SMILES C(=O)(CCCCCOCC)NC1C2CN(C(CC(C=C)C)=O)C1C2 N1(C(CC2(C)CC2(Cl)Cl)=O)CCC(CNC(=O)CCCC2CCC2)CC1 C1(C(=O)NCC(C(C)C)(C)NC(C2OCCC2C(F)(F)F)=O)CC(=O)C12CCC2 C(=O)(CCCN(C(C)CNC(=O)CNC(C1CC12CCC2)=O)C)NC c1(C(=O)NCCC(C)NC(CCc2cnc(C)o2)=O)ccncc1OC(C)(C)C c1(C(=O)NC2C(CNC(c3c(OC)cc(C)cn3)=O)C2)sccc1S(N)(=O)=O CC(O)CCCCCC(=O)NCC(CNC(=O)CN(C)CCN(C)C)C(F)(F)F C1(C(=O)NC(C)(C)C(c2ccc(Br)cc2)=O)CCC(F)(F)CO1 c1(C(=O)NCCN(C(C)C)CCO)cc2oc(Cl)cc2[nH]1.C1CC(=O)N1C C(=O)(C(CC)(CC)CO)NC(CC=C)CNC(C1OC2CCC1C2)=O N1(C(Cn2ccc(C)n2)=O)CC2(CCC2CNC(=O)CCN2CCC(F)C2)C1 N1(CCCC)CCC(C(=O)NCCC(CNC(=O)CC)O)CC1 C#CC1CCC(C(=O)NC2CCC(NC(C3CC4CC3CC4O)=O)C2)CC1 C12(C(=O)NCCC3CCC(C)O3)COCC1CN(C(c1nc(=N)cc[nH]1)=O)C2 c1(CC(=O)NC(C2CCN(C(=O)CCc3nccs3)C2)C)ccncn1 c1(CNC(C(F)NC(=O)OC(C)(C)C)=O)ncncc1Cl c1(NC(c2n(CCCSC)nnn2)c2csnn2)ccc(Br)c2c1OCCO2 C1(O)(CNC(CC2(C)CCN(C(C)=O)C2)=O)CCCN(C(c2occc2C)=O)C1 C(=O)(N=c1[nH]nc(-c2ccc3c(c2)OCO3)s1)CC(C)CSc1ccccc1 N1(Cc2cn(-c3c(C)cccc3)nn2)C(C)CN(C(=O)CCc2cn[nH]c2)CC1C Cc1cc(F)ccc1C(N1CC(NC(c2nc(Cl)ccc2F)=O)CC1CO)=O C1(C(=O)NCCC(=O)NCC2(CC(=O)NC(CC)C3CC3)CC2)CCCO1 N1(C(Cn2nc(C)oc2=O)=O)CCN(C(c2cc(Cl)cc(C)c2O)=O)CC(O)C1 N1(C(C2C(C(C)C)(C(=O)O)C2)=O)CCn2c(cc3c(Cl)cccc23)C1 C1(OCC)CCCC(c2nnnn2CCCF)(NCC(C2CC(F)(F)C2)(F)F)C1 C1(CC(=O)NC2(C(=O)OC)CC2)CCN(C(=O)Cc2cc(C)on2)CC1 C1(CCC(=O)N(CC(CNC(COCC(=O)NC)=O)O)C)CCCCO1 c1(C(N2CCC(NC(=O)NCC(n3ncc(C)c3)C)C2)=O)ccc(N(C)C)nc1 CCC(C)(CN=c1[nH]c(=NCCc2ccc(Br)s2)[nH]c2c1COC2)C(N)=O N1(Cc2ccn(C)c(=O)c2)CC(C)(CC)CC1=O C1(CNC(C2CCCS2)=O)CCCN1C(=O)CC(O)C1CCCC1 C1(C(=O)NCc2c(C(C)C)ocn2)CN(C(=O)C(O)C2CCC2)CCO1 c1(CCCN)ccc(F)cc1.C#CCCCN(CCCCO)CC=C Cc1ccc(NCC(=O)NCCCNC(C2(Cc3cncs3)CC2)=O)cc1 C1(C#N)(COC)CN(C(=O)NC2CCC=CO2)C1 c1(C(=O)NC2C(NC(c3scc(C)c3Cl)=O)C2)c(F)ccc(F)c1O C(=O)(C1=CCC(C)CC1)NC1CC2(CC(NC(Cc3c(OC)cccc3)=O)C2)C1 N1(C(c2cnc(C(C)C)o2)=O)CCC(C(=O)NC(CO)CCC2CC2)(C(C)C)C1 C(CC(O)C(=O)NCCCCCC1CC1)NC(Cc1scc(C)c1)=O c1(C(=O)NC2(C)CN(C(c3cccc(CC)c3)=O)C2)ccc(C#N)c(O)c1 c1(CCNC(c2nnnn2CC2(C)CC2)CCC)cc(CC)no1 N1(C(CCOCC#C)=O)CCC(NC(=O)CC2CCC3CC23)C1C(C)(C)C O=C(CC(C(F)(F)F)NC(c1cnsc1)=O)NCCN1C(=O)CNC1=O CCC(C(=O)N1CC2CCC(CNC(c3c(C)ncnc3C)=O)C2C1)C(F)(F)F c1(C(=O)NCCNC(c2ncc(C)cc2Br)=O)oc2c(C)cccc2c1C c1(C(N2CCN(C(c3c(O)nc(=N)[nH]c3)=O)CC2)=O)ccc([N+](=O)[O-])cc1F C1(N(C)C(C2CCC(C)(C)C2)=O)CCC2CN(c3ccnc(C4CC4)n3)CC2C1 C1(C(C(N2CC(CN(C(CCOC)=O)C)C2)=O)O)CCCCC1 CCCCCC(O)CC(=O)NC1CC(C)N(C(=O)Cc2ccc(F)cn2)C1 c1(C(=O)NC2CCN(C(CCOC)=O)C23CC3)ccc2nc(C)c(=O)n(C)c2c1 c1(OC)ccc(C)cc1C(N1C(C(=O)Nc2ncc(O)cc2Cl)CCC1C)=O c1(CC)nonc1C(=O)NCc1cc[nH]c1C(=O)O.C12(CC1)CC(=O)NC2 N1(C(CC(=O)NCC#C)=O)CCC2(CCCN(C(c3ccn(C)n3)=O)C2)C1 C#Cc1cccc(C(=O)NC(C(=O)NCC(c2ccccn2)O)C(C)(C)C)c1 C(=O)(C(=O)CCC(C)C)NC1CCC(C(=O)NCC(COC)(C)O)C1 Cn1cnc2c1CCC(C(=O)NC(C)(C)CNC(c1cnc(S)n1C1CC1)=O)C2 C#CC(C)N(C)N1CCN(CCOS(C)(=O)=O)CC1 CCC(COC)C(=O)NCCN(C(c1ccccc1OC)=O)Cc1ccccc1 c1(C(C)(C)C)cc(C(=O)NCCCCCNC(=O)Cn2cc(C(O)C3CC3)nn2)on1 C1(C(=O)NCC(CN(C(=O)CCC2CC2)C)O)CC12CCSCC2 c1(C(=O)NCC2N(C(C3CC(CC(=O)OC)C3)=O)CC2)cc2cccn2cn1 C1(C(=O)NCC(c2ccccn2)NC(C2CC(=O)C2)=O)CC(F)(F)C1 C1(CNC(COC(C)(C)C)=O)CCC(C)(C)CN1C(=O)CCCc1ccncc1 C1(C(=O)NCC2N(C(C3=CCCC3C)=O)CCCCC2)CN(C)C(=O)CCO1 N1(C(c2c(C)c[nH]n2)=O)CCN(C(c2cn(C)nc2Cl)=O)C2CS(=O)(=O)CC12 CC1=NC(C)(C(=O)NCCC2CCCN(C(=O)C(O)C(C)C)C2)N1CC1CC1 N1(C(C2CCC(=O)NC2)=O)CCC2C(C1)CN2C(c1cncnc1)=O N1(C(C2C(OC)C2)=O)CC2CCN(C(c3noc(C4CC4)c3C)=O)C2C1 C1(C#N)(CC)CCN(C(=O)CN(C(c2cc(C#N)ccc2N)=O)CC2CC2)CC1 C(CCC(=O)NC(C)CCCNC(=O)C(c1ccn(C)n1)C)N(C(C)=O)C N1(C(c2nc(CC)oc2)=O)CC(C)(C)CC1CC(=O)NCc1c(O)cccc1F C(C(=O)N1CC(NC(C2CC(C)(C)C2)=O)C(C(F)(F)F)C1)(C(C)C)OCC(C)C CC1(C)C(NC(=O)CC2CCCOC2)CCN1C(=O)C1=CSCS1 c1(C(=O)NC2C(NC(C(CC)N3CCCC3=O)=O)C2)cc(NC(C)=O)cnc1O c1(-c2ccc(CN3C(CC)CCCCC3)o2)c[nH]c2ccccc12 C=CC1CN(C(=O)C2=CCCC2C)CC1NC(c1cscc1C(N)=O)=O C(CCC(=O)NC1(C(=O)NC2CC(O)C2OC)CC(O)C1)SC C1(N(C(=O)C(C)C)CC#C)CCCCN1NC(=O)C1CCC1.C1(=O)CCN1 C12(CNC(C34OCC(NC(c5occ6c5CCC6)=O)(C3)C4)=O)COC(C1)C(O)C2 C1(N(C(=O)CN(C2CCC2c2ccccc2)C)C)Cc2ccccc2C1 c1(C(=O)NC2(CO)CC2)cccc(S(=O)(=O)N2CCCCC2)c1 N1(C(c2ccc(C(C)C)cc2)=O)CCN(C(=O)C2CC2)C(C2CCC2)C1 c1(C(=O)NCC2(C)CCCN2C(=O)CCC2CCC2)cc2ccc(O)cc2[nH]1 CC(CNC(C1(N(C)C)CCC1)=O)C(=O)NCC1(O)CCOC1 C=CCC(C)(C)CC(=O)NC(C1(O)CCN(C(c2cc(C(C)C)oc2C)=O)C1)C C1(C(=O)NCCOCCCN(C(=O)Cc2ccco2)C)CC2CC1C2 c1(CCC)sc(C(N2CC(CNC(C3(C)CCCC3)=O)CC2C)=O)cc1CC O=C(C1=NOC2COCC12)NC1(CC(N2CCCC(C(F)F)C2)=O)CC1 c1(C(=O)NCC2(NC(=O)C(F)(F)F)CCCC2)cnc2sc(Br)cn2c1=O C1(OC(C)C)CCN(C(C2CC(C)N2C(=O)COc2cccnc2)=O)C1 c1(C(N2CC3C(NC(=O)NC(CC#C)C(N)=O)(C3)C2)=O)c[nH]c2nccc-2c1 N1(C(CCOC(c2ccccc2)C)=O)CCOC(C(=O)O)(C(=O)O)C1 C(c1csc2ccccc12)=CC(C)NC(C1(OCC)CC=CC1)c1nnnn1C C#CCCCCCC(=O)NCC1(O)CCN(C(c2cn3c(n2)CCCC3)=O)CC1 c1(CN(CCN)CC)ccc2nonc2c1 N1(C(C(C)SCCCC)=O)CCN(CCN(C)C(C2C(C)(C)C2(F)F)=O)CC1 c1(C(=O)NC2CC(N(C(C3N(CC)C(=O)CC3)=O)C)C2)cn(C)c2ncccc12 C1(CNC(C2(C(=O)NC)CC(C)(C)C2)=O)CC(C)(C)CN1C(C1CC1COC)=O C(=O)(C1SCCc2sccc21)NC(CCCC)CNC(c1cnn(C)c1SC)=O C1(NC(c2c(C)nc(C)o2)=O)CCCC(NC(C2CC(=O)C2C)=O)CC1 c1(N(C(C)=O)C)ncc(Cl)c(C(=O)NCC2(F)CC2)n1 C1(CC(=O)NC2(CCNC(CCOCC(C)C)=O)CCC2)CCC(C2CC2)O1 c1(C(=O)NCC2N(C(C3OCCC(=O)C3)=O)CC(O)C2)cc[nH]c2nccc1-2 c1(CNC(C=CC(=O)NC)=O)cccc(C)c1.C12(O)CN(C1)C(=O)C=CC2 c1(C(=O)NC(C)CNC(=O)C(C)OCC#N)cnn(C2CCC2)c1 C1(C(=O)NC2(COC)CN(C(C3(CF)CC4(CCC4)C3)=O)C2)CCCCOCC1 N1(C(C(COC)O)=O)CC(=O)NCC1C(=O)NCCc1ccncc1C C(=O)(CC1=CCOCC1)N1CCC(NC(=O)C(O)C2CCC2)C1c1ccccc1 C(CCCCCCC)NC(C1CCCN(C(COCC=C)COC)C1)=O N1(S(CC)(=O)=O)CCCC1C(N1CC=CC1CN(C)CCn1cc(C)cn1)=O Cn1cc(Cl)c(C(=O)NCC(CO)NC(c2cccn2C)=O)n1 C(C)(C)(CC(=O)N1CC(CNC(c2sccc2CC#N)=O)(OC)C1)OC Cc1[nH]c2ccccc2c1C1=CCN(C(C2CC(C)(C(C)(C)C)C2)=O)CC1 N1(C(COCCCC)=O)CC(CNC(=O)CC2CC(F)(F)C2)N2CCC1C2 C1(C)(C(C)(C)CNC(C2CCCC2O)=O)CCCN1C(c1cc(Cl)cs1)=O c1(-c2n(C(COC)C)nc(C3CCCO3)n2)nn(-c2ccccc2)cc1[N+](=O)[O-] C#CCC(C)C(=O)NC(C)CNC(=O)COc1ccc(C(C)C)cc1 N1(C(Cc2c(OC)ccnc2)=O)CCC2CCN(C(=O)Cc3csnn3)CC2C1 N1(C(CC2C(C)CCN(C(C3(CC(C)=O)CC3)=O)C2)=O)CC2(CNC(=O)C2)C1 C1(NC(c2c(C(=O)OC)coc2)=O)CCOCC1NC(=O)Cc1cc(C)nn1C C1(CC=C)(NC(C2CCOCC2)=O)CCN(C(C2CC(=O)N(CC)C2)=O)C1 C(=O)(CCCCC(=O)N1CC2(CCC(NCc3c(Br)cnn3C)C2)C1)OC N1(C(CC2N(C(C3(C)CC4(CC4)C3)=O)C3C2CCC3)=O)CCC2CCC(C2)C1 c1(N2CCCC(N3C(=O)NCC3)C2)nc(=NCCC(F)F)[nH]c2c1CCCCC2 c1(C(=O)NC2CC(C(=O)NCc3ccc(Cl)nc3)C2)ccccc1C1CC1 N1(C(C=CC2N(C)CCC2)=O)CCCC(C)(C)C1CNC(c1cccc(Cl)n1)=O C1(C(C)C)CN(C(=O)C(C)n2ccnc2)CCN1C(=O)CCNC(=O)CO c1(C(N2C(CNC(C3CC4C=CC3CC4)=O)CC2)=O)cc(F)ccc1Br C1(C(N(C)CC2COCCN2C(c2cccc(=O)o2)=O)=O)Cc2ccncc2C1 c1(OC)ccc(C)cc1-n1cc(-c2cscn2)nn1.C12CN(CC1C)C2=O C12(CN(C(c3cc(C)no3)=O)C1)C(=O)NC2.CCC(CSC)OC N1(C(CC(C=C)(C)C)=O)CCC2(CNC(c3coc(SC)c3)=O)CCCCC12 C=CCCC(C)(C)C(=O)N1CCCC(NC(c2ccc(C(F)(F)F)cc2)=O)C1 Cn1cc(C(=O)NCC2CCCOC2C(C)(C)C)c(=O)c2cnn(C)c12 S(=O)(=O)(c1nc2c(s1)C(=O)CCC2)Nc1cccc(C2C(C)(C)C2(C)C)c1 Cc1cc2cccnc2nc1C(=O)NC1CCC(NC(=O)Cn2cnnc2)CC1 C1(OC)COCCC1CC(N1CCCC1CCCNC(c1coc(O)n1)=O)=O C(CO)(CO)N(C(C=CC(C)NC(C1CC(OC2CC2)C1)=O)=O)C c1(CNC(C(C(C)C)F)=O)nnc2n1CCN(C(=O)Cc1nc(C3CC3)cs1)C2 c1(C(=O)NC2CC3(C2)CC3C(=O)NCC2CC3(CCC3)C2)c(F)cccc1F c1(C(N2CC(C=C)C(NC(c3cnc(C)[nH]3)=O)C2)=O)sc2ccccc2c1Cl C1(CC(=O)NCC2(CO)CCCC2)C=CC(NC(c2cncs2)=O)C1 C(=O)(C(C)(C)C1=CCN(C(c2cccnc2S)=O)C1)N1C(C)C(C)(C)CC1 CC(C)C(CCNC(=O)C(C)(C)c1ncco1)NC(=O)C(F)C1CCC1 C(=O)(C(C(C)C1CCOCC1)N(C)Cc1ccccc1Br)NCCCCCC Cc1cc(C)c(C(=O)N(CC(O)CN(C(=O)C(c2cccnc2)O)C)C)s1 C1(C(N(CCC(C)(C)NC(Cc2c(C)nccc2)=O)C)=O)CC2CCCCN2C1 c1(C(=O)NCC2(C(C)NC(C(CC(C)C)C)=O)CC2)cccc2c1OCC2(C)C c1(C(N(C(CNC(C2CC(CC(F)(F)F)C2)=O)C2CC2)C)=O)ccc(Cl)[nH]1 CC1(C)CCOC1CC(=O)NCC1CC(NC(=O)C2=CCSC2)C1 c1(CC)ncc(C(=O)NCCC2CCN(C(C3(CC(=O)OC)CNC3)=O)C2)[nH]1 c1(C(C)NCc2c(N3CCN(C(=O)OCC)CC3)cccc2)ccc(Cl)nc1Cl Cc1cnc2c(cnn2CC(N2CCCC(C(C)(C)O)C2)=O)c1 c1(C(N2CC(NC(C3CCSC3)=O)CC3(C2)CC3)=O)cc2cc(Cl)cnc2o1 c1(OC)cc(C)nc(N2CCC(O)(CNC(C3CCCC(F)(F)C3)=O)CC2)n1 N(C(=NCCC(C)C)NCC1CCC2(COC2)O1)C(c1ccccc1)C Cc1n[nH]c(C)c1C(C)C(N1CCC(C(C)NC(c2ccc(F)cn2)=O)C1)=O c1(C(=O)NC2(C)CCN(C(C(C(C)C)C#N)=O)C2)ccsc1S(N)(=O)=O C1(C(=O)NC(C(=O)OC)C2CCC2)CCCN(C(c2cn(C)nc2OC)=O)CC1 Cc1cn2cc(C(=O)NCC(C)NC(=O)Cn3[nH]cc4c(=O)ncnc3-4)sc2n1 CN(C)N=Nc1ccccc1CN1CCOCC(O)(CO)C1 C1(c2cccc(OC)c2)CN(C(=O)COCCF)CCN1C(C1(C)C=CCC1)=O c1(C(N2C(CNC(C(C)SCCC(C)C)=O)C=CC2)=O)cc(C(C)C)ccc1O C1(N(C(C2C(C(C)C)CCC2)=O)C)CCCN(C(c2cnc(F)c(Cl)c2)=O)CC1 c1(C(=O)NC2COCCN(Cc3cc(C)[nH]c3C)C2)c(Br)ccc2cccnc12 C1(O)(CNC(CCC2CC(NC(C=CCCC)=O)C2)=O)CC2CCC1O2 C1(C(=O)NCC2CCCC(NC(=O)Cc3ccsc3C)C2)(CC)CCCCC1 C1(C(=O)NC(CNC(Cc2ccn(CC)n2)=O)CC)COCCN1CC(F)(F)F N1(C(CC2CC(NC(CC3COCC(C)O3)=O)C2)=O)CCC(F)(F)C(O)C1 c1(CCC)ncc(C(N2CC(O)(CNC(c3coc(C)n3)=O)C2)=O)s1 C1(C(N2CCN(C(C(C(C)O)C)=O)CC2C)=O)OCC2CCCC1C2 CC(C)CC(C)CC(=O)NCCCC1(O)CN(C(=O)C(C(C)C)NC=O)C1 c1(CC(N2CC3CCC2C3)=O)ccncc1Cl.C12(CC=CC1)C(=O)NC2 n1(CC(=O)NC2C=CCN(C(c3ccc(CC)[nH]3)=O)C2)[nH]cc2c(=O)ncnc1-2 N1(C(c2c(OC)n(C)nc2)=O)CCC2CCCC(C1)N2C(C1CSCCS1)=O N1(C(c2ccc(F)nc2)=O)CC2CCC(Nc3ncncc3Cl)CC2C1 C=C=CC(C)C(=O)N1CC(F)CC1C(=O)N(C)OC C12(CNC(C3N(C(C4C(C)C4C)=O)CCOC3)=O)CCN(CC1)CC2 C12(CC(=O)Nc3c(CNC(C=CC)=O)ocn3)CC1CN(C(=O)OC(C)(C)C)C2 Cc1cc(=NCC(C(C)C)N(C)C)[nH]c(N2CCC(CS(C)(=O)=O)CC2)n1 C1(NCC(=O)NC(C)C)CC2CC(NC(C3CSC3)=O)C1C2 C(=O)(C(C)(F)C(C)(C)F)NCc1ccc(CN(C(c2nc(C)nn2C)=O)C)cc1 c1(C(=O)NCCC(CNC(C2C(C)N(C)CC2)=O)O)cc(F)c(F)c(Cl)c1F C1(C(=O)NCCc2n(CC)cnn2)(CC)CCN(C(c2sccc2OC)=O)CC1 C1(C(=O)NCC(C)(C)CCO)(COC)CCCCCC1 c1(C(N(CC(CC)NC(C23CC(CO2)C3)=O)C)=O)csc(CSC)n1 CCCC(C)(CC)C(=O)N1CC=CC(NC(=O)Cc2ccc(OC(F)F)cc2)C1 C1(C(=O)NCC=C)CC(F)(F)CN1Cc1ccc(C2CC2)cc1 N1(C(C(=O)NC2C(NC(c3ccn(C(CC)CC)n3)=O)C2)CC)C(=O)CCC1=O C1(CC(=O)NCC(CC=C)NC(c2[nH]cc3c2CCC3)=O)CCC(C)(C)CO1 C1(NC(c2cccc(S(=O)(=O)NCCC=C)c2)=O)COc2cccc(Br)c2C1 c1(C(=O)NCC2(C)CCN(C(C3CC(C(F)(F)F)C3)=O)C2)cc(Cl)ncc1O c1(OCCCC(=O)N(CCNC(CSCCCC)=O)C)ccc(C)cc1Br N1(C(C2CN(CCC)C(=O)C2)=O)CCC2(CCC2NC(=O)CN(C)CCC)CC1 N1(C(C2CCN(C(C(CN(C(C)C)C)C)=O)CC2F)=O)CCC(C)(C2CC2)C1 C1(CNC(C2CCN(CC=C)C2)=O)CCCCN1CCC(C)C N1(C(C(CCCC)(C)F)=O)Cc2n[nH]cc2C1C(=O)N1CC2CCC1C(CO)C2 N1(C(C2CC(OC)C23CCC3)=O)CCCN(C(=O)CC2CCC=CCC2)CCC1 N1(C(C(CCF)NC(c2nn(C)c(Cl)c2)=O)=O)CCOCC(C)(C)C1 c1(OC)nc(=NCC2CN(C(c3nc(O)sc3C)=O)CCCO2)[nH]c2[nH]cnc12 c1(CC(=O)NC(C(C)C)(C)CNC(=O)CN2CCC2C)cc2cc(Cl)ccc2[nH]1 N1(C(C2CCC(CC)O2)=O)CC(NC(=O)CCc2cn[nH]c2)C2CCCC12 C(C1CCC(C)CC1)=C(C)C(N1CC(O)(C(C)NC(c2ncoc2C2CC2)=O)C1)=O CC1CC2CN(CC3C(=O)NCCN3Cc3ccccc3)CCN2C1 c1(NC(c2scc(OC)c2)=O)cccc(F)c1CSC c1(NC(C(=O)N(CCC(=O)O)Cc2ccccc2)=O)c(F)cc(OCF)cc1F c1(C(=O)NC2CN(C(CCCCOC)=O)CC2O)nn(C)c(C)c1Br CCCCCC(=O)NCC(N1CC(CNC(=O)COCCF)C(O)C1)=O n1(CC)nccc1C=CC(=O)NC(C1(O)CN(C(C2CC(C)OC2C)=O)C1)C c1(CC(N2CCC(N(C(c3nnnn3C)CC)C)C2)=O)cc(F)cc2c1OCC2 C1(NC(C(CCOC)C)=O)CC1C1CCCN(C(c2coc(C3CC3)n2)=O)C1 N1(C(C(CC)=CCCC)=O)C2CCC1C(CC(N1CCC13CCOC3)=O)C2 C1(CNC(c2cnc(C)s2)=O)C2CN(C(=O)CCCNC(N)=O)CC12 c1(CNC(C2=CCCC2C)=O)nn(C)c2c1CN(C(C1CN(C)C(=O)N1)=O)CC2 C(C(CO)C(F)(F)F)NC(C(C)OCc1ccoc1C(N1CC=CC1CF)=O)=O C(=O)(C1=NOC2(CCC2)C1)N1CCC(NC(C(CCCC)(C)C)=O)C(C)C1 Cc1cc(C(=O)N(C)CCC2CCCCN2C(=O)CN2CSCC2=O)cc(N)c1 CC1CCN(C(c2ccc(CN=[N+]=[N-])cc2)=O)CC1NC(c1ccc(F)cc1)=O N1(C(Cc2cn(C)nc2)=O)CCC(NC(C2CC3CCCC2C3)=O)CC(C)(C)C1 C1(C(=O)NCC2C=C2C)(OC)CCN(C(=O)C(C(C)C)OC(C)=O)CC1 C1(C#N)(C(N(C2CCN(C(CCOCC#C)=O)CC2)CCC)=O)CC2CCC1C2 N12CC3CCCN(C3C1)Cc1nccc2n1.c1(C(=O)OC)cc(Cl)nc(Cl)c1 C=CCC(C(=O)NC1COC(C)(C)C1)NC(=O)CC1CC(=O)C1 c1(C(=O)NCC(C2(O)CN(C(CSCC)=O)C2)(C)C)cscc1C#N C(=O)(C(C)CCCC(C)C)N1CCC(CNC(C(CC2CCC2)OC)=O)C1(C)C CN1CCN(CC(=O)NCCN2CC3C=CC2C3)CC1.C1(NC(CC)=O)CCCC1 c1(C(N2CCC(C(C(=O)N(C)CCOCCO)(C)C)C2)=O)cccc2cc[nH]c12 C1(C2CCC2)C(=O)N1.C1(C)(OCCNC(C2(CO)CC2)=O)CCC1.CC C1(NC(C=CC(C)C)=O)CC2(C1)CN(C(C1CCC(F)(F)CO1)=O)C2 C=CC(C)(C)C(=O)Nc1ccc(C(C)NC(=O)C(=O)NCC2CC2)cc1 C(CC1CCC1)(C(=O)N1CC(O)(CCNC(C23CCCC2C3)=O)C1)OC CC(CCl)(CCl)CS(=O)(=O)N1CCC(NC(=O)CCOc2ccccc2)C1 c1(N2CCCC(NC(C(C)N3CCC3)=O)CC2)nccn2nnnc12 Cc1ccccc1C(=O)NC1CC(NC(C2(NC34CC(C3)C4)CC2)=O)C1 c1(C2(C)CC2)cccc(C(=O)NCC2CC2CNC(=O)CO)c1 C(CO)(C(=O)NCn1cc(CNC(=O)C(C)O)nn1)OC c1(NC(C)=O)ccc(CC(=O)NCC(C)(O)CNC(=O)C2=CCCS2)cc1 c1(OCC)ccc(C(N2CCC(O)C(C(=O)NCC3CCC(F)C3)C2)=O)cc1Br N(C1CCCc2ccccc21)CCC(=O)NC1CC(C(=O)OC)C12CCC2 c1(C(=O)NCC(CN(C(=O)COC(F)F)CC)(C)C)ccc(C(C)C)nc1 C(CS(=O)(=O)CC)NC(c1n(CCC)nnn1)C1CC1Cc1ccccc1 Cc1cncc(C(=O)NC2CCCN(C(=O)Cc3ccnn3C)C2C)c1Cl n1(C(C)C(=O)NC(C)(CNC(=O)C=CC2CC2)C2CCC2)ccc(C(F)(F)F)n1 CC(CC(=O)NCc1ncccc1NC(C1CSCC(=O)N1)=O)C(C)(C)C N1(C(CCCOc2cn(C)nc2)=O)CCC(O)C(NC(=O)C#CC2(C)CC2)C1 Cc1ncc(C=CC(=O)NCCC2CC(NC(c3cnc(N)cn3)=O)C2)s1 c1(C(N2C(C(N(C3CCOCC3)CC)=O)CC(OC(C)=O)C2)=O)cc(Br)ncc1Cl c1(C(=O)Nc2c(C(=O)NC)nccc2)nc2ccc(-c3cnc(O)nc3O)cc2s1 c1(OC)cccc2c1OCC2NC(=O)C(C)=CCSC CC1(NC(C2CCC2c2cccnc2)=O)CN(C(=O)C(C2CCOCC2)=O)C1 N1(C(C2C(=C)CC2)=O)CC2(CC2)CC1C(=O)NCC1CCCC1 N1(C(C2OCCC(NC(CCCN(C(C)C)C)=O)C2)=O)CC2(CCOC(=O)N2)C1 Cc1ccc2oc(C(N3CCCC(CN(C(=O)C=CC(N)=O)C)C3)=O)cc2c1 c1(C(=O)NCC(C)N(C(C2=NOC(C)C2)=O)C)cc2cc(Br)cn2cn1 C1(CC)CCc2sc(C(=O)NC3CC(C)(NC(C4CCN(C)C4=O)=O)C3)cc2C1 C1(C)(CC(N2CC(C(C(=O)N(C(C)C)Cc3ccsc3)O)C2)=O)CCCO1 CC(C)C(C)C(CNC(=O)CCC(=O)N1CCOCC1)NC(c1ccccc1F)=O C(=O)(C(C#N)C(C)(C)C)C1C2(C(N3C(C)CC(C(=O)N)C3)=O)CCC(C1)C2(F)F Cc1cc(C(=O)NC2C3CC2N(C(C2CC(C)(C)CN2C)=O)C3)nc(O)n1 CCS(=O)(=O)CC(=O)NCC1CC(C)CN(C(=O)C2=CCSC2)C1 CC(C)CC(O)CC(=O)NCCCC(C)NC(C1(C)CCCNC1=O)=O CCC(CC(C)C)C(=O)N1CCC(NC(=O)CC2CSC2)CC1C c1(C(N2CC(C3(NC(=O)CC(F)(F)F)CC3)C2)=O)cnc2ccoc2c1 C1(CNC(C(CNC(c2cnc(OC)s2)=O)OC)=O)CC(=O)N(C)C1=O N1(C(C2N(C(C(C)c3cc[nH]n3)=O)CCC2C)=O)CCOC(C2(C)N=N2)C1 c1(OC)ccc(C(=O)NCC2CCC2NC(c2cc(Cl)cnn2)=O)c(F)n1 N1(C(c2cc(C)oc2)=O)CC(NC(c2ccccc2CC(C)(C)C)=O)CC1C C(N=c1cc(CC2CC2)nc[nH]1)C1CCC(NC(CC2OCC(C)(C)C2)=O)C1 N1(C(C2(C#N)CCC2)=O)CC2C=CC1C(C(=O)NCC1CC3(CCC3)C1)C2 C(=O)(CC(C)(C)NC(=O)CSc1ccc(SC)cc1)NC C1(C(=O)NCC2CCN2C(C2CCc3n[nH]cc3C2)=O)CCn2ccnc2C1 CN1CCC(O)C(C(=O)Nc2cc(CNC(=O)CC3CCCSC3)no2)C1 C1(N(C(c2cc[nH]c2C)=O)CC)CCCN(C(C23CC(C)(CO2)C3)=O)C1 c1(C(=O)NCCCNC(COCC=C)=O)cc(F)cc(C)c1N c1(C(=O)NC23CN(C(C(CCC)CC)=O)C(C2)C3)cc(C)c(CC)nc1O C(CC(C)(C)CNC(=O)C(c1cccs1)NC(C1(C)C=CCCC1)=O)OC C(CCCCCCCCCCO)N.O=C1CCO1.C(C(F)(F)F)C=O N1(C(C(C)N(C(C)=O)C)=O)C(C(N2CC(C)CC(C)C2)=O)C2CC(F)C1C2 c1(NC(N2CCC(c3[nH]nc(N(C)C)n3)CC2)=O)c[nH]c2cccnc12 S(=O)(=O)(c1ccc(Br)cc1Cl)N1CC(CC)C1.c1(N)ncnc(-c2ccccc2)c1N C(=O)(CC(CN(C)C)C(F)F)NCC1N(C(COC(C)C)=O)CC(C)(C)C1 CCC(C)C(C(=O)N1CC(CC)(OC)C1)NC(=O)CN(CCO)CCOC N1(C(C(CC)Cc2ccccc2)=O)CC2CC(C1)N(C(=O)CSCC(=O)OC)C2 C(Cc1cn[nH]c1)(C(=O)N1CCCO1)NC(CC1N(CC)CCOC1)=O C(CCCCC(=O)NC(C)(CNC(c1c(C)c[nH]c1CC(N)=O)=O)CO)SC CCCC(C(=O)NCc1ccsc1C(=O)NCC1(OC)CCC1)NC(N)=O c1(C(=O)NC2(CO)CN(C(c3occ(C(N)=O)c3)=O)C2)csc2c1CCCC2 CCCCCC(C)CC(=O)N1CCCC1C(C)(C)C(=O)NC(C)COC(F)(F)F CCC(C)(C)CC(=O)NC1CCN(c2cc(CCOC)ncn2)CC1F Cc1cccc2c(CC(=O)NC3CCC(NC(=O)C(C)(C)CF)C3)c[nH]c12 c1(NC(C#C)=O)cccc(CCC)c1Br.C12(C)CCCN1C(=O)OC2=O C12(NC(c3cncc(C(C)=O)c3)=O)CCN(C(C3CCSCC3)=O)CC1C2 C1(CN(C(c2ccc(C#N)s2)=O)CC)CCN(C(C2CCC(F)C2)=O)CC1 C1(CC=C)(C(N2CC(NC(C)=O)C2)=O)CCN(C(C2CC=CCC2)=O)C1 C(=O)(CC(C)C)N.C(CC(=O)N(C)CCNC(=O)CCOCC1CCC1)N(C)CC Cc1nn(CC(=O)NCCN(C)C(c2ncncc2Cl)=O)c(=O)o1 N1(C(C(n2ncc(C)c2)C)=O)CCC(NC(c2ccon2)=O)C1C Cc1c(CN2CCC(C(CNC(=O)CCF)(C)C)CC2)ccn1C C#CC1(C(=O)NCCC2CCCCC2)CN(C(=O)CC2C=CS(=O)(=O)C2)C1 c1(C(=O)NC2CN(C(C(CC)C)=O)CC2CC)nnc2ccccc2n1 C1(C(=O)NCCOCCNC(C(=O)OCCN2CCOCC2)OC)CCOC1=O c1(C(=O)C(N2CCN(C(C3CCCO3)=O)C(CO)C2)=O)ccc(F)c(F)c1F Cc1ccc(CNC(C2CC(NC(=O)CC3CCN(C(C)C)CC3)C2)=O)nc1 CCCC(C(=O)OC)C(=O)N1CCC(N(C(=O)CCc2scnc2C)CC)C1 c1(C(C(=O)N(CC(=O)N(c2ccccc2)CC2CC2)C)=O)ccc(Cl)cc1 CC1(NC(=O)Cc2cncc(O)c2)CCCN(C(c2cc(C3CC3)[nH]n2)CCl)C1 Nc1c(C(=O)NC(CNC(=O)CN2CCC2C)CO)cccc1F c1(C(C(=O)OCC(=C)C)N(C)Cc2cc(Br)ccc2OC)cc2ccccc2s1 N1(C(C2CN(C(C)C)C(=O)CC2)=O)CC2CC(NC(=O)C(=O)OC(C)C)C(C2)C1 S(=O)(=O)(c1ccc2c(c1)CCC2)Nc1ncc(-c2ccc(C)cc2)cc1C C(CN=c1cc(NCCc2ncccn2)nc(CC)[nH]1)NC(=O)NCC c1(C(=O)OC2CCC(C)S(=O)(=O)C2)ncnc2c1CCC2 C1(NC(c2c(C)c[nH]n2)=O)CCN(C(c2cc(C(F)F)on2)=O)C(C)C1 CC1CC(C(N2CCC(N(C)C)(CNC(c3ccn(C)n3)=O)C2)=O)CC(=O)N1 c1(C(=O)NCC2(C(C)NC(=O)C=C3CCCC3)CC2)ccc(C(C)(F)F)nc1O C(=O)(C(C)CS(C)(=O)=O)N1C(CNC(c2ncc(C)c(C)c2)=O)CC1 N1(c2nc(O)nc(C)c2C#N)CCCC1C1CCCCN1C(c1nocc1Cl)=O c1(NCc2cnc(CCC)s2)ccc(S(=O)(=O)N2CCC(CO)C2)cc1Cl O=C1CC(NC(C2(F)CCCN(C(=O)CC3CCCNC3=O)C2)=O)CC(=O)N1 c1(C(=O)NC2C(CNC(c3c(C(C)(C)C)n[nH]c3)=O)CC2)ncnc2sccc12 N1(C(C(C)OCC=C)=O)CC(C)(C(=O)N(CC(F)F)C)CC1(C)C Cc1[nH]c2ccccc2c1CCC(N1CCC(NCc2cncc(Cl)c2Cl)C1)=O C1(NC(CSCC(C)C)=O)CC(C(=O)N(C)Cc2ccc(F)cc2)C1(C)C C1(NC(CC2CCCC(C)O2)=O)CC(F)CN(C(=O)Cn2ncnn2)C1 N1(C(CC2N(C(C3C4CC(=O)CC43)=O)CCC2)=O)CC2(CCC(=O)O2)C1 N1(C(c2c(C(C)C)scn2)=O)CC2CN(C(=O)Cn3nnc(=N)[nH]3)CC2C1 c1(CNC(C(CC)COC)=O)n[nH]c2c1CN(C(=O)C1=C(C)CCCC1)C2 c1(C(=O)NCCn2cc(CNC(C3CCCC(C)C3)=O)nn2)cc([N+](=O)[O-])c[nH]1 Fc1c(Cl)ccc(Br)c1NCC(F)C(F)F c1(C(=O)NC2C(CNC(c3c(=N)[nH]cnc3)=O)C2)ccc2c(c1)CCCCS2 N1(C(c2cnc(CC3CC3)s2)=O)CCOCC1c1ccc(Br)cc1 c1(C(N2CC(NC(=O)Cc3nnc(O)s3)C(F)C2)=O)ccc(F)c(C(F)(F)F)c1 CC(C)C(F)(CNC(c1cc(C(F)F)[nH]n1)=O)C(=O)N1CCC2(CC(CO)C2)C1 c1(OC)ncc(Br)c(NCCCC(C)NC(C2CCCC(O)C2)=O)n1 C(CC(C(=O)NC1CC1NC(=O)Cn1nnc(-c2ccsc2)n1)NC(C)=O)OC CC1(CCO)CCN1C(c1n[nH]cc1CNC(=O)Cn1ncnn1)=O c1(C(=O)NCC2CC(COC)CN2C(=O)COC(C)=O)cc(=O)n(C)cn1 c1(C(N2CCN(C(c3cn(C)c(O)n3)=O)C3C2C3)=O)cc2ccc(Cl)c(F)c2[nH]1 c1(N(c2c(F)cnc(NC3CCCCNC3)n2)CC)ccc(O)c2ncccc12 c1(C(=O)NC(CNC(CC(C=C)C)=O)CC)ccc(C)nc1C(C)C c1(C(=O)NC(C)C(=O)NCc2ccc(N)cc2)c(Cl)cccc1Cl N1(C(c2cc(C(=O)NC)no2)=O)CC2CCC1C2NC(COCC)=O N1(C(=O)CCCCC(F)F)CCC2(CCN(C(=O)C(C3CC(F)(F)C3)O)C2)C1 C1(CN(C)CC2(NC(=O)Cc3coc(C(F)F)n3)CC2)CC(O)C(O)C1 c1(NC(C(CC)NC(=O)CCC2CCN(C(C)=O)C2)=O)cnc(F)nc1 Cc1c(C(=O)N(CCO)CCNC(C23CCN(CC2)C3)=O)ccc(C(F)(F)F)c1F C#Cc1ccc(C(=O)NCC2(F)CC(NC(c3ccncc3OC)=O)C2)nc1 N1(c2c(C)n(C3Cc4ccccc4CO3)nn2)CC2C3CCC(C3)C2(C)C1 C12(C(=O)NC3C(NC(C4(c5ccncc5)CC4)=O)C3)CC3CCC(CC(C3)C1)C2 C1(C(=O)NCC2(C)CCN(C(c3ccc(SC)o3)=O)C2)OC2CCC1CC2 N1(C(C(=O)NCCCOCCC2CC2)C2C(C)C2)CCCC(C(N)=O)C1 C1(C(N2CC(C(N)=O)(CNC(c3c(C)c(N)ccc3)=O)C2)=O)CCCCC(C)(C)C1 C(=O)(C1CC(C)(C)C1)N1CC(OC2C=CC(C(NOC(CC)(C)C)=O)C2)C1 CCCC(C)(C)CC(=O)N1CCC=CC1C(=O)NC(C12CCC(CO1)C2)C CCCC(CC)CC(=O)NCc1cc(C2CCN(C(C3CC3CF)=O)CC2)no1 N(C1c2ccccc2CC1O)C(C1CC(O)CN1Cc1ccncc1O)=O CC1CCC(NC(c2cnn3ccsc23)=O)CN1C(=O)CC12CCCC1C2 c1(CNC(=O)NCC(=O)NCCN(C(C2CCC(=C)C2)=O)C)cccc(C)c1 c1(C(=O)NC(CC)CC(=O)NC2COC(C)(C)C2)ccc(O)nc1C C(=O)(C1CCOc2ccccc21)NCC1C(NC(CCCN=[N+]=[N-])=O)CCC1 C(CNC(=O)CSC)(CC)(CC)NC(C(CC)OC)=O.c1(CC=CC=O)ccccc1 CCCCC(=O)NCC1(O)CC(C(=O)NOC2CCOC2)C1 c1(C(=O)NCC2(F)CCCN(C(CCCSC)=O)C2)cc2c(Cl)cc(F)cc2[nH]1 C(=O)(NNC(=O)c1ccc(C)s1)N(CCCOCC)Cc1ccccc1 C1(NC(c2cncc(Cl)c2)=O)COC2(C1)CN(C(c1cn3cccnc3n1)=O)C2 CCC(C)(C(=O)NC(C1CCN(C(c2ccc(CO)cn2)=O)CC1)C)OC C(C(=O)NC(c1cnc[nH]1)C)(C(C)(C)C)NC(c1c(C)cc(F)s1)=O N1(C(c2c(OC)ccs2)=O)CCCC2CN(C(c3cnc(C)cn3)=O)CC12 N1(C(c2c(CC)ncs2)=O)CCC(C(F)(F)F)C(CNC(C2(C#N)CCOC2)=O)C1 O=C(CC1COc2cc(O)ccc21)N1CCC(N(C(=O)CCC2CC2)CCO)C1 C(C(CNC(C1CC12CCC2)=O)S(C)(=O)=O)NC(C=C(C)C)=O C(=O)(C1CCCc2ncccc21)N1CCCC(NC(c2ccc(=N)[nH]c2)=O)C1 C(=O)(CC(C)CNC(=O)CN1CCN(C(=O)Cc2nocc2C)CC1)NC Cc1ncc(CCC(=O)NCC(=O)N(CC(=O)N(C2(C3CC3)CC2)C)C)o1 c1(OC)ncc(C(N2CC(O)(CN(C)C(c3ccnn3C3CCC3)=O)C2)=O)cn1 C(=O)(CCCC(C)(C)CC)NC(CCCC)CNC(c1cc(Br)no1)=O C1(NC(c2cnc(C)n2C)=O)CCC(C)N(C(c2cc(C(C)C)ccc2O)=O)C1 N1(C(C2C(C)CC(C)O2)=O)C2CCC1CN(C(c1cccc(C(N)=O)c1)=O)C2 C(=O)(CC1CCCNc2ccccc21)N1CC=CCC(C)(C)C1.c12ccc(cc1)o2 c1(C(=O)NCCCN(C(C(C=CC)O)=O)Cc2ccccc2)ccncc1O N1(C(C(C)OCCOC)=O)C(C(=O)N(C2(CC(=O)OC)CC2)C)CCC1C1CC1 C1(NC(Cc2ccc(C)s2)=O)CCCN(C(c2cn(C(F)F)nc2C(F)F)=O)CC1 N1(C(CC(C=C)(C)C)=O)CCCC2(CCCN2C(C2CCCOC2C)=O)C1 c1(C(N2CC(C(N(C)CC3(C)CCCO3)=O)C3(C2)CC3)=O)ccc2cncn2c1 c1(CNC(c2c(-c3c(C)ccnc3F)cncc2)=O)cccc2ccnn12 n1(CCNC(C2(CCC=C)CN(C(=O)CCC3CCCOC3)C2)=O)nc(C)nc1C C1(COC)CN(C(c2ccc(Cl)nc2N)=O)CCN1C(C1CNC(=O)N1)=O CC(C)C(F)(F)CC(=O)N1CC2CCC1C2NC(=O)C=CCN1CCCC1 N1(C(C2(OC)CCOC2)=O)CCC(CNC(C2(C)CNC(=O)C2)=O)C(F)(F)CC1 C1(C(=O)NCCN(C(c2c(C)csn2)=O)CC2CC2)CC2CCC2C1 CCC(C)CC(=O)NCC(C1CCN(C(=O)C(C)CC2CCCCC2)CC1)C n1(C(C=CC(=O)OCC)C)cc(CCC2CCOCC2)nn1 CC(C)C(C)CC(=O)N1CCCN(C(C2CCN(C)CC2)=O)CC1 C1(C(=O)NCC(C)CO)CCCCN1C(=O)CN(C)C(=O)Nc1ccccc1 CN1CCN(C(c2coc(CO)c2)=O)C(CNC(C2CCSC2)=O)C1 c1(C(N2CCC(NC(c3nc(C)c(C)s3)=O)CC2)=O)cnc2n1CCS2 C1(CNC(C2(C=C)CC2)=O)C(C2CC2)CCN1C(=O)Cn1cnc(=N)[nH]1 CC(C)CC(=O)C(=O)NC1CCN(C(C2CC2C(C)O)=O)CC1 C1(CNC(=O)C=CCOc2ncccn2)CC12CCN(C(C1CCCO1)=O)CC2 c1(C(N2CCN(CCO)CC2)C(=O)NCCC)ccc2ccc(Br)cc2c1 C(S(=O)(=O)C(F)F)CC1C(C(N(CC)Cc2csc(-c3occc3C)n2)=O)C1 n1(CCCC)ncc(C(=O)NCC2CCN2C(=O)CC(C)O)c1CC C1(C(=O)NC2CC=C(C)CC2)CC2(CC(NC(C3(Cl)CC3)=O)C2)C1 C(C)(CNC(=O)C(CC1CC1)N(C)C)(CC(C)C)NC(C(=Cc1ccco1)C)=O CC(CCCc1ccccc1)C(=O)N1CC(NC(C2(O)CC2)=O)C(C(F)(F)F)C1 C=C=CCC(=O)N1CCC(N(C(=O)CCCNC(c2sccc2C)=O)C)C1 c1(C(=O)OC)ccc(CO)c(OC)c1.N12CCCC(C1)C1(CC1)C2=O C1(CNC(C(C(C)C)NC)=O)CN(C(=O)CSCc2ccccc2)C(C)(C)C1 CCC(C)(C#N)C(=O)NC(CNC(c1cc(O)cc(F)c1)=O)C(C)C N1(C(C2(CC)COC2)=O)CCC2(CC1)CN(C(=O)CC1CCCN1CC)CCO2 c1(C(C)C(=O)N(CC(C)CNC(=O)CN(C)C(=O)C2CC2)C)cnn(C)c1 CCCCCC(O)CC(=O)NCC1CN(C(c2cccc(O)c2[N+](=O)[O-])=O)C1 CC(=O)CC(C)C(=O)NCC1CCCN(c2cc(C#N)ncn2)CC1 C(c1cn(C)nn1)=CC(=O)NCC1(NC(Cc2c(C)ocn2)=O)CC1 C1(CNC(CCCSCC)=O)CCCN(C(c2ccc(CC)s2)=O)C1 N#CC1CCCC(C(=O)NCCCCCCNC(c2ccc(CCF)cc2)=O)C1 C12(C(=O)NCC3CN(C(C4CCC(C)(F)C4)=O)C3)CC3CC(C)(C1)CC(C)(C3)C2 C(CC(F)F)(C(=O)NCC1CCC(=O)N1)NC(c1ncc(N)nc1)=O C1(C)(NC(C(C)CNC(=O)CO)=O)CCCN(C(=O)COC)C1.c1(OC)ccccc1 C1(CNC(C(CCC2CCC2)OC)=O)CN(C(c2csc(CO)n2)=O)CC1(F)F c1(NC2(c3n(CCC4(C)CC4)nnn3)CCCC2)nnc2ccccn12 S(=O)(=O)(c1c(Br)cc(F)c(Cl)c1F)NCc1cc2ccc(C)cc2cc1 c1(NC(C2(C(F)F)CCN(CC(=C)Cl)C2)=O)cccc(OC)c1 N1(C(c2n[nH]c(C)c2C)=O)CCC(C2CC2)C1CNC(C1CCC(C)CC1)=O C1(NC(CC2CC(C)C2)=O)CCCC2CN(C(=O)C=Cc3ccc(Cl)cc3)CC12 O=C(N=c1c(Cl)c[nH]cc1Br)C1(c2ccccc2)CCN(Cc2ccnc(Br)c2)C1 C(=O)(C1CC2(CCN(C(C3(C#N)CC34CCC4)=O)C2)Oc2ccccc21)NC c1(C(=O)NCC(CC)(CC)NC(c2nn[nH]c2Cl)=O)cc(O)nc(N(C)C)n1 c1(CC(N2C(C(=O)O)COC(C(F)(F)F)C2)=O)cccc2ccncc12 C1(C(=O)NCCOCC(=O)NC)C(C)OCCN1C(C1CC2(C1)CC21CC1)=O C(=O)(C(=O)C(C)(C)CC)NCc1cc(C(N2C(CC)C(C)(C)C2)=O)sc1 N1(C(=O)NC(c2cccc3ccccc23)CCC)Cc2ccccc2CCC1C N1(C(c2n(CCC)nc(C)c2)=O)CCC2(CCCN2C(c2cccc(=O)o2)=O)C1 c1(Cn2ncc(C)c2)nccc(=NCCC(C)N(C)Cc2ccccc2)[nH]1 C1(C(C(=O)NCCCCNC(=O)C(C)c2ccco2)OCC)CC(F)(F)C1 C1(C(=O)NCCCN(CCCNC(c2c[nH]nc2C(F)(F)F)=O)C)CNC(=O)N1 N1(C(CN2CCCC2)=O)CCc2ccccc21.CC1CCCN1C(=O)NC.C1C(=O)N1C c1(C(N2C(C)C(C)C2)=O)cc2oc(Br)cc2[nH]1 c1(C(N(CCN(C(=O)Cc2cccc(C(F)F)c2)C)C)=O)c[nH]c2cnc(Cl)cc12 c1(C(=O)OCC)cccc(C(=O)NC2(CF)CCN(C(=O)CCSC(C)C)C2)c1 CCCC(C(=O)NCCCCCCNC(c1ccc(N(C)C)nn1)=O)C(C)C C1(O)(C(=O)OC)CCN(C(C2C(C(=O)NCc3cnnn3C)CC=CC2)=O)CC1 c1(CCC)sc(C(N2CC(CNC(c3occc3F)=O)C2)=O)cc1CC c1(CC(C)C(=O)NCC2CN(C(=O)C(O)c3ccsc3)C2)cccc(Br)c1 c1(C(=O)NCC(CNC(C2C3CC(=O)CC32)=O)O)cnn2c1OCC2 CC(C)CC(CNC(C1CC1C)=O)NC(C1(Sc2ccccc2)CCOCC1)=O C(=O)(C(F)(F)C1=CCOCC1)N1CCC(NC(C(CCC)OC)=O)C(CC)C1 C(C(C(C)C)C(C)C)NC(N1CCCC(n2c(C)ncc2)C1)=O C12(CNC(C3(CC=C)CC=CC3)=O)CCC1CN(C(c1cnc(C)c(Cl)c1)=O)C2 CCCC(O)CC(=O)NCC1CCCCCN1C(c1cnn(C(C)C)c1N)=O c1(C(N2CC(NC(c3c(C)cnnc3)=O)C(O)C2)=O)ccc2c(c1)NC(=O)C2 C1(CC)(NC(c2c[nH]c(=NC)o2)=O)CCN(C(=O)CC(C)COC)CC1 C(C1OCCc2sccc21)N(C)C(C1CCCCN1CC(F)(F)F)=O N1(C(C(CO)N(C)C)=O)CC(CNC(C2CC(=O)CCO2)=O)C(C)(C)C1 CC(C)C(CCNC(C1CC(C)(F)C1)=O)NC(=O)Cc1nc(=N)[nH]s1 Cc1cc(C)c(S(=O)(=O)Nc2ncc(CC(=O)Nc3ncco3)s2)c(C)c1 C1(CNC(CN(CC(C)(C)C)C)=O)(NC(=O)CC2OC(=O)N2C)CCCCC1 c1(CC(=O)NC2CC(CNC(C(C(C)C)NC=O)=O)C2)cccc2c1OCCO2 N1(C(c2cc(C)oc2)=O)CCCC2(CCCN2C(C23CC4CC2C3C4(F)F)=O)C1 CCCCC(CC)N=c1nc2ncn(C)c2c(NCC2Cc3ccccc3CO2)[nH]1 c1(C(N2CC(CC)C(NC(c3scnc3C)=O)CC2)=O)cc2cnn(C)c2s1 C(=O)(CCCC1CCC1)N(C(CCNC(C1(OC(C)=O)CC1)=O)C)C Cc1ccc(Cl)c(C(=O)N(C2CCCCN(C(=O)C#CC3(C)CC3)C2)C)c1 N1(C(C(c2cccc(C)n2)(F)F)=O)CCCCC(CNC(=O)CCC(F)F)CC1 C1(C(=O)NCCCN(C(C)=O)C)CN(C(c2ccc(OC)nc2)=O)CC1C(C)C N1(C(Cc2cc(C)nn2C)=O)CC2CCC1C1CN(C(=O)C=CBr)CC21 N1(C(C(=O)NC)=O)CCCCC(NC(=O)C(=O)Nc2cc(Cl)ccc2OCC)C1 C(c1ccc(F)cc1F)=CC(=O)NC(C)CCCNC(c1ccn(C(F)F)n1)=O c1(C(=O)OC)cn(C)[nH]c1=NC(=O)NC(c1nc(C2CC2)no1)C C1(C(=O)NCC(C)CN(C(=O)Cc2csc(SC(F)(F)F)n2)C)CCCCS1 c1(CNC(c2cnn(C)c2F)c2n(CC)nnn2)cc2ncccc2s1 C=CCC(C(=O)OC)NC(=O)C(O)C1CN(C(=O)C(C)OC)C1 N1(C(C(C)C)=O)CCC2(C(=O)O)CC2C1.c1(CC2CC2)cc(Cl)c(N)cn1 c1(-n2cc(CN3CC(Br)=C(C)CC3CO)nn2)cnc2c(CC)c1CCOCC2 c1(CNC(CN(CC(C)(C)C)C)=O)ccc(Cl)c2c1OCCO2 C1(NC(COCCC(C)C)=O)CCCC12CCN(C(=O)C=CS(C)(=O)=O)CC2 c1(OC)ccc(C(c2nnnn2C2CCC2)NC23CC(F)(C2)C3)cn1 C1(C(=O)NCC(C2CCCC2)C)CCC2CCC1N2C(c1cc[nH]n1)=O C1(NC(c2cnc(C3CC3)o2)=O)COCCN(C(C23CCCCC2C3)=O)C1 C1(NC(C2CC(n3cc(CCc4nn[nH]n4)nn3)C2)=O)CC2CC3CC(C2)CC1C3 c1(N2C(C(=O)Nc3ccc(C)nc3I)C=CC2)nc(C)c2cc(Br)ccc2n1 Cc1ccc(C(N2CCC2CC(=O)Nc2c[nH]ccc2=O)=O)nc1 C(=O)(C1=CCC(C)CC1)NC(c1ccnn1C)C(N1CC2CC(C)C2C1)=O C=C(C)C(CC(=O)NC1CCCC(NC(=O)C=C2CCCCC2(C)C)C1)OCC C(=O)(C1OCCc2ccccc21)NCC(C)NC(C1CC2CC1OC(=O)N2)=O C(=O)(C(C)CCOC)NC(C(CO)NC(c1c(CC)ncs1)=O)C c1(C(=O)NCCCNC(C2(C)CCC(=O)C2)=O)ncc2ccccn12 C1(CC=C)(NC(=O)C(C)OC)CCCN(C(=O)CC2(O)CCOCC2)C1 C(=O)(C(O)(C(C)C)C(F)(F)F)N1CCC(NC(c2sc(C)c(O)n2)=O)C(C)(C)C1 C1(CONC(C(c2cnn(C)c2)NC(CCCCC#C)=O)=O)CCC(=O)N(C)C1 C#CC1CC2CCC1N(C(c1cc(COC)on1)C(=O)NC1CCCC1)C2 N1(C(c2c(F)ccc(C#C)c2)=O)CC2CCN(C(C3CC(C)OC3=O)=O)C2C1 NC1c2ccccc2CC1C(=O)NCc1cnn(-c2ncc(Br)cn2)c1 C=Cn1nccc1C(=O)NCC(F)CNC(=O)C=Cc1ccc(Br)s1 C1(C)(CC)CCCN(C(=O)CC=CCNC(=O)Cc2nccn2C)C1 c1(OC)cc(C(=O)NC2CCN(C(C3(C4CCC4)CC3)=O)C(C)C2)c(F)c(Cl)c1 C1(CC=C)(CNC(=O)C(N2CCC(CC(N)=O)C2)=O)CCS(=O)(=O)CC1 c1(C(N2CCC(NC(=O)CC3CC4(CC4)C3)C2)=O)cc2cccn2c(O)n1 C1(=O)CC(CC(C)C)CN1.c1(C(C(C)C)NC(=O)OCC)ccc(Cl)cc1 CC(C)C(O)C(C)C(=O)N1CCCC(C)(C)C1C(=O)NCC(Cl)=CCl N1(C(C2COCC(C)O2)=O)CCC(F)(C(=O)NOCCc2ccccc2)CC1 CC(CCCc1ccccc1)C(=O)NC1CN(C(c2cn(C)nc2O)=O)C1 n1(CCOC)nnc(C(=O)NCCNC(=O)C(c2cnn(C)c2)O)c1C(F)(F)F C1(CNC(CCc2cnn(C)n2)=O)CCN(C(c2ccnc(Cl)n2)=O)CC1(F)F N1(C(=O)Cc2cccc(OCF)c2)CC(C2CN(C(C3CC3C3CCCCO3)=O)C2)C1 c1(C(=O)NCC2(NC(c3csc(Cl)n3)=O)CCC2)coc2ccccc12 CCC(CC)C(F)C(=O)NCCC1CC(NC(=O)C(c2ccccc2F)C)C1 c1(C(N(C2CCCN(C(c3cn(C)[nH]c3=N)=O)C2)C)=O)cc(Cl)cc2c1CCC2 C1(NC(=O)CC2COCC2O)CCOCC1NC(c1cscc1Cl)=O CC1=C(C(=O)N2CCCC(CCC(=O)NC3CCN(C)CC3C)C2)SCCO1 CC(C)C(C)C(CNC(c1nnc(O)nc1O)=O)NC(c1cn2c(n1)SCC2)=O CCN=c1ccc(C(N2CC(NC(=O)C=Cc3nccs3)CC(O)C2)=O)c[nH]1 C(=O)(CCCC(=O)NCCCOCCNC(=O)CN1CCCCCC1=O)NC c1(CC)ccc(F)c(C(=O)NC2CC(C)CN(C(=O)CC3(CO)CC3)C2)c1F c1(OC)cc(O)ncc1C(=O)NC1CCN(C(c2csc(F)c2)=O)C1C N1(C(C(C)OC(C)=O)=O)CCOCC(NC(c2cccc(O)c2Cl)=O)C1 c1(CC(=O)NCC(CNC(c2ccc(OC)c(O)c2)=O)O)ccn2cncc2c1 N1(C(c2cc(C(C)C)on2)=O)CCC2(C1)CN(C(c1cnncc1O)=O)CCO2 C1(CNC(CNS(N)(=O)=O)=O)CCCOC1C1CCN(C(=O)CC2CSC2)CC1 N1(c2c(OC)cncn2)CC2CC(NC(=O)CCC(N)=O)CC2C1 c1(CC(=O)N(CC(C)NC(C2CC2(C)C(=O)OC)=O)CC)ccc(OC)cn1 C1(NC(c2c(CC)noc2)=O)CCC12CN(C(c1ccc(C3CCC3)nc1)=O)C2 n1(CC)ncc(C(N2CCCC(CN(C(=O)C(c3cncnc3)C)C)C2)=O)c1Cl CC1CCC(C(=O)NCC2(F)CN(C(=O)CNC(C3CCC3)=O)C2)O1 CC(C)(C)CC(O)C(=O)NC1CCC1CC(N1CCCC(O)(CO)C1)=O CCC(CC)C(C(=O)N1CCSCC1C(=O)NC1CCn2ccnc2C1)OC C1(C(=O)NC2CC(CNC(C(CCSC)NC=O)=O)C2)CCc2nncn2CC1 c1(OC)cc(O)ncc1C(N1CCC(CNC(C2COCCN2C)=O)(OC)C1)=O C=CCC(CC)C(=O)NCCOC1CN(C(c2cc(C)c[nH]2)=O)C1 c1(OCC)cc(C(N2CC(N(C(=O)Cn3c(C)ccc3C)C)C(O)C2)=O)ccn1 c1(C(=O)NCC2CN(C(CC(C=C)C)=O)CC23CC3)occ2c1CCOC2 CCC(CCCC(=O)N(CC(C)(F)F)C)NC(c1cc(CO)n(C)n1)=O CC1(C)OC(C)(C)C1C(N1CC2C(C1)N2C(c1cc2n(n1)CCO2)=O)=O c1(SCC)ccc(Cl)cc1C(=O)NCCCNC(c1cc(C#N)no1)=O C1(NC(=O)NCCN(C)C(=O)OC(C)(C)C)C2CCC1(C)C2(C)C C1(F)(C(=O)NCC(C)(C2CC2)NC(c2csc(=N)[nH]2)=O)CCC(F)(F)CC1 C1(C)(C(=O)Nc2cccc(NC(C#CC(C)(C)C)=O)c2)CCCNS1(=O)=O C1(C(C)NC(=O)CCN2CCOC2=O)CCCN(C(c2cnoc2C(C)C)=O)C1 Cc1ccc(Br)c(CN(C(=O)CCC2CCC(=O)NC2)C)c1 C(=O)(CC(=O)N1CCCC1C(C)(C)NC(C1CNC(=O)N1)=O)NC c1(C(=O)NCCCCCNC(CSC(C)C)=O)ccc(C2CCCO2)cc1 C(=O)(CCCC(C)(C)C#N)NC1(CCC(=O)NCCCCC=C)CCCC1 c1(C(N2CC3(C(NC(C(C)OC)=O)CCC3)C2)=O)cc2cc(C)ccc2nc1C CCC(O)(CC)CCNC(=O)NC1(C(=O)OCC)CSC(C(=O)O)C1 C1(C(N(CC(CN(C(CCNC(=O)OCC)=O)C)O)C)=O)CCCC(C)CC1 c12ccc([N+](=O)[O-])cc1N2.N1(C(C2CCC(C(N)=O)S2)=O)CCC(F)(F)C(CO)C1 C1(NC(C2CCCCC2(F)F)=O)CC2CCC(C1)N2S(=O)(=O)c1cccs1 N1(C(c2c(N)cncc2)=O)CCN(C(c2n[nH]cc2F)=O)C(c2ccncc2)C1 N1(C(c2cncc(C)c2)=O)CCC2CCC(NC(c3ccc(F)cc3Cl)=O)C12 C12(CC(=O)NC3CN(c4n(C)nnn4)CC3(C)C)CC3CC(CC(C3)C1)C2 C1(NC(C(c2ccc(C)o2)C)=O)CC1C1CCCN(C(C2CC3(C2)CC3F)=O)C1 c1(C(CNC(CC2(C#N)CC2)=O)NC(C2CC2(F)F)=O)cc(F)cc(Cl)c1 S(=O)(=O)(c1ccc(F)cc1Cl)NC1CCC(NC(c2ccc(C)c(Br)c2)=O)C1 c1(C(=O)NCCC(C)N(C(=O)C(C)C#N)C)cccc2scnc12 Cc1c(CC(=O)NOCCCCC(=O)NCC(CC2CC2)CO)cnn1C C(=O)(CC(C)P(C)(C)=O)N.C(=O)(C(C(C)C1CCCCC1)N(C1CCOC1)CCF)OC Cc1ncc(C#N)c(N2CCC(CNC(c3coc(C)n3)=O)C2)n1 Cc1ccc(C)c2sc(COC(=O)C(C)Cc3cnn(C)c3)nc12 c1(CN(C(=O)NCC2(C(=O)OC)CCCC2)C)ccc(O)c(OC(F)(F)F)c1 c1(C(=O)NCC2CCN(C(C(C)OCCCCCC)=O)C2)c(Cl)ccc(F)c1C N1(C(C(C#C)(C)C)=O)CC2(C1)OC1(C)CC2(NC(c2ccn3c2CCCC3)=O)C1 c1(C(=O)NC(C)(CNC(=O)CCc2cnc(O)[nH]2)CO)cnc2[nH]cnc2c1 Cc1cc(C(=O)NC2(CCCNC(C3CCC4(CC4)C3)=O)CC2)c2c(c1)CCO2 C#CCC(CC)NC(=O)C(C1(O)CN(C(=O)C(C)n2ccnn2)C1)F c1(C(=O)NC(CCNC(C(CC)F)=O)C(C)C)ccc2nc(N(C)C)sc2c1 C(=O)(CC(C)C(=O)NCCCCC(N1CC(=O)NCC1C(C)C)=O)OC Cc1cn(CC(=O)NC2CCC2NC(C2CCc3nncn3C2)=O)c(=O)nc1O C1(NC(c2cnc(C(=O)OC)c(C)n2)=O)CN(C(=O)CN)CC1C1CC1 CC1CCC(C2CCC2)CN1C(=O)C(=O)Nc1ccc(S(C)(=O)=O)cc1 C1(CNC(C(C)C2CC2)=O)CCN(C(=O)C=Cc2cccc(F)c2)C12CCC2 C1(C(=O)N(C2CCN(CC(C)(C)C)C2)CCO)CC2(CCO1)CC(F)(F)C2 N1(C(CC(=C)C)=O)CCC(c2ccccc2)C(NC(C2(CO)CCCO2)=O)C1 N1(C(C2(CC#C)CC2)=O)CCC(C)N(C(C2CCCN2C2CC2)=O)CC1 c1(OC)cccc2c1OCC(C(=O)NCCCCCNC(=O)CC(C)OC)C2 C1(CC#C)CCNCC1.c1(OCCN(C=O)C)ccccc1C(C)C c1(C(=O)NC(C(C)(C)NC(C(Cc2c(C)nc[nH]2)O)=O)C)cnn(C(C)C)c1C N1(C(C(c2ccc(Cl)s2)C)=O)CCN(CC2CN(C(C3CC3(F)F)=O)C2)CC1 CCS(=O)c1ccccc1C(=O)NCC1CC(F)CN1C(=O)CN1CC2CC2C1 c1(C(N2CCCC(F)(CNC(C(CC)OC)=O)C2)=O)cc2cc(F)ccc2cn1 C1(C)(C(=O)NCCC(CNC(c2sc(F)cc2C)=O)OC)CCC(=O)NC1 C(CCCCCN(C(=O)Cn1nccn1)C)NC(C1CC(OC)C1)=O c1(C(=O)NC(C2(O)CCN(C(c3nccn3C)=O)C2)C)cc(Cl)cc(Cl)c1 CC(Cc1cccs1)N=c1[nH]c(=N)[nH]c(=NC2CCCN(S(=O)(=O)N(C)C)C2)[nH]1 C1(C(=O)NC2CC(N(C)C)C2)CN(C(C2CCS2(=O)=O)=O)CC1(C)C N1(C(C(C(C)O)C)=O)CC2CC(NC(c3cc4n(n3)CCO4)=O)C2C1 CC#CCCC(=O)N(CC(=O)N(C)CC1CCCS1)C(C)C Cc1[nH]c2c(C(N3CCN(c4cc(C#N)ncn4)CC3)=O)cccc2c1C N1(C(C(C)OCCOCC)=O)CC2(CC(NC(=O)Cc3coc(C)n3)C2)C1 CC(O)CC(C)(C)CNC(c1ccc(CNC(C2CC(CF)C2)=O)s1)=O C1(O)(CNC(COCCOC)=O)CCN(C(=O)Cn2cccc(N)c2=O)CC1 C(=O)(CCS(C)=O)N(C1CCN(C(=O)Cn2ncn(C)c2=O)C1)CC(C)C Cc1coc(C(=O)NC(C)CCN(C(=O)CSCc2ccccn2)C)c1C N1(C(C2C(C)(C)CO2)=O)CC2OCCN(C(c3cc4cccc(F)c4o3)=O)C2C1 Cc1cc(C(N2CC(NC(c3cnnn3C)=O)CC(C)C2)=O)c(F)cc1Cl c1(C(N2CCCC(C)(CNC(C(C(COC)C)C)=O)C2)=O)cncc([N+](=O)[O-])c1 c1(OC)ccccc1NC(C1CN(C(C)=O)CC1C)=O N1(C(c2cc(C)nc(O)c2)=O)CC2(CCN(C(c3ccoc3Br)=O)CC2)C1 N1(C(CCNC(=O)CO)=O)CC=CC1C(=O)NCC1(F)CCC1 C12(NC(CCCCOC)=O)CCN(C(=O)C(=Cc3cscn3)F)CC1C2 c1(C(=O)NCC(C2CCC2)OCC)cc(CNC(C2CC(C)CO2)=O)nn1C N1(C(C=CCN(C)C)=O)CCC(CF)(NC(C2(C)CC2(Cl)Cl)=O)C1 CC1=NOC2(C1)CC(C(=O)NC1CCN(C(C3CCC(=O)O3)=O)C1C)C2 C1(NC(c2c(N)n(-c3ccccc3)nc2)=O)CS(=O)(=O)CC1NC(C1(F)CC1)=O c1(COC)nc(NCc2nccs2)cc(N(C)Cc2ccoc2C)n1 c1(CCC(=O)N(C(CNC(C2CCCC2)=O)C2CC2)C)cc(F)ccc1F C(CC(C)(c1nnnn1C)NC)SC.C1(OC)CCOC1.C1CS1 C1(F)(CNC(C(n2ccc(C3CC3)n2)C)=O)CC(CNC(=O)Cn2ncnn2)C1 C#Cc1cc(C(=O)N(C2CCN(C(=O)C=COCC)C2)C)ccc1C Cc1ccc(Cl)cc1C(=O)NC1CCCC1CNC(c1sccc1C(F)F)=O C1C(C(F)(F)F)CC(=O)N1.Cn1cc(S(=O)(=O)N2CCOCC2)c(-c2ccccc2)n1 C(=O)(C(C)(COC)CC)N(CC(C)NC(c1cnc(OC(C)C)c(Cl)c1)=O)CC C1(NC(C2(CC(C)=O)CC2)=O)CCC(C(=O)Nc2cncnc2O)CC1 C1(OC)CC(CNC(C2CC(F)C(=O)N2)=O)N(C(c2cnns2)=O)C1 C1(NC(CC(=O)NCC2CCCO2)=O)CC(=O)N(C2CN(CCOCF)C2)C1 C(=O)(C#CC1CCN(C(=O)NC(c2c(C(=O)OC)occ2)C)CC1)OC(C)(C)C C1(C(N2C(C3CCN(C(CC(CC)O)=O)CC3)CCC2)=O)CCC(=O)N(CC)C1 C1(C(=O)NC(CN(C(COCC)=O)C)CC)CCC2(CC1)OCCO2 CS(=O)(=O)C1CCCCN(N2CCC(N=c3cc[nH]c4ccccc34)C2)C1 c1(N2CCCCC(SC)C2)nc(NC2CC3CCC2O3)c2ncn(C)c2n1 N1(C(C2CCCN2C(=O)Sc2ccccc2)=O)CCC(O)C1C(F)(F)F C1(N(C(=O)CCOC2CCC2)CC)CCCN(C(=O)CNS(=O)(=O)N(C)C)C1 C1(N(C(CSCCOC)=O)CCO)CCN(C(C2(C)CC=CC2)=O)C1 N1(C(CCC=CC)=O)CCCc2cc(CNC(=O)CCCC(F)(F)F)ccc21 c1(C2(C(=O)NC(C3CN(C(=O)CC4CSC4)CCO3)C)CC2)c(Cl)cccc1Cl C1(C)(C(=O)NCC(C)N(C(=O)COCC(=O)NC2CC2)C)CCC(=O)C1 c1(OCC(=O)OCC2C(C)CCC2)ccc(CO)cc1 C1(CC)C(NC(C2C3CC4C(C3)C24)=O)CCN1C(=O)C(c1ccc(F)cc1)CO c1(CC=C)cccc(C(=O)NCCn2c(C)csc2=O)c1.C12CC1C(=O)NC2 c1(CCC(=O)NC2CC(C(=O)NC(C)C(N)=O)C2)ccccc1Cl C=C(CNC(C1CCCN1C(=O)C1CC1)=O)CCNC(C1(n2cccn2)CC1)=O c1(COC2CCN(C)CC2)cnn2c1CN(C(=O)C(Cl)=CCl)CC2 C1(C(=O)NC(C)(C)CNC(=O)CCC(=O)c2ccncc2)CCCCC1(C)C CCC(Cl)(Cl)C(=O)NCC(C)(C)CN(C(=O)C(C)OCC(F)(F)F)C c1(CC(=O)N(C2CCC2)CCC)c(C)ncnc1C N1(C(c2cccc(OCOC)c2)=O)CCOCC(NC(C2CC2F)=O)C1 C1(NC(C(C)SC(C)C)=O)CCC(C)N(C(=O)CCOCC(F)(F)C(F)F)C1 C(=O)(C(CO)C(F)(F)F)N1C(C2CN(C(c3cc(COC)no3)=O)C2)CCCC1 N1(C(c2c(C)c[nH]n2)=O)CCS(=O)(=O)C(CCNC(=O)CCOCCC2CC2)C1 Cc1cc(C(=O)NCC2(F)CCCN(C(c3cnc[nH]c3=N)=O)C2)nc(O)n1 Cc1c(F)ccc(C(=O)NC2CC(CC(=O)Nc3cc(Br)cnc3O)C2)c1F c1(OC)cccc(C(N2CCC2CNC(=O)C(C)(C2CC2)NC(C)=O)=O)c1N C(=O)(CC(O)CC(C)C)N1C(C(N2C(COC)CC2)=O)(CO)C1 C1(CC(C)NC(c2coc3c2C(O)CCC3)=O)C2C3CC4C1C1C2CC3C41 C(=O)(C1CCCc2nn[nH]c21)NCCCNC(c1cnn2ccn(C)c21)=O C1(O)(C(N(C(c2ccccc2)CC)C2CC2)=O)CCN(C(=O)CCN2CCCC2)C1 N1(C(Cc2nc(=N)[nH][nH]2)=O)CCC(NC(=O)CCOC2CCC2)C(F)C1 C(=O)(C(CC(C)(C)C)NC(=O)OC(C)(C)C)N1CC(N(OC)C)C1 C1(NC(N2CC(c3c(C)nccn3)C2)=O)CC2CC(N(C3CC3)C3CC3)C1C2 Cc1ccc2c(C(=O)NCC3CC4CCC3N4C(C3CCCOC3)=O)coc2c1 CC(CC(=O)NCCC1CN(C(c2n[nH]c3c2CC(C)CC3)=O)C1)CC(F)(F)F C(C(C)(C)CC(=O)NCC(N1CCN(C)CC1)(C)C)N(C)C(=O)OC(C)(C)C N1(C(C(C)N(C)C)=O)CCC2(CCCN2C(C2COC3COCC23)=O)CC1 C1(NC(c2cnc(S)[nH]2)=O)CCN(C(c2scnc2Cl)=O)CCC1CO C(C(N=[N+]=[N-])C(=O)NCC1(NC(C2CNC(=O)N2)=O)CC1)OCC CC(=O)C(C(C)C)NC(=O)C(C(C)C)NC(=O)OC(C)(C)C c1(C(=O)NC(CNC(=O)C(O)c2cnc[nH]2)CO)ccc2c(c1)NC(=O)CS2 Nc1cc(C(=O)NC2(C3CC3)CCN(C(C3CC34CCCC4)=O)C2)cc(Cl)n1 Cc1cc(C(O)C(=O)NCC2CC(F)CN2C(c2cc(Cl)cs2)=O)ccc1F C(C(CC(=O)NCCCN(C(=O)CCn1cncn1)C)C(F)F)N(C)C C(C(=O)NCC=CCNC(c1c(-n2ccnc2)cccc1F)=O)(C(C)(C)C)SC Cc1nc2ccccc2nc1N(C)C(C1COCCN1C(C1CC(O)CN1)=O)=O N1(C(c2ncc(CC)cn2)=O)CCCC2(CCCN2C(C2CCCC2)=O)C1 n1(CC(=O)NCC2CCC2C(=O)NCC23CCCC2C3)c(O)nnc1O [N-]=[N+]=NC1CCCCC1C(=O)N(C1CCN(C(=O)C=Cc2nccs2)CC1)CCO N1(C(=O)NCc2ccccc2)CCCC(CO)C1C1(OC)C(CCC)COC1 Cc1cnn(CC(=O)NCC(C(=O)N(C(C)CCO)C)N(C)C)c1 N1(C(CC(=C)C)=O)CCC(C2(NC(=O)C(C)CN(C)C)CC2)C1 C12(NC(Cc3cn(CC)nc3)=O)CCCC1(F)CN(C(C1(SC)CCC1)=O)C2 c1(OCCC(=O)NCC2CN(C(=O)C=CBr)CCO2)ccc(F)cc1F c1(OC)cc(NCc2c(-c3ccc(O)nc3C(C)C)ccnc2OC)ccc1I c1(OC)cc(Cl)c(I)cc1NC(C1(CCOC)CCCC1)=O c1(NC2CC(F)(COC)C2)ncnc(C)c1C#N.C12(CCSC1)C(=O)N2 CCC1=NOC(C(=O)NC2COCCC2C(=O)N(C)C(C)C)C1 CCCC(CC)C(=O)NC1CN(C(=O)CCn2cncn2)CC1C(F)F N1(C(C2C3(CC(NC(C(C)N(C(C)=O)C)=O)C3)C2)=O)CCCCC(F)(F)C1 Cc1cc(F)c(C(N2CCC(F)(C(=O)Nc3cccc(F)c3F)C2)=O)cc1F c1(C(N(CC(O)CN(C(=O)CSc2cncn2C)C)C)=O)cn2ccncc2n1 C=CCC(C)(C(=O)NC1CCC1NC(=O)CCCCCOC)N(C)C N12CC(=O)CCC1C(=O)NC(C)C2=O.Cc1nc(C2(NC(C)C)CC2)n[nH]1 c1(C(C)NC(CC2(CC)CC2)=O)c(C(=O)O)n(C)c2c(C)cccc12 C1(NC(CN2CCC(C)CC2)=O)CCC12CCN(C(C1CCS(=O)CC1)=O)CC2 CCCCC(O)C(=O)NC(c1ccc(C2CC2)o1)c1nnnn1CCC1(C)CC1 C(c1cncn1C)=CC(=O)N(C1CCN(C(C(C)NS(C)(=O)=O)=O)C1)C CCCCCC(F)C(=O)NCC(C)(C)C#CC(=O)NCCN(CCC)CCC n1(CC)ncc(Br)c1C(N1CC(OCCNC(C2(C#N)CC2(C)C)=O)C1)=O C1(N(CCC)C(c2ccccc2CC(C)C)=O)C2CN(Cc3cn[nH]c3)CC12 O=C(N=c1ccc(C2CC2)n[nH]1)NC1CC2COCC2C1 c1(C(=O)NC2COCCN(c3ncnc(CC)c3F)C2)ccc2nsnc2c1 Cc1cc(C(N2CC(NC(=O)Cc3cncs3)C(C)C2)=O)sc1-c1ccccc1 c1(NC(C)C(=O)NC2CC(CNC(=O)CCn3cccc3)C2)ccc(C#N)cc1 Cn1cc(C(=O)NCC23CC2CN(C(=O)COc2ccc(Cl)cc2)C3)ncc1=O N1(C(CCNC(=O)OCC)=O)CCC2(CNC(c3cnn[nH]3)=O)CCCCC12 c1(NC(C(c2cccnc2)NC(C2C(=C)C2)=O)=O)ccccc1C(N)=O C(=O)(CCCC(C)(C)C)N(CC(=O)NCC1CC1Cl)C CCCC(C)(C)C(=O)N(C(c1ccnn1C)C(N1CCCC2CC12)=O)CC c1(NC(C2CC(CF)C2)=O)ccc(OC(F)F)cc1.C1(C(=O)N)C=CCC1 c12ccccc1CNC2=O.C1(C)(C(=O)OC)C=CCN1C(=O)CCCF Cn1nc(C(=O)NC2CCCCC2CNC(=O)CSCC#N)c2c1CCCC2O C1(NC(COCC(=O)OC)=O)CCOCC1NC(=O)CCc1ccccc1C Cc1nc2cccc(C(=O)Nn3cc(CCN4CCCC4C(C)O)nn3)n2n1 C1(F)(c2cn(CC(=O)OCC)nn2)CCN(C(c2cnc(C3CC3)s2)=O)C1 c1(C(N(CCCCNC(CC(C=C)C)=O)C)=O)cnc2n1CCC(C)C2 c1(C(=O)NC2CC(C)(NC(C3CC34CC4)=O)C2)cnn2c1S(=O)(=O)NCC2 CC1CC(=O)NC1C(N1CCC(NC(c2cc(-c3ccns3)on2)=O)CC1)=O c1(N(C(=O)CC=CC2CCCN2C(=O)COCC(C)(C)C)C)ccc2[nH]ccc2c1 N1(C(C(C(C)(C)C)O)=O)CCC2CN(C(=O)CN3C(=O)CCC3=O)CC2CC1 c1(C(=O)NCC(C)NC(C2CC2c2cccnc2)=O)cc2c(nc1O)CCCC2 c1(C(N(C(C(=O)OCC)C)C)=O)cc([N+](=O)[O-])cc(C)n1 C(=O)(CC(C)C(F)(F)F)N1CCC(CCOC)(NC(C2CCC2C)=O)C1 N1(C(c2c(C#C)cnn2C)=O)CCCC(C2(NC(C3CC(C)(C)CO3)=O)CC2)C1 c1(C(=O)NCCC2CCCN(C(C(C3CC3)SC)=O)CC2)cnc2c(c1)COC2 Cc1cc(C)c(C(=O)NCC2CC3CCC2N(C(=O)CNC=O)C3)cc1N N1(C(C(CC=C)C)=O)CCCC(CO)(CNC(C2(CCCC)CCC2)=O)C1 C1(CC)CC(C(N2CC(NC(c3cccnc3S)=O)CC(C)C2)=O)CC(=O)N1 C1(CC)CCN(C(c2coc(CNC(c3scc(C)c3C)=O)n2)=O)C1C C1(NC(C(C)C2CC2)=O)CCCCN(C(c2scnc2C2CC2)=O)C1 N1(C(c2cc(C)oc2C)C(=O)NCc2cccc(Br)c2)CCOC(C)C1CO N1(CC(=O)NC(C2CCN(C(C(COC)C)=O)C2)(C)C)CCN(C)CC1 O=C1CCC(S(=O)(=O)Nc2ccsc2C(N2C3CCC2CC3)=O)CC1 N1(C(C(C(C)C)c2cnc(C)s2)=O)CCCC(NC(=O)COCC2CC2)CC1 O=C1CC(CNC(=O)C(Cc2cn[nH]c2)NC(=O)CN2CC(F)(F)C2)CN1 c1(CC)cc(C(=O)N(CC(O)CN(C)C(c2cncnc2)=O)C)cc(Cl)c1 Cn1nc2c(c1C(=O)NCC(O)CNC(C13CCC1C3)=O)CCCC2 C1(F)(C(=O)NCC(=O)N(C)C2CC2)CN(C(c2cc(C(N)=O)[nH]n2)=O)C1 c1(C(c2n(C(CC)C)nnn2)NCc2cn(C(C)C)nn2)ccc(Cl)c(F)c1 C1(C(N2CCC(NC(C(C)(C)OCC)=O)C(F)C2)=O)CC(c2cnn(C)c2)=NO1 C1(C(=O)NC(CNC(c2cccc(OC)n2)=O)CO)Cc2ccccc2C(=O)O1 C(=O)(C1=CC2(CCN(C(=O)CN3CCN(C)CC3)C2)C1)NC(CCCC)C C12CN(CCO1)C2=O.N1(C(C=CC(=O)N(C)CC2C3CCCC23)=O)CCOCC1 N1(C(c2n(CC)nnc2C)=O)CCCN(C(=O)CP(C)(C)=O)CC1C C1(C(=O)NC(C(C)NC(=O)CCNC(C2CCC2)=O)CO)CCC(C)(C)O1 CC(C(O)C(=O)NCCCOCCN(C(=O)CO)C)c1ccccc1F C1(CC(NOCCC)=O)CC(NC(=O)C(O)C2CC2)C1(C)C N1(C(C2CC(C(C)C)C2)=O)CCN(C(C2CN(C(N)=O)C2)=O)C(CC(F)F)C1 C1(CC(=O)N(CCN(C(=O)CC2CCCC2)CC)CC)CC(=O)NC1=O C(=O)(C1=CS(=O)CCC1)N1CC(CNC(c2occ(OC)c(=O)c2)=O)CC1(C)C S(=O)(=O)(c1ccc(N(CCCC2CCCC2)C)c(Cl)c1)NCC1C(C)C1(F)F CCC(Cc1ccccc1)C(=O)NCCNC(=O)COC(F)F C1(C(=O)NC(C(C)C)C)COCCN1C(C)C.C12(CCCO1)C(=O)NC2 N1(C(c2c(CC)non2)=O)CCC(F)(CNC(c2cnc(O)o2)=O)C1 C1(CC(N2C(CNC(C=CC(=O)OCC)=O)CCC2)=O)CCCC12CC2 Cc1nc(C)n(C2CCC2)n1.c12cn(-c3ccccc3)nc1-c1nc-2no1 C1(C(=O)NC2CCOC(C(=O)NCCc3c[nH]nc3C)C2)(CC)CCCC1O C1(NC(C)=O)CCC2(CC1)CN(C(=O)CCNC(c1ccccc1C)=O)CCO2 N1(C(C2C(C=C)CC2)=O)CCC(CNC(=O)CCC(=O)NCC)(CC)C1 c1(C(=O)NCC2C3CN(C(CCC(C)(C)OC)=O)CC32)c(F)ccc(Cl)c1N c1(OC)ncc(C(=O)NCCC(C)(C)NC(=O)CC2CCC(C)CC2)cn1 C1(C(=O)N(c2cccc(CO)c2)C)(OC)CCN(C(=O)C=Cc2nc(C)co2)C1 N1(C(c2c(OC)csc2)=O)CCC(C)(NC(c2nnsc2C)=O)C1 N1(C(c2cc(CCC)[nH]n2)=O)CCCC1(C(=O)N(C)Cc1cn(C)nn1)C(C)C Cc1ocnc1C(c1nnnn1Cc1cccs1)NCCc1ccc(Cl)s1 c1(C(N2CC(NC(c3c(CCC)[nH]cc3)=O)C(O)C2)=O)cn2cc(Cl)cnc2n1 n1(CC(=O)NCC(C2CCC2)NC(C2CC(n3cccn3)C2)=O)ccccc1=O C1(C(=O)NCC2CC(CF)C2)C=CCN(C(c2ncc[nH]2)=O)C1 C1(C(N2CCCC(NC(C(C)Sc3ncccn3)=O)C2)=O)CCCC12OCCO2 C#CC1CN(C(=O)C(O)C=C)CCN1C(=O)COC1CCCC1 c1(OC)cc(C(=O)NC2CC(C)N(C(=O)CCn3cncn3)C2)cnc1C C1(C(N(CCNC(C(C)C)=O)C)=O)CC(O)CN1C(=O)CCCF C1(C(N2CCC(N(C(=O)C=CS(C)=O)CCCC)CC2)=O)CCCCC1(F)F C(=O)(C1=C(Cl)CCC(C)C1)N1C(C(C)NC(COCCCCC)=O)CCC1 N1(C(C(CC=C)C)=O)CC(CNC(c2cnn(C3CC3)c2C)=O)C(C)(C)C1 C1(C(N(c2c(C)cccc2)C)=O)CC2(CC2)CN1C(=O)CC1CCCOCC1 Cc1n[nH]c(=NC2CCCN(C(c3cnc(CO)nc3C)=O)CC2)s1 c1(C(=O)NCCN(CCOC)C(C2(C)CCCO2)=O)cn(C)c(C(F)F)n1 C(=O)(CCC(=O)NN(C)C)NC1CC2(C(C(N(C(C(C)SC)C)C)=O)C2)C1 C1(CNC(c2cnn(CCO)c2)=O)CCC2(CCC2)CN1C(C1CC(O)C1)=O C1(CC)CCCN(C(=O)C(C)OCCC(C)C)C1C(=O)NCc1ccncc1Cl c1(C(CC(=O)NCC2N(C(c3c(CCC)nns3)=O)CC=C2)C)ccc(F)cc1 Cc1coc2ccc(C(N3CC(NC(=O)C(O)CC(N)=O)CC3CO)=O)cc12 C(=O)(CC(O)C(C)C)N(C(C)CNC(C1COCCN1C1CCCC1)=O)C N1(C(CSCCC(C)C)=O)C(C(N2CCN(C)C(=O)C2)=O)CC2CCCC12 C1(C(=O)NC2CN(C)C2)C2CC1N(C(=O)Cc1cccnc1Br)C2 c1(C(=O)NCCNC(C2CCN(CCF)C2)=O)ccc(OC2CC2)cn1 C1(C(N2CCC(O)(CNC(c3ccc(=N)[nH]n3)=O)C2)=O)CCC2(CCC2)O1 N1(C(=O)C(Cl)=CCl)CCN(C(c2cc3n(n2)CC(O)CO3)=O)C2COCC12 C1(CCNC(C(C)(C)OCC)=O)CCCN(C(=O)C=CI)CC1 CCC(C)(C)CCCC(=O)N1CCC(=CCNC(C2CC2F)=O)CC1 Cc1c(O)ccc(C(=O)Nc2ccc(NC(c3cncn3C)=O)cn2)c1C C1(CNC(C(C)C=O)=O)CC2CC2N1C(=O)C(C)(F)F.c1(SC)cccc(Cl)c1 C#Cc1ccc(Cl)cc1NC(=O)C(C1CCCC1)N(C)CC Cc1ccc(C)c(COC(c2ccccc2SCC(=O)Nc2ccsc2Cl)=O)c1 C1(c2c(CC)ncs2)NC(=O)N(C(C)CC)C(Cn2cnnc2C)=C1C(=O)OC C(C(C(=O)NCCC1CCCN1C(c1ccn(C(F)F)n1)=O)N(C)C)OC Cc1cccc(OCCC(=O)NC2(CNC(c3cnc(C(C)C)o3)=O)CC2)c1F S(=O)(=O)(c1ccc(C(=O)NCC23CC2CN(C(C2(C)CC2)=O)C3)cc1)NC C1(C(=O)NCCOCCCNC(c2ccc(C#C)o2)=O)CCn2c(C)nnc2C1 c1(SC)cccc(NCC2CCCN2C(c2ncoc2C)=O)c1 C1(CCOCCOC(C)(C)C)CSCCN1C(C1CC(=O)N1)=O.C1CCC(=O)N1 N1(C(C(C2CCN(C(C(C(=O)OCC)(C)F)=O)CC2)C)=O)CC2CC(C1)C2(C)C N1(C(CCC=CC)=O)CCC(C)C(CNC(C2(CO)CCOCC2)=O)C1 CC(C)CCC(F)C(=O)N1CCC(CNC(=O)CC2CC3C=CC2CC3)C12CC2 C1(NC(C2(COCC)CC2)=O)CCC(N(C(=O)C(C)n2ccnn2)C)CC1 N1(C(C=CC)=O)CC(NC(C2CC(=O)N(CCOC)C2)=O)C(O)C1 C(c1ccc(SC)cc1)=CC(=O)NC1CN(C(c2cnc(OCC)s2)=O)CC1O c1(C(C)=O)ccc(CC(N2CCN(C(=O)Cc3cnc(C)[nH]3)CC2)=O)cc1 c1(C(N(C2CCCC2)CCNC(=O)CCCC2CCC2)=O)cc2ncccc2o1 CCN=C(NCCC1CCC(OC)(OC)C1)N1CCCC(OC(=O)C(C)C)C1 c1(CNC(C2C(c3n(C)ccn3)OCC2)=O)cc(Cl)ncc1O c1(C(=O)NCCN(C(C=CC(=O)OC2CC2)=O)C2CC2)cc(F)cc2nc[nH]c12 N1(Cc2c(-c3cc(F)c(F)c(F)c3)ccc(Br)c2)C2CCC1CC(O)(C1CC1)C2 c1(CONC(Cc2cc(OC)c(Br)cc2)=O)cc(OC)c(OC)c(I)c1 C1(NC(C(CC2CCC2)NC(C2C(=C)C2)=O)=O)CCCC1N=[N+]=[N-] Cn1nnc2cc(C(=O)NCC3(C)CN(Cc4cc(Cl)cnc4F)C3)ccc12 C1(NC(c2c(C)ncnc2)=O)CS(=O)(=O)C12CCN(C(c1cnoc1)=O)CC2 Cc1ccc(CC(N2CCOC(C(C)NC(=O)CC3CCOC3)C2)=O)cc1F Cc1ccc(C(=O)NC2CC(CNC(=O)C(C(C)C)n3cnc(C)c3)C2)c(C)n1 CCC(C)(COC)C(=O)NC1CC(NC(c2nc(C3CC3)n[nH]2)=O)C1 c1(CN2CCCC(C(=O)NCC(c3ccc(Br)cc3)(C)O)C2)cccc(Br)c1Br N1(C(C(=O)NCC(F)F)=O)CC2CC(C1)N(C(C1CCOC1C1CC1)=O)C2 N1(C(c2nc(CC)oc2)=O)CCC(F)C(NC(c2ccccc2CC)=O)C1 N1(C(C2CC(N(C(C3CN(C(C)C)C3)=O)C)C2)=O)CCCC(F)(F)C1 N1(C(C(F)=C(C)C)=O)CCC2(CCCCC2NC(c2cc(C(N)=O)[nH]n2)=O)C1 c1(OC(c2nsnc2N2CCCC2)=O)ccc(F)c2c1C(=O)C(=O)N2 c1(C(N2CCC(CN(C)C(C3OCC4CCCC34)=O)C2)=O)cscc1S(C)(=O)=O C(=O)(C(C)CC(C)C)N(CC(CNC(C=Cc1cc(C)no1)=O)(C)C)C C1(CNC(C(c2ccc(F)cc2F)(C)O)=O)CC2C(C1)C2(F)F C1(C(N2C(C(N(C)C)=O)CC2)=O)CN(C(C2COC(=O)N2C)=O)C2(CCC2)C1 c1(-c2cc(OC(C)(C)C)cc(F)c2)cc2c(s1)CCN(Cc1ccnc(O)c1)C2 CCC(C)(C)COC(C)(C)C.C1C(CC)NCC2CC12 C1(C(N(CCNC(c2csc(C)c2C)=O)CCOCCO)=O)CN=C2N=CNN2C1 c1(C(=O)NCC2CN(C(CC(C)F)=O)C3(C2)CCC3)cc2ccccc2cc1F C=CCCCC(C)(C)C(=O)NCC1C(O)C(O)CN1C(=O)CNS(C)(=O)=O c1(C(N2CC(CC(C)NC(c3cnnc(O)c3)=O)C2)=O)cc2c(O)cccc2[nH]1 C(=O)(CCCC(F)(F)CO)N1CCC(C(C)NC(c2nn(C)cc2Cl)=O)C1 C(CC(C)(C)C)(c1n(C(CC)C)nnn1)(C1CC1)Nc1cnc(F)cc1C c1(C(N2CCC(NC(C3C4CC5C(C4)C35)=O)C(F)C2)=O)ccc(F)c(Cl)c1F Cc1ccc(C(C)C(=O)NC2CC2NC(c2ccncc2F)=O)cc1 c1(SC)ccc(N2CCN(C)CC2)c(F)c1.C1C(=O)N(C)CCOCCN1C N1(C(C(c2c(NC(C)=O)cccc2)(F)F)=O)CCC(O)(CNC(=O)C(C)C)CC1 c1(C(=O)NCC2OCC(CNC(C3C(=C)C3)=O)C2)cc(N)cnc1Cl c1(C(=O)NCCC2CN(C(COCCCCC)=O)C2)cccn2cnnc12 C(=O)(CC(F)(F)C(F)(F)F)NC1CC(CNC(c2cnc(CC)s2)=O)C1 c1(OC)cnccc1C(N1C(CSC2CCN2C(=O)CC(C)(F)F)CC1C)=O N1(C(CC(CC)SC)=O)CCCC2(CC(NC(C3(F)CCOCC3)=O)C2)C1 c1(CN2CCCC(C(N3CC(n4cccn4)C3)=O)C2)ccc(F)c(S(=O)(=O)N)c1 C1(C2CCN(C(=O)CC3CC3)C2)(NC(c2n[nH]cc2Cc2ccc(F)cc2)=O)CC1 C12(CNC(=O)C(F)F)CCCC(CN1C(c1ccc3nc[nH]c3n1)=O)C2 c1(C(=O)NCCN(C(C2(C(O)C(F)(F)F)CCC2)=O)CC)cc(CO)[nH]n1 CC1CC(NC(=O)CCc2nnc(C3CC3)o2)CN1c1cc(C(F)(F)F)ncn1 N1(C(C2(CNC(c3cnc(Cl)s3)=O)CCCO2)=O)CCOC(CC2CC2)C1 N1(C(C(C)NC(c2ccc(C)s2)=O)=O)CCc2ccncc21 n1(C(C)C)cc(C(=O)NC2(CNC(=O)CCCCOC)CCCC2)c(Br)n1 Cc1ccc2c(C(N3CCC(C(C)NC(c4occc4F)=O)CC3)=O)csc2c1 c1(C(N2CC(NC(C(C)c3cc[nH]n3)=O)(CO)C2)=O)cc2c(cn1)CCCC2 C#Cc1cccc(CC(N2CC=C(C(=O)NC(c3ncccn3)CC)C2)=O)c1 Cc1c(C(N2CC(n3cc(C(N4CCCC4)C4CC4)nn3)C(O)C2)=O)noc1 c1(CC(=O)NC(CNC(COCc2onc(C)n2)=O)(C)C2CC2)cc(Cl)n(C)n1 C(=O)(CCN(OC)C(=O)C(C)C(O)C(C)C)N1CCC(C(C)C)(COC)C1 c1(C(N2CC=C(CNC(c3ncn(C(C)C)c3)=O)CC2)=O)cc(O)c(F)cc1N C(=O)(C1=CC2CCC(C1)C2)NC(C(=O)NCC1(O)CCC(C)(C)C1)Cc1ccco1 c1(-c2ccc(CNC(C3CCOC3c3nc[nH]n3)=O)s2)ccc(Cl)cc1 c1(COC)cnn(C)c1C(=O)NC(C)CCN(C(=O)C(c1ccccc1)O)C c1(C(N(CC)CC2CCN(C(C3(CO)CC3)=O)CC2)=O)cc2sc(Cl)cc2s1 c1(CN(CCC)C(=O)Nc2cncc(C(F)(F)F)c2)cn2ccccc2n1 c1(NCc2ccc(OC)nc2)ncnc(N2CCCC(c3cc(O)n[nH]3)C2)c1C CC1(C)CCN(C(=O)CSCc2cccs2)C1CNC(C1CC=CCO1)=O c1(NC(CN(C)S(N)(=O)=O)=O)cccc(NC(=O)CC2CCC3CC23)c1 c1(C(N(C2CN(C(c3c(C)nns3)=O)C2)C)=O)cncc2ccccc12 c1(C(=O)NCC2(CO)CCN(C(COCCCC#C)=O)C2)cnc2[nH]cncc1-2 O=C(C#CC1CC1)NC(C(=O)NCCCF)C1(O)CCC1 N1(C(C(C)SCC)=O)CCC(C)(C)C1CNC(c1c[nH]nc1-c1ccncc1)=O c1(C(N(CCCCCC)CCNC(=O)C=C2CC2)=O)ccc(F)cc1OC c1(C(=O)NC2(CC(=O)NCCc3ccnc(C)n3)CCC2)c(Cl)cncc1Cl C1(CNC(c2ccc(C)cn2)=O)CCN(C(C2C=CCC2)=O)C1(C)C c1(-n2c(C(c3onc(C)n3)Nc3cnn(C(F)F)c3)nnn2)ncccc1Br C1(C(=O)NC2CC(NC(CC(c3ccccc3Cl)C)=O)C2)CCN(C)C(=O)C1 c12cccc(c1)C(c1ccc(F)cc1)NC2=O.C=CCCCN C1(CC=C)(NC(=O)C(C2CC2)OCC)CCN(c2nnn(C)n2)CC1 N1(NC(c2cccc(C)c2)=O)CCCC(C)(C#N)C1.C(C(C)C)SC N12CCN(C(C)C1)C(C1CC1)c1nsc2n1.C1(C(=O)OC)CCCC(C)CC1 N1(C(CC(C=C)(C)O)=O)CCc2ccc(CNC(C3CCCCS3)=O)cc2CC1 C(=O)(C1=CCCCC1)NCC(C1CCCC1)NC(C1CCC12CCC2)=O c1(OC)ncc(Cl)cc1C(=O)N(CCCN(C(=O)Cc1ccco1)C)C C1(CC(C)NC(C2(OCC)CCC2)=O)CCN(C(=O)CC2(C#N)CC2)CC1 C(=O)(CCC(O)C(C)(C)C)N1C(CN(C(c2c[nH]c(=NC)s2)=O)C)CCC1 C1(NC(C(CC)OCC)=O)CN(C(c2cnc(Br)s2)=O)CC(F)(F)C1 C(CC(=O)NCC12CCC(CC1O)C2)(C(F)(F)F)NC(C1C(C)CCOC1)=O C1(NC(C2(NC(c3c(C(C)C)c[nH]n3)=O)CC2)=O)CCCCCC1CO N1(C(c2c(COC)noc2)=O)CC(C)CCC1CNC(=O)C(F)(F)C1CCCC1 CC1(C)OC(C(=O)NCC(C)(O)CNC(c2csc(Br)n2)=O)C(C)(C)O1 C1(C)(CNC(CC2C(CC)C2(F)F)=O)CCCN(C(c2c(C)nsc2C)=O)C1 Nc1ccc(F)cc1C(=O)NC1CCCC1CNC(C1CC12CC2)=O N1(C(=O)CC2CC=CC2)CC2(C1)CN(C(C1CC13CCOC3)=O)CCO2 N1(C(COCCOCC#C)=O)CCC2OCCN(C(c3ccsc3C#N)=O)C2C1 C1(C(=O)NC(C)Cn2cc(-c3ncc(F)cc3F)nn2)CC2CC(C1)C(=O)N2 N1(C(c2cnc(CCC)s2)=O)CC(CNC(C2CC(=O)N(C)C2)=O)C(C)(C)C1 C1(C(=O)NCc2nc(CNC(c3cc(C4CC4)on3)=O)sc2)CCCC(F)C1 c1(C(N2C(CNC(c3c(C)ccs3)=O)CC2)=O)cnc2c(C)cnn2c1 c1(N2CCN(C3CCN(C(=O)C(F)(F)c4ccco4)C3)CC2)c(SC)cccc1C.CO C1(NC(c2ccc(O)cn2)=O)CC(C(=O)NOCC(O)COCCO)C12CCC2 c1(-n2c(C3(NCC4(SC)CC4)C(C)(C)C3)nnn2)ccccc1-c1cc[nH]n1 N1(C(CN(C(C)C)C(c2ccncn2)=O)=O)CCC2(C1)CC2(F)F S(=O)(=O)(CCC(=O)N1CCC(O)(CCNC(=O)CCC=CC(C)C)C1)NC C1(CC(=O)NCCCN(C)C(c2ccnnc2)=O)CCCC2CCCCC12 N1(CC)CCC2(CC1)CN(C)C2.C(=O)(C(C)CC=Cc1ccccc1)N Cc1[nH]nc2ccc(C(N3CCCC(F)(CNC(=O)CSC(C)C)C3)=O)c(Cl)c12 c1(C(=O)NCC2(F)CCC(NC(C)=O)C2)c(OC(F)F)cccc1Cl C1(N(C)C(c2ccn(C(F)F)n2)=O)CN(C(c2c[nH]nc2C2CC2)=O)CC1F N1(C(C=CC2(C)COC2)=O)CCC2CN(C(=O)CC3CC(C(F)F)C3)CC12 c1(C(=O)ONCC)cc(C)c(C)nc1C.C12CCN(C1)C2=O CCC(CNC(c1cc(CC2CC2)on1)=O)(CC)NC(=O)C(=O)NC1CC1 O=C(C#CC1CCOC1)NCC1COCCN1C(c1cc2cnccc2[nH]1)=O c1(N2CCC(C)(F)C2)ccc(S(=O)(=O)NCCc2cc(Cl)cc(Cl)c2)cc1C#N CC1CC2CN1C(=O)OCc1ccc(s1)NC2=O.C(C)(C)(C)SC1CC1 C1(NC(C(COC)c2ccccc2)=O)(CO)CCCN(C(=O)C(C)SC(F)(F)F)C1 c1(OCC(=O)NCC2CC(F)(CNC(C=C)=O)C2)cc(F)ccc1F CCC(C(=O)NCC#CC(N1CCC(C2CCC2)C1)=O)C(C)(C)CC C(=O)(C#CC(=O)N(C)C)N1CC(CC(C)NC(c2c(CC)ccs2)=O)C1 c1(C(N(CCNC(C(CC)n2nccc2C)=O)C)=O)ccnc(OC(F)F)c1 c1(CN(C(=O)NCCCC2CCCN(C)C2)C2CC2)c(O)cccc1F C#Cc1ccc(C)c(NC(=O)C(C)NC(c2cnc3n2CCC3)=O)c1 c1(C(=O)NCC2CC(NC(C3OCCCO3)=O)C2)ccc(-c2ccccn2)o1 CCC(N=c1nc2sccc2c(NC2CCCCCC2F)[nH]1)C(C)C N1(CC)CCCN(C)CC1C.C12CC(C1)SCC2 N1(C(CN2CC(C)(OC)C2)=O)CCC2CCN(C(=O)CCC(C)N(C)C)C2C1 C1(C)CCN1CC(F)Cl.C(C(C)C)NC(=O)OC.CCO C1(C(=O)NC(C(=O)NCC2CCCCCC2)C2CCC2)C2CCC(F)C12 N1(C(c2c(C(C)C)nns2)=O)CCC(CNC(=O)Cc2nnc(O)s2)C(C)C1 CC(=O)CCCC(=O)NCC1CN(C(=O)CCOC2CCCC2)CC1C CCCCCC(CC)C(=O)N1CCC(CC(C)NC(c2csc(C)c2N)=O)CC1 Cc1ccc(C(N2CCCCC2CNC(=O)Cc2conc2C)=O)cc1CO N1(C(CNC(N)=O)=O)CCC2(CCC2)C(NC(=O)CN2CC(=O)NC2=O)C1 c1(C(N2C(C)CN(C(CC)=O)C(C)C2)=O)cc2c(s1)C(C)(C)CCC2 c1(C(N2CCC(NC(C(CCSC)OC)=O)C(C)C2)=O)ncnc2sccc12 N1(C(CC(C)(C)OC)=O)CCCC12CCCN(C(C1(CC3CCC3)CC1)=O)C2 Cc1cc(C(N2CCC(NC(c3ocnc3C)=O)C2)=O)c(C(F)(F)F)o1 CC(CO)C(=O)N(C)CC=CC(N1CC(CCN(C)C)C1)=O c1(OC)ccc(C=CC(=O)N(C2CCCN(C(c3csc(CO)n3)=O)C2)C)nc1 c1(C(=O)NCc2scc(CNC(c3c(CC)nn[nH]3)=O)n2)cc(Cl)ccc1C C(CC1CC1)(C(=O)N1CCC(CC2CC2)C1)NC(=O)C=CCn1cncn1 CC1(NCC2(C)CCCCO2)CCOC12CC2(F)F C(C)(CO)(C(=O)N(C)CC1(CNC(c2csc(C)n2)=O)CC1)OC c1(CC(=O)NC)ccc(F)cc1.N12CC(C1)C(=O)NCC2=O.CC(C)(C)OCCCC N1(C(c2cncc(C(=O)OC)c2)=O)CC=C(CCNC(C2CNC(=O)N2)=O)CC1 c1(C(N2CCC(NC(c3ccc[n+]([O-])c3)=O)C2)=O)c[nH]c2nccc-2c1 CCCCC(CNC(=O)C=Cc1ccc[nH]1)NC(=O)C(C)NS(=O)(=O)CC N1(C(c2cccc(C)c2)=O)CC(CNC(c2cc(N)ccc2Cl)=O)C2(CCC2)C1 c1(C(N(C2CCCN(C(=O)CCc3ccccc3O)C2)CC)=O)cc[nH]c(=N)c1 c1(C(=O)NC2CCCN(C(=O)CN3CCCC3)C2)oc2ccccc2c1CO C(=O)(C(C)(C)C(F)F)N1CC=CC(C(=O)NC(COC)C(C)C)C1 C1(CNC(CC2(C=C)CC2)=O)CCC2(CN(C(c3nocc3C(=O)NC)=O)C2)O1 c1(C(=O)NC2CC(CNC(=O)C(F)=CCCF)C2)csc2cncn12 c1(OC)cc(CN2CCC(C)(C(=O)NCCCN3CCCCC3)CC2)ccc1Cl c1(NC(=O)NC(CNC(C(C)NC(=O)OC)=O)(C)C(C)C)cc(Cl)ccc1C N1(C(C(CC)CC2CCCCC2)=O)CCCN(C(C2CCCS2(=O)=O)=O)CC1 c1(C(CNc2ccc(SC(CC)(C)C)cc2)(F)F)cccc(F)c1F C1(C(=O)NC2CN(C(C(CC)SC)=O)CC2(C)C)CCc2nncn2CC1 Cc1c(C(N2CCC(F)(CNC(C3(CCO)CC3)=O)C2)=O)ccc2ccccc12 C1(OC(=N)O)CCN(C(C2(N(C)C(C3C=CCC3)=O)CC2)=O)C1 CC(C1=CCN(C)CC1)OC(=O)C(O)CCOCC(C)(C)C Cc1[nH]nc(C(N2CC3C(C(N4CCCC4C4CCCC4)=O)C3C2)=O)c1Cl Cc1cccc(OCC(=O)NC2CCC(NC(C3CCCC3C(F)F)=O)CC2)c1 CC1(C)C(NC(C2CCCN(C(c3occ4c3CCC4)=O)C2)=O)C(C)(C)C1O CC(c1ccsc1)=CC(=O)NC1COCCC1NC(=O)C(C)(C)c1ncco1 C1(C(C(=O)N(CC(CC)NC(C2CC2OC(C)(C)C)=O)C)O)CCOCC1 C1(CC(N2CCC(NC(C(C(C)C)(C)C)=O)CC2)=O)Oc2ccccc2NC1=O C1(C(=O)OC)(C(=O)N(CC(C)NC(=O)C(O)CC(C)C)C)CC2(CCC2)C1 c1(OC)ccc(C(=O)Nc2ncc(CC(=O)Nc3cnc(Cl)cn3)s2)cc1F Cc1cc(C2CCCN2C(=O)C(=O)NCCN(C(F)C(F)(F)F)C(C)C)cnc1C C1(C(=O)NC2CCSC23CN(C(C2CC2CF)=O)C3)CC(c2cccnc2)=NO1 N1(C(Cc2cnc(C)[nH]2)=O)CCOC(CCNC(=O)CCN(C)CCO)C1 CC(c1ccccc1)=CC(=O)NCC1CCC(C)CN1C(=O)CN(CC(C)(C)C)C CC(C(=O)N(CC(C)(C)NC(=O)CC1CCCC(C#N)C1)C)C(C)(C)C C#CCC(C)C(=O)NCC(C1CC1)NC(c1ccc(Cn2ccnc2)cc1)=O c1(N(CCCCC)CC)ccncc1C#N.C1(C(=O)N)CCCN1C1CCCC1 c1(C(C)NCC(O)Cc2cccc(Br)c2)cc(F)ccc1OC(F)(F)F c1(OC)ccc(C(=O)NC2CCCCC2NC(=O)C(C)OCCC(C)C)nc1 C1(CC(=O)N(C(CC(=O)NC)C2CC2)C)CN(C(=O)C(C)OCC2CC2)C(C)(C)C1 c1(C(=O)NC2(CO)COC(C(=O)O)C2)ccn2ccnc2c1.n12cc(nn1)C2 C(=O)(C1=CCOCC1)NCCC1(NC(C23CC(C(=O)OC)(C2)C3)=O)CCC1 C=CCC(C(=O)N1CC(CNC(=O)C(=Cc2cccs2)C)C(O)C1)C(C)C CCC(CCC(=O)NCC1(C(F)F)CCN(C(=O)C(F)(F)c2nccs2)C1)OC c1(N2CC(N(C)C(C3CCOCC3)=O)C2)nc(C2CCC2)ns1 N1(C(Cn2cc(CCC(CC)C)nn2)=O)CCC(O)C(F)(F)C1 c1(OC)nc(C)ncc1C(=O)NCCC(C(C)C)NC(c1cc(C)cc(Cl)c1)=O C1(C(=O)NCC(C)(C)NC(C(c2ccc(F)c(Cl)c2)C)=O)CCc2ncnn2C1 C1(C(=O)NCc2nccc(C)c2)CC12CCN(C(=O)Nc1ccccc1)C2 c1(OC)cc(C)ccc1C(=O)OCC(=O)N(C)CCNC(C1CC(F)C(=O)N1)=O N1(C(c2c(C)coc2C(C)(C)C)=O)CCC(C)C(NC(C2C3COCC23)=O)C1 C(=O)(CC(C)(C)c1cccc(Br)c1)NC(C(C)NC(C=C(CC)CC)=O)C C(C(=O)NC1CN(C(=O)Cc2conc2C)CC1O)(C(C)C)(C(C)C)NC(C)=O N1(C(CCCOC)=O)CCCC12CCN(C(C1CCc3ncccc3C1)=O)CC2 C1(C(N(CC(=O)NCc2coc(C)n2)CC#C)=O)CCOC1C(C)C C1(NC(CC(C(C)C)(F)F)=O)CN(C(=O)C(F)CC2CC2)CC12CCOCC2 CC(=O)CCCC(=O)NC(CNC(=O)C(C)Oc1cccnc1)C(C)C C1(NC(c2c(C)n(CCO)nc2)=O)CCC(C)N(C(c2ncccc2CO)=O)C1 S(=O)(=O)(c1ccc(Br)cc1N1CC2CCCN2C1)N1CCC(CCC=C)C1 C12(C(=O)NCCC(C)N(C(c3cnn(C(C)C)n3)=O)C)CCC(CC1)C(C)(C)O2 c1(C(N2CCC(NC(c3nccnc3Cl)=O)C2)=O)cnc(Cl)cc1Cl C1(C(N(CCCCC=C)C)=O)CCCN(C(c2ccncc2Cl)=O)C1 CC(F)(F)CCCC(=O)NC1C2COCC1CC(NC(=O)CCNC(=O)CO)C2 c1(CN2CC(NC(Cn3ccc(C)n3)=O)C(F)C2)cnn2ccncc12 c1(CC(N2C(C(=O)NCC(C=C)(F)F)CC2C)=O)cccnc1F C1(CC(=O)NC)CCNC1=O.C12CCN1C(=O)NC2 c1(OC)ccc2c(c1)CN(Cc1ccnc(Cl)c1F)C(C)C2 C1(NC(c2n(CC)ncc2)=O)CCN(C(c2cnc3[nH]cncc2-3)=O)C12CCC2 c1(C(=O)NCC2(F)CC(NC(C(C)NC(C)=O)=O)C2)cncc(C(F)F)c1 c1(NC(C2N(C(C=C(C)C3CC3)=O)CC(F)C2)=O)cccc(N=[N+]=[N-])c1 CC(=O)CCN=C(NCCCC(F)(F)F)NCC1CC(=O)N(C(C)C)C1 N1(C(c2n(C)cnc2)=O)CCCC(CNC(c2ccc(Br)cn2)=O)C1 Cn1ccc2ccnc(N(CCC3CC4(CCCC4)CO3)CCOc3ccccc3Cl)c12 CC(CC(=O)NC12CCC(CC1)N(C(=O)C(c1ccc(Cl)s1)=O)C2)CC(F)(F)F C(=O)(CCCCCCCCCO)NC1(CO)CCN(C(Cc2nc(C)sc2)=O)C1 N1(C(C(C)NC(C2CCCC2)=O)=O)CC=CC(NC(C2(S(N)(=O)=O)CC2)=O)C1 N1(C(C2CC(C)(F)C2)=O)CCCC2(C1)CN(C(=O)CSCc1ccccc1)C2 C1(C(N(CC(COCC)O)C)=O)(NC(=O)CC(C)O)CCCC1C CC(CCCC(=O)NC1(C)CCCN(C(=O)Cc2ccns2)C1)c1ccccc1 c1(C(=O)OC)ccc(C(=O)NC23CCC2CN(C(=O)CCS(C)(=O)=O)C3)c(F)c1 c1(CC)cc(C(=O)NCC2C(CC)CCN2C(C2C=CCCC2)=O)oc1CC C1(NC(C(F)=CCC)=O)CC2CCC(C1C)N2C(c1ccc(CC(C)C)cc1)=O C(=O)(C(CN(C)C)NC(=O)CCc1nccn1C)N(CCOCC)C c1(C(=O)NC2CCCN(C(CC3(NC(C)=O)CC3)=O)C2)cc2cc(Cl)ncc2[nH]1 c1(C(=O)OCC(CC)(C)Cl)cc(COC)cn1C CCCCCCC(CC)C(=O)OCC(=O)NOc1ccc(F)c(F)c1F.C(C(C)(C)O)O c1(CN2CCC(C(=O)NC3CC(=O)N(C4CC4)C3)C2)cccc2[nH]ncc12 N1(C2CC3C(NC(C)(C)C)C3C2)CCN(CCCCC(=O)NCC(F)(F)F)CC1 CCCC(O)CC(=O)NC(C)CNC(c1cn(-c2cccc(F)c2)nc1C)=O c1(C(=O)NCCN(C(c2c(C)nc(C)n2O)=O)CC)ccc(F)cc1N N(C1CCc2cccn21)C(c1nnnn1CC1CCCO1)Cc1ccc(C)o1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCCC1CN(C(Cn2nc(C)n(C)c2=O)=O)C1 C1(F)(C(N(CC(CNC(c2c(C(C)C)[nH]cc2)=O)C)C)=O)CCN(C)CC1 CCCCC(C(=O)N(CCC(C)NC(=O)C(C)O)C)ON=C(C)C S(=O)(=O)(C(C(F)(F)F)N1CCC(n2ccc3ccccc23)C1)NC(C)C C1(C2CN(C(=O)CCCNC(c3ccsc3)=O)C2)(NC(CN(C(C)C)C)=O)CC1 C#Cc1cccc(C(=O)N(CC(=O)NCC2CC2Cl)C(C)C)c1C CC1Cc2sc(C(=O)N(C)CCN(C)C(C3(n4cncn4)CC3)=O)cc2C(C)C1 CC1=CC(C(=O)NC(C)C(CO)NC(=O)CCOC2CCC2)SC1 c1(C(c2n(CC=C)nnn2)NCC(Cc2ccco2)CO)cncc(C=C)c1 c1(C(C)F)ccc(C(=O)NCC2(CN(C)C(C3COCCOC3)=O)CC2)cc1 Cc1cc(NC(C(C)NC(C2(C)CC3(CC3)C2)=O)C(C)C)nc(C(F)(F)F)n1 C(=O)(C(F)(F)C(F)F)N1CCC(C(C)(C)NC(=O)CC(O)C2CC2)CC1 S(=O)(=O)(c1cccc(=NC(CC)C2CCCCC2)[nH]1)N1CC(OCC)C1 c1(C(N2CC3(C(C(=O)NC(CC)C(=O)OC)C3)C2)=O)cccc(O)c1[N+](=O)[O-] Cc1ccc(F)cc1C(N1CCC(O)(C(=O)NC(C2CCOC2)C)C1)=O C1(NC(C(=O)NC(c2cccc(Cl)c2Cl)COC)=O)CCC2(CCCOC2)C1 C1(CCNC(c2cc(-c3ccc(C)s3)[nH]n2)=O)C(C)CCCN1C(=O)C=CCO C1(NC(=O)C=CCc2ccco2)CC(N=c2cc(Cl)nc(C3CCCO3)[nH]2)C1 C1(C(=O)NC2(CNC(=O)COc3ccc(Cl)cc3)CCOC2)CC2C(C1)C2(F)F CC(C)C(C)(C)C(=O)NC(CNC(=O)Nc1cccs1)C(C)C.C1(=O)C(C)N1 c1(OCCOC)cncc(C(=O)NC2CCC(N(C(=O)C=C3CCC3)C)CC2)c1 C(=O)(C(C)(C)CF)NC1CCC(CCC(=O)NCCCCCN(C)C)C1 c1(C(=O)NCC#CCNC(c2ccc(SC3CC3)s2)=O)cccc2nc(S)oc12 C(=O)(C(C)(C)C(=O)N(CC(C)N(C)C(c1cc(C(C)C)oc1C)=O)C)NC C1(NC(COc2cccc(C#C)c2)=O)CC2CN(C(C3(C)CC3)=O)CC2C1 c1(CNC(CCC2(NC(CC(C)n3ccnc3)=O)CCCC2)=O)cccc(F)c1 C1(C(N(CCCNC(=O)C(C)(F)F)CC)=O)CCCCC12CCC2 c1(C(=O)NCCC=C(C)C)ccc(CN(C)C)o1 C1(C(=O)NCCN(C(c2sc(COC)cc2C)=O)CC)CCCCC1F C=CC(C)(O)C(=O)N1CC(CN(C)C(c2c[nH]nc2C2CCOC2)=O)C1 C1(NC(CC=CCC)=O)CN(C(=O)CCCCC2CC2)C2(CCCCC2)C1 CC1c2cc(Cl)c(Cl)cc2CCN1C(=O)C(c1ccccc1Cl)N C(=O)(C(F)CC(C)(C)NC(C1CCC(C)(O)CC1)=O)NCC1CC(C)(C)OC1 C1(CC(c2cccc(C(O)C(N3CCN(C)CC3)=O)c2)C)CC(C)(C)OC(C)(C)C1 C1(NC(c2cc(C)nc(C)c2)=O)CCC12CCN(C(c1cc(C)oc1C)=O)CC2 Cc1c(Cl)ccc2[nH]c(C(=O)NCC(O)CNC(c3c[nH]c(=N)o3)=O)cc12 c1(N)nccc2occc12.c1(CC(N2CC(C(=O)OCC)(C)C2)=O)ccc(C)cc1 C1(CNC(C2C(C)=C2)=O)CN(C(=O)C(O)C(C)(C)C)CC1(F)CO Cc1cccnc1CC(=O)NC(C)C(CO)NC(c1cc(C(C)(C)C)c[nH]1)=O c1(NC)snc(C)c1C(=O)NC(C)CCNC(=O)C(c1cccc(C)c1)(F)F c1(CC)cccc(F)c1C(N1CCC(COC)(NC(=O)C=C(Cl)Cl)C1)=O C(=O)(C(C)C(C)S(C)(=O)=O)NCC1(C(N)=O)CN(C(c2c(C)nccn2)=O)C1 Cc1cccc2[nH]c(C(N3CC(O)CC3C(=O)NCCc3ccccn3)=O)cc12 c1(C(=O)NC2CN(C(=O)C(=O)C=Cc3cccs3)C2)ccc(SC(F)(F)F)nc1 C#CCC(CC#C)C(=O)N(C1CC2CCC(C1)N2C(C12CCCC1C2(F)F)=O)C N1(C(c2cc(C)nn2C2CC2)=O)CC2CC(NC(c3cncc(Cl)c3Cl)=O)CC2C1 Cc1c(NC(=O)CC2CCCC2NC(=O)CSC2CC2)cnn1CC CCC(C(=O)NCC(C)NC(c1n[nH]c2nccc(Cl)c12)=O)C(C)(C)CC CN(C1CCCC1c1ccccc1C(F)(F)F)N1CCC2(CCC2)C1 N1(C(CCCCNC(N)=O)=O)CCN(C(C2CCCC(F)C2)=O)CC12CC2 C1(CNC(CC2OCC(C)(C)C2)=O)CCN(C(C2C=CC=CC=C2)=O)C12CCC2 c1(NC(C(C)OCCC=C)=O)ccc(C(=O)NC)cc1 C1(OCC)(CNC(=O)Nc2cc(N)ccc2Cl)Cc2ccccc2C1 c1(C(=O)NC(CC)CNC(=O)C(CC(C)C)C(C)C)cnc(P(C)(C)=O)cn1 c1(C(N(C(C)CNC(c2csc(C(C)OC)n2)=O)CC)=O)ccnnc1O c1(C(N2C(c3cccc(OC)c3)CC(O)C2)=O)c[nH]c2ccc(F)cc2c1=O N12CCC(CC1)NC2=O.c1(CN(CC(C)OC)CCCC2CC2)cccs1 c1(C(C(=O)NC(CC)CN(C(=O)C=CSCC)C)(C)C)ccc(C(C)(C)C)cc1 Cc1cc(CC(=O)NCCC(O)CNC(c2cccn2-c2ccccc2)=O)n[nH]1 CCC(CC(=O)N1CCOCC1CNC(=O)CC1CC2(CCCC2)CO1)C(F)F CCC(CC)C(=O)N1CCNC(C(N2CCN(c3ccccc3Cl)CC2)=O)C1 C#Cc1cccc(C(C(N2CC3CC3C2)=O)NC(=O)OC(C)(C)C)c1.C1CN1 c1(OC)ccc(F)c(C(=O)NCC(C2CC2)NC(C2CCSCC2)=O)c1F c1(C(N2C(CNC(CC(C)c3cccnc3)=O)C=CC2)=O)ccn2ccnc2c1 Cc1ncc2ccc(C(=O)NC3CC4CC(NC(c5nccn5C)=O)CC34)cn12 CC1(C)CCCC1C(=O)NCC1(CNC(=O)C(F)(F)CN2CCCC2)CC1 C(CC(C)CC)(C(=O)N1CCCC(O)(CO)C1)NC(Cc1c(CC)con1)=O O=C(CCCCc1ccccc1)NC1(CNC(c2cocn2)=O)CCOC1 c1(C(=O)NCC23C(CN(C(Cc4cnc(C)s4)=O)C2)C3)cnc2[nH]cc(C)c2c1 C1(C)(CNC(C=COCC)=O)CCN(C(=O)CC2CC(F)(F)C2)C1 C1(NC(CCCCSC)=O)CS(=O)(=O)CC1NC(=O)C(=Cc1ccccc1)C C1(CC)CN(C(C2CCCSC2C)=O)CC1C(=O)Nc1cnc(O)nc1 C(=O)(C(C)(C)C(=O)N(C1CCN(C(=O)C(F)=CC2CC2)C1)CC1CC1)OC N1(CC(N2CC3C(C2)N3C(c2cc(-c3ccccn3)[nH]n2)=O)=O)C(=O)CNC1=O c1(SC)cscc1C(=O)N(CC(C)(C)CNC(c1cc(Cl)cs1)=O)C C1(C(=O)NCc2cn(CCC)nn2)C=CCN(C(=O)CCC2OCCO2)C1 c1(C(=O)NC(CC)CCOC)cccnc1CNC(=O)CC1CC2CC2C1 c1(NC(C2CN(C)CN2Cc2ccc(C(N)=O)nc2)=O)ncc(Cl)cc1F C(C(CC(=O)NCC1CC(O)CCO1)C1CC1)NC(C1CCCC2CC12)=O N12CCC(CC1)C(=O)N1CCC(C1)n1cc(nn1)CC2.c1(N)ccccc1.CCO c1(C(C(=O)NCC(C)C)N(CC=C)CC2CC(C(=O)NCCO)C2)ccn(CC)n1 n1(CCCC)nc(C)c(NC(=O)C(F)C2CC(NC(c3ccnn3C)=O)C2)c1C c1(C(N2CCN(C3CCCC3)C(=O)C2)=O)cc2c(s1)-c1ccccc1CC2 C1(NC)CCN(C(c2c(F)cncc2Br)C(=O)NC(C2CCCC2)C)CC1C N1(C(c2cccnc2)=O)CCC2CC2(C(=O)NCc2cccc(O)n2)CC1 N1(C(C(C)N(C(C)=O)C)=O)C2CC=C(C(=O)N(CCCN=[N+]=[N-])C)C1CC2 C(CC(=O)Nc1cnccc1N(C)C)(C(C)C)NC(C(CC#C)O)=O C1(NC(CCNS(CC)(=O)=O)=O)CC2CC1CN2C(c1cccn2cnnc12)=O C(CO)(CCCCNC(c1ccc(CF)cc1)=O)NCCC(=O)OC c1(COc2ccccc2CN(C(C)CC2CCC(C)O2)CC)cccc(Cl)c1OC c1(CN2CCC(CNC(C(COC)C)=O)C2)ccc(Br)c2nsnc12 c1(OC)cc(C(N2CC(NC(=O)Cc3cc(C)no3)CC2C)=O)cc(C)c1 c1(C(=O)NCC2C3CC2N(C(=O)CCCc2ccncc2)C3)cc(F)cnc1O C=CCC(CNC(=O)CCc1nc(C)no1)NC(C1CCOC1)=O C(Cc1cn[nH]c1)(C(=O)N(c1ccsc1)C)NC(CCN(CC)CC)=O c1(C(=O)NCC(CC)(CC)NC(=O)CC(=O)NC2CC2)cc(Cl)c(C)cn1 C1(C(N2CCC(N(C(=O)Cn3ccc(Br)n3)C)C2)=O)CCc2nn[nH]c2C1 c1(C(=O)OC)cnn(C)c1C(=O)NC(C)C(C)NC(c1cn(C2CC2)cn1)=O C1(c2nnnn2C)(NC(C(C)C)c2cccs2)CCC(P(C)(C)=O)C1 c1(C(=O)NCCC(C)NC(CS(CC)=O)=O)nc2ccccn2c1F CC1CN(C(=O)CCc2cnn[nH]2)CC(C)N(C(=O)CC23CCC(CC2)CC3)C1 c1(CC)c(C(N2CCC(CN(C(=O)C(C)C(=O)OC)CC)C2)=O)[nH]c2ccccc12 c1(OC)nc(C(=O)NCC2CCCCN2C(=O)C=Cc2nnn(C)n2)sc1C N1(C(C2(CC=C)CC=CC2)=O)CC2CCCC(C1)N2C(C1CCCN(C(C)=O)C1)=O C(CC(O)C(F)(F)F)NC(C1CN(C(C2CCN(C(=O)OC(C)(C)C)CC2)=O)C1)=O CCC(C)CC(C)C(=O)NCCOCCOC(=O)Nc1ccc(OC)cc1 C(=O)(C1=NNC(C(F)(F)F)C1)N(CCC(C)NC(C1CC(CCC)C1)=O)C N1(C(C(C(C)C)O)=O)CCOCC(C)(CNC(c2ccc(C(C)(C)C)cn2)=O)C1 C1(CN(C)C)C(NC(=O)CCOCCNC(=O)CC2(O)CCC2)C1(C)C C1(NC(C=CC=CCC)=O)CN(C(c2ccc(C)nc2O)=O)C2(CCCOC2)C1 c1(C(N2CCC(O)(C(C)NC(c3cc(Br)n[nH]3)=O)CC2)=O)ccc(F)c(Cl)c1N CC(CCC(C)(C)C)C(=O)NC1CCCC(NC(=O)CN(CC(C)(C)C)C)C1 Cc1cnc(C(N2CC(F)CC2CN(C)C(C23CC(C2)S(=O)(=O)C3)=O)=O)c(C)c1 N1(C(C2C(CC)C2)=O)CCN(C(=O)CCC(N)=O)C(CC(F)F)C1 C12(C(N(CCOC(=O)NC(C)C(=O)NC3CCCC3)C)=O)CCC(C)(CO1)C2 c1(C(=O)NCCCCCCN(C)C(C2COCCO2)=O)cncc(C(F)F)c1 C1(C(N2CCC(NC(c3c(CC)con3)=O)(CF)C2)=O)CCC(C2CC2)CC1 Cc1cc(C(=O)NCC(C2CCN(C(=O)CSC(C)C)CC2)(C)C)c(C(F)(F)F)o1 C1(NC(C(C)C2CC2)=O)COC2(CNC(c3c[nH]ccc3=N)=O)CC1C2 C(C1CCC(C)CC1)=CC(N1C(CN(C)C(C2CCOC2)=O)CCCC1)=O CC1(C(=O)NCC(CO)OCC2CC2)CCN(C(c2cc(=N)[nH][nH]2)=O)C1 C12(CNC(CCSCC)=O)CC(NC(c3cnc(SC)[nH]c3=N)=O)(C1)C(C)(C)O2 c1(CCC(=O)NCC2CCC(NC(COCC=C)=O)CC2)ccc(C(F)F)cc1 C1(CC(=O)Nc2cccc(C(c3ccco3)=O)c2)CCC2(CNC2)OC1 C12(CNC(CCCNC(C)=O)=O)COC(CNC(=O)C(c3cccs3)N(C)C)(C1)C2 Cc1cc(C(=O)NCCc2ocnc2CNC(C2CCCC23CC3)=O)nc(O)c1 Cc1c(CC(N2CC=CC(NC(c3cc(Br)oc3C3CC3)=O)C2)=O)ncn1C Cc1cc(F)ccc1CC(=O)N(CCCNC(C1CC1C(F)(F)F)=O)C CC(C)C(C)C(CNC(=O)CNC=O)NC(c1cnc(S)n1-c1ccccc1)=O CC1CC(NC(c2ccc(F)s2)=O)CCN1C(C1CC2CC2CC1C)=O c1(C(=O)NCCC2CCCN(C(=O)C=Cc3cc[nH]n3)C2)cc(O)nc(O)c1 C(=O)(C(O)C(C)(C)C)N(C)CC1CN(C(=O)C(N2CCOCC2)C2CC2)C1 CCCC(C)CC(=O)N1CCCC(N(C)C(c2c[nH]nc2OC)=O)C1 Cc1ccc(C(=O)N(C)CC2CCCN2C(C2(F)CCCCC2)=O)nc1O C1(NC(c2cncc(N)n2)=O)CCCCN(C(=O)Cc2cc(C(F)F)no2)C1 C1(CNC(c2nc(CC)oc2)=O)CC(C)CN(C(c2cc(C3CCC3)no2)=O)C1 c1(CC(=O)NCCN(C(C2CC2C2CCC2)=O)CC)cccc(OC)c1Cl N1(C(=O)NCCC2CC(C)(C)OC2)CCCN(CC2CCCCCC2)CC1 c1(C(N2CCC(C(N(C)Cc3c(CC)noc3)=O)C2)=O)cncc(OC)c1 c1(C(=O)NC(C)CCCNC(c2cnsc2)=O)cnc2ccccn12 O=C(C1OCCn2ccnc21)NC12CC1CN(C(=O)CCn1cnnn1)C2 C1(C(=O)NC2CON(CC)C2=O)CC2(CCN(C(=O)C(C)O)C2)C1 N1(C(C=C(COC)C)=O)CCC2C(C(=O)N(C(C)C(C)C)C3CC3)C2C1 c1(C(=O)NCC2C3CN(C(C4CCCCO4)=O)CC23)ccccc1[N+](=O)[O-] CC1CCC(CNC(=O)CCSC(F)(F)F)CN1C(c1nnc(O)nc1O)=O Cc1nc2c(O)cc(C(N3CCC(O)C(NC(=O)C(C)C(C)C)C3)=O)cc2n1C n1(CC(=O)NC(CC)(C)CNC(C2Cc3nccn3C2)=O)c(C)cc(O)cc1=O C(=O)(C(O)C1=CCCCC1)N1CC(CNC(CCn2c(C)ncc2)=O)N(C)CC1 c12nc(cc(Cl)n1)N1CCC(C1)NC2=O.c1(COC(C)(C)C)cnsn1 c1(OC)cccc(C(F)F)c1C(=O)NCC(C1CCC1)NC(C1(C#N)CC1)=O C(=O)(C(CCC1OCCO1)NC(c1snnc1C)=O)OC C1(C(=O)NCC(C(C)C)(C)NC(c2cn[nH]c2)=O)CCC2(CCC2)O1 C1(C(=O)N(CCCNC(=O)C(F)(F)C2CC2)C2CC2)CC2CCCC12 c1(OCC)ccc(C(=O)NCC2(N(C(=O)C=CCO)C3CC3)CCOC2)cc1 N1(C(C(C)CSC(F)(F)F)=O)CC2CCN(C(c3snc(Cl)c3Cl)=O)CC12 C(CCOC)(C(=O)N1CC(N2CCOC2=O)C1)NC(CSC)=O c1(OC)ccc(C(N2CCC(C(=O)NCC3CCC(O)C3)C2C)=O)cn1 c1(C(=O)NCC2CCCN(C(=O)CC3CCC(=O)NC3)C2)cnc2cccnn12 CCCCCCC(C)CC(=O)N1CCCCC(NC(=O)C(F)(F)c2cnnn2C)C1 N1(C(CC(c2ccc(CC)cc2)C)=O)CCC(NC(=O)C(C)OC)C(F)C1 c1(SC)ccc(N)cc1C(=O)N(C)CC1(O)CCN(C(=O)C2CC2)CC1 c12cc(C(=O)OC)ccc1[nH]c(=O)[nH]2.N1(CC)CCCC1C(N)=O c1(C(N2CC(CN(C(=O)CCCC3CC3C)CC)C2)=O)cc(O)ncn1 CC1CCN(C(C2CCC=CC2NC(=O)Cc2cnoc2)=O)CC1O c1(CNC(C)CCS(C)=O)nc2cc(Cl)ccc2n1C C(=O)(N=S(C)(=O)C1CC1)c1onc(-c2cc(OC(C)(C)C)cc(Cl)c2)n1 Cc1cc(N)c(Br)cc1C(N1CCC(C(C)NC(=O)C=CC2CC2)CC1)=O c1(CC)c(C(=O)NCC2CC3CCC(C2)N3C(=O)C(C)O)cnc2ncnn12 C1(CC)CN(C(=O)C(F)C(C)(F)F)CCN1C(=O)CC1CCC(F)(F)C1 C#Cc1ccc(F)c(NC(CC(c2nnnn2CCSC)NCC)C2CC2)c1 C=Cn1nccc1C(=O)NCC1(C(=O)NCC2CC2c2ccoc2)CC12CCC2 S(=O)(=O)(c1cccc(C(C)C)c1)Nc1c(C)ccc(C(=O)OC)c1 C12(NC(CCSCCC)=O)CCC(CC1NC(C13CCC(CC1)OC3)=O)C2 Cc1ccc(C(N2CC(=O)NCC2C)C(=O)NC2CC(C(=O)OC)C2)c(F)c1C c1(Cn2c(C(=O)NC(CCNC(c3c(C)ncs3)=O)C)ccc2)cccc(F)c1 C(=O)(C(CCC(C)C)NC(c1ccc(C)cn1)=O)NCC(CCC)O C1(COC)(NC(=O)C=CC2CCCO2)CN(C(C2CCN(C)C2)=O)C1 c1(NC(C2(C)CCCN(C(c3cccc(C#N)c3)=O)C2)=O)ccc2oncc2c1 CC(c1ccccc1F)=CC(=O)NCC1(O)CC2C=CC1C2 Cn1cc(CN(c2ccccc2Cl)C(=O)NCCO)c(C2CCOC2)n1 C1(NC(c2ccc(C)c(Br)c2)=O)CN(C(C2C=CCC2)=O)C2(CCC2)C1 N1(C(c2c(Cl)cn(CC)n2)=O)CC2CC(NC(c3ncccc3OC)=O)CC2C1 C(=O)(CC(C)CCCCCC)NC(CC(=O)N(CC#C)CC)CC c1(C(=O)NC(CNC(CC(C(C)C)OCC)=O)C)ccc(=O)n2c1CCCCC2 C12(NC(C3(C=C)CCN(C(c4nc[nH]n4)=O)C3)=O)CC3CC(CC1C3)C2 CCC(CC1CC1)C(=O)N1CC(NC(c2cc(=O)cc[nH]2)=O)C(F)C1 c1(C(CC)NC(C2(CCO)CNC2)=O)cc(F)ccc1F N1(C(c2n[nH]c(C)c2C)=O)CCC2CN(C(c3cc(F)cc(F)c3)=O)CCC2C1 C1(NC(C(CC)COC)=O)CC2CC1CN(C(C1(CC(F)F)CCOCC1)=O)C2 C1(CC(=O)NC2C(CSC)COC2)CN(C(=O)CN2CCCCC2=O)CCC1C c1(OC)nc(N2CCC(C)(NC(=O)CC3CC(F)(F)C3)CC2)cc(C)n1 c1(C(N2C(C(=O)Nc3nnc(C)o3)CSCC2)=O)ccc(Br)cc1C(F)(F)F C(=O)(CC(C)(C)c1nc(C2CC2)no1)NCC1N(C(C(C)OCCCC)=O)CC1 C1(C(C)NC(=O)COC2CCOC2)CCCN1C(=O)Cn1ccnn1 N#Cc1ncc(C(=O)NC2CCCC(CNC(=O)CCCn3cccn3)C2)s1 CC1(NC(c2ncsc2Br)=O)CCN(C(=O)Cn2cnc(C#N)n2)C1 c1(NC(CCC)(c2nnnn2CCC2CC2)C2CC2)nc2ccc(Br)c(C)n2n1 CC1CN(C(=O)C=Cc2ccc[nH]2)CCN1C(C1CC(=C2CCC2)C1)=O CCCCC(CC)CC(c1nnnn1-c1ccccc1CC)NCC1C=CCC1 N=c1cc2n([nH]1)CCN(CCN1CCC(c3ccc(Br)cc3)CC1)C2 c1(NC(=O)CCCN(C(=O)C(C)C(C)(C)C)C(C)C)nc2ccccc2s1 C1(NC(COc2cn(C)nc2)=O)CCC(C)(CNC(=O)C2=CCCCO2)CC1 c1(C(=O)NC2C(NC(CC3(CC)CCCC3)=O)CCC2)ccc2ccncc2c1 c1(CNC2CC(NC(c3ccsc3Br)=O)C2)cnc2[nH]ccc2c1 C1(NC(c2ccnnc2S)=O)CCN(C(c2cn(C(F)F)cn2)=O)CCC1CO C1(C(N2CC3C(NC(=O)C(O)C4CCC4)(C3)C2)=O)CC2(CCCCC2)C1 C1(CCN(C(c2c(C)noc2)=O)C)CCCN(C(=O)CC2CCN(C(C)C)CC2)C1 c1(OC)ccncc1C(=O)NC1CC1NC(=O)CC(C)c1cccnc1 N1(C(COC2(C)CCCC2)=O)CC2(NC(=O)CCc3cncc(F)c3)CC1C2 N1(C(CC(C)F)=O)CCC2(CC1)CN(C(=O)Cc1cccc(C(F)(F)F)c1)C2 c1(CCOC)n[nH]c(=NC(=O)C2(C#N)CC3C=CC2C3)s1 c1(CCCNC(C(C)Nc2ccc(Cl)cc2Cl)=O)cccc2ncccc12 C(=O)(CCCC(C)(C)C)NCC1CCN(C(c2n(C)nnc2)=O)CC1O C(CCCCC(C)C)OC.N12CCC1C(=O)NCC1CC1C2=O c1(C(N2CC3(CC(CNC(C)=O)OC3)C2)=O)nn2c(c1I)OCCC2 c1(OC)ccc(C(c2ccc(Cl)c(I)c2)Nc2ccccc2)cc1OCC(C)(C)O C1(C(N2CCC(CN(C)C)C2)=O)(CO)CCN(C(=O)Cn2cc(Br)cn2)C1 N1(C(C)C)CCCC1C(=O)NC(C(=O)NCc1cccnc1)C1CC1 c1(CCCC(=O)NC2CN(C(C(C)NC(C)(C)C)=O)C(C)C2)ccc(F)c(F)c1 c1(CCC(=O)NCCCC(C)NC(=O)COCCF)cccc(Cl)c1Cl C12(CNC(Cc3cn(C)nc3)=O)CCCCC1N(C(=O)CC1CSCCS1)CC2 CC(C)CC(C(=O)N1CCCCC1CF)NC(=O)C(Cl)Cl CN=C(NCC(C)CSc1ccccc1)NCC1COC(=O)C1 c1(C(N2C(C)CCC(NC(Cc3scc(C)c3)=O)C2)=O)cccc2c(C)c(C)[nH]c12 c1(CC)cc(C(N2CCC(C(C)NC(=O)C(C)C(O)CC)CC2)=O)cc(C)c1 C1(CC(=O)NCC2(C)N(C(COC)=O)CCC2)CC(c2ccccc2)=NO1 C12(N3CC(CC)C3)CCCC(C1)NCCn1c2nnn1.C(C)(C)(C)OC(N)=O Cc1cc(C)n(CC(N2CC(C(C)NC(c3cnn(CCO)c3C)=O)C2)=O)n1 CCC(CC(=O)N1CCCCC1c1n[nH]cc1C(N1CC(n2ccnc2)C1)=O)C(C)C c1(C)nc(O)c2c(C)c(C)sc2n1.S(=O)(=O)(CCCNC(=O)N(C)C)N(CC)CC c1(OC)cc(OC)cc(CN2CC3CC3(C(=O)Nc3cccc(Br)n3)C2)c1 c1(OC)cc(CN(C(C23CCC(CC2)C3)C(=O)Nc2ccoc2)C)ccc1F Cc1cccc(OC)c1.c1(CNC(C(C)O)C)ncc(C2OCCO2)s1 C1(CNC(C2(C)CC2)=O)CC(CNC(c2cnoc2C2CCOCC2)=O)CO1 C(C1=NOC(C)C1)NC(C(CC1CN(C(CCSCCC)=O)C1)F)=O c1(C(=O)NCC2CC2CNC(C2CCOCC2)=O)cccc(F)c1F c1(C(N2CCN(C(=O)C(O)CCl)CC2)=O)cc(Cl)nc(Cl)c1 c1(CC)oc(C(=O)NCC2(NC(=O)C3=C(C)CC3)CCC2)cc1C(=O)OC N1(C(CC(COC)(C)C)=O)CCOC2(C1)CN(C(c1cncc3c[nH]nc13)=O)C2 S(=O)(=O)(c1ccc(N2CCN(C=O)CC2)c(Cl)c1)NCc1c(C)cc(N)cc1 c1(CC)ncc(C(=O)NC2CC2CNC(c2cc(C3CC3)[nH]n2)=O)s1 c1(C(=O)NCCN(C)C(c2cccc(F)c2)=O)ccccc1OC(C)(C)C Cn1nc(C(=O)NCCCOCCNC(C2CCCC2(C)C)=O)cc1F c1(OC)cccc(C(C)(C)C(=O)NCC(C)CNC(C2(CC(F)(F)F)CC2)=O)c1 Cc1ccc(C(=O)NC2(CCNC(c3cnc(Cl)c(N)c3)=O)CCCC2)cc1Cl C(C(C)(C(=O)NC(C)C(CO)NC(=O)CCc1nc(C2CC2)no1)OC)OC N1(C(CC2CC(C)(C)CN2C(=O)CSc2cn[nH]c2)=O)C2CCCC1COC2 N1(C(C(CC)NC(C)=O)=O)CC2CCC1CN2c1nccc(C(F)F)n1 C1(c2ccccc2F)(CNc2nnc(-c3c(C)cccc3)s2)CCCCCCC1 Cc1cnc(C(=O)NCC#CCNC(=O)C(C(C)(C)C)n2ccnn2)cc1C#N C1(NC(C2C(C(=O)OC)C2)=O)CC2(C1)CC(NC(=O)CC1(O)CCOCC1)C2 Cc1ccc(O)c(NC(=O)C(C)N(C(=O)CCc2cncnc2)C2CC2)c1 c1(OCC)cc(Br)c(C(=O)NC2(C)CN(C(C3CC3C(F)F)=O)C2)cc1OC C1(C(=O)NC(CC2CN(C(c3cc(SC)oc3)=O)C2)C)CCS(=O)(=O)C1 N1(C(c2nccc(CC)c2)=O)CCC2C(CCCN2C(=O)CC2CNC(=O)C2)C1 N1(C(C2(Cl)C(C(C)=O)C2)=O)CCC(C(=O)N(CC(C)C(C)(C)C)C)C1(C)C CC(CC(=O)N1CC(O)(CNC(c2cnn(CC(F)(F)F)c2)=O)C1)c1ccsc1 c1(C(=O)NC2CCCN(C(CCc3c(C)noc3C)=O)C2)ncc2n1CCCC2 C1(C(OC(c2nc(CC)[nH]n2)=O)OC)CCCN(C(c2ccccc2)CC)C1=O N1(C(CCOC)=O)CCCC(C2CCCCN2C(=O)CN(S(=O)(=O)CC)C)C1 c1(N(CC(CC)C)C)nc(N(C)Cc2ncc(C)s2)c2c(n1)CSC2 c1(N(C(C2N(C(C(CC)C)=O)CCCC2)=O)C)ccc(C)c(Cl)c1 Cc1nc(C(=O)NC(C)CC(C)NC(=O)C(C)SC(F)(F)F)ccc1C(F)F C1(C)(CNC(C=COCC)=O)CN(C(c2scnc2C)=O)CC1C.C12CN(C1)C2=O N1(C(Cc2c(SC)cccc2)=O)CC(NC(c2cc(O)nc(Cl)c2)=O)CC(F)C1 c1(CNCC(C(C)(F)F)Cl)cc(Cl)c2cccnc2c1O c1(C(N(C(C)CNC(c2c(Cl)cccc2Cl)=O)C)=O)cc(F)cc2ccncc12 C(=O)(CC(C(F)(F)F)c1c(C)nn(C)c1C)NC(CN(C(COCCC)=O)C)C C1(C(N2CCC(NC(C3=C(C)OCCC3)=O)(CF)C2)=O)CCOCC12CCCC2 Cc1ncccc1CN1CCOCC1C(=O)Nc1cnn(-c2cccc(Br)c2)c1 C1(NC(C(COC)C)=O)CN(C(C2(Cc3ccc(F)cc3)CCC2)=O)CC1O N1(C(C(=O)NC)C(C)C2CCC2)CCc2c(F)ccc(OC)c2C1 C1(C)(n2c(C)ncc2)CCN(N(C)Cc2ccccc2Cl)CC1 C(=O)(C(C)C(CC)CC)NC1CN(C(c2cc(CCC)ncc2)=O)CC1CC1CC1 N1(C(C2C(C)C2)=O)CCC(CCC2CCCN2C(=O)CCc2csc(=N)[nH]2)CC1 c1(CC)ccc(CC(O)C(N2CC3C(NC(=O)CN(C4CCC4)C)C3C2)=O)cc1 C1(NC(=O)CCOCC(F)(F)F)CN(C(C2CCCNS2(=O)=O)=O)CC1C1CC1 c1(C(=O)NC)cccc(Cn2cc(CCN3CCCCC3C)nn2)c1.C(CN)SCC N1(C(C2(NC(CCc3n(C)ccc3)=O)CCC2)=O)CCOC2COCC2C1 C1(NC(C(CC)C)=O)CCCC12CCN(c1snc(CS(C)(=O)=O)c1C#N)CC2 N1(C(CCC(C)NC(C2(CSC)CC2)=O)=O)CCn2c(cnc2C)C1 N1(C(C(CC)C)=O)CC(OC)CC1CCNC(=O)COC1CCCC1 CC(C)C(C(=O)NS(=O)(=O)C1(C)CC1)NS(=O)(=O)C1CC1 C(=O)(CCCCC(=O)N1CC2(COC(CNC(=O)CSCC(N)=O)C2)C1)NC N1(C(C2CC(C#N)(O)C2)=O)CCc2ccccc2C1CNC(C1(CO)CCC1)=O N1(S(CC2CCC(C)CO2)(=O)=O)CCC2NCCCC2C1 C(C1CCCCCC1)=CC(=O)NCC(C)(C)CNC(=O)COCCF c1(C(=O)NCC2CN(C(Cc3c(C)ccs3)=O)C2)ccnc(NC(=O)C2CC2)c1 C1(C(=O)NCc2c(C)coc2)CCN(C(=O)C2=COCC2)CC1C N1(C(C(C)OCC#C)=O)CCN(C(=O)C(C)(C)CF)CC1C1CCCC1 C1(C(=O)NCC(CNC(C(CCC)OC)=O)OC)Cc2cscc2C1 N1(N2CCC(C)C(CC=O)C2)CCC(C)(C#N)CC1.C(=O)CN(C1CC1)C(C)C C(CC(C)C(=O)NC1CC1NC(=O)CN(CC=Cc1ccccc1)CC)=CCC C1(C(=O)OC)(NCC=Cc2ccco2)CC2NCCC12 c1(C(C)=O)[nH]c2ccccc2c1C(=O)Nc1ccc(-c2ccco2)cc1 C(=O)(CCCCC(N)=O)NCC1CC(NC(C(C(C)C)NC(C)=O)=O)C(O)C1 N1(C(C(C)(C)NC(=O)C=Cc2ccsc2)=O)C(CO)CCC12CCC2 C1(NC(C(CC2CN(C(c3c(C)n[nH]c3)=O)C2)F)=O)CC2CC1CC21CC1 Cc1c(C(=O)NCC2CC2NC(=O)C2=COCCO2)nc2sccn12 C1(NC(c2scc(C)c2)=O)CCCCC1C(=O)NCCC1CCCCC1O C(C(=O)NC(C)(C)CCNC(c1snnc1C)=O)(C(F)(F)F)OC(C)=O C1(NC(CNC(CC)=O)=O)(CNC(c2coc(C(C)C)n2)=O)CCC(F)(F)CC1 N1(C(C(=Cc2ccccc2)C)=O)CCN(C(=O)C2CC2)CC1c1ccco1 C1(O)(CNC(C2(CC(=O)OC)CC2)=O)CCN(C(C2CC3(CC3)CO2)=O)C1 N1(C(COc2ccn(C)n2)=O)CC2CC(NC(=O)CCCN=[N+]=[N-])C1C2 C1(NC(Cc2cc(C)sc2)=O)CCCCC12CCN(C(C1CCN1S(C)(=O)=O)=O)C2 Cc1ncnc(C)c1C(=O)NCC(C)(C)OCC(=O)NCCn1cncc1C(N)=O c1(C(=O)NCCN(C(C2CCCC2)=O)CC)ccoc1C(F)(F)F N1(C(CNC(CCC)=O)=O)CC2(CCC2)CC1CNC(=O)Cc1ccc(C)nc1 c1(C(=O)NCC(C2CCCC2)NC(CN(CCC#C)C)=O)c(N)sc2c1CCC2 C1(CC)C(NC(=O)CS(N)(=O)=O)CCN1C(=O)C=Cc1cc[nH]n1 c1(N2CCCC(OC)CC2)nc(NC2CCN(C3CC3)CC2)nc2c1cnn2C Cn1cc(C(=O)NCC2(NC(C3C4CC4C4CC34)=O)CC2)c(O)nc1=O C1(NC(C2CCC=CCC2)=O)CCCN(C(=O)Cc2ccn(C3CCCC3)n2)C1 C(CSC)(C(=O)N1CC(=C(F)CNC(=O)Cc2cc(C)cs2)C1)OC C1(NC(C=CCOCCOC)=O)CCOC2(CCN(C(=O)CCC(=O)NC)CC2)C1 c1(C(=O)NCc2nc(CNC(C3(CC=C)CCOC3)=O)sc2)cc(C)c(F)cn1 c1(C(=O)NCCN(C(C2C(OC)CCC2)=O)C)cccc(NC(C)=O)n1 c1(C(N2CCC(CCNC(c3nnc(C)s3)=O)C2)=O)cc2n(n1)CCN(C)C2 C(=O)(C(=O)N(CCN(C(=O)C1CC1)Cc1ccco1)CC)N(CCCC)C c1(OC)c(Br)ccc(CNC2CCC(C(=O)Nc3ccc(C#N)c(Cl)c3)C2)c1F C1(NC(CCC(=C)Cl)=O)CCCC12CN(C(=O)C(C)OC)C2 C1(CNC(c2cnc[nH]2)=O)C2CCC(C2)N1C(=O)C=CC1CCCCC1 C1(C(=O)NCCCOCCNC(CC2CC(OC)C2)=O)CCCC2CC12 O(C=CC(=O)NCC1(F)CC(C(=O)NC2CC2)C1)CC.C12(CC1)C(=O)N2 CN1C(=O)COc2ccc(C(N3CCC(CNC(C4(C)CC=CC4)=O)C3)=O)cc21 CC(C)S(=O)(=O)CC(=O)N1CC(NC(=O)CCS(=O)(=O)N(C)C)CC(C)C1 C1(C(=O)NCCN(C(C(CC)NC(N)=O)=O)CCOC)CCCC1(C)C c1(C(N2CC(NC(C3C(=C)C3C(=O)OC)=O)C2)=O)ccc(F)c(C(F)F)c1 C1(C)(C(N2CCC(N(CC)Cc3ncoc3C(C)(C)C)C2)=O)CCC(=O)N1 c1(C(=O)OC)ccc(NC(=O)Cc2cc(N(C(C)=O)C3CC3)no2)c([N+](=O)[O-])c1 N1(C(c2nccc(CC)c2)=O)CCCC2(C1)CN(C(=O)C(C)CC(=O)OC)C2 C1(C(=O)OCC)C=CCN1C(=O)NCc1ccc(C)s1 C1(C(=O)NCC2CCCN(C(C=COCC)=O)C2)Cc2ccc(F)cc2C1 C1(NC(COCCN(C)C)=O)CN(C(=O)C2=CCC2)C2(CCC2)C1 c1(C(=O)NC2CC(F)(CNC(C(C)NC(=O)NC)=O)C2)nn(C)cc1[N+](=O)[O-] C1(NC(C=C(C)C)=O)CC(C)CN(C(c2cccc(-c3ccco3)c2)=O)C1 N1(C(c2cn(C(C)C)nn2)=O)CCC(C2CC2)C1CNC(C1(C)CCOCC1)=O CCC(O)CC(=O)NC1CCC(C(N2CCN(S(C)(=O)=O)CC2)=O)C1 C1(CC)CN(C(c2cccc(N)c2O)=O)CCN1C(=O)CC(C)c1cccnc1 N1(CC(=O)NCC2CN(C(c3n(C)nc(C4CC4)c3)=O)C2)CCCC2(CC2)S1(=O)=O c1(OCCC(=O)NC2CC(CCNC(=O)CC3CC=CCC3)C2)cccc(F)c1 C[Si]1(C)CCC(C(=O)NC2CCOCC2O)CC1 C12(NC(CS(=O)(=O)N(C)C)=O)CCCC1CN(C(C1(F)CC3(CCC3)C1)=O)C2 CCC(C(=O)N1CCCCC1C(N1CCCC(O)CC1)=O)C(C)(C)CC N1(C(C=C(CC)C)=O)CC(C)(CNC(c2cc(C3CC3)ccn2)=O)CC1(C)C N1(C(CC2(C=C)CCOCC2)=O)CCN(C(=O)CCCN=[N+]=[N-])CCC1C c1(CN2C(C)COCC2)ccc(S(=O)(=O)N2CCC(OCCN(C)C)C2)cc1C#N c1(C(N2CCN(C(CC(CC)C)=O)CC2)=O)ccc(S(=O)(=O)N2CCCC2)o1 CCC(C)(C)C(C(=O)N1CCC(O)(CNC(c2cncc(Cl)c2C)=O)C1)OC c1(C(=O)OCC)ccc(CC(=O)NC2CCC(C)N(C(=O)C(=O)NC)C2)c(Cl)c1 CCC(C(=O)N1CCC(NC(c2ccccc2C(C)(F)F)=O)CC1)C(C)O C#CCCCC(=O)NCC1C2CN(C(=O)CSCc3cccc(C)c3)CC12 Cc1cc(N2CCCC(CNC(=O)Nc3c(C(F)F)c(C)nn3C)C2)nc(Cl)n1 C1(C(N2CCC(CCN(C)C(C3CC(=O)NC3=O)=O)CC2)=O)C(F)(F)C12CCC2 c1(CC(=O)NCC2(Nc3cccc(F)c3)CC2)cccc(OC(F)F)c1F Cn1nc(C(F)F)c(CN2CCC3(CC3C(N3CCC(O)C3)=O)C2)c1Cl C(=O)(CCC(c1nnnn1CCCSCC)NC(C)Cc1ccc(C)nc1)NC c1(C(N2CC(NC(C3(CCC)CCC3)=O)C(C)CC2)=O)oc2ccccc2c1Cl C1CC(=O)N1.C(C(C)NC(=O)CN(C)C(C)=O)NCCOC N1(C(C(CC2CN(C(=O)CSc3nc[nH]n3)C2)F)=O)CCC(C2CC2)C1 N1(C(C(CCOC)NC(CN(C(=O)OC)C)=O)=O)CC2(CC(C)CO2)C1 C(=O)(NCC)OCC#N C1(C(N(C)Cc2ccco2)=O)CC(CO)CN1C(=O)CN1C(=O)CNC1=O C(C(=O)NCC1CN(C(=O)Cc2ccn(C(C)C)n2)CC1O)(C(C)(C)C)OC Cc1cc(CC(=O)NCC2CN(C(C34CCCC3C4)=O)CC2C)n(C)n1 C1(CNC(NC(C(C)(C)C)Cl)=NCC2CC3(CCC3)C2)CC2(C1)C(F)(F)C21CC1 C1(C)(CC)C=C(C(=O)N2CCC(O)(CCNC(=O)CCC(F)F)CC2)C1 c1(CC)ncc(C(=O)NCC(c2ccn(C)n2)O)s1.C12CCCC1CNC2=O N1(C(C)=O)CCN(C(c2cc(C3(CC)CCC3)c[nH]2)=O)C(C2CCCC2)C1 N1(C(C(C(C)C)N(C)C)=O)CCC(O)(CNC(C2CC2CC(C)(C)C)=O)CC1 c1(OC)ccnc(OC)c1C(=O)NC1CCN(C(=O)C(C)n2cncn2)CC1F N1(C(=O)CC2(N(C)C)COC2)CCCC2CCN(C(C3(F)CCCCC3)=O)CC12 C12(NC(C3N=C(C)SC3)=O)CCCN(C(c3ccncc3OC(C)C)=O)CC1C2 C1(C#N)(C(=O)NCCOCC(=O)NCC(CC2CC2)OC)CCCCC1 C(=O)(C(C)C(O)C(C)C)NCC(C1CCCC1)NC(c1cc(C)ncc1C)=O c1(C(N2CC(N(CC)CC)C2)=O)ccc2c(n1)CN(C(=O)Cc1n[nH]c(C)n1)CC2 c1(NC(N2CC(CC(=O)NCC(=O)OCC)C23CCC3)=O)ccc(Cl)c(F)c1 N1(C(CNC(C)=O)=O)CCC(CNC(C2CCCN2C(C)=O)=O)C1 c1(C(=O)NC2CCN(c3nc(C)c(C)s3)CC2O)cccc2nc(C)sc12 C(C(CC(=O)N1CC(OCCO)C(O)C1)NC(c1cccnc1)=O)OC N1(C(c2ccc(C#C)cn2)=O)CC(NC(=O)CS(=O)(=O)NC2CC2)CC(C)(C)C1 C1(NC(c2ccccn2)=O)CCN(C(C2CCC3(CC3)C2)=O)CC1 N1(C(CC2N(C(C)=O)CC2)=O)CCC(NC(=O)CCc2ncccn2)C1(C)C c1(CC(=O)NC(C)CCN(C)C(C2CC2(Cl)Cl)=O)cccc2ccccc12 C(=O)(C1=CC2(CN(C(c3cn(CCO)nn3)=O)C2)OC1)N1C(CO)CCC(C)C1 c1(C2C(C(=O)NCC(C)CNC(C3CCCCC3)=O)C2)ccncc1F CCC(C(=O)N(C1CCN(C(=O)CC2(N(C)C)CC2)CC1)CC)C(F)(F)F n1(CCC(C)C)cc(C(N2CC(O)(CNC(=O)CCOCC3CCCO3)C2)=O)nn1 CN1N=C(CC(=O)NC2CC3CC(NC(C4CCC(C)(C)OC4)=O)CC23)CC1=O C1(NC(c2nc(CC)oc2C)=O)CCC(C)N(C(=O)Cc2nnc(O)s2)C1 c1(C(N2CC(OC)(CNC(=O)Cn3nc(C)cc3C)C2)=O)cnc2c(c1)CCC2 Cc1cc(NC2CCN(C(C3CCCC3)=O)C2)nc(S(C)(=O)=O)n1 c1(N2C3CN(C(C4C(C)(C)CCC4)=O)C(CC3)C2)ncnc2[nH]ccc12 C1(C)(CC)C=C(C(=O)N(CC(C)NC(c2ccc(NS(C)(=O)=O)c(C)c2)=O)C)C1 CC(C)CC(CN(C)C(c1ccoc1)=O)NC(=O)C(C)OC1CCCC1 Cc1nn(Cc2cccc(CNC(c3ccc(C(N)=O)nc3)=O)c2)c(C)c1Br c1(C(N(CCNC(=O)C(C)C(C)C)CC)=O)c(OC)ccc(OC)c1N c1(C(=O)NCCOCCNC(C(C=C)O)=O)csc(C)c1C n1(CC)nccc1C=CC(N1CCOCC1CN(C(=O)CNS(C)(=O)=O)C)=O CC1(C#CC(=O)NC2CN(C(=O)C(O)c3ccsc3)C2)CCCO1 C(=O)(C1=CC2CCCCCCC12)NCC(CNC(c1c(N)cn(C)n1)=O)O C1(C(=O)NC(C2CN(C(C=C(C)C(C)(C)C)=O)C2)C)CCC2(CC1)OCCO2 c1(C(=O)NC2CC3(CN(C(CC(=O)OCC)=O)C3)OC2)cnc2snc(C)c2c1 C(C(O)CC(=O)NCC1CC(NC(=O)C(c2cccc(Cl)c2)O)C1)N(C)C C=Cc1cncc(C(=O)NCC2CN(C(c3coc(CO)c3)=O)CC2C)c1 C1(C(=O)OC)C2CCN(C(c3cc(OC)cc(OC)c3NC(C)=O)=O)CC12 CC1(C(F)(F)F)CN(C(C2CCCO2)C)CC1C(=O)O N1(C(c2c(C)csn2)=O)CC(C(=O)NCC(c2ccncc2)C)C2(CC2)C1 CCC1CC(=O)N2CC1C2.C(Cc1ccoc1)(C(=O)OC)Nc1nnnn1C.C1CCC1 C(c1ccnc(Cl)c1)=CC(=O)NCC(C(C)(C)C)NC(=O)C=C1CC1 c1(NC(C)=O)cccc(CC(=O)NC2CCN(C(=O)CN3CCOCC3)C2C)c1 CC1C2CCC(C2)C1C(=O)NC(C(=O)NCC=Cc1ccc[nH]1)C1CC1 CC1CCCN1CC(=O)NCC1(CNC(=O)CNC(N)=O)CC1 Cc1nc(C#N)c(NCCC(=O)N(C)CCN(C)C(C2CC2C(F)(F)F)=O)o1 c1(OC)cc(C(N2CCCC2C(C)(C)NC(c2cnn[nH]2)=O)=O)ccc1Cl N12CC3(CN(C3)C(=O)CC3CCCN(C3)CCC1)C2.c1(NC)cccc(O)c1C C(=O)(C1=CCCC1C)NC(CNC(C(C)N(CC)CC)=O)C c1(OC)ncc(C(=O)NCC(C2CCCN2C(C2(CN(C)C)CC2)=O)(C)C)s1 c1(CN2CC3CN(C(c4cnc(Cl)c(F)c4)=O)CC32)cc(F)c(F)cc1Cl C1(NC(C(C)NC(=O)OC(C)(C)C)=O)(CNC(N2CC3C=CC2C3)=O)CCCCC1 N1(C(c2ccc(CC)cc2F)=O)CCCN(C(C2CC2C(F)F)=O)CCC1 n1(CCC(N2CCC(NC(=O)Cc3csc(S)n3)C23CC3)=O)cc[nH]c(=O)c1=O N1(C(=O)CC2CC=CCC2)CC2CN(C(C3CC4CCCC34)=O)CC2C1 CON(C(=O)C(CNC(=O)C(C)CC(C)C)C(F)(F)F)C1CCOCC1 c1(C(N2C(C(N(CCOC)CC3CC3)=O)CSC2)=O)cn(C)c(=O)n1C c1(C(=O)NCC(CC=C)NC(C2CC(C(=O)OC)C2)=O)cc(C)ccc1Br c1(NC(C(=O)Nc2cccc3occc23)=O)cc([N+](=O)[O-])cc([N+](=O)[O-])c1 c12c[nH]c3c(c1=O)CN(CC3)C2.n1(C(C)CNC(N)=O)c(O)nc2ccccc12 n1(CC(=O)NC2C(NC(c3c(C)oc(Cl)n3)=O)CCC2)ccc(=O)n(C)c1=O C1(O)(CNC(=O)CC2CCOC2)CC2CCC(C1)N2C(C1(O)CCCC1)=O c1(C(CNC(=O)CC2CCOC2)NC(C2CC(F)C2)=O)ocnc1C1CC1 C1(CC(N2CCC(N(C(COCC)=O)C)C3(C2)CC3)=O)Cn2ccnc2NC1=O CCCC(O)CC(=O)NCCC1(O)CCN(C(=O)COCCOC)CC1 C(=O)(CC1=NNC(=O)C1)NC(CC)CN(C(=O)CCn1c(C)csc1=O)C N1(C(C2(OC)CCCC2)=O)CCC(c2ccccc2)(CNC(=O)C(C)(O)CSC)C1 C(=O)(C1=NOCC1)N1CCC(C(C(=O)NCCN(CCC)C(C)C)F)C1 Cn1cc(CN2CCC3(CC3C(=O)NCc3ccc(Br)cc3)C2)c2ccccc12 c1(CN(C(=O)CCn2ccnc2)C)ccc(CNC(c2cccn2C)=O)cc1 C12(CNC(Cc3cccc(COC)c3)=O)CCC1CN(C(=O)C(F)(F)CSC)C2 C1(OC)CCC2(C(=O)NC3CCCCC3NC(C3C4COCC34)=O)CC12 C1(C(C(=O)OC)O)CCN(C(=O)Nc2cccc(-c3ccco3)c2)CC1 C(CNC(c1ncoc1C1CCC1)=O)(C(C)(C)C)NC(C=CC(C)C)=O Cc1cc2nc(NCC(C)(C3CC3)NC(C3CCCS3)=O)cc(=O)n2o1 O=S(=O)(c1cccnc1NCc1cc(Cl)cc(Cl)c1F)NC(CO)CCF n1(CC(=O)NC2C3CN(C(C(CC)(C)C(N)=O)=O)C2C3)ccc2ccc(F)cc12 N1(C(C2N(C(CCC)=O)CCC2)=O)CCCC(C)(NC(c2cc(Cl)c(Cl)s2)=O)C1 N1(C(c2n(C)cc(C(N)=O)c2)=O)CC(NC(=O)CCC(F)(F)F)C2(CCC2)C1 c1(C(=O)NC(CNC(c2cccc(N)c2)=O)CO)cc(F)cc(F)c1 C1(C(N2CCC(N(C(CC(=C)C)=O)CC)C2)=O)CN(C)CCO1 C1(NC(C2(C#C)CC2)=O)CCC2(CC1)CN(C(=O)CCCC(C)C)C2 C1(N(C(=O)Cc2cc[nH]n2)CC)CCCN(C(c2ocnc2C2CC2)=O)C1 c1(C(=O)NCC23N(C(=O)CNC4(F)CCOC4)CC(C2)C3)ccc(C2CC2)cc1 O=C(CCCCCn1cc(C2C3CCCCCC23)nn1)NC1CC2(CCOC2)C1 CC1CCN(C(C2C3(CC3)C23CC3)=O)CC1NC(=O)CCC(N)=O c1(C(N2CCOCC2(C)C2CC2)C(=O)NC(CC)C)ncc(Br)cc1C C=CC(C)(CC)C(=O)N1CC(CNC(=O)COCC2CC2)C(C(F)F)C1 C1(NC(c2cncc(CO)c2)=O)CCN(C(c2cc(CF)on2)=O)C12CCCC2 N1(C(C(C(C)C)NC=O)=O)CCC2(CC1)CN(C)C(=O)O2 Cc1ccc(Cl)c(N)c1C(N1CC2CCCN(C(c3cccs3)=O)C2C1)=O c1(C(=O)NC2CC2CNC(c2n[nH]cc2[N+](=O)[O-])=O)cc(F)c(Cl)c([N+](=O)[O-])c1 c1(C(N2C(CNC(c3c(C)nsc3)=O)C=CC2)=O)nc2ccccc2[nH]1 Cc1ccc(S(=O)(=O)NCC(N2CC3(CC(N(C(=O)CO)C)CO3)C2)=O)cc1 N1(C(c2cc(OC)no2)=O)CCC(C(O)CNC(C2C3COCC23)=O)CC1 C1(F)(CNC(C2C(CC)C2)=O)CN(C(C2CCN2S(C)(=O)=O)=O)C1 c1(C(N2CC3C(n4cc(-c5cccnc5)nn4)C3C2)=O)cccc(Cl)c1.CO C(C(C)(O)C(C)(C)C)OC.C(=O)(C1=NOC(C)C1)N1CC2(C1)C(=O)NC2 C1(C(=O)NC(CNC(CCCC#C)=O)C(C)C)CC2C(C1)C2(C)C Cc1cccc2c1CC(C(N1CCN(C(=O)C(F)C(C)C(F)(F)F)CC1C)=O)N2 C1(CC(N2CC(NC(N)=O)C2)=O)CCN(C(c2nnc(O)nc2O)=O)C1(C)C C1(N(C(=O)C=CC(F)(F)F)C)CN(C(=O)C(F)CC2CCOC2)CC1F N1(C(C(Cc2ccccc2)NC(C)=O)=O)C(C(=O)NCCCF)CCC1C1CC1 N1(C(C2C(=C)C2C(=O)OC)=O)CCC2(CCN(C(C3CCCCNC3=O)=O)CC2)C1 C1(NC(C2(C(C)C)COC2)=O)CCCN(C(C2COC(C)C2)=O)C1C CC(C)CC(C(=O)NC1CN2CCCC1C2)ONC(=O)C=CCF Cc1ncc(CC(=O)N(CC(C)O)CCNC(=O)CC2COC(=O)N2)[nH]1 c1(C(=O)NC2(CC(=O)NCC(CC(=O)NC)C)CCC2)cncc(F)c1C C1(CNC(c2n[nH]c(C)c2Cl)=O)COC(C)(C)CN1C(=O)C(C)NC(N)=O c1(CC)c[nH]c2ccc(OC(F)(F)F)cc2c1=O.C12CCN(CC1)OC2=O c1(C(N2CCC(C(C(=O)NC(C(=O)NC)C)C)CC2)=O)cc([N+](=O)[O-])ccc1C N1(C(c2cc(C(C)(C)C)on2)=O)CCC(CNC(=O)Cn2cc(CO)nn2)C12CC2 N1(C(C2OCCC(C)C2)=O)CC2(CC2)CC1CC(=O)N(C1CC1(F)F)CC(F)F c1(COC(C2CCCCC2Cc2ccccc2)=O)cc(Cl)c(O)c(Br)c1 C(=O)(CCN(C(=O)CSCCC#N)CC1CC1)NCC(C)OC C1(O)(CNC(c2cc(C)sc2C)=O)CCCN(C(c2ccc(C(F)(F)F)s2)=O)C1 c1(C(=O)NCCCCCNC(C23CCC(CC2)C3)=O)ccc(Cl)c(F)c1F CCCC(C#N)C(=O)NCCOC1CN(C(c2cnn(C3CC3(F)F)c2)=O)C1 CC(CN)C(F)C(=O)NCC1CC2CCC(C1)N2 c1(C(N(CCCNC(c2ncc[nH]2)=O)CCO)=O)cc2n(n1)CC(F)C2 Cc1cc(C(=O)NC(Cn2ccnn2)C(=O)N2CC3CC3C2)cnn1 c1(CC)ccccc1C(N1CC=CC(NC(c2cccnc2NC(C)=O)=O)C1)=O C1(C(N2CC(C)C(CNC(=O)C(C#N)C3CC3)C2)=O)C2C3CC4C1C1C2CC3C41 C(=O)(C(O)(CN(C)C)C(F)(F)F)N1CC(CNC(c2c(OC)scc2)=O)C1 N1(C(C(CC)NC(N)=O)=O)CCN(CC2(NC(=O)C(CC)SC)CC2)CC1 C(c1ccncc1)=CC(=O)NCC1(CC=C)CN(C(=O)C(C2CCOC2)OC)C1 C1(CC(C)C)CCN(C(c2csc(Cl)c2)C(=O)NCc2ccco2)C1 C(=O)(C(C)(C)N=[N+]=[N-])NCC(CN(C(C1OCCN(CC)C1)=O)C)(C)C C(CC(C)CC)(C(=O)NC(c1nccc(O)n1)C)NC(C1CC(CCC)C1)=O N1(C(c2nccc(CC)c2)=O)CC(NC(=O)CNC(=O)CCC(C)C)CC1(C)C C1(C(=O)NC(CC)C(N)=O)CN(C(c2ccc(O)cc2)=O)CC1F C#CC1CN(C(c2nccn2C)=O)CCN1C(c1csc(C(F)F)n1)=O Cc1c(C(=O)CN2CCOC(c3cccc(F)c3)C2)[nH]c2ccccc12 C(=O)(C(C)(C)C(C)C)NCC(C1CC1)NC(C1CN(CC(C)C)C(=O)C1)=O C1(C(=O)NC(C)C(=O)NCC(=O)N(C)O)CCCC(=O)CC1 CC(C(C)(C)NC(c1cnn(CCO)c1)=O)NC(=O)CCOC1CCOC1 C1(NC(=O)C2=CCCCC2)CCN(C(=O)C2=CCOC2)CC(O)C1 c1(COC2(C)CCN(C(CNC(COCCC=C)=O)=O)C2)ccc(F)cc1O CCCC(C)(CC)C(=O)N(C(CNC(=O)COC(F)F)CC)CC Cc1ccncc1C(=O)NC(C1CCCC1)CNC(=O)CCc1cncc(F)c1 c1(CSCC(=O)NCCCN(CCO)C(C2CC3CC3C2)=O)ccncc1 N1(C(C(N2CCCCC2=O)C)=O)CCC2C(CCCN2C(c2cc[nH]c(=N)c2)=O)C1 C1(C)(C(C)(C)C)CC(C(=O)NCC2CCCN2C(c2cnc(Br)s2)=O)C1 C(=O)(C(=O)CCC(C)(C)C)N(CCCN(C(CCn1nc(C)c(C)c1C)=O)C)C n1(CC=C)nc(CCCN2CCCCC2)nc1C1(C)CC1 c1(C(N(CCOCCN(C(CC)=O)C)C)=O)cccn(C(C)(C)C)c1=O N1(C(C(c2cncnc2)C)=O)CCC(C)(C)C1C(=O)NC1CC2CC(O)C1C2 C1(NC(C(CC=C)NC(=O)CC2CCOC2=O)=O)CCCCCC1C(N)=O C1(C(=O)NCCCN(C(C(C(C)C)C)=O)C2CC2)CCN(C)S1(=O)=O C1(NC(CCN(C(C)=O)C)=O)CCN(C(=O)C=Cc2ccc(C)o2)CC(C)(C)C1 Cc1ccc(O)c(C(N2CCC(CNC(=O)CC(C)c3ccncc3)C2(C)C)=O)c1 C1(NC(c2c(CC)c[nH]c2)=O)CC2CCC(C1)N2C(C1CCC(=O)N1C)=O C1(C(N2CCC(C)(NC(C3CCC(C)(C)C3)=O)C2)=O)(COC)CCCCC1 C#Cc1cc(C(=O)NCCCCCCNC(c2coc(COC)n2)=O)cc(F)c1 Cn1c(=O)ccn(CC(=O)NC2C=CCN(C(C3CCNC3=O)=O)C2)c1=O C1(CCOCC)CCN(C(C2(C)CC2(F)Cl)=O)CC1.C1(C(=O)NCC)(CF)CC1 C(=O)(CCCCCNC(c1cnn(C)c1)=O)NC(CC(=O)NC)C N1(C(COC)=O)CCC1CNC(C1(C(C)(F)F)CC1)=O c1(CC)c(C(N2CCC(CN(C(=O)CC(C)(C)OC)C)C2)=O)cccc1C CC(C(=O)NCC(C)NC(c1ccc[nH]1)=O)NS(C)(=O)=O C1(C(N2CCC(C(=O)NCCO)C2)=O)CCCCN1C(c1ccsc1)=O c1(C(C(=O)NCCN(CC(C)O)C(C2CC2C#N)=O)(F)F)c(F)cccc1F N1(C(C2C(=C)C2)=O)CCCCC(C2CN(C(=O)C(O)C(C)CC)C2)C1 c1(C(=O)OC2CC(C)CC(C)C2)ccc2ncn(C)c(=O)c2c1 c1(OC)cccc(C(C)CC(=O)N(CC(C)CNC(c2ncccc2F)=O)C)c1 C1(CC(=O)NCCC(C)NC(c2cn3c(n2)SCC3)=O)CC2C=CC1CC2 C(=O)(C1CCCc2ccnn21)N1C(CNC(C(C(C)C)O)=O)CCCC1 C1(NC(C(CCN(C)C)NC(C(CCOC)N(C)C)=O)=O)CC2(CCCO2)C1 C1(C(=O)NCCC(C)N(C(C(CC)NC(N)=O)=O)C)CCC2(CC2)C1 N(C1CCCc2ccc(Cl)cc21)CC(CO)CC1CCOCC1 S(=O)(=O)(c1cc(C(=O)NC2CCCC2Cn2cccn2)co1)NC C1(NC(c2c(C)ccc(C)n2)=O)CCN(CCc2cccc(O)c2)CC(C)(C)C1 CCCC(O)C(=O)NC1CN(C(=O)CN2CCOCC2)CC1C(F)F c1(NC(CNC(C2CCC(C(C)O)CC2)=O)(C)C)ncc([N+](=O)[O-])cc1F CC1(NC(C2(C)CN(C(=O)CNC=O)C2)=O)CC2CCC1C2 C1(C2CCC2)(C(=O)NC(CCCNC(c2n(CCOC)ncc2)=O)C)CC1 N1(C(c2cnc(CNC(C(C)NC=O)=O)o2)=O)CC2C(C)C2C1 CN=c1nc(NC(=O)COCC(F)(F)F)cc(C)[nH]1.c12cnc(I)c(n1)N2 C1(CNC(C(CSC)OC)=O)(CNC(C2(C(C)C)CCOCC2)=O)CC12CCC2 c1(C(C)(C)C)cc(=NCC2CC2CNC(c2cnn(C(F)F)c2)=O)[nH]cn1 N1(C(C(CC)(C)OC)=O)CC(S(=O)(=O)N2CCN(CC=C(Cl)Cl)CC2)C1 c1(C(=O)NC2CCN(C(CC(C)OC)=O)C2C(C)C)ccc(Br)c(F)c1C C#CCCCC(C)C(=O)NC(COC)C(=O)Nc1cccc(OC)c1C c1(C(N2C3CC(NC(=O)C4=CCCC4)C(C3)C2)=O)nn2cccnc2c1Cl C1(NC(=O)NC23C(C)OC(CC2)C3)C2Cc3cc(F)ccc3C12 C(=O)(C(C)(C)C(N)=O)NC(C)CN1CCN(C(C2CC2c2ccccc2)=O)CC1 c1(C(N(CCC(=O)NC(CC)C(=O)O)CC2CC2)=O)cnc(O)nc1O N1(C(CC2(CC)CCC2)=O)CCC2CN(C(=O)C(C(=O)OC(C)(C)C)OC)C2C1 CCC(C(C)C)C(C(=O)Nc1cccc(OC)c1)N(C)Cc1cccc(O)c1 C(CC(CNC(C1CCS1(=O)=O)=O)NC(C1(N2CCCC2)CC1)=O)OC C1(O)(CCNC(CCCCN(C)C)=O)CCN(C(C23CCC(CC2)O3)=O)CC1 Cc1[nH]c(=N)ccc1C=CC(N1CCC1CNC(c1cc2c([nH]1)CCCC2)=O)=O N1(C(C2(COC)CCC2)=O)CC2(CCCC(CNC(C3(F)CC=CCC3)=O)O2)C1 C=C=CC1CCCCN1C(=O)CN(CC(=O)OC(C)(C)C)C(C)=O CCCCC(F)C(=O)NCCCC(O)C(=O)NCC1CC2(CCC2)CO1 C(C(C)C(C)C(=O)NC1COCCN(C(c2cc(F)cnc2Cl)=O)C1)OC c1(OC2(C(=O)NC(C)CCCNC(c3nn[nH]c3F)=O)CC2)cccc(F)c1 c1(C(N2C(CNC(C(CCC)C)=O)C=CC2)=O)ccc([N+](=O)[O-])c(NC)c1 S(=O)(=O)(c1cnccc1N1CCn2ncc(Cl)c2C1)NCC(CO)OC Cc1ccc(CN2CCSCC2)cc1NC(c1cc(C(=O)O)co1)=O N1(C(C2N(C(=O)NC)CCC2)=O)CC2CC(NC(=O)CCCN=[N+]=[N-])C(C2)C1 C1(C)(C(=O)NCC2C(NC(C(N3C(=O)CCC3=O)C)=O)CCC2)CCN(C)CC1 c1(CNC(c2cccs2)=O)nc2c(s1)CCN(C(C1CC3C=CC1C31CC1)=O)C2 Cc1cncc(C(N2CC=CC2(C)C(=O)NCC[Si](C)(C)C)=O)n1 N1(C(C(C(C)C)O)=O)CC2CCCC(CNC(=O)CS(=O)(=O)C(C)(C)C)C2C1 N1(C(CCCC(C)C)=O)CC(NC(C2CCCS2(=O)=O)=O)C(N=[N+]=[N-])C1 C1(C)C(=O)NCCC(C)NC(=O)C(NC(C)=O)COCCN1C.C(C)(C)C CC1CCC(C(=O)NCC2CCCC2NC(=O)CCc2ncc(C(C)(C)C)o2)O1 N(C1c2ccccc2CC1NC(=O)COc1ccccn1)C(CS(C)(=O)=O)=O N1(C(Cc2c(C)ccs2)=O)CC(NC(C2CCN(CC(F)F)CC2)=O)C(O)C1 N1(C(c2cc(C)n(C)c2C)=O)CCC(C)N(C(c2cc3c(s2)COCC3)=O)CC1 CCC(C)(CNC(c1csc(C#N)c1)=O)C(=O)NCC(C)NC(C)=O C1(NC(c2cnsn2)=O)CN(C(c2ccc3nc[nH]c3n2)=O)CC1C1CC1 c12ccc(cc1)NC(=O)CO2.c1(OCC(=O)NC2CCCC2F)cccnc1 C1(C(N2CC(C)C(CNC(=O)C=CS(C)=O)C2)=O)CCOC(C)(C)C1 C12(CC(=O)NCC(N3CC(C)C3)c3cccs3)CC3CC(C1)CC(O)(C3)C2 O(N(C)C(=O)CC(C)C(C)(C)NC(C1CN(C)C1)=O)CC c1(C(N2CCC(CNC(C(CCC)OC)=O)CC2)=O)nnc(O)c(Br)c1O CCC(CO)C(=O)NCCC(C)N(C(=O)C(C)n1ccnc1)C C1(C(=O)NCCOC2(C)CCC2)CCCN(C(C2COC(=O)N2)=O)C1 C12(C(=O)NCC=C(C(=O)NCCC(C)OC)C)CC(C#N)(C1)C2 N#Cc1cc(Cl)c(NC(C2CCC(NC(=O)CC3CC3)CC2)=O)c(Cl)c1 c1(OC)cc(N)c(C(=O)NCC2CCCCN2C(C2CC3C=CC2C3)=O)cc1F c1(NC(C(CN(C(c2cccc(CC)c2)=O)CC)OC)=O)cccc(F)c1O c1(C(C)=O)ccc2c(c1)C(=O)N(C)C2=O.C123CCCC1(C2)C(=O)N3 C(=O)(C1CCc2nccn21)NC1CCCCCN(C(C(CC)(CC)CO)=O)C1 C1(NC(=NCC)NC(c2ccc(F)cc2)C2CC2)CC1C1CCCC1 C(=O)(CC(F)(F)C(F)(F)F)N1CCC(NC(C=C(C)c2cccs2)=O)CC1C C#Cc1ccccc1CC(N1CCC(C)(CCNC(=O)C(N)=O)C1)=O c1(C(=O)NCC(c2ccccc2)NC(CC=CC)=O)nn[nH]c1Cl c1(OCC)cc(NCC(CCNC(c2cc(C(N)=O)n(C)n2)=O)OC)ncn1 C1(NC(CC2N(C)CC=CC2)=O)CCCCCC1NC(c1ccc(Cl)cc1)=O c1(C(=O)NCC(C2CCCC2)NC(c2c(C)ocn2)=O)c(F)ccc2c1OCC2 CC1(C)CCCN(C(=O)CC2C=CCCC2)C1C(=O)NCc1ccc(C#N)cn1 Cc1cc(CN2CCCC(C(=O)NC(C)C(F)(F)F)C2)cnc1C Cc1nc(C(=O)N(CC(C)NC(=O)C(C)(O)C2CC2)C)sc1C c1(CC(=O)NC2CCN(CCNC(C3C(=C)C3)=O)CC2)ccc(C)c([N+](=O)[O-])c1 c1(C(=O)NC(C)C(C)(C)C(=O)NC(C2CCOCC2)CO)cc2cccnc2[nH]1 C1(C(=O)NC(CNC(=O)CCc2cnc(C)o2)CC)(COC)CCCCO1 N1(C(c2c(CNC(Cn3c(C)nnn3)=O)n[nH]c2)=O)CCC2(CCCO2)C1 C1(CN(C(CCN(C(=O)Cn2nc(C)oc2=O)CC=C)=O)C)CCCC1(C)C c1(C(=O)NC(CNC(CSCCOC)=O)CO)cscc1C#N Cc1cccc2c1OC(C(=O)NC1CN(C(C3(n4cc(C#N)cn4)CC3)=O)C1)C2 C1(C(=O)NC2CC(CNC(CCc3ccc(NC)cc3)=O)C2)CC(=O)NC(=O)N1 Cc1cc(C(=O)NCC(O)CNC(=O)C=CSc2nc[nH]n2)cnc1OC(F)F c1(C(N(CC(CC)OC)C)=O)cnn2c1CN(C(=O)C(CC(C)C)N(C)C)CC2 c1(C(N2CCC3(NC(C=CCOC)=O)C(C2)C3)=O)cc2c(OC)cccc2[nH]1 C1(CNC(C2CC2(F)F)=O)CCC12CN(C(c1ccc(-c3ccccn3)o1)=O)C2 CC1(C)CC(C(N2CCCC(CO)CC2)=O)CCN1C(=O)Cn1cc(Cl)cn1 C1(C(N(CC(C)NC(=O)COc2ccccc2)CC)=O)CCCN2CCCC12 C1(C(=O)NC(CCCNC(C2C(COC)C2)=O)(C)C)COc2cc(O)ccc2C1 c1(OC)ccc2[nH]c(C(N3CCC(NC(=O)Cc4cc[nH]n4)C(F)C3)=O)cc2c1 c1(C(=O)NCCCCC2(NC(Cn3ncc(C)c3)=O)CC2)cc(C)c(C)c(C)c1 C1(NC(C23N(C(c4cc(C)nnc4C)=O)CC(C2)C3)=O)C(C)(C)C(O)C1(C)C C12(NC(CCCc3onc(CC)n3)=O)CCN(C(c3c[nH]nc3C)=O)CC1C2 c1(C(N2CC=CC(OCC)C2)C(=O)Nc2ccccc2)c(F)cc(Cl)cc1Cl C12(C(N3CC(C)N(C(c4cnnn4C)=O)CC3)=O)C3C4C1C1C2C3C41C(N)=O c1(C(=O)OC2CC(CN)C2)cnn2c1S(=O)(=O)NCC2 C1(C(=O)NC(CC)C(C)O)CC2(CCN1C(c1ccns1)=O)CC2 C#CCCCC(C)C(=O)NC1(C)CN(C(=O)CNC(=O)CCC(C)C)C1.C1CO1 N1(C(c2c(C)coc2C2CC2)=O)CC2(C1)CN(C(C1CC1C(N)=O)=O)CCO2 C(=O)(N=c1cc(C)n(CCO)[nH]1)NC1(O)CC(NC(c2ncc(C)c(C)c2)=O)C1 C12(C(N3C4CC(CC(C(N5CCCCC5)=O)C4)C3)=O)CCCC1CS(=O)(=O)C2 C1(NC(c2ccc(C#C)o2)=O)CC2CC1N(C(c1c(Cl)cnn1C(C)C)=O)C2 c1(C(=O)NC(C(C)C)CCNC(=O)CCCn2cncn2)cc2c(s1)CCOC2 C1(NC(CCC(C)OCC)=O)CCN(C(c2cc[nH]c2C(=O)NCC)=O)CC1O C1(C(=O)Nc2cnc(OC)nc2)N(C(=O)C(O)Cn2cncn2)CCCC1(C)C c1(C(=O)NCC(C)NC(=O)C(N2C(=O)CCC2=O)C)c(N)sc2c1CCC2 C(=O)(C1OC(=O)c2ccccc21)N1C(CNC(CCC(=O)OC)=O)CC(C)(C)C1 C1(O)(CC(=O)NCC2C(C)CCN2C(c2cc(C(N)=O)[nH]n2)=O)COC(C)(C)C1 N1(C(C(C(C)(C)C)SC)=O)CCN(C(c2csc(C)c2C)=O)CC(C)C1 N1(C(C2C(=C)CCC2)=O)CCC(C2CCN(c3cc(CCC)ncn3)CC2)C1 CC1(C)COC(C)(C(=O)NC2CCN(c3ccc(C#N)nc3)CC2F)CO1 C(C)(C(CC(=O)N1CCSCC(C)C1)NC(C1COCCN1C)=O)OC C(CN1CCCC1)(C(=O)N(CC1CC1)OC)NC(C(C=C=C)C)=O C1(C(N2CC3N(C(C=COCC)=O)CC(C3)C2)=O)CCc2c(nnn2CC)C1 C#CC1(C(=O)NC(CO)CCC=C)CCN(C(c2nc(=N)cc[nH]2)=O)C1 c1(C(N2CC(OCCNC(CC3CCN(C)C3)=O)C2)=O)ccn2[nH]c(=N)nc2c1 c1(C(N2CCC(N(C(C(CC(=C)C)C)=O)C)CC2)=O)cc2c(s1)CCC(C)(C)C2 c1(Cn2c(C(C)(C)C)cc(-c3nc(C4CC4)nn3C)n2)ccc2c(c1)C(=O)OC2 N1(C(c2n(CCC)c(C)nn2)OC)CCOC(C)(CCOC)C1 C(=O)(CS(=O)(=O)c1ccccc1Cl)N(C)CC1N(C(C(CC)F)=O)CC(F)C1 c1(C(=O)NCC2CC(NC(c3n(C(C)C)nnc3)=O)C2)cc(Cl)ccc1F c1(C(=O)NCC(=C)CCNC(C2COC(=O)N2)=O)cc(Cl)cc(Cl)c1Cl N1(C(Cc2cnc(C)o2)=O)CCC(NC(c2c(C)nc(C)n2O)=O)CC1C C(=O)(N=c1cc(CCO)[nH][nH]1)c1nc(NC(c2ccc(C)c(C)n2)=O)sc1 N1(C(C2C(C)(C)C2)=O)CCC(C)(NC(=O)C=CC(=O)NCc2cccs2)C1 CN1CCN(C(=O)Cc2ccsc2Cl)CC1CNC(=O)CCCc1ccncc1 C1(OC)CC2(CCC(NS(=O)(=O)C3CC3)CC2)C1.N12CCN(CC1)CC2=O C1(CN(C)C(c2coc(Br)n2)=O)CCCN(c2cc(O)ncn2)C1 C(C(C)CCCO)NC(C(C1(O)CN(C(CC2(CCC#C)CC2)=O)C1)F)=O c1(CC)nc(=O)cc(OCCCCOC2CCC(F)(F)C2)[nH]1 c1(OC)ccc(C)c(C(=O)N(CCNC(c2ccc([N+](=O)[O-])s2)=O)CC2CC2)c1 c1(C(=O)NC(C2(O)CN(C(c3nc(C(C)OC)sc3)=O)C2)C)ccccc1Cl C1(N(C(CNC(=O)OC)=O)C)CN(C(C2(n3cccc3)CCCC2)=O)CC12CC2 S(=O)(=O)(c1ccc(Cl)c2nonc12)N1C(CC(=O)OC)COC(C(F)(F)F)C1 CC1(NC(=O)C(O)CC2CCCC2)CCCN(C(c2cnc(N(C)C)cn2)=O)C1 N1(C(c2cn(CC)nn2)=O)CCOC(C(=O)NCCc2ncccc2F)C1 N1(CC(=O)NC(CNC(c2ccnn2CC)=O)CCOCC)CCCCC1CC C(C)(CCC(=O)Nc1csnc1C)NC(C=CCCC)=O N1(CCNC(C(CC)C)=O)CCC(NC(=O)CC2CCC2(C)C)C(C)(C)C1 Cc1ccc(C=CC(N2CCC(CF)(NC(=O)CN3CCSCC3)C2)=O)cn1 c1(NC(CC2N(C(CN(CC)CC)=O)CC2)=O)ccc(F)cc1F c1(C(=O)N(c2cc(Cl)cnc2Cl)C2CC2(F)F)cc2ccc(Br)cc2s1 C1(NC(c2cccc(C(=O)OC3CC3)c2)=O)CCNCCC1c1ccccc1 Cn1nc(CNC(=O)CC2(C#N)CCC2)c2c1CCN(C(C1CS(=O)(=O)C1)=O)C2 C1(C(N2C(CNC(=O)CCc3ccc(F)cc3)C=CC2)=O)CCC2(CCC2)OC1 c1(C(=O)Nc2cccc(C(=O)Nc3c(C)cc(CC)s3)c2)cc(Cl)c(Cl)nc1Cl C1(NC(c2n[nH]c3c2CCSC3)=O)CC2CC(C1)N(C(C1CCCCS1)=O)C2 CC1CCCC(C(=O)NC(C2CN(C(c3cccc(F)c3)=O)C2)C)CC1 CC1CN(C(c2nccnc2Cl)=O)CCC1CNC(c1c(Cl)cnn1C)=O C1(NC(c2nc(CCC)oc2)=O)CC2CCC(C1F)N2C(C1CC(C)(O)C1)=O CC(C)CC(C(=O)NCC1=CCCN(C(C2CCCC(F)(F)C2)=O)C1)C(C)C c1(C(=O)NC2CN(C(C(C(C)C)(C)O)=O)C2)noc2c1CC(C)(C)CC2 N1(C(=O)CCC2CCCC2)CC2C(NC(=O)C(F)(F)c3cccnc3)C2C1 c1(NC(C(N2CCC(CCC=C)C2)=O)=O)ccc(F)cc1OC c1(CNC(C2(CC#C)CCN(C(=O)C(C3(C#N)CC3)C)C2)=O)c(F)cccc1F n1(CC(=O)NCCCNC(=O)CC2CCCCC2O)c(=O)cnc2ccccc12 C12(CC(=O)NC(C(=O)NC)(C)C)CCC1CN(C(c1ccoc1C(C)C)=O)C2 Cc1ccsc1C=CC(=O)NCC(F)CNC(=O)CNc1nnnn1C N1(C(Cn2ccc(C)n2)=O)CCCC(CNC(=O)C=CC(N2CCC(C)C2)=O)C1 N1(C(CSCC)=O)CCC2CN(C(=O)C(C)(O)CCc3ccccc3)CC12 c1(C(=O)NC(C(C(C)C)C)CNC(c2cnsc2)=O)ccc2c(c1)NS(=O)(=O)C2 c1(OC)ccc(-c2cnccc2CNC(c2ccccc2Cl)C(=O)O)c(OC)c1 CCC(C)(C#N)C(=O)NC(C)CN(C(=O)Cc1sccc1C)C(C)C N1(C(CC(C(F)(F)F)NC(c2c(OC)csc2)=O)=O)CCc2cccnc2C1 CCCCC(CCCC)C(=O)N1CC(CN2CC(C(=O)NCCC(C)SC)C2)C1 n1(CCC)cccc1C(N1CCC(CC(=O)NCC2C3COCC23)C1)=O C(CCCC(=O)NCC(c1ccc(C)cc1)NC(=O)C=C(C)C(F)F)(OC)OC c1(OCC)cccnc1C(=O)NCC1CCCN(C(C2(O)CCOC2)=O)C1 c1(OCC(=O)NC(CNC(C(C)=C2CCCC2)=O)CC(C)C)c(F)cccc1F CCCCCC(O)CC(=O)NC(C)C(C)C(=O)N1CC2(CSC2)C1 N1(C(c2cccc(N)c2Br)=O)CCC2(CCN(C(c3ccccn3)=O)CC2)C1 c1(C(=O)NCC(CC)NC(=O)C(CC)NS(C)(=O)=O)cc2cccnn2c1 N1(C(c2cc(C)nc(Cl)c2)=O)CCCC2(CCN(C(c3cn[nH]c3)=O)C2)C1 C1(C(=O)NCCNC(=O)OC)CN(C(c2ccc(C#N)cn2)=O)CCN1C C1(NC(c2ccc(-n3cc(C4CC(C)OC4=O)nn3)cc2)=O)CCS(=O)(=O)C(C)C1 C(=O)(C1=C(C)CCOC1)NCC(C(=O)N(C(C(=O)OC)C)C)O C1(CNC(C(C)OCC=C)=O)CCC2CN(C(=O)C(C#N)CC)CC12 c1(N(C)C)ccc(C(=O)NCCC2CCN(C(C3(Cl)CC3(F)F)=O)C2)cn1 CC(CC(=O)NC(C(N1CCC(CCCO)CC1)=O)c1ccoc1)CC(C)(C)C c1(N(CCCOC)C)cc(C)c(S(=O)(=O)N2CCCC(CCO)CC2)cn1 C(C(C)CC(=O)N1CCC(Oc2ncccn2)CC1)OC c1(CNCCN2CCOC(C)C2)ccccc1N.C(C(C)C)OCC C1(OCC)CCCC(NC(N2CC(N3CCNC3=O)C2)=O)C1 c1(C(=O)NC(CNC(C(COCC)(C)C)=O)CC)cc(F)c2[nH]nnc2c1 C1(CNC(CN(S(C)(=O)=O)C)=O)CN(C(c2cc3c(s2)CCC3)=O)CCC12CCC2 n1(CC)ncc2c1CC(C(N1CCC(CNC(=O)CN(C)C)C1)=O)CC2 c1(OCCCCCC)ccc(CN2CCCC2C(N2CCC3(CC3)C2)=O)cc1 c1(C(=O)NCC(C2CCN(C(=O)C=CS(C)=O)CC2)C)cc2c(=O)[nH]ccn2n1 C1(NC(C(C=CCCC)O)=O)CCCN(C(c2ccc(C(C)C)s2)=O)CC1 CCC(C)(COC)C(=O)N1CCCC(CO)(NC(c2cc(OC)no2)=O)C1 c1(C(C)=O)ccc(C(N2CCCC2CN(C)C(C(F)C2CCC2)=O)=O)o1 C(C)(C(C)(C)C(=O)NC1CCN(C(=O)CSC(C)C)CC1)NC(C)=O c1(NC(CC(CC)C2CCC2)=O)cc(C)c(Br)cn1 C1(N(C(c2cc(C)c(Cl)s2)=O)CC)CCCN(C(=O)CC(C)(C)O)C1 c1(C(=O)NC23CCCC2CN(C(=O)C2=CCCCC2)C3)nncc2c1CCCC2 c1(C(N2CCN(C(CN(C)C)=O)CC(C)(F)C2)=O)cccc2c1OC(C)(C)C2 c1(-c2nc(C(c3c(F)ccc(C)c3)C(C)C)on2)cc2c(s1)CCCC2 c1(C(=O)NCC2C(NC(C(=O)N(C)CC3CC3)=O)CC2)cocc1Br c1(C)ccnc(O)c1C.c1(CCC)nc(C)c(C(=O)N)s1.C1CC(=O)OCC(=O)N1 C1(CNC(c2ocnc2C2CC2)=O)CC2(CCN(c3nnc(O)s3)C2)CO1 Cc1cc(Br)c(C(=O)NCC(C)NC(=O)COC(C)(C)C(F)(F)F)s1 CC(C)S(=O)(=O)CC(=O)N1CCCC1C1CSCCN1Cc1ccc(Cl)cc1 C1(N=[N+]=[N-])(C(=O)NCc2c(C)cccc2F)CCN(C(=O)CC2CCOC2)C1 C(=O)(C(C)C(C)(F)F)N(C1CCN(C(CCn2c(C)ccc2C)=O)CC1)C C(C(C)C(F)C(=O)NCC1OCCC1(C)C)NC(C(CC)C#N)=O C=Cn1nncc1C(=O)NCC1(CCNC(=O)COCC2CCCC2)CC1 C(N=c1nc2sccc2c(N2CC(C#N)C3(CCC3)C2)[nH]1)CC(C(C)C)C N1(CC2(NC(Cc3nnc(C)o3)=O)CC2)CCN(C(=O)C(C)(Cl)Cl)CC1 Cc1ccc(OCC(N2CC(NC(=O)C(C(C)C)c3cnc(C)s3)C2)=O)cc1C Cn1ncc2c(NCc3cn4c(n3)SCC4)[nH]c(=NCCC3(CCO)CCC3)nc12 C(CC(O)C(F)F)NC(CCOCCNC(c1c(C)noc1)=O)=O c1(OC)ccc(S(=O)(=O)N)c(C(F)(F)F)c1.C(C(=O)O)(C1(CC(C)C)CC1)N c1(CC)ccccc1NN1CCN(C(N2CC(COC(C)(C)C)C2)=O)CC1.C S(=O)(=O)(c1cc(C(=O)OC)n(C)n1)Nc1cccc(C2C(C(=O)OC)C2)c1 Cc1ncc(C(N2CCCC2CCNC(=O)CC(O)C(C)C)=O)cc1N n1(CC)ncc(C)c1C(=O)N(CCC(N1CC2C(C1)C2(C)C)=O)C(C)C C123CCC(CC1)(CO2)C(=O)NC3.C1(C(=O)NC2C(COC)C2)CC(C(C)(C)C)C1 C1(NC(c2cc(C)sc2)=O)CCN(C(c2nsc3ccccc23)=O)CC1(C)C C(N=c1nc(N2CCN(CC3CCCO3)CC2)c2[nH]ccc2[nH]1)C1SCN=CC1 C1(C(N2CC=CC2C(=O)NCC2CCCO2)=O)C2C3CCC(C3)C12.n12cc(nn1)C2 N1(C(CC=CCC)=O)CCCC(N(C(=O)CC(C)CC)CCO)C1 c1(C(=O)OC)cnc(C)c(C)n1.C1(N(CCC(C)F)C)CCN(C(=O)CC2CC2)CC1 Cc1nn2c(C)c1C2C1CC1.c1(NCCN2CCCC2C)nnnn1CCCF c1(CCCC(=O)NC2CN(C(C3C(C)C3)=O)C2)ccc2c(c1)Cc1ccccc1-2 c1(CSCC(=O)NCCN(C(C2CCCN2N=O)=O)CC)ccc(Cl)cc1 CC(C)C1=CCC(C(=O)NCC2(NC(=O)COCc3nc[nH]n3)CCOC2)CC1 c1(N(C)Cc2cn(-c3cnccc3Cl)nn2)cccc(Br)c1Cl C1(NC(C=CC)=O)CCCN(C(=O)C(C)NC(=O)OC(C)(C)C)C1c1ccccc1 c1(N2CCC(C)(C(F)(F)F)CC2)ccc(F)c(F)c1-c1nn[nH]n1 C1(CNC(CN(C(c2ccc(C(N)=O)[nH]2)=O)CC)=O)CCCCS1 c1(C(N2C(C3(NC(COCCOC)=O)CC3)CCCC2)=O)ccc(F)cc1C N1(C(C2C(C)CC2)=O)CCN(C2CN(C(=O)Cn3ncccc3=O)C2)CC1 CC#CC1(C(=O)NC(C)CCC(=O)N2CC3C=CC3C2)CCC1 c1(C(N2C(C)CC(CNC(C3CCCC3O)=O)C2)=O)c(Cl)oc2ccccc12 C(=O)(NNc1cc(I)ccn1)NC(CC(=O)O)c1cncs1 C(=O)(C1=COCCO1)N(C1CCN(C(C=C(COC)C)=O)C1)C.C12CCC(C1)N2 c1(OC)ccc(Cl)cc1CC(=O)NCc1c(C)nn(C)c1C N12CCN(CC1)C(=O)NC1CN(C1)C(=O)C2.C1(NCCO)CCOC1 N1(C(C)=O)CC(NC(c2c[nH]nc2C2CCOC2)=O)C(C2CC2)C1 C=CCC(CC(=O)N(C1CN(C(C)C)C1)C)NC(=O)C(C)COC c1(NC(C2C(C)(C)CCN(C(C(CCC)C)=O)C2)=O)cnc2ncnn2c1N CC(C)(C)C(CNC(C12CC(CO1)C2)=O)NC(C1CN(N2CCCCC2)C1)=O C(CC(F)CN=[N+]=[N-])NC(C(C)(CO)NC(C12CC(C)(C1)C2)=O)=O c1(C(=O)NCCOC2CCN(C(C(CCC)OC)=O)CC2)cccc2c1COC2 c1(OC)cc(C)c(C(N2CC3CC2CC3CNC(c2cnoc2)=O)=O)cc1OC c1(CC2N(CC(=O)N(C(C)(C)C)CC(=O)OC(C)(C)C)CCC2)ccccc1Cl N1(C(c2c(C)nns2)=O)CCC(C)(CC(=O)NCCNC(=O)CO)C1 C1(C(=O)NC(C#C)C)CC12CCN(Cc1ncc(Cl)cc1Cl)CC2 C1(NC(C(CC)SC)=O)CC2CN(C(=O)CCC3CC(c4ccccc4)C3)CC12 c1(C(=O)Nc2c(C#N)ccc(Cl)n2)csc2c1CCOC2 C1(C(N(CCC(=O)NCCn2ncc(CC)c2)C(C)C)=O)CC2(CCO1)CC2 c1(C(N2C3C(C(=O)Nc4ncc(C)c(Cl)n4)C(C3)C2)=O)ccc2c(c1)NC(=O)C2 N1(C(CCC(=O)NC(Cc2cccc(C)c2)C(=O)O)=O)C2C=CCC1CC2 C(CCCCCC(=O)NC1CCCCC1O)NC(CCC(C)(C)OC)=O C1(CNC(c2c(CC)con2)=O)CCN(C(C2CC(OC3CC3)C2)=O)C12CCC2 Cc1cccc(N2CCC(CNC(=O)C(C)(C)N(C)C)C2)c1C C(=O)(C(F)C(C)(C)O)N1CCC(N2CCN(C)CC2)C1.C12CCCN1C2=O C(C)(C)(C(=O)NCCN(C)C(C1(O)CC(c2ccccc2)C1)=O)OC(C)C C1(C(C)C)CCCCC1CNC(=O)NC1CC(NC(=O)OC(C)(C)C)C1 c1(C(=O)NC(C)CCCNC(=O)CC2CC2)ccc([N+](=O)[O-])cn1.C1(C)C=CCCC1 C1(NC(=O)C(=Cc2cscn2)F)CCCCN(C(C2CCC23CCC3)=O)C1 C12(CNC(C=CCC)=O)CCC(CC1)N(C(=O)C(C)(Cl)Cl)C2 c1(CNC(COCCN(C)C)=O)ccccc1CNC(=O)CN(C)C(N)=O CC1CCN(C(c2nccc(C(F)F)n2)=O)C1CNC(=O)CC1CCSC1 c1(OC)ncnc(C(=O)NC2(CN(C(=O)CCOc3ccccc3)C)CC2)c1F C(c1c(C)noc1C)=CC(=O)NCC(CCOC)NC(c1cc(C(N)=O)c[nH]1)=O C1(CNC(N(C)Cc2ccc(C(F)(F)F)cc2)=O)CC2CCCCC2O1 CCC(CC(=O)N1CC(C2CC2)C(F)(C(=O)O)C1)C(C)(C)C C(=O)(C(CC(C)C)C(N)=O)NC(C(N1CC2(CC(OC)C2)C1)=O)c1ccoc1 Cc1ccc(F)c(C(=O)NC2(CNC(=O)Cc3cc(Cl)cs3)CCC2)n1 CCCCCCCCN(C)C(C1(CNC(c2cnc(C)[nH]c2=N)=O)CC1)=O c1(C(=O)Nc2cc(C(=O)O)ccc2C(F)(F)F)c[nH]c(=O)c2ccnn12 c1(C(CSCC(=O)N(CC(C)C)C(C)C)=O)ccccc1.C1(C)C(=O)N1 c1(OC)cncc(C=CC(N2CC(C)C(C)(CNC(C3(N=[N+]=[N-])CC3)=O)C2)=O)c1 c1(N(C)C)c(C(N2CC=CC(NC(c3csnn3)=O)C2)=O)cnc2ccccc12 N1(C(CSCC#C)=O)CCOCC(C)(CNC(c2nc(C)sc2CC)=O)C1 c1(CN(CC(C)C(C)C)CCOCC)cc(Br)cs1 C1(NC(C(C)Sc2ccccc2)=O)CC(F)CN(C(=O)C(C)NC=O)C1 c1(C(=O)NC(CC=CC)C(=O)NCC(C)(C)COC)cc([N+](=O)[O-])no1 Cc1cn2c(n1)CCC(C(=O)NC1COCC1NC(c1ccc([N+](=O)[O-])[nH]1)=O)C2 CC1CCCc2nc(C(=O)NCC3(CO)CN(C(=O)C(=O)NC4CC4)C3)cn21 C1(CC(=O)NCC(CC)C)CC(C)(C)CN1C(=O)C(CC)C(=O)OC Cc1[nH]nc(C(C)C)c1C(=O)NC(C)C(C(C)C)NC(C1CCCS1(=O)=O)=O C1(N(C(C)C(c2ccccc2)O)C(c2cc(C)no2)=O)C2CCC1CNC2 Cc1nnccc1C(=O)NC1COCCC1NC(c1cc[nH]c1C1CCCC1)=O c1(OC)cc(C(=O)NC(C)CC2CN(C(C3(CF)CCC3)=O)C2)ccn1 Cc1ccnc(O)c1C(=O)NCC1CCCCC1NC(c1csc(C2CC2)n1)=O CC1(C(=O)NCCN(C2CCCCC2)C(C2(C(F)F)CCCO2)=O)CCNC1=O C(=O)(CCC(=O)NC1CC(CNC(c2coc(Cl)n2)=O)C1)NCCC C(CN=C(NCc1c(F)cccc1Cl)NCC1(C)CCCCC1O)OCC N1(C(C(C)n2cncn2)=O)CCC(CNC(C2(O)CC(C)(C)C2)=O)CC1 C12(CNC(CCNC(=O)OC)=O)CC1CN(C(C13CC(F)C1C3)=O)C2 C(=O)(C1CCCc2ccnn21)NCCN(C(CC(C)P(C)(C)=O)=O)C n1(C2(C)CC2)nnnc1CC1CN(CC2CCSC2)C1 c1(N(CCNC(C=CCC)=O)CCC)cc(C(=O)NC2CC2)ncn1 c1(C(=O)OC)ccc(C(=O)N(C)CC2CN(C(c3c[nH]c(Br)c3)=O)C2)o1 C(C(C(=O)NCC1CC(F)(F)CO1)C(C)C)NC(C(COCC)C)=O Cc1scc(C(=O)N(CC(C)NC(=O)C(c2ccc(Cl)cc2)C)C)c1N CCC(CN(C)C(C1CC(NC(C2(N(C)C(C)=O)CC2)=O)C1)=O)OC c1(N(CCC(=O)N(CCC=C)C)C2CN(C(=O)CC)C2)c(F)cccc1F CCCC(O)(CCC)CC(=O)NCC(CO)NC(c1cccc(C)c1N)=O CC1(NCc2ncc(-c3ccc(Cl)cc3)n2C2CC2)CCOC1C1CC1 c1(C(=O)NCC2CC(F)(CNC(=O)Cc3ccoc3)C2)cc2cccnn2c1 c1(Cn2cc(C3CCCC3)nn2)ncc(N)o1.C1(CCCC)(C(=O)N)CCC1 c1(C(=O)NC(CN(C(=O)CS(N)(=O)=O)CC)C)ccc(-n2cccn2)c(Cl)c1 C1(CNC(C2CC(C#C)(O)C2)=O)CC2CCCC2N1C(c1ccn(C)c(=O)c1)=O c1(NC(C2C(CC(C)C)C2)=O)cc(Cl)cnn1.C12CC(F)(C1)CNC(=O)CSC2 c1(CN(C)CC2CCS(=O)CC2)nc2ccccc2[nH]1 Cc1ccc(-c2cn[nH]c2)cc1.c1(C(NOCC=O)=O)ccccc1-c1ccccc1 C1(C(=O)NCC2N(C(c3nc(C)n(C)c3)=O)CC2)CC(O)c2ccccc2O1 O=C(CCCCCF)NC1(CNC(=O)CC2CCC3CC23)CCCOCC1 C12(C(N(CC(C)(C)NC(C3COCC3C(N)=O)=O)C)=O)CCN(CC1)CC2 n1(CC)nc(C(=O)NCC(C2CCC2)NC(=O)C(=O)NC(C)C)cc1C c1(NC(=O)CCC2CCCO2)cccc(CNC(C2CC2F)=O)c1 CC1CC(C(=O)NCC2CC3CN(C(=O)C(C)CC4CCCO4)CC23)=NO1 Cn1ncc(C(N2CC(NC(=O)C=Cc3cc[nH]n3)C(O)C2)=O)c1N c1(C(=O)NCC2(NC(c3ccc(-n4ccnc4)cc3)=O)CCC2)cncc(O)c1 N1(C(C=C)=O)CCCC1(C)CNC(c1cc(C(F)(F)F)nn1CC)=O C1(CC)CCCN1CCn1cc(CN2CCNCC2)nn1 N1(C(c2cccc(COCCCOCC)c2)=O)CC2C3CCC(C(OC)C3)C2C1 c1(CC(=O)OCC(C(CC)C)OC)cc(S(=O)(=O)NC(C)C)ccc1Cl N1(C(=O)CCCN2CCCC2)CCC(CCNC(=O)C=Cc2ccoc2)C1 C(CCN=C(NCc1cccc(C(C)C)n1)N1CCC(c2cccnc2)C1)SC C(=O)(C#CC1CCCOC1)N1C(CNC(c2cc(C)c(N)cc2F)=O)CCC1 CC1(C)CCN(Cc2cc(-c3cscn3)ccc2F)CC1C(=O)O C(=O)(C1=NOC(C)(C)C1)N(C1(C(=O)NC(C(C)(C2CC2)OC)C)CC1)C c1(C(N2CC(CN(C(Cc3c(C)n[nH]c3)=O)C)C2)=O)cc(O)nc2c1CCCN2 CC(C)CCCCCC(=O)N1CCC(CCNC(C2CCC3(CCC3)OC2)=O)C1 Cc1cccc(C(N2CCC(NCc3c(Br)cnn3C)C(O)C2)=O)c1I C1(O)(N2C(=O)NC(CCSC)C2=O)C=C(c2cccnc2)CCC1 CC1(F)CCC(NC(=O)Nc2nc(Nc3ccc(F)cc3)cs2)CC1 c1(C(N(C)Cc2nnc(CC)s2)=O)cc(CNC2CC=CCC2)ccn1 c1(CC(=O)NCC2CCC(CNC(COC)=O)CC2)[nH]c2cc(C)ccc2c1C c1(NC2C3N(C(c4ccc(C)cn4)=O)CC(CC3)C2)nc(C)c([N+](=O)[O-])cc1Cl C1(C(=O)NC(c2ccoc2)=O)CC2CC2N1C(N1CSCSC1)=O CCCCCCC(CNC(=O)NC(C1CC=CCC1)CC)CC CCS(=O)CC(=O)N(C1CCCC1)CCNC(c1ccc(Cl)cc1)=O CCC(CC(=O)N(C)C(c1cccnc1)C)NC(C1CCC(F)CC1)=O N1(C(COCCC=C)=O)CCCC(O)(CNC(C2Cc3ccccc3S2)=O)CC1 N1(C(CN(CCC)C(=O)OC)=O)CCC(C(C)(C)C(=O)NCCCO)C1 N1(C(CC2CN(C(c3c(C)nn[nH]3)=O)CC2C)=O)CC2C=CC1CC2 C1(CC(=O)NCCCNC(C(C=C)c2ccccc2)=O)SC2=NCCN2C1=O CC1=NNC(=O)C1CC(=O)NCCCC1CCCCN1C(c1cccc(N)n1)=O C(=O)(C1Cc2ccccc21)NC1CC(CNC(C2(F)C(C)(C)C2(C)C)=O)C1 C(=O)(CCCCC(N)=O)NCC(CNC(c1ccc(OC)c(Cl)n1)=O)(C)F n1(CC)nncc1C(=O)NC1COCC1NC(=O)COC1CCOC1 Cc1sc(Cl)nc1C(=O)NCC#CCNC(=O)CC(O)c1ccccc1 n1(CC)cnnc1C(=O)NC(C1CC(NC(=O)CCN2CCCCC2)C1)C Cc1cn(C)nc1C(=O)NCCC1CCN(C(c2ccccc2CO)=O)CC1 C1(C)(C(=O)OC)CCN(C(C)(CNC(=O)Cn2cc(C3CC3)nn2)C2CCC2)C1 c1(C(N2CCN(CCC3CCCO3)CC2)=O)c(Cl)cnc2[nH]nc(C(F)(F)F)c12 C(C(C)(C)C#CC(=O)NC(C)Cc1ccccn1)NC(c1cc(COC)on1)=O C1(F)(CNC(C(CC)(C)O)=O)CCCN(C(=O)C(c2cncn2C)O)CC1 N1(C(c2cnc(C)s2)=O)CC=C(C(=O)NC2(C(F)F)CCCC2)C1 c1(C(=O)NC(CC(C)NC(CSCCCC)=O)C)cc(C)c(C)c2ncccc12 C1(C(N2CCN(CCCNC(C3C(C)C3C)=O)CC2)=O)CC2(C1)CC(C)(C)C2 c1(C(N2CC(F)(CNC(COCCCCC)=O)C2)=O)cnc2c(ccn2C)c1 c1(CC)ocnc1C(=O)NC(C)C(CO)NC(C1CC(N(C)C)C1)=O N(C(=NCC1CC2CCC1O2)NCc1sc(C)cc1Br)C(CC)CC CC(C)C(C)CCNC(C1CCCN1C(c1ccn(C2CC2)n1)=O)=O N1(C(C2(OC)CC2)=O)CCCC2C1CCN2c1nc(C2CCC2)ns1 Clc1cccnc1C(c1ccccc1)NCCC1COCCO1 CC1CCC(C)(C(=O)NCC2CN(C(=O)CCC=CC(C)C)CC2C)C1 CCC(C)(C)C(=O)NC1(C(=O)N(CC(O)CN(C)C)C)CSC1 Cc1cnc(C(N2CCN(C(c3cccnc3C)=O)C(C3CC3)C2)=O)c(F)c1 C1(C(C(=O)NCC(n2cc(C3CN(C(C)=O)C3)nn2)COC)C)CC2CCC1CC2 N1(C(c2n(C)c(Cl)c(Cl)c2)=O)CCOC2(C1)CN(C(c1ccc(F)cc1Cl)=O)C2 C1(C(N2C3(CNC(CCN(S(C)(=O)=O)C)=O)CC(C2)C3)=O)CCC2(CCC2)O1 c1(NC)cnncc1C(=O)NCC(C1CC1)N(C)C(c1sc(CO)nc1C)=O c1(C(N2CCCC(N(C)CC)C2)C(=O)NC)ccc(OCCO)c2oc(C)cc12 c1(NC(C2CN(Cc3cc(Br)cnc3Cl)CCC2(F)F)=O)ccc(Br)c(Cl)c1Cl c1(C(CF)NC(c2c(C(=O)OC)occ2)c2nnnn2CC2CC2)ccc(F)cc1 c1(C(N2CCN(C(C3C(=C)CC3)=O)CC2CCO)=O)ccc2c(c1)B(O)OC2 c1(OC)cc(OC)c(C(N2CCCCCC2CNC(C2(O)CCC2)=O)=O)cn1 c1(C(N2CCC(C3CCN3C(C3CCCO3)=O)C2)=O)cc2c(Cl)nccc2o1 c1(C(=O)NCCCNC(C(C(=O)OCC)OC)=O)cncc(Cl)c1C C1(NC(=O)NCc2cc(C(C)C)on2)CCC2(CC1)CNCCO2 C1(C(N(C(C)CNC(c2cc(F)c[nH]2)=O)C)=O)C2CCC1(C1CCCO1)C2 Cc1cc(N(C)CCNC(C(C)C(N2CCCCCC2)=O)=O)ccc1F CC1C(C(=O)N2CC(C)C(NC(=O)CCS(C)(=O)=O)C(C)C2)=NOC1C Cc1cnccc1C(=O)N(CC(C)NC(C1CCC(C(N)=O)CC1)=O)C c1(C(N(c2ccc(-c3cc4sccc4s3)cc2)CCC)=O)cnc(OC)c(Cl)c1 C12(C(=O)NC(C3CN(C(c4cc5cscc5s4)=O)C3)C)CCCN(CC1)C2 C1(C(=O)NC2CC(NC(c3n[nH]c4c3CSCC4)=O)C2)CCc2[nH]nc(O)c2C1 c1(OC)ccc(C(c2nnnn2C2CCCC2)NCCCCS(C)(=O)=O)c(C)c1 CCS(=O)(=O)C=CC(=O)N1CCC(C2CCCN2C(C2CC2C(C)O)=O)CC1 C(=O)(C1CCCn2cc(C)nc21)NC1(COC)CN(C(=O)C(F)C2CCCC2)C1 c1(C(N2CC(C3CN(C(c4cc(Br)cs4)=O)C3)OCC2)=O)ccc(F)c(Cl)c1 C1(C#N)(C(N2CCCC(O)(CNC(CCC(C)OC)=O)C2)=O)CCN(C)CC1 c1(C(=O)NCC2CCC2NC(=O)CCc2cccc(Cl)c2)ccc(Cl)c(F)c1 Nc1c(Cl)c(C(=O)NCC2CCC2NC(=O)C=Cc2ccco2)cc(F)c1Cl c1(C(N2C(CNC(C3CC3C(F)(F)F)=O)CCCC2)=O)ccc(F)cc1OC(F)F C1(NC(C=CC)=O)CCN(C(C2CCCC3(C2)CC3(F)F)=O)CC(C)(C)C1 C1(C(N2CC(C)C(C)C2C)=O)CC2CCC(C1)N2C(C1CCCOC1)=O c1(C(N2CCC(C)C(N(C(=O)CCc3nc[nH]n3)C)C2)=O)ccnc2cc[nH]c12 S(=O)(=O)(c1[nH]c(=NC(Cc2ccncc2)CO)ccc1Br)NCC1(C)CC1 C1(NC(C(N2CCC(C)CC2)C)=O)CCN(c2nccc(CO)n2)CCC1CO c1(CN=c2ccnc(NC3CC(C)SCC3)[nH]2)cccn2c(CO)nnc12 N1(C(C(C=C)(C)O)=O)CCC(C2(O)CC(NC(=O)CC3CCC(=O)N3)C2)CC1 C1(C(=O)NC(C(C)NC(c2[nH]cc(C(C)=O)c2)=O)(C)C)CCc2n[nH]c(C)c2C1 C1(CCC)CN(C(=O)CN(C)C(c2cccs2)=O)CCN1C(C1CSCCS1)=O C(=O)(C(C(C)(C)O)NC(=O)CC1(C)CCC1)NCc1nnn(C)n1 C(CCNC(C1C2CCC(F)C12)=O)(C(=O)N1CCC(C(C)C)CC1)OC N1(C(C=CCCC)=O)CCN2C(=O)C(NC(C3CCN(CCC)CC3)=O)CC2C1 Cc1cc(-c2ccccc2)nc(CNCN2CC(C#N)(SC3CCC(F)C3)C2)n1 C1(C(=O)NC2(C(=O)NCC(N3CCCC3)=O)C(C)(C)C2)CC2CCC2C1 N1(C(C(C)C2CCCC2)=O)CCN(C(c2ccc(C(F)(F)F)cn2)=O)CC(O)C1 c1(C(=O)NC2C=CC(CNC(C3C=CCC3)=O)C2)cc(F)cnc1O C(=O)(C1CCOc2c(F)cccc21)N(C)Cc1ccc(NC(CC=C=C)=O)cc1 c1(C(=O)NC2CCN(C(CC)=O)C2c2ccccc2)nn(C)c(=O)cc1C C(C1=NOC2CN(C(c3cnc(S)nc3)=O)CC12)NC(Cc1cn(C)nc1Cl)=O N1(C(CC2CCCC(NC(C3C(C)CC3)=O)C2)=O)CCC2(CSC2)C1 C1(NC(c2ccc(C)c(OC(F)F)c2)=O)CCN(C)C12CCCNC2 CN=c1cc(C(=O)NC2CCC(CC(C)C)C2)cc[nH]1.C12(CCC1)CCC(=O)N2 C12(CCNC(Cn3ncc(C#C)c3)=O)CCC(CC1)N(C(=O)CC=C)C2 CC(C)(C)C(CNC(=O)C=Cc1cnc[nH]1)NC(=O)CSCc1cscn1 C12(c3cn(CC(=O)NC(CC)C(=O)OC)nn3)CCC(CC1)N2C(=O)C=CCOC N12CC3(C1)CN(C3)C(=O)CCC1CCC(O1)C2=O.c1(CC)ncccc1OC N1(C(CC=CCC)=O)CCC(N(C(=O)CC2CCOC2C)CCOC)C1 C1(CNC(C2C(C(C)C)(CC)C2)=O)CCCC(CNC(c2nsnc2O)=O)C1 N1(C(C2ON=C(C)C2)=O)CC(C(=O)NCCC(C)C(F)(F)F)CCC1C C(CCCC(=O)N(C1(CC(=O)N(C)Cc2cccnn2)CC1)C)(OC)OC N1(C(CN(C(c2n(CC#C)cnn2)=O)CC)=O)CC(C)CCC1C C1(NC(c2c(CNC(=O)CC3CCOC3)cco2)=O)CCCC2(CC2)C1 n1(CCCNC(C2CCCCC2C(=O)NC2CN(CCF)C2)=O)ccccc1=O c1(C(=O)NCC(=O)Nc2ccc([N+](=O)[O-])s2)cc(F)cc(Cl)c1 C1(C(=O)OC(C#C)C)CCN(C(c2c(C)c[nH]c2C)=O)CC1.C1CO1.C1CO1 c1(C(N(CC(C)NC(CSCC#C)=O)C)=O)ccc(OCC(F)(F)F)cc1 n1(CCC)cc(C(N2CC(F)(CNC(=O)CC(C)O)C2)=O)cn1 n1(CC(=O)NCCN(C(=O)CSc2cn[nH]c2)CC2CC2)ncc2ccccc12 c1(C(N2CC(NS(CC=C)(=O)=O)C(C=C)C2)=O)ccc2nc[nH]c2n1 C12(C(=O)NCC(CNC(c3ccc[nH]3)=O)OC)CCC(C1)S(=O)(=O)CC2 C12(CNC(c3cnc(Br)s3)=O)CCC1CCN2C(c1cn(CCO)nn1)=O N1(C(c2ccc(C(C3C4(CC4)C34CC4)=O)s2)=O)CC2CC(NOC)C(C2)C1 C1(C)(C(=O)NCC23C(CN(C(c4c(C)nncc4)=O)C2)C3)CCN(C)CC1 Cc1ccnc2sc(C(=O)NC(C)CNC(c3nscc3N)=O)c(C)c12 c1(C(=O)NCC(C2CCCC2)NC(c2cscc2C(F)F)=O)ccc([N+](=O)[O-])s1 NS(=O)(=O)CCCCCCC(=O)NCC1CCNCC1F C1(C)(C(=O)NCCC2CCN(C(CNC(C(CC)C)=O)=O)C2)CC(C2CC2)=NO1 C1(CCNC(=O)C(O)Cc2cnc[nH]2)CCN(C(=O)C=Cc2ccco2)CC1 N1(c2c(C#N)cncc2)CCc2sc(C(=O)Nc3cc(Br)c(F)cc3O)cc2C1 c1(C(=O)NCC2CCCN(C(C3C=CCC3)=O)C2)c(Cl)ccc2c[nH]nc12 N1(CCOCCOC)CCC2(CC1)CN(C(=O)CCC1CC1(C)C)CC(C)O2 C1(C(=O)NC2CCCC(NC(c3c(OC)c[nH]n3)=O)C2)CCCCC(F)(F)C1 c1(C(N2C(CCNC(C(CCC)O)=O)COCC2)=O)nn(C)c(Cl)c1Br CCC(C)CCC(=O)NC1(CCC)CCCN(C(c2ncc[nH]c2=O)=O)C1 C1(CC)(NC(=O)CC2CC2)CCCN(C(c2cccc(F)c2SC)=O)C1 C(=O)(C(O)CCCNC(c1cncnc1)=O)N(CC(COC)(F)F)C C(=O)(C(CC)C(C)C)NC1(CC=C)CCN(C(c2cnc(Cl)[nH]2)=O)C1 N1(C(c2c(CC)n(CC(C)C)nc2)=O)CC(NC(C2CC(O)C2)=O)C(C)(C)C1 c1(C(C)(C)C)ccc([N+](=O)[O-])cc1NC(=O)CCCCCF CCCCCCC(C)C(=O)N1CC(C(N2CCC3(CC2)CN(C)C3)=O)C(C)C1 Cc1ccn(CC(=O)NC23CC2CN(C(=O)CC2(C)CCS(=O)(=O)N2)C3)c(=O)c1 C(=O)(C1=CNC2=NCCC2=C1)NC1(CN(C(=O)Cc2cnns2)C)CC1 c1(CC(N2CCC(N(C(CC(C)(C)OC)=O)C)C2)=O)cc(Br)ccc1C c1(C(=O)NCCC(CNC(C(C)n2ccnc2)=O)O)ccncc1C(F)(F)F C=C(C)CCCC(=O)NC1CCCC1NC(=O)Cn1nc(C)n(C)c1=O CC(C)(C)C(CNC(C1(c2ccccc2)CCOC1)=O)NC(C1(CCO)CC1)=O C1(OC)CC(c2nnnn2Cc2ccccc2)(NCc2scnc2Cl)C1 c1(OCCOC)cccc(CSc2cccc(NC(=O)OC(C)(C)C)c2)c1 CN1C2CC(CNC(=O)CCc3ccc(Cl)cc3Cl)C1CCC2 C1(NC(CCc2cc(C)sc2C)=O)CCN(C(c2coc(C(C)C)n2)=O)CC1F C1(NC(c2c(C)scc2)=O)CN(C(=O)CNC(N)=O)CC1C C=CCC(C)(CC)C(=O)N1CC(C)(OCCNC(=O)CCC(C)(F)F)C1 Cc1ccccc1C(C)CC(=O)NCCN(C(c1cnc(C2CCC2)s1)=O)C1CC1 C(CCC(=O)NCC(C)(C)OCCNC(C1CC(C)(F)C1)=O)OCCOC C1(NC(c2c(C)n(C)cc2)=O)CC=C(C(=O)NC2COCCN(C)C2)C1 N1(C(C(C)c2cccs2)=O)CC2CC1CC2NC(=O)Cn1cc(C2CC2)nn1 C1(NC(C(C)NC(CC)=O)=O)CC2CC(NC(c3noc(CC)c3C)=O)CC12 c1(C(=O)NC2COCCN(C(c3nncc(C)c3)=O)C2)cccc2oc(O)nc12 C1(CNC(=O)CO)CN(C(c2cnn3ccsc23)=O)C2(CCOCC2)C1 C1(NC(C2CCCN2C2CCCCC2)=O)CCC(N=c2[nH]nco2)CC1 c1(CC)c(C(=O)NC2CC2C(=O)Nc2cnn(CCOC)c2)ccn1C C1(CNC(c2c(C)nncc2)=O)CC2CCC1N2C(c1cccc(C)c1Br)=O C1(NC(c2cc(COC)no2)=O)CN(C(=O)C(C)=CC(C)(C)C)CC1n1ccnn1 c1(NC23C(O)CCC2C3)nc2ccccc2nc1NCCCOC(F)(F)F C1(C(=O)NCC#CCNC(=O)CCCc2ccsc2)CN2CCN1CC2 c1(C(=O)NCCC(C)(C)NC(c2n(CC)cc(Br)c2)=O)ccc(F)c(C)c1C c1(OC)cc(CN2CCC(C)(C(=O)NCc3ccccn3)C2)c(Br)cn1 O=C(C1CCCc2ccccc21)NC1CC(NCc2cn3cc(F)ccc3n2)C1 N1(C(CCOC)=O)CCC(CNC(C2CCCN2CC(C)C)=O)(OC)C1 N1(C(C(C)(C)SC)=O)CCC2CCN(C(=O)C=Cc3ccc(F)cc3)C2C1 c1(OCC)cnc(C(N2CC(C3(NC(=O)CC4CC(C)(C)C4)CC3)C2)=O)c(Cl)c1 N1(C(C(CCC)NCC)=O)CC2CCC2(C(C(=O)C=CCOC(C)(C)C)=O)C1 C1(C(=O)NC(CNC(c2cn(CC)nc2OC)=O)C2CC2)CC(C2CC2)=NO1 CCCCCCC(C)C(=O)N1CC2CCCN(C(C3CCCC(F)(F)C3)=O)C2C1 C1(C(N(CCOCCC(=O)N(C)CC2(C)CCCO2)C)=O)C2CCCC(=O)C12 c1(C(=O)NC(CC(C)NC(c2cccc(CC)n2)=O)C)ccc(C)c(Cl)c1N c1(C(=O)NC(CC)CNC(c2cnnc(Cl)c2)=O)ccc2oc(O)nc2n1 C1(NC(c2ccnc(C3CCC3)c2)=O)CCCC(NC(C2CC=CC2)=O)C1 C(=O)(C(C)N=c1cncc[nH]1)N1CC2CN(C(C(CC=C)(C)C)=O)CC2C1 N1(C(CC=C)=O)CCCCC1C1CCCN1C(c1cc(OC)ccc1N)=O c1(C(=O)NCCN(C(=O)C(c2ccccc2Cl)OC)CC)cn(C(F)F)c(C)n1 C=Cc1cncc(C(=O)NCc2cc(C(N3CC(n4cccn4)C3)=O)n(C)n2)c1 C(=O)(CN1C(=O)CCc2ccccc21)NCC1N(C(CN=S(C)(C)=O)=O)CCC1 C1(C(N(CC(=O)N(C)C)CC)=O)CC(NC(=O)C(C)c2cccs2)C1 c1(SC)ncc(N)c(C(=O)NCC(C)(C)CNC(=O)CNS(=O)(=O)C2CC2)n1 c1(C(=O)NCC(CC)NC(C2CC2C(F)F)=O)sc2ccccc2c1CC(N)=O c1(CC)cccc(C(=O)NC2CC(NC(c3c(C)cnn3C)=O)C2)c1 C12(NC(C3C(CCC)C3)=O)CC1CCC2CCn1cc(CCC)nn1 c1(CC(N2CCC(CNC(CCCC#C)=O)C(O)C2)=O)ccc(O)c([N+](=O)[O-])c1 c1(CN2CC(CC(=O)NCCOCC)OCC2)cccc(-c2noc(C)n2)c1 N1(C(CCC=C)=O)CCOC(CCNC(C2(C)CC(C)=N2)=O)C1 CN1CC=C(C(=O)NCC2CN(C(=O)CCNc3ccccn3)CCO2)C1 c1(C(=O)NC(C2CCN(C(C(C)SC)=O)C2)(C)C)nnn(C)c1C(F)F C1(C(=O)NC2C3CC2N(CC)C3)CC2(C1)CC(O)C2.C12CC3(C1)CC3C(=O)N2 C(CC(C)(C)C(=O)NC1CCC(CCNC(c2nn(C)cc2C(=O)OC)=O)C1)SC C(=O)(C1=NN2CCCN=C2N1)N1CC(O)(CNC(Cc2cc(C)cc(C)c2)=O)C1 C1(C(C)(C)C)(CO)CCN(C(=NCC2CCCC23CCOCC3)NC2CCCC2)C1 c1(C(=O)NCCCC(C)NC(c2c(C)n(C)nc2Cl)=O)cc2cc(Cl)sc2[nH]1 CP(C)(=O)C(O)C(=O)N1CC(CNC(c2cccnc2C(=O)N(C)C)=O)C(O)C1 O=C(NNc1cc(Br)ccn1)NCCC1CC2CCC1C2 c1(OCC)cccc(C(=O)NCC2CC2CNC(c2cc[nH]n2)=O)c1N C(C(C)(C)CC(=O)N1CCCC(F)C1)NC(C(c1ccn(C)n1)(C)C)=O C1(C(N(CCCN(C)C)C)=O)CC2(CC2)CN1C(=O)C(C(C)(C)C)OC(C)(C)C c1(C(=O)NCCN(C(=O)CC(=O)NC2CC2)CCC)ccc(C2CC2)o1 N1(C(Cn2nc(C)c(Cl)c2)=O)CCC(NC(C2CC(F)(F)C2)=O)C12CC2 C1(C(N(C2CCN(C(C3CCCCO3)=O)C2)CC)=O)C2CCC(C2)C1C Nc1cnc(Cl)cc1C(N1CC(CNC(c2ccc(F)cc2Cl)=O)C(F)(F)C1)=O C12(C(NOCC(=C)Cl)=O)CCC(CC1NC(C1(C#N)CCOC1)=O)C2 C=CC(O)C(=O)N1CC(CNC(C2CCCN2C(=O)OCC)=O)C1 c1(CC)noc(C)c1CNC(C1C2CN(C(c3cc(=N)[nH][nH]3)=O)CC12)=O n1(CC)ncc(C(N2CCC2C2CCC2)C(=O)NCC2CCOC2)n1 c1(C(=O)NCC(CNC(C2C(CC)C2)=O)OC)cccc(C2CC2(F)F)c1 c1(C(=O)NCCCN(C)C(C2(CO)CC2)=O)cc(C(F)F)nn1C c1(C(=O)NCC23C(CN(C(CC=C=C)=O)C2)CCCC3)ccnc(S(N)(=O)=O)c1 CCCC(C)(O)CC(=O)N1CCC(NC(c2ccnn2CC(F)(F)F)=O)C(O)C1 Cc1cnccc1C(=O)NCCC1CCCN(C(=O)CNc2ncccn2)C1 Cc1c(C(N2CCCC(C(N3CC(O)CC3CO)=O)C2)=O)cnn1C c1(-c2c(C(=O)NC)nccc2)ccc(S(=O)(=O)N2CCC23CCCCC3)cc1 CC1CC2CN(C(=O)Nc3ccc(Cl)c(I)c3)CCN2C1=O C1(C(N(C)CCN(C)C(C2(C(F)(F)F)CNC(=O)C2)=O)=O)CCCC(C)(C)O1 C12CCCN(C)C1c1cn2nn1.CCCCCN(C)CC.C1(=O)CCN1 CC(C)C(F)(CNC(=O)C(C)S(C)(=O)=O)C(=O)N1CC(c2nncs2)C1 c1(NC(c2ccc(C)cc2)C)ncnc(NC(C2CSC2)C2CCC2)c1C c1(C(=O)NCC(CN(C)CC2CC2)O)sc(NC2CC2c2cccnc2)cc1C CC(C)C(C)C(CNC(=O)C(C1CC1)C1CC1)NC(c1cccc(F)c1CO)=O c1(-c2cn(C)nc2)ccccc1C(c1ccccc1)NCc1ccsc1Cl Cc1nc(C#N)ccc1C(=O)OC1Cc2cccnc2C1 Cc1cc(C(=O)NC2CCC(C(=O)NCC3CC4CC4C3)CC2)cc([N+](=O)[O-])c1 c1(C(=O)OCC)cc(NC(=O)C(N)CSC2CCCCC2COC)n(C)n1 c1(C(=O)NC2CC(C)(NC(C=C(CC)C)=O)C2)cc(N(C)C)c2ccccc2n1 C(=O)(C(F)(F)C(F)(F)C(F)F)N1C2C(NC(=O)CSc3cncnc3)CC(C2)C1 c1(C(=O)NCC(CO)NC(C2C(C(=O)OC)C2)=O)cc2c(C)cc(Cl)cc2[nH]1 C(=O)(C1=NN(C)C(=O)CC1)NCCC1OCCN(C(c2onc(C)c2C)=O)C1 C12(C(=O)NCCC3(COC)CCC3)CCC1CN(C(=O)C(F)(F)C1CCCC1)C2 N1(C(C)=O)CCCCC1CC(=O)NC(C)(C)CCNC(C1CC(CF)C1)=O C1(N(C(C(C)CC2CCCC2)=O)C)CCCN(C(C23CC(C#N)(C2)C3)=O)C1 c1(-c2cc(C)cc(C)c2)ccc2c(c1)CCN(C(=O)CNC(N)=O)C2 C#CCCCCCC(=O)N1CCC2CN(C(C3CCCCCCCC3)=O)C2C1 N1(C(CCn2c(C)cc(C)n2)=O)CCC(CO)C(NC(c2cnc(S)n2C)=O)C1 N1(CCC(C(C)N)=O)CCc2c(C(N)=O)cccc2C1 C12(NC(c3cc(O)ncc3Br)=O)CCC(CC1)N(C(=O)C(c1ccccc1)O)C2 c1(CN(C2C3CCCC23)C(c2cccc(C)n2)=O)oc2ccccc2c1C Cc1nn(C)c(Cl)c1C(c1nnnn1C1CCC1)NCC1COC1 C(CCCC(OC)OC)(C(=O)NC(C)CCCCO)NC(C(CSC)OC)=O Cc1cnn2cc(C(=O)NC3CCCC4CN(C(c5cnn[nH]5)=O)CC34)cnc12 N1(C(CSCC(C)C)=O)CCC2CN(C(c3ccc(Br)cn3)=O)CC2C1 C(CCCN=c1[nH]c(=NCc2ncc(-c3ccccc3)o2)c2ccccc2[nH]1)OC C1(OC)CC(C(N2C(CC)C=CC2)=O)N(C(c2cc(C#N)c[nH]2)=O)C1 C(CCCCC(=O)NC1CCN(C(=O)CCS(C)=O)C1)=CC C1(N(C)C(C2CCCCC2)=O)CC2CCC(C1)N2C(=O)C(=O)CC1CCCO1 c1(C(=O)NCC(CC)NC(=O)CN(C)CC)cc(=O)c2ccc(O)cc2o1 c1(C(NOCCOC)=O)coc2c1CN(C(=O)COc1ccsn1)C2 c1(C(=O)NCCCCN(C(=O)CCCC2(C)N=N2)C)cnn2ccncc12 N1(C(C(=O)NC2CCCC(C)C2C)=O)CCNC(=O)CC12CCC2 C12(CC(N3C(Cn4cc(NC(c5ccoc5Cl)=O)nn4)CCC3)=O)CCC(CC1)C2 c1(C(C(=O)NCc2nnn(C)n2)N(CCCN(C)C)C)cc(Cl)ncc1Br N1(C(=O)C(F)C2CCC2)CCC(C2CC2)C1C(=O)NCc1ncnn1C1CC1 CCC(C(=O)NCC1CC2(C1)CN(C(=O)CC(C)=C(C)C)C2)C(C)O c1(OCC)cc(S(=O)(=O)NC(C)CCN2CCN(C)CC2)ccc1C(N)=O C1(C(N2CCC(CC(N)=O)CC2)=O)CCN(C(=O)C=CCc2ccccc2)O1 c1(C(=O)NC)cc(F)c(NCc2csc(C(=O)OC)c2)c(F)c1 N1(C(CN2C(C)CC2)=O)CC2C(CNC(=O)C=Cc3ccc(C(N)=O)o3)C2C1 Cc1nc2cc(C(=O)NC3CCN(C(c4ncccc4C)=O)C(C)C3)cnc2[nH]1 CCS(=O)(=O)C=CC(=O)NCCCCC1CN(c2ncc(C#N)cc2F)C1 c1(OC)ccnc(CN2CCN(c3cc(NCCNC(C)=O)ncn3)CC2)n1 n1(CC(=O)N(C(C)CC(=O)NC(C2(CO)CC2)C)C)c(O)nnc1O c1(C(N2CCC(C(C)NC(COC)=O)C2)=O)cc(N(C)C(C)=O)ccc1Cl N1(C(c2scc(COC)c2)=O)CCC(CCN(C)C(C2(F)CCOC2C)=O)CC1 c1(C(N(C2CN(C(C3(C)CC3F)=O)C2)C)=O)cc2oc(Br)cc2[nH]1 c1(N2CCC(CCOC)(NC(C(CC)n3ccnc3)=O)C2)nc2cccnc2s1 c1(C(C2CCCC2)NCC(c2nncn2C)C)nnnn1C1CC(F)(F)C1 Cc1nc2c(C(=O)NC(C)CC(C)NC(=O)CCC(C)C)ccnc2[nH]1 CC(C)C(O)C(=O)NCc1nc(CNC(C2CCCN(C)C2)=O)cs1 Cc1cc(C(N2CCCC3C2CCN3C(=O)C(C)C(C)C)=O)c(N)c([N+](=O)[O-])c1 C(CCCCC(=O)NC1C2CC1N(C(c1cnc(C)cn1)=O)C2)NC(C)=O C(=O)(C(F)Cc1ccccc1)N1CC(C(C(=O)NCCCO)O)C1 N1(C(c2c(C)nsc2Br)=O)CCC2(C1)CN(C(=O)COCCCF)C2 c1(OCC)cc(N2CCCCCC2CNC(C2CC3CC3C2)=O)ncn1 C1(CNC(C(CCOC)C)=O)CCCN(C(c2ncn(CC(F)(F)F)n2)=O)CC1 c1(CC)onc(C(N2CC3C(CC(=O)N(CC(O)CN(C)C)C)C3C2)=O)c1C C(=O)(C#CC1CCCCC1)N1CC(NC(CCCCCCC)=O)C2(C1)CCC2 N1(C(c2c(C)nc(C)o2)=O)CCC(C(=O)NCC2CCN(C(N)=O)C2)CC1(C)C C1(NC(C(C)OCC2CC2)=O)CCCC12CN(C(=O)C(F)=C1CCC1)C2 N1(C(C(C)OCCC=C)=O)CC2(C1)C(NC(C1CC3CC3C1)=O)CCS2(=O)=O c1(C(=O)NCC(CC)(C)NC(c2ccc(CN(C)C)o2)=O)cnccc1Cl C1(C(=O)NCCn2c(CC)ncc2)CCN(C(=O)C(C)C2CCC2)C12CC2 c1(CNC(=O)NC2C3CCCC23)ccnc(-c2ccccc2)n1 N1(C(CC2(C=C)CN(C(=O)CC3CC4(CC4)CO3)C2)=O)CCCN(CC)C(=O)C1 c1(OCC(=O)N(CCCCCNC(=O)C(C2CC2)C2CC2)C)cccc(F)n1 C1(CN(C(=O)CC2COCCN2C)CC)CCN(C(c2snnc2C)=O)CC1 C1(C(C)C)CN(C(C23COC(CF)(C2)C3)=O)CCN1C(=O)CCn1cccc1 N1(C(C=NOC)=O)CC(O)CC1C(=O)NCC1(O)CCCC1 N1(CC(=O)NCC(CC=C)NC(=O)C(CCC)NC(C)=O)CCC(CC)CC1 c1(OCC)cccc(C(=O)NC2CC(O)CN(C(=O)CCCF)C2)c1N c1(C(=O)NC2(CNC(c3cn(CC=C)nc3)=O)CCC2)cccc2[nH]ncc12 N1(C(C2CCC(NC(c3nc(C)sc3)=O)C2)=O)CCN2CCCC2C1 c1(C(=O)NC(C(C)NC(c2sccc2Cl)=O)(C)C)ccc(N)c(F)n1 C1(C(C)C)CN(C(c2cnn(C)c2)=O)CCCN1C(c1cnc(O)c(F)c1)=O C1(NC(C2OCCN(C(C)C)C2)=O)CCN(C(C2CC3(CCC3)C2)=O)CC1O c1(C(=O)O)ccnc(CC(=O)N(O)Cc2cn(C3CCC3)nn2)c1 C1(NC(C(C(C)C)C)=O)CN(C(C2(c3ccccc3F)CCC2)=O)CC1(C)C C1(OC)CN(C(C2(S(N)(=O)=O)CC2)=O)CC1NC(c1coc(C)n1)=O c1(C(=O)NCC(=C)CCNC(C2(C)CCOC2)=O)cc(Br)cc(Cl)c1F C1(NC(c2cncc(N(C)C)c2)=O)CC1C1CCN(C(c2scnc2Cl)=O)CC1 C(=O)(C(C(=O)NC1(C(=O)NC(c2ncc[nH]2)C)CCN(C)C1)OC)OCC C1(CNC(C(C(C)(C)C)OC)=O)CC2CCC(C1)N2C(=O)C(C)(C)c1cncs1 N1(C(c2cccc(CC)c2)=O)CCC(CNC(=O)Cn2ccccc2=O)C(C)C1 CCC(CC(=O)N1CCN(C(=O)Cc2cnns2)CC1C(C)C)CC(F)(F)F C12(NC(C(c3cccc(Cl)c3)CC)=O)CCCC1N(C(=O)CCC(N)=O)CC2 N1(C(CC(C)c2ccccc2)=O)CCc2c(-c3cn(-c4cc(F)cc(F)c4)nn3)cccc2C1 N1(C(C(=O)NCCOc2cc(Cl)cc(Cl)c2)=O)CCC(O)C(CO)C1 c1(C(N2C3CN(C(C(C)=CC4CC4)=O)CC2C3)=O)cc(C)cc([N+](=O)[O-])c1 c1(NC(C2C(C(=O)OC)C2)=O)cc(Cl)ccc1CNC(=O)Cc1ccon1 c1(N2CC(C)SC(C)C2)ccc(S(=O)(=O)N2CCC3(CC(F)C3)C2)cc1 C1(C(=O)NC2C(NC(CNC(=O)COC(C)=O)=O)C2)(CC)CCNC1=O Cc1ccc(-n2c(C)cc(C(=O)C(=O)N(C3CCC4(CC3)CC4)C)c2C)c(C)c1 CCCCCC(O)CC(=O)N1CCC(CCCCC(N2CCOC(CC)CC2)=O)C1 C1(C)(CCN(C)CCNC(C2(C(=O)Nc3ccccc3)CC2)=O)CCCC1N CCC(C)CCCCC(=O)N(CC(=O)NCC(F)(F)C(F)F)C c1(SC)cc(C(=O)N(CCCn2cc(CC3CCC(C)(C)C3)nn2)C)ccc1F c1(C(=O)NC(C)CCCNC(c2ccoc2)=O)ccnc2ccccc12 C1(C(=O)NC2C(C)(C(F)F)C2)(NC(c2ccc(CCF)cc2)=O)CC(F)(F)C1 c1(CC(=O)Nc2cc(C)nn2C)cnn2c1CCCC2 Cc1ccc(C(N2CC(NC(=O)C(C)(C)c3cnc[nH]3)CC(C)C2)=O)c(O)c1C C1(C(=O)NCCN(CC(C)O)C(c2ccc(Cl)[nH]2)=O)CCCCC1 N1(C(C2C(C=C)C2)=O)CC(NC(=O)C(c2ccc(CC)cc2)(F)F)CC1(C)C c1(C(=O)NCC2N(C(c3c(OC)ccs3)=O)CCOC2)cccc(C)c1Cl C1(NC(C2C(C(=O)OC)C=C2)=O)CC(C)CN(C(C2CC3CCC(C2)S3)=O)C1 c1(CC(=O)NCCN(C(=O)CCn2cc(C)cn2)CC)cc(C(=O)OC)no1 c1(CCC(=O)N(CC(C)NC(=O)CC2CCC(C)CO2)C)ccc(Br)cc1 C(=O)(C(C)(C)C1=CCS(=O)(=O)CC1)NCCNC(c1c(C)cc(CC)o1)=O c1(C(=O)NC(C(=O)OCC)(C)C)c(CNC(=O)CC2CCOCC2)nnn1C c1(C(=O)NCC(c2ccccc2)N(C(C=C(C)C2CC2)=O)C)ccnnc1O CC1CN(C(=O)C=Cc2cccc(Cl)c2)CCCN1C(=O)C(CO)N(C)C N1(C(CC2ON=C(C)C2)=O)CCC2(CCN(C(C34CCC(C3)C4)=O)C2)C1 N1(C(=O)Cc2cncnc2)CC2CCCC(C1)N2C(c1ccc(Br)cc1CO)=O C1(CNC(C(CC)Sc2ccccc2)=O)CCN(C(C2(CCO)CC2)=O)CC1 c1(C(N(C2CCc3[nH]c(=N)sc3C2)CCC)=O)cnc2c(c1)c(O)nc(=O)n2C N1(C(C=CC(C)C)=O)CC(C2CCCN(C(=O)C(C)OCC3CCCO3)C2)C1 C(N=c1nn[nH]n1C)C1(F)CC(NC(C(C)C2CC2)=O)C1 N1(C(c2c(C)c(=O)cc[nH]2)=O)CCC(C)(C)CC1C(=O)NCC1=CCCN(C)C1 N1(C(C(C)=C(C)C)=O)CCN(C(c2cc(C)[nH]n2)=O)CC1c1nccn1C c1(C(N(C)CC2CCN(C(CC(CC)SC)=O)C2)=O)ccc2ncccc2n1 N1(C(C(COC)(F)F)=O)CC2CC(NC(=O)Cn3nc(C)cc3C)C(C2)C1 c1(C(=O)NCC(CO)NC(C2(OCC)CCCC2)=O)cccc2c1NCCC2 CN1C(=O)CCCC1CNC(=O)CC1COCCN1C(C1(F)CCCC1)=O N1(CCOCC)CC(C(=O)N(C)CCN(C)C(c2sccc2C)=O)CC1=O C1(CCn2cc(C3OCCC(C)C3)nn2)COc2ccccc2O1 c1(C(=O)NC2C(OC)CN(C(=O)C(O)CC(N)=O)C2)cccc2ncnc(O)c12 c1(C(N2CC(CNC(C3(OC)CCCOC3)=O)C(C)C2)=O)ccc(C)c(F)c1N C(=O)(CCC(=O)N(C1C(C)(C)C1(C)C)CCC)N(C1CCN(C(C)=O)C1)CCC C(=O)(C1=CCS(=O)(=O)C1)N1CCC(COC)(NC(=O)CCCN(C)C)C1 C(CC)(C(=O)NC(C)C(CO)NC(c1ccc(C2CC2)s1)=O)=CC C(=O)(C(O)C(F)(F)F)N1CCN(NC(C(C)(C)O)C2CCCC2)CC1.c12cn(nn1)C2 C1(CCNC(Cc2nc(C)oc2)=O)CSCCN1C(c1cc(CO)c(C)o1)=O c1(N2CC(OC)C(C)(C)C2)nc2c(c(=NCC34CCN(CC3)CC4)[nH]1)CCC2 CC(C)C(C(=O)NC(CCC1CC1)C(=O)NC1CC12CC(O)C2)n1ccnc1 Cc1cc(CNC(C2(c3ccc(Cl)cc3)CC(N)C2)=O)c2c(n1)CCCC2 c1(CC)ncc(Br)cc1C(=O)NCC1CCN1C(c1ccc(O)cn1)=O c1(C(N2CC(NC(c3cnc(N(C)C)o3)=O)CC2(C)C)=O)cc(F)c(F)c(F)c1 c1(C(N2C(CCCC)CN(C(C3CCC3)=O)CC2)=O)ccc2[nH]ccc2c1 C(=O)(C1=CCC(NC(=O)C(c2cccnc2)O)C1)N1CC2C(COC)C2C1 c1(C(N2CC(O)(C(C)NC(=O)CC3CCCCC3O)C2)=O)cnc2ccoc2c1 N1(C(c2ccc(NC)cc2)=O)CCC(C)(NC(=O)C(O)CC2CC2)CC1 CC1CCCCC1CNC(C1CN(C(=O)C(c2ccccc2F)(F)F)CCO1)=O C(CN=c1[nH]cnc(Cl)c1CO)(C1CC1)NC(Cc1c(SC)cccc1)=O c1(C(=O)NCC(CO)NC(c2cn(C)nn2)=O)cccc2c1CCCC2=O c1(CNC(C(CCCC#C)N2CCOCC2)=O)sc(S(N)(=O)=O)c(OC)c1OC C1(NC(CC(C)(F)F)=O)CC2(C1)CN(C(c1nc(-c3ccccc3)ncc1Cl)=O)C2 C(CC(=O)N1CC(C)CC(O)C1)(C(F)(F)F)NC(C(CCC)C)=O CC(CN1CCCCC1)CN=c1cc(CN2CCNC(=O)C2)nc[nH]1 C=C(C)C1OCCC1C(=O)NCCCCC1CN(C(c2cc(C(N)=O)cn2C)=O)C1 N1(C(c2occ(C(C)=O)c2)=O)CCC(O)(C2(NC(c3ccsc3C)=O)CC2)CC1 CCC(CC)(C(=O)N(C)CCOCCNC(C1CC2CCCC2C1)=O)OC c1(OCCC)ccc(C(C)NC(=O)C(=O)Nc2cc(O)n[nH]2)cc1 Cc1cccc(C)c1NC(=O)C(C(C)C1CCCC1)N(CCCCO)C CCC(F)C(=O)NCC(C)(C1CC1)NC(=O)C(C)(C)C1CCCCC1 CCC(CC(=O)NC1CCCC1N(C(=O)CCc1cnn[nH]1)C)OC c1(C(=O)NCCN(C(c2ccsn2)=O)CC2CC2)ccc(O)c(F)c1 N1(Cc2c(C)onc2)CCC2(CC1)CC2(C)C(N1CCNC(=O)C1)=O N1(C(c2c(C)ncs2)=O)CC2CC1CCN2C(c1cc(CO)on1)=O c1(C(=O)NC2C(OC)CN(C(=O)Cn3cnc(C#N)n3)C2)ccc(S(N)(=O)=O)o1 C(C)(C)(C(=O)NCC1(F)CN(C(C2(C)CCCO2)=O)C1)OC(C)=O C(=O)(CCCCCC(=O)NC(CCSC)C(=O)NCc1nccn1C)OC c1(C(=O)NC2C=CC(C(=O)NCc3c(C)nn[nH]3)C2)c[nH]c2cnccc12 N1(C(=O)C#CC2CC2)CC(CO)C2(CCN(C(C3CCC3)=O)CC2)C1 Cc1nc(C2CC2)sc1C(=O)NC12CC(C1)N(C(C1(C)COC(=O)C1)=O)C2 Cc1ccn(CC(=O)NCCC2(O)CN(C(=O)Cn3cccc3)C2)c(=O)c1 C12(NC(C(CCC#C)O)=O)CC(C)(C1)OC21CN(C(=O)C(CC)N(C)C)C1 OC1CCNCCC1NCc1ccccc1.c12nccc(n1)C2 Cc1ccc(C2CC2C(=O)Nc2ccc(C(=O)Nc3nc(Br)cn3C)nc2)cc1C C(C1COCc2ccccc21)NC(=NCC=C)NC1CC(OC(F)F)C1 c1(C(N(C(C(=O)NCC(C)(C2CC2)OC)C)C)=O)cc2cc[nH]c2cn1 N1(C(C2(OC)CC2)=O)CCCC2(CC(NC(c3ccnc(C(C)C)n3)=O)CO2)C1 C(=O)(C(C)(F)C(=O)NC1CCC(CNC(c2scnc2C(F)(F)F)=O)C1)OC C1(NC(=O)C(C2CC(F)(F)C2)O)C2CC1CN(C(c1c[nH]c(=O)cn1)=O)C2 N1(C(C=CCOC)=O)CCC2CCN(C(=O)C(C3CCOCC3)C)C2C1 C(=O)(C(CCC(C)C)NC(=O)CC(C)C(C)C)NCc1c(C)ncs1 C1(C(=O)NC2(CNC(=O)C(C)Cn3ccnc3)CC(OC)C2)CCCCCCC1 c1(N(C)CC2(NC(C3(C)CC(C)C3)=O)CC2)ccccc1C.C12COCC1C(=O)N2 c1(C(=O)NCCN(C(=O)C=Cc2ccoc2)CCC)cccc2c1nnn2C N1(C(C(C)OCCOCC)=O)CCC(C)(CNC(C2CC3CC2C2CC32)=O)CC1 C(CC(C)C(F)F)NC(C1C(CNC(c2c(C)snn2)=O)OCC1)=O c1(C(=O)NC(CC=C)CNC(C2(CO)CCCO2)=O)nnn(C2CC2)c1CCC C(C(C)(C(=O)NCC(O)(CO)CO)NC(=O)Cn1cnnc1)SC N1(C(c2c(CCNC(C(C)=C3CCCC3)=O)n[nH]c2)=O)CCC(CC2CC2)CC1 c1(C(N2CCC(F)(CNC(C=C(COC)C)=O)CC2)=O)cc2c(s1)CCC(C)C2 C(=O)(C(C)(C)CSC)NCC(CCC)NC(c1cnn(C(C)C)c1F)=O n1(CC)ncc(C)c1C(C(=O)NC(C)C)N(CC(=O)OC)C Fc1cc(Cl)c(Cl)cc1CC(c1cn(C2CC2)cn1)c1nnnn1CCN C1(CCNC(COCCSC)=O)CN(C(=O)C=C2CCN(C)CC2)CCCO1 CCCCCCC(=O)NCC(C)CNC(c1ccc(F)cc1NS(C)(=O)=O)=O C1(CC(=O)NCC(CNC(c2n(C(CC)CC)ncc2)=O)C)CCCC2(CC2)C1 c1(OC)c(C(=O)OC)nnn1CC(C)CC(=O)O N1(C(C(C(C)O)C2CCC2)=O)CC2CN(Cc3cn[nH]c3)C2C1 c1(C(N2CC(OCC)C(CNC(C3(F)CC3C)=O)C2)=O)ccc([N+](=O)[O-])c(Cl)c1 C1(C(=O)NCC2(CN(C(CSCCCC)=O)C)CC2)CCCCC1OC c1(C(=O)NCC(C)NC(=O)CS(=O)(=O)N(C)C)cncn(C)c1=O c1(COC(c2cc(F)c3cn[nH]c3c2)=O)ccc2nc(Cl)sc2c1 c1(CC(=O)NCC2C(CNC(C(CC=CC)C)=O)C2(F)F)ccc(NC)c(C)c1 c1(C(N(CC(C)NC(C2(O)CCSC2)=O)C)=O)ncc2[nH]ncc2n1 c1(C(=O)NCC(CC)(C)NC(c2csc(C)c2)=O)cn2c(n1)C(C)CCC2 C1(CNC(C=CCOCCOC)=O)CCCN(C(=O)CCc2cncn2C)C1 c1(C(=O)NCCCCC(C)NC(c2nc(OC)c(C)s2)=O)cc(N)c(O)c(F)c1 c1(C(=O)NC2CCN(C(C3CCNC3=O)=O)CC2F)nc2ccccc2[nH]1 C(=O)(C(C)CCCC(C)C)NCC1(OC)CN(C(C2(C)CCCO2)=O)C1 C(CNC(C1CCCN(C)C1)=O)(CC(=O)NCc1c[nH]nc1C(C)C)OC N1(C(CC(CCC)CC)=O)CCC2(CCCN2C(c2nn(C)c(C)c2N)=O)C1 O=C(CC(F)(F)Br)NCC1CN(C(=O)CC2CCOCC2)CC1O c1(C(=O)NCC#CC(=O)N(C)Cc2n(CC)cnn2)ccnnc1C CCC(C)CCC(=O)N1CC2CC(NC(c3cnn(C)c3C(F)(F)F)=O)C1C2 c1(C(=O)NC2C(CNC(C=Cc3ccc(C)s3)=O)CC2)cnc2[nH]cnc2c1 c1(C(C(N2CC(CCNC(CCCCOC)=O)C(C)C2)=O)=O)ccc(F)c(Cl)c1 c1(C(N(C2CCCN(C(=O)CNC(c3cccs3)=O)C2)CC)=O)cncnc1C C(=O)(CC1COc2cc(O)ccc21)N(CCNC(C(CC)(C)O)=O)C(C)C C1(C)(CC)CC(NC(C)=O)CN1C(=O)CCc1ccncc1 C12(C(=O)NCCNC(CCC3(C#N)CCC3)=O)CCCC(=O)N1CCC2 c1(C(=O)NC2CC(N(C(=O)CN3CCOCC3)C)C2)cc(N)c(Br)c(F)c1 n1(CC(=O)NC2CN(C(C3CCC3)=O)CC2CO)sc2ccccc2c1=O C1(C(N2C3(CNC(c4cc(C(F)(F)F)no4)=O)CC(C2)C3)=O)CCCNS1(=O)=O CC1CN(C(c2ccc(CN(C)C)[nH]2)=O)CCC1NC(=O)C(O)C1CC1 C1(C(=O)Nc2ncc(C#N)s2)CN(Cc2cccc(-n3cccn3)n2)CCC1O c1(C(N(C2CN(C(C3(COCC)COC3)=O)C2)C)=O)cc2ccccc2n1C Cc1ccc(C(=O)NCC2(C)CCCN2C(=O)C(C)S(N)(=O)=O)c(C)c1 C=Cc1ccc(C(=O)N(CCNC(c2c(C(F)(F)F)cnn2C)=O)CC)cc1 c1(OC)cccc(-n2c(SC3CC(F)C(=O)N3)nnc2-c2ccc(C)cc2)c1 CC1CC(=O)NCC1C(=O)NCCCCCNC(c1cscc1C(N)=O)=O C1(C(=O)NC2CCN(C)C2=O)CC(C)(C)CN1C(c1csc(Cl)c1)=O N1(C(c2c(CC)[nH]cc2)=O)C(C(=O)NCC(C(C)(C)C)OC)CC2CC12 CCC(C)CC(=O)N(CC(CC(=O)N1CCC(OC)C1)OC)c1cccnc1 c1cc(-c2nc(CN(C)C)nn2C2CCOCC2)ccn1.c1(CCS)ccccc1 c1(OC)ccc2cc(C(=O)NCC(C)(O)CNC(=O)C#CC(C)(C)O)ccc2n1 C1(C(=O)NCC2COCC2O)CC12CCN(C(=O)CN1CCNC1=O)C2 C1(CNC(Cn2c(C)ncc2)=O)CCC(C)(C)CN1C(=O)CCC1CCCN1C CC1(C)Cc2cc(Br)ccc2C1NC(C1CCC2(CCCNC2)C1)=O N1(C(=O)NCC2CCN(CC(F)(F)F)CC2)CC2(CCSCC2)C1 Cc1cc(C)c(NC(=O)CC2CCCCC2NC(=O)COCCCN=[N+]=[N-])cn1 N1(C(=O)Cn2cnnc2C)CCC2(CNC(=O)O2)C1.C(C)(C=O)NCCC c1(COC)ncc(C(=O)N(C2CCCC(O)C2)C)cn1.C12(CC1)C(=O)N2C Cc1cc(CN(CCCC)CC)no1.C12(CC(=O)O)CCCC1C2 Cc1coc(C(=O)NCC=CCNC(C2(C(=O)Nc3ocnc3CC)CC2)=O)c1.C(N)=O C=C1CCN(C(=O)C=CC(C)(C)SC)C(C(=O)NCCC(C)(C)OC)C1 c1(C(=O)NCC2CC(C)SCC2)cnc2sc(Br)cn12 c1(C(=O)NCC(c2ccc(OCC)cc2)O)ccc2c(c1)c(C#N)cn2C Cc1ncc(N)cc1C(=O)N(CC(O)CN(C)C(c1csc(Br)n1)=O)C CCCCC(F)C(=O)NCCC(C)(C)C(=O)NCCC(=O)N(CC)CC C1(CC(=O)OCC)CCCN1C(C1CC1C(=O)NCCn1nnc(C(=O)OC)n1)=O C(=O)(CCN=[N+]=[N-])N(C(CNC(=O)C(N1CCOCC1)C1CC1)CO)C N1(C(C2N(C(CC3CC(=C)C3)=O)CCC2O)=O)CCCCC(CO)C1 S(=O)(=O)(CCc1cnn(CC(F)(F)F)c1)NCC(n1cccn1)C Cn1cnnc1CCC(=O)NC1CCC(C(=O)NCCSCCO)C1 c1(C(=O)NC2CN(C(c3cn(CC=C)nn3)=O)C(CO)C2)cc(O)nc(O)n1 N1(C(C(C(C)C)CNC(C2CCN(C)CC2)=O)=O)CCC2CC1C(=O)O2 CC1CCOCCN1N1CCCC(Cc2ccc(F)cc2)C1 C12(C(=O)NC3C(CNC(c4nc(N(C)C)oc4)=O)C3)CCC(CO)(CC1)C2 C1(C(NCP(OCC)(C)=O)=O)C(C)CCN1C(=O)CC1CC1 C1(C(=O)Nc2ccccn2)CC12CCN(C(=O)CCN1CCOC1=O)CC2 C(C(=O)N1CC(C)(O)CO1)C1(NC(Cc2c(C)cccn2)=O)CC1 C1(CC(=O)NC2CC(OCCNC(C(c3ccccc3)C)=O)C2)CCC2(CCC2)O1 c1(CCCC(N2CCC(c3cn(CC4CC(=O)OC4)nn3)C2)=O)cccc(Cl)n1 Cc1ccc(Cl)cc1C(=O)NC1CCN(C(C2(c3ncccn3)CCC2)=O)CC1 N1(C(c2ccc(OC)o2)=O)CC(C(=O)NC2CC23CCOC3)C2(CCC2)C1 C(=O)(CC(C(C)C)C(C)C)C(C)=O.C(CCN)(C(C)(C)C)N(c1ncns1)C c1(NCCCC)ccc(N)c(C(N2CCC(CO)(NC(=O)CSC(F)F)CC2)=O)c1 c1(SCC(N2CCOCC2)=O)cnn2c1CCC2.c12cn(nn1)C2 c1(OC)ncnc(C(=O)OCCCS(N)(=O)=O)c1O C(CC(C)C)(C(=O)NCCc1ncccn1)N(C(C(CC)OCC)=O)C N1(C(CSCC(N)=O)=O)CC2ON=C(CNC(=O)C=C3CCSCC3)C2C1 CC1(C)CCC=C(C(=O)NCCCC(C)(C)NC(=O)CCc2ccoc2)C1 CC1CC2(CCN(C(=O)CCCN3CCCCC3)CC2)CN1C(C12COCC1C2)=O C1(C(=O)Nc2cccc(NC(c3n(CCC)ccc3)=O)c2)CC12CC(C)(C)C2 Cc1cc2[nH]c(C(=O)NCC3CC(C)(C)CN3C(=O)CSCC(F)F)cc2o1 C(CN=c1[nH]c(=NCC(C)(C)CC(C)C)[nH]c2cccnc12)SCC=C c1(C(N(CC2N(C(C3C(=C)C3C(=O)OC)=O)CCC2)CC)=O)cc(Cl)cn1C N1(C(C(C)SCCCC)=O)CCC(CNC(=O)CCc2ccco2)(COC)C1 Cc1nc(=NCC(CC(C)C)NC(=O)CCC2CCCC2)s[nH]1 CC1CC(F)(F)CN1C(=O)CN(C1CCC1)C(c1cnn(CCN(C)C)c1)=O CCC(C)C(O)C(=O)N1CC(F)(F)CC1C(N1CCS(=N)(=O)CC1)=O c1(C(=O)NCC2C(C(N)=O)CN(C(C(C)(C)OC)=O)C2)cc2cnccc2[nH]1 CC1CN(N2CCCCC2c2ccccc2-c2ccccc2)C1 c1(C(N2CCCOC(CO)C2)C(=O)NCCCSCC)cc(F)c(F)c(F)c1F Cc1cc2nc(n1)N(C)C2.C1(CC2CC2)CC(F)C1 Cc1nc(C(C)C)ccc1C(=O)NCC12CCC1CN(C(c1cccc(N)n1)=O)C2 c1(OC(CC(=O)NCC(C)CNC(C2CC2[N+](=O)[O-])=O)=O)ccc(Cl)cc1 CN1CCN(C(=O)CC2(C)OCCO2)C(C(=O)NCCC2CCC(C)(C)O2)C1 C=C(Br)CCC(=O)NCC1(n2ccnn2)CC1.c12cn(nn1)C1CN(C1)C2=O Cn1cc(C(C2CC2)NC(=O)Cc2cn(CC(=O)O)nn2)c(Cl)n1 N1(C(c2c(OCC)nccc2)=O)CC2CCN(Cc3occc3Br)C2C1 C1(NC(C2(OC)CC2)=O)COCCC1NC(c1sc(C)nc1CC(C)C)=O N1(C(c2c(C)c(F)ccc2)=O)CC2(CCCCN2C(c2cn3c(n2)SCC3)=O)C1 N1(C(C=CC(CC)=CC)=O)CCC2CCN(C(c3ccc(C)nn3)=O)CC12 c1(C(N2CCC(NC(C(CC)(C)C)=O)C2)=O)ccc(NC(C)=O)cc1O c1(NS(CC)(=O)=O)cccc(F)c1C(=O)Nc1cc(OC)cc(Br)c1 C1(C(=O)NCCC(CCNC(c2n(CC)cnn2)=O)C)CCCC(C)(C)CC1 c1(C(N2CC3(CCC3)C2)C(=O)NCC(F)F)cccc(C2CCCCC2)c1 c1(C(N2CCN(C(CC(C=C)C)=O)CC2C)=O)cc(C)c(C)cc1C c1(OC)cc(NC(c2ccoc2)=O)ccc1OC.C123COC(C1)(C2)C(=O)NC3 C1(c2nnc(N3CC(C)SCC3)n2CC)CC2CCC1N(C)C2 Cc1nc(C)n(CC(=O)NCC2CC2CC(=O)NCCc2cnco2)n1 C12(C(=O)NC3C(CNC(C4=C(C)CCC4)=O)COC3)CC3CC(CC(C3)C1)C2 C1(NC(CC=C=C)=O)CCCCCN(C(c2ncc(Br)cc2F)=O)C1 C1(C(=O)NC23CC(NC(c4c(C(N)=O)c[nH]c4)=O)(C2)C3)COCCN1C(N)=O N1(CCC(=O)NCC(=O)NCC(=O)NCc2ccoc2)CCCCC1 C=C(Cl)CC(C(=O)NCCN1CCCCCC1)NC(c1ocnc1C)=O C1(CCC)CC(C(=O)NC2(C3CCCN3C(C3CC(C)=NO3)=O)CC2)CCO1 C1(C(=O)NCCOC(CNC(C(C)Cc2ccco2)=O)(C)C)OCCCC1(C)C C1(C(=O)NC(c2ccc(O)cc2)C(C)C)C(O)CCN1C(c1ccc(F)cc1)=O c1(NCc2nnn(C)n2)ncccc1S(=O)(=O)NCC1C2CCCCCC12 N1(C(c2c(CCC)cccc2)=O)CCC2(CCC2)C(NC(=O)C=CC(C)(C)C)C1 CC(C)C(=O)C(=O)NC1CCOCC1C(=O)Nc1cccc(C(N)=O)c1 CON=C(C(=O)NC(c1nccnc1C)C)c1ccco1 N1(CC(C)C)C(=S)NC(c2ccc3cn(C)nc3c2)C2=C1C1(CCOC1)NC2=O C=CC(C)(CC)NC(=O)C(C)(C)NC(c1ccn(C)c1)=O c1(CC)c[nH]nc1C(=O)NCCCN1CCC(NC(c2cc(Cl)c[nH]2)=O)C1 c1(C(CN(c2nnc(C)s2)CC2CCCC2)O)ccc(C(F)C(F)(F)F)cc1 n1(CCC)nc(-c2cccc(OC(C)(C)C)c2)nc1C(CC1CC1)OC N1(C(c2c(C)nc(O)cc2)=O)CC(C)CN(C(=O)C(C)n2ccnc2)CC1C c1(C(C(=O)NC2COC2)N(CCc2c(C)noc2C)C)ccc(S(N)(=O)=O)s1 C(CC(C(C)(C)C)NC(=O)C(c1ccc(C)cc1)(F)F)N(C(CSC)=O)C C1(C(=O)NCc2nc(CNC(C3CC3c3cccs3)=O)cs2)CC(=O)NC(=O)C1 C1(NC(c2cccc(OC)c2F)=O)CC2CC(NC(C3CC=CCC3)=O)CC2C1 N1(C(COCCC=C)=O)CCC(C)(NC(=O)CCn2cccn2)C1 C1(N(C(c2ccc(Cl)o2)C(=O)NCCCF)CC)CCC(=O)NC1=O N1(C(C2(CCNC(C(c3ccccc3)C)=O)CCC2)=O)CCC2CCCC2C1 C1(N(CC(=O)N(C2CC(NC(C3CCCCC3O)=O)C2)C)C)CCOCC1(C)C C(C(N=[N+]=[N-])C(=O)NC1CCCCC1NC(c1cncc(Cl)c1)=O)OCC C(CCO)(C(F)(F)F)NC(CC1CCN(C(CCCC2C(C)C2)=O)C1)=O C(CN=c1ccnc(C2CC2)[nH]1)C1CCN(C(C2CCN(CCC)CC2)=O)C1 CN1CCCC1(C)C(=O)NCC1CCN(C(=O)Cc2ccnn2C2CCCC2)C1 C1(C(N(CCN(C(C)C)C(c2cc(Cl)n(C)n2)=O)C)=O)CCN(C)C(=O)C1 C(=O)(C1=CC2(CCOC2)C1)NCC(CCCC)NC(CCCC#C)=O C1(C(=O)Nc2nnc(CC)s2)CCCN1NC(=O)COCC1CCC1 n1(C(C)C)ccc(CNC(c2nnnn2C2(C)CC2)C2(C3CCCO3)CCC2)n1 CCC(C)(C)C(C)CC(=O)NCC1CC(C)(C)CN1C(=O)CCC1OCCO1 C1CC(=O)N1.C1(C(=O)N(CCOC)C)(CC)CC1 C1(CC(=O)NC(CCC=C)C)CCCC(NC(c2cccnc2O)=O)C1 CC(C)(C)C(C(=O)N1CC(C#N)(CCF)C1)NC(C1CC(C)(O)C1)=O C1(SC(C)CC(O)c2cccnc2)CCN(C(=O)C(=O)NC2CCOCC2)CC1 C1(NC(c2ccc(Nc3ccncn3)s2)=O)CCCCC1NC(N1CCCC1)=O c1(CCC)cc(-c2nc(C3CC3)nn2C)cc(OC)c1OC c1(C(C(=O)OC)Nc2cc(N3CCOCC3)ncn2)ccc(Cl)cc1Br C1(NC(c2cc(NC(C)=O)ncc2)=O)CN(C(C2CC23CC3)=O)CC2(CCC2)C1 c1(C(N2CCC(C(CNC(CSCCC)=O)C)CC2)=O)c(F)cc(O)cc1F c1(C(=O)NCC2C(NC(c3ccc(C)cc3Br)=O)C2)cc(F)c(C)cc1N C1(CNC(C=Cc2n(C)ncc2)=O)CCN(C(c2cc[nH]c2)=O)CCC1(F)F N1(C(CC=CC=C)=O)CCCC(N(C(=O)C(C)N(CC(F)(F)F)C)C)CC1 Cc1nn(C)c(Cl)c1C(=O)NC1CCCCN(C(=O)C2=CCSC2)C1 Cn1nccc1CCNC(=O)CCC1CC(NC(C2CCC2C#N)=O)C1 C12(NC(C3CC(=O)N3)=O)CCCN(C(=O)C=CCCc3ccccc3)CC1C2 C(CC(C(=O)NC(C)CC1CC1)NC(=O)CC1CCSCC1)OC c1(OC)ccc(C(=O)NC2CCC2NC(c2c(C)cccc2C)=O)cc1F C12(CNC(CC(C)(C)OC)=O)CN(C(=O)C=C3CCOCC3)CC1(C(F)(F)F)C2 Cc1cc[nH]c1C(=O)NCCC1CCC(NC(=O)CSc2n[nH]c(O)n2)C1 N1(C(c2cc(CC)sn2)=O)CC2CCC2(NC(=O)C(CO)NC(N)=O)C1 C1(C2CCC2)(CNC(=O)C(N2CCC(N3CC=CC3)C2)=O)CCNCC1 N1(C(C(C)OCC(F)(F)F)=O)CCOC(CNC(=O)Cc2ccn(C(F)F)n2)C1 c1(C(=O)NCC2(C#N)CCOCC2)ccc2c(n1)CN(C(C1C=CCC1)=O)CC2 C1(NC(CN(C(C(C(CC)C)OC)=O)CC)=O)CCn2ccnc2C1 N1(C(c2ncn(CC)n2)=O)CC(C2CN(C(c3coc(-c4ccsc4)c3)=O)C2)C1 c1(C(=O)NCC2(C(=O)NC3CC(C)(CC)C3)CC(F)C2)nc2ncccn2n1 S(=O)(=O)(c1ccc2c(c1)C(=O)NC2=O)Nc1ncc(C)[nH]1 c1(C(N2CCC(CNC(c3cnc(CC(C)C)s3)=O)C2)=O)cccc2c1OCC2 C=C1CN(C(=O)NC(C)(C)C)C1C(=O)NC1(CO)CN(C(=O)C=C(C)C(C)C)C1 C(C(C)(C(C)C)NC(=O)C(C)SC)NC(CCOCC)=O c1(C(N(C)Cc2ccccc2)=O)nc2ccccn2c1-c1cccc2c1ccn2C C1(CNC(C=CCC)=O)N(C(C23CC4CC2C3C4)=O)CCCC1(C)C C=C(C)CC(C(=O)NCC(c1ccco1)O)NC(c1sccc1C)=O C12(CNC(c3cc(C)sc3)=O)CCCN(C(=O)COc3cccc(C)c3F)C1C2 C1(C(=O)NC(C)CN(C)C(c2n[nH]nc2Br)=O)Cc2ccccc2N1 CCC(CNC(c1ccc(C(C)(F)F)cc1)c1nnnn1C1CCCC1)CCO C1(C(=O)NCC(CN(C)C)O)COCCN(C(c2ccc(C#N)cn2)=O)C1 C1(NC(=O)CCn2ccnn2)CCC2(CC1)CN(C(c1cnco1)=O)CCO2 c1(C(=O)NCCCCN(C(COC)=O)CCO)cc([N+](=O)[O-])cc(C)c1Cl N1(C(C2C3(CN(C(c4c(C)noc4C)=O)C3)C2)=O)CCCN2CCCC2C1 c1(-n2cc(C(CCC)=O)nn2)ccc(OC)c(Cl)c1.C12CN(CC1C)C(=O)C2 C1(C(C)C)CN(C(C2CCC2(C)C)=O)CCC1NC(=O)CCCn1ccnc1 c1(NCC(Cc2ccccc2)NC(c2ccc(C)[nH]2)=O)cc(O)ncn1 CC1CN2CCN1C(C(=O)NCC#CCNC(=O)CC1CCOC(C)(C)C1)C2 N1(C(c2cc(C)oc2C)=O)C2CCCC1CC(NC(c1ccnc(C)c1N)=O)C2 N1(C(C(CN(C)C)NC(c2ccc(C)nn2)=O)=O)CCCC(C)(CC2CC2)CC1 c1(SC)ccc(C(=O)NC(C)C(C)NC(c2ncnc(O)c2F)=O)cc1[N+](=O)[O-] c1(C(C)C)ccc2occ(C(N3CCC3CNC(=O)C(C)(C)C(C)(F)F)=O)c2c1 c1(C(=O)NC2CCCC(N(C)C(c3ccc(F)s3)=O)C2)csc2ncnc(O)c12 C(=O)(C(CCF)NC(c1cccs1)=O)N(C1CCC(F)(F)C1)C C(C)(C)CC(F)(F)CC.C(C(=O)NCCSC)(OC)OC C1(C(=O)Nc2ccc(C(=O)OC)c(O)n2)COC2CCCCC12 N1(C(c2cccc(OC)n2)=O)CC(C)CCC1C(=O)NCc1sccc1C N(C(=NCCN1CC2CC2C1)N1CCCC2(CCOC2)C1)Cc1cccc(O)c1 C(C(=O)Nc1ccc(-n2cnnn2)cc1)(C(C)C)OCC(C)C c1(C(=O)NC(C)(CC2CC2)N(C)C(=O)OC(C)(C)C)ccc(C(F)(F)F)c(Cl)c1 C1(C(N2CCN(c3ccccc3[N+](=O)[O-])CC2)=O)Cc2cncn2C(=O)N1 c1(CC)cncc(C(=O)NCCC(C(=O)NC2(CO)CCSC2)OC)c1 Cc1cccc(C)c1C(=O)NCCCC(=O)NC1CC1NC(=O)C(C)S(C)(=O)=O c1(N(C)CC2CCCC2O)nc(N(CCCc2ccco2)C)c2sccc2n1 C1(C(N(CCN=[N+]=[N-])CC)=O)COCCC1NC(=O)CCCNC=O c1(OC)cc(OC)cc(C(=O)NC(C)CN(C)C(c2c(C)ccnc2Cl)=O)c1 Cc1cccc2[nH]cc(C(=O)NC3(C)CN(C(=O)CCc4n[nH]c(=N)s4)C3)c12 c1(CC(=O)NC(C(=O)NCCN2CCCCC2)c2ccoc2)ccc(O)cc1 c1(C(N2C(CNC(c3cc4n(n3)CC(F)C4)=O)CC2)=O)cc2nc[nH]c2cc1F C1(OC)CC2CCC(C1)N2C(c1coc(C(C)NC(c2ccc(C)o2)=O)n1)=O O(NC(=O)CC1CC(NC(c2c[nH]cc2C2CC2)=O)C1)C(C(C)C)O C(=O)(C#CC1CCCOC1)NCC1N(C(c2ccc(OC)c(N)c2)=O)CCC1 CCC(CC)CCNC(=O)CNC(=O)CSC.c1(C(N(C)C)C)ccccn1 N1(c2ccccc2)CCC(N)CC1.Cn1cnc(C(=O)N(C2CCCC2)C2CC2)c1 C(=O)(C(C(=O)NCC1(C(=O)NC)CC1)OC)OCC.c1(C2CC2)ccsc1 c1(C(=O)NC2(CF)CCN(C(CC(C)(C)C)=O)C2)cc2ccccc2nc1O c1(OC)cnc(C(=O)NC(C)(C)CCNC(C2(CO)CC2(F)F)=O)nc1 N1(C(CCC)=O)CCC(c2nnnn2C)(NC2CC(=O)N(C)C2)CC1 c1(C(=O)NCC(CNC(C2CC2CSC)=O)OC)coc(C(C)C)n1 C1(C(=O)NCc2cc(OC)ns2)CN(C(C2CCCC2)=O)CC12CC2 C(C1c2ccsc2CCN1C(=O)C(c1cnn(C)c1)=O)NC(C1ON=C(C)C1)=O Cc1cc(C(=O)NC(C)CNC(c2cncnc2)=O)c2c(O)n[nH]c2n1 c1(C=O)cc(CO)oc1C.c1(CC)ncc(C(N2CC(CN)(COC)C2)=O)s1 CCC(C)(CC)C(=O)N1C(C(=O)N(C2CC(C)CC(C)C2)C)CCC12CC2 N1(C(c2ccc(Cl)cn2)C(=O)Nc2ccc(OCC)cc2)CCOCC12CCC2 C#CC1CN(C(=O)C(c2nnn(C)n2)OC)CCN1C(c1cc(Cl)cs1)=O C#CC1(O)CN(C(=O)CCC2CC(NC(=O)C(CC)OCC)C2)C1 N1(C(C2=CCN(C(c3cnc(CC)s3)=O)C2)=O)CCCC[Si](C)(C)C1 CCCCC(C(=O)NCC12CC1CN(C(=O)C(CO)N(C)C)C2)N(C)C Cn1ccc2cc(C(=O)NC3CCCCN(C(C4(CO)CC4)=O)CC3)cnc12 c1(CC)nc(C)ncc1C(=O)NC1CCCCC1NC(=O)C#CC(C)C CN1CCN(C(C2CCCN2C(N2CC3CC2CN3C)=O)=O)C(CO)C1 N1(C(C(=O)NC(C(C)(C)C)Cc2ccccc2)=O)CCOCC12CC2 C1(C(=O)NCc2cc(C)ncn2)C2CCN(C(c3cc(O)n(C)n3)=O)CC12 c1(NC(C2CCCC(NC(c3nccc(CC)c3)=O)C2)=O)cc(Br)c(C)nc1O C(=O)(C(Cc1cn(-c2ccc(O)nc2)nn1)CC(C)C)N1CC(COC)C1(C)C C1(NC(c2ncoc2Br)=O)CCN(C(c2nocc2Br)=O)CC1O C1(CNC(C(C)(C)c2cc[nH]n2)=O)CN(C(=O)CCC2OCCO2)C2(CCC2)C1 CN1N=C(CC(=O)N2CC(CCNC(C3CCC(C)(C)OC3)=O)C2)CC1=O C12(C(N3C(CNC(=O)CSc4ccncc4)CC(OC)C3)=O)CCCC1C2(F)F c1(C(=O)NC2(C)CC(NC(c3cnc(COC)s3)=O)C2)c[nH]c2nc(F)ccc12 N1(C(=O)CC2CCCN(C(c3ccc(O)cn3)=O)C2)CCC2(CCCO2)CC1 N1(C(c2[nH]cc(C(=O)OC)c2)=O)CC(NC(=O)CCCF)C(F)(F)C1 C(CC(C)C)(C(=O)NC1CCN(CCNC(C2(C)CC(C)(C)C2)=O)CC1)OC C(=O)(C1=CCCSC1)NC(C1CC(F)(Cn2cc(CNc3ccc(=N)[nH]c3)nn2)C1)=O N1(C(CCC=CCCC)=O)C(CNC(C2CN(C)C2)=O)CC2CC12 CC1=NN(C)C(=O)C1CC(=O)NC(C)CCN(C)C(c1cc(Cl)cs1)=O N1(C(C(C)(C)SC)=O)CC(NC(C2(O)CCOCC2)=O)C(n2ccnn2)C1 C1(N2CCC2)CN(CC)CCN1C(=O)CC1CC2(CC2)CO1.c1(N)ccc(CO)cn1 c1(C2C(Nc3ccc(OCC)cc3)N(C(=O)NC)CCC2)ccc(F)c(C)c1F C1(NC(c2c(C)ncn2O)=O)CC2CC(C1)N(C(c1scnc1Cl)=O)C2 N1(C(C2(CCNC(CCOCC)=O)CC2)=O)CC(=O)NC(C)(C)C1 C1(C)(CNC(c2c(C)n(C)nn2)=O)COCCN(C(=O)C2=NOC(C)C2)C1 C1(OCC(N2CC3C(NC(=O)CCc4nccs4)(C3)C2)=O)CCC(F)(F)CC1 c1(CC(=O)N(C)CC2CN(C(C3C(CC)OCC3)=O)C2)ccc(CO)cc1F C(=O)(CC(CCC)=CCC)NC(CC=C)CNC(C1CCOC1)=O C(=O)(C1Cc2c(Cl)cccc21)N1CCCC(C(=O)NC2(NS(=O)(=O)C3CC3)CC2)C1 c1(C(=O)NCC(CC=C)NC(=O)Cn2nccn2)ccc(F)cn1 C(=O)(C1=NN(C)C(=O)CC1)NCC(C(=O)N(CC#CC)C(C)C)CC(C)C c1(CN(CC)CC2C3(CCC3)C23CCC3)nc2cc(C)cc(C)c2[nH]1 O=C1CCC(C(=O)N2CC3CC3(C(=O)Nc3nccc(C(F)(F)F)c3Br)C2)=NN1 CN1CCN(C(=O)C2=CCC(NC(=O)CCc3cnoc3)C2)CC1C(N)=O c1(-n2ncc(C(=O)NCCCN(C(C(C)=C(C)C)=O)C(C)C)c2)ncc(Cl)cn1 C1(NC(C2(C)CCC(F)(F)CC2)=O)Cc2ccccc2C1NC(C1CCC1)=O C(CCSC)(C(=O)N(CC(F)F)C(C)C)NC(c1cn(CCC)nn1)=O c1(CCC)ccccc1C(=O)NCCC1CCN(CC(=O)NC(C)C2CC2)C1 N1(C(C2N(C(Cc3cc(C)on3)=O)CCCCCC2)=O)CCC(C2=NOCC2)C1 C(N=c1[nH]c(Cl)ncc1C(=O)OCC)C1(OC)CN(C(C(C=C)O)=O)C1 CC(C)C(O)CC(=O)N(CC(C)(C)NC(c1ccc(C(F)(F)F)[nH]1)=O)C N1(C(C(=O)NCc2ccco2)C2CC2Cl)CC(OC)CC2CCCCC12.CO CCC(C)C(O)C(C)C(=O)N1CCC(NC(c2c[nH]nc2CC)=O)CC1C C(C)(CCC(=O)N1CCCC1(C)CNC(=O)CC(C)c1ccccc1)SC C1(C(N2CC(NC(C3C(C=C)C3)=O)CC2(C)C)=O)CCC(=C(F)F)CC1 CN1CC(=O)N(CC(N2CCC(NC(=O)CC34CC(C(=O)O)(C3)C4)CC2)=O)C1=O C(=O)(CC(C(F)(F)F)NC(C12CCCC1C2(F)F)=O)N(C1CC2CCC1O2)C C1(C(N(C(C(N2CC(O)(C(C)C)C2)=O)C2CC2)C)=O)CC2(CC2)CN1C N1(C(CC(C)c2cnn(C)c2)=O)CCN(C(=O)CC2(O)CCC2)C(CCO)C1 C1(NC(=O)CCOC2CC2)CCCC(N=c2[nH]nc(CCO)s2)C1 c1(C(N2CC(F)(CNC(C3=CCCCC3C)=O)C2)=O)cnc2c(ncn2C)c1 C(=O)(C(CC(C)C)NC(C1CC2CCC1CC2)=O)NC(CCSC)C C#CCC(C(=O)NCCOC1CCN(C(=O)CCc2ccnn2C)C1)NC(C)=O C(=O)(CC(C)CC(C)(C)C)NC(C(N1CC(CC#C)OCC1)=O)c1ccco1 C1(NC(C=CCC2(NC(c3c(C)n(C)cn3)=O)CCC2)=O)CC2CSCC(C1)C2 N1(C(C(C)Cn2ccnc2)=O)CCC(C(=O)NC(Cc2cnc[nH]2)CO)CC1 C1(N(C(c2c(C)csc2Cl)=O)C)CN(C(=O)C(F)C(F)(F)F)CC1(C)C c1(C(=O)NCCOCCNC(C(CC#C)CC#C)=O)ccc2[nH]ccc2c1F C(=O)(C(F)(CNC(C1(O)CCCC1)=O)C(C)C)NC1C(SC)CCC1 C1(CNC(C(=O)NCC)=O)CN(C(=O)COc2cccc(C)c2)CCC1C C=CC(CCC)CC(=O)NC1CCN(C(c2cnn(C(C)C)c2)=O)CC1 CC1CCC(CC(N2CC(CCN(C(=O)Cn3ccc(C4CC4)n3)C3CC3)C2)=O)O1 C1(CCNC(C(CC)OC)=O)CCCN(C(c2cn(Cc3cccs3)cn2)=O)C1 C(=O)(CC(C)(O)C1CC1)NS(C)(=O)=O.CC(C(=O)N(CCOC)CCO)NC=O CON(C)C1CCN(C(=O)C(C)(CO)NC(C2CCCCC2F)=O)CC1 Cc1nc(C(C)NC(=O)C(Cc2cn[nH]c2)NC(=O)CC2CC(C(C)C)C2)c(C)o1 Cc1cn2c(n1)CC(C(=O)N(CCCCN(C)C(C1COC3COCC13)=O)C)C2 C1(C(N(C(CN(C(C(C)=C(C)C)=O)C)C)C)=O)(CF)CC1(F)F C1(NC(c2cc(Cl)ccn2)=O)COC2(CNC(C3(CF)CCNC3=O)=O)CC1C2 c1(OC)ccc(NC(N2CC(Nc3nccc(C(F)(F)F)n3)C(O)C2)=O)c(Cl)c1 Cn1c(C(N2CC(NC(=O)CO)C(O)C2)=O)ccc1C1CCCC1 CCC1=NOC(CC(=O)NC(CO)C(=O)N(C)Cc2ccon2)C1 c1(C(=O)NC2C3CN(C(C4(C)CCC(=O)NC4)=O)C2CC3)cnc2[nH]nnc2c1 c1(CCC)cc(C(=O)NCC(C2CCCC2)NC(=O)C(C)CC)n(C)n1 S(=O)(=O)(c1cccc(=NCC(=O)NC(C2CCCC2)C)[nH]1)NC1C(C2C(C)C2)C1 N1(C(c2c(C)coc2)=O)CCC2(CCCN(C(=O)CC3CCCOCC3)C2)C1 c1(OC)ccc(CN2CCCC(C(=O)NC3CCC(F)(F)C3)CC2)c(Br)c1 c1(CCn2c(C)ncc2)nc(-c2ccco2)nn1C.C12CCN(C1)CCC(=O)C2 C1(C(N(C)CC2(NC(=O)Cc3ccccc3O)CC2)=O)CCC12CCOCC2 c1(C(=O)NCCNC(=O)CC2CCOC2)cc2n(n1)CC1(CC1)CO2 C=CCCC(C(=O)N1CC(=O)NC(CC)C1)NC(c1ccnn1C(=O)OC)=O N1(C(c2n(CC)ccc2)=O)CCC(F)CC1C(=O)NCc1c[nH]nc1CC1CC1 C1(NC(COC)=O)CN(C(c2cccc(C#N)c2)=O)Cc2ccnn2C1 C1(C(=O)NC2CC2)(CC)CCCN1C(C1CCCN1C(C)C)=O C1(NC(c2cc(SC)oc2)=O)CC(OC)CN(C(=O)COCC2CCCCO2)C1 C(CS(=O)(=O)CC(=O)NC(C1(C(=O)NC2CCC(=O)N2)CC1)C)OC C1(CC#C)(NC(c2cc(CSC)on2)=O)CCN(C(=O)CC(C)C)C1 C1(CCNC(c2cc(C)nn2C)=O)CC(F)(F)CN1C(=O)CCN1CCC(F)C1 N1(C(C2N(C(C(C)(C)C)=O)CC2)=O)CCCC12CCN(C(c1cnc[nH]c1=N)=O)C2 C1(CC(=O)NCCOCCN(C(CSC)=O)C)CC=CCC1.C1CO1 N1(C(C(C2CN(C(=O)CCCc3cc[nH]n3)C2)OC)=O)CC2CCC(C1)C2C#N c1(N2CC3OCCN(Cc4c(F)nccc4)C3C2)cc(Br)cc2cn[nH]c12 C1(C(C)C)(C(=O)NCCCOCCO)CCN(C(=O)Cc2ccccn2)C1 N12CCC(C1CNC(C1CC(OCc3nncn3CC)C1)=O)CCC2=O.CC.CC C1(CC(=O)Nc2n[nH]c(-c3ccccc3)n2)CCN(C(=O)CC2(O)CCCC2)C1 CC(C)C(O)C(F)(F)C(=O)N1CCC(CCNC(C2CCC(=O)N(C)C2)=O)CC1 N1(C(c2ccc(SC)o2)=O)CC(NC(C2CSCC(=O)N2)=O)C(n2ccnn2)C1 C1(N(C)C)CC(N=c2[nH]c(=NC(C)c3cccc(Cl)c3Cl)[nH]c3ncn(C)c23)C1 C1(C(=O)NC2(CNC(CCC(C)OC)=O)CCCC2)CCCCC1(F)F c1(CCCC(=O)NCCN(C(c2ccccc2OC)=O)CC)ccc(Cl)cc1 C1(C#N)(C(N2CCC(N(C)C3CC3)CC2)=O)CC2CC2C1.C12CN(C1)C2=O C12(NC(COCCC(C)C)=O)CCC(CNC(=O)CCC(C)CN(C)C)(C1)OC2 C1(C(=O)NCC#CCNC(C2N(C(C)=O)CCCC2)=O)CCc2nc(O)[nH]c2C1 C(C)(CO)(C(C)(C)O)NC(c1c(C)nc(CNC(=O)CN2CC(C)(C)C2)o1)=O c1(C(=O)NC(CN(C(C(F)OC)=O)C)C)cc(N)cc(O)c1 c1(CC(N2CC3CC(CNC(C4(CCC)CC4)=O)C3C2)=O)c(C)nc(O)nc1C c1(C(=O)OC)ccc(S(=O)(=O)N2CC(N(C)C(C3CCCCNC3=O)=O)C2)n1C C(=O)(C1=NOC(C)C1)NC(C(=O)OC)CC1CC1 c1(OCC(C)C)ccc(CNCc2c(C(N3CCC3)=O)csc2)cc1 c12nocc1C(=O)NC2.C(C(C)(C)CSC)NC(C1(OC)CCC1)=O N1(C(c2cc(C(=O)OC)no2)=O)CC(OC)CC1NC(=O)COC1(C)CCCC1 Cc1cc2cc(C(=O)NC3CN(C(=O)Cc4ccc(F)cc4)CC3F)ccc2[nH]1 C(=O)(C1CCCc2ncnn21)N1CC2(CN(C(c3ccn4nccc4c3)=O)C2)C1 CC(C)CCC(=O)NCC1(NC(=O)CC2CCCN2C)CCOCC1 CC1C2CCC(C2)C1C(=O)NC1CC2(C1)CC2C(N1CC(n2ccnn2)C1)=O C(CCCC(C)(C)C(=O)NNC(=O)CCCC1CCC1)NC(c1c(C)occ1)=O CC1(C)C(NC(=O)CN2CC3C(NS(=O)(=O)c4ccccc4)C3C2)CCS1(=O)=O c1(C(N2CCC(C(C)NC(c3nc(C)oc3)=O)CC2)=O)cc2c(cc1Br)OCO2 C(=O)(C1=C(Cl)CCCC1)C(=O)CC1CC(O)C12CCC2.C12CC3CCC1N3CC2.N C(=O)(C1=CC2C=CC1C2)NCC1CCN(C(CCc2c(C)cccn2)=O)C1(C)C c1(NC(C2CC(NC(c3cncc(C=C)c3)=O)C2(C)C)=O)ccc(F)c(F)c1F C1(C(=O)NC2CN(CCC)C(=O)C2)CCC(C)(C)N(C(c2scc(C)c2C)=O)C1 N1(C(c2cncc(C)n2)=O)CCN(C(c2ccc(C(F)(F)F)nc2)=O)C2CC12 C1(OC)CCCCC1N=c1cccc(S(=O)(=O)NCc2cnn(CC(C)C)c2)[nH]1 CN1CCOC(C(=O)NC2COCC2CNC(=O)CN(C)C(N)=O)C1 CN1CCC(C(=O)N(CC(C)(C)NC(c2cc(-c3cnn(C)c3)[nH]n2)=O)C)C1 N1(C(C=C2CCC(C)C2)=O)CCC2CN(C(=O)C(C)Cc3ccco3)C2C1 C(C1(C)CCOCC1)=CC(=O)N(CC(CC)NC(C1COCCN1CC)=O)C C123CC4CC(C1)CC(C4)(C2)N3C(C=CC=CCC)=O.C(=O)(C(C)COC)OC c1(COC)ccc(C2CC2(F)F)cc1.n12cc(nn1)C(C)NC(=O)C21CC1 C12(CNC(C3C(C)=CCS3)=O)CCC(CC1)N(C(C1(C)CCC3CC3C1)=O)C2 C(CNC(Cc1ccc(C(=O)NC)c(C)c1)=O)(C(C)C(C)C)NS(CC)(=O)=O C=CCC(CNc1cn(C)nc1C(N)=O)C(=O)NC(c1ccn(C(F)F)n1)=O Cc1ccc(F)cc1C(=O)NCC1CC(NC(=O)CN2CCCCS2(=O)=O)C1 c1(CCC(=O)NCC#CCNC(CC(C)SC)=O)ccc(O)c(Cl)c1 N1(C(c2c(C)nn(CCO)c2)=O)CC(CNC(C2CCCO2)=O)C(F)(F)C1 CC1OC(=O)NC1C(=O)NCC12COC(CNC(=O)C3=COCC3)(C1)C2 CC1CC(C(=O)NC(C)C(=O)Nc2ccc(SC3CC3)cc2)CCC1=O C#Cc1ccc(C(=O)NC(C)(C)C(C)NC(=O)C(O)Cc2ccccc2Cl)nc1 C(=O)(CCC(=O)C(C)(C)C)N1C(C(=O)NCc2c(C)ccc(OC)c2)CSCC1 c1(C(=O)NCC(CC=C)NC(=O)CCCN2CCCCC2)cnnc(O)c1 C1(NC(c2cn(CCOC)nc2C)=O)CCCC12CN(C(c1sc(=N)[nH]c1C)=O)C2 CC1CCCN(C(C2C3CCC2CC3)=O)C1CNC(=O)CN(C1CCC1)C C1(CNC(c2cn(C)c(O)n2)=O)CC2CCC1N2C(c1cccc(C2CC2)c1)=O N1(C(=O)NCCc2onc(C)n2)CC2(CCCCC2)c2ccccc21 c1(C(N(CCN(C(=O)CCC2CCC(=O)N2)C)C)=O)nc2ccccc2s1 C1(CNC(CNC(CCCCC)=O)=O)CC2(CCC2)CN1C(C1CC1C(C)O)=O N1(C(C2CC(C)OC2)=O)CCC2(COC(CNC(c3c(F)cccc3F)=O)C2)C1 C1(CN(c2cc(N3CC(C)OC(C)C3)ncn2)C2CC2)CC(F)(F)C12CCC2 c1(NC(C(C)N(C(c2c(C)n[nH]c2)=O)C)=O)ncccc1C(C)C c1(OC(C(C=Cc2ccc(OC)cc2)=O)=O)ccc(F)c2occc12 C1(NC(=O)Cc2ccncc2)CCC2(CC1)CCN(C(=O)CC1CC1)CC2 c12ccc(cc1)COc1cccc(c1)OCCC(=O)N2.N1(CC=C)CCC(CO)C1 c1(C(N2CCC(NC(C3CC4(C3)CC4(F)F)=O)C(F)C2)=O)cc[nH]c2nccc1-2 C1(NC(C(C(C)(C)O)F)=O)(CNC(c2ccc(F)cc2N)=O)CC2CCC1CC2 C(=O)(C1=CC(O)CCC1)N1CCC(CNC(CNC(=O)OCC=C)=O)C1(C)C C(=O)(C(CC=CC)NC(c1c[nH]c(=NC)o1)=O)N(CCN(C)C)CC CCC(O)C(C)C(=O)NC1CC2(C1)CC(NC(=O)C(O)COC)C2 C1(C(=O)NCCCC(C)NC(=O)C(=O)NC2CC2)COCCC1(F)F c1(CCSCCC(=O)N(CC)CC)nc(NC(c2ccccn2)=O)n[nH]1 C1(C(N(C2C3CN(C(CN(C4CC4)CC)=O)CC32)C)=O)CCc2c(cnn2C)C1 CCCC(C(=O)NCC(C(F)(F)F)OC)NC(=O)C(CC1CCC1)OC N1(C(=O)C2=CCC2)CCC2OCCN(C(C3CC4CCC(C3)S4)=O)C2C1 Cc1nonc1CC(=O)N(CCNC(C1COC(C)C1)=O)CCOCCO C1(CCC)CC(C(=O)NCC2CC2NC(=O)C(C2CCCC2)OC)C1 C(=O)(C#CC1CCCCC1)N1CCC(=CCNC(=O)C=Cc2ccccn2)CC1 C(CCNC(=O)C(=O)NCCO)(C(=O)N1CCCC(F)C1)SC c1(C(N2CC(C3CN(C(C(C)CC4CCC4)=O)C3)C2)=O)ccccc1S(C)(=O)=O C(C1CN(C(=O)CN2CCNC2=O)CC1C(=O)NC(C)CCCCCO)=CC C1(NC(CCCCC#C)=O)CCCCCN(C(c2cnc(CCCC)s2)=O)C1 C1(C(N(C(C)CO)CC)=O)COC2(CCN(C(c3ccno3)=O)CC2)C1 C12(C(=O)OC)CCC(CN(C(C3(C)CCCC3(F)F)=O)C1)C2 C(c1nnn(C)n1)=CC(=O)N(CCCCN(C(=O)CCCN1CCCC1)C)C Cc1cc(C)c(CNC(C2C=CCN(C(=O)C(C)(C)n3cnnn3)C2)=O)s1 C1(CCNC(C2CCN(C(C)=O)C2)=O)CC(F)(F)CN1C(C1CCCN1C)=O N1(C(C(C)CC(F)(F)F)=O)CCC2CN(CC(=O)N(C(C)C)C(C)C)CC2CC1 N1(C(=O)NCc2cc(N3CCOC3=O)ccc2F)CCC2(CCNC2=O)CC1 C(=O)(C(C)(CC)CCCCCC)NCC1(NC(C2(OCC#C)CCCCC2)=O)CC1 C1(C(=O)NC(CCCOC)(C)C)CC(C)CN(C(c2sccc2C)=O)C1 C1(OC)CC2CC(C1)N(C(C1C3CC1N(C(c1cncc(N(C)C)c1)=O)C3)=O)C2 c1(CCNC(C(C)C2CCCO2)=O)ccc(CNC(=O)Cn2ccnn2)cc1 C(C(C)C(C)C(=O)N(CCNC(=O)CCP(C)(C)=O)C(C)C)SC Nc1ccc(C(=O)NCC2CCN(C(=O)Cc3cccnc3F)C2)nc1 O(NC(=O)C(CC(C)(C)C)NC(c1ncnc(O)c1F)=O)CC C12(C(=O)NCCC(C)(C)NC(c3cc(C#N)c[nH]3)=O)CCCC(C1)C(=O)NC2 C1(CC(=O)NCC2(CNC(C=CC(C)(C)SC)=O)CCC2)CCCCN1C C1(OC)CC(NC(=O)CCCNC(C)=O)CN(C(C23CCCC2(C(N)=O)C3)=O)C1 Cc1cc(C(N2CCCCC2CNC(c2nccnc2C(F)(F)F)=O)=O)ccn1 c1(C(=O)NC2C(CC(N3C(COC)(CO)C=CC3)=O)CCC2)cc(C)nnc1O C(C(NC(=O)NCCOCC1CCC1)NC1CC1)OC C1(CC(C)C)CCN(c2cc(NC(=O)C(C)OC3CCCC3)ncn2)CC1 C1(CC(=O)NC2(CCCC)CC2)C2CCCC2N1C(=O)CC1CCCC2CC12 c1(CCC(=O)NC(C2CN(C(C3CCCN3C)=O)C2)C)ccc(F)cc1 C1(CC)(CC)C(OC)CC1NC1(c2cccc(F)c2)CCOCC1 N1(C(C2CC(C#N)C2)=O)CCC2(CCC2NC(c2ccc3ncccc3n2)=O)CC1 CCCCCCC(C(=O)N1CCC2C(N(C)C)CC12)NC(=O)OC(C)(C)C c1(C(=O)NC2CC(F)(CNC(=O)C(F)C3CCOC3)C2)cnc2cc[nH]c2c1 N1(C(c2ccc(C(=O)OC)o2)=O)CCC(F)(CNC(c2oncc2C)=O)CC1 C(=O)(C(CNC(=O)Cc1ccccc1C)C(C)C)NCC(C#C)C(C)C N1(NC(c2c(C)cccc2)c2c(-c3ccccc3)ncn2C)CC2CC2C2CC12 c1(C(=O)NC2CCC(CNC(CSc3c(C)ccs3)=O)C2)cnc2nccn2c1 CCCC(C)(O)C(=O)N1CCC(CN(C(=O)CCOCCC)C)C1 C1(C(=O)NCC2C(NC(Cc3ncc(C)o3)=O)CCC2)CCCC1C1CC1 CCCCN=C(NCc1cc(N(C)C)ccc1Br)NCC1CCSC1 C1(CNC(CC2C(C)(C)C2)=O)CCC(NC(=O)C(F)(F)C2CCCC2)C1 C1(C)(C(N2CC(OCC(=O)NCC=CC(=O)NC)C2)=O)CCC(=O)NC1 C1(CCOC)CN(C(=O)CC2SC(=N)NC2=O)CCN1C(=O)Cc1cnnn1C CCCC(C)(CCC)C(=O)NC1CN(C(C2CC2CC(C)C)=O)CC1CC1CC1 C1(C(N(C2CCOC2)CC#C)=O)CCN(C(=O)COCC(C)(C)C)C12CCC2 Cc1cc(Br)ccc1-c1cn(CC2CCCN(C(c3csnc3Cl)=O)C2)nn1 N1(C(C(C)C2CCC2)=O)CC2CCCC(C1)N2C(c1cc(Cl)on1)=O C1(C(=O)NC(C2CCOC2)CO)(SC)CN(C(=O)C(C)c2cccs2)C1 C1(NC(c2cccc(SC(F)(F)F)c2)=O)CN(C(=O)C=CC2(C)COC2)CC12CC2 c1(OC)cc(C)c(C(=O)NC2(CF)CCN(C(c3ccc(C(N)=O)o3)=O)C2)cn1 Cc1cccc(C(N2CC(C)(C3CCCN3C(=O)CCCn3cccn3)C2)=O)n1 C(=O)(C1CCCc2scnc21)NC1CC(CNC(c2cc(C)c(N)cc2Cl)=O)C1 Cc1nn(C)c(Cl)c1C(=O)NC1CC(C)N(C(C2CC3(CCC3)C2)=O)C1 c1(CC(N2CCCC(Cn3cc(C4(C)CCCC4)nn3)C2)=O)cc(F)cc(F)c1 C1(OC)CN(C(=O)CCC(C)C)CC1NC(c1ccc(C(F)(F)F)cn1)=O C(CC(C)C)(C(=O)NCC1(NC(C2CCCC(C)(C)C2)=O)CCOCC1)OC N1(C(c2c(C(N)=O)csc2)=O)CCCC(NC(C23CSCC2C3(F)F)=O)CC1 C1(NC(c2cc(OC)nn2C)=O)C(C)(C)CN(C(=O)CP(C)(C)=O)CC1(C)C S(=O)(=O)(c1cccc(=NCCC(C)SC)[nH]1)N(CCCSc1ccccc1)CC#C C(CC(=O)N1CCC(NC(=O)CC2CS(=O)(=O)C2)C(O)C1)(C(C)C)OCC N1(CC#CCOCC)C(=O)c2ccccc2C1=O.C1(C(F)(F)F)CN1 N1(C(COC)=O)CCCC(C)C1C(C1(NC2CCC2)CC1)CNc1cc[n+]([O-])cc1 c1(CC(N2CC(CNc3ccc(C(=O)NC4CC4)cc3)C2)=O)ccc(F)c(F)c1 C(=O)(CCCC(=O)OCC)NCC(C(=O)NC(CC#CC)CO)N(C)C C12C3CN(CC13)C2=O.C(=O)(CCCC1CCNCC1)NCCCOC N1(C(C(C)N(C(c2c(C)ccc(C)n2)=O)C2CC2)=O)CC(C)OC2(CCC2)C1 c1(CNC(C(CC)=CC)=O)cc(O)nc(CNC(=O)C(F)CC2CCOC2)n1 CC1CCCCC1C(=O)NCCCNC(=O)CCc1csc(=N)[nH]1 C(=O)(C(F)(F)C(F)F)NCC1(C)CCN(C(C2(C#N)CCOCC2)=O)C1 S(=O)(=O)(c1c(C)ccc2ncccc12)NCC1C(CCC)C1 C1(CC(=O)NC(CS(=O)(=O)N(CCCNC)C)=O)CNC2CCCCC12 c1(C(N2C3CC(CC(NC(C4CC5CC5C4)=O)C3)C2)=O)cc2c(F)cccc2s1 c1(C(=O)NCCN(C(COC(C(CC)C)=O)=O)CC(C)O)cccc(OC)c1F c1(NC(C2(C(C)(F)F)CC2)=O)csnc1-c1ccccc1 Cc1cc(C(N2CCCC2CNC(=O)CSc2cnn(C)c2)=O)on1 C(=O)(C(C(C)C)N1CCSCC1)NCC(=O)N(C1CC1)CC C#CCCCCC(=O)NCC(C)(C1CCC1)NC(=O)Cc1ccc(F)c(C)c1 C1(CCOC)(NC(=O)CCCF)CCN(C(c2cnn(CC3CC3)c2)=O)C1 c1(C(=O)NC2(C)CN(C(c3c(C)n[nH]c3)=O)C2)ccc2c(n1)CCC(C)C2 N1(C(C2N(C(c3c(OC)nsc3)=O)CCC2)=O)CCCN(CCO)CC1 Cc1cocc1C(=O)N(C)CC1(C(=O)NCC(C)CC2CCCC2)CC1 Cc1cccc(CC(=O)NCC(C2CC2)NC(c2conc2C)=O)c1Br Cc1cnc(C(=O)NCCN(C(c2cc3n(n2)CCC3)=O)C2CC2)cc1C c1(N(C)Cc2cc(Cl)cc(Cl)c2F)nc(N2Cc3cncnc3C2)nc2c1CSC2 C12(NC(C3(COC)CCCN3C(=O)CNC=O)=O)CCCCC1OCC2 Cc1noc(C)c1C(C)C(=O)NC1CN(C(c2conc2C2CCC2)=O)CC1C Nc1cncnc1C(=O)NCCc1n[nH]cc1C(=O)NC1CC(CO)C2CC12 Cc1ccnc(C(=O)NCC2CC(F)CN2C(=O)Cc2ccccc2F)c1Br CCC(C(=O)N(C)CC1(CNC(c2c[nH]nc2C)=O)CC1)C(F)(F)F Cc1cc(F)cc(Cl)c1NCC1CN(C(=O)OC(C)(C)C)C1 C(=O)(C(C)C(=O)OC)NCCN(C(C1CCC(c2ccccc2)O1)=O)CC C1(CC(=O)N(C2C3CN(C(=O)C(C)CC)CC23)CC)CCCN(S(C)(=O)=O)C1 Cc1ccnc(C)c1CNC(=O)CC1CCCN(C(=O)CCP(C)(C)=O)C1 C(=O)(C(C)(C)C(F)F)N1CC(C(C)NC(C(C(C)O)NC(C)=O)=O)OCC1 C123CN(C(=O)COC(F)F)C(C1)(C2)CNC(=O)C(OC)C3.C1(OC)CC(F)C1 N1(C(CC=C)=O)CCC2(CC1)CC(NC(=O)C(C)C(O)CCCC)C2 c1(OC)cccc(C(C)C(=O)N(CCCNC(=O)C(C)N2CC(C)C2)C)c1 c1(C(=O)NCC2(OC)CN(C(C3Cc4nncn4C3)=O)C2)cc2sccc2n1C C(=O)(C(F)(F)Cc1ccccc1)NCC1N(C(C(c2nc(C)sc2)=O)=O)CC1 c1(OC)ccc(CC(=O)NCC2C=CCN2C(=O)CN2CCCC2=O)c(Cl)c1 C1(CC(=O)NCCCNC(c2cncc(Br)c2)=O)Cc2ccccc2NC1=O c1(CC(=O)NC23CCCC2N(C(=O)C(F)=C(C)C)CCC3)cccc2c1OCCO2 c1(C(C(N2CC3CCC3(OC3CCOCC3)C2)=O)O)cc(F)ccc1F C1(CNCc2cnc(C(F)F)s2)CCCN(CSCCl)C1.c1(C(=O)O)ccc(CO)o1 N1(C2CCCN(C(C3C(=C)C3)=O)C2)CCN(C(=O)COCC(=O)OC)CC1=O C1(CC(=O)N(C2CCCC2)CCCNC(C(COC)C)=O)CCN(C)C1=O c1(C(=O)NC2C(C)N(C(=O)CC3=CCCC3)CC2)ccc([N+](=O)[O-])cc1O c1(CC)cc(C(=O)NC(C2CN(C(=O)CCc3cnn[nH]3)CCO2)C)cc(O)n1 c1(C(=O)NCCN(CC)CC)c(Cl)cc(OC)cc1Cl c1(C(N2CCN(C(c3oc(C)c(CO)c3)=O)CC2)=O)cccc(C(N)=O)c1C C1(CC(=O)NCC2(F)CN(C(c3cc(C(C)(C)C)n[nH]3)=O)C2)COCCOC1 C1(C(=O)NC2CC(C)(NC(=O)CC(C)n3ccnc3)C2)(OC)CCSC1 C#CC1(C(=O)NC2CC(O)(CNC(c3nccnc3C)=O)C2)CCOCC1 C12(C(N(C3C(C)(C)C3(C)C)C)=O)CC(CCO1)N(C(c1cccc(O)c1)=O)C2 CC(CNC(=O)C=Cc1cncs1)CC(=O)N1CCC1CC1CC1 C1(C(=O)NCC(C)(Cc2ccccc2)NC(C2CC(F)C2)=O)CC12CC(O)C2 N1(C(CNS(N(C)C)(=O)=O)=O)CC(C(N2CC3(CCC(=O)N3)C2)=O)CC12CCC2 C(N=c1[nH]c(=NCC(C(C)(C)C)N(C)C)[nH]c2c1COCC2)C1(COC)CC1 C(=O)(C(C)(C)CC(=O)OC(C)(C)C)NC(CC)CNC(c1c(N)sc(C)c1C)=O C12(CC13CCC3)C(=O)C2.c1(COC(=O)Nc2cc(OCC)n[nH]2)cccc(Cl)c1 c1(C(=O)NCC(CC=C)NC(c2c(Cl)n[nH]c2C)=O)cnc(C(F)(F)F)cn1 N1(C(c2cccc(C#C)c2Cl)=O)CCC2CN(C(C3CCCS3)=O)CCC12 C=Cc1cc(C(=O)NCC2(F)CC(CNC(C3(C)CCC3)=O)C2)cc(F)c1 N1(C(C2(OC)CCC2)=O)CCC12CN(C(c1cccc(C)c1N)=O)C2 c1(CC(=O)NC2CN(Cc3cc(Br)ncc3F)CC2O)cc(F)c(Br)cc1F N1(C(C)=O)CCC(C)(NC(c2ccc(C(=O)Nc3ccccn3)cc2)=O)C1 CCCCC(C(=O)NCC1(N(C)C)CCC1)NC(=O)Cc1cc(C)nn1C C12(C(N(c3ncccn3)C)=O)CCC(NC(c3ccc(F)cn3)=O)(CC1)CC2 C1(NC(c2c(OC)ccnc2)=O)CCCN(C(c2cc(Cl)n(C)n2)=O)C1C C(=O)(C1CCCc2nncn21)NCCCCC(=O)NC(CC)CNC(N)=O CC1(C(=O)NC2C3CC2N(C(c2cccnc2C2CC2)=O)C3)CCC(=O)NC1 c12ccccc1-n1cc(nn1)COC2.c1(C(=O)OC)cncn1C(C)C(=O)OC C(=O)(C(CC)C(=O)NC1CCN(C(c2ccn(CC(F)(F)F)n2)=O)C1C)OCC CCCCC(CC(=O)NCC(c1cnccn1)C)NC(=O)Cc1sccc1COC CCC(CC(=O)NCc1cccc(OC)c1)NC(=O)CC(C)(C)OC N1(C(C(=O)NCC2C(c3onc(C)n3)C2(CF)C)=O)CCC(C2CC2)C1CO C(=O)(C1=CCC2(COC2)OC1)N1CC(O)CCC(NC(=O)C=CC2CCCC2)C1 CC1CCC(NCC(c2ccccc2)N2CCC(N3CCCCC3=O)C2)C(C)C1 C1(NC(C(CC)CO)=O)CCCCC12CCN(C(c1ncoc1C1CC1)=O)C2 CC(C(=O)OC(C)(C)C)C(=O)NCCC(C)N(C(=O)CCCn1ccnn1)C CC(C(=O)NCC(C1CCCC1)NC(c1ccc(-n2cnnn2)cn1)=O)C(F)F C1(CNC(C(C(C)C)n2ccc(C)c2)=O)CN(C(c2cc(F)n[nH]2)=O)CC12CC2 c1(C(N2CCC(CNC(c3ccc(C#N)cc3)=O)C2)=O)ccc2c(c1)CCO2 C(=O)(C1=CCN(C(c2cnccn2)=O)CC1)N1CC(OC(=N)O)C1 c1(SC)cc(C)ccc1C(=O)NCC1(O)CCN(C(C2C3(CC3)C23CC3)=O)CC1 C1(C(=O)NCC2CC(C)(C)C2)CCCN(C(C2CC23CCC3)=O)C1 N1(C(=O)NC2CC2)CCC2(CC2N(c2ccc(Cl)cc2)CCC(C)(F)F)C1 Cc1c(NC(=O)CC2CC(C)N(C(=O)NCC(F)(F)F)C2)cccc1Br C1(F)(CNC(CSCCC)=O)CCN(C(=O)C(c2cnn(C)c2)OCC)C1 Cc1cc(C(F)(F)F)nc(NC(=O)CN2CCSC(CN3CCN(C)CC3)C2)n1 c1(C(=O)NCCCC(=O)NCc2n(C)ncc2C2CC2)cnc2[nH]cnc2c1 CCCCC(C)CCC(=O)NC(C)(CSC)C(N1CC2CC(O)CC1C2)=O c1(OC)ccc(-c2cnc(NC(=O)C(n3ccnc3C)c3ccccc3)o2)cc1 c1(C(N2CCCC(COC)C2C)C(=O)NCCOC)cccc(OC)c1Br c1(C(=O)NC(C)CN(C(=O)CC2CC=CCC2)C)ccc2nc(O)[nH]c2c1 C1(NC(c2cc(C(C)(C)C)no2)=O)CN(C(=O)CC2NC(=O)NC2=O)CCC1(F)F CC(C)(C)CC(=O)Nc1ccccc1NC(C1(CNC(=O)C(N)=O)CCC1)=O N1(C(CSCC(=O)OC)=O)CCC(C)C(NC(=O)Cc2cc(Cl)cs2)C1C N1(CC)CC(NC(=O)C(C2(O)CN(C(C3CC=C(C)CC3)=O)C2)F)CC1=O c1(C(=O)NC(C)CCN(C(=O)Cc2csc(C3CC3)n2)CC)cc(O)c(F)cc1N N1(C(c2nc(COC)sc2)=O)CC(NC(=O)C2=CCCC2C)CCC(O)C1 C1(C(N2C(CO)CC(NC(C(C(C)C)N(C)C)=O)C2)=O)CC2(CCCCC2)C1 CCCC(F)C(=O)N1CCC(C(C)NC(=O)Cc2cc(C)on2)CC1 Fc1ccc2ncnc(N3CC4(CF)CC4(C(F)(F)F)C3)c2c1 N1(C(c2cc(SC)c(C)o2)=O)CCC2(CCC2)C(NC(=O)CSCC2CCCO2)C1 CCC(C#N)C(=O)N1CCC(CNC(c2nc(C)oc2C)=O)C1 c1(C(=O)NCc2ncc(OC)nc2)c(C)ccc(C)c1O N1(c2ncnc(CC)n2)CCC(F)(CNC(=O)Cc2n[nH]c(C)n2)CC1 N1(C(C2N(C)C(=O)CC2)=O)CCC(C#N)(NCc2cccc(SC(F)(F)F)c2)C1 CCC(C)C(C(=O)NC1(C)CC(C(=O)NCC2CCOC2=O)C1)OC Cc1cc(NC(C2CC(C(=O)Nc3ccc(CC#N)nc3)C2)=O)ncc1Cl C1(CCC)CCCN(C(C2(C)CCN(C(c3nn(C)cc3Cl)=O)C2)=O)C1 c1(CC(=O)N(C2CN(C(C3CC(C)C3)=O)CC2O)C)ccc2[nH]ccc2c1 c1(C(=O)NCC(C)CNC(=O)CN2CC=CC2)ccc(C#N)c([N+](=O)[O-])c1 N12CCc3c(n[nH]c3C1)C2=O.Cc1cc(CNc2cccc(Cl)c2C)ccc1Br c1(OC)c(C(=O)NC(c2cncnc2)C)cnn(C)c1=O c1(C(=O)NCCCN(C(CC2CC(=C)C2)=O)C2CC2)cc(Cl)c(Br)cn1 c1(C(=O)NC2(C)CCN(C(C34CC(F)(C3)C4)=O)C2)cccc(Br)c1Cl c1(N2CCC(C(=O)NCc3ccc(C)cn3)C(C)C2)cnc(C#N)c(C#N)n1 C1(C(C)C)(C(N2CC(O)(CCNC(c3ccns3)=O)C2)=O)CNC(=O)C1 C1(C(N2CCCC(O)(OC)C2)=O)CN(C(=O)C2=CCCC2C)CCC1(C)C C1(NC(C2(COC)CCCC2)=O)CCCC(CNC(=O)Cn2cc(Br)c(=N)[nH]2)C1 CCCCCC(c1ccccc1)N(C)C(C1CC(n2cc(CN)nn2)C1)=O c1(C(=O)NC2CCC(CNC(c3nccs3)=O)C2)cc2ccncc2o1 N(C1c2ccccc2CC1(F)F)C(=O)NCc1c(CCC)nns1 c1(-c2n(C)ncc2)ccnc2c(C(=O)Nc3cc(Cl)cc(F)c3O)cnn12 C1(COC)COCCN1NC(=O)CCC(O)c1ccccc1Br N1(C(C(C2(O)CN(C(c3c(C(C)C)noc3)=O)C2)F)=O)CCCC(C)(C)C1C C1(O)(C2(c3cn(C4N(C(C(N5CCCCCC5)C)=O)CC4)nn3)CC2)CCCCC1 CON(CCC(=O)NC(c1cncc(F)c1)C)C(=O)Cc1ccccc1N(C)C C12(C(=O)NC(C(=O)OCC)CO)CC1CN(C(C1CC13CCCC3)=O)C2 C1(NC(CCc2nc(C)sc2)=O)CN(C(=O)CCC(=O)c2ccncc2)CC1O c1(C(=O)NC(CNC(=O)COc2cccnc2)CO)cn(C(F)F)nc1C(F)F Cc1c(C)c(C)c(C(=O)NCC(C)(O)CN2CCOCC2)c(C)c1C C(C)(CCC(=O)NCC(CC(C)C)NC(=O)C(O)Cc1ccccc1)OCC C1(CNC(c2ccccc2)=O)CCCN1C(c1csc(C(F)F)n1)=O C(=O)(C1=NN(CC)C(=O)CC1)NC1C(NC(C(CC)=CC)=O)CCOC1 CC(CC(=O)N1C2CCC1CN(C(c1cnn(C)c1Cl)=O)C2)CC(F)(F)F C1(CNC(CCCC(=C)C)=O)CCC2CN(C(=O)C(CC)=Cc3cn[nH]c3)CC12 C1(NC(=O)C(N2CCN(CCC(=O)O)CC2)=O)CCC12CCCC2 C#CCC(O)C(=O)NCC(C)C(=O)NCC(C)CCO CC(C)CC(C(N)=O)NC(C1(F)CCCN(C(c2cn(C(C)C)cn2)=O)C1)=O c1(SCCC(=O)N(C2CCC(NC(=O)Cn3nccc3F)C2)C)ccccn1 C(CC(=O)NC1CC(F)CN(C(=O)C(=C2CCCCC2)F)C1)(C(F)(F)F)OC C1(CC=C)(NC(=O)CC(C)(C)O)CCN(C(=O)COC2CCOC2)CC1 CC(C)CC(CCC(=O)O)NC(c1c[nH]c2nccc-2c1)=O CC(O)C(C)C(=O)NCCCC(C)(C)NC(=O)CCNC(c1ccncc1)=O N1(CCNC(c2c(NCc3c(CCC)cccc3)cccc2)=O)CCCCCCC1 C12(CNC(C(C)OCCCC)=O)CCC(CC1)N2C(=O)C(C)Oc1ccccn1 c1(C(C)C(=O)NCC=C2CN(C(=O)C(F)(F)c3cscn3)C2)ccc(F)cc1F C1(CNC(c2ccc(OC)cc2)=O)CCN(C(=O)C=Cc2cc[nH]c2)CC1(F)F C(=O)(C(F)(F)C(C(C)C)NC(C1CCCCC1CC(F)(F)F)=O)OC C=CC(CC)CC(=O)N1CC(CCNC(=O)CCOCC(C)C)C(C)C1 N1(C(c2c(C)csc2)=O)CCC(C(=O)NCc2cnnn2C)C(C)(C)C1 N1(c2nc(C)c(Br)cn2)CCC2CCC(C1)N2C(c1cc2nccc(Cl)n2n1)=O C1(C(N(CC(N2CCC(C#C)C2)=O)CCOC)=O)CCCCCN1C CC1(C(=O)NC2CC(NC(=O)CCCNC(=O)C3CC3)C2)COc2ccccc2O1 C1(NC(C2CC(=C)C2)=O)CCN(C(C2CC(C)(C)CCO2)=O)C1(C)C C(=O)(CC(CC1CC1)NC(c1c[nH]c(=NC)o1)=O)N(CC(C)O)CCOC CC1(NC(c2cc(C(N)=O)co2)=O)CCN(C(c2cnc(C(C)(F)F)s2)=O)CC1 c1(SCCCC)c(NC(=O)NC2CC(NC3CCC(F)(F)C3)C2)nc(=N)[nH]c1C c1(NC(C2CCCCN(C(C(C)OCC#C)=O)C2)=O)c(C)cccc1[N+](=O)[O-] C1(NC(CCC(C)SC)=O)CCOC12CCN(C(c1cc(C(N)=O)[nH]n1)=O)CC2 CCC(O)C(C)C(=O)NCc1c(C)coc1-c1ccc(C)cc1.CC1=CC12CN2 C1(C(=O)NCC2(C)CCN(c3snc(CC)n3)C2)Cc2ccccc2O1 N1(C(CC2(COC)CC2)=O)CC(NC(c2cnn(C(C)(C)C)c2N)=O)C(SC)C1 c1(C(N(CC(CC)NC(=O)C(C)(C)SC)C)=O)ccc(F)c(O)c1F c1(CC)cc(C(N2CCCC2CNC(=O)C(C)(C)CNC(C)=O)=O)ccc1OC C1(CC)CN(C(C2(C(F)(F)F)CC2)=O)CCC1CNC(=O)Cc1ncc[nH]c1=O c1(C2(C(=O)NC3C(CNC(COCC)=O)C3)CCC2)c(F)cccc1F N1(C(CC2N(CCOCC)CC2)=O)CCCC(NC(c2ccc(F)c(C)c2)=O)CC1 c1(C(N2CCCC(C(N3CCCC(CC)C3)=O)C2)=O)cc(C)c(O)nn1 c1(C(=O)NCCC2OCCN(C(C(C)(F)F)=O)C2)ccc(F)cc1-c1ccsc1 C(CCCCCC(=O)NC1CC12CCC(NC(=O)CCc1cocn1)CC2)SC n1(CC)c2ccccc2c2cc(CNC3CCCOC34CCOCC4)ccc12 N1(C(c2nnc(C)s2)=O)CC(C(=O)NCC2CC(C)CC(C)C2)C(C2CC2)C1 N1(C(c2nc(OCC)sn2)=O)CCN(C(c2cc3occc3s2)=O)CC1C C1(NC(CSc2n(C)nnn2)=O)CCN(C(c2nc(-c3ccccc3)no2)=O)CC1 Cc1nc2cccc(C(=O)NC(C)CCNC(C3CCCSC3C)=O)c2[nH]1 C(CCCCNC(=O)Cc1cn(CC2CCCOC2)nn1)N(C)C C1(NC(c2c(OC)scc2)=O)(CNC(C2(C#N)CC3(CC3)C2)=O)CCCCC1C c1(C(C(=O)NC(C)C=CC(=O)NC(C)COC(C)(C)C)O)ccc(C#N)cc1 c1(NC(C2(F)CN(C(C3C(C#N)C3)=O)C2)=O)ccc2nn[nH]c2c1 C1(CN(C)C(C2(O)CC(CF)C2)=O)CN(C(C2CCC2)=O)CCO1 C1(C)(CNC(C2(CC)CC(F)(F)C2)=O)CC(OC)CN1C(C)=O c1(C(=O)NCC2(CNC(C3CCCO3)=O)CC2)cnc(Cl)cn1 C1(CCNC(CCC=C)=O)CN(C(=O)CCCn2cncn2)CCS1(=O)=O c1(OC(C)C)ccc(C(O)Cn2cc(-c3noc(C(F)F)n3)nn2)cc1 c1(CN(C)Cc2noc(C3CCCCC3)n2)ccccc1.c12ccc(s1)[nH]c2=O C1(NC(c2c(C)scc2)=O)CCN(Cn2nnnc2C)CCC1c1ccccc1 n1(CC(N2CCC(CNC(C3CC(C(F)F)(OC)C3)=O)C2)=O)nc(C)c(Cl)c1C C1(NC(c2cc(C)[nH]n2)=O)CC1C1CCN(C(c2ccncc2O)=O)CC1 CCC(C(=O)NC(CCC1CC1)C(=O)N(C)Cc1nc(C)cs1)C(C)C N1(C(c2n(C)cc(Cl)c2)=O)CCCN(C(=O)C(C#N)CC2CC2)CC1 N1(CC(=O)NC2CC(CNC(C3(C=C)CC3)=O)OCC2)C(C)=CC(C)=NS1(=O)=O c1(OC2CCN(C(=O)NCC3C(COCC#C)C3)C2)cccnc1Br C(CCCCC(=O)NC1C(=O)NCc2cccnc2C1CCOC)NC(C)=O c1(C2N(CCC3(C(=O)OCC)CCCC3)CCOC2)cccc(F)c1F C1(C(=O)NC2CC(CNC(C3CC4C=CC3CC4)=O)C2)CCCCC12CCC2 c1(COCC(=O)N(C)CCNC(c2cnc(N(C)C)o2)=O)ccncc1 C(=O)(CC1OCc2ccccc21)N1CC=C(COC)CC1.C12(C)CC1C(=O)NC2 C1(c2cn(OC(COC)(C)C)nn2)CN(C(C2CCC(C)C2)=O)CCO1 C(=O)(C(C)CC(=O)N1C(CNC(c2ccc(F)cc2F)=O)CC2CC12)OC c1(C(=O)NC(CC)CNC(=O)C(C)c2ncco2)cc(C)ccc1Br C1(NC(C(C)OCCCC)=O)CN(C(C23CC(C(=O)OCC)(C2)C3)=O)CCC1(F)F C1(O)(CNC(=O)CC(F)F)CCN(C(c2ncc(Cl)cc2Cl)=O)CC1 Cc1cc(C(=O)NCC2(CNC(c3nc(C4CC4)c(C)s3)=O)CC2)n(C(F)F)n1 C#CC1CCC(NC(=O)CCn2cc(CO)nn2)CC1 C1(CC=C)(NC(c2cc3n(n2)CCO3)=O)CCCN(C(=O)CN(C2CCC2)C)C1 CC(C)C(O)CC(=O)NC1CN(C(=O)C(N2CCCCCC2)C)CC1C N1(C(CCC(C)OCC)=O)CCC(C)CC1C(=O)NCC=Cc1ccccc1 C1(C(=O)NC2CC(NC(c3ccc[nH]3)=O)C2)CCC(Oc2ccncc2)C1 c1(CC(C)C(=O)NC2CCN(c3cncc(C#N)n3)CC2O)ccc(F)cc1Cl C1(NC(=O)NC(C)(C)C(F)(F)c2ccccc2)NCCC1C1CC1 C1(CC(=O)N(CC(C)NC(C(C)C(C)(C)C)=O)C)CCCCCC1(F)F c1(OC)cccc(C(=O)NC2CCC(NC(c3coc(CC4CC4)n3)=O)C2)c1F c1(C(=O)NC(C)CNC(=O)C(F)(F)CN(C)C)ccc(NC(N)=O)cc1Cl c1(C(=O)NCC2CCN(c3nccc(OCC)n3)C2)cnc2cccc(Cl)c2c1 C1(C(=O)NC(C2(C(=O)NCC3N(CC)CCC3)CC2)C)CC2CC(=O)C1O2 c1(CCN2CCC(O)(C(=O)N)C2)cccc([N+](=O)[O-])c1.N1(CCC2CC2)CCOCC1 CC1CCCC=C1C(=O)NC1(CO)CCN(C(=O)Cc2ccsc2)C1 c1(CC(=O)N(CC(C)(C)CNC(C2C=CCC2)=O)CC)cccc(C#N)c1OC C(=O)(CC(CC)N(C)C(c1cncc(Cl)c1)=O)N(CCCO)CCC C=CCC(CC(F)F)C(=O)NC(C)CC(C)NC(=O)C(C)OC(C)=O C(C(CC)N=c1nc(CC)[nH]s1)NC(Cc1c(SCC)cccc1)=O c1(C(=O)NCCCCCC(=O)OC)c(Cl)ccc(N2C(SC)CC3CC32)c1F C(=O)(C(C(C)CCC(=O)OC)N1CC(C)C(S(C)(=O)=O)C1)NCCCSC C(c1ccccc1C#N)=CC(N1CCCC(CN2CCN(C(C)=O)CC2C)C1)=O C(=O)(C1CCCc2nn[nH]c21)NC1CN(C(CC=CCC)=O)CC1(C)C c1(CN(C(=O)C2=CCOC2)CC(C)O)cc(C(N)=O)cc(F)c1 C12(C(=O)NC3(c4nc(C)[nH]n4)CC3)CCCC1N(C(c1coc(CO)c1)=O)CC2 N1(C(Cc2snc(C)n2)=O)CCCCC1C1(CNC(=O)CSC(C)C)CCOCC1 C1(C(=O)N(C)Cc2nnc(O)o2)(CC)CCCN1C(=O)CN1CCCNC1=O c1(OC)cncnc1C(N1CCC(C)(C(=O)NC(C)CC2CCC2)C1)=O N1(C(C2N(C(CC(OCC)OCC)=O)CCOCC2)=O)CCCC(N=[N+]=[N-])C1 c1(OC)ccc2cc(C(=O)N(C3CCN(C)CC3)C(C)(C)CO)ccc2n1 C1(NC(C2CCCC2(F)F)=O)CCN(C(c2cncc(F)c2Cl)=O)C12CC2 c1(NC(C(CSC)(C)NC(=O)CC2CC(F)(F)C2)=O)cc(C)cnc1C C#CCCN=C(NCc1ccc(CN(c2ccccn2)C)cc1)NCC C=C(C)CCCC(=O)NC(C)C(C1CCCCC1)NC(c1cncc(O)c1)=O N1(C(c2occ3c2CCC3)=O)CCC2(NC(=O)COC3CC3)CCCCCC12 N1(C(C(c2cccc(Cl)c2F)NC(=O)OC(C)(C)C)=O)CCCOCC1(C)C C(=O)(C=C1SCC(=O)N1C)N1CC(CN2CCC(NC(c3c(C)nc[nH]3)=O)CC2)C1 Cc1cccc(C)c1CCNC(=O)C(C)(C)NC(=O)Cc1cn(C)cn1 N1(C(=O)CC2CCCC23CC3)CCC2(CCCN2C(c2cccc(Cl)c2O)=O)C1 c1(C(N(C2CC(NC(=O)CCc3csc(Br)c3)C2)C)=O)cnccn1 N1(C(C=C(CC)C)=O)CC2CCCC(CNC(=O)C=CC(C)C)C2C1 N1(C(C(C)n2ccnc2)=O)CC(C(=O)NCCCOC(=N)O)C(F)C1 N1(C(CC(=O)OC)=O)CCc2ccc(C(=O)C3CC3)cc2CC1 C1(CC(=O)N(C(COC)C)C2CC2)CN(C(=O)C(C)(C)N(C)C)CCO1 Fc1c(CNC(=NCC2COC2)NCC2CCCO2)ccnc1Br Cc1cnc2n1CC(C(=O)NCC(C1CCC1)NC(=O)C(F)(F)C(F)(F)F)CC2 CC1(C)CC(NC(=O)C=CC2CCOCC2)CN1C(c1cc(CO)ccn1)=O c1(C(=O)NC2(CC=C)CN(c3ccnc(-c4nccs4)n3)C2)nnc(O)nc1O Cc1cn(C)nc1C(=O)NC(C)C(C)(C)NC(C1CC(=O)N(c2nccs2)C1)=O Cc1cc(C(=O)NC2CC(F)CN(C(C3CC3C)=O)C2)n2ncnc2n1 c1(C(=O)NCC2(C)CCN(C(CC(=O)N(C)C)=O)C2)cnc2[nH]c(=O)ccc2c1 Cc1cc(C)n2nc(C(N3CCCC3C3CCCN3C(=O)CN(C)C)=O)cc2n1 c1(C(N(CC(C)(C)NC(C=CCOC)=O)C)=O)cc(CCO)on1 C(=O)(C1=C(Cl)CCCC1)N1CCN(C)CC1CNC(C1CCCC1F)=O n1(CCC)ncnc1CN(C1CCN(C)C1)CCNC.C(C)(=O)N C#Cc1cc(C(N2CCC(NC(=O)COc3ccc(C)cc3F)C2)=O)cc(F)c1 c1(NC(CCCNC(C2C(=C)C2)=O)C)ncc(C(=O)OCC)cc1Cl c1(C2C(=O)N2CCCO)cccc(C(F)(F)F)c1.CC(C)C(=O)NCC(F)F c1(C2C(N(C(CNC(c3n(CC)nnn3)C3CC3)=O)C3CCC3)C2)ccc(F)cc1 N1(C(CCC2CCN(C(C)=O)C2)=O)CCOC(C)C1C(N1CC(F)(F)CC1C)=O C1(C(N(C)Cc2cscn2)=O)CCC2CCC1N2C(c1ccncc1)=O Cc1cscc1C(=O)NCC1CCN(C(c2nnc(C(C)(C)C)s2)=O)C1 C(C(=O)NC(C)CN(C(=O)COc1cccnc1)CC)(C(C)(C)C)SC C1(C(=O)NCC2N(C(Cc3c(C)nc(C4CC4)s3)=O)CCC2)CCC2CC2CC1 C1(NC(C(C)c2cncs2)=O)CCCN(C(=O)CSc2n[nH]c(=N)s2)C1 C1(SCCNC(C(N)C2CCCC2)=O)CC=CCC1 n1(CC)cnnc1C(=O)NCC12CC(C(=O)N(C(C3CCCC3)C)CC)(C1)C2 CS(C)(=O)=NC(=O)C(=O)NC1CN(C(C23CC(C(F)F)(CO2)C3)=O)CC1CC1CC1 N1(c2c(OC)c(Cl)ncn2)CC2CCC(NC(c3cc(F)n(C)n3)=O)CC2C1 C(=O)(C(C)C(C)S(C)(=O)=O)N1CCC(O)(C)C1.Cc1cccc(C)c1 CN(OCc1ccccc1)C(=O)C(CCOCCO)NC(C1CCOC1)=O C1(C(C)C)CN(C(=O)C(N2CCOCC2)C)CCCN1C(=O)CC1(C)CCOC1 Cc1nn(C)c(C)c1C(=O)C(=O)NCC(CO)NC(=O)C(O)CC1CCCCC1 c1(C(CNC(C=[SH]C2CC2)=O)N(CC)CC)cc(F)cc(Cl)c1.C12(CC1)C(=O)N2 Cc1cc(O)c(C(=O)NC2CCCC(CNC(=O)Cc3cnc[nH]3)C2)nn1 C1(CNC(=O)C=CC(F)(F)F)CCCN(C(C2CCCCS2(=O)=O)=O)CC1 Cc1ccc2ncnc(N3CCC(CN(C(=O)CC4CC5CCC4C5)C)C3)c2c1 CN1CCCCC1C(=O)NC1CCCCC1NC(=O)CCc1cccc(O)c1 C(=O)(C(C(C)(C)C)NC(c1cccc(O)c1)=O)NCC(C)N(C(=O)CN(C)C)C CC(C)C#CC(=O)NC(Cc1cn[nH]c1)C(=O)NC1CC1c1cccnc1 c1(C(=O)NCC2CC(CC(=O)NC(C3CCOC3)C#C)C2)cc(CC)[nH]n1 N1(C(c2cnc(C)cn2)C(=O)NCCCC)CC2OCC(C(=O)OCC)C2C1 C#CC1(C(=O)NCC(O)CC(=O)NCC(c2ccccn2)C)CCCCC1 C1(CNC(C(C)CF)=O)CN(C(c2cccc(Br)c2Cl)=O)CC12CC2 C(=O)(CC1=CCCCC1)NC1CC(C)N(C(=O)CN2CC=CC2)CC1 N1(CC)CCC(N(C)C(=O)NCCN2CCOCC2)C1 CCCCCC(O)C(=O)NC1CCCC1NC(C1CCC(CC)CC1)=O N1(C(CC(C=C)CC)=O)CC2CCC(C1)N2C(=O)CN(c1ccc(Cl)cc1)C N1(C(C(C(C)C)(C)O)=O)CCN(C(c2ccc(C#N)[nH]2)=O)CC12CCC2 C1(CC(N2CCC(CC(C)C)C2)=O)CC2(CC2)CN1C(=O)C=Cc1cncn1C CC1COC2(CCC2)CN1C(=O)C(Cc1ccoc1)NC(=O)C(Cl)Cl CCC(C)(CC)C(=O)NC(C)CCNC(c1cccn1CC1CCCC1)=O Cc1cc(=NC(=O)C(=O)N2CC(O)(C(C)NC(=O)CC(C)C3CCCC3)C2)[nH]o1 c1(N(CCCC)C(=O)OCC2CCOC(c3cccnc3)C2)ccc(Br)cc1 CC(C)(CCC(=O)N1CCC(CNC(c2ccc(Cl)nc2)=O)C1)[N+](=O)[O-] C(=O)(C1CCCc2sc(C)nc21)NC1C2C(NC(C(F)=CC)=O)CC(CC2)C1 c1(OC)ccc(-c2cccc(CN3CCC(O)(Cn4ccnn4)C3)c2)c(CO)c1 c1(C(N2CC3(CCN(C(c4nc(Cl)c(Cl)s4)=O)C3)C2)C)ccc(S(C)=O)cc1 CCCC(C(=O)NC1CCCC(CNC(=O)CCC2CC2(F)F)C1)S(N)(=O)=O c1(C(=O)NC(c2nccs2)Cc2ccccc2)coc2c(F)c(Cl)ccc12 C(CC(C)(C)C)(C(=O)NC1CCC(OC)C1)NC(C(CC)CC)=O Cc1nc2cncc(C(N3CC=CC3CNC(=O)COCC3CCCC3)=O)c2[nH]1 c1(C(=O)NCC(C2CCCC2)NC(C(C)(C)OC)=O)ccn2ccnc2c1 CC1CN(C(=O)C(C(C)O)NC(c2ccsc2C#N)=O)CC1F N1(C(C)C)CCCCC1C(=O)NCCN(C)C(C1CC1C(N1CCOCC1)=O)=O C1(C)(CNC(CCn2ncc(C)c2)=O)CN(C(c2c[nH]c(C#N)c2)=O)CCO1 C(c1ccc(Cl)nc1)=CC(=O)NCCNC(c1ccn(-c2ccncc2)n1)=O c1(OC(C2(CC#N)CCC(C)(C)C2)=O)ccc2c(c1)OCO2 C12(NC(C=CC)=O)C(C(=O)O)C3CCC1C2C3.c12cccc(c1)C=CC(=O)N2 N1(CC=CC(=O)NC2CCC2CNC(c2ccc(C(F)F)s2)=O)CCOCC1 C=C(C)C(C)(C)C(=O)N(CCC(C(C)C)NC(=O)CCc1ccc[nH]1)C S(=O)(=O)(CC(=O)NCC(C)(O)CNC(c1ccc(SC)cc1)=O)NC C(=O)(C1=CC2(CCN(C(c3c(F)cccc3F)=O)C2)C1)N(C(C(C)C)C)C N1(C(C(CC)(C)F)=O)CCC(CCNC(=O)CC2(C(F)(F)F)CC2)C(F)(F)CC1 c1(N2CCC(SC)CC2)[nH]c(=NCc2cccc([N+](=O)[O-])c2C)nc2scnc12 C1(COC)(NC(=O)Cn2ncccc2=O)CCN(C(=O)C(C)=C2CCCC2)CC1 CC1(C2CN(C(=O)CC3CCCC3NC(=O)CC3CCCNC(=O)C3)C2)CC1 Cc1ccc2c(c1)CC(C(=O)NC1CCC(CNC(=O)C3=COCC3)C1)S2(=O)=O C1(CC(=O)NCCNC(CC2(CC(=O)OC)CC2)=O)CCC(C(F)(F)F)N(C)C1 C=C(C)CC(C(=O)NC(C)C(=O)C(=O)OC)NC(c1cccc(C)n1)=O C(C(C)(C(F)F)NC(C1CCC(NC(C)(C)C)C2CC12)=O)SC c1(C(N(CC(C)N(C)C(c2cc(C#N)no2)=O)C)=O)cc2c(F)c(Cl)ccc2[nH]1 Cc1cc(C(=O)NCC2CCCN(C(c3cc(C#N)on3)=O)C2)nc(Cl)c1 C1(C(C2CC2)NC(N(C)Cc2cnc(C(C)(C)C)s2)=O)CC(F)(F)C1 CC1CC=C(C(=O)N2CCC(CC(=O)NCC3OC(=O)CC3(C)C)C(O)C2)CC1 N1(C(c2c(C)nc(C)s2)=O)CCN(C(=O)COCCCC(C)C)CC(C)C1 C(=O)(C(C(C)C1CCCC1)N(C(c1ccccc1)C(C)C)C)NC1C(CC)COC1 c1(OCC)cc2c(c(OC)c1OC)CN(C(CC)CCNC(C)C(C)C)CC2 c1(C(N2CCC(CNC(C34CCC(C3)C4)=O)C23CC3)=O)cc2ncccc2o1 Cc1ccc2c(CC(N3CC(NC(=O)CC4(O)CCOC4)C3)=O)coc2c1 c1(C(N2CC(CC(NOCCCOC)=O)OCC2)=O)c[nH]c(C)cc1=O C1(NC(CNC(CCC)=O)=O)CC(F)CN(C(C2(CC(=O)OC)CCCCC2)=O)C1 c1(C(N2CCC(C(C)NC(C=CCCC)=O)CC2)=O)c(OC)ncc(Cl)c1C CN1CCN(C)C2(CCCN(C(C34COCCN3CCC4)=O)C2)C1 C1(C)(NC(C(C)OCCOC)=O)CCCC12CCN(C(=O)C(=O)NC1COC1)CC2 c1(C(N(CCNC(CCSCCC)=O)C)=O)coc2cc(OC)ccc12 N1(Cc2ccc(N(C(=O)Nc3cnc(C(C)C)s3)C)cc2)CC2(CC(CO)C2)C1 C1(CNC(C2CC(C#C)(O)C2)=O)CCCCN(C(=O)C(F)(F)C2(OC)CCC2)C1 N1(C(C(c2ccccc2)C)=O)CC(F)CC1CN(C(=O)C=CSc1nc[nH]n1)C C1(C(N2C(CC)CCCC2)=O)CCN(C(=O)c2cc(C(N)=O)co2)O1 CC1CC2(CCN(C(=O)CC3(O)CCOC3)CC2)CN1C(=O)CC(C)N(C)C c1(CC(C)NC(c2cc(C)sn2)=O)ccc(CNC(=O)COC2CCOC2)cc1 c1(CNC(c2scc(C)c2)=O)ccc(C(=O)NCCCC(O)CO)nc1 c1(NC(C2N(C(C=NOC)=O)CCC2)=O)cn(CCF)nc1C#N c1(C(=O)NCC(=C2CN(C(=O)CCCC3CCOC3)C2)F)cc(O)cc(Cl)c1 C(=O)(CCC(=O)NCCCCC1CCCN(C(=O)CC(C)(C)OC)C1)NCCC c1(C(N2C3CCN(C(C(CC)(F)F)=O)C(C3)C2)=O)cnc(O)c([N+](=O)[O-])c1 N1(C(CCCNC(C)=O)=O)CCC2CCN(C(=O)C3CC3)C2C1 c1(C(N2CCN(C(C3CCN(CC#C)CC3)=O)C(C)C2)=O)ccc(Cl)c(C)c1O C(=O)(CCCCCC(C)C)NC(C(=O)NC(CC#C)(C)C)C c1(C(N2CC(NC(c3cc(CC)cc(Cl)c3)=O)C2)=O)c(C)ccc2nsnc12 Cc1cnc2c(C(=O)NC(C)(C)C(C)NC(C3CCC(C)(C)C3)=O)cccn12 c1(C(=O)NC2CCC(CCNC(c3c(Cl)cn(C)n3)=O)C2)nc2cnccc2s1 C1(C(=O)NCc2ncc(Cl)cn2)C2CC2CN1C(=O)COC1CCOC1 N1(C(=O)CC2CCCOC2)CCN(C(c2cnc3n2CCS3)=O)C(CC(F)F)C1 C1(CCC)(NC(=O)C(C)CC(C)C)CCCN(C(=O)C=Cc2ccc(SC)s2)C1 c1(OC)sc(C(N2CCn3c(C(C)(C)C)nnc3C2)=O)c2c1CCCCC2 N1(C(C(c2ccc(Cl)cc2)C)=O)CCC2C(CCN2C(C2C(C)C2C)=O)C1 C1(C(NOCC(=C)C)=O)CC(OC(C2(N(C)C)CC2)=O)C1(C)C c1(CN2CC3C(C(=O)Nc4c(C(=O)OC)ccs4)(C3)C2)c(F)cncc1F N1(C(C(C)SCc2ccccc2Cl)=O)CCC2CN(C(=O)C(C)(C)CO)CC2C1 C1(CCC(=O)N(C2COCC2O)C)CCN(C(=O)CCC2(C#N)CCC2)C1 c1(CNC(CC)=O)ccc2c(c1)CCCC2NC(C12CCN(C1)S(=O)(=O)C2)=O n1(CC#C)c(C)cc(C(=O)N(CC(C)NC(c2ocnc2C(C)C)=O)C)c1C C1(NC(C)=O)CCC12CN(C(c1ccn(-c3cccc(F)c3F)n1)=O)C2 Nc1cc(F)c(O)cc1C(=O)NC1CCC(CCNC(=O)CC(=O)NC2CC2)C1 CCC(CC(C)O)NC(=O)CC1(CO)CC1.c12ccccc1NC(=O)CO2 C1(C(=O)NC2C3(CC(NC(C4CN(C(C)C)C4)=O)C3)C2)CC(=O)NC(=O)N1 CCC(CC)(CO)C(=O)NCCCOCCC(=O)NCSC(C)CC(=O)OC CCCC(CNC(=O)C(C)c1ccsn1)NC(c1cnc(C)[nH]1)=O c1(C(C)(C)C)ccc2c(S(N)(=O)=O)cccc2c1.C1(=O)CCC2CC(C2)N1 C1(C)(CC(=O)NC2C(NC(Cc3cn(CCOC)nc3)=O)CC2)CCCCC1 c1(CC(=O)NCC(C)N(C)C(c2cccn2C)=O)ccnn1-c1ccccc1 C#CC(CNC(=O)C(Cc1cn[nH]c1)NC(c1ccc(O)cc1)=O)C(C)C C1(CC(=O)NCC(N(C(CN(C2CC2)CC)=O)C)C2CC2)CCCCC12CC2 C1(C(=O)NCCC2CCCC2O)CCCCN1C(c1c[nH]nc1Cl)=O C1(C(N(C)CC2(CO)CC2)=O)CCN(C(=O)C2(C#N)CC2(C)C)O1 C1(C(C)NC(c2c(CC)scc2)=O)CCN(C(=O)CCOC)CC1 C(=O)(C(CC(C)C)C1CCC1)NC(CC)CN(C(=O)C=CC(c1cccnc1)=O)C C(=O)(CC(O)CC(C)(C)C)N1CCC(CN(C(c2cc(C)n(C(C)C)n2)=O)C)C1 c1(C(N2C(NC(COC3CN(C(=O)NC)C3)=O)C=CCC2)=O)cccnc1S C1(N(C(CSCCOC)=O)C)CN(C(c2cn(C(F)(F)CO)nn2)=O)CC1F C1(N(C(CCCC)=O)C)CCCC2CN(C(c3ccncc3N)=O)CC12 C1(C(N(CCCN(C(c2c(OC)nsc2)=O)C)C)=O)CCC(=O)N(CCOC)C1 N1(CCN(C(C(=O)NC(C)C)CCc2ccccn2)C)CCC(C#N)(CC)CC1 Cc1cc(Cl)cc(C(=O)N(C)CC2CCN(C(C34CC5CC3C4C5)=O)CC2)c1O c1(C(C(=O)NC2CCC(NC(c3n(CC)ccn3)=O)C2)F)cccc(C)c1 c1(C(CC)C(=O)N(C)CCOCCCNC(=O)C=CC(N)=O)cccc(Cl)c1 C(=O)(C(CNC(=O)C=CC(C)C)N(C)C)NC(c1ccn(C)n1)CC C12(C(N(CCCNC(C3CCCN3c3ncccn3)=O)C)=O)CCCN(CC1)C2 N1(C(C2C(C)CC(=O)NC2)=O)CCC2CCN(C(c3ncc(Cl)s3)=O)CC12 c1(C(N2CC(CC=C)(NC(c3csc(C)n3)=O)C2)=O)csc2ccccc12 Cc1cc(C(N2CCCN(C(c3cc[nH]n3)=O)CC2)=O)c2c(C(C)C)noc2n1 C(=O)(C1=CCCC(C)(C)C1)N1C(C(C)C)CN(C(=O)CCSCC(N)=O)CC1 C1(NC(CC2OCC(C)(C)C2)=O)CCN(c2nnc(CO)s2)C12CCC2 N1(C(C2(C(C)C)CC2)=O)CCC(C(C)(C)C(=O)NCC2CCC(=O)O2)C1 C1(C#N)(NC(CNC(CNC(C(C)n2cncn2)=O)=O)=O)CCCC1 C1(CNC(C(C(C)(C)C)O)=O)C2CCCC1N(C(c1ccnn1CC#N)=O)C2 C1(NC(C2CCN(C(C)=O)CC2)=O)C2CC1CN(C(c1cc(C)c(C)o1)=O)C2 C(=O)(CC1=CCN(C)CC1)N(CC(C(=O)NC(CC)(C)CN(C)C)C)C Cc1n[nH]c(C)c1CC(C)C(=O)NCC1(NC(=O)CC23CCC(CC2)C3)CC1 N1(C(c2n(C(C)C)nnc2)=O)CC(CNC(c2c(N)cccc2Cl)=O)C(C)(C)C1 C1(C(=O)NC(C2N(C(Cc3c(C)n[nH]c3C)=O)CCC2)C)CCC=CCCC1 C1(C(=O)NC(C(=O)NCCCC(F)F)Cn2ccnn2)CC2C=CC1O2 CCCC(C)CC(=O)NC(Cc1ccco1)C(=O)N(C)Cc1cncs1 CC1CCOC(C(=O)NCC2(F)CC(NC(c3ccc(C4CC4)cc3)=O)C2)C1 CC(C)(C(=O)NC1CC(NC(=O)CC2CC2C)C1)n1cccn1 c1(C(=O)NC(CCSC2C(C(n3nccn3)=O)CCC2)CC2CC2)cncn1C c1(NC(c2n(C=C)nnc2)=O)cccc(Cl)c1C(=O)NC c1(C(=O)NCC2N(C(C(C)c3cc[nH]n3)=O)CC=C2)noc2c1CCCCC2 CC(C)C(CC(=O)NC1C(O)CC1O)NC(C1CCC1C#N)=O c1(CN(C2CNCC(F)(F)C2)C(CC(C)C)=O)cc(F)c(F)cc1O C1(C(C)C)C(C(=O)NCC2CC3CCCC23)CCN1C(=O)Cc1ccccc1 N1(C(=O)Cc2cn[nH]c2)CC2(CNC(C3CCC([N+](=O)[O-])CC3)=O)CC(F)(C1)C2 C12CCCCN1C(=O)NC(C)(C)CC2.c1(CCCOCCO)ccc(F)cc1 C(=O)(C(C)CN(C)C(c1cc(C(C)C)no1)=O)N1CC(=CC)C1 C1(NC(c2c(C)sc(Cl)n2)=O)COCCN(C(C2CC3CCC2CC3)=O)C1 c1(C(N2C(CCNC(C(C)C(C)(C)C)=O)COCC2)=O)ncn2c1CCCC2 C(CNC(=O)C(C)(C)C1CCN(C(c2cnn(CCO)c2)=O)C1)(C(C)(C)C)OC C(=O)(CCCCCC#N)NCCCC(c1ccccc1)OCC.N1(C)CCCCC1=O CCCC(C(=O)NC(C)(CNC(=O)C(COC(C)(C)C)N(C)C)CO)OC CCCCC(CC)C(=O)N1CCC(N(C(=O)C(c2cnn(C)c2)OC)CCO)C1 N1(C(CCCC(C)O)=O)CC2CCCC(NC(=O)CCc3ccn(C)n3)C2C1 CCC(CO)(C(=O)NC1CC=C(C(=O)NC2CCCCCCC2)C1)OC c1(OC)ncc(C(N2CCC(C(=O)NCCCCN3CCC3)C(C)C2)=O)cc1Cl C1(OC(CNC(CN(C(=O)OC)C)=O)=O)(NNCCC(C)c2cn[nH]c2)CCC1.OC C1(C(=O)NC2(CNC(=O)CCC3CCCC3)CC2)CCn2c(O)nnc2C1 N1(C(c2n(CC)cnn2)=O)CC(CNC(=O)CCc2nnc(C(C)C)o2)CC1C N1(C(C2C(C)CCC2)=O)CCN(c2ncnc(Cl)c2[N+](=O)[O-])CC12CCC2 C1(CC)C(C(=O)NCc2cccnc2)CCN1C(=O)C(O)C1CCC1 C1(NC(C2(C)CC2(Cl)Cl)=O)CC(NC(=O)Cc2cnsc2)C12CCC2 N1(C(C(=O)NC2(NC(C3CC4CCC3CC4)=O)CC2)=O)CC2CN(CCF)CC2C1 CC(O)C(C)(C)C(=O)N1CCC(N(C(=O)CC2(CS(C)(=O)=O)CC2)C)CC1 c1(C(=O)NCC(CC=C)NC(=O)COC2CCOC2)cc(N)ccc1SC c1(OC)c(C(=O)NCCN(C(C2CCOCC2C)=O)C2CC2)cc(F)cc1F c1(C(=O)NCCN(C2CC2)Cc2nc(C)on2)snc(O)c1Cl Cc1cc(F)cnc1C(=O)NC(c1cn(CC2(CC(=O)O)CC2)nn1)C c1(OC)ccc(C)cc1-n1cc(CNC(=O)C(C)SC)nn1 C(C(=O)N1CCC(=CCNC(=O)COC(C)C)CC1)(C(C)C)NC(=O)OC C(=O)(C1CCC(=O)c2ccccc21)NCC1N(C(CNC(N)=O)=O)C2CCC1C2 C1(SCC)CCC(C(N2CCC(C)(CNC(C3(F)CCOC3C)=O)C2)=O)CC1 N1(C(C2CC3CN(C(C4C(C)(C)C4C#N)=O)CC3C2)=O)CC2(COC(C)(C)C2)C1 c1(C(=O)NCC2CN(C(c3cc(C)ncc3C)=O)CC2C)c(O)cc(F)cc1F c1(OC)cc(Cl)ccc1C(=O)NC1C2CCN(C(=O)C(O)Cc3ccccn3)C12 C12(CNC(C3(OCC)CCOCC3)=O)CC(CC)(CN1C(=O)C(O)C(F)F)C2 Cc1cc(Br)cc(C)c1CC(=O)OCC1CCC(=O)C1 N1(C(C2CC(CC)C2)=O)CCCC(C)C1CCNC(c1cnc(O)cc1OC)=O C1(F)(C(=O)NC(C(C)OC)CO)CCN(C(c2cc(C)ccc2C)=O)CC1 C#CCCC(O)C(=O)NCC1CCC1NC(c1cccc(CS(C)(=O)=O)c1)=O n12nc(-c3cnn(CC(F)(F)F)c3)nc1C2.c1cc(CC2CCC(O)C2)ccn1 c1(CC)cc(C(=O)NCC2CCN2C(=O)C(C)OCOC)c(Br)s1 c1(OC)ccc(O)c(C(N2CCCCCC2CNC(C2CC2F)=O)=O)c1 C1(CC(=O)NCCCN(C(C#CC(C)C)=O)C2CCCC2)CCCC2(CCC2)O1 CCC(C)CCCC(=O)N1CC2(CC(C(=O)NCC3Cc4nccn4C3)CO2)C1 c1(SC)ncc(N)c(C(N2CC3C(N(C)C(c4ccc(F)s4)=O)C3C2)=O)n1 c1(NC2CCC(NC(c3c(C)occ3)=O)CC2)ncnc2[nH]ccc12 C1(C(=O)NC2CCC(NC(c3n(CC)ccc3)=O)C2)CCCS1(=O)=O N1(C(c2ccc(C)o2)=O)CCCCC1C1(NC(c2cnn(C(C)C)c2)=O)CC1 CCCC(C(=O)NC1CN(C(c2cc(C)oc2C)=O)CC1C)OCC C(=O)(C1CCCc2c[nH]nc21)N1CCC(CNC(c2c(C)nsc2N)=O)C1 N12CCC3(CC1)CC3C2=O.C(CC(=O)N1CCC1C(=O)NC(C)(C)C)=C(C)C N1(C(C2CC(OC)C2)=O)CC2CCCC1(CNC(=O)C(C)(C)c1cccs1)C2 C1(CN=[N+]=[N-])CCCN(C(c2cc(CNC(=O)Cn3ccnn3)no2)=O)C1 Cc1cnc(Cl)c(C(=O)NCC2(O)CCCN(C(=O)C(C)NC=O)C2)c1 Cc1ccc(C(N2CCC(O)(COC)CC2)C(=O)NCC2CCCO2)c(C)c1 C1(CCCC)CN(C(=O)C(C#N)C2CC2)CCN1C(=O)C1=CCCC1 c1(C(N2CCC3(CC2)CC(=O)O3)C(=O)NCC=C)ccc([Si](C)(C)C)cc1 C1(C(N2CCC(c3cnn[nH]3)C2)=O)(OC)CCN(C(c2nc[nH]n2)=O)C1 Cc1ccc(C(N2CC3(CNC(=O)C(C4CCC(=O)N4)C)CC2CO3)=O)nc1F c1(-c2n(CCC)c(SCc3nn(C)c(=O)n3C)nn2)ncnc2ccccc12 Cn1cnc2cc(C(=O)NCCOCCNC(C3CCCC(F)(F)C3)=O)cnc12 C1(CNC(C2N(C)CC(O)C2)=O)CCN(C(c2ncc[nH]c2=O)=O)C1(C)C C1(CNC(c2n[nH]c(C)c2Cl)=O)CC2(CC2)CN1C(=O)CCc1nc(O)n[nH]1 c1(OC)ccc(C(C)NC(=O)NC(CC(N)=O)c2ccccc2)cn1 c1(OCC(=O)N(C2CN(C(CCSCC)=O)CC2F)C)ccc(Cl)cc1F C(=O)(C1c2ccccc2C2CC1C2)NC(C)C(C)NC(=O)C(F)(F)C1CC1 c1(OCC)ccc2[nH]c(C(N3CCCC(NC(=O)C(C)C#N)C3)=O)c(C)c2c1 C1(CNC(C2N(C(C)C)CCC2)=O)(CNC(C2CCCO2)=O)CCCCC1.C c1(CCC)ccc(S(=O)(=O)N2CCSCC2C(=O)NCc2cncnc2)cc1 CCCC(CC(=O)NC(C)CF)NC(c1cnc[nH]c1=N)=O N1(C(C2(C)CCC2)CC)CCC(C(F)F)(CNC(=O)CCCCn2ccnn2)C1 N1(C(CCC(=O)NC)=O)CCC2(CC1)COC(CNC(=O)C(C)(C)C)C2 Nc1ccc(F)c(C(N2CCC3C(NC(=O)CCn4ccnc4)C23)=O)c1F c1(NC2(CO)CCN(C(c3cccn(O)c3=O)=O)CC2)cc2nncn2cn1 N1(C(c2c(CC)cns2)=O)CC2CC(C1)CN(C(c1conc1C(C)C)=O)C2 C(CCCCC(=O)N(CC(O)CN(C)C(c1cn2ccsc2n1)=O)C)=CCCC Cc1ccc2nc(C)c(CN3CCC(CNC(c4cncc(Cl)c4)=O)C3)n2c1 CCCS(=O)(=O)CC(=O)NCC1(NC(c2cn(C)c(C(F)F)n2)=O)CCCCC1 CCCCCC(F)C(=O)N1CCC(NC(=O)CCC=CC(C)C)C1COC C(C(C)C(=O)NCC1CCN(C(=O)Cc2ccc(Cl)s2)C1)OC c1(C(=O)NC2(CC=C)CN(C(c3cnn[nH]3)=O)C2)ccc(F)c(OC)c1 c1(C(=O)OC)ccc(C=CC(=O)NC(C)CCNC(C2CCS2(=O)=O)=O)o1 C1(C(=O)NCCC(C)(C)OC)COC2(C1)CN(C(=O)CCOC1COC1)C2 CCCC(C)CC(=O)NNC(=O)c1nn(C)cc1P(C)(C)=O C1(C(=O)NCCOCCNC(c2c(C)nc(Br)o2)=O)CCOCC12CCCC2 C1(C(N(CC(CN(C)C(c2n[nH]c(C3CC3)n2)=O)O)C)=O)CCC(C(C)(C)C)O1 C1(NC(=O)C(O)c2ccsc2)CCCC12CN(C(=O)C(N1CCCC1)C1CCC1)C2 CCC(CNC(=O)C(C)NC(c1ccc(CO)s1)=O)C(C)(F)F N1(C(N(c2ccsc2)CC)=O)CCC(C2CCN(C)C2)C1 C1(OC)CN(C(=O)C(c2ccc(Br)cc2Cl)(F)F)CC12CC2 N1(C(C2CC(C)=C(C)CC2)=O)CC2CCC1CN(C(c1cc(Cl)c(C)cn1)=O)C2 N1(C(c2c(OCC)nccc2)=O)CCC(O)(CNC(C2C3CC4C(C3)C24)=O)CC1 c1(CC)cc(C(N2CCCCC2C(C)NC(=O)CC(=O)NC)=O)c2c(c1)CCO2 c1(C(CNC(COCC=C)=O)NC(c2cc(CC)[nH]n2)=O)cccc(Cl)c1 N1(C(CC(C)(C)CNC(c2cccc(F)c2O)=O)=O)CC2(C)CC1CCO2 c1(-c2ccc(CNC(C3C4(CC(=O)NC4)C3)=O)cc2)cnc2c(c1)CNC(=O)N2 CC(C)CC(=O)C(=O)N1CCC(OCC(N2CCOC(C3CC3)C2)=O)C1 N1(C(C2CN(CC)C(=O)CC2)=O)CCN(c2nnc(CO)s2)CC(O)C1 Cn1cc(C(N2CCC(C3CCCN3C(=O)CC(F)(F)Cl)C2)=O)c(O)n1 CC(C)(C)S(=O)(=O)CC(=O)N1CCOC2(C1)CN(C(C1CCCC(O)C1)=O)C2 c1(OCC)cnc(C(N2CCCC(N(C(=O)CC3CCCC3(F)F)C)C2)=O)cn1 O=C(C1=CC2CCC=CCCC12)NCC1CC(O)CN1C(=O)C=Cc1nccs1 C(=O)(CCN=c1[nH]ccs1)NCC(CNC(C1CCC(N=[N+]=[N-])CC1)=O)CO c1(NC(C2C(OCC)CC2)=O)cc(C(=O)N(C)CCO)ccc1C N1(C(c2c(NCC)cccn2)=O)CCC2CC1CN(C(=O)C=Cc1cscn1)C2 c1(N(CCCNC(COCC)=O)CC)snc(Cl)c1C#N C1(C)(NC(C2CCC(CCNC(c3ncn(C(C)C)n3)=O)C2)=O)CC2(CCC2)C1 C=C(Br)CCC(=O)N1CC(NC(=O)CN2CCCCC2=O)C(SC)C1 N#CC1(C(N2CC(CNC(=O)CNC(c3cccnc3)=O)C(O)C2)=O)CCCOC1 c1(OC)nsc(OC)c1C(=O)NC(C1(O)CN(C(=O)Cc2csc(C)n2)C1)C C(=O)(C(C)(C)C(=O)NCC1COCC1NC(=O)C1=CCCCO1)N(C)C C(=O)(C#CC1(C)COC1)NCCSCCNC(C(C=C)(C)CC)=O c1(CNC(C(C(C)NC(C=CC(CC)C)=O)C)=O)ccc(C)nc1O N12CCC3CC13C2=O.CC1CCCN1CC(=O)NCCCN=[N+]=[N-] C1(C(C)(C)NC(c2cnc(C)[nH]2)=O)CCCCN1C(c1nnsc1C)=O c1(C(=O)NC2C(C)CN(C(C3CC=CC3)=O)C2)ccc2nnn(O)c2c1 CC1c2ccccc2CC1C(=O)NCC(C)(C)CNC(c1[nH]cnc1Cl)=O c1(OC)ccc2c(c1)C(C(=O)N1CCN(C(C)C)C(=O)C1)CC2 c1(CC)cc(C#N)ccc1OCCCNC(=O)Nc1c[nH]c2cnccc12 C1(O)(C(=O)NCCC(C)NC(C2CC3OC(=O)OC3C2)=O)CCCCCC1 C(N=c1[nH]c(=NC2CCCC(C)C2)[nH]c2c1COC2)c1ccc(CC)cc1 c1(CC(=O)NC(CC=C)CNC(c2cnccc2Br)=O)cc(F)ccc1F CC1COC2(C1)CN(Cc1ccc(-n3cccc3)cn1)C2 N1(C(c2c(C)snc2)=O)CCC(C2CC2)CC1.C12(CC(F)(F)C1)C(=O)N2C1CC1 CC1Cc2ccccc2CC1NC(=O)COC(C)(C)CNC(C1(Cl)CC1(F)F)=O c1(C(N(CCCNC(COCCC)=O)C(C)C)=O)cnc2ccccc2c1OC C1(CNC(C2N(CCC)CCC2)=O)CCC2(CN(C(=O)CC3(OC)CCC3)C2)O1 c1(NC(CC)=O)cccc(C(=O)NC2CN(C(=O)C(C)(C)OC(C)C)C3CC23)c1 C1(NC(=O)NC23CC(NC(CC(C)C)=O)(C2)C3)CC(=O)N(c2ccccc2F)C1 Cc1ncccc1C(=O)NC(CNC(C1CC(C)(F)C1)=O)C(C)(C)C N1(C(CC2CC(C)(C)OC2)=O)C2CCC1C1CC1(NC(=O)COCCCF)C2 C1(NC(=O)C(O)Cc2cnc[nH]2)CCC(NC(=O)CCCC2CCCC2)CC1 N1(C(CCc2ccc(C)o2)=O)CCC2OCCN(C(c3nc(C)sc3C)=O)C2C1 C1(C(=O)NCC(C(C)O)C)CCC(C)(C)N(C(C2CC2(C)C)=O)C1 Cc1ccc([N+](=O)[O-])cc1C(=O)NC(Cn1cc(C(C)(C)C(C)C)nn1)CC(C)C C1(NC(c2c(CC)cccc2)=O)CCCCN(C(=O)Cc2ncoc2C)C1 c1(C(N(C)CC2CCCN(C(C(=O)NC)=O)C2)=O)cc2ccc(Cl)nc2s1 CN(C)NC(=O)CCC(=O)NC1CN(C(C2C(F)(F)C23CC3)=O)C1 c1(N(CCNC(C(CC)C)=O)C2CC2)ccc(C(F)(F)F)cc1[N+](=O)[O-] c1(C(=O)NC2CC(NC(=O)CC3CCC(O)C3)C2)ncc([N+](=O)[O-])cc1Br C(=O)(CC(C)CC(C)(C)C)NC1CC(C)(NC(CSCC(=O)OC)=O)C1 Cc1cc(C(=O)NCC2CCC2NC(c2nc(Cl)ccc2N)=O)cc(C)c1Cl C(C(CCNC(C1CCCN1C(=O)CCN1CCOCC1)=O)OC)OC C(N=c1[nH]c(=NCC2(Br)CC2)c2c(F)cccc2[nH]1)c1c(C)ccc(S(N)(=O)=O)c1 CS(=O)(=O)CCCC(=O)N1CCN(C(=O)CC=Cc2ccc(F)cc2)C(CF)C1 c1(N2CCc3n(cc(C)n3)C2)nc(=NCc2cnc[nH]2)[nH]c2c1CCCCC2 CC#CCCC(=O)N(CC(C)CNC(c1ccccc1CC(=O)OC)=O)C Cc1cc(C(=O)NCCCCNC(C2CCC(=O)C2)=O)cc(F)c1C c1(CC)cnn2ccc(C(=O)NC(CNC(=O)C(F)(F)C(C)O)C3CCC3)nc12 c1(C(=O)NC(c2ccccc2Br)C)cc(F)ncc1NCc1ccc(F)cc1O C(=O)(CCCCN1CCC(C(=O)NCCN(C(=O)C(=O)NC(C)C)C(C)C)C1)NC C12(NC(C(C)NC(=O)CC=C(Cl)Cl)=O)CCC(n3cc(CNC4CC4)nn3)(CC1)C2 C#Cc1cccc(C(=O)NCC2CN(C(=O)C(CO)C(F)(F)F)CCO2)c1F c1(-c2cn(-c3c(CNC(c4cc(C)sc4)=O)scc3)nn2)cc2cn[nH]c2cn1 C12CN(CCO1)C2.n1(CCCN(C(C(C)n2cccn2)=O)C)cc(C(C)O)nn1 c1(SC)cc(C)c(C(=O)NC2CC(F)(CNC(C3CCC3c3nc[nH]n3)=O)C2)s1 c1(C(N2CCC(C(=O)NCCCCC#C)(CO)C2)=O)nccc(C)c1N C1(NC(C(OC)OC)=O)CC2(C1)CN(C(c1cc(F)ccc1C(F)F)=O)C2 Cc1cn(CC(N2CC3CC3(NC(c3coc(C(F)F)c3)=O)C2)=O)c(=O)nc1O N1(C(C2CCN(C(c3cnns3)=O)C23CC3)=O)CCc2ccccc2C1 c1(NC(c2n(CC)ccn2)C)cc(NCc2nc(=N)[nH][nH]2)ncn1 n1(CC)cc(Br)cc1C(=O)NCC(CO)NC(=O)C(c1cccc(Cl)c1)(F)F N1(C(COC)=O)CCN(CC(F)Cn2cc(CNC(CSC)CO)nn2)CC1 C(=O)(C#CC1CCCC1)N1CC(F)CC(NC(=O)Cn2cc(C3CC3)nn2)C1 N1(C(c2ccc(C)o2)=O)CCCCC(N(C)C(c2nn(C)cc2Br)=O)C1 N1(C(C(CCCC)C)=O)CCOC2(C1)CN(C(c1cc(C(C)=O)c[nH]1)=O)C2 N1(C(C2(SC)CC2)=O)C2CCC1CC(F)(CNC(=O)C(C1CC1)SC)C2 C12CCN(CC1C)C(=O)NC2.C(CCC(=O)Nc1n[nH]c(O)n1)OCC C(CN=c1[nH]c(N2CCNC(=O)CC2)nc2c1CSC2)(c1cccc(C)c1)OC C12(C(=O)NC3CC(CCNC(C(C4CCC(O)CC4)C)=O)C3)CC(C)(CCO1)C2 c1(NC(CC)CNC(c2ccc(C(C)(C)C)cn2)=O)c(Cl)cc([N+](=O)[O-])cc1Cl C(=O)(C(C)(C)C(N)=O)NC(Cc1cn(Cc2cc(C(C)(C)C)sc2)nn1)CCO C(=O)(C(CCC1CCC1)NC(=O)CCc1ccsc1)NCc1ccc(CC)s1 C12(CNC(C(C)=C3CC3)=O)CCCCC1N(C(=O)CCc1ccc(Cl)nc1)CC2 c1(N2CCC(CNC(CCCC(C)(C)C)=O)CC2)[nH]cnc2nc(Cl)cc1-2 c1(C(=O)Nc2cccc(OCCC=C)c2)cccc(Cl)c1-n1cncn1 CC1(C)CC(C(N2CC(O)C(O)C2)=O)CN1C(=O)CC1CCCC12CC2 C1(C(C(=O)NC)(CO)N(CC(C)(C)C)CCCO)CCC(C)CC1 C1(CNC(CCC=C)=O)CCCN(C(c2cc(C(C)(F)F)ccn2)=O)C1 n1(CCCS(C)(=O)=O)nc(C(F)(F)C(F)(F)F)c2ccccc2c1=O c1(CC)ncnc(N2CC3(CC3)CC2CNC(=O)CCCc2nncn2C)c1F c1(CCC)[nH]ccc1C(N1CC(CNC(c2cncnc2)=O)(COC)C1)=O N1(C(C(CC)OCC)=O)CCC2(CC1)CCN(C(=O)COC1CC1)CC2C C1(NCC)CCCC(C(=O)N(CC=CC(=O)Nc2cncn2CC(C)C)CC)CC1 c1(CC(=O)NC2CC3(NC(=O)CCF)COC2C3)n[nH]c2c1CCCC2 Nc1c(Cl)ccc(Br)c1C(=O)NC1(CNC(C2C=CCC2)=O)CCCC1 C1(C(=O)NCC2C3CN(C(c4nonc4N)=O)CC23)(CC)CCCCC1 c1(C(N(C2CCN(CCOCC3CCCO3)C2)CCC)=O)ncccc1Br Cc1cc(Br)cc(C)c1C(=O)NC1C=CCN1S(=O)(=O)CC1CC1 C1(CNC(c2ccc(OC)nc2Cl)=O)CN(C(=O)CCC2CC2)CCC12CCC2 C1(CC(=O)NCCCC=C)CCCCN1C(=O)Cn1cc(C)cn1 C1(N(C(CCC)CNC(=O)CC(C)F)C(c2cc(Cl)cn2C)=O)CCC(F)(F)CC1 c1(C(=O)NC(C(=O)NCC2C(CC(C)(C)C)C2)C2(C)CC2)ccc(C#N)o1 c1(C(N2CC(CNC(c3c(OC)ccnc3)=O)C2)=O)cc(O)cc(O)c1 C1(C(N(C)CC=CC(=O)NCc2cnsc2)=O)C2CCCCCC12 c1(OC)cc(C(N2CCN(C(=O)C(C)(C)C3(C)CC3(F)F)CC2C)=O)nc(C)c1 Cc1cccc(=S)n1CC(=O)NC(c1ccc(O)cc1)CC1CC1 N1(C(CCC(C)OC)=O)CCCC2CN(C(c3cncc4sccc34)=O)CC12 c1(CC(C)C(=O)N(C(C)CNC(C2(n3ccnn3)CC2)=O)C)cccc(F)c1 N1(C(c2cnc(OC)s2)=O)CCC2C(C1)NC(=O)CCN2C(=O)CSCCOC C(=O)(CCCCC(=O)N1CC(O)CC1C(N1CCC(C)(O)CC1C)=O)OC CC(C)(C)C(O)C(=O)N1CCCC(CCC(=O)NCC2(C)CCC(O)CC2)C1 c1(CNC2C(C(N3CC(C(F)(F)F)C3)=O)C2)nc(CSc2cccs2)no1 c1(N(C)C)cn(C2CC(C(c3ncoc3-c3ccccc3)=O)C2)nn1 c1(NC2CCC(CC)CC2)ncc(C)cc1S(=O)(=O)N1CCOC(C2CC2)C1 N1(C(c2c(C)nc(NC(c3ccnc4c3OCO4)=O)s2)=O)CCNC2(CCC2)C1 c1(SC)cncc(C(=O)NC(C)CCNC(c2ccncc2)=O)c1 C1(F)(C(=O)NC2(C)CC(NC(=O)CCCN3C(=O)CCC3=O)C2)CC12CCCCC2 c1(SCC(C(=O)NC)N2CCCC2COC(C)(C)C)ccc(F)cc1.CCN(C)C N12CCCC(C1)C(=O)N(C)CC1(O)CCN(C1)NC2=O.C1(C)CC2CCC1O2.CO c1(NC(=O)NC(C(=O)NCc2csc(C3CC3)n2)C2CCCO2)ccc(Br)cc1 C=CCCC(C)(C)CNC(=O)C(CC(C)C)ONC(c1cc(C)nnc1O)=O C1(C(N(CC(=O)NC2CCCC2N(C)C)CCC)=O)CCCN1C CC1CCCC1C(=O)NC(CCCNC(c1ccc(CO)s1)=O)c1ccccc1 C1(C(N2CCC(CCNC(C34CCC(CC3F)C4)=O)C2)=O)CC2(C1)CC2(F)F CC1CC(C(=O)NCC2(C(=O)NC3(CF)CC3)CC2)=NO1 Cc1ccc(CCC(=O)NCC2(NC(=O)C(F)C3CC3)CC2)cc1C C1(CNC(C2(C)CCC2)=O)CN(C(=O)CCCc2ccccc2)CCC12CCC2 Nc1c(F)ccc(Cl)c1C(N1CCC2C(C1)CN2C(=O)C(=O)NCC(F)F)=O CC(O)CCCCCC(=O)N1CC(O)(C(C)NC(c2cnc3[nH]cncc2-3)=O)C1 C12(CC(=O)NC3(CCNC(C(c4cn(C)nc4)=O)=O)CCC3)CCC(CC1)CC2 c1(CNC(C2C(NCc3cc(C)oc3C)C2)=O)ccc(Cl)c(Cl)c1 N1(C(=O)Cn2cnnc2)CCN(C(=O)C2=CCCC2)C(c2cccs2)C1 C=CC(C)(C)C(=O)NC(CNC(=O)CCC1CCC(C2CC2)O1)CC C12(CNC(C3CCCN(C(C(CC)C)=O)C3)=O)CCC(CC1)CN2C(C)=O N1(C(C2CN(C(CCC)C)C(=O)C2)=O)CC(NC(c2nnsc2C)=O)C2(CC2)C1 N1(C(c2ccncc2)C(=O)NC)CCN(CC(C)O)CC1 C(C(Cc1ccco1)CC(=O)N1CCN(C)CC1C)c1c(OCCC)cccc1 c1(C(N2C(CCNC(=O)C(O)C(F)F)CC(F)(F)C2)=O)cc2c(s1)CCCCC2 C(N=c1[nH]c(Cl)ncc1F)C1CC(NC(C2CCC(CC)O2)=O)C1 C=CC(C)CCS(=O)(=O)NC(CC)C(=O)OCC1CC1 C1(NC(c2cc(C3CCCC3)no2)=O)CCN(C(=O)Cc2ccsc2)C1 N1(C(C(C)NC(CC)(C)C)=O)CCC(NC(C2CCC(F)(F)CC2)=O)C(C)(C)C1 N1(C(=O)NCC2CC(C)(C)OC2)CCCSCC1c1ccccc1 c1(OC)c(-c2cccc(NC(c3cnn4c3OCCC4)=O)c2)cccc1C#N c1(C(N2C(C(=O)Nc3c(C)nccc3)CSCC2)=O)ccc([N+](=O)[O-])cc1 CC1CC(NC(C2(CCF)CC2)=O)CCN1C(=O)CCN1CCCS1(=O)=O CC1=NNC(=O)C1CC(=O)Nn1cncn1.c12cn(nn1)CCN(CC(C)O)C2 c1(C(N(C2CCN(C(C3CC(C)OC3C)=O)C2)CC)=O)cncc(O)c1 C(=O)(C(CC(F)F)N(C(=O)CC(C)F)C)NC(CSC)(C)C C(=O)(CC(C)C(=O)N1CCN(C(=O)C=Cc2scnc2C)CC1C(C)(C)C)OC c1(CC)noc(CC)c1CC(=O)NCC1C2CN(C(=O)CN3CCOC3=O)CC12 N1(C(C2(NC(CC3CC(SC)C3)=O)CC(F)(F)C2)=O)CCCC(C=C)C1 C1(C(=O)NC(CC)C(F)(F)F)COCCN(C(=O)CC(=O)NC2CC2)C1 N1(C(Cc2ncn(C)c2)=O)CC(C2CC2)(C(=O)NCCC2(C)CC2)C1 CC1CCCC(NC(=O)CCNC(C2OCCC2C)=O)C1C C#CC1CC2(CC(CNC(=O)N(C(C(=O)OC(C)(C)C)CCCC)C)C2)C1 C1(CCC)CN(C(c2nc(C)oc2C)=O)CCN1C(=O)C1=CCCC1C c1(C(=O)NC2C3CN(C(CC(CC)O)=O)CC32)cccc2c1CCCO2 c1(C(N)=O)ncnc2c1cnn2CC(N1CCC1(CO)CO)=O C(=O)(CCCC(=O)NC1CCN(C(C)(C)C)C1)N(CCC)C(C1(C)CCCC1)=O C(CCCCCNC(c1cscc1Cl)=O)NC(=O)C(C1CCCCC1)c1cccs1 CCC(C(C)C)C(C(=O)NC(C)C)N(C(CC(C)C)C(=O)NCCCF)C CC1(C(=O)NCC2COCCN2C(=O)Cc2nc([N+](=O)[O-])n[nH]2)CCC(=O)NC1 C1(CC)C(=O)NCCN1C(c1n[nH]c(C)n1)C(=O)Nc1ccc(F)cc1C C1(CC(=O)NCC(C)C#N)C2CCCC2N1C(=O)Cc1cnn(C)c1 c1(C(N2CCC(C)SCC2)=O)cc(O)nc2c1CN(C(=O)CCCF)CC2 N1(C(c2n(C)cnc2)=O)CC(CNC(=O)C(O)CC(F)F)CC12CCC2 N1(C(Cc2ccc(C#C)cc2)=O)C2CCC1C(C)C(NC(C1(CCO)CC1)=O)C2 C1(CN(CC(C)NC(=O)COCC2CC2)C(=O)CC2CC2C(F)(F)F)CCCCCC1 Cc1ncc2n1CCN(C(=O)C(C1CCN(C(C3CNC(=O)C3)=O)C1)C)C2 CCCC(CCCNC(=O)Cc1cc(Cl)n(C)n1)NC(=O)C=CSc1nc[nH]n1 C(CNC(=O)CCC1CCOC1)(CC)(CC)NC(CC1CC(=C)C1)=O C1(C)(COC)CC(NC(c2cncc(OC)c2C)=O)CN1C(c1cnc(C)s1)=O N1(C(C=CCN(C)C(C2CC3C(C2)C3(F)F)=O)=O)CC(S(N)(=O)=O)C1 Cc1ccc(C(=O)NCCCCNC(=O)C(F)(F)c2cncs2)o1 C12(CNC(CC3CC(C)N(C(=O)CNC(C4CC4C)=O)C3)=O)CCCN1CCC2 c1(C(=O)NC2CC(NC(c3c(O)cccc3F)=O)C2)ccc([N+](=O)[O-])s1 Cc1cc(C(=O)N(CC(C)NC(c2n[nH]cc2C)=O)CC)n2ncc(C#N)c2n1 C=CCC(CC(=O)NC12CC(F)(C1)C2)NC(=O)CCCCCF C1(NC(C(C(C)C)F)=O)CN(CCc2ccc(F)cc2)CC1(C)C N1(C(c2c(C)snn2)=O)CCC(C(=O)NC2COCC2CO)(CO)C1 c1(C(=O)NCCCCNC(C(C)OCC#C)=O)n[nH]c(C(C)(C)C)n1 O=S(=O)(c1ccc(Br)cc1)NN1CCC(O)(C(F)(F)F)C1 c1(NC(=O)OCCCc2cc(F)ccn2)cc(Br)cc([N+](=O)[O-])c1 N1(C(C(CC#CC)NC(=O)C(C)OCOC)=O)CCC2(CC1)CC2C#N C(=O)(C(N)CNC(N1CCCC1)=O)N(c1cccs1)C Cc1ncc(N)cc1C(N1C(C(=O)NCC(C)(O)CN(C)C)CC1)=O Cc1nc2ccc(C(=O)NC(C)(C)CCNC(C3CCC(C)CC3)=O)cc2[nH]1 N1(C(C2CC(C)(C)OC2)=O)CCCC(C2(NC(=O)C#CC3CCCCO3)CC2)C1 C(C)(N=c1[nH]c(=NCc2ncoc2C2CC2)[nH]c2c1COC2)c1nc(C)[nH]n1 Cc1cc(C(N2CCC(C(=O)NC3(CN(C)C)CC3)(CF)C2)=O)ccn1 c1(C(=O)NC(CNC(c2c(CC)csc2)=O)CO)cnn2ccc(C)cc12 C(=O)(CS(=O)(=O)C12CC(C1)C2)N1C2CC(NC(C(CC(C)C)(C)O)=O)CC1CC2 CCCC(C(=O)N(CCC(=O)NC1(C2CCC2)CC1)OC)N(C)C C1(CC)C(=O)NCCN1C(c1ccn(CCNC(=O)CS(=O)CC)c1)=O C1(C)(CNC(CC(CC)NC(=O)C(C)(C)N2CCCC2)=O)CCC(CO)CC1 C1(C(N(CC(Cc2cccc(Cl)c2)CO)CCC)=O)CCC(C(=O)OCC)CC1 CC(=O)CCCC(C)C(=O)N(C1CN(C(c2cncc3[nH]ccc23)=O)CC1O)C c1(C(N(C2CCC(NC(=O)C3=CCC3)CC2)CC)=O)ccc2c(c1)NC(=O)C2=O c1(-c2ccn(CCc3c(OC)cccc3)n2)[nH]nc2c1COC2 N1(C(c2n(CC)nc(C)c2)=O)CC2CCCCC2(NC(=O)Cc2sccc2C)C1 C(C(C)(C(F)(F)F)c1ccccc1)OC.N12CCC(CC1C)NC2=O C1(C(=O)N(CC(CC)OC)C)(NC(C2CC(C(=O)OC)C2)=O)CCOC1 c1(-c2cn(C3CC4(C(CN5CC(CN(C)C)C5)=O)C3C4)nn2)ncc[nH]c1=O C1(CC)CCCCC1C(=O)N(C)CC1CN(C(c2ncc(F)cn2)=O)C1 CC1(CNC(c2ccc[n+]([O-])c2)=O)CCCN(C(C2CCC(C3CC3)C2)=O)C1 C=C(C)CCCC(=O)N1CC2(CC2)CC1C(N1CC(C)CC(O)C1)=O Cc1ncc(CCC(=O)N(CC(C)CNC(c2ccc[nH]2)=O)C)o1 C(=O)(CC(C)(O)CNC(=O)CSc1cn[nH]c1)N1CCC(NC(=O)OC)C1 C1(NC(C=CC(C)NC(=O)Cc2ccccc2)=O)CC(C)CC(C)(C)C1 C1(C(=O)NC2(C)CCCN(C(C3=C(C)CCC3)=O)C2)COc2ccccc2O1 C1(NC=O)(CNC(C2CC2C(=O)OCC)=O)CCOCC1.C#CCOCC N1(C(C(C)OCCC(C)C)=O)CCN(C(=O)CCCCCO)CC1CO N1(C(CCCCNC(N)=O)=O)CC2ON=C(CNC(c3coc(Cl)n3)=O)C2C1 C1(NC(C2(C)SCCCS2)=O)CC(C(N2CCC3(CC2)N=N3)=O)C12CCC2 c1(C(=O)NC2C(NC(=O)Cc3ccccc3)COC2)c(F)ccc(F)c1Br Cc1nn(C)c2sc(C(N3CCC(NC(=O)C(C)C(F)(F)F)C3)=O)cc12 N1(C(c2cn(C)nn2)=O)CCN(N2CC3CCC3(CO)C2)CC1 C(C1=CCCN(C(C2C3CC4C(C3)C24)=O)C1)NC(COC1(C#C)COC1)=O N1(C(C(n2cc(Cl)cn2)C)=O)CCCCC1CN(C(=O)C(F)=CCCF)C n1(CC(=O)NC2CCCCC2NC(=O)CC2NC(=O)NC2=O)nc(C)cc1CC c1(C(=O)NCC(CC=C)NC(C2CN(CC(F)(F)F)C2)=O)ccc(Cl)cc1OC c1(C(=O)NCC(CNC(=O)CCCN2CCOCC2)O)cc(F)cc(F)c1 N1(C(C(=O)NC(C)C)C)CCC2(CC1)COC(=O)N2 CC1CN(C(=O)CN2CCCC2C)CC1NC(C1CC1C#N)=O CC1CN(C(c2sccc2CC#N)=O)CCN1C(=O)CCCC(=O)NC1CC1 N1(C(C2CC3(CCCO3)C2)=O)CCN(C(C2CCCC2O)=O)CC(O)C1 c1(CN2CC3CN(C(c4cc(C)c(Cl)c(C)c4)=O)C3C2)oc2ccccc2c1C N12CC3OCCN(C3C1)C(=O)C1CN(C1)CC2=O.C1(CC)CC1OC C1(OC)(CNC(=O)C(C)n2cccn2)CCN(C(=O)CCOCC(C)(C)C)C1 S(=O)(=O)(CCC(=O)N1CCOCC1CN(C(=O)COCC1CCCO1)C)NCC Cc1n[nH]cc1CC(=O)NCCOC1CCN(C(c2ncnn2C(C)C)=O)C1 C(C)(C)(CCC(=O)NC1CN(C(=O)C(F)(F)c2cccnc2)CC12CC2)N(C)C C1(C(=O)NCC(O)CO)CCC(CNC(C2CC2(F)Cl)=O)CC1 C1(CC(=O)NSc2ccccc2)CCN(CC2(O)CCSC2)CCC1(F)F c1(CC)ccc(-n2nc(CC(c3ccccc3)O)nc2C2CC3CC2C3)cc1 C1(CCN(C)C)CN(C(c2cocc2Br)C(=O)NCC2CCCO2)CCO1 c1(C(=O)NCC2CCC(C)=C(C)C2)cnc(O)c(Cl)c1.CC1=NOC(=O)C1CC CN1CCCC(C(=O)NC2(C3CCCN3C(=O)CC3CCCCC3O)CC2)C1 N1(C(=O)Cn2nccn2)CC2CC(C(=O)NCCN3CCCOCC3)C(C2)C1 Cn1cc(S(=O)(=O)NCC2(CC(=O)O)CCC2)cc1-c1ccccc1 N1(C(CC2(N(C)C)CCC2)=O)CCC2(CCCN2C(=O)CC2CCC(=O)N2)C1 C(=O)(C(N=[N+]=[N-])C(C)C)NC1(C(=O)NCCn2c(C)nnc2)CCOCC1 Cc1[nH]nc2c1CCC(C(N1CCC1CNC(=O)Cn1cccn1)=O)C2 c1(COC)ccc(OC)cc1.c1(C(CC)N(C(C(=O)N)=O)CCC)ccc(Br)cc1 C1(CC)(NC(c2ccoc2C)=O)CCN(C(=O)C2CC2)C1.N12CC(C1)C2=O c1(OC)ccccc1OCC(N1CC2CC2(C(=O)NCC=C2CCNCC2)C1)=O c1(C(=O)NC2CC(N(C(c3[nH]cc(CC)c3)=O)C)C2)c(C)cnnc1O Cc1c(O)ccc(C(N2CCC(O)(CN(C)C(C34CCC3CC4)=O)C2)=O)c1C CC1CN(C(c2cc(F)n[nH]2)=O)CC1CNC(C1CCOC1)=O Cc1ccc(C(=O)N(C)CCC2CCN(C(=O)CCF)CC2)nc1C c1(CC(=O)NCC(CNC(c2n(C)cnc2)=O)(C)C)coc2cc(F)ccc12 N1(C(CSCCC)=O)CC(C)N(C(C2CC3C=CCC(C2)C3)=O)CC1C CC(C)C(C(=O)N(C(C)CNC(=O)CCCn1ccnn1)C)NS(N)(=O)=O N(C(=NCC#CC1CC1)NCc1ccc(CO)cc1)C(COC)C C1(NC(c2cn3cccnc3n2)=O)CC(N=c2nc[nH]c3[nH]c(Br)cc23)C1 CC1CN(C(c2c[nH]nc2[N+](=O)[O-])=O)CC(C(=O)NCC(c2cn(C)cn2)O)O1 N1(C(Cc2cccc(C)c2F)=O)CC2CCN(C(c3ncccc3C)=O)C2C1 N1(C(C(C)OCC(C)C)=O)CC2(CC(NC(C3CCCC34CC4)=O)C2)C1 c1(C(=O)NC2CC(F)(CNC(c3sccc3CO)=O)C2)cc(Br)ccn1 c1(C(=O)NC(CNC(c2sc(C)c(Br)n2)=O)C)cc(C(C)C)cnc1O N1(C(c2ncn(C(C)C)n2)=O)CC2(C(=O)NCC3CCCC(C)(C)C3)CC1CO2 c1(SC(C)C)cc(C(N2CCC(CNC(=O)C(F)(F)C(C)O)C2)=O)ccc1F C(Cn1cc(COC(=N)O)nn1)(CCC(F)(F)F)NC(C(CCC)O)=O c1(OC)ccc(N(CCS(=O)(=O)N)C)c(C)c1.C(CC(C)C)OCC(=O)OC c1(C(N2CCC(C(C)NC(COCC=C)=O)C2)=O)cccnc1N(C)C N1(C(C2C(=C)C2)=O)CC(NC(c2cc(-c3ccc(Cl)cc3)[nH]n2)=O)CC(C)(C)C1 N1(C(C(C2CCC2)SC)=O)CC(NC(=O)COC2CCOC2)CC12CCOCC2 CCCC(CC)CCC(=O)N1CCC(N(CCC)C(C2(COC)CCC2)=O)C1 N1(CCOC)CCN(CC(N2CCC(C3CCCN3C(C3CCC3)=O)C2)=O)CC1 c1(C(=O)NC2CC(CNC(CN(C)C)=O)C2(C)C)ccnc2ncnn12 C#Cc1cccc(CC(=O)NCC2CCN2C(=O)COc2c(F)cccc2Cl)c1 c1(C(N2C(CNC(CCC(=O)OC(C)(C)C)=O)CC2)=O)ccc(F)c(F)c1 Cc1cc(C#N)sc1C(N1CCC(O)(CNC(=O)CCCNS(C)(=O)=O)C1)=O c1(CNC(C(=O)NCC(C)N(c2ccc(Br)s2)C)=O)ccccc1 C1(N(C(C=COCC)=O)C)CC2CCC(C1)N2C(=O)CSc1ccccc1O N1(C(c2cscc2Cl)=O)CCC(F)(F)C(Cn2ccnc2)C1.N12CCCC1C2 C1(CNC(CSCC)=O)CC2CC2N1C(=O)C(C)Cc1cnc[nH]1 Cc1nc(C)c(C(=O)NC2CCCN(C(c3nn(C(C)C)nc3Br)=O)C2)o1 N1(C(c2cn(CC)nc2C)=O)CCC(NC(c2cc[nH]c2C2CC2)=O)C(CC)C1 C(=O)(C(F)(CNC(=O)C(C)CC(N)=O)C(C)C)NC(c1nc[nH]n1)CC c1(C(N2CCN(C(CNC=O)=O)CC2CO)=O)ccc2ncccc2c1Cl c1(C(=O)NC2C(NC(c3c(C)ccnc3)=O)CC2)nc(C)n2ccccc12 C(=O)(C(O)CCc1ccccc1)N(C(CNC(c1cc(OC)ns1)=O)C)C c1(C(N2CC(C(C)C)N(C(C3CCSC3)=O)CC2)=O)cc(F)c(F)c(Cl)c1F C1(C(=O)NCc2onc(C)n2)CC(C)(C)CCN1C(C1CC1C1(N(C)C)COC1)=O N(C1CCc2cccc3cccc1c23)N1C(C(N(C(C)(C)C)C)=O)CCC(O)C1 c1(-c2c(C)c(Cl)ccc2)nc2ccc(O)nc2s1 C1(C(=O)NCC2(CC)CC2)CC2(C1)CC(CNC(c1n(C=C)ncc1)=O)C2 C(CCN=C(NCC1(O)CCC1)N1CCOC(C2CCCO2)C1)OC(C)C Cc1nn(C)c(C)c1CC(=O)NC1(C2CN(C(=O)C=Cc3ccncc3)C2)CC1 C1(NC(=O)Cc2ncccn2)CN(C(=O)CC2CNC(=O)O2)CC12COC2 C1(C)(C(N2CC3C(NC(C=C(CC)C)=O)(CC3)C2)=O)CCCCC1(F)F C#Cc1cc(C(=O)NCC2CN(C(=O)C(C)OCCOC)CCO2)cc(F)c1 Cc1ccc(C(=O)NC(C)C(C)NC(c2cnoc2C)=O)c(O)c1C C(=O)(C1CCc2ccccc21)NC1CCCN(C(C2CN(C)C(=O)C2)=O)CCC1 S(=O)(=O)(c1cccc(F)c1)NC(c1c(CNCCCOC)nc2n1CC(C)O2)=O c1(NC(=O)NC2C(C3(C(=O)NC)C(=C)CC3)CCC2)c(F)cc(Cl)cc1F.CC N1(C(c2c(CC)c[nH]n2)=O)CCCN(C(=O)CCCCCOCC)C(C)C1 C(=O)(C1=NOC(C)(C)C1)NCCC1(NC(CC2CCCC(C)C2)=O)CCCC1 N1(c2nnc(C(CC)(C)C)o2)CCC(NC(=O)CC(C)C2CCCO2)C(C)(C)C1 n1(CC)nc(C(N2CCC(NC(c3c[nH]cc3Br)=O)C2C2CC2)=O)cc1C N1(C(c2c(-c3n(C)ncc3)n[nH]c2)=O)CC(C(N2CC([N+](=O)[O-])C2)=O)C2(CCC2)C1 c1(C(=O)NC2C3CN(C(CCCC=C)=O)C(C3)C2)ccc2ncnn2c1 c1(C(N(C)Cc2nccs2)=O)cc(C2CC2)[nH]n1 C(N=c1cc(Cl)nc[nH]1)C1CCCN(C(=O)C(F)(F)Cl)C1 C1(C(=O)NCC2N(C(CCCS(N)(=O)=O)=O)CC2)CCc2[nH]nc(C(F)(F)F)c2C1 c1(OC)cccc(C(=O)NC2CN(C(=O)C=Cc3ccoc3)CC2O)c1C c1(C(N2CCN(C(=O)Cc3cncs3)CC2C2CCC2)=O)cc2ccncc2o1 C1(CNC2C(NC(CC(CC)c3ccccc3)=O)CCCC2)CCS(=O)(=O)CC1 N1(c2c(C)c(N3CCC3)ncn2)CC2CCC1CN2C(c1ccnc(Cl)c1)=O Cn1cc(C(N2CC(NC(=O)Cc3ccccc3C(F)(F)F)C2)=O)c(O)nc1=O c1(C(N2CC(C)C(NC(c3ncnn3C)=O)C2)=O)ccc(Cl)c2cc[nH]c12 S(=O)(=O)(c1cc(C)c(F)cc1Br)NC1(N(C(=O)C(CC(=O)OC)SC)CC)CCOC1 Cc1csc(C(C(F)(F)F)N(C(=O)C(C2(N)CCCC2)O)C(C)C)n1 c1(C(C2CCC2)SC)ccc(Cl)cc1OC.c12nnnn1C(CC=C)N2 C1(N(C(=O)C(Cl)=CCl)C)CCCCN(C(C2(CF)CC2)=O)C1 C(=O)(CC1=NNC(=O)C1)N1CC(C(C)NC(c2cnccn2)=O)OCC1 CCCCC(CNC(=O)Cc1c[nH]nc1C)NC(C1CCC(=O)N1C1CC1)=O C(=O)(CC(C)CN(C)C)NCC(CNC(c1cnc[nH]c1=N)=O)OC C1(F)(C(=O)NCCc2cnc(C)[nH]2)CCN(C(c2sncc2C)=O)CC1 C1(C(=O)OC)CC(=NO)N1S(=O)(=O)CCOCCOC(C)(C)C c1(CC(=O)NCC(C)NC(c2scc(C(=O)OC)c2)=O)ccc(C(C)(C)C)cc1 N1(C(CCC)=O)CCC(NC(=O)CNC(=O)CCc2nc(C)no2)C(CO)CC1 C1(C(F)F)(CNC(c2cc(C)[nH]n2)=O)CCN(C(=O)Cc2ccccn2)C1 C1(C(=O)NCCOCCNC(C2(CC=C)CC2)=O)C2(CC2)C12CC2 C(=O)(C(CC(=O)OC)c1ccccc1)N(CCCNC(C1(Cl)CCC1)=O)CC CC1CCNC(=O)C1NC(c1cc(CNC(c2cc(Cl)ns2)=O)ccn1)=O N1(C(c2cccc(OC)c2O)=O)CCCC2(CC(NC(c3sccc3Cl)=O)C2)C1 c1(C(N2CC3(CC(Nc4ncn(C)c(=O)c4)C3)C2)=O)c(Br)ccc2c1OCO2 c1(C(=O)NCC(C)(C)NC(C(COCC)C)=O)cc2c(C)cc(Cl)cc2[nH]1 C(=O)(CCN1C(=O)COc2ccccc21)NC(COC)(C)CC(C)C C1(COC)CC(O)CN1C(c1cc(CNC(C2CCC(=O)NC2)=O)no1)=O CCC(C)CC(=O)C(=O)NC(C(N1CCCCC(C)(F)C1)=O)C1CCOC1 C(=O)(CC(CC(C)C)NC(c1ccc(C#N)cn1)=O)NC(C#C)C C1(C(=O)NCCC(C)(C)SC(C)C(=O)NCc2ccccn2)CC12CCOCC2 Cc1coc(C(C)C)c1C(=O)NCC1CCN1C(c1cc(O)nn1C)=O C#CC1CC2CCC1N(C(=O)CC1CC1CNC(=O)Cc1cc(C)[nH]n1)C2 C1(NC(CCc2cc(C)[nH]n2)=O)CC2CC(C1)N(C(c1c[nH]cc1C(C)C)=O)C2 c1(CC(=O)NC2C(CNC(C(C)c3ccsc3)=O)CCC2)ccc(F)c(Cl)c1 C(=O)(CCCCCCCCCO)NCC1(OC)CN(C(C2(C)COC(=O)C2)=O)C1 C(C(C)(C)CCC#N)(c1nnnn1C1CC1)NCCOCCNC(=O)NC N1(C(C(CC#C)O)=O)CCN(C(c2ccc(Cl)c(OC)c2F)=O)C2COCC12 c1(C(N2CC(NC(=O)C(F)CC3CC3)C3C(C2)C3)=O)cc2c(Cl)cccc2s1 C(=O)(C(F)(CC)C(=O)OC)N1CCC(C)(CNC(C(c2ccccc2)SC)=O)C1 c1(C(C)=O)cncc(C(=O)NCCOCCNc2sc(N3CCCC3)nc2Cl)c1 C(C(=O)NC(c1ccsc1)C)(C(C)(C)O)NC(Cn1c(C)ncc1)=O N1(C(C2C(CCC)C2)=O)CCC(C(F)C(=O)NCCN(C)C2CC2)C1 C1(CCC)CCC(NC(C2(CNC(=O)C(n3nccc3C)C)CC2)=O)CC1 C(=O)(C1=CSCCO1)NCCC1N(C(c2cc(C3(C)CC3)on2)=O)CCC1 C(N=c1[nH]cnc2ccsc12)C1(F)CCN(C(C2CC23CC3)=O)CC1 c1(C(=O)NC2CCN(C(c3nc(OC)oc3)=O)C2)oc2cc(Cl)ccc2c1C CC1(C(=O)NOCc2cn(CCCO)nn2)CC(c2ccccc2)=NO1 Cc1cc(N2CCC(CC(C)NC(c3sccc3N(C)C)=O)CC2)nc(C)n1 c1(CSC)ccc(C(=O)NCCC(C)N(C)C(C2(C)CC(C)=NO2)=O)cc1 N1(C(C2C3CCCC23)=O)CCCN(C(c2ccoc2C2CC2)=O)C(CO)C1 C1(C(=O)NC(Cc2cc(C)no2)C)CC(F)CN(C(=O)Cn2cccn2)C1 N1(C(c2c(C)occ2)=O)CCOC2CCN(C(=O)CN3CCOCC3)CC12 c1(OC)cccc(C(N2CC3CN(C(=O)C(Cl)(Cl)Cl)C3C2)=O)c1Br c1(OC)cccc(C(=O)NCC(C(C)C(C)C)NC(=O)COc2ccsn2)c1F c1(C(N2CCC(O)(C(C)NC(COC)=O)C2)=O)cc(COC)nnc1C C=C(Cl)CCC(=O)N(CCNC(C1CCN(C(C)=O)C1)=O)CCOCCO c1(CN(CCOC)CCNC(C2CCCO2)=O)ccc(F)cc1 CON1CC(C(N2CCN(C)C(CNC(=O)C=Cc3ccccc3)C2)=O)CC1=O c1(CC(C)C)ccc(C(=O)N(C2CCN(C(=O)CC(Cl)Cl)C2)CCO)cc1 C1(C#N)(C(=O)NCC(C)CNC(c2cn(C)nc2Br)=O)CCCOC1 C(=O)(C1=CC(O)C(NC(=O)C2=NOC(C)C2)C1)NC(c1nc(C)[nH]n1)CO c1(C(N2C(CCN=c3[nH]nc(CC)s3)CCCC2)=O)cccc2c1C(=O)NC2=O c1(C(=O)NCC2(O)CN(C(c3c(C)coc3)=O)C2)sc2ccc(C)cc2c1C Cc1cnc2c(C(=O)NCC3COCCN3C(=O)CC3(C)CC3(F)F)cnn2c1 C=CC1CN(C(=O)CCSC(F)(F)F)CC1NC(=O)CC1CCCC1(F)F C1(NC(C(C)=C(C)C)=O)CN(C(=O)CCC(F)F)CC1C1CC1 C(=O)(C(C)(C)C(O)C(C)C)NC1CCCN(C(c2c(OCC=C)cccn2)=O)C1 N1(C(c2[nH]cc(CN(C)C)c2)=O)CCC2(CCCN(C(=O)CN3CCC3C)C2)C1 C(=O)(CCCCCC(C)O)NC1(C2CN(C(c3c(CC)oc(C)c3)=O)C2)CC1 C1C(C2CCC2)N=C2NN=C(O2)C2CC12.Cc1ccc(C(=O)NN2CCOCC2)[nH]1 c1(OC)ncc(-c2ccc(F)c(O)c2)cc1C(=O)N(c1ccc(C)cn1)C1CC1 C1(N)C=CCN(C(=O)C=CC(C)(C)NC(C(C)Sc2ccccn2)=O)C1 C1(CNC(c2c(S(C)(=O)=O)ccs2)=O)CC(N=c2c(Cl)c[nH]cc2[N+](=O)[O-])C1 n1(CC(=O)NCC2(COC)CN(C(=O)C=CC3CCOC3)C2)ccccc1=O CCC(C)(O)C(=O)NC12CC1CN(C(=O)CSc1cc(C)on1)C2 C(N=c1ccc(C(F)(F)F)c[nH]1)C1CCCN(C(c2ccc(C(C)(C)C)s2)=O)C1 N1(C(C(C=C)O)=O)CC2(CCC2NC(c2cc(SC)oc2C)=O)C1 C1(C(N2CC(CNC(c3c(=N)cc[nH]c3)=O)OCC2)=O)CCC12CCOCC2 C=CCC(C)(C)CC(=O)NCC1CCC(CNC(c2cc(F)ccc2F)=O)CC1 N1(C(C(C(=O)OC)OC)=O)CC2CC(C(N3CCN(C)C(=O)C3C)=O)C(C2)C1 c1(CN2C(C(=O)Nc3cccc(C)c3O)CCCC2)cc(Cl)c(Cl)c(Cl)c1 C1(NC(c2c(CNC(c3ccon3)=O)noc2)=O)CC(CO)CC1O Cn1nc2ccccc2c1CN=C(NS(=O)(=O)CCN1CCCC1)NC1CCS(=O)(=O)C1 C(=O)(C1=NOC(CO)C1)N(C)C.C(=O)(C(F)(F)CC#N)NCCCN1CCC1 N1(C(c2ncc(I)cn2)=O)CCC2CN(c3ncnc4cc(Br)ccc34)CCC12 CCC(CC)CCCC(=O)NCCCC(C)NC(=O)CC1(O)CCCOC1 N1(CCCNC(C(C)C2CC2)=O)CCC(NC(=O)Cc2cnccn2)C1 c1(C(=O)NCCCCCNC(C2CC3CCCC3C2)=O)ccc2ncccc2n1 c1(CC)ccc(C(=O)NC(CSC)C(=O)N(C(C)C(C)C)C2CC2)[nH]1 N1(C(CCCCNC(C)=O)=O)CCC2CCCN(C(=O)C(C#N)=CC(C)C)C2C1 C(=O)(CC(=O)N1CCCCC1)OCCN(C(C)C(=O)NC(C)C)CC#C N1(C(C(C)OCCCC)=O)CCCCCCC1CNC(=O)Cc1csc(CC)n1 C1(NC(c2nc(C(=O)OCC)sc2)=O)CC2(NC(=O)CC(O)C(C)C)COC1C2 C1(C)(CNC(c2nccc(C)c2)=O)CCN(C(c2ccc(CC#N)cc2)=O)CC1 CC1(C)CCCC(C(N2CC(F)CC2CNC(=O)CCOC2CC2)=O)O1 c1(C(N2C(CNC(=O)COc3ccsn3)CC(OC)C2)=O)cnc2ncccn12 N1(C(c2c[nH]c(=N)s2)=O)CCCC(NC(=O)C(O)Cc2ccccc2)C1 N1(C(CC23CC(C(=O)OC)(C2)C3)=O)CCC2CN(C(=O)C(C)C(F)F)CC2C1 N1(CCCC)CCCC1(C)CNCc1ccc(NS(C)(=O)=O)o1 Cc1ccc2ncccc2c1C(=O)NC1CCC1CNC(=O)CCC(C)C#N CN1CCN(CC(N2CC(Cc3ccccc3)C2)=O)CC1.C123CC(C1)(C2)C(=O)N3 c1(SCC)ccc(C(=O)NCC(C)CN(C)C(C2(CF)CC2)=O)o1 c1(C(C)NC(CC2CC(OC)CN2C(=O)C(C)C)=O)ccc(F)c(Cl)c1 c1(C=O)n[nH]c2nccc(Cl)c12.Cc1nocc1CC(=O)NCC1COC(C)C1 Cc1cc2c(C(=O)N(CCCN(C)C(c3ccnc(Cl)c3N)=O)C)cccc2o1 CCC(C)(CCNC(C1CC2(CC2)CO1)=O)NC(=O)CCC1CCC1 N1(C(CSc2cccc(C)c2)=O)CC2CCC1CN2C(C1CNC(=O)CC1C)=O c1(C(=O)NC2(CO)CCN(C(C(CC)(C)OC)=O)C2)ccc(C)c(N)c1 N1(C(c2ccc(C(C)C)s2)=O)CC2CCC1C(NC(C1(Br)CC1)=O)C2 C1(NC2CC(C)NC2=O)CCCN1NC(=O)C1Cc2ccccc21 Cc1c(F)ccc(C(=O)NCC2CCN2C(c2ccc(Cl)c([N+](=O)[O-])c2)=O)c1F C1(OC)CN(C(=O)CC(F)(F)CC)C(C)(CNC(c2ncc(F)cc2F)=O)C1 N1(C(CSCC)=O)CC(CO)C2(C1)CN(C(=O)COc1cccc(Cl)c1)C2 C1(C(N2CC(C(N3CC(CCC)C3)=O)C(F)C2)=O)C2CCCCCC12 N1(C(c2sc(CC)c(Br)c2)=O)CCN(C(=O)C(O)CC)CC1CC#N c1(NCn2ccc(NC(CC(C)C)=O)n2)cc2ccc(C#N)cc2[nH]1 n1(CC(N2CCN(C(=O)Cn3nnc(=O)[nH]3)C(CO)C2)=O)ccc2ccccc12 c1(C(=O)NCCN2CCN(C(CCCC#C)=O)CC2)c(C)ccc2ncccc12 N1(C(CCNC(C)=O)=O)CCOCC(C(=O)NCC=CC2CC2)C1 C(=O)(CS(=O)CCC(F)(F)F)N(C1CCC(CNC(C(C(=C)Cl)(C)C)=O)CC1)C N1(C(C2C(OCC)C2)=O)CCOC(C)(CNC(c2cnc(C)cc2C)=O)C1 c1(CC(=O)NCCCN(CCCCNC(C(C)CC2CCC2)=O)C)ccccc1O N1(C(COCCCC#C)=O)CCCC(C(=O)NCCN2CCCCCC2)C1 Cc1nc(C(F)(F)F)oc1C(=O)NCC(c1ccco1)NC(=O)CC(C)C C(=O)(C(C)(C)CONC(=O)CC1CCCCC1NC(=O)CN1CCCCC1=O)OC N1(C(C2N(C(C(C)=C(C)C)=O)CCC2)=O)CCN(CCC2CCSCC2)CC1.C=O Cc1cc(Cc2nc(-c3ccnn3C)nn2C2CCCCC2)ccc1Br C(=O)(C#CC1(C)CC1)N(CCCN(C(=O)C(C1CCC(C(C)(C)C)CC1)O)C)C CC1C2CCC(C2)C1C(=O)NCC1CC(C(=O)NCC2(O)CCCCC2)C1 N1(C(C=C(CCC)C)=O)CCC(NC(c2cc(C)ccc2OC)=O)C(C(N)=O)C1 C1(C(N2CC(CC(C)NC(C3CC=C(C)CC3)=O)C2)=O)Cc2ccncc2N1 N1(C(=O)OC(C)(C)C)CCC2(CC2)CC1NCCC1C=CCC1 n1(CC(=O)NC2CC(NC(c3c(N)cccc3F)=O)C2)ccc2ccccc12 C(=O)(C(F)(F)C(F)(F)F)N1CCCC(C(=O)Nc2cc[nH]c2-c2ccccc2)CC1 N1(C(c2nccc(C)n2)=O)CCN(C(c2nc(Br)cnc2N)=O)C(C)C1 C(=O)(C1CCCc2ccccc21)NC1C(C)N(C(=O)CC2COC(=O)C2)CC1 c1(C(=O)NC2CN(C(C=C(C)C3CC3)=O)CC23CCC3)cc(Cl)ccc1[N+](=O)[O-] CC1(C)CC(C)(CNC(C2C(C)(C)C2(C)C)=O)CN1C(C1CC(=O)CCO1)=O N(C1CCCn2nccc21)C(C1C(NC(c2cnccc2Cl)=O)C2CCC1C2)=O Cc1cn2c(n1)CCC(C(N1CCCN(C(=O)OCc3ccccc3)CC1)=O)C2 C1(NC(c2c(CC)ccs2)=O)CC2CCC1(NC(=O)CC1CCC(=O)NC1=O)C2 c1(C2CCCN(CC(CF)F)C2)nnc2n1CCCC2 c1(CNC(COCCOC)=O)ccc2c(c1)CCN(C(=O)C(C)NC(C)=O)C2 C12CCC(CC1)C(=O)N2CC1CC1.C(=O)(C(C)(C)CF)NCCNC(C)=O C(CC(C(=O)N(C1CCCCCC1)CCNC(=O)CP(C)(C)=O)NC=O)SC n1(C2(C(=O)NC3CCC(N(C(c4c(C)[nH]cn4)=O)C)C3)CC2)cc(C#N)cn1 CC(C)C(O)C(F)(F)C(=O)N1CCC(NC(=O)C(C)Cc2ccccc2)C(O)C1 N1(C(C(CC#C)O)=O)CCC2CN(C(c3ccc(C(F)F)o3)=O)CCC12 Cn1ncc(C#N)c1C(=O)NC1CCC(C(=O)NCC2C=CCOC2)CC1 N1(C(C(C(C)C)n2cnnn2)=O)CCCCCC(NC(c2cnc[nH]c2=N)=O)C1 C1(CNC(c2cnc(C)[nH]2)=O)CN(C(c2cc(O)nc(O)n2)=O)C2CCN1C2 C(=O)(CCC(=O)NC(C)CNC(=O)CN1CCSCC1)OC O=C(C1=CCCCCC1)NC1CCC1CNC(=O)CCC1CC(CF)C1 CCCCCS(=O)(=O)CC(=O)NC1CCN(C(c2cc3cc(F)ccc3[nH]2)=O)CC1 N1(C(C2(OC)CCC2)=O)CC(C)(C)C(NC(C2CCC(C)S2)=O)C(C)(C)C1 C(=O)(C1=NOC2(CCOC2)C1)NC1(CNC(c2nncc(OC)c2)=O)CCOC1 N1(C(C(CC)(C)CNC(c2cscn2)=O)=O)CCCC(O)(C2CC2)C1 c1(-n2cc(CCC(=O)N(C(CC=C)CO)CC)nn2)c(CC)cccc1C c1(NC(C)CC2CC2)ncccc1S(=O)(=O)N1CCN(C(=O)NC(C)(C)C)CC1 c1(C(=O)NCC2C(NC(c3cc(COC)on3)=O)CCCC2)ccc(C)c(C)c1 Nc1c(Cl)cc(NC(=O)NCc2ccncc2Nc2ccc(Cl)cc2)cc1Cl N1(C(C(=O)N(CC(CC)C)C)C)CCCC(C(c2ccncc2)=O)C1 c1(N(C)CC2CCC=CO2)nc(N(C)Cc2nncn2C)nc2c1CCC2 C=CCCC(CO)NC(C1CCN(C(=O)CN(C)CCC)C1)=O CC(C)C(O)C(C)(C)C(=O)N1CCOC(CNC(c2ccc(C(F)(F)F)s2)=O)C1 C(=O)(CCCS(C)(=O)=O)N1C(CNC(c2cn(C)c(Br)c2)=O)CC2CC21 N1(CC(=O)NCCCN2CCOC2=O)CCCCC1NC(=O)CCc1cscn1 c1(C(C)NC(C2CC2)=O)ccc(F)c2cnccc12.Cc1ccc2c(c1)C(=O)N2 c1(C(=O)NC(C(F)=CC)=O)cc(F)c(CO)c(F)c1.C12CCCC(C1)N2C c1(CCNC(C(C)(F)F)=O)ccc(CNC(=O)CCc2n[nH]c(=N)s2)cc1 C=CCCCNC(C1(CC)C(C(=O)NCCCCN(C(=O)OC(C)(C)C)CC)C1)=O C1(CNC(c2ccnnc2O)=O)CN(C(C2(C3CCCO3)CCC2)=O)CC1(F)F C=C1CCN(C(=O)CCN(CCCO)C(c2cnn(C(F)F)c2)=O)C1 c1(OCC(=C)C)ccccc1C(N1CC(CCNC(=O)C(C(C)C)SC)C1)=O C(=O)(CCCC(=O)NC(C)(C)C)NCC(C(=O)NCC1CC(C)(C)CCO1)OC Cc1ccc(Cl)cc1OCC(N1CCCCC(NC(c2c(C)[nH][nH]c2=N)=O)C1)=O N1(C(CCC(C)O)=O)CCC(C)(CNC(c2cn(C)nc2-c2ccco2)=O)CC1 C1(CNC(c2ccc(F)s2)=O)CC2(CC2)C(=O)O1.C1(CC2CCOCC2)C(=O)N1 CC1CN(C(=O)CC(C)(C)CN(C)C)CCC1NC(C12CCC(CO)(CC1)C2)=O CCC(C)CCCC(=O)N1CC2CN(C(=O)C(=O)NOC)CC2C1 C12(C(=O)NCCN(C(C(C)=CC)=O)C3CCCC3)CCC(OC)C1C2 c1(SC)ccc(C(=O)NC(C)CNC(C2C=CC(C)(C)C2)=O)cc1 N1(Cc2cccc(OC)n2)Cc2c(C(=O)N(CCO)CCO)n[nH]c2C1(C)C c1(C(ONC(=O)C2(NC(=O)C(O)C3CC3)CC2)C)ccn(C)c1 C12(NC(COC)=O)CCCC1N(C(=O)Cn1cccn1)CC2.c1(O)cccc(SC)c1 c1(C(=O)NC2CC3CCC2(NC(c2ccc(Cl)s2)=O)C3)cnc2c(n1)CCCC2 c1(CC(=O)NC(CCN(C(C2(CC#C)CCCC2)=O)C)C)c(F)cccc1Cl c1(CC)ccc2cc(NC(=O)C(CNC(=O)OC(C)(C)C)C(C)C)cn2c1 c1(OC)nsc(C(=O)NC(C)CNC(=O)C=Cc2cocn2)c1Br c1(C(=O)OCC)ccc(=NCC(C)NC(c2ccnc3[nH]c(C)nc23)=O)[nH]c1 C=CCCCC(C)(C)C(=O)NC1CC2(C1)CN(C(=O)C(N1CCCCCC1)C)C2 c1(C(C)C)c(C(=O)NCC(C2CC2)N(C)C(c2cnc(N)cn2)=O)cccc1F c1(CCC)cc(C(N2CC(N(C(=O)C(C)Sc3nncn3C)C)C2)=O)no1 c1(C(N2CC(C(C)NC(c3c(SC)cccc3)=O)C2)=O)cc(O)cc(F)c1 CCC(C)C(C(=O)NC1CC(C)(NC(=O)CC2(COC)CCC2)C1)OC C1(C(N2CCN(C(C(C=C)O)=O)CC2)=O)CC(C)CC(C)(C)C1 c1(CC)ccc(CNC(C2NCCCC2c2ccccc2)=O)nc1C C1(CC(=O)NCC(C#C)OC)CC(F)CN1C(=O)C(CO)OC c1(C(=O)NCC2CC2N)cc(C)nn1C1CC1.c1(C(=O)OCC)scnc1C1CCCC1 C(C(=O)N(C1CN(C)C1)C)(C(C)C)NC(c1cc(C)no1)=O C1(NC(C(C(C)C)SCC)=O)CCCC2CN(C(=O)C=Cc3ccncn3)CC12 c1(NC2CN(C(=O)CCc3nc(O)n[nH]3)CC23CCC3)ncc2c(n1)CCOC2 N1(C(COCC=C)=O)CCC(CO)C(NC(=O)CNC(=O)C(CC)CC)C1 C1(n2c(C(c3cc(C4(OC)CCC4)n(C)n3)NC(C)C)nnn2)CCC(C)(C)CC1 c1(C(=O)NC23CC(CNC(CNC(C(CC)C)=O)=O)(C2)C3)cc(C)ccc1Cl c1(C(=O)NC2COCC2NC(=O)CCC2CC2CC2CC2)coc(C(N)=O)c1 C(C(CC)(CC)NC(C1CN(C)CCO1)=O)NC(C1CC(C)(C(=O)OC)C1)=O c1(OC)coc(C(N2CC(C)(C)CC2CNC(C2(SC)CC2)=O)=O)cc1=O C#Cc1cccc(NC(=O)CC2(CNC(c3ncccc3F)=O)CC2)c1 Cc1cc(Cl)ccc1OCC(=O)NCC=CCNC(=O)C(n1cnc(C#N)n1)C C1(C(N2CCN(CC#N)CC2)=O)CC1N=c1[nH]cnc2cnccc12 CCCC(CCCNC(C1CC2(CCC2OC)C1)=O)NC(=O)CN1CC(CC)C1 C1(CC)CCCCCN1C(=O)C(=O)NCc1ccnc(C(=O)NC2CC2)c1 c1(CN(C(C2CCN(C3CCCCC3)C2)=O)CC2CCCO2)ccnc(CO)n1 Cc1cccc2c(C(=O)NCC3CN(C(c4cnn5c4CCC5)=O)C3)c[nH]c12 CC1(C)CN(C(C2CC23CC(NC(c2ccsc2)=O)C3)=O)CCO1 C1(C(=O)NC2C(NC(C(c3n(C)ncc3)(F)F)=O)COC2)CCC(CO)CC1 c1(C(=O)NCC2(O)CN(C(c3cn(COC)nc3)=O)C2)cccc2c1CNC2=O c1(C(=O)NCCC2CCN(C)C2=O)cc2cccnc2nc1O C1(CNC(c2c(C)cc(=O)n(C)n2)=O)CN(C(=O)C(Cl)=CCl)CCC12CCC2 Cc1cnc(NCc2cnc(F)cc2C)c(S(=O)(=O)NCCN2CCCC2C)c1 C(c1ccc(Cl)c(Cl)c1)=CC(=O)NCC(C)(C)CNC(c1ccccc1)=O c1(C(C(=O)NC(C)CCCNC(c2ccsc2C)=O)OC(C)=O)cccc(Cl)c1 C(C)(C)(CCCNC(=O)CC1CCCC(C)C1)NC(c1ccc(CCC)[nH]1)=O CC1=NN(C)C(=O)C1CC(N1CCC(C(=O)NCCc2ncc(C)cn2)C1)=O C1(C(=O)NC2CC(CCNc3cc(OC)ncn3)C2)COCC2(CCC2)O1 C(=O)(NNC(=O)C(F)(F)c1cccc(O)c1)C1C(C#N)C1 N1(C(c2c(C)c[nH]c2)=O)CCCC(NC(=O)C(C)Cc2c(C)noc2C)CCC1 c1(NC(=O)NC(Cc2cnc[nH]2)CO)cccc(NC(C2CCC(F)C2)=O)c1 N1(C(COCCC=C)=O)CC(N(C(=O)CCSCCOCC)C)C(O)C1 c1(C(=O)NCC2CN(C(C3C=CCCC3)=O)CC23CC3)nccc2c[nH]nc12 c1(CC(C)C)ccc(C(=O)NC2CN(C(c3cncn3C(C)C)=O)CC2C)cn1 N1(CCC(=O)N(CC(CC)NC(=O)CC2C=CCN2C)CC)CCCCC1C C1(NC(C(C(CC)C)O)=O)COC2(C1)CN(C(=O)C(C(C)C)N(C)C)C2 C1(NC(C(c2cn(C)nc2)(F)F)=O)CCCN(C(=O)CCc2cnccn2)C1 C1(C(=O)NCCN(C(c2cccc(C)c2C)=O)CC)CCc2ncccc2C1 C(CN=c1cc(C)c(C#N)c[nH]1)=CCN(C(CC(C=C)(C)C)=O)CC1CCCO1 CC(C)S(=O)(=O)CC(=O)N1CCN(C(c2cc(Cl)cnc2O)=O)C(CO)C1 n1(CCOC)cccc(C(=O)N(c2ccccn2)CCO)c1=O.C1(=O)C(C)(C)O1 C(CC(C)(C)CC(=O)N(C1CN(C(C2CN3CCCN2CC3)=O)C1)C)OC N1(C(CCC2CCC(=O)NC2)=O)CCCCC(NC(=O)COCCF)CC1 C1(C(=O)NCC2C(CNC(Cc3cc(C)[nH]n3)=O)C2)CC(C)(C)C(C)(C)C1 C1(C)(CNC(C2CC(c3onc(C)n3)C2)=O)CCCN1C(=O)CC(C)(C)C C(=O)(C(C(C)(C)C)NC(C)(C)C)N(C1CCCC1)CC(=O)N(C1CC1(C)C)C c1(C(C)C)c(NC(=O)CC(C2CC2)NC(c2cnn(C)c2)=O)cnn1C C1(NC(=O)NC(C2CN(C(=O)OC(C)(C)C)CCO2)C)CCCN(CC(F)F)C1 N1(C(C(C=C)C)=O)CCN(Cc2conc2C2CN(C(=O)OC(C)(C)C)C2)CC1 c1(C(=O)OC)cocc1C(=O)NCCCCCNC(=O)Cn1nccc1C CC(C)CC(CNC(c1cc(Cl)no1)=O)NC(C1CC1c1ccncc1)=O Cc1ccc(CCC(N2CCC(NC(c3c(C(C)C)nnn3C)=O)C2C)=O)cc1 C(=O)(C1OCCc2ccccc21)NCCNC(c1cnc(-c2cn(C)nc2)s1)=O c1(C(=O)NC(CNC(c2c(C)ncs2)=O)C(C)C)cccc2nccnc12 C1(C(=O)NCC2CN(C(C(C)(C)C)=O)CC3(O2)CCC3)CCc2nnc(O)n2C1 CCC1C(=O)Nc2ccc(C(=O)NC3CC[Si](C)(C)C3)cc21 c1(C(=O)NC(CC)CC(=O)NCC2(COC)CCC(=O)N2)c(C)oc(C)c1C c1(C(N(CC(=O)NCC2CC3CCCC3C2)CCOC)=O)ccc2ccoc2c1 c1(CN2CC3CN(C(c4cccc5nc[nH]c45)=O)CC32)cccc2ncccc12 CC(C)CC(C)C(=O)N(CC(=O)NCCN(C(=O)CO)C(C)C)C.C(C(C)(C)O)O n1(CC)cc(C(=O)N(CC(C)NC(c2coc(C(C)C)n2)=O)CC)c(C)n1 c1(N2C(=O)CCC2)ccccc1S(=O)(=O)N1CC23CCCCCC2(C1)C3 c1(C(=O)NC2C3CCN(C(c4cccc(OC)c4C)=O)C32)nccc2cc[nH]c12 c1(C(N(CC(O)CN(C)C(C2(Br)CC2(C)C)=O)C)=O)ccc2c(c1)COCO2 Cn1cc(C=CC(=O)OC)nn1.C12CCC(O1)CC(=O)NCC1N(CC1)C2=O c1(C(=O)NCCC23C(CN(C(CC(=O)OC)=O)C2)CC3)cnc2n1C(C)CCC2 c1(C(=O)NC(C(C)NC(c2c(C)cnnc2)=O)CO)c(Br)sc(C)c1C C1(C(N2CCC(NC(C34CC(C)(OCC3)C4)=O)CC2)=O)CC1C1CC(F)(F)C1 C(=O)(CCCN(C)N=O)NCC1CCN(C(c2cnc(CC(C)C)s2)=O)CC1C CC1CN(C(=O)C(c2ccccc2)NC(=O)CCP(C)(C)=O)CCN1C1CC1 c1(CN=c2scc(C(=O)NNC(S(=O)(=O)c3cn[nH]c3)=O)[nH]2)cc(Cl)nc(Cl)c1 C#CCC(C(=O)N1CCC(OCC(N)=O)C1)NC(=O)Cc1csnc1C N1(C(C(C)OC(c2cc(C(N)=O)c[nH]2)=O)=O)CCN(CC)CC1.C(C)(C)(C)O CP(C)(=O)CC(=O)N1CCN(CCNC(=O)CCCC#N)CC1 N1(C(CN(C)C)=O)CCOC(C(=O)N(CC(C)(O)C2(N(C)C)CC2)C)CC1 N1(C(C2CC(OCC)C2)=O)CCCCC(NC(c2sccc2SC)=O)C1 CC1CN(C(C2(Cl)CC2)=O)CCC1NCC=Cc1cn[nH]c1 C#CCCCCC(=O)NCC1(F)CCN(C(=O)C(F)OC)C1 c1(C(=O)NC2CC(CC(=O)N(CCCOC)C)C2(C)C)cc[nH]c2nccc1-2 N1(C(C(COCC)C)=O)CCC(O)C(NC(=O)C(C)(C)CSC)C1 c1(C(=O)NC2C(C)(NC(c3c(C)nccn3)=O)CCC2)coc2c1COC2 c1(NC(C2C3CC2N(Cc2ccc(N4CCC4)cc2Br)C3)=O)cnc(O)nc1O C(=O)(C(C)(C(C)C)OC)N(CCCNC(c1cccc(CC)n1)=O)C(C)C c1(OC)cccc(Cl)c1CC(N1CCN(CC2CC2)C(=O)C1)=O C1(NC(C=CCCC)=O)CC2CC1N(C(c1nn(C)c(C(=O)OC)c1Cl)=O)C2 C12(C(N(C(C=C)C)C)=O)CC1CN(C(=O)CN1CCC(C)CC1)C2 c1(C(=O)NCCN(CCC)C(C2CN(C)CC2C)=O)ccnc2ccsc12 N1(C(Cc2ccc(C)cc2)=O)CC2CCN(C(c3cn(C)c(=O)n3C)=O)C(C2)C1 N1(C(c2nccc(CSC)c2)C(=O)NCCC2CC2)CC=CCC2(CCCC2)C1 n1(CC(=O)NC(C)C(C)NC(=O)CNC=O)cc(CO)nn1 CC(C)C(C)(CNC(=O)Cc1nc(C2CC2)cs1)NC(C1CC2CCC1C2)=O C1(NC(c2nc(C(N)=O)sc2)=O)(CNC(c2cncc(F)c2)=O)CC2CCC1C2 C=C1COc2c(C(=O)NCC(C3CCCC3)NC(c3sccc3C)=O)cnn2C1 C1(C(N(CCCNC(C2CC(=O)N(C)C2)=O)CC)=O)CCc2ncc(C)n2C1 CC1CC=C(C(=O)N(C2CCOC(C)C2)C)CC1.c12cc(on1)C(=O)NC2 Cc1cccc(COC(C)C(=O)NCCC2(NC(=O)CC(C)O)CCC2)c1 c1(C(N2C(CCC(=O)NCC(C)(C)CC3CCOCC3)CC2)=O)ncc(CC)[nH]1 C(=O)(C(C)(C)C(=O)NC(CCN(C)C(C1Cc2nccn2C1)=O)C(C)C)NC CC(C)(C(=O)N1CC(F)(CNC(=O)CSC2CC2)C1)c1cncs1 CCCC(C)(O)CC(=O)NC1CC2(C1)CC(C(N1CCOC(C)(O)C1)=O)C2 N1(C(c2ccc(Br)c(C)c2F)=O)CCn2nnc(C(=O)NC(C)CN(C)C)c2C1 C(=O)(C(C)(O)CCC)N1CC(CCC)C(NC(c2c(C)nsc2C)=O)C1 c1(CC(=O)OC)cnn(C)c1NC(=O)NCCC(C(=O)NC1CC1)OC C1(C)(CNC(CCCC)=O)CCN(C(=O)C(N2CCC(O)CC2)C)C1 C1(NC(C(C=C)C)=O)CC2CC(C1)CN(C(=O)CCc1cccc(C)c1)C2 Cc1ccc(C)c(CNC(C2CCCN2C(C2CCC(C)O2)=O)=O)n1 CC1CCN(C(c2nc(C3CC3)cs2)=O)CC1NC(c1ccc(C(C)(C)C)[nH]1)=O c1(C(=O)NC2C(NC(C(C(CC)C)O)=O)CCCC2)cc(F)cc(Cl)c1O Cc1nn(C)c(=O)c(C(N2CC3(C2)C(NC(=O)C(N)=O)CCS3(=O)=O)=O)c1C N1(C(C(C2CC2)SC)=O)CCCC(C)(CNC(=O)CCCCCNC(C)=O)C1 CC(C)CC(C(=O)N(CC(O)CNC(c1ccn2ccnc2n1)=O)C)C(C)C C1(NC(c2c(CC)n(C)nc2)=O)CC2CC(NC(=O)C(F)(F)C(O)C3CC3)C1C2 N1(C(C(C)N(C(C2CN(C(C)=O)C2)=O)C)=O)CCCC(CCF)C1 CC(C)C(O)CC(=O)NC(C)(C(=O)NCC1(S(C)=O)CC1)C1CCC1 c1(C(N2CCC3(CC2)CN(C(=O)CC2CC2)C3)=O)c[nH]c2cccc([N+](=O)[O-])c12 C1(NC(=O)C=CCO)C2CN(C(=O)COC3CC=CC3)CC12 C12(COC)CCC(C(=O)NCC3CCOCCN3C(=O)CC(C)CF)(CC1)CO2 C1(NC(COC(CC)(C)C)=O)CC2CCC1(C(=O)N(CC(O)CN(C)C)C)C2 Cc1cnc2n1C(C(=O)N(CC(O)CN(C(=O)CSCC(F)F)C)C)CCC2 c1(C(=O)Nc2c(C(N(CCCOC)CCO)=O)c[nH]c2)c[nH]c(C#N)c1C C(CCC(=O)NCC(=O)N1CCC1)OC(C)=O.C(=O)(C(C)S)N(C)CCO c1(NC(=O)NC(c2ccc(Cl)cc2Cl)C)ncc([N+](=O)[O-])cc1O C12(NC(=O)CSCC(F)(F)F)CCCN(C(c3cc(O)nc(O)n3)=O)CC1C2 C(CCN=c1nc(Cc2ccccc2)cc(N2CCCCCCCC2)[nH]1)NC(C)=O C1(C(N(CCN(C)C(c2cccs2)=O)C)=O)CCN2CCOCC12 Nc1ccc(C(N2CC(NC(C3CC(=C4CC4)C3)=O)C3(CC3)C2)=O)c(F)c1 C(=O)(C(C)(C)CNC(=O)CCC1(C)N=N1)NC(C)CN1CCOCC1 C=CCC(C(=O)N1CCC(CNC2CCN(c3ccccc3)C2)CC1)NC(C)=O C1(C(=O)NC2CC(CCNC(c3cc(CSC)c(C)o3)=O)C2)(CC)CCNC1=O C(=O)(C1=NOC2(CCN(Cc3ccc(NC(C)=O)s3)C2)C1)NC(CC)C(C)O c1(SCC2C(CC(=O)N(CCCC)CCOC)C2)sccc1Cl C=CC1CN(C(c2cc(Cl)cc(Cl)c2)=O)CC1NC(=O)CCCC(C)=O c1(C(CO)NC(=O)NC23CC(CCC(=O)OC)(C2)C3)cccc(F)c1Br C#CCC(CC(=O)NC(c1cnsc1)C)NC(=O)C(C)=C(C)CC N1(C(c2n(C)nc(CC)c2Cl)c2nnnn2CCCF)C2CCC1CC(F)C2 C1(CNC(CN(C2CCC2)C)=O)CC(C)(C)CN1C(C1C=CCCC1)=O C1(NC(CC(C)(F)F)=O)COC2(CCN(C(c3sccc3C(F)F)=O)C2)C1 Cc1ccc2n[nH]cc2c1C(=O)NC(CNC(=O)CC1CCCC1(F)F)C(C)C N1(C(CCN(C(=O)CS(C)(=O)=O)C)=O)CCCc2sccc2C1 N1(C(CC2CC(C)(C)C2)=O)C2CCC1CC(CNC(=O)C(F)(F)CC1CC1)C2 C1(NC(c2cc(C)cc(O)n2)=O)CCCCCN(C(=O)CSc2ccncc2)C1 Cc1cc(OCC(=O)NC2CCC(NC(=O)Cn3cc(Cl)cn3)CC2)ccc1F N1(C(C(N2CCC(c3ccccc3Br)C2)=O)C2(C)CC2)CCCNCC1 c1(C(=O)NC(C)CCN(C(=O)CC2(C(F)(F)F)CC2)C)ccsc1Cl c1(CN(C)C(=O)NCCN(c2cnccn2)C)cnnn1C CC1CCCC1(C(=O)N(C1(CCO)CC1)C)NC(=O)CN(C)C(N)=O C1(O)(CCNC(c2cc(CF)on2)=O)CCCN(C(C2COCCC2(F)F)=O)C1 c1(C(N2C(CNC(CC=C(C)C)=O)CC(O)C2)=O)csc(S(C)(=O)=O)c1 N1(C(=O)Cc2ccc(C#N)s2)CCC2(C=Cc3ccccc32)CC1.C1(=O)CO1 C=C(C)C1CN(C(=O)CC2C(NC(=O)C=Cc3cc[nH]n3)CC2O)CCO1 S(=O)(=O)(c1cn(C)nc1C)Nc1ccc(C(=O)Nc2c(C)ccc(Br)c2)nc1 C(=O)(CC(F)(F)F)NC(C)C(=O)NCCC1CCCN(C(c2ccno2)=O)C1 C1(CCC(N2CCCC2Cn2cc(C3CCC3CC=O)nn2)=O)CCCCC1 C#CCCCCCC(C(=O)Nc1ccc(Cl)cc1F)N1CCC(C(=O)OC)CC1C N1(C(C2(CC(C)C)CC2)=O)CC=CC(NC(c2cc(-c3cnn(C)c3)no2)=O)C1 c1(OC)c(C(=O)N(C2CN(C(c3cnn(C(C)C)c3C)=O)C2)C)ccc2c1CCC2 c1(CN(CCC)C(=O)NC2CC(C(N)=O)C2(C)C)ccc(Cl)cc1Cl C1(C(=O)NCC(CNC(CC(C)(C)F)=O)F)Cc2nncn2C1 C#CCC(C)(C(=O)N(C)CC1CCCC1(C)C)NC(=O)C(COC)N(C)C C1(CC)CN(C(c2cccc(Br)c2)=O)CCN1C(c1cc(C)cc(Cl)c1)=O C1(CCC)(CNC(C2C=CCN2C(=O)Cc2ccsn2)=O)CC(=O)C1 Cc1cc(F)c(C(N2CCC(NCc3cn4ccsc4n3)C(C)C2)=O)c(F)c1 Cc1ccc2sc(C(N3CCC(NC(c4c(C)cncc4C)=O)C3)=O)c(C)c2c1 c1(C(C)C)cccc(C(=O)NCC2CCC(C(=O)Nc3nnc(Br)s3)CC2)c1O CCC(CC(=O)N(CCC(=O)NCC(N1CCCCC1)C)C1CC1)OC C1(C(=O)NCCCOCCCNC(C(C)n2cccn2)=O)CNC(=O)N1 C1(C(N2C(C(=O)NC3(C)CC(C)C3)CCC2)=O)(OCC)CCCC1 N1(C(COCC)=O)C2CCC1CC(CNC(=O)CC1(C)CCOC1)C2 c1(C(=O)NCC(C)N(C(CC2CC(OCC)C2)=O)C)cc(F)ncc1C(N)=O O=S1(=O)CCCN1C(c1ccc(Cn2cc(C3(O)COC3)nn2)cc1)=O C1(CC)(NC(c2cc(O)cc(=O)o2)=O)CCN(C(=O)C(CC)n2cncn2)CC1 C(=O)(CCCCCOCC)NCC1CC(CNC(C(C)OCCC=C)=O)C1 CC(CCNC(=O)Cc1cccc(NS(C)(=O)=O)c1)CCNC(C1CC(O)C1)=O c1(CCC(=O)NCCN(C(=O)CCOC2CCC2)C(C)C)ccncc1.C(C)(=O)O CCC(C)CC(C)C(=O)N1CCC(c2cn(-c3ccccc3Cl)nn2)C1(C)C C1(NC(CN(C)C(=O)C2CC2)=O)CCCCN(C(C2(n3cc(Cl)cn3)CC2)=O)C1 C(C(=O)N(CC1CC2CC2C1)OC)N(C(C(C)SCCCC)=O)CC N1(C(C2N(C(c3c(OC)ccs3)=O)CCC2)=O)CCC(O)CC1C(F)(F)F CCCCC(C(=O)N=c1cc(C(N)=O)n(C)[nH]1)NC(=O)CC(C)CC(C)C O=C1CN(C(N2CCc3ncccc32)=O)c2ccccc2N1 C1(C(=O)NC(C2CCCCC2)CNC(C2C(=O)NCC2)=O)Cc2cccnc2C1 CN1N=C(C(=O)N2CCC(C(=O)NCCCn3cncn3)C2C(F)F)CCC1=O c1(NC(C)=O)cccc(C(C)NC2CCOC(c3ccccn3)C2)c1 c1(COC(C2(CO)CC2c2ccccc2)=O)ccc(Br)cc1I C(C)(C(=O)N1CCC(C(=O)NC(C)CCC(C)(C)C)O1)OCC(C)C C1(C(=O)NC(CCNC(c2c(C)oc(C(C)C)n2)=O)C(C)C)CCC2CCC1O2 C=CC1CCN1C(=O)C(C)N(C(=O)CC1CCC(C)O1)C C1(N(S(C)(=O)=O)CC)C2CN(C(c3csc(-c4ccsc4)n3)=O)CC12 c1(CNC(C2(NC(C(COC)N(C)C)=O)CC2C)=O)ccncc1Cl C1(CC(=O)NC2(CNC(=O)COCC3CCOC3)CC2)C=CS(=O)(=O)C1 N1(C(C2C(C)C2)=O)CCC(F)C(NC(c2ccc(CCF)cc2)=O)C1 C1(C(=O)NCC(C)CNC(=O)Cc2cc(F)ccc2F)CCC2(CCC2)CC1 N1(C(C=CC(C)=O)=O)CC(F)CC1CN(C)C(c1ccccc1CC=C(C)C)=O CC1(C)CC(NC(c2ccsc2Cl)=O)CN1C(=O)CNC(C1CCC1)=O c1(C(N2CC3C(C2)N3C(C2CCC(F)(F)C2)=O)=O)cccc([N+](=O)[O-])c1O CC1COCCN(C(=O)C=CCC2(NC(C3CC(=O)CS3)=O)CCC2)C1 Cc1cc(Cl)c(C(=O)NCC(CC(C)C)NC(C2CCN2S(C)(=O)=O)=O)s1 C(=O)(C(C)(C)CCS(C)(=O)=O)NC1CN(C(COCC(=O)NC)=O)CC(O)C1 c1(C(=O)NCC2C=CCN2C(=O)C2=CCCS2)ccc(F)c(C2CC2)c1 N1(C(C2NC(=O)OCC2)=O)CC(NC(c2cc3ccncc3[nH]2)=O)CCC(O)C1 CCCCC(O)CNC(=O)C(Cn1cccn1)NC(=O)CSC(C)C CCC(C)(C(=O)N1CC2CCC2(NC(=O)C=CCCC=C(C)C)C1)C(F)F N1(C(C(c2ccc(Br)cc2)(C)C)=O)Cc2[nH][nH]c(=NC(=O)c3cnnc(O)c3)c2C1 C12(NC(C3(c4ccc(F)cn4)CC3)=O)CCC(=O)N1CCS2.C12CC1C(=O)N2 c1(C(=O)NC2C(CNC(C3CC(C)(C)OCC3)=O)CCC2)cc(F)cc(N)c1F N1(C(c2cccc(OC)c2)=O)CC2CCC(NC(c3sccc3C#N)=O)(C2)C1 C(=O)(C(Cc1ccccc1)C(F)(F)F)NCC(C)N(C(C(C)OC)=O)C c1(C(=O)NCCC2CC(NC(c3nc(COC)oc3)=O)C2)cccc(Br)c1 c1(COC(N2CC(C(=O)OCC)C(N(C)C)C2)=O)cc(Br)c(C)cc1F C(=O)(C1CCc2nnc(C)n21)N1CC(C2(NC(c3c(CC)csc3)=O)CC2)C1 Cc1cc(C(N2CCCC2C(=O)NCC(F)F)C(=O)NC(C)(C)C)ccn1 c1(CC)cc(C(N2CC(OC(C)=O)C(NC(=O)CS(C)(=O)=O)C2)=O)sc1C C=C(C)CCCC(=O)N(CC(C)NC(=O)C=Cc1ccc(Br)cc1)C CC(CNC(C1(C)CC(NC(C2CN(C)CCN2C)=O)C1)=O)CC(F)(F)F Cc1cn2c(n1)C(C(=O)NCCCCNC(C1CC13CC(C)(C)C3)=O)CCC2 N1(C(c2c(NC)cccc2)=O)CC2CC1CN2C(=O)CCc1ccn(C)c1 C12(CNC(C(C(C)O)C)=O)CCC(C(F)(F)F)(CC1)C2.C12(F)CN(C1)C2=O n1(CC(N2CC3C(CNC(c4ncn(C)n4)=O)(C3)C2)=O)ccc(O)nc1=O c1(C(=O)NC(Cn2cc(-c3cc(C)c(F)cc3)nn2)C)ccc([N+](=O)[O-])cc1 Cc1c(C(=O)N(C(CNC(=O)C(C)(C)C(C)(F)F)C2CC2)C)cc(O)cc1N N1(C(CCc2scc(C)n2)=O)CCCC(NC(C2CN(C3COC3)C2)=O)C1 C#CC1CN(C(=O)CC(O)CN(C)C)CCN1C(c1cnn(C(C)(C)C)c1)=O C(N=c1[nH]c(Cl)nc2c1SCC2)C1C(NC(c2cncnc2)=O)CCCC1 C(CC1CCCCC1)(C(=O)NC(C)(C)C)NC1CC(CCC)C1 c1(C(N2CCC(N(C(CSCCOC)=O)C)CC2)=O)cnc2n1CCC(C)C2 N1(C(C(c2scc(C)n2)(F)F)=O)CCC2C(NC(c3coc(C)n3)=O)C2CC1 N(C(=NCc1ncccn1)NCc1nc(C2CC2)n[nH]1)C(C#C)CCC C(=O)(C1=NOCC1)N(CCCNC(=O)Cc1cc(-c2ccco2)on1)CCO c1(C(=O)NC(C)CN(C)C(c2nccc(Cl)c2F)=O)ccn2c1CS(=O)(=O)CC2 N1(C(=O)Nc2c(C)nn(C)c2CN2CCCC2)CCc2cccc(C)c21 C1(C(N2C3(C(=O)NCCC(C=C)C)CC(C2)C3)=O)CC2CCCC2C1 C1(=O)C(F)CC(C)(C)N1.CCC(C)C(CNC(=O)CCSC(F)(F)F)CO N1(C(CCOCCOCC)=O)CCN(CC(C)(CC)NC(=O)C(C)OC(C)=O)CC1 C(C(O)C(F)(F)F)N(C)C(=O)NCc1nc(-c2ccncc2)cs1 C1(C(=O)NCc2cc(COC)on2)CCC(O)CN1C(c1ccccc1F)=O CCC(CC)C(C)C(=O)N1CC(O)CC1CNC(C12CCC(CC1)C2)=O c1(C(C)C)nc(C(=O)NC2COCC2NC(=O)C(C)CN(C)C)co1 C1(C(=O)NC2CC(CNC(C(C)(C)c3ccccc3)=O)C2)Cc2ccccc2S1 C1(C(N2CC(CCCCNC(C3CCN(C4CC4)C3)=O)C2)=O)CC(=C(F)F)C1 CCCC(F)(F)C(=O)NC(CC(N1CCC(C)C1C)=O)C1CC1 CC(=O)CC(C)(C)C(=O)N1CC2C(C(=O)NCC(O)COC(C)C)C2C1 c1(C(N2CCC(N(C(=O)C3=COCCO3)C)C2)=O)cnn2c1CCCN2 C1(C(=O)NC2CC(C(F)C(=O)NCCc3cc(C)[nH]n3)C2)(CC)CCCC1O O=C(CCS(=O)(=O)c1ccc(Cl)cc1)NC1(F)CCN(C(=O)CO)C1 c1(C(N(CC(CNC(CCCN(C(C)=O)C)=O)O)C)=O)cnc2c(ccn2C)c1 CCCCCC(CC)C(=O)N1CC(C(=O)Nc2cc(Cl)ccc2F)CC(C)(C)C1 c1(CC(=O)NCC(C)(C)NC(c2cncc(OC)c2)=O)c(F)c(F)cc(F)c1F Cc1c(CN2CCC2C(=O)NCc2ccc(SC(F)(F)F)cc2)cnn1C CCCC(C(=O)NCC1(C(N)=O)CN(C(=O)Cc2cc(Cl)n(C)n2)C1)N(C)C c1(C(=O)NCC(CNC(C(C)N(C(=O)CC2(OC)CC2)CC)=O)OC)nccn1C CC(C)CC(=O)C(=O)N(C)Cc1ccc(SC(F)F)cc1 CCCC(C)(C)CC(=O)N1CC(NC(c2cc(N)nc(Cl)c2)=O)C(n2ccnn2)C1 c1(N2CC3(C(N)CC3)C2)cc(Br)c(I)c(Cl)c1 c1(C(=O)NC(CC(C)C)CNC(=O)C=C2CCCCC2)ccc(N)cc1Cl N1(C(C2C(CC)N(C)CC2)C(=O)NCc2cc(C)nc(C)c2)CCC(C)(C2CC2)C1 c1(C(=O)NCC2COCCN(C(C(C)NC(CC)=O)=O)C2)cc2ccccn2c1 CC(C)(CCCNC(C1CCN(C(=O)C=Cc2nccs2)C1)=O)NC(N)=O C1(NC(C2C(NC(c3ccc[n+]([O-])c3)=O)CC2)=O)CCn2ccnc2C1 Cc1cc(F)cnc1C(N1C2CCC(C2)C1CC(=O)NC(C)CC(C)C)=O c1(C(c2nnnn2C2CCCC2)CCC=CCCC)c(OC)ncc(Br)c1F c1(C(=O)OCC)ccc(NNC(=O)C2CCN(c3ccccn3)CC2)cc1 c1(CC)ncnc(CC)c1C(=O)NC(CCN(C(=O)COCCF)C)C(C)(C)C c1(C(=O)NCC2C(NC(C3(CC=C)CCOC3)=O)CC2)ccc(C)nc1C N1(C(CSCCCC)=O)C2CCC(C2)C1N(C(=O)CCCCCF)C.C1(C)(C)CN1 N1(C(c2n(CCC)ncc2)=O)CCC2(C1)CN(C(=O)C(C)CSC)C2 C1(C(=O)NCC2(CNC(c3ccc(C4CC4)o3)=O)CC2(F)F)CCC2(CC1)CC2 Cc1nn(C)c(CNc2cccc(SCCc3ccccc3)c2)c1Cl c1(OC)c(F)ccc2[nH]c(C(=O)NC(CNC(C3CCCS3)=O)C(C)(C)C)cc12 C1(NCC(C)C(=O)N(C)C)COCC1(C)C.C(C=O)C(=O)NCCOCCCN c1(C(=O)OCC)ocnc1C(=O)N(C1CCC(NC(C2=CC=C(CC)C2)=O)C1)C C1(NC(c2cnnc(-c3ccccc3)c2)=O)CN(C(=O)COCCF)CCC1F C(=O)(C(C)(C)O)C(=O)CC1CC(C(N(CCC(N)=O)CC)=O)C1.N CC1CC(NC(C2CCC2)=O)CN(C(=O)C(C)(CO)CO)C1 c1(CC(=O)NCc2cccc(NC(C(C=C)(C)C)=O)c2)ccc2c(c1)CC(=O)N2 C1(NC(=O)NCC(C)CNC(=O)CSCCN(C)C)CCC(F)C1 C1(O)(CC)CCCN(C(C(=O)NCCCC2CC2)C(C2CC2)OC)C1 C(=O)(CC(C(C)C)NC(=O)CC1CC2CCC1O2)NC(c1cccnc1)CC C1(CNC(COCC(=C)C)=O)CC2CCC1N2C(=O)CC1CCN(C)C1 c1(CC)nc2sc(C)cn2c1C(=O)NCC=CCNC(C1CCCCCC1)=O C=CCC(C)(C)C(=O)NC1CC(NC(=O)CCCC(=O)c2ccc(F)cc2)C1 C12(CN(C)C(c3cn[nH]c3)=O)COCC1C2.C1CCOC(=O)C2(CC2)C(=O)N1 C(=O)(C1=NOC(C)C1)NC(CCCNC(C1(CC(C)C)CC(=O)C1)=O)C N1(C(=O)NCC(c2ccc(F)cc2F)C)C2CCC1CC(CCOC(C)(C)C)C2 c1(C(=O)NC(c2ccc(Cl)c(Cl)c2)CC(=O)OC)ccc(C)cc1C N1(C(c2cc(OC(C)C)n(C)n2)C(=O)NC)CCCC(O)(CN(C)C)C1 C(=O)(C(O)CC[S+](C)C)N1CC(CN(C)C(c2cccc3ccoc23)=O)OCC1 N1(C(CCC(N)=O)=O)CC2CCN(C(=O)C(O)CN3CCOCC3)CC12 c1(C(=O)NCCNC(c2cnn3c2CCC3)=O)cc2c(ccc3ccccc23)o1 c1(OC)cccc2cc(C(=O)NC3(CCCNC(=O)C(C)=CC)CC3)c(=O)oc12 C1(CNC(C=CC=CCC)=O)CCN(C(c2cc(C)[nH]n2)=O)CC1(F)F C1(NC(CCC#CC)=O)CN(C(=O)CSc2cccc[n+]2[O-])C(C)(C)C1 c1(-c2cn(C3CCN(C(=O)CSC4CC5CC5C4)C3)nn2)cccc2ccsc12 c1(C(=O)NC(C(N2CC(C(C)C)(CO)C2)=O)c2cccs2)cnc2cc[nH]c2c1 N1(C(=O)OC(C)(C)C)CCc2nn[nH]c2C1.c12noc(n1)CCC(=O)NC2C c1(C(=O)NC(C)CNC(c2coc(C3CC3)n2)=O)cc(O)nc2[nH]c(=N)ccc12 C1(CC(N2CC(NC(c3cnc(CC)[nH]3)=O)C(F)C2)=O)CCC2(CCC2)O1 N1(C(=O)Cc2cnns2)CCN(C(c2ccc([N+](=O)[O-])o2)=O)C2CCC12 C=CC(CC)CC(=O)N1CCOC(CN(C(=O)C(F)(F)CC2CC2)C)C1 C1(C(=O)NCC(C2CC2)NC(C2(COC)CCCO2)=O)CN2CCCN1CC2 C(C)(C)(CCN=c1ccnc(NC(C)(C)C)[nH]1)NC(C(C)(C)C1CCCCO1)=O C(=O)(CC(C)CNC(C1(C)CC(C)=NO1)=O)NC(C#C)CC c1(SCC(=O)NCC2CN(C(CC=CC=C)=O)C3C2C3)ccc(F)c(F)c1 Cc1ccnc(O)c1C(=O)NCC(C)(C)NC(=O)C(c1cccc(Cl)c1)C C1(N(C)C)CC(C(=O)NC2CC=CCC2NC(=O)C(O)C2CCCC2)C1(C)C N1(C(CCc2n(C)ccn2)=O)CCOCC1CC1CC1.C12CCCN1C(=O)NC2=O C(=O)(C(C)(C)C(F)(F)F)N1CC(C)(C)C(CNC(=O)C(F)=C2CCC2)C1 CN1CCN(C(c2scnc2C(F)F)=O)CC1CNC(c1cc(C(N)=O)[nH]n1)=O N1(C(CNC(CC)=O)=O)CC(NC(=O)C(=O)NC(C)C)C1 C1(C(=O)OC)CC2CN(C(=O)NC(c3ccc(C(C)C)cc3)C)CC2C1 C(=O)(C(CC(F)F)C1CCC1)NCC1CCC(CNC(C2CN(C)C2)=O)CC1 C1(CC(=O)NC(Cn2cc(CC(=O)NCC(=O)NC)nn2)C)CCCNC(=O)C1 C(c1ccc(Cl)cc1F)=CC(N1CCC(NC(C2CCC(=C)CC2)=O)C(F)C1)=O C1(CNC(c2c(CC)noc2)=O)CN(C(=O)C(CC)SC)CCO1 c1(NCC(CCC)OC)ccc(S(=O)(=O)NCC2CCCC(F)(F)C2)cc1F c1(C(N2CCC(NC(C3ON=C(CC)C3)=O)C2(C)C)=O)cccc2c1CCC2 N1(C(CC2CC(=C)C2)=O)CCC(NC(c2cc(C)oc2CC)=O)C(O)C1 c1(-n2cc(C(CC(N)=O)NC(Cn3ccc(C)n3)=O)nn2)ncccc1C(=O)O C1(NC(c2cncc(F)n2)=O)CCCCN(C(c2scnc2Cl)=O)C1 c1(CC(N2CC3CC(NC(C4(C5CC5)CC4)=O)C(C3)C2)=O)cnn2c1OCCC2 C1(C#C)(C(=O)NC(C2CCCC2)C#C)CCN(C(=O)C(CC(C)(C)C)OC)CC1 C1(CCc2cn(C(C)C(=O)N(C3C4CCCC34)C3CC3)nn2)SC(=N)NC1=O N1(C(C(C)C(F)F)=O)CC2CC(C1)CN(C(=O)C(C)Oc1ccccc1F)C2 N1(C(Cn2c(C)nc(C)n2)=O)CCCCC(NC(=O)CN2CCCNC2=O)CC1 c1(CC(C)C)ccc(C(N2CC(CO)(NC(C3(C4CC4)CC3)=O)C2)=O)cc1 C(N=c1[nH]cnc(Cl)c1Br)C1(OC)CN(C(c2ccc(COC)[nH]2)=O)C1 N1(C(C2(OC)CCSC2)=O)CCC(=CCNC(=O)C(n2cnc(C#N)n2)C)CC1 C1(C(N2CCC(NC(=O)CCc3ccc(Cl)s3)(CO)C2)=O)CCC(F)(F)CC1 C12(C(=O)NCC(CN(C(C3(COC)CCC3)=O)C)(C)C)CCCCC1C2(F)F O=C1CC(CC(=O)NCC(c2ccccc2)NC(C2CSC2)=O)CCCN1 c1(C(C)C)ccc(C(=O)NC(C)CCCNC(=O)CC(C)C(C)C)cc1[N+](=O)[O-] C1(C)(C(=O)NCCNC(C2C(C)(C)C2C(=O)NCCCCSC)=O)CCCC1O C12(NC(c3cc[nH]c3C3CCC3)=O)CCC(CF)(CC1)CC2.C12CC(C1)CNC2=O C1(CN(C(CCNC(=O)OCC)=O)C)CCCN1C(=O)CC1C=CCC1 c1(CC(=O)NCC=CCC(=O)NCC2(C)C(C)(C)C2)ccc(F)cc1 Cc1cc(C(=O)N(C2CCCC(NC(c3nc(Cl)oc3C)=O)C2)C)n(C2CC2)n1 C1(NC(c2c(CC)scc2)=O)CN(C(C2(C)C=CCCC2)=O)CC12CC2 N1(C(C)C)CCCC(C(=O)NCC2CC(NC(=O)C(C)(O)C3CCC3)C2)C1 Cc1cc(F)ccc1C(O)C(=O)NC(C)C(C)(C)NC(=O)C=CC(C)(C)C c1(OC)ccc(Cl)cc1C(N1CCOC(CN(C(=O)COCCF)C)C1)=O Cc1cnccc1-n1cc(CCCNC(C2CCCN(C(N)=O)C2)=O)nn1 c1(CC)noc(C(=O)N(C)CCN(C)C(C2CCN(C(C)CC)CC2)=O)c1C CC1CN(C(=O)C(F)(F)c2ncc[nH]2)CCN1C(=O)C(F)=C1CCCC1 c1(CNC(C(=O)NCC)=O)cnn2c1CN(C(c1cnc(C3CCC3)s1)=O)CC2 c1(NC2CC(C)N(Cc3ccccc3)C2C)cc2c(nn1)CCCC2 Cc1nc(C)c(C(=O)N(C2CCN(C(C3CCOC3)C)C2)C)o1 C1(C(=O)NC2C3CN(C(C(c4ccccc4)OC)=O)C2C3)CC2CCC1CC2 C1(CC)C(C(=O)NC2COCCOC2)CCCN1C(C1CCSC1)=O N1(C(c2nc(CC)oc2C)=O)CCC(NC(c2coc(C3CCC3)n2)=O)CC1C c1(CCCNC(C2(OC)CCC2)=O)cnn(CC(=O)NCC2(CC)CC2)c1 C(CC(C(=O)N(CCS(C)(=O)=O)C)OC)NC(c1c(CC)ccs1)=O c1(C(=O)NC(C)CCCNC(C2(Cl)CC23CCC3)=O)cnc2ccoc2c1 Cc1cc(C(=O)NC2CCCC(CN(C)C(c3cc(CO)[nH]n3)=O)C2)cc(C)c1 Cc1ccn2cc(C(=O)NC(C3CCN(C(=O)C(F)CC4CCC4)C3)C)nc2c1 Cc1cc(P(C)(C)=O)oc1C(=O)NC(C1CCN(C(C2(F)CC=CC2)=O)C1)C n1(CCCC)ncnc1CNCCc1cccs1 c1(NC(C2CCC(NC(C3(F)CCOCC3)=O)C2)=O)ncc2c(n1)NC(=O)C2 c1(C2(C(=O)NC3CCCC3NC(C3(C(F)F)CCCO3)=O)CC2)nnc(S)n1C C1(O)(CNC(c2ccoc2C2CC2)=O)CCN(C(C2CCC2)=O)C1 [N-]=[N+]=NC1CC(C(N2CC3(CC(F)C3)C2)=O)N(C(=O)C(C#N)CCCF)C1 Cc1cn2cc(C(=O)NCC3CCCN3c3ncc(C(N)=O)cc3Cl)sc2n1 C1(COC)CCCC1C(=O)NC1CC1CNC(c1conc1C(C)C)=O C(C)(C(F)(F)C(F)(F)F)NC(C(C)Oc1ccc(Cl)cc1)=O Cc1cnc(N2CC=CC(OC(F)(F)F)C2)c(S(=O)(=O)N2CC3CCOC3C2)c1 N1(C(=O)Cc2ccco2)CCC2C(CCCN2C(c2cccc3[nH]ccc23)=O)C1 c1(C(=O)NC2COCCN(C(=O)C(F)(F)CO)C2)ccc2c(c1)S(=O)(=O)NC=N2 C1(N(C(c2c(SC)ccs2)=O)C)CCCN(C(=O)C(C2CC(F)(F)C2)O)C1 Cc1nc2ccc(C(N3CC4CC(C3)N4C(c3cc[nH]n3)=O)=O)cc2[nH]1 C(CC(C)C(=O)NCC(CC(C)C)NC(=O)Cc1c(Cl)cnn1C)OC C=CCC(CCC=C)NC(=O)CN(C(=O)C(C=C)CC)C(C)C C1(C)(C(N(CCCCCC=C)C)=O)CCCN(C(=O)C(COC)OC)C1 Cc1nn(C)c(Br)c1C(N1CCCC1Cc1ccco1)=O CS(=O)(=O)c1ccc(CC(=O)OCCCCCN2CCOCC2)cc1 Cc1coc(C)c1C=CC(=O)Nc1cccc(NC(=O)C(=O)N(C)C)c1 CC1(C)CCCCC1NC(=O)CCCCCNC(=O)C(F)C1CCCC1 C1(C)(C(=O)NC(C2CCCC2)CNC(C2CC(OC(C)C)C2)=O)CCC2CC2C1 N1(C(=O)Nc2cn(CCOC)nc2)CCC2(CC1)CC2(C#N)CO c1(CC)cc(C)ccc1C(=O)NC(CNC(=O)C=CCN1CCOCC1)(CC)CC C(CNC(C1CCC1CNC(=O)CC1OCCC1C)=O)(C(F)(F)F)OC N1(C(C2(C#C)CCCC2)=O)CCCC(NC(=O)C(C)(O)c2ccccc2)CC1 c1(C(=O)NCCOCCNC(c2ccn(C)c2)=O)cncc(P(C)(C)=O)c1 C12(OC)CCC(C(=O)N(CCCCC(=O)NS(C)(=O)=O)CCC3CC3)(CC1)C2 c1(N(CCC(=O)NC)C)ccc(C(=O)NC2CC2CNC(=O)C(C)CCOC)cc1 C1(O)(C(=O)NCC2C(NC(C3(O)CC(c4ccccc4)C3)=O)C2)CCSCC1 c1(C(=O)NCCCCCNC(C(C)C(F)F)=O)cc(N)c2ncccc2c1 C1(CCNC(=O)Cc2ccccc2)(CNC(C=CC(CC)C)=O)CCCC1 C=C(C)C1OCCC1C(=O)NCC1CCCCCN1C(=O)CCC1CC(OCC)C1 Cc1ccnc(O)c1C(N1CCN(C(c2cccc(Br)c2Cl)=O)CC1)=O C1(C(=O)NCC2N(C(c3c(C)[nH]c(C(F)(F)F)c3)=O)CCC2)CCC2CC2CC1 C1(CNC(C2(SCC)CC2)=O)CN(C(c2ccc(C(C)F)cc2)=O)CCO1 C1(NC(Cc2c(C)con2)=O)CCN(C(c2c[nH]nc2C2CC2)=O)C(C)C1 c1(C(=O)NCCC(C)NC(=O)Cc2cscc2F)n[nH]c2ccc(Cl)cc12 S(=O)(=O)(c1ccc(NCc2cnc(C)s2)c(Cl)c1)NC1C2(CC(OC)C2)C1 C(=O)(C1=CCCCC1P(C)(C)=O)NC(CNC(c1cc(C(C)C)no1)=O)C1CC1 CC1CC(NC(=O)CC2(CS(C)(=O)=O)CC2)CCN1Cc1cc2ccsc2[nH]1 N1(C(C(C)=CC)=O)CCC(CNC(c2oc(C3CC3)nc2C)=O)(OCC)C1 C1(C(=O)NCc2c(C3CN(C(c4c(C)nco4)=O)C3)ocn2)CC(O)CN1C c1(C(=O)NCC=CCNC(C2(C)CC(C)(C)C2)=O)cc(C2CC2)nc(O)c1 Cc1nn2ncccc2c1C(N1CC2CCC(C1)N2C(c1sc(F)cc1Cl)=O)=O C1(CNC(c2n(CC)ncc2Cl)=O)COC(C)(C)CN1C(=O)Cc1cscn1 C1(C(N(C)Cc2nnc(C)s2)=O)CC(C)N(C(c2nccn2C)=O)C1 N1(Cc2cc(C(=O)O)c(O)cc2)CCC2(CC1)CC2C(=O)Nc1cn[nH]c1 O=C1CN(CCC(=O)N2CCC2c2ncccn2)CCN1.C12(CCCC1)C(=O)N2 Cc1cccc(Cl)c1CC(=O)Nc1cccc(CNC(=O)C(C)CF)c1 c1(C(=O)NCC2(NC(=O)Cn3cnnc3)CCC2)c(OC(F)(F)F)cccc1Br C(=O)(C(F)C(F)(F)F)N1CCCC(n2cc(CNC(CCCC=C)=O)nn2)C1 c1(C2(C(=O)NCCNC(C3CCC(CN4CCOCC4)O3)=O)C(C)C2)ccccc1 C1(NC(C2CCC(=O)N2)=O)CC2CN(C(=O)CC3CC3(Cl)Cl)CC12 N1(CC)CC(NC(=O)CSc2ccncc2)CC1=O.C1(=O)CCCN1 C1(C(=O)NCCNC(CCN(c2ccncc2)C)=O)COC2(CCC2)CO1 c1(CN2C(C(=O)NC(COc3cccc(OC)c3)=O)CC2)ccc(C)cc1Cl c1(OC)ccc(CC(=O)NC(C2(O)CN(C(C3CC(=C(F)F)C3)=O)C2)C)c(Cl)c1 C1(C(=O)NCC2N(C(c3nccc(C#C)c3)=O)CC(O)C2)CCC2(CCC2)CC1 C1(=O)C(CC2CCC2)N1CC1(CC(C)C)CCC1.C(=O)(CO)N.C(CN(C)C)OC c1(OC(C)C)ccc(Cl)cc1C(=O)NCC1CCN(C(c2cnsc2)=O)C1(C)C n1(C(C)C(N2CCC(C#N)C2)=O)ccc(=NC(=O)c2cc3ccoc3s2)nc1O c1(C(N2CC(C)(NC(Cc3ncc(CC)[nH]3)=O)C2)=O)ccc2ncsc2c1 c1(CC(=O)NCC2(C(C)(C)O)CN(C(C3C(C)OCC3)=O)C2)ccc(N)cc1 c1(CC(C(=O)NCC=CCSC)NC(=O)CNC(=O)C2CC2)ccc(Cl)cc1Cl C1(C(N2CCC(NC(N)=O)C2)=O)CC2(CCN1C(=O)C#CC1CCC1)CC2 C1(N(C(=O)CC2CC2(Cl)Cl)C)CCCN(C(=O)CC2(c3ccccc3)CC2)C1 Cn1cc2c(n1)CCC(C(=O)NCCOCCCNC(c1cncc(Br)c1)=O)C2 N1(C(c2c(C)cccc2F)=O)CCC2(CC1)CC2(C)C(=O)N(CCC#N)C C=CC(C)(O)C(=O)NCC(C)NC(c1ccc(-c2cscn2)nc1)=O c1(NCC(=O)NC2CCN(C(C3(NC(C)=O)CC3)=O)C23CC3)ccccc1[N+](=O)[O-] c1(OC(Cc2c(Br)cc(C)s2)=O)cc(Cl)c(Cl)cc1Cl C1(NC(CCCNC(CC)=O)=O)CC2(C(=O)OC(C)(C)C)CC1C1CC21 N1(C(C(n2cc(CN3CCCN(C)CC3)nn2)C)=O)CC2CC(F)CC2C1 O=C(C1=CC2CCCCCCC12)N1CCOC(c2n[nH]c(C3CC3)n2)C1 C(=O)(C(F)(F)C(F)F)NC1C(NC(C(c2cccc(O)n2)C)=O)CC1 CCC(CC(C)C)C(=O)N1CCC2C(C1)CN2C(c1cncc(C)c1)=O c1(C(C)=O)ccc(C(=O)NC2CCCN(C(C3CC(=O)OC3(C)C)=O)C2)cc1F c1(C(N(CC(C)N(C(CCNC(COC)=O)=O)C)C)=O)nccc(Cl)c1O C1(CNC(COC(CC)C)=O)CCC(CNC(=O)C(c2ccc(Cl)cc2)O)CC1 C1(CNC(C2(CCOC)CCC2)=O)CC2(CC2)CN1C(=O)CCc1cc(C)no1 Cc1nc2c(s1)C(NCC(=O)NCc1cc(Br)c3c(c1)OCO3)CCC2 Cn1ncc(CC(=O)NC2CCC(NC(=O)CCc3nc(=N)[nH][nH]3)CC2)c1C(F)F C(=O)(C(=O)C(C)CC)NCC1CC(Cn2cc(CCSCC)nn2)C1 c1(C(N(CCOC)CCNC(=O)C(O)CC(F)F)=O)cn2ccnc2cn1 CCCC(CC)CC(=O)N(C1CN(C(=O)COC2CCC(F)(F)CC2)C1)C C(=O)(C(F)(CC)C(=O)O)NCC(C)(CC(C)C)n1cc(CN(CC=C)CC)nn1.CC c1(CNC(C2(NC(=O)OC(C)(C)C)CCS(=O)(=O)C2)=O)cc2nn[nH]c2cc1F c1(C(=O)NCC2(CNC(C3CC4(CSC4)C3)=O)CCCC2)cccc2cnnn12 C(CC(C)C)(C(=O)NC1CCCC2CC12)NC(C)=O.c12c[nH]nc1C(=O)N(C)C2 C=C1CC(C(=O)N(C)CCc2ccccn2)(CNC(=O)Cc2ccoc2)C1 C1(NC(=O)CN2CC3CC3C2)C=CCN(C(C2(c3ccccc3)CC2)=O)C1 N1(C(C(CC)n2cccn2)=O)CCC(CN(C)C(C2CCC23CCC3)=O)CC1 C1(CNC(C(Cc2ccoc2)NC(C(C)c2cc[nH]n2)=O)=O)CCCOC1(C)C c1(C(=O)NC(CNC(CC2CC(OC)C2)=O)C)ccc(CO)cc1 C1(C(N(CCCC(F)(F)F)C)=O)CC(C)(C)CCN1C(=O)CCCCCF C1(C(C(=O)NCCOCCC(=O)NCC(C)(C)OC2CCC2)O)CC(F)(F)C1 C1(CCNC(C=CCC)=O)CN(C(c2cc(N)ccc2Cl)=O)CCS1(=O)=O c1(C(=O)NC(C)C)ccc(CNC(c2cnc(CN)o2)=O)cn1 Cc1cc(=NC(C)c2nncs2)[nH]c(=NCc2cnc(C(F)(F)F)s2)[nH]1 CC1CCC(CNC(c2ncoc2CNC(=O)CC2COCC(C)O2)=O)CC1 c1(OC)ccc(OC)c(C(N2CC3(CC3)CC2CNC(c2c[nH]c(C)c2)=O)=O)c1 Cc1cc(F)cc(C(N2CCC(CNC(=O)CCCc3nccs3)C2)=O)c1C N1(CCCC(C)=O)CCC(CCSc2nncn2C)CC1 S(=O)(=O)(c1ccc(F)cc1)N1C(C(=O)Nc2c(OC)cccc2)CCCC1 c1(CCC(=O)NCC2C=CCN2C(C2CCC(=O)N2)=O)ccc(F)cc1Br C(=O)(C1=C(c2ccccc2)CCCC1)NCCNC(c1csc(C)c1C1CC1)=O c1(C(N(CC(CC)NC(=O)C(F)F)CC)=O)coc2c(C)cccc12 C1(F)(C(=O)NCC(C)CN(C(=O)C(C)OCC2CCCO2)C)CC2(CCC2)C1 CC1CCn2ncc(C(=O)NC(C)CNC(=O)C(F)C(F)(F)F)c2C1 c1(CNC(=O)Nc2c(C(=O)OC)nc(-n3cccc3)s2)ccc(O)c([N+](=O)[O-])c1 c1(C(=O)NCC2CN(C(C3C(OCC)C3C)=O)C2)ccc2[nH]ccc2c1F N1(C(c2cc(-n3ccnc3)no2)=O)CCOCC1c1cn(CC2CCCO2)nn1 N1(C(C(C)C(C)O)=O)CCC(F)(F)C(CNC(C2(C#N)CC=CC2)=O)C1 CCC(CC)(CCNC(=O)CC(C)(O)C1CC1)NC(C1CC1(Cl)Cl)=O c1(C(=O)NC2C(C)CN(C(c3ccc(Cl)c(F)c3)=O)C2)ccc2c(c1)NC(=O)C2 c1(NC2(CNC(CNc3c(C)cccc3C)=O)CCC2)ccc(Cl)c(C#N)n1 S(=O)(=O)(CCC(=O)NCC1C(C)CCCN1C(=O)CC1CCC(=O)NC1)NC Cc1ncc2n1CC(C(N1CCCCC1CN(C)C(c1cnco1)=O)=O)CC2 C(c1ccc(C)nc1)=CC(=O)OC(COC)CC(C)C Cc1cc(C(=O)NC2C3CC4C(C3)C24CNC(=O)C(O)CC(C)C)cnc1O c1(CC)c[nH]cc1C(N1CC(N(C)C(c2cc(C(C)C)[nH]n2)=O)C1)=O N1(C(CN(CCC)C)=O)CCN(C(c2c[nH]c(C#N)c2)=O)CC1c1ccccn1 C1(C#N)(C(=O)NCC(=O)NC(C(C)SC)C)CCOC1 CC(C)C(C)CC(=O)NCc1ccc(C(=O)NC2CC(=O)N(C3CC3)C2)cc1 N1(C(C)C(=O)Nc2ccccc2)CC(COC(c2cnccn2)=O)OCC1=O c1(CC)cnccc1C(=O)N(CCCCN(C)C(C1CCC2CC12)=O)C N1(C(CC#N)=O)CCC2CCCN(C(N3CC(CC4CCOCC4)C3)=O)C2C1 c1(CN2CCC(CNC(c3nn(C)c(O)c3)=O)C2)ccc(F)c(S(C)(=O)=O)c1 C1(C(=O)NCCc2cn(-c3c(C)cc(I)cc3)nn2)Cc2ccc(F)cc2C1 c1(CC(N2CC(NC(C3C(C)(C(F)F)C3)=O)C2)=O)cc(C(F)(F)F)co1 C(C(C(=O)N(CC(=O)NCC(C)(O)CO)CC(C)C)NC(N)=O)OC c1(CC(=O)NC2CCC(CN=c3cnc(F)c[nH]3)C2)cn2c(n1)CCCC2 C12(C(N3CCC(NC(C(CCC)CC)=O)C(O)C3)=O)CCCN(CCC1)C2 C1(C(=O)NC(C(N2CC(COC)C2)=O)C2CCCO2)CC(C)(C)CCO1 c1(SC)ccncc1-c1nc(C)nn1CC(C)(C)O.SCO c1(C(N(C2CCCN(C(=O)C(C)(C)C3CCCO3)C2)CC)=O)cn(C)nc1O c1(NC(C2(C)CCN2C(=O)CSc2ccccc2)=O)cccc2c1OCC2 C(=O)(C1=CCC(N(C(C23C(=O)C4CC2C3C4)=O)CCO)C1)C(c1ccc(F)nc1)=O c1(NC)ncc(Br)nc1NC(=O)NCc1ccc(OC2CCCCC2)nc1 S(=O)(=O)(c1ccc(NC(c2ccccc2Br)C2CC2)c(F)c1)NC(C1CC(C(N)=O)C1)=O C1(C(=O)NC(C(C)NC(c2ccc(CC)o2)=O)C(C)C)C2CCC(F)(F)C12 N1(C(c2cnccn2)=O)CCN(C(C2CC2)=O)CC1.C12(CCCC1)CCCN2CC Cc1cccc(F)c1C(=O)NCC1CC(C)N(C(=O)Cn2ccnn2)C1 CCCS(=O)(=O)NC(C)C(=O)NCCC1(OC)CN(C(C2(O)CCSC2)=O)C1 N(C(=NCCc1nccc(C(F)(F)F)n1)NCC(C)(C)C)CC(COC)C C(=O)(C1=NOC(CNC(=O)Cc2ccc(O)nc2)C1)N1CC(OC(C)=O)C1 c1(CN2CCC(CNC(c3cnc4n3CCS4)=O)C2)cc(O)nc(C2CC2)n1 C1(C(=O)NCCCCc2cn(-c3cccc(C)c3N)nn2)CN(C)C(=O)CCO1 C1(C)(C(N(C)Cc2ccc(C)nc2)=O)CCCN(C(=O)C(=O)O)C1.N12CCCC1C2 c1(-c2nnc(C(N3CCC(CCC(=O)OC)CC3)=O)s2)cc(CO)ccc1OC c1(C(=O)NCCCN(CCCCl)C(=O)O)cccc(OCC)c1.c1(CC)ccccc1 C(=O)(C(CC(C)C)N(C(C1CC(OC(F)(F)F)C1)=O)C1CC1)NCCOC C(=O)(C(C)(C)C(O)C(C)C)NCC1C(NC(Cn2nc(C)c(Cl)c2C)=O)CC1 Cc1cc(C(=O)NC(C2CCOC2)CNC(c2ccnnc2O)=O)cc(C)c1F N1(C(C(C)=CC)=O)CC(C)(NC(=O)C(C)Cc2ccccn2)C1 c1(C(=O)OCC)ccc(Oc2ccccc2Sc2n[nH]c(C)n2)nn1 c1(C(=O)OC)ccc(N(C)C)nc1.C1C(C)CN1.C1(=O)C(C2CC2)O1 [N-]=[N+]=NCCCCNC(c1csc(CNC(=O)C(O)C2CC2)c1)=O N1(C(c2ccn(CC)c2C)=O)CCCC(C2CC2NC(C2(C)CC2)=O)C1 c1(N2CC(F)CC(NC(C3CCS(=O)(=O)N3)=O)C2)nc(Cl)nc2ccccc12 C1(C(=O)OC)CCC2(CCOCC2)N(Cc2cccc(OC(F)(F)F)c2O)C1 c1(OC)nccc(C(=O)NCC2CN(C(c3c[nH]c(-c4ccccc4)c3)=O)C2)n1 N1(C(CCC(C)N)=O)CC2OCCN(C(c3ccco3)=O)C2C1 N1(c2ncc(C#N)cc2Cl)CC2CCCC(NC(=O)C(N)=O)C2C1 CC1(C(=O)NCCCCNC(c2nnsc2C(F)F)=O)CCCCC1(F)F C1(CNC(c2c(F)ccc(C)c2)=O)CN(C(C23CC(C2)C3)=O)C2(CCC2)C1 C12(C(N3CC(NC(C(C)c4cc[nH]n4)=O)C3)=O)CC1COC21CCC1 c1(OC)csc(C(=O)NCC2CN(C(c3cc[nH]c3)=O)C2)c1OC C1(NC(c2c(OC)n[nH]c2)=O)CN(C(c2ncoc2C)=O)C(C)(C)C1 N1(CCC)CCCCC1C(=O)NCCCC(C)NC(C1(c2ccno2)CC1)=O n1(CCCCC#C)c(N2CCC(c3ccnc(O)c3)CC2)nnc1-c1cnccn1 N1(C(CC(C)n2ccnc2)=O)CCC(C)(CCNC(C2(CF)COC2)=O)C1 c1(C(N(C2CCCN(C(C3C(C)C3C)=O)C2)CC)=O)ccncc1Br c1(C(=O)NC2CCC(CCNC(c3cc(Cl)cs3)=O)C2)cc(F)c(O)c(F)c1 CC1CN(C(C2(NC(=O)C=CC3CCCC3)CCN(C)C2)=O)CC2(CCC2)O1 C(=O)(C(C)(C)C(=O)OC)NCCC(C)NC(CCCC=C)=O c1(C(N(C(C)CNC(=O)C(F)(F)C2CCCCC2)C)=O)ccc2c(c1)OCO2 S(=O)(=O)(c1ccccc1C1(C)N=N1)NCC=CC(=O)NC c1(C(=O)NCC2CN(C(c3ccnc(CC4CC4)c3)=O)C2)cncc2[nH]ccc12 C1(OCCNC(=O)Cc2cscn2)CCN(C(c2cnc(-c3ccsc3)s2)=O)C1 CC1(C)CN(C(=O)C2=CCSC2)CCC1NC(=O)CC1SC(=N)NC1=O C1(C(N(CCNC(C2(CC)CNC(=O)C2)=O)C(C)C)=O)CC2(C1)CC(C)(C)C2 CCCC(CC)CCC(=O)NCCC1(C(=O)N(C)CCc2ncon2)CC1 CC(C)C(F)(CNC(C1CCC(C)C1)=O)C(=O)O N1(C(C2OCCC(=O)C2)=O)CC(F)C(F)(F)C1.C12C(C1(F)F)n1cc2nn1 C1(NC(CNC(C)=O)=O)CCCCC1.C1(CC(=O)NC(CCOC)CO)CCCC1 C(=O)(C1=CCCCC1C)N(C1(CC(=O)NCC(CC2CC2)OC)CC1)C CC(C)C(C#N)C(=O)NC(CC(=O)N1CC=C(Cl)C1)C(C)C c1(C(=O)NCC(C)CNC(c2coc(C3CCC3)n2)=O)ncccc1Cl CC1(CNC(c2cc(C3CCC3)on2)=O)CCCN1C(c1sccc1Cl)=O N1(C(CCOC)=O)CCCC1C(=O)NCc1cnn(CCF)c1 c1(C(CNC(N(C)Cc2ccn(C)c2)=O)(F)F)cccc(Cl)c1 N1(C(C2CCN(C(CC)=O)C2)=O)CCC(O)(CNC(c2nc(C)sc2C)=O)CC1 c1(C(=O)Nc2c(C)n(C(C)(C)C)nc2)ccc(Br)cc1O c1(C(N2CCCC(NC(Cc3nc(C)sc3)=O)C2)=O)cc(C)nc2c1cnn2C CC1C(NC(CCC(=O)NC)=O)CCN1C(=O)CN(c1ccc(Cl)cn1)C C1(O)(CNC(C2CCC(F)(F)C2)=O)CCCN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CC1 c1(OC)cnc(C(=O)NCCC2(O)CCN(C(C3CC3F)=O)C2)nc1 c1(C(=O)NCCN(C2CC2)CC2(C(C)OC)CC2)csc(CC(F)(F)F)n1 C(=O)(C1=NOC2(CCOC2)C1)N(CCCNC(C1(C)C(C)(C)C1(C)C)=O)CCO c1(-c2cc(CC(=O)NCCC(F)(F)F)ncc2)cccc(Cl)c1O n1(CC)c(C(=O)NCc2csc(C(N3CCCC3CF)=O)c2)cnc1O c1(C(=O)NCC(CN(C(C(c2cnccn2)C)=O)C)O)cc(-c2ccco2)on1 c1(SC)cc(C(N2CCC(NC(=O)CC(C)c3ccco3)C2)=O)cc(Cl)c1 Cc1nsc2ncc(C(=O)NC(C)(C)CN(C)C(C3(C)CCCC3O)=O)cc12 c1(CCC(=O)N(CC2(CCNC(C(C=CC)O)=O)CC2)CC)ccc(=N)[nH]c1 Cc1cc(C(=O)N(C2CCCC2)CCNC(C2C3CCC23)=O)ccc1F Cc1ccc(CC(N2CCC(C)CC2CNC(=O)CC2COCCO2)=O)cc1C C(C(C)(C)CCO)NC(c1cccc(Cl)c1)c1n(CCC(=O)OCC)nnn1 N1(C(C(C)NC=O)=O)CC2(CCN2C(=O)C(C)Sc2ncccn2)C1 N1(C(C2N(C(C(CC=C)C)=O)CCC=C2)=O)CC2(CCOC2)C1 C(=O)(C1=C(C)CCOC1)NC(CCNC(C1CC(C)=C(C)CC1)=O)(C)C N1(C(c2cnc(C)[nH]2)=O)CCC(O)C(C(=O)NC(c2ccccc2C)C)C1 N1(C(CCc2n(C)ccn2)=O)CCC(C(=O)NCCCC(F)(F)F)(CO)C1 c1(C(C)=O)cc(NC(C2CC3CC3N2Cc2cn(C)cn2)=O)ccc1F c1(NC(C2CC(NC(C3C(OC)C3)=O)C2)=O)cc(Cl)nc2ccccc12 CCC(C)(O)C(=O)N(C)CC1CCN(C(C23COCC2C3)=O)CC1 C#CCC(C)(C(=O)N1CC(N2CC(F)C2)C1)NC(=O)C(C)S(C)(=O)=O N1(C(C(C)c2ccco2)=O)CCC(NC(=O)CC2(N(C)C)CCCC2)C(F)C1 C(c1c(C)cc(C)cc1C)=CC(=O)NCC1CN(C(CC(C)SC)=O)C1 c1(C(=O)NC(CN(C(=O)CC2CC(C)(C)CO2)CC)C)ccc(OC2CC2)cc1 c1(NC(=O)NCCNC(C2C(NC(c3ccccc3)=O)C2)=O)ccccc1 c1(C(=O)NCC2C(NC(c3cc(OC)n[nH]3)=O)C2)cc(F)cc([N+](=O)[O-])c1 CCCC(CCC)=CC(=O)NC1(C(=O)Nc2cnc(N(C)C)nc2)CC1(C)C N1(C(C=CSC)=O)CCN(C(=O)CC(O)C(C)C)C2(CCC2)C1 Cc1nc(C(=O)C(=O)NC2CCC2NC(c2ccsc2Cl)=O)cs1 C1(C(N(CC(CNC(C(C)OCC)=O)C)C)=O)Cc2cc(C)ccc2S1 C(=O)(CC(O)CN(C)C)NCCCN(CCCNC(C1CC(C)(CC)C1)=O)C Cc1cc(CCC(=O)NC(C)CCNC(=O)CCc2ncc(F)cn2)cc(C)n1 CC1=CC(C)CN(N2CCCN(c3ccc(C)c(C)c3)CC2)C1 CCCCCC(O)CC(=O)NC1CCCCC1NC(c1cn(C)c(C)cc1=O)=O Cc1cccc(C(=O)NCCCC=CC(N2CCCCC2C2(O)CC2)=O)c1 C(=O)(C1CCCc2nc[nH]c21)N(C1CCCC1)CCNC(c1ccc(Cl)cn1)=O C1(NC(C(C2CC2)OC)=O)Cc2ccccc2C1N=c1[nH]nc(C)s1 C1(CC(=O)OCC)CCN(S(=O)(=O)NC2CCC3CCCCC3C2)C1 c1(NC(CCCOCC=C)c2nnnn2CCCC2CC2)ccccc1O C(=O)(CCCCCNC(=O)CSC)NC1(CC=C)CC=CC1 N1(C(C(CC=CCSCC)NC(=O)OC(C)(C)C)=O)CCCN(C=O)CC1.CC=C C(C)(CC1CCC1)(C(=O)NCC1(CNC(=O)CCCCO)CC1)OC C#Cc1ccc(N(C)C)cc1NC1(c2nnnn2C)COCC1COC c1(C(=O)NCC(CNC(C(C)(C)OCC)=O)(C)O)cnn(CCC(C)C)c1C c1(C2(COC(C3CCCC(=O)N3)=O)CC2)ccc2c(c1)OCO2 c1(OC)cc(C(=O)NCC(O)CNC(=O)C(C)(C)C(C)C)cc(OC)n1 c1(C(=O)NCC2OCCC(NC(c3ccc(C)o3)=O)C2)cc(S(N)(=O)=O)co1 c1(COC)cc(NC(=O)NC2CCN(C(=O)OC)CC2)c2c(c1)OCO2 Cc1c(CCC(N2CC(NC(c3ccnc(O)c3)=O)CC2CO)=O)cnn1C c1(C(=O)NC(c2ccccc2)CC2CC2)cccc2ccc(C(=O)O)nc12 C1(C(=O)NC(CNC(C=C2CCN(C)CC2)=O)(C)CO)CCS(=O)(=O)C12CCC2 CC1=CCC(CNC(=O)CCC2CCN(Cc3cnc(Br)s3)C2)CC1 c1(OCCOC(C)C)ccc(S(=O)(=O)N2CC3CC(CCCC3)C2)cc1 C1(C)(NC(C2C(C)(C)C2)=O)CCN(C(C2(F)CC=CC2)=O)CC1 C(CCF)(C(=O)NOCC(C)C)NC(C(CC)(C)N(C)C)=O c1(C(N(C2CCN(C(C(C(C)(C)C)N(C)C)=O)C2)CCO)=O)cc(Cl)c(F)cc1F C(=O)(C1=CC2CCCCCC12)NCC1N(C(Cc2cncc(C)n2)=O)CC(C)(C)C1 C1(C(N2CC3C(CNC(CCn4ncc(C)c4)=O)(C3)C2)=O)CC12CCSCC2 c1(C(=O)NC(CC(C)C)(C)CNC(C2CCCC2)=O)cccc2cc(O)ncc12 c1(OC(c2nnnn2C2CC2)C(C)OC)ccc(F)cc1.C(C1CC1)N c1(OC)ncnc2c1ncn2CC1CCCC2(CCC2)O1.C12(C)CCCN1C2 C1(C(=O)NCC(C)N(C(=O)Cc2cc(C(F)(F)F)n[nH]2)C)CCCC12OCCO2 c1(C(N(C2CCN(Cc3sccc3Cl)C2)C)=O)cccc(NS(C)(=O)=O)c1 C(C(C)(C)C(=O)NC(C1CCOC1)CNC(=O)CCc1cccc(Cl)c1)OC c1(C(C(=O)NC2C(C)C2C)NC(C(COCC)C)=O)cnc(OC)cc1C c1(C(C(=O)NC2COC2)N(C(C(=O)OC)C)C)ccoc1C C1(C(c2ccc(C(C)=O)cc2)=O)CC2CCC(C1C)N2 N1(C(C(N2CCC(O)CC2)C)=O)CC2(CCCC2NC(=O)CCC(C)(C)C)C1 Cc1cn2cc(NC(C3CCN3C(=O)C(C)n3cnnn3)=O)ccc2n1 c1(N2CC(C)OC(C3CC3)C2)nccc(=NCc2cnc(O)c(F)c2)[nH]1 C(CCCCNc1cn(C(C)CO)nn1)N(C(=O)CCc1ccc[nH]1)C(C)=O CC1(C)CN(C(=O)Cn2[nH]cnc2=N)CCC1NC(c1[nH]nc2ncccc12)=O c1(C(=O)NC2CC(NC(Cc3nc(C)[nH]n3)=O)C(O)C2)ccc(N)c(F)c1 Cc1cnc2nccc(C(N3CC4CC4(CNC(=O)C(O)C(C)C)C3)=O)c2c1 n1(CC#C)cccc1C(=O)NCC(C)CN(C(=O)C(CC1CCCCC1)OC)C CCC(Cc1ccccc1C)C(=O)N(C1CC(NC(=O)C=Cc2ccoc2)C1)C C1(CCCC#C)CCCN1C(C1CC(F)(C(=O)OC)C1)=O C=CC1CCN(C(C2CN(C(=O)CCCCSC)CC2CCC)=O)C1 C1(C)(NC(C(CCC)C)=O)CCCN(C(C2CCN(C(=O)C3CC3)CC2)=O)C1 C1(CNC(C2C(C)CC2)=O)CC2(CO1)CN(C(C1(c3ncco3)CCC1)=O)C2 CCC(C)C(=O)ONC(=O)N(C(COC)COC)CCOCc1ccccc1 c1(SCC)cccnc1C(=O)N(C1CN(C(=O)COCC2CCCCO2)C1)C C12(CNC(c3cc(CC)c(CC)o3)=O)CCC(C1)N(C(=O)CC(C)(C)OC)C2 C1(C(=O)NCCOCCNC(=O)CCc2c(Cl)cncc2Cl)CC2C(C1)C2(F)F CC(C(F)(F)F)N(C(=O)C(F)CC1CN(C(C2COC(=O)N2)=O)C1)C1CC1 CCCC(CCC)CC(=O)NC(C)(C)C(C)NC(=O)C(C)(C)COCC N1(C(C2(CCOC)CCC2)=O)CCC2(CCCN2C(=O)COc2cnccn2)C1 Cc1c(C(=O)NCC(F)CNC(c2cc(C(N)=O)[nH]n2)=O)nnn1C1CCOC1 C1(C(=O)NC(C(C)C)(C)C)CCN(C(C2OCCCC2(C)C)=O)CCO1 c1(C(=O)OC)ncccc1NC(c1cncc(NCC2CNC(=O)C2)c1)=O N1(C(CCC)=O)Cc2ccccc2CC1CNC(c1nnn(C)c1C(F)(F)F)=O c1(C(C)=O)cc(CN2CCC(C)C2)n(C)c1.c1(C(CN)O)cccc(Cl)c1 N1(C(CCSCCCC)=O)CCC2CCN(C(=O)C(CC)NC(C)=O)C2C1 N1(C(c2ccn(C(C)C)n2)=O)CCCC(C)(CNC(=O)C(C)(C)CF)C1 CCCCC(C)(F)C(=O)N1Cc2[nH]nc(C(=O)NCC3(O)CC3)c2C1 N1(C(CCC(C)(C)C)=O)CCC(NC(c2nc(C(C)(F)F)cs2)=O)C(C)(C)C1 C1(COC)(NC(C2CC3CC3C2)=O)CCCN(C(c2csnc2C)=O)C1 CC1CCSC1C(=O)N(C(C)CNC(c1csc(NC(=O)NC2CC2)n1)=O)C C(=O)(CC(C(F)F)NC(=O)CC1CC2(CC2)C1)NCCCC(=C)Cl C=CCC(C)(C)C(=O)N1CCC(N(C(=O)C(C)OCCCCCC)C)C1 N1(C(C(CC)SC)=O)CC(NC(c2ncc(C)cc2C)=O)C(S(C)(=O)=O)C1 c1(CNC(C2CC(Nc3cc(-c4nn[nH]n4)ccn3)C2)=O)cccc(O)c1 C1(CC)(OC)CCN(C(C2C(C(=O)NC3(C(=O)OC)CCC3)COC2)=O)C1 Cc1ccc(C(=O)NC23CC(C2)N(C(=O)C(C)NC(=O)CC(F)(F)F)C3)c(F)c1 c1(C(=O)NC(CCCNC(C2CCC(C)C2)=O)(C)C)cc2ncccc2[nH]1 C(CC(=O)NC(c1ccoc1)C)(CC(C)C)NC(C1(CC=C)CC1)=O c1(C(=O)OCc2cccc3c2CCCC3)ccc(Cl)c2ccncc12 C1(C(=O)Nc2c(CCC(=O)OCC)nn[nH]2)CCCCC1CF.C1(C(=O)N)CC1C C1(NC(C(COC(C)C)NC(C)=O)=O)CN(C(=O)C(F)(F)CO)CC1C Cc1ncc(NC(C2CCN(C(=O)Cc3ccccn3)C2(C)C)=O)c(C)n1 CN=c1[nH]c(C(=O)NC(C)C(C)(C)NC(c2csc(-c3cnc[nH]3)n2)=O)cs1 c1(CC)ncc(NC(N(C)CCC2CC2)=O)o1 N1(C(c2nc(CC)sc2)=O)CCCN(C(=O)CCCC(C)(F)F)CC1C N1(CC)CCN(C(=O)C=CCN(CC(F)(F)F)C)CC1C.N12CCCC(C1)C(=O)N2 CCCCCCC(C)C(=O)N(CCC(=O)NC(c1ccccc1)CF)C(C)C C1(NC(=O)NC2C(C(C)C)(CC)C2)CCC(=C(F)F)CC1 c1(CC(Cn2cc(C3(C(=O)OC)CCOC3)nn2)O)ccc(Cl)cc1 CN1CC=C(CC(=O)N2CC3CCC(CNC(=O)CNC4CCCC4)(C3)C2)CC1 c1(CC(N)=O)ccc(C(=O)NCC(O)CCNC(=O)CSc2ccccc2)cc1 C(=O)(C(C(C)(C)C)OC(C)(C)C)NC1CN(CC(=O)NCC(C)C)CC1C C(=O)(C1=CCC(C)(C)CC1)N1CC(C(C(=O)NCC(C)(C)N(C)C)OC)C1 c1(C(=O)NCCN(C(c2c(C)oc(Cl)n2)=O)C)ccccc1[N+](=O)[O-] N1(C(COCC(=C)C)=O)CC(CCNC(=O)CCCC2CCC2)OC(C)C1 c1(CC(=O)NC2CN(C(c3c(C(C)C)cccc3)=O)C2)cc2c(cc1Br)OCO2 n1(CC)ccc2cc(C(=O)N(CC(C)CNC(=O)C(F)C3CCC3)C)ccc12 N1(C(CSCc2ccc(C(=O)OCC)cc2)CC)C(=O)c2ccccc2C1=O C1(C(=O)NCC(C2CCN(C(=O)COC(F)(F)F)C2)(C)O)CC2(CCC2)C1 c1(C(N(CCOC)CCNC(C2C3CCC2CC3)=O)=O)cccc(C)c1Br N1(C(CN(C)C(=O)C2CC2)=O)CCC2(C1)CN(C(C1CCCC3CC13)=O)C2 c1(C(c2nnnn2C)NC(c2c(C)nn(C)c2C)C)ccc(C#N)c(Cl)c1 c1(OC)ccccc1C(C)C(=O)NCc1ccc(C(C)(C)C)nc1 N1(S(CC2C(C)CC2)(=O)=O)CCCCC1c1ccc(F)cc1 N1(C(CNS(CCOCC)(=O)=O)=O)CCN(C(=O)C(C2CCC2)OC)CC1CC C1(C)(C(=O)NCC(C)N(C(C2CCN(CC)C2)=O)C)CCNC1=O C12(C(=O)NCC3(O)CC(CNC(C4CS(=O)(=O)C4)=O)C3)CCC(CC1)CO2 C(=O)(C(CC(C)C)C(N)=O)NC1C(CNC(c2cc(C)c(O)nn2)=O)CC1 CC1CC(C(=O)N(C2CCC2C)C)CCN1C(C1CC2(C1)CC(O)C2)=O c1(C(N2CC3C(CNC(CN4CC(=O)NC4=O)=O)C3C2)=O)c[nH]cc(F)c1=O CC1(C)CC(O)(CC(N2CCC(O)(CNC(C3CCC=CO3)=O)C2)=O)CO1 N1(C(CSCCOC)=O)CC2CCN(C(C3CC(=O)N(CC(F)(F)F)C3)=O)C2C1 Cc1cc(C(=O)NCC2CCN(C(C3CC(F)(F)C3)=O)CC2C)ccc1Cl c1(C(=O)NCC(CC=C)NC(c2cccc(C(C)C)n2)=O)c(C)ccc(C)c1O N1(C(c2c(C)oc(C#N)c2)=O)CC2CN(C(=O)C=Cc3cncc(F)c3)CC2C1 C(=O)(C=CS(F)(F)(F)(F)F)N1CC2C(NC(=O)Cn3cc(CN4CCC4)nn3)(C2)C1 N1(C(C(CC=C)(C)C)=O)CCC2(CCCC2NC(=O)CCNC(=O)NC)CC1 Brc1ccccc1C1(NCc2noc(Cc3ccco3)n2)CC1 C1(C(N2CC(CC)OCC2)=O)CCN(C(=O)CC2CNC(=O)O2)O1 c1(C(=O)NCC2N(C(CSC)=O)CC=C2)ccc(OC(F)(F)F)cc1Br C1(NC(CC2(OCC)CCC2)=O)CCN(C(=O)C(C)OC)CC1F N1(C(C(CC=C)C)=O)C2CCC1CC(c1cn(-c3cncc(F)c3)nn1)C2 n1(CC(C)NC(c2cn[nH]c2)=O)cc(CNC(C2(O)CCSC2)=O)nn1 N1(C(CCSCC)=O)CCOC2(C1)CN(S(=O)(=O)c1cccc(C(F)(F)F)c1)C2 C(N=c1ccc2c([nH]1)CCCC2)C1(C)CCC(NC(=O)C=C(Cl)Cl)CC1 N1(Cc2cn(C)nn2)CC2C3CCC(C2C1)N(C(c1ccc2nonc2c1)=O)C3 CC(CNC(=O)CCc1cnn[nH]1)C(=O)NCc1nc(C2CC2)n[nH]1 C1(NC(C2(n3cnnn3)CC2)=O)CN(C(c2cnsc2)=O)CC1C1CC1 c1(CCC(=O)N(CCNC(C2CCCCN2C)=O)CC)cccc(F)c1Cl N1(C(COC)=O)CC2(CC(C(=O)NCC3(C)COCCO3)C2)C1 C1(NC(CC2CN(C)C2)=O)CN(C(C2(C)CNC(=O)C2)=O)CC1C(F)(F)F CC1CCCCCC1SCc1cc(Cl)cc(Br)c1.c1ccc(Br)cc1 Cc1ccc(F)c(N)c1C(N1CCN(CCNC(C2CCCSC2C)=O)CC1)=O N#Cc1ccc(C(=O)NCC2(F)CCN(C(c3ccc(Cl)cn3)=O)CC2)cc1Cl CCC(CCC(=O)Nc1cnccc1CO)NC(=O)C=Cc1cc[nH]n1 N1(C(C2(C(F)F)CC(=C)C2)=O)CCC(CN(C)C(c2c(Cl)n[nH]c2C)=O)CC1 C(=O)(C(C#N)C(C)(C)C)NCC1(c2cn(CCC(=O)OC)nn2)CCCC1 c1(OC)ccc(N=c2scc(CC3CCCO3)n2-c2ccc(SC)nc2)c(F)c1 C(=O)(C(F)(F)CCSC)N(C(CNC(CCCCOCCC=C)=O)C1CC1)C C=CC(C)(O)C(=O)NCC1CC(F)CN1C(=O)C(C)OC(C)=O c1(C(=O)NC2CC(C)CN(C(c3cncn3C)=O)C2)cc([N+](=O)[O-])cnc1O C1(CC(C(=O)NCCCF)N(CC(CC)CC)C)CCC(F)(F)CC1 C1(O)(C(=O)NC(C2CCCN(C(c3c(C)n(C)cn3)=O)C2)C)CCOC1(C)C C1(C(=O)NC(C#C)C)C=CCN1C(=O)C(n1ccnc1C)C c1(C(=O)NCC(CO)NC(=O)CC2CC(CF)C2)ccc2cccnc2n1 C(=O)(C#CCNC(=O)C(=O)C1CCCC1)NC(C#C)(C)C1CCCC1 c1(C(C)(F)F)ccc(NC(=O)NCC2CCCN2CCCc2ccccc2)cc1 C1(NC(C(C)NC(C)=O)=O)CCN(C(c2ccc3cnsc3c2)=O)CC(C)(C)C1 C1(CC(=O)NC)CN(C(=O)C(c2ccccc2)O)CCN1C(=O)CCC(C)(F)F CC(C)C(CNC(=O)C=Cc1ccccc1)C(=O)N1CC2CC2C2CC12 c1(C(=O)NCC2COCCN2Cc2cnon2)cccn2ncnc12 C(=O)(C1Cc2c(Cl)cccc21)NCC1CC(NC(C(CC(C)C)C(N)=O)=O)C1 N1(C(=O)Cc2ccsn2)CCN(CC2CCCN(C(C3CCS3(=O)=O)=O)C2)CC1 c1(C(N2CC(C(=O)NCCSc3ccc(C)cc3)OCC2)=O)cnc(F)c(C)c1 O(NC(=O)C(C)Cn1cccn1)CC(=O)N(C(CCCC)C)C1CC1 N1(C(CS(CC)=O)=O)CCC2CCN(C(c3ccc(C(F)(F)F)cc3)=O)CC2C1 c1(C(C(=O)NCCCN(C(=O)C(F)(F)C(C)(C)O)C)=O)c[nH]c2ccccc12 CC1(C)CC(=O)OC1CNC(=O)CCC1CC(NC(=O)CC2CC3CC3C2)C1 c1(OC)ccccc1CCNC(c1cncc(-c2ccncc2)c1)=O C1(C(C(=O)NCC2(NC(C3C(CC(C)C)C3)=O)CC2)F)CCOCC1 N1(C(c2n(CCOC)ncc2)=O)CCCN(S(N)(=O)=O)CC1 Nc1sc2c(c1C(=O)NCC1CC1CNC(c1ccc(=O)oc1)=O)CCC2 C=C(C)C(C)(C)C(=O)NCC1CN(C(=O)C(C2CCC2)OCC)CC1C C1(CNC(C2N(C(C)C)CCC2)=O)CC(N=c2[nH]c(Cl)ncc2C(N)=O)C1 C(=O)(C(=O)CCC(C)(C)C)NCCN(C(=O)C=Cc1ccncc1)CC N1(C(c2cccc(C)c2N)=O)CC2CC1CCC2NC(=O)CC(C)C n1(CC)nc(C(=O)NC2(CNC(=O)C(CCc3ccccc3)OCC)CC2)c(C)n1 CCC(CC)C(=O)NC(C)Cn1cc(CNC(C23CC(F)(C2)C3)=O)nn1 c1(C(N2C(C3(O)CN(C(CC=CC)=O)C3)CCC2)=O)cc(C)ccc1C1CC1 N1(C(C(C)n2ccnc2)=O)CC2CCC(NC(c3ncc4ccccn34)=O)C2C1 Cn1ccc2ccc(CNc3ccc(NC(c4c[nH]c(=O)cn4)=O)cc3F)cc12 c1(C(=O)NC23CCC(CC2NC(=O)CC2(O)CCC2)C3)ccc(F)c2c1CCC2 C1(NC(C(CSC)O)=O)C2CN(C(=O)CCOCC(C)C)CC12 C1(O)(C(C)NC(C(C)C)=O)CCN(C(c2cccnc2-c2ccnn2C)=O)C1 C1(C(=O)NCCC2(O)CN(C(C3CCCN3C(C)C)=O)C2)(CC)CCCC1 N1(C(c2sc(CCC)c(CC)c2)=O)CCC2(C1)CN(C(C13CCCCC1C3)=O)C2 Cc1nc(C(N2CC(CCc3cn(C(C)C)nn3)C2)=O)n(C)n1 N1(C(=O)Nc2nc3ccccc3s2)CCC2CCCN(C(c3ccccc3)=O)C2C1 N1(C(CCC2(C)N(C(C(C(C(C)C)O)C)=O)CCC2)=O)CCCC2NC(=O)CC12 C(=O)(CC(C(C)OC)NC(c1ccc(O)cc1F)=O)NC(C=C)C1CCC1 c1(C(N2C(C)CC(CNC(c3occ4c3CCC4)=O)C2)=O)cccc2ncnn12 c1(C(N2CC(C(=O)Nc3c(F)cccc3F)OCC2)=O)ccc2c(c1)C(=O)CC2 N1(C(CCOC)=O)CCN(CC(C)(C)NC(=O)Cc2nnnn2CC(F)F)CC1 CCCC(O)(CCC)CC(=O)NC(C)CCCCNC(c1nn(C)cc1C)=O C1(CC=C)(SC)CN(C(C2(CNC(C3CC3CC(C)(C)C)=O)CCC2)=O)C1 C1(SC)CC(CO)ON=C1NC1CCCCC1C#N C1(NC(Cn2ccc(C)n2)=O)CC2CC(NC(=O)CN3CSCCSC3)C2C1 c1(OCC2(C(=O)NCCn3ccnn3)CC2)ccc(O)cc1 c1(CC(=O)NC23CCC(C(=O)NCC4CCCOC4)(CC2)C3)c(F)cccc1Cl C(=O)(C(F)C(C)CNC(C1(C(C)C)COC1)=O)NC1C(C=C)OCC1 N1(C(C(CCOC)OC)=O)CCCCCC(NC(c2cc(C(F)(F)F)n[nH]2)=O)C1 Cc1noc(C)c1C=CC(=O)NCC(C(C)C(C)C)NC(=O)C=CC1CCCCC1 C(CC(=O)NCC1COC(C)(C)C1)(C(F)(F)F)NC(CC=CC(C)(C)C)=O C1(CC=C)(NC(=O)CSC(F)F)CCCN(C(C2CCCC3(CC3)C2)=O)C1 CC(CN(C)C(C1CC2(CC2)C1)=O)C(=O)NC(C)C(C)(C)O CCS(=O)CC(=O)N(C)CC1CCCN1C(=O)CCOc1cccc(OC)c1 C(=O)(C(=O)NC1CC1)N(CCCN(C)C)CCN(C)Cc1ccco1 N1(C(CC2N(C(C(C)(C)n3cccn3)=O)C3C2CCC3)=O)CC2COC(=O)C2C1 CC1(C)CCN(CC(=O)NC(C)(C)CCCNC(=O)CC2CSCCO2)CC1 Cc1ccc2c(c1)CC(C)N(c1ncnc3cc(-c4ccccc4)ccc13)C2 c1(OC)ccnc(O)c1C(=O)NC1CC2(C1)CN(C(=O)CC1CCC(C3CC3)O1)C2 c1(C(=O)NCC2(CCNC(CCC=CC)=O)CC2)cccn2ncc(Br)c12 n1(CC)nnc(C)c1C(=O)NCC1C(C)CCN1C(c1ccc(C)cn1)=O C(=O)(CC(F)(F)C(C)C)NCCn1cc(CCNC(CCC)=O)nn1 C1(CCC)CCOCC1(c1nnnn1-c1ccccc1)NC1CCC(=O)N(C)C1 N1(C(CCNC(CC(CC)CCCOC)=O)=O)CCC(O)C(C)C1 c1(OC)ccc(C)cc1C(=O)N(C1CCN(C(=O)CCCC2CCCO2)C1)C c1(CNCc2scc(C)n2)ccnc(NCCOC(C)C)c1 C=CCCCCC(=O)NCC(C(C)C)NC(C1CC2(CC(OC)C2)C1)=O C(C)(CCC(=O)N1CC(OC2CCC2)C1)NC(CCOCC(C)(C)C)=O c1(CN(C(CC(C)C)CO)C(C2C3CN(CCO)CC23)=O)ccc2cccnc2c1 C1(C(=O)NC2CN(C)CC2F)(CC)CNCCS1(=O)=S CCC(CC(=O)NCCCCc1ncc[nH]1)NC(C1CCCSC1)=O C(=O)(CC1CC(=O)Nc2ccccc21)N(CCCNC(C1CC=CCC1)=O)CC N1(C(CC(C(CC)C)NC(=O)COC(C)C)=O)CCC2C(=O)NCC2C1 N1(CC(CCCC)C)CC2CCCN(C(=O)Nc3ccccc3)C2C1 C12(C(N(C3CCN(C(C4CC(C)C=C4C)=O)CC3)CC#C)=O)COCC(C1)OC2 C1(C(=O)NC(CCCNC(c2cncc(OC)c2)=O)(C)C)CCCC2(CC2)C1 N1(C(C(n2ccc(C)n2)C)=O)CCC2C(NC(c3cc(C(F)F)ncn3)=O)C12 C=CCC(C(=O)N1CC(CNC(c2scc(C)c2OC)=O)C1)C(C)C c1(CCCC=C)nc(-c2cnn(C)c2)nn1C1CCS(=O)(=O)C1 n1(CCC)nccc1C(N1CCCC1CC(=O)NC1CC(F)C1)=O C1(CNC(C2C=C(C)CS2)=O)CC(C)N(c2nnc(CC(F)(F)F)s2)C1 C(=O)(C(CCC1CCC1)NC(C1CC2(CC2)CO1)=O)NCC1CCC(C)C1 N1(C(C=CC(=O)OCCCC)=O)CCC(CNC(=O)Cc2cnn(C)c2)C1(C)C N1(C(Cn2c(C)ncc2)=O)CCN(C(c2ccnc(C(F)(F)F)c2)=O)C(C#N)C1 N1(C(c2ccc(OC)nn2)=O)CC2CCCC1C2CC(N1CCC(CF)CC1)=O c1(OC)ccc(CN2CC(NC(C3CCCC3OC)=O)C(F)C2)cc1Br Cc1nc2ccnn2c(C)c1C(N1CCN(C(=O)C(F)CC2CCC2)CC1C)=O N1(C(Cc2c(C)nc(C)s2)=O)CCCC(NC(C2COC(C)(C)C2)=O)C1C Cc1cc(Cl)c(C(N2CC=CC2CNC(C2CCC(=O)N2C2CC2)=O)=O)s1 C(=O)(C1=NOC2(CCC2)C1)N1CCC(C=C)(C(N2CCOC3CCCC23)=O)C1 C1(C(=O)NCC(CNC(C(C)C2CCC2)=O)O)CCn2c(O)nnc2C1 C(=O)(C(C)C(C)NC(C1CCCC1)=O)NCCOCCCNC(CC)=O C(CCCC(=O)OCc1csc(Nc2c(C(F)(F)F)coc2C)n1)OC c1(C(N(CC(C)CNC(=O)C(C)(C)C2CCCCO2)C)=O)ccnc2ccsc12 C1(C(N(C2CC(F)(F)C2)C)=O)CCCCN(C(=O)CCc2cnn(C)c2)C1 C1(C(N(CC(COC)C)C)=O)CCN(C(c2cnc(N)cn2)=O)CC1C C1(=O)C(C)(C)CN1.c1(C(C)NC(=O)CN2CC3CC3C2)ccc(CNC(N)=O)cc1 c1(CNC(=O)NC(c2ccc(C)cc2)C(C)(C)C)cn2ccc(Br)cc2n1 N1(C(CC(C(F)(F)F)OC)=O)CC2CC(NC(c3cnsn3)=O)CC(C2)C1 c1(OC)cccc(CCC(=O)NC(CNC(c2ccc(SC)o2)=O)CO)c1F C1(NC(C(NOC)=O)=O)CN(C(=O)C(C)(C)NC(C)=O)CCN1C(=O)C(F)(F)F c1(NCc2n(C(C(=O)OC)C)nnn2)ccc(-c2cnn(C)c2)c(F)c1 c1(OC)ccc(C(C)C(=O)NCC(C2CC2)NC(C2CC2F)=O)c(C)c1 N1(CCC(=O)NC(CC(C)C)CNC(C2(C)CC3CC3C2)=O)CCSC(C)(C)C1 N1(C(C2(C(N(C(C)C)C)=O)CC2)=O)CCN(C(=O)C(F)C2CC2)C(CN(C)C)C1 C1(c2n(CCSC)nnn2)(NC2CC(CC#N)C2)CSC(CC(=O)OC)C1 C(=O)(C#CC1CC1)NCC(CNC(c1oc(Br)cc1C)=O)OC Cc1[nH]nc(C(=O)NC(Cn2ccnn2)C(=O)NCCc2ccccc2O)c1C c1(OCC)cccc(CC(=O)NCCC(C)NC(=O)CCc2ccoc2)n1 c1(C(N2CCC(O)(CN(C)C(C3CC3Cl)=O)CC2)=O)cnc2c(n1)CCCC2 C(=O)(CCCCSC(F)(F)F)N(C1CCN(C(=O)C(C)(F)F)C1)C c1(C(N2CC(NC(Cn3c(C)cc(C)n3)=O)C(F)C2)=O)c(Cl)cccc1Cl Cc1nc(C)c(C(=O)NC2(C(=O)NOCC3CC4CCC3C4)CC(F)(F)C2)s1 N1(C(c2nccc(C)n2)=O)CCCC2(CNC(=O)C3=NNC(=O)CC3)CCCC12 N1(C(C(CCC)(C)C)=O)CC2CCOCC2(NC(c2sccc2OCC)=O)C1 c1(CCC(=O)NCCCCCNC(C=CC(C)C)=O)nc2ccccc2[nH]1 N1(C(CCc2c(C)cc(F)cc2)=O)CCCC2CN(Cc3ccc(F)cc3)CC12 C1(OC)CN(C(=O)C(C)C)CCC1NC(C1(c2cc(C)no2)CCOCC1)=O c1(C(=O)NCC2(C)CCN(C(C3(C)CCC(=O)C3)=O)C2)cc2n(c1)CCCC2 CCC(O)C(C)C(=O)N1CCC(NC(=O)C(C)Oc2ccc(C#N)cc2)C(C)C1 C1(C(N(CCN(C(c2c(C)oc(C)c2C)=O)C)C(C)C)=O)C2CCCCCCC12 N1(C(CCOC)=O)CCC(CO)C(NC(=O)CC2CCSCC2)C1 c1(NCC)cccnc1C(N1CCC(C)(NC(=O)Cc2ccco2)C1)=O Nc1c(C(N2CCN(C(c3cnc(Br)s3)=O)C3CC23)=O)cccc1F C(C(=O)NOCc1cccnc1)(C1CCCC1)NCCSC(CC)C(=O)OC C(CC1(O)C(=O)Nc2ccccc21)NC(=O)NC(c1ccccc1Cl)C c1(C(N(C)CC2C3CN(C(C=C(COC)C)=O)CC32)=O)c(C)[nH]c2ncccc12 C1(CC(=O)N(C2CN(C(=O)Cn3cnnn3)CC2F)C)CC2(CCCC2)CO1 c1(C(N2CC3C(NC(CCCOCC)=O)(CC3)C2)=O)ccc2c(C)noc2n1 c1(C(C(N2CC(CNC(c3c(C)ccnn3)=O)C2)=O)C)c(F)cccc1F Cc1cc(C)c(C(=O)NC(C)CCCNC(c2cccc3c2NCC3)=O)c(C)n1 C(=O)(C(C)(C)CN(C)C)NCC1OCC(CNC(CNS(CC)(=O)=O)=O)C1 C1(C)(C(=O)NCC2(NC(c3ncn(C)n3)=O)CC2)CC2(CC2)C1 C1(Cc2cccs2)CCCCN1C(=O)C(C1CC1)OC.C1(=O)CSCN1CC C(=O)(NNC(=O)OC)C1(C(=O)OC)CC(c2ncc(C(F)(F)F)[nH]2)C1 C1(NC(=O)Cn2cncn2)CCCCCC1NC(c1ccc(OC(F)(F)F)cn1)=O C=CC1(C(=O)NCCc2nc(CC)no2)CCN(C(=O)Cn2nccc2C)C1 C(=O)(C(F)(F)C(F)(F)F)N1CCC(NC(c2c(C(C)C)ncnc2)=O)C(CO)C1 Cn1ccc(=O)c(C(N2CCN(C3CCN(c4nnn(C)n4)C3)CC2)=O)c1 C1(C(N(C(C)C)CCN(c2nnc(C#N)s2)C)=O)CCCC(C)CC1 CCCCCC(C)(C)C(=O)N(C)CCNC(c1c(C)sc(Br)c1C)=O N1(C(C2ON=C(C)C2)=O)C2CCC1CN(C(c1ccnc(N3CCC3)n1)=O)CC2 c1(C(C(=O)NC(CNC(=O)CN2CCOC2=O)C2CC2)OC)ccc(F)cc1F c1(C(N(CCC(C)NC(C2CC3(C2)CC3(F)F)=O)C)=O)ccc2n[nH]cc2c1Cl C(CCCCOC(=O)C(C)NC(=O)CCSC(C)C)OC c1(Nc2ccc(C(=O)NCC(CNC(C=NOC)=O)C)cc2)ccc(C)c(O)n1 c1(COC)nc(NCC=CC2CC2)cc(=NC2CCCc3[nH]ccc32)[nH]1 CN1CCCC1(C)C(N1CCCC(Nc2ccccn2)C1)=O c1(C2C(C(=O)NC(CCN(C(c3c(C)scc3)=O)C)C)C2)ccc(F)cc1 N1(C(CCNC(N)=O)=O)CCOC2CN(C(c3ccc4nc[nH]c4n3)=O)CC12 c1(NC(C2(OCC)CC2)C(=O)C2CC2)cnn(C(=O)NCC2C=CCC2)c1 C1(COc2cccnc2)CCCCC12CC2.C12CCCCN1C(=O)COC(=O)C2 N1(C(C(CCN(C)C)NC(C2CCCC(=O)N2C)=O)=O)CCCC(C2(C)CC2)C1 c1(C2(NC(=O)NC(CS(C)(=O)=O)CC3OCCO3)CC2)cc(Br)ccc1[N+](=O)[O-] C(=O)(CC(C)CC(C)(C)C)NC1CN(C(c2nc(CC)sc2N)=O)CC1O c1(NCCC=CC)ccc(S(=O)(=O)N2CCC(C3CCCCO3)C2)cc1F C1(NC(CCCN(C(=O)OC)C)=O)CCCN(C(=O)CN2CC3CCC2C3)CC1 N1(C(C(C)N(C(c2nccc(C#C)c2)=O)CC)=O)CCc2ncncc2C1 C1(C(=O)NCCC2(NC(=O)CC3C=CCC3)CC2)CCCN(C(=O)C2CC2)C1 C12(OC)CCC(CNC(c3cc(C)c(Br)cc3F)=O)(CC1)CC2 C1(NC(c2c(CCC)n[nH]c2)=O)CC(F)CN(C(c2ccc(C)[nH]2)=O)C1 N1(C(C(C)CC2CCC2)=O)CC(CNC(c2ccccc2CC#N)=O)C(C)(C)C1 CC(C#N)C(=O)NCC(C)(C)CNC(=O)CC1CS(=O)(=O)C1 C1(CNC(CCCOC(C)=O)=O)CN(C(=O)CCCCC(F)F)C2(CCC2)C1 c1(C(N(C(C)C(C)NC(n2cccc2NC)=O)CC)=O)ccnc(CC(C)C)n1 CC1(C(N2CCCCC2c2cccc(Br)c2)=O)CCC(N)CC1 C1(C(N2CCC(OCC#C)C2)=O)CNC(=O)CN1C(=O)C(CC)CC Cc1csc(Cl)c1C(=O)NCC(O)CCNC(=O)C(C)C1CCCC1 c1(Cn2cc(CNC(C3CCn4ccnc4C3)=O)nn2)nc2cc(Br)ccc2s1 N1(C(c2cc(C)nc(O)c2)=O)C2CCC1CC(NC(c1cn(C)nc1O)=O)C2 N1(C(c2c(C)cc(F)s2)=O)CC2CCC(C1)N2C(c1cscc1C#N)=O c1(CC(=O)NCC(C)NC(CC(F)(F)F)=O)ccc(-n2ccnc2)cc1 CCC(CNC(c1cnc(CC(C)C)s1)=O)(CC)NC(=O)C(C)SC(F)(F)F C1(C(N(CC(C)CNC(=O)CN(CC(C)(C)C)C)C)=O)CCS(=O)(=O)C(C)C1 Cc1cnc(C(=O)NC(C(=O)Nc2cc(Cl)ccc2C)C2CCC2)c(F)c1 c1(C=O)ccc2sccc2c1.N12CC(CC(C)(C)C1)C(=O)N(C)CC1(CC1)N2C C1(O)(c2cn(CCC)nn2)CCN(C(=O)NC(c2c(Cl)cccc2Cl)C)CC1 N1(C(C2N(CC)CC2)=O)CCCC2(CC(NC(C3CCC(=C4CC4)CC3)=O)C2)C1 C1(NC(C(C2CCN(C(c3c(CC)nns3)=O)CC2)C)=O)CC2(C1)CN(C)C2 Cc1oc2ccccc2c1Cc1ncnn1C.N1C(=NCC(C)C)NN(C)C(=O)C1 CCS(=O)CC(=O)N1CC(COC)(NC(=O)Cc2cccc(Br)c2)C1 C(=O)(C1=CCN(C(C2COCCN2C)=O)C1)NCCC(C)N(C)C C(=O)(C(CC1CCCC1)CC)N1C(CNC(C(C=C)O)=O)CC1 N1C(NC2CCCC2)=NCCC2(CC2)C1.N1(C2C(C(N)=O)C2)CCOCC1 N1(C(c2c(C)nn(C)c2)=O)CCCC(C2CN(C(c3cc(C(C)C)on3)=O)C2)C1 c1(C(N(CCOCCNC(CC(CC)(C)C)=O)C)=O)cc2ccncc2s1 Cc1nc(CC(=O)NC2(C)CC(NC(C34CC(C)(C3)C4)=O)C2)n[nH]1 C1(NC(c2c(CC)cno2)=O)CCCN(C(C2CCC(=O)NC2)=O)CCC1 C1(NS(CC)(=O)=O)CCOC12CCCCC2.c12cn(nn1)C(C)C(=O)N2 c1(C(=O)NC2CCCC(NC(C3(CO)CCC3)=O)C2)coc(=O)c2ccccc12 CC1(C)C2CCC1(C(N1CCC3C(NC(=O)CC4(O)CCOC4)C3C1)=O)C2 c1(CCC(=O)N(CC(C)O)CCNC(C(C(C)C)SC)=O)cnc(C)nc1O C(CCC(O)CO)N(C(=O)CC1CC(NC(=O)CC(O)CN(C)C)C1)C N1(CCC(=O)N(C2CCN(C(c3c(CC)noc3)=O)C2)CCO)C(=O)CCC1=O S(=O)(=O)(c1cnccc1N1CCC(F)(CF)C1)N(CCN(CC)CC)CC c1(C(=O)N(Cc2ccncc2)Cc2ccsc2)csc(-c2ccco2)n1 c1(CC)ccoc1C(=O)NC(CC1CCCC1)C(=O)NCC(F)(F)Br C(=O)(C1=CCCO1)NCC1(C(=O)NCCCCC#C)CCCO1 C1(CC(=O)NC2C(C(=O)OC)COC2)(NC(=O)CC(C)C2CC2)CCN(C)C1 C(C)(C)(CCC(=O)NCC(C)CC(=O)NC(CC1CC1)C(O)C(C)C)OC C1(C)CC(C)(C)CN1C(=O)C.c1(CC)c[nH]nc1C(=O)NCC(C1CCCCC1)O C(=O)(CC(CN)C(F)(F)F)N1C(c2c(C)c(Br)ccc2)CCC1 N1(C(C(C)n2cncn2)=O)CCC(NC(=O)C(C)SC(F)(F)F)C(C)(C)C1 CC1CC12NC(=O)N(C1CCC(CC(F)(F)F)CC1)C2=O c1(N(CC(C)CNC(c2c(F)ccnc2F)=O)C)ncnc(N(C)C)c1[N+](=O)[O-] CCCCC(CC(=O)N(C1CCN(OC)CC1)C)NC(C1CCC(=O)CC1C)=O n1(C(C)C)ncc(C(=O)NCCC(C)NC(c2nnsc2C(F)F)=O)c1F c1(C(c2nnnn2C(C)(C)CC)NCCCCSC)ccn(CCF)n1 Cc1c(C(=O)NC2CCCC(C(N3CCC(n4ccnn4)C3)=O)C2)c[nH]c1C#N Cc1c(C(=O)CN2CCOC3CC23)nnn1Cc1ccccc1 CCCCC(CNC(=O)C(c1cccc(OC)c1)C)NC(c1ccc(SC)o1)=O C(C(C)(C)n1cccn1)NC(CN(C)C(C1CCOC1)=O)=O N1(C(CC2C(C)C(=O)CC2)=O)CCC2(CC2)CC1C(=O)NCc1ccnc(CO)c1 N1(C(c2ccn(CCCC)n2)=O)CCN(C(c2cnc(O)c(Cl)c2)=O)C(CF)C1 C(=O)(C#CC(C)(C)CNC(C1CCC(F)C1)=O)N1CC(C)N(C2CC2)CC1 Cc1sc(C)c(C(=O)NC(C)C(C)NC(=O)CCn2cnnn2)c1C#N N1(C(CCC2(C)CC2)=O)CC(NC(c2sc(C#N)cc2Cl)=O)C(C)(C)C1 n1(CC(N2C(CNC(C(C)(C)CO)=O)CC(F)C2)=O)ncc(C#N)c1N C(=O)(CC(C=C)CCC)N1CC2C(CNC(CCc3ccc(OC)cc3)=O)C2C1 N1(CC2(NC(C(N3CCC(C)C3)=O)=O)CC2)CCN(C(C2COC(=O)C2)=O)CC1 c1(C(N2CC3CN(Cc4cc(C)c(O)cc4C)C3C2)=O)c[nH]c2ncc(Br)nc12 C1(NC(Cn2ncc(C)c2)=O)C2CC(NC(C3(F)CCOC3C)=O)CC12 c1(C(=O)NCC2N(C(C=CC(=O)OCCCC)=O)CC2)ccc2c(c1)C(=O)NCC2 CCC(C)CC(=O)N(C1CCCN(C(=O)Cc2cnn(CC)c2)C1)C C1=NN(c2ccc(C(=O)NCCn3cc(C4CCOC4)cn3)cc2)CCC1 c1(CN(C(c2n[nH]cc2NC(=O)CC2CC3CC3C2)=O)CC)c(C)cccc1Cl C1(C(N2C(CNC(C3(C(=O)OCC)CCO3)=O)CCC2)=O)C(Cl)(Cl)C12CC2 N1(C(CC(c2ccc(C)cc2)C)=O)C(C)C2CC1C2NC(=O)C(O)C(C)(C)C C1(NCCCCC(C)N(C(CCc2nc(C)c(C)o2)=O)CC)CC1C1CCCC1 C1(NC(=O)CC2C=CCC2)CS(=O)(=O)C12CCN(C(c1cnns1)=O)CC2 C1(CC)C(NC(=O)C(C)CO)CCN1C(c1cc(C)n(-c2ccccc2Cl)n1)=O CC1(C)COCCC1NC(=O)C=CC1CCCN1C(=O)CN1CCCCC1 C(=O)(C1CCCc2ccc(O)cc21)N1CC(NC(=O)OC(C)(C)C)CC(C)C1 c1(C(N2CCC3(NC(=O)C=Cc4cocn4)C(C2)C3)=O)ccc2c(n1)OCCO2 C1(NC(C(CCC)C)=O)CCN(C(=O)C(CC)CCc2ccccc2)CC1C N1(C(C(C2CC2)SC)=O)CCC=C(C(=O)NCCOCC(C)C)C1 C(=O)(N=c1ccnc2[nH][nH]cc1-2)C1N(C(C)C)CCC1.N1C=CCSC1=O C(=O)(C(C)C(C)NC(c1cnnc(C)c1)=O)Nc1occ(C)c1 N1(C(CCSCCCC)=O)CCC(n2cc(NC(C34CCC(C3)C4)=O)nn2)CC1 c1(CN(C)C(c2cn(C(F)F)cn2)=O)cnn2c1CN(C(=O)CCC(N)=O)CC2 C(=O)(C1CCCn2cc(C)nc21)N(C1(O)CCN(C(=O)CC2(C)CC2)CC1)CC N1(C(C2(NC(C)=O)CC2)=O)CC(NC(=O)C(C(C)C)NC=O)CC1C c1(C(=O)NC2(C)CN(C(CC(CC)OC)=O)C2)cnc(Cl)cc1N N1(C(c2ccc(C)nc2)=O)CCN(C(=O)Cc2cncnc2)CC1CC(C)(C)C c1(N(C)CC2C(C)C2)nc(N2CCCC(C3(C)CC3)C2)nc2c1CCCCC2 c1(C(N(C2CN(C(c3cc(OC)nn3C)=O)C2)C)=O)coc2c1C(O)CCC2 c1(OC)ccc(C(=O)NC2(CCNC(=O)C3=NOC(C)C3C)CC2)c(F)c1Cl CC(C)C(CO)C(=O)NC(CNC(c1cc(F)cnc1O)=O)CC(F)(F)F N1(CC)CC(C(N2CCC(NC(=O)CC3(OC)CCCCC3)CC2)=O)CCC1=O C1(C(=O)NCC2C(NC(=O)CCc3ccc(F)cc3F)C2)CCC2(CCC2)CC1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CNC(c1ccc(NC(=O)OC)cc1)=O)CO CC1=C(C(=O)N2CCN(C(=O)CCCNc3ccccc3)C3CCC23)CCCC1 C12(CNC(=O)Cn3ccc([N+](=O)[O-])n3)CCCC1CCN2C(c1nncs1)=O N1(C(Cc2c(C)ncnc2C)=O)CCC2(CC1)CC(NC(=O)C(F)=CCCF)C2 Cc1nc2ccc(Br)cc2c(=O)n1NC(=O)C(C)SCC(C)C O=C(C1=NN(Cc2ccc(Cl)cc2)C(=O)CC1)N1CC2OCCOC2C1 C1(N(C)CCn2cc(C3(O)CCOC3)nn2)CCOC1(C)C c1(OCCNCC(C2CCCC2)OC)ccc([N+](=O)[O-])cc1C c1(C(=O)NCC2(F)CC(NC(CNC(=O)NC)=O)C2)ccc(S(C)(=O)=O)cc1Cl Cc1nc(CC(=O)NCCC2CCC(NC(c3cc(F)cs3)=O)C2)cs1 N(C(=NCCCN1CCOCC1)NC1CC(n2cccn2)C1)CC1N(C)CCC1 c1(C(N(C(CNC(C2CCCS2)=O)C2CC2)C)=O)c[nH]nc1-c1ccncc1 N1(C(c2[nH]cc(C)c2)=O)CCC(NC(c2cc3n(n2)CCC3)=O)C(F)C1 C1(NC(c2cc(CCC)on2)=O)CCN(C(=O)Cc2cc(F)ccc2C)C(C)C1 S(=O)(=O)(c1cccc2c1NC(=O)CO2)N(c1cnnn1C)C C1(C(=O)NCC(n2cc(CC(CC)O)nn2)C)CC2(C1)CS(=O)(=O)C2.OCC n1(CC(=O)NCC2(C)N(C(CN3C(C)CCC3C)=O)CCC2)cnc([N+](=O)[O-])n1 CC(CN(C)C)CC(=O)NCC1(NC(=O)Cc2cccs2)CCOC1 Cc1cccc(N(C(c2cc(Br)ccn2)C(=O)NC(C)CC#N)C)c1 C(=O)(CCCC(C)(C)NC(=O)CCc1cnn[nH]1)NCC1(CC)CCOC1 C1(CNC(c2c(C)nccc2)=O)CCC2CN(C(C3COC(=O)N3)=O)CC12 n1(C)ncc([N+](=O)[O-])n1.N1(CC)CC(CN(c2ccccc2)C(C(=O)NCC)=O)OC1=O CC1(O)CCCN(C(c2cc(C3CC3)nc(C3CC3)c2)=O)CC1 C1(C(=O)NC(c2nccs2)C)CN(Cc2ccncc2O)CCC1O C(=O)(CC(CC)C(C)(C)C)NCCCCC(C)NC(c1ccc(OCC)nc1)=O N1(c2n(Cc3ccccn3)c(-c3nscc3Br)nn2)CCCC(O)CC1 C1(CC)CN(C(c2cnn(CCO)c2C)=O)CCN1C(=O)C(C)P(C)(C)=O c1(N2CCC(c3nc(C)[nH]n3)C2)nccc(=NCC(O)CN2CCC(O)CC2)[nH]1 C12(NC(c3cc(SC)oc3)=O)CCCC1N(C(C1CCc3nccn3C1)=O)CC2 C1(OC)CC(C(N2CCC(N(C(=O)Cc3ccns3)C)C2)=O)N(S(C)(=O)=O)C1 c1(OC)coc(NCC2(C(=O)NCc3cccc(I)c3)CC2)cc1=O C(C)(C(=O)N=c1ccn(CC(=O)NC2CCCC(C3CC3)C2)[nH]1)N(C(C)=O)C C1(C(=O)NC23CC(NC(C4CCC5(CC4)CC5)=O)(C2)C3)CCC2(CCOC2)O1 c1(OC)ccc(C(N2CCOCC(CNC(c3sccc3C)=O)C2)=O)c(OC)c1 C1(C(=O)NC(CCC)C)CCCN(C(c2cnn(C)c2N)=O)C1C N1(C(C)=O)CC(C(N2CCCC2c2noc(C3CC3)n2)=O)CC2OCCC12 CC(C)C(C(C)NC(=O)CC1OCCO1)NC(c1csc(-c2cccs2)n1)=O C1(S(=O)(=O)N)(C(=O)OC)CC1C.C123CC(CN1C(=O)c1nccc2n1)C3.OC CC1CC(NC(C2(NC(c3cnccn3)=O)CC2)=O)CN1C(=O)C1CC1 N1(C(C(C2CCN(C(CN(C3CC3)CC)=O)C2)C)=O)CC(C)(C#N)C1 Cc1cnc(C2CN(C(=O)C=Cc3cnccn3)C2)[nH]c1=NC1CC1 N1(C(C(CCC#C)O)=O)CCCC2(C1)C(NC(c1ocnc1CC)=O)CCN2C c1(N2CCN(C(c3ccc(C#C)o3)=O)CC2C)ncnc2cnn(C)c12 Cn1c(O)nc2cc(NCN3CCC(OC4CCOC4)C3)ccc12 N1(C(C(CCC)CCC)=O)CCC(C2CCCN(C(c3cncn3C)=O)C2)CC1 C1(C(N(CCCNC(CCSCC)=O)C)=O)CCCN1C1CCCC1 c1(OC)cc(Cl)c(C)cc1C(=O)NCC1CC1NC(=O)CC1(O)CCC1 CN1CCN(CC(=O)NCCC2CN(C(C3(C(F)F)CCCO3)=O)CCO2)CC1 C1(NC(c2cnc(CCC)s2)=O)CN(C(=O)CCc2c(C)n[nH]c2C)C2CC12 c1(NC(C2C=C(C)CN2)=O)cccc2c1oc(=O)n2C C(CC(C)C(=O)N(C)CCN(C)C(c1cccn1Cc1cccnc1)=O)OC C=CC1(C(=O)NC2CCC(NC(=O)COCCc3cccs3)C2)CCC1 CC1C2CCC(C2)C1C(N1CC(C(C(=O)NCc2nc(C#N)cs2)N(C)C)C1)=O N12CCC(C3CN(C3)C(=O)C3C(C3)C1=O)CC2.C1(C(=O)OCC)CN(C(C)=O)C1 N1(C(c2ccc(OC)c(OC)c2)=O)CCC2CCN(C(=O)CCCC#N)CC2C1 c1(CC)ncoc1C(=O)N(CC(=O)N(CC(O)CO)C)CC(C)C c1(C(=O)NCCCN(C(C(C)OCC)=O)C(C)C)cc(OC)c2nc(C)oc2c1 C(c1cc2ccccc2o1)=CC(=O)NC1CCCCN(C(=O)C2=COCC2)CC1 C1(C(=O)NCCC2(NC(=O)COc3ccon3)CC2)CCC2(CCCCC2)C1 c1(C(=O)NCCCCCn2cc(CC(OCC)OC)nn2)ccc(Cl)cc1Br c1(CC)nc(=N)[nH]cc1C(=O)NC(CCNC(c1cc(Cl)cnn1)=O)C(C)C C(=O)(CC(C)CC(C)(C)C)NCC(C)(C1CCC1)NC(C#CC(C)C)=O CCC(C)CC(=O)C(=O)NC(COC(C)C)C(=O)NC1CCC2CC1CO2 C1(C(N(CCNC(c2cc(C3CCOCC3)[nH]n2)=O)CC)=O)CCC2CC1CO2 c1(NC(C)=O)ccc(Cl)c(C(=O)NC2C=CCN(C(c3cnc(C)[nH]3)=O)C2)c1 CC(C)CC(=O)N1CCCC1CN(C)C(c1ccnnc1)=O CC1CN(C(c2cn(C)nn2)=O)CCC1C(=O)NCCc1nccc(O)n1 C=CCC(C(=O)NCC(O)CC(=O)N1CCCC(CCOC)C1)OC C(C1CCN(C(C2(F)CCCOC2)=O)CC1)=CC(=O)NCCCc1cccnc1 c1(C(N2CCC=C(C(=O)NCc3cc(Br)ccn3)C2)=O)ccc2ccccc2c1 C#CC1CCC(C(=O)NC(C2CN(C(c3cccc(F)c3CC)=O)C2)C)CC1 N1(C(c2c(C)nc(C)o2)=O)CC2CCCC2(NC(=O)CN(C(=O)C(C)C)C)C1 c1(C(N(CCNC(C2CC2CC2CCCCC2)=O)C2CC2)=O)c(C2CC2)noc1C C1(NC(C2(CNC(=O)CCC3CCOCC3)CC3(CC3)C2)=O)CCCCCC1F CC(CC(=O)N(C(C)CCNC(c1[nH]ccc1C1CC1)=O)C)c1ccco1 CCC(C(=O)OC)C(=O)N(C(C)(C)CC(=O)N(C1CC1(C)C)C)C Cc1c(N)ccc(C(=O)NC2CCCC2NC(C2CCS2(=O)=O)=O)c1C C1(NC(C=C(COC)C)=O)CC(F)CN(C(C2CC(=O)N(C3CC3)C2)=O)C1 C1(NC(C(CC)n2ccnc2)=O)CN(C(=O)CN2CCCCC2=O)CC1N=[N+]=[N-] c1(CC(C(C)C)C)ccc(C(=O)NCCNC(=O)CCc2ncc(F)cn2)cc1 CC(C)CC(C(=O)N(C)CC1CCC(NC(=O)CC(C)N(C)C)CC1)N(C)C c1(CNC(C2CCN2Cc2ccc(C3CC3)o2)=O)ccc(-n2cncn2)cc1 C1(N(C(=O)NC)C2CC2)CCCN(C(=O)NCCOC)C1 CCC(CC(F)(F)F)C(=O)NC12CC(NC(c3cnn4c3N(C)CC4)=O)(C1)C2 Cc1ccc(N2CCCCC(CNC(C3C4CCCC34)=O)C2)c([N+](=O)[O-])c1 C(=O)(CC(F)(F)C(C)C)N1CCCC(CC(=O)NCc2nc(C)sc2)C1 Cc1cc(C(F)F)nn1CC(=O)NC1(CNC(C2(C)CCC(=O)C2)=O)CC1 c1(C(=O)Nc2ccc(Br)cc2I)cccc2c1CN(S(=O)(=O)C(F)(F)F)CC2 N1(C(C2ON=C(C(C)C)C2)=O)CCCC2CN(C(C3CCCS3)=O)CCC12 C1(NC(CCCC(C)=O)=O)CCN(C(=O)C(=CC2CCCCC2)F)CC1(C)C C1(CNC(C2CCCCN2S(C)(=O)=O)C)COC(C)(C)O1 c1(OC)cc2ccccc2cc1NC(=O)CC1CN(Cc2ccnc(CO)c2)C1 c1(C(=O)NCCCC(C)(C)NC(c2cncc(C)n2)=O)cc(C)c(C)nc1O c1(NC(C2CCCCC2F)=O)ccnc(OCC(F)(F)F)c1 c1(C(=O)NCC(=O)OC)ccc(C(C)NC(=O)C(C)OC)cn1 N1(C(CCCOC(C)C)=O)CCC(NC(=O)C(C)CC2CC2)CC(C)(C)C1 C12(C)CC13CCN(CC3)C2=O.C1(OC)CC2CCC1CC2 C1(C(=O)NCc2ccnc(C)n2)CCN(C(C2C3CCC(F)(F)C23)=O)C12CC2 C12(CNC(C(CO)N(C)C)=O)CC(C1)C(NC(c1ccsc1)=O)CO2 N1(C(C2(C)CCCS2(=O)=O)=O)CCCCC(NC(=O)CSCC(N)=O)CC1 c1(C(N2CC(CCCCNC(C(C=C)(F)F)=O)C2)=O)ccc([N+](=O)[O-])c(C#N)c1 c1(SC)ncc(C#N)c(N2CC(NC(c3ccoc3)=O)C(C#N)C2)n1 C(C1=CN(C(=O)OC(C)(C)C)c2ccccc2OC1)=CC(=O)OCCN(C)C C(=O)(C#Cc1ccccc1)N1C(C(=O)NCCNC(c2ccccc2)=O)CC(O)C1 C1(NC(CC2(C#N)CC2)=O)CC2CN(C(c3c(F)cccc3Cl)=O)CC2C1 CC1CN(C(c2c(Cl)cnn2C)=O)CCC1CNC(=O)CN(S(C)(=O)=O)C N1(C(C2(CCNC(C(CC)CC)=O)CCCC2)=O)CCN2CC(C)CC2C1 N1(C(c2ccc(COC)cc2)C(=O)NCC(C)C)CCOC(C)(C)C1(C)C c1(C(N2CCC(CNC(C34CC(F)(C3)C4)=O)C(F)(F)C2)=O)ccc2oncc2c1 CC(F)(F)CCC(=O)NC1CC(F)(F)CC1NC(=O)Cc1ccc(O)nc1 S(=O)(=O)(c1c[nH]c2ccc([N+](=O)[O-])cc12)N1CCN(c2cc(C)[nH]c(=N)n2)CC1 c1(OCCCC)ccnc(NCC2CCC(NC(=O)C(O)C3CCCC3)CC2)n1 CC(C)C(O)C(F)(F)C(=O)NCC1(C)CCCN(C(=O)CSCc2cccnc2)C1 n1(C(C2CCCO2)C)nc(C2CC2)nc1-c1ccc(-c2ccccc2)[nH]1 C(=O)(C(CO)C(C)(C)C)N(C)CC1CCCCN1C(c1cnc(O)o1)=O CCCC(C)(O)CC(=O)N(C)CC=CC(N1CCOCC(C)C1)=O c1(NCC(CCC)(C)C)ccc(S(=O)(=O)NC(C)Cc2ccc(C)s2)c(Cl)c1 c1(OC)ccc(C(C)C(=O)NC(C2CCN(C(=O)C3=CCC3)C2)(C)C)cc1OC C(=O)(C(COC)C(F)(F)F)NCC1(C)CC(NC(C2C(CC)CCC2)=O)C1 c1(OC)cccc(C(=O)N(C2CC2)CC2CCCCN2C(c2ncnn2C)=O)c1 c1(N(C)CC2CCCS2)nccc(=NCCNCCN2CCCCC2)[nH]1 C1(CC(=O)N(C2CCN(Cc3csc(Br)c3)C2)C)CCC(O)C1 c1(C(=O)NCC(CNC(CC(C)N2CCCC2=O)=O)C)ccc2sccc2c1 C(=O)(C(C)(CC#C)NC(=O)CC1CCCC12CC2)NCCC(=O)NCC#C C1(SC)(NC(c2ncc(CO)n2C)=O)CCCN(C(=O)C(C)(C)OCC(F)(F)F)C1 C(CC(C)(C)C(=O)N1CC2(NC(=O)COC3CCCOC3)CC1C2)SC N1(C(c2cc(SC)c(F)cc2)=O)CCC2(CC1)CC2NC(=O)C=Cc1cn[nH]c1 c1(NC)ccccc1C(N1CCC(C(C)NC(=O)Cc2cnc(C3CC3)[nH]2)C1)=O N1(C(CCNC(c2cc(O)ncc2F)=O)=O)CCC(=C(F)F)CC1 Cc1cc(CN=C(NC2CCc3nccn3C2)N(C)C2CC2C)ccc1O c1(C(=O)NC2(C)CC(NC(c3c(CC)non3)=O)C2)cn2cccc(C)c2n1 N1(C(CCSCCCC)=O)CC(C(=O)NCC2CCC(=O)O2)C2(CCC2)C1 CC1(CC(N2CCCC2CCC2CCCN2C(=O)CC2CC(=O)C2)=O)CCCC1 C1(CNC(C(COC(C)C)(C)C)=O)CCN(C(C2CC2C(N)=O)=O)C12CC2 S(=O)(=O)(c1ccc(Br)cc1[N+](=O)[O-])N(C)CCOCc1ncccn1 C12(C(N(C)CC3CCN(C(c4cccs4)=O)C3)=O)CCC(C)(C1)OC2 N1(C(C2C(CNC(C=C(CC)CC)=O)OCC2)=O)CCOCC1C1CC1 CC(CC(C)NC(c1ncoc1C1CCC1)=O)NC(=O)CCn1cnnn1 C1(NC(=O)CCN2CCOCC2)CCN(C(c2cc(Br)ncc2F)=O)CC1O n1(CC(=O)NC(C)Cn2cc(CN)nn2)cnc([N+](=O)[O-])n1 c1(CC)noc2ncc(NCC3CCCN(c4ncnc(C(=O)O)c4C)C3)cc12 C1(NC(Cc2c(C)occ2)=O)CCCN(C(=O)Cn2cccnc2=O)CCC1 N1(C(CSCCOC)=O)CCOC(C(C)NC(c2csc(SC)n2)=O)C1 c1(C(=O)NCC2C3CN(C(c4ncc(CC)s4)=O)CC32)cc2ccccc2s1 N1(C(c2cnco2)=O)CCC2CCN(C(=O)Cc3nccs3)C2C1 c1(OC)ccc2c(=NC(C)C3CCCO3)[nH]c(=NCC3(CCOC)CC3)[nH]c2c1 c1(C(=O)NC2CCN(C(CCC#C)=O)C(C3CC3)C2)csc2cc(Cl)ccc12 c1(C(N2CC(NC(C3C(CC)CCO3)=O)C(C)C2)=O)c(N)cc(Cl)cc1F C(CO)(C(=O)NCC1COCC1NC(=O)CCCOC(C)=O)OC c1(NC(c2ccc(C)cc2C)C(=O)OC)nc2cnc(Cl)cc2s1 C(CN=c1[nH]c2c(c(=NC3CCCC3C)[nH]1)CCCCC2)NC(=O)NC Cn1c(C(=O)NCC2CN(C(C3CS(=O)(=O)C3)=O)CCO2)cnc1Cl c1(N(C)Cc2cccnc2)cc2[nH]c(-c3ccco3)nc2cn1 CC1(C(N2CCCC(C3CCCN3C(=O)Cc3cnccn3)C2)=O)CCCCC1 c1(C(=O)NC(C(=O)N(CC=C)CC=C)c2ccoc2)ccnnc1O c1(C(=O)NC(C)(CNC(=O)Cc2c[nH]ccc2=O)C2CC2)ccc2snnc2c1 C1(C)(CNC(C2C(OCC)CCC2)=O)CCCN(C(c2conc2C(C)C)=O)C1 c1(OC)ccc2c(=NCc3ccc[nH]3)[nH]c(=NCc3csc(O)n3)[nH]c2c1 Cc1cc(C(N2CC3CN(C(c4cc5n(n4)CCC5)=O)C3C2)=O)ccc1O CC(=O)CCCC(=O)N1CCCC(CCNC(=O)C(O)Cc2cnc[nH]2)C1 C12(NCCNC(C)=O)CC(NC(=O)C(C)NS(C)(=O)=O)(C1)OC2(C)C N1(C(c2cc(C)nc(O)n2)=O)CC2CCCC2(NC(c2nnc(C)s2)=O)C1 c1(C(N2C(C)(C(=O)NC(C3(CO)CC3)C)CCC2)=O)ccc2cncn2c1 c1(C(=O)NC2CC(O)CN(C(c3ccc(Cl)nc3O)=O)C2)cccc2cc[nH]c12 CC(CCCCNC(c1cn(C)nc1-c1cccs1)=O)NC(=O)CSCC(N)=O N1(C(c2cc(C)c(F)nc2)=O)CCC(C2CC2)C1CNC(c1c(C)noc1C)=O c1(N(c2ccccc2)C(=O)CCC2CCCO2)ccc(C(=O)CF)cc1 C1(CC(=O)N(CCC)CCNC(c2cc(C(F)(F)F)no2)=O)CN(C)CC1O c1(OC)cc(C)c(CN2CCC(CC(=O)NCc3cccnc3)C2)cc1OC c1(C(=O)NC2C(C)CN(C(C3(CC=C)CC3)=O)CC2C)cc(Cl)c(N)c(Cl)c1 c1(OCC)nccc(C)c1C(N1CCC(NC(c2csnc2Cl)=O)C(O)C1)=O C(=O)(C1CCc2cccc(Cl)c21)NC12CC(NC(C3CC3c3ccccc3)=O)(C1)C2 C1(C(=O)Nc2cc(-c3ccc(C)s3)[nH]n2)CCCN(C(=O)C2=CCCC2)CC1 N1(C(c2ccn(C)n2)=O)CCN(C(=O)CC2CC2c2ccccc2)CC1CCO CCCN=C(NCC1CCCSC1)NCC(C)Oc1ccccc1 c1(C(=O)NC2(C)CCN(C(=O)C(Cl)=CCl)C2)cc2c(Cl)cncc2s1 CC1(C(=O)NCC2CCCC2NC(=O)CN(c2ccc(Cl)cn2)C)CCC(=O)N1 N1(C(C)=O)CCC2CN(C(c3cc(S(C)(=O)=O)ncn3)=O)CC2C1 N1(C(c2c(CC)scc2)=O)CCN2CCOCC2(CNC(=O)CC2CC23CC3)C1 C1(C(=O)NC)=CN(C2c3ccccc3N(C(=O)C3CC3)C2(C)C)C1.C(C)(C)(C)O N1(C(CC(CC=C)(C)C)=O)CCC(O)(C2(NC(C3CC34CCCC4)=O)CC2)CC1 C(c1ccncc1)=CC(=O)N(C1CCC(NC(c2cncn2C(F)(F)F)=O)C1)C c1(NC(C)=O)ccc(S(=O)(=O)N2CCCN(C)CC2C)cc1 C(=O)(C(F)(F)CC(C)C)N1C(C)CCC(NC(C(C2CC2)OC)=O)C1 C#CCCC(O)CCNC(=O)C(C)(C)CNC(C1CC=CCC1)=O C1(NCCn2nnnc2C(c2cccc(CO)c2)OCC)COCCC1(F)F C1(CCC)(NC(C2CCOC(C)(C)C2)=O)CCN(C(=O)C(C)(C)OC(C)C)CC1 Cc1n[nH]cc1CC(N1CCC(N(CCO)C(C2CCOC2C(F)(F)F)=O)C1)=O C1(C#N)(CNC(CCC2CCN(C(C3C(C)CC3)=O)C2)=O)CC(C)(C)C1 C1(C(=O)NCC2OCC(CNC(c3ccc(OC)s3)=O)C2)COCCC1(F)F N1(C(C2C(=C)CC2)=O)CCC(CO)C(NC(=O)COCC(c2ccccc2)=O)C1 C(CN=C(NC1CCCSC1)NC1CCS(=O)(=O)C1)OC.C1C(=O)O1 Cc1cc(=NCC2CCOC(C)C2)[nH]cc1S(=O)(=O)NCCS(=O)(=O)NC1CC1 c1(CCC(=O)NCCNC(C(c2ccc(OC)cn2)(F)F)=O)ccc(OC)c(O)c1 n1(CC)ccc(C(N2CC3(CC3C(=O)NCc3ccc(C)cc3)C2)=O)c1C c1(SC)cn(C)nc1C(=O)NC1CC(NC(C23CCCC2CC3)=O)C1 c1(C(=O)NCCCC2(CNC(C3C(COC)C3)=O)CC2)cc(Cl)no1 N1(C(CCc2c[nH]c(=N)[nH]2)=O)CCC(O)(CNC(C23CCC(CC2)O3)=O)C1 CC(C(C(=O)NC1CC(=O)N(C)C1c1cncn1C)N(C)CCF)C(C)(C)C N1(C(c2c(C)nsc2)=O)CCC(O)(CN(C)C(c2cc(C(C)(C)C)n[nH]2)=O)C1 c1(OC)cc(N)ccc1C(=O)NCC1(CO)CCN(C(C2C=CCS2)=O)C1 Cc1nn2cc(C(=O)NC3CC4CCC3N(c3ccncn3)C4)nc2s1 CC(C(=O)NC1CCCCC1CNC(c1cc2c(s1)CCC2)=O)C(C)(C)C C12(NC(=O)CC34CCC(CC3)C4)CCOCC1CN(C(=O)C(F)(F)C(F)(F)F)C2 Cc1cc(F)cnc1C(=O)NC12COC(C1)C(NC(c1ccncc1F)=O)C2 c1(C(=O)NC23CC(NC(c4ccn(C(F)F)n4)=O)(C2)C3)cc([N+](=O)[O-])ccc1O CC1=NC(C(=O)NCCCOCCNC(c2ocnc2C(F)F)=O)CS1 c1(SCC)cnc(O)c(C(=O)NC2CCN(C(=O)C(F)OC)C2C)c1 N1(C(c2ccc3nc(C4CC4)sc3c2)C)CCCC2CCCN(C)C12 N1(C(CC(=O)OCC)=O)CC(C)CN(C(C2CCCN2C2CC2)=O)CC1C C1(C(N2C(C(=O)NC3CCCOC3)CC3CC32)=O)CCc2ccccc2C1 N1(CC(=O)N(C2(NC(=O)C=Cc3cccnc3)CC2)C)CCC2CN(C)CC2C1 c1(COC)cncc(C(=O)NC2CCCC2NC(=O)CCCc2cc[nH]n2)c1 C=CCCCC(C(=O)N(C)Cc1noc(CC)n1)NC(=O)Cc1cnns1 N1(C(COCCC#C)=O)CC2CC2(C(N2CCOCC2CC)=O)C1 C(=O)(C1CCCc2nn[nH]c21)NCCOCCNC(Cc1cc(C)c(O)cc1)=O c1(OC)nccc(C(=O)NC2CC(NC(c3ccnc(OC)c3F)=O)C2)c1F C1(N(C(C(CSC)C)=O)C)CCCN(C(c2csc(-c3nc[nH]n3)n2)=O)C1 N1(C(C(=O)NCCOC)c2cc[nH]n2)CC(C)C12CCOCC2 N1(C(CCCSC)=O)CCC(C)(CNC(=O)Cn2nnc(C3CC3)n2)C1 c1(C(=O)NC2CCC(C)N(C(c3ccc(C#N)[nH]3)=O)C2)ccc2c(c1)CCOC2 C(CCC(F)(F)F)ONC(C1CCCN(C2CCC(O)CC2)C1)=O Cc1cccn2c(=O)c(C(=O)NCC3CCC3NC(=O)CC3CC3(C)C)cnc12 N1(C(C2CCCCS2)=O)CCC2(CCCN2C(=O)CSc2ccc(Cl)cc2)C1 N1(C(CC)=O)CCc2c(CNC(c3cc(Cl)c(C)cn3)=O)cccc2C1 C(CCCCC(=O)N1CC2C(CNC(C3CC(=O)N(CC(C)C)C3)=O)C2C1)SC C1(CC(=O)NCC2CC(NC(=O)CCN3CCC3)C2)(OC)CCC1 c1(C(N2CCCC(C(C)NC(c3nnc(C)s3)=O)C2)=O)ccc(Cl)cc1C c1(NC(C2CC(n3cccc3CN(C3CC4CC4C3)C)C2)=O)cc(C)c(C)nn1 c1(C(=O)NC2CCC(NC(c3cccc(C(N)=O)c3)=O)C2)cnc2occc2c1 c1(NC(C2CN(C(=O)CC3CCCO3)C2)=O)n[nH]cc1CNc1ccccc1 N1(C(CSC)=O)CC2CC1CN(C(C1OCCC1c1nn[nH]n1)=O)C2 c1(C(=O)NCC2(CNC(C(CO)OC)=O)CC2)[nH]c(C)nc1C CC1OC2(CNC(C3CC3C#N)=O)CC1(NC(=O)C(C(C)O)N(C)C)C2 c1(C(=O)NCC2(OCC)CN(C(c3ccoc3)=O)C2)cc([N+](=O)[O-])ccc1NC C(=O)(CC1=NNC(=O)C1)N1C(CCCC)CN(C(C2(C)CCCS2(=O)=O)=O)CC1 C1(NC(C(C)(N(C)C(C2CCCCO2)=O)C2CC2)=O)CCC2(CC1)CC2 C(CCN=C(NCCC1CC1C(N)=O)N1CC(C)N(C)C(C)C1)SC c1(N(C)C)ncc(C(N2CC(NC(C3NC(=O)C4CC34)=O)C2)=O)cc1Cl c1(NC(C2CN(C(CC)=O)C2)C(=O)N(C)C(c2ccccn2)C)cccnc1S C(=O)(CCC(C)(F)F)N1CC(OC2CCN(C(c3n(COC)ncc3)=O)CC2)C1 N1(C(CCC2N(C)CCC2)=O)CC2CC(O)C1C2NC(=O)CCOC1CCC1 C(=O)(CCC(C)NC(C)=O)N(CCc1cn(CCC2CCCC2)nn1)CC N12CCC(C(C)(C)C1)C2=O.CCC(C)CC(=O)OC.N12C(CC1C)C2=O c1(C(=O)NCCCn2cc(C3C(C)C3)nn2)ccc(C(=O)NCCO)nc1 c1(C(C)NCC(C(F)F)n2cccn2)cc(Cl)cc(Cl)c1F CCCCC(C)C(=O)N(C1CC2CCC(C1)N2)C(C)(C)C C1(NC(C(c2ccn(C)n2)(C)C)=O)CCN(C2CN(Cc3cnccn3)C2)CC1 CC(C)CC(CNC=O)CC(=O)NCC1(CNC(C2CC2C)=O)CC12CCC2 C1(CNC(C2(C#C)CN(C(=O)C(C)n3cncn3)C2)=O)OCC2CCC1C2 C12(CNC(CCCCC=CC)=O)CCC(CC1)N(C(c1coc(SC)c1)=O)C2 c1(C(=O)NCCCC(C)(C)c2noc(C3CCCC3(F)F)n2)ccc(Cl)c(N)c1 C1(C(=O)Nc2c(C)cc(Oc3ccccc3)cc2)CN2CC3CC2(CO1)C3 C1(NC(C23C(CN(C(c4[nH]cc(C#N)c4)=O)C2)C3)=O)CCS(=O)(=O)CC1 N1(C(C2CNC(=O)N2)=O)CCC(C(F)F)(CNC(c2cnc(Cl)s2)=O)C1 c1(NCc2c[nH]c3cccc(C)c32)cc(Br)c(C)c([N+](=O)[O-])c1 C1(NC(c2ccc(CNC(c3cccc(C)c3)=O)cn2)=O)C(C)CCCC1C C1(CNC(C(COC)OC)=O)CCN(C(=O)CC(C)(C)c2cccs2)CC1C c1(C(=O)NC2C3(CC(NC(C(CC#C)O)=O)C3)C2)cccc2ccsc12 C1(CNCc2scc(CC)c2)CC(C2CCCCC2)CN1C c1(C(=O)NCCCOCCNC(c2c(C)snn2)=O)ccc2c(c1)NCCC2 N1(C(Cc2c(C)noc2Cl)=O)CCC2(CC1)CC(NC(=O)C1=CCCOC1)CO2 N1(C(c2n(C)nc(O)c2)=O)CCC2C(C1)CN2C(c1nc(Cl)c(Cl)s1)=O c1(C(=O)NCC2(NC(C(C)OCCCC)=O)CC(F)(F)C2)cnc2ccccn12 CCCC(C)(CC)C(=O)N1CCC(=O)C(NC(C)=O)C1 N#Cc1ncc(C(=O)NC2CN(C(c3cncc(-n4cccc4)c3)=O)C2)s1 N1(C(CC2C=CC(NC(CSS(C)(=O)=O)=O)C2)=O)CC2COC(=O)C2C1 C1(CC(=O)NCCOCC(C)C)C2CCC(C2)N1C(C1CC2C=CC1C2)=O c1(OC)ccc(C(=O)C(=O)NCCc2c(C)cccc2C)cc1Br N1(C(=O)OC(C)(C)C)CC2CCC2(C(N2CC(C)(COc3cnn(C)c3)C2)=O)C1 C1(NC(c2c(C)sc(O)n2)=O)CC2CC(NC(c3nnsc3C)=O)CC2C1 N1(C(c2n[nH]c(C)c2O)=O)CCN(C(=O)C(C)CCN(C)C)CC(O)C1 c1(C(N2CC(NC(C34CC3CCC4(F)F)=O)CC3(CC3)C2)=O)cnn2cnnc2c1 Cc1ccccc1CNC(C1CCCC1CNC(=O)CCc1cncs1)=O Cc1cc(CC(n2c(-c3cccc(C)c3)nnc2S)C(=O)OC(C)C)ccc1F C(=O)(C(C)C1=CCCC1)N(C1CC2CN(C(c3n(CC(C)C)ncc3)=O)C1C2)C c1(C(=O)NC(CC(C)NC(=O)CNC(C2CCOCC2)=O)C)cncc(CO)c1 C1(C)(C(=O)NCCC(CCNC(c2c(COC)cco2)=O)C)CCC(C)=C(C)C1 CCCCC(C)CCC(=O)N(C)CC1OCCC1C(=O)OC.C12(CC1)C(=O)NC2 c1(COCC(=O)N(C(C)C)CCN(C)C)ccc(Sc2ccccn2)cc1 c1(N2CCC(C)(C)C(CO)C2)ccc(S(=O)(=O)NCc2cncc(F)c2)c(Br)c1 CC(C)(O)CCCCCC(=O)NCCN(CCOCCO)C(C1CC2CC1C2)=O N1(C(CC(CC)O)=O)CCCC(N(C(c2cc(F)ccc2N)=O)CC)CC1 C1(NC(COC(C)C)=O)CC2CN(C(c3cc(C4CC4)[nH]n3)=O)CC12 Nc1cnc(C(N2CCC(CCNC(=O)CSc3cn[nH]c3)C2)=O)cn1 N(C1c2cc(Br)ccc2CC1)C(CCCCCN(C)C)=O C1(CC(=O)NCCCN(C(C(CCC)OC)=O)C(C)C)CC2(CCOCC2)CO1 C(=O)(CC(C(F)F)NC(=O)C(C)=C(C)C)NC(C=C)C N1(C(C=CCC)=O)CC(C(F)(F)F)OCC1CNC(c1occc1C1CC1)=O Cc1[nH]cc(C(=O)NC2CC3CCC2N3C(C2CC=CC2)=O)c(=O)c1Cl CN1CC2CCN(C(c3ccoc3CNC(c3sccc3Cl)=O)=O)C2C1 C1(NC(c2cc(Cl)cs2)=O)CN(C(=O)C(F)(F)c2ccncc2)CC12CC2 Cc1ccn(CC(=O)NC(C)C(C)NC(c2cccs2)=O)n1 c1(N(C(C(=O)N(CCCO)CC#C)=O)C(COC)COC)ccccc1 CCC(CC(Cl)Cl)C(=O)N1CC2C(NC(c3cncc(C(F)(F)F)c3)=O)C2C1 Cc1cc(O)c(C(N2CCC(C)C(NC(=O)C=CC3CC3)C2)=O)cc1Br C(CCC(C)(C)C(=O)NC1CN(C(c2oncc2C)=O)CC1C)OC N1(C(CCC)=O)CC2(CCN(C(c3cnn(C(C)CC)c3CC)=O)CC2)C1 c1(C(=O)OC)ccc(C(=O)NCC(C(C)(C)C)NC(=O)C=CCCC=C(C)C)nc1 c1(OC)ccn2c(C(=O)NC3CCC(N(C)C(C4CC4CF)=O)CC3)cnc2c1 C1(CC(=O)NC(CN(C(c2snc(O)c2Cl)=O)CC)C)COCC1(C)C N1(C(C(=O)Nc2c(C)c(Cl)ccn2)=O)CCc2ccsc2C1 C12(CCN(C)C1)C(=O)N2.C1(CC(=O)NC(CC=C)C2CC2)CC2CC2C1 Nc1cc2c(cc1CNc1ncccc1-c1ccncc1)OCO2 N1(C(C2CC23CCC3)=O)CCCC2(NC(C3(C4CCCO4)CCC3)=O)CC2C1 c1(CC(N2CC3C(CN(C(C(C)NC(CC)=O)=O)C)C3C2)=O)cccc(F)c1O CCC(C)(CNC(=O)C(Cc1cnc[nH]1)NC(c1ccc(=N)[nH]n1)=O)C(N)=O N1(C(c2c(C)n[nH]c2)=O)CCC(C)C(NC(C2CCCS(=O)(=O)C2)=O)C1C C1(C(CN(C)CCn2cnnn2)C=O)CCCN(C(=O)C(O)Cc2cnc[nH]2)C1 C1(C(=O)NCC(CCC)NC(C2(N(C)C)CCCCC2)=O)CCc2nn[nH]c2C1 C1(NC(C(C)CN(C)C)=O)C=CCN(C(c2ccccc2C2CC2)=O)C1 N1(C(C2C(C)C2C)=O)CCC2C1CCCN2C(c1cc(C2CCC2)[nH]n1)=O CCC(COC)C(=O)NC(C(=O)NCC(O)C1CC1)C1(C)CC1 C1(NC(C(C)SC)=O)CC2CCC1C(NC(c1csc(C(C)(C)C)n1)=O)C2 n1(CC(N2C(CCC(=O)Nc3ccc(F)s3)CCCC2)=O)ccc(O)nc1=O N1(C(Cc2nc(C)on2)=O)CCC(O)C(CC(=O)NC(C)(C)CC(C)C)C1 C(c1ccccc1)=CCN(C(CN(C(c1cc(C)on1)=O)C)=O)CC1CC1 c1(C(=O)NCc2c(CN(C)C(C3CCSC3)=O)cccc2)ccc2occc2n1 c1(OC)cc(F)ccc1SC(c1noc(CC(C)C)n1)c1nnnn1C(C)C.CCN C=C(C)C1OCCC1CNC(=O)CN(C(c1ncoc1COC)=O)C1CC1 CN1CC(C(=O)N(C)CCN(C)C(c2cnc(C(C)(C)C)nc2)=O)OCCC1=O c1(C(N2CCC(C)(CNC(c3ccc(C(C)C)cc3)=O)C2)=O)cc2sccc2s1 N1(C(C2ON=C(CC)C2)=O)CC2CCCC1(CNC(=O)Cn1cccnc1=O)C2 C1(C(c2nnnn2CCCSC)CCOC)(NC2CCC3CCC23)CCCOC1 CCCCCC(=O)NCc1nocc1C(=O)NCCC1(C)CCCC1 C(=O)(CCCC(F)(F)CO)N1CC(CNC(COc2cccc(C)c2F)=O)C(O)C1 C(C(CC(C)C)C(=O)NC(COC)CC(=O)N(C)CCn1cncn1)OC C1(C(N2C(C)CNC(=O)C2)=O)CCN(C(c2ccc(=N)[nH]n2)=O)C12CCC2 c1(C(N2CCC(NC(C3COCCC3(F)F)=O)CC2)=O)ccn2ncccc12 C(=O)(CCC(=O)N1CC(NC(C2(OCC3CC3)CCCCC2)=O)C1)NC Cc1ccc(Cl)c(S(=O)(=O)NCC(=O)Nc2ccccc2F)c1 c1(CC(N2CC(CC)N(Cc3cc(Cl)cnc3Cl)CC2)=O)cc(Br)cc(Br)c1O Nc1c(F)cc(F)c(F)c1C(=O)NCCCCCNC(C1(C2CCC2)CC1)=O CC1CCC(CNC(c2cnccn2)=O)N(C(=O)CCOc2cccnc2)C1 Cc1cnc2cc(C(=O)NC(CNC(=O)C(C(C)C)N(C)C)C(C)C)ccn12 c1(OCCC=C)ccc(F)cc1COC(=O)CNC(=O)Oc1ccc(Cl)cc1 c1(NC(CN(CC(COCCO)C)C)=O)ccc(Cl)c(Cl)c1.C=CCOC Cc1cc([N+](=O)[O-])cnc1C(=O)NC1CN(C(c2ccc3[nH]c(=N)oc3c2)=O)C1 C1(CNC(c2n(CC)nnc2)=O)CCC2(CN(C(=O)CC3CCCCN3C)C2)O1 C1(NC(CS(=O)(=O)NC)=O)CCN(C(c2cc(C)[nH]c(=NC)n2)=O)CCC1CO c1(N(C2CCS(=O)(=O)C2)Cc2ccc(Cl)cc2)ccc(S(=O)(=O)C(F)(F)F)cc1 C1(CNC(CC(CC)C)=O)CCN(C(c2ccnc(C)c2)=O)C1(C)C c1(C(N2CCC(C3N(C(C(C)=C4CC4)=O)CCC3)C2)=O)ccc([N+](=O)[O-])cc1Cl CN(CCCC(=O)N1CC(O)(CCNC(=O)Cc2cccnc2Cl)C1)N=O CCCCCCCCC(C)C(=O)NC1CN(C(c2cncnc2C)=O)C1 c1(C(=O)NC(c2cccnc2)C(=O)N(CC)Cc2ccccn2)ccnnc1O C(=O)(C(C)(C)C1CCCCO1)NCCC1CN(C(C(C)=CC2CC2)=O)C1 c1(CC(=O)NCCC2CC(C)N(C(=O)CC3CCC3)CC2)nc(F)c(F)cc1F Cc1cc(N)c(C(=O)NC(CNC(c2cc(C)c(C)o2)=O)C(C)C)c(F)c1 n1(CC(N2C(C(C)NC(CCC#C)=O)CCCC2)=O)cc(Cl)c(O)nc1=O c1(C(=O)NC2CC(CNC(C3(C)CC3(F)Cl)=O)C2)ccc(F)c2[nH]ccc12 c1(C(=O)NCC(CN(C(C2CCCN(CCC)C2)=O)CC)(C)C)cccc(F)c1O O=S(=O)(c1ccc(Cl)cc1Cl)N(c1nc2ccccc2o1)C1CC1 c1(CCC(=O)NC(C2N(C(C=CC(C)C)=O)CCC2)(C)C)cc(F)ccc1F S(=O)(=O)(c1[nH]c(=NCC2CC3(CO2)CC(F)(F)C3)ccc1Br)NCC(C)C CCCCC(C)C(=O)NCC(O)CCNC(c1cccc(C(=O)NCCC)c1)=O C1(C(N2CCC=C(CNC(C3CC(=O)NC3)=O)C2)=O)CCC([N+](=O)[O-])CC1 Cc1ccc(CC(=O)NCC2(C(=O)Nc3ccc(OC(F)F)nc3)CC2)c(C)c1 N1(C(Cn2c(CCC)ncc2)=O)CC2CC1CN2C(c1csc(COC)c1)=O c1(OC)cc(C)c(Cl)cc1C(N1CC2CCCC1C2c1ccco1)=O CC(=NOCC#N)C(=O)N(CC(C)C(=O)NC(c1ccccc1)CO)C C=C1Cn2c(C(N3CCC(CO)(NC(=O)C=CC4CCOCC4)C3)=O)nnc2S1 C(=O)(CC(C(F)F)C(C)(C)C)NC1C(C)(C)CN(C(=O)CCCC2CC2)C1 c1(-c2c(C(=O)NC(CNC(CC(C)(C)C3CC3)=O)CO)nco2)ccc(Cl)cc1F c1(-c2nc(-c3cc(CC(C)C)on3)on2)ccc(S(C)(=O)=O)nc1 C1(N(C(=O)C(=O)NC2CC2)C)CN(C(c2c[nH]c(-c3ccsc3)c2)=O)CC12CCC2 CCCC(C)CC(=O)NCCOCCCNC(c1cc(C)cnn1)=O C1(CNC(C(CC)n2ccnc2)=O)CC(C)(C)CN1C(=O)CCc1nnc(S)n1C c1(NCCOC)ccc(CNC(c2sc(C3CCCCC3)nc2C)=O)cc1 C#CC1(C(=O)NC2CCC(O)CC2)CCN(C(=O)CC2CC=CC2)C1 c1(C(=O)Nc2ccc(-c3cn(C4CCOC4)nn3)c(F)c2)cc(Cl)c(Br)cc1F Cc1ccc(C(N2C(C(=O)NOCC(F)F)CC2C)=O)o1 C(CC(C(=O)NCC(C1CCCCC1)(C)C)NC(C1CCC1)=O)=CC O=C(C1CCCc2scnc21)NC1CN(C(C2CCC3CC23)=O)C1 C(=O)(C(C)(O)CC)NCC(CC)NC(=O)C=Cc1ccc(C(F)F)o1 C1(NC(c2n(C)ccn2)=O)C2CCCC1N(CCOc1cccc(F)c1)C2 c1(CNC(CCN(CCC)C)=O)cnn(C)c1C(=O)NCCC(C)CO c1(C(=O)NCC2C(NC(CSS(C)(=O)=O)=O)CCC2)cc(C2CC2)nnc1O c1(C(N2CC(N(C)C(c3ccc(C4CCCO4)[nH]3)=O)C2)=O)ccn2ccnc2n1 c1(NCc2c(C(=O)OCCS(C)=O)nccc2)nc2c(cc1C#N)CC(C)CC2 C1(CNC(c2c(C)nn(C)c2)=O)N(C(=O)CSc2nncn2C2CC2)CCC1(C)C CCCCCS(=O)(=O)CC(=O)N1CCCC(N(C(c2ccc[nH]2)=O)CC)CC1 C1(C(N(CC(CC)(C)OC)C)=O)CC=CCN1C(c1nscc1C)=O S(=O)(=O)(c1cnn(C(F)(F)F)c1)C(C(=O)OCCC)C C1(CNC(C(C)=CC)=O)CCCN(C(=O)CC2COCC2O)CC1 N1(C(CC=C=C)=O)CCN(C(c2ccc(Br)c(C)c2N)=O)C(C)C1C C1(C(N2C(CNC(c3cnco3)=O)CC2)=O)COCC1n1cccn1 N1(C(C2CCC(CC)CC2)=O)CCOC(C(=O)NCCCCCCF)CC1 CC(C)(C)CCCCC(=O)NCCN(CC(C)O)C(C1(C)CC2CC2C1)=O C(=O)(C1CCc2c[nH]nc21)N(C(C)CNC(=O)CSCCC(c1ccco1)=O)C C(=O)(CC(C)(C)CN(C)C)NC1(C)CCN(C(CC(C)c2ccncc2)=O)C1 C1(C)(c2cn(CC)nn2)CCCCC1NC(C1CC(=O)N(c2nccs2)C1)=O c1(C(=O)NC2CN(C(CC(=O)OC)=O)C2)cn2c(n1)CCCC2 C1(CC(=O)NCCCSC)C2CCC(C2)N1C(=O)CN1CCNC1=O c1(C(=O)OC(C2(c3ccc(OCC)cc3)CC2)C)nc(F)ccc1Cl C1(C(N2C(CNC(=O)Cc3cccc(F)c3)CC(O)C2)=O)CC2C=CC1CCC2 c1(C(N(C)C(C2CCCOC2)C2CC2)=O)cn2c(n1)CCN(C1CCOCC1)CC2 N1(C(=O)Nc2c(C)cc(I)cn2)C2CCC1CC(N1CCOCC1)C2 Cc1cn(C)nc1C(=O)NC1CCC1NC(=O)Cc1ncccc1C C12(C(N3CCC(N(C(C(CC=C)C(C)C)=O)C)C3)=O)C3CCC(CC13)C2(F)F N1(C(c2cncc(OC)c2)=O)CCCC(N(C)C(c2cnc(Cl)cc2N)=O)CC1 C1(NC(c2cn(CC)nn2)=O)CCCN(C(c2ccnc(CC(C)C)c2)=O)C1C Cc1cc(C(=O)NC(C)(CNC(C2CC2CF)=O)C2CC2)cs1 N1(C(CCC(=O)NC)=O)CCN(C(=O)CC2CC(=O)NC(=O)C2)C(CC(F)F)C1 CCC(CC)N(CCC(=O)NC(C)CN(C)C(C1CCCC1)=O)C C12(NC(=O)COc3ccccn3)CCC1CN(C(C13C4C5C1C1C3C4C51C)=O)C2 Cc1ccc2c(C(=O)NC3CCC(CNC(c4csc(C)c4C)=O)C3)c[nH]c2c1 c1(C(N2CCC(C)(C(N3CCC(C#N)C3)=O)C2)=O)cccc2[nH]ccc12 C1(NC(C(CCC)O)=O)CCC2(CC1)CN(C(=O)C1CCc3ccccc31)C2 C(=O)(C(CNC(=O)C=CC=C(C)C)C(C)(C)C)NCC1(C)ON=C(C)C1 c1(C(=O)NCCNC(C=C(CC)c2ccc(C)cc2)=O)cn2ccc(OC)cc2n1 N1(C(C(=C)CC(C)N(C(c2ccccc2)=O)CCC)=O)CC(C)(C)C(O)C(C)(C)C1 C1(CN(C(c2c(CC)cccc2)=O)CCNC(=O)C(CC)SC)CCCC(C)(C)C1 N1(C(CC2CCN(C(c3cc(CC)sn3)=O)C2)=O)CC2CC1CS2=O N1(C(CCCN(C(=O)OCC)C)=O)CC2(NC(=O)CN(C)C)CCC1C2 CC(C)CC(C(=O)N1CC(N(C(=O)CC23CC(C2)C3)C)C1)NC(=O)C1CC1 c1(NC(c2cn(CC3CCCO3)nn2)=O)cc(Cl)cc2c1OCCC2 C1(NC(c2cn3c(n2)CCC3)=O)CC2CCC1CN2C(=O)CC1CC1(Cl)Cl C1(CNC(C(COC)O)=O)C(C)CCN1C(C1(c2ccc(F)cn2)CC1)=O Nc1ccc(C(N2CCN(C(c3ncc(F)cc3F)=O)CC2C(F)F)=O)nc1N Cc1cnc2[nH]cc(CN3CCC(C(=O)NCCc4ccccn4)C(F)C3)c2c1 c1(CNC(c2c(C)c(Cl)c(Br)cc2)=O)ccc2c(c1)C(C)C(C)O2 N1(C(Cn2c(C)ncc2)=O)CCC2(COCCN2C(c2cccc(F)n2)=O)C1 c1(CC)c(C(=O)NCC(CO)NC(c2nncn2CC)=O)cccc1C(F)F c1(CC(=O)NC2CC3(CN(C(CNS(NC)(=O)=O)=O)C3)C2)cn2c(C)csc2n1 c1(C(N(C2CN(CCC)C2)C)=O)[nH]ccc(=O)c1C.c12c[nH]nc1NC2=O Cc1ccc(-n2cc(C3CCC(CNC(=O)C(C)O)CC3)nn2)c(F)c1F CC1(C)CCC(C(N2CC(C(N3CC(CO)(CF)C3)=O)C(F)(F)C2)=O)CO1 c1(C(O)C(F)(F)F)ccc(NCc2ncc(-c3cc[nH]n3)s2)cc1 C1(NC(CC=C=C)=O)CC2(NC(=O)CSc3ccc(COC)cc3)COC1C2 C1(OC(c2cc(C(C)OCC)on2)=O)CCN(c2cc(C)nn2C)C1=O N1(C(c2n[nH]c(C)c2O)=O)CC(N(C)C(c2cnn(CCO)c2N)=O)C2(CC2)C1 c1(-n2cccn2)ccccc1.S(=O)(=O)(CC1COC1)NC(=O)NCCC1CC1 O(NC(=O)C(CC1CC1)NC(C1CC=CC(O)C1)=O)CC N1(C(c2ncc(C)s2)=O)CCN(C(c2ccc(=O)oc2)=O)C2CC12 S(=O)(=O)(c1ccc(F)c(C(N2CCC(CO)(NC(=O)CSC)CC2)=O)c1F)NC C(C)(CC(C)CC)NC(C1C(CNC(C2(CC=C)COC2)=O)CC1)=O c1(NCCc2n(CC(=O)OCC)c(S)nn2)ncc(C)c(-c2ccccc2)n1 c1(CNCCC(=O)NC2CNCC2O)ccc2c(c1)OCCO2 c1(NC(C)=O)ccc(C(=O)NC(CCCNC(C2(C(C)(C)OC)CC2)=O)C)cc1 c1(C(=O)NC2CCCN(C(C(C)=C3CC3)=O)C2)cccc2[nH]c(=N)oc12 C(=O)(C(C(CC(C)C)OC)N1CC(CSC)OC(C)C1)NCCCCCCCC c1(C(=O)NC2CCN(C(c3ccnc(C)n3)=O)C(C)C2)cc2ccccc2o1 C1(CNC(c2ccc(O)nc2)=O)CC(F)CN1C(c1ccon1)=O C(CC(F)F)(C(=O)NCCc1nn[nH]n1)N(C(C1C(=C)C1)=O)C CC1(CNC(=O)COc2ccc(Cl)cc2)CC(F)(F)CN1C(=O)C(=O)NC1CC1 C(=O)(C1=NOC(c2ccccc2)C1)NCCNC(C=C(CC)C)=O N1(C(C2=NOC(CNC(=O)CCC3CCCOC3)C2)=O)CC2(CNC(=O)OC2)C1 Cc1noc2ncc(C(N3CCC(NC(C4CCn5cnnc5C4)=O)C3)=O)cc12 C1(CC)C(=O)NCCN1C(=O)C(N1CCC(OCCC(C)O)CC1)=O c1(C(N2CC(C(=O)NCc3cc(Cl)ccc3Cl)OCC2)=O)c(F)ccc(Cl)c1Cl C1(C(N(CCCNC(c2cc(N)cc(F)c2)=O)C)=O)CC2COCCN2C1 C1(CCC)CCCCN1C(=O)CN(C(=O)Cc1ccn(C)n1)CCC c1(C(=O)NCC2(COC)CN(C(c3coc(CO)c3)=O)C2)cc(Cl)c(Cl)n1C N1(C(CN(S(N(C)C)(=O)=O)C)=O)CCC=C(C(=O)NC2CC3CC3C2)C1 c1(OCC2CCN(Cc3c(N)cccc3)CC2)ccc(F)cc1Cl N1(C(Cc2nccc(OC)n2)=O)CCCC2C(NC(=O)CN(C)CCO)CC2C1 Cc1cc(N(C(C)(C)CNC(c2nnn(C(C)(C)C)n2)=O)C)nc(CO)n1 C12(C(=O)NCC3N(C(COCC(=O)NC)=O)CC3)CCCCC(=O)N1CCC2 C1(C(=O)NCCCOC=C)CC12CN(Cc1ccc(C(F)F)nc1)C2 C=C(C)CC(C)C(=O)N1CCC(O)(CCNC(=O)C(F)=CC2CC2)C1 N1(C(C(CCC)O)=O)CC(O)(C2CCN(C(=O)CSc3nc[nH]n3)CC2)C1 N1(C(CC(C)OC)=O)CC2(C=C(C(=O)N3CC4(CC(F)C4)C3)CO2)C1 C(C(=O)Nc1ccc(F)cc1C)(C(C)CC1CC1)N(C(CC)C(=O)OC)C C1(C(N2CC(N(C(=O)CCC3OCCO3)C)C2)=O)CS(=O)(=O)CC(=O)N1 C1(C(N2C(C)(COC)CCC2)=O)CC(NC(C2CCCC2(C)C)=O)C12CCC2 CC(C)(O)C#CC(=O)N1CCC(N2CC(NC(=O)CCc3nccs3)CC2=O)C1 Cc1nc(NC(C2C3CC2N(C(=O)Cc2nc(C)sc2C)C3)=O)ccc1Br CC1CCN(C(C2CCCN2N=O)=O)C(C)C1NC(c1cncc(Cl)c1)=O C1(CNC(COCc2cc(C)on2)=O)C(C)CCN1C(c1ccc(C#N)s1)=O C(CC)(CCC(=O)N1CCCC1CCO)NC(C(CC)=CCCC)=O.OC(=N)O c1(OCC)ccc(NC(N2CC(NC(=O)NCc3ccc(F)cc3)C2)=O)cc1 C1(NC(CCOC(C)=O)=O)CC(F)(CNC(=O)C(C2CCCCC2)O)C1 C1(C2(O)CCC2)(CNC(CC2CCN(C(CCC(C)O)=O)C2)=O)CC1 N1(C(C23C(CN(C(=O)OC)C2)C3)=O)CCC2(CCCN2C(=O)CN2CC=CC2)C1 C1(NC(c2ccn(C)c2)=O)CN(C(c2cc3c([nH]2)CCCC3)=O)C2CCCCC12 N1(C(COC(CC)=O)=O)CCC(C=CC(=O)NC2CCCN(CC)C2)CC1 CC1(C)CCn2cc(C(=O)NC34CCN(C(=O)Cc5ccco5)CCC3C4)nc21 c1(C(N(C)CC2CCN(C(C3CCC(=O)O3)=O)C2)=O)ccn(C)c(=O)c1 N1(C(c2nc3ncccn3n2)=O)CCC2(CO)CCN(c3ncns3)CC2C1 c1(N2CCCC(C(=O)NC3C=CCS3)C2)cc(Cl)nc(-c2ccccn2)n1 C1(C(=O)NC2CC(CNC(CSCC(N)=O)=O)C2)C2COCC12 c1(C(=O)NCC2(OCC)CN(C(=O)CCc3cnco3)C2)ccc(C)nc1 C1(NC(CC=CC=C)=O)C=CC(C(N2CCC(C(CC)CC)C2)=O)C1 c1(NC(=O)CC2CN(C(C3CC3F)=O)C2)cccnc1I N1(CC)OCC(NC(=O)C(c2cn(C)nn2)NC(=O)CC(C)COC)C1=O Cc1cnn(C)c1CC(N1CC(CNC(=O)CSCC(N)=O)CC1C)=O C1(CNC(C(C#C)(C)C)=O)COCCN(C(c2cccnc2OCC)=O)C1 CC1(C)CC(c2ccccc2)N(C(=O)C(c2cc(F)cc(F)c2)F)C1 c12nccc(n1)Cc1cn-2nn1.Cn1cc(CC(N2CC(CC3CC3)C2)=O)cn1 C1(NC(C2(CC)CCCC2O)=O)CCN(C(=O)CCN2CCOCC2)CC1OC c1(C(N(CC(C)N(C)C(c2ccc(Cl)cc2)=O)C)=O)ccc(Cl)nc1N CC(C(=O)NC1CCC1C(=O)N(CC(F)Cl)C)=C1CCC1 [N-]=[N+]=NC1CCC(C(N2CCC(O)C2C(=O)NCc2cc(O)ccc2F)=O)C1 C1(NC(C2CCC(C)O2)=O)CC2CCC(C1F)N2C(C1COCCOC1)=O C1(CC=C)(NC(=O)CC(C)C2CC2)CCN(C(C2(C)CCCC2C)=O)C1 N1(C(CNC(CNC(C)=O)=O)=O)CCC(NC(=O)C#CC2CC2)C1c1ccccc1 N1(C(C2(OC)CCSC2)=O)CCCC(C2CC2NC(c2cncn(C)c2=O)=O)C1 C1(C(N(C(CNC(c2scc(C)c2)=O)C2CC2)C)=O)CC(C)CC(=O)N1 c1(C(=O)OC)[nH]nc(C(=O)OCC(N2CCCC2C2C(C)(C)C2(F)F)=O)c1Br N1(C(C2(F)C(C)C2)=O)CC2OCC(NC(c3ccsc3C(F)F)=O)C2C1 N1(C(CCC=CC)=O)CCN(C)CC1CNC(c1cnccc1Cl)=O C1(N(C)C)CCCN(CCC(=O)NCCN(C(=O)Cc2cncn2C)C2CC2)C1 CC(C)CC(C(=O)N(C)CCNC(c1cc2scc(Cl)c2[nH]1)=O)C(N)=O N1(C(c2ccc(-c3nc4c(s3)CCCC4)cc2)=O)CCC(C2(O)CC2)C1 C1(C(N2CCC(CCOC)C2)=O)(NC(=O)Cc2ccon2)CCC(C)(C)C1 C(=O)(CCO)N(CCCO)CCC.C1(N)CC(OCCCN(C)C)C1 CCN=c1nc(C(N2CCCC2CN(C(=O)CC(C)F)C)=O)cc(C)[nH]1 C1(CC)CN(C(C2(CCOC)CCCC2)=O)CC1CNC(=O)COCP(C)(C)=O c1(C(N2CCC(C)(NC(CCOCC#C)=O)C2)=O)cc2c(s1)CCC(C)C2 CCCCCCCCC(C)C(=O)NCC1(CCNC(=O)C(O)CCC2CC2)CC1 c1(C(=O)NC2(C)CCCN(C(C3(C(C)C)COC3)=O)C2)cnc2n1CCCCC2 C1(C(=O)NC(C)C(C)NC(c2cncc(N)c2)=O)(OC)CCCCCCC1 C1(CNC(c2ccc(CC)nc2)=O)COC(C)(C)CN1C(=O)C=C(C)C(C)(C)C c1(C(=O)OC)ccc(Br)nc1CS(=O)Cc1nc(C2CC2)cs1 C1(c2ccccn2)(Cc2nc(CS(=O)(=O)CCN3CCCC3)no2)CCOCC1 CC(C)CS(=O)(=O)CC(=O)NC1CC1NC(C1CC(O)C1)=O C1(C(C)C)CN(C(=O)C(C)C2(O)CCC2)CCN1C(C1CC1C(C)(F)F)=O C(=O)(C(C)(C)c1cscn1)NCC1C(NC(CN2CC(C)C2)=O)CC1 c1(NC(C2OCCN(Cc3ccc(C)cc3F)C2)=O)cccc2nc(O)oc12 S(=O)(=O)(c1cc2sc(=NC(CCO)C3CC3)[nH]c2cc1Cl)NCC(C(=O)O)F N1(C(C(CCC)(C)C)=O)CCC(NC(C2(C)CCCS2(=O)=O)=O)CC(O)C1 c1(NC(C2OCCN(C(C3ON=C(C)C3)=O)C2)C)cc(S(C)(=O)=O)ncn1 N1(C(c2ccc(OCCOCCC)cc2)=O)CC(NC(=O)CC(C)CF)C(C)(C)C1 c1(OCC(=O)O)ccc(CCNC2CCC(NC(c3ccc(Cl)cn3)=O)C2)cc1 c1(C(N2CCC(CNC(CNC(=O)OC)=O)(CC3CC3)C2)=O)c(C)cc(C)nc1C c1(OC)ccc(-c2nc(CC3(C)CC3)nn2-c2ccncc2C)nc1OC c1(C(=O)NC(C2N(C(CSCC)=O)CCC2)C)ncnc2sccc12 c1(CC(=O)N(CCNC(C2CC(CC)C2)=O)C)ccc(OC)c(OC)c1Cl c1(C(N2CCC(CNC(C(CCC)OC)=O)C2)=O)cc(OC)c(OC)c(Br)c1 c1(C(=O)NC(C)CN(C(=O)Cc2ncc(Cl)n2C)C)c(C#N)cnn1C C1(NC(C2CC(F)(F)C2)=O)CC2CCC1N(C(=O)C(c1ccc(F)cn1)(F)F)C2 c1(CC)c(C)cc(C)cc1N.c12ncsc1C(=O)NCCOCCNC2=O C1(CCNC(C)(CCC#N)c2n(CCOC)nnn2)CCC(C)(C)CO1 C1(NC(C(CNC(C2(CC(C)C)CC2)=O)O)=O)CCN2CCC1C2 c1(C(=O)NCCn2c(SCC)ncc2)cc(F)ccc1C(=O)O C(C)(C)(CC(=O)N1CCC(CSC)C1)n1cc(C)nn1.c1(O)cccc(C#N)c1 c1(N(C(CC)=O)C(C)CN(C(=O)C=C(C)C(C)C)C)ccc2nn[nH]c2c1 c1(CC(=O)NCC(C)N(C(=O)C(C)C(C)C)CC)ccc(O)c(Cl)c1 c12cc(on1)CC(=O)NC1CCN(C1)CCCSC2.c1cncn1C1CC1 CC1CN(C(c2ccc(C(N)=O)nc2)=O)CCC1NC(c1cc(O)cc(O)n1)=O c1(N(C)CC2CCN(C(C(CCCC)O)=O)C2)nc(Cl)nc2c1COCC2 C1(CCNC(=O)CC(F)(F)F)CN(C(=O)COC2CCCOC2)CCCO1 Cc1cc(O)cc(=O)n1CCC(=O)NCCC1CN(C(C2(CF)CC2)=O)CCO1 C(=O)(CCCCN)N(C)C.C12C3CC1CN(C3)CCC2=O.C(C)(C)(C)O c1(OCC)ncccc1CN(c1cnc(C(N2CC(NC)C2)=O)cn1)C C=C(C)C(C)(C)C(=O)NCC1CC1NC(C1CCNC1=O)=O Cc1csc2nc(CN3CCN(C(c4ccc(F)nc4)=O)CC3)cc(=O)n12 c1(-c2nnc(C(N3CCC(CC=C)C3)=O)n2CCC#N)cc2c(s1)CCC2 N1(C(c2c(C)coc2)=O)CC2CCN(C(C3CCC(=O)C3)=O)CCC2C1 c1(CC)cccc(CC)c1C(=O)N(C)CC1CN(C(c2cncc(O)c2)=O)C1 CCC(CC)CC(=O)NCCC1CN(Cc2coc(-c3ccc(C)c(C)c3)n2)C1 CCCC(C)(C)CC(=O)NCC(CC(C)C)NC(c1cnn(C2CC2)c1C)=O C=CC1OCCC1N=c1nc2c(ncn2C)c(N2CCN(C(C)(C)COC)CC2)[nH]1 C1(CNC(c2scc(C)c2)=O)CC2CCC1N2C(=O)C(C)NC(=O)NC1CC1 CC(C)C(CCN(C)C(c1occc1C1CC1)=O)NC(=O)C=CCO C1(C(C)(C2CC2)NC(C=CC(C)NC(=O)CCc2cccs2)=O)CCCO1 C(=O)(CC(C(F)F)C(C)(C)C)NCCCN(C(c1ccnc(C)n1)=O)C1CC1 C1(CNC(C2(N(C)C)CCC2)=O)CN(C(C2CCC3(CC3)C2)=O)C2CCCCC12 C1(C(=O)NC(C(C)C)C(C)C)CN(C(c2cccc(CC#N)c2)=O)CCN1C N1(C(=O)CN2CCCNC2=O)CCC2CC2(C(=O)NCCC(F)(F)CO)CC1 C(C)(CCC(=O)NC1CC=CC(O)C1)NC(C(C1CCOCC1)C)=O N1(C(C(C)(C)C2CCC2)=O)CCCCC(CNC(c2ncsc2Br)=O)C1 C12(C(=O)NCCCC(CO)NC(c3cnc(C4CC4)o3)=O)CCCC1CCC2 CC(CC(=O)NCCC1(C)CCN(c2nnn(C)n2)C1)CC(C)(C)C C=CCC(C)(C(=O)N1CCOCC(CCC)C1)NC(=O)NCc1scnc1CC Cc1noc(N)c1C(N1CCCCC1CCN(C(=O)Cc1cccnc1F)C)=O C=CCC(C)C(=O)N1CCOC(CNC(=O)Cn2ccccc2=O)C1 C1(C(=O)NCCC(Cc2ccccc2)NC(c2cc(C)cs2)=O)(CC)CCOC1 N1(Cc2c(C)ccc(C(=O)OC)n2)CCNC(=O)CC1C C1(CC=C)(NC(=O)Cc2coc(C)n2)CCN(C(c2nnn(C)c2C)=O)C1 C#CC1(CO)CCN(C(c2cnc(-c3cccs3)nc2)C(=O)NCCOC)C1 C1(C)(C(=O)NCCC(C)CCNC(=O)CCCc2cccs2)CCCC(F)(F)C1 c1(C(N2CC(NC(C(C)Cc3ccccn3)=O)C(O)C2)=O)nc2c(s1)CCC2 c1(NC(C2N(Cc3c(C)noc3C)CCC2)=O)ncc(Br)nc1CO CC(C(C)(C)CN(C)C)NC(C1CC=CC(NC(C2(CO)CCC2)=O)C1)=O N1(c2cc3nnc(C)n3cc2)CCCC(C)(C)C1C#N c1(SCC)ccccc1C(=O)NC1CN(C(=O)C(C)Cn2ccc(C)n2)C1 c1(C(=O)NCCCOC(C(=O)NC(CC)CC)C)conc1C(C)C c1(C(=O)NC2CN(C(COCC#C)=O)CC2n2ccnn2)ccc(OC)cc1 Cc1c(C(N2CCC2CC(=O)NCCC2(C)CC2(F)F)=O)cccc1O CC(CC(N)=O)C(=O)N(C)CC1CCN(C(=O)Cc2cc(F)ccc2O)C1 C1(NC(C(CCC)NC(c2ncn3c2CCC3)=O)=O)CCc2n[nH]cc2C1 N1(C(C=C(C)C(C)C)=O)CC=CCC1C(=O)NC(CO)C(C)(C)C C12(C(=O)NC3(C)CCCN(C(Cc4nc(C)sc4)=O)C3)CCCCC1OCC2 c1(OC)ccc(Cl)cc1C(N1CC2CC(NC(C3CC(=O)NC(=O)N3)=O)C1C2)=O c1(C(C(=O)Nc2ccccc2)N(C2CCN(CCOC)C2)C)ccc(Cl)s1 C1(CCS(C)(=O)=O)C(=O)N1.CCC(O)CC(=O)N1CCC(c2cncs2)C1 n1(CCCNC(c2cn(C3COCC3CC3CCOC3)nn2)=O)cccnc1=O C(c1ccccc1C)=CC(=O)NC(CNC(CCC(C)SC)=O)(C)C(C)C CC1(C)CC(CO)CN(C(=O)C(C)(CO)NC(c2ccc(C#N)cn2)=O)C1 C1(NC(C2C(C)OC(C)C2)=O)Cc2ccccc2C1NC(c1cc(Cl)n(C)n1)=O C1(C(=O)NC2CC(NC(C3(COC)CCC3)=O)C2)CCOCC1 Cc1cc(Cl)c(C(=O)NC2CCC2NC(C2CC2C(c2ccccc2)=O)=O)cc1N c1(OC)c(C(=O)NC(CNC(c2sncc2C)=O)C(C)C)ccc(Br)c1F c12cn(cn1)C2.C(CC(=O)N(C(C)C(=O)NCC)C)OCC c1(C(=O)NCCCOCCN)ccc(C)c(C)n1.C1(CC(C)=O)(C(=O)OCC)CCC1 N1(C(c2cc(CNC(CCOCCC)=O)on2)=O)CC2CCCC2(COC)C1 C(COC(C)(C)C)(C(=O)NC(C)CC(C)NC(c1cnsc1)=O)N(C)C C(=O)(C(CN(C)C)N(C)C)NC(CC)CN(C)C(C1(C(C)C)CCC1)=O CCCC(C(=O)NCC12CC1CN(C(=O)C=Cc1cccnc1)C2)OCC c1(CC(=O)NC(CC2CN(C(CC(C)OC)=O)C2)C)cccnc1N1CCCC1 N1(C(c2nc(=N)[nH]cc2)=O)CC2(NC(c3cc(-c4ccns4)on3)=O)CCC1C2 n1(CC(N2C(CNC(CCC=C=C)=O)CCCC2)=O)cc2ccccc2n1 C1(CC)CN(C(c2coc(SC)n2)=O)CCC1NC(c1nc(=O)n(C)[nH]1)=O C1(C)(CC)CCC(C(=O)NC2(C)CC(O)(CO)C2)O1.c1(C2C(=O)N2)cccnc1 C1(CNC(c2c(C)c(N)ccc2)=O)(NC(=O)C=C2CCC2)CCC(F)(F)CC1 C(=O)(CCCCCN(C)C)N(CC(=O)NC(C)CF)CCC CC(C#N)CCC(=O)N1CCCN(C(C2(C)C=CCCC2)=O)CC1 C1(NC(C2CC(OCC)C2)=O)CCCC(C(=O)NCC2(CO)CC=CC2)C1 c1(C(N2CC=C(CO)CC2)C(=O)NC)ccc2c(c1)OCC(=O)N2 C(=O)(C(CC1CCCC1)NC(c1nc[nH]n1)=O)NC(C1CC(C)(C)C1)C Cc1cc(N)c(C(N2CC(C3(NC(=O)COCCN(C)C)CC3)C2)=O)nc1C Cc1nc(NC2CCCN(CC3(c4ccc(Cl)cc4)CCC3)C2)nc2ccccc12 c1(C(N2C(C)CC(NC(=O)CSc3ccc(Cl)cc3Cl)C2)=O)csc2ccccc12 N1(C(C(CCSC)OC)=O)CCN(C(=O)C#CC2CCC2)CC1c1cn[nH]c1 C(=O)(C1=CCCC1)N1C(C(=O)NCC(CC)C)CSC1 CCC(CC)CCC(=O)NCCN(CC(C)O)C(c1cnc2c(c1)COC2)=O CC1C(C)N(C(c2nocc2Br)=O)CCN1C(c1ccc(C#N)n1C)=O c1(CCNC(=O)NC(CC(C)O)C)cccc2c1OCCO2 C1(C(=O)NCC2OCCCN(C(c3nc(C)n(C)n3)=O)C2)CCC(N=[N+]=[N-])CC1 C1(C(=O)NCC2(COC)CN(C(C3CC(=O)N(C(C)C)C3)=O)C2)CC1C1CCC1 C1(NC(CCc2c(C)nn(C)c2)=O)CCN(C(c2ccoc2C)=O)C12CC2 c1(C(N2CCC(N(C(=O)CSC)CC#C)CC2)=O)ccc2cc(C)ccc2n1 n1(CC)c(CNC(=O)C(CN(C)C)NC(=O)CC2(C)CCC(=O)N2)cnc1C c1(N2CCN(C(=O)NCc3c(C)[nH]nc3F)CC2)cccc(Cl)c1O c1(OC)cc(C(=O)NCC(C2CCCC2)NC(=O)C(C)n2ccnn2)cc(F)c1 C1(CC)CN(C(=O)Cc2cncc(Br)c2)CCN1C(c1cc(=O)cc(Cl)[nH]1)=O CC1(C(=O)NCCCC(O)C(=O)N2CCC3CC23C)CCCC(=O)N1 C=CCC(CNC(c1cnn(-c2ccccc2)c1)c1nnnn1CC)CC(C)C C=Cc1cnn(C)c1C(=O)NCC1CCC(C)CN1C(=O)CC1CC(C)(C)C1 C(=O)(C1=NNC(=O)C1)N1CC(C(C(=O)N(CCOC)CC2CC2)O)C1 C(CCNC(=O)Nc1ccc(CC)cc1)(C(C)C)OCCNC(C)=O CC(C)CC(F)C(=O)N1CCCCC1C1CCCN(C(=O)C=CC2CCCO2)C1 C1(NC(=O)Cc2cnoc2)CC1C1CCCN(c2cc(C(F)F)ncn2)C1 C1(NC(C2CC=CC2)=O)CCN(C(c2coc(C3CC3)n2)=O)CC(O)C1 CCC(CNC(C1CCN(C(C2C3CC4C(C3)C24)=O)C1)=O)(CC)C(N)=O C1(NC(c2cnco2)=O)CN(C(C23CCCC2C3Br)=O)C2CCCC12 C(=O)(CC(C)(F)F)NCC(C1CCCCC1)NC(C1N(C(CCC)=O)CCC1)=O C1(NC(COCCNC(Cc2cc(C)sc2)=O)=O)CC2C=CC1C2 C1(CC(=O)N(C2CC2)CC2C(C)C2)COCCN1C(c1cc(=O)cc[nH]1)=O Cc1ncsc1C(=O)NCCC(C)NC(c1ncoc1-c1cccs1)=O Cc1cn2cc(C(=O)NCC(C)(C)CNC(=O)Cn3nnc(C)n3)nc2s1 C1(NC(CCCOCC)=O)COC2CN(C(=O)Cc3ccc(C)nc3)CC12 c1(C(=O)NC(CC)CN(C(=O)C(O)CC(C)C)C)cc2c(s1)CCCCC2 Cc1c(F)c(C(N2CC3CC3(C(N3CCCC(O)C3)=O)C2)=O)nn1C C#CC1CC2CCC1N(C(c1cnn(CCNC(C3CCCOC3)=O)c1)=O)C2 C1(OC)CC(NC(=O)CCC(=O)N(C)C)CN(C(c2cn(CCO)nn2)=O)C1 N1(C(c2cn(C)nc2)=O)CC2CC1CC2NC(c1cccn(C2CCC2)c1=O)=O CC(C)(C)C(C(=O)N1CCC12CN(C(=O)CC1NC(=O)CNC1=O)C2)N1CCC1 Fc1ccccc1Cc1ccc(NC(C(F)(F)F)C2CC2)o1 N1(C(CCC(C)SC)=O)CC2CC1CN2C(c1cnn(C(C)C)c1N)=O C(=O)(CCCCC(N)=O)N(CCCNC(COCCC)=O)Cc1ccccc1F c1(C(=O)NCCCC2(NC(C(CC)n3cncn3)=O)CC2)cc(Cl)cn1C N1(CCC(=O)N(CCC(=O)NC(c2ccc(C)s2)C)CC)CCOCC1=O C1(CCC)(NC(c2ccsn2)=O)CCN(C(c2ccc(O)c(Cl)n2)=O)CC1 C12(NC(CCCCCN(C(C(C(C)(C)C)OC)=O)C)=O)CCC(CC1)C2(C)C N1(C(c2onc(CC)n2)C)CCC(NC(C2C(C)OC(C)C2C)=O)CC1C C(=O)(CCC(F)(F)F)N1CC(SC)C(NC(=O)C(C)SCC2CCCO2)C1 N1(C(c2ccn(CC)n2)=O)CC2CCC(C1CC1CCN1C(=O)OC)N2CCSC C12CC(CCO1)NC2=O.C1(CCOC)CCN(C(=O)CNC(N)=O)C1 C1(CNC(C(N2CCC(C)C2)=O)=O)C2CC2CN1C(=O)CN(C(=O)C(C)C)C C1(NC(C2N(C=O)CCC2)=O)CCN(C(=O)CSc2cn[nH]c2)CCC1(F)F Cc1ccc(F)c(C(=O)NCC2CC2C(=O)NCc2nn[nH]n2)n1 c1(CC(N2C(CCOC)CCCC2)=O)cc2ccccc2n1C C(C(CC(C)C)C(=O)NC1CCCCC1F)OC.C1C(=O)NCCS1 c1(C(=O)OCC)noc2c1CN(C(=O)NC1CCCC13CCC3)CC2 C12(C(=O)NCC(C)CNC(c3cc(C(F)F)ncn3)=O)CC(C)(CO1)C2 Cc1nn(C)c(Cl)c1C(=O)NC1CCCC1CNC(=O)CN1C(=O)CCC1=O N1(C(c2c(C)nc(O)cc2)=O)CC(NC(C2C3CCCC23)=O)C(C2CC2)C1 N12CCC3(CCC(C3)C(=O)N3CCC3CC1=O)CC2.c1(C(=O)O)cc(Cl)ncn1 N1(C(CSCC)=O)CCCC1(CC)CC.c12ccccc1CNC2=O O=C(CCCC(F)F)NCC1(F)CN(C(c2ccc(C3CCCOC3)cc2)=O)C1 Fc1ccc(-c2ncccc2OCCOC2CCC2)c(F)c1 C(C)(C)(CC(F)C(=O)NCc1cnco1)NC(C(C)NC(=O)OC)=O N1(C(c2cnc(C)s2)C(=O)NCCCF)C2CCC1CC(C(=O)NCC(C)C)C2 N#Cc1nccc2cc(NC(c3ccc(Cl)c(C(F)(F)F)c3)C(N)=O)ccc12 C(=O)(C1=CCC(NC(C2CCCOC2)=O)C1)N(CC(C)(C)C)CCOC CCCCC(=O)C(=O)NCc1nnn(C)c1C(=O)Nc1cccc(CC)c1 C(=O)(CCCC(C)(C)C)NC(CNC(C(C)Cc1ccncc1)=O)CC(F)(F)F C=CCC(CC(C)C)C(=O)N1CCC(N(C(=O)C(CC)(CC)CC)CC2CC2)CC1 N1(C(c2cc(C#N)[nH]c2)=O)CCOC2(CCN(C(C3CC3(F)Cl)=O)CC2)C1 c1(OC)cccc(Br)c1C(N1CCN(C(=O)Cc2ccccc2Cl)C(CO)C1)=O n1(CC(=O)NCCNC(C(CN(C)C)c2ccccc2)=O)ccc(Br)cc1=O C(C(C)(O)C(=O)NC1C=CC(CC(N2CCC(C)(O)C2)=O)C1)OC C1(CCC(=O)NC(C#C)(C)C)CCCCN(C(=O)C(CC(C)C)N(C)C)C1 C1(NC(=O)OC(C)(C)C)CC2CCC1CC2C(=O)Oc1cccc2cncn12 N1(C(CCOCC#C)=O)CCC(=CCNC(=O)C(F)=CCC)CC1 CCCCC(C(=O)NCC(C)N(C(=O)C(F)(F)CC)C1CCCC1)NC(N)=O C1(C)(C(N2CC(NC(CC3C=NN(C)C3=O)=O)C3(C2)CC3)=O)CCS(=O)(=O)CC1 C1(CNC(CC(C)(C)SC)=O)CCN(C(c2cnc(N(C)C)cn2)=O)CC1(F)F C1(C(N2C(C(C)NC(=O)CC3CC3C(F)(F)F)CCC2)=O)CCc2ccccc2C1 C1(NC(C(COCC)N=[N+]=[N-])=O)CCCCC1N=c1[nH]ccnc1F.C(C)=O C(=O)(C1CCCc2scnc21)N1CC2(CN(C(c3cc4c(s3)CCC4=O)=O)C2)C1 N1(C(C(CC)N(C)CC)=O)CCC2(CC1)CC2C(N1CC(N2CC(F)C2)C1)=O C1(C(=O)NC(C(=O)NC2CN(CC)CC2C)Cn2ccnn2)CC(C)(C)CCO1 C1(NC(c2ccc(CCC)s2)=O)CN(C(=O)CSC(C)C)C2(CCOCC2)C1 c1(C(N(CC(CC)NC(=O)C#CC2(C)CC2)C)=O)cccc(Br)c1Cl C1(CC)(NC(=O)CCCOC(C)C)CCCN(C(C2(C(=O)N(C)C)CC2)=O)C1 C(=O)(C(C#N)C(C)(C)C)N1C2(CC(COC)C2)CC1.C1(=O)CCCO1 N1(C(C=C(C)C)=O)CC(F)(F)CC1C(=O)NCCCC1(O)CC1 N1(C(C2CCC(CNC(C(C=C=C)C)=O)C2)=O)CC2C3CCC(C3)C2C1 C(C(C)(O)CNC(=O)COCCc1ccccc1)NC(C1C(COC)C1)=O C(=O)(C(CNC(C1COCCC1C)=O)C(C)(C)C)NCc1cncc(CC)c1 c1(C(N2CC(C(=O)NC(CCOC)(C)C)C(O)CC2)=O)cnn2cccnc12 c1(C(C)=O)cc(C(=O)N(CC(C)NC(c2ccc(CC(N)=O)cc2)=O)C)oc1C Cc1cc(NC(N2CCN3C(=O)NCC3C2)=O)cc2cccnc12 C1(NC(c2ncc(CC)cn2)=O)CC1C1CCN(C(=O)CC(C)(C)C)CC1 O=C(C1=C(Cl)CCC1)NC1CCC(CNC(c2cc[nH]c2)=O)C1 N1(C(CC2(C)CCC2)=O)CCN(C(=O)CCC2CCC2)C(C(C)(C)C)C1 c1(C(=O)NC(CCNC(C=C(C)C2CC2)=O)(C)C)cc(C(F)(F)F)c(C)s1 CC(N=[N+]=[N-])C(=O)N(C)CC1CCCCN1C(=O)CCCC1CC1 CCC(O)C(C)C(=O)NC1(COC)CN(C(=O)C2=CCCS2)C1 C1(NC(CCCOCC=C)=O)CC(OC)CN(C(=O)C(C)CC)C1 Cc1cc(C(=O)N(C(Cc2cn[nH]c2)C(=O)NC2CCSC2)CCO)nn1C N1(CCC(=O)NC(CN(C(CSCC#C)=O)C)(C)C)CCc2ccccc21 C1(NC(C(C#C)(C)C)=O)CCC(C)(C)CC1CNC(=O)Cc1ccc(O)c(F)c1 C1(O)(CNC(C(C)OC)=O)CCN(C(c2ccc(C(=O)NC(C)C)cc2)=O)C1 C1(NC(c2cc(C)c(C)s2)=O)CCCN(C(=O)CCc2ncc(F)cn2)CC1F c1(OC)cc2ccccc2cc1C(=O)NCCN(C(C1CCNC1=O)=O)C1CC1 O=C(N=c1cc(-c2cccs2)[nH][nH]1)c1cnccc1-c1ccc(OC(F)(F)F)cc1 C(=O)(C(C)C(C)NC(c1oc(CNC(C2CC(=O)C2)=O)nc1C)=O)OC Cc1cc[nH]c(=N)c1C(=O)NC1CC(NC(=O)CS(C)(=O)=O)C12CCC2 C(c1ccc(Cl)s1)=CC(=O)N(C)CCN(C)C(c1c[nH]nc1O)=O c1(CNC(C2CCS(=O)CC2)c2n(C3(C)CC3)nnn2)ccnc(F)c1F C1(NC(C(CCC)O)=O)Cc2ccccc2C1NC(=O)CC(C)(C)C1CC1 c1(OCCC(=O)N)ccc(Cl)cc1.C1(NC(CN(C(C)C)C)=O)(COC)CCC1 C1(CNC(c2cnc3nccn3c2)=O)CN(C(c2ccc[nH]2)=O)C2COCC2O1 C(CC(=O)N1CC(OC(F)F)C1)N(C(=O)C(C)N(CC)CC)CC#C N1(C(c2c(C)nc(CC3CC3)o2)=O)CCCC(NC(=O)CCC2CC2)C(F)C1 C1(NC(C2C3CC4C(C3)C24)=O)CC2CC(C1)N(C(c1ccn3nncc3c1)=O)C2 c1(OC)cc(F)c(F)cc1C(=O)NCc1cnc(OC)nc1 N1(C(C2=C(C)CCC2)=O)CC2CC(CNc3ncnc(C(C)(C)C)n3)CC1C2 C(N=c1[nH]c(=NC)[nH]c(=NC2COCC2O)[nH]1)C1N(CCC)CCCC1 C(=O)(C(F)CCC(C)(C)C)NC1(C(=O)NC(CCC(=C)C)C)CC1 C(CO)(C(C)(C)CO)NC(C1C(C(C)NC(C2C=CCCC2)=O)C1)=O c1(N2CCC(CC(=O)NC3CC(=O)NC3=O)C2)ccn2nccc2n1 C1(NC(CCN(C)CCO)=O)COC2(C1)CN(C(c1ccns1)=O)C2 C=CC1(CNC(=O)C(Cc2cnc[nH]2)NC(C2CC=CC(O)C2)=O)CCOCC1 CCC(C(=O)N1CC(CNC(=O)CN2CCCC2=O)C2(CCC2)C1)C(F)(F)F C=CC(C)(CC)C(=O)NCCN1CCN(C(c2sc(C3CC3)nc2C)=O)CC1 CC1=NN(C)C(=O)C1CC(N1CCC(NC(C2COCCO2)=O)C12CC2)=O C1(C(N(C2CCN(C(=O)Cc3cccc(SC)c3)C2)CC)=O)(CF)CCOCC1 CCCC(O)C(=O)NCC1(C(=O)N(CC(C)COCC)C)CC=CC1 C(=O)(N=c1ccn(CC2CC2)[nH]1)c1cc(CNC(C2CC3(CSC3)C2)=O)sc1 c1(C(N2CC(C(C(=O)NCC3CCC3CO)OC)C2)=O)csc(Cl)n1 N1(C(c2c(C(C)C)ncs2)=O)CCC(CNC(C2(O)COC2)=O)C(C)C1 C(=O)(C(C)(C1CCCC1)NC1CCC1)N(C(C)C)CCNC(=O)OC(C)(C)C C1(C(=O)NCc2c(CC)nco2)CCCCN1C(c1ccc(OC)s1)=O N1(C(C(C=CC)O)=O)CC(O)CC1(C)C(=O)NOCc1ccccc1 Cc1cc(OCC(=O)NCC23CC2CN(C(=O)CC2CC=CC2)C3)ccc1NC CC1(C)OC(=O)NC1CNC(=O)NC1(Cc2ccccn2)CCOC1 C(CCC(C)C(c1nnnn1CC1CCOCC1)NCCNC(=O)OC)=CC c1(CNC(C(CC)(C)OC)=O)ccc2c(c1)CCC2NC(c1cscc1F)=O CC1OC2CCC1(NC(=O)Nc1ccccc1-c1ccccc1I)C2 Nc1cccc(CNC(c2ccc(-c3ccncc3)nc2)=O)c1 N1(C(C(C)OCC(C)C)=O)CCCC1(C)CNC(=O)CNC1(C)CCC1 C(=O)(C(CO)C(C)(C)C)NC(C1(CNC(C2CCN(CC(C)C)CC2)=O)CC1)C C(N=c1[nH]c2c(c(=NC3CCC4CC34)[nH]1)CCCC2)c1c(Cl)nccn1 c12cc(no1)CNC(=O)C21CC1.c1(OCC)cn[nH]c1.c1(C)nccs1 C(N=c1[nH]c(=NC2CCCCC2C#N)c2ccccc2[nH]1)C1C(C)(C)NC(=O)O1 c1(C(=O)NC(CC(C)C)CNC(=O)CC2CC(C)OC2C)cccc2cnnn12 c1(C(=O)NCCCC(C)(C)NC(COC(CC)C)=O)nc(C)ccc1Br C(C#Cc1cn(CC2CC(F)(F)C2)nn1)NCC1C(C)CC(=O)N1 c1(CCS(C)(=O)=O)ncc2c(n1)CCN(C(c1c(F)cc(Br)cc1Cl)=O)C2 N1(C(Cn2ccc(C)n2)=O)CCC(F)(CNC(C2CCN2S(C)(=O)=O)=O)C1 N1(C(C(CCC)OCC)=O)CC(N=c2[nH]cnc3cnn(C)c23)C1 C1(CNC(C(C)(c2ccco2)NC(CCSC)=O)=O)C2CCCCCC12 CN1CCCC(O)(CC(=O)NCC(C)(CO)NC(c2ccnc(C(F)F)c2)=O)C1 c1(C(=O)NCCOCCNC(C2(CC(C)(C)C)CC2)=O)cc2c(s1)CCC2=O Cc1cc(Br)cc2c(C(=O)NCC3(O)CN(C(=O)C4=CC=NC(=O)C4)C3)coc12 N1(C(C(C)C2CC2)=O)CC(F)(F)CC1C(=O)NCC=CC1CC1 Cc1cc(C(=O)NC2CCCC23CN(C(C2CCN(C)C2=O)=O)C3)c(O)nc1C Cc1ccc2sc(C(=O)NC3(CNC(c4ccc(Cl)cc4N)=O)CC3)cc2c1 C1(C(=O)NCC2CC(NC(CSCCC#N)=O)C2)CCCCC1N=[N+]=[N-] c1(CC)nc(C)sc1C(=O)NC1CC(F)(CNC(c2ccccc2Cl)=O)C1 c1(CCC(=O)N(C)CC2(NC(=O)CC3CCCCC3)CC2)ccccn1 N1(C(C2(OC)CCCCC2)=O)CCCCC(NC(C2OCCOC2(C)C)=O)C1 C1(CN(C)CC)CCN(C(c2sccc2CNC(=O)C(C)NC=O)=O)C1 C1(CNC(C2C(COC)(COC)C2)=O)CN(C(=O)Cc2cc[nH]c(=N)c2)CCO1 N1(C(C(COC)OC)=O)CC(C(=O)NC2CCN(C)C2)C2(CC2)C1 c1(C(N(C(CNC(C=Cc2n(CC)ccn2)=O)C2CC2)C)=O)ncc(Cl)cc1Cl C(=O)(C(=O)CC(C)C)N1C(C(CNC(C2CC(C)(CC)C2)=O)(C)C)CCC1 N1(C(c2c(OC)nsc2OC)=O)CC(C)(C(N2CCOC(CO)C2)=O)CC1(C)C C1(CNC(=O)CCC(F)F)CN(C(c2nncs2)=O)CC(C(F)(F)F)O1 C1(CNC(c2c(C(C)(C)C)ncs2)=O)C2CN(C(c3cc(Br)n[nH]3)=O)CC12 c1(N(CC(=O)NC(C2(O)CN(C(C(COC)O)=O)C2)C)C)ccccc1[N+](=O)[O-] c1(CNC(c2c(C(C)C)ocn2)=O)cccc(NC(C2CC2(C)C(F)F)=O)c1 CN1CCCCC(NCC2CCCN(c3cc(N4CCCCC4)ncn3)C2)C1 Cc1cc(CNC(=O)COC2CN(C(C3(CO)CC34CCC4)=O)C2)cc(C)n1 C(=O)(C(C)(C)CC(=O)OC(C)(C)C)N1CCN(C(C(CO)OC)=O)CC1C N1(C(c2c(C)cco2)=O)CC(NC(c2sc(C)c(C)c2C(N)=O)=O)CC(O)C1 CCCCCC(=O)NCC(N1CC(CNC(=O)C(C)CC2CC2)C(C)C1)=O C1(C(N(CCCNC(=O)Cc2csc(S)n2)CC)=O)COCCN1C C=CCC(C(=O)N(CC(=O)N(C(CC(C)C)C(=O)NC)C)C1CC1)C(C)C c1(OC)ccnc(C(=O)NCCC(C(C)C)NC(c2cccc(N)n2)=O)c1OC Cc1cnc[nH]c1=NCCC1CCCN(C(=O)C(O)C(C)C)C1 N1(C(C(CC(C)C)NC(C)=O)=O)CC2CC(C1)N(c1ncc3ccnc-3[nH]1)C2 C1(C(=O)N(CC(C)CO)C2CC2)CCN(C(=O)CCOCC2CC2)O1 C(=O)(C(C)(C)CC(=O)N1CCCC(N(C(=O)CC2(C)CCCO2)C)C1)OC N1(C(C(C)C)=O)CCCC2(CCCN2C(c2cnn3c2N(C)CC3)=O)C1 C1(C2(O)CCCOC2)(C(=O)NCC2CCN(C(=O)CC3CCOC3)C2)CC1 N1(C(=O)C=Cc2cc[nH]n2)CCC(N=c2c(Br)c[nH]cc2[N+](=O)[O-])(CO)C1 C1(C(=O)NCC2(CSC)CCC2)CCN(C(=O)C2(C)CC2(C)C)O1 c1(C(=O)NC2CC3(CC(NCc4ccc(OC)nn4)C3)C2)cc(Br)c(O)c(Br)c1 c1(C(=O)NCC2CCC(NC(C(C)=C3CCC3)=O)C2)cc2cc(C#N)ncc2[nH]1 C(=O)(CC(F)(F)C(F)F)N1C(CN(C)C(C2CC2C(C)(C)C)=O)CC1 n1(CCNC(Cn2cc(CCC)nn2)=O)cc(S(C)(=O)=O)cn1 C1(C(N2CC(C(C)NC(CCC(C)O)=O)OCC2)=O)NC(=O)OC1(C)C Cc1cc2c(C(N3CCC(C)(CNC(=O)C(C)O)C3)=O)nccn2n1 N1(C(CNC(=O)OCC)=O)CC(NC(c2csc(C(C)(F)F)n2)=O)C2(CCC2)C1 C1(C(=O)N(CC(C)C#N)CC2(CC(=O)OCC)CC2)CCCC1F C1(CC(C)C)CCCN(C(c2ccc(CC3NC(=O)NC3=O)cc2)=O)C1 C12(C(=O)OCC)CCN(C)CC1CN(C(=O)Nc1ccn3nccc3c1)C2 C1(C(=O)NCCC2CCN(C(C(C)NC(C)=O)=O)C2)C(=O)ON=C1C CC(CCc1nc(-c2ccc(F)cc2)nn1Cc1cccc(Br)c1)C(C)(C)C CC(CS(C)(=O)=O)C(=O)NCc1cccc(NC(=O)CCC2CCCN2C)c1 C1(C(=O)NCCc2cc[nH]n2)(OC)CCN(C(=O)Cn2nnc(C)n2)C1 N1(C(C(C)(C(C)C)OC)=O)CCC2(COCCO2)C1 N1(C(CC2C(C)OCC2)=O)CCCC(C(=O)NC2CC(Cl)C2)CC1 C1(NC(C=Cc2cc(OC)ns2)=O)COC2(CCN(C(C3CCCN3C)=O)C2)C1 C(=O)(C(F)(F)C(F)(F)C(F)(F)F)NC1C(CNC(CCCCOCCC=C)=O)CC1 CC(CCOc1ccccc1)C(=O)NC1CC(NC(=O)Cn2cnnc2)CC1O N1(C(CSCCOC)=O)CCCC(C(N2CCC(C)(C)C2C)=O)CC1 C=CC1CN(C(=O)CC(CC2CC2)NC(C2CCC2C#N)=O)CC1O c1(C(N2CCOCC2c2ccc(CN(C)C)o2)C(=O)NCCC)ccncc1C c1(C(=O)NC(Cc2ccc(Br)cc2)C(=O)O)ccc(NC(C2CC2)=O)cc1F C1(NC(C2(OCC)CCOCC2)=O)CC2CC1N(C(C1CC(F)C1)=O)C2 Cc1cc(C(=O)NC2CC3(C2)CC3C(N2CCOC(C)(C3CC3)C2)=O)cc(C)n1 N1(C(C(C)N2CCCC2)=O)CCCC(O)(CNC(C2(C)CC=CC2)=O)C1 c1(C(=O)NC(C)C(CO)NC(c2ccc(Cl)o2)=O)ccccc1Br CC1CCN(C(c2cc(-c3cnn(C)c3)on2)=O)CCN1C(C1CCCCC1)=O c1(C(=O)NC(C)CCCNC(=O)C=Cc2cc[nH]n2)cccc(-n2cnnn2)c1 N1(C(c2n(C)c(C#N)cc2)=O)CCC2CCCC(C1)N2C(C1SCCCS1)=O c1(C(=O)NC(C2CCOC2)CNC(c2nncc(OC)c2)=O)cc(O)ncc1F C1(C)(CC(=O)NCCCC(C)NC(=O)CCn2cc(Cl)cn2)CC(F)(F)C1 Cn1cc(Br)c(C(N2CC3(CCN(C(=O)C(C)(O)C4CCC4)C3)C2)=O)cc1=O N1(C(Cn2ncc(C#C)c2)=O)CCN(C(c2cncc(CO)c2)=O)C(C(F)F)C1 C(=O)(C(C)c1ccsn1)N(CCCNC(C1(C(F)(F)F)CC1)=O)CC C1(CC)CN(C(C2C3CCC(F)C23)=O)CC1C(=O)NCC1CN(CC)CCO1 C1(NC(C2CC(C(F)(F)F)(OC)C2)=O)CN(C(=O)CCn2ccnn2)CC1O c1(CC)nc(C)n(C)c1C(N1CCC(O)(c2cn(Cc3ncon3)nn2)C1)=O c1(C(C(=O)NCC2CC2CNC(c2cncnc2C2CC2)=O)=O)ccc(Cl)cc1 N1(C(c2c(C)cn(C)c2)=O)CCCC2C1CCN2C(C1CN2CCN1C(C)C2)=O C1(C(C)(C)C)CCCCC1C(N1CC(NC(=O)Nc2ccccc2)C1)=O C1(C(N2CCC(CC)(CC)C2)=O)CN(C(c2cc(C#N)c[nH]2)=O)C(C)(C)C1 c1(C(N(C)CC2CCCN2C(C2CC23CCCC3)=O)=O)cnc(O)c2ccsc12 C1CCCC1(C)OC.n12cnc(n1)C(=O)CNC(=O)C2.C1CCC2(CC2)O1.CC C(=O)(CC(COC)COC)N(C1CCN(C(=O)CC2CCOC2=O)CC1)CC#C O=C1CC(C(=O)N(CCCN=[N+]=[N-])CCO)N(C(C2C=CCS2)=O)C1 C=C1CCC(C(=O)N(CCC(=O)N2CC(CN=[N+]=[N-])C2)CC2CC2)CC1 CC(C)CCC(C)NC(C1(NC(=O)C=CCN2CCC2)CCCC1)=O N1(C(C=Cc2c(C)ccnc2)=O)CCC(NC(=O)Cc2cn[nH]c2)CC(C)(C)C1 C(C1=Cc2ccccc2OC1)NC(c1cccc(CCC=C)c1)=O C(=O)(CCCC(C)(C)C)N(C)CCOC1CCc2nnnn2C1 C(=O)(C(C)C(F)(F)F)N(C1CCN(C(c2c(CC)ocn2)=O)CC1)CC1CC1 C1(NC(c2ccncc2C2CC2)=O)CCCCC1NC(C1CC1CF)=O c1(C(=O)NCC2C3CN(C(C(CC)C(C)C)=O)CC32)c[nH]c2cccc(F)c12 N1(C(CCOCCNC(CCCC(CC)=O)=O)=O)c2ccccc2CC1C N1(C(c2ccc(CC)cc2)=O)CC(NC(=O)CCn2cc(C)cn2)CC(O)C1 c1(C(N2CCC(N(CCCC(C)c3ccccc3)C)CC2)=O)c(C)nc(C)n1O N1(c2ccnc(CC)n2)CCC(C2CC2)(CNC(c2cnc(C3CC3)s2)=O)C1 c1(OC)ccccc1CC(C)=CC(=O)OC1(F)CC1(F)F c1(-c2cccc(C(N(c3ccccn3)CCCC)=O)c2)nnc2n1CCC2 c1(OC)ncc(C(=O)O)cc1C(=O)NC(C(=O)O)C1CCCC1 c1(NC(CC)=O)oc2ccccc2c1C(=O)O.c12ccccc1N1CCCCC1C2 C(=O)(C1CNC(=O)c2ccnn21)NC(C)(C)Cc1ccc(Br)cc1 C1(CNC(C(CC2CCCCC2)OC)=O)C2CN(C(c3ccc(F)cn3)=O)CC12 C1(CNC(c2c(C(C)C)nns2)=O)COCCN(C(c2nncn2C)=O)C1 C1(CC(=O)NCC2(NC(C(c3ccccc3)SC)=O)CCC2)CSCCS1 c1(C(N2CC3C(NC(CCCC)=O)(CC3)C2)=O)ccc2c(c1)nc(O)n2C1CC1 C(=O)(C(C(C)(C)O)NC(C12CCC(CC1)C2)=O)N1CC(CC(C)C)C1 C1(CC)CN(C(c2cc(C3CC3)ns2)=O)CCC1NC(=O)CCC1CC1C(C)C Cc1cc(Br)c(C(=O)NCC2CN(C(=O)CCCC3CCC3)C3CC23)s1 C1(CSC)CC(N=c2cc(NCCc3ccccc3C)nc(C(C)C)[nH]2)C1 Cc1ccn2c(C(=O)NCC3CC4CCC34)cnc2c1 c1(C(=O)NC(CC=C)CNC(c2cncc(CC)c2)=O)nc2cc(O)ccc2[nH]1 c1(OC)cc(NC2CC(NC(=O)C(n3cc(Cl)cn3)C)C2)nc(OC)n1 C12(NC(C3CCCC3)=O)CC(CNC(c3cnc(C4CCCO4)s3)=O)(C1)C2 c1(C(=O)NCC2(O)CC(NC(C(C)NC(=O)NC)=O)C2)c(Cl)c([N+](=O)[O-])nn1C c1(NC(C2(C)N(C(CC3N(C)CCC3)=O)CCC2)=O)cccc2cncn12 CCC(C(=O)N1CC(F)(CNC(=O)CCSc2ccc(F)cc2)C1)C(C)C Cc1cc(C)c([N+](=O)[O-])c(C)c1C(N1CC(NC(=O)C(O)C2CCC2)C(C)C1)=O N1(C(C(C=C)(C)C)=O)CCC2C(NC(c3ccccc3OCCC)=O)C2CC1 N1(C(C(CCC)NC(C)=O)=O)CCC(NC(=O)C(C)=C(C)CC)C(C)C1 C(c1ccoc1)=CC(=O)NC1CC(F)(CNC(=O)Cc2c[nH]nc2Br)C1 n1(CC)ncc2cc(C(=O)NCCN(C)C(C3CCC4CC3CO4)=O)c(C)nc12 c1(CCC(=O)NCCC2COCCN2C(=O)CCOC2COC2)ccc(F)cc1F C(=O)(N=c1nc2c(I)cccn2[nH]1)Nc1c(Cl)cc(C)nc1 c1(C(N(C2CCN(C(=O)C(C)(C)c3cncs3)C2)C)=O)cc2n(c1)CCCC2 C(C)(C(=O)N(CC(C)CNC(c1cn[nH]c1)=O)C)NC(COC)=O N1(C(c2c(Cl)cn(CCC)n2)=O)CC(NC(C2CCCC2)=O)C(S(C)(=O)=O)C1 C1(CC)C(NC(=O)C(C2CC2)OC)CCCN1C(=O)NC1CCCCCC1 N1(C(C=C(C)CNC(=O)Cc2nnnn2C)=O)CCC(=C(F)F)CC1 c1(C(=O)NC(C2CCN(C(Cc3c(CC)cccc3)=O)C2)C)cc(C)ncc1C N1(C(Cc2ccc(C)cc2)=O)CC2CC1CCC2NC(=O)CC1CC2CC2C1 CC(C)C(C)(O)C(=O)NC1CN(C(c2cc(C#N)cs2)=O)CC1n1ccnn1 c1(C(=O)NC2(CC#C)COC2)sc(F)cc1I N1(C(C=C(C)c2ccco2)=O)CCC2CC2(NC(=O)Cc2ccc(Cl)nc2)CC1 c1(CNc2cncc(C(N(C)CCc3cccc(Cl)c3)=O)c2)ccc(F)nc1F C1(C(N2C(CC)CC2)=O)C2CCCC2CN1C(c1coc(CO)c1)=O C(C(CC)(CC)NC(C1CC(O)C1)=O)NC(CN(CC)CC)=O CCC(C)CCC(=O)NCC(C)(C)C(=O)N1CCCC1CN(C)CC CCCCC(CC(=O)NCc1nccc(C)n1)NC(C1CC2C=CC1CC2)=O n1(CC(N)=O)cc(NC(C2CCN2C(=O)CC2CC2)=O)cn1 CN1CCC(CC(N2CCC(CF)(NC(c3cnccn3)=O)C2)=O)C1=O c1(CCC)ccccc1C(=O)N(CCC(C)NC(c1cccc(C)c1)=O)C C1(C(=O)NCC2CCCC(CNC(C(C(C)C)O)=O)C2)CN2CCCC2CO1 C(=O)(CC(C(F)(F)F)n1cccn1)NCC(CNC(c1cncn(C)c1=O)=O)OC CC1CN(C(c2cnn(Cc3ccccc3)c2)=O)CC1CNC(=O)C#CC(=O)O c1(CNC(=O)N(C2CCCCC2)Cc2ccccc2)ccc(C(F)C(F)(F)F)cc1 C1(CC)(CNC(=O)CCC2CCCN2C(c2cc(C3CC3)[nH]n2)=O)CCC(=O)N1 C1(C#N)(CC)CCN(C(C2C=CCCN2C(C2CC3CC3C2)=O)=O)CC1 N1(C(CCCN(C)C(C2CCCN2c2ccccc2)=O)=O)CCN(CC(=O)O)CC1 C1(NC(c2cc(OC)ns2)=O)COCCC1C(=O)N(C1CCCC1(F)F)C C1(NC(C(CC)NC(c2ccco2)=O)=O)CC2C1CCN2C(=O)CC1OCCO1 N1(C(C(CC#C)(C)NC(c2cnn(C)n2)=O)=O)CC2CC(C1)N(C)C2 C(=O)(C1CCc2c[nH]nc21)N(CCNC(c1c(C)cccc1)=O)CC1CCCC1 c1(OCCOC)cccc2c1CN(c1nccc(=NCC3(CSC4CC4)CC3)[nH]1)C2 N1(C(CC2C(C)=NOC2=O)=O)CCCC(C)(NC(=O)C2=COCC2)C1 C(C(CC(C)C)C(=O)NCC(C(C)(C)C)NC(C1CC(=O)C12CCC2)=O)OC c1(CNC(C2(F)CCN(Cc3cc(C)cc(F)c3)C2)=O)cc(F)c(Cl)cc1C C1(C(=O)N(C(C)CNC(=O)CSc2cscn2)CC)(OCC)CCOC1 C=CCCCCCC(=O)NC1CC(F)(F)CC1NC(=O)C(N1CCOCC1)C c1(C(=O)NCCCCC(C)NC(C2CC(C)OC2C)=O)nnc2ccccc2n1 C=CC(C(=O)N(CCC(=O)NC1CCC(O)C1)C)OC N1(C(C(CC)n2cncn2)=O)CCCN(C(c2cc(C)c(C)nc2C)=O)C(C)C1 c1(C(N2CCC(C)(CNC(C(CC)C#N)=O)C2)=O)cc(Br)cc2scnc12 C1(CC)C(=O)N(C)CCN1C(=O)C(=O)NC1CCOC12CCOC2 C1(C(F)F)(OC)CCN(C(=O)C(CNC(=O)OC(C)(C)C)CC2CCCCC2)C1 c1(C(=O)NCC(c2ccc(OC(C)C)cc2)O)ccc2c(c1)CCN2 CC1(C)CCC(C(=O)NCCCOCCC(=O)NCCC(Cl)Cl)CO1 N1(C(C(CC(CC)CC)F)=O)Cc2n[nH]cc2C1C(=O)N1CCCC1CC(N)=O CCC(C)C(O)C(C)C(=O)N1CCCC1CCC(=O)NC1CC=CC1 C(=O)(C(C)P(C)(C)=O)N1CCC(CN(C(C=CC(=O)OCC)=O)C)C1 N(C(=NCCCC1CCCO1)NCC1CCCCO1)CC1CCS(=O)(=O)C1 Nc1ccc2c(NC3CCC(=O)N4CCCCC34)nccc2c1 C1(NC(=O)OC)CN(C(=O)CCOCc2ccccc2)CC(C)(O)C1 C(=O)(C(CC)C(F)(F)F)NC1(CC=C)CCN(C(=O)Cc2ccn(C(F)F)n2)C1 c1(NCC)cnn(C)c1CC1(CC(=O)NC(c2n(CC)ccc2)=O)CC1 C(=O)(CC(O)(C(F)(F)F)C1CC1)NCC(C(C)C)NC(CN(C)CC)=O c1(C(N(CCOCCN(C(c2c(CC)con2)=O)C)C)=O)cc(Br)ccc1C C(=O)(CCCCCC#N)N1CC(C)OC(CCNC(=O)COCC2CC2)C1 Cc1ccc(C(=O)O)cc1C(N1CC2C(C(N3CCCC(O)C3)=O)C2C1)=O CC1=C(C)CC(C)(NC(=O)C(CO)NC(=O)CCc2ccccn2)CC1 Cc1[nH]c2ncnc(N(C)Cc3nnc(S)n3C)c2c1C C=C1CCN(C(c2c[nH]nc2OC)=O)C(C(=O)NCC#CC)C1 C(C(C)(CC(C)C)NC(c1cncn1C)=O)NC(COCCCC(C)C)=O C1(NC(c2cc(SC)oc2C)=O)CCN(C(c2ccn(C(C)(C)C)c2)=O)C(C)C1 C(=O)(CCCCC(F)F)NC(c1cccc(C)c1)CNC(c1csc(C)n1)=O C(C(=O)N1CCN(C2(NC(=O)CCP(C)(C)=O)CC2)CC1)(C(C)C)n1ncc(C)c1 CCC(C)CCC(O)CC(=O)N(C)CCN(C(=O)COc1cccc(F)c1)C C12CCCN(C1)C(=O)C(c1ccccc1)NC(=O)CC(=O)N2.C(C)(=O)NCC c1(C(=O)NC2CC3CN(c4nc(SC)nc(C)c4)CC32)cc(C#N)ccc1Br N1(C(C2N(C)CSC2)=O)CCN(C(c2ccc([N+](=O)[O-])s2)=O)CC1CCO C1(NC(N2CC(OC)(NC(=O)OC(C)(C)C)C2)=O)C2Cc3ccc(Br)cc3C12 N1(C(c2c(COC)cco2)=O)CCC(NC(C2(CO)COC2)=O)C(C)C1 N1(C(c2c(C)ccc(O)c2)=O)C2CCC1CN(C(c1cnn(C)n1)=O)CC2 N1(C(CC2CC(OC)C2(C)C)=O)CC2(C1)CN(C(=O)CC(C)C(C)(C)C)CCO2 C1(C(N)=O)(C(=O)NCC(O)CCC2CC2)CN(C(=O)CCC2CC(OC)C2)C1 n1(CC(=O)NC2C(CNC(C3C(C)COCC3)=O)C2)cnc2ccccc2c1=O C1(C(=O)NCC2(O)CC(CNC(C34CC5CC3C4C5O)=O)C2)CCCC12CCC2 C1(C(N2C(C(N3CC(n4ccnn4)C3)=O)CSC2)=O)CC2CCCCC12 c1(NC(C2C(C(=O)Nc3c(Cl)ncc(OC)c3)C2)=O)ncc([N+](=O)[O-])cc1I c1(C(N2CCC(O)(CCNC(=O)C3=CCCCC3)C2)=O)cc(Cl)cc2ccccc12 C1(n2cc(C(C=C)(C)O)nn2)CN(C(C2(C)COCCO2)=O)CC1O CCCC(C(=O)NCC1CCCN1C(C)CN1CCCC1)NC(C)=O CC1(CNC(=O)CCSC(F)(F)F)CCN(C(c2cnc(C3CCCO3)s2)=O)C1 c1(C(=O)NCCC(C)N(C(=O)CN(C)C(=O)C2CC2)C)ccc(F)cc1OC(F)F N1(C(C2N(C(=O)NC)CCC2)=O)CC2(CC(NC(=O)CCC(C)C)CO2)C1 c1(C(N2CCN(C(CCC(C)OC)=O)C(CCO)C2)=O)ccc(Cl)c(C)c1Cl c1(NC(C2CCCN(C(CSc3c(C)ncs3)=O)C2)=O)nc(N(C)C)nc(=N)[nH]1 c1(C(=O)NCCC(CNC(C2CCC(C)(C)OC2)=O)O)cc2cccnc2[nH]1 C(CNC(c1cc(F)ccc1OC)=O)(C(C)C(C)C)NC(c1ccn(CC)n1)=O C1(CC)C(NC(=O)CSC(F)F)CCN1C(C1CCCC1SC)=O c1(C(=O)NC2CCC(CNC(C3(SC)CC3)=O)C2)cc2cc[nH]c(=O)c2s1 N1(C(c2c(C(C)C)occ2)=O)CCC(NC(=O)CC2CC(C)(C)CCO2)C(C)C1 c1(NC(C(CC)N2CCCCC2)=O)ccc2c(C(=O)NC3CC3(C)C)ncn2c1 C(=O)(C#CC1(C)CC1)N(C(C)(C)CCNC(C1CN(C2CCOCC2)C1)=O)C c1(C(C(=O)NC)N(C)C(C2CC(CO)C2)C)ccc(Br)cn1 c1(NCC(CN2CCN(C(C)C)CC2)(C)C)nccc(=NC2CCCOC2)[nH]1 N1(C(c2n(C)c(S)nn2)=O)CC2CC(NC(c3csc(C4CC4)n3)=O)CC1C2 N1(C(c2cc(C)nn2C)=O)CCN(C(c2cc(CO)oc2C)=O)C(CO)C1 N1(C(c2ccc(CC(=O)OC)cc2)=O)CCN(C(=O)C(C)CCN(C)C)C(C)C1 C1(C)(C(=O)NCCN(C(c2cnc(C3CCCCC3)s2)=O)CC)CC(C(C)C)=NO1 N1(CC(N2CCC(C(C(=O)NC(C3(CO)CCC3)C)C)C2)=O)CCC(=O)CC1 N1(C(C2(CC)CC2(F)F)=O)CCC2(CC1)CC2NC(c1ccc(C2CC2)nc1)=O C(CN=c1[nH]c(N2CCOCC(C)C2)nc2c1CSC2)n1c(C(C)C)nnc1 CC1(C)C(CNC(C2(CO)CCN(C(c3ccc[n+]([O-])c3)=O)C2)=O)C1(C)C C1(CNC(c2cc(CNC(C3(SC)CC(=O)C3)=O)ncc2)=O)CCCC(C)(C)O1 CC(C)(C)C(C)(C)C(=O)N1CCC(NC(c2cccc(I)c2)=O)C(F)C1 C1(CC(N2CCC(CCO)CC2)=O)C2CCCC2N1C(=O)Cn1cc(CO)nn1 c1(CN(C(CCC2(C)CC2)=O)CCNC(C2CC2Cl)=O)cccc(Cl)c1 CC(CCC(=O)NCC1CCCC1NC(c1ccncc1C1CC1)=O)S(C)(=O)=O c1(CNC(C(CNC(c2c(CC)con2)=O)N(C)C)=O)cccnc1O Cc1cc(C#N)sc1C(N1CCC(N(C)C(C2CCC(C)(C)OC2)=O)C1)=O N1(C(c2c(CC)ncs2)=O)CCOCC1C(N1CCOC(COC)C1)=O Cc1cccc(C=CC(N2CCC2CNC(=O)CN2CCC(CO)CC2)=O)c1 CCC(C)CCC(=O)NCC(CNC(c1ccnn1CC(F)F)=O)C(F)(F)F C(=O)(C1CCCn2ccnc21)N1C(CN(C(CC(CCC)C)=O)C)CCC1 c1(C(N(CCNC(c2cc(Cl)cs2)=O)CC)=O)cnn(C)c1C(C)=O N1(C(C(CC)n2cncn2)=O)CCC(CCC(N2C(C)CC2(C)C)=O)CC1 c1(C(=O)NC2C(C)CCN(C(C3(C(=O)OC)CC3)=O)C2)occ2c1CCOC2 CCC(C(C)(F)F)NC(=O)C(C1CCCO1)NC(c1cc(OC)nn1C)=O N1(C(CC=CC)=O)CCC(CO)C(NC(c2snc(C)c2N)=O)C1 N#CCC(C(F)(F)F)NC(N1CCC(C(F)(F)F)CC1)=O c1(C(=O)NCC(=C)C)n[nH]c2cccc(-c3ccc(O)c(NC(C)=O)c3)c12 C=CC1(CC(=O)NC2CCCC(NC(=O)Cc3ccc(C)cc3)C2)CCCCC1 C=C=C(C)CC(=O)NCCN(C(=O)CCCc1ccc(Cl)cc1)C Cc1cc(C#N)ccc1C(N1CCCC1CN(C)C(C1CC(C)(F)C1)=O)=O C=CCCCCCC(=O)NCC1(F)CC2CCC(C1)N2C(=O)Cc1ccco1 c1(CSCC)ccc(NCc2n[nH]cc2C)cc1O c1(C(=O)NCC(CNC(CN(C)S(N)(=O)=O)=O)(C)O)ccn2cccc2c1 c1(CC)cnoc1C(=O)NC1CCCC1NC(c1nnc(C)s1)=O c1(CC(=O)NCCC2CCC(NC(C3(N(C)C)CCCC3)=O)C2)cnccc1Cl c1(SC)cnn(CO)c1.C(=O)(C(F)(F)C1CC1)N1CC(OCC(=O)NCCS)C1 C12(CNC(C3=NOC(C)C3)=O)CCCC1N(C(=O)CC1(C)CC1)CCC2 c1(CC(=O)NCC(CN(C(c2n(CCOC)ncc2)=O)C)O)noc(C)c1C#N c1(C(=O)NCC(C2CCCC(C)C2)(C)O)ccc(OC(F)F)c(F)c1 C1(NC(c2ccc([N+](=O)[O-])s2)=O)CN(C(=O)CC(F)F)C2(CCOC2)C1 C1(OCCC)CCCN(C(C2(CC)CCCN2C(c2ccc(C#N)[nH]2)=O)=O)C1 Brc1cn2c(CNC(c3nnnn3C3CCC3)C3CCCC3)cnc2s1 c1(OCC(=O)NC2C(NC(CSCCN(CC)CC)=O)C2)ccc(Cl)c(Cl)c1 N1(c2[nH]c(=NCCc3c(C)nn(C)c3O)[nH]c(=N)n2)CC(C)(C)C12CCOCC2 C#Cc1ccc(C(=O)NC(Cn2cccn2)C(=O)NC2CC(OC(C)C)C2)nc1 N1(C(c2n(C)c(S)nn2)=O)CC2CCCCC2(CNC(=O)CC2(O)CCCC2)C1 C1(NC(=O)C(F)C2CCOC2)CN(C(Cc2c(C)nccc2)=O)CCC1CO C1(C(C)C(=O)NC2CCN(C(=O)CCC=C(C)C)C2C)CCC2(CC1)OCCO2 c1(-c2cn(CCCC(=O)NC3(O)CCC(COC)C3)nn2)cc(C)c(F)c(F)c1 c1(-c2ccc(C(N3CCC(C(C(=O)O)OC)CC3)=O)cc2)ccc2cnccc2c1 N1(C(c2c(C)oc(Br)c2)=O)CC2CC(NC(C3CCC3(F)F)=O)CC2C1 C=C(COC(C)(C)C)C(=O)N1CCC(N(CC(C)C(C)C)C)C1 c1(C(N2CC(C)C(CNC(=O)CSCCC(F)(F)F)C2)=O)cccn(C)c1=O C(=O)(C1CC(C)Nc2ccccc21)NCCCNC(c1c(C(C)=O)cccc1)=O Cc1cc(=NC(=O)C(=O)N2CC(NC(=O)C=C3CCCC3)CC2C)[nH]o1 C(=O)(CC(C)C(C)C)N(C(CNC(c1c(C(=O)OC)nccn1)=O)C)C C1(CCNC(C(C)OCCCC)=O)COCCN1C(c1nn(C)nc1C)=O N1(C(CC(=O)NCC)=O)CCC(NC(c2ccoc2C)=O)C(O)C1 C(=O)(C1=CCCCC1C)N(CC)CC1CCN(C(=O)CC2(C)CCOC2)CC1 C(C(C)(C(=O)N1CC2CC1CS2)NC(=O)CSCCCOC(F)(F)F)SC CC1CN(C(=O)N(C)CC2CCO2)c2ccc(Br)cc2O1 CC(CCC(=O)NC1CCCC(C(=O)Nc2cccc(C(F)F)c2)C1)N(C)C c1(OCC#C)ccc(C(=O)NCCN(C(C2CC2Cl)=O)CC)cc1CC c1(C(=O)NCCC(C)N(C(=O)C2=CCCC2(C)C)C)cc2sccc2n1C c1(OC)cc(C(=O)NC(C)C(C(C)C)NC(c2ccc(=N)[nH]c2Cl)=O)ccc1Cl c1(CN(C2CN(C(c3c(C(F)(F)F)cccc3Cl)=O)C2)C)c(O)cccc1O Cc1ccc(S(N)(=O)=O)c(C(N2CC3(CCN(C(C4CC4[N+](=O)[O-])=O)C3)C2)=O)c1 C(C(CC(=O)O)C(F)(F)C(F)(F)F)NC(c1c(C)c2c([nH]1)cccc2)=O C(=O)(C1CN(CCC2CCC2)Cc2n[nH]cc21)OC O=S(=O)(c1ccc(NCC2C3CCCOC23)c(F)c1)N1CCCC(F)CC1 C1(NC(C(C)SCC)=O)(CNC(=O)CC(C)(C)CC)Cc2ccccc2C1 CC(C)CC(C)(CN(C(C1C2CC1N(C(=O)OC(C)(C)C)C2)=O)C1CC1)CC c1(OC)cc(C(N2CC(OC)CC(NC(c3c(C)n[nH]c3C)=O)C2)=O)cc(Cl)n1 Cc1ccc(C(N2CC(N3CCN(C(C4(O)CCSCC4)=O)CC3)C2)=O)nc1C C(CCCCC(=O)N(C)CC1CCCN1C(C1CC2CC1CO2)=O)SC c1(C(C)NCCNC(=O)NCC(C#C)O)ccc2ccccc2c1 N1(C(CC=C)=O)CCC(C)(C)C(CNC(=O)CC(C)c2ccncc2)C1 C1(CNC(Cc2cnc(C)[nH]2)=O)CC2(CO1)CN(C(=O)Cn1cc(CO)nn1)C2 C1(n2cc(C(CCC)NC(=O)Cc3ccc(Cl)cc3)nn2)CC2C=CC1C2 C(CC(C)CCNC(c1c[nH]c(Br)c1)=O)NC(C(C1CCC1)OC)=O Cc1cc(CNC(C2SCCS2)=O)oc1C(=O)N(CC(C)C)CCO C(=O)(CCCCCOC)N(C1CCN(C(=O)C=CCOCCO)CC1)CCC N1(C(C2N(CCC)CCCC2)=O)CC(NC(c2ccn(CC)n2)=O)C(C2CC2)C1 N12CCCC(C1)C2=O.CC1(NC(=O)CN2CCCC2)CCC1 c1(CC(=O)N(CCC(C(C)C)NC(C(C)SCC)=O)C)ccc(F)cc1Cl c1(OC)cc(CCNC(C2CC2c2ccc(C(F)(F)F)cc2)=O)ccc1C c1(CNCC(CC)n2cccn2)cc(S(N)(=O)=O)c(C)nc1C(=O)O Cc1cc(C(=O)NC(C)(C)CCNC(=O)CC2CC3C=CC2C3)cc(N)c1 N1(C(CSC)=O)CCCC2(CNC(C3CCC(C(N)=O)CC3)=O)CCCC12 C(C(=O)N=S(=O)(c1ccccc1F)C(F)F)c1cccc(OC)c1 N1(C(=O)NCCc2cccc(Br)c2F)CCC2CS(=O)(=O)CC2C1 C(=O)(C1=CCCN(C(C2C3CCC(F)C23)=O)C1)NC(C)C(C)n1cncn1 c1(OC)nc(C(=O)NC(C)CNC(c2cn(C3CCOC3)cn2)=O)ncc1F CCC(CC(=O)NC1CON(CC)C1=O)NC(=O)Cc1ccccc1 C(=O)(C(C)(C)CC(C)(C)C)NC1CN(C(c2cncc(OC(C)C)c2)=O)C2C1C2 c1(OC)c(C(N2CCCC2(C)C(=O)NCC2(C(F)(F)F)CC2)=O)cccc1F c1(CS(=O)(=O)NC2(C)N(C(C(N3CCCCC3C)C)=O)CCC2)ccnc(F)c1 c1(CC(=O)N(C2CCCN(C(C(C)OCCC#C)=O)C2)C)ncc(F)cc1F c1(C(N2CC(C)N(C(=O)CS(C)(=O)=O)CCC2)=O)cccc2nc(O)ccc12 N1(C(C(CNC(C2N(CCC)CCC2)=O)OC)=O)CC2CC(O)CC2C1 C1(C(N2CCCC(c3ccccn3)C2)=O)CCn2cnnc2C1 C12(OCC)CCC(C(N3CCCC(CN(C)C(c4nnsc4C)=O)C3)=O)(CC1)C2 N1(C(C2C(C)CCO2)=O)CCC2CCCC12C(=O)Nc1cncnc1O N1(C(=O)OC(C)(C)C)CCC2(CC1)CC2(CO)NC(=O)Nc1ccc(Cl)nc1 C(=O)(C1CNc2ccccc21)N1CCC(NC(C(C)C2CCC2)=O)C(CO)CC1 CCCCCC(O)C(=O)N1CCN(C(c2ccn(CC)n2)=O)CC1CCCC c1(C(N2CCC(OC)(CNC(C3CCCC3O)=O)C2)=O)cc(F)ccc1F c1(C(=O)NCC(CCNC(=O)Cc2cncs2)O)nccc2ncccc12 C1(NC(COC2CCN(C)CC2)=O)CC2CCCC(C1)N2C(=O)CC(F)(F)F c1(C(=O)OC)c(F)cc(Cl)c(C(=O)NC(c2cn(C3CCOC3)nn2)C)c1Cl C12CCC(C1)N2.c1(C(=O)NCC(C)(C)C)cc(C2CC2)ns1.C1C(=O)NN1C C1(C(=O)NC2CC(NC(c3c(N(C)C)nccc3)=O)C2)C2CC3CC(C2)CC1C3 c1(C(N2CC(NC(C3C(C#C)C3)=O)CC23CCC3)=O)cncc2cc(Cl)ccc12 c1(C(=O)NCCCn2cc(C(C)OC)nn2)cc2sc(C)cc2s1 c1(C(=O)NC(C2CN(C(c3cc(CC4CCC4)on3)=O)C2)C)nc(Cl)cs1 C1(C(=O)OC)CCC(n2nnnc2C(c2coc(Br)n2)NCc2ncnn2C)C1 C=CC(C)(CC)NC(C1CC1C(F)(F)F)=O C(c1ccccc1)(C(F)(F)F)=CC(=O)NCC1CC(NC(C2CC2(F)Cl)=O)C1 C1(CNC(C(COC)C)=O)CC(NC(c2cc(N3CCCC3)ncn2)=O)C(O)C1 C#CCCCCCCCC(=O)N1CCN(C(C2CCC(C)(C)C2)=O)CC1 CC1CCN(C(c2cnc(Cl)s2)=O)C1C(=O)NC(C)Cc1nc[nH]n1 N1(C(C(C)SC)=O)CC(F)CC1CC(=O)NC12CC(F)(C1)C2 C1(CC(=O)NC(CN(C(=O)CCCOC(C)(C)C)CC)C)C=CCCC1 CC1=CCN(Cc2cccc(C(=O)NCC3N(C(N)=O)CCC3)c2)CC1 C1(O)(CNC(CCN(CC#C)C(C2C[SH](CCC)C2)=O)=O)CCCC1 Cc1cc(NC(=O)C(=O)NCC2CSC2)n(C2CCC2)n1 N1(C(=O)CN2CCOCC2)CC2CCC1CN2C(c1cc(Cl)ncc1Cl)=O C(=O)(CCCC(=O)NC1CCOC1C(=O)NCc1ncc[nH]1)N(C)C Cc1ncccc1C(N1CCC1CC(=O)N(C1CC1)Cc1ccoc1)=O c1(-c2nc(-c3ccc(C(C)=O)nc3)on2)ccc(C(F)F)c(C)c1 c1(CCC)ccc(C(N2CCC(C(C)NC(c3[nH]cnc3C)=O)C2)=O)s1 N1(C(C(C2(OC)CCSC2)(F)F)=O)C2CCC1CC(Oc1sc(C)cc1Cl)C2 c1(N(S(=O)(=O)CC2CCCC2)C)cccc(NC(c2cccc(Br)c2)(F)F)c1 C(=O)(CCC(CF)CF)Nc1c(C(N2CCN(C(=O)NC)CC2)=O)c(C)ccc1 N1(C(CCC=CC(C)C)=O)CCC2(CC1)CN(C(c1cc3c([nH]1)CCOC3)=O)C2 S(CS(=O)(=O)CCOCC)NC(c1cn(CC=C)nn1)C1CC1 c1(C(N2CC=CC(NC(CN(CCOC)C)=O)C2)=O)cnc2c(c1)CCCC2 C(c1ccc(C)nc1)=CC(=O)NC(CC=C)CNC(c1ccc(C2CC2)nc1)=O c1(N2C3C(NC(C=CCCC)=O)(CCC3)CC2)c(F)cc(C#N)cc1[N+](=O)[O-] Cc1cc(C#N)ccc1C(=O)NCCC(C(C)C)NC(c1cnc(O)c(F)c1)=O C1(NC(C(c2cccc(C)c2)F)=O)CC2CC1N(C(c1[nH]nnc1C)=O)C2 Cc1cc(Cl)cc(Cl)c1OCC(=O)NCCC1COCCN1C(=O)C(C)CO c1(NCC2(C)CCC(NC(C=C(C)C)=O)C2)cc(C)c([N+](=O)[O-])cc1Br C(=O)(C1=CCC(F)(F)CC1)N1CCC(NC(c2n(CC)ccn2)=O)CC1C n1(CCC)nc(C)cc1C(=O)NC1(CC(=O)NC2CCCC2(C)CO)CCC1 c1(OC)cc(C(=O)NC23CC(C2)N(C(=O)CC(C)c2ccco2)C3)c(F)cc1N C=CCCCCCCCC(=O)NCC(CC=C)NC(=O)CC12CC(C1)C2 c1(C(C)C)ccc(NC(C2CN(C(=O)CSc3nnnn3C)CCO2)=O)c(Br)c1 N1(C(C2OCC(C)C2)=O)CCOC2(CCN(C(c3nc(C4CC4)no3)C)CC2)C1 CC(C)(C#N)CCC(=O)NCC1(NC(C2OCCCO2)=O)CC1 c1(C(N2CC=C(CNC(c3c(C)nsc3)=O)CC2)=O)cccc2cc[nH]c12 C1(NC(C(C2CCOC2)OC)=O)CCN(C(c2cc(N)c(F)cn2)=O)C(C)C1 C1(CC)CN(C(c2cncn(C)c2=O)=O)CCN1C(c1cnc(CC(C)C)s1)=O CCCC(CCCNC(=O)COCC(=O)NC)NC(c1sc(NC(C)=O)cc1C)=O N1(C(CC(OCC)OCC)=O)C2CC1CN(C(c1ccc(O)cc1C)=O)C2 c1(CC)ccc(C=CC(=O)NCC2(NC(=O)C(C3CCCCC3)OC)CC2)cc1 Cc1cc(C(=O)NCCc2n[nH]cc2C(=O)NCC(C)(F)F)no1 CCCC(CCCNC(C1CCc2cc(Br)ccc2C1)=O)N=c1nc(C(C)C)[nH]s1 c1(NC(c2cnn(CC(F)(F)F)c2C2CC2)=O)cc2cccc(O)c2[nH]1 C(C(CC(F)(F)F)NC(=O)C(C1CCCCC1)F)NC(c1cncc(O)c1)=O CCCCCCC(=O)N1CCCCC(NC(c2cnc(NC(C)=O)o2)=O)C1 N1(C(c2c(C)nco2)=O)CCN(C(C2CCC(=O)N2C)=O)C(CC(F)(F)F)C1 c1(C(=O)NCC2(C)CCCN(C(C3(C)C=CCC3)=O)C2)ccc2c(c1)CCOC2 C1(C(N(C)Cc2cccc(CNC(C3CC(F)C3)=O)c2)=O)CC2C(C1)C2(F)F CC1CCC(NC(=O)Cc2ccc(Cl)c(Cl)c2)CN1C(c1cc(O)ccc1N)=O C(=O)(CS(=O)(=O)C(C)C)N1CC(CC)C(NC(=O)C=Cc2cccc(C)c2)CC1 C1(C)(CCNC(C(COC)N(C)C)=O)CCN(C(c2c[nH]nc2F)=O)C1 C(=O)(C1CCc2nccn21)NC(c1ccc(C)cc1)CNC(=O)C=CC1CC1 C1(CCO)(NC(c2cn(CC)nn2)=O)CCN(C(=O)C(C)NCCC(C)C)CC1 C(=O)(C1=CC(O)C(NC(c2cnc3ccccn23)=O)C1)N(CC=C)CC=CCC c1(SC)ccc(Cl)c(C(N2CCC(CNC(=O)C(CO)NC(=O)C(C)C)C2)=O)c1 N1(C(CCOCC(C)C)=O)CC2CC1C2NC(C1CC(CC(C)(C)C)C1)=O Cc1cc(NC(c2csc(CNC(c3c[nH]c(=N)c(C)c3)=O)c2)=O)c(C)cc1F c1(C(=O)NC2C(C)CN(C)S2(=O)=O)ccc2c(c1)C1(CCCC1)CN2C(=O)CC#N C1(NC(c2c(OCC)cccc2)=O)CN(C(=O)C=C(CC)CC)CCC1CO C1(C(N2CC(COC)(CNC(C3CC3CC(C)(C)C)=O)C2)=O)CC(=O)NC(=O)N1 CN1CCC(N)(C(N2CCCC2(C)c2nncn2C)=O)C1 C1(CNC(C(CSCC)N(C2CC2)CC)=O)CC2CCC1C2 N1(C(=O)Nc2nccc(COCCOC)c2)CC2CCCCN2CC1C c1(C(=O)NCC2(C(C)NC(C3C(=C)C3)=O)CC2)cnc(C(F)(F)F)cn1 C(=O)(C1=CS(=O)(=O)CCC1)NC1C(NC(CNC(CNC(C)=O)=O)=O)CC1 Cc1n[nH]c(C)c1C(=O)N(CC(N1CC(NC(=O)CSCC(N)=O)C1)=O)C O(NC(=O)C(CN(C)C)NC(=O)Cc1csc(C)n1)CCOCC#C c1(OC)cc(Cl)c(Cl)cc1C(=O)N(C(C)CCNC(C1CCCC(=O)O1)=O)C N1(C(C2N(C(C3CC(=O)C3)=O)CCC2)=O)CCCC2(CCNC2=O)C1 c1(C(N2CC3C(CNC(c4ncn(C)n4)=O)(C3)C2)=O)cc2cccc(F)c2o1 N1(C(C2C(C)C2)=O)CC2(CC(NC(c3cc(-c4cn(C)nn4)on3)=O)CO2)C1 c1(C(N(CCCNC(=O)C=Cc2ccccn2)C)=O)ccc(Cl)c2c1OCCO2 c1(C(=O)NC2CCN(C(C=C(C)C(C)C)=O)CC2C(C)C)cc2c(nn1)CCC2 CCCC(C)CC(=O)N1CC2(CC2)CC1NC(=O)CCNC(=O)C1CC1 c1(-n2c(-c3nc(CC)oc3C)nc(C3CC3C)n2)cc(COC)cc2ccccc12 N1(C(C2(C(C)C)CC2)=O)CCCC(N(C)C(c2cnn(C)c2Br)=O)C1 C1(CNC(CC2(CC)CCC2)=O)CN(C(=O)CN2CC(=O)NC2=O)CC1(C)C c1(-c2cc(CC(C)NC(c3cc[nH]c3)C)no2)ccc(F)cc1F N1(C(CCCOCC)=O)CCC2(C1)CN(C(c1nccc3occc13)=O)C2 C1(CNC(c2c(C)cc(F)s2)=O)CC(NC(=O)Cc2cc[nH]n2)C12CCC2 c1(N2C(=O)CC(C(=O)NC(c3cnn[nH]3)CC)C2)ccc(OC)cc1C CC1(C)C2CC1C(=O)N2.c1(NCC(=O)NCC2CN(CC(F)(F)F)C2)ccccc1 N1(C(c2ccc(C)cc2O)=O)CCC2CCC(NC(=O)C(C)C3CCCO3)C1C2 Cc1nc2ccnn2c(C)c1CCC(=O)NCC(CO)C(F)(F)F C1(c2nnnn2Cc2cccs2)(Nc2cncc(F)c2)CCCN(C)C1 C1(NC(c2c(C)nc(C(C)(C)C)s2)=O)CC(F)CN(C(=O)CN2CSCC2=O)C1 C(CCCCC(=O)N1CC(C(N2CCOC(C3CC3)C2)=O)(COC)C1)SC c1(C(=O)NCCCN(C(=O)CCc2cccc(Cl)c2)CC)cc(C)cnc1F N1(C(C(CC)NC(N)=O)=O)CCC(=CCN(C(C2C=CCC2)=O)C2CC2)CC1 C1(CC(=O)N(CCNC(Cc2cn(CC)nn2)=O)CC2CC2)CCCC(=O)C1 C1(C(=O)NC(C(=O)OC)C(C)C)CC(C)CN(C(=O)CC2C=CCCC2)C1 c1(C(=O)NC2CCC(NC(c3c(CCC)nns3)=O)C2)ccc2c(n1)OCCO2 C12(NC(c3c(Cl)ccc(CC)c3)=O)CCCC1N(C(=O)CCCC1CCC1)CC2 N1(C(CCC)=O)CCCC(NC(=O)CN(C(=O)C(F)=C2CCCC2)C)C1 C1(CNC(C(C2CCCCC2)C)=O)C2CCCC1N(C(=O)CC(C)(C)C1CC1)C2 C1(Nc2cc(NC(=O)NC)ncn2)CCCC2(CCCCC2)C1 CC1(C)CCC(CNC(C2CCSC2)=O)(NC(=O)CC2CCCC(=O)N2)CC1 CC1Cc2c[nH]nc2CC1NC(c1ccc(NC(=O)C(=O)N(C)C)c(F)c1)=O C1(C)(C(=O)NCC2(NC(c3ccnc(CC(C)C)n3)=O)CCC2)CCCNC1=O N1(C(CS(CCOC)(=O)=O)=O)CCC2CN(C(c3ccc(C(N)=O)o3)=O)CC2C1 c1(N2CCC(COC)C2)nnc(-c2ccc(C)o2)n1CCC(C)=O CC1(C)CN(C(=O)CCCCn2cc(CO)nn2)CCCO1.C1(S(N)(=O)=O)(C)CC1 CCC(CC(=O)N1CC2(CCN(C(C3CCC(F)(F)CO3)=O)C2)C1)C(F)F N1(C(c2c(OC)cc(C)s2)=O)CCC2C(NC(=O)C(c3ccncc3C)C)CC12 C1(OC)CC(CNC(=O)CC2CN(C(=O)Cc3cscn3)C2)C1 N1(C(c2cnc(CC)nc2O)=O)C2CCCC1CN(C(C1CCCOC1)=O)C2 c1(C(N2CCC(C(C)(C)NC(C(C)NC(CC)=O)=O)C2)=O)cc(O)nc(O)n1 c1(CC(=O)NCC2(C(N)=O)CN(C(C(C)OCC#C)=O)C2)n[nH]c2c1CCCC2 O(NC(=O)CCOC1CNC1)CCCN(CC(F)OC)C C1(CNC(C(C)CO)=O)(NC(=O)C=CC(C)(C)C)CC(F)(F)C1 N1(C(C2CCC(C)O2)=O)CCCC2(C1)CN(C(=O)CN1CCOC1=O)C2 C1(C(=O)NCCCOCC=C)C(C2CC2)CCN1C(C1CCC1)=O C=CC(C)(C)CCNC(=O)CC1CC(C)N(C(c2cnc(Cl)s2)=O)C1 C1(NC(c2cc(C)cc(Cl)c2)=O)CCN(C(C2CCCSS2)=O)C12CCCC2 C#Cc1ccc(OC)c(C(N2CCC(C)C(NC(=O)Cn3ccc(C)n3)C2)=O)c1 CC(C)CCCCCC(=O)NCC(C1CCCCC1)NC(c1coc(C(N)=O)c1)=O c1(CCC(N2C(C(N(C(C(F)=CC)=O)CC)(C)CC)CCC2)=O)ccc(O)nn1 c1(NC(CC2N(Cc3c(C)cncc3)CCC2)=O)ccc(Br)cc1F C1(C(N(CCCNC(CCCCCC)=O)CC)=O)CCc2c[nH]nc2C1 c1(CC(=O)N(C2(CC(=O)NCC(CC)n3ccnc3)CC2)C)ncc(C)s1 N1(C(C(CC(C)C)C)=O)CC(C(=O)NC2(CN(C)C)CCC2)C2(CCC2)C1 N1(C(C(CC)C(=O)OC)=O)CC2(C=C(C(=O)N(C)CCn3cnnc3)CO2)C1 C1(C(=O)NCC(C(C)C)NC(C2OCCO2)=O)CCN(c2ccccc2Cl)C1=O C1(NC(=O)CCc2cn[nH]c2)CCCC(CNC(=O)CN2CCCCC2)C1 c1(COC)ccc(C(N2C3CCC2CN(C(c2occc2CO)=O)C3)=O)cc1C#N N1(C(c2c(CCC)nco2)=O)CCC(C)(C)C(CNC(C2COCCOC2)=O)C1 CC1(CNC(=O)COCCN(C)C)CCCN1C(=O)Cn1nccn1 c12ccc(c(Br)c1)[nH]c2=O.N1(c2snc(COC)n2)CCOC(C(C)C)C1 Cc1nc(C(N2CCC(C(C)NC(c3ccn(C)c(=O)c3)=O)C2)=O)cc(O)n1 c1(N(C(=O)Nc2ccc(C)cc2)C2CC2)cc(C#N)nc(C)n1 N1(C(CC2CCN(Cc3ncc(C)cc3F)CC2)=O)CCc2cc(F)ccc2C1 C1(CNC(c2cnn(CC)n2)=O)CCC(NC(=O)CCCc2n[nH]c(=N)s2)CC1 N12CCC(C(O)C1)C2=O.Cc1c(C(F)(F)F)n[nH]c1NC(=O)CCSC(F)(F)F N1(C(C)CC(=O)NCCN(C(=O)CC#N)C2CC2)C(=O)NC2(CCCC2)C1=O C1(F)(C(=O)NC2(CNC(=O)COc3cccc(F)c3)CCOCC2)CCCCC1 C1(C(C(=O)NCC(C)NC(=O)CCc2ccsc2)OC)CCCCC1 N1(C(c2cc(F)cc(F)c2)=O)CC2CCCCC2(CNC(C2CC(O)C2)=O)C1 c1(-c2ccc(C)cc2COC)cccc2c(C(N3CC(F)CC3C#N)=O)[nH]nc12 N1(C(CC2CCN(C)CC2)=O)CCN(C(=O)Cc2c(O)ncnc2O)C(CF)C1 c1(C(C)C(=O)NCC2CCCN2C(=O)Cc2nc[nH]n2)nc(F)ccc1Cl c1(C(N2C3C(NC(CCC#C)=O)C(C3)C2C)=O)ccnc2[nH]c(C)nc12 Cc1nn(C)c(S(=O)(=O)NCC(c2cncn2C)=O)c1Cc1ccccc1 Cc1cc(OCC(=O)NCC(C)(CO)NC(=O)CN2CC3CC3C2)ccc1Cl c1(OC)ncc(CCC(=O)NCC2CC(NC(=O)Nc3ccccc3)C2)o1 c1(C(=O)NC(C2OCCN(C(C(CCC)O)=O)C2)C)ccc2c(c1)OCC(=O)N2 C1(C#N)(C(N2CCC(C(C)NC(=O)Cc3cc(F)ccc3F)C2)=O)CC12CCCC2 CC(CC(=O)NCCCN(C)C(c1csc(C(F)(F)F)n1)=O)c1cccnc1 c1(C(=O)NCCNC(C2N(C)C(=O)CC2)=O)cc(Cl)cc(Br)c1 N1(C(C(N2CCCCC2)C)=O)CC(NC(C2(N(C)C)CCCC2)=O)C2CC12 c1(CC=C)ccc(OCC)c(S(=O)(=O)NCCC2(O)CCCNC2)c1 C1(NC(C(CC)(C)CO)=O)CN(C(c2ccc(F)c(Cl)c2)=O)C2(CCOCC2)C1 O=S(=O)(c1ccc(NCc2cnoc2)nc1)NCc1ccnc2c1CCC2 C1(CN(CCCC)C)CCCN(C(C2COCC2(C)C)=O)C1 Cc1cc(C#N)sc1CC1CC(NS(C)(=O)=O)C1.C12CCCC1NC(=O)N2 c1(NCCOC(CC)C)nccc(=NCCCCCNC(C)=O)[nH]1 C(=O)(CC(C)CC(C)C)NCC(CC=C)NC(c1cc2n(n1)CCO2)=O c1(C(N2CCN(C(c3c[nH]c(=N)s3)=O)C3C2C3)=O)cncc2nc[nH]c12 c1(CC)cccc2c1OCCC2N=c1[nH]c(CCCCC(F)(F)F)cs1 c1(CN(C)C(C2(N(C)C(C3CCOC3)=O)CC2)=O)cncnc1 c1(OCC(=O)NCCNc2c(C#N)nc(C)o2)ccc2c(C)cc(=O)oc2c1 c1(C(=O)NCCN(C(c2nc(OC)cc(OC)n2)=O)C)cc(F)cc2nn[nH]c12 Cc1cccc(C)c1NC(=O)CCNC(=O)Nc1cc(O)cc(Br)c1 C=C(C)CC(Cc1cccs1)NC(C1CC1(C)CSC)=O N1(CC(=O)N(CCNC(=O)CC#N)CC)C(C)=CC(C)=NS1(=O)=O C(c1cocn1)=CC(=O)NCCCN(C(=O)C(O)CC1CCCC1)CC C(CCCCN=[N+]=[N-])NC(CC1C(NC(C(C)n2cccn2)=O)CC1)=O C1(O)(C(=O)NC2CC3CN(C(Cc4cncc(C)c4)=O)C2C3)CCC(C)(C)CC1 c1(C(=O)NC(C2CCN(C(C3CCOCC3)=O)C2)C)cc2cccnc2[nH]1 S(=O)(=O)(c1ccc(N2CCC(C)(C)C2)nc1)NCCC(C)N(CCC)CC c1(C(=O)NC2(CC#C)CCC2)coc(CNC(=O)CC(C2CC2)C2CC2)c1 C1(COC(c2cc(C(C)(F)F)n[nH]2)=O)COc2ccccc2O1 CCCC(C)(C)CC(=O)N1CCC(CNC(C2CC3CC3C2)=O)(OC)C1 Cc1cc(C)c(C(=O)NC(CNC(C2CN3CCC2CC3)=O)C(F)(F)F)cn1 c1(C(C)O)ccc(C(=O)NCCC2(NC(=O)CC(C)N3CCCCC3)CC2)cc1 C1(N(C(CSCCOC)=O)C)C2CN(C(=O)C(CC3CC3)CC3CC3)CC12 N1(C(c2nccc(CNC(Cc3ccn(C)c3)=O)c2)=O)CC(C#N)C2(CCC2)C1 Cc1nc(C2CC2)ncc1C(N1CCC(CNC(c2cnn3c2OCC3)=O)C1)=O C1(NCC)CCCC(C(=O)NC2CC(NC(c3ncccc3C(=O)OC)=O)C2)C1 C1(COC)CCN(N2CCC(C3CCCOC34CCC4)CC2)C1 N1(C(C2CC(C)(O)C2)=O)CCC2(NC(=O)Cn3nnc(C4CC4)n3)CC2C1 N1(C(C2CN=CCC2C(F)(F)F)=O)CC2(CCN(C(=O)CCOCC3CC3)C2)C1 c1(C(=O)NC2C3CN(C(C4C(C(=O)OC)C4)=O)C2CC3)cc2nccc(Cl)c2s1 c1(C(=O)NCC(CNC(C2(C)N(C(C)=O)CCC2)=O)(C)O)ccc2nnnn2c1 C1(NC(c2cnn(-c3ccccc3)c2)=O)CCN(CC2CC(N3CC(F)C3)C2)C1 C1(NS(CCCC)(=O)=O)CCCS(=O)(=O)C1.c12nc(cs1)CC(=O)N2 C(=O)(C1OCCc2ccccc21)NC1C(CC)N(C(=O)CC(C)SC)CC1 c1(C(=O)NCC2(NC(C34CCC3C4)=O)CC2)cccc(C2CC2(F)F)c1 c1(NC(c2scnc2-c2ccc(C(F)(F)F)nc2)=O)cc(F)ncc1F C(=O)(C(C(C)(C)C)n1cc(Cc2ccccc2)nn1)NCCC1(C)CNC(=O)N1 c1(C(N2CCC(CN(C)C(c3cnc(C4CC4)o3)=O)C2)=O)cc(Cl)c(F)cc1O C1(NC(CSCC(N)=O)=O)CC2CCC1(CNC(=O)Cc1cc(F)cc(Cl)c1)C2 C(=O)(CS(=O)(=O)CC(=O)NC1CN(C(=O)CC2CCCC2(F)F)CC1(C)C)OC N1(C(C(CC)SC)=O)CCC(F)CC1C(=O)N(CC(OC)OC)C c1(CC)ccc(C(=O)N(C2CCN(C(=O)CCc3ccc(C)o3)C2)CCO)nc1 C1(c2nnnn2CC2CCCO2)(Nc2cc(CC=C)sn2)CC2(COC(C)C2)C1 N1(C(CC2CCC(C)(C)CO2)=O)Cc2nccn2CC(NC(c2cc[nH]n2)=O)C1 c1(C(=O)NC(C(=O)NCC2(CC)CCCO2)c2ccoc2)cc2n(n1)CCO2 CCC(CCC(=O)NOCC(=O)OC)OC1(C(O)CO)CC1 c1(C(=O)NC2CCC(CNC(c3cc(C)n(C)n3)=O)C2)ccc2ocnc2c1 C1(OC)CC(C(=O)N(CC(O)C(C)(C)C)C)N(C(=O)CCOC)C1 c1(OC)ccc(F)c(CN2CCN(S(=O)(=O)CC3CC3)CC2)c1OC N1(C(c2c(OCC)ccs2)=O)CC(NC(c2nc(C)nn2C)=O)C(O)C1 N1(C(c2ncnn2CCC)C(=O)NCCCC)CCC2CC3CC(C2)CC1C3 C1(CC)CCCCC1C(=O)NC(c1ccnn1C)C(=O)N(C)CCOC1CC1 c1(CCC(=O)NCC(CNC(C2CNC(=O)N2)=O)OC)ccc(Cl)c(F)c1 C1(O)(CCNC(C2CC(OCC)C2)=O)CCN(C(C2OCCC2C)=O)CC1 C1(C(=O)NC23CC(CC)(C2)C3)C2C3CCC(C3)C12.c12cc(no1)C(=O)NC2 N1(C(C(C=C)c2ccccc2)=O)CCC(COC)(NC(=O)C(CC(C)C)OC)CC1 N1(C(C(c2cc(F)cc(F)c2)CC)=O)CC(OC)CC(NC(=O)C=CC(C)(C)C)C1 N1(C(c2c(C)nccn2)=O)CC(C)(C)OCC1CNC(C1CSCCS1)=O c1(OC)ccnc(C(=O)NCC2CCCC2NC(C2(C)CCCO2)=O)c1 C1(OCCOC)CCCN(C(=O)NC2(C)CNC(=O)N2)CC1 C1(CC)(CC)CC(C(=O)NCC2CC(NC(=O)CCC3CC3(Cl)Cl)C2)C1 c1(C(C)(F)F)ccc(C(=O)NC2CCCCC2NC(=O)CCc2nc[nH]n2)cn1 N1(C(CC2(C)CC2(F)Cl)=O)CCN(CC2CN(C(=O)CNC(N)=O)C2)CC1 C1(C)(C(N(CCC#C)C)=O)CCN(C(=O)C=CC2(C)COC2)C1 C1(C(N2CC(C(=O)NCCN(CCC)C(C)C)OCC2)=O)CC2CCCC2C1 c1(C(=O)NCC2CCC(NC(C3ON=C(C)C3)=O)C2)c(C)csc1Cl C=CCCCCCCCC(=O)NC1CCCCC1NC(=O)Cc1cncnc1O CC1CN(C(c2ncc(Br)cn2)=O)CCCN1C(c1cnc(O)s1)=O C1(C(C)NC(=O)Nc2nc(C)c(Br)nc2)CCN(S(N)(=O)=O)CC1 C(=O)(CCCC(C)(F)F)NC(CNC(C(COC(C)=O)C)=O)C(C)C C1(CNC(CC(C)SC)=O)CN(C(=O)CC=CCc2ccccc2)C(C)(C)C1 c1(OC)ccc2c(C(=O)N(C3CCN(C(C4(C)CC4(F)Cl)=O)CC3)C)n[nH]c2c1 C1(NC(CCCCC#C)=O)CCCC12CCN(C(c1cnc(CC)s1)=O)CC2 C=Cn1nccc1C(=O)NCc1cnn(C)c1C(=O)N(CC(C)(C)COC)C C1(CC)CC(CC(N2CCC2CNC(c2cscn2)=O)=O)CCO1 C1(CC)CN(C(=O)OC)C(C2CC2)CN1Cc1c(OC)nc(OC)cc1Br c1(C(=O)NC2CC(CNC(CNC(=O)NC)=O)C2)ccc(S(N)(=O)=O)cc1Cl c1(C(N2CC(CNC(C(CC)OC3CCCC3)=O)(OC)C2)=O)cc(F)c(F)cc1O N1(C(C2(COC)CCC2)=O)CCCC(NC(=O)CCc2cnc[nH]2)C1C C1(CC)CCCC(NC(C2(CC)CN(C(c3n[nH]cc3C(C)C)=O)C2)=O)CC1 C1(NC(C(COC)COC)=O)CCCN(C(c2cccnc2)=O)C1C C1(CNC(=O)NC(CC#CC)C)CCC2(CCCCC2)O1 Cc1sc(CC(N2CCCC2CN(C)C(C2CCCS2(=O)=O)=O)=O)nc1C(C)C C(=O)(C(=O)CC(C)C)NCCN.C=C1CC2(C1)C(=O)NC2.C1(C)CCOC1 c1(OC)ccc2nc(C(=O)NCC3CN(C(=O)CC4CCCCC4O)C3)cn2n1 C1(NC(CC2CCCC(C)C2)=O)CN(CC2CCCOC2)CC2(CCOCC2)C1 c1(OC)cc(OC)cc(C(F)C(=O)NC2CCC2C(=O)O)c1.C(C)(C)C C1(C(=O)NC2C(CNC(c3c(C)nns3)=O)CCC2)CCc2nnnn2CC1 C1(CC)CCC(C(=O)NOCC(=O)NCCC2COCC2C(=O)OCC)O1 C1(NC(CC2(C=C)CCCCC2)=O)CC1C1CCN(C(C2CCC(O)C2)=O)CC1 C1(CC=C)(NC(c2cn(CCCC)nn2)=O)CCCN(C(=O)C(C)(CC)CC)C1 N1(C(CCCCOC)=O)CC2CCC1C(NC(c1ncccc1Cl)=O)C2 c1(C(=O)NCCCCS(=O)(=O)CCO)ccc2[nH]c3c(c2c1)CCCC3C C1(CNC(C2CC3CCC2O3)=O)CN(C(c2c[nH]nc2C2CC2)=O)CCCO1 N1(C(c2ccc(NCc3cn(C)nc3C)cc2)=O)CCCC2CN(OC)CC12 C1(C(=O)NCC(C#C)OC)C2CC2CN1C(=O)CCc1ccccc1 c1(C(=O)NCCCC(C)NC(C2C(F)(C(=O)OC)C2)=O)cc(C(F)(F)F)cn1C c1(CC(=O)NC(CCCCNC(c2ccc(OC)s2)=O)C)cccc(F)c1Cl N(C(=NCc1ccccc1Br)NCC12CC(C1)C(C)O2)C(C=C)C C(c1ccncc1)=C(C)C(=O)NCC1(F)CC(NC(c2scnc2C(C)C)=O)C1 C1(NC(CCCc2n(C)c(S)nn2)=O)CC2CC(NC(C3CC(F)C3)=O)CC2C1 c1(C(N(CCCNC(C2CCC(=O)NC2)=O)CCC)=O)cc2scnc2[nH]1 c1(C(=O)NC2(CF)CCN(C(c3c(C)nn(C)c3)=O)C2)ccc(Cl)c(Cl)c1 Cc1ncc(CCC(=O)NC(CNC(c2ccsc2Cl)=O)C2CCC2)s1 CC1(C)CN(C(=O)OC(C)(C)C)C(C)(C(=O)NC2CCC2)CO1.C123CC(C1)(C2)N3 C(C(C)C(C)(C)C)NC(C(CC)N(C)C(c1ccc(COC)o1)=O)=O c1(C(=O)NC(C(C)NC(c2cn(CCC)nc2)=O)C)ccc(OC(C)C)cc1 N1(CC(=O)NCCNC(CC2CC(C)(C)OC2)=O)CCN(S(C)(=O)=O)C(=O)C1 N1(C(c2onc(C)n2)=O)CCC(C2CCN(C(c3c(C)nsc3N)=O)CC2)CC1 c1(C(=O)NCCCNC(C(c2ccc(Cl)cc2)OC)=O)cccc(Cl)c1N CC1CC=C(C(=O)N2CCC(F)(C(=O)NOCC(CO)C(C)C)C2)CC1 C12CC3CCCC3N1C(CC)C(=O)NC2.c1(SCC)cccc(C(=O)NCC)n1 N1(C(c2cncc(C)c2)C(=O)NCCOC)CC(C)C(C)C1C C(=O)(CCC(=O)N(CCCCCCNC(=O)C(F)(F)C1CCC1)C)N(C)C C1(NC(c2cnc(C)[nH]c2=N)=O)CN(C(C2(C#N)CC2)=O)Cc2nccn2C1 c1(C(=O)OCC)ccnnc1C(=O)N(CC(C)(C)NC(C1(C(F)F)CCC1)=O)C C1(CNC(CCCN(C(C)=O)C)=O)CN(C(=O)CCOC2CC2)C2CC12 C(=O)(C#CC1(CC)COC1)NCC(CNC(=O)CCc1nncn1C)OC C(=O)(C(C)S(N)(=O)=O)NCCC1(NC(C(n2c(C)ncc2)C)=O)CC1 C1(CNC(c2c(C)cn(C)n2)=O)CCN(C(c2ccc([N+](=O)[O-])o2)=O)C12CC2 C12(CNC(c3n(CC)ccc3)=O)CC1CN(C(=O)CCc1nc(CSC)no1)C2 CC1C(=O)CCC1CC(N1CCCC(C(N2CCC(O)(C(N)=O)C2)=O)C1)=O O=C(CCS(=O)(=O)C(F)(F)F)N1CCC(O)(c2ccccc2C(F)(F)F)C1 c1(CC(=O)N(CCCNC(C(N2C(=O)CCC2=O)C)=O)C2CC2)ccc(Cl)cn1 C(C(CNC(C1(C)CCCCO1)=O)C(F)(F)F)NC(CC(=O)NCC#C)=O C12(CNC(c3cc(C)no3)=O)CCCC1N(C(=O)CN1CC3C=CC1C3)CCC2 c1(C(=O)NCC2CC(C)N(C(c3cnn(C)c3Cl)=O)C2)n[nH]c2ccc(Cl)cc12 C1(C(=O)NC(C2CCCO2)(C)C)CC2CCCC2N1C(=O)CC1NC(=O)NC1=O Cc1sc(C(=O)NC2CC(NC(=O)C(C)Cn3ccnc3)CC2O)nc1O C1(C(N2CCC(N(C(=O)CC3CNC(=O)C3)CC)C2)=O)CCC2(CCCC2)C1 c1(C(=O)NC(CNC(c2nc(C)sc2)=O)C(C)C(C)C)cc(Cl)cc2c1CCC2 O=C1CNc2ncc(-c3ccc(NCc4cc(Cl)cnc4O)s3)c(=O)cc2N1 C1(NC(C2CC(C)(C)N(C(=O)C=CCN3CCCC3)C2)=O)CCC2CCCC1O2 c1(C(=O)NC2CCN(C(c3c(SCC)cncc3)=O)C2)ccnc2ncsc12 N1(C(c2c(C)cc(F)cc2)=O)C2CCC1CN(C(=O)CSC(F)(F)F)C2 C=CCC(C(=O)NC(C1CCCN1C(c1cnc(O)n1C)=O)(C)C)C(C)C C(CCCC(=O)N1CC(F)(F)CC1C(=O)NCCc1cn(C)nn1)(OC)OC C1(NC(=O)NCC2CCCC2N2CCCC2=O)CC2(CCC(CO)O2)C1 C=CC(C)CCNC(=O)C(C)N(C(=O)CC1(CC)CCC1)CC CC1CN(C(c2cc(F)ccc2O)=O)CCN1C(=O)CCC1CC(C)(C)CO1 C1(CNC(C=CC=CCC)=O)C2CN(C(c3cnn(C)c3C)=O)CC12 n1(C(C)C)cc(-c2cn(C(C)CNC(C3CCC3C#N)=O)nn2)cn1 c1(C(N2C(C(=O)Nc3c(OC)ccc(C)n3)CC(O)C2)=O)ccc(Br)c(F)c1F N1(C(CC2CCN(C(C(C=C)(F)F)=O)CC2)=O)CCC(C)C(O)C1 Cc1nc(N2C3CCC2C(CNC(=O)Cc2coc(C(F)F)n2)C3)ccc1C#N c1(C(=O)NCC2CN(C(CC(C)OC)=O)CC2(C)C)cnc2c(c1)NC(=O)CS2 C1(NC(=O)C2=CCCC2)CN(C(c2ccn3ccnc3c2)=O)CC1C1CC1 O=C1CC(c2cn(C3COC3)nn2)NC(=O)N1c1ccc(N2CCC(O)C2)cc1 C1(NC(Cc2c(C)noc2C)=O)CC(O)CN(C(c2ccnc(N(C)C)c2)=O)C1 CN1CC2OCCN(C(C3CN(C(c4ccc(=N)[nH]c4)=O)CCC3(C)C)=O)C2C1 C(CCC(c1ccccc1)N(C)C)OCCCN(C1CCCC1)C(=O)NC Nc1cc(CC(=O)NCCOCCNC(C2OCCO2)=O)c(Br)cc1[N+](=O)[O-] N1(C(c2cc(C)ncn2)=O)CC(C2CCCN(C(=O)CCC3CCC(=O)N3)C2)C1 N1(C(CC2CCN(C)C2)=O)CCCN(C(c2cccc3c2CCC3)=O)C(CO)C1 CC(C)CC(F)C(=O)N(C)CCC1CCN(C(C2CCCC2)=O)CC1 C1(C(N2CCN(C(c3c(OC)cccc3)=O)CC2CO)=O)CCc2cncn2C1 c1(C(=O)NCc2scc(C(N(CCCC)C(C)CC)=O)c2)c(C)nsc1N c1(C(=O)NC(C2(CNC(C(C=C)O)=O)CC2)C)cc(Br)c(O)nc1C c1(OC)cnc(NC(=O)NC(C2CCCCC2)CSc2ccccc2O)c(F)c1 C1(NC(C(C)SCC)=O)CC2(C1)CC2NC(c1coc(C(F)F)n1)=O C1(C(=O)NCCOC2CCN(C(c3c(CC)nc[nH]3)=O)C2)CC(O)CN1C C1(O)(CNC(=O)COC2COC2)CN(C(C2CC(O)C2)=O)C1 c1(SC)nccnc1C(=O)NCC(O)CCNC(=O)C(C(C)C)c1cnc(C)s1 C1(CC)C(C(=O)Nc2cncnc2C)CCN1C(=O)CCn1cnnn1 N1(C(c2ncc(C)cn2)=O)CCOC2(CCCN(C(=O)C(C)(C)CF)C2)C1 C1(CC)CN(C(=O)CCOCC(F)(F)C(F)F)CCC1CNS(=O)(=O)CCC c1(OCC)ccccc1C(=O)NC(c1cn[nH]c1)C.C12(CC1)C(=O)N2 C1(CC)CN(C(=O)C(F)(F)CO)CCC1CN(C(=O)CC1CCCC1)C1CC1 C1(CCNC(CSC(C)C)=O)CN(C(=O)CCCCN2CCCC2)CCCO1 C(=O)(C1CCCc2ncc(C)n21)N1CCN(C(CC2CN(CC)C2)=O)CC1 N1(C(c2nnnn2C)C)CC2CC1CN2C(c1ccc(-n2ccnc2)cn1)=O C(=O)(C1=CCS(=O)(=O)C1)NC1(C2CN(C(c3cc(C)ns3)=O)C2)CC1 C1(C)(C(=O)NC2CCC(NC(C3CN(C)C(=O)CC3)=O)CC2)CCCCC1(F)F N1(C(C(c2ccc(C)o2)C)=O)CCOCC(CNC(c2ncoc2C)=O)C1 N1(C(C2(OC)CCCC2)=O)CCC2(CC1)CN(C(C1(C)CC1(F)F)=O)C2C(C)C CC1(C)CCCC(O)(C(=O)NCC2CCC(NC(C3CCCCO3)=O)CC2)C1 C1(C(N(C2CCN(c3ccccc3)C2)C)=O)CCN(C(=O)NC2CCOC2)CC1 C1(CC)C(NC(=O)CC(O)CN(C)C)CCCN1C(C1CCOCO1)=O C1(NC(CC2CCN(C(CCCCCC)=O)C2)=O)C2CCC(C2)C1(C)C c1(CC(=O)NC2CCC(CNC(C3(COC)CC3)=O)C2)c[nH]c2cccc(Cl)c12 Cc1c(CC(=O)NC(C)C(=O)NCC(N2CCCC(C(N)=O)C2)=O)cnn1C c1(C(N(C2CCCCCC2)CCNC(C2C(C)CCS2)=O)=O)cccc2nsnc12 C12(NC(C=CCOC)=O)CCCC1CN(C(c1cnc(-c3ncccn3)s1)=O)C2 c1(C(=O)NC(CN(C(C2CCCC(OC)C2)=O)C)(C)C)cnc2[nH]cnc2c1 C1(CC)CC(C(N)=O)(CO)C(C)C1.C1CCCC(C2CC2)NC(=O)NC1.C(C)(C)(C)O C12(NC(CC=CCC)=O)COCCC1CN(C(=O)C1=NN(C3CC3)C(=O)CC1)C2 C1(CC)CCN(C(C2CN3CCC2CC3)=O)C(C(N2CCC(C)(CCO)C2)=O)C1 Cn1cc(CC(O)C(=O)N2CC(CCNC(c3ccsc3N)=O)C2)cn1 C1(=CC(=O)NCC(C2CCCC2)NC(c2n(C(C)C)nnc2)=O)CCN(C)CC1 C(=O)(C(C)(O)C(C)(O)C(=O)N1CC2C=CC2C1)OC C1(NC(C2(C#N)CC2)=O)CC2(C1)CC(NC(c1n[nH]cc1C(F)(F)F)=O)C2 C1(NC(C(c2ccccc2)OC)=O)CCC2(CC1)CC(NC(=O)C1=CCOCC1)C2 Cc1cc(=NC(C)(c2cccc(Cl)c2Cl)c2nnnn2C)[nH]n1C(C)(C)C c1(C(=O)NC2(C(=O)OC)CCCOC2)cc2c(s1)CCC(C)(C)C2 N1(Cc2c(C(=O)NCc3noc(C4CC4)n3)cccc2)CC(=O)Nc2ccccc21 CC1(C)CN(C(c2cc(N)ccn2)=O)CC1NC(C12CC3CC1C2C3)=O Cc1c[nH]c(=NCCCC2CCCCO2)cc1O CC1CCC(CC(=O)N(C)C)C1.n1(CC(=O)OC)nnc(C2CC2)n1 Brc1cnc(-c2nc(C3CCC3)nn2Cc2ccncc2)nc1 N1(C(C2OCC(C)C2)=O)CCC2(CCN(C(=O)C(=O)NCC3CC3)CC2)C1 C(=O)(CC(C(C)C)NC(=O)CCCCOC)N(C(c1cn(C)nn1)C)CC c1(C(=O)NCCC(CNC(c2cc(OC)n(C)n2)=O)O)cccc(Cl)c1C C=C1CC2(C1)CC(C(N1CCC1CNC(c1c(C)nn(C)c1C(F)(F)F)=O)=O)C2 C1(C(N2CC3CC2(c2ccncc2)C3)=O)CC2(C1)CC2F C1(C(N2CCC(NC(c3cnc(S)nc3)=O)(CO)C2)=O)Cc2cc(F)ccc2O1 C(CN=c1cc(C)nc(N(C)CC2CN(C)CCN2C)[nH]1)N(C1CC1)CC N1(C(CCCNC(C)=O)=O)CC(CNC(=O)NC2(CS(C)(=O)=O)CCC2)C2(CC2)C1 c1(C(N2C(CN(C(CC(C)C)=O)C)CCC2)=O)ccccc1SCCC(F)(F)F C(C)(CC(=O)N1CCC(NC(=O)C(C)(C)c2cccs2)CC1)(C1CCC1)N(C)C S(=O)(=O)(c1cccc(Cl)c1)NCC(=O)NCCCNC(CC(=O)NCC)=O c1(N(CCC#N)C)[nH]c(=NCCNC2(OCC)CCOCC2)nc2c1ncn2C C1(CNC(CCOC(C)C)=O)CCC2(CCC2)CN1C(C1CCCCN1N=O)=O c1(C(=O)NCC2N(C(C3CC(C)N(C)C3)=O)CC(C)(C)C2)[nH]nc([N+](=O)[O-])c1Cl N1(C(C2(F)C(C)C2)=O)CCCCC(NC(c2ccccc2-n2cnnn2)=O)C1 C#Cc1ccc(C(N2CCCC2CNC(c2occc2CC)=O)=O)c(OC)c1 Cc1cc(C(N2CCC(NC(=O)C3CC3)C(O)C2)=O)c(C)n1C1CCCCC1 c1(C(=O)NC2CC(C)N(C(c3nnc(O)cc3O)=O)C2)cc2cc(Cl)ncc2[nH]1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(C1CN(C(C2CCCS2)=O)C1)C C1(C(=O)NC(c2ccc(-c3ccc(F)c(F)c3)s2)C)CCCN(C(=O)C(N)=O)CC1 Cc1ccc(C(=O)NC(C)CC2CCN(C(C3(CO)CCC3)=O)CC2)nc1O N#CCCCC(=O)N1CCC(OCCN(c2cnn(C3CCCC3)c2)CC2CC2)C1 C1(C(=O)NCc2cccc(C(=O)NCCCO)c2)CC2CCC(C1)S2 N1(CCC)C(=O)CCC1C(=O)NCCCCCN(C)C(C1(CF)CC(F)(F)C1)=O Cc1cncc(C(=O)NC(C(=O)NC(c2cnc(C)s2)C)c2ccoc2)n1 N1(C(=O)CCOc2cccnc2)CCC2C(CCCN2C(C2CC=CCO2)=O)C1 C(C)(C)(C(=O)NCCNC(=O)CC1CCCN1CC1CCCC1)NC(=O)NCC Cc1cc(N)cc(C(N2CCN(C(=O)C=CC3CCCO3)CC2C2CC2)=O)c1F C(=O)(C1=CNS(=O)(=O)N=C1C)NCC1CC(CNC(C2N(CC)CCCC2)=O)C1 c1(OC)ccc(Cl)c(C(N2CCOCC(NC(c3cn(C)ccc3=O)=O)C2)=O)n1 c1(C(=O)NC(C(C)NC(C2CCCN2S(C)(=O)=O)=O)CO)ccc2sncc2c1 C(CCCCC(=O)N1CCCCC1C1CCN(C(C2CN(C)CC(C)O2)=O)C1)OC c1(C(=O)NC2CN(C(C(C3CCCOC3)OCC)=O)C2)c[nH]nc1Cl C(CC(C)CC)(C(=O)NCC(C)(C)CCOC)NC(C(CCC)OC)=O C1(O)(C(C(N2CCOC(CNC(C3CC4C=CC3C4)=O)C2)=O)F)CCCCCC1 Cc1cc(-c2cn(CCN(C(c3cccn3C3CCCC3)=O)C3CC3)nn2)cc(F)c1 c1(C(=O)O)cc(OCCOCC(N2CCCC2NC(C)=O)=O)cc(COC)c1 C1(CNC(CN2CCN(C)C(=O)C2)=O)CCCC2CN(C(=O)C(=O)N(C)C)CC12 C(=O)(C(C)C(C)C(C)(C)C)NC(CNC(c1ccc(C(=O)NC)nc1)=O)C1CC1 Cc1ccc(CCCC(N2CC(C)CCC2CNC(=O)CSC(C)C)=O)cc1C C1(CCC)(C(=O)N2CC(=O)N2C(C)C)CC1.C(COC)OC.C1(C)CC1 Cc1noc(CCC(=O)N(CC(=O)NC(c2ncc(C)o2)C)C2CC2)n1 C1(NC(c2c(CC)c[nH]c2)=O)(CC)CCCN(C(=O)C(N2CCC(C)C2)=O)C1 CP(C)(=O)c1ccc(CNC(=O)C(N2CC3(CCC(CO)O3)C2)=O)s1 c1(C(=O)NC(c2nccs2)C)ccc(CN(C)Cc2nccs2)o1 C1(C(=O)NC(C)(C)CN2CCOCC2)CCC(NC(c2ccsc2Cl)=O)C1 C(N=c1[nH]c(=NCCCOC2CC2)[nH]c2cc[nH]c12)C1CC(C)(C)C1 N1(C(C(C)Cc2ccc(Cl)cc2)=O)CC2CC(C1)CN(C(=O)CC1CC(=O)C1)C2 C1(C(N)=O)CN(C(=O)C(c2ccccc2)O)CC1CNC(=O)CCC1CCCC1 c1(NC(C(N(OC)C)=O)C)cc2c(c([N+](=O)[O-])c1)OCO2 C1(C(=O)NC(CNC(CSCC(C)=O)=O)(C)CC(C)C)CC(C(C)(C)C)=NO1 C12(NC(C(C)(C)C3CCCO3)=O)CCCC1CN(C(=O)C(C)(C)S(C)(=O)=O)C2 Cc1cc(Cl)c(C(=O)NCC(C2CCC2)NC(=O)C(C)(C)N2CCOCC2)s1 CCCCCCC(CC)C(=O)NC(C)CC(C)NC(=O)C(C(C)C)SC C1(CC(=O)N(C(C)C(=O)N2CC(n3cccn3)C2)CC)CCCCC1 N1(C(C2=C(C)CCC2)=O)CCC2CN(C(=O)CC(C)(C)C(F)F)CC2C1 c1(CC(=O)NC2C(NC(C(CO)NC(N)=O)=O)C2)cccc2nonc12 C1(CNC(c2cnc(SC)s2)=O)CCCC(NC(c2n[nH]cc2C)=O)C1 N1(C(C(C(CC)C)O)=O)CCC(C2(NC(=O)CCNS(C)(=O)=O)CCC2)CC1 N1(Cc2cc(C)c(Br)cc2C)CCC2(CCN(C(=O)C(F)(F)c3ccccc3)C2)C1 c1(OCC(C)C)cc(C(=O)NCCNC(C2CC2(F)Cl)=O)ccn1 C(c1ccc(=N)[nH]c1C)=CC(=O)NCC(CC)(C)NC(C1CC1F)=O c1(-c2ccc(OC)cc2)n[nH]c(=NC(=O)N(C)C(c2nnc(C)o2)C)s1 N12C3CCC1C(C3)NC1CCC3(C1C3)C2=O.C1(C(=O)OC)CCC(C(N)=O)N1C C12(C(=O)NCCOCCNC(C3(O)COC3)=O)CCN(CC1)CC2 n1(CC)nccc1C(=O)NC(C1CCN(C(C2(c3ncco3)CC2)=O)C1)C C1(CNC(c2ccnc(N3CCC(O)C3)c2)=O)CC(O)CN1C(=O)C1=CCCS1 C(=O)(C(C)(C)CCCNC(=O)C1=CCN(C)C1)NC1C(C#C)CCC1 c1(C(=O)NCC(CCNC(CC=C)=O)O)cnc2c(c1)NCC2 C(N=c1[nH]c2c(c(=NC(C)c3c[nH]c4ccc([N+](=O)[O-])cc34)[nH]1)CCC2)C1C(C)C1 Cc1cccnc1-c1cn(C2CN(C(C3(C4CC4)CC3)=O)C2)nn1 C12(CNC(=O)C=C3CCC3)CCC(CC1)N(C(=O)C(F)C1CCCC1)C2 c1(OC)ccc(F)c(CNC(=O)Cn2cc(C(N3CCN(C)CC3)(C)C)nn2)c1 C(=O)(C1=CC2C=CC(C1)C2)NC(CN(C(=O)CC(C)(C)CC)CC)C Cc1ccc(Cl)c(CC(=O)NC(C)CC(C)NC(=O)CN2CCCCC2)c1 C1(O)(CNC(C=CC=CCC)=O)CCCN(C(=O)CCOC2CCC2)C1 c1(C(N2CCC(C)(CNC(C3CCC(=O)C3)=O)C2)=O)nc2c(Br)cncc2[nH]1 N1(C(Cn2c(C(C)C)ncc2)=O)CC2C(CNC(c3conc3C3CCC3)=O)C2C1 C(=O)(CC(C)(O)COC)N1CCC(NCC(N2C(CC(=O)NC)C=CC2)=O)C1 O(N(C(=O)C(F)C1(O)CN(C(=O)CC2CCCO2)C1)C(C)C)CC N1(Cc2c(OC)cc(Cl)cc2)c2ccccc2C(C)C1C Cc1oc([N+](=O)[O-])cc1C(=O)NC1CC(NC(c2cccc(C(N)=O)c2)=O)C1 Cc1nn(CC(C)C)c(Cl)c1C(=O)NC(C)C(CO)NC(=O)CCOC1CCC1 C12(C(=O)NC3CC(NC(C4(CC(C)C)CCC4)=O)C3)CCN(C1)S(=O)(=O)C2 Cc1ccc2c(C(=O)NC(C)CNC(=O)CCC3CC3C)ccnc2c1 c1(N2CCN(C(CC3CC(C)(C)OC3(C)C)=O)CC2)nc2c(F)cc(Cl)cc2s1 N1(C(C23CC(C)C2C3)=O)CC(NC(C2(N(C)C)CCC2)=O)CC(C)C1 c1(CNc2c(F)ccc(Br)n2)cc2cc(Br)ccc2s1 N1(C(C(C)c2ccsc2)=O)CC(C(C2CC2)NC(=O)Cc2cccs2)C(O)C1 CCCCC(C)CC(=O)N1CCN(C(=O)C(C)n2ccnc2)C(C)C1 CC(C)CC(=O)NCC1CN(C(=O)CCC2CC(C)C2)C1 N1(C(C(c2cncnc2)C)=O)CC2CCC1CN2C(=O)CCC(=O)N(C)C(C)C c1(CC)cc(C(=O)NC2(CCNC(=O)C(C)(C)C3CCOCC3)CCC2)ncn1 C(=O)(CC(C)(C)C(=O)N(CC)Cc1cn(C2CCC(C(=O)O)C2)nn1)OCC c1(ONC(CN2C(C)CCC2C)=O)ccc(N=Nc2ccccc2)cc1 C1(NC(c2c(C)nc(C)s2)=O)CCCCCC1C(=O)NC1CC(O)C1OC C=CCCC(F)(F)C(=O)N1CC(C(=O)NC(c2ccn(C)n2)CC)(COC)C1 c1(C(N(C2CC3CN(CC)CC23)c2nc(C)ncc2Cl)=O)cccc2ncoc12 c1(CCC(N2C(C(C)NC(c3cc(C)ncc3)=O)CCC2)=O)ccc(O)c(Cl)c1 c1(C(=O)NC2CCCCC2CNC(C2CC23CCCC3)=O)csc([N+](=O)[O-])c1 N1(C(c2c(OC)scc2)=O)CC(NC(=O)Cc2c(F)cccc2Cl)C(C2CC2)C1 CC12CC(C(=O)NCCCN(C(c3cc[nH]n3)=O)C3CC3)(C1)C1(CCC1)O2 c1(CNC(=O)N(C2CC2)Cc2ccccc2)cc2ccccc2s1 Cc1ncc(COCC(=O)NC2CC(C)(NC(=O)CCOC3CCCCC3)C2)s1 c1(C(=O)NCc2nnc(CNC)s2)cccc2c1nnn2C N1(C(C(C)OCC#C)=O)CCC(C(=O)NOCC)CC1Cc1ccnc(O)c1 c1(C(C)NC(C(c2ccn(CCC)c2)N(CC=C)CC#N)=O)ccc(Cl)cc1 C1(NC(C(=O)N(C)C)=O)COC2(CCCN(C(=O)CCc3cccnc3)C2)C1 N1(C(CCC=C=C)=O)CC2(C1)CN(C(=O)CCC(C)OCC)CCO2 c1(C(=O)NC(C(C)NC(C2CCOC2=O)=O)CO)cc(Cl)cn1C N1(C(C2COCCC2NC(=O)Cn2ccnc2)=O)CCN(CC(=O)OCC)CC1 c12ccc(cc1OC)CC1(CC3(CSC3)C1)c1nnnn1CCCCO2.CO C(=O)(CCCCSC)N1CC(C(N)=O)(CNC(c2ccc(C(C)(C)OC)o2)=O)C1 CC(CC(=O)Nc1cncnc1O)C(C)(C)N1CCC(C)(OC(F)F)C1 c1(-c2cnc(SC)nc2)cn(C)[nH]c1=NC(=O)C12CCC(CO)(CC1)C2 CC(C)CC(C)(O)C(=O)Nc1cccc(NC(C2CC(=O)N(O)C2)=O)c1 c1(C(=O)NCC(CNC(c2nccnc2C)=O)OC)ccc(C(C)C)c(C)c1 c1(OC)ccccc1C(=O)NC1CC(CCC(=O)N(CC(C)CC)C)C1 C1(NC(c2ccc(C)nn2)=O)CCC(C)N(C(C2CCC(C)(C)O2)=O)C1 C(C(CC(F)(F)F)NC(=O)C(C)OC1CCOC1)NC(c1c(C)occ1)=O C=C1CCC(C(=O)NC2CC(NC(c3ccc(NCCC)cc3)=O)C2)CC1 C(=O)(C(CNc1cccc(N)c1)CCCC(F)(F)F)OCc1cccc(OC)c1 c1(C(NOCC(C)C)=O)coc(C2CCCN2C)n1.c12ccn(n1)CC(=O)N2 CS(=O)(=O)c1cccc(C(=O)NCCOCCNC(C2CC3CC2C3)=O)c1 c1(OC)cc(C)c(C(=O)NC(C2CCN(C(c3ccc(O)nn3)=O)C2)C)c(F)c1 c1(CC)cc(N2CCCC2(C)CNC(=O)COCCOC)ncn1 CCCCCC(F)C(=O)NCC(C)CNC(C1(CC(F)F)CC1)=O Cc1nc2cnn(C)c2cc1C(N1CCC(NC(=O)C(=O)N(C)C)C(C)C1)=O N1(C(=O)CC2CC3CCC2O3)CCN(C(c2nc[nH]n2)=O)C(C2CCC2)C1 C(=O)(C(C)(C)C(=O)Nc1ccn2ccsc12)OC(C)(C)C C(N=c1[nH]c2c(c(=NCc3cccnc3O)[nH]1)COC2)c1c(CC)nn(C)c1 C1(CNC(C(C=C)(C)C)=O)CC2(CCC2)CN1C(C1CCC(=O)NC1)=O Cc1c(Cl)c(C(=O)NCC(C)(CC(C)C)NC(c2csnn2)=O)nn1C N1(C(CC=CCNC(C2(C)CCC(=O)NC2)=O)=O)CC2CCC(O)C2C1 c1(CCC(=O)NCCN(C(C2CCC3CC3CC2)=O)CC)cnc2n1CCCC2 c1(Nc2c(C)nc(NC(=O)C(C)(C)CC(F)(F)F)nc2)cc(C)c2cc[nH]c2c1 C(=O)(C1CCCc2c[nH]nc21)N1CC2C(CCNC(=O)CSC(F)(F)F)(CC2)C1 C1(NC(C(=Cc2ccncc2)C)=O)CC(O)CN(C(c2cnccc2Cl)=O)C1 CCC(O)C(C)C(=O)N1CCC(O)(Cc2nn[nH]n2)CC1 N1(C(c2nnc(C)s2)=O)CCN(CC(C)(C)NC(=O)CCN2CCC(F)C2)CC1 c1(C(CCCC(N(C2CC3CC2CN3)S(C)(=O)=O)=O)=O)c(F)cc(F)cc1F N1(C(C(C(C)O)C)=O)CC2CC(C)C(C1)N2c1cc(S(C)(=O)=O)ncn1 c1(SC)cccc(C(=O)N(CC(O)CN(C(=O)CC2(C)CCC2)C)C)n1 CC1(NC(c2ccc(Cl)c(O)c2)=O)CCN(C(=O)C=Cc2ccc(Cl)s2)CC1 C1(NC(CC(=O)NCC)=O)CCN(C(c2cccc(C(C)(F)F)c2)=O)C12CCC2 C1(C(=O)NC23CC(NC(C=CC)=O)(C2)C3)CCC2C1C2(F)F Cc1ccc(-c2cn[nH]c2)cc1.c1(C2C3C(C3)C(=O)N2)ccccc1 Cc1ncccc1CC(N1CCCC(CCC(=O)NC2CC(C)C2)C1)=O c1(OC)ccc(N(CC(=O)NCC(Cc2ccoc2)CO)C)cc1 N1(C(CC(CC)C(C)C)=O)CCC2CCC(C1)N2C(=O)C(C)(COC)OC c1(CC(=O)N(C2CCN(C(=O)Cc3cnccc3Cl)C2)CC)ccc(C)cc1C C1(N(C(C(C)P(C)(C)=O)=O)C)CCN(C(c2ccn(C3CC3)n2)=O)CC12CC2 C#CC1(C(=O)NCC2CCC(C)(C)O2)CCN(C(C2CCCSC2)=O)C1 c1(C(=O)NCC(CC)NC(c2ccc(Cl)[nH]2)=O)c(C(F)(F)F)cccc1Cl c1(C(N2C(C(C)C)CN(C(=O)CSC3CC3)CC2)=O)cccc2c1CNC2=O C1(CN(C(CN(C(C2CC(=C)C2)=O)Cc2ccccc2)=O)C)CC(C)CO1 N(C1CCc2c(Br)ccc(Cl)c21)Cc1ccc(S(=O)(=O)N2CCOCC2)cc1 N1(C(C)C)CCCC(C(N2CC(C)(C)C2)C(=O)NCC(F)F)C1 c1(OC)ccc(CCC(=O)NC(C)CCNC(=O)C(C)c2ccon2)cn1 c1(C(N2CCC(C3N(C(C(C)n4cncn4)=O)CCC3)C2)=O)ccnn1C C1(NC(C2(C(N(C)C)=O)CC2)=O)CCN(C(C2CC3CCC2C3)=O)CC1(C)C c1(CNC(C(=O)NC2(CSC)CCNCC2)=O)sc2[nH]cnc(=O)c2c1C N1(C(=O)C=Cc2cn3c(n2)CCCCC3)CCc2nc[nH]c2C1c1ccncc1 C1(NC(CC)=O)C(C(=O)NC(C)C2CC2)C1(C)C c1(CC)cc(C)ccc1NC(=O)C(F)C1CC(NC(c2c[nH]nc2C)=O)C1 N1(C(C(CCC)N(C)C)=O)CCCC(CNC(c2c(C)n[nH]c2C)=O)CC1 N1(C(c2c(C)nsc2)=O)CC(CNC(=O)C=Cc2cnc[nH]2)CC12CCC2 C1(C(=O)NCCSCC(=O)OC)CC1C1CN(C(=O)CCC(=O)NC)C1 C(=O)(C(C)(C)CC(F)(F)F)NCC1CN(C(C2(C=C)CC2)=O)C1 C1(N(C(C(C)=C2CC2)=O)C)CCC(NC(=O)Cc2cc(C)cs2)C1 CS(=O)(=O)c1ccc(Cl)c(C(=O)NCC2CN(C(c3cnns3)=O)CC2O)c1 c1(OC)cc(Br)ccc1C1(C(N2CC(O)(CCNC(C3CC3F)=O)C2)=O)CC1 c1(OC)ccncc1C(=O)NCC(C(C)(C)C)NC(c1cnn(C(C)C)c1F)=O C1(C(=O)NCC(CN(C(=O)CC(=O)NC(C)(C)C)C)O)CCC(C2CC2)CC1 C1(C)(OC)CC(NC(=O)NCCCN(C2CCCC2)C)C1(C)C c1nc(Cl)sc1Cl.N1(CC(=O)OC)CCC(N(CCCC)C(=O)COC)C1 N1(C(CCCC)=O)CC(NC(=O)CN(C)CC)C(Cc2cccc(F)c2)C1 C1(NC(=O)Cc2ccc3nn[nH]c3c2)CC(C2CCN(C(C3C=CCS3)=O)C2)C1 n1(CCC=C)cc(C(=O)NCCC2(O)CN(C(c3cnc(C4CC4)o3)=O)C2)nn1 CCCC(CCC)CC(=O)NCC(CO)NC(C1CCC1C(=O)OC)=O CC1CCCCN1CCCNC(C(=O)CN1CCCCC1C)=O.C(COC)O C1(C(=O)NC(C)Cc2ccsc2)CCCCCN1C(=O)CSC(F)F Cc1cncc(C(=O)NC(C(=O)NCC2(C)CC=CCC2)c2ccco2)c1 C(C)(C)(CC(F)C(=O)NCCc1cnccc1C)NC(C(F)=C(C)C)=O C1(CNC(CC2CCN(C(C3(c4c(C)cccc4)CC3)=O)C2)=O)CC2CCCC2C1 C12(CNc3nc(C)nc4c3ccs4)CCCC1N(C(=O)C=CI)CCC2 C(=O)(C#CC1CCCOC1)N1CC(COC)(CNC(C23CCN(CC2)CC3)=O)C1 C=CCC(C)(CNC(=O)CC(C)NC(=O)CCC(C)(F)F)CO C1(NC(CSc2ccc(C)cc2)=O)CCSC12CN(C(=O)CCc1cnn[nH]1)C2 CCCC(C(=O)NCC1CCC(CN(C)C(C2C(C)C2C)=O)CC1)NC(N)=O c1(-n2cc(CN(C)C(C(C)(C)CC3CCOC3)=O)nn2)cnn2c1NCC2 C(=O)(CC(O)(CC)N1CCC(Cc2cccc(O)c2)CC1)NCCCC C1(C)(C(=O)NCC(CC)NC(c2sc(NC(C)=O)nc2C)=O)CCC(C)C1(C)C C(C(=O)NC(C1CC(F)(F)C1)C)(C(C)(C)C)NC(c1n(C=C)ncc1)=O CCCCCC(O)C(=O)N1CCCC(CCNC(c2c(C3CC3)cnn2C)=O)C1 CCC(CC)CC(=O)N(CCSC)CC1CCN(C(C)=O)CC1O N1(C(CCCC#N)=O)CCC2CC2(NC(=O)CSc2cc(Cl)ccc2Cl)CC1 C#CCCC(=O)NC(CN(C(=O)C(C)(C)NC(=O)Nc1ccccc1)C)CC c1(CC)cc(C(=O)N(CC(CC)NC(c2sc(C3CC3)nc2C)=O)C)cc(O)n1 C(=O)(CCCCCNC(N)=O)NCC(C)(CO)NC(C12CC(C)C1C2)=O N1(C(C(c2[nH]c(=N)sc2)O)=O)CCCC(NC(=O)CCc2nncs2)CC1 C1(NC(CSCCN(C)C)=O)CN(C(=O)C2=NOCC2)C2(CCCCCC2)C1 c1(-c2ccc(C(N(C)CC3CCN(C(C4CC4CF)=O)C3)=O)s2)ccc(F)cc1 C12(CNC(C3(OC)CCOC3)=O)CC(C1)C(NC(c1cc3n(n1)CCO3)=O)CO2 C#CCC(C)C(=O)NCC=CCNC(=O)C(C1CCCCC1)Nc1ccncc1 C1(C(N2C(C(=O)NCCC(C)CO)CC2)=O)CCCN1C=O c1(C(=O)NCC2(C(C)NC(=O)CC(C)N(C)C)CC2)cnc(Cl)c(N)c1 C1(NC(C(CC(=C)C)C)=O)CC2CC(C1)CN(C(C1C3CCC1CC3)=O)C2 N#Cc1ccccc1C(=O)NCC1CN(C(=O)CCOc2ccccc2)CCO1 Cc1cc(CNC(C2(N(C(=O)Cc3cnnn3C)C)CC2)=O)oc1C C1(=CC(=O)NC2C(CNC(C3CCC(=O)N3)=O)CCC2)CCOc2ccccc21 C1(NC(C(C)CC2CCC2)=O)CC12CCN(C(c1ccc(C3CCCO3)[nH]1)=O)C2 c1(CN2CCN(C(C3CCc4cnnn4C3)=O)CC2)ccc(Cl)cc1[N+](=O)[O-] C1(CNC(c2cscc2F)=O)CCCCN1C(c1conc1C1CCCO1)=O c1(CC(=O)NC23C(CN(C(c4c(C)ccs4)=O)C2)C3)ccc2n[nH]cc2c1 N1(C(c2n(C)cnc2)=O)CC2(CCCN(C(C3CC3c3ccccc3Cl)=O)C2)C1 N1(C(c2n(C)nnc2)=O)CC2COCC2(C(=O)NC2CCCC(C(N)=O)C2)C1 N1(C(c2nc(C(C)=O)sc2)=O)CCC(NC(c2cc(C)n(C)n2)=O)C1(C)C c1(C(N2C(CNC(c3cccc(OCC)c3)=O)CCC2)=O)cnc(OC)c(C)c1 C1(CN(C(C(C)OCCC(C)C)=O)C)CCCN(C(=O)CN2CC3CC3C2)C1 c1(NC(C2CC2c2ccccc2)=O)cc(Cl)cc(Cl)n1.C12CC1C(=O)NC2 C(CC(C)C(=O)NC(CCOCC)C(=O)NCc1ncnn1C)=CC N1(C(CCc2n(C)cnn2)=O)C(CC(=O)NCCn2cnccc2=O)C2CCCC12 Cc1ccncc1C(=O)NC1CCC(C(=O)Nc2cncc(C(F)F)c2)C1 CC(C)CCC(O)C(=O)N1C2CCC1CC(NC(c1c(F)ccc(F)c1N)=O)C2 c1(Cn2cc(CNC(C3CCC(SCC)CC3)=O)nn2)ccc2c(c1)CCO2 C1(C2CCCN(C(=O)C(O)C3CC3)C2)(NC(c2n(C)c(C(F)(F)F)cn2)=O)CC1 c1(CC)nccnc1C(N1CCCC1C=CC(N1CC(n2cnnn2)C1)=O)=O CC(CS(C)(=O)=O)C(=O)N1CCC(CNC(c2cc(C(F)F)no2)=O)C12CCC2 N1(C(C2C(C)CCS2)=O)CCN(C(c2ccc3cc(F)ccc3n2)=O)CC12CCC2 c1(C(C(=O)NCCCF)N(CCCC)C)ccc(OC)cc1.C(CO)O C12(C(N(CC)CC3CCCN3C(=O)CSC(C)C)=O)CCCC1C2(F)F C(=O)(C(C)C(O)CC)N1CC(CNC(c2ccc(C(=O)OCC)cc2)=O)C1 c1(OC)cc(C(=O)OCC(C2(O)CN(C(=O)CCC(F)(F)F)C2)(C)C)cc(F)c1 C12(C(N3C(C(=O)NC)CC3)=O)CCCC1CCN2C(=O)C(n1cc(C)cn1)C N1(C(c2cc(C#N)[nH]c2)=O)CC2CCN(C(=O)CCc3cccc(F)c3F)CC12 N1(C(c2c(C)oc(Br)c2)=O)CCC(O)(CNC(=O)C=C2CCC(C)C2)CC1 C1(O)(C(=O)NC2C(NC(C(=O)NCC)=O)CCC2)CCCC(C)(C)C1 C1(C(=O)NC(C)CCCNC(=O)C(N2CCOCC2)C)NC(=O)OC1C C(C(C(=O)NC1CC=CC1)NC(C1CSC1)=O)OC(C)C C1(NC(C2(COC)CCCC2)=O)CCN(C(c2ncc(C)cc2OC)=O)CC1C C=CCC(CC)C(=O)N1CCCCC1CNC(C1CN(C(C)C)C1)=O C1(C2=CCOCC2)(c2onc(CN3CCCC(NC(=O)NC)C3)n2)CC1 N1(C(C2NCCN(C(c3c(OC)ccs3)=O)C2)=O)CC(O)C(O)C(O)C1CO c1(NC(C(N2CC(C)C2)C)=O)csc2c1CCOC2 CC1(CNC(=O)COCCF)CN(C(C2CCC3(CCC3)C2)=O)CCO1 C(CC(C(=O)N1CCC1C1CCOCC1)NC(C1C=CC=CC=C1)=O)=CC N1(C(c2c(C)con2)=O)CCN(C(c2cc(Br)cnc2O)=O)C2CC12 C(=O)(C(F)C(=O)NC1CN(C(=O)CN(CC(C)(C)C)C)CC1OC)OCC c1(NCC(CC(C)C)NC(C)=O)ccc(S(=O)(=O)NCCC(=O)OC)cc1Cl C(=O)(C1=CCC(C)(C)CC1)NCC=CC(N1C(C)CC1CO)=O C1(C(N2C(C)(C(=O)OC)CC2)=O)CCCC(NC(=O)CC(C)c2ccco2)CC1 C#CC1(OC)C(N(C)Cc2cc(Br)cn2C(C)C)C1C[Si](C)(C)C C1(C(C)C)CN(C(C2CC2C)=O)CCN1C(c1cc(Cl)no1)=O N1(C(C(CC)(CC)OC)=O)CCC2CC(NC(C3CC3(F)F)=O)CCC2C1 Cn1ncc2c1CN(C(C1CCCCN1Cc1ccc(O)cc1Br)=O)CC2 C1(C(N2CCCCC(N(C)C(C3CCOC(C)(C)C3)=O)C2)=O)C2CC(F)(F)CC12 C(=O)(C(C)(C)c1cnsc1)N(CC(O)CNC(=O)C1CC1)C N1(C(CCCCCCC)=O)CCCC2CN(C(C3(C)CCN(C)CC3)=O)CCC12 N1(C(=O)NCCOC)CCC(C(=O)NC(C)C)C(C)C1.c1(CCN)cc(C)ccc1F C1(NC(=O)Cc2cc(Cl)ccc2O)CC12CCN(C(C1(Cl)CC1(F)F)=O)CC2 C1(NC(CCC#C)=O)CCCCCC1NC(=O)COc1ccc(F)cc1Br Cc1c(C(N2CC(O)CC2C(N2CCC3(CC2)CC3)=O)=O)ccc2c1OCO2 c1(C(C)C)cc(C(=O)NCC2C(C)CCN2C(=O)C(=O)C(C)(C)C)ccc1F C(N=c1nc2c(ncn2C)c(NCCC2SCCS2)[nH]1)c1cc(C)cc(C)n1 CN1CCOC(CNC(C2OCCC2NC(=O)CCCn2cncn2)=O)C1 CCCCCCCC(=O)N1CCSCC1CCNC(c1cc(C)c(F)cn1)=O CCC(C(=O)NC(CCF)C(=O)Nc1cccc(O)c1)C(C)C CCCCC(CC(=O)NCC1(C)CCCC(=O)N1)NC(=O)CCNC(=O)NC C(=O)(C(C)(C)CCCF)NCC(C(=O)N(CCCC)CCCO)O C(CC(C(C)(C)C)NC(c1coc(C(F)(F)F)c1)=O)N(C(=O)C(C)(C)F)C c1(C(N(C2CCN(Cc3cc(C4CC4)on3)C2)C(CC)CC)=O)sc(C)cc1C CC(C)(C)CCCC(=O)NCC(CNC(C1C(C)(C)OC1(C)C)=O)CO N1(C(C(CCC)O)=O)CC2CCOC2(CNC(c2c(SC)cccc2F)=O)C1 c12cc-1ccc2F.C(C(=O)N(CCO)C(=O)C1CC1)=CCC C1(NC(c2n(CC=C)nnn2)C(OC)OC)CCN(c2ccccc2)C1=O C1(NC(C2CC(=C)C2)=O)CN(C(=O)Cc2nc(C3CC3)cs2)CC12CCC2 CC1(C)COCC1C(N1CC(NC(c2ccc(-c3ncon3)cc2)=O)C1)=O C(C)(C1=NOC2COCC12)NC.c1(C(CNC=O)N(CC)CC)ccc(Cl)cc1 C(=O)(C(CC)(CC)CC)N1CC(CCCC)N(C(C2CCOC2CC)=O)CC1 n1(CC)ncc(C(=O)N(CCCNC(=O)C(=O)Nc2ncc[nH]2)CC)c1Cl C1(NC(C2CC(C)(O)C2)=O)CC(C(N2CC(N3CC(F)C3)C2)=O)C12CCC2 C1(NC(CN(CCOC)C)=O)CC2CCC1CN2C(=O)CCc1cccc(O)n1 C#CCCCC(=O)N(CC(C)O)CCNC(=O)Cc1coc(C(F)F)n1 c1(C(=O)NCC(C(C)C)C(=O)NC2CCC=CCCC2)cccc2cncn12 c1(C(N(CCCN(C(=O)Cc2cc(Br)cs2)C)C)=O)ccc(Cl)cc1N C12(NC(C3CC(C)(C)C3)=O)CC(C1)N(C(=O)C(=O)NCc1ccc(F)cc1)C2 S(=O)(=O)(c1cnccc1N1CCC(O)CC1(C)C)NCc1cnc(OC)c(C)c1 CC(c1cnn(C)c1)=CC(N1CC(NC(=O)CSCc2ccccn2)CC1C)=O C1(NC(C2(OC)CCSC2)=O)CN(C(C2SCC=C2C)=O)CC1(C)C n1(CC)cnc2c(NC(C)(C)COC)[nH]c(=NCCNC(C)=O)nc12 c1(C(=O)NCC2(OC)CN(C(=O)Cn3nnc(C4CC4)n3)C2)cc(C)cnc1C CC(C1=CCN(C)CC1)NC(=O)C(C1CC1)NC(c1ccc(O)nc1C)=O c1(N2CCCC(NC(c3c(C)ncn3C)=O)C2)nc2ccccc2[nH]1 N12CC(C(C(=O)N(C(CSC)CO)C)C1)OC(=O)NCC2=O.CNCC C1(C(=O)NCC2(OC)CC2)C2CCCC2CN1C(=O)C(=CC1CCCC1)C C(C)(C(=O)N1CCC(C(=O)NC2CC(OC(C)C)C2)O1)OC N1(C(C2CN(CC)C(=O)C2)=O)CC(C)N(C(c2nc(OC)cc(C)n2)=O)CC1C c1(CC(=O)NCC2CCCC2C(F)(F)F)nnc(C(=O)O)s1 c1(NS(C(C)C#N)(=O)=O)ccnc(N=c2cncc(Cl)[nH]2)c1 C1(OC)(NC(CCn2cc(CNCCNC(C)=O)nn2)=O)CCOCC1 C1(NC(=O)Nc2ccc(Cl)c(Cc3nn[nH]n3)c2)Cc2cccnc2NC1=O C(C1CCCN1C)=CC(=O)NC(C1CN(C(c2coc(C(F)F)c2)=O)CCO1)C Cc1cc(C(=O)NCC2CC(NC(=O)C(C)c3ccsc3)C2)nc(N(C)C)n1 c1(C(N(C)C)=O)ccc(Br)c(C(=O)NCCCCc2cccc(Cl)n2)c1 C1(NC(Cc2n[nH]c(=N)s2)=O)CC2(C1)CC(CNC(=O)CC1CC(F)(F)C1)C2 Cc1oc(C(=O)Nc2ccc(CCn3cc(C(C)O)nn3)cc2)cc1Br Cc1ccc(C(=O)N(C)Cc2cn(Cc3ccc(Cl)cn3)nn2)c2c1NCCC2 CC(F)(F)CCCC(=O)N1CC(c2ocnc2CNC(c2ccc(O)o2)=O)C1 c1(C(=O)NCC2(O)CCCN(C(CCCC(C)=O)=O)C2)c(Cl)nc2sc(C)cn12 c1(C(=O)NC(C2CN(C(C3(C)CC3C(F)(F)F)=O)C2)C)nccc2cc[nH]c12 CC1C(NC(C2CCc3nn[nH]c3C2)=O)C(C)CCN1C(=O)CCC1(O)CCC1 C1(NC(C(C)NC(N)=O)=O)CCC12CN(C(=O)CN1CCNC(=O)C1)C2 N1(C(CC(CCCC)NC(=O)C=Cc2ccoc2)=O)Cc2ccc(O)cc2C1 C(c1ccc(F)cc1F)=CC(N1CC2C(NC(C3N(C)CCOC3)=O)(C2)C1)=O CCC(C)C(O)CC(=O)NC(C)C=CC(=O)NCC(F)(F)CC C1(C)(C(=O)NCCN(C(C(CC)(C)CC)=O)C)CCC(F)(F)CC1 c1(OC)cc(F)c(C(=O)NC2CC(NC(=O)CC34CCCC3C4)C2)c(F)c1 n1(CC(N2CC(CC(C(=O)NC3C(C)(C)OCC3)F)C2)=O)cc([N+](=O)[O-])cn1 c1(C(N(C2CCCOC2)CC#C)=O)cc(-c2cc(OC)ccc2OC)ccc1F C1(NC(c2cncc(CC)c2)=O)CCN(C(c2cocn2)=O)CC12CCC2 O=C(Cc1cn2c(n1)SCC2)N=c1ccc2ncc(Br)n2[nH]1 c1(CC(N2C(CNC(C3CC(F)(CO)C3)=O)CC(O)C2)=O)ccccc1[N+](=O)[O-] c1(C(=O)OC)cccc([N+](=O)[O-])c1CN1CCCC(CN=c2cc(C)nc[nH]2)C1 C1(C(N(C)Cc2ccns2)=O)CCC(C2CC2)N1C(c1ccnc(O)c1)=O c1(C(=O)NC(CNC(CC(CC)C)=O)(C)CO)cc(C)cc2c1OCC2 Cc1ccnc2nc(C(=O)NC(C)C(C)NC(C3(C#N)CCSCC3)=O)nn12 C1(CNC(=O)C(Cl)=CCl)CCN(C(c2cnc(-c3ccccn3)s2)=O)C12CCC2 C1(C(N2CCCCC2C2CCCN2)=O)CNc2cc(F)ccc2C1 C(=O)(C(C)(C)C(C)(F)F)NC1CN(C(C(C(C)C)F)=O)CC1(F)F N1(C(C2(COC)CCCC2)=O)CCC2CN(C(=O)CC3CCC(C)(C)O3)C2C1 n1(CCN2C(=O)CN(Cc3cc(C(F)F)on3)C2=O)ncc(=O)c2ccccc12 c1(C(=O)NCC2CCC(NC(c3csc(Cl)n3)=O)C2)cnc(O)c2ccccc12 C(=O)(C1CCCc2ccccc21)N1CC(NC(c2nn[nH]c2Cl)=O)CC2(C1)CC2 CC1C(NC(=O)Cn2nccn2)CCCN1C(=O)C(C)SC(F)(F)F c1(CN(C(c2c(CC)scn2)=O)C)cccc(CNC(C2OC3CCC2C3)=O)c1 c1(C(=O)NC(C(C)NC(C2CC(SC)C2)=O)C)ccc(C(C)=O)cc1F CC1CN(C(=O)C(C)c2ccco2)CCCN1C(=O)CCCc1ccccc1Cl c1(C(N2CCCC2)CNC(=O)NC(C=C)(C)C)cccnc1C c1(CC(N2CCC(CNC(=O)Cc3ccnc(O)c3)C2)=O)nc2c([nH]1)CCCC2 Cc1cc(=NC(=O)C(C2CCCO2)NC(=O)CC2SCCS2)[nH]n1C(C)C CC1C(C(=O)NC(C)CN2CCN(C(=O)C3=CCCC3)CC2)CCN1C c1(Sc2cccc(C(=O)OC3C(OC)CS(=O)(=O)C3)c2)nccn2nccc12 c1(C(N(CC(C)NC(=O)Cc2ccsc2)CC)=O)ncc(OCCOC)cn1 c1(C(=O)NCC2N(C(C(F)OC)=O)CCCC2C)ccnc2nccnc12 c1(C(=O)Nc2c(OC(C)C)nccc2)c[nH]c2ccc(F)cc2c1=O N1(C(C2CCCO2)=O)CCN(CCCNC(C2CC2c2ccccc2)=O)CC1 c1(C(=O)NCC2C3CN(C(C(CC4CC4)OC)=O)CC32)ccc(Cl)cc1F C(CCC(=O)N(C(C)C(=O)N(C)C(c1ncccn1)C)C)OC(C)C C1(O)(CCNC(C2CC(=C)C2)=O)CN(C(=O)C(C)(C)N2CCOCC2)C1 Cc1cc(C)c(CNC(C2CCC(CNC(=O)CC3CCC(=O)C3C)CC2)=O)cn1 n12nc(C3CC3)cc1C(=O)N2.C1(N(C2CN(CC)C2)C)CC(=O)N(CC)C1 C1(C(N2C(CCNC(C(c3ccnn3C)C)=O)CCC2)=O)CCCN1C=O C1(NC(CC(C)(C)OC)=O)C(C)(C)C(NC(=O)C(CCO)N(C)C)C1(C)C CN(C)S(=O)(=O)N(C)CC(=O)NC1(CNC(c2cnc(S)[nH]2)=O)CCOC1 Cc1ccc2c(c1)CC(C(N1CC(O)(C(C)NC(C3CCCC(=O)N3)=O)C1)=O)S2 C(=O)(CS(=O)(=O)CC(=O)NC1CCC(CNC(=O)C(C)(C)OC)CC1)OC CCC(C)C(O)C(=O)N(C1CC2CC1N(C(=O)C=Cc1ccccc1)C2)C C1(CC)C(NC(=O)C(C)CC(N)=O)CCCN1C(=O)CC1CC(C)(C)CO1 C(CCCOC)(C(=O)N1CCOCC(O)C1)NC(C(COCC)C)=O C1(N(S(C)(=O)=O)CCN2CC(NC3CC3)C2)CCN(Cc2cccnc2)CC1 c1(C(=O)NC23CC(NC(C(C4CCOCC4)C)=O)(C2)C3)cncc2nnn(C)c12 c1(C(N2CC=CC(NC(C3CCC(C)(CCOC)O3)=O)C2)=O)cc([N+](=O)[O-])cn1C c1(C(=O)NC2CC3(C2)CC(NC(=O)C(O)C2CCC2)C3)ccc2ncncc2c1 C1(C(N(CCNC(CN(S(CC)(=O)=O)C)=O)C)=O)CC(=O)N(OC)C1 N1(c2snc(SC)n2)CCC2(CCCN(CC(c3cnn(C4CC4)c3Br)=O)C2)C1 N1(C(C2=CC(O)C(NC(C3(C)CCSCC3)=O)C2)=O)CCC(O)(C2CC2)CC1 C=C(C)C(CC(=O)N(C)CCN(C)C(C1(CC)CN(C(C)=O)C1)=O)OCC C=CCCCC(C(=O)NCc1c[nH]nc1C1CC1)NC(C1CC(C2CC2)=NO1)=O c1(C(N2C(CNC(c3ccnnc3)=O)COCC2)=O)ccc2ncsc2c1 C(C(=O)NC(C)(C)CCCO)(C(C)O)NC(C1CC(CCC)C1)=O c1(C(=O)NC(C)C(C)NC(c2ccn(C(F)F)n2)=O)cc(=O)cc(Cl)[nH]1 CC(C)C(CCC(=O)NCc1nnn(C)n1)NC(=O)C(C)(C)CCC#N C1(NC(C2(OC)CC2)=O)CCC2(CCN(C(C3CCSC3C)=O)C2)C1 c1(SC)cccc(CC(N2CC3CC3(NC(C3CC=CCC3C)=O)C2)=O)c1 C1(C(=O)NC(C)(CNC(C2CCCC(C)C2)=O)C2CC2)(CC)CCOCC1 N1(C(CC2C(C)CCO2)=O)CC2CCCN(C(C34CCOC(C)(C3)C4)=O)C2C1 c1(CC)nc(C)c(C(=O)NC2CC(CNC(=O)C(C)OCc3ccccc3)C2)s1 C12(C(N3CC(NC(C4=C(C)CCC4)=O)C(CO)CC3)=O)CC3CC(CC(C3)C1)C2 CC(C)CC(O)C(=O)NCC1CC(CNC(=O)Cc2cccc(C(C)C)c2)C1 C1(NC(C(=O)NC2CCC(C)CC2)=O)CCN(C(C2CSC2)=O)CCC1CO C1(C(=O)NC(C)(CO)C2CC2)C2CCN(C(C3CN(C)C3)=O)CC12 N1(C(C=C(C)C)=O)CCC(NC(c2ccc(NC(=O)NC(C)C)cc2)=O)CC1C c1(OCCOC(C2OCCC2c2nc[nH]n2)=O)ccccc1F c1(C(=O)NC2(CC)CN(C(C(CC)O)=O)C2)ccc(Br)c(OC)c1 c1(N2CC(CNC(c3c(C)ocn3)=O)C(F)(F)CC2)ccc([N+](=O)[O-])c(C#N)c1 C(=O)(C1=NNC(C(F)(F)F)C1)N(CCCN(C)C)CCNC(C1COCCN1C)=O c1(C(=O)NCCCCNC(C23CC(C(C)C)(C2)C3)=O)cc2c(F)cc(F)cc2o1 n1(CCN2CC3CCC2C3)nc(C(=O)NC(C2CCCC(CC)C2)=O)cc1C1CC1 C1(CNC(Cc2c(C)scc2)=O)CN(C(=O)CCCNS(C)(=O)=O)CC1O C(=O)(CCC(C)(C)NC(C1C(C)(C)C1(C)C)=O)NC(c1ccccc1)C C#Cc1cc(NC(C2(C#C)CN(C(=O)C(C3CCCC3)OCC)C2)=O)cc(F)c1 C(c1cnn(C)c1)=CC(=O)N(CC(=O)NC1C(C)OCC1)C1CCC1 N1(C(CC2C(OC(C)(C)C)COCC2)=O)CC2CC1CN(C(c1cccs1)=O)C2 C1(C(C)C)COCCN(C(c2ccc(C(N)=O)o2)=O)C1.C12CN(CCO1)C2 N1(C(c2cn(C3CCC3)nn2)C(=O)NCC2CCCO2)CCCS(=O)(=O)CC1 N1(C(c2c(C)cc(CC)o2)=O)CC(C)C(Nc2nccc(C)n2)C(C)C1 CN1C(=O)CCCC1C(=O)NCC1CC(F)(F)CN1C(C12CCC(F)(CC1)C2)=O c1(CCCCC)nc(CN2CCC(C(=O)NCCO)C2)n[nH]1 C(=O)(CC(C(F)F)NC(C12CCC(C1)OC2C)=O)NCCC(COC)OC CC(C)CC(CNC(=O)C(C)S(N)(=O)=O)N=c1[nH]nc(C(C)C)o1 c1(CC(=O)NC2CC3CN(C(COCC(=O)OC)=O)C2C3)ccc2nonc2c1 c1(NC(C2CC3(CN(C(c4c(C)nco4)=O)C3)OC2)=O)ccc2ncccc2c1 C12(C(=O)NCC3N(C(C4CCOC4)=O)CCC3)COCC1CS(=O)(=O)C2 CCCCC(C)CCC(=O)N1CC=CC1(C)C(N1CCCC(C(C)(C)O)C1)=O C=CC(C)C(C)C(=O)NC1(c2cn[nH]c2)CCN(C(c2csc(C)c2)=O)CC1 N1(C(C2N(C(C(C)=NOCC#N)=O)CC=CC2)=O)CCC(F)(F)C(O)C1 N1(c2c(OC)cncn2)CCC(NC(c2c(Br)c(C)nn2C)=O)C(F)C1 C1(CNC(C=C(CCN(C)C)Cl)=O)CN(C(C2CCCCS2)=O)CC1C(F)(F)F N1(C(CSC(C)C)=O)CC(CNC(C2CCCN2CC(F)(F)F)=O)CC1(C)C C(C(=O)NOOCCOCCOCCOC1CC1)OCC#C c1(CN2CC(C(N(CCCOC=C)CCO)=O)OCC2)cc(C#N)n(C)c1 n1(CC)c(=O)oc2cc(NC(N3CCOCC(CO)C3)=O)ccc12 Cc1noc(CCC(=O)NCC(=O)NCc2ccco2)n1 C1(NC(CCSCC)=O)CC2CCC1CN2C(c1ncc(Cl)cc1Cl)=O N1(C(C2CC(=C)C2)=O)C2CCC1CC(CNC(=O)CCn1cc[nH]c(=O)c1=O)C2 Cc1nc(Cl)c2c(n1)CN(C(=O)Nc1cccc(CCO)c1)C2 c1(NC(C(CNC(CC2C(C)(C)CCO2)=O)CC2CC2)=O)cccc2c1CCC2 CN(C)S(=O)(=O)N(C)CC(=O)NC(C1(O)CN(C(C2CNC(=O)N2)=O)C1)C C1(CCCC)CN(C(=O)C=C=C(C)C)CCN1C(=O)C(C1CCOCC1)OC Brc1ccc(C=CCN(CCn2cccn2)Cc2cccnc2)cc1 c1(CCCC(N2CC3CC3(NC(C3(O)CC3)=O)C2)=O)ccc(Cl)c(Cl)c1 Cc1ccc(C(N)=O)cc1C(=O)N(CCC(C)NC(=O)CCc1cccs1)C c1(NC(C)(CCNC(=O)C(F)C(F)(F)F)c2ccccc2)cncc(C#N)n1 C=CCC(C(=O)N1CCCC(CC(=O)Nc2cc(C)cnc2OC)CC1)C(C)C N12CCCC(CC1)N(C(C1(c3nnco3)CCC1)=O)CC2=O.CCC(=O)NC1CC1 c1(C(N2CCC(CC)C2CNC(C2CCCCC2O)=O)=O)cccc(F)c1C c1(CC(=O)NC(CC(C)C)CNC(=O)CC2(CS(C)(=O)=O)CC2)cn2ccsc2n1 C1(NC(CCC(=O)NC)=O)COCCN(C(C2CC(C)=NO2)=O)C1 C1(C(=O)NCCN(C(C)C)C(C2(C(=O)OC(C)(C)C)CCC2)=O)CC2COCC2C1 c1(C2N(C(C(=O)NC(c3ncc(N)nc3)C3CC3)=O)CC2)cc(F)cc(F)c1 c1(C(N2CC3C(CNC(C(CC#C)C4CC4)=O)(C3)C2)=O)cc(F)c(C)cc1O CC(CC(C)(F)F)C(=O)NCC1(C)CCN(C(c2cnc(O)c(F)c2)=O)CC1 C1(NC(C=C(CCN(C)C)Cl)=O)(CO)CCN(C(=O)C(O)CC2CCCC2)C1 C12(C(N(CCN(C(=O)C(F)C(C)(C)O)C)C)=O)CC(C)(C1)OC2(C)C CN1CCCCC12CCN(C(c1cc(Br)n3c1CCC3)=O)CC2 c1(C(=O)NCCN(CCCCCC)C(C2CCCOC2)=O)ccc(OC)nc1F C1(F)(C(=O)NC(C#CCC)(C)C)CCCN(C(C2(C)CC(=O)N(C)C2)=O)C1 C1(CNC(c2c(C)nn(C(C)C)c2)=O)CCN(C(=O)CC2CC(F)C2)C1(C)C C(=O)(CCCCCO)NC1CCC(CNC(CCNC(COC)=O)=O)C1 c1(OC)cccc2c(CCNC3CC(C)CC(C)C3)c[nH]c12 N#Cc1ccc(NCCCNC(=O)Cc2nc(F)c(F)cc2F)c([N+](=O)[O-])c1 c1(N(C)CC)ccc(C(=O)NCCCCNC(=O)CCc2cccnc2C)cc1 C12(NCC(C)(C)SC)CC3CC1CC3ON(CCOCC)N=NN=C2 N1(C(C(CC(CC)C)NC(=O)CCc2nccs2)=O)CCC(C2CCCC2)C1 c1(NC(=O)NCC2CCC(F)(CC#N)C2)cc(F)cc2cccnc12 CS(=O)(=O)c1ccccc1CNc1cc(=NCC23COC(CC4CC4)(C2)C3)[nH]cn1 N1(C(c2cnc(C3CC3)s2)C(=O)NC2CCC2)CCOc2cc([N+](=O)[O-])ccc2C1 C1(F)(C(N(C)C)=O)CCN(C(c2cccc(-c3cccc(CO)c3)c2)=O)C1 c1(C(=O)N(CC2OCCN(C(CCNC(=O)OC)=O)C2)CCC)cccc2c1COC2 CCC(Cc1ccccc1)C(=O)N(C1CCCC1)CC1CCN(C)C1=O C1(=O)CC(O)CN1.c1(C(=O)NCCN(CC)CC)ccn(C2CC2)n1 N1(C(C(C(C)OC)NC(c2cnn(CCF)c2)=O)=O)CCCC(C(N)=O)C1 CCCCC(C(=O)NCC(C(C)C)NC(=O)CCOc1ccccc1F)OC N1(CC)CCOCC1C(=O)NCCCCCNC(c1scnc1C(C)(C)C)=O c1(C(=O)NC2C(CNC(c3cc(C)sc3Br)=O)C2)cnc2[nH]nnc2c1 c1(CCC)nc(=NC2CC(NC(C3CCC4CCCCC4C3)=O)C2)s[nH]1 C1(CCOC)(NC(=O)C#CC2CC2)CCN(C(C2(S(N)(=O)=O)CCCC2)=O)CC1 c1(CC)nccnc1C(=O)NCC(c1ccccc1)CNC(=O)C(F)CC N1(C(N2CCC(CC#C)(C(=O)OC)CC2)=O)CCNC(=O)c2c(Br)cccc21 Cc1cccc(N2CCC(NCCCC3CC(C)OC3=O)C2=O)c1 N1(C(C2N(C(C3CC(OC)C3)=O)CC2)=O)CCC(OC2CCCCC2)C1 C1(CN=[N+]=[N-])CCCN(C(C2CCCCN2C(=O)C=CC2CCCC2)=O)C1 CN1CC(NC(c2ccc(CNC(=O)CCn3ccnn3)cn2)=O)CC12CCC2 CON(CCCO)C(=O)C1(NC(c2cccc(OC)c2)=O)CCN(C)C1 c1(C(C)=O)[nH]c(C)c(C(=O)NC(CNC(C2(C)CC(O)CN2C)=O)C(C)C)c1C N1(C(c2c(C(C)C)con2)=O)CCC(C)N(C(c2conc2C)=O)CC1 Cc1cn2c(C(=O)NCCC3CSCCN3C(c3cnn(C)c3C)=O)cnc2s1 N1(C(c2c(-n3c(C)cc(C)n3)cccc2)=O)CCCC12CCN(C(=O)C1CC1)C2 C1(C(=O)NC2CCCCCN(C(CCCCOC)=O)C2)CC2COCC(C1)C2=O Cc1ccc(C)c(C(N2CC3(NC(C4CCCOC4)=O)CCC2C3)=O)c1O N1(C(c2c(COC)noc2)=O)CC(Nc2ccc(SC(F)(F)F)nc2)CC(F)C1 c1(NC(=O)NC2CCC2C(F)(F)F)ccccc1OCc1cnsc1 N1(C(C(CCCC=C)NC(=O)C(C)CC(=O)OC)=O)CCc2oc(C)nc2C1 Cn1cc(C(=O)NCC(CNC(=O)Cc2cccn2C)CO)nn1 c1(C(=O)NC(C(C)(C)C)C2CC2)ccc2cccc(F)c2n1 N1(C(C=CCOCCOC)=O)CCCC(C(C)N(C)CCC)C1.C(C)(=O)N C(=O)(CCCCCC#N)NC(c1cn(CCC2(CN(C)C)CCOCC2)nn1)C C1(C(=O)NCCCCSC)N(C(C2CCC(F)(F)C2)=O)CCC1(C)C CC1(C)CC(Nc2ccc([N+](=O)[O-])cc2)CN(C(c2ccc3scnc3c2)=O)C1 N1(C(c2cn(CC=C)nn2)=O)CCOC(C(=O)Nc2conc2C2CC2)CC1 N1(C(C(CC(=O)OC)NC(C)=O)=O)CC(NC(=O)CCCCOC)C2CCCC12 C(=O)(CCC(=O)N(C)C)NC1N(C(=O)NCC2C(c3c(C)ncs3)C2)CCC1 c1(CC)cc(C(=O)NC2CCCC(CF)C2)cc(Cl)c1.N12CC(C)(C1)NC2=O c1(C(=O)NCC(CC)NC(C2(C#N)CC3CC3C2)=O)c(F)ccc(C)c1F c1(C(N2CCCC(C(=O)NC34CCN(CC3)CC4)C2)=O)c(F)cccc1F c1(C(=O)OC)nnc(S(=O)(=O)N2CCN(CC(=O)OC3CCCC3)CC2)s1 CCC(C)(C)C(O)C(=O)NC1CCCCCN(C(=O)C=Cc2cccs2)C1 c1(SC(CC)C(=O)NC(c2ccccn2)CO)cccc(Br)c1 c1(C(N(CC(CC)NC(c2ccc(Br)o2)=O)C)=O)ccc(-c2nc[nH]n2)cc1 C(C(C(C)(C)C)NC(c1ocnc1C(F)F)=O)NC(C(C=CC)O)=O CCCCC(CC)CCCNC(=O)C(=O)N(c1ccc(C)c(C(F)(F)F)c1)C N1(C(c2nc(CCC)oc2)=O)CCCN(CCNC(c2ccc(F)nc2F)=O)CC1 c1(CC)ccc(C(N2CC(NC(=O)C(C)n3cncn3)C3(CC3)C2)=O)cc1Br c1(C(N2C(C(=O)NCCc3n(C)cnc3)C=CC2)=O)cccc(CO)c1 N1(C(CC(C)(C)OC)=O)CCOCC(C)(CNC(c2cncc(C)n2)=O)C1 c1(C(N2CC3C(CNC(C4C(C)C4C)=O)(C3)C2)=O)occ2c1CCC2 c1(C(=O)NC(CC)CNC(=O)CCc2nc(O)n[nH]2)cc2c(o1)CCCNC2=O c1(NC(CC(=O)NCC#C)=O)ccc(C(=O)NCCN(C)C(=O)N(C)C)cc1 N1(C(C(CC)C)=O)CCC(C(=O)Nc2ccc(NC(C)=O)c(C)c2)C(F)(F)C1 c1(NC(C(C2CCOC2)NC)=O)cccc(CNc2nnnn2C2CCC2)c1 c1(C2(C(=O)NCC(C)N(C(=O)COC3CC3)C)CCCC2)ccc([N+](=O)[O-])cc1 C1(C(=O)NCC(C)CNC(c2cnc(S)[nH]2)=O)CC2(C1)CC(O)C2 C1(CC(=O)N(C)CC2CCCN(C(=O)C(C)CCO)C2)CC2CCC(C1)C2 C(CCCCC(=O)N(C(CC(F)F)C(=O)N1CCC(C(C)(C)COC)C1)C)OC C(=O)(C(CC(C)C)NC(=O)CSc1cc(F)ncc1F)OC c1(C(N2CCN(C(c3ccoc3)=O)C3CC23)=O)cccn2cncc12 C(=O)(CC(C)(C)C(F)F)NCCC(CNC(C(CC)n1ccnc1)=O)O N1(C(C(C2CC2)OCC)=O)CCCN(C(=O)C(C)C(C)C)CCNC1 CCC(CNC(c1cc(C(F)F)[nH]n1)=O)(CC)C(=O)N1CCC2(CCC2)C1 c1(C(=O)NCC2C(NC(c3cc(OC)nn3C)=O)COCC2)cnc2n1CCS2 CCC(CC)C(C(=O)NCC1CCCN1C(c1sccc1C#N)=O)OC N1(C(C(=O)Nc2ccccc2)=O)CC2C(N)CS(=O)(=O)C2C1.CC1CCN1 C1(CC)CCCCC1C(N1CCC(CO)(CNC(=O)C(C)SC(F)(F)F)C1)=O C(CC(CNC(=O)CC1CNC(=O)C1)NC(=O)Cc1csc(C(C)C)n1)OC N1(C(C(C)(C)NC(c2cnc(C)c(Br)c2Cl)=O)=O)CCC2COCC2C1 C1(N(C(CC(C)F)=O)C)CCC2(CC1)CCN(C(c1cnc3occc3c1)=O)C2 C1(F)(CNC(CCSCC(C)C)=O)CCCN(C(C2CC(C)(C)CO2)=O)C1 CCCCCCCC(=O)N(C)CCC1CCCCN1C(C1CC(=O)CCO1)=O c1(OCC)ccc2c(c1)CC(C(=O)NC1CC(NC(=O)C(C)(CC)OC)C1)CO2 C1(N(C(=O)CC(C)(O)C2CC2)C)CCCN(c2nnc(C#N)s2)CC1 c1(C(=O)NC2(CNC(c3cc(CC)[nH]n3)=O)CCCCC2)ccc2nn[nH]c2c1 C(=O)(C(C)(C)C1CC1)NCC(CN(C(CNC(CCC)=O)=O)C)C C(=O)(C#CC1CCCOC1)N1C(COC)CN(C(c2cccn(C)c2=O)=O)CC1 N1(C(CCc2n(C)ccc2)=O)CC(O)CCC1C(=O)NCC1OC(=O)CC1(C)C N1(C(C(COC)O)=O)CCn2ncc(CNC(c3cc(Cl)ccc3Cl)=O)c2C1 C1(N(C(c2ccn(C(C)C)n2)=O)C)CCCC(NC(c2cnc(N)cn2)=O)C1 CC1(C)CC1(C#N)CNC(C1CC(n2cc(Br)nn2)C1)=O C1(C(N2CCC(C(F)F)(CNC(CP(C)(C)=O)=O)C2)=O)CCCCC12OCCO2 c1(CCC)cc(C(=O)NC(C2CCCN2C(C2C=CCCC2)=O)C)n(C)n1 O=C(C#CC1CCCCO1)N1CC2(CCC2)CC1CNC(=O)CC1CCCC1 CCC(CCO)C(C)NC(C1C2CC1(c1ccc(OC)cc1)CO2)=O O=C(C1=CCCCCC1)N1CC(C(=O)NCCc2ccon2)C2(CCC2)C1 N1(C(C2C(C)CCCC2)=O)CCC(C)C(CNC(C2CCC3CC3C2)=O)C1 c1(C(N2C(C)(C(N(C3CCCC3C#N)CC)=O)CCC2)=O)cccc(Br)c1O c1(C(N(CCNC(C2CC(C)(F)C2)=O)CC)=O)ccc(N(C)C)c(F)c1 c1(OC)ccc(Br)c(CN2CC(C)(CC(=O)NCc3cnc(Cl)cc3Br)C2)c1F c1(CNC(c2cn(CCNC(C(C)(C)NC(=O)OC)=O)nn2)=O)cnc(C)cn1 O=C(CC1CCOc2ccccc21)OCC1(c2ccccc2)CC1(F)F C1(CC)CCC(C(=O)NC(C)C=CC(=O)NCC2(C3CC3)CC2)O1 CN1C2CCCC1CN(C(c1cnc(C3CC3)[nH]1)C(=O)NCCC1(C)CC1)CC2 CC1=CCN(C(C2(NC(=O)CNc3cccnc3)CC2(C)C)=O)CC1 C1(N(CCCC=C)CCc2ccc(Cl)cc2)CCOC(C)(C)C1 c1(CC)cc(OC)ccc1C(N1CCOCC1)C(=O)NCc1ccc(C)n1C N1(C(=O)Cc2cnsc2)CC2=C(C1)CN(C(=O)C(c1ccc(Cl)cc1F)O)C2 N1(C(c2cn(CC=C)nn2)=O)CCC(NC(c2sccc2F)=O)C12CC2 c1(OC)cnc(Cl)cc1C(N1CCN(C(=O)CCOC2CC2)CC1COC)=O c1(NCC(S(=O)(=O)NCC)C)ncccc1S(=O)(=O)NCc1csc(CC)n1 C1(CC)CCCN(C(C2CC(O)CN2C)=O)C1C(=O)NCC1CCN(C)C1 N1(C(C)C(=O)ON)CCN(C)CC1.c1(Cc2cc(C(C)(C)C)on2)ccccc1 C(=O)(C1CCCc2c1ncn2C)N1CC(NC(C(C)SCC)=O)CC12CCC2 c1(CNC(c2ccc(CNC(C3(SC)CC3)=O)nc2)=O)cnc(O)c(F)c1 O=C1NC2(CCN(Cc3ccccc3)CC2)Nc2ccccc2N1 c1(OC)ccc2[nH]c(=O)c(NC(c3cc(C)sc3N3CCOCC3)=O)cc2c1 C1(CNC(=O)CCn2ccnn2)CCC2(CCC2)C1NC(=O)C(Cl)=CCl N1(C(c2cc(C)cc(O)c2)=O)CCCC2(CCCCC2NC(c2cnc[nH]2)=O)C1 n1(C(C(=O)N(CCC2CC(NC(CCC3C(C)C3)=O)C2)C2CC2)C)cnc(C#N)n1 CC(CCCNC(=O)CCc1cncs1)NC(=O)C(F)C1CCC1 N(C1CCOc2c(Cl)cc(Cl)cc21)C(C(=O)Nc1cccc(Br)c1)=O N1(C(C(CC)C(C)C)=O)CCC2(CC1)CC(NC(C1CCCCS1)=O)C2 C1(C#N)(C(=O)NC(C(C)NC(Cc2c(C)cnn2C)=O)C)CCOCC1 c1(CC)ccc(Cc2nc(C)n(CC)c2C)c(C(c2noc(CC3CC3)n2)=O)c1 O=C(C(Cc1ccccc1)CC(F)F)Nc1cc(-c2ccccc2)nn1CCO Cc1cc([N+](=O)[O-])nn1C(C)C(=O)N(CC(O)C1(Cl)CC1)C N1(C(c2c(CC)c[nH]n2)=O)CCOCC(NC(c2oc(C3CCC3)nc2C)=O)C1 C1(=O)C(C)C(C)N1.C(=O)(C(C)C)NCCNC(C)=O.C(CCO)CCC c1(C(=O)NCC2C(C(=O)NC(CCC)C)OCC2)cc(CC)nn1C C1(OC)(CNC(=O)C(C)SCC2(Br)CC2)CN(C(C2CCCC2)=O)C1 C(=O)(C(O)(C(F)(F)F)c1cn[nH]c1)N1CCN(C(C(c2n(C)ccc2)=O)=O)CC1 C1(NC(COCC=C)=O)CC(NC(=O)C(C)Cc2ccnn2C)CC1O c1(COCCN(CC=C)CCC)ccc(C2(F)COC2)cc1 c1(C(=O)NCC2N(C(C(CCCC)O)=O)CCN(C)C2)c(F)ccc(C)c1Cl N1(C(C(CC(=C)Cl)NC(=O)CC2CCC(=O)N2C)=O)CCC2(CCC(O)C2)C1 C1(CCNC(N2CCSCC2C2CC2)=O)CC12CCOC2 N1(C(C(C)OCCCC)=O)CCOCC(CNC(C2CN3CCN2CC3)=O)C1 Cc1ccc(Br)c(C(N2C3CCC(C3)C2C(=O)NC(C(C)(C)C)C2CC2)=O)c1F c1(SC)ccc(Br)cc1C(=O)NCC1C=CCN1C(c1cccnc1)=O Cc1nc(O)ccc1C(N1CCC(C)CC1C(=O)Nc1c[nH]ccc1=O)=O Cc1cc(C(=O)NC2(C)CCN2C(=O)COc2nc(C)ncc2F)c(Cl)cc1F C(N=C(NCCNS(C)(=O)=O)NC1CC1)c1c(C(C)C)ncs1 CCC(C)CCCCC(=O)N1CCCC(Cc2cn(Cc3cnns3)nn2)C1 CCC(CCOC)C(=O)N1CC(n2cc(C(C)(C)C(=O)NC(C)=O)nn2)CO1 c1(C(N(C2CCN(C(=O)CCc3cncnc3O)C2)CCC)=O)ccc(Cl)cn1 C1(C(=O)NCCCOC(C)C)CC(C)(C)CCN1C(=O)CC1CCOCC1 CC1CN(C(=O)NCCOc2cccc(C(c3ccccc3)=O)c2)CC(C)(C)C1 N1(C(C2CC(NC(c3occ(C)c3)=O)C(O)C2)=O)CCCC(C)(C)C1C C1(C(N(CCC)C)=O)CN(C(C2CC3(CC3)CO2)=O)C2(CCC2)C1 c1(C(=O)NCCOCC=C)cnc2c(c1)CCN(Cc1cnc[nH]1)C2 c1(C(N(CC(=O)NC2(CCCC)CC2)CC#C)=O)ncccc1N(C)CC c1(C(N2C3CC(CNC(c4c[nH]c(=O)cn4)=O)C(C3)C2)=O)n[nH]c2ccc(F)cc12 N1(C(COc2cccc(CC)c2)=O)CCN(C(c2ccnnc2C)=O)C(C)C1 c1(C(=O)NCC(C2CCCCC2)NC(=O)CCc2cnoc2)sccc1Cl N1(C(c2c(CCC)[nH]cc2)=O)CC(NC(c2ccsc2C(F)F)=O)C2CCCC12 Cc1nccn1CCN(C(=O)CN(C(=O)CCc1nccn1C)C)C C(=O)(C(CN(C)C)NC(C1CCOCC1)=O)N(C(C#C)C1CCC1)C NS(=O)(=O)C1(C(=O)NC2CCN(C(=O)CCCCc3ccccc3)CC2)CCC1 c1(C(=O)NC(CNC(c2nc(C(C)OC)oc2)=O)(C)C)ncc(Br)cc1N Cc1cc(C)n2nc(COC(c3csc(Cl)c3)=O)nc2n1 c1(C(N(C)CC2(O)CCN(C(=O)CCF)CC2)=O)n[nH]c2cccnc12 c1(C(=O)NCCN(C(=O)CC2CC2(Cl)Cl)CC2CC2)cccc2c1CCO2 N1(C(c2c(CC)cc[nH]2)=O)CCCCCCC1C(=O)NC1COCC1OC C(=O)(CCCCCCCCCc1ccccc1)N(C(c1cc(C)on1)C)C N1(C(c2c(Cl)cnc(OC)n2)=O)CC2CC(NC(c3cnc4sccn34)=O)CC1C2 C#Cc1ccnc(C(=O)OC(C)=O)c1.C(=O)(C1CO1)OC Cc1cc(CNC(C2CCCCS2)=O)oc1C(N1CCC(CO)C1)=O C12(C(N(CCNC(c3csc(COC)n3)=O)CC)=O)CCCC(C1)OC2 C1(CNC(c2cc(C)c(C)o2)=O)CN(C(c2ccc(N)c(O)c2)=O)CCC1(C)C CCCC(C)(CO)n1nnnc1C1N(C2(c3ccccc3F)CC2)CC1(C)C C=Cc1cc(C(=O)N(C2CCCCN(C(=O)C3=CCCCC3C)C2)C)cc(F)c1 CC(C)CC(C(=O)N(C1(CNC(=O)CC2CC3(CC3)CO2)CC1)C)NS(C)(=O)=O CC(C)C(O)CC(=O)N(C(C)CC(=O)NCCn1cncn1)C C1(C(=O)OC)C(C)OCCN1C(c1cn(-c2cc(F)cc(F)c2)nn1)=O CCC(C)(F)C(=O)N1CCC(NC(=O)Cn2cc(-c3ccccc3)nn2)C1 C1(CC(C)NC(CC(=C)C)=O)CC2CCC(C1)N2C(=O)CSc1ccc(C)cc1 Cc1[nH]c2cccnc2c1CNC1CCN(CCC(C)C)CC1 N1(C(c2ccnc(C)c2N)=O)CCC2(CC1)CN(C(=O)C(C)C(C)C)C2 N1(C(C2CC(C#N)C2)=O)CC(F)CC1CNC(C1(N(C)C)CCC1)=O C(=O)(CCCCCN(C(=O)CC1(OCC)CC1)C)N1C(CCC)CCC1 Cc1cc(CC(C)NC(=O)C(C)CNC(c2scnc2Cl)=O)n[nH]1 C1(CNC(C2(CO)CCOC2)=O)COCCC1(F)F C12(NC(C(C)NC(N)=O)=O)CC(CNC(=O)CC(F)F)(C1)OC21CCOCC1 c1(NC(C(N2C(CS(C)(=O)=O)CCC2)=O)=O)c[nH]c2cc(Cl)ccc12 c1(OC)ccc2c(c1)CCC(C(=O)NC13CC(NC(C4CCCC4O)=O)(C1)C3)C2 c1(OC)ccc(C(=O)COC(c2[nH]nnc2C(=O)Sc2ccc(Br)cc2)=O)cc1Cl c1(C(=O)NCC(CC)NC(=O)CCOC(C)(C)C)cc2n(n1)CCN(C(C)=O)C2 C=CC(C)C(=O)N(C(C)CC(=O)NCC(C)(C)COC)C C1(C)(C(=O)NCC(CC)(C)NC(=O)CN2CC(F)(F)C2)CC2CCC1C2 N1(Cc2cn(CC)nc2)c2ccccc2CC1C(N1CCC(O)C(C(=O)OC)C1)=O C(N=c1nc2c(ncn2C)c(NCCCS(N)(=O)=O)[nH]1)c1cnn(CCC)c1C C(CC(C)(C)C(=O)N1CCCC(C(N2CCC(CCC)C(C)C2)=O)C1)OC N1(C(COC(CC(CCC)c2ccccc2)=O)=O)CC(=O)NC(C)(C)C1 C12(CO)CCC(CC1)N(C(C1(NC(c3cc(C)nc(C)n3)=O)CCC1)=O)C2 N(C1COc2cc(Cl)ccc21)C(=O)CC(C(F)(F)F)N1CCOCC1 S(=O)(=O)(c1ccc(NC(c2ccccn2)C)s1)N1CC(C(=O)OC)C(F)(F)CC1 C(=O)(N(C)OCC(F)(F)F)C1C(C(c2ccccc2)C2(C(=O)OC)CCC2)CC1 CC1CC(C(=O)NCc2ccc(Cl)nc2)CCN1C(c1cc(CN(C)C)n[nH]1)=O N1(C(c2c(CC)cccc2)=O)CCC(F)CC1C(=O)NCCCP(C)(C)=O C1(C(N2CCCC(N(CCO)Cc3cncc(C4CC4)c3)C2)=O)CCCC1(F)F N1(C(c2c(F)ccc(C)n2)=O)CCC2(CCCC2NC(=O)CCc2ccon2)C1 C12(CCO)CN(C1)C2=O.c1(C(C(=O)C=CC2CC2)=O)cnccn1.N C(=O)(CCCCCCCC(=O)OC)NCC1C(NC(C2C(OC)C2)=O)C1 N1(C(C=CC)=O)CCCOC(CNC(=O)C(C)CC(F)F)C1 c1(OC)cccc2c1C(C(=O)NC1CCN(C(=O)C=C(C)Cl)CC(C)(C)C1)CC2 C(=O)(C(C)CC(C)C(C)=O)NC(COCC)C(=O)NCc1conc1CN(C)C c1(C(N2CCC(O)(C(C)NC(=O)C=CS(C)(=O)=O)C2)=O)cccc2c1NCCC2 C1(N(C(=O)CC2CC2(Cl)Cl)CCC)CCN(c2nc(CC)ns2)C1 c1(NCC2NCCC(C(=O)OCC)C2)cc(Cl)c(OC(F)F)cc1Cl C1(C(N(C)Cc2cnsc2)=O)C=CCN1C(=O)CCc1nncn1C N1(C(C2CCCC2Nc2ccccc2S(C)=O)=O)C2CCC1CC(N(CC)CC)C2 C1(C(=O)NCc2c(CC)ccnc2)CCN(C(=O)C(C(C)CC)NC(C)=O)O1 C(=O)(C(F)C(F)(F)F)N1C(CNC(C(C=C)C)=O)CCC1 C(=O)(C(COC)CC(C)C)N1CCC(O)(CCNC(CC(C=C)(C)C)=O)C1 N1(C(c2ccccc2SC2CCCC2)=O)CCC(F)(F)C(Nc2ccncn2)C1 Nc1cc(C(N2CC(CO)(NC(=O)Cc3cscn3)C2)=O)cnc1N O=C(C1=CCCOCC1)NC1CC(NC(=O)Cc2ccc3c[nH]nc3c2)C1 c12nc(C)oc1NCCC1CC(C1)NC(=O)c1cc([nH]n1)CC(=O)OC2=O.CC N1(C(C2CCC(C)C2)=O)CCCC(C2CC2NC(=O)C(C)OCCN(C)C)C1 Cc1nnc2n1CCC(C(=O)NCC1(NC(c3ncc(C#N)cc3Cl)=O)CC1)C2 c1(CCC(=O)NC2(CCO)CN(C(C=CCN(C)C)=O)C2)cccnc1Br C1(C#N)(C(N(CCNC(=O)CCNC(c2cccc(Cl)c2)=O)CC)=O)CCOC1 Cc1ccccc1C(C)(C)C(=O)NC(C)CN(C)C(C1CCN(C)C1)=O N1(C(C(COC)OC)=O)CCOC2CCN(C(c3cccc[n+]3[O-])=O)CC12 c1(OC(C)(C)C(N2CC(NC(c3cccs3)=O)C2(C)C)=O)c(F)cccc1F Cc1cn2c(CC(N3CC(C(=O)NCC(C)(C)N(C)C)CC3(C)C)=O)csc2n1 C(=O)(C(C)(C)COC(C)(C)C)NCC(CN(C(=O)CC1SC(=N)NC1=O)C)(C)C C(C1OCCc2ccccc21)(C1CC1)NC(=O)Nc1cnc(O)c2ccsc12 CCC(CC)CCCC(=O)NCC1CCC(C(=O)NOCc2ccncc2F)O1 C1(C#N)(C(CNC(=O)OC)(F)F)CCN(C(=O)OC)CC1.C1(C(F)F)CCN1 c1(C(=O)NC(CC)CNC(=O)CCC#N)ccc(C2CCC(=O)N2)cc1 CC(C)C(O)C(F)(F)C(=O)NC1C=CC(CNC(=O)CCCC(F)F)C1 CCCCS(=O)(=O)CC(=O)NC1CC12CC(NC(=O)CNC(=O)NC)C2 C1(CNC(CCN(C(=O)Cc2cnn(C)c2)CC=C)=O)CC=C(C)CC1 C(=O)(CCCCCc1nn[nH]n1)NC1CCN(CCOC)C1 c1(C(=O)NCC2(C)CC(NC(c3nscc3Br)=O)C2)coc(C#N)c1 c1(-n2c(C3CCSC3)nc(-c3ccc(N(C)C)cn3)n2)ccc2c(c1)OCCO2 CC1CCC(CNC(C2CCCC(O)C2)=O)N(C(=O)CC2(C)CCC2)C1 c1(C(N2C(C)(CNC(C(CC)NC(N)=O)=O)CCC2)=O)cnc2ncccn12 CC1CN(C(=O)CCc2cscn2)CC1CNC(c1cccc(C2CC2)c1)=O CC(CC(=O)NC1(CNc2ccccc2)CC1)CC(F)(F)F c1(N2CCC(C)(CC)C2)nc(=N)[nH]c(=NC2CC2CC)[nH]1 c1(CCNC(C2(CC)CC2)=O)cncc(C(=O)NCC2=NOC(C)C2)c1 C1(NC(=O)CC(F)(F)Br)CN(C(c2c[nH]ccc2=O)=O)CCC1F C1(c2c(C)c(I)ccc2)CCC2(CC1)CNC(=O)C2 N1(C(c2ccc(C)c(C(F)(F)F)c2)=O)CCC(C)(C)C(CNC(=O)C(C)SC)C1 N1(C(CN2CCC(N(C)C)CC2)=O)CCC(NC(C2CC2C2CC2)=O)C(C)(C)C1 C1(C(=O)NCC(C)(C2CC2)NC(C(=O)NCCOC)=O)CC(C2CC2)=NO1 c1(-c2cccc(OC)c2C)ccc2cc(C(N3CCC(C)C3)=O)cn2c1 C1(C(N2CC3C(CNC(c4coc(C(F)F)n4)=O)(C3)C2)=O)CS(=O)(=O)CCO1 C1(NC(CSCC#C)=O)CN(C(=O)CCSc2ccccn2)C2CCCC12 c1(OC)ccc2c(C(C)(C)O)cc(C(=O)NC3CC3C(=O)NC3CCC3)nc2c1 N1(Cc2ccc(C)o2)CCC2(CC2C(=O)O)C1 CCCC(O)(CCC)CC(=O)NC1(C)CCN(C(c2coc(COC)n2)=O)C1 Cc1nc(O)ccc1C(N1CCCC(N(C)C(C2CC3(CCC3O)C2)=O)C1)=O C1(C(N2C(CNC(c3c(C(C)C)ocn3)=O)CC2)=O)CC2(C1)CC2(F)F C1(NC(C2C3CCCC23)=O)CCN(C(c2ccsn2)=O)C12CCC2 c1(OC)c(NC(=O)C(C)N(C)C(C2(C)CCC2)=O)cccc1F n1(Cc2ccc(C(C)N)cc2)ccc2c(C(F)(F)F)cccc12.C1(C)CCCN1 O(P(C)(=O)CNC(C1CC(C)CN1C(=O)CCC1CCOC1)=O)CC N1(C(CCC(C)C)=O)Cc2ccccc2C(NC(C2CCC=CCCC2)=O)C1 N1(NC(C2(CC)CCN(C(CNC(=O)OCC)=O)C2)=O)CCc2ncncc2C1 n1(C(C)C)nncc1C(=O)N(C)CC1CCN(C(C2CC(O)(C(F)(F)F)C2)=O)C1 C(=O)(CC(O)CC(C)(C)C)N1CCC(COC)(NC(c2[nH]cc3c2CCC3)=O)C1 C1(C(=O)Nc2c(CC)cccc2)CCN(C(=O)CCCCCNC(C)=O)C(C)C1 N1(C(C(C(C)C)O)=O)CCN(C(=O)C=Cc2nccs2)C2COCC12 CCC(C)(C)C(O)C(=O)NC(C12CCC(CC1)C2)CNC(=O)Cc1ccccn1 CC(CN=C(NCc1cc(OC)ncn1)NC1CCOCC1)N1CCOCC1 CC1CN(C(C2CN(C(c3cccnn3)=O)CC2(C)C)=O)CC(C2CC2)O1 N1(N2C(C(C)C)CC2)CCCCC1C1(C=O)CC1.C(=O)CCCC1CCCO1 C(CC(C)C(=O)NC1(C(N2CCSCC2C)=O)CC(C(=O)OC)C1)=CCC c1(COC)cc(F)c(N2C(CC(CCC)C(=O)OC)CCCC2)c(F)c1 C(CNC(C1CCN(C(=O)CC)CC1)=O)(C(C)C(C)C)NC(CCOCC#C)=O c1(NC(C2CC(N(C(C(COC)OC)=O)C)C2)=O)ccc(O)cc1F C(=O)(CCCCCN(C(=O)C=CC1CCOCC1)C)NC(C=C)C(F)(F)F c1(N(C)C(C2CC3(CC(NC(C4CC5CCC5C4)=O)C3)C2)=O)cccc(C#N)c1 S(=O)(=O)(c1cccc(Cl)c1F)N1CC(OC)C(NC(C2CCCCO2)=O)CC1 N1(CC)CCC(NC(C2CCN(C(=O)Cc3cc(C)[nH]n3)CC2)=O)C1=O C1(NC(C=CCN(CC#C)C)=O)CCCC1CNC(=O)CC1C=CCC1 Cc1c(CC(=O)NC(C)C(C)NC(c2ncn(C)n2)=O)ncn1C N1(C(c2c(C)scn2)=O)CCCCC(CNC(c2ccc(=N)[nH]n2)=O)C1 C1(C(=O)NC(C2CCCCC2)CNC(CC=C(C)C)=O)CCCC(=O)N1C C(=O)(C1=C(C#N)CCC1)N(CCCNC(c1cc(C)n(C)c1)=O)CC c12cccc(c1)N2.c1(CC(=O)NC(CNC(C=CC)=O)(C)C2CC2)[nH]cnc1C CCC(CC)C(F)C(=O)N(C1(CC(=O)NC2COCC2(C)C)CC1)C N1(Cc2c(Br)ccc(C#N)c2)CCc2cc(F)ccc2C1 CC(CC(=O)NCC1(O)CCN(C(c2ccc(C(F)F)cn2)=O)CC1)P(C)(C)=O CN1CC2CCC(C1)N2c1nccc(-c2n[nH]c3c2CN(C(=O)C(F)F)C3)n1 C1(CC=C)(NC(C2CCCOCC2)=O)CCN(C(=O)CCCn2ccnc2)C1 N1(C(C(=O)NC(c2cnc3sccn23)=O)=O)CC(N)CC2(CCOCC2)C1.CC=CC N1(C(C2(C(C)NC(CCC=C)=O)CC2)=O)CCC(C)(O)C(O)C1 C12(NC(C(CC)OCC)=O)CC3CCC(C1C2)N3C(=O)C(c1ccc(Cl)s1)=O Cc1ccc(C(N2CCN(C(=O)C=CC3CC3)CC2C)=O)c(N)c1C C12(C(N3CCC(=CCNC(c4c(C)nco4)=O)CC3)=O)CCC(C)(CC1)OC2 N1(C(c2csc(C)n2)C(=O)OCC)CCOC(C(=O)Nc2nnc(COC)s2)C1 c1(CC(=O)NCC2CC(O)(CNC(=O)C3CC3)C2)cncnc1O C1(NC(C2C3(N(C(c4cccc(C)c4O)=O)CC3)CC2)=O)CCN2CCCC2C1 N1(C(COC(CC)(C)C)=O)CC2CCC1C(NC(c1ccc(NCC)cc1Cl)=O)C2 C(N=c1[nH]cnc(Cl)c1C#N)C1CCCN(C(Cc2n(C)nc(C(F)F)n2)=O)C1 CP(C)(=O)c1cccc(NC(=O)C(=O)NC2CC3CCC2CC3)c1 N1(C(C(C)CC(F)(F)F)=O)CCC2CN(C(c3cc(O)cc(O)n3)=O)CC2C1 c1(C(=O)NC(C)CN(C(=O)CC2COCCO2)C)cc(Cl)c(F)c(Cl)c1 C1(C(=O)NC2CC3N(C(CC(=O)OC)=O)C(CC3)C2)CC(F)(F)CCC1(C)C N1(CC(=O)NCC2(CNC(C3N(N=O)CCCC3)=O)CC2)CCCCCCC1=O N1(C(c2c(C(=O)OC)noc2C)=O)CCC(O)C(NC(=O)CCCC(N)=O)C1 N1(CC(COC)O)CCCC(CCNC(=O)Cc2ccccc2OC(F)F)CC1 Cc1nc(C(F)(F)F)c(C(=O)NCC(C2CCCN(C(C3(F)CC3)=O)C2)(C)O)o1 c1(C(=O)OC)cnc(N2CC3CC(NC(c4ccc(OC)c(Cl)n4)=O)C3C2)c(C)c1 CC(CC(=O)NC1(C2CCN(C(=O)CC(C)c3ccco3)C2)CC1)C(F)(F)F C(=O)(C(C(C)(C)C)OCc1ccccc1SC)N1CCC(N(CCC)CCC)C1 c1(NC(C(CNC(C2C(CCC)CCC2)=O)C)=O)cn(CC)nc1C#N C(=O)(CCCNC(C)=O)NCC1CC(C(C(=O)N(CC(COC)O)C)F)C1 C12CC3(CCCN(C3)C1=O)C2.C(=O)(C=CSc1nc[nH]n1)C(=O)CC1(CO)CC1 c1(C2C(C(=O)N(CCO)CCCCO)C2)ccccc1F.C(CO)OCC C1(O)(CC(=O)NC2CC(C(=O)NCC3C=CCOC3)C2)CCCCC1 c1(CNC(CC2(C)CN(C(C(C)Sc3ccccn3)=O)C2)=O)cc(O)ccc1Cl Cc1ccc(OCC(=O)NCC23CCC(C2)N(C(=O)CC2CCOC2)C3)cc1C C(=O)(C(CC(C)C)N(C(=O)C=Cc1nc(C)co1)CC)N1C(C)CCCC1 N1(C(CC(=O)N(C)C)=O)CCCC(CC(=O)NC2C(C)(C)C2(C)C)CC1 c1(C(=O)NCCOCCNC(C(C(C)C)n2cnnn2)=O)cnc2[nH]c(O)nc2c1 N1(C(COC)=O)CCC(C2(O)CCN(C(=O)CC3COC4(CCC4)CO3)C2)CC1 N1(C(C(C)SC)=O)CC2(C1)CN(C(c1ccn(C3CCC3)n1)=O)CCO2 C1(OCC)COCCC1NC1CCC(OC(=O)OC(C)(C)C)C1 C1(NC(=O)Cc2ccon2)CCN(C(=O)C=Cc2ccncc2)C12CCCC2 C(CC(C)(C)F)NC(CNCCC(C(CCC)=O)C1(C)CNC1=O)=O C1(NC(CC(=O)NCCC)=O)(CC)CCN(C(C2CCCSC2)=O)CC1 C1(CC(N2C(CN(C)C)COCC2)=O)CCCN(C(C2CCOC2C2CC2)=O)CC1 N1(C(CCCCC)=O)CCN(C(c2c(C)nsc2NC(C)C)=O)CC1CCC Cc1nn(C(C)C)c2sc(NC(=O)C3=CCCC3)cc12.c12nnc(o1)C2 c1(C(C)=O)ccc(C(=O)NC(C)CCCNC(C2(c3ccccc3)CCC2)=O)[nH]1 Cc1nsc2ncc(C(N3CC(NC(=O)CC(F)F)CCC3C)=O)cc12 C1(NC(CN(C2CCC2)C)=O)CCCN(C(c2cnn(CC3CC3)c2)=O)CC1 CCC(C(=O)N(C)CC1CC(F)CN1C(c1cc(C)on1)=O)C(C)(C)CC N1(C(COCCC=C)=O)CC2CC(C(N3CCCC(CC(C)C)C3)=O)(C2)C1 C(=O)(C(F)(F)CCn1cc(-c2ncoc2C)nn1)NC(C(=O)OC(C)C)C c1(C(=O)NC2(C)CN(C(c3c(CCC)nsc3N)=O)C2)ccc2scnc2c1 C(=O)(CCC(C)(C)C#N)NCc1c(C(N2CC(C)S(=O)CC2)=O)n[nH]c1 N1(C(c2c(C)onc2)=O)CC2(CCCC(CNC(C3CC(=O)NC3(C)C)=O)O2)C1 c1(C(C(=O)N(C)CC2CCN(c3nc(C(C)(C)C)ns3)C2)O)cccc(F)c1 C1(N(C)C)CN(C(=O)C(C2CC2)NC(=O)CN2C(=O)CNC2=O)CC1F C1(c2cn(CC)nc2)CN(C(c2nc(C3CC3)no2)C)CCO1 C(c1ccc([N+](=O)[O-])cc1)=CC(C1(F)C(C(=O)OC(C)C)C1)=O NS(=O)(=O)CCCC(=O)NC1COCC1NC(=O)CCOc1ccc(Cl)cc1 C1(C)(C(=O)NC(C)CCNC(=O)CC2CSC2)CCCCC1 c1(CNC(=O)NCC(C)(C)CCCO)cccc2ncccc12 c1(OC)ccc(C(=O)NCCC(O)CNC(c2nocc2Cl)=O)nn1 N1(C(C(CC)n2ccnc2)=O)CCN(C(C2CCC(=O)N2)=O)C(CCOC)C1 C#CCC(CC(F)F)C(=O)NCCN(C1CCCOC1)C(=O)COCCOCC N(C(=NCc1ncc(Br)s1)N1CCC(OC)C1)C(C=C)C Cc1csc2ncnc(N3CCC(O)CC3C(=O)Nc3ccccc3)c12 O=C1CCOC(COC(=O)CCc2ccc(C(F)(F)F)cc2)C1 c1(C(C(=O)NCC=C)N(C2CCCCC2)CCN(C)C)cccc(Cl)c1Br Cc1cccc(Cl)c1C(=O)NC1CN(C(C23CC(C)(CO2)C3)=O)CCC1C c1(C(=O)NCC2CN(C(C(CCOC)OC)=O)C(C)C2)nc(Cl)ccc1F c1(CNC(=O)Nc2nc(Cl)ccc2Cl)c(O)cc(O)cc1O CCCCC(C)(F)C(=O)N1CCC(CNC(=O)CC(COC)COC)C(O)C1 N1(C(CCCCCC)=O)CCC2(CC(CNC(=O)OC(C3(F)CCC3)=O)CO2)C1 c1(OC)ccc(F)c(C(N2CCC(C)(C(N3CCC(C(C)(C)O)CC3)=O)C2)=O)c1 c1(COC)cc(CC(N2CC(C(N3CC=C(C)C3)=O)(CO)C2)=O)on1 n1(CC(=O)NCCC2CCN(C(Cn3ncc(C)c3)=O)C2)nnc2c1CCCC2 c1(CCCC(=O)O)cnc(NC(=O)CNS(=O)(=O)c2cccs2)c(C=O)c1 CCCCCC(O)CC(=O)NC1CCCCC1CNC(=O)CCC(N)=O NC(=O)CCCCC(=O)N1CCCC(NC(C2CC(n3ccnn3)C2)=O)C1 C(=O)(C(CCC1CCC1)NC(=O)CCC=C(C)C)NCC(C)(C)SC N1(C(CN(C2CCC2)C)=O)CC2CC(NC(C3CNC(=O)N3)=O)CC(C2)C1 c1(CN(C(=O)C(C)CN(C(=O)CN2CC(C)(C)C2)C)CC)ccncc1 c1(CCC(=O)N(C)CC2(NC(C3CC(CC)OCC3)=O)CC2)cccc(F)c1Cl Cc1cnccc1C(C)C(=O)NCCCCNC(=O)C(C)c1ncco1 CCC1=C(C(=O)N2CC3(C2)CN(C(=O)COc2nc(C)ccc2Br)C3)CCCO1 c1(NC(C)C(=O)NC2(C(=O)NC3CCCC3C(N)=O)CCCC2)cc[nH]c(=N)n1 Cc1c(O)cccc1F.N1(C(C2(C)CCN(C(=O)CC3CC3)C2)=O)CCN(C=O)CC1 C1(CCNC(=O)CC=CCNC(c2ccn(C3CC3)n2)=O)CCCCCC1 N1(C(C2CN(C(C)=O)C2)=O)CCC2CCN(C(c3c[nH]cc3Br)=O)CC2C1 Cn1cc(C=CC(N2CCC(C)(CNC(c3cccc(C(N)=O)c3)=O)C2)=O)cn1 N1(C(c2c(C)c[nH]n2)=O)C2CCC1CC(NC(c1ccc(CN(C)C)cc1)=O)C2 c1(CC)nn(C)cc1C(=O)NCC(O)CNC(=O)COc1ccccc1O c1(NC(C(C)NCCN(CCCF)C)=O)cncc(Br)c1 c12nc(cc(O)n1)CN2.N1(C(C)=O)CCC(C)C(CNC(=O)C2=CCCCO2)C1 N1(C(CCOCCOC(C)(C)C)=O)CCC(C(=O)NC2(C#N)CC2)C1 C1(C(N2C(CN(C(=O)CC3(O)CCCOC3)C)CCCC2)=O)CN2CCN1CC2 c1(CCC(=O)NC2CC3CC2N(c2ccncn2)C3)ccc(F)c(F)c1 C=CCCCCCC(=O)NC(C)(C(=O)NCCc1ccn(C)n1)C1CCC1 c1(OC)ccc2ncccc2c1C(N1CCCC(CCNC(=O)CC(C)O)C1)=O C1(NC(C2C(C(C)NC(C=CC(C)C)=O)C2)=O)CCCC1C#N C1(NC(CNC(=O)OC)=O)CC(NC2CN(C(=O)CCn3ccnn3)C2)C1(C)C c1(C(N(C(CNC(CC2(OC)CCCC2)=O)C)C)=O)ccccc1CC#N c1(N(CC(C)NC(c2cnn(CC)c2C2CC2)=O)C)ccc([N+](=O)[O-])cn1 c1(C(=O)NCCOCCC(=O)NCCCN2CCOC2=O)conc1C1CC1 c1(CNC2C(C(N3CCS(=O)(=O)CC3)=O)CCC2)c(F)ccc([N+](=O)[O-])c1F c1(-c2cn(CCCC)nc2)ccc(C(=O)Nc2ccc(C3CC3)s2)c2[nH]ccc12 c1(OCC2CCC(NC(=O)C(F)C(F)(F)F)C2)cccc2ncccc12 c1(C(=O)NCC(CNC(C2N(C(C)=O)CCOC2)=O)C)c(C(C)C)nn(C)c1CC C(c1cnn(C)c1)=C(C(=O)NC1C(CNC(C(C)=C2CCC2)=O)C1)F C(=O)(C1=NN(C)C(=O)CC1)NC1C(C)CN(C(=O)Cn2nnc(=O)[nH]2)C1 c1(C(=O)NCC2(CNC(C3(C)CC3(F)F)=O)CCCC2)cc2cnccc2[nH]1 C1(C(=O)NC(C)C(F)(F)F)CC12CN(C(C1(C(F)(F)F)CCC1)=O)C2 C1(C(=O)NCC2(CNC(c3cn(CC)nc3)=O)CC2)CC1C1CCCC1 N1(C(CC(=O)OCC)=O)CCCC12CCN(C(=O)CSCc1cccnc1)C2 c1(C(=O)NCC2OCCN(C(CSCCN(C)C)=O)C2)ccc2nc(S)oc2c1 C1(CC)CC(C(=O)NCC(C)(C)NC(=O)Cc2c(C)noc2Cl)CCC1=O Cc1cnc(N2C(CC(CNC(=O)C(O)CC(C)(C)C)O)CC2)nc1S(C)(=O)=O C1(O)(CC(=O)NCC2(CCC)CC2)CN(C(=O)C=C2CCC2)C1 O=C(C1=C(Cl)CCC1)N1CCN(C(c2ccc(Cl)o2)=O)C(CC(F)(F)F)C1 C1(C(=O)NCCOCCCNC(C(CC)F)=O)OCC2CCCC12 c1(C(=O)NC2CC(NC(c3nc(C)oc3)=O)C23CCC3)cc(C#N)c(C)cn1 N1(C(C(C)S(C)(=O)=O)=O)CC=C(CC(=O)N(C2CCCN(C)C2)C)CC1 CC1(C)CN(C(=O)CC(O)C2CC2)C1C1CCN(C(C2CCS(=O)(=O)N2)=O)CC1 C1(CNC(C(C)=CC)=O)CCCN(C(=O)CCN(c2ccnc(Cl)n2)C)C1 C1(C(=O)NCC(C)N(C(C2CCC2)=O)CC)CCOC1 C1(C(=O)NCC(=O)NCCC(=O)NC2(C)CCSC2)Cc2nccn2C1 CC(C)(C)C(C)(C)C(=O)N1CCCCC1CNC(c1ccc(Cl)c(F)c1O)=O c12ccc(cc1Br)ONC2.c1(COC)ccc(CCCCC2CCCN2CC2CC2)o1 C1(CCOC)(N(CC(=O)NCC(=O)NCC2(N(C(=O)OC)C)CC2)C)CCC1 C1(CN(CC(C)C)C)CC2COCC(C1)C2(F)F.C12CC1C2.C(C)(C)(C)OC=O N1(C2CC3(CN(S(C(CCC)C)(=O)=O)C3)C2)CCC(F)(F)C(C#N)C1 Cc1c(C(N2CC(F)(CNC(C3CCOC3)=O)C2)=O)sc2cc(F)ccc12 C1(NC(C(C(C)C)NC(=O)C2CC2)=O)CCC2(CC1)N=N2 C1(C(=O)NCC2C(NC(c3ccc(C)cc3O)=O)C2)CC(C)(C)OC(C)(C)C1 C1(NC(CC(=O)NC)=O)Cc2ccccc2N(C(=O)COc2cc(F)cc(F)c2)C1 CC(C)(C(=O)NCC(O)CNC(C1CCCN(S(=O)(=O)C(F)(F)F)C1)=O)C(N)=O N12CCc3ccc(cc3C1)Cn1c2nnc1-c1nccs1.N1(CC)CCOCC1 C(=O)(C1=CCC2CCC1N2C(=O)C(C)CC(C)C(C)=O)N(C)Cc1c(CC)noc1 C1(CC(N2CCN(CC(C)(C)NC(=O)CO)CC2)=O)NC(=O)CN(C)C1=O Cn1ccc2ccnc(C(=O)NC3(C)CC(NC(c4cnc[nH]4)=O)C3)c12 c1(OC)ccc(C)cc1CC(=O)NC1CC(O)CN(C(c2csc(C)c2)=O)C1 C(=O)(C(CCCCOC)NC)NC(CCC(OC)OC)C(C)C C1(C(=O)NC)CN(c2nnnn2C(=O)NCCn2nc(C(F)(F)F)cc2C)CCO1 c1(C(C(=O)OC)NC(CCC(C)OC)=O)cc(C)c(C)nn1 N(C1CCc2cccnc21)C(C12N(C(CC(C=C)(C)C)=O)CCC1C2)=O Cc1cccc(F)c1C(N1CCC(NC(C2CCC2(F)F)=O)CC1)=O C12C=CCCN1C2=O.C(c1ccccc1)=CC(N1C(C2CCCC2)CCC1)=O c1(C(=O)NC(CNC(c2scc(C)c2Cl)=O)CO)c([N+](=O)[O-])cnn1CC(F)F c1(C(=O)NCCOC2CCN(C(C3(O)CC(CF)C3)=O)C2)cc(F)cc(Cl)c1 N1(c2nc(SC)nc(C)c2)CC(C2CCCN(C(c3ncccc3C)=O)C2)C1 Cn1nc(Br)nc1C(=O)NCc1cn(CC2(F)CCOC2)nn1 C(=O)(CC(C)F)NCCN(C1CC1(C)C)CC N1CC(N(c2nccc(SC)n2)C)C(C)(C)C1.C1(C=O)CC(C(C)C)=NO1 C1(C2CCC2)(C(N(C)CC2CCN(C(c3cncs3)=O)C2)=O)CC1(F)F C1(=O)C(CC)CCNCC(CSCC)N1.C=CCCC1(CN)CC1 c1(C(=O)Nc2ccccc2CCO)cc(C(N2CCCC2)=O)cnc1C(F)(F)F c1(CC(=O)NC(C(C)(C)C)CNC(c2cc(C3CC3)no2)=O)cc(O)nnc1O N1(C(C(C)OCC)=O)CCC2(CCN(C(c3cnns3)=O)C2)C1 CCC(CC)CCCC(=O)NC(C)(C)COCCNC(C1(CSC)CCCO1)=O c1(C(=O)NCC(C(C)C)NC(C2(C)CCCS2)=O)cnc2[nH]cnc2c1 C1(NC(CS(CCC)(=O)=O)=O)CC2(CCCCN2C(C2CSC(C)=N2)=O)C1 C1(NC(C(C)C)=O)CCN(CCNC(c2ccnn2C(C)(C)C)=O)CC1 C1(NC(=O)C2=COCCC2)CC2CCC(C1)N2C(C12COCC(C1)OC2)=O C1(CNC(C(C)OCC=C)=O)CC2CCC1N2C(C1(O)CN2CCC1CC2)=O c1(NC2C(NC(c3onc(C)c3[N+](=O)[O-])=O)CCCC2)ncccc1S(C)(=O)=O N1(C(COCCOCCOC)=O)CCCC(O)(CN(C(=O)C2=CCCS2)C)C1 N#Cc1ccc2cc(C(N3CCN(C(c4csnn4)=O)C4CCC34)=O)ccc2c1 C1(NC(C(=O)NCCCc2ccc(C#N)cc2)=O)Cc2cccnc2C1 c1(C(N2C(C(N3CCCCC3)=O)CC(O)C2)=O)ccc([N+](=O)[O-])cc1Cl N1(C(C(COC)(C)C)=O)CC2(CCCN(C(=O)CS(=O)(=O)CC(=O)OC)C2)C1 Cc1cccnc1C=CC(N1CCCC(N(C(=O)C2=CCCCC2)C)CC1)=O Cc1ccc(CN(C(=O)C(CCN(C)C)NC(C2CC(O)C2)=O)C)nc1 N1(C(C(C)NC(COC)=O)=O)CC(NC(C2C(C)C2(F)F)=O)C(COC)C1 C12(CNC(c3scc(C)c3C)=O)CCC(C1)N(C(=O)C(C1CCC1)C1CCC1)C2 C=CC1(C(=O)NC2CCN(C(=O)C(=O)CCc3ccccc3)C(C)C2)CCOCC1 C1(C(N2CCN(C(c3cnn(C)n3)=O)C(CO)C2)=O)CCCCCC1(F)F C1(C)(NC(c2nc(C(C)C)sc2)=O)CCN(CCO)CC1 Cc1cc(C)c(C(=O)NCC2(C)CCN(C(c3ccco3)=O)C2)s1 c1(CC(=O)NC2CN(C(=O)C=Cc3cccnc3)C2)ccc2c(c1)CCO2 C1(CCNC(CCC=C(C)C)=O)CN(C(=O)C(F)C(C)(F)F)CC(C)O1 C1(SCCC(=O)NC2C(NC(c3c(CC)c[nH]n3)=O)CCC2)CCS(=O)(=O)C1 N1(CC(=O)N(CCC(=O)NCc2ccc[nH]2)CCC)CCCNC1=O CCCC(CNC)C(=O)NCC(C)C(=O)OC.C(c1cc[nH]n1)=C c1(NCc2sc(Br)nc2Br)c(Cl)cc(C#N)cc1Cl.Cn1cc2cc1C(=O)N2 C=CC1(C(N2CCC(C(O)CNC(C3(C)CCCC3O)=O)CC2)=O)CCOCC1 CCCCC(CC)CC(=O)NCc1ccc(C(C)NC(c2ccncn2)=O)cc1 c1(OC)ccc2c(c1)n(C)c(=O)n2C.C12CCN(C1)C(=O)N2C C1(NC(C(CC)Oc2ccccc2)=O)CC=C(C(=O)N2CCC(OC)C2)C1 N1(C(C(CCC)O)=O)CC(C2CC2)(C(N2CC(NC(C)=O)C2)=O)C1 c1(C(N2CC(N(C(C3CCC(OC)C3)=O)C)C2)=O)nc(C)c(C)[nH]c1=O CCN=C(NCCS(=O)(=O)NC1CC1)NCc1ccc(-c2ccccc2F)o1 c1(C(=O)NC2C(CNC(CCc3ccc(C)cc3)=O)C2)nnc(O)nc1O C1(C)(C(=O)NCC2C(OC)CN(C(c3c(COC)ncs3)=O)C2)CC2(CCC2)C1 Cc1ccc(O)c(CNC(=O)C(CO)NC(c2ccc(CO)s2)=O)n1 n1(CC(=O)NC(C)CC(C)NC(c2cc(C(N)=O)co2)=O)ccc(=O)n(C)c1=O C1(OC)CN(C(C2CC2C2(C)COC2)=O)CCC1NC(c1cc(C)cc(C)c1)=O c1(C(=O)NCC2(O)CN(C(c3cc(COC)no3)=O)C2)cncc2c1CCCC2 C(CN=c1[nH]nc(C(C)(C)C)s1)C1N(C(CCC(=C)Cl)=O)CCCC1C CC(C)C1=NOC(C(N2CCC(CF)(NC(=O)CCCc3cccnc3)C2)=O)C1 C(=O)(C#CC1CCCOC1)NCC1N(C(c2cccc(CC)c2F)=O)C2C(C1)C2 N#Cc1ncc(CC2CC2)nc1N1CCC(C(N)=O)CC1 C1(NC(c2nc(C)oc2)=O)CN(C(c2cn(CC(F)F)nc2C)=O)CCC1C C1(NC(c2c(C)[nH]c(C(C)(C)C)c2)=O)CC12CCN(C(=O)CO)CC2 Cc1[nH]nc(C(N2CC(NC(c3cc(Cl)c[nH]3)=O)CC2C)=O)c1O c1(CC)ccc(C(C)=CC(N2CCCC(NC(C3CCN3C(C)=O)=O)CC2)=O)cc1 CCCCC(CCC)NC(=O)CCN(C(=O)C(F)CC1CCOC1)CC N1(C(CC(=C)C)=O)CC(NC(C2CCC(=O)N(CCC)C2)=O)C(C)(C)C1 c1(C(=O)NCCCC(C)NC(=O)Cc2cc[nH]c2)cc(OC(F)F)ccn1 C1(CNC(=O)Cc2cc[nH]c2)COCCN1C(=O)CC1CC=CC1 Cc1cc(CO)oc1C(=O)NCCCCNC(=O)C(O)CCc1ccccc1 C=CCC(C(=O)N(C)CC1(C#N)CCC1)NC(=O)C(N1CCOCC1)C CC1(C)C=NN1C(=O)C(CN=[N+]=[N-])NCc1ncccc1OC(F)F c1(OCCCC)ccc2cc1-2.N12CC3CC(C1C3)NC2=O.O(C)CC C1(C(N2CCN(C(c3c(CC#N)cccn3)=O)CC2)=O)CC2CCC(C1)C2O C#Cc1ccc(C(C)(C)NC(=O)C(N)CNC(C(C)(C)C)=O)cc1 C(CC(C(C)(C)C)NC(c1cnc(Br)s1)=O)N(C(=O)C1=CC(C)(C)C1)C c1(CC)ncc(Cl)c(C(N2CC(CCO)(NC(C3CNC(=O)CC3C)=O)C2)=O)n1 Cc1cn2nc(N3CCN(C(c4ccnn4C)=O)CCC3C)sc2n1 N1(C(c2cc(C)oc2)=O)C2CCCC1CC(NC(=O)Cc1c[nH]c(=N)nc1O)C2 C1(NC(c2ncn(CNC(C(N3CCOC3=O)C)=O)c2)=O)CC2CCC(C1)N2C C(=O)(C(C)CCCc1ccccc1)NCC(C)NC(c1cc(Cl)c(Cl)s1)=O N1(C(CCSCC(C)C)=O)CCCC(C2CC2NC(c2csnn2)=O)C1 C(=O)(C(=O)C(C)(C)C)NC(C)CCCCNC(c1cccc(C2(O)COC2)c1)=O CC1(C)C(CO)CCN1C(c1ccnc(CNC(c2cc(O)cc(=O)o2)=O)c1)=O n1(CC(=O)NC2C(CNC(c3c(CCC)n[nH]c3)=O)C2)nc(C)n(C)c1=O N1(C(CC(c2ccccc2Cl)NC(CC(CC)OC)=O)=O)CCC(C)(F)CC1 c1(C(C)=O)ccccc1C(=O)NCCCCCNC(=O)Cc1ccccc1 CN1CC(C)(C(=O)N(C)CCOCCCNC(C23CCCC2C3)=O)CCC1=O C1(C(=O)NC(C2CSC2)C)CCOCCN1C(=O)Cc1nc(=N)[nH][nH]1 Nc1c(C(N2CCC=C(CNC(=O)CC3CCCC3)C2)=O)cnc2ccnn12 c1(C(=O)OCC(CCNC(=O)OC(C)(C)C)O)cc2c(nc1N)CCCC2 Cc1cccc2nc(N(C3CN4CCCC4C3)Cc3ccc4c(c3)CCOC4)sc12 C(=O)(C(F)(CNC(c1cc(C)c(C)s1)=O)C(C)C)C(C(CC)CNC)=O c1(C(=O)NC(CNC(CC(C=C)C)=O)C2CCC2)ccc(C(F)(F)F)c(O)c1 C1(CCCC)CN(C(=O)C(C2CCC2)OC)CCN1C(C1CC1C(C)C)=O c1(N(c2cccc(OCC)c2)Cc2ccccc2)c(OC(C)=O)cncc1Br C1(C(=O)NCC2C(C)CCCN2C(c2cnc(Cl)cn2)=O)CCc2nncn2C1 N1(C(c2cc(F)ccc2F)C(=O)NCCCSCC)CCC2(CC1)CNC(=O)C2 N1(C(c2nccc(C)n2)=O)CCCC(O)(CCNC(=O)CCC(C)(F)F)C1 c1(C(=O)NCC(C)N(C(CC2CCC(C)O2)=O)C)cc2c(=O)[nH]ccn2n1 c1(OC(C)C)ccc(=NC(=O)CCCc2ccc(Br)cc2)[nH]n1 c1(C(=O)NCC2C(C)CN(C(C3CC4(C3)CC(O)C4)=O)C2)c(F)ccc(O)c1F c1(C(=O)NCC(C)N(C(CC(CC)O)=O)C)c(N)cccc1[N+](=O)[O-] c12[nH]ccc1CNC2=O.c1(C2(CC(=O)NCC3C=CCC3)CC2)ccon1 C#CCCCCC(=O)NC(C1CCCCC1)C(=O)NCC1CC(C)=NO1 c1(C(C(=O)N(CCC(C)NC(c2cc(C(F)F)n(C)n2)=O)C)C)cncc(F)c1 c1(OCCC(=O)NC2C(C)(C)C(=O)C2)ccc(F)c(F)c1F C#CC1CN(C(C2CC(O)C(F)C2)=O)CCN1C(=O)CCCSC(C)(C)C c1(OC)ccc(F)c(NC(C2CC2C2CN(C(C3CC4CCC4C3)=O)C2)=O)c1 N1(C(c2c(C(=O)OC)con2)=O)CC(NC(C2CCN2S(C)(=O)=O)=O)C(C)(C)C1 N(C1CC2(CCCC2)c2ccccc21)N1C2(C(=O)NCC2)CCC1 N1(C(C(C)(CC2CCC2)OC)=O)CC2CC(NC(=O)CC3C(C)(C)C3(C)C)C(C2)C1 Cc1cc(Cl)cnc1C(=O)N(c1nccc(C(F)(F)F)n1)CC1CCCNC1 c1(N(C(CN(C(C2(SCC)CC2)=O)C)C)C)nc(C#N)ncc1Cl CCC(C(=O)N1CCCC1CC(=O)NCc1ocnc1C1CC1)C(F)(F)F C(=O)(CC1C(=O)Nc2cc(OC)ccc21)NCC1C(NC(COCC)=O)CC1 N1(C(CCC(C)SC)=O)CC(NC(c2cn(C)c(O)n2)=O)CC12CCCC2 CCCCC(C(=O)NC(CC)C(C)(C)CC)NC(=O)C(C(=O)NC)N(C)C C1(NC(C(C)(C)NC(=O)NCC)=O)CCCC(CNC(=O)C(C)=C2CCC2)C1 N1(C(c2coc(C(F)F)c2)=O)CC(O)CC1C(=O)NC1CCN(CC2CC2)C1 c1(C(N(CCN(C(=O)CCN2CCCCC2=O)CC)CC)=O)nn(C)c(N)c1C C(=O)(C1=CCCOCC1)N1CC=CC(NCc2nc(CC)sc2)C1 c1(C(C(C)C)NCC(C)NC(C(=O)NC)=O)ccc(Br)c(F)c1 CCC(CN1CCC(Cc2cnn(C)c2)C1)(CC)OC C1(NC(c2onc(COC)n2)=O)CCN(C(=O)C=Cc2ccco2)CCC1CO c1(C(N2CCC(NC(C3CC3c3ccccn3)=O)CC2)=O)cc(Cl)nc(Cl)c1 C1(NC(C(CC)N(C)C)=O)CC2C(NC(C3(c4cnc(C)s4)CC3)=O)C2C1 C1(NC(C(CC)SC)=O)CCCCN(C(=O)C(c2ccc(F)cc2C)(F)F)C1 C1(C(N2CC(N(CC=C)C)C2)=O)(CC)CCCN(C(=O)CCCCSC)C1 c1(C(=O)NC23CC(CNC(=O)CSc4cccnc4)(C2)C3)onc2ccccc12 c1(C(c2ccccc2)C)cnc(NC(C2CCC(C(C)(C)C)CC2)=O)nc1 N1(CC(=O)NCCC(C)CNC(c2ccnnc2)=O)CCCCC1C N1(CCC(=O)NC2C=CCN(C(C(CC)OC3CCC3)=O)C2)CCSC(C)(C)C1 c1(C(=O)NC2(C)CN(C(C(COCC)N=[N+]=[N-])=O)C2)cnc2[nH]nnc2c1 c1(C(=O)NCCC(C)N(C(c2ccn(CC(C)C)n2)=O)C)ccccc1S(C)=O C1(=CC(=O)NCC2CCC(NC(=O)C(F)(F)C3CCCC3)C2)CN2CCC1CC2 Cc1ccc(C(CN(C(=O)CC2CCCC(O)C2)C2CC2)NC(=O)C(C)(C)O)cc1 C(=O)(C(F)C(C)(F)F)NC1C(C(=O)NC(CSC)C)COC1 N1(C(C2(CC=C)CCC2)=O)CC2CCC2(CNC(=O)CN2CC(C)(C)C2)C1 N1(C(C=CC=CC)=O)CCN(C(C2CCN(c3ncccn3)C2)=O)CC(C)(F)C1 C1(C(NOCC=C(C)C)=O)C(CO)CCN1C(=O)C(C)n1ccnc1 CC1CCN(C(c2c[nH]c(C(=O)NC)c2)=O)CCN1C(c1cccc(F)c1Cl)=O C(=O)(C1=CS(=O)(=O)CCC1)NC(CC(C)NC(=O)C(C)(C)CCC#N)C CC1(CNC(C23CCC(CC2)CC3)=O)CCCN(C(C2CCCN2C2CC2)=O)C1 c1(C(N2C(C(C)NC(c3csc(C4CC4)n3)=O)CCC2)=O)ccsc1S(N)(=O)=O O=C(CC(C(F)(F)F)NC(C1CCC2(CCC2)C1)=O)NC1CC(O)C1O c1(-c2nc(-c3ccc(C)o3)nn2C(C)C2CC2)cc(C)c(OC(F)F)c(C)c1 C1(C(N2C(CC(=O)N(C3CC4CC4C3)C)CC2)=O)CC=CCN1C C(=O)(CCCC(C)(C)CC)NCC1CCC(C(=O)NC2C(OCC)C2C)C1 C(=O)(C(C)(CNC(=O)CC1(C)CCOC1)CC)NC(CSC)C c1(C(=O)NC(CCOC)CNC(=O)COc2cnc(Cl)cn2)ccnc(Cl)c1O C1(CC(=O)NCC2(C)CCN(C(c3ncc(Cl)cc3F)=O)C2)CN2CCN1CC2 C(=O)(C(F)(F)C(O)C1CC1)Nc1cccc(CNC(C=Cc2n(C)cnn2)=O)c1 c1(CC(=O)NCC(=O)NCC2CC(NC(CCCC#C)=O)C2)cc(O)ccc1C N1(C(c2snc(C)c2N)=O)CCn2ncc(CNC(C3C=CC=CC=C3)=O)c2C1 c1(C(=O)NC2CC(O)CN(C(=O)Cc3csnn3)C2)ccc2ccccc2c1 C12(NC(CSCCC)=O)CCCN(C(=O)CSc3ccc(OC)cc3)CC1C2 C(=O)(C(C)CN1CCOCC1)NCCN(C(=O)CC1(CC(=O)OC)CC1)CC C1(NC(C=Cc2cc(OC)ns2)=O)CN(C(=O)C=C2CCOCC2)CC1N=[N+]=[N-] c1(C(N2CCC(NC(c3cccc(C)n3)=O)C(F)C2)=O)sccc1S(C)(=O)=O C1(O)(C(=O)NCCn2cccc2)CCN(Cc2cccc(F)c2)CC1 CC1=C(C(=O)NC2CCN(C(c3csc(-c4cnn(C)c4)n3)=O)C2)CCCC1 C1(NC(c2c(CCC)nco2)=O)(CNC(=O)C(C#N)CC)CCC(F)(F)CC1 N1(C(C2CCCN(Cc3cc(C)c(F)cc3)CC2)=O)Cc2nn(C)c(N)c2C1 C1(CCC)(NC(=O)C(C(=O)OCC)OC)CCN(C(=O)C(O)CC2(O)CCC2)CC1 CC1CC(C(=O)NC2C3CCN(C(=O)Cc4ccnn4C)C23)=NO1 c1(C(N2CC(CCNC(C(C)(C)OC)=O)C(C)C2)=O)ccc(C)n(C)c1=O C(CCC(C)CC(=O)NCC1(F)CCN(C(=O)Cn2ncn(C)c2=O)C1)=C(C)C C(=O)(N1OC2CC1C(O)C2O)C1(C)N(C(Cc2n(C)cnc2)=O)CC(O)C1 c1(C(=O)NCC(C(C)C)NC(c2scc(C)c2Cl)=O)cc2cnccc2[nH]1 N1(C(CNC(N)=O)=O)C2CCC1CN(C(=O)CN1CCCCC(O)C1=O)CC2 c1(CN2C(C(=O)Nc3cc(C)no3)CC(F)C2)ccc(I)c(F)c1F Cc1nccc(C(=O)NC(C(=O)NCCc2c[nH]nc2C)C2CCOC2)n1 Cc1nc2sccn2c1C(N1CC2CCC1C2NC(C1CC2(CCOC2)C1)=O)=O Cn1cc(NC(=O)CC2CCN(C(N)=O)C2)nc1C(=O)Nc1cc(C(F)F)no1 C1(C(N2CCC(N(C(=O)Cc3cn(C)nc3C)CC)C2)=O)CC(C)CC(C)(C)C1 C(=O)(N=c1nc(O)[nH]c(O)n1)c1ncc(-c2c(OC)ncc(C#N)c2)nc1 c1(C(=O)NCC2(C)N(C(c3cn(CC)nc3)=O)CCC2)cc(F)ccc1Br CCC(CC)(C(C)C)NC(c1ccc(CNC(=O)C(=O)C(C)(C)C)s1)=O c1(C(N2CCC(O)(CNC(C(C)C3CCC3)=O)C2)=O)cnc(O)c(Br)c1 N1(C(Cc2c(C)ccs2)=O)CC2CCC2(CCNC(C2CCS2(=O)=O)=O)C1 C(=O)(CC(=O)N(C)C)NCCCN(C(=O)CCNc1nccs1)CCOC N1(C(C(CN(C)C)(F)F)=O)C2CCC1CC(NC(=O)CCCc1ccsc1)C2 C1(NC(c2[nH]c(=N)sc2)=O)CCN(C(=O)CC2CCCCC2)CC1C(N)=O N1(C(C(C(C)C)NC(C(N2CC(C)C2)C)=O)=O)CCCC(F)(C(N)=O)C1 N1(C(CCC=C)=O)CC(NCc2cnc(C)cn2)C(C#N)C1 Cc1cc(-c2nc(CNC(C)Cc3cc(Cl)ccn3)co2)c(C)o1 Cc1ccc(OCC(=O)NCC2CC(C)N(C(=O)CC34CCC(C3)C4)C2)cc1C N1(C(C(C)O)=O)CCC(C(=O)NCCCCC(C)(C)C)C12CCC2 c1(C(N2CCOCC2NC(=O)NC)C(=O)NCC=C)cc(Cl)c(F)c(Cl)c1 C1(C2(O)CCN(C)CC2)(C(N2C3(CNC(C(CC)(C)CC)=O)CC(C2)C3)=O)CC1 CCC(C(=O)N1CC(C2CCCN2C(=O)CCC2CCC(=O)C2)C1)NC(N)=O N1(C(C=C(CCC)C)=O)CCN(C(=O)CC2(OCC)CCCC2)C(CC(F)F)C1 S(=O)(=O)(c1ccc(N2CCCC3(CCCO3)CC2)c(Br)c1)NCC=C CCCC(C)(O)C(=O)NC(Cc1ccco1)C(N1CC2CCC(C2)C1)=O CCC(CC)C(C)C(=O)NC1CCOC1C(=O)NC1COCCN(C)C1 C1(N(C(C=CC=CC)=O)C)CCN(C(=O)CCC2CCC(O)CC2)CC1 C1(C(=O)NC(c2cccc(Br)c2)CC)CC(F)(F)CN1C(c1sccc1C)=O c1(OC)ccc(NC(C2CCCN(C(C(C)CC3C=CCC3)=O)C2)=O)cc1 O=C(C1=CCC2CCC1N2C(=O)CCCC1CC1)N(CCCO)C1CC1 c1(OC)ncc(NC(=O)C(=O)NOCc2ccccc2F)cn1 C1(C(N2CCC(NC(C3CN(CCOC)C(=O)C3)=O)C2)=O)CC12CCOCC2 N1(Cc2ccc(C)c(C)c2)Cc2ccccc2C1C(=O)NC(c1ccccc1)C N1(CC2C(OC)COC2)CCC(=O)N(c2n[nH]c(C(C)C)n2)C1=O C=CC(N)C(=O)N1CCC(NC(C2CCOC2)=O)C1 c1(NC)cccc(C(=O)NCC(C)(C)CC2CN(C(=O)C=C(C)Cl)C2)n1 CC1CCC=C1C(=O)N1CCC(O)(CNC(=O)COc2ccccc2Cl)C1 c1(C(N2CCC(C(C)NC(c3cn4c(n3)SCC4)=O)C2)=O)ccc2nccn2c1 C1(NC(C=C(C)C)=O)CCCOC12CCN(C(C1CC(C)(F)C1)=O)CC2 C(CN=c1ccc(C)c[nH]1)NC(=O)NC(CCOC)CO N1(C(C(C)N(C(c2c(OC)cncn2)=O)C2CC2)=O)CCC(CO)C12CC2 c1(SC)cc(Cl)c(N)c([N+](=O)[O-])c1.c1(OC)ccc2c(c1)NC(=O)CCC2=O c1(C(=O)NC(C2CCCNC2)C)cc(=O)n2nccc2[nH]1 c1(CC(CCC)NC(C2(C)CC(=C)C2)=O)c[nH]c2ccccc12 c1(C(=O)NC2C3OCC(NC(c4c(CC)ncs4)=O)(C3)C2)cc2c(s1)CCCCC2 Cc1ccc(C(=O)NCC2CCC(NC(=O)CCOC3CCCC3)C2)c(O)c1C CC1CN(C(=O)COc2cc(O)nc(O)n2)CCC1C(=O)NC1CCN(C)CC1 N1(C(CC)=O)CC(NC(=O)C(N2CCC(c3cccc(C)c3)C2)=O)C(C)C1 c1(Cc2cn(CC(CCNC(C3(C)CCCCO3)=O)F)nn2)cc(F)cnc1Br c1(OC)ccc(NC(=O)C(c2c(C)cnn2C)N(C2CSC2)C)cc1 CN1CCN(C(C2CC(Cl)(Cl)C2)=O)C(CNC(=O)CCC2OCCO2)C1 c1(CC)cc(C(=O)NCCNC(c2noc(C)c2I)=O)c(C)o1 C(=O)(C(F)(F)c1nccs1)NCC1CC(NC(CCSCC=CC)=O)C1 c1(SCC(=O)NC(C(C)NC(C2(C3CCCO3)CC2)=O)(C)C)cc(F)ccc1Cl C1(C(=O)NC(C(=O)N(C)Cc2ccco2)(C)C2CCC2)CCCCN1C C(CC(Cc1ccccc1)NC(C1CCOC1)=O)NC(CC#C)=O c1(CC)nc(C(=O)NC2(C(=O)NC(C)Cn3cncn3)CCSC2)co1 c1(C(N2C(C(=O)NCCC(=O)OC(C)(C)C)C(C)C2)=O)ccc2cccnc2c1 CC(CC(=O)N1CC(NC(C2(C#N)CC3CCC2CC3)=O)C(C)C1)CC(C)(C)C C(C)(C)(CCC(=O)NCCCOCCC(=O)N(C1CCCC2CC12)C)NC CN=c1cc(NC(C)C(=O)Nc2ccccc2N2C(=O)CCC2=O)cc[nH]1 c1(C(=O)NC2CC(CNC(=O)Cc3ccsn3)C2)cnn2c1OCC(F)C2 c1(C(N2C3CC(NC(CN(C)CCO)=O)C2CC3)=O)ccnc2[nH]cnc12 C1(N(CC#C)C(N2CCC(CC(C)(C)C)C2)=O)CCN(C(C)=O)CC1 c1(C(=O)NCC(CCOC)NC(C(C)OCCOC)=O)cnc2[nH]ncc2c1 C(=O)(CCCCCCCBr)N1C(C(=O)Nc2nc(C)c(Br)s2)CC(C)C1 CC1(C(=O)NCC(C2CCCC2)NC(=O)CCc2csc(=N)[nH]2)COCCO1 C=CC(C)(CCOC)C(=O)NCC1CC(O)CN1C(c1ccc(C)c(C)c1)=O N1(C(C2C(C(C)C)OCC2)=O)CCC(OCCN(C(c2nc(Cl)cs2)=O)C2CC2)CC1 c1(C(C)C)cc(C(=O)O)n(C(C)CCCN2CC(C(=O)OC(C)(C)C)C2=O)n1 c1(C(NC2CC2)=O)ccccc1OC.C(=O)(CC=O)OC.C1CC(=O)N(C)CCN1 C12(C(=O)NC3CCC(NC(CC(C)C)=O)CC3)CCC(C1)C(=O)NC2 CC(C)CC(C(=O)NC1(CNC(=O)CN2CCCCCC2=O)CCCC1)C(N)=O C1(NC(C2C(CC)C2)=O)CN(C(=O)Cn2c(C)n[nH]c2=N)CCC1C N1(C(CCSC)=O)CCN(C(c2ccnc(OC3CC3)c2)=O)CC1CO Cc1ccnnc1C(=O)NC(C)CCCCNC(=O)C(C1CC(F)(F)C1)O N1(C(C(C)C(F)F)=O)CC2CCN(C(=O)CCc3ccc(F)c(F)c3)C2C1 CC(CC(F)F)C(=O)N1CC(C(C(=O)NCC(c2ncc[nH]2)C)N(C)C)C1 C(=O)(CC(C(C)OC)NC(=O)CCC(N)=O)NCCC(=O)NCC c1(CC)cc(F)c(NC(c2ccc(CN)cc2C)=O)c(F)c1 CC(C)CC(C)CC(=O)N1CCOCCC1C(=O)N(C)Cc1cn(C)nn1 N1(C(C(OCC)OC)=O)CCC2CN(C(c3ccnc4c3CCO4)=O)CC12 C(=O)(C(CC(F)F)NC(=O)C=C1CCC1)NC(CC=C)CNC(C)=O c1(N2CC(C)C(NC(c3cc(Cl)nc(Cl)c3)=O)C2)ncnc2c1CCCC2 C=CCC(C)C(=O)NCCCCNC(c1sccc1Cn1cnnn1)=O N1(C(CC(CC)O)=O)CCN(C(=O)Cc2cc(Br)ccc2Cl)CC1CO CC1CC2(CC(C(N3CCN(C(=O)CCCC4OCCO4)C(C4CC4)C3)=O)C2)C1 c1(C(=O)OCc2cccc(-c3c(C)cc(C(N)=O)s3)c2)c[nH]cc(Br)c1=O c1(C(CC)CC)cc(C(=O)N(C(C)CCNC(c2sccc2COC)=O)C)on1 c1(OC)csc(C(=O)N(CCCCNC(=O)CC2CC(O)C23CC3)C)c1OC C(C(C)(O)C(=O)NCC1(CNC(C2CCN(CC(C)C)C2)=O)CC1(F)F)OC c1(N2CCC(N(C(CC3C(C)=NNC3=O)=O)C(C)C)C2)cccc(F)c1[N+](=O)[O-] N1(C(c2n(C)nnc2)=O)CCN(C(=O)C2=COCCO2)CC1CO N1(C(c2c(CC)c[nH]n2)=O)CCCN(C(C2CCC3CC3CC2)=O)CCC1 C1(NC(=O)C=CCF)CN(C(c2ccc3n[nH]cc3c2Cl)=O)Cc2nccn2C1 CCC(F)(F)C(=O)NCCC(C)NC(=O)CN1CCCC(N(C)C)C1 c1(C(N(CC(=O)N(CC(F)F)C)C(C2C(=C)C2C(=O)OC)=O)C)ccncc1 C1(CNC(c2cc(CC)on2)=O)CC(C)N(C(=O)C(C)=C2CCC2)C1 N1(C(CS(CC)(=O)=O)=O)CC2CCC1CC2NC(c1ccc(C)o1)=O C(=O)(C1CCCc2nn[nH]c21)N1CC(C)(C)C(NC(c2ccc(C(N)=O)o2)=O)C1 C(C(CC1CC1)C(=O)NC1CCCC1)N(CC(=O)NC(C)Cc1cnc[nH]1)C C1(CNC(C(CNC(CSCCCC)=O)O)=O)CNC(=O)CO1 C=CC(C)CC(=O)NC1CCCN(C(=O)CCc2ccc(CO)cc2)C1 C1(NC(C(C)(C)NC(C=COC)=O)=O)CC2CC(NC(=O)CCC3CCC3)C1C2 c1(C(=O)NCC(CNC(C(c2cccc(OC)c2)O)=O)O)ccc2c(c1)CCN2 N12CC(CC(F)(F)C1)C2=O.c1(CC(OCC)OC)ncc(F)c(OC)n1 C(=O)(C1=CCc2ccccc21)NCC1CCCC(NC(C(C(C)(F)F)(C)C)=O)C1 Cc1ncc(Br)c(C(=O)N(C(C)CCNC(=O)COCC2CCC2)C)n1 N1(C(C)=O)CCCCC1C(=O)NC(c1ccc(CN(C)C)cc1)C C1(C(N(CCCCN(C(C(C=C)C)=O)C)C)=O)C2CCC(=O)C12 CC1(C)CCCN(C(=O)COC2CC2)C1C(=O)NCC1CCCCCC1O c1(CC(=O)NC(C)(C)CNC(C2CCCN2C)=O)ccnnc1O CCCCCC(O)CC(=O)NN1CCCC1C(=O)N(CCCC)C(C)C N1(C(CCc2ccc(C)s2)=O)CC(NC(c2cc(O)nc(Cl)c2)=O)CC(C)(C)C1 C=CCN=c1[nH]cc(C(=O)N(C(C)CN(C)C(C2CN(C)C2)=O)C)s1 C1(CNC(CC=C)=O)CN(C(=O)Cn2ccnn2)CCC1C(F)(F)F C1(CC(=O)NCC2N(c3ncn(C)c(=O)c3)CCC2(C)C)CC2(CCCC2)CO1 CC(CNC(c1cocn1)=O)C(F)C(=O)NC1CCC1 C(=O)(C(C(CC)CC)OC)N1CCCC(CC)(NC(=O)CCCc2cc[nH]n2)C1 C=CC(CC)CC(=O)N1CCC(C(N2CCC3C(C(N)=O)C3C2)=O)C1CC c1(CNC2(c3nnnn3C3(C)CC3)C(CC=C)CCC2)cc(C)ccc1OCC c1(C(=O)NCCn2cc(C(=O)OC)nc2)cnc2sc(C)cn2c1=O N1(C(CC(=O)OCC)=O)CCCC(NC(=O)C(COC2CC2)N(C)C)C1C c1(C(=O)NCC(C2CC2)NC(Cn2cc(C(C)=O)nn2)=O)c(C)nsc1C C(=O)(CCCC(N)=O)N1CC(NC(c2ccc(OCC)cc2)=O)C(C)C1 C(=O)(C(C)(O)C(C)C)NCC(c1ccccc1C(C)C)NC(c1cc(C)ns1)=O CCC(CC(=O)NC1COCCC1NC(C1CCC1c1ccccc1)=O)C(F)F c1(C(N(C2CCN(C(CC3CC(C)C3)=O)C2)C)=O)cc(=O)c2ccncc2o1 CC(CC(N)=O)C(=O)N1CCCN(CCC(=O)N2CC(O)CO2)CC1 c1(CCCNC(C(c2cccc(Cl)c2)NC)=O)cc(=NC(=O)OC(C)(C)C)[nH][nH]1 c1(CCC)onc(C)c1C(=O)NCCC(C)NC(C1CCOC1=O)=O c1(CC)c[nH]c2ncnc(N3CCOC(CNC(=O)C(CC)N4CCCC4)C3)c12 Cc1ccc(C(=O)NC2CCN(C(=O)C(C)NC(C3CCCC3)=O)C(C)C2)nc1F c1(C(N2CCC(N(C)C(C3CNC(=O)N3)=O)C2)=O)cc2cc(Cl)sc2[nH]1 Cc1cc(OCCCC(=O)NC(CNC(=O)CNC(N)=O)CC(C)C)ccc1Cl C#CC1C(C(=O)NCCN(C(=O)CCCc2ccccn2)C(C)C)C1(C)C CCC(CNC(C1CC1C(C)(C)C)=O)(CC)NC(=O)CN1CCC(=O)CC1 C(=O)(CS(=O)(=O)CC)N(CCC(=O)N(CC)Cc1cccnc1)CC#C Cc1ccc(Br)c(C(=O)NCC2CCN2C(=O)Cn2ccc(C)n2)c1 N1(C(C2C(c3cn(C(C)C)nc3)C2)=O)CCC(C2CCN(C(C3CCC3)=O)CC2)C1 c1(OC)ccc2[nH]c(C(=O)NCCN(C(=O)CC3CC3(C)C)C3CC3)cc2n1 N1(CCNC(C(=O)NC(C(c2cccc(Cl)c2)OC)C)=O)CCCCCC1 C1(Cc2ccccc2)CN(C(=O)CO)CC12CC2.C(=O)(CCCOC)N(C)C1CC1 C1(CC(NOCC=C)=O)CCCCN1C(=O)COC1CC1 C1(CC=C)(NC(=O)CCCC2(C)N=N2)CCN(C(=O)C(C)(C)Cc2cnn[nH]2)C1 c1(C(=O)NCC2CC(F)(CNC(C(C(C)O)C)=O)C2)c(F)cncc1Br C1(OCC)CC(NC(c2cccnc2NCc2cnn(C3CC3)c2)=O)C12CCC2 C(=O)(CCC(F)F)NCCCO.c1(C(N(C)CCCCS)=O)cn(C(C)(C)C)nn1 Cc1cn2c(n1)C(C(=O)N1CCC3CN(C(C4(O)CC4)=O)CC3C1)CCC2 C1(C(=O)NC(CNC(C2(C=C)CC2)=O)(C)C2CCC2)CCn2nnnc2C1 C1(CC(=O)NCC(CN(C2N(CC)CC2)C)O)SC(=Nc2ccccc2)NC1=O C(C(O)(CNC(=O)C(CCN(C)C)NC(=O)C(c1ccn(C)c1)C)CO)OC Cc1nn(C(C)C)cc1C(c1nnnn1C)NCC(C)OC(C)(C)C C12(CNC(C(CC#C)O)=O)CCCCC1N(C(=O)C(C)C1CCC1)CCC2 O=C(C1CCc2c[nH]nc21)NCC1(O)CCCN(C(=O)C2=CCCC2)CC1 C1(C)(NC(C(Cc2c(C)nc[nH]2)O)=O)CCN(C(c2cccc(C(N)=O)c2)=O)C1 N1(C(C2(COCC)CC(=O)C2)=O)CCC(F)(CNC(C2CCC2OC)=O)C1 CCC(=O)CCC(=O)NOCC(N1CCCC12CCOC2)=O N1(C(C2(CC#C)CC2)=O)CC(NC(C2CC(O)C2)=O)C(C2CC2)C1 c1(CC)nc(CC)c(C)s1.C(=O)(C(C)N1CCN1CCOC)NC(CC)C CC1(C(=O)NCC2CCCC2NC(c2cnn(CC3CC3)c2)=O)CCNC1=O CCC(C(=O)N1CCN(C(c2ccccc2I)=O)CC1)C(C)O C12(CNC(C(C)SC)=O)CCCCC1N(C(c1cc[nH]c1C)=O)CC2 N1(Cc2c(C)ccs2)CC(OCc2cn(C3COC(=O)N3C)nn2)CC(C)(C)C1 c1(C(C(=O)NCC(C(C)C)NC(C2(C)CCCN(C)C2)=O)O)cccc(Cl)c1Cl C(=O)(CCC(C)(C)C)NC(C1CCN(C(=O)CCc2ccc(Cl)s2)C1)C c1(NC(C2CC2CNC(=O)OC(C)(C)C)=O)cc(Cl)c([N+](=O)[O-])cc1O Cc1nc(NC(c2ccc(F)cc2Cl)C)cc(N2CCCC(OCC3CC3)C2)n1 C(=O)(C1=NNC(=O)CC1)N(C(C)CNC(=O)Cc1csc(-c2nc[nH]n2)n1)C c1(SC)cccnc1C(=O)NCCCCNC(=O)CCn1ncn(C)c1=O c1(C(=O)NC(C2(CNC(=O)C#CC3CCCO3)CC2)C)ccc2cnnc(O)c2c1 Cc1cccc(C(N2CC(NC(c3nccc(Cl)c3C)=O)C3(CC3)C2)=O)c1C#N C1(C(=O)NCc2ccc(F)c(O)c2)CC2(CC2)CN1C(=O)Cc1cncnc1 C12(CO)CC1CN(C(c1cc(CNC(C3(N4CCCC4)CC3)=O)on1)=O)C2 C(CC(C)C(=O)NCCN(CC(C)O)C(=O)Cc1cnsc1)=CC c1(C(=O)NC2CCC2c2ccc(F)cc2)ccc(OC(C)(C)C)cc1.C1(=O)CN1C.C C1(O)(N(C(C(=O)NC(COC)C)=O)C)CCN(C(=O)CN(C2CC2)C(C)C)C1 N1(C(C(c2ccc(CC)s2)=O)=O)CCC2CN(C(C3CCCC(=O)N3)=O)CC12 C1(C(=O)NCCCC(C)NC(CCC=C)=O)CC2CC(=O)C1C2 C=C1CC(C(=O)NCc2ccc(Cl)s2)N(C(c2ccnc(F)c2)=O)C1 C(=O)(CC(C)CC(C)C)NCC(CC)NC(=O)C(CO)N(C)C C1(C(=O)Nc2ccc(O)nc2)C2CC1N(C(c1cc(-c3ccco3)no1)=O)C2 Cc1nc2cccc(C(=O)N(C3CCCCC3NC(C3CC4CC4C3)=O)C)c2s1 c1(OCC)ccc(Cl)cc1NC(c1cccc(Cl)c1)c1nnnn1C1COC1 C(=O)(C1=Cc2ccccc2C1O)NC1(C)CCN(C(COC(CC)(C)C)=O)C1 N1CCC=C(c2cccnc2)C1.c1(-c2cccc(Br)c2)cc2c(n1C)CCNC2 N1(C(C2N(C)C(=O)NC2)=O)CCN(C(=O)C(F)C(F)(F)F)CC1c1ncc[nH]1.C1CC1 CCC(C)(C)CC(=O)NCC(=C1CN(C(=O)Cc2ccsc2)C1)F CCC1=C(C(=O)C(=O)CCCCN(C)C(=O)OCC2C(N)CCC2)SCCO1.NC C(CCC)(C(=O)NCCC#CC(C)C)NC(c1c(CC)c[nH]c1)=O C1(C(=O)NCC(C(C)C)C)C2CCC(C2)N1C(=O)CCC1(C)N=N1 CN1CC(C)(C(=O)NC2CCC(NC(c3ccc(Cl)cc3)=O)CC2)CC1=O Cc1c(C(N2CCCC(NC(c3cnc(C#N)s3)=O)C2)=O)cncc1Br C1(NC(C2(OCC)CCCC2)=O)CC2CC(NC(=O)C=Cc3ccc(Cl)s3)C2C1 C(=O)(CCC(=O)c1ccc(Cl)cc1)N(CC(CNC(C(C)c1ncco1)=O)O)C CCCCCCC(C)N(C(=O)C(CCC)c1nn[nH]n1)C c1(C(=O)NCC(C)NC(c2c(NC(C(C)C)=O)scn2)=O)ccc(C(=O)CF)cc1 C1(CNC(C(COC)(C)O)=O)CN(C(=O)C(Br)=C(C)C)CC12CCC2 N1(C(c2n(CC)ccn2)=O)CCC2(C1)CN(C(C1CC13CCCC3)=O)C2 CC1(NC(=O)C(N)=O)CCCCC1C(N1CCC(F)(CF)C1)=O CCC(C)(C)CCN=c1[nH]c(NC2CCn3cncc3C2)nc2c(F)cccc12 C=CCCC(C(=O)NCC(C)(C)C1CCC1)NC(C1CC2(CCC2O)C1)=O N1(C(CN2CC(C)C2)=O)CCC(C2CCN(C(=O)C(CO)N(C)C)C2)C1 CC(C)(C)C(O)CNC(c1ccc(-n2cc(C3CC3C(=O)O)nn2)cc1)=O CCC(C)(CO)C(=O)N1CCC(CCNC(c2cnc(-c3ccccc3)[nH]2)=O)C1 C(=O)(C1Cc2ccccc21)NC1C(C)CCN(c2nccc(C(C)C)n2)C1C C(=O)(C1CCCc2cccnc21)NCC(C(C)C)NC(c1ccc(C)c(F)c1)=O C(C)(C(=O)NCCCCN(C(=O)COC1CCOC1)C)OCC=C c1(C(N2C(CNC(C(F)=CC)=O)CC2)=O)cn(C)nc1-c1ccc(Cl)s1 C1(C(=O)NC(C(=O)NC)C)CC(F)CN(Cc2cc(C)cs2)C1 C(=O)(C(F)CC1CCCCC1)N(C(C)C)CCN(C(=O)C=CC(=O)N(C)C)C1CC1 C1(CN(C)C(C2CCCSC2)=O)C2CN(C(=O)CC3CCCCN3C)CC12 C1(CC)CCCCCN1C(=O)CC(F)(F)c1cccnc1Br C1(CCNC(C2C(COC)C2)=O)CC(F)(F)CN1C(c1cc(C2CC2)no1)=O c1(C(=O)NCC2(NC(C3CCC(CC)O3)=O)CC2)c(Cl)cccc1[N+](=O)[O-] NC1CC(CNC(=O)C(N2CCN(C(=O)C(F)(F)F)CC2)=O)C(O)C1 C1(O)(CNC(C2C(COC)C2)=O)CCN(C(=O)C(C)(C)C#N)C1 c1(C(=O)NC2(CC)CN(C(=O)CC(C)N(C)C)C2)ccc(C(C)C)c(C)c1 Cn1nnc(C=CC(=O)NC2CCCC(NC(c3csc(Cl)c3)=O)C2)n1 C12OCCC1NC2=O.C(CCO)N(C)C(N)=O.C1(=O)CSCCN1 CCCCCC(O)CC(=O)N1CCN(C)C(CNC(c2occ(C)c2C)=O)C1 C1(C(=O)NCCN(C(C2CCCC23CCC3)=O)CC)CC2(CCO1)CC2 N1(C(c2c(N)cc(Cl)nc2)=O)CCC2(CCOCC2)CC1 N1(C(C(CCC)NC(C)=O)=O)CCC(C)(C)C(C(=O)NCCC(C)(C)N(C)C)C1 c1(CC)ccnc(C(=O)NCC(C)N(C(=O)CC)C)c1.c1(C(=O)N)cnn(CC2CC2)c1 N1(C(C(=O)N(CCCO)C(C)C)=O)CCN(C2CCCN(C)C2)C(=O)C1 C1(CCOC)(NC(c2c(C)csc2Cl)=O)CCN(C(c2nc(O)c(C)s2)=O)C1 c1(C(=O)NC(C)(C)C)cc(OCC(=O)N(CCCNC=O)CC)on1.C(C)(C)C Cc1nn(C)c(Cl)c1C(=O)NCCC1CCCN(c2ccnc(C3CC3)n2)C1 c1(OC(C)C)ccc(C(=O)NCC2C=CCN2C(=O)C(O)C(F)F)cc1 CC1OCCC1C(=O)NC(Cc1ccoc1)C(=O)NC(CC1CCC1)CO c1(C(N2C(CCNC(C(CCC)C(C)C)=O)CCC2)=O)nccn2nc(C)cc12 c1(CC)onc(C)c1C(=O)NCC(C1CN(C(=O)COCC(=O)NC)C1)(C)O c1ccc2ocnc2c1.c1(C(=O)OCC)nc(C)c(N)s1.C12C3CC1N(C3)C2=O C12(CNC(c3n(CC)ncc3)=O)CCC(NC(=O)C#CC(C)C)(CO1)C2 N#Cc1cc(F)c(CN2CCCC2CCC(=O)Nc2ccsc2C(N)=O)c(Cl)c1 CC(C)(C(=O)NCC(C)(F)CNC(c1cc(C(F)F)[nH]n1)=O)c1cccs1 CCC1c2ccccc2CCN1C(c1coc(CN)n1)=O n1(CC)nnc(C)c1C(C(=O)NC(C)C)N(CCOC)Cc1ccccn1 n1(CC=C)ncc2c(O)nc(=NCC3(C)CCN(C(=O)C=CBr)C3)[nH]c12 C1(C(=O)NC(CC)C(=O)OC)CC(F)(F)CN1C(C1CCC(C(=O)OC)C1)=O N1(C(CCOCCCOC)=O)CC(C(N2CCC(C)(CO)CC2)=O)C(C2CC2)C1 c1(NC2(CNC(c3cc(CC)no3)=O)CCCCCC2)ncnc2c1ncn2C c1(OC)ncc(C(N2C(C(=O)NCCn3cc(C)cn3)CC3CC23)=O)cn1 C12(NC(c3occ(C)c3)=O)CCC1CN(C(=O)CN1CC(C)C1)C2 c1(CN2CC(c3onc(-c4c(N(C)C)cccc4)n3)C2)c(F)cccc1Cl c1(CC(C)C)cccc(C(=O)NC(c2cn(C3CCC(=O)NC3)nn2)C)c1 N1(c2c(-c3cc(C)[nH]n3)ocn2)CCCC(CCCO)C1 O=C1COC(CNC(=O)C(Cc2cn[nH]c2)NC(=O)Cn2ccccc2=O)CN1 C1(NC(CCCC)=O)CCCCC1NC(C1CCOC1=O)=O CCC(CC)CC(F)C(=O)N(CCC(=O)Nc1cccc2c1CCCC2)OC C(=O)(CCCCCCCC1CC1)NC(CNC(C1CN(CCC)C(=O)C1)=O)C c1(-n2c(Cc3c(C)cco3)nc(C3CC34CC4)n2)ccc(F)cc1C C(CC(C)C)(C(=O)N1CC(CNC(c2nnc(Cl)cc2N)=O)(OC)C1)OC N1(C(CCC2CCC(NC(=O)CNC(=O)C3CC3)C2)=O)CCc2ncncc2C1 c1(CCOC2(CC(=O)NC3CN(C(c4sccc4Cl)=O)C3)CC2)ccccc1 Cc1cc(=NCCC2CCCC3(CCC3)C2)[nH]c(=NCc2ccc(N(C)C)nc2)[nH]1 c1(OC)cc[n+]([O-])c(C(=O)NCC2(O)CC(NC(C3CCCCC(=O)N3)=O)C2)c1 C(=O)(CCCC(C)(C)C)NCCCN(C(=O)CCc1cncn1C)CC CCC(CC)CCC(=O)N(C)CCN(CC(C)C(C)C)C(=O)CCSC N1(C(Cc2c(C)nc(S)s2)=O)CCCC(C)C1CNC(=O)CSC(C)C CC1(C)CN(c2nc(Cl)c(C#N)s2)CCC1NC(=O)CC1CC=CCC1 CC(CN(C)C)CC(=O)N1CCC(F)(C(=O)NCc2ncoc2C2CC2)C1 CCCCC(CC)C(=O)NCC1(C)CC(NC(c2cccc3ncsc23)=O)C1 CC1Oc2ccc(C(=O)NC3CCCN(C(=O)CCc4ncc[nH]4)C3)cc2C1C C1(NC(c2c(Br)ccc(OC)c2)=O)CCCC2CN(C(=O)CC(C)F)CC12 N1(C(c2c(COC)scc2)=O)CCCC(N(C)C(c2cnc3sccn23)=O)CC1 N1(C(c2cccc(CSCC)c2)=O)CCC(NC(=O)Cc2csc(=N)[nH]2)C(C)C1 C1(C(=O)NCc2c(C(=O)NCC3CCC(C)C3)c[nH]n2)CC2(CC(=O)C2)C1 [N-]=[N+]=NC1CCN(C(=O)C(c2cccnc2)NC(=O)C=CC(F)(F)F)CC1O Cc1cnc(C(=O)NCCCC2(NC(C3CCOC3C(F)(F)F)=O)CC2)c(C)c1 c1(C(=O)NCCN(C(CC(C)c2ccco2)=O)C2CCCC2)cc2ncccc2o1 c1(C(=O)NCC2CC(O)CN2C(C2CC(O)CCO2)=O)ccn2ncnc2c1 c1(NC(=O)CCOc2ccc3c(c2)CCC3)nc2cc(F)c(O)c(F)c2s1 C1(NC(CN2C(C)CCC2)=O)CN(C(c2cc(Cl)sc2Cl)=O)CCC1F C1(C(=O)NCCC(C(=O)OC)O)C2CC3C(C2NC(=O)Cc2cn[nH]c2)C13 N1(C(CC2CC(CC)C2)=O)CC2(CCN(C(C3CSCCS3)=O)CC2)CC1C C1(C(=O)NCC(CC)(C)OC)C(C2CC2)CCN1C(c1ccc(C)nc1O)=O c1(C(N(C)CC2CCN(C(=O)CCNS(C)(=O)=O)C2)=O)cnc(N)cn1 c1(C(N(CCC(C)NC(CCCCCC)=O)C)=O)cccc2sncc12 CC(C)CC(F)C(=O)NC1CC(NC(C2(c3cccc(F)c3F)CC2)=O)C1 Cc1cc(-c2nc(CC3(C(F)(F)F)CC3)n(Cc3cnccc3Cl)n2)ccc1F N1(C(C2CCC(=O)NC2)=O)CCC2(CC1)CC(NC(C1CCCOC1)=O)CCO2 C=CCC(CC=C)C(=O)NCC#CC(=O)N(CC(CC)OC)C CCC(C)C(C(=O)N1CC(NC(C2CC2c2cccc(Cl)c2)=O)C(C)C1)OC C1(COC)CC(CNC(c2c[nH]c(=N)s2)=O)N(C(=O)C(C)n2cccn2)C1 CC(CCCNC(C12COCC1C2)=O)NC(=O)CSS(C)(=O)=O N1(C(CSC)=O)CCC(N(C(=O)CCCNS(C)(=O)=O)CC2CC2)C1 C1(C(=O)NC(C)C(C)(C)NC(=O)CC#N)Cc2ccc(Br)cc2C(=O)O1 c1(CC)c(C(=O)NCC2CC2NC(c2ccoc2C)=O)cnn1-c1ccc(C)cc1 CCC(CC(=O)NC1(C)CCN(C(=O)CCCCNC(C)=O)C1)SC C(=O)(N=c1cc[nH]c2ccc(I)cc12)c1ncc(-c2cccc(-n3c(C)ncc3)c2)nc1 CCC(C)(C)C(O)C(=O)N1CCCC1C(C)(C)NC(=O)CC(C)(C)CN(C)C CCCCC(=O)NCCN(C1CCCCC1)C(=O)CC1CCC1(C)C C(=O)(C1=CNS(=O)(=O)N=C1C)NC(CC)CNC(=O)CN(C)C(c1cccs1)=O C1(N(C(=O)CCC2CCC2)CCC)CCN(C(=O)CC(C)C2CCCCC2)CC1 c1(CC=C)cn(CC2CCC(NC(=O)CCN(C)C)C2)nn1 Cc1ccnnc1C(=O)NC(C)C(c1ccccc1)NC(=O)C(C)N(C)C CN1CCCCC1CCC(=O)NC1CCOCC1NC(c1cnsn1)=O C1(C)(CC)CCC(C2CC(F)(CN(C(=O)OC)Cc3ccccn3)C2)O1 C1(NC(c2c(OC)cc(Cl)cc2)=O)CN(C(C2CC3CC2C3)=O)CCC12CCC2 c1(C(N2C3(CCC3)CC(=O)Nc3cnc(s3)C2=O)=O)[nH]c(C)nc1C.CCO.OC Cc1c(NCCc2csc(C3CC3)n2)ncnc1NCC1C(F)(F)C12CCC2 c1(SCC)nccnc1C(N1CCC(O)(CN(C)C(C2CC3CCC3C2)=O)C1)=O C1(NC(c2c[nH]c(=NC)o2)=O)CN(C(c2ccc(OC)nc2OC)=O)CC1(C)C c1(C(=O)NCC2(C)CCN(C(C3CC(C#C)(O)C3)=O)C2)cc(F)c(O)c(F)c1 CCCC(CCC)CC(=O)NCC1C=CCN1C(c1c[nH]cc(F)c1=O)=O Cc1nscc1CC(N1CCCC1C1(NC(c2cnn(C)c2)=O)CC1)=O c1(C(=O)NCCNC(C(C(C)SC)O)=O)ccc2nc(C(F)F)[nH]c2c1 CCC(CC)(C(=O)N1CCCC(NC(=O)CN2CCP(C)(=O)CC2)C1)OC C(CCC)(C(=O)NCC1CC(O)CN1c1ccncn1)=CC(=O)NC CC1CN(C(=O)Cc2cn(C)nn2)CC1CC(=O)NC1(C(N)=O)CC1 C1(NC(C)=O)CCN(C(c2csc(-c3ccco3)n2)=O)CC1.c12cn(nn1)C2 C(=O)(CC(C)NC(C1CCN(CCCO)C1)=O)OC CC1(C)C(CC(=O)NCCc2cocn2)CCN1C(c1cnc(S)nc1)=O c1(CC)cc(C(=O)NCC(C2CC2)NC(C2CC2CF)=O)cc(O)n1 C1(CC(=O)NCCC(=O)OC(C)C)C2CN(C(c3cncn3C)=O)CC12 C1(C)(CC)CC(C(N2CCN(C(C3C4CC5C(C4)C35)=O)C(C3CC3)C2)=O)CCO1 CC(C)CCC(=O)NC1COCC1NC(c1cnn(C)c1Br)=O C1(NC(C2(C=C)CCCCC2)=O)CC2(CCCCC2)C1.c12sccc1CNC2=O C(=O)(CCCCCCCCCO)NC1CC(C)N(C(C2CC(C)(O)C2)=O)CC1 C1(OC)CN(C(C2(CC=Cc3ccccc3)CC2)=O)CC1NC(=O)C(C)(F)F Cc1c(C(N2CCCC2C2CCN(C(c3nnn(C)c3CO)=O)C2)=O)cccc1O N1(C(COCC#C)=O)CCOC(C(C)NC(=O)Nc2cc(CCC=C)on2)C1 C(=O)(C(C(C)C)Nc1ccccc1)NCCCC1(NC(c2c(C)cco2)=O)CC1 N1CCCC(F)(CO)C1.C#CC1(C(=O)NCCNC(=O)C(C)C)CCCC1 c1(C(N(C)CCOCCCNC(c2cnc(S)nc2)=O)=O)cc(F)cc(N)c1F Cc1ccnc(C(=O)N(CCC(=O)N)CCCO)c1F.N1(CCO)CCC1 C(=O)(C#CC1CCCCC1)N1C(CNC(=O)Cc2ccno2)CC(COC)C1 C#Cc1cc(F)c(C(=O)NCCC(C)NC(c2cnnn2C)=O)c(F)c1 N1(C(c2cc(C)c(S(N)(=O)=O)s2)=O)CCc2c(ccc(Cl)c2F)C1 CC1C(C(=O)N(CCO)CC2CC2)CCN1C(c1csc(Cl)c1)=O N1(C(C(CC2CC2)NC(Cc2c(CC)con2)=O)=O)CCCC12CCCC2 C1(NC(c2ccc(F)cc2)=O)CN(S(=O)(=O)Cc2ccc(Br)cc2F)CC1(F)F C=CC(C)(C)CCNC(=O)C(C)(CSC)NC(=O)C=C1CCC1 Cc1ccc(CN2C(=S)NC(c3cnn(C(C(=O)O)C(C)C)c3)C2)c(C2CC2)n1 Cc1noc(C(C)C)c1C(=O)NC1CCCN(CCC2CCCN2C)C1 C1(NC(C(C)=C(C)C)=O)COC2(C1)CN(C(=O)C(C)(C)C(=O)N(C)C)C2 c1(N(C)CC2CCN(OCc3ccccc3)CC2)cc(F)ccc1N1CCCC1 c1(CNC(C(CCOCC)NC(=O)C(C)CO)=O)cc(C)cnc1O Cc1nn(CC(N2CC(CNC(C3CCC(F)CC3)=O)C(C)C2)=O)cc1Cl C(=O)(C(C)(O)COC)N1CC(CCNC(c2sccc2Cl)=O)(OC)C1 C(N=c1ccnc(Nc2ccc(C)c(C#N)c2)[nH]1)c1c(C)nc(OCC)s1.n1(C)nnnn1 C1(c2ccccc2)(NC(C(COC)C)=O)CCN(C(c2cnsc2)=O)C1 c1(N(CC)CC)ccc(C(=O)NCc2cnc(Sc3c(C)csc3C)s2)c(O)c1 c1(OCC)ncc(C(=O)NC2(CNC(=O)CCc3cc[nH]n3)CCCC2)cn1 C(C)(N=c1[nH]c2cc(F)ccc2o1)C1N(C(C2C(CCC)CCC2)=O)CCCC1 C(=O)(C(CCC)S(N)(=O)=O)NCCC(=C)CNC(C1CCC(C)(C)C1)=O N1(C(C(COC)OC)=O)CCCCC1CNC(=O)CCCCN(C)C C(CC(=O)C1=C(c2cccc(F)c2)CCC1)N(C)C(c1ccc(C#N)cc1O)=O C#Cc1ccc(C(=O)NCCN(C(=O)C=C(Cl)Cl)CC(C)O)cc1C c1(CNS(N(CC)CC)(=O)=O)cc(F)cc2c1CCC2 Cc1nc2cccc(C(N3CCCC3C(C)NC(C3COCCO3)=O)=O)c2[nH]1 N1(C(CC2CN(C)C2)=O)CC(NC(=O)CC=C(Cl)Cl)C2CCCC2C1 N1(C(C#CC(C)(C)O)=O)CC2(CCC2)CC1CNC(=O)CCCn1cncn1 Cc1c[nH]nc1C(=O)NCC(C)(Cn1cccn1)NC(=O)CCc1ccncn1 C#Cc1ccc(C)c(NC(=O)C(CCOCCO)NC(=O)C(C2CC2)SC)c1 c1(C(N2CC3(N(C(c4c(COC)nn[nH]4)=O)CC3)C2)=O)c(C)c(C)cc(C)c1C C(=O)(C1=NN(C)C(=O)CC1)NCC12CC(NC(c3oc(C)c(Br)c3)=O)(C1)C2 N1(C(c2nc(C(=O)OC)oc2)=O)C2CCC1CN(C(c1cc(Cl)cnc1C)=O)C2 Cc1cnc(C(=O)NCC2CCN(C(C3CCCN(S(C)(=O)=O)C3)=O)C2)c(C)c1 Cc1c(C(N2CC(NC(c3ccccn3)=O)C3CC23)=O)sc2[nH]cnc(=S)c12 C1(C(=O)NCCN(C(c2c(CC)[nH]cc2)=O)C)C2CC3C(C2)C13 CCC(C)C(C)C(=O)NCCN(C(C1CCCC1CC)=O)C1CC1 c1(-n2cc(CC(C(=O)O)NC(C3C(F)(F)C34CCC4)=O)nn2)cccc(F)c1F Cc1cncc(CCC(=O)N(CCCCCNC(=O)CC2CCC(F)(F)C2)C)c1 CC1(C)CN(C(=O)CCC2CCCCN2C(=O)C#CC2CCC2)CCS1 c1(C(=O)NC2CC(CCNC(C3(CC#C)CCOC3)=O)C2)cccc(N(C)C)c1 c1(C(C(=O)NCC(C2CCC2)NC(C(C)=CC)=O)(F)F)ccc(C)cc1 N1(C(CNS(N)(=O)=O)=O)CCN(C(=O)Cc2ccns2)C2(CCC2)C1 N#CC1(C(N2CC(CC(F)C(=O)NCC3(C4CCC4)CC3)C2)=O)CC2CC2C1 CC1(CNC(C2(C)CCCO2)=O)CCN(C(C2(C3CCCCO3)CC2)=O)C1 N1(C(CC2CCCN(C)C2)=O)CCC2C1CCN2C(c1cc[n+]([O-])cc1)=O CC1(C)CC(CNC(=O)Cc2c(F)cccc2Cl)N(C(=O)Cc2cnc[nH]2)C1 c1(C(=O)NC2CCN(C(C3(CF)CCC3)=O)CC2F)n[nH]c2c1CCSC2 N(C(=NCCn1cccn1)NCCc1nccs1)C(C)CC1CCCO1 N1(C(c2c(CC)ncs2)=O)CCCN(C(C2CS(=O)(=O)CC(=O)N2)=O)C(C)C1 C12(C(N3C4CC(NC(Cc5c(C)cccc5)=O)C(C4)C3)=O)CC(C)(C1)OC2(C)C c1(OC)ccc(OC)c2[nH]c(C(=O)NCCNC(=O)C(F)(F)c3cncs3)cc12 C1(=CCNC(C2C(CC)C2)=O)CCN(c2nccc(-n3ccnc3)n2)CC1 CC(O)C(F)(F)C(=O)N1CCN(C(=O)C=Cc2cc[nH]n2)C(CC(F)F)C1 CCCC(C#N)C(=O)NC1CC2(C1)CC(C(N(C)CC1(OC)CC1)=O)C2 C(CCC(O)C(=O)NCc1cccc(CO)n1)NC(c1cc[nH]c1)=O c1(C(=O)NCC23C(CN(C(C(C)C)=O)C2)C3)cc(NC(C2CC2C)=O)ccc1Cl N1(C(C2CCN(C(c3cn(CCC)nc3)=O)CC2)=O)CC(C)CCC1CC c1(C(N2CC(CCNC(C=C(CC)C)=O)C2)=O)ccc(Br)cc1OC.C1CC1 c1(CC(=O)N(CCNC(CC2(C)CC2(F)Cl)=O)CC2CC2)ccc2nn[nH]c2c1 N1(C(=O)Cc2cncnc2O)CC2CCCC(C1)N2C(c1ccsc1C1CC1)=O N1(C(C(CC)C)=O)CCC(C)(CNC(c2cc(Cl)ccn2)=O)C1.C1(=O)CN1 c1(NC(C(CC)(C)C(N)=O)=O)cc2c(cn1)OCCC2.C12CC3CN(CC13)C2=O C1(C(=O)NCC2(O)CCN(C(=O)C(Cl)=CCl)C2)CC2CCC(C1)C2 N1(Cc2c(OC)cccc2)CCC(=O)N(Cc2ccoc2)C1=O C#Cc1ccccc1CNC(=O)C(N1CCC(C(=O)NC)CC1)c1ccon1 CCCCCC(O)CC(=O)N1CCCCCC1CNC(C1CCN2CCOCC12)=O Cc1nc(NC(c2[nH]cnc2C#N)=O)ccc1-c1cncc(O)c1 N1(c2cc(N3CCC(C#C)C3)ncn2)CCN2CCCC2C1 Cc1cc(C(N2CC(N3CC(NC(=O)OC(C)(C)C)CC3=O)C2)=O)ccc1Cl c1(CNC(CCC(C)NC(C2(CN)CCCC2O)=O)=O)cc(Cl)cc(Cl)c1 C(CN=c1ccnc(N2CCC(C3CCC3)C2)[nH]1)OCC(c1ccccc1)C Cc1cc(NC(c2ccncc2Cl)c2nnnn2C(C)(C)C)ccc1F N1(C(c2ccnn2CCF)=O)CC2CCC1CN2C(C1CCn2nncc2C1)=O Cc1c(-c2ccccc2)c(C(=O)NC(C)CC(C)(C)O)nc2[nH]nc(O)c12 c1(C(=O)NC(CC)CNC(=O)COc2cccc(Cl)c2Cl)cccc2scnc12 CCC(CCC(=O)NCCCN1CCCC1=O)NC(c1ccc([N+](=O)[O-])o1)=O c1(-c2ccc(C(=O)NC(c3ccc(OC(C)C)cc3)CC)nc2)ccc(F)cc1C N1(C(CCNC(=O)OC)=O)CC(OC)CC1(C)C C=CC(C)(O)CC(=O)NCC1CC(NC(=O)CCNS(C)(=O)=O)C1 CC1CC(CNC(C2CCC23CCC3)=O)CCN1C(c1ccco1)=O C1(CCNC(C=CC(=O)N(C)C)=O)CN(C(=O)CSC2CCOC2=O)CCO1 c1(C(=O)NCCCNC(=O)Cc2cnccc2Cl)cc(Cl)cc([N+](=O)[O-])c1 N1(C(c2c(C)nc(=N)[nH]c2)=O)CC2CCOC2(CNC(c2cnoc2)=O)C1 CC1CC2(CCN(C(c3ccc(Cl)[nH]3)=O)CC2)CN1C(c1coc(CO)c1)=O C1(NC(COCCOCC#C)=O)CCCCC12CCN(C(=O)Cc1cnc[nH]1)C2 N1(C(CC2(C(=O)OC)CC2)=O)CC2CCC1(CNC(C1CCC(OC)C1)=O)CC2 CCC(O)C(C)C(=O)N1CC2CC(C1)C2NC(=O)CCCCCN(C)C c1(C(=O)NC(C)CCN(C)C(c2cnn(C)c2F)=O)ccc(N)cc1[N+](=O)[O-] CC(C1Cc2ccccc21)Nc1ccccc1OC(F)(F)F CCCC(CCC)=CC(=O)NCCCC1CCCN1C(c1cnoc1C1CC1)=O N1(C(C2(C)CC(=C)C2)=O)CCN(C)CC1C(=O)NC(C)Cn1cncn1 c1(OC)ccc(C(F)(F)C(=O)NCC2CCN(C(c3cc(C)c[nH]3)=O)C2)nc1 CCCCCC(O)C(=O)N1CCCC1(C)CNC(c1cccc2ccoc12)=O N1(C(C2(OC)CC(C)C2)=O)CCOCC(NC(c2ccn(C3CC3)n2)=O)C1 c1(NC(C(C)N(CCC)C(c2ccc(C#N)cc2)C)=O)ccc2ccccc2c1 c1(NC(C(c2cccnc2)C)=O)cc2[nH]ccc2cc1-c1cc(OC)ncc1F O=C(CCOCC1CCCO1)NOC1CCCCC1.C1C(=O)O1 CCN=C(NCC(c1sccc1C)OC)N1CC2CC(C1)C1CCCCN1C2 C1(NC(c2c(CC)ocn2)=O)CCCN(C(=O)C2=C(Cl)CCCC2)CCC1 CCCCC(CNC(C1CC(C)(C)CO1)=O)NC(=O)Cn1cc(CO)nn1 c1(COC)cccnc1.C12CC(C1)C(=O)N(C1COC1)CCCNC(=O)C(C)O2 C1(CC(=O)NCCCOCCN(C(CN(C)CC)=O)C)CCCCO1 C(c1ccc(Cl)cc1F)=CC(=O)NC12CCC(C1)N(C(C1CC(=C3CC3)C1)=O)C2 C1(N(C(c2scc(CC)c2)=O)CC)CCCN(C(C2C(C)C2C)=O)CC1 C1(C(=O)NC2CC2CNC(=O)Cc2cncc(F)c2)(OC)CCSCC1 c1(C(=O)NC(CNC(CSCC#C)=O)(C)C2CC2)cc([N+](=O)[O-])ccc1NC c1(C(=O)NCCC2N(C(C(CO)NC(N)=O)=O)CCCC2)nccc2n[nH]cc12 c1(C(=O)NC(CC)(C)CNC(=O)C(C)(C)N(C)C)cc2c(o1)CCCC2 N1(C(C(C(C)C)(C)O)=O)CCC2(CC1)CN(c1ncc3ccsc3n1)CCO2 c1(C(N(C2CCN(C(C3(CCN(C)C)CC3)=O)C2)CCC)=O)n[nH]c(C2CC2)c1Cl C(N=C(NCc1nc(-c2ccco2)n[nH]1)N1CCCCC1)C1C(O)CCCC1 C12=NC(=NCCN1C)Nc1ccccc12.C1(=CCSC)CC(=O)N(C(C)C)C1 N1(C(C)C(=O)N(c2nc(Cl)c(C#N)n2C)C2CC2)C(=O)NC2(CC(C(F)(F)F)C2)C1=O O=S(=O)(c1cccc(=NCCC=CBr)[nH]1)N1CC2CCC(C1)O2 C1(NC(C2C(CCOC)C2)=O)CCN(C(c2cnn3c2OCCC3)=O)CC(O)C1 C1(N(C(c2cccc(C(C)=O)c2)=O)C)CCN(C(c2ocnc2C)=O)CC1C CC1=C(C(=O)NC2CCC(C)N(C(=O)C(N3CCCCC3=O)C)C2)CCS1(=O)=O C1(C2CC2)(C(=O)NCc2c(C)cccn2)CN(C(c2cc(=N)[nH][nH]2)=O)C1 Cc1cc(C(N2CCCC2CNC(C2CCCC(F)C2)=O)=O)c2c(c1)CCCN2 N1(C(CCOCC)=O)CC(N=c2[nH]ccn3nnnc23)C(C)(C)C1 c1(CC)nc(C)ncc1C(=O)NC1CN(C(c2c[nH]cc2C(C)(C)C)=O)CC1O C1(NC(c2cc(C)nc(O)c2)=O)CCCOC12CCN(c1nnco1)CC2 CCCC(C)(C)CC(=O)NC1CC(NC(C2(F)CCCN(C)C2)=O)C(O)C1 c1(C(=O)NC(C)CN(C)C(C2CCC(C)(C)OC2)=O)cc(Cl)c(Cl)cc1N c1(N(C2CC3CNC2C3)C(C2CC(O)C2)=O)ccc2c(c1)OCCO2 CCCC(C)(O)C(=O)N1CC(C(C)NC(c2ncncc2OC)=O)C1 C#CC1(O)CCN(C(C2CCN(C(c3c[nH]nc3CCC)=O)C2C)=O)C1 c1(C(=O)NCC(CNC(C2(CN3CCCC3)CC2)=O)O)nn(CC(C)=O)cc1C C1(C(NOCCCOC)=O)(CNC(c2c[nH]c(C)c2)=O)CC12CCC2 Cc1ccc(C(N2CC(F)(F)CC2CNC(C2CCN(C)C2=O)=O)=O)c(N)n1 c1(C(=O)Nc2c(C)cc(OC(C)C)cc2)ccc2cccnc2c1 c1(CCC(=O)NCCC(C)NC(=O)C(C)NS(C)(=O)=O)nnc(-c2ccco2)o1 CC(C(=O)NC(C)(C)CCNC(C1CC(n2cnnc2)C1)=O)C(F)(F)C(F)F Cc1nn(C)c(-n2cncn2)c1C(=O)N(C)CCN(C(=O)CCCC1CCC1)C C1(C(=O)NCC(Cn2cc(-c3c(C)scc3)nn2)(F)F)CCC2CC(=O)CN12 c1(C(N2CCC(NC(COCCCC)=O)C(C)C2)=O)c(F)cc(C)cc1Cl C1(CC)CN(C(=O)C2=CCCC2)CCC1NC(c1ccc(OC(F)F)c(C)c1)=O C1(C(=O)OCC(=O)Nc2cc(Br)ccc2Cl)CC2(CCOC2)C1 Cc1sc2ncn(CCC(=O)NC(C)CCNC(C3C(C)C3C)=O)c(=O)c2c1C c1(C(=O)NC(CCN(C(C(C)OCCC=C)=O)C)C)cc(C(C)C)nc(O)c1 N1(C(C(CCSC)NC(C)=O)=O)CC(C(=O)Nc2ccc(F)c(C)n2)C2(CC2)C1 Cc1cc(C)c(C(N2CCCCC2CN(C(=O)CCNc2ccccn2)C)=O)s1 CCCC(C#N)C(=O)NC(C1CCN(C(=O)C=CCF)CC1)(C)C c1(C(=O)NC2C(NC(C3(SC)CCC3)=O)CCC2)cc(C#N)ccc1Br C(=O)(C(C)S(C)(=O)=O)NCC(N1CCCC(C(CC)CC)C1)=O c1(C(=O)NC(C)CN(C)C(c2ccn(CC#N)n2)=O)ccc2nc[nH]c2c1F C1(CNC(=O)CCn2ccnn2)CCCC1C(=O)NCC(N1CCCC1)C Cc1cc(N2CC3C(C2)C3(C)C)ncc1S(=O)(=O)NC1CCc2ccc(Br)cc21 O=CN1CCCC1C(=O)NC(Cc1ccco1)C(=O)NC1CC(CCF)C1 C(CNC(=O)CCCc1ncco1)(C(=O)NCCCCC1CC1)N(C)C N1(C(C2C(CC(C)(C)C)C2)=O)CC2CCC(C1)N2C(C1(C)COC1)=O Cn1c(CNC(=O)NCc2conc2C(C)(C)C)cnc1[N+](=O)[O-] CC(C)C1C(=O)NC1=O.C(=O)(CC(C)(C)c1ccccc1)OC(C)(C)C Cc1cc(=O)c(C(N2CCC(C(C)NC(=O)CSc3ccccn3)CC2)=O)c[nH]1 c1(OC)nc(Cl)ccc1C(=O)NC1CCCN(C(c2ccc(CO)nc2)=O)CC1 c1(C(=O)OCC)nc(C(=O)NCCC(C)NC(c2ccn(C3CCC3)n2)=O)cs1 N1(C(c2cccc(Cl)c2)C)CC2CC1CN(C(c1cc(CC3CC3)[nH]n1)=O)C2 C1(F)(CNC(C(c2nc[nH]n2)OC)=O)CCCN(C(c2ccn(C)c2)=O)C1 CC1=CCC(C)(C(=O)NCc2nnc(C)s2)CC1 N1(C(C(C)CSC(F)(F)F)=O)CCC(NC(=O)C(=O)NC2CC2)C1c1cccnc1 c1(CO)ccc2c(c1)COC2.N1(C(c2ccccc2)C=C)CC2OCC1C2 C1(NC(=O)Cc2cnns2)CCCN(CCN(C(c2c[nH]c(Br)c2)=O)C2CC2)C1 c1(CC(=O)N(C2CCC(NC(C=NOC)=O)CC2)C)ccc2ccccc2c1 Cc1ccc(C(N2CC3C(CNC(c4cnc(Cl)s4)=O)C3C2)=O)c(F)c1F N1(C(c2c(NC)cncc2)=O)CCCN(C(c2ccc(F)cc2F)=O)C(CO)C1 C1(C(N2CC3C(CO)C3C2)=O)CCN(C(=O)C2COCC2O)O1 C1(CC#C)(C(=O)Nc2ccc(C(=O)NC3CCCC3NC=O)s2)CCCCC1.SCC Cc1cn2c(CC(N3CC(C(=O)Nc4cccc(NC)c4)CC3C)=O)csc2n1 N1(c2nc(N3CC4CCC(C3)O4)cc(C)n2)CC2(CCOCC2)CC1CO N1(C(C2OCC(C)C2)=O)CCC2(CC1)CN(C(=O)CCCC(C)(C)C)C2 c1(C(=O)NC(C2N(C(c3occ(C)c3)=O)CCCC2)C)c(C)nn(C)c1F N1(C(C(C)=C(CC)C)=O)CCC(C2CC2NC(=O)C(N2CCCC2=O)OC)CC1 N1(C(C(C=CC)O)=O)CCN(C(c2cncnc2C)=O)C2CS(=O)(=O)CC12 C1(NC(c2ccc(CC)s2)=O)CN(C(=O)Cn2cc(F)ccc2=O)CCC1F C12(C(=O)NC(CNC(c3c(C)cccc3)=O)CO)OCCCC1C2(F)F c1(OC)cc(N)ccc1C(=O)NC1CCC(CNC(C2CC=CCC2)=O)CC1 c1(C(C)(C)C)nccc(C(N2CCN(C(c3ccccc3Br)=O)CC2)=O)n1 c1(CN(CC(C)NCC2CC2)C)ccc(C(N)=O)nc1 c1(C(=O)NCC2C(C)(C)CCO2)cc(O)nc2c1CN(C(=O)Cc1nc[nH]n1)CC2 Cn1cc(NC(=O)C(N2CCC(c3nc(NC(c4cccs4)=O)n[nH]3)C2)=O)cn1 c1(C(N2CC(C)(CNC(=O)CN3CC=CC3)OCC2)=O)ccc2nccnc2n1 CC1NC(=O)OC12CN(C(=O)CC(C(F)(F)F)NC(=O)CC(Cl)Cl)C2 c1(C(N(C(CNC(COCCC#C)=O)C2CC2)C)=O)cc(Cl)c(Cl)s1 C1(NC(=O)C(=O)Nc2ccccc2)CN(C=O)CCC1F.C(CCC1(O)CC1)NC Cc1c(N)cc(C(N2CCCC(NC(c3[nH]cnc3C)=O)C2C(C)C)=O)cc1Cl Cc1nn2c(C(=O)NCCNC(=O)C(C)Cc3cccc(Cl)c3Cl)c(C)nc2s1 c1(C(=O)NCCC2OCCN(C(CCc3onc(C)n3)=O)C2)ccc(Br)c(O)c1 C(C(CCC)C(=O)N1CC=CC1CN(C)C)NC(C1C(=C)C1)=O c1(C(=O)NC(CN(C(C(Cc2c(C)nc[nH]2)O)=O)C)(C)C)cc(F)cc(Cl)c1N c1(C(CC(=O)NC(CCNC(C(C)n2cnnn2)=O)(C)C)O)cc(Cl)cc(Cl)c1 N1(C(c2ncn(CC)c2)=O)CCC(O)C(C(=O)NC2(CC(=O)OC)CCC2)C1 N1(C2CCN(C(C(N3CC(O)(Cc4[nH]c(=N)sc4)C3)=O)=O)C2)CC(=O)NC1=O N1(C(C2CN(CC)C(=O)C2)=O)CCN(C(=O)Cc2cnsc2)C(C)C1 C#CC1(C(=O)NC(C2CCCO2)CNC(=O)CN(C)C(=O)OC)CC(=O)C1 C1(NC(c2cc(OCC)ns2)=O)CN(C(C2CCOC2(C)C)=O)CC2(CCC2)C1 Cc1ccc(C(N2CCC(NC(=O)Cc3nonc3C)CC2)=O)nc1 c1(C(N2CC(NC(C(c3ccc(CC)cc3)O)=O)C2)=O)nc(C)ccc1C#N C1(CNC(c2c(C)cncc2)=O)CC2(C1)CN(C(=O)Cn1ccnn1)C2 N1(C(c2cnc(C)o2)=O)CCOC(C(C)NC(C2CNC(=O)N2C)=O)C1 N1(C(Cn2c(=N)nn[nH]2)=O)CCN(C(=O)CC2CC2(Cl)Cl)CC1 N1(C(C=CC(=O)NC2CC2)=O)CC(NC(C23COC(CCO2)C3)=O)CC(O)C1 C(C(CO)(CO)NC(=O)C(C)OC1CCCCC1)N(C(CCCOCC=C)=O)C N1(C(C2(OC)CCCC2)=O)CC2(C1)C(NC(=O)CC(=O)NC1CC1)CCS2(=O)=O C12(C(=O)NC(C3CCN(C(=O)CCc4cncn4C)C3)C)CCCC1C2(F)F N1(C(CCCC(=O)OCC)=O)CCC(NC(c2ccncc2)=O)C(CO)CC1 c1(C(=O)NCC2CN(C(c3cnc(CC)s3)=O)C(C)C2)cc(O)cc(N)c1Cl N1(C(C2(CCOCC)CCCC2)=O)CC(NC(=O)C(F)(F)CN(C)C)CC(O)C1 CC(O)CCN=c1nc2c(ncn2C)c(NC2CC2c2cccc(Cl)c2)[nH]1 C12(C(=O)NC(C)CNC(c3ccc(C4CC4)c(F)c3)=O)C(=O)C3CCC1C2C3 N1(C(C(C)CSC(F)(F)F)=O)CCC(NC(c2ncoc2C(F)(F)F)=O)C12CC2 C(=O)(CCC(C)(F)F)N1CCC(C(N(CC(C)C)C)=O)(C(C)C)C1 c1(CC(N2CCC(O)(CN(C(C(C)NC3CC3)=O)C)C2)=O)cnn2c1OCCC2 n1(CC(N2CCN(C(C3C(C=C)CC3)=O)C(CC)C2)=O)nc(C)c2cccnc12 N1(C(C(COC)COC)=O)CCN(C(=O)CNc2cccc(C)c2C)C(CF)C1 c1(C(=O)NC(C2CCCC2)CNC(c2cc(Cl)on2)=O)sccc1C1CC1 C1(F)(C(=O)NC2(COC)CCC2)CCCN(C(C2(C)CCCCO2)=O)C1 c1(-c2cn(CC3N(CC(N4CCC(C(=O)O)C4)=O)CCC3)nn2)cc(Cl)ccc1F c1(CC(=O)NCCC2(C)CCN(C(C3CC(C)C3)=O)C2)ccc2c(c1)OCO2 C(=O)(CC1=CCOCC1)NCC1(C(C)NC(c2ccn(C3CCC3)n2)=O)CC1 C(=O)(CCCCC(C)(C)C)N1C(C)(C(=O)NC(C)CCC2CCCC2)C=CC1 CC1CCN(C(=O)NC(C)(C)C)C(NCc2ccc(Oc3cccnc3)cc2)C1 N1(C(C=CCCC)=O)CC(NC(=O)Cc2cnn(C)c2)CC12CCCC2 CCCC(CNC(=O)C=Cc1cc[nH]c1)C(=O)NCCc1c(O)n[nH]c1C c1(CC)nc(C(N2CCCC2(C)CNC(C2CCN(C)C2)=O)=O)c2ccccn12 c1(NC(C2CC3CC3N2S(=O)(=O)CCCCl)=O)ccc(Cl)cc1I N1(C(c2ccnc3ccncc23)=O)CCc2ncc([N+](=O)[O-])cc2C1 c1(NCCC(=O)NCC)ccc(S(=O)(=O)NCCC2SCCS2)cc1Cl Cc1cc(=NC(=O)C2CC(C)CN2C(c2cccc(Br)n2)=O)[nH]c(C)c1C#N N1(C(C(C)(C)Sc2ccccc2)=O)CC=C(CCNC(C2CCCS2)=O)CC1 C12(CNC(=O)C3=CCCC3)CCC(Nc3ncc(O)cn3)(CC1)CO2 c1(OC)ccc(-n2nnnc2C2(NCCS(N)(=O)=O)CC(C(N)=O)C2)c(C)c1 C1(CNC(CC(C=C)C)=O)CN(C(=O)C(C2CCCCCCC2)O)CCCO1 N1(C(c2cc(C(C)=O)on2)=O)C2CCC(C2)C1CNC(c1ccc([N+](=O)[O-])o1)=O c1(C(=O)NC2CCC(C(=O)Nc3ncc(C)cc3I)C2)cc(Cl)c(O)cc1F c1(C(CCOC)C2CC2)cn(CC2CCCN2C(C2CC(C)(CO)C2)=O)nn1 Cc1ccc2c(=NCCN(CC(C)C)C)[nH]c(=NCC3(COC)CCC3)[nH]c2c1 CC(c1cccc(Cl)c1)=CC(N1CC(NC(c2ccoc2C)=O)CC1C)=O N1(C(C2N(C)CC2)=O)C2CCC(C2)C1CC(=O)NCCC(O)CO c1(C(=O)NCC2CCC(F)C2)cc(-c2ccccn2)cnc1O CN1CC2OCCN(C(=O)CN(c3ncn(C)n3)C(=O)CC(Cl)Cl)C2C1 c1(C(=O)NC2CCC(C)(NC(C3C(COC)C3)=O)CC2)c(OC)ccc(Cl)c1C C1(NC(C(COC)C)=O)CCN(C2CCN(C(c3csc(CO)n3)=O)CC2)CC1 CC1=C(C(=O)NC2CCN(C(C3CCCN3C)=O)C2)CCC1 N1(C(C(C)=CCC)=O)CCCC1C1(NC(=O)CCCc2cccs2)CC1 C(=O)(C1=CCC(C)CC1)NCC(C(C)C)NC(c1cnc(C(C)OCC)s1)=O c1(CC)c(NC(C2(NC(=O)C(CO)N3CCCC3)CCCC2)=O)cnn1C CCCCCC(C)CCNC(C)C(=O)NC1CCCCC1 C=CC(CC)C(=O)NCC(CC1CC1)C(=O)NC1CCCC1CCC C(c1cccc(F)c1)=CC(=O)NCC1N(C(c2c(CC)n(C)nc2)=O)CCCC1 N1(C(c2nc(CC)oc2)=O)CCOCC1CN(C(=O)COc1ccon1)C1CC1 Cc1cnc(Cl)c(C(=O)NCCN(C(=O)CNC(c2ccc(C)c(C)c2)=O)C)c1 CC(C)CC(C(=O)NCC1(C)CCCO1)NC(=O)CC1(C)CCOCC1 c1(C(N2CCC(C(=O)NCCCC(=O)NC)CC2C)=O)cccn2nccc12 N1(C(c2n(CC)nnc2)=O)CCCC(C)(NC(=O)CCc2cnco2)C1 C(=O)(C(C)(C)C(F)(F)F)N1CCN(C(c2cncc(NC)n2)=O)C(C2CC2)C1 c1(C(N(C)CC2N(C(C3C(OCC)CC3)=O)CCOC2)=O)cn2c(n1)SCC2 N1(C(C2C(CC)OCC2)=O)CCCC2(CCN(C(c3n[nH]c(C)c3F)=O)C2)C1 C(CC)(CC)(CCNC(c1ccc(C(C)=O)cc1)=O)NC(C(CC=C)C)=O C(C(O)C(=O)NC(CO)C(C)NC(c1cnn(-c2ccncc2)c1)=O)=CC Cc1nn(C)c2c(NCCN3CCCC3C)nc(N3CC4C(C3)C4(C)C)nc12 c1(C(N2C(CNC(=O)CCOC3CCCCC3)CC2)=O)cccc2c1NCCC2 N1(C(C(C)OC)=O)CCC(NC(=O)CCOc2ccccc2O)C12CC2 N1(C(COC)=O)CCC(O)(C(F)(F)C(N)=O)CC1.OC C(=O)(C(C)(C)CCCF)N1CC(C(C)NC(=O)CN2CCSCC2)OCC1 C1(C(=O)NC(CN(C(=O)C(F)OC(F)(F)F)C)(C)C)CCCC(O)C1 C(CCO)(CC(C)C)NC(C1(NC(c2c(OC)nn(C)c2)=O)CC(O)C1)=O C1(C2CCCN(C(c3nnsc3C(F)F)=O)C2)(NC(C(CC)C(C)C)=O)CC1 c1(C(C)(C)OC)nc(=NC2CCCCC2CNC(C2CCC(=O)N2C)=O)s[nH]1 CCC(O)C(C)(C)C(=O)N(CC)CC1CCN(C(=O)CC2CCCOCC2)CC1 C1(CCNC(c2ccn(CCN(C)C)n2)=O)CCCN(C(c2coc(Cl)n2)=O)C1 N1(C(C(COC(C)C)NC(c2nc(CCC)oc2)=O)=O)CC=CC(O)C1 C1(C(N(CCOC)CCNC(C2(n3cncn3)CC2)=O)=O)CC2CC2C1 c1(C(N2C(CNC(C(C(C)C)OCC)=O)CCCC2)=O)cc(=O)n2ccsc2n1 C1(C(=O)NCC2(NC(C3OCCO3)=O)CCCC2)(OC)CCCOC1 c1(C(=O)NC2C(NC(Cc3nc(C(C)OCC)sc3)=O)C2)ccc(OC)nc1C C(C)(CCCC(=O)N1CC(C)(O)CO1)NC(C(CC)CCOC)=O N1(C(=O)OC(C)(C)C)CCCC(CC(=O)NCC(C(F)(F)F)N2CCCC2)CC1 C(=O)(CCC(C)CN(C)C)NC1CN(C(COc2cc(C)on2)=O)CC1C c1(C(N2CCC(C)(O)C2)=O)cn2c(n1)CN(C(c1cc(F)c(Cl)cc1F)=O)CC2 N1(C(c2n(COC)ncc2)=O)CCCCC1CNC(=O)C(C)c1ccsn1 C1(C(N2CC=CC(C(=O)NCc3ncn(C(C)C)n3)C2)=O)(OC)CCCCC1 c1(CNC(C(C(C)(C)C)c2nn[nH]n2)=O)cn2cc(Cl)cc(Cl)c2n1 c1(C(=O)NCC2C(NC(C(CSC)C)=O)CCC2)ccc2ncnc(O)c2c1 C(CCC(N)=O)(C(=O)NC1CCN(Cc2cc(F)c(Br)cc2C)CC1F)SC c1(NCC2(OCC)CN(C(=O)NC3CCC(N=[N+]=[N-])C3)C2)nc(C)c(C)nc1C c1(CN2CC(O)(CC(=O)N(c3nccs3)C)C2)cnccc1C(F)(F)F c1(CC)cn2c(n1)CCC(C(=O)NC1CC(NC(=O)C3CCc4c[nH]nc43)C1)C2 c1(C(C(=O)NCC(=C)C)N(c2ccccc2)CCCO)cncc2ccccc12 c1(C(=O)NC2C(OC)CN(C(c3ccc(C#N)o3)=O)C2)cc(F)c(F)cc1Cl N1(C(C(C)(C2CCC2)OC)=O)CC2CC(NC(=O)C=C(C=CCC)CC)CC2C1 n1(CC(=O)NC2CCC2)ccc(=NCc2cc(F)cc3cccnc23)nc1O Cn1ccc2ccnc(C(=O)NCC3CCCN(C(C4(C)CC=CC4)=O)C3)c12 N1(C(c2cccc(OC)c2)=O)CCN(C(=O)CCN2CCCC2)C2CCC12 N1(C(COC(C)C)=O)CC(C(=O)NC2(C(C)C)CC2)C2(CCC2)C1 N1(CC)CCOC(C(=O)NCC=CCNC(=O)CCn2cccc2)C1 C(CSc1ncc[nH]1)(C(F)(F)F)Oc1ccccc1.C1(=O)C(=O)N(C2CC2)N1C C1(F)(CNC(=O)CCc2nc(-c3ccsc3)no2)CN(C(C2CCCCS2)=O)C1 c1(C(=O)NC23CC(C(=O)NCCc4cccc(C)c4F)(C2)C3)c(Br)cc(F)cc1Br CC1CCN(CCC(N2CC3C(CNC(C4CC(Cl)(Cl)C4)=O)C3C2)=O)CC1 C1(OC)CCOCC1N=c1cc(C)nc(NC2CN3CCC2C3)[nH]1 c1(C(=O)NCC(C)(O)CNC(=O)C=CC(=O)N(C)C)ccc(Cl)c([N+](=O)[O-])c1 C1(CC(=O)NC2(C(N(CC(CC)OC)C)=O)CCCC2)CCCC12CC2 Cc1ccc2c(N3CCC4(CC3)CC(NC(=O)C(Cl)(Cl)Cl)C4)ncnc2c1 c1(CC(=O)NCCCOCCCNC(C2COC(=O)N2)=O)ccsc1Br C12(NC(CC3C(C)=NOC3=O)=O)CCC(CNC(c3cnn(CF)c3)=O)(CC1)OC2 c1(CC)c(C(=O)N(C2CCCC2)CCCC2(CC#N)CCCC2)cnn1CCO C1(C(=O)NCC(CN(C)C(C2C=CCCC2)=O)(C)C)Cc2ccccc2O1 C1(C(N2CCC(C)C2(C)C)=O)COc2cccc(F)c2O1 c1(C(N(CCNC(C2CC2(C)C)=O)CC)=O)cnc(C(F)(F)F)s1 c1(C(C(C)C)NC(C2CCC3(CC2)CC3)=O)nc2ccccc2s1 N(C(=NCCSC1CCOCC1)NCC1(C#N)CC1)C(CC)C C(=O)(C1=C(CC)OCCC1)NCCCN(CCC)C(C1(C#N)CCCOC1)=O c1(C(N2CCC(C(C)(C)OC)C2)=O)[nH]c(Cl)c(Cl)c1Br C1(NC(C(C)(C)CF)=O)COC2(CCN(C(C3CC3c3cccnc3)=O)CC2)C1 Cc1csc2ncc(C(=O)NC3(CO)CN(C(c4ccc(C(=O)OC)[nH]4)=O)C3)n12 c1(C(=O)NC2C(C)(C)CN(C(=O)CCc3ccco3)C2)cnc2ccncc2c1 C1(C(=O)NCCN(C(=O)C=C2CCN(C)CC2)C(C)C)CC12CCOC2 c1(C(N2CC3C(C(=O)Nc4c(C)cc(F)cc4)(CC3)C2)=O)cc2cccnc2[nH]1 c1(OC(C(=O)N(CC(=O)OC)CCC(C(=O)NC)(C)O)C)ccc(Cl)cc1 n1(CCCC)nc(-c2ccnn2C)nc1CC1CCC1 C1(NC(C2CN(C(C)C)C2)=O)C2CCC1N(C(=O)C(c1ccc(F)cc1)(F)F)C2 c1(CC(=O)N(C(CC)C(=O)OC)CCC)csc2nccn12 C12(CC)CN(C(c3cn(C)nc3C(C)(C)C)=O)C(CNC(C3CC3F)=O)(C1)C2 N(C1CCc2cccnc21)C(C1N(C(c2ccc(OCC)cc2I)=O)C2C(C1)C2)=O C1(NC(C(C)NC(CC)=O)=O)CN(C(c2cc3ncccc3s2)=O)CC12CCC2 C=CC1CCCN(c2nnc(C3(OC)CC3)n2CCC=C(C)C)C1 C(=O)(C1CCCc2nccn21)N(CC(CN(C(C(C=C)(C)C)=O)C)O)C N1(C(CCc2cnc(C)s2)=O)CCCN(C(C2CC3(C2)CC(C)(C)C3)=O)CCC1 C1(O)(CC(=O)NCc2cnc(Br)s2)CCCN(C(c2cc(Br)ncc2Br)=O)C1 Cc1ccc(C(=O)NCCOCCN(C)C(c2cc(C3CC3)cs2)=O)cc1C n1(CCCC(N2C(CN(C(C3CC3(F)F)=O)CC)CCC2)=O)nc(C)cc1C CC1CCC(C2CCC2)CN1C(=O)C(N1CC(C)(Cc2ccccc2)C1)=O C1(C(=O)NC2CCN(CC)C2)C2CC3C(C2=O)C13.c1(C(=O)N)c[nH]c(C(N)=O)c1 C(=O)(C(=O)NOC)NCC(C(=O)NCc1ccc(SC)o1)N(C)C c1(CN2CCCC(NC(c3cccc(Cl)c3Cl)=O)C2)cc(F)c(Br)cc1[N+](=O)[O-] CCC(C)(C)C(=O)N1CC(NC(=O)CCc2ncco2)C(c2cncn2C)C1 c1(C(=O)NCC2(N(C(C(c3ccccc3)SC)=O)C)CC2)cc(F)cc(F)c1F CC1C(C(N2CCOC(CCNC(c3ccnn3CC(F)F)=O)C2)=O)CCN1C C(=O)(C(C)CCCC(C)=O)NC(CCC=C)C(N1CCCC2(C=CCO2)C1)=O c1(C(=O)NCc2cc(OC)ncc2-c2ccn(C)n2)cc(F)c2cc[nH]c2c1 C(=O)(C(C)(C)C(C)C)NCC(CC)NC(c1cc(Cl)ccc1Cl)=O CC(F)(F)CCC(=O)NCC(F)CNC(=O)COCCCc1ccccc1 N1(CC(=O)NCCCCCC)CCC(=O)N(CC(c2csnn2)OC)C1=O c1(CC)ccc(C(=O)NCC2CC(O)CN2C(=O)CCC2CC(C)(C)CO2)nc1 C(C(=O)N(CCSC)NC(C1CC1C)=O)N(CC)CC Cc1cc2c(cc1C)OC(COC(C1CC(=O)CO1)=O)C2 N1(C(c2c(O)cccc2Cl)=O)CCCC2C1CCN2Cc1cc(O)cc(F)c1 C1(CNC(C(C)(C)C2CCOC2)=O)CN(CC2(O)CCCCC2)CCO1 c1(NCC2(C)CC2)[nH]c(=NCCN2CCNC2=O)nc2sccc12 C1(NC(c2ccc(OC)c(C)c2)=O)CC2CC1CN(C(=O)C(C(C)C)NC=O)C2 N1(C(c2nc(C(=O)OC)sc2)=O)CC(CNC(c2scnc2C(C)C)=O)CC1C C(=O)(CS(=O)(=O)Cc1cccs1)NCC1CN(C(c2cc(C)no2)=O)CC1O O=C(C(Cc1ccc(O)cc1)C(F)(F)F)NC1CC2OC1C1CC21 C1(NC(C(=O)N(C)Cc2ccc(OC)cc2)=O)CC2(CCCCO2)C1 C1(NC(C(C)SC(C)C)=O)CN(C(c2ccc(CN(C)C)o2)=O)C2CCCCC12 C1(NC(C2CCC(C)O2)=O)CN(C(=O)Cc2ccoc2)CC12CCCC2 C(=O)(CCCC(=O)NC(C)C)NC(CC=C)CNC(=O)C=CC(=O)N(C)C C1(CCNC(c2nccc(CC)c2)=O)CN(C(C2CCCN2C)=O)CC(C)O1 C1(SC)CC(N=c2nc3scnc3c(NCCc3ccc(C)c([N+](=O)[O-])c3)[nH]2)C1 c1(N2C(CCNC(C3CCC(OC)CC3)=O)CCC2)nc(Cl)nc2c1ncn2C Cc1cc(NC(=O)N(C2CCC(C(=O)OC(C)C)CC2)C)cnc1O N1(C(C2CNC(=O)N2)=O)CC(NC(C2(O)CC2)=O)C2CCCCC12 CS(=O)(=O)c1cccc(C(N2CCC(NC(C3CCSC3)=O)C(O)C2)=O)c1 N1(C(c2c(CCC)nns2)=O)CCC2CN(C(c3ccc(N(C)C)nc3)=O)C2C1 C#CCCCC(C)C(=O)NCC(C)N(C(=O)CCCN1C(=O)CN(C)C1=O)C Cc1cc(CCCC(=O)N(C)CCOCCNC(c2nnc(S)n2C)=O)c(C)s1 N1(CC)C(=O)CCC1C(N1CC(NC(c2ccn(CC(F)(F)F)n2)=O)C(O)C1)=O CN1CC(C(=O)NCCCC2CCN(C(C3CC(O)(C(F)F)C3)=O)CC2)CC1=O Cc1ccc(F)c(C(=O)NC2CC(CCNC(c3nnc(S)n3C)=O)C2)n1 c1(C(N(CCCNC(=O)CC2OCCC2(C)C)C)=O)cccn2[nH]c(=N)nc12 C1(C2(O)CN(C(=O)CC(F)(F)C(F)F)C2)(CNC(CC23CC(C)(OC2)C3)=O)CC1 c1(C(=O)NC(CC)CN(C)C(C2CCCCN2C(C)=O)=O)cc(Cl)c(Cl)cc1N CC1CCCC=C1C(=O)NC1(CN(C(=O)C2=CCCCCC2)C)CC1 C1(CN(CC(=C)C)CC)CCCCN1C(=O)CCCOCCOC N1(C(c2cc(C)nn2C2CCC2)=O)CCC2(NC(C3CC(F)(F)C3)=O)CCCC12 C=CCC(C(=O)NC(C(N1CCC(OCCO)C1)=O)c1cccs1)C(C)C C1(CNC(C(CC)CC2CCCCC2)=O)C(C)CCCN1C(=O)COc1ccsn1 N1(CC(C)N(C)C)CCCC1C1CCCCN1C(C12CC(C)(C1)OC2(C)C)=O CC1(F)CCC(C(=O)NNC(=O)c2ccccn2)CC1 C1(C(N(CCCNC(C(c2cccnc2)C)=O)C)=O)CC(Cl)(Cl)C1 c1(C(=O)NCC(C)=CC(=O)NCC2CC3(C2)CC32CC2)cc2cc[nH]c2cn1 C=CCCC(F)(F)C(=O)NCC1(O)CCN(C(=O)C(C)NC(=O)NC2CCC2)C1 c1(C(=O)NCC2C(C)CCN2C(C2C(C)(C)C2(C)C)=O)cc(Br)c(C#N)s1 c1(C(=O)NCC2(F)CC(NC(CS(CC)(=O)=O)=O)C2)cc2ccc(F)cc2o1 c1(C(C)C)oncc1C(=O)NCC1(CNC(c2ccc(C)s2)=O)CCC1 N1(C(C2CC(=C)C2)=O)CCOC(CNC(C2CC(C)(O)C2)=O)C1 C12(OC)CCCCC1CN(C(c1sc3cncn3c1C)=O)C2 C(CCCCCS(N)(=O)=O)NC(c1nn(CC)nc1C)c1nnnn1C(C)(C)C C1(c2n(CCOCC)nnn2)(NC(CC)C(C)(C)C)CCOC(C(F)(F)F)C1 C12(C(=O)Nc3cc(C)c(NC(C4CC(O)C(F)C4)=O)cc3)CCC(CC1)C2(C)C C(=O)(C1=NOC2(CCOC2)C1)N1CC(C)(NC(c2c(Cl)cccc2[N+](=O)[O-])=O)C1 C1(NC(c2ccsn2)=O)CCN(C(c2ccns2)=O)CC1O N1(C(C2(C)CCCN2C(c2cccc3nccn23)=O)=O)CCC(CO)C(F)(F)CC1 C1(C(N(CCC(=O)NCC2(C)CC3CC3C2)CC2CC2)=O)CC2(CCC2)CO1 N1(C(CNC(=O)CC2CCc3nc[nH]c3C2)C2CC2)CCC12CCC(CO)CC2 C1(C(=O)NCCNC(=O)CO)C2CC1N(C(=O)CC1CCCSC1)C2 C(CCC(C)C)(C(=O)NC(C)(C)CCCC1CC1)NC(CCOCCOC)=O C(=O)(N=c1ccn(C(C)C)[nH]1)C1C2CN(C(C(CC(=C)Cl)OC)=O)CC21 c1(C(C)NC(=O)Nc2ccnn2CC2CC2)nccc2ccccc12 n1(CC)cc([N+](=O)[O-])c(C(=O)NC2(COC)CN(C(=O)COCCCF)C2)n1 C(C)(N=c1cc[nH]c(=NCCC2CCC3CC23)[nH]1)c1cccc(COC)n1 N1(C(COc2cc(C)on2)=O)CC2CC(NC(=O)Cc3ccc(Cl)c(F)c3)C2C1 C(=O)(C1CCCc2nncn21)N1CCN(C(CNC(C(C)CC(N)=O)=O)=O)CC1 c1(C(N2CCC(CN(CCC)C)C2)=O)c(C)nn(CC(F)F)c1C Cc1cc(F)c(CC(=O)NCC(O)CCNC(=O)CCS(C)=O)cc1F C1(CCC)CN(C(c2nc(SC)cn2C)=O)CCN1C(=O)Cc1c[nH]ccc1=O c1(CNCC2C(F)(F)CCN(C(=O)CC(F)(F)F)C2)cc([N+](=O)[O-])cc(Br)c1O CC1CCN(C(c2ncoc2C2CCNC2)=O)CC1Cc1ccc(Br)o1 C1(CNC(CCS(=O)(=O)N(C)C)=O)CCC2(CN(C(C3CCOCC3)=O)C2)O1 Cc1cnc(Cl)[nH]c1=NCCCCNC(C1CCC(CCOC2CCC2)CC1)=O C1(NC(C(C)CC#N)=O)CN(C(=O)CC2CCC2)C2(CCC2)C1 Cc1cc(C(N2CC3CC3(CNC(c3nnn(C)c3N)=O)C2)=O)cc(F)c1 C=CCCCCCCN=c1[nH]c(=NCc2cnn(CC=CC)c2)c2ncccc2[nH]1 c1(C(=O)NC(CN(C(C2CC2F)=O)CC)C)ccc2c(n1)OCC(=O)N2 c1(C(=O)NCC(C2CC2)NC(C(c2ccc(OC)cc2)O)=O)cc2c(ncn2C)[nH]1 C1(CC)(CC)CC(NC(=O)CCc2ccc(F)cc2)CN1C(=O)C=CC(C)C C1(C(N2CC(COC(C)C)C2)=O)(CNC(c2cccnc2O)=O)CC12CCC2 C(C)(C)(CC(=O)N(C1CN(CC)C(=O)C1)c1nccs1)NC(c1snnc1C)=O N1(C(CC=CC=C)=O)CC2(C1)CN(C(=O)C(n1ccc(C3CC3)n1)C)CCO2 N1(C(C(CCC)F)=O)CCC(NC(c2ccc(OC)cc2F)=O)C(CO)C1 c1(OC)cc(C)cc(C(N2CC(NC(=O)C(F)=C(C)C3CC3)CC(F)C2)=O)c1C C1(C(=O)OC)CCN(C(C2(CNC(c3cc[nH]n3)=O)CC=CC2)=O)C1C N(C1CN(C(=O)COCCSC)Cc2ccccc21)C(CC(C=C)CC)=O C(N=c1[nH]c(N2CCC(SC)C2)nc2c(F)cccc12)C1CCN(C(C)=O)C1 CC1(C)CN(C(=O)C(F)C(C)(C)O)CC1NC(C1CCC2CC2C1)=O c1(C(=O)OC)c(C)ccnc1NC1CN(C(C2(C3CC3)CC2)=O)CCC1CO c1(C(N2CCCC(CNC(CCCCOC)=O)C2)=O)nn2c(c1C)CCCC2 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CC)(CC)CCNC(=O)C(C#N)CC N1(C(C(=Cc2ccco2)C)=O)CCN(C(=O)Cc2csnn2)C2CCCC2(C)C1 C1(NC(CNC(=O)OCC=C)=O)CCCC(C(=O)NCc2csc(C)c2C)C1 C1(CNC(C2CC3CCCC23)=O)CC2CCC1N2C(C1CC1(F)F)=O c1(C2N(C(C3CNCC(C)C3)=O)CCC2)ccc([N+](=O)[O-])cc1 Cc1ccc(C(=O)N2CCC(C(=O)NCC34CC(CCO3)C4)O2)cc1F C1(O)(C(=O)NC2CC(NC(C(C(COC)C)C)=O)C2)CN2CCC1CC2 CCC(C)(C)C(O)C(=O)N1CC2CN(C(=O)C(C)OC)CC2C1 C(=O)(C1=NOC2(CCC2)C1)NC1(C)CCN(C(CC2CCCC(C)O2)=O)CC1 C1(CNC(Cc2cnc(C)s2)=O)COCC2(CCN(C(=O)C=CCF)C2)O1 C12(NC(c3cc(C)[nH]n3)=O)CCCN(C(=O)Cc3c(C)cc(F)cc3C)CC1C2 N1(C(Cn2cnc(=N)[nH]2)=O)CC2(C1)CN(C(c1csc(C3CC3)n1)=O)CC2CO c1(NCc2c(S(C)(=O)=O)cccc2)nccc(=NCC2=CCCC2)[nH]1 Cc1nc(C(C)C)ncc1C(=O)NCC1(C)CCCN1C(=O)CC(C)CF c1(CN2CCCC(C(=O)Nc3nnc(Br)s3)CC2)ccc(F)c(Br)c1F N1(C(c2c(CCC)nco2)=O)CCC(C(=O)OC(C)(C)C)C(CO)C1 Cc1cc(C)c(-c2nc(C(c3ccccc3F)O)no2)cn1 c1(CC)cc(C(=O)N(CCN(C)C(c2ncnc(C)c2C)=O)C(C)C)cc(F)c1 O=C1CC(CC(=O)NC23CC(NC(C4CCCCC4(F)F)=O)(C2)C3)=NN1 C=C1CC2CC1CN2C(=O)C(C)(CSC)NC(=O)CC1CCC(C)(C)O1 c1(NC(c2cc(C(C)C)nn2CCO)=O)ccccc1C#N.n12cc(nn1)C2 C(=O)(C1=NOC2(CCC2)C1)N1CC(COC)(CNC(c2ccn(C)n2)=O)C1 C(=O)(C(C)CC(N)=O)NC(C1(O)CN(C(CC2(OC)CC2)=O)C1)C C(C(N=c1[nH]nc(C#N)s1)c1ccccc1)NC(c1c(F)ncc(OC)c1)=O c1(C(N2CCC(C(C(=O)NCC(C)OCC#C)(C)C)C2)=O)ccc(CC#N)cc1 Cn1cc(C#CCNC(=O)NC2(c3cccc(Br)c3)CCC2)cn1 c1(CN2C3CN(C(c4n[nH]c(C)c4C(F)(F)F)=O)C(C3)C2)ccc(C#N)c(F)c1 c1(CC(=O)NCCC2CCC(NC(C(CC)(C)F)=O)C2)ccc([N+](=O)[O-])cc1 c1(C(N(C2CCCN(C(=O)CC3CC3(C)C)C2)C)=O)c[nH]c2cnccc12 N1(C(C2CCC(=O)N2)=O)CCOC(CCNC(c2cccc(C(F)(F)F)n2)=O)C1 c1(C(N(C2CCC(NC(c3ccc(CO)cc3)=O)C2)C)=O)ccn2nnnc2c1 Cc1c(C(=O)NCC2CCC2NC(=O)CCCc2ccccn2)cncc1N C12(CNC(c3nn(C(CC)C)c(C)c3)=O)CCC(CC1)N2c1ncns1 N1(C(CC(C(C)C)C)=O)CCC(CNC(=O)Cc2cccs2)C(F)(F)C1 c1(C(=O)NCC(CC(=O)NCCC2(COC)CC2)C)ncc(C)cc1C C1(C(N(C)CC2CCCN(C(COCC#C)=O)C2)=O)CN2CCN1CC2 C1(CCn2ncc(Cl)c2)CN(N2CCC(CN3CCCCC3)CC2)C1 c1(C(N(CC(C)NC(COC(CC)(C)C)=O)C)=O)cc(OC)c(OC)c(N)c1 S(=O)(=O)(c1cc(C(=O)NCC2CC3(CCC3)CN2C(=O)C(C)O)c(C)o1)NC C1(NC(Cn2c(C)ncc2)=O)CCCN(C(c2scnc2C(F)(F)F)=O)CC1F Cc1ccc(N)cc1C(=O)N(CC(C)NC(c1coc(-c2cnn(C)c2)n1)=O)C C12(C(=O)NCC3(F)CC(CNC(C(CC)(C)C)=O)C3)CC1COC2(C)C N1(C(CCC(C)(C)NC(Cc2cnc(C)s2)=O)=O)Cc2n[nH]cc2C1CO C1(C(=O)NC2(CCNC(=O)CCCC3CCCCC3)CCC2)COC2(CCC2)C1 CC1CC(C(=O)NCC2CCCCC2NC(C2CCOC(C(C)C)C2)=O)=NO1 C1(NC(C(C)S(N)(=O)=O)=O)CCN(C(c2n[nH]cc2Br)=O)CC1(C)C CC(CC(C)NC(c1ccn(CC(F)F)n1)=O)NC(C1CC(F)(CO)C1)=O c1(C(N2CCC(C)(C(=O)Nc3c(OC)nccc3)C2)=O)c(C)cccc1C N1(C(CC(CC=C)(C)C)=O)CC2CC(C)N(C(C3CCCN3C3CC3)=O)C2C1 CCCC(CCCNC(c1ccc(CC(C)(C)C)cc1)=O)NC(=O)C=CC1CC1 N1(C(CCOCC)=O)CCN(C(=O)CC2OC(C)(C)OC2=O)CC1C1CCCC1 CC1CN(C(c2coc(Cl)n2)=O)CC1NC(c1cnc(OC2CCOCC2)cn1)=O c1(N(CC(=O)NC)C)nnc(-c2cnc(SC)nc2)n1Cc1cccc(OC)c1 N1(C(C(C(C)C)O)=O)CCN(C(c2cc(=O)n(C)o2)=O)C(c2cccc(Cl)c2)C1 C1(COC)CN(C(c2ccccc2-c2nc(S)n[nH]2)=O)CCN1C(=O)C(C)SC CON1CCC(C(=O)NC2CC(O)C2CC(=O)NCC(F)C2CCC2)CC1 C1(O)(C(N(C2CCC3CC23)CC)=O)CCC(NC(=O)OC(C)(C)C)CC1 CC(C)C(C)C(C)CC(=O)N1CCCC1CN(c1nccc(S(C)(=O)=O)n1)C N12CCCC1C2.C(C(=O)N(CC(=O)N(CCO)C1CC1)C)NC(=O)NC CN1CCCN(C(=O)C(C(C)(C)C)NC(c2ccc[nH]2)=O)CC1 C1(CC)(CC)CC(NC(c2cc(O)n(C)n2)=O)CN1C(=O)CSC1CCOC1=O C1(C(N(CCCNC(=O)C(F)(F)c2ccccc2)C)=O)CCc2ncccc2C1 C(CN=c1[nH]ncn2ccc(Br)c12)(C1CCCC1)OC CC(C)C(F)(CNC(=O)CCC(CF)CF)C(=O)NC(C)(C)CCC1CC1 C=CCCC(F)(F)C(=O)N(CCCCCNC(c1cc(Cl)cs1)=O)C(C)C N1(c2nnc(C3(OC)CCC3)n2Cc2ccccc2)CCc2c(ccnc2Cl)C1 Cn1cnc2c1C(C(=O)N1CCOC(CCNC(=O)CS(N)(=O)=O)C1)CC(=O)N2 N1(C(C(CC)NC(c2ccccc2)=O)=O)CC2CC(C)N(C(=O)CSC(F)F)C2C1 c1(C(=O)NC2CN(C(=O)Cc3ccnc(Br)c3)CC2F)cc(Cl)c(Cl)cn1 N1(C(C2CCC(C)(C)OC2)=O)CC2(CCCC2NC(=O)C2=CCCOC2)C1 C(=O)(CC(C(C)CC)NC(=O)C(c1ccnn1C)C)NC1CC(C#C)C1 C(c1ccc(Cl)cc1F)=CC(=O)N(C(c1cn(CCCCCC)nn1)C)C c1(C(=O)NCC2CC(OC)CN2C(c2cccs2)=O)csc(=NC2CC2)[nH]1 N1(C(C2(OC)CC2)=O)CC(CNC(c2oc3c[nH]nc3c2C)=O)N2CCC1C2 C123CCCC1N(CCC2)C3=O.c1(OC)ccccc1NC(c1ccncc1F)=O c1(OC)ccc2c(n1)NC(C(=O)N(CCCCNC(=O)Cn1ccnn1)C)C2 c1(SCC)ccc([N+](=O)[O-])cc1C(=O)NC1CN(C(=O)C(C)N(C)C)CC1F Cc1ccc(NC(=O)NC2COC(CSc3ccccc3F)C2)cc1.C1C(=O)N1 CC1CCCC(C(=O)NCc2ncccc2C(F)(F)F)O1 CCC(CC(=O)NC1(CO)CCCCC1)NC(=O)C(C)C(C)NC(C)=O c1(C(=O)NC2(C)CN(C(c3ccnc(O)c3)=O)C2)cc2n(n1)CCCNC2=O C(=O)(C(C(C)C)NC(c1ccc(OC)cc1)=O)NC1(COCC)CC1 N1(C(C(CC(=C)C)C)=O)c2ccccc2C(C(N)=O)CC1C C12(CNC(C(c3cccc(O)c3)C)=O)CCCC1CN(C(=O)Cc1ccon1)C2 c1(NC(CC(CC)NC(=O)C(C(C)C)N(C)C)=O)cccc2c1CCC2 C1(N(CC(=O)NC2CCCNC2)C)CCN(CC(F)F)CC1 c1(C(N2C(CC)CN(C(=O)COC(F)(F)F)CC2)=O)coc2c1CCCC2 Cc1nc2ccnn2c(C)c1C(=O)NCCC1COCCN1C(=O)COC(C)C C1(CC)CN(C(c2ccccc2Br)C(=O)NC2CCC2)CC(C)O1 N1(C(CN(C)CC)=O)CC(NC(C23CC(CF)(CO2)C3)=O)C(F)C1 N1(C(C2CC3(CC3)CO2)=O)C2COCC1C2.c12nocc1C(=O)NC2C c1(CN(CCNC(c2nc(CCC(C)C)oc2)=O)C(C)C)nc2ccccc2[nH]1 c1(CN(CC(C)C)Cc2ccc(I)cc2)ccc(Br)cc1 C1(CC)CN(C(=O)CCSC)CC1NC(=O)CC(C)(C)OC(C)=O c1(OC)ccc(Cl)cc1C(F)(F)C(=O)NCC(CO)NC(C1CCSC1)=O C(=O)(N1CCCc2ccnn21)C1OCCC(NC(c2cnc(C)s2)=O)C1 N1(C(c2ccn(CC)n2)=O)CCN(C(=O)CCC=C2CCCCC2)CC1 N#Cc1nccc2cc(NC(C3CCN(Cc4cccc(Cl)c4Cl)C3)=O)ccc12 C(=O)(CC(F)(F)C(C)C)NCCOC(CNC(C1CCCN(C(C)C)C1)=O)(C)C C(C(C)(C)CC(=O)N1C2(CC2)C1)N(C)C.c1(NCCC(C)O)cccc(C#N)c1 C1(C(=O)NC(C)CC2CCCCC2)CC2(CCN1C(=O)C(C)C(F)(F)F)CC2 N1(C(C2NCCC2C2CCC2)=O)Cc2ccccc2CC12CCC2 N1(C(C(CC=C)OC)=O)CC(C)(C)OCC1C(=O)Nc1csnc1OC N1(C(CCC2CC(OC)C2)=O)CCCN(C(c2cnc([N+](=O)[O-])n2C)=O)C(C)C1 C=CC(C)(CCOC)C(=O)NCC(CCNC(c1cc(C(F)(F)F)no1)=O)OC C(CCN=C(NC(C)C1CC1)NC1CC(=O)N(C(C)(C)C)C1)=C(C)C c1(CN(C)C(=O)NCC2CCC3COC2O3)ccc2sc(=N)[nH]c2c1 Nc1cc(C(=O)NC2CC(CO)N(C(c3cnsn3)=O)C2)cc(F)c1 Cc1ncncc1C(=O)NOC1(CO)CCN(C(=O)C=CC(F)F)C1 N1(C(C(CCC=C)(C)C)=O)CC2COCCC2(NC(C2CCCN(C)C2)=O)C1 C1(C)(NC(c2nc(C(C)NC(C=C(C)C)=O)oc2)=O)CC=CCC1 C1(OC)(CO)CN(C(C2(CCNC(=O)C(C)CO)CCCC2)=O)C1 c1(C(C)C)ccc(C(C)CC(=O)N(C)CCNC(=O)C=CC2CCCN2C)cc1 c1(CC)c(C(=O)NC2CCCCC2NC(=O)CC2CCCCN2C(C)=O)nnn1C Cc1nc(C(=O)NC(C)(C)CC(=O)N2CC=CC(O)C2)sc1C C1(S(N)(=O)=O)(C(N2C(CNC(c3c(C(=O)OC)coc3)=O)COCC2)=O)CC1 N1(C(c2c(CC)nn(C3CC3)c2)=O)CC2CN(C(=O)CC(O)C(C)CC)CCC12 c1(CC)cc(C(=O)NC2CC(C)(NC(=O)Cc3csc4nccn34)C2)ccc1C c1(C(N2C(C)CC(NC(C(CC)CC3CCCCC3)=O)C2)=O)c[nH]c(=N)cc1C C1(NC(C2C(CCC)C2)=O)CC2(C1)CC(C(=O)NOCC1CC1)C2 c1(-c2nc(C(C)C(F)(F)N3CCCCC3)sc2)ccccc1Br Cc1cc(Cl)ccc1OCC1CN(C(=O)C2=NOC(CC3CCC(=O)C3)C2)C1 C1(NC(c2ccc(CC)s2)=O)CC2(C1)CC2C(N1CC2CC2(CC)C1)=O Cc1ccc2c(c1)C(C(=O)N1CCC3(CC1)OCc1ccncc13)CC2 c1(CN2CCC(NC(c3c(C)nc(Br)cc3)=O)C(F)C2)ccc(Br)c2nsnc12 c1(C(=O)NCC(C)(C)NC(c2cc(CNC3CCCCO3)on2)=O)ccncc1Cl c1(C(N2CCCC2C(N2CCC3CC23)=O)=O)ccc(Br)c(Cl)c1F N1(C(C2C(C)(C)C2)=O)CC2CCN(Cc3c(O)cccc3Cl)CC2C1 C#CC(CNC(=O)CCN(C(=O)CC1CCCO1)CCO)C(C)C C1(C)(C(=O)NCCSCc2ccc(C)cc2)CCCN(c2cc(C#N)ncn2)C1 CC(CCCNC(=O)C(C)(F)c1ccccc1)NC(C1(O)CCCC1)=O CCC(C)CCC(O)CC(=O)N(CCNC(=O)C1CC1)CCOC N1(CC(=O)N(C)C2CC2)C2CCC1CN(C(c1cnon1)=O)C2 c1(C(N(C2CCC(NC(c3ncccc3Cl)=O)C2)C)=O)cn2c(n1)SCC2 C(N=c1cc(NCCn2cnc(Br)n2)nc[nH]1)c1c(C)sc(Br)n1 c1(C(=O)NCCN(C(CC=C(C)C)=O)C2CC2)ccnc(OC2CC2)c1 N1(C(c2[nH]ccc(=N)n2)=O)CCC2CC1CN(C(C1CCC3(CCC3)CC1)=O)C2 C1(OCC=C)CCN(C(=O)CC2C3CN(C(=O)CC(Cl)Cl)CC23)CC1 CC1CC2(CC2)CN1C(c1cc(CNC(c2cncs2)=O)on1)=O c1(C(N2CC(CCNC(C(C)C3CC3)=O)OCC2)=O)cc2n(n1)CCC2 C(C)(CCC(=O)NCC(C)NC(=O)C(C)Cc1ccncc1)OCC C(C)(N=c1[nH]n(C)c(C(=O)NCC)c1[N+](=O)[O-])C1N(C(C=CC)=O)CCCC1 C(=O)(C1=C(Cl)CCC1)NCC1(C(N2CC(C)SCC2)=O)CCCC1 N1(C(CN2CCC(OC)C2)=O)CCCCC(CNC(=O)CCC2OCCO2)C1 Cc1c(N)cc(C(N2CCC(NC(C3CCS(=O)(=O)N3)=O)C(C)C2)=O)cc1N C1(NC(C2CC(OC)C2)=O)CC2CC(NC(c3cncc(C(C)(C)C)c3)=O)C2C1 c1(C(N(C2CCCC(NC(c3c(C#C)c[nH]n3)=O)C2)C)=O)cccn2nccc12 Cc1sccc1C(c1nnnn1CCOCC1CC1)NCC(=O)N(C)O c1(C(=O)NCC(CNC(c2cnc(O)o2)=O)OC)cc(CN2CCCC2)ccn1 C1(NC(CCCCC)=O)C2CC3CC(C2)CC1(CNC(=O)C(F)(F)CC)C3 C1(NC(C2C(=O)NCC2)=O)CN(C(c2ccc3occc3c2)=O)C2(CCC2)C1 N1(C(C(COC)O)=O)CCC2(CCCN2C(=O)C=Cc2ccoc2)CC1 N1(C(C(C2CC2)NC(c2oc(CC)c(C)c2)=O)=O)CCC2(CNC(=O)N2)C1 C1(C)(CNC(Cc2ncc(C)o2)=O)CCCN(C(c2cc(Cl)no2)=O)C1 C1(OCC)CC2(C1)CC2C(=O)NCC(O)CNC(=O)Cc1cnccc1Cl c1(SCC)ccc(C(=O)N(CCNC(C2CCC(=O)NC2)=O)CC2CC2)cn1 CC1CN(C(=O)C=Cc2ncco2)CC1NC(=O)C(c1ccc(Br)cc1)C C(C(=O)N(CCCNC(C1(C)CCC1(C)C(=O)O)=O)C)(C(C)C)c1cc(C)no1 C1(CC(=O)NCc2ccc(COC)o2)COCCN1C(=O)CC1CC(OC)C1 Nc1c(F)cc(C(=O)NC2CCC(NC(C3(CO)CCCCC3)=O)C2)cc1F C(CNC(C1CC2CC2N1C(=O)CCC(C)N(C)C)=O)(C(C)(C)C)OC C(=O)(CCC1=NNC(=O)CC1)N1CC(NC(c2nc(OCC)sn2)=O)C(O)C1 C=C=CC(C)C(=O)N1CCC(CC(=O)N(CC(C)CC)C)C1 N1(C(c2cc(CC)nnc2C)=O)CC(C2CN(C(C3(C(C)(F)F)CC3)=O)C2)C1 CC(C)C(C(=O)NCC1CC1CNC(=O)CSC(C)(C)C)C(F)(F)F C(CNC(=O)COCC1CCOC1)(CCNC(=O)Cc1nonc1C)OC C1(N(C)C)CN(C(C2CC(NC(=O)CCC(N)=O)C2(C)C)=O)CC1O C1(COC)(CNC(=O)C(C)(O)C2CC2)CCCN1C(c1cc(C(C)C)n(C)n1)=O c1(C(=O)NCCN(C(=O)Nc2cc(CC3CC3)[nH]n2)C2CC2)c[nH]nc1F c1(CC(N2CCN(C(c3cccc(=O)n3O)=O)CC2)=O)ccc(Cl)cc1[N+](=O)[O-] C(CC1=CCN(C(=O)Cn2ncn(C)c2=O)CC1)NC(CN(C)S(N)(=O)=O)=O C(=O)(CC(C)CCC(=O)NC1CCC1NC(=O)CCCc1nc(C)cs1)OC C=CC1(C(=O)NCCCCCNC(=O)Cc2cccn2C)CCC1 Cc1cc(C(=O)NCC(C)CNC(=O)CC2CCCC2O)ns1 C1(NC(CS(N)(=O)=O)=O)CC2CC(NC(c3csc4nnsc34)=O)C1C2 c1(CN2CCC(C(=O)Nc3n(C)nc(O)c3)C(O)C2)c(F)ccc(Cl)c1Br c1(C(CNC(C2CC2Cl)=O)NC(=O)CCCCN2CCCC2)cccc(Cl)c1 C(=O)(C(CCC1CCC1)NC(=O)C=CC(F)(F)F)Nc1cn(CCOC)nc1 C(=O)(CCC(CC)NC(c1cnccc1OC)=O)N(C1CCOC1)CC#C N1(CCC#C)CC2CCN(C(c3csc(C(C)C)n3)=O)C2C1 C(=O)(C#CC1(C)CCCO1)NC(CN1CCN(C(CC(CCC)C)=O)CC1)(C)C C1(NC(C(C)CN2CCOCC2)=O)CC(=O)N(C)C1=O N1(C(c2c(C)ccc(O)c2)=O)CCC2CC2(NC(N2CC3CCC(C2)O3)=O)CC1 CC(C)CC(O)C(=O)N1CCN(C(c2ccc(-c3nc[nH]n3)cc2)=O)C(CO)C1 C(=O)(C(C)(C(F)F)c1ccccc1)NCC(C)(C)NC(c1n(C(C)C)cnc1)=O c1(C(=O)NC(C2CCOCC2)CCc2nc(C)[nH]n2)cc2c(cn1)NC(=O)CO2 CC1CCN(C(c2cnccn2)=O)CCN1C(C1CC2(C1)CC(O)C2)=O c1(CNC(CN(CCOC)C(c2ccc(C)nn2)=O)=O)ccncc1Cl c1(CC(=O)NC(C2CCN(C(c3cc(CO)[nH]n3)=O)C2)C)cccc(S(C)(=O)=O)c1 C1(C(=O)NC2C=CC(C(=O)NC)C2)CN(C(=O)CCCCN(C)C)CC12CCC2 CC1(C(=O)NCC2(CNC(c3cc(C#N)no3)=O)CC23CCC3)CCOCC1 CC1CCN(C(c2ccc(C#N)s2)=O)C1c1cccc(F)c1 N1(C(CC(CC)(F)F)=O)CCC2CCN(C(C3CC(OC(F)F)(OC)C3)=O)CC2C1 N1(C(c2c(C)nns2)=O)CCC2C(NC(=O)CSCCN(C)C)C2C1 C(=O)(C=C1SCC(=O)N1C)N1CC(CC)C(NC(=O)Cc2ccsc2)CC1 CC1C(NC(c2cc(Cl)ccc2Cl)=O)CC2CCC1N2C(C1(CO)COC1)=O c1(CC(N2CC(NC(C3CC(=O)N3)=O)C(C3CC3)C2)=O)cccc2c1OCCO2 CON1CCC(C(=O)NCCN(C)C(c2nocc2CC(C)C)=O)CC1 N1(C(Cc2n(C)cnc2)=O)CC(C(=O)NC(c2cscn2)CO)C(F)(F)C1 c1(C(C(=O)NC(C)(C)C)N(C)CC2(C)CCCO2)cc2c(cc1C)OCO2 C(=O)(CCCC(F)(F)C(F)(F)F)N1CCCC(CNC(C2C(C)CCO2)=O)C1 C(=O)(C(O)CC(N)=O)NCCC1N(C(c2c(OC)cccc2)=O)CCOC1 c1(CC)cccc2ccc(C(N3CC(O)CC3(C)C)C(=O)NC3CC3)nc12 S(=O)(=O)(c1cccc(CC(=O)NCc2nc3c(s2)COCC3)c1)N(C)C C1(C(=O)NCC(CN(C(Cc2ccc(C(C)=O)cc2)=O)C)O)CC(=O)NC(=O)C1 C12(CCCN1C(C1(C=C)CCC1)=O)C(=O)NOC2.C1(C(=O)OC)CCCS1 n1(CC)ncnc1CCC(c1nnnn1C1(C)CC1)C1CC=CCC1.NC CC(C)(CO)C(=O)NCCC(C)(C)NC(=O)Cc1sc(S)nc1-c1cccs1 N12CCC(C(O)C1)C2=O.C(=O)(CCCCC)NC1(C(=O)OC(C)(C)C)CC1(C)C c1(C(=O)NCC2(C)CCCN(C(C(CC)F)=O)C2)cc2c(s1)CC(C)(C)C2 N1(C(C)C)CCCC1CC(=O)NCC(C1CC1)NC(=O)CC(F)F c1(C(N2CCC(N(C(Cc3c(C)con3)=O)C)C(C)C2)=O)ccc2cncn2c1 c1(C(N2CC3C(NC(c4cccc(=O)n4O)=O)C3C2)=O)nccc2occc12 N1(C(C(C)Cn2ccnc2)=O)CC2=C(C1)CN(C(=O)C(N1CCOCC1=O)C)C2 c1(OC)cnc(F)c(C(N2CC(C)(C)CC2CNC(c2cncc(F)c2)=O)=O)c1 c1(C(=O)NCCN(CCCN(C)C)C(=O)Cc2cccnc2)onc2c1CCCC2 Cc1c(F)ccc(Cl)c1C(N1CC2OCC(NC(C3CC3F)=O)C2C1)=O c12ccc-1nn2.Cn1nccc1C(O)CNC(=O)CSC1(F)COC1 N1(C(C(N2CCN(C(C)CO)CC2)=O)=O)CCn2cccc2C1C c1(C(=O)NC2C(CNC(C3C(=C)CC3)=O)C2)cnc2c(F)cc(C)cc2c1 c1(C(=O)OC)nccc2c1CCCN2C(=O)Cc1coc2ccccc12 c1(C(=O)NC2CC(C)(NC(CCOC)=O)C2)cnc(O)nc1O c1(CC)cc(CN2CC(C3C(=O)N3)C2)ncn1.C(=O)(CCc1nccs1)NC C1(C(N(CC)OC)=O)CN(C(C2CC(=O)CO2)=O)CC12CCC2 C1(NC(Cc2cc(C)[nH]n2)=O)CCC(CNC(C2CCOC2C(C)C)=O)CC1 CC1CCCC1(C)NC(C1CCC(NC(=O)C(C)NC=O)CC1)=O C1(C(N2C(CCNC(c3ccno3)=O)CSCC2)=O)Cc2nccn2C1 c1(CC(=O)NCC2C(C(=O)NCC(=O)OCC)C2)cc(F)cc(F)c1Br Cc1ccc(C2CC2C(=O)NCCCN(C)C(C2CCO2)=O)cc1C N1(C(c2n[nH]c(C3CC3)c2Cl)=O)CCCN(C(C2C3CCC(=O)C23)=O)CC1 c1(C(=O)NC2C(CNC(=O)CCc3cnn[nH]3)CCCC2)cc2cscc2s1 c1(C(=O)NCC2(CNC(C3(C)C(CC)CCC3)=O)CCC2)cncc2c1CCC2 C=CCC(C(=O)N1CCC1CSC)C(C)C.c12cc(nc(O)c1)CNC2=O c1(OC)ccc(COC(=O)CC(C(=O)O)N2CCOCC2)cc1C#N CC#CCCCCNC(=O)C(C)N(C(c1cc(CCC)on1)=O)C1CC1 N12CCCC(C)(CC1)OCC2=O.C#Cc1cnn(CC(=O)NC2CC(OC)C2)c1 C1(NC(CC2C(C)(C)C2)=O)CCOC12CCN(C(c1ccc(F)c(Cl)n1)=O)CC2 C1(CCC)CN(C(c2c(C(F)(F)F)ncn2O)=O)CCN1C(C1CC12CC2)=O C12(C(=O)N(C3CCC3)CCO)CCCN(C(=O)CCN3CCCCCC3=O)CC1C2 c1(CC)cc(C(=O)N(C2CC(NC(c3nccc(Cl)c3F)=O)C2)C)cn(C)c1=O C12(CNC(=O)CC3CCCC(=O)N3)CC(CO1)N(C(=O)CCCc1ccsc1)C2 Cc1ccc(Cl)c(C(=O)NCC#CCNC(=O)CC2CCCC2S(C)(=O)=O)c1O c1(SC(C(=O)NC2(CCO)CN(C(CC(C)(C)OC)=O)C2)C)ccc(F)c(F)c1 N1(C(CSC)=O)CC(C(=O)OC)C2CC12.c1(SCC)cc(C(F)(F)F)oc1C c1(CNC(CC(CCC)CC)=O)nn(C)c2c1CN(C(=O)CNS(N)(=O)=O)CC2 C1(NC(Cc2ccc(OC)c(F)c2)=O)CN(C(C2CC23CC3)=O)C2(CCCC2)C1 c1(C(=O)NCC2N(C(C(CCC)CC)=O)CC=C2)ccc(F)c2c1OCC2 C1(CC)(CC)CC(NC(C2CC2(C)C)=O)CN1C(c1cc(Cl)ccc1N)=O N1(C(C(N(C)C(c2nnc(S)n2C)=O)C2CC2)=O)CCC(F)(F)C(O)C1 C(=O)(C1=CCc2ccccc21)NCCCCCN(C)C(c1cncnc1)=O c1(CC(N2C(N(C(=O)C(C)SC)CC(=C)C)CCC2)=O)cc(F)ccc1O c1(OCCC)cccc(CCC(C)NC(c2ocnc2-c2ccccc2)=O)c1 N1(C(C=CCC2(NC(c3c(C)c(F)ccc3)=O)CCC2)=O)Cc2cccc(F)c2C1 C1(C(=O)NC2CC(N(C(C(C)c3cc[nH]n3)=O)C)C2)CNC(=O)C(C)(C)C1 C(C(C)C(=O)NCCCN(C(C12CC(N)C1C2)=O)C1CC1)OCC c1(C(=O)NCC(C2CC2)NC(c2cn(C(C)C)nc2)=O)cncnc1C(C)(C)C c1(C(=O)NC2(CF)CCN(C(C3(C#N)CC34CCC4)=O)C2)cccc2c1CCO2 CC(C)C(CC(=O)NC1(CCO)CCC1)NC(C1CC(F)C(=O)N1)=O C(=O)(CC(CC)OC)NCC(N(C(c1cnc(CC)s1)=O)C)C1CC1 N1(C(COCC(=C)C)=O)CC(F)CC1CNC(c1csc(-c2cnc[nH]2)n1)=O N1(C(c2ccc(N)cn2)=O)CCC2CCN(C(c3cc4n(c3)CCOC4)=O)C2C1 C(=O)(C1CCCc2sc(=N)[nH]c21)NCCOCCCN(C(=O)C(O)CC(N)=O)C S(=O)(=O)(c1ccc2c(c1)CC(C(=O)NC1CC1)O2)N1C(S(C)(=O)=O)CCOCC1 C1(NC(CCC2N(C)CCC2)=O)CCN(C(=O)CN=S(C)(C)=O)CC1F N1(CC(=O)N(c2cnc3n2CCC3)CCN2CCCC2)CCSC2COCCC12 C(C)(C)(CCC(=O)NC1CC1CC(C)C)OC.C12CC1CNC2=O Cc1cc(C(=O)NCCC(O)CNC(c2ccns2)=O)cc([N+](=O)[O-])c1O C1(NC(C(COC)OC)=O)CCCC(N(C(=O)COC2(NC(=O)CSC)CC2)C)C1 c1(C(=O)NC(C(=O)NCC(=C)F)Cn2cccn2)ccc(CO)cc1F N1(C(c2cc(OC)ns2)=O)CCN(C(=O)C(OC)OC)C(c2nccn2C)C1 C1(C(N2CC3(CC(NC(COCC(=O)OC)=O)C3)C2)=O)CC2CC(O)CC(C1)C2 c1(C(C)C)cccnc1NC(c1ccc(Nc2cc(C(F)(F)F)ncn2)nc1)=O C1(CC(N2CCCCC(CO)C2)=O)C2CCCC2N1C(c1coc(C(F)F)n1)=O Cc1cc(NC2(CNC(=O)C(C)CF)CCCC2)cc(C#N)c1[N+](=O)[O-] N1(CC(=O)NCC(COC(=N)O)CO)CC(=O)NC1=O.C1(C(=O)N)(CO)CCCC1 C1(N(CCOC)CCn2cccn2)CCS(=O)(=O)CN1 N1(C(C(CC)(C)C)=O)CCC2(CC1)CC2c1cn(CCC2(C(C)(F)F)CC2)nn1 N1(C(C(C2CCOCC2)OCC)=O)CCC12CN(C(=O)C=Cc1cnc[nH]1)C2 C1(O)(CN(C(=O)C(=O)NCC(F)(F)F)C)CCCN(C(=O)CC2C=CCCC2)C1 N1(C(Cn2[nH]c(=N)c(Br)c2)=O)CCCC2(NC(=O)CCC(F)F)CC2C1 Cc1cc(CC(=O)N(C(CNC(=O)CCOCC2CCC2)C2CC2)C)cc(F)c1 C(C(CC1CC1)CO)NC(CN(C(=O)Cc1ccnn1C)CCC)=O C(N=c1[nH]c(=NCCOC2CC2)[nH]c2c1SCC2)CS(C)(=O)=O.C1(C)CCCCO1 CCCCC(CC)CC(=O)NC1CN(Cc2sccc2-c2ccccc2)CC1C S(=O)(=O)(c1cccc(NC(=O)CN2CCC(C3CC3)C2)c1)NCC c1(C(N(CCNC(c2cc(C)c[nH]2)=O)CC)=O)cc2ccccc2cc1C C12(NC(c3c(C)coc3)=O)CCOCC1CN(C(C1(C#N)CC=CC1)=O)C2 CC(CCC(=O)NCCCOCCO)NC(=O)Cn1nnc(=O)[nH]1 N1(C(C2CN(CC)C(=O)C2)=O)CCCC2C1CCN2C(c1ccncc1)=O c1(C(=O)NCC2N(C(c3c(O)ncc(CC)c3)=O)CC2)cccc2c1CC(=O)N2 Cc1cccc2c1CCCC2N=c1[nH]c(=NCCCSC(F)F)[nH]c2ncn(C)c12 C1(C(c2nnnn2CCCF)NCc2n(CC)ccc2)CC(C)(C)OC(C)(C)C1 O=C(CCCCCCCC1CC1)NCC(C1CCC1)NC(C1CC2CCC1O2)=O C(CC(C(F)(F)F)N1CCOCC1)NC(c1cccc(-c2ccc(O)nn2)c1)=O c1(COC)nn[nH]c1C(=O)NC(CNC(C1CC1c1csc(C(C)=O)n1)=O)CC c1(C(N2CC(OC)C(NC(=O)C=CC3CCCC3)C2)=O)c(C)ccnc1C N(C(=NCCC1CCN(C)C1)NCC(c1ccc(F)cc1)(C)C)C(COC)OC C(=O)(C1=NOC(C2(C)CC2)C1)NC1CC(NC(CN(C)CCO)=O)C1 CCCC(O)C(CO)NC(C1CCCN(C(c2ncccc2F)=O)C1)=O Cc1nc(N2CC(NC(C3CC4CC4C3)=O)CC2C)c2c(C)c(C)sc2n1 N1(C(CC2(C)CC2F)=O)CC(C2CN(C(=O)C(F)(F)Oc3ccccc3F)C2)C1 CC1(C)CC(NC(c2ccc(F)cc2)Cn2cncn2)CS1 N1(C(C(C)NC(=O)OC)=O)CC(C)(NC(=O)C=CC2CCOC2)C1 C(c1cc(Cl)ccc1OC)=CC(=O)NCCC(CCNC(C=C(COC)C)=O)C C1(NC(c2c(NC)cncc2)=O)CC2CC(NC(=O)C(C3CC3)SC)CC12 C1(NC(C2N(C(CC3ON=C(C)C3)=O)CCC2)=O)CCOCC1CN(C)C c1(CC(=O)N(C(C)C(=O)N(C)C(c2ccco2)C)CC)cc(C)on1 N1(C(C(CCC)F)=O)C2CCC1CC(C(=O)Nc1c[nH]c3cccnc13)C2 CC1CON(Cc2cccc(C(F)(F)F)c2)C1 c1(CC(C(=O)NCCC(=C)CNC(C2(n3cncn3)CC2)=O)C)cccc(F)c1 N1(C(C2(CCCC)CC2)=O)CC2ON=C(CNC(=O)Cn3ccc(C)n3)C2C1 C(=O)(C(C)(C)CC(C)(C)C)N1CCC(NC(COc2ccc(C)cc2C)=O)CC1 C1(OCCC)CCCN(C(C2C=CCCN2C(=O)CCc2cncnc2)=O)C1 c1(C(N2CC(C)(NC(c3onc(CC)n3)=O)C2)=O)cc(C#N)c[nH]1 C1(CNC(C(C=C=C)C)=O)CN(C(C2CCC3(CC2)CC3)=O)CCC12CCC2 C(CO)(CCCCNC(=O)CCC1CCC(O)CC1)NC(CCC)=O c1(C(=O)NC2CCN(C(CC3CC(=O)NC3=O)=O)C2)cnc2c(c1)CCCCC2 C1(C(N2CCC(CNC(C(N3CCC(O)CC3)C)=O)C2)=O)CCC2(CCC2)CC1 C1(CCC)CN(C(C23CCC2C3)=O)CCN1C(=O)CCn1ccnc1 c1(C(N2CC3N(c4nc(CC)cc(CC)n4)C3C2)=O)ccc([N+](=O)[O-])cc1C C1(C(=O)NCC(OC)OC)CN(C(c2ncccn2)=O)CCS(=O)(=O)C1 N1(C(c2n(C=C)nnc2)=O)CCOCC1(C)C CC1=C(C)CN(C(=O)CN2CC(N(C)C(C34CCCC3(C(N)=O)C4)=O)C2)CC1 c1(C2(CN3CCC(C)(c4onc(C)n4)C3)CC2)ccc(Cl)c(Cl)c1 CC(C)(C)C#CCCNC(C1CC(O)CN1C(=O)Cc1cnns1)=O C1(NC(Cc2n(C)ncc2)=O)CCC(F)(CNC(=O)CNC(c2cccs2)=O)C1 c1(C(=O)OCC=CC)cc2c(cnn2C)nc1C Cc1cnc(N2CC(=C(F)CNC(=O)CCc3nccs3)C2)nc1 c1(CNC(=O)NC2CCN(CC(=O)OCC)CC2)cnc(C#N)c(Cl)c1 n1(C(C)C)ncc(C(=O)NC2CC(N(C(=O)COCC3CCCCO3)C)C2)c1Cl c1(C(=O)NC(C)C(C)NC(C2CCCC2)=O)ccnc2c(C(N)=O)cnn12 c1(CNCC23C(CN(C(c4cc(C)c(F)cn4)=O)C2)C3)ccc(F)c(C#N)c1 c1(C(N2CCC(CNC(CCCNC(=O)OC)=O)C2)=O)nnccc1C c1(C(=O)NC(C(C)C)C(=O)NC2CC=CC2)ccc(=O)n(C)c1 c1(C(CNC(C2C3CCC23)=O)NC(CC2(OC)CCC2)=O)ccc(C)cc1 C(=O)(CC(=O)NCC(C)(C)OCC(=O)NCCCC1CCOC1)N(C)C N1(C(C2CC(OC)C2)=O)CCC2(CNC(C3(NC(C)C)CCC3)=O)CCCC12 c1(CNCCO)ccnc(Cl)c1.C(=O)(C(F)(F)N1CC(N)C1)C(c1ccccc1)=O c1(C(N2CCC3C(NC(CCCC#C)=O)C3C2)=O)ccc2cc[nH]c2c1 C1(C(=O)NCCC2(NC(C3CC(CC(=O)OC)C3)=O)CC2)CCCOCC1 N1(Cc2nc(C)on2)CCC(C(=O)N2CC(CO)C2)c2cc(O)ccc21 N1(C(CCC(C)N(C(C2CC(C)(C)CN2C)=O)C2CC2)=O)CCC12CCSCC2 CCC(C)CC(C(=O)NCC12CCC(CC1O)C2)NC(=O)CCCNC(C)(C)C CCCC(C(=O)OCC)NC(C1CCC=CO1)c1nnnn1CC1C(C)(C)C1(F)F CCCCC(CNC(=O)C(c1cnn(C)c1)O)NC(=O)C(COC)COC C(CCCCC(=O)NC1CCCN(C(=O)COCCCF)C1)OC C(CCCCCC1CC1)NC(C1(NC(C2N(CCC)CCC2)=O)CC1(C)C)=O CC(C(C)(O)C(=O)N1CCC(NC(=O)C(C)(C)C2CCCC2)C1)c1ccccc1 c1(C(=O)NC2C(NC(c3cccc(Br)c3F)=O)CC2)cc(Cl)ccc1F N1(C(CC(CCC)(C)C)=O)CC2CC(C1)CN(C(C1(C#N)CC13CCCC3)=O)C2 N1(C(CC2(C)CCN(C(C(C=CC)O)=O)C2)=O)CCc2nc[nH]c2C1 N1(C(CNC(c2cnc(C)n2C)=O)=O)C2CCC1CC(F)C2.C1C(=O)N1 C(=O)(C1=CCCCCC1)NC(CN(c1cc(OC)nc(OC)n1)C)C c1(C(N2CCCC(N3CCCCC3)C2)C(=O)NCCC)ccc2c(c1)CCCO2 Cc1ccc(C(N2CC(C(=O)Nc3cn(C)nc3C(N)=O)C3(CC3)C2)=O)cc1F O=C(C1=CCCCC1)NC1(C(N2CCC(C3CCCO3)C2)=O)CC1 c12cc(c[nH]1)SC1CN(C1)C2=O.C1(C(=O)OC)CSCN1C(C1CCCCC1)=O CC(C)CCC(C(=O)NCC1CCC(=O)NC1C)NC(=O)C(C)CO N1(C(Cc2cc(C)cc(F)c2)=O)CCC2CCC(C1)N2C(C1CCC1)=O c1(SC)cc(C(=O)NCCCCC(C)NC(C2(CF)CC(F)(F)C2)=O)n(C)n1 CC1CN(C(c2cc(CNC(=O)CCCn3cncn3)on2)=O)CCN(C)C1 C(=O)(C(COC)COC)NCCC1(C(=O)NC(C#C)CC)CCCC1 C1(OC)CCCC(C(=O)N(C)CCN2CCN(C(=O)CC(C)O)CC2)C1 c1(OC)ccc(CC(=O)NC2CCN(C(=O)CN3CCC3C)C23CC3)c(Cl)c1 c1(C(=O)NCC(CNC(CC(C=C)C)=O)F)ccc(OC)c2occc12 c1(CNC(C2N(C(Cc3ccn(C)c3)=O)CC(F)C2)=O)nnc2n1CCC2 c1(C(N(CCCNC(C2(C)CCOC(C)C2)=O)CC)=O)ccc2cnc(C)n2c1 C1(NC(C(CC#C)C)=O)(CNC(=O)CC2OCCCO2)CCC(C)(C)CC1 C(CCCC(C)NC(C1(c2ccc(O)nc2)CCC1)=O)NC(C(O)SCC)=O C1(Cn2cc(CNC(CNC(C(COC)C)=O)=O)nn2)Cc2ccccc2O1 C1(CC)CC2(C1)CN(C1c3[nH]c(CC)cc3C(=O)NC1=O)C2.C(CCF)C(=O)OC O=C1NCCC1CNC(=O)CC1CCCN1C(c1c[nH]nc1Cl)=O C1(CN(C(C(C2CCCCC2)OC)=O)C)CN(C(=O)C(COC)N(C)C)CCO1 c1(OC)ccc(CNC(C2CC2C(=O)Nc2sccc2C(C)=O)=O)c(Cl)n1 N1(C(C(c2ccccc2Cl)OC)=O)CC(NC(=O)C=C(C)C2CC2)C2(CCC2)C1 c1(C(N2CC3C(NC(C(=Cc4ccco4)C)=O)(C3)C2)=O)cccc2[nH]cc(Cl)c12 S(=O)(=O)(c1cccc(C#N)c1)NCC1(C)CN(C(c2c(Cl)cc(F)c(F)c2F)=O)C1 N1(C(CC(C)(C)C)=O)CCC(F)C(NC(=O)C(=Cc2cccc(F)c2)F)C1 CCS(=O)(=O)CC(=O)N1CCC(CCCCNC(C2CCNC2=O)=O)CC1 c1(OCC(=O)NCC2(C)CCN(C(C(CCC)OC)=O)C2)cc(C)c(Cl)c(C)c1 c1(C(=O)NCC2(O)CCN(C(CCCCN(C)C)=O)C2)nn(C)c2ccccc12 c1(SC)onc(C)c1CC(=O)NCC(C)NC(C1CC1C)=O C1(C2CC2)(C(=O)NCCN(CCOC)C)CN(C(c2ccc(SC)o2)=O)C1 C(=O)(C(C(C)(C)C)n1ccnn1)N1CCC(N(C)C(c2cn(CCF)nn2)=O)C1 Cc1nccc(CCC(=O)NC2CC(NC(C3(c4cccc(Cl)n4)CC3)=O)C2)n1 c1(C(=O)NC2C(CCC)CN(C(=O)C=C(C)C(C)C)C2)cncc2[nH]ccc12 C(=O)(C(F)(F)C(O)C(C)C)NCCC1(OC)CN(C(C(CCOC)C)=O)C1 C1(OC)CC(NC(c2snnc2C)=O)CN(C(c2c(C)[nH]c(C)c2C)=O)C1 Cc1cn2nc(C(N3CC(NC(=O)CCC4(C)CC4)C4(CC4)C3)=O)cc2c(=O)[nH]1 c1(C(=O)NCC(CO)NC(C(C)P(C)(C)=O)=O)cccc2c1COCC2 C1(C(=O)NCc2nccs2)CCN(C(=O)CC23CCCC2C3)CCO1 N1(C(c2ccc(COC(C)C)nc2)=O)CC2CCCC2(NC(=O)CCC(C)(C)F)C1 N1(CC)CCOCC1CC(=O)NC1CN(C(C2(n3cccn3)CC2)=O)C1 N12CCOCC1C1C(=C)C1C2=O.n1(CCCNC(=O)C2CC2)cc(C)cn1 N1(C(c2cc(CNC(c3n(CCC)ccc3)=O)[nH]n2)=O)CC(C)(C)C1CC C1(OC)CN(C(=O)OC(C)(C)C)C2(CCCC2)C1.C12CC(C)N(C(C)C1)C2=O N1(C(CC(CC)C)=O)CCCC(NC(=O)CN2CSCC2=O)C1C C(=O)(C(C)CC(C)(F)F)N(C1CCN(C(c2nccc(C)c2N)=O)CC1)C c1(CN(C(C)C)C(=O)NC(C)CN(c2ccncc2)C)ccccn1 CC(N=[N+]=[N-])C(=O)NCC(CC(=O)N1CCC=C(F)C1)C1CCC1 c1(C(=O)NC(CC)CN(C(=O)C(C)Sc2ccccn2)C)c(C)cc(C)oc1=O C(=O)(C1=NNC(=O)C1)NCC(C)N(C)C(C1CCOC1)=O n1(C(=O)OC)nnc(NC(=O)C(=O)Nc2ccc(CC(F)(F)F)cc2)c1N N1(C(CC=CC=C)=O)CC2(CCOCC2)CC1CNC(=O)CCCc1cccs1 N1(C(c2ncc(OC)nc2)=O)CCC(C(N2CC(F)(CO)C2)=O)C(C)C1 c1(CC)noc(C)c1C(=O)NCCCCC(C)NC(C1COC(=O)N1C)=O c1(OCC(=O)N(CCNC(C2(O)COC2)=O)CC)ccccc1[N+](=O)[O-] N1(C(c2c(CC)nncc2)=O)C2COCC1CC(NC(C1CCCC1SC)=O)C2 N1(C(C2(CCCC)CCC2)=O)CCC(NC(=O)CCC2CCCN2C)C(C)C1 N1(C(C(C2CC2)SC)=O)CC(CNC(=O)Cc2cc(C)cs2)C(F)(CO)C1 c1(-c2nnc(NC(N3CCC(CC(=O)NC)CC3)=O)o2)c(F)cc(F)c(Br)c1F C1(C(=O)NCC2(NC(c3ccc(C)cc3F)=O)CC(OC)C2)CC2(C1)CC(C)C2 C(N=c1[nH]c(=N)[nH]c(=NC2CCNC3(CCC3)C2)[nH]1)C12OCCC(C)(C1)C2 C=C(C)C(O)CC(=O)NC(C1CCCN(C(=O)C(C)(C)CCSC)C1)C C1(C(=O)NC2CC(C(=O)NCC(C)C(F)F)C2)CC(=O)C12CCC2 c1(C(=O)NC(C2N(C(c3ccc(CC)s3)=O)CCC2)C)cc2[nH]ccc2s1 C(=O)(C(O)CC(C)C)N(CCC)CCNC(=O)C(CC1(C)CC1)c1ccccc1 CC(C)CC(COCN1CN1C(=O)C(C)(C)Sc1ccc(F)cc1)N=c1nnn(C)[nH]1 c1(OC)ccc(F)c(C(N2CCC(NC(c3sccc3OC)=O)C(F)C2)=O)c1 CCS(=O)CC(=O)NC1CCCC1NC(C1C=CCCN1C(=O)OC(C)(C)C)=O C1(NC(C=CC(CC)C)=O)CCN(C(c2cccc(Cl)c2N)=O)C1(C)C N1(C(Cc2n[nH]c(=NC)s2)=O)CCN(C)CC1CNC(=O)COC(C)(C)C C1(CC=C)(C(=O)NC2(c3cn(CCO)nn3)CCCOC2)CCCN1C(C)=O N(C1c2ccccc2CCC1N(C)C)C(N1CCC2(C(C#N)C2)CC1)=O N1(C(C(C(C)C)SC)=O)CCOC2(CCN(C(c3ncccc3F)=O)C2)C1 c1(C(=O)NCC2C3CN(C(CC(CC)C4CC4)=O)C2C3)cccc2nc[nH]c12 N1(C(C(C(C)C)SCC)=O)CCC(C2(O)CN(C(C3CC3(F)F)=O)C2)CC1 Cc1ccc(C(C)C(=O)NCC2CCCC2NC(=O)CCn2ccnn2)s1 N1(C(c2ccc(CC)s2)=O)CC2CCCC2(C(=O)NC2CNC(=O)C(C)(C)C2)C1 C12(CC)CCCN1C(=O)C1(CCCC1)C(=O)c1nnc(o1)CNC2.OC C1(NC(=O)CCc2ccncc2Br)CCN(C(=O)C=Cc2cnc[nH]2)CC1O CCCCC(C(=O)NCCc1ncccc1C)NC(=O)CCP(C)(C)=O C(=O)(C1Cc2ccc(F)cc21)NCC(C(C)C)NC(=O)CNC=O C(c1c(C)coc1C)=CC(=O)NCCCCCCNC(c1c(CC)ncs1)=O c1(CC(=O)NC(CC2CC2)(C2CC2)OC)cn(C)nc1C(F)F c1(OC)ccc(-c2noc(C(C(=O)NC3CCC3)N(C3CCC3)CC)n2)cc1Br c1(C(N(C(C)CNC(=O)C(N2C(=O)CCC2=O)C)C)=O)cccc2c1OCCO2 CC1(C)CN(C(C2(C#N)CCC2)=O)CC(CNC(=O)CN2C(=O)CNC2=O)O1 c1(C(N(C(CC(=O)OCC)c2cnn(C)c2)CCC)C)ccncc1 CCC(CC(=O)NCc1nccs1)NC(c1cn(C)nc1CC)=O N1(C(CC(C)(C)n2cc(-c3c(=O)cc(C)[nH]c3)nn2)=O)CCc2ccc(C#N)cc2C1 c1(NC(=O)Cc2ccc(NC(c3n[nH]cc3[N+](=O)[O-])=O)cn2)ncc(F)cc1Br C1(NC(C=C(C)C)=O)CCC(C)(CNC(=O)C(O)CN2CCCC2)CC1 CCC(C)(C)CC(=O)N1CCCCCC1C(=O)NC1CC(N(C)C)C1 CC1CN(C(=O)C(C2CCOCC2)=O)CCC1C(=O)NC1CC2CCCC2C1 N1(C(C2CCC(OC)CC2)=O)CC2CCN(C(c3cccc4nccn34)=O)C2C1 C1(C(N2CC(COC)(CNC(c3cc(C(C)C)no3)=O)C2)=O)CCOC1(C)C C1(C(=O)OC)(OC)CCCN(C(=O)C(c2cccc(Cl)c2)NC(C)=O)C1 C(=O)(C#CC1CCOCC1)N1CC(CCNC(C2CCC(F)CC2)=O)OCC1 c1(NC(C2OCCN(C(c3n(CC)ccc3)=O)C2)=O)ccc2c(c1)CCO2 c1(C(=O)NC2(CCNC(CC3CN(C)C3)=O)CC2)cnnc(-c2ccccc2)c1 C=CC(C)(CC)C(=O)NCC12CC(C1)C(NC(=O)CC1(C)CCOCC1)CO2 C1(NC(C2C(c3n(C)ccn3)C2)=O)CN(C(=O)CS(C)(=O)=O)CCC1O C1(C(N(C2CN(C(=O)CC3=NN(C)C(=O)C3)C2)C)=O)CCc2nc(=N)[nH]cc2C1 c1(C(N2C(CN(C(CCOCCOC)=O)C)COCC2)=O)cc([N+](=O)[O-])nn1C CC1CN(C(c2cc(C(C)(C)C)no2)=O)CCC1CNC(=O)COCC1CCOC1 C1(NC(C2CC(OC)C2)=O)(CNC(c2csc(C)c2)=O)CCCCC1C Nc1cnc(Br)c(C(=O)NCCNC(C2CCCS(=O)(=O)N2)=O)c1 CC1C(NC(c2cccc(-c3cccs3)n2)=O)CCCN1C(=O)CCCN(C)C c1(CC(=O)NC2(CNC(CSC)=O)CCCCC2C)csc2sc(C)cc12 C1(CNC(C=CC(=O)OCC)=O)CC(C)(C)CN1C(=O)CC1CC(C)C1 n1(CC(N2CCC(C(C)(C)NC(C3(F)CC=CC3)=O)C2)=O)ncc2ccccc12 C12(C(=O)NC(C(CCC)C)C)CCC(CC1)N(C(=O)Cc1cc(C)ns1)C2 C(=O)(CC(C)n1cc(Br)cn1)NCC(C)NC(CCN(C)CC)=O C1(CCC(=O)NCCC(C)(C)NC(C2COCCN2C)=O)CC2C=CC1C2 c12cccc(c1)-c1cnc(nc1)NC2.N1(S(C)(=O)=O)CCC(N2CCCC2)CC1 c1(OCC(=O)NCC(CC)NC(=O)C(C)(F)F)cccc([N+](=O)[O-])c1 Cc1ccc(CC(N2CCC(OCCNC(C3(Br)CC3)=O)CC2)=O)cn1 O=S(=O)(c1cccc(=NC2CCSCC2)[nH]1)NCc1ccc(Br)cc1F c1(C(CC)(C)C)ccc(C(=O)NC2(CO)CN(C(=O)C(C)c3cccs3)C2)cc1 c1(CCCC)nc(C)c(CC(=O)NC2CN(C(C3CC(C)CO3)=O)CC2O)s1 C(=O)(CCCC(F)(F)CO)NC(CNC(C1N(C(C)=O)CCOC1)=O)CO C(=O)(C(O)C(F)(F)F)N1CC(CC(C(=O)NCCC2(C)CCOCC2)F)C1 c1(OC)c(NC(=O)C=C2CCN(Cc3c(F)cc(O)cc3F)CC2)cc(Cl)cc1Cl Cc1nc2cc(C(=O)NC(C)CN(C)C(C3(C)CCOC3)=O)[nH]c2s1 c1(C(N2C(CC(=O)Nc3nccc(Cl)c3Cl)CCC2)=O)c(Br)cncc1F Cc1ncn(O)c1C(=O)NCCCCCCN(C)C(c1c[nH]c(=O)cn1)=O c1(CC)c[nH]nc1C(=O)NC1CC(NC(C2CCC(C(=O)OC(C)(C)C)C2)=O)C1 CC1CCC(CO)(NC(=O)NC(C2CCCC2C2CC2)C2CC2)c2ccccc21 C(C(C)(C)C(F)(F)F)NC(CCOCCCN(C(=O)C(c1ccnn1C)C)C)=O S(=O)(=O)(c1ccc(NCC2CC2c2ccccc2)c(Cl)c1)NCc1c(C)cco1 C12(C(N(CC(C)OC)C)=O)CC(CO)(CN1C(=O)C(O)C(C)(C)C)C2 C1(NC(C2CN(C(CNC(=O)NC)=O)C2)=O)CCCC(C(N)=O)CC1 c1(C(N(CC(C)CNC(C2(CF)CCOCC2)=O)C)=O)cccc(F)c1F Cn1cc(C(=O)NC2(C3CCCN3C(=O)COC3CC=CC3)CC2)c(O)n1 C1(NC(C(C(C)C)SC)=O)CCN(C(C2CN3CCN2C(C)C3)=O)CC12CCC2 C1(CCC(=O)NCCC#CCC)CCCCN1C(c1cc(C)nn1C)=O N1(C(=O)NCCO)CCC(c2cccc(NC(=O)C(F)(F)F)c2)C12CC2 N1(C(c2cccc(CC#N)c2)=O)C2CCC(C2)C1C(N1CCCC(CO)C1)=O C1(CC)(NC(c2nnn3c2CCC3)=O)CCCN(C(=O)CCOC2CC2)C1 N1(c2snc(CC(C)C)n2)CCCC2(NC(=O)CC3CCC4CC4C3)CC2C1 N1(C(C(C)SCC)=O)CCCC(F)(C(=O)NCC2CCCSC2)C1 c1(OC)ccccc1C(=O)N(C(CC)C(=O)NCc1ccc(C2CC2)cc1)C C1(C(=O)NCC2C(C)CC2)CNC(=O)CN1C(c1ccncc1N)=O c1(C(=O)NCC2N(C(c3c(C)sc(C#N)c3)=O)CC2)c[nH]c2c(C)cccc12 N1(C(C(C)(C)c2cnsc2)=O)CC(NC(=O)COCC2CC2)CC(C)(C)C1 CC(C)C(O)CONC(C1C(C)CN1C(=O)CC(=O)N(C)C)=O CS(=O)c1ccccc1C(N1CCC2(NC(c3ncccc3F)=O)CCCC12)=O c1(CC)ccccc1CC(N1CCC(C(C)NC(c2ccc(CC)nc2)=O)C1)=O C1(NC(CCNC(=O)OCC)=O)COCCC1NC(C1CC1F)=O C1(NC(c2c(C)cc(Cl)cc2N)=O)CN(C(=O)Cc2nc[nH]n2)C2(CCOC2)C1 CCC(C(=O)N(N(CCn1ncc(CC(N2CC(C)C2)=O)c1)C)C1CC1)SC CCC(C)(C)C(O)C(=O)NCC1COC(C)(C)CN1C(C12CSC(C1)C2)=O c1(CNC2C(C(=O)Nc3c(OC)cc(O)cc3)CCC2)n[nH]c2ccc(Cl)cc12 C1(O)(C(C)CNC(c2cncnc2)=O)CCN(C(=O)CCCC2(C)N=N2)C1 N1(C(=O)Cc2ccc(Cl)cc2Cl)CCC2CN(c3cc4ncnn4cn3)CCC12 C(N=c1[nH]c(N2CC3CCC3(CO)C2)nc(=N)[nH]1)C1CCN(C(C=CC)=O)C1 C=C(Cl)C(C)(C)C(=O)NCC1CN(C)CCN1C(c1ccn(C(F)F)n1)=O c1(CC(=O)NC2CCCC(NC(c3c(CC)csc3)=O)C2)cc(F)cc(F)c1 C1(C(=O)NCC2(NC(C3C(C)(C)CC3)=O)CCC2)Cc2cc(F)ccc2C(=O)O1 C#CC1(O)CC(C(=O)NC2CCN(C(=O)C(C)n3cccn3)C2C)C1 c1(C(C(=O)NCCOCCCN(C(C2C(C=C)C2)=O)C)CC)c(C)noc1C C1(C(=O)NCCC(O)C2CCCC2)(CC)CCCN(C(C2CC(F)(F)C2)=O)C1 C1(CC)CC(CC(=O)NCCC(C)(C)CNC(=O)Cc2ccsc2)CCO1 C1(NC(CN2C(C)CCCC2)=O)CCC2CCN(C(=O)COc3ccsn3)C12 c1(SC)cccc(C(=O)N(CC(O)CN(C)C(c2ncccc2C(C)=O)=O)C)c1 CCCCC(CNC(C1(C)CCCOC1)=O)NC(=O)C(=O)Cc1cccs1 c1(NC(=O)CC2CCCN2C(c2cccc(F)c2)=O)cccc(C(F)(F)F)c1Cl c1(C(N(CCN(CCNC(CCC)=O)CC)C(C)C)=O)cc2c(Cl)cncc2s1 CC1CCC(C(N2CC(F)(CNC(C3(C4(C)OCCO4)CC3)=O)C2)=O)C1 c1(CC(=O)N(C(C)C)CCNC(=O)Cn2cncn2)c[nH]nc1O C=Cn1ncc(C(=O)NCC(O)CC(=O)N2CCC(C(C)C#N)C2)c1N C1(CCNC(COCC(C)C)=O)CN(C(C2(C)CC=CCC2)=O)CCS1(=O)=O N1(CCNC2CCOC2)CCC(NC(C2N(C(CSC)=O)CCC2)=O)CC1 c1(CNC(=NCC(C)C)NCC2(SC)CC2)ccc2c(c1)C(=O)NCC2 c1(C(N(CC(C)NC(CC(CC)C2CC2)=O)C)=O)nnn(CC2CC2)c1C c1(C(N2CC(CC3C(=O)NC(=O)N3)C2)=O)ccc2c(n1)CCCC2 N1(CC)CCCC1Cn1cc(C2CN(C)C2)nn1 N12CCCC1C1CCCN1C(=O)C2=O.c1(OC)ccc(CSC)c(C)c1 CC1CCN(C(=O)CC2(O)CCC2)C(C(=O)NC(C)Cc2nncn2C)C1 Cc1cc(CN2CC3C(C(=O)NCCCN4CCOCC4)C3C2)c2cc[nH]c2c1 c1(NC(CC(=O)NCCC2CCC(C)C2)C)cn(C)ccc1=O C(C(C(C)(C)C)NC(C1CN(C)C1)=O)NC(C1CC(CC)(CC)C1)=O c1(OC)ccc(-c2cnccc2NCCC(=O)NCCC(C)C)cc1F C1(C(C)C(N2CC=CCC2)=O)CCCN(C(=O)CC2COCC2(C)C)C1 C(=O)(CCCCC#N)NC(C1N(C(CCc2cnc(C)s2)=O)CCCC1)C N#Cc1cscc1C(=O)NC1(CNC(=O)CCOc2ccccc2Cl)CC1 C(=O)(C(CNC(=O)CCn1ccnc1)C(C)C)Nc1c(C)ncnc1 C1(C#N)(C(N2CCCC(CC(=O)N(C3CCC(C)(C)C3)C)C2)=O)CCCCC1 CC(CSC(F)(F)F)C(=O)NC1CCC1CNC(C1CC=CCC1)=O CCC(CC(=O)N1CCCC1C(=O)NCc1cc(OC)ncn1)C1CCC1 CC1(C(=O)NC(C2CCOC2)CNC(=O)C2=NNC(=O)C2)CCS(=O)(=O)CC1 c1(C(C(=O)NC(C)CCNC(=O)CN2CCCCC2)C)ccc(F)cc1 CCCCC(C)C(=O)N(CC(=O)Nc1cncc(F)c1)CC1CC1 c1(C(N(CCCN(C(CCCc2nc(C)sc2)=O)C)C)=O)nsc2ccccc12 C1(CNC(C(C(C)C)NC(C)=O)=O)CCC2(CCNCC2)CO1 Cc1cc(CNC(=O)CCN(C(C2COCC(C)O2)=O)C(C)C)oc1C C1(C(N2CCCC(CC=C)C2)=O)CCC2CCC1N2C(c1cn2c(n1)CCC2)=O Cc1oc(C)c(C(=O)NCC(C2CC2)NC(C2CCCN2C(N)=O)=O)c1C N1(C(C(CC)OC2CCCCC2)=O)CC(NC(=O)CCCCO)CC2(CCC2)C1 c1(C(=O)NC2(CO)CCOC2)ccc(Oc2ccccc2)c(Cl)c1 C1(CNC(C(CC)(C)O)=O)(CO)CCCN(C(c2ccc(C)cn2)=O)C1 C1(n2cccc2)(C(=O)NCC(C)NC(C2CC(CN(C)C)C2)=O)CCCC1 Cc1cc(N2CC(C)OC(C)C2)ncc1S(=O)(=O)N(C)Cc1ccc(Cl)cc1Cl C1(NC(c2scc(C)c2)=O)CN(C(C2COCCC2(F)F)=O)C2CCCC12 CC(C)(CCOC(c1ccc(Cl)c(CN2CCCCC2=O)c1)=O)C(F)(F)F c1(C(=O)NC2CC3CC(NC(C45CCC(C4)C5)=O)C2C3)cc2sccc2cn1 CC1CCCN(C(c2ncc(F)cn2)=O)C1CNC(=O)Cn1ccccc1=O C1(NC(c2nc(CCC)oc2)=O)CN(C(c2cn(C)cc2C)=O)CC(C)(C)C1 CC1CN(C(=O)Cn2cnnc2)CC(C)N(C(=O)CCn2ccnc2C(C)C)C1 CCC(C)CCCCC(=O)NC(CN(C(c1ccc(P(C)(C)=O)cn1)=O)CC)CC Cc1nn(CC(=O)NCC2CC(NC(C3SCCCS3)=O)C23CCC3)c(C)c1C N1(C(CSC)=O)CC(NC(c2cnc(O)cc2C)=O)CC(O)C1.c1(S)cccc(Cl)c1 Cn1c(CCOC(c2cc([N+](=O)[O-])c[nH]2)=O)nc2cc(Cl)ccc12 N1(C(CNC(CNC(C)=O)=O)=O)CCC(F)(F)C(CNC(C2CC23CCC3)=O)C1 C1(NC(C(COC)N(C)C)=O)CCCCC1CNC(=O)C(C)Sc1ncccn1 c1(C(N2CCC(C(=O)NCc3c(CC)c[nH]n3)(C(C)C)C2)=O)cnc2n1CCC2 c1(-c2cn(CC3N(C(=O)C=CC(F)(F)F)CC=C3)nn2)ccc2ccccc2c1 C=C(Br)CCC(=O)N1CC(N(C(=O)C(C(C)C)SCC)C)C(F)C1 c1(CC(N2CC(OCC)C(=O)C2)=O)c[nH]c2cc(Cl)ccc12.c1(=O)c(=O)[nH]1 N1(C(Cc2nccc(OCCC)n2)=O)CCC(NC(=O)C(CCO)NC)C1(C)C Cc1nc(C(=O)NC(C2CCN(C(=O)CCCCC3CC3)CC2)CO)c(C)o1 c1(C(=O)NCc2cc(NC(C3(COC)CCC3)=O)no2)nn(C)cc1C C1(C(N2CCC(CNC(C3CC(SC)C3)=O)C2)=O)CCCC(C)(C)C1 C(=O)(C1CC(=O)c2ccccc21)NCC(C(C)(C)C)NC(C(C)OC)=O c1(CC(N2C(CN(C(C=CC)=O)CC)CCCC2)=O)cc(F)c(F)cc1F c1(CCC(N2CCC(C(C)NC(CCOCCC)=O)C2)=O)ccc(N)nc1 N1(C(COCCCCC)=O)CCOCC(NC(=O)C(=O)NCCNC(C)=O)C1 C(=O)(C(C)(CC)CCCCCC(Cl)(Cl)CO)Nc1ccc(OC)c(Br)c1 c1(C(N2C(C(=O)NC(c3c(OC)cccc3)C)CCC2)=O)ncc(F)cc1C C1(C)(NC(C2(NC(C)=O)CC2)=O)CCN(C(=O)CC2CCOC(CF)C2)C1 N1(C(c2c(CC)occ2)=O)CCC2(CC1)CC(NC(C1CCCC(=O)N1C)=O)CO2 Cn1cc(Cl)cc1C(=O)NCCOC1CN(C(=O)C(=O)C2CCCC2)C1 C1(C(=O)NCC2=CCCOC2)(CC)CCCN(CCO)C1.C1(C)CC1 Cc1c(C(=O)N(C2CN(C(C34CC(C)(CCO3)C4)=O)C2)C)sc2ccc(Cl)cc12 c1(C(N(C2CCN(C(c3cncn3C3CC3)=O)C2)CCC)=O)cn(C)cc1C N1(C(c2ccc(OCCF)[nH]2)=O)CCC2CN(C(=O)C(F)(F)C3CC3)CCC2C1 C12(CNC(C3C(C)CCC3)=O)CCC(CN(C(c3cc([N+](=O)[O-])nn3C)=O)C1)C2 C1(C(N2CCOCC(NC(c3c(C)ocn3)=O)C2)=O)CCC(S(N)(=O)=O)CC1 N(C1=NCCN(C)C2(N1)CC2)C(CC)C.C(=O)(C(C)(C)C)NCCSC(F)(F)F c1(C(=O)NCC2OCCN(Cc3scc(C)n3)C2)cc2n[nH]cc2cc1Cl CC(C)C(C(=O)N(CC(C)(C)C#N)C)C(C)NC(=O)CCCn1cccc1 C(=O)(CC(C)(CN)C(F)(F)F)NCCNC(COCCC#C)=O C1(CNC(Cc2nc(C)oc2)=O)CCC(F)(NC(c2nn(C(F)F)cc2Cl)=O)C1 c1(OCC(=O)NC(CN(C(=O)C=C(Cl)Cl)CCCC)C)cccc(C(C)(C)C)c1 N1(C(=O)CC2(CNC(=O)OC(C)(C)C)CC2(F)F)CC(S(C)=O)C1 C(=O)(CCC(C)OC)N1CC(OCCNC(=O)NC)C1 CC(C)CC(CNC(=O)CC1CCCOC1)NC(=O)C(C)CO c1(CC(=O)NC2CCN(C(C3CC3F)=O)CC2)ccc(Cl)cn1 CC12CCC(C(=O)NCCCC3(C(=O)NOC(C)(C)C)CC(F)(F)C3)(CC1)CO2 CC1(C)C(CNC(=O)Cc2csc(Cl)c2)CCN1C(C1Cc2nncn2C1)=O c1(NC(CC)(CNC(=O)CC2CC3CC3C2)CC)ccc([N+](=O)[O-])cc1C CCC(C)CCC(O)CC(=O)NCCCCCCN(C(=O)C1=CCCS1)C C1(CNC(C2(OC)CCC2)=O)CCCCN(C(C23CCC2C3)=O)C1 c1(C(=O)NCC2CC(NC(=O)C=CCO)C2)cnc(OCC(F)F)c(Cl)c1 Cc1cc(F)ccc1C(O)C(=O)NCCCC1(NC(c2cnc(S)[nH]2)=O)CC1 c1(C(=O)NCC2CN(C(C)=O)C(C)(C)C2)ccc2c(c1)C=CS2(=O)=O CC1(C(=O)NC2CC(NC(=O)C(O)Cc3ccccn3)CC2O)CCCCO1 C(=O)(CC(C)(C)CNC(=O)C=CC1CCCCC1)N(CC=C)C(C)C C=C(Cl)CCC(=O)N1CCC(N(C(=O)C(C2CC2)OCC)C)CC1 C1(C(N2CCC(C3CC3)(NC(=O)CSC(F)F)C2)=O)CCC2(CC1)CC(O)C2 c1(OC)ccc(Cl)cc1S(=O)(=O)N1CCC(C)C1c1ccccc1NC(C)=O CC(C)CC(CN=c1cc[nH]c(C#N)n1)NC(=O)C(C1(O)CCCC1)F CC1C(NC(c2cnnn2C)=O)CC2CCC1N2c1nnn(C)n1 N1(C(C(CC)O)=O)C(C(=O)NCc2cscc2OC)CC2CC12 C#CCCC(=O)N(C1CC1)Cc1cn(CC(C)NC(=O)C(C)(C)C)nn1 Cc1c(CNC(C2CC2F)=O)cccc1-n1cc(-c2cccc(F)c2Br)nn1 Cc1cc(C)c(C(=O)N(CCCN(C)C)CCNC(c2ccc(F)nc2)=O)cn1 N1(C(COC)=O)CCC(C(C(C)C)NC(c2nocc2CC2CCCC2)=O)CC1 C(=O)(CCCCCCC(C)C)NCC(CO)NC(CCCC(=C)C)=O c1(C(N2CC(C(C)NC(C(C)(C3CC3)OC)=O)OCC2)=O)nnc2ccccn12 n1(CCC(=O)N(CC(C)O)CCNC(=O)CS(C)(=O)=O)ncc2c1CCCC2 N1(C(=O)NCC)CCC(NNCCNC(=O)C(C)C)CC1C.N1(C(=O)O)CCC(C)C1.C C(C)(C(=O)NC1CC(NC(=O)CCc2cocn2)C1)NC(C)=O c1(C(=O)NC(C(C)C)CCNC(C2CC3CC3C2)=O)ccn2ccnc2n1 CCCCCC(C)(C)C(=O)NCc1ocnc1C(=O)NC1(C)CCC(=O)NC1 C1(CC(=O)NCC(C)NC(c2nc(COC)oc2)=O)CCCC(=O)N1 S(=O)(=O)(c1cc(F)ccc1C)N(CC(CC)O)Cc1ccccc1Cl c1(C(=O)NC2(CCNC(C(C(C)OC)O)=O)CCC2)cccc2nccn12 C1(NC(COCc2ncc(C)o2)=O)CCN(C(C2(CO)CC(F)(F)C2)=O)CC1(C)C C1(C(=O)NCC(c2ccc(SC(CC)C)cc2)N(C)C)CCCCS1(=O)=O c1(CNC(C)(C)CCC2CCOC2)cccc2oc(CC(F)(F)F)nc12 CCC(CC(=O)Nn1ccccc1=O)N(C(=O)CC1CCOC1(C)C)C CN1C2=NC(=O)CCCC1(C(=O)O)CN2.c1(S)cccc2ncccc12 CCCC(CNC(=O)C(C)C#N)C(=O)NCC1=NOC(C)C1 C1(CNC(C2(SCC)CC2)=O)CCCCN(C(c2cccc(CC)c2N)=O)C1 N1(C(C(c2cnn(C)c2)C)=O)C2CCC1CC(NC(=O)C(C1CCCCC1)F)C2 C1(NC(C(F)OC)=O)CN(C(C2CC2c2ccccc2)=O)C2(CCC2)C1 c1(C(=O)NCC2(CNC(C(C)SCCCC)=O)CCCC2)cc2cnccc2[nH]1 CCC(C)C(C(=O)N1CCC1(C)CC(=O)Nc1ccc(CO)nc1)N(C)C Cc1cc(C2CC2)ncc1C(N1CCCN(C(=O)CNC(=O)C2CC2)CC1)=O C1(C)(NC(C(C)CC2CCCC2)=O)CCCC1NC(=O)CN1CSCC1=O C(=O)(C(C)(O)C1CC1)NC(C1CCCN1C(=O)C(C)NC(C)(C)C)C C(=O)(C(C)(F)CCCC)NC1CCC(NC(c2cc(CCCCC)[nH]n2)=O)CC1 c1(C(C)(C)NC(CCn2cc(CCNC(N(C)C)=O)nn2)=O)cc(F)cc(F)c1 c1(CC)ncc(Cl)c(C(N2CCC(C3CCCN3C(C3(C4CC4)CCC3)=O)C2)=O)n1 S(=O)(=O)(CC(=O)N(C)CC1C(C)CCN1C(=O)CCCCC1CCCCC1)NC Cc1nc(Cl)c(NC(C2CN(C(c3ccc(CCO)cc3)=O)CCN2)=O)c(Cl)n1 CC(F)(F)C(C)(C)C(=O)NCC1CCC1NC(c1ccc(-c2cc[nH]n2)cc1)=O N1(C(c2c(OC)scc2)=O)CCC(C(F)(F)F)C(CNC(=O)CC(C)SC)C1 C(=O)(CC(C=C)CCC)NC(CC=CC(=O)NC(C1CCOCC1)C#C)(C)C N1(C(C(CC(C)C)O)=O)CCN(C(c2ccccn2)=O)CCC1C CC(C)(C)C(CO)C(=O)NCC1(NC(=O)C(c2ccc(F)c(Cl)c2)O)CC1 C(CS(=O)(=O)CC(=O)N1CCCCC1CCC(C)(C)NC(=O)C(C)O)OC N1(C(C2N(Cc3ccc(C)c(Cl)c3)C3C(C2)C3)=O)C(C)(C)CCCC1(C)C C1(NC(c2ccn(C)n2)=O)CCCC(NC(C2CCC(C)(C)CC2)=O)CC1 O=C1CCCCC1CC(=O)NCC1CN(C(=O)CC2CC3CCC2O3)C1 N1(C(Cn2c(C(F)F)cc(C)n2)=O)CCC(C)C(NC(=O)CNc2cccs2)C1 C(c1c(F)ccc(Cl)c1F)=CC(=O)N(C(c1cn(CC(=O)OCC)nn1)C)CC c1(C(=O)NC2(c3cccc(Cl)c3F)CC2)ccn(O)c(=O)c1 CC12CCC(NC(=O)C=Cc3cnc[nH]3)(CC1)OC2 c1(OC)ccc(NC(C2CCCC2NC(C2CC(=O)CCO2)=O)=O)cc1 C1(C(N(CCCNC(C2C(C=C)C2)=O)CCO)=O)CCCN1Cc1ccccc1 C(CCCCCN=c1[nH]nc(-c2ccccc2)o1)N(C(C(C(CC)C)OC)=O)C C1(C(=O)NCC(C=C)O)CC2CC1CC2NC(C1CC2CC(=O)C1C2)=O C1(C(=O)NC(c2noc(=O)n2C)C)CC2COC(C)CN2C1 C1(C(C)NC(C2(C)CC(C)C2)=O)CN(C(c2nn(C)cc2N)=O)CCO1 CC(CC1CCCC1)C(=O)NCCCN(C(C1CC(F)(F)C1)=O)C1CC1 C1(OC)CC(CNC(c2cn(C)c(C)n2)=O)N(C(=O)CC2CCCN2C(C)C)C1 Cc1cccc(Br)c1CNC(=O)CCc1nccn1C.N12CC(C1)C(=O)NCCC2 c1(NC(=O)C2=CCC2)cccc(NC(C2C3CCCOC23)=O)c1 C1(O)(CC(=O)NCCOCC(C)C)CCN(C)CC1 N1(C(CSCC)=O)CCC2(CCC(CNC(c3ocnc3C)=O)OC2)CC1 C=CC1(C(N2CCCC(N(C)C)CC2)=O)CCN(C(C23CSCC2C3)=O)C1 c1(N2CCCC(C#C)C2)ncc(S(=O)(=O)NC2CC(OC)CN(CC)C2)cc1Cl C=CCC(C(=O)NCCC1(NC(=O)C(O)C(C)C)CC1)C(C)C C(=O)(CC1OCc2ccccc21)N(CCN(C(c1cc(CC)cc(F)c1)=O)C)C C1(OC(CCCN(C(=O)C(=O)NC2CC(OC(F)F)C2)C)=O)CCC2CC12 N1(C(C2(C)N(C(c3c(C)cc(C)s3)=O)CC(O)C2)=O)CCc2nc[nH]c2C1 Cc1cnn(C(C)C(=O)NCCN(C(=O)CCc2ccc(Cl)s2)CC2CC2)c1 c1(C(=O)NC(C2CC(C(=O)NCC(F)(F)F)C2)C)cccc(=O)n1C c1(C(N2CCCC(CNC(c3cccc(OC)n3)=O)C2)=O)cc2n(n1)CCO2 c1(C(=O)NCCCCC2CN(C(C(C3CC3)SC)=O)C2)ncc2ccccn12 Clc1ccc(-c2cc(NCCC3CC=CCC3)on2)cc1 C(CNC(c1csc2cncn12)=O)(CC(F)(F)F)NC(CC(C=C)C)=O C1(NC(C2(C)CCCOC2)=O)CC2CC1N(C(c1c[nH]nc1C1CC1)=O)C2 C1(NC(C(C(CC)O)C)=O)CC2CCCC(C1)N2C(=O)CCSc1ccccn1 C(=O)(C1=CCC2CCC1N2C(c1cncc(Cl)c1)=O)N(CC(CC)O)C C1(C)(CNC(c2c(C)coc2C)=O)CC(F)(F)CN1C(c1ccnn1C)=O C(=O)(NNC(=O)CCCCCCN)c1c(C(C)(F)F)ccc(Br)c1 c1(C(N2CC(O)(CNC(c3nc(CC)oc3)=O)C2)=O)n[nH]c2cc(OC)ccc12 C1(NC(Cc2cc(COC)on2)=O)CN(C(c2cnn(C)c2N)=O)C(C)(C)C1 C(C)(C(C(=O)NC1(CNC(=O)CCCSC)CCCC1)N(C)C)OC n1(CCCC(=O)NC(CC)CNC(=O)CCC2(CO)CCCO2)c(O)nnc1O C1(C(N2CC(CNC(c3ncc(CC)nc3)=O)(OC)C2)=O)CCc2cnnn2C1 C1(NC(C(C2CCOC2)OC)=O)CCCN(C(=O)CC2OC(C)(C)OC2=O)CC1 C1(OC)CC(CCNC(c2csnc2OC)=O)N(C(=O)COC2CC(F)(F)C2)C1 C=C(C)CC(C(=O)NCC(CC(C)C)OC)NC(c1cnn(C2CC2)c1)=O C1(NC(c2c(CC)occ2)=O)(CNC(=O)C(F)OC(F)(F)F)CC(F)(F)C1 N1(C(=O)CNC(c2ccc(F)cc2[N+](=O)[O-])=O)CC2(CC2)c2ncccc21 CN1C(=O)CC(NC(N2CCN(C(=O)N=S(C)(C)=O)CC2)=O)C1c1ccncc1 N1(C(=O)CN2CCN(C(=O)C=C(Cl)Cl)CC2)CC2CCC(C1)C2O N1(CC(=C)C)CCc2cc(OC(F)F)c(F)cc2C1 N1(C(c2c(C)noc2)=O)CCCC(CCCCNC(=O)CN2CC3C=CC2C3)C1 C1(CNC(=O)CN2CC3CC3C2)CCC(C(N2CCC3CC23)=O)CC1 C1(=O)C(Cc2cnc[nH]2)CN1C.C12(CC(=O)NC3CCC3)CCCC1C2 N1(C(c2n(C(C)C)ccn2)=O)CCN(CCCNC(C2CCCN2C=O)=O)CC1 C1(CC)(CC)CC(O)CN1C(=O)C(CNC(C1OCCC1C)=O)N(C)C C1(C(=O)NC2CC(CNC(COCC(=C)C)=O)C2)CCCCC(C)(C)C1 c1(NC(=O)NC(c2c(F)cccc2F)C(F)(F)F)cnc(O)c(F)c1 N1(C(CC(CCC)(C)C)=O)CCC2(CC1)CCN(C(c1ccc(C(F)F)o1)=O)C2 C1(C(=O)NCCC2N(C(COCCCC#C)=O)CCC2)C(F)(F)C12CCC2 c1(C(=O)NCC2C(NC(C3(CC=C)CC3)=O)C2)cc2ccc(F)cc2nc1O Cc1cc(C(F)(F)F)ccc1C(=O)NC(C1CCCCCC1)c1nnnn1C C1(C(=O)NC2C(C)CCC2)CC2OCCC2N(C(=O)Cc2ccsc2)C1 c1(C(N2CC(NC(C(C(=C)Cl)(C)C)=O)CC3(C2)CC3)=O)ccc2c(cnn2C)c1 CC1CC(NC(C2C3CCCCC23)=O)CN(C(=O)C(c2ccc(F)c(F)c2)=O)C1 c1(CNC2(c3nnnn3CCOC)CCC(F)(F)C2)cnn2c1OCCC2.C1CC1 CC1CC(NC(C2(O)CCSC2)=O)CN(C(c2cnn(C(F)(F)F)c2)=O)C1 N1(C(c2ccc(Cl)[nH]2)=O)CCC2OCCN(C(=O)CCc3cn[nH]c3)C2C1 c1(C(=O)NCCCNC(C2CC3(C2)CC(F)C3)=O)cc2cccc(Cl)c2s1 C(c1ccoc1)=CCNC(C12CC(CO1)C2)C.CCO C12(CN)CCC(CN(C(=O)CCc3ccn(-c4ccccc4)n3)C1)C2 c1(C(N2CCC(C(=O)NCC3CC(F)C3)O2)=O)cccc2[nH]ncc12 C1(CNC(c2cc(SC)oc2C)=O)CC2(CC2)CN1C(=O)CC1OCCC1(C)C N1(C(CCCC)=O)CC2(CC(NC(=O)CC3CCC(C)C3)CO2)C1 Cn1nc(C(N2CCCC(CCNC(c3ccncc3F)=O)C2)=O)cc1C#N C(CCN(C(=O)CCc1ccccc1)C)(C(C)(C)C)NC(CSCC#C)=O N1(C(=O)OC(C)(C)C)CCC2(CNC(c3cc(F)c(F)c(F)c3)=O)CCCC12 c1(CC(N2CC(C(=O)NOCC(F)CO)(CC=C)C2)=O)cnccc1C c1(SC(C)CC#N)cccc(C(N2CC(F)(CO)C2)=O)c1 Cc1cccc(CC(=O)NCC2(O)CC(NC(=O)C(c3ccccc3)F)C2)c1 O=S(=O)(c1c[nH]ccc1=NCC1(S(=O)(=O)CC)CC1)NCC(O)C1(Cl)CC1 c1(CCCC)ccc(Oc2ccc(N(S(C)(=O)=O)Cc3nncn3C)cc2)cc1 c1(NC(C23CCC(NC(CSC)=O)(CC2)CC3)=O)cc(Br)cnc1[N+](=O)[O-] C12(OC)CCN(CC1)C2.c1(NCC(=O)OC)cn(C)nc1C C1(C(=O)NC(C)C(CO)NC(C2C=CCS2)=O)COCCN1C C1(NC(C2C(C(=O)OC)CCC2)=O)CCC(O)CN(C(c2nccc(C)n2)=O)C1 c1(C2(C(N(C(CNC(c3cc(C)[nH]n3)=O)C3CC3)C)=O)CC2)cccc(Cl)c1 c1(COC(C(=O)NCC2C(NC(CC(=O)OCC)=O)CCC2)C)ccccc1F Cc1cc(Cl)ccc1C(=O)NCCC1CCCN1C(c1cnc(S)n1C)=O C1(CNCCC(CC)CC)CCC2C(CC1)C2(F)F n1(CC(C)C)[nH]c(CC(=O)NCC=CCNC(=O)CCc2cncn2C)cc1=O N1(C(C2CN(C(c3c(C)ccn3C)=O)CC23CC3)=O)CC2(COC(C)C2)C1 CC(C)(C)CC(C)(C)C(=O)N1CCC2CC12C(N1CCc2c(nnn2C)C1)=O C(=O)(CC(O)CNC(=O)OC(C)(C)C)NC1C(NC(C)=O)CC1 CC(C)(O)C(F)C(=O)N1CC2CC1C2NC(=O)CC1=CCCC1 N1(C(c2cc(C)nc(C)n2)=O)CC(NC(C2(C(F)F)CCCC2)=O)CC(C)(C)C1 c1(OC)c(-c2nc(Nc3cc(C)c(-c4c(C)n[nH]c4C)cn3)cs2)cccc1Br N1(c2ncc(CC)cc2C)CC2CC(NC(=O)C(C)(C)C(O)C=C)CC2C1 C1(CCC)(NC(=O)C(C)CO)CCN(C(c2cccc(F)c2SC)=O)CC1 C12(NC(C(CC(=O)OC)C)=O)CCCC1CN(C(c1nccc3occc13)=O)C2 C1(C(=O)NCC(C)(C2CC2)NC(COCC=C)=O)CCC(C(N)=O)CC1 c1(C(=O)NC(C2CN(C(=O)C(C)(C)C3CCC3)C2)C)cc(Oc2ccon2)n[nH]1 C(=O)(C(F)(CNC(c1cc(O)nc(C)n1)=O)C(C)C)N(C(CC)C)CCO N1(C(c2ncc(C)cc2C)=O)CCC(NC(c2cnn3c2OCC3)=O)C12CCC2 N1(C(c2c(C)nn[nH]2)=O)CCCC(C)(C(=O)NC2C3C=CC(C3)C2CO)C1 c1(C(N2C(C)(C(=O)Nc3ccc(O)cc3F)CCC2)=O)cccc(C#N)c1F CN1C(=O)CSC1=CC(=O)NC12CC(CNC(C3(F)CCCOC3)=O)(C1)C2 C1(COC)(NC(=O)Cc2ccc(Cl)nc2F)CCN(C(=O)CC2CCCC2)CC1 N1(C(c2cc3sccc3[nH]2)=O)CCC2OCCN(C(=O)Cc3cn(CCO)nn3)C2C1 C1(C(=O)NCC2CCC(CN(C(=O)Cn3ncnn3)C)CC2)(OC)CS(=O)(=O)C1 C1(C(=O)NCC=CCNC(c2ccc(C(C)C)o2)=O)CCCCN1C1CCCC1 c1(C(=O)NC2(COC)CN(C(C3CCCCC3(C)C)=O)C2)ccc(C#N)cc1C CC1(NC(c2cc(=O)cc[nH]2)=O)CCN(C(C2(C3CC3)CCCO2)=O)CC1 C(=O)(CC(C(C)C)c1ccccc1)N(CCNC(C1(C)CC1C)=O)CC CCC(CC(C)C)C(=O)N1CCC2(C1)CN(C(c1cc(C)c(F)cc1O)=O)C2 c1(C(N2C(CNC(C#CC(C)(C)C)=O)CC2)=O)cccc2c1C(=O)NC2 C1(C)(C(=O)NCC(c2ccc(NC(=O)OC(C)(C)C)cc2)C)CCCN1C c1(-c2cn(C3(CC)CCCN3C(=O)C(C)CCCOC)nn2)cncc(C#N)c1 N1(C(c2c(C)nc(C)o2)=O)CC2C=CC1C(C(=O)NC1CN(C(N)=O)C1)C2 C(=O)(CC(C)C(F)(F)F)C(C)C(N1C(C)COCC1(C)C)=O CCC(C)C(O)C(C)C(=O)N1CCCC1(C)CCC(=O)Nc1cc(Cl)n(C)n1 c1(NC(C)CC#N)nccc(NC2CCN(c3ccccn3)C2)n1 N1(C(CC(=O)N(C)C)=O)CCCC(C2CN(C(C3CCO3)=O)C2)C1 CC1(C)CC(NC(=O)Cc2csnn2)CN(Cc2cc[nH]c2-c2cccnc2)C1 c1(C(=O)NC(C2OCCN(C(C3(C=C)CCCC3)=O)C2)C)cc(OC)ccc1F Cc1c(C(N2CC3CC(NC(c4ccncc4N)=O)C3C2)=O)cnc2ncnn12 Cc1cc(=NC2CCN(C(C3CCC34CCC4)=O)CC2)[nH]c(C(C)C)n1 c1(N2Cc3c(nc(C)s3)C2)nc(=NCc2cccnn2)[nH]c2c1COC2 c1(OC)cccc(CNC(C2CSCCN2C(=O)COC2CCC2)=O)c1F N1(C(C(C)CO)=O)CCC(CNC(=O)CC2CC(F)(F)C2)C(F)(F)CC1 c1(C(=O)NCC(CC(F)(F)F)NC(C(CCOC)C)=O)c(C)cc(C)oc1=O Fc1ccc(CCNC2CC23CCSCC3)c(F)c1 C1(C(=O)NC2(C#C)CC2)CC12CCN(C(=O)CCOCC(F)F)CC2 CC1(C)CN(C(=O)C(CNC(C2(C)C=CCC2)=O)CC2CC2)CCS1 N1(C(C2C(C=C)C2)=O)CCCC12CCC(NC(=O)C=C(C)CCC)CC2 Cc1cccc(F)c1C(=O)N(c1nccc(C(F)(F)F)n1)C1CC2CC1CN2 C1(CNC(C(COC)NC(C)=O)=O)CCC2(CN(C(c3ccnn3C)=O)C2)O1 Cc1ccc(OCC(N2CC3(NC(=O)CO)CCC2C3)=O)c(C)c1 C1(NC(=O)CSC(F)(F)F)CCCC12CN(C(=O)Cn1cc3ccccc3n1)C2 n1(Cc2occ(CO)n2)cnc2c(N3CCC4(CCCO4)C3)ncnc12 N1(C(c2c(CC)scc2)=O)CCC(O)(C(C)NC(c2ccccc2COC)=O)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])N(CC(CC)NC(C1(C(=O)OC)CC=CC1)=O)C C(=O)(C(C)(CC1CCC1)Nc1ccc(C(C)C)cc1)OCC n1(C(C)C)cc(C(N2CC(CNC(=O)CCF)C(C)(C)C2)=O)c(O)nc1=O N1(C(C(C2CCOC2)OCC)=O)CCCCC1CNC(=O)CCCCF c1(C(=O)NCCN(C(c2ncnc(C)c2C)=O)CC)cc(N)cc([N+](=O)[O-])c1 C(=O)(C1=NOC2(CCC2)C1)N(C(C(=O)NCc1ccc(C#C)cc1)C)CC c1(CNC(NCC(CO)Cc2ccccc2)=NCC2CC2)nc2c(s1)CCCC2 c1cc(F)ccc1F.CC(C(CO)NC(=O)C(F)(F)C1(O)CCC1)NC(=O)COC c1(CC(N2CCC(NC(C3C4C=CC3CC4)=O)CC2)=O)ccc(Cl)cc1O Cc1cnc(C(=O)NCCCN(C(C23CCCC2C3(F)F)=O)C2CC2)cc1Cl c1(C(=O)C2CC2)ccccc1-n1cc(C2CC(C(=O)O)C(O)C2)nn1 c1(CC(=O)N)cccc(OC2(CCCCCNC(C(C=C)O)=O)CCC2)c1 C1(NC(c2cnc(C)n2C)=O)(CNC(C2(C)CCOC2)=O)CCCCC1C CC1CN(C(C2CN(C(=O)CCC(C)(F)F)CCO2)=O)c2ccccc21 c1(C(N(C(C)C(N2CCCCC2C2CC2)=O)C)=O)cccc(F)c1 c1(C(N(CC(O)CN(C)C(C2(c3cc[nH]n3)CC2)=O)C)=O)cc(Cl)cc(Cl)c1F c1(C(N2C(C(C)OC)CN(C(=O)CNC(C)=O)CC2)=O)nc2c(s1)COCC2 c1(C(C)NC(N2CCC(C(N3CC4CC4C3)=O)C2C(C)C)=O)ccc(Cl)cc1 c1(C(=O)NC(CC)CNC(c2nn(C(F)F)cc2Cl)=O)cccc(C)c1CC CCCC(CCC)=CC(=O)NC1(CO)CCN(C(C2CCCO2)=O)C1 C(=O)(CCCCCCCNc1cc(O)nc(Cn2cncn2)n1)OCC C(=O)(CCC(C)CN(C)C)NC1CC(CC(=O)Nc2cnc(CC)nc2)C1(C)C Cc1cc(C(=O)NCC2CC(NC(=O)CCc3cnc[nH]3)C2)cnc1C(F)(F)F Cc1ccc2c(c1C(N1CC3CC3(CNC(=O)CC(C)(C)C)C1)=O)CCCN2 C(=O)(CCCN(C(=O)CC1C=CCCC1)C)N(C1C(C)CC1)C C1(CC(=O)NC2CC(NC(C=C(CSC(C)(C)C)C)=O)C2)CC=CCC1 Cc1noc(Cl)c1CCC(=O)N(CC(C)CNC(=O)C(N1C(=O)CCC1=O)C)C Cc1cc(C(N2CC(NC(c3nn(C)cc3Br)=O)C3CC23)=O)ncc1F c1(C(=O)NC(CNC(CCC=C)=O)(C)C(C)C)sc(C)c(C)c1Br N1(C(CCOCC)=O)CCC(CNC(=O)C(C)N2CC(C)C2)C(C)C1 N1(C(C2C(CC)CCO2)=O)CC(C)(C)CC1C(=O)NC(CO)C1(C)CC1 c1(N(CCCc2ccc(C)s2)C)ccncc1S(=O)(=O)NCC1COCC1CO C1(NC(C(C(=O)OCC)(C)C)=O)CC2(CCN(C(=O)C=Cc3sccc3C)C2)C1 C1(CCC)(NC(C2CCCN(CC)C2)=O)CCCN(C(C2CCC3CC3C2)=O)C1 C(=O)(CS(=O)(=O)CCO)N1CC=C(CNC(C=Cc2occ(C)n2)=O)CC1 C(=O)(CCCC(C)C)NC(C1N(C(c2c(C)nc(CC(C)C)s2)=O)CCC1)(C)C C(=O)(C1=CC2(CCOC2)C1)NCc1c(C(N2CC3C(C)(CSC3)C2)=O)con1 n1(C(N(CCN(C(=O)CCOC2CCCC2)CC)CC)=O)nc(C)c(C)c1C N1(C(CSCC=C)=O)CC(CNC(=O)C(C2CC(F)(F)C2)O)C(C)C1 CC1CCC2(CC2)N(C(C2CCC(C)N(C(=O)C=Cc3ccoc3)C2)=O)C1 C12(CNC(=O)Cc3cnc[nH]3)CCC1CN(C(c1ccc(-c3cscn3)nc1)=O)C2 Cc1cc(C(=O)NC2CCCCC2NC(=O)CO)cc(C)c1F N1(C(Cc2c(C)nc(CCCC)s2)=O)CCN(C(=O)C(Cl)=CCl)C(C)CC1C N1(C(C2CC(=C)C2)=O)CC(CNC(c2cc(O)nc(OC(C)C)n2)=O)C(F)(F)C1 c1(C(=O)NC2C(C(=O)Nc3cc(C(C)=O)cc(F)c3)C2)ccc2cnccc2n1 c1(C(N2C3CN(C=O)CC32)=O)ccc(Br)cc1I.c1(C(N)=O)cccc(Cl)c1 C1(NC(C2CCS(=O)(=O)C2)=O)CC2CCC(C1)N2C(=O)CCC1CCCC(O)C1 c1(C(N2CC(N(C(=O)Cc3cn(CCCF)nn3)C)C(O)C2)=O)ccc(Cl)nc1N C#Cc1ccc(OC)c(C(=O)NC2CC2NC(=O)C(c2ccc(F)cc2)C)c1 Cc1ccc(CNC(C2CCN(c3ccccc3)CC2)C2CC2)c(Cl)c1 Cc1cccc(C)c1CC(N1CC(C)(C)CC1CNC(=O)C(c1cccnc1)O)=O C=C(C)CCCC(=O)NCC1CCC(NC(=O)CCCC2CCCO2)C1 C12CC(=NO1)C(=O)NC2.Cc1conc1CC(=O)NCCCC1CCCCO1 C1(O)(C(CNC(C=C(C)C(C)C)=O)(C)C)CCN(C(C2CCC(=O)N2C)=O)CC1 C=CCCCCCCCC(=O)NCC(O)CCNC(=O)Cc1ccccc1OC C(CC(C(=O)NCCOCC1CSC1)NC(=O)CSC)OC CC1(CNC(=O)COC2CCN(C(C3CC4(CCC4O)C3)=O)C2)CC2C=CC1C2 C1(C(=O)NOC)(CC)CCCN(C(=O)Cc2ccc(OC(F)F)cc2)C1 C(C(C)N=c1[nH]c2ccccc2nc1C#N)(C1CC1)NC(C(C(C)C)C)=O O=C(CCCC(=O)NC1(CC(N2C3CSCC2C3)=O)CCC1)C1CC1 C(=O)(C(C)CC1CCC1)N(CCC(=O)NCC1CC12CC2)CC=C c1(C(=O)NC2CN(C(CC3(C=C)CCC3)=O)C(C)C2)cn2ccnc2s1 C1(C)(C(=O)NC(CC=C)CNC(=O)C(C)C)CCC(O)CC1 C(C)(N=c1[nH]c2cc(F)cc(F)c2o1)C1(NC(c2c(OCC)nsc2OC)=O)CC1 c1(C(=O)NC(CSCC)C(=O)N2CCC2(C)C)cc(C)sc1N C1(C(=O)NC(C)CF)CN(C)CCN1C(=O)CCS(C)(=O)=O c1(NC(=O)NCC2C(OC)CC2)cc(F)c2nc(C)cn2c1 c1(CCC(=O)NC2CCN(C(CCC#C)=O)C2)cncc(F)c1 CC1(C)CC(C(N2CCC(OCC(N)=O)C2)=O)CN1C(c1coc(CO)c1)=O C1(C(=O)NCCC2CC(OC)C2)CN(C(=O)C2=COCC2)CC1c1ccccc1 C(=O)(C1=CCC2(CC1)CC2)N(C(C)CNC(c1csc(C#N)c1)=O)C N(C(=NCc1ccncc1Cl)N1CCC(CC2CCOC2)C1)C(C)C N1(C(c2c(C)nccn2)=O)CCCC(N(C)C(C2C=CCC2)=O)CC1 c1(OC)cccc2[nH]c(C(=O)NCC(CO)NC(=O)CCCCC(C)C)cc12 Cc1cc(C)cc(C=CC(=O)NC2CCN(C(c3cc[nH]c3)=O)CC2(C)C)c1 c1(CN2CCCC(C(N(CC=C)CC3CC3)=O)C2)c(OC)cccc1F N1(C(Cc2occ(C)c2)=O)C2CCC1CN(C(c1cnc(Cl)cn1)=O)CC2 N1(C(c2c(C)nccn2)=O)CC(NC(=O)C(c2ccc(Cl)c(F)c2)=O)C(C)(C)C1 C(=O)(CC1=CCCC1)NC1C(NC(CCC=CCC=C)=O)CCC1 N1(C(CSCC(N)=O)=O)CCC(COCCC2(NC(C3COCCO3)=O)CC2)C1 c12ccccc1C(=O)N1CC(C1)OCC(=O)N2.N1(CC)CCC(CC(=O)OC)C1 c1(C(=O)NCC2CN(C(C3C(OC)C3)=O)C2)cc(-c2csc(C)n2)cn1C C1(NC(c2n(CCOC)ncc2)=O)CCCN(C(=O)C(n2nc(C)cc2C)C)C1 c1(NC(CNC(Cn2c(NC(C)=O)nnn2)=O)CO)cn(C)c2ccc(F)cc12 C(=O)(CCCCC#N)NC(c1ccc(C)cc1)CNC(C1(Cl)CC12CCC2)=O C=CC(C)(O)C(=O)NCCN(C(=O)CC1CCN(CC(F)(F)F)C1)CCC C1(C)(C(=O)NC(C2CCN(C(C(C=C)(F)F)=O)CC2)C)CCC(=O)NC1 CC(C)CC(C)(O)C(=O)N1CCC(F)(C(=O)NCCC2=CCCCC2)C1 c1(C(N2CCC(N(C(c3cnc(CC)o3)=O)C)CC2)=O)cnn2c1CN(C)CC2 N1(C(C(C)C(C)(C)C)=O)CC2(CCN(C(=O)CCC3NC(=O)NC3=O)CC2)C1 Cc1cnncc1C(=O)NC(C1(CNC(C2CC2C(C)O)=O)CC1)C CN(C)S(C)(=O)=NS(=O)(=O)N1CC(O)(C(c2ccccc2F)c2ccccc2)C1 CCC(CC)C(C(=O)NC1(COC)CCN(C(c2cc(CO)[nH]n2)=O)CC1)OC CC1=C(C(=O)NC2CN(C(c3onc(C)c3C)=O)CC2O)CCS1(=O)=O N1(C(C(C)OCC)=O)CC(CNC(c2csc(C(F)F)n2)=O)C(O)C1 CC(O)C(C(=O)NC1CC(NCCC(=O)NC2COCCC2O)C1)N(C)C C(=O)(C(C)(C)C(=O)OC(C)(C)C)NC1C2CCN(C(c3cc(CCC)on3)=O)C21 c1(C(N(CC(CNC(C2(OC)CC2)=O)O)C)=O)nc(Br)sc1C C(C)(C)(CCC(=O)NC1CCCC(COC)C1)NC(C(COC)COC)=O C1(C(=O)NCC2N(C(c3ccc(NC)cc3C)=O)CC2)CN2CCCN1CC2 N1(C(CC(C)c2ccco2)=O)CC2CC(C1)CN(C(=O)CN1CCC(O)CC1)C2 C=CCC(CC=C)C(=O)NCC(c1cccc(C)c1)NC(c1csnc1OC)=O Cc1ccnc(O)c1C(=O)NC1CCCC(N(C(=O)CC2CSC2)C)C1 C1(C)(CN(C)C(c2ccc(CC#N)cc2)=O)CCCC1NC(c1ccoc1Cl)=O C1(NC(=O)C(=Cc2c[nH]cn2)F)CCOCC1NC(=O)CC1CCCC12CC2 c1(C(=O)NCC(C2CC2)NC(C(C)N2CCCC2)=O)ccc(=O)n2c1CCCC2 C(=O)(CC(C)(C)OC)N1C(CN(C(=O)CC2CC3C=CC2C3)CC)CCC1 Cc1cnc(Cl)c(CN2CCSC(C(=O)Nc3ccccc3-c3ncc[nH]3)C2)c1 C1(CC2CC2)CC2N(C1)CC(=O)NC2=O.c12ccc(cc1)o2.C1(OC)CC1 CCC(C)(C#N)C(=O)NCCC1CN(C(c2cn(C)nc2C(C)(C)C)=O)CCO1 C1(C(C)=O)CC(CC(=O)NCCN(C)C(c2ccnnc2)=O)C1(C)C c1(CN2CC(F)CC(C(=O)Nc3cc(O)ncn3)C2)ccc(F)c(F)c1O C1(NC(c2cc(OC)nc(Cl)c2)=O)CN(C(C2(CCO)CC2)=O)CC2(CC2)C1 c1(OC)ccc(C(CNC(=O)C=CC2CC2)NC(C2OCCO2)=O)cc1 N1(C(CCC(C)N(C)C)=O)CCn2nc(CNC(=O)CC(C)(F)F)cc2C1 N1(C(C(C(CC)(C)C)=O)=O)CC2CCCC(NC(=O)Cc3ccno3)C2C1 C1(CC)(CC)CN(C(C2CC(CCNC(c3ccnn3C)=O)C2)=O)CCO1 C1(C(=O)NCC2CCCC(NC(C(F)=C(C)C)=O)C2)CCN(CCO)C(=O)C1 Cc1cc(C(=O)NC2CC(CNC(C3CCC(C)(C)CC3)=O)C2(C)C)nc(C)c1 N1(C(c2[nH]cc(C)c2)=O)CCC2(CC1)CC(NC(=O)Cc1cnn(C)c1)C2 C(N=c1[nH]nc(C(C)(C)C)o1)C1C(NC(c2cc(CC)no2)=O)CCCC1 C1(NC(=O)C=CC(F)(F)F)C2CCN(C(=O)Cc3cccc(F)c3F)CC12 c1(OC)cccc2c(C(N3CCCC(NC(=O)CCC(F)(F)F)C3)=O)c(C)[nH]c12 C1(NC(c2c(CC)oc(C)c2)=O)CN(C(c2cc(CSC)c(C)o2)=O)C2(CCC2)C1 C1(N)CCc2c(nnn2C)C1.C(=O)(CC(C)C)N1CC(c2cccs2)(CC)C1 c1(C(=O)NCCC(CNC(Cc2c(C)scc2)=O)O)cnn2c1CCC2 CC(O)CCCCCC(=O)NCC(CO)NC(c1cn(C)[nH]c1=N)=O C1(=O)C(O)C(CCC)N1.C(=O)(C(C)C(O)C(C)C)N(CC#C)CC=C C1(OC)Cc2cc(F)ccc2N(C(=O)CCc2ccccc2NC2CC2)C1 N1(C(COCC=C)=O)CCC2(CC1)CC(NC(c1cccc(C)c1)=O)CCO2 C(C#CC(=O)NC(C1CCCN(C(c2cccnn2)=O)C1)C)(OCC)OCC C1(CC(=O)NCc2cn(CCN(C)C)nn2)CCCN(c2ccc(OC)cc2)C1 c1(C(N2CC(F)(CNC(c3c(C(C)C)onc3)=O)C2)=O)cccc2c1NCCC2 N1(C(C2N(C(c3c(C)nsc3N)=O)CC(=O)NC2)=O)CCCN(C)C(=O)C1 c1(C(N2CCC(OC)C23CC3)=O)nn(C)c2ccc(F)cc12 N1(CCCNC(=O)CC2C=CCC2)CCN(C(=O)C2=CSCS2)CC1 C1(CNC(c2cnc(C(C)C)[nH]2)=O)CCCCC1NC(=O)C1=CCCC1 c1(C(N2C(C(C)NC(c3c(C)nc(CO)s3)=O)CCC2)=O)nc2sccn2c1C c1(OC)cc(F)c(C(=O)NC(C)C(C)NC(=O)Cc2cccnc2)cc1Br c1(C(C)C)ncsc1C(=O)NC(C)CN(C(=O)C(C)Oc1ccccn1)C C1(CC)C(C(N2CC(O)(CNC(C3(OC)CCOCC3)=O)C2)=O)CCN1C C1(NC(C(CCC)F)=O)CN(C(=O)Cc2ccsc2C)CC2(CCC2)C1 N1(C(=O)C(F)=C2CCC2)CCC2CCN(C(c3cccc(O)c3Cl)=O)C2C1 Cc1cc2c(C(N3CC(CNC(C4CNC(=O)N4)=O)C4(CC4)C3)=O)cccc2o1 c1(C2(NCC3CCCN(C4CCC4)C3)NCC(=O)C2)nnc2n1CCC2 C1(C(N(C2CCCC2)CCNC(C(N2CCCCCC2)C)=O)=O)CCC(C)(C)O1 c1(CNC(C(=O)NC2CCN(C3CCN(C)CC3)C2)=O)ccn2c1CCCC2 C(c1cccnc1)=C(C)C(=O)N(C)CC1CCCN1C(=O)C(c1cnn(C)c1)C C1(C)(NC(c2cc(CC)[nH]n2)=O)CCN(C(=O)CCc2ccc(Cl)s2)CC1 CC1(CCNC(=O)CCF)CCN(C(=O)C(O)c2ccsc2)CC1 c1(CNC(CSCCCC)=O)ccc(C(=O)Nc2oncc2CC)cn1 c1(CC(=O)NCCN(C(COCC)=O)CC(C)O)cnn2c1OCCC2 C1(NC(C2CCCC(C)C2)=O)(CO)CCCN(C(=O)COC(F)F)C1 c1(C=O)cc2nc[nH]c2cn1.CC1(C[N+]2([O-])NC2CC)CC2CCC1O2 n1(CC(N2CCCC(N(c3ncc(C#N)cc3Br)C)C2)=O)cc2ncccc2n1 c1(C(=O)NCC2(F)CCCN(C(CC3C(C)(C)C3)=O)C2)ccc(Cl)c(Cl)c1N N1(C(CSCC#C)=O)CC(NC(c2nc(Cl)sc2C)=O)CC2(CC2)C1 Cc1nc(SCCC(Cc2ccccc2)CC(=O)NCCc2nocc2Cl)n[nH]1 C(C1CN(C(C2(CC)COC2)=O)CC1C(N1CC(F)(CF)C1)=O)=CC N1(C(CCc2ccc(C)s2)=O)CCC(NC(=O)C=CCN2CCCC2)C(O)C1 C1(C(C)(C)C)CC(=O)N1.C1CC(=O)OCCCO1.C(CCF)OCC N1(C(c2c(C)cccc2F)=O)CCOC2(CCN(C(c3cc(C)n(C)c3)=O)C2)C1 c1(OC)cc(CNC2CCCC2C(=O)NC2CCCOC2)cc([N+](=O)[O-])c1 Cc1ccc(C2CCN(C(CCCc3nc(-c4ccncc4)n[nH]3)=O)C2)c(C)c1 C1(C)(NC(C=C(C)C(F)F)=O)CCC(NC(c2cccc(C3CCC3)c2)=O)CC1 N1(C(c2n(C)ncc2Cl)=O)CCC2(CC1)CCN(C(c1cnnc(O)c1)=O)CC2 C1(CC#C)(C(N2CC=CC(NC(=O)C3=CCSC3)C2)=O)CCOCC1 CC1CN2CCN1C(C(=O)NC1CCCN(C(C3(N(C)C)CCC3)=O)CC1)C2 C12(NC(c3n(CC)ncc3)=O)CC3CCC(C1C2)N3C(=O)Cn1nc(C)oc1=O C(=O)(C#CC1CCOCC1)NC(C1CCCCC1)C(=O)NC1CCC(OC)C1 c1(C(=O)NC(CNC(c2cn(CCOC)nn2)=O)C(C)C)c[nH]cc(C)c1=O c1(C(C2CN(C(c3c(C)nns3)=O)C2)N(CC(O)CO)C)ccc(Br)cc1 C(=O)(C(C(F)(F)F)C(F)(F)F)N1C(C)CCN(C(=O)CCc2ncccn2)CC1 C1(C(N2CCC(N(C(=O)CN(C)S(N)(=O)=O)CCC)C2)=O)CCC(=O)N1CC N1(C(c2nc(C(C)NC(CC(=C)C)=O)oc2)=O)CCC(CO)CC1 c1(C(=O)NCC(C)N(C(c2cccc(C)n2)=O)C)ccc2c(c1)NC(=O)C(C)O2 C1(C(N(CCCCNC(C2(C(=O)NCCCOC)CC2C)=O)C)=O)CC(=O)N(C)C1 c1(CC)c(C)sc(NC(C2CC3(CCNC3)C2)=O)c1C(N)=O C1(CC=C)(NC(=O)C=C(C)I)CC2CCC(C1)N2C(c1c(C)cc(C)nc1O)=O N1(C(C(C)CO)=O)CC(CNC(=O)C=C2CCOCC2)CC1(C)C c1(OC)cccc(F)c1C(=O)NCCCCNC(=O)C=Cc1ncc(C)[nH]1 CN1CCc2cc(C(N3CCC3C(N3CCC4(CCC4)C3)=O)=O)ccc21 c1(C(N(C2CCN(C(C3(C#C)CC3)=O)C2)C)=O)cc(N)cc(S(C)(=O)=O)c1 N1(C(c2c(C)n(C)nc2)=O)CCN(C(=O)Cc2nn(C)cc2Cl)C(CC(F)F)C1 C1(C(N(C(C)CNC(=O)C(C)=C2CC2)CC)=O)CCCN1c1nccs1 S(=O)(=O)(c1ccc(NC2CCC(F)(F)CC2)c(F)c1)N1CC(C)OC(C)C1 c1(OC)cnc(C(=O)NCC2(O)CCN(C(C34CCCC3C4)=O)C2)c(F)c1 Cn1ccnc1C(=O)NC(CCCNC(=O)CCOCCF)c1ccccc1 N1(c2nccc(C)n2)CCN(N2CCc3ccccc3C#CC2)CC1 c1(CC)oc(C)cc1C(N1CCC(C(C)C(=O)N(C2CC(COC)C2)C)C1)=O c1(C(=O)NC2(C)CN(C(c3ccc4n[nH]cc4c3)=O)C2)nccc2ccn(C)c12 c1(C(=O)NCC2CN(C(C(CCC)(C)O)=O)CC2C)ccc2c[nH]nc2c1 C(=O)(CCS(=O)(=O)c1ccccc1)NCCC(CCNC(C(COC)(C)O)=O)C c1(C(N2C3CC(CNC(C4C(C)(C)CO4)=O)C2CC3)=O)cccc2c1NCCC2 CC1ON=C(C(=O)NC2C3CC(NC(C4C5COCC45)=O)CC23)C1C c1(OC)cc(C(=O)NC2CN(C(c3cnoc3C3CCOCC3)=O)C2)ncn1 C(=O)(C1COc2ccccc21)N(C1CCN(C(C2(CN(C)C)CC2)=O)C1)CCC N1(C(C(C)Sc2ccc(C)cc2)=O)CCN(C(=O)C(O)C(C)(C)C)CC12CCC2 N1(C(CSCC)=O)CCN(C(C2CCCCN2C(C)C)=O)C(c2cn[nH]c2)C1 c1(C(=O)NCC(CC)NC(C2CCC(F)CC2)=O)cc(N)ccc1Br N1(C(C(CC(C)C)O)=O)CCC(C(=O)NCC2CC[Si](C)(C)C2)C12CCC2 N1(C(C2=CCC(NC(c3ccoc3)=O)C2)=O)CCCC(C2CC2)CC1 CCN=c1[nH]cnc2cc(C(=O)NC(C)CCNC(c3cncnc3)=O)ccc12 C#CCCC(C(=O)NCCc1ncc[nH]1)NC(c1cc(O)cc(F)c1)=O C(=O)(CC1C(=O)Nc2c(F)cccc21)NC(C)CNC(c1cc(C(F)F)[nH]n1)=O c1(C(C)C)nc(N)cc(N2CCC(c3ccns3)CC2)n1.N1(CCF)CCOCC1 N12CC(C(C)(C)C1)NC2=O.c12cc(ccc1F)CC(C(C)C)O2.C(C)(C)(C)ON c1(C(=O)NCC2CCCN(C(C3CC(=C)C3)=O)C2)ccc(Cl)c(C)c1 CS(=O)CCC(=O)NCC1CCCCC1NC(=O)C(C1CCOCC1)F c1(COC)cc(C(N2CC=CC2C(N2CC(NC(=O)C3CC3)C2)=O)=O)no1 C1(OC)CCCC(CNC(=O)C(CN(C)C)NC(c2cn[nH]c2)=O)C1 Cc1ccc(CC(=O)NC(C)CCCNC(c2ccc(Cl)nc2O)=O)cc1Cl C1(CNC(C2=NOC(C)C2)=O)CN(C(=O)CSc2cnn(C)c2)CC2(CCC2)O1 C1(C(N(C2CCN(C(=O)Cc3cc[nH]c3)C2)CC)=O)CC2C=CC1CCC2 C12(C(N(C3CCOC3)CC)=O)CC1CN(C(=O)CCc1cnoc1)C2 C1(NC(c2scnc2C(F)F)=O)CCN(C(C2CC2F)=O)CC12CCC2 C1(NC(CC2C(C)(C)C2)=O)C(C)(C)C(NC(c2ccc(C3CC3)cc2)=O)C1(C)C N1(CCN(C(c2ncc(Br)s2)C(=O)NCCC#N)C)CC(=O)Nc2ccccc21 C1(NC(CCCCOC)=O)CN(C(C2SCCCS2)=O)C2CCCCC12 N1(CC2C(C)CCN(C(=O)OC(C)(C)C)C2)CCOCC(C)(CCS(=O)(=O)NC)C1 N1(C(CCC(C(C)C)NC(C2C(C(C)C)C2)=O)=O)C2CCCC1CN(C)C2 Cc1ncc(C(N2CC(CCNC(C3CC3F)=O)C2)=O)c(C)n1 CC1CC(C)(C(=O)NC2CC(CNC(c3nc(Cl)c(=O)[nH]c3N)=O)C2)CC(C)O1 C1(C(=O)NCC)CCN(C(c2ccncc2F)C(=O)NCCCF)CC1 c1(C(N2CCC(N(C(C=NOC)=O)CCO)CC2)=O)c(C)n(C)c2ccccc12 Cc1cccc2c1ccn2CC(N1CCC(CNC(=O)COCCOCCO)C1)=O c1(OC)cnc(F)cc1C(=O)NCC1CC(NC(c2cc(C)ccc2O)=O)C1 c1(C(=O)NCC2(C(F)(F)F)CC2)ccccc1C(F)(F)C(F)(F)F C#CC1(O)CCCN(C(=O)CC2CC2CNC(C2CC23CCOC3)=O)C1 C(=O)(C(C)(C)CC(F)F)NCCC1CCN(C(c2scc(C)c2C)=O)C1 c1(C(c2nnn[nH]2)(C)CC2CCC2)cc(F)ccc1C.C#CCCCN C1(NC(C(c2ccccc2)NC(=O)CC2OCCCO2)=O)COC2(CCC2)C1 C1(C(=O)NC(CNC(C(C)(C)OC(C)C)=O)C(C)C)CCC(C)C(C)C1 c1(C(=O)NCC2CCCN(C(CC3CC(=O)NC3=O)=O)C2)ncnc(O)c1Br N1(C(CN(C(=O)OC(C)(C)C)CC)=O)CC2(C1)CN(C(c1cc(Cl)ncc1O)=O)C2 O(NC(=O)C(C1CCOCC1)NC(=O)CC1CCC(=O)C1C)CC(=C)Cl c1(C(=O)NCC2N(C(C(CC)(C)C)=O)CC(OC)C2)ccc(F)c(F)c1C N1(C(C(C)n2cccn2)=O)CC(CNC(c2cc(=O)ccn2C)=O)CC(C)(C)C1 CC(C)(CC(=O)NCC1(NC(c2cc(C3(C)CC3)n[nH]2)=O)CC(F)(F)C1)C1CC1 N1(C(c2c(CC)c[nH]c2)=O)CC(CNC(C2CS(=O)(=O)C2)=O)C(O)C1 C1(C(F)(F)F)(C(=O)NCCCCN(C(C(CC)n2cncn2)=O)C)CCCCC1 N1(C(c2ccn(CC)c2C)=O)CC2(CNC(C3CC3(C)C(C)C)=O)CCC1CC2 C(=O)(N=c1[nH]ccn2ncc(Br)c12)NCc1c(C(N(C)C)=O)cccc1 N1(C(C2CCC2C(=O)OC)=O)CC(C2(NC(=O)CCCc3ccc(C)s3)CC2)C1.CCOC C1(N(C(CSCCCC)=O)CC)CCN(C(=O)C(C)C=C=C)CC1 S(=O)(=O)(c1c[nH]c(=NCCn2ncnn2)cc1C)NCC1C(CC)CCCC1 C1(NC(C=CC=CC)=O)CC(CNC(=O)Cc2ccc(O)nc2)C12CCC2 Cc1ccnnc1C(=O)NC1CN(C(c2cc[nH]n2)=O)CC1CC(C)(C)C C12(NC(CCC=C)=O)CC1CN(C(=O)C(C1CCOCC1)OCC)C2 c1(OCC)cc(Cl)ccc1NC(=O)C=CC(=O)NC(c1cncs1)C c1(C(C(=O)NCC(C)N(C)C(c2ccnnc2)=O)O)ccc(C2CC2)cc1 C1(C(N2CCC(C)(CCNC(C(c3ccnn3C)C)=O)C2)=O)CCS(=O)(=O)CC1 c1(C(N2CCC(CCNC(c3ccnc(S)c3)=O)C2)=O)ccc2cnoc2c1 N1(C(C2CC(C#C)(O)C2)=O)CC(C(N2CCC(CO)C(O)C2)=O)C(C)(C)C1 CC(O)C(C)C(=O)N1CC(CCCCNC(=O)C(=Cc2cccnc2)F)C1 CC(Cc1ccco1)C(=O)NCC1(NC(=O)CCc2nc(C3CC3)no2)CC1 CC1=C(C(=O)NC(C(=O)NCC2CCCCN2CC)C2CCCO2)CC1 N(S(=O)(=O)N(C)C)CC1CCN(C(CN(C)CCN2CCOCC2)=O)C1 C(=O)(C(C)(C=C)CCOC)NC(CCCC)CNc1ncc(C(=O)OC)cc1Cl C(CCCCC(=O)Nc1ccc(F)cc1OC1CCCN(C)C1)NC(C)=O c1(C(=O)NCC(C)OC)ccc2c(n1)CN(C(=O)C1=NOC(C)C1)CC2 c1(C(=O)NCC(CNC(CC2C(C)(C)C2)=O)O)cc(Cl)cc(Cl)c1O C1(NC(CCC=CC)=O)CC(CNC(=O)CCCN2C(=O)CCC2=O)CC1O C1(NC(CSCC=C)=O)CCC(NC(C2(COC)C=CCC2)=O)C1 N1(C(C2(F)C(C)(C)C2(C)C)=O)CCCC(C2CN(C(=O)COC(F)(F)F)C2)C1 N1(C(C2N(C(C=C(CCC)C)=O)CCC2)=O)CCCC(C)(COCC)C1 CC1CCN(C(=O)C#CC(C)(C)C)CC1CNC(c1cnn2c1CCC2)=O C(C(CC(C)C)NC(c1cnc(S)nc1)=O)NC(Cc1cn(CC)nn1)=O C(=O)(C(C)(C1CC1)OC)NC(C(=O)N(CCC(=O)OCC)C)C1CCOC1 c1(COC)ccc(C(=O)NCC(C)(F)CNC(c2n[nH]cc2C)=O)o1 S(=O)(=O)(c1ccc(N2CCC(NCC(C)C#N)C2)c(Cl)c1)N(CC)CC c1(OC)cc(C(=O)N(CC(C)O)CCNC(c2cc(C(C)C)nn2C)=O)ncn1 c1(C(N2CCC(=CCNC(=O)Cc3ccon3)CC2)=O)cc(O)cc([N+](=O)[O-])c1 CS(=O)(=O)CCC(=O)N1CCC(OCCCNC(C2OCC3CCCC23)=O)CC1 c1(N2C(C(=O)OC)CCCC2)ncnc2cc(NCCSC)c(OC)cc12 c1(NC(C2(N(C(c3c[nH]c(=NCC)s3)=O)C3CC3)CCC2)=O)cccc2c1CCC2 C12(NC(=O)CCc3cccnc3Cl)CCC1CN(C(c1cn3ccnc3s1)=O)C2 N1(C(C(C)CCN(C)C)=O)CCC(NC(C2CC23CC3)=O)CC1C N12CCCCCC(C1)NC(=O)C1(CC1)C2=O.c1(C2(F)C(C)C2)ccccc1 C1(C(N(C)Cc2cn(CC)nn2)=O)CC(O)CCN1C(C1CCCO1)=O N1(C(=O)NC(C)C(CO)N(C)C)CC(c2ccccc2)C(C)(C)C1 C=CC1(C(=O)NC2C=CCN(C(=O)CSCC)C2)CCOCC1 C1(C2CCC2)(C(N2CC(O)(C(C)NC(C3CCC(F)C3)=O)C2)=O)CC1(F)F N1(C(CSC)=O)Cc2ccccc2C1CNC(=O)C(N1C(=O)CCC1=O)C Cc1ncc2cc(C(=O)NC3CCC(CNC(=O)C(C)(C)S(C)(=O)=O)C3)ccn12 Cc1ccc(N)c(C)c1C(=O)N(C)CC1(CNC(c2cc(Cl)no2)=O)CC1 c1(C(N2CC(N(C3CC3)CC3CC3)C2)=O)ccnc2ccccc12.c1(NCC(C)N)ncc(Br)cn1.CC c1(OC)ccc(F)c(C(=O)NCCC(C)(C)NC(=O)CC2CCCC(O)C2)c1OC C(C(C)(C)CCNC(=O)CCC(C)(C)C)NC(CCNC(COC)=O)=O Cc1c(CNC(C23CCC2CN(C(c2cc(Cl)no2)=O)C3)=O)cccc1F Cc1ccc(C(C)NC(=O)NC(C2CCC3(CCC3)O2)C2CC2)c(F)c1 c1(C(=O)NCCN(C(=O)C(O)C(F)(F)F)C2CC2)cncc(F)c1C(F)(F)F c1(NC(C2CC(F)(CN3CC(CO)C4(CCC4)C3)C2)=O)ncnc2ccccc12 N1(C(CC(COC)C)=O)CCC(N(C(=O)CCc2cccc(O)n2)C)C2(CC2)C1 c1(C(N2CC(CCNC(C(CC)=CC)=O)OC(C)C2)=O)cc(CC)c(=O)n(C)c1 N1(C(C=C(C)C(C)C)=O)CC(O)(CCNC(C2(Cc3cnn[nH]3)CCC2)=O)C1 C1(C(=O)NCC(C)CNC(c2ccnc(C(F)(F)F)c2)=O)CCc2nncn2C1 CCCCC(O)C(=O)NCC(C)(Cn1cccn1)NC(=O)CCC(=O)N(C)C CCC(C)(CCO)NC(=O)C(CO)NC(=O)CC1CC(F)(F)C1 n1(CC(=C)C)nc(CCCC)nc1-c1ccn(Cc2ccc(OC)cc2)c1C c1(CC(C)C)n[nH]c(=NC(CNC(c2ccc(F)nc2)=O)C(C)C)s1 N#CC1CN(C(c2ccc(-c3nnco3)cc2)=O)CCN1c1ncnc2sccc12 c1(CCC)c(C(=O)NCCC2CCCC3CC23)nnn1CC c1(C(N2CCC(C#N)(NC(c3cncc(Cl)c3)=O)C2)=O)c(O)cccc1[N+](=O)[O-] C1(NC(C(CC2CCC2)NC(C2CCN(C)C2=O)=O)=O)CCn2cnnc2C1 C12(C(=O)OCCC3(C)CCN3)CCOCC1C2(F)F C1(C(=O)NCC2(C)CCN(C(C3C(C(=C)C)OCC3)=O)C2)C2CCCCCCC12 c1(C(N2CCC(COC)(NC(=O)C=CSC)C2)=O)c(C)nn(C)c1F C1(NC(C(=O)NCCCCNC(COCC=C)=O)C2CC2)(CSC)CCCCC1 Cc1cncc(C(N2CCCC(N(C(=O)C=CC3CCCO3)C)C2)=O)c1 C(=O)(C(C(=O)N1CCC(CCNC(=O)C(F)CC2CCC2)CC1)OC)OC C1(C(=O)NCC2(CC(=O)NCC(C#C)OC)CC2)CCC(=O)C1 n1(CC)nc(C(=O)NCC(C)(O)CNC(=O)C(C(C)C)n2ccnc2)c(C)n1 N1(C(COC2(C)CCC2)=O)Cc2ccccc2C(NC(=O)Cc2nc[nH]n2)C1 C1(C(=O)NC2C(NC(Cc3c(C)nsc3)=O)CCC2)C2CCCCC12 C(C(C(=O)NC(C)Cc1ncc(C)[nH]1)NC(=O)CNC=O)OCC CCC(CN=c1cc(NCc2ccoc2)nc[nH]1)N(C)C Cc1ccc(C(N2CCC(c3c(Cl)cccc3Cl)C2)C(=O)NC2CC2)c(F)c1C N#CC1(NCc2cnc(C(F)(F)F)s2)CCNC1 CC1CN(C(C23CC4CC2C3C4)=O)CCC1CNC(c1cncnc1)=O C1(C(=O)NC)CC(C)CN1C(=O)C(C)C.C12CCC(CC1)NC(=O)C2 C(=O)(C(C)C(C)(F)F)NC(C)CN(C)C(c1ccnc(N(C)C)c1)=O O=C(N=c1cc(Cl)cn[nH]1)c1cccc(-c2cccc3c2COCC3)n1 CC1CCC(CNC(=O)CC=CC(C)(C)C)CN1C(=O)C(=O)C(C)(C)C c1(NC(=O)NC)ccc2c(cnn2C(F)F)c1.c1(C(C)C)cc(CC2CC2)n(C)n1 c1(COC)nc(N2CCCC(CNC(=O)CC3CCCCC3O)CC2)cc(C)n1 O=S(=O)(c1cnc(Nc2c(F)cccc2Cl)c(Cl)c1)N1CCC12CC(CO)C2 CN1CC(C(=O)N(C)CC2(O)CN(C(c3csc(Cl)c3)=O)C2)C(C(F)(F)F)C1 c1(CCC(N2CCN(C(N(CC(=O)O)C)=O)CC2)=O)c[nH]c2ncccc12 Cc1cc(C(=O)NCC2CC(C)N(C(c3cccn3C)=O)C2)c(C)n1CC1CC1 Cc1cc(C(=O)NC2CCC(C)N(C(c3oc(Br)nc3C)=O)C2)cc(O)c1 c1(C(N2CC(CCNC(CCOCC)=O)(OC)C2)=O)ccc2n[nH]c(C)c2c1Cl C(=O)(C(N)CCN(C)C)N(CCC(=O)N(C1CCCC1)CC(C)C)C C1(N(C(Cn2c(C)nnn2)=O)C)CN(C(C2CC2Br)=O)CC1(C)C Cc1ccc(CNc2ccc(NCc3ccccn3)cc2F)c(C)c1 N1(C(C2CCN(C(C)=O)CC2)=O)CCN(C(c2csc(C)c2)=O)C(C(C)C)C1 C1(C)(NC(C(CCSC)NC(c2cc(CCO)on2)=O)=O)CN2CCC1CC2 C1(NC(COCC=C)=O)CC(C(=O)NCCn2ccc(=O)cc2)C1(C)C CC1(C)Cc2cc(CNC(=O)NCc3ccccc3I)ccc2O1 c1(C(=O)NC2(COC)CCCN(C(c3cc[nH]n3)=O)C2)nn2c(c1C)OCCC2 n1(CCC(N2CCN(C(C3(C)C(C)CCC3)=O)CC2)=O)cc[nH]c(=O)c1=O c1(C(N2C(C(C)NC(C(CC#C)C)=O)CCC2)=O)occ2c1CCCC2 C=C(C)CCN=c1cc[nH]cc1S(=O)(=O)N(N1CCCCC1)Cn1cc(C)cn1 c1(C(=O)NCC(CNC(c2cc(Cl)c[nH]2)=O)OC)c(F)cncc1Cl c1(C(=O)NCCOC(C(C)C)C)cccnc1Sc1ccccc1 N(C1CCc2ccc(Cl)cc21)CCS(CC1C(C)(C)CC1)(=O)=O Cc1nnc(CN(C(=O)CN(C2CC(C#N)C2)C(=O)C(F)C2CCCC2)C)o1 c1(C2C(C(=O)NC3C(CC)CCC3)C2)ccc(F)cc1F CC1=CCC(C(N2CC3CC2(CNC(=O)CCC(C)C)C3)=O)CC1 c1(C(=O)NCCN2CCN(C(C3(C)CC(=C)C3)=O)CC2=O)cccc2nonc12 CC1CN(C(=O)Cn2cc([N+](=O)[O-])cn2)CCCN1C(=O)CCC1CNC(=O)N1 c1(C(=O)NC)cccc(S(=O)(=O)NC2CC(OCc3ccc(F)cc3)C2)c1 C1(CNC(Cc2cc(C)no2)=O)CCCCN1C(c1ccnnc1)=O CCCC(C)CC(=O)N1CC=CC(NC(=O)C(=O)C(C)(C)C)C1 CCC(C)(O)C(=O)N(N1CCN(C(=O)C(F)(F)C2(OC)CCCC2)CC1)C CCS(=O)(=O)c1ccccc1CC(=O)NC1CC2CCC1N2C(c1ccoc1)=O N1(C(CC2C(C)CCC2)=O)CCC2CN(C(c3csnc3Cl)=O)C2C1 C1(CN(C(=O)CC(=O)OC(C)(C)C)C)CC(O)CN1C(c1cn(C)cn1)=O c1(C(N2CCC3(NC(CCCCNC(C)=O)=O)C(C2)C3)=O)cc(C#N)ccc1O C(CC(C(=O)NCCc1ncn(C)n1)NC(=O)C=C(C1CC1)C1CC1)OC CCCC(C)CC(=O)NCC(CC)NC(=O)C(F)CC1CCOC1 n1(CC)cc(Cl)c(C(=O)N(CC(=O)NC(CO)(CO)CO)C(C)C)n1 N1(C(c2cnn(CCC)c2)C(=O)NCCOCC)CC(C)CCC1CCO C12CN(CC3CC13)C2.O=C(CSc1ccccc1)NOCc1ccccc1 N12CCC(CC1)CC2=O.Cc1nc(SCC(=O)OC)n[nH]1.N12CC(C1)N(C)CC2=O c1(C(=O)NCC(CNC(CCc2c(C)cccn2)=O)(C)C)cc(Cl)cnc1C C(=O)(C(C)CC(F)(F)F)N1CCN(C2CCN(C(C3CC(CC)C3)=O)C2)CC1 C1(C(=O)NC2CCC(C(=O)OCC)C2)(NC(=O)C(O)O)CS(=O)(=O)C1 C1(CC(=O)NC2(NC(C3CCC(NC(N)=O)CC3)=O)CC2)SC2=NCCN2C1=O N1(C(c2c[nH]c3ccccc23)=O)CCC2(CC1)CC2C(N1CCCC(Br)C1)=O C1(C(=O)NCC2(NC(CCOCC=C)=O)CC2)(COCC)CCCC1 c1(C(C(=O)NC2CCN(C(CCSC)=O)C2)(F)F)ccccc1C(=O)C(F)(F)F C(=O)(C(Cc1cccnn1)NC(=O)NC(C)COC(C)(C)C)OCC N1(C(C=CC)=O)CCN(C(=O)C(C)N(C)C)CC1CS(C)(=O)=O O=C(C1=NOCC1)N1CCC(NC(C2CC(c3ccccc3)C2)=O)C1 c1(OC)cc(C(=O)N(C)CC2CCCCN2C(=O)C(n2ccnc2C)C)n(C)n1 N1(C(C2C(C)OCC2)=O)CC=C(CC(=O)N2CC3CC(C2)CN(C)C3)CC1 c1(COCC(=O)NCCC2CC(NC(C3CC(C(C)C)C3)=O)C2)nnc(S)n1C CN1CCC2CCC(C1)N2C(c1coc(CNC(=O)COCCN(C)C)n1)=O C1(CC(=O)NC2(CSC)CC2)CCCC1NC(C1CC=CCO1)=O C1(NC(C(CC)C(C)O)=O)CCN(C(c2ccccc2C2CC2)=O)CCC1CO c1(-c2cn(CC3N(C(C4C(c5c(C)nco5)C4)=O)CCC3)nn2)ccc(F)cc1 N1(C(C(CC(=O)OCC)(C)C)=O)CC2COCCC2(NC(c2ccco2)=O)C1 N1(Cc2c(C)n(-c3ccccc3Cl)nc2)CCNC(=O)CCCC1 N1(C(c2n(CC)nnc2)=O)CCCC(NC(C2CCCC2(F)F)=O)C(F)C1 C#CCCCCCCC(=O)N1CCCCC1C1(NC(=O)Cc2cc(C)ns2)CC1 C(C)(C)(CCCC(=O)NC1CC1c1cncs1)NC(C1C(C)(CC)C1)=O C1(CNC(C2C(=C)C2)=O)CN(C(C23COCC2C3)=O)CC1N(C)C Cc1cc(C(=O)N(C)CCOCCNC(=O)C(O)C(F)(F)F)c(N)c([N+](=O)[O-])c1 CSC=CC(=O)NCCCN(C(C1COCC1c1ccccc1)=O)C1CC1 Clc1ccc2c(c1)C(NCc1ccc3c(n1)CCC3)CCC2 CN1CCC(C)(C(N2CCC(C)(NC(c3cccc(C4CC4)c3)=O)C2)=O)CC1 N1(CC)CCN(C(=O)C(Cn2cncn2)NC(=O)CN2CC(=O)NC2=O)CC1 Cc1ccc2c(C)c(C(N3CC4CC3CN4C(=O)Cc3ccsc3)=O)[nH]c2c1 CCCCCC(C)(C)CN.C1(c2ccn(CC3C(C)CCN3C)n2)CC(C)(C)CCO1 C1(C(=O)NC23CC(F)(C2)C3)(CNC(C(C)n2ccnn2)=O)CC12CCC2 C(=O)(CCC(C)(C)CNC(c1cccc(C(C)N)n1)=O)OC N1(C(c2cc(C(F)F)no2)=O)CCC2CC12C(=O)NCc1ccncc1Cl Cc1ncncc1C(=O)N(CCCN(C(=O)C(CO)c1ccccc1)C)C c1(C(C2CC=CCC2)(C)NCC2CC3(CC3)C2)nnnn1-c1ccccc1 c1(C(=O)NCC2OCCN(c3nccc(CC#N)n3)C2)ccc2cnsc2c1 CCC(C)(C)C(O)C(=O)NCC(=O)NCC1CCN(C2CC2)C1 N1(C(C(CC)F)=O)CCN(CC2CCCN(C(=O)COC)C2)CC1 CC(C)CC(C)(C)C(c1nnnn1CC(F)F)NCc1ccccc1F N1(C(C2C(=C)C2)=O)CCCN(C(=O)CC2CC2C2CC2)CC1C Clc1cccc(CCOC2CCC(N3CCCC3)CC2)c1 CCCC(C(=O)N1CCC(C)(NC(=O)CC2CC(N(C)C)C2)CC1)C(C)C C1(C(=O)NC(CNC(C(C)NC(CC)=O)=O)CO)CCC(NC(=O)C2CC2)CC1 CCCCC(CNC(=O)CC(C)F)NC(c1ccc(F)o1)=O C1(CCOC)(NC(c2ncn(CC)n2)=O)CCN(C(=O)C(n2nccc2C)C)C1 CCCCC(CNC(C1CC2CC1C2)=O)NC(=O)C(C)(C)CC1CC1 c1(NC(C2N(C(c3ccn(C)c3)=O)CC=C2)=O)cc(F)c(Cl)nc1Cl c1(C(=O)NCCCCCNC(CCc2ncc(C)[nH]2)=O)ccccc1OC(C)C Cn1ncc2cc(C(N3CCCC(CNC(=O)CC(C)(C)O)C3)=O)sc12 C1(NC(C2C=CCN(C(C(C)c3cccs3)=O)C2)=O)CN(C)CCC1O CC(C)S(=O)(=O)C(C)C(=O)NCC(C)(CC(C)C)NC(c1cscn1)=O c1(C(=O)NCCC2(NC(C3CC=CCO3)=O)CC2)cc2c(s1)CCC2=O C1(CN=C(NCC2C(CC)C2)NC2CCCCC2)CCc2cnn(C)c2C1 c1(CCCCSC)nc(-c2cccc(C(N)=O)c2)nn1CCCCO c1(C(N(CC(CC)NC(C2(CC(F)F)CC2)=O)C)=O)nn(C)nc1Br Cc1cc(C(=O)N(C)CCn2cc(-c3cccc(Br)c3F)nn2)c(C)cn1 Cc1cc(=NCc2cc(Cl)ncc2Cl)[nH]cc1S(=O)(=O)NCC(Cl)Cl C(=O)(CCCC#CC)N(C)CC1CN(C(C(CC=C)NC(C)=O)=O)C1 N1(C(COCC(OC)OC)=O)CCCN2CCCC2C1.c12cn(nn1)CC(=O)NC2 CC(C)CC(C)C(=O)NCC(C)NC(C1CCC(=O)N1)=O c1(C(N2CC(NC(=O)COCC3CCCOC3)C(O)C2)=O)cc2c(s1)CCSC2 N1(C(=O)COC2CCCNC2)CCC12CCCOC2 c1(C(=O)NC2(COC)CCN(C(=O)C(C)OCCC(C)C)C2)cnc(O)cc1C C1(C(=O)NC(C)C(C)NC(c2cccc(C3CCC3)c2)=O)C2CC3C(C2)C13 C1(CNC(c2sc(CCC)c(CC)c2)=O)CCN(C(=O)C(C#N)CC)C12CC2 Cc1cc(C(N2CCN(C(c3n[nH]cc3Cl)=O)C3CC23)=O)c2nccn2c1 C1(NC(CC2ON=C(CC)C2)=O)CC(NC(c2[nH]cnc2C)=O)C12CCC2 C12(CNC(C3(C)CCC3)=O)CCCC1CN(C(C1CC3CC1CC3O)=O)C2 C1(NC(C=CC(CC)=CC)=O)CCOCC1NC(c1cccc(C(C)C)n1)=O Cc1ccc(Br)c(S(=O)(=O)CSc2cccc(OC3CCCC3)c2)c1Br N1(C(CN(C(CCSCC#C)=O)C2CC2)=O)CC2CCC(C1)C2C#N CC1CC(C(=O)NCc2cccc(Cl)c2)CN(C(=O)C(O)Cc2ccc(O)cc2)C1 C=CCC(CC(=O)Nc1cc(CC)ccc1C)NC(=O)C(COC)OC C(=O)(CN=c1ccc(Cl)n[nH]1)N1CC(NC(CC(CCC)CC)=O)C(F)C1 c1(C(N(C(CNC(C2C(=C)C2)=O)C)C)=O)cc(C(F)(F)F)[nH]c1C c1(CNC(C2CCc3nc[nH]c3C2)=O)ccc2c(c1)CCCC2NC(=O)CCF n1(C)nc(NC(=O)OC(C)(C)C)cc1O.C(=O)(C=CC(C)CC(=O)O)OC c1(OC)cc(C2(NC(=O)COCc3ccncc3)CCC2)ccc1F c1(C(=O)NCCCN(C(C2(C(C)C)C(C(=O)OC)C2)=O)C)c(Cl)cncc1Cl CC(O)CCCCCC(=O)NCC1CC2(CO1)CN(C(c1ncccc1N)=O)C2 C12(C(=O)NCC(CSC)OC)CC(CN(C(=O)CC3CCCCN3C)C1)C2 C1(C(=O)NCC(C)F)(NC(CC2CC(=C)C2)=O)CCC(C)(C)C1 c1(C(=O)NCC2CC(NC(C(C(C)O)(F)F)=O)C2)cc2cc([N+](=O)[O-])ccc2o1 C(=O)(C(C)(CCF)c1ccccc1)N1C(C(c2ccccc2)C)CCC1 O=C(CCC(CF)CF)NC1(C(=O)NCC2CC23CCOC3)CC(O)C1 C1(C(=O)NC2(C(C)C)CC2)CC(NC(=O)CC2CCCSC2)CCO1 Fc1ccc(C(CCc2ccc(Cl)cc2)NCc2noc(C3CCCC3)n2)cc1 CC12CN(C(C3(C#N)CC3)=O)CC1(C)CN(C(c1ccc3oc(O)nc3n1)=O)C2 CS(=O)(=O)c1ccsc1C(=O)NCC1CCCCN(C(=O)C(F)F)C1 C(=O)(CC(C)CC(=O)O)N1CCCC(CNC(C2CC3(C(OC)CC3)C2)=O)C1 c1(C(N2CC=CC(NC(C34CC3CCC4(F)F)=O)C2)=O)ccc2nnn(O)c2c1 O=C1COc2ccc(-c3cscc3C(=O)Nc3ccc(Cl)cc3Br)cc2N1 C(=O)(CCCC(=O)NC(C)(CSC)C(=O)NCCC1CCCNC1=O)OC N1(C(C(CC)NC(N)=O)=O)CCN(C(=O)C2=COCCO2)C(COC)C1 c1(NCC(c2cccnc2)C)ccc(-c2cccnc2)s1 c1(C(N)=O)ccc(C(=O)NCC2(CN=c3[nH]nco3)CCC2)cc1 c1(C(=O)NC2C(NC(C3N(CCC)CCC3)=O)COC2)ccccc1SC C1(C#N)(C(C(=O)NCCC)N(C(=O)OC(C)(C)C)C(C)C)CCOCC1 Cc1cc(Br)ccc1-n1nc(C(=O)OCCC23CCC(C)(C2)OC3)cc1C Cc1cccc(C(C)NC(C2(CCNC(c3ccnn3CCF)=O)CC2)=O)n1 c1(OC)cccc(C(=O)NCC2CC2CNC(=O)CCc2cnco2)c1O C1(O)(CCNC(=O)CC2CCOC2)CCCN(C(C2CCC3(CC2)CC3)=O)C1 CC1CC2(CC(C(=O)NC3(C(=O)NCCS(N)(=O)=O)CCOCC3)C2)C1 CC1CC=C(C(=O)NC2CC=C(C(=O)NCC(C)C(F)(F)F)C2)CC1 c1(OC)cccc(Cl)c1CC(=O)NCC1(C)CCCN1C(c1n[nH]c(C2CC2)n1)=O c1(CC)ccc(C(=O)NCC2CCN2C(C2(C(C)(C)OC)CC2)=O)[nH]1 C(=O)(C#CC1CCOCC1)N1CC2=C(CN(C(C3C(C)(C)CCC3)=O)C2)C1 C12C(C)CCCN1C(=O)CCCOC(=O)C2.c1(OC)cccc(OC)c1.C(CSC)O C(=O)(CC(C)C(=O)N(CC(C)CNC(=O)C(C)(C)c1csc(C)c1)C)OCC CC1CCCCC1(CNC(c1nncs1)=O)NC(=O)Cc1cnccn1 C1(NC(CC)=O)CCN(C(=O)Cc2nc(-c3ccccc3Cl)oc2C)C1C N1(C(C=C2CCC(C)C2)=O)CCC2(NC(c3cncc(C4CC4)n3)=O)CCCC12 C12(NC(C=Cc3c(C)ccs3)=O)CCN(C(=O)C(c3ccccc3)F)CC1C2 c1(CC)ncc(C(=O)NC2(COC)CN(C(=O)CCOC3CCCC3)C2)c(C)n1 Nc1ccc(F)c(F)c1C(N1CCN(C(C2CCCS2)=O)C(C2CC2)C1)=O N1(C(CCc2cnc(C)o2)=O)CCC2(CC2)CC1C(=O)Nc1conc1C N1(C(C2CCC(=O)N2)=O)CCC2(CCC(C(N3CCOC4CC34)=O)CC2)CC1 N1(C(Cc2c(C)non2)=O)CCN(C(C2CCCC(C)(C)C2)=O)C(c2cn[nH]c2)C1 CN1CCC(NC(C2CCCC2C(=O)Nc2ccc(CO)nc2)=O)(CO)C1 C(CC(C(C)C)NC(=O)C=C1CCC(C)C1)N(C(C(CC)SC)=O)C C(c1ccncc1)=CC(=O)NCC(C)(CO)NC(c1ccnnc1S)=O N1(C(c2csc(Br)n2)=O)CC2CCC1C(CNC(C1(CC3CC3)CC1)=O)C2 C12(NC(CC3C(C)CC3)=O)COCCC1CN(C(c1cc(C(F)F)ncn1)=O)C2 C1(NC(C(C)(C)O)=O)CN(c2nccc(-c3ccccc3F)n2)CC1(F)F C1(NC(C2(C(C)NC(c3cc4ccccn4n3)=O)CC2)=O)CN(C)CCN(C)C1 C(CC(C(=O)NCc1cccnn1)NC(=O)C=CC1CCCN1C)OC N1(C(CC2CC(=C)C2)=O)CC(NC(=O)CCc2cc(F)ccc2Br)CC(O)C1 c1(C(N(CCCNC(C2CCC2(F)F)=O)C2CC2)=O)n[nH]c2c1COC2 Cc1cnc(C(N2CC(CNC(c3nccnc3-n3ccnc3)=O)C(C)C2)=O)nc1 Cc1ncnc(C(=O)NCC2CCN(C(C3C(C)(C)C3(F)F)=O)CC2)c1C CC(C)(CC(=O)N1CCCC(C)(NC(=O)COCCO)C1)CC(F)F N1(C(C2N(C(c3cc(CC)[nH]n3)=O)CC(OC)C2)=O)CCC2CCN(C)CC12 CCC(C)CC(C(=O)NCCC(C)(C)COC)NC(=O)C1=C(Cl)CCC1 N1(C(COC(C)(C)C)=O)CCC12CN(C(c1c(Br)cnn1C)=O)C2 CCC(CC(=O)N1CC(NC(=O)Cc2ccn(C(C)C)n2)C2(CC2)C1)C(C)(C)C C1(NC(CSCC)=O)CCS(=O)(=O)C12CN(C(=O)C=C1CCSCC1)C2 Cc1ncc2ccccc2c1C(=O)NCC1(NC(=O)CCC(C)(C)C)CCCC1 c1(CCCC(=O)NCCCNC(C(C)C(F)F)=O)nc2ccccc2[nH]1 N1(C(C(C)SC(C)C)=O)CC(NC(=O)C(C)OC(C)(C)C)C(S(C)(=O)=O)C1 c1(CC)ccncc1C(=O)NC(C1CCCN(C(c2cc(Cl)cnn2)=O)C1)C C(CC(C)C)(C(=O)NCC(F)CNC(c1cccc(F)c1Cl)=O)NC(C)=O C(C)(C)(C(C)NC(c1cn(C2CCCC2)nn1)=O)NC(C(C)O)=O c1(C(=O)NC2CC(NC(CC3CC(SC)C3)=O)C2)ccc(SC2CC2)cc1 c1(C(C)=O)ccc(C(=O)NCC2CCC2NC(=O)CC2CCC(=O)N2)o1 C1(NC2(c3n(CC(=C)C)nnn3)COC2)CC(C(=O)OC)C12CCC2 C1(CCc2cn(CCC(C)C)nn2)CN(C(=O)C#CCc2ccccc2)CCO1 c1(OC)ccc(OC)c(CNC(C2CCC(n3cc(C4CC4(Cl)Cl)nn3)C2)=O)c1 c1(C(=O)NC2CCCC(CC(=O)NCc3ccnc(F)c3)C2)c(O)cccc1F C(CN=c1[nH]cnc2c(Br)nn(C)c12)C1CCC(NC(C(CCCCC)O)=O)C1 c1(N2C(C)C(NC(c3cc(Cl)ccn3)=O)CCC2)nc2c(cc1C#N)CCOC2 Cc1cc(CN2CCC(C#N)(NC(C3CCN(S(C)(=O)=O)CC3)=O)C2)cc(Br)c1 N1(CC(=O)NCc2cccc(C#N)c2)CCC2(CC1)CSC2 N(C1CCCn2ccnc21)C(c1c(CNC(C(CO)OC)=O)nccc1)=O CC1CC(C(=O)NC(CO)C2(C)CC2)CN(Cc2ccc(C(=O)O)cc2)C1 c1(C(=O)NCC2(NC(C(C=CCCC)O)=O)CC2)c(F)cc(F)c(O)c1F c1(CC2C(C(=O)Nc3cscc3Br)C2)ccnc(Br)c1 C1(N(C)C)C2CN(C(=O)C(C3CC3)N(c3cccnc3)C)CC12.O=C1CCN1 C(=O)(CC(C)(C)CC(=O)OC)NC(CN(C(c1ccc(C#C)cc1F)=O)C)C CC(F)(F)CCC(=O)NC1CS(=O)(=O)CC1NC(=O)COc1ccc(Cl)nc1 c1(OCC)ncc(C(=O)NCC2CC(NC(C3CC3[N+](=O)[O-])=O)C2)cn1 Cc1cc(C(=O)NCC(C)NC(C2CC2c2ccccc2)=O)nnc1C C(CC(C)(C)CC(=O)N1CCC(C)(NC(=O)C(C)(C)C(F)(F)F)C1)OC CC1(C(=O)NCCCOCCNC(=O)CC2C=CCCC2)CC2(CCC2)C1 CC(C)C(C(=O)N1CCC1CNC(c1cncc(Cl)c1)=O)NC(c1cccs1)=O CCCCC(O)C(=O)NC1CC2C1CCN2C(c1cnc(SC)nc1OC)=O C1(NC(=O)CCC2CC(F)(F)C2)CC2CC(C1)N(C(C13CCCC(C1)OC3)=O)C2 CN1CCN(c2ccccn2)CC1.C12CN(C1)CCCN2C(C1CCC1)=O Cc1c(C(=O)NC(C2CCCCN2C(=O)COCCOC)C)nn(C)c1N N1(C(CSCCC)=O)CCCC1C1CCCN1C(c1cnc2c(cnn2C)c1)=O c1(C(=O)NCC(C)N(C)C(c2cnc(C(F)F)s2)=O)coc(Cl)c1 Cc1noc(Cl)c1CCC(=O)NC(C)CC1CN(C(c2cnn(C(C)C)c2)=O)C1 C(C1=CCCN(C(C2(C3CCCC4CC34)CC2)=O)C1)NC1CC(OC)C1 c1(OC)ccc(-c2c(Br)n[nH]c2NC(N2CCN(CC3CCSC3)CC2)=O)cc1 Cn1cc(Cl)cc1NC(N1CCN(CCCNC(=O)Cn2cncn2)CC1)=O c1(-c2cccc(C#C)c2)ccc2[nH]cc(C(=O)Nc3ccc(OC)c(F)c3)c2c1 Cc1cc(C(=O)N(CCNC(=O)CC(C)(F)F)CC)cnc1OC(F)F c1(C(=O)NCCC(C(=O)NCCC(C)N2CCCC2)O)ccc2cc[nH]c2c1 CC1CN2CCN1CC2C(=O)NCC(CNC(c1nnn(C)c1N)=O)C(F)(F)F C1(C(N(CCCC(=O)NCC(c2ccco2)O)C)=O)CCCC(O)C1 c1(C(N(C2CC(F)CN(C(c3cncn3C)=O)C2)C)=O)cc2cccnn2c1 CCC1=C(C(=O)NC(CC(=O)NCC(c2ccsc2)O)C(F)(F)F)CCCO1 N1(C(C(C)C(C)(C)C)=O)CC(C)(C)OCC1CNC(=O)CCC1CCCCCC1 C1(C(=O)NC2CN(C(=O)C(C)(C)COC(C)C)CC2C)(OC)CCC(F)(F)CC1 Cc1cnn(C)c1C(=O)N(C)C(C1CCCCN1C(=O)CCCC1CCC1)N C1(CCNC(C(C2CCOC2)OCC)=O)CCN(C(=O)Cc2ncc(C)s2)CC1 N1(C(C(CCC)O)=O)CC(CNC(c2cc(NC)ccc2Cl)=O)C(F)(F)C1 CC1CC(NC(c2nn(C)c(Cl)c2Cl)=O)CN(C(c2scnc2C(C)(C)C)=O)C1 c1(OC)nc2c([nH]1)CCCC2.C12CCCN(C(=O)OC(C)(C)C)C1OC2=O Cc1cnc2n1CCC(C(=O)NC1CCN(C(c3n[nH]cc3F)=O)C1)C2 c1(C(=O)OC)cccnc1NC1C2CN(C(=O)C(N)=O)CC12.C(C)(C(F)(F)F)O C1(C(N(CCOCCNC(C2CC(C)(C(C)C)C2)=O)C)=O)CC2CC(=O)C1O2 CC1CCC(NC(=O)C=CC2CC2)CN1C(c1ccc(-c2ccsc2)s1)=O c1(C(C)C(=O)N(CCO)Cc2nc(C(F)(F)F)n[nH]2)cccc(C#N)c1 CC1CN(C(C2CCC(NC3CCCC3)CC2)=O)CCN1C(C1CCS1(=O)=O)=O C=CC1OCCC1C(N1CCC1CC(=O)NC(CC)CCOC)=O C(C(C)(C)CC(=O)NC1CCC(C)(CNC(=O)C2=NOCC2)C1)N(C)C C12(NC(c3c(C)coc3)=O)CCN(C(c3cccc(SC(F)(F)F)c3)=O)CC1C2 c1(C(=O)NC2CCCN(C(C3CC(=O)NC3)=O)C2)ccnc(O)c1F c1(C(N2C(CNC(C(C)OCCN(C)C)=O)CCC2)=O)cc(N)cc(O)n1 c1(SCC(N2C(C)CCC(N(C)C(=O)NC3CC3)C2)=O)cc(C(F)(F)F)ccc1O CCC(C)(O)C(=O)N1CCC(NC(c2ccnc(N3CCOCC3)n2)=O)C1 C1(C2CCN(C(=O)C(F)C(F)(F)F)CC2)(NC(Cc2cnc(C)[nH]2)=O)CC1 C1(C#N)(C(=O)NCC(CNC(c2n(CC(C)C)ncc2)=O)O)CC2(CC2)C1 C1(NC(CCOCC)=O)CCN(C(c2cncc(Cl)c2)=O)C1c1cccnc1 c1(CCC(=O)NC(C)C(C)(C)NC(C2CC3C=CC2C3)=O)ccc2c(c1)OCO2 CC(C)C(O)CC(=O)NCC(CNC(=O)CSCC(N)=O)CO C1(F)(CNC(COCCC#C)=O)CC(NC(=O)CC2(C)OCCO2)C1 C(=O)(C1=C(C)S(=O)(=O)CC1)NCC1(C)CCC(NC(C=CCC)=O)CC1 N1(C(c2c(C)ccc(OC)n2)=O)CC2CCN(C(c3nc(C)nn3C)=O)CC2C1 c1(C(N2CCN(C(=O)COCC3CC3)CC2CC2CC2)=O)ccc2occc2c1 C1(CC=C)(NC(C2CCCCN2CCC)=O)CCN(C(=O)C=CCCC)C1 C1(C)(CC)CC(NC(C23CC(F)(C2)C3)=O)CN1C(c1ccc(C#N)cc1)=O c1(SC(c2cc(Cl)c[nH]2)=O)ccncc1Nc1ccc(CO)cc1 Cc1cc(Br)cc(CNCC2(OC(C)C)CCOC2)c1O c1(C(N2CCC(CC(N3CCCC(C(=O)OC)C3)=O)CC2)=O)c(I)ccnc1Cl CC1(C)CCCCC(CNC(=O)NC(C(=O)OC(C)(C)C)(C)CO)C1 C(CCC(F)(F)F)N(C(CC1(NC(C(C)c2ccco2)=O)CCCCC1)=O)C Cc1ccc(CC(=O)NCCCN(C(C2CCN(C)C2)=O)C2CC2)c(Cl)c1 Cc1ccc(F)c(C(N2CCN(CC(=O)Nc3nc4c(s3)CCC4)CC2)C)c1 CCCC(C(=O)NC1COCCC1NC(c1ccc2nonc2c1)=O)P(C)(C)=O C1(CNC(c2cccc(CO)c2)=O)CC12CCN(C(=O)CNS(N)(=O)=O)CC2 CC1CN(C(c2csc(Cl)n2)C(=O)NC2CC2)C=CC1C(=O)Nc1ccccc1 C1(OC)CC2CC(NC(=O)CC(COC)NC(=O)C#CC3CC3)CC12 n1(C(c2ccccc2)(F)F)ccc(=NC(c2ccc(Cl)c(F)c2)C2CC2)[nH]1 C1(C(=O)NCCCC(C)NC(=O)CCOc2ccccc2)CCC(N(C)C)CC1 CCC(CC(=O)N1CCC(CCO)C1)N(C(=O)CC1CCCC2CC12)C N12CC(C)OC3(CCN(C3)CC(=O)N(C)CC1=O)C2.c1(NC(C)=O)ccccc1 C=C(F)C1(CC(=O)NCc2ccc(C(N3CCC3C(=O)OC)=O)s2)CCC1 C1(C(=O)NC(CCN(C(C=C(CCC)C)=O)C)C)CCCC(F)(F)C1 N1(C(C2(CC)CCNC2=O)=O)CCOCC(NC(=O)C(C)SC(F)(F)F)C1 c1(C(=O)NCCC2(O)CCN(C(CC(CC)OC)=O)C2)cc2c(Cl)cncc2s1 C1(CC(=O)NCCC(=O)NCC)C(NC(c2nccn2C)=O)CC1O c1(NCc2ccc(C)c(C)c2)ncnc2c1CCCC2 CS(=O)(=O)c1sccc1C(=O)NCC1(NC(=O)CC2CCOC2=O)CCC1 Nc1c(Cl)cnc(C(N2CCN(C(=O)CCCC(F)(F)F)CC2CCO)=O)c1Cl N1(Cc2ccc(OCC=C)cc2)CCC(O)C(C(=O)Nc2cnn(CCF)c2)C1 c1(C(N2CCC(NC(c3c(C)nc[nH]3)=O)C(F)C2)=O)cnc2cc[nH]c2c1 N1(C(CCN(C(=O)CCc2ccccn2)CC=C)=O)CCCC2NC(=O)CC12 CCCCCCCCCCCC(=O)N(C)CCN(C)C(C1CC2(CC(=O)N2)C1)=O c1(C(=O)NC2CCC(N(C(c3cnc(CCC)s3)=O)C)C2)cc(Cl)ncc1N Cc1ccc(C=CC(=O)NCC(C)(CO)NC(=O)C(N2CCSCC2)C)c(C)c1 CC(C)(CS(N)(=O)=O)C(=O)NC1CCCN(c2ccnc(Cl)n2)CC1 CCCC(CNC(=O)C(C1CCCCC1)=O)C(=O)NCc1ncc(C)o1 c1(CC)ccc(C(=O)NC2CC2CNC(c2cn(C)nc2CC)=O)c(F)c1 CC1CN(C(=O)Cn2nnc(-c3ccsc3)n2)CC1NC(=O)Cc1cncnc1 C(=O)(C1=CCCCO1)NC1CC(C(C)NC(c2n[nH]c(C3CC3)n2)=O)C1 Cc1ncnc(O)c1C(N1CCCN(Cc2ccccc2)CC1)C1COC(C)C1 C(=O)(CCC(N)=O)N(C(CNC(CN)=O)C)C.C(C=O)N(C(C)=O)C C1(NC(=O)CC2CCCC2NC(=O)Cc2ccc(O)nc2)CC2CC3C(C2)C13 CCCC(C#N)C(=O)NCCC(O)CCOC.C1(C)(CO)C(=O)N1 N12CC3=C(C(=NC(=O)c4csc1n4)NN3)C2.S(=O)(=O)(C1CCCCC1)S(CC)(=O)=O C1(CNC(=O)CCSC2CC2)COCCN1C(C1(F)CC1c1ccccc1)=O C12(C=O)CCC(C(=O)O)(CC1)CC2.C1(SCNC)CNC2(CCC2)C1 C(CN=c1[nH]c(=NCCCN2CCCOCC2)[nH]c2c1CCC2)(C(C)C)OC Cc1c(CCNC(C2CCN(C(c3ccoc3)=O)C2C)=O)cnn1C N1(C(CCOC)=O)CCOCC1C(=O)NCCc1ccc(F)nc1 C#CCC(C)(C)C(=O)N1CC(OCCC(=O)N2CC(c3nn[nH]n3)C2)C1 N1(c2ncnc(C)c2C#N)CCC2CCCC12CNC(=O)C(C1CCCCC1)O C1(NC(COCCOCC)=O)CCCC(N(C)C(c2cccc(F)c2)=O)C1 c1(C(C)C)ccc(F)c(C(=O)NC(C)CCCNC(C2(CO)CCOC2)=O)c1 c1(OC(C)C)cncc(C(=O)N(C2CCCCC2N(C(=O)C(C)CO)C)C)c1 c1(CC)nn(C)cc1C(=O)NC1(CN(C(=O)Cc2ccc(OCF)nc2)C)CC1 C=CCCC(F)(F)C(=O)NC1CN(C(=O)C(C)C2(O)CC2)CC1c1ccnn1C C1(CNC(C(C)NC(=O)NC)=O)CN(C)CCN1C(C1CC1C(C)O)=O C12(NC(CC=C)=O)CCCCCC1N(C(=O)CCC1CCCO1)CC2 C1(NC(C(CC#C)C2CC2)=O)CN(C(c2ccc(Cl)c(OC)c2)=O)C(C)(C)C1 C1(NC(c2ccc(C)s2)=O)CCC(C)N(Cc2snnc2C)C1 N1(C(CSCCOC)=O)CCC(C)N(C(C2CC(=O)N(CC(F)(F)F)C2)=O)CC1 N1(C(c2n[nH]c(C)c2C)=O)CCC2(NC(C3CC3C3CCCC3)=O)CCCC12 C1(NC(CC(C)C2CC2)=O)CCCN(C(c2csc(C(C)(F)F)n2)=O)C1 N1(C(c2ccc(OC)c(F)c2)=O)CC2(CC1CNC(=O)CCC(N)=O)CC2(F)F c1(C(=O)NCC2(C)CCN(C(C3(COC)CCC3)=O)CC2)cccc2ccsc12 c1(C(N2C(C)C(NC(=O)CCc3cnc[nH]3)CC2)=O)cc2ccnn2cn1 c1(C(N(C)Cc2nc(O)n[nH]2)=O)cc(Br)cc(Cl)c1O C#Cc1cnn(C)c1C(=O)NCC1CC1CNC(=O)Cc1ccc(F)cc1F C1(NC(C(N2C(=O)CCC2=O)CC)=O)CC(C)N(Cc2ccccc2)C1 CCC(C)C(=O)C(=O)NC1CN(C(=O)C(C)OC(C)(C)CC)CC1CC C1(NC(c2cc(=N)[nH]cc2)=O)CC2CC(NC(c3cc(Br)no3)=O)C2C1 N1(C(=O)CO)CCC(n2cc(COc3cncc(Br)c3)nn2)CC1 CON1CCC(C(=O)N(C2CCCCC2N(C(=O)Cc2n[nH]c(=N)s2)C)C)CC1 N(C1c2cccc(F)c2CCC1C)C(=O)NCc1cc(SC)c([N+](=O)[O-])cc1 N1(C(CC2CC(=O)NC2=O)=O)CCCN(CCNC(c2ccc(F)s2)=O)CC1 N1(C(CC)=O)C2CC=C(C(=O)NC3CCC3O)C1CC2 CS(=O)(=O)C1CCCCC1NC(=O)Nc1ccc(O)c(Cl)c1 c1(C(N(CC(CC)NC(c2c(CO)noc2C)=O)C)=O)cncc(C(C)(C)C)c1 c1(NC(N2CCC(c3nocn3)C2)=O)nccc2cc[nH]c12 C(C1CCCCC1)=CC(=O)N(CCCNC(C1CCOC1)=O)C1CC1 Cc1cc(COC(C2CCCN2NC(C)C)=O)ccc1F.c1(=O)c(=O)[nH]1 C1(CN(C(C(C)C)c2cncs2)C(C2CCCN2)=O)CCCC2CCCCC12 CCCC(C#N)C(=O)NC1(CNC(c2ccc(-c3sccc3C)s2)=O)CC1 C12(C(N3CCCC(F)(CNC(c4csc(Cl)n4)=O)C3)=O)CCC(CO)(CC1)CC2 c1(C(=O)NCC2(F)CN(C(C=CC)=O)C2)cnn(-c2cccc(SC)c2)c1C C(C)(CC(=O)N1CCC1C(=O)OC)OCCCC.C1(C)C(=O)N1 c1(NC(c2n(CCSC)nnn2)c2nccs2)cccc(S(=O)(=O)C(F)(F)F)c1 c1(C(N2C(C)CCN(C(C3CCCCS3)=O)CC2)=O)cnn2c(N)ccnc12 c1(C(C)NC(=O)NCc2cnnn2-c2ccccc2)ccc(Cl)c(Cl)c1Cl C1(CC(=O)Nc2nccc(C(N(C)CCC(=O)N)=O)c2)CC2CCC1CC2.C1(C)CC1 C=CCC(C(=O)Nc1ccco1)NCC1CN(c2ccccc2)C(=O)O1 CC(C)C(C(=O)N(C)CC1CCCN(C)C1)NC(c1ccncc1Cl)=O c1(NC(C=CC(C)NC(C2(SC)CC2)=O)=O)cc(C#N)ccc1O c1(C(=O)NC2CCN(C(C(C)OC)=O)C23CC3)cc2ccccc2cn1 c1(C(=O)NCC(CN(C(c2cc(C)sn2)=O)C)(C)C)cc(C)n(C(C)C2CC2)n1 C1(OCc2scc(CC(=O)OCCCCOC)n2)CCCC(C)C1 c1(CNC(C)CC2(O)CCCC(C)(C)C2)n[nH]c2c1CCCCC2 Fc1ccc(N=c2scc(-c3ccoc3)n2CCOc2cccc(Cl)c2)cc1Cl N1(C(CCCOC(C(C)C)=O)=O)CCC2C1CCCN2C(C1C=CCCC1)=O c1(C(=O)NC(CNC(=O)Cc2cnc[nH]2)C2CC2)cc(C(F)(F)F)c[nH]1 N1(CC(=O)NCC2CN(C(C3CCC=CCC3)=O)CCCO2)CCCCCC1=O c1(CCC(=O)NCC(C2OCCN(C(CC)=O)C2)C2CC2)ccc(N)c(F)c1 c1(-c2scc(NCCC(C)C)c2)ccnc(-c2ccn(C(C)C)n2)c1 Cc1ccc(C)c(CN2CCC(NC(c3c(Cl)cncc3Cl)=O)C(O)C2)c1O C1(NC(c2c(C)csn2)=O)CCCC(C(=O)NCc2c(C)cncc2C)CC1 N1(C(Cc2c(C)nsc2)=O)CCC(C2CC2)(CNC(=O)Cc2ncoc2C)C1 C(=O)(CCN=C(NC1CN2CCCN1CC2)N1CCCC(C)C1)NC CC1(C)CN(C(=O)CC23COCC(C2)C3)CC1NC(c1ccc(Cl)c(O)c1)=O N1(C(CCc2cn(C)nn2)=O)CC2(CCC2)CC1C(=O)NCC1NC(=O)NC1=O c1(C(c2nnnn2CC2CC2)NCc2snc(CC)n2)ccnc(Cl)c1F c1(CC(=O)N(CC(N(C(=O)CCCN(C)C)C)C2CC2)C2CC2)ccc2[nH]ccc2c1 C1(C(N2CCC(CN(C)C(c3cscc3C#N)=O)CC2)=O)CC(=O)C12CCCC2 Cc1nnc(CCC(=O)NC2C(CNC(C3CN(C(C)C)CCO3)=O)C2)n1C c1(NC2CC(C)NC(=O)C2)cc(Br)ccc1S(=O)(=O)N1CC2CSCC(C2)C1 c1(N(C)CC2CCCCN2C(C2CC2C2CCCC2)=O)ncnc2c1CCC2 C=CC(C)(C)CC(=O)N(C1CCN(C(c2cn(C)nc2Cl)=O)CC1)CC c1(C(N2CCC(CC#C)C2)=O)ccc(C)c(OCN)c1.C1(N)CCOCC1 c1(C(=O)NC(CCOC)CNC(=O)C(C)(O)C2CCC2)ccc(C#N)c(F)c1 C1(C(=O)OC(C)(C)C)(C(F)F)CCCN(C(C(c2ccccc2Cl)C(=O)OC)=O)C1 CC#CCC(C(=O)NC1(C(O)COC)CC1)NC(=O)Cc1cncn1C CC1CC(C)N(C(=O)CNC(=O)CC(F)(F)F)CCN1C(=O)C=Cc1cn(C)nn1 C1(CNC(C(=O)NCc2c(C)ccc(Br)c2)=O)COC2(COC2)C1 CC1CC(C(=O)N(C)CC2CCC(CNC(c3cccc[n+]3[O-])=O)CC2)CCO1 S(=O)(=O)(c1ccc(-c2nccs2)cc1)N1CCC(COC)C1 c1(N2CCC(NC(c3c(CCC)n[nH]c3)=O)C(C)C2)ncnc2ccc(Cl)cc12 c1(C(=O)NC(CCC)C(=O)NCC2CCC(CO)CC2)cc([N+](=O)[O-])c[nH]1 c1(C(N2CCN(C(C(C(=O)OC)C)=O)C3(C2)CC3)=O)cn2ccc(CO)cc2n1 CC1(C(N)=O)CCN(C(=O)CC2CCN(C(=O)Cc3ccon3)C2)C1 c1(OC)ccc(C=CC(N2CC3CC2CN3C(=O)C=CCF)=O)c(OC)c1 CC(C)(C)CC(O)CC(=O)NC(C(=O)Nc1ccc(F)c(C#N)c1)C1CCOC1 C1(n2cc(-c3n(C)c(S)nn3)nn2)CC2(CCCCC2)CO1 CC(C)C(C)CNC(C1CCCN1C(=O)C=CC1CCC1)=O C1(CC(=O)N(CC(C)(C)CNC(c2coc(C)c2)=O)CC)CCC2(CCC2)O1 Cn1nc(-c2ccco2)cc1NC(c1sc(Br)cc1Cl)=O C(=O)(C1=COCCO1)NCC1(OC)CCN(C(=O)C(C)c2ccco2)C1 N1(C(c2ccc(N(C)C)cc2)=O)CC(CNC(=O)Cn2ncnn2)C2(CC2)C1 CC1CCc2ccccc2CN1C(=O)C(N1CCC(C(=O)Nc2nccs2)CC1)=O C1(NC(C2(CNC(CN(C3CCC3)C)=O)CC(C)(C)C2)=O)C=CC(C)(C)CC1 C(CCC)(C(=O)NC(C1CCN(c2nc(CCOCC)ns2)CC1)C)=CCC C#CCC(CC#C)C(=O)NC(CN(C(=O)C=C1CCOCC1)CC)CC Cn1ccc(C(=O)NCCOCCNC(c2csc(CO)n2)=O)c1 C12(NC(CCCC(=O)NCC)=O)CCCCC1N(C(=O)CC1CCC(=O)N1)CC2 CCC(CNC(C1CC(=C2CC2)C1)=O)NC(=O)CSc1cn[nH]c1 CC1CCCC(C(N2CCCC3(C2)N=N3)=O)CC1.C1CC(=O)N1 c1(N(C2CCOCC2)C)[nH]c(=NCC2CC23CCC3)ccc1[N+](=O)[O-] C1(NC(c2c(C)sc(C(F)(F)F)n2)=O)C2CCC1N(C(=O)Cc1nc(CO)cs1)C2 c1(NC(c2cnn(C3CC3)c2)=O)cnc(C2CCC2)o1 CCCC(C)(O)CC(=O)N1CC(F)(C(=O)NCC23CCCC2CCC3)C1 S(=O)(=O)(c1ccc(C(=O)NC(=O)C(n2ccc(C)n2)C)o1)NC.C12CC1NC2 CC(CCC(=O)NC12CCN(CC1)C2)NC(C1CC(=C2CC2)C1)=O c1(N2CC(OC)OCC2)nc(NCCS(=O)(=O)C(C)C)c2ncn(C)c2n1 C(C)(CCN=c1[nH]cc(C#N)c(C(F)(F)F)c1C#N)C1c2c(C)ccnc2C1 N1(C(c2c(CC)cno2)=O)CCCC(C)(C)C1CNC(c1ccc(O)cn1)=O Cc1cc(CC(=O)NCC(CNC(C2CC(O)(C(F)F)C2)=O)CO)ccc1CO N1(C(CC(C)OC)=O)CCC(CF)(NC(c2cc(C)cnn2)=O)C1 C1(C(=O)NCC2CCCN(CC)C2)CCN(C(c2ccncc2)=O)C12CCC2 c1(C(=O)OC(c2ccccc2)C(=O)N(C)C)cn2ccnc2s1 c1(C(N2C(C)CC(NC(c3sccc3OC(F)F)=O)C2)=O)ccn2ccccc12 N1(CC2CCC(N(C)C)C2)CCCC(C2OCCO2)C1 c1(N(c2ncc3sccc3n2)Cc2c(C)nc(Cl)cc2)cc(C)c2nnc(C)n2c1 C(=O)(CC(C(F)(F)F)n1cccn1)NC1CC(C)(CNC(C(C2CC2)SC)=O)C1 C1(NC(c2scc(C)c2Cl)=O)CCC2CC1CN2C(c1ccc(C#N)[nH]1)=O c1(C(=O)NCC(C)N(C(=O)C(C)SC)CC)cn(CC)c2ccccc2c1=O CCC(C)(C)CCNC(C1CC12CC(NC(=O)Cc1ccoc1C)C2)=O c1(CCC(N2CC(NC(=O)C(C)N(C)C)CC(C)C2)=O)ccc2cnn(C)c2c1 C=CCC(CC)C(=O)N1CCC(C)(CCNC(=O)CN(C)S(N)(=O)=O)C1 C1(c2cn(C(c3ccccc3)C(CC)O)nn2)CCCN(S(=O)(=O)C(F)F)C1 c1(OC)c(C(N2CCC(O)C(NC(C3CC3F)=O)C2)=O)oc2ccccc2c1=O CCCCC(F)C(=O)NC1CC(C)(C(=O)NC(CC)C(=O)N(C)CC)C1 c1(CNC(=O)OCC)cccc2c1CCN(C(=O)CSc1ccsc1[N+](=O)[O-])C2 c1(C(N2C(C)CC(NC(c3c(CCC)n[nH]c3)=O)C2)=O)cc(C)cc(Br)c1F c1(C(=O)NC2CC(NC(C3C(C(=O)OCC)C3)=O)C2)cc(O)nc2ncn(C)c12 N1(C(CC2C(C)CCO2)=O)CCC(C(=O)NC2CN(C3CCC3)C2)C(C)(C)C1 C12(OC)CCN(CC1)C2.c1(SC(C(=O)N(CC(=O)OC)C2CC2)C)n[nH]c(=N)s1 C1(NC(C(CCC2CC2)NC(C(CC)n2cncn2)=O)=O)CCn2nccc2C1 c1(OC)ccc(O)cc1C(=O)N(C(C(N1CCC(OC)C1C)=O)C1CC1)C C1(C(N(CC(CC)NC(=O)CNC(C)=O)C)=O)CCCN1C(=O)C=CSC N1(C(C(CC)C#N)=O)CC(OC)CC(NC(=O)Cc2ccn(C3CCCC3)n2)C1 C1(N(C(CCOCCC)=O)C)CN(C(=O)CCN2CCC(F)C2)CC12CC2 N1(C(C2C(=C)C2C(=O)OC)=O)CCCC(CC(=O)N(CC)Cc2cn(C)nn2)C1 c1(NC(c2c(OC)cccc2)Cc2cccnc2)cc2ccccc2s1 Cc1ccc(C(N2CC=CCC2C(N2CC(CF)C3CC23)=O)=O)cc1F C(=O)(C(O)CC(F)(F)F)N(C)CCO.C(c1ccccc1OC(F)F)=CC(=O)NCC c1(SCC(N2CC3C(NC(C=NOC)=O)C3C2)=O)nnc2ccccn12 c1(OC)ccc(C(=O)NCCCN(C)C(c2cocc2C)=O)nn1 c1(OC)c(F)ccc(F)c1C(=O)NC1CCN(C(C2CSCCS2)=O)C(C)C1 C1(C(=O)NCC(CCOC)NC(C=C(CC)CC)=O)CCC(N=[N+]=[N-])CC1 N1(C(=O)OCC)CSCC1C(=O)NC1CCN(C(c2cc(C3CC3)[nH]n2)=O)C1 C1(CCC(=O)OC(C)(C)CCOCCNC(CCCSC)=O)CCC(=O)NC1=O c1(C(N2CC(NC(CCOC(C)C)=O)C(O)C2)=O)ccc(F)c(O)c1F C1(NC(c2c(C)[nH]nc2Cl)=O)CC2CC1N(C(c1cc(Cl)ccn1)=O)C2 N1(C(C(CC)SC)=O)CC(CNC(=O)C=Cc2ccc(OC(F)F)cc2)CC1(C)C N1(C(CCC=CC)=O)CCOC(CC(=O)NC2CC23CC(O)C3)C1 Cn1ccc2nc(N3CC(CCNC(=O)C=CCOC(C)(C)C)C3)ncc12 CC1COCC(CC(N2CC(F)(CNC(=O)Cc3ccccc3Cl)C2)=O)O1 CC(C)CC(C)(O)C(=O)N1CC2C(C(=O)Nc3ccc(CO)nc3)C2C1 N1(C(CC(C=C)(C)O)=O)CCC(C(=O)NC(c2[nH]c(C)nc2C)C)C(C)(C)C1 C(=O)(C(CSC)NC(=O)CCn1ccnn1)NCC1(C(C)(C)OC)CC1 c1(N(CCn2cc(N3C(=O)CCC3)nn2)CCN2CCOCC2)c(F)cccc1Cl c1(CC)noc(CC)c1CC(=O)NC(C1(O)CN(C(=O)COCC2CC2)C1)C CCC(CCN(C)CCC(C)COC)CC(=O)OC c1(C(=O)NCC2CCC(NC(c3c(C)n(C)cc3)=O)C2)cc2n(c1)CCCC2 CCC(C)(CNC(c1cnc(C)nc1C)=O)C(=O)N1CC2(CC(F)C2)C1 c1(C(=O)NC2C(NC(c3ccc(C(C)=O)o3)=O)CCCC2)ccnc2c1CCC2 c1(Cc2cnn(C)c2C(=O)NC(=O)NC2C3CN(CCF)CC23)cccc(F)c1F c1(-n2cc(C(CC)O)nn2)ccc(C(C)C)cc1.N12CCC(C1=O)NC(=O)C2 n1(CC)nnc(C(N2CC=CC2(C)C(N2CCC2C)=O)=O)c1C C(CC(=O)NC(c1cccnc1)C)(C(F)F)NC(C(c1ccc(C)o1)C)=O c1(C(N(CCCCCNC(C(C)(C2CC2)OC)=O)C)=O)cnc2cccc(C)n12 Cc1nnc(CC(N2CCCC(Cc3cn(C(C)C)nn3)C2)=O)n1C C1(CNC(C=C(C)Cl)=O)CCN(C(c2ccc(-c3ccccn3)o2)=O)CC1C CCC(CC(=O)N1CCCC1CCNC(c1ccc(OC)cc1)=O)SC c1(C(=O)N(c2ccccc2)CCCO)cc(C(F)(F)F)cc(C(F)(F)F)c1 CC1CC2CN(C(=O)C(O)c3ccsc3)CC2N1C(C1CC2CC2C1)=O N1(C(c2c(CC)c[nH]c2)=O)CCCC1(C)C(=O)NCC(C)(C)OC Cc1cc(C(N2CCSCC2CCNC(C2CC2CF)=O)=O)sc1C C(C)(CO)(CN=c1ccc(C(=O)N(CCCN2CCCC2)C)c[nH]1)OC C(=O)(CC1CCOc2ccccc21)NC(CCCC)CNC(=O)C(Cl)=CCl N1(C(Cc2c(CC)n[nH]c2CC)=O)CC2(CC(NC(c3cnsc3C)=O)CO2)C1 N1(C(C(CC)CNC(c2c[nH]nc2Cl)=O)=O)CCOC(C)(C2CC2)C1 C1(C(=O)OCC)CCCCN1C(=O)CC1CCCN1Cc1ncco1 C1(C(=O)OCC)CC2C(CCC(C)N2CC2C3CCCCC23)O1 CC1=NN(C)C(=O)C1CC(N1CCN(C(c2[nH]cnc2C#N)=O)C(C2CC2)C1)=O N1(C(C(C)NC(CC)=O)=O)CCCC(NC(c2cncc(C)n2)=O)C1CC c1(CCC)ccc(S(=O)(=O)NC2CCCC(Nc3ccnc4ncnn34)C2)cc1 C1(C(N(C(C)CN(C(=O)CC(=O)N(C)C)C)C)=O)CCCC(=O)C1 c1(C(N(CC(CO)(CO)NC(=O)C=Cc2cnc[nH]2)C)=O)csc([N+](=O)[O-])c1 CC1(CNC(=O)Cn2cnnc2)CC(F)(F)CN1C(c1n[nH]c2c1COC2)=O N1(C(CCC=C(C)C)=O)CCN(C)C(CNC(c2ccncc2)=O)C1 c1(CNC(=O)CNC(c2ccc(O)nn2)=O)cccc(F)n1 C1(C2CCCNC2)(C(=O)OCC(=O)NC2CC2)CC1 C1(CC)(NC(C2CC3CCC2CC3)=O)CCCN(C(=O)C(C(=O)OC)OC)C1 C1(NC(C(C2CCCC2)OC)=O)CC2(CCCCN2C(=O)CCNC(=O)CO)C1 c1(CC(=O)NC2CCC(NC(=O)Cc3cccs3)C2)cccc(OC2CCC2)c1 C1(C(=O)NC2(F)CC(NC(C(CCCC)NC(N)=O)=O)C2)Cc2nnc(C)n2C1 Cc1ccc(F)c(CNC(c2c(I)c(C)nn2C)c2nnnn2C2CCCC2)c1 Cc1cc(C(=O)NC2(C(=O)NC(CO)CCC3CC3)CCN(C)C2)cnn1 C(=O)(CC(C(=O)N1CCC(NC(=O)CCC(=O)N(C)C)C1C)N(C)C)OC c1(C(=O)NCC2(NC(C=C(C)C)=O)CC2)cccc(Br)c1CC#N C1(NC(COc2ccc(C(CC)C)cc2)=O)CCCCN(C(=O)CC(F)F)C1 CCC(C)(C#N)C(=O)NCC(O)CNC(c1nc(C)ccc1Br)=O c1(C(N2C3C(NC(c4c(C)cn(C)c4)=O)C(C3)C2)=O)ccc(F)c(C(F)(F)F)c1 CN=c1[nH]c(C(N2CCC(C)C2CNC(=O)CCOCCN(C)C)=O)cs1 c1(C(=O)NC(C=C)C2CCC2)cc(CCNC(=O)C(C2CCC2)C2CCC2)on1 N1(C(CCNC(CC(C)C)=O)=O)CCCN(C(c2ncccc2Cl)=O)CC1C c1(C)c(C)cccc1C.N12CCCC1(C)C2=O.N1(CC)CCCC1CNC CC(C)CCCC(=O)N1CCC(NC(c2cn(C(C)C)nn2)=O)C1 CCC1c2cc(Cl)cc(Cl)c2CCN1C(C1(NC(C)C)CC1)=O Cc1nn(CCO)c(C)c1C(=O)NCC(C)CN(C)C(C1COC(=O)C1)=O Cc1cc(C(=O)NC2CC(F)(CNC(c3cc(C(C)C)on3)=O)C2)c(N)cc1F N1(C(C2C(C)(CC)C2)=O)CC(C2CN(C(c3ccc(Cl)c(NC(C)=O)c3)=O)C2)C1 C1(C(=O)NC2(C3CN(C(c4occc4C4CC4)=O)C3)CC2)CCCCC12CCC2 C1(C(N2C3C(C(N(CC=C(C)C)C4CC4)=O)C(C3)C2)=O)CCCC1C1CC1 c1(NC2C(NC(c3c(NC(=O)OCC)cccc3)=O)C2)nc2ccc(I)cc2s1 C=CCN=C(NCc1cc(Cl)cn1C)N1CCC(CCC(=O)C(F)(F)F)CC1 c1(CC(COC(c2cc(C3CCC3)ns2)=O)O)ccccc1F C(=O)(CC1=CCCCC1)NCC(C1CCC1)NC(C(C(COC)C)C)=O N1(C(CCOCC#C)=O)CC(C)C(C)(CNC(c2cc[nH]n2)=O)C1 c1(NCCOc2c(C)cccc2)ccc(S(=O)(=O)NCC2CC2)c(Cl)c1 c1(C(=O)NCC2CCCC2C(F)F)cc(NC(=O)C(F)C2CC2)ccn1 N1(C(c2nn(C)c(Cl)c2Cl)=O)CCC2(NC(=O)C=CC=C(Cl)Cl)CCCC12 c1(C(C)C(=O)NCC(C)(C(C)C)NC(C2CC2C(F)(F)F)=O)cncc(F)c1 c1(C(=O)NC2C3N(C(CC(C)CF)=O)C(CC3)C2)cc(Br)cc([N+](=O)[O-])c1 N1(C(C2(OCC)CC2)=O)CCc2ncc(NC(C3CCCN3C)=O)cc2C1 c1(C(N2CCC(OCCNC(=O)Cc3cncs3)C2)=O)cncc(C(F)F)c1 c1(C(=O)NC2C(C)(CN(C(=O)CC3CC3)C)CCC2)cc(O)c2cnn(C)c2c1 N1(C(C2(CC#C)CCCCO2)=O)CCC(C)N(C(C2CC3CCC2CC3)=O)CC1 Cc1ccc(O)c(C(=O)NCC2CN(C(=O)C(O)CN(C)C)CC2C)c1 c1(C(N2C(CNC(Cc3n(CC)ccc3)=O)C=CC2)=O)cncc2ccccc12 C(=O)(C(CNC(C1(C)CC(C)(C)C1)=O)C(C)C)NC1C(CC(C)C)C1 C1(CCNC(CC2(OC)CC2)=O)CCCCN1C(c1cc(C2CC2)on1)=O C1(C)(C(N2CCCC(CNC(C(=O)NCCOC)=O)C2)=O)CC2(CCC2)C1 Cc1nc(CNC(C2(NC(=O)CCc3ccsc3)CCOCC2)=O)c(C)o1 C(=O)(C1=CN(C)S(=O)(=O)N=C1C)N1CCC(NC(C(COCC)(C)C)=O)C(C)C1 CC(C)(CC#N)C(=O)NCC1(F)CCC(CNC(c2ccccc2Cl)=O)C1 N1(C(CC(N2CCCC(C)C2)=O)=O)CCN(C(C2(C(=O)NC)CC2)=O)CC(O)C1 C12(OC)CCC(C(=O)NC3(CO)CN(C(=O)Cc4nc(C)oc4C)C3)(CC1)CC2 CCCCCCC(C)(CC)C(=O)NC(CNC(c1n[nH]cc1Br)=O)CC(C)C CC1Cc2c[nH]nc2C(C(=O)NC2CN(C(=O)C(F)(F)C(F)(F)F)C2)C1 N1(C(C2(C)COC(=O)N2)=O)CCCC(C)(C)C1C(=O)NCC=C(Cl)Cl c1(C(N2CCC(NC(C3CC3c3cccnc3)=O)C2)=O)cccnc1S C(=O)(C1CCCc2n[nH]cc21)N1CCC(CC)(Cc2cnn(CC(F)F)c2)C1 c1(C(=O)NC(CNC(CC)=O)C2CC2)ccc(CNC(C2CCOCC2)=O)cc1 N1(C(C(C=C)CC)=O)CCC(C)(C)C1CC(=O)NC(C(C)(C)O)C1CC1 C(=O)(C#CC1CCCOC1)NC(C)(C)CNC(=O)C(C)(C)C(C)(C)C C1(CNC(Cc2scc(C(=O)OC)c2)=O)C2CN(C(=O)C(C)CCN(C)C)CC12 N1(C(C=CCN(C)C)=O)CCC(C(C)(C)NC(C2CC(=O)N(C)C2)=O)CC1 Nc1ccnc(C(N2CCCC(CCNC(C3C4COCC34)=O)C2)=O)c1 c1(C(C)NCc2cn(CCCCCO)nn2)ccc(O)cc1 C1(C(=O)NC2(CCNC(c3c(C)snn3)=O)CCC2)CC1C1CCCCC1 c1(N2CCN(CCOC(C)(C)C)CC2)nc(=N)[nH]c(=NCCc2cnco2)[nH]1 c1(C(N2CCC(NC(Cn3ncc(C#C)c3)=O)C2)=O)cc2c(=O)[nH]ccn2c1 N1(C(c2cc(CC)n(C)n2)=O)C2CCCC1CN(C(=O)C(N)=O)CC2 C(=O)(CCC(F)(F)C(=O)NCC1CCN1c1nc(C)c(F)c(C)n1)OCC CC1(C)CN(C(C2CC(NC(=O)C=Cc3cc[nH]n3)C2)=O)CCO1 CCCC(CC)CC(=O)NCC(C)N(C(c1cc(Cl)cn1C)=O)CC c1(C(=O)NC(CN2CCCC2)Cc2ccccc2)cccc2ccnc(Cl)c12 C1(C(=O)NC(C(=O)NC)C2CC2)C2CC3C(C2NC(c2cc(F)ccc2C)=O)C13 C1(C(N2CC(CNC(C3C(C)N(C)CC3)=O)OCC2)=O)CCC(C2CCCO2)O1 CCC(CC)CC(F)C(=O)NC1CCCN(C(c2snc(C)c2N)=O)C1C Cc1c(NC(=O)C(CCC2(C#N)CC2)N(C2CC(F)(F)C2)CC2CC2)cccc1Cl C(=O)(C(O)CC(C)(C)C)NC(CNC(c1n(CC)nc(C2CC2)c1)=O)CC C(=O)(C1=NN2CCCN=C2N1)N1CC(CNC(CN2C(C)CSCC2)=O)C(C)C1 c1(CC(=O)Nc2c(COCC#C)cccc2)cc(Cl)c(Br)c(Br)c1 C1(NC(CCN2CCN(C(C)C)CC2)=O)CC(F)CN(C(c2cnns2)=O)C1 N1(C(CN(C(=O)CCN2CCCC2)C)=O)CC2(CC(N(C)C)C2)C1 C1(NC(CCN(C)C(C2CC3(CCC3=O)C2)=O)=O)CCCCCCC1O c1(C(N(C(C)CNC(C2CCCN2C2CC2)=O)C)=O)cc2cc(O)ccc2[nH]1 c1(CN2CCN(C(C3(C4CCC4)CC3)=O)CC2)cc(N2CCOCC2)cc(F)c1 C(=O)(C(CC)C(=O)OC)NCC1CC(C(=O)N(C)Cc2ccc(CC)cc2)C1 c1(OC)ccnc(C(=O)NC2CCCN(C(c3csc(COC)n3)=O)CC2)c1F CCC(CC(=O)N1CC(N(C(=O)CCCCSC)C)C1)c1ccc(NS(C)(=O)=O)cc1 C(c1ccc(-c2ccccc2F)s1)=CCCCc1onc(N(C)C)n1 c1(CN(C)C)ccc(C(N)=O)nc1.c12ncc(o1)C(=O)NC1CN(C1)C(=O)CC2 c1(C(=O)NCC(N(C(=O)CC2CCC(C)(C)C2)C)C2CC2)cc(S(N)(=O)=O)c[nH]1 c1(NC(C2CC(NC(c3ccn(CC)n3)=O)C2)=O)cc(C#N)c(Br)cn1 CC(C)CC(O)C(=O)NC1(C)CCN(C(=O)C(C)C(F)F)CC1 N1(C(C2OCCC(=O)C2)=O)CCC(NC(=O)C=Cc2ccco2)C(F)C1 c1(OC)cc(N2CCCC(NC(=O)NC3CC(C(=O)O)C3)C2)nc(=N)[nH]1 CC1(CNC(c2n[nH]cc2-c2ccc(F)cc2)=O)CN(C(=O)C(N)=O)CCO1 c1(C(=O)Nc2cccnc2O)nnc(O)nc1O.C12CCN(CC1)CCNC2=O c1(CCC(=O)NCC2C=CCN2C(=O)C2=COCC2)cccc(F)c1 C(=O)(CCCC(=O)NC1CC1)NCC1N(C(C(CCC)F)=O)CC(O)C1 N1(C(=O)Nc2nc(OC)oc2)CCOCC1CC(=O)NCCc1ncoc1C Cc1cc(C(=O)NCC2COCCN2C(c2cc(Br)ccc2Cl)=O)ncc1F C1(CNC(C(c2ccc(C(F)F)cc2)C)=O)CCC(NC(=O)C(F)(F)CO)CC1 N1(C(C(c2c(C)noc2C)CC)=O)CCCCC12CN(C(c1ccn(C)n1)=O)C2 N1(C(C(CC(C)C)ONC(CC2ON=C(C)C2)=O)=O)CCCC(C)(C#N)C1 C(C(C)(C)C1=CCCC1)NC(C(C1CN(C(CC2CC(SC)C2)=O)C1)OC)=O Cc1sc(C(=O)NC2CCN(C(c3ccoc3Cl)=O)C2C)nc1Br CCC(C)(C(=O)N1CCN(C2CCCN(C(=O)C(=O)NC3CC3)C2)CC1)C(F)F CC(CN=c1[nH]c(N2CCCN(C)CCC2)nc2c1COC2)N(C)C C1(C(N2CCC(N(C)C(c3sccc3Cl)=O)C2)=O)CC2CCC(C1)S2 c1(OC)cccc2c1OCC(C(=O)N1CCC(NC(c3csnc3OC)=O)C1)=C2 c1(C(=O)NC23CN(C(CCC(C)C)=O)C(CC2)CC3)c[nH]c2cc(F)ccc12 Cc1cn(C)cc1C(N1CC(NC(=O)CC2CSC2)CC1C)=O C(CCC(C)C(=O)N1CCN(C(=O)CCc2cn(C)nc2C)C(C)C1)OC CN1CCC(C)(C(N2CC(NC(=O)C(Cl)=CCl)C(CC(C)(C)C)C2)=O)C1 N12CCC(CC1)N(C(c1csc(O)n1)=O)C(=O)C2C.c1(NC)ccccc1 c1(OC)ncc(Br)cc1NC(C1CC1C(=O)Nc1cccc(C2CC2)n1)=O N1(C(C(C(=O)OC)SC)=O)CCOCC(C(=O)N(C)CC2CC(F)(F)C2)C1 c1(C(=O)NC2C(NC(c3ccc(NC(N)=O)cc3)=O)C2)ccc(N)c(F)c1 CCCCCCCC(=O)NC(C)(CNC(c1ccnc(O)c1F)=O)CC C=C(C)CCCC(=O)NCC1CCCN1C(c1ccc(OC)cc1C(=O)OC)=O c1(SCC(=O)NC2(C(F)(F)F)CC(O)(C(=O)O)C2)nc2ccccc2s1 c1(C(=O)NCC(C)N(C)C(C2C=CCCC2)=O)cc(C(F)(F)F)cnc1O N1(C(C2=CC(C)(CC)C2)=O)CC2(CCN(C(c3occ(C)c3C)=O)C2)C1 C(C)(C)(CC(=O)Nc1ccc(C(C)=O)cn1)N(C(CSC)=O)C c1(C(=O)NCC2CCCC(NC(CSCC)=O)C2)c[nH]c2c(F)cccc12 c1(C(N2CCC(NC(C=CC)=O)C2)=O)cc2ccccc2cn1 CN1CC(O)CC1C(N1CC(O)(CCNC(C2(C)CCC2)=O)C1)=O CC(C)CCCCC(=O)NC1(CNC(C2CCC3(CCCC3)C2)=O)CCC1 C1(C(CNC(C(C2(O)CCCC2)OC)=O)(C)O)CCN(C(=O)CCS(C)=O)CC1 N1(C(C(n2ccc(Br)n2)C)=O)CCOCC(C)(CNC(=O)Cc2ccoc2)C1 N1(C(C)=O)CCC(C(N2CC(NC(C3(C)CSC3)=O)C2)=O)CC1 NS(=O)(=O)c1ccsc1C(=O)NC1CCCC1NC(C1CC(N2CCCC2)C1)=O c1(C(=O)OC)ccc(C(=O)N(CC(O)CN(C(=O)CN2CCC2C)C)C)c(F)c1 c1(CC(=O)NC2(CO)CCN(C(=O)CC3CC(C4CC4)C3)C2)cccc(F)c1Cl C1(N(C(C(C(C)C)C)=O)C)CC2CCC(C1)N2C(c1cc(=O)cc[nH]1)=O Cc1ccc(C(C)C)cc1OCC(=O)NCC1CCC1NC(c1ccc[nH]1)=O N1(C(C2ON=C(C)C2)=O)CCC2(CC1)CN(c1nccc(SC)n1)CCO2 N1(C(c2cnccn2)=O)CCC2(CC1)CN(C(c1cccnc1)=O)CC2CO N1(C(c2cncc(OC)c2)=O)CC2CN(Cc3cc(F)ccc3I)CC12 C=CC(CC)CC(=O)N1CCC2C(C(=O)Nc3cccc(OCF)c3)C2C1 C(=O)(C1=CSCCO1)NC1CCCC(NC(CCCCOC)=O)C1 CC(C)(C)C(CO)C(=O)NCC1CC2COCC2N1C(c1cccc(F)c1N)=O Cc1ncc(C(N2CC(NC(=O)CCc3ccc(Cl)cc3)CCC2C)=O)cc1Cl c1(N(C(=O)C(F)(F)F)CC(N2C(CNC(=O)C(O)C3CC3)CC2)=O)cccc(Cl)c1 Cn1c(=O)cc(C(=O)NC2CCCC2NC(=O)C=Cc2ccoc2)c2ccccc12 n1(CC(C2CCC(C#N)CC2)=O)cc(-c2ccccc2)cc(C(F)(F)F)c1=O N1(C(c2cc(OCC)no2)=O)CCN(C(=O)C(C)(C)CC2(CC)CC2)C2(CCC2)C1 c1(CC)cc(C(=O)NCC(C(C)(C)C)NC(=O)CCNC(=O)C(C)(C)C)sc1C C1(=O)CCCC(c2nnnn2CCNC)NCCCN1.C(C(=O)OC)NC(C)=O c1(OC)c(Cl)ccc(C(N2CCC(F)C(NC(=O)C(F)=CCCF)C2)=O)c1F C(=O)(CCCCCC(C)O)NC1C(OC)CN(C(=O)CC2OCCC2(C)C)C1 c1(CC)ncnc(NC2CCCC(CNC(=O)CCc3c(C)c[nH]c3C)C2)c1F c1(OC)cccc2c(C(N3CCC(N(C(=O)C(C)=C4CC4)CCO)C3)=O)coc12 C1(C(=O)NCCCC2CC(C)C2)CCN(C(=O)C2=COCC2)CC1(C)C c1(C(=O)NCCN2C(C)CCC2C)cccc2c1ccn2C C1(C(=O)NCC(CC(=O)N(CC(C)C#N)C)C2CCC2)CCC(=O)CC1C CC1(C)C2CCC1(CC(=O)NC1CCCC(NC(c3cc(F)n[nH]3)=O)C1)CC2 N1(C(c2cc(OC)ncc2)=O)CCN(C(C2CCN2C2CCCC2)=O)CC1C C1(C(=O)NCCCOCCCNC(COCCCOC)=O)CCOC1C C(CN=c1nc2sccc2c(NC(C)(C)C)[nH]1)=CCN1CCN(c2cccs2)CC1 N1(C(c2ncc(OCC)nc2)=O)CCN(C(=O)C=CSC)CC1CC(F)F C1(CCC)(NC(c2sccc2C(C)=O)=O)CCN(C(C2COCCO2)=O)CC1 N1(C(c2sc(CC)c(C)c2)=O)CCC(NC(c2cnccn2)=O)C(C)C1 O=C(C(F)C(F)(F)F)N1CC2CC1(c1cn(CCC3CC34CC(O)C4)nn1)C2 c1(NC(C2(F)CCN(C(=O)Cn3ccnc3)C2)=O)cc(Br)cnc1[N+](=O)[O-] C1(CC=C)(NC(c2coc(Cl)n2)=O)CCN(C(=O)CCN2CCOC2=O)C1 C1(NC(CCC(=O)NCCC)=O)CCC2CN(C(C3(C4CC4)CCC3)=O)CC2C1 C1(NC(c2cc3ccccn3c2)=O)CCCCC12CCN(C(=O)CCCF)C2 N1(C(c2ccc(Cn3ccnc3)o2)=O)CC2(CCN(C(C3CC(F)C3)=O)C2)C1 c1(C(N2CCC(NC(C(C)OCCN(C)C)=O)C2(C)C)=O)cc2ccccc2o1 Cc1cc(C(=O)NC2CCCC(N(C(=O)CC3CCOCC3)C)C2)ncc1F c1(C(=O)NC2CC(NC(C3CC(CCC)C3)=O)C2)cc(N)cnc1Cl C(=O)(C1=C(F)CN(C(=O)CC(C)(C)CC(F)F)CC1)N(CCCCCCC)C C1(C(=O)NCC(=O)NC(C)C)(CC)CN(C(C2C=CCCC2)=O)C1 C1(CNC(COCCC#C)=O)CC(OC)CN1C(C1CCCN1C1CC1)=O c1(-n2cc(CN(C3CC3CN)CC)nn2)c(C)cccc1Br.C12CCCN1C2=O CC(C)(C(=O)NCCC1CCC(NC(=O)CCC2CC2)C1)C1CCC1 c1(OC)cccc(C=CC(=O)N(CC(=O)NC2CC2)C)c1OC.c1(N)ccccc1C c1(CC)nn(C)c(CC)c1CC(N1CC(O)CC1CNC(=O)C(C)O)=O c1(C(=O)NC(C)(C)CNC(c2coc(Cl)c2)=O)ccc2c(c1)CC(C)(C)C2 C1(CNC(=O)CCn2nc3c(n2)CCC3)C2CCC(C2)N1C(=O)C#CC1CC1 C1(OC)CN(C(c2nn(C)nc2Br)=O)CC1NC(c1ccc(C)cn1)=O C1(OCC(=O)NC)CCN(C(C2CCC(F)(F)C2)=O)C1CC.C1C(=O)NCCO1 C1(N(C)C)C2CN(C(=O)C(C3CC3)N(C(=O)C(C)(C3CC3)N(C)C)C)CC12 c1(OCC)cc(Cl)ccc1C(N1CCC(CNC(C2(C)CC3CCC2O3)=O)C1)=O n1(CCC(N2CCC(NC(CNC=O)=O)C2)=O)sc2ccccc2c1=O c1(N(C2CCCN(C(C34CC=CC(C3)OC4)=O)C2)C)nc2ncc(Cl)cc2s1 C1(C)(CC)CC(C(=O)NC(C2(O)CN(C(c3cnccc3C)=O)C2)C)CCO1 CC12CCCCC1CN2c1nnc(C(F)(F)F)s1 c1(C(N2C(CNC(CS(CC)(=O)=O)=O)CC2)=O)ccc(F)c(Cl)c1F C(=O)(C#CC(C)(C)CNC(C1C2CCCCC12)=O)N1C(C)C(O)CC1 C1(c2n(C)ccn2)CN(C(C2(O)COC2)=O)CC1NC(c1ccsn1)=O CC(C)CCC(O)C(=O)N1CCCCC(NC(C2CC(C)(O)C2)=O)C1 C(=O)(C(=O)C(C)(C)C)N1CCC(C(=O)NCCC(C)(C)C)(OC)C1 Cc1cccc(CC(=O)NCC2CN(C(C3(CCC4CCC4)CC3)=O)CC2C)c1Cl c1(C(N(C)CC2CCN(C(C(CCCC)(C)F)=O)C2)=O)cc2cccc(C)n2n1 N1(C(c2c(Cl)ccc(C)c2)=O)CCN(C(C2CC(C)(F)C2)=O)C2CS(=O)(=O)CC12 C1(CNC(=O)Cn2cnc(Br)c2)C2CN(C(=O)Cc3cccc(Cl)c3)CC12 C12CCC(CC1)CNC2=O.C1CCCCC1F.C(CNCC1CC1)OC C1(C(C(=O)NC(C2CCCC2)CNC(=O)CCOC2COC2)F)CCCCC1 C1(C(N(C)CC2C(C)C2)=O)CN(C(=O)CCn2cncn2)CC1F Cc1ccnc(C(N2CCCCC(CNC(=O)Cc3c[nH]nc3O)C2)=O)c1Br c1(CCC(=O)NCC2(CCNC(CSC)=O)CC2)cncnc1 Cc1cccc(CC(N2CC(CNC(=O)CN3CC=CC3)CC2C)=O)c1 C1(C(N2CCC(NC(C(CCCC)O)=O)C2C)=O)CC(=O)CC12CCC2 N1(CC(=O)NC(C)C(CO)NC(c2cc(O)cs2)=O)CCCCS1(=O)=O C1(CC)CN(C(=O)NCC2(n3cc(Br)cn3)CCC2)CCO1 CC(C)(CCNC(=O)C(O)CCC1CC1)C(=O)NOCC1CCCCC1 c1(CC)ccccc1C(CNC(=O)C(CO)N(C)C)NC(C1CCCS1)=O n1(CC(=O)OC)nnnc1C(c1ccn(C(F)(F)F)n1)NCC1CC1(C)C c1(NCc2c(CC)n[nH]c2)cccc(OC(C)(C)C)c1 C1(NC(C(C)OCCOC)=O)CC(F)CN(C(c2cnc(C)nc2)=O)C1 CC(C)CC(C(=O)NC1CCCC(O)CC1)N(C)C(c1cnn(C2CC2)c1)=O c1(C(=O)NCC(CC=C)NC(=O)CC(C)F)c([N+](=O)[O-])cnn1CC c1(C(=O)NC2CN(C(c3nc(C)oc3)=O)CC2C)c(Cl)cncc1Cl CCCC(C(=O)NC(C)CN(C(=O)C=C(Cl)Cl)C)C(C)C N1(C(C2C(C)CCO2)=O)CCC(C)(NC(c2nn(C)cc2N)=O)C1 c1(OC)ccc(C(C)C(N2CC(NC(=O)C(F)F)C(C)(C)C2)=O)c(C)c1 c1(OC)cc(C(C(=O)NCc2cncs2)N(C2CCS(=O)(=O)C2)C)ccc1Cl c1(C(N2CCN(C(CNC(=O)NC)=O)C(COC)C2)=O)ccn2nccc2n1 N1(c2ccnc(C)n2)CC(NC(c2coc(Br)n2)=O)C(C)(C)C1 C12(CC(=O)N(C(CCNC(C3CN(C(C)=O)C3)=O)C)C)COC(CF)(C1)C2 C(=O)(C(CC(F)F)N(C)C(c1nc(Cl)cs1)=O)NC(c1scc(C)n1)C C1(C(N2CCCC(n3cc(CCC(C)(C)CO)nn3)C2)=O)CCCCC1(C)C c1(NC(=O)CN2CCC(CC(=O)N(CC3CCCO3)CC3CC3)C2)cccc(Cl)c1 C12(C(=O)NC(CC)CNC(=O)CC3(O)CCCOC3)CCCN(CC1)C2 C(=O)(C#CC1CCCCO1)N1CCC(C)(CC(=O)NCCCOCC(F)F)C1 c1(CNC2(CC(=O)NC3CC(=C)C3)CCC2)cc(Cl)cc(Br)c1O C12CCN(C1(C)C)C(=O)c1cccc(c1)NC2=O.C1(N)CCC(CO)CC1.COC C1(NC(Cc2c(CC)cccc2)=O)CC2CN(C(C3CSC(C)=N3)=O)CC2C1 Cc1ccnc(C)c1C(=O)NCC1(F)CCC(NC(=O)C(C)Cc2ccsc2)C1 C1(N(C)C(C2CC(OC(F)F)C2)=O)CCCCN(C(c2cn3ccnc3s2)=O)C1 N1(Cc2cc(CC)c(O)cc2)CC2CCN(C(=O)C(C)Cc3ccc(Br)cc3)C2C1 C(=O)(CCCC(C)(C)C)NCC1(F)CCCN(C(C(C)OCC2CC2)=O)C1 C1(CNC(C2(CCNC(C3C(C(C)C)CC3)=O)CC2)=O)CCOC1(C)C.C1CO1 N1(C(=O)OC)CCCC(C(=O)NCC(CO)NC(c2onc(OC)c2Br)=O)C1 c1(C)c[nH]c2ncc(Cl)cc12.N1(C(c2nc(C(=O)OC)[nH]c2)=O)CCN(C)CC1 Cc1nc2c(s1)CN(C(C13CC1CN(c1ncnc4c(Br)c[nH]c14)C3)=O)CC2 C1(CNC(C(=O)NC)=O)CN(C)CC1(C)C.c12ccc(cc1)NC21CC(O)C1 S(=O)(=O)(CC(C)c1ccccc1)NC(NOCC)=O c1(OCC(=O)NC2C(C)N(C(c3csc(Cl)c3)=O)CC2)nc(O)nc(O)n1 C=C1CC(CC(=O)NCCCN(C(=O)COC2CC=CC2)C(C)C)C1 N1(C(c2c(C)coc2)=O)CC2CCC(C1)N(C(=O)Cc1cc(C3CC3)on1)C2 CCCC(O)CC(=O)N1CC2CC2(CNC(c2ccc(C)cc2Cl)=O)C1 CC1CC=C(C(=O)N2CCC(N(C)C(c3cccc(F)c3C(F)F)=O)C2)CC1 c1(C(=O)NC2(C)CCN(C(C3C(C)C3(F)F)=O)C2)ncc(C(F)(F)F)cc1N C1(NC(C(C)=C2CCC2)=O)CC2(C1)CC2NC(c1cc(CCCO)on1)=O C(c1ccccc1Cl)=CC(C(=O)NC(CC(C)NC(=O)Cc1nnn(C)n1)C)=O c1(CC)ccc2c(c1)CN(C(c1ccc(C)c(I)c1)C(=O)NCCCSC)CC2 C1(C(=O)NCCC)N(C(=O)CN2CSCC2=O)CCC1(C)C c1(C(=O)NC2C(CNC(c3cn(C4CC4)nn3)=O)C2)cc(F)cc(Br)c1O Cc1ccnn1C(C)C(=O)NCc1cc(C(=O)N(C2CCC3CC23)C)co1 CCC1=NOC(C(=O)NCC(C)C(=O)NC2(CCF)CC2)C1 CON1CCC(C(=O)NC(CNC(=O)CSC(F)F)CO)CC1 c1(C(=O)NC(CC)CC2CCOC2)cccc(COCC(=O)O)c1 N1(C(C=C(CC)CC)=O)CC2(CCC2)CC1CNC(c1nnn2c1CSCC2)=O c1(CC)cnccc1-c1ncsc1C(=O)NCCOc1ccccc1C.C1CO1 c1(CCC(=O)N(CC(C)N(C(C(CC)O)=O)C)C)ccc(O)c(OC)c1 c1(C(N2CC(C(C)NC(C3C(C=C)OCC3)=O)C2)=O)cc2cccn2cn1 C1(NC(C2C(C)C2)=O)CN(C(=O)CCCCOC(C)=O)CC1F c1(C(=O)OC)cc(C(=O)N(C)CCN(C)C(c2nnc(C)s2)=O)ns1 N1(C(c2c(C)snn2)=O)CC2COCCC2(NC(c2csc3nnsc23)=O)C1 C(=O)(CCCCCSCCC(C)C)N(CCNC(CCCOCCC)=O)C C1(C(N2CCCC2CN=[N+]=[N-])=O)(CNC(C(C)N(C)C)=O)CCCCC1 c1(C(=O)NC2C(CNC(Cn3ncc(C)c3)=O)CC2)c(Br)cnn1C(C)C Cc1ccncc1NC(c1ccc(CNC(=O)C(O)CC2CCCC2)s1)=O c1(OC)cc(C(N2CCC(NC(=O)C(C)C#N)C2)=O)cc(Cl)n1 C1(NC(=O)Cc2cccs2)CCC2(CC1)CN(C(c1ccnnc1)=O)CCO2 c1(OC(c2nc(C)no2)C(=O)OC)ccccc1N(CCCN(C)C)C Cc1cccc(C=CC(N2CCC2CNC(C2CCN(C)C2C)=O)=O)c1 c1(OC)ccc2c(c1)CC(NC(c1cccc(-c3ccc(=N)[nH]c3)c1)=O)CCC2 c1(OC)ccc(NC(C23CC2CN(C(=O)CCn2ccnn2)C3)=O)c(OC)c1 CCC(COC)C(=O)N1CCCC1(C)C(=O)NCc1ncn(C2CC2)n1 Cc1[nH]c(C)c(C(=O)NC(C)CCNC(=O)CC2NC(=O)NC2=O)c1C O=C1CCC(C(=O)N2CC(CNC(=O)COCc3ccncc3)C3CC23)=NN1 N1(C(C(C(C)(C)C)O)=O)CC=C(CC(=O)NC2CC3(COCCO3)C2)CC1 C(=O)(N=c1nc[nH]n2cc(Br)cc12)c1nc(Cc2c(C)ccc(F)c2)[nH]n1 N1(C(c2c(NC)scn2)=O)CC2(CCCCN2C(=O)C(C)SCC2CCCO2)C1 C1(CNC(C(C)=C2CC2)=O)CC2COCC2N1C(=O)Cc1ccccc1Cl N1(CC(N2CC=CC(NC(C(C(CC)(C)C)O)=O)C2)=O)C(=O)c2ccccc2C1=O Cc1csc(C)c1C(=O)NC(C)C(C)C(=O)NCC1(CN(C)C)CC1 C1(O)(CN(C)C(c2cn(C3CC3)nn2)=O)CN(C(c2cccs2)=O)C1 Cc1c(C(=O)NNC(=O)c2nn[nH]n2)cc(C(C)(C)C)n1C O=C(CC1CCc2ccc(O)cc21)OC1(Cc2ccccc2)CCCC1 CC1(O)CC(C(=O)N(C2CCN(C(=O)CC3CCOC3=O)C2)CCO)C1 C(=O)(C(O)P(C)(C)=O)N1CCCC(N(C(=O)COCCF)C)C1 N1(C(CC2CC(OC)C2)=O)CC(OC)CC1CNC(C1CCC(=O)N1C1CC1)=O C1(C(N(C)Cc2nnnn2C)=O)CCN(C(C2CC2[N+](=O)[O-])=O)C(C)(C)C1 CC1CCCN(C(=O)COCC(C)(C)C)C1.C(C)(CC)NC(C1CN(C(C)=O)C1)=O c1(CC)ocnc1C(=O)NC1CCC(N(C(=O)Cc2cc(C)cs2)C)C1 C(=O)(C(F)C(C)C(F)(F)F)N(CCNC(=O)CC(c1cccs1)n1cccc1)CC CC1(C)CC(C(=O)NC2CC(O)C2(C)C)CCN1C(=O)CSC(C)(C)C CC1=C(CNC(=O)C(C2CCN(C(C3CC3(F)Cl)=O)CC2)C)COCC1 N1(C(c2ccc(COC)[nH]2)=O)CC(C)(C)CC1CNC(c1cccc(OC)n1)=O N1(C(=O)Nc2c(C)n(C(F)(F)F)nc2)CCn2nnc(Br)c2C1 Cn1ccc2nc(N3CCC3(C)C(=O)Nc3ccc([N+](=O)[O-])c(Cl)c3Cl)ncc12 CC1(C)CC(NC(c2ccc(C#N)cc2)=O)CN1C(=O)C=CI C(=O)(C(C)CC(=O)c1ccc(F)cc1)NCC(C)N(C)C(c1ccns1)=O c1(C(=O)NCC2(F)CCC(C)CC2)cccc2c1C(=O)CC2 C12(NC(c3c(COC)scc3)=O)CCOCC1CN(C(=O)C(C)=C1CC1)C2 c1(SC)cccnc1SC.C12(CCC1)CCNC(=O)N2.C1(S)CCC1 Cc1sc(S(=O)(=O)Nc2ccc(OC3CCCCC3)nc2)cc1[N+](=O)[O-] C=CCC(CNC(=O)COCCCN(C)C)NC(=O)CCC1CCC(C)O1 c1(C(=O)NC(CNC(CS(CC)=O)=O)C(C)(C)C)cnn2c(N)cc(C)nc12 c1(C(=O)NCCOCCC(=O)N(C)CC2(C)CCC2)cccc(=O)o1 CC(C(=O)N1CC(CNC(C2(CC(F)F)CC2)=O)C1)NC(C)(C)C C=CCCC(C(=O)NCC1CC1C(N)=O)NC(C1CCCC(C(=O)OC)C1)=O c1(C2C(NC(N3CCOC(CC(F)F)C3)=O)C2)cc(Cl)ccc1Cl c1(C(C)C(N2CC(NC(C3CCCC(=O)N3)=O)C(O)C2)=O)noc2ccccc12 C1(C)(C(=O)NCCCCN(C(C2(CCC)CCC2)=O)C)CC(C2CC2)=NO1 N1(C(c2c(C)nc(C(C)SC)s2)=O)CCN(C(=O)COc2cnn(C)c2)C(C)C1 C1(CC(=O)NCC(CC)NC(=O)Cc2cc(C)sc2C)CCCC2(CC2)C1 N1(C(C2C(C)(C)OCC2)=O)CCOCC(NC(=O)C(c2cc(F)cc(Cl)c2)=O)C1 C(=O)(C1CNc2ccccc21)NCC(CNC(c1n(C)nnc1-c1ccco1)=O)F c1(OCC(CN2CC(O)(CCNC(=O)CCCOC(F)F)C2)O)ccc(Cl)cc1 C1(C(N(C2CCCN(C(=O)C(c3c(C)noc3C)C)C2)CC)=O)C=CC=CC=C1 N1(c2snc(OC)n2)Cc2nccn2CC(CNC(=O)OC(C)(C)C)C1 O(NC(=O)C(C1(C)CC1)NC(=O)CC1(C)OCCO1)CCC(CC)C C#Cc1cccc(CC(=O)NCC2CN(C(=O)CNS(N)(=O)=O)CCC2F)c1 N1(C(CCSC)=O)CC2(CCCC2)C1C(N1CCC(CO)C(C)C1)=O C(=O)(CC(C)(C)CN(C)C)NC(C)CCNC(c1cncc(Cl)c1)=O Cc1nn(C)cc1-c1nonc1C(=O)OC1CCC(=O)NC1 C1(C(N(C(CC)C(=O)OC)C)=O)C=CCN(C(=O)CCc2nc(C)no2)C1 Cc1nc(C(=O)NC2(CCNC(=O)C=CC3C(C)C3(Cl)Cl)CC2)c(C)o1 Cc1cnc2n1CCC(C(=O)NCCN(CCOCCO)C(C1CCCN1C)=O)C2 C=CC1(C(=O)NCCC(=O)N(C)C)CCN(C(C2CC(N(C)C)C2)=O)C1.CCO S(=O)(=O)(c1ccc(NCS(C)(=O)=O)cc1Cl)NC1C(C(C)C)CN(C)C1 Cc1cccc(NC(C2CC23CCN(C(c2ccccc2Br)=O)C3)=O)c1[N+](=O)[O-] Cc1cc(C(=O)N(C)CC2(NC(C3CNC(=O)CC3C)=O)CC2)c2c(c1)CCO2 c1(C(N2CC(NC(C34CCCC3C4)=O)C2)=O)ccc(Cl)c(C(F)(F)F)c1 CC1CCN(C(=O)C(O)Cc2cnc[nH]2)CC1NC(c1n[nH]cc1Cl)=O CC(C)(F)CCCCC(=O)NCCC1CCCN(C(=O)CC(O)C2CCCC2)CC1 c1(C(N(CCCNC(=O)C(C)(F)CC2CCCC2)C)=O)cc(Cl)c(F)cc1F c1(CC(CNC(=O)C(C2CC2)SC)NC(=O)CNC(=O)C2CC2)ccccc1 c1(CC(=O)NCCCN(C(=O)CC2CC23CC3)CCO)ccccc1O c1(C(=O)NCc2c(C(=O)NC3C(CCOC)C3)scc2)cc(Cl)ccn1 c1(NCCOCCCC#C)noc(-c2ccn(CC(=O)OC)n2)n1 N1(C(CCN(C2CCCCC2)C)=O)CCC12CN(C(=O)CC1CS(=O)(=O)C1)C2 CC(CC(Cl)Cl)NC(C1CC1c1cn[nH]c1)=O C(=O)(C(F)(F)CCn1ccnn1)NC(CC(C)NC(COC)=O)C n1(CC(=O)N(CC(C)N(C(c2cc(C)ncc2C)=O)C)C)cnc2ccccc12 C#CCCCCCC(=O)NCC(C1CCCC1)NC(=O)CC1COCC(C)(C)O1 CC(C(C)(C)C(=O)NCCC(F)F)NC(=O)C(C)C1(O)CCC1 c1(C(C)C(=O)NC2CCCC(NC(C34CC(CO3)C4)=O)C2)c(F)cccc1F Nc1ccc(C(N2CC(F)(CNC(C3(CO)CC3)=O)C2)=O)nc1N Cc1ccc2c(C(N3CCC(CNC(C4NC(=O)OC4C)=O)CC3)=O)coc2c1 N1(C(CCN(C2CCCCC2)C)=O)CCC(NC(C2(F)CCOCC2)=O)C(F)C1 CC1=CCC(C)(C(=O)NC(C2CN(C(=O)C(C)N3CCCC3)C2)C)CC1 CC1COCC(CC(N2CCCC2C(C)(C)NC(C2CCCN2C)=O)=O)O1 C(c1cnn(C)c1)=CC(=O)N(C(C(=O)NC1C(COC)CCC1)C)C1CC1 CC1(CN)CCC(NC(=O)CCC(=O)C2CC2)C1.N1(C2(C(=O)N)CC2)CCCC1 C(C1=NOC2CN(C(=O)C3=CCCCCC3)CC12)NC(c1cc(C)nc(O)c1)=O n1(CC(=O)NC(CNC(=O)CC2CSC2)CC2CCCC2)cccn1 N1(C(c2ccc(Cl)nc2C)C(=O)NCC=C)CCCC(C2CCCC2)C1 C(=O)(CC(C)NCCN(C(=O)COC1CCC1)CCSC)OC.C(C)C N1(C(C(CC)C(C)O)=O)CCCN(C(c2cc(C)cs2)=O)CCC1 N1(NC(C(CC2CN(C(CCCC(=O)CO)=O)C2)F)=O)C2CCC1CCSC2 C#CCC(O)C(=O)NC1CCC(CC(=O)NCC2CC(N(C)C)C2)C1 C(=O)(C(C)(O)C(F)(F)F)N1CC(C(N2CCC(O)(CC#C)CC2)=O)OCC1 CC(C(C)(C)C(=O)N1CCC(c2ccco2)C1)NC(=O)CO c1(C(N2CC(C(=O)Nc3cnc(C)nc3)C(C)C2)=O)c[nH]c(=N)c(C)c1 C=C(Cl)CCC(=O)NCc1ncccc1CNC(c1ccc(F)cn1)=O c1(C(c2n(CC=C)nnn2)NCc2ccsc2)cnn2c1CCC2 c1(C(=O)NC(C2(C(N(C)CC3(OC)CCC3)=O)CC2)C)cn(C)c(=O)cn1 c1(C(N(CCOCCNC(CS(C(C)C)(=O)=O)=O)C)=O)ccc2oc(=O)oc2c1 C1(C(=O)NC2C(CCC)CCC2)CC(F)CN1C(c1sccc1COC)=O C1(CCCC)CCCN(C(C2C(C)CN2C(=O)CCC)=O)C1 CC(C)(F)CCC(=O)NCC12CC(CN1C(c1cnc(N)c(-c3ccsc3)c1)=O)C2 Cc1nn(C)c2nc(O)cc(C(=O)NC(C)CNC(c3snc(Cl)c3Cl)=O)c12 N(C(=NCc1ccccc1C1CC1)NCC1CC1(F)F)C(c1ncn(C)n1)C C(=O)(C(=O)C(C)(C)C)N(C)CC1CCN(C(c2c(CC)ncs2)=O)C1 c1(OC)ccc(F)cc1C(=O)NC1CC(NC(c2cn(C)nc2C2CCC2)=O)C1 C1(N(C)C)CCCN(CC(=O)NC(CNC(=O)Cn2cc(Cl)cn2)C2CC2)C1 C(=O)(C1=C(C)OCCC1)NC(CC(=O)N1CC(C)(OC)C1)C(F)F c1(CNC(C2CC3CCC2O3)c2n(CCCSCC)nnn2)ccc(CC)cc1 CC(C(=O)NCc1cc(C(N2CC(C)OCC2C)=O)on1)C(C)(C)C c1(OCC)c(C(N2CCCC(O)(CNc3cncc(Cl)c3)C2)=O)cccc1C N1(C(C(CC)(C)C)=O)CC2CCC1CN2C(=O)C(=O)NC1CCCC1 N1(C(c2c(C)snc2)=O)CCCCC1C(C)NC(c1csc(-c2nc[nH]n2)n1)=O C12(NC(Cc3ccc(C)cc3)=O)CCC(C(N3CCOCC3CO)=O)(CC1)CC2 CCCN=C(NCCc1cc[nH]n1)NCc1nnc(C(C)(C)C)s1 C(CC(=O)NNc1ncccc1SC1CC1)(c1cccs1)NC(=O)OC(C)(C)C c1(C(=O)Nc2cccc(NC(C(C)n3cncn3)=O)c2)n[nH]c2c1COCC2 N1(N(C(C)CCCl)Cc2cccs2)CCC(O)CC1.C12(CCCC1)C(=O)NOC2 CC1CN(C(c2ccc(Cl)nc2N)=O)CCN1C(c1ccc(C(F)F)c(F)c1)=O C=CCCCCCC(=O)NCCCN(C(c1ncc(C(=O)OC)s1)=O)CC Cn1nnc2cc(C(N3CC(O)CC3C(=O)NCC3CCC3)=O)ccc12 N1(CCOC)CCC(C(=O)NC(Cc2ccccn2)C(F)(F)F)c2ccccc21 C(=O)(C1=CC2C=CC(C1)C2)Nc1c(CNC(C2(CO)CCCCC2)=O)cn(C)n1 Cc1ccc(C(N2CC(NC(C3CNC(=O)C3)=O)C3(CCC3)C2)=O)c(N)c1Cl C1(C(=O)NCCN(C(C(C)C2(O)CCC2)=O)C)CC2(CCC2O)C1 c1(C(=O)NCC(F)(F)F)cc(NC(c2cccc(C3CC3)n2)=O)ccc1F C(=O)(C1CCCc2scnc21)NC1C(C(C)C)CN(C(=O)Cn2nccn2)CC1 N1(C(C(=O)Nc2ccc(OC)cc2)c2ccco2)CCS(=O)CC(C)C1 N1(C(C23N(C(c4n(COC)ncc4)=O)CC(C2)C3)=O)CCn2nc(C)cc2C1 C(C(C(=O)Nc1cccn2cncc12)C(C)(C)C)NC(CCC#C)=O N1(C(CCc2ccc(C)c(Cl)c2)=O)CCC2CCC(NC(c3[nH]cnc3C)=O)C12 C=CCC(CC(C)C)C(=O)NC1COC2(C1)CN(C(c1cnccn1)=O)C2 Cc1cc2cccc(C(N3CCCC(O)(CN=c4[nH]nc(O)s4)C3)=O)c2o1 C(=O)(CCCSC)N(C1CCN(C(=O)CC(O)C2CC2)C1)CC#C N1(C(C(C)(C)CO)=O)CC2CCC1C(NC(C1CC(=O)N(CC(F)(F)F)C1)=O)C2 C(=O)(C1CC(=O)Nc2ccccc21)NC1CC(CNC(c2c(C)cnn2C)=O)C1 c1(C(N2C(CNC(c3ccn(C(F)F)n3)=O)CC2)=O)cc2ccccn2c1C(F)F CCC(C(=O)N(C1CN(C(=O)CCC2CCCOC2)C1)C)n1cncn1 C(N=c1[nH]c(Cl)ncc1[N+](=O)[O-])C1CCN(C(C2CC(C)OC2C)=O)C1 N1(C(CCC=C(C)C)=O)CC(N=[N+]=[N-])CC1C(N1CCC2CC12C)=O Cc1nc(SCC(=O)NC(c2ccc[n+]([O-])c2)C)c(C#N)c(C)c1C C(=O)(CCCCC(=O)NC)NC1CC(O)(CNC(c2c(O)ncc(CC)c2)=O)C1 c1(C(=O)NCCN(CCC)C(c2csc(CC(F)F)n2)=O)cccc([N+](=O)[O-])c1 c1(N(CCCNC(CC(C)n2cccc2)=O)Cc2ccccc2)ncc(F)cn1 C1(NC(C2CN(C(C)C)C2)=O)CN(C(c2c[nH]nc2C)=O)CCC12CCOCC2 CCC(CCCC(=O)NCC=CC)NC(=O)C(F)C(C)(F)F N1(C(C(=Cc2cccs2)C)=O)CC(CNC(=O)CC2OCCO2)C(C)C1 c1(NCCCNC)ccc(C(C)C)cc1S(=O)(=O)NCCF C(=O)(CCCOC)NC1(C(N(CC)CC)=O)CC1.C1(=O)C(C)N1 c1(C(N2C(C(=O)NCCOCCC)CCC2)=O)cccc2c(Cl)cccc12 c1(C(N(C(C)CNC(=O)C(c2cnccn2)C)CC)=O)c[nH]c2c(F)cccc12 CC#CCCCC(=O)NCC1CC2CC2N1C(=O)C(CC)(CC)OC CCCC(O)CC(=O)N1CCC(CN(C)C(C2(C#N)CC3CC3C2)=O)CC1 C1(CN(C)C(C2(CO)CCN(C(=O)CCCN3CCCC3)C2)=O)COCC1(C)C N1(C(C2(C(N(C)CC3(O)CCC3)=O)CCC2)=O)CC2C(C(N)=O)C2C1 C(=O)(C(O)CC(C)(C)C)N1CC2C(CNC(C3N(C)CC(F)C3)=O)(C2)C1 c1(C(N(CC(CNC(C=CCOC)=O)O)C)=O)cnc(C2CCOCC2)nc1 c1(NC(=O)NC2CC(NC(Cn3nnc(C)n3)=O)C2)nnn(C)c1SC(C)C N1(C(c2c(CC)ccnc2)=O)CC(C2CN(C(=O)C(F)(F)c3cccnc3)C2)C1 c1(NCC2C(C3C(C)C3)C2)cc(Br)ccc1S(=O)(=O)NC12CCC(CC1)OC2 C1(C(N(CC(CC)OC)C)=O)CCCCCN1C(c1cc(C)cc(C)n1)=O c1(C(=O)NC(c2ccc(Br)cc2)(C#C)C)ccnc2ccc(Cl)cc12 C(=O)(C(CCN(C)C)NC(C1CC12CC2)=O)NCC1CC(OC)C1 c1(C2C(NC(C=C(CCC)C)=O)C2)cn(-c2ncc(C(=O)OC)s2)nn1 N1(C(C2CN(C(=O)NC)C2)=O)CCC(C2CC2)(CNC(=O)CC2(C(F)F)CC2)C1 C1(CCC)CN(C(=O)C(CC)N(C)C)CC1C(=O)NC(CO)C(=O)OCC N1(C(C2(CCC=C)CC2)=O)CC(NC(=O)CCc2nc(C)c(C)[nH]2)C2(CCC2)C1 c1(C(=O)Nc2c(NS(CCOCC)(=O)=O)c[nH]n2)cccc2cn(C)nc12 N1(C(=O)CC2CN(C(c3ccnc(O)c3)=O)C2)CCC2(C1)CC2(F)F C1(C(N(C(C(CC)C)C)C2CC2)=O)CCN(C(=O)Cn2ncnn2)C(C)(C)C1 Cc1ncc(C(=O)NCCNC(=O)C(COC(C)(C)C)N(C)C)[nH]1 c1(C(N(CCN(C)C(=O)OC(C)(C)C)C2CC2)=O)cn(-c2ccccc2)cn1 C(=O)(C1CCCc2nncn21)NCCCCCNC(=O)C(F)C(F)(F)F c1(C(N(CC(C)N(C)C(C2CCC(=C(F)F)CC2)=O)C)=O)n[nH]c2cccnc12 C(=O)(CCC(C)(C)F)N1CC(OC2CCN(C(C3C(C=C)C3)=O)CC2)C1 C(C(=O)NCc1cnc(F)c(C)c1)(C(C)(C)O)NC(C(C)NC(C)=O)=O C(=O)(C(C)(C)CNC(C1C(C)C1C)=O)NC(c1snnc1C)C c1(C(N(CCCNC(C(CC)SC)=O)C(C)C)=O)cnn(C)c1Br N1(C(C2CCC(CC)O2)=O)CCC(CCNC(=O)C(N)=O)C(F)(F)C1 N1(C(C(C)SCc2ccc(F)cc2)=O)CCCC1(C)C(N1CCC(N(C)C)CC1)=O C1(NC(CCN(CC)CC)=O)CC(O)CN(C(c2nc(OC)cc(OC)n2)=O)C1 C1(C(N2CCC(NC(CC(=C)C)=O)C2c2ccccc2)=O)CC(C2CC2)=NO1 n1(C(=O)NNC(C)=O)ncc2c(C3CC3)cc(CCOC)nc12.CC CCC(CC(=O)NC(C)CN(C(=O)CCNC(c1ccccn1)=O)CC)C1CC1 CN1CCN(C(=O)C=CC2CCC2)CC1C(N1CCN(C)C2CC12)=O n1(CC)nc(CN(C)C(C2CCN(S(=O)(=O)C(F)F)CC2)=O)c(Br)n1 C1(NC(c2nc(C)oc2)=O)CC(F)CN(C(c2cnn(C3CCC3)c2C)=O)C1 C1(C(=O)NCc2occ(C)n2)C(C)CCN1C(=O)CC1(C)CCOCC1 N1(C(C2CCCN(CCC)C2)=O)CCC(C2(NC(c3nccn3C)=O)CC2)CC1 C1(C(=O)NC(COC)COC)CCCCCC1NC(C12CCC=C1C2)=O N1(C(C2CC(OCC)C2)=O)CCCN(C(c2ccc([N+](=O)[O-])cc2)=O)CC1C c1(C(=O)N(CCC(=O)NC(C2CCCC2)CO)CCO)n[nH]c2ccccc12 c1(C(=O)NCC(C2CC2)NC(CC=C)=O)c[nH]c2nc(F)ccc12 N1(C(CC(C)n2cccn2)=O)CCN(C(c2cc(N)cnc2Cl)=O)CC(C)C1 CC1(CNC(=O)CCCCNC(C2(CO)CCCO2)=O)CCCC(=O)N1 Cc1cc(C)c(C(=O)NCC2CCN2C(c2csc(S(C)(=O)=O)c2)=O)c(=O)o1 N1(C(C2=C(C)CCC2)=O)CC2OCC(NC(=O)C(C)(C)N(C)C)C2C1 CC1(C(N2CCCC2CNCC(O)CN2CCOCC2)=O)CC=CCC1 C1(OC)(OC)CCC1C(=O)NCC1CCC1NC(C1CCN(C)C1)=O C1(CNC(=O)CC2CC3(CCC3)C2)COCCN(C(C2CC3CCC(C2)O3)=O)C1 c1(C(N2C(C)CC(CNC(c3cncc(Cl)n3)=O)C2)=O)coc2ccc(Cl)cc12 C1(CNC(C(C)OCC(C)C)=O)CN(C)CCN1C(c1cn2c(n1)CCC2)=O C(=O)(CCC(N)=O)NCC1(CNC(CN(C)CCO)=O)CCCC1 c1(C(N(C)CC2(NC(C=Cc3scc(C)n3)=O)CC2)=O)cnc(N(C)C)c(Cl)c1 C1(C(CO)NC(c2ccccn2)=O)CCN(C(=O)C(F)n2ccnc2)CC1 O=C(CCCCCF)NC1(C(=O)NC23CC(F)(C2)C3)CCSC1 N1(C(C=NOC)=O)CC2CCN(C(c3cccc(F)c3Cl)=O)C2C1 C#CCCCC(C)C(=O)N1CC=CCC1C(N1CCC(C(N)=O)C1)=O.C(=O)CC CC1(C)C(O)C(O)CCN1C(c1cccc(S(C)(=O)=O)c1)C(=O)NCC1CCOC1 C1(NC(c2c(OCC)c(F)ccc2)=O)CN(C(c2cnc(C)o2)=O)CC12CCC2 C(CCC(C)(C)C(=O)NCC1(C)CCCO1)NC(C1CC(CC)C1)=O C=CC(C(=O)N1CC(O)(C(F)C(=O)NC(CC)C2CC2)C1)OC CC(C)CCCCCC(=O)N1CC(C)CN(C(=O)CC2CCCSC2)C(C)C1 C1(NC(C(n2ccc(C)n2)C)=O)CCCC(C(N2CCCC2)=O)C1 C1(C#N)(CC(=O)NCC=CCNC(c2ccc(OC)o2)=O)CCCCC1 c1(C(=O)NCC2(CN(C)C(C3CCC4CCCCN34)=O)CC2)ccc(S(N)(=O)=O)s1 c1(C(N2C(CNC(c3cc(COC)cn3C)=O)CCC2)=O)cn2cccnc2n1 c1(C(N(CC(C)Sc2n(CC#C)cnn2)C)=O)ccc2c(N(C)C)ncnc2c1 N1(C(C)=O)CCC(C)(OC(C)(C)C2CN(C(c3sccc3C)=O)C2)CC1 Cn1ccc(C(C)(C)C(=O)NCC(C)(C)CNC(c2ccc(Cl)[nH]2)=O)n1 C=C(C)C(CC(=O)N(C)CC1CCCC1NC(c1cnc(N(C)C)s1)=O)OCC c1(OC)ccnc2c1CN(C(N1CCN(CCCO)CC1)=O)CC2 C1(C)CCC2(CC1)CC2.c1(SC)cncc(C(=O)NCC2CC2CNC(=O)C2CC2)c1 Cc1ccc(C(=O)NC2CCC(C)N(C(c3ccc(F)s3)=O)C2)nc1C C1(CCNC(c2c(C)onc2)=O)CCN(C(=O)CCCCC(C)C)CCC1(F)F c1(C(=O)NCC(CNC(c2cccc(OC)n2)=O)OC)nc2c(s1)CCCC2 C(=O)(CCP(C)(C)=O)N1CC(C)C(CCNC(c2sccc2CO)=O)C1 N1(C(Cn2cc(C(C)=O)nn2)=O)CC(CNC(=O)COC(C)C)CC1C N1(C(C2C(CC)N(C)CC2)=O)CC(NC(c2cccc(C(F)F)c2)=O)C2(CC2)C1 CC1=C(C(=O)N2CCCCC2CCNC(=O)Cc2cn[nH]c2)CCC1 c1(C(=O)NCC(CCOC)NC(C2CCCCS2)=O)cc2c(n1C)CCOC2 c1(C(=O)NCCCOC2CCN(C(CC(C)F)=O)CC2)cnc2sccn12 C(C(CC(C)C)NC(C1(C)CCN(C)C1)=O)NC(CCCOC(C)=O)=O C(=O)(CC(C)(C)C(F)F)NC(CC)C(=O)NCCOCCCC(C)C CCCC(C#N)C(=O)N1CC(N2CCN(C(C3CS(=O)(=O)CCO3)=O)CC2)C1 C1(C(N2CC(CCOC)C2)=O)(CC)CCN(C(c2c[nH]c(C)cc2=O)=O)CC1 c1(C(N2CC3C(NC(CC(CCC)(C)O)=O)C3C2)=O)cc([N+](=O)[O-])ccc1NC CC(C)(O)C(C)(C)C(=O)NCC1(F)CN(C(c2ccn3c2CCCC3)=O)C1 C(C(CNC(c1nc(Br)c[nH]1)=O)C(F)(F)F)NC(c1c(C#N)scc1)=O N1(C(C2CCN(C(C)=O)C2)=O)CCCC(F)(C(=O)NC(C)(C)CCCF)C1 C#Cc1ccnc(C(=O)NCC2(NC(=O)C=CC3CCCC3)CCCCC2C)c1 C#CCCCC(C)C(=O)N1CCCC(F)(CNC(C)=O)C1 c1(C(=O)NC(CN(C(C=C(C)C(C)C)=O)C)C)cc(F)cc(C)c1N N1(C(C2(C)CCCN(C(c3cccnc3F)=O)C2)=O)CC2CSCC(C2)C1 N1(C(CS(=O)(=O)N(CC)CC)=O)CCC(C)(C)C(NC(c2ccnn2C)=O)C1 N1(CC)CCOCC1C(=O)NCCCC(C)NC(c1cnoc1C1CCC1)=O c1(C(N2C(C)CCC(NC(C3(OC)CCOCC3)=O)C2)=O)cn2cccnc2n1 C1(CCNC(C2CCCO2)=O)CCCN(C(c2ccc(C(F)(F)F)o2)=O)CC1 c1(C(=O)NC2(CF)CCN(Cc3c(C)cccc3)C2)ccc(F)c(C(F)(F)F)c1 Cc1nccc(CNC(C2(CNC(=O)CCCF)CC(C)(C)C2)=O)n1 N1(C(C2N(C(c3c(O)ccc(C)c3)=O)C3C(C2)C3)=O)CC2CCCC(C1)N2C C1(OC(c2ccc(OCC#C)cc2)=O)CCC(C)N(CCOc2ccccc2)C1=O C(=O)(C(F)(F)C(C)O)NCC=CCNC(C(C(C)C)N1CCN(C)CC1)=O C1(NC(CN(C(C(C)C)=O)C)=O)CCCC(CNC(=O)C(=Cc2cccs2)F)C1 c1(C(=O)N(C)Cc2cc(Br)ccn2)oc(C(=O)OC)cc1C(=O)O N#Cc1c(F)ccc(S(=O)(=O)N2CCC(=O)C23CCCCC3)c1F CC(O)CCCCCC(=O)NC(c1ccccc1)CNC(=O)C(C)(C)CF C1(C(=O)NC2CCN(C3CC3)C2)(COC)CCCN1C(=O)C(N1CCC(C)C1)=O C#CCCCC(C)C(=O)NCC12COC(C1)C(NC(=O)CC(=O)O)C2 N1(CCSC)CCCN(c2ccc(Cl)cn2)CC1.C1(C2C(=O)N2)CC2C=CC1C2 N1(C(C(CC(C)C)OC)=O)CCC2CCCC(C1)N2C(=O)Cc1cncnc1 N1(C(C2=C(C)OCC2)=O)CCC2(CC1)CN(C(C1CCCC(C)CC1)=O)C2 c1(OC)cc(C)nc(NOC2CCN(C3CCOC3)CC2)n1 c1(-c2cc(O)ncc2)nncc2ccoc12 Nc1c(C(=O)NCCCC2CCCN2C(=O)C=CC2CCOC2)cccc1Cl C12(NC(C(C)NC(CC)=O)=O)CCCC1N(C(c1ccc(Br)cn1)=O)CC2 C=C(C)C(C)(C)C(=O)NC1CC(CC(=O)NCCOC)C1 Cc1cc(Br)cc(S(=O)(=O)NC2CC3CC2CN3C(c2ccncc2)=O)c1 N1(C(C=CS(C)=O)=O)CCC(NC(=O)Cn2ncc3ncccc23)C12CCC2 C(=O)(CCCCN(C)C)NCC(CO)NC(C(c1ccccc1Cl)OC)=O C(CC(C)(C)C)(C(=O)NCCCCCC(=O)N(C)Cc1cc(C)cc(C)n1)OC C(=O)(CC(C)(C)CNC(C1CCCN1C(C)C)=O)NCCC(C(=O)OC)C C(=O)(C(F)CC(C)(C)NC(=O)C(C)(C)C#N)Nc1ccc(OC)cc1C CCCCCC(O)C(=O)NC(CNC(=O)C(c1cnn(C)c1)C)(CC)CC N1(C(C=C(C)c2ccco2)=O)CCC2C(C1)CN2C(=O)CNS(=O)(=O)N(C)C Cc1cc2occ(C(=O)N(C3CN(C(C4CCNC(=O)C4)=O)C3)C)c2cc1C N1(C(CC2(C)CC2)=O)CC2CN(C(=O)CC3(O)CCOCC3)CCC2(CO)C1 N1(C(COC(C2CC(=C)C2)=O)=O)CCCC(NC(C)(O)C(C)C)C1 C1(CC(=O)NC(C(=O)NC2(c3cnn[nH]3)CC2)C2CCOC2)CCCC1 C1(C(=O)NCC2CCC(NC(c3ccccc3C(N)=O)=O)CC2)(CC)CCNC1=O c1(N(CCC)CCN(C(=O)C(C)(C)CC)CC)ncnc2cccc([N+](=O)[O-])c12 Cc1c(C(N2CCC(NC(=O)CC3CCC3)C(CO)CC2)=O)nn2ccccc12 C1(C(=O)NC2(CCC)CCN(C(C3CCCO3)=O)CC2)CC2(CCOCC2)CO1 C(C(C)(CC(C)C)NC(=O)Cc1cccc(Cl)c1)NC(CCC=CCC=C)=O C1(C)(C(=O)NC(C)CCCNC(c2c[nH]ccc2=N)=O)Cc2ccccc2C1 N1(C(CN(CCCCCC)C)=O)CC2CCC(N(C(=O)CN3CCC3)C)C2C1 C1(C(=O)NC2CCC(NC(C(c3ccc(C)s3)C)=O)CC2)CN(CP(C)(C)=O)C1 CC(C)CC(C(=O)NCC1CSC1)NC(=O)C1=CCCC1 c1(NC(C=CC(C)(C)C)=O)ccc(CC(=O)NCCCCO)c(F)c1 CC1CC1C1CC1C(N1CC(NC(c2coc(C)c2)=O)CC1C)=O.n1(CN)cccn1 c1(C(=O)NCCCC(C)NC(CC2(CSC)CC2)=O)coc2cc(F)cc(F)c12 CN1CC(C)(C(=O)NCC(C)(C)NC(C2C(C(F)F)C2(C)C)=O)CCC1=O C(=O)(CC(C(C)C)NC(=O)Cc1ccoc1)NC(CCC)CCC C12COCC1NC(=O)CN(CCCC)C2=O.C(=O)(CN(C)C(C)C)NC C1(C2CCN(C(C3CNc4ccnn4C3)=O)C2)(NC(c2ccco2)=O)CC1 c1(C(N(CCCNC(=O)C(F)CC2CC2)CC)=O)[nH]c2c(C)cccc2c1C c1(C(=O)NCC(C)NC(CN2CCC(C)C2)=O)[nH]ncc1C#N C1(NC(=O)Cn2cccn2)CCN(C(c2ccc(CO)cc2F)=O)CCC1(F)F c1(C(=O)NC(CC)CNC(c2cnc(C)cn2)=O)cc(C)cc([N+](=O)[O-])c1 c1(NC(C2CCN(C(c3c(CC)nccc3)=O)C2)=O)ccc(C#N)cn1 c1(CNC(CCN(CC#C)C(C2CCCS2)=O)=O)nn(C)cc1CO c1(C(=O)NC(CNC(CC2(C=C)CCC2)=O)(C)C(C)C)cn2c(n1)CCC2 n1(CC(=O)NCCC2CCN(C(C3(F)CCC3)=O)C2)nc2c(n1)CCCC2 CC#CCC(C(=O)Nc1csnc1OC)NC(=O)Cc1cn(C)nc1C Cc1cc(C)c(C(N2C3CCC2CN(C(=O)CC2(C(F)F)CC2)C3)=O)cc1C N1(C(CCc2onc(CC)n2)=O)CCCN(C(c2coc3c2COC3)=O)CC1C C1(NC(c2ccc(CO)cc2F)=O)CC2CCC1N2C(=O)CC1CCCCCC1 c1(C(=O)NCCOCC(=O)NC2C(C)(OC)COCC2)cc(O)nc(O)n1 C1(OC)CN(C(=O)CC2CCCC2NC(=O)CC2(NC(C)=O)CC2)CC(C)(C)C1 N1(C(C(C(C)CNC(C2CC23CCC3)=O)F)=O)CC=C(C(C)(C)C)CC1 CC(C)C(C(=O)NCCCOCCNC(c1ccncc1)=O)c1cccc(Cl)c1 C1(CNC(=O)C=Cc2cccnc2)CCCCCN1C(C1(F)CCOC1)=O N1(C(CCC(C)O)=O)CCCC12CCN(C(c1cc3ncccc3s1)=O)C2 CCC(C)CCCC(=O)NCC1(CC(=O)NCC(O)C(C)C)CC1 C12(NC(Cc3c(C)cco3)=O)CCN(C(c3cnn(CCO)c3N)=O)CC1C2 N1(C(C=C=C(C)C)=O)C2CCC(C2)C1CNC(C1CC(C)(O)C1)=O C1(NC(CC2(C=C)CC2)=O)CCC(C)N(C(=O)CN2CCOC2=O)C1 c1(C(=O)NC2CC(C)N(C(c3cc(CO)nc(Cl)c3)=O)C2)c[nH]nc1S(N)(=O)=O c1(CNC(N2CCNC(=O)C23CC3)=O)ccc2c(Cl)ccnc2c1 CC1(C2CN(C(C3(C)CN(C(c4cc5ccccc5[nH]4)=O)C3)=O)CCO2)N=N1 c1(C(=O)NCCC2(O)CCN(C(c3ccc(OC)nc3)=O)C2)c[nH]cc(C)c1=O c1(C(N2CC(C)(NC(c3ccc(=NC)[nH]c3)=O)C2)=O)cnc(O)c([N+](=O)[O-])c1 Cc1cccn2nc(C(N3CCCC(C)(NC(c4ncncc4Cl)=O)C3)=O)cc12 c1(C(=O)NC(C2(O)CCN(c3nccc(SC)n3)C2)C)cnc2ccccc2n1 c1(SC)cc(F)ccc1C(N1CCC(O)C(C(=O)NCCn2ccnn2)C1)=O CC1C(C)C1N=c1[nH]c(-c2ccccc2)nc(=NCC(F)C2CCCCC2)[nH]1 CN1CCN(C(=O)CCCN=[N+]=[N-])CC1CNC(=O)C(C1(O)CCCCC1)(F)F c1(C(N(CC(C)CNC(=O)C(C)Cc2ccco2)C)=O)ccc2c(n1)CCCC2 c1(N2CC(CN(C(C=CC=CCC)=O)C)C2)nnc(Br)s1 c1(C(N2CC(O)(C(C(=O)NC(c3ccco3)C#C)F)C2)=O)cncnc1C C(=O)(C1CCCc2scnc21)NCCCNC(C1N(C)S(=O)(=O)CC1)=O CCC(CC(=O)NCCOCCC(=O)N(C(C)C(=O)NC(C)C)C)SC c1(C(=O)OC)c(NC(c2sc(NC(=O)CCCCN)nc2C)=O)sc(C)c1C N1(C(c2n[nH]c(CC)c2C)=O)CC=C(C(=O)NCC2CCOC(C)(C)C2)C1 N1(C(c2n(C)cc(Cl)c2)=O)CCC(NC(c2ccn(C(F)F)n2)=O)C(C(N)=O)C1 C(=O)(C1=CCCCO1)Nc1cn(CC23CC(NC(C4CNC(=O)O4)=O)(C2)C3)nc1 c1(C(c2nnnn2C2CCCCC2)NC(CC)CSC)ccccc1OC(F)F CC(c1ccccc1)=CC(=O)NCCC1(NC(=O)C(C)SCC=C(C)C(=O)O)CC1 Oc1cccc(SCC=Cc2ccc(N3CCOCC3)cc2)c1Br N1(C(C2(c3cccc(C)c3)CC2)=O)CC(CO)C2(CC2)C1.C12(CC1)C(=O)N2 C1(NC(C(C=C)(C)CC)=O)CN(C(C2CCC(C(=O)OC)CC2)=O)C2CCCCC12 N1(C(C(CN(C(c2nn(CC)c(C)c2)=O)C)(C)C)=O)CCS(=O)CC1C C1(C(C(N2CCC(NC(=O)COCCCF)C2C2CC2)=O)O)CCCCCCC1 n1(C(C)C)ncc(C(=O)NCC2(NC(=O)C(c3ccc(Cl)s3)C)CCOC2)c1N N(C(=NCCCN1CCCOCC1)NC1CCCCC1)Cc1c(C)scc1 c1(C(N2CCC(C)(NC(CN3C(=O)CC(C)(C)O3)=O)C2)=O)cn2ncccc2n1 C1(NC(C2CCCC(F)C2)=O)(CNC(C2Cc3nccn3C2)=O)CCCCCC1 N1(C(c2ncn(CC)n2)=O)CC2(CC2)CC1CNC(=O)Cc1c(F)cccc1F C1(CNC(CNC(N)=O)=O)CCCN(C(=O)CCCOc2cccc(Cl)c2)C1 C(=O)(C1=C(C)CCCC1)NC12CC(NC(c3ccc(OC)c(N)c3)=O)(C1)C2 C(=O)(C(C)(O)C(F)(F)F)N1CCN(C(COC2(C)CCC2)=O)C(CO)C1 N1(C(C(c2c(C)n(C)nc2)N)=O)CC(C)C(CO)C(C)C1 C1(C(=O)NCC2(C(=O)OC)CC2)CCCC1NC(C1CC12CC2)=O C(=O)(CC(C)C(F)(F)F)NCCN1CCN(C(CN2CCC(C)C2)=O)CC1 c1(C(=O)NC2(C)CCCN(C(Cc3c(C)nsc3)=O)C2)cc(F)c(C(C)C)cc1F C=C(C)CCCC(=O)N(CCC(C)(N)C(F)F)C Cc1csc(C)c1C(=O)N(C(C)CNC(c1coc(C(N)=O)c1)=O)C CN1CC(C(=O)NC(Cc2ccccc2)CCNC(=O)C(C)(C)F)CCC1=O C1(CN(CCCS(C)(=O)=O)C(C)C)CCC(C)NC1=O N1(C(C(=O)NC(C)C)=O)CC(NC(=O)C=CS(C)=O)CC(C(F)(F)F)C1 C1(NC(C2(NC(=O)CC3CCC(=O)N3)C(C)C2)=O)CC2CC(C(N)=O)CC12 C1(O)(CNC(c2ncc(F)cc2F)=O)CCCN(C2CCc3c(F)cccc32)C1 c1(C(=O)NC2CCCN(C(C(C)P(C)(C)=O)=O)C2C)nc2ccccn2c1F C(C1CC(C)(C)Oc2ccccc21)NC(=NCC)NCC(CC)(CC)CC CN1CC(NC(C2(C)C=CCN2C(c2nonc2N)=O)=O)C2(CC2)C1=O C1(C(=O)NCc2c(CC)onc2C)CCN(C(=O)CCCN(C)C(C)C)C(C)C1 CC(C)C(C(=O)N1CC(CNC(c2ccoc2)=O)C(O)C1)c1ccccc1 CCC(CC(C)C)C(=O)N1CC(CNC(c2ccc(C(C)C)nc2O)=O)C(C)C1 N1(C(C2COCC(C)O2)=O)CC2CC1CN2C(=O)Cn1cccc(O)c1=O N1(C(Cc2c(C)scc2)=O)CC=CC(NC(=O)C=Cc2cc[nH]n2)C1 c1(CC(=O)NCC2CN(C(c3c(C)nc[nH]3)=O)CC2(C)C)cccc2c1OCO2 N1(C(C(C2CCCO2)NC(C(CC=C)NC(C)=O)=O)=O)CC(CO)C2(CC2)C1 CC(C)C(CO)C(=O)NC1CC(CNC(C2(O)CCOCC2)=O)C1 Cc1cccc(C)c1C(=O)NCC1CCCCN1C(c1cc(O)nn1C)=O C(C(=O)N1CCC(C)(NC(c2cnn(CCO)c2)=O)CC1)(C(C)(C)C)N(C)C C1(NC(c2cc[nH]n2)=O)(CO)CCCN(C(c2ccc(-c3ccco3)s2)=O)C1 C#CCCCCCCC(=O)N1CCN(C(=O)C#CC2CCCOC2)C(C(C)C)C1 Cc1c(C(N2CC=CC2C(=O)N(C)CC2CCC2)=O)ccn1C c1(C(=O)NCCCN(C(=O)CC2CC=CCC2)C)ccsc1Br c1(C(=O)NCC2CN(C(C3CC3(F)F)=O)CCCO2)cc2n(n1)CCCO2 c1(C(N2C(C(=O)NC3CC=CC(C)CC3)CCC2C)=O)ccc2c(c1)CCC2 N1(C(C(CSC)(C)C)=O)CC2OCC(NC(C3COCCN3C)=O)C2C1 c1(C(=O)NCC2N(C(CC)=O)CC=C2)cccc(-c2cnccn2)c1 C1(CC)CCN(C(=O)CC#N)C1CNC(=O)CCc1cc(C)[nH]n1 C(=O)(C1=CCN(C(=O)CNC=O)C1)N(C(C)CCO)C c1(C(=O)OC(C)(C)C)sccc1NC1CCC1C(=O)NS(C)(=O)=O c1(NC(CC2CCN(Cc3cccc(C)c3Br)CC2)=O)cccc2nccnc12 O=C(C1=NOC(n2cccn2)C1)NC1CC(NC(=O)CC2CCCS(=O)(=O)C2)C1 CC(c1ccco1)=CC(=O)NCC(c1ccc(Br)cn1)=O C(=O)(C(C)CC(C)C(C)=O)N1CCC(C(=O)NC(CC(=O)NC)C)CC1C C1(CC(=O)NCC(C)CNC(=O)CC2CC(=O)NC2=O)C(C)(C)C1(C)C CCCC(C)C(=O)NCCCN(C(=O)CC1CCCCC1C)C(C)C C=CC(C)C(=O)NCCN(C(=O)CC1CC(F)C1)C c1(NC(CCNC(C)CC(N2CCCC(CC(N)=O)C2)=O)=O)cccc(N)c1 S(=O)(=O)(c1ccc(F)cc1C(=O)O)N1C2CN(Cc3c(CC)nccn3)CC21 N1(C(C2N(C(C=C(COC)C)=O)CC3(CC3)C2)=O)CCC(CO)C(C)(C)C1 n1(CCC)cc(C(=O)N(C)CCN(C)C(c2coc(C)c2)=O)c(C)n1 c1(CSC)cc(C(=O)NC(C)CCNC(c2cc(O)cc(O)n2)=O)ccc1F N1(C(c2ccc(SC)o2)=O)CC2(CCCCN2C(c2nccn2C)=O)C1 C1(O)(CN(C(C(C=CCCC)O)=O)C)CCN(C(=O)C(C)(C)c2ccccc2)C1 c1(CC)ccnc(C(N2CCC(CCC(=O)NCC3CCCC(CF)C3)C2)=O)c1 CCCCC(O)CC(=O)NC(C)C(C)(C)NC(=O)C=C1CCN(C)C1 C1(C(N2CCC2C(C)O)=O)(NC(CNC(=O)OCC=C)=O)CC1(C)C c1(C(=O)NCC2N(C(CC=CC)=O)CCC2C2CC2)ncn2cc(Cl)ccc12 c1(CC)c(Cl)nc(C)[nH]c1=NC(C)CNC(c1cnsn1)=O C=CCCCC(C(=O)NCc1ncccc1O)NC(c1cc(C)c(C)o1)=O C12(C(=O)NC(CNC(C(C(C)C)O)=O)(C)CO)CCC(=O)N1CCS2 C1(NC(C2(CC=C)CCOCC2)=O)CCN(c2nnc(C3CC3)s2)C(C)C1 N1(C(COCC(=O)NC)=O)CC(CNC(c2cccc(O)n2)=O)OC(C)(C)C1 C1(CNC(C2C(C)CC2)=O)CN(C(c2ccnc(OCC(F)(F)F)c2)=O)CCO1 c1(NC(C(C2CC(F)(F)C2)OC)=O)sc(Br)cc1F C1(CCC)CN(C(C2CCC3(CC2)CC3)=O)CCN1C(=O)C(O)CCn1cncn1 C12(NC(c3cnc(C)n3C)=O)CCCC1N(C(=O)C=Cc1ccc(O)cc1)CC2 C1(O)(CCNC(C(C)SC(F)(F)F)=O)CN(C(c2ccnn2C2CCC2)=O)C1 C=C(C)CCCC(=O)N1CC2CC1C2NC(c1cn2ccsc2n1)=O CC(CC(=O)NCCN(C)C)n1cccn1.C12(C)CN(C1)C(=O)C1CC1C2=O c1(-c2cc(C(=O)NC3C(NC(=O)CC45CCCC4C5)C3)no2)ccc(Cl)cc1 C1(CNC(C2CCC(CC)CC2)=O)CN(C)CCN1C(C12CCC(CO1)C2)=O C(=O)(CC(C)CC(=O)NC(=O)CCCCN(CC)CC)NCC1(C)CC(CC)C1 C(=O)(CC1=CCOCC1)NS(CCc1n(C)ncc1)(=O)=O Cc1c(Cl)ccnc1C(=O)NCC(C(C)(C)C)NC(C1CCN(C(C)C)CC1)=O N1(Cc2ccc(OCC#C)nc2)CCNC(=O)C1CC(F)(F)F c1(C(=O)NCC(C(C)(C)C)NC(C2CCC3CC2CO3)=O)ncn2c1CCC2 N1(C(C(CNC(C2OCCC(C)C2)=O)O)=O)CC2(CCC(=O)N2)C1 c1(-c2ccc(CNC(=O)CCCC(F)(F)F)cc2)ccc2c(=O)ccoc2c1 N1(C(C=CCCC(C)C)=O)CCN(C(c2ccc(=N)[nH]c2)=O)C(C2CCC2)C1 Cc1cc(C2CCCN2C(=O)NCCC2CC23CCOCC3)ccc1Br c1(C(=O)NCC2CCCCN(C(C(C)=C3CC3)=O)C2)ccc(N=[N+]=[N-])cc1 N1(C(COC(C)=O)=O)CCCC(C(C)NC(=O)Cc2sc(C)cc2Br)C1 c1(N2CCC(c3c(C)nc(C)s3)C2)ncnc2c1ncn2C1CCCC(O)CC1 Cc1cc2ncn(CC(O)CNC(c3cccs3)=O)c2cc1C C#CCCCC(=O)N1CC(NC(=O)CC2(N3CCCC3)CC2)C(O)C1 C(=O)(C(COCCCN(C(COCC)=O)C)OC(C)C)NCCCCS C(=O)(NNC(=O)c1cccnc1-n1cc(C(=O)O)nn1)c1ccn(C)n1 C1(C(C)C)CCC(C)CC1Cn1cc(-c2cncc(Cl)c2)nn1 C1(C(=O)NCc2onc(CC)n2)CC(F)CN1C(C1CCO1)=O C1(CC=C)(NC(c2cnc(C)s2)=O)CCN(C(C2CCCC2CCC)=O)C1 N1(C(=O)NC(c2nc(C(C)C)cs2)CC)CC(C)C(C)(C(F)(F)F)C1 N1(CC(=O)NC(CN(C(c2cnc(C)s2)=O)C)(C)C)C(=O)NC(C)(C2CC2)C1=O C(=O)(CCCCC(=O)NCC1(O)CCCN(C(=O)C(C)NC(C)=O)C1)OC C1(CCC)C(=O)NCCN1C(=O)C=CCC(C)(C)NC(c1coc(CO)c1)=O c1(NC(C2CC=CCC2)C)ccc(S(=O)(=O)N(C)CCn2cnnn2)cc1Br C1(NC(N)=O)CCN(C(=O)NC2CCN(C(=O)NC3CCC3)CC2)CC1 C#CCCCC(C)C(=O)NC(C)CC1CCN(C(c2[nH]cc(C)c2C)=O)CC1 c1(C(N2C(CNC(C(N3CC(C)C3)C)=O)CCC2)=O)ccc(SC(F)(F)F)cc1 C(CCNC(=O)CCC1CCCO1)(C(=O)NCCN1CCC1)OC Cc1cc(C2CCCN2C(=O)NCc2ccnn2C#N)ccc1Cl N1(C(C(C=C)(F)F)=O)CC(O)(C2(CNC(=O)COCC3CCOC3)CC2)C1 C1(C(=O)NCC(CNC(C2(COC)CCCO2)=O)O)CCCC2(CCC2)O1 Cc1scnc1C(=O)NCCOCCCNC(c1cnn(C2CCC2)c1)=O N1(C(=O)OC(C)(C)C)CC(CCNC(N2CCCC2c2nnc(O)o2)=O)C(C)C1 CC(C)C(C#N)C(=O)N1CCOCC(NC(=O)CCCOc2cccnc2)C1 N1(C(c2nc(CC)oc2)=O)CC(NC(=O)Cc2ccn(C(F)F)n2)C(O)C1 c1(C(=O)NCC(CCCC)NC(=O)COCC)cc2c(cnn2C)nc1C N1(C(CN2CC(CC)C2)=O)CCN(C(=O)CC2(COC)CC2)CC(C)(F)C1 C1(CNC(c2c(C)cc(F)s2)=O)CC(C)(C)CN1C(C1CCC(F)(F)CC1)=O c1(C(=O)NCC(C(C(C)C)C)NC(=O)Cc2ccsc2)cnc2c(c1)nnn2C C1(C(N2CCC(O)CC(C)C2)=O)(NC(=O)OC(C)(C)C)CC2(CCCCC2)C1 C1(N(C)C)CCC(C(=O)NC(CCCNC(=O)COC2CC2)c2ccccc2)CC1 N1(C(c2c(CC)ncs2)=O)CC(NC(C2CC2c2ccn(C)n2)=O)C2(CCC2)C1 CC(C)C(O)C(F)(F)C(=O)NCC1(F)CCCN(C(=O)COC(C)(C)C)C1 c1(C(=O)NC(C2(O)CN(C(C3CC(C)(F)C3)=O)C2)C)cscc1-c1ccccc1 c1(C(=O)NC2CN(C(C(C)OCOC)=O)C2)cnc(-c2ccccc2)s1 c1(C(O)CF)nnc(C(F)(F)F)o1.c12noc(n1)C2F C12(COC)CCC1CN(C(=O)C(O)CN1CCCC1)C2.c12ccoc1CNC2=O c1(COC)cc(C(=O)NCCC(C)NC(C2(C#N)CC23CCC3)=O)ccc1F c1(C(N2CC(C3CC3)C(NC(=O)C(O)C3CC3)C2)=O)ccccc1[N+](=O)[O-] N1(C(CONC(C2CCOC2CNC2CCCSC2)=O)=O)CCc2sccc2C1 N1(C(C2C(=C)CC2)=O)CC2(C1)CN(C(c1cc(C)ccn1)=O)CC2CO N1(C(C#C)=O)CCCC(C2CN(C(c3cc(C)c(Br)cc3Cl)=O)C2)C1 C1(OC)(CNC(=O)C(C2CC2)NC(C)=O)CCN(C(C2CN(C)CCO2)=O)C1 CN1c2ccccc2C(NC(=O)NCC23CCC(CO2)C3)CS1(=O)=O N1(C(CCCOCCOC)=O)CCC(F)CC1C(N1CCCN(C(C)C)CC1)=O c1(CCC(=O)NCCN(C(COC)=O)CCOC)cc(Br)ccc1C C(=O)(C(CC)C(=O)NCc1ccc(CNC(=O)CS(N)(=O)=O)cc1)OCC C(C(C(=O)N1CCC(OC(C)C)C1)NC(=O)CC1CC1)SCC.C1(OC)CCOC1 C(=O)(CN=C(NCC(C)(C)C(F)(F)F)NCC1(OC)CCC1)NC C1(CCNC(c2nnn(CC)c2C)=O)CCN(C(c2ccccc2F)=O)C(C)C1 N1(C(c2cnc(SC)s2)=O)CCC(C(=O)NCc2ccc[n+]([O-])c2)C(O)C1 Cc1ccn2cc(CNC3CNCCCC3C(F)(F)F)nc2n1 C1(C(=O)NCC2CCCC2CNC(c2ccc(Cl)nn2)=O)(OC)CCSCC1 N1(OC2(COC)CC2)CC(=O)N(CCc2ccc(Cl)cc2Br)C1=O Cc1cc(F)ncc1-c1cn(CCCN(CC(=O)NC(C)C)C(C)C2CC2)nn1 C1(NC(C(Cc2c(C)nc[nH]2)O)=O)CCN(C(C2CN(C(N)=O)C2)=O)CC1C C12(CN3CCN(c4nc(SC)nc(C(F)(F)F)c4)CC3)CCCCCC1OCC2 c1(C(=O)NC(CNC(CC2(C=C)CCC2)=O)C(C)C)cc2c(F)cc(Cl)cc2[nH]1 c1(C(=O)NC2CCC(NC(=O)C#CC3CCC3)CC2)ccc2ccsc2c1 C(=O)(NNc1ccc(S(=O)(=O)CC)cc1)C1CCC(C)(C)O1 N1(C(Cc2cc(C)sc2)=O)CC2CC(NC(=O)Cc3ccnc(F)c3F)C(C2)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])N1CC(CC)N(C(c2ccn(C3CCC3)n2)=O)CC1 C1(C(N2CCCCC2C2(C(F)(F)F)CC2)=O)COC2(CCC2)CO1 CS(=O)CCC(O)C(=O)NCC1(F)CC(CNC(=O)C=CBr)C1 C1(NC(C2OCCN(CC)C2)=O)CCC2(CC1)CN(C(=O)C1=NOCC1)CCO2 C(=O)(C(C)C(F)F)N(CCOCCC(=O)N(CCCOCC)C)C c1(C(=O)NCC2C(NC(c3cc[nH]n3)=O)CCC2)cnn2c(=O)cc[nH]c12 N1(C(C2C(OC(C)=O)C2)=O)CC(C(N2CCOCC3(CC3)C2)=O)C2(CCC2)C1 N(C1CCc2ccccc21)C(CCC1C(NC(c2c(C)ocn2)=O)CCC1)=O c1(C(=O)NCC(CO)ON)cc(C2CCCCC2)cc(Cl)c1O N1(C(c2cncc(SCC)n2)=O)CCC(C)C(CNC(=O)CC(C)C)C1 Cc1cc(Cl)cc(C(N2CCN(C(=O)Cc3cnc(C4CC4)[nH]3)CC2C)=O)c1O C(c1c(Cl)cccc1Cl)=CC(=O)NCC(CNC(C=CCOC)=O)C(F)(F)F C12(NC(C#C)C3CC3)CCC(NC(C3(c4cc(C)ccn4)CC3)=O)(CC1)CC2 c1(C(CNC(C2CCC(C)(CC)O2)=O)N(CC)CC)ccc(Cl)cc1 CC12CN(C(C3CCCCCN3C(=O)NC)=O)C(C(=O)NC(C)(C)C)(C1)C2 C1(CNC(CCC(=O)NCC)=O)CC2CCC1N(C(=O)C(C)CSC)C2 c1(C(=O)NCC2(O)CCN(C(C3(C)CCCS3)=O)C2)ccc(Br)c(F)c1 c1(CCC(=O)NCC(=O)NCc2cn(CC#N)nn2)nc2ccccc2s1 c1(OC)cc(C)cc(C(=O)NCC#CCNC(=O)CC2C(C)(C)C2(C)C)c1C N1(C(C2(OC)CCCC2)=O)CC(NC(=O)Cn2nnc(=O)[nH]2)C(O)C1 c1(CC)cc(CC(=O)N(C2CCN(C(=O)C(c3cnn(C)c3)OC)C2)C)n(C)n1 C1(C(N2Cc3ccncc3C2)=O)C2CC(CC2F)N1C(c1cc(Cl)cnc1F)=O C(=O)(C(F)C(F)(F)F)N1CC(C)(NC(C2CC(C)(F)C2)=O)C1 C(CC(C(=O)NCc1nnc(CO)s1)NC(=O)C(c1cccn1C)=O)N(C)C C(=O)(CC(C)CCC(=O)NC1(C)CN(C(C2CCS(=O)(=O)N2)=O)C1)OC N1(C(C(COC)(C)C)=O)CCC2(CCCCN(C(=O)CNC(C)=O)C2)C1 C=CC(C)C(C)C(=O)NCCN(C1CCCC1)C(=O)C=Cc1sccc1C c1(CC(=O)NC2CC3CC(NC(C(C=CC)O)=O)C2C3)c[nH]c2cccc(C)c12 N1(C(c2cc(C)sc2Br)=O)CCC2(NC(C3CC3(F)F)=O)CCCC12 c1(C(c2nnnn2C2CC2)N2CC2)cc(OC(C)C)n[nH]1.CO C1(C)(NC(C2C(C(c3nnc(-c4ccco4)o3)NC(C)=O)CC2)=O)CCCOC1 CC(C)C(C)C(=O)NCC(C(N1CCC(OC)CC1)=O)N(C)C N#CC12CC(C(=O)NCc3ccc(C(=O)NCC(c4ccco4)O)s3)(C1)C2 c1(C2ON=C(c3ccccn3)C2)ccnc(-c2nccc(C(F)(F)F)n2)n1 CC1CCC(CC(=O)N(C(=O)CN2CCCC2CCn2cccnc2=O)CCl)CC1 c1(CNc2c(C)c(NC3C(C)CC3C)ncn2)n[nH]c2c1CCCC2 N1(C(COCC(C)C)=O)CCC2C1CCCN2C(=O)CN(C)C(C)C n1(CC(=O)NCC(CNC(C(C)OC2CCC(C)CC2)=O)O)cnc([N+](=O)[O-])c1 c1(C(N2CC3(C(NC(=O)CC4CC45CC5)CC3)C2)=O)c(F)cc(Cl)cc1[N+](=O)[O-] N1(C(CCCC(CC)CC)=O)CC(=O)NC2CN(C(C3CCS3(=O)=O)=O)CCC12 N1(C(c2ccc(C)cn2)=O)CCC(NC(=O)Cc2cnoc2)C12CC2 CC(C)(C)CC(O)CC(=O)NCC(O)CNC(=O)Cc1ccc(C(N)=O)cc1 C1(CC)CCCN1C(=O)C(=O)NC(C)(C)C.C12(CN(C(=O)CC(C)C)C1)C(=O)NC2 C(C(C)(C(C)C)NC(=O)CSC(F)F)NC(c1cnc(CC(C)C)s1)=O S(=O)(=O)(c1ccccc1N(C)Cc1cn(C2C=CCCC2)nn1)NCC c1(C(=O)NC2CCCC2)nc(C(F)(F)F)n2ccncc12.C1CCC2(CC2)N1 c1(C(N(C2C(C)CCN(C(CCOCCOC)=O)C2)C)=O)cc2ccccn2c1 C1(CNC(=O)CCc2ccc(Cl)s2)CC2(C1)CN(C(c1ccnc(CO)c1)=O)C2 N1(C(c2n(CC)ccn2)=O)CCC(NC(=O)CC(C)(C)O)CC(O)C1 c1(CN2C(CCC(=O)NCCCCO)CCC2)ccc(C(F)(F)F)cc1I C1(n2c(-c3ccnc4ccnn34)nc(CCC3(C)CC3)n2)Cc2cccnc2C1 N1(C(CNC(=O)NC)=O)CCCC2(C1)CN(C(c1ccc(CF)cc1)=O)CCO2 c1(C(N2CCN(C(CCOC(C)C)=O)CC23CC3)=O)c[nH]c2ccc(O)cc12 C(=O)CCCN(C(C1CS(=O)(=O)C1)CO)CCO.C(C)(C(C)C)SC C(C(=O)N1CC(O)CC1C(=O)NCC1CN(C2COC2)C1)(C(C)C)SCC CC(O)CC(=O)NCC(O)CCNC(=O)CC1CCSC1 c1(C(=O)NCC(CNC(C2(C)CCCO2)=O)O)cc2[nH]ccc2s1 C=Cc1nc(Nc2nc(C(=O)OC)ns2)n(C)n1 c1(NC)c(C(=O)NC2CC(NC(C3CCCS3(=O)=O)=O)C2)sc2nccnc12 c1(CC(=O)NCC(C)CNC(=O)C(C)(C)C)nccc2ccccc12 CCC(C)(CNC(c1cccc(F)c1Br)C)C(C)O C(CNC(=O)C=CCOC1CCOCC1)(CC(F)(F)F)NC(C1(C#C)CCC1)=O c1(NC(C(C)(C)Br)=O)cnc(F)cc1CNC(c1ncncc1Cl)=O C(c1ccccc1)=C(OC)C(=O)N(C)CCN(C(=O)CCCOC1CCCC1)C C1(C(=O)NC2(C)CN(C(C3CC4(CSC4)C3)=O)C2)CC(c2ccccc2)=NO1 c1(C(=O)NCC2CC(F)(CNC(C(CC)SC)=O)C2)cn2cc(C)nc2s1 CC(C)CC(F)C(=O)N1CCC(CN(C)C(C2(C)CCCCC2)=O)C1 N1(C(CCCN(C(C)=O)C)=O)CCN(C(C2CS(=O)(=O)C2)=O)CC1C C1(C)(NC(c2c(OC)scc2)=O)CCCC1NC(C1CCCN1C=O)=O C1(CC=C)(NC(=O)CCC(F)F)CCN(C(c2cc(CC)no2)=O)C1.CCO C(=O)(C1CCCc2ccnn21)N(C(CC)CNC(=O)CC1(CO)CC1)C C#CC1(C(=O)Nc2cccc(CC)c2)CN(C(=O)CCOCC)C1 C(=O)(CCCCCSCC)NC(CC(=O)N(CCC)CC)CC1CC1 N1(CCN(C)C(C23CC(n4cc(C(c5nccs5)O)nn4)C2C3)=O)C(=O)CCC1=O N1(CCNS(CC)(=O)=O)CCC2C(CCCN2C(=O)Cc2cc(C)ccn2)C1 C1(NCC2(C(=O)Nc3c(C(F)(F)F)nc(OCC)[nH]3)CC2)C2CCOC2C1(C)C C(CCCCC(=O)NC1CCN(C(c2cc(C)ccc2Cl)=O)CC1CO)=CC CC(C(=O)Nc1cccc(CNC(=O)Cn2ccc(C(F)(F)F)n2)c1)C1=CCCC1 CCCC(O)(CCC)CC(=O)N1CCCC1Cc1ccc(F)cc1 c1(NC(C2N(Cc3cc(C)nn3C)CCC2)=O)cc(F)cc(Br)c1 S(=O)(=O)(c1ccc(NCCCC2CCC2)c(F)c1)NCC(C(C)O)(C)C CC1=C(C(=O)N2CCC(c3ccccc3)(CNCC3CCC4CC4C3)C2)CCCO1 N1(C(C(C)OCC#C)=O)CCC(C)CC1CNC(=O)CCCOCC C1(CS(=O)(=O)NC23C(CN(C(C(C(=O)NC)(C)C)=O)C2)C3)CC2(C1)CC1(CCC1)C2 C1(C(=O)NCC(=O)NOCc2ccc(Cl)cc2)(CO)CC12CCOCC2 C1(CNC(=O)CN2CCCC2=O)CCN(C(c2nnc(O)cc2O)=O)CC1(F)F c1(C(C(=O)OC)NC(c2sc3[nH]cnc(=S)c3c2C)=O)ccc2nc(O)[nH]c2c1 c1(CC)cccc(C(=O)NC(C(=O)N(C)CC2CCCS2)C2CC2)c1 C(CC(=O)N(C1CCCNC1=O)C)(C(F)(F)F)NC(C1CCN(OC)CC1)=O C(=O)(C(O)CCC(C)C)NCC1(OC)CCN(C(CC)=O)C1 C1(NC(=O)CCC2CC2)CC2CN(C(c3cccc(CO)n3)=O)CC2C1 C(=O)(CCCCC(C)(C)C)NC1(CNC(C(CC(C)C)=O)=O)CC1 C12(NC(CCCOC)=O)COCCC1CN(C(c1cnn3ccn(C)c13)=O)C2 c1(C(N2C3CN(C(C(CC#C)(C)C)=O)C(C3)C2)=O)cc([N+](=O)[O-])cnc1N N1(C(C2(C)CCCS2)=O)CCCC(NC(c2ccnc(C(F)(F)F)c2)=O)CC1 C1(N(C(=O)Cc2cnc[nH]2)C)CCC(NC(C2(c3ccccc3)CC2)=O)C1 N1(C(c2c(CC)c[nH]c2)=O)CC(N(C(=O)CS(=O)(=O)NC(C)(C)C)C)C(C)(C)C1 C(CNC(c1ccccc1F)=O)(CC(C)C)NC(CSCC#C)=O CC1C(C)CCC1NC(=O)CC1CCCC2CC12 C(C(COC)CC(=O)NCc1ncccc1OC)OC.C12CCN1C(C)C(=O)N2 C#CCC(CC(=O)N(C(CC)CC)C)NC(c1ncccn1)=O C#CC(C)(C)C(=O)N1CCC(C(C)NC(=O)C(C)(C)SC)C1 c1(C(=O)NCC2N(C(C3ON=C(C)C3)=O)CCC2)cc2ccccc2nn1 C1(C(N(C(C(=O)NCC(n2cccn2)C)C)C)=O)CN2CCC1C2 Cc1ccc(C(=O)NCCN2CCC(CCN(C)C)CC2)c(OCC(C)C)c1 N1(CC(=O)NCc2c(C(=O)NCC3(C)CCCO3)cco2)CCC(O)CC1 c1(C(N2CCCCC(CNC(C3C(C)C3)=O)C2)=O)ccc(Br)c(F)c1N C(=O)(C1CCCn2ccnc21)N1CCOCC(NC(C=NOC)=O)C1 N12CCC(C)(C1)CN(C)C2C(=O)NCc1cc(CSC)no1.c1(CC)ccco1 c1(C(=O)NC2C3(CC(NC(C(C)(C)O)=O)C3)C2)c[nH]c2nc(Cl)ccc12 c1(CNC)ncc(F)cc1OC.N1(c2ccccc2)CCCC1(C(=O)NCCOC)CO c1(C(=O)NCC2(CO)CCN(C(c3c(CC)ncs3)=O)C2)c(F)cc(O)cc1F N1(C(c2cc(C)n(C)c2)=O)CC2CCN(C(c3cc[nH]c(=N)c3Cl)=O)C2C1 Cc1cc(C(=O)NC(CNC(C2CCCC2(F)F)=O)C(C)C)c(N)c(F)c1 C#CC1CCCC(CNC(=O)C(Cc2ccoc2)NC(C2SCCS2)=O)C1 c1(NCCCc2ccc(C(=O)OC)cc2)c(Cl)cnc2[nH]nnc12 N1(C(c2c(N)non2)=O)CC2(C1)CN(C(C1CC1(Br)Br)=O)C2 N1(C(CCOCCC)=O)CCN(C(c2coc(C#N)c2)=O)C(C)C1C CC1(CNC(C23CCCC2C3)=O)CC12CCN(C(c1cc3cccnc3[nH]1)=O)CC2 CCCC(O)C(=O)NCC(C1CC1)NC(c1[nH]ccc1-c1ccccc1)=O C=CCC(C(=O)NC(C1CCOC1)CNC(c1sccc1CO)=O)OC Cc1cc(C)c(CN2CCCC(CNC(=O)CC(C)(C)O)C2)[nH]1 c1(OC)c(C(N2CCCC2C2CC2(F)F)C(=O)NC2CCOC2)cc(Cl)cc1Cl c1(NC(=O)Nc2cccc(NC(C=CCCCCC)=O)c2)cc(Br)ccc1F C(=O)(CC1=CCCCC1)N(CC(CC)NC(C(CCC)CC)=O)CC C(=O)(C(C)CC(N)=O)NCC1C(C)CCN1C(c1cc(CN(C)C)on1)=O C1(CC(=O)NCCSCC(=O)NC(CC=C)CO)CCCC(=O)C1 C1(CC(=O)N(CC2(OCC)CCCC2)CC)CC(F)CN1C(=O)C=Cc1cscn1 C(=O)(C(C)(C)C(=O)Nc1nnc(C)s1)NC.N12CCN(CC1)CCN(C)CC2 C(c1ccc(F)c(F)c1)=CC(=O)N.N1(C(CCC)=O)CCC2C(NC(C)=O)C12 C(=O)(CC(C(F)F)NC(C1OCCC1(C)C)=O)NCCn1c(C)ncc1 C1(c2cn(CCCC(=O)NC3(c4cccnc4)CCC3)nn2)(OCC)CCOC1 C1(C(=O)NCCN(CCOC)C(C2(C)CCC(=O)N2)=O)CCC(C)(F)CC1 Cc1cc(C)n(C(C)C(N2CCC(CNC(c3cc(Br)c(C)s3)=O)C2)=O)n1 c1(C(=O)NCC(CNC(CCN(CCC)C)=O)C)cnc[nH]c1=N Cc1cc(C(N2CC(OCCC(=O)NCC3(O)CCN(C)C3)C2)=O)nn1C c1(C(=O)NCC(C)CNC(c2c[nH]nc2C(C)(F)F)=O)cc(Cl)ccn1 N1(C(C2C(=C)C2)=O)CCN(C)CC1CNC(=O)CN(C(=O)CCC)S(C)(=O)=O c1(C(N2CC(COC)(NC(=O)C(F)=CC3CC3)C2)=O)cccn2c(C)nnc12 N1(C(C(CCC)OC)=O)CCC(C)N(CC2CC2)CC1 C1(CN(C(COCC#C)=O)C)COCCN1C(=O)C(C)NC(=O)NC CCC(C)CCC(O)CC(=O)NC1CCCN(CC(O)COCc2ccco2)C1 c1(C(=O)NC2CC(C)(c3ccccc3)C2)cc(CNC(C2CC2F)=O)cc(F)c1 C(C)(CC(F)(F)F)NC(c1n(CC=C)nnn1)c1ccncc1 C1(CC=C)(NC(=O)C(=O)NC2CC2)CCN(C(=O)C(c2ccccc2)N(C)C)C1 C(=O)(CCC1=NNC(=O)CC1)N1CC2OCC(NC(CNS(CC)(=O)=O)=O)C2C1 C(c1ccc(F)c(F)c1)=CC(=O)NC(C(C)NC(=O)CCC1CC1(F)F)CO c1(C(N2CC(NC(=O)CC3CCOC3)C(F)C2)=O)cc2c(cn1)OCCC2 c1(C(N2CC(C(=O)OC)C(O)C2)=O)cc(C)c(I)cc1C Cc1cc(Cl)ncc1CC(=O)NC1CC(C)N(C(=O)C(F)=CCCF)C1 C1(C(=O)OCC)CCCS1(=O)=O.C1(=O)CCC(=O)N(C2CC2)C2(CC=C)CN1C2 C1(CNC(Cc2c(C)ccnc2)=O)CN(C(=O)C(F)C(C)(F)F)CC12CC2 Cc1nn(C)cc1NC(=O)C(c1ccccc1)NC(=O)C(C)c1ccsc1 C(=O)(CS(=O)(=O)CC(=O)N1CCCC1C(C)NC(C1COC2(CCC2)C1)=O)OC C1(C(F)F)(CNC(C(C)=CC2CC2)=O)CCN(C(C2(C(C)C)CCC2)=O)C1 Cc1ncnc(C)c1C(=O)NCC12CC(NC(C3CCC(C)C3)=O)(CO1)C2 C#CCC(C(=O)Nc1cnn(CCC)c1)NC(=O)CCc1cscn1 C1(CNC(C2C(C=C)C2)=O)C(O)C(O)CN1C(c1sc(C)cc1Br)=O C(C(=O)NNc1nc2ccccc2s1)N(C(C1(C)CCC1)=O)C1CC1 C(CCC(=O)NC(C)C(C)C)SC.n1(CC(=O)N)cc(CO)nn1 c1(CN(C(=O)NCCc2cccnc2)CC)ccc(-c2cccc(Cl)c2)cc1 c1(OC)cc([N+](=O)[O-])ccc1C(=O)NCC(C)CNC(C1CC(C(F)F)C1)=O C(=O)(C(CCC)NC(=O)CC1CCC(C)(C)O1)NCC(COCCC)(C)C c1(C(C(=O)NCC(C(C)C)NC(C2CCC3CC3CC2)=O)C)ccc(F)cc1F c1(NCC2(OC)CCOC2)ccc(S(=O)(=O)NCc2nc(C)ccc2Br)c(Cl)c1 c1(C(N(CC)CC2CCCN2C(=O)CC2(C)CCC2)=O)ncc[nH]c1=O C(=O)(C1(C)CCc2ccccc21)Nc1c(C)cc(NC(c2nonc2N)=O)cc1 Cc1cc(C(=O)NC(C)CCCNC(c2nsnc2O)=O)ccc1O N1(C(CC2C(C)C2)=O)CC2(C1)CN(C(c1nn(CCn3cccn3)cc1Br)=O)C2 Cc1ncccc1CC(=O)NCCN(C(=O)CCCc1cnccn1)CC1CC1 C1(C(=O)NCC(C(C)C)NC(=O)CCc2cnccn2)CCn2c(O)nnc2C1 N1(C(CC(CC)NC(=O)CCOC2COC2)=O)CCCC(C)(O)C1 c1(CC)nc(C)c(C(=O)NCCNC(c2cc(Cl)sc2Cl)=O)o1 N1(C(C(C)(C)NCCC)=O)C=COCC1NC(=O)OC CC(C)(C)CCCC(=O)NC1CC(NC(C2CCOC(=O)N2)=O)C1 C1(C(=O)NCCOC2CC(NC(C(C)O)=O)C2)CCC(n2cccc2)CC1 CCCC(C)(CCC)C(=O)N(C)CC1(O)CCN(C(C2CC2c2cccs2)=O)C1 C(=O)(C(C)(C)CCC(=O)OC)N1CCCC(CNC(CCSCCCC)=O)C1 N1(C(C2CC2F)=O)CCC(C2CCCN(C(C3Cc4c[nH]cc4S3(=O)=O)=O)C2)C1 c1(CC(=O)NCC(CN(C)C(c2cc[nH]c(=N)c2)=O)O)ccc(Cl)c([N+](=O)[O-])c1 c1(CN(C(CC)C)C(c2ccc(NC(=O)C(C)CC)cc2)=O)cccc(F)c1F CCCC(C(=O)N1CCOCC(NC(c2cnc(COC)s2)=O)C1)C(C)C CCCCCCCC(=O)NCC(CC(=O)Nc1cc(C)cc(C)c1)C1CCC1 C1(F)(C(=O)NCC(COC(C)C)O)CCN(C(c2occc2C2CC2)=O)C1 CCC(CNC(=O)CC1CN(C)C1)(CC)NC(=O)Cc1ncn(C)c1C C1(O)(CCNC(C2CN(C)C2)=O)CCN(C(C2CCCC(C)CC2)=O)CC1 C1(C(N2CCC(NC(C=CSC)=O)(CO)C2)=O)CC(O)c2ccccc2O1 CCCCC(C)(F)C(=O)N1CCCN(C(c2cnc(OC)s2)=O)CC1 CC(CCNC1CCCC1)N=c1ccnc(N2CCOC3(CCCC3)C2)[nH]1 C(C(F)(C(=O)N1CCC1CC1CCCC1)C(C)C)NC(CC(COC)COC)=O C(=O)(C1=CC2CCCC12)NCCCN(C(=O)CCCC1CC1)C n1(CC(=O)NC2CC(C)(CNC(C3CCN(CC)CC3)=O)C2)cccc(O)c1=O c1(OC)cccc2c(C(=O)NCC(C3CC3)N(C(=O)CCS(C)(=O)=O)C)n[nH]c12 c1(C(=O)NCC2OCCC(NC(c3cnsc3)=O)C2)ccc2c(n1)CCC2 c1(NC(C(=O)NC(C#C)C(C)C)=O)ccc(OCCC)c(OC)c1 c1(NC(C2CCN(C(c3cc(C4CC4)on3)=O)CC2O)=O)cccc2occc12 c1(C(C)=O)csc(C(=O)NCC(C2CC2)NC(c2ncoc2C(C)C)=O)c1 N1(C(c2scnc2C)C(=O)NCCOCC)CCCC(C)(C(=O)OC)C1 C1(C(=O)NCC(CC#C)(C)C)CCCCCN1C(=O)CCc1cnc(C)o1 Cc1sc(O)nc1C(N1CC(NC(c2nccn2C(C)C)=O)C(C(N)=O)C1)=O c1(C(N2CCCN(C(C3C(C=C)CC3)=O)C(CO)C2)=O)nnc2n1CCCCC2 c1(CC)cc(OC)ccc1C(N1CCCC1C(C)NC(=O)C1=CCC1)=O CC1CN(C(=O)CCCc2cncs2)CCC1NC(C1CC(OC2CC2)C1)=O CC1(C#CC(=O)N2CCC(Nc3ncncc3Cl)C(F)(F)CC2)CCCO1 c1(OC)ccccc1NC(=O)C(c1cc(C)oc1C)N N1(C(CC(CC)(C)C)=O)CC2(CC(NC(=O)C(c3ccccc3)F)CO2)C1 N1(C(C(C)c2ccsn2)=O)CCCC12CCN(C(C1(C#N)CC1)=O)C2 c1(C(N2CCCC(C)C2CNC(=O)CCc2nncs2)=O)ccc(C#N)cc1F C1(NC(CS(=O)(=O)NCC)=O)CCCN(Cc2coc(C)c2)CC1 CC(=O)CCN=C(NCc1ccc(C)cc1C)NCc1cccc(S(C)(=O)=O)c1 c1(C(N(C(c2cccc(F)c2)C)C2CC2)=O)cccc(C2(F)CC2)c1 N1(C(C2(C(F)(F)F)CC(=C)C2)=O)CCCC(NC(=O)CCOCCC)C(F)C1 c1(OC)c(C(=O)NC(C)C(C)NC(=O)COCCF)cccc1F.c1(O)ccccc1 N1(C(C2CC2NC(c2cnc3sccn23)=O)=O)Cc2cccc(F)c2C1 N1(C(c2cc(C)cc(F)c2)=O)CCC(NC(c2cnsn2)=O)CC(C)(C)C1 C(=O)(C1CCCc2nn[nH]c21)NC(C1CCCCC1)CNC(C1C(=O)NCC1)=O C(=O)(CS(=O)(=O)CCc1ccccc1)NCCC1N(C(C2C(=C)C2)=O)CCCC1 C(Cn1nccn1)(C(F)(F)F)NC(=O)NCc1ccccc1OC.C1CCCO1 C#Cc1ccc(C(=O)NC2CC(CC(=O)OC)C2(C)C)cn1.N12CC(C1)CC2=O N1(C(C2CC(NC(=O)CC3CCCC(O)C3)C2)=O)CCC2OCCC2C1 c1(CN2CCC(C(=O)NC(CC)C)C(O)C2)cc(C)c(OC)c(C)c1 C1(NC(CN2CC(C)C2)=O)CN(C(c2cc3c(F)cccc3[nH]2)=O)C2(CCCC2)C1 C1(C)(C(=O)NCC2CCCC(NC(CN(C(C)=O)C)=O)C2)CC2CCC1O2 C1(C(=O)NCCNC(C2(C(C)=O)CCC2)=O)C2C3CCC(C3)C12 CS(=O)(=O)C(CNC(=O)CC1CNC(=O)C1)CNC(=O)COCCC(F)(F)F c1(CCC(=O)NC(C(=O)NCC(C=C)O)c2cccs2)cc(C)[nH]n1 N1(C(C2(CC#C)CCCC2)=O)CCN(C(C2OCC2(C)C)=O)C(C2CC2)C1 N1(C(=O)OC(C)(C)C)CCC2=C(C(=O)Nc3c(C)cc(O)c(Cl)c3)CN2C1 C1(C(C)C)CC(OC(c2ccnn2Cc2ccccc2S)=O)CCO1 C(C(C)C(=O)N1CCC(CCNC(c2cc(C(F)(F)C(F)(F)F)on2)=O)C1)SC CON1CC(C(N2CCC(CNC(=O)CCSc3ccccc3)C2)=O)CC1=O CCCCC(C)C(=O)NCC(C)(C)CN(C(c1cn(C)c(C)n1)=O)CC C1(CNC(CCOC)=O)CN(C(c2cc(N(C)C)ccn2)=O)CCO1 c1(CNC(C)=O)ccc(C(=O)NC(C)C(C)NC(C2(C(C)(F)F)CC2)=O)s1 N1(C(c2nn(CC)nc2C)=O)CC(C)OC2(CCN(C(=O)CCS(C)(=O)=O)C2)C1 N1(C(CC)=O)CC2(CC(C(=O)Nc3csc(C)c3)CO2)C1 C1(NC(c2cc(CC)[nH]n2)=O)CCCC(CNC(C2CCN(CC(F)(F)F)C2)=O)C1 c1(OC)c(Cl)cc(CN2CCCC(F)(CNC(=O)CCc3ccsc3)C2)cc1Cl C(CCCCCS(=O)(=O)CCCCCO)NC(c1cc(-c2ccc(C)o2)n[nH]1)=O N1(C(C=C(CC)CC)=O)CCCN(C(c2cc(C(N)=O)cn2C)=O)C(C)C1 c1(C(=O)NC2C(NC(c3c(C)ncn3O)=O)C2)cc(F)ccc1S(C)(=O)=O N1(C(c2c(Cl)ncn2C)C(=O)NCCCC)CC=CCC2(CCC2)C1 N1(Cc2cc(C)no2)CCC(C)C(NC(=O)CC(C2CC2)C2CC2)C1 C=CCCCC(C(=O)NCC(O)CC(C)C)NC(=O)C(c1cccn1C)=O N1(C(CN(CCC)C)=O)CCCCCC1C(N1CC(O)C(O)C1)=O N1(C(C)=O)CCC(O)C(F)C1.c12cc(co1)C(=O)NC2.C12(CC1)C(=O)NC2 C(=O)(N1CCC(C(N2CC3CCC(C2)O3)=O)O1)C1C(C#N)C1 C1(C(=O)NCc2oc3ccc(OC)cc3c2)COc2ccccc2O1 c1(C(=O)NC2CC(CCNC(C3(C)CC=CCO3)=O)C2)cncc(S(C)(=O)=O)c1 C(C(CC(C)C)NC(C1CCC(C(C)(C)O)CC1)=O)NC(C(F)OC)=O Cc1cc(F)ncc1C(N1CC2CC(NC(C3CCC4(CCC4)O3)=O)C2C1)=O C1(c2nnnn2CCCC(=O)OC(C)(C)C)(NCCCSC)CCSC1C C(=O)(CCC(=O)N1CCC(=CCNC(=O)C=CC2CCCO2)CC1)NCCC C1(OC)(CNC(=O)C(C(C)C)OCC(C)C)CCN(C(=O)CC2(C#N)CC2)C1 N1(C(C2N(C(C(C)SCCCC)=O)CC(=O)C2)=O)CCC2(CCCO2)C1 CCC(CCC(=O)N1CC(CO)C1)NC(=O)CC1CCCCN1C C1(CNC(c2cn(CC)nc2)=O)(OC)CCN(C(=O)Cc2ccsc2C)C1 c1(C(=O)Nc2c(C#N)n[nH]c2)cc2cc(-c3ccn4cnnc4c3)ccc2o1 CC(C)C(C(C)C)C(C(=O)NC1(C)CC1)N(c1ccc(F)cc1)C1CCOCC1 CC1CCC=C1C(=O)N1CCC2(CC2NC(c2cccc(F)c2F)=O)C1 c1(C(=O)NC2C(CNC(C3(OCC)CCC3)=O)CCC2)occ(C)c1C N1(C(CCCCN(C)C)=O)CCN(C)CC1CNC(=O)C(F)CC1CCCCC1 C1(CC)C(=O)N(C)CCN1C(=O)C(CC(F)F)N(C(=O)COCC(F)F)C C#Cc1cnc(C(=O)NCC2CC(F)CN2C(=O)CC2CNC(=O)O2)c(C)c1 c1(C(C)N(CCOCCC(=O)NCCN(C)C)C)nnc(C(F)(F)F)s1 CC1C(C(=O)NCC2CCCC2)CC2CCC1N2C(=O)CCSc1ccn(C)n1 NC1(C(=O)NC2CN(C(=O)CCCC(=O)O)CC2(F)F)CC2(CCOCC2)C1 N1(C(=O)C=CC2CCOC2)CC(NC(C2(O)CC2)=O)CC(O)C1 CC(C)C(C(=O)N1CCCC(CN(C)C(C2CC2)=O)C1)S.n1(C2(N)CC2)cccn1 Cc1oc(C(=O)NC(C)(CNC(=O)CS(N)(=O)=O)C(C)C)cc1Br CC1CN(C(C2CC23CC(O)C3)=O)CC1(C)CNC(c1cc[nH]c1)=O N1(C(CC(C=C)C)=O)CCCC(C)(NC(=O)C=CCOC)C1 N1(C(C(C)C(C)C)=O)CC=CC1CNC(=O)CCc1nc(-c2cccs2)no1 n1(CC#C)c2nnc1C1CC1C(=O)N2C1CC1.c1(CC)ccc(Cl)s1 c1(-c2n(C)nc(-c3nccn3C3CCOCC3)n2)cnn2ccc(O)nc12 C1(OC)CC2CC1CN(C(=O)C(CC(F)F)N(C(=O)CCn1cccc1)C)C2 Cc1nc(NCc2nc3c(s2)CCCC3)cc(=NCC(C)CC(F)(F)F)[nH]1 N1(C(C(C)NC(=O)OCC)=O)CC(O)(CNC(C2(C3CC3)CCCO2)=O)C1 c1(NC(C)=O)cc(C(N2C(C(=O)NCC3(O)CCC3)CC3CC23)=O)ccc1F Cc1cc(O)ccc1CNC(=O)C(C(N)=O)NC(C1CC1C#N)=O c1(C(=O)NCc2nccc(C(=O)NC(CCC)CCC)c2)cc(N)cc(F)c1 c1(C(=O)NCCC(C)NC(Cc2cnc(C)[nH]2)=O)cc(N)c(OC(F)F)cc1F C1(C(=O)NCC(C2(O)CN(C(C(C3CCCC3)OC)=O)C2)(C)C)NC(=O)NC1=O N1(C(CC=C)=O)CC(NC(=O)CC23COC(C2)C3)CC1C CC(C)C(O)C(=O)NCCCOC1CCN(C(=O)CN(C2CCSC2)C)CC1 C1(C)(NC(CN(C2CCC2)C(c2cnc(CC)nc2)=O)=O)CC(C)(C)OC1=O Cc1nn(C)c(Cl)c1CN1C(C(=O)NCC2CC(=O)N(C(C)C)C2)CCC(O)C1 C1(NC(CSCC(C)C)=O)CC2(CCCN(C(=O)CSCc3cccs3)C2)C1 CC(C)CC1C(=O)NC2C(CC)N1C(CC)CCC2C(=O)NC(C)C CC1CCCN(C(=O)C2=NOC(C)C2)C1CNC(c1ccc(CO)nc1)=O C1(NC(CCC2COC(C)(C)O2)=O)COCCN(C(C2CC(n3cnnc3)C2)=O)C1 Cc1cn2c(n1)C(C(=O)Oc1nccc3ncccc13)CCC2 c1(N2CC=CC(NC(c3c(C)nc(O)nc3C)=O)C2)nc(Cl)nc2cnn(C)c12 N1(C(c2nnn(CC)c2C)=O)CC(F)(F)CC1CNC(=O)CS(=O)(=O)CC C1(C(=O)NCc2cnn(CC)c2C)CC2CC1CN(C(=O)CC(F)(F)F)C2 C(=O)(C(C)(CC)C(=O)OC)N1CCCC(C(N(CC)Cc2cccnc2)=O)C1 c1(C(=O)NC2C(C)CCN(C(CCCC#CC)=O)C2)nc2ncccn2n1 C1(C(=O)NCCC2ON=C(C)C2)CCN(C(c2cc(C)[nH]n2)=O)CC1C c1(OC)ccccc1C=CC(=O)NC(C)CCCCNC(C1(F)CC=CCC1)=O c1(C(N2CCC(C)(CNC(C3(C)CC=CCC3)=O)C2)=O)ccc2c(c1)COC2 c1(CCC(=O)NCC(CO)NC(C2C3CCCOC23)=O)cc(Cl)cc(Cl)c1 C1(NC(c2nnc(C(C)(C)C)s2)=O)CCC2CCN(C(C3CSCCS3)=O)C1C2 C(=O)(C(=O)N=S(C)(C)=O)C(C1(OC)CCCCC1)=O.N1CCCCC1CN c1(C(=O)OCC)cnc(=NC(C)CCCNC(=O)CCc2cncs2)[nH]c1 C(=O)(CCCCC(F)(F)F)NCCCCCN(C(=O)C(c1cncn1C)O)C C1(C(=O)NCC2(CNC(CC=C(C)C)=O)CCCCC2)CC(=O)CC12CCC2 CCC(C)C(C(=O)N1CC(NC(=O)COC2CCCC2)C1)NC(=O)OC.C1CC1 Cc1nc(CC(F)(F)F)sc1C(=O)NC(C)COc1cccc(F)c1 c1(CCC(=O)NCCC(C)NC(c2cccc(C3(C)CC3)c2)=O)cncc(F)c1 C1(C(=O)NC2(CO)CN(C(CN(C(COC)=O)C)=O)C2)CCCCC12CC2(F)F c1(C(N2C(CNC(Cc3ccc(C)nc3)=O)CC2)=O)c[nH]c2nccc-2c1 Cc1nn(C)c(C(=O)NCC2CCN(C(c3cc(C)n(C)n3)=O)C2(C)C)c1Cl C(=O)(C1CCCc2ncnn21)NC(C)CCNC(c1cnc(C(F)(F)F)nc1)=O N(C(=NCC(C)C)NCc1ncccc1Cl)C(Cc1ccc(C)s1)C c1(C(=O)NC2C(CC)CN(C(=O)C(Cl)=CCl)CC2)cc2cc(OC)ccc2[nH]1 Cc1cccc2c(C(=O)NCCCCC(C)NC(c3cnns3)=O)n[nH]c12 c1(C(=O)NCCN(C(=O)CC2CCN(C)CC2)C(C)C)nnc(O)cc1O C1(F)(CNC(=O)Cc2ccc(F)cc2)CCN(C(C2CC3(CCC3)C2)=O)CC1 c1(C(=O)NCC(CNC(c2cccc(OCC)n2)=O)F)cc([N+](=O)[O-])ccc1O CC1CN2CCCC2CN1C(c1ccc2c(c1)CCC2)C(=O)NC1CCCCC1 C1(C(C)C(=O)NCCCC2CCCCC2)CCN(C(c2cc(O)ncn2)=O)CC1 S(=O)(=O)(CC1=NOCC1)NC(c1nnc(-c2ccccc2)s1)C N1(C(C2C(C)CCS2)=O)CC(C2(NC(c3cnc(C4CCC4)nc3O)=O)CC2)C1 n1(-c2n(C)ccn2)nc(-c2cccc(F)c2)nc1C1CCN(CC2CCCO2)C1 c1(COCCNC(c2n(CC(=C)C)nnn2)C2CCOC2)cccc(C)n1 Cc1cc(C)c(C(=O)NC2(C)CCN(C(=O)CCC3CCCCO3)C2)s1 C(=O)(CS(N)(=O)=O)N(C1CN(C(c2ccccc2SCC#N)=O)CC1O)C c1(C(N(C(C)C)CCN(C)C(C2CC2F)=O)=O)cnc2c(F)cccc2c1 C1(CCNC(=O)Nc2cnn(-c3ccccc3F)c2)CCCNC1=O c1(C(C)=O)ccc(C(N2CC3(CC3)CC2CNC(=O)C(C)CN(C)C)=O)c(C)c1 c1(C(N(CC(CC)NC(c2ccccc2Cl)=O)C)=O)cc2n(n1)CCO2 c1(N2CC(CNC(c3cc4n(n3)CCO4)=O)OCCC2)ccn2nccc2n1 N1(CCc2cn(C3C(OC)COC3)nn2)C(=O)C2CCCCC2C1=O c1(OCC(=O)N(C)C)cccc(C(N2CCOC(CNC(=O)C(C)(C)C)C2)=O)c1 c1(C(=O)NCC(CN(C(c2[nH]cc(CC)c2)=O)C)C)cc(C)c2occc2c1 C(=O)(C1CN(Cc2ccnn2C(F)(F)F)c2ccccc21)OC c1(C(=O)N(CC(CC(C)C)NC(CN(CC)CC)=O)CC)noc2c(F)cccc12 C1(NC(CS(N)(=O)=O)=O)CC2CN(C(=O)CCc3cncs3)CC12 C12(C(N3CCC(N4CCC(NC(C(F)=CC)=O)CC4)C3)=O)CCC(CC1)OC2 c1(N(C)CC2CC(O)C2)nc2cccnc2c(=NC2CC2c2ccsc2)[nH]1 C=CCC(C(=O)N(C1CCCN(C(c2ccc(CO)cc2)=O)C1)CC)OC N1(C(CC2N(C(c3cncc(OC)c3)=O)CCC2O)=O)CC(OC)C2(CC2)C1 CCC(CC(=O)NC1CC(CC(N2CC(OC)CC(C)C2)=O)C1)CC(C)C c1(C(=O)NCC2(O)CCN(C(C3CCC=CO3)=O)C2)csc([N+](=O)[O-])c1 Cc1cc(C(N2CC3(CCN3C(=O)C(C)n3ccnc3)C2)=O)nnc1C C1(NC(C=NOC)=O)CN(C(=O)C(c2ccc(F)cc2)=O)C2CCCCC12 C1(C(=O)NCC(CC(C)C)NC(=O)CC2(O)CCCOC2)CCCCCCC1 N1(C(C(CCSC)O)=O)CC(NC(C2CC3(C2)CC32CC2)=O)C(C)(C)C1 C12(C(N3CCC(C(C)NC(c4ns[nH]c4=O)=O)C(C)C3)=O)CCCC(C)(C1)OC2 c1(CC(=O)NC2C(NC(C(CC)NC(N)=O)=O)CCCC2)c[nH]c2c(Cl)cccc12 c1(CC(C)C(N2CCCC(C)(CNC(=O)CC3CC3)C2)=O)cc(F)cc(F)c1 C12CCCN(C1)C(=O)NCCCNC(=O)C2.c1(C(C)C)nc(C(C)C)no1 C1(CCOC)(NC(=O)CCCO)CCN(C(c2ccc(CNC(C)=O)o2)=O)CC1 c1(C(N2CC(C)(C)C(NC(=O)CCC3(O)CCC3)C2)=O)ccc2ocnc2c1 Cc1c([N+](=O)[O-])c(C(=O)NC2CC3CN(C(=O)C(C(C)C)N(C)C)CC23)nn1C N1(C(C2C(C)C2)=O)CCN(C(=O)C(F)C2CCC2)CC1.C(C)(C)(C)NC=O N1(C(c2c(OC)ccc(Cl)c2)C(=O)NCCC(C)C)CCCCC2CCCCC12 C(=O)(C#CC1CCOCC1)N(CCN1CCN(C(c2cc(C)ncc2)=O)CC1)C C(=O)(C(C)(O)CNC(c1cccc(OC(C)(C)C)c1)=O)OC c1(CC(=O)N(CC=C)CC2CCCN2)ccccc1OC(F)F C1(CC(N2CCC(N(C(CNC(=O)OCC=C)=O)CC)C2)=O)CC(=O)NC1=O CCCC(C(=O)NCC1(C)CCCN1C(C1CC(N2CC(O)C2)C1)=O)OC C=CCCN=C(NC(=O)Cc1ccccc1)NCC1(O)CCOC1C c1(C(=O)NCC(CCNC(C2C(C)C2)=O)(C)C)cc2c(s1)C(C)(C)CCC2 C1(NC(C(CCC)OC)=O)CCOC12CCN(c1ncc(C)c(O)n1)CC2 c1(C(=O)CC2C(C(=O)NCC3(CO)CC(=C)C3)OCC2)ccc(OC(C)C)cc1 N1(C(C2(CCCC)CC2)=O)CCOC(CCNC(=O)Cc2cncn2C2CC2)C1 Cc1ccc2[nH]nc(C(=O)NCCC3CN(C(=O)CC(C)P(C)(C)=O)C3)c2c1 Cc1ccc(CO)cc1NC(=O)C(F)CC1CN(C(C2CCCCCN2C)=O)C1 CCCCCCCCC(=O)N1CC(C2CCN(C(=O)CN3CCOC3=O)O2)C1 C(=O)(CC(C)(C)C1CCCCC1)NC(CCC=C)C1CC1 O=C1CC(C(N2CCN(C(c3ccco3)=O)CC2CC(F)(F)F)=O)NC(=O)N1 c1(C(N2CC(CNC(c3cc(CCOC)on3)=O)C2)=O)cccc(Cl)c1[N+](=O)[O-] N1(C(c2c(CNC(CC(C)(C)C3CC3)=O)noc2)=O)CCC(C2=NOCC2)C1 N1C(=NCC(F)(F)F)NCc2ccc(cc2)CC2C(CCO2)CN1.N(C)(C)CC c1(NC(Cc2n(C)nnn2)=O)cc(C#N)ccc1Br C(=O)(C(O)CC(N)=O)NC(CSC)(C)C(=O)N(C)Cc1csc(C)n1 C1(NC(C(CC)C2CCC2)=O)CC2CCC1CN(C(c1ncn(C)c1C)=O)C2 C(C(O)CC(=O)N1CC(C)(C#N)C1)NC(Cn1ccc(C)n1)=O c1(OC)cc(C)c(C(N2CCCN(C(=O)C=C(C)C(C)C)C(C)C2)=O)cc1Cl C1(NC(=O)NCC2OCC(C)C2)NC(=O)OC1(C)C c1(OC)ccc(C(=O)NC2CC(F)CN(C(=O)C=CC3CCCC3)C2)nc1N C(=O)(C(C)(C)S(C)(=O)=O)NCCN(CCCN(C)C)C(c1cccc2c1NCC2)=O C1(NC(=O)CN2CCCC2=O)CC2CC1N(C(=O)CC(O)C1CCCC1)C2 C1(OCC)CC(C(=O)On2cc(Cl)c(C)n2)C1(C)C C1(C(=O)NC2C(CNC(=O)CCOc3cccnc3)C2)CCC2CC2CC1 c1(C(N2CC(CCCNC(c3cnc(CC)[nH]3)=O)OCC2)=O)ccc(F)c(Cl)c1 c1(C(N2CCC(NC(C=C(CCC)C)=O)C(F)C2)=O)cc(=O)c(OC)cn1C C(N=c1[nH]c2c(c(=NC3CSC3)[nH]1)CSC2)c1c([N+](=O)[O-])ccc(N)c1 Cc1nc(C(N2CCC(NC(=O)Cn3ncccc3=O)C(C)C2)=O)ccc1C#N C(=O)(CCCCCCN=[N+]=[N-])N(C)CC1CCN(c2cc(C)ncn2)C1 C1(F)(CNC(C(C)(C)C)=O)CCN(C(C2(Cl)CC2(C)C)=O)CC1 C(=O)(C(F)CC(C)(C)NC(=O)CCOC1CCCC1)NC(c1n(CC)ccn1)C C#CC1CN(C(C2CCN(C(=O)C(C)OCC3CC3)CC2)=O)CCN1C CC1(C)CC=C(C(=O)N2CC(CCCCNC(=O)Nc3ccccc3Br)C2)CC1 C#CCC(CC(=O)N1CCC(C(N)=O)C1)NC(c1oc(C)nc1C)=O c1(C(=O)NCC2(NC(c3cc(Cl)c[nH]3)=O)CCOC2)ccccc1[N+](=O)[O-] N1(C(c2[nH]cc(C(C)=O)c2)=O)CC=C(C(=O)NC(c2ccccc2O)C)CC1 c1(C(N2C(C)(CNC(C(COC)(C)OC)=O)CCC2)=O)sc2ccsc2c1C Cc1ccc(N(C)C(c2cc(CNC(C3CC34CC4)=O)cs2)=O)c(C)c1 C(=O)(C(C)(O)Cn1cc(Br)cn1)OCC(C1CCC(CCCCC)O1)=O CCC(C)CC(C)C(=O)NC1CC2CC(NC(C3CC(F)(CO)C3)=O)C1C2 C1(C(N2CCC(OC)C2)=O)CC2CC1CC2NC(=O)Cc1ccc(O)cc1 CC1(C)CCCC(CNC(=NCCc2cccs2)NCC2CCC=CO2)O1 C(=O)(CC(F)(F)C(C)C)NC1CCN(C(C2C(c3cc(C)on3)C2)=O)C1C(C)C CCCC(C#N)C(=O)NCC1(CNC(=O)CCc2nnc(C(C)C)o2)CC1 c1(C(N2C(CC)CN(C(c3csc(=NC)[nH]3)=O)CC2)=O)cc(C)c(=O)n(C)c1 c1(C(N(C2CCN(C(c3n(CC)ncc3)=O)CC2)C)=O)c[nH]c2cccc(F)c12 N1(C(CC(=C=C)C)=O)CCC2C(CCN2C(c2ccc(NC)c(F)c2)=O)C1 C(C)(C(=O)NC1CC(CCNC(=O)CCc2cnoc2)C1)OCC#C CCC(CC)(CCNC(C1(CCOC)CC1)=O)NC(c1ccnc(OC)c1)=O C(=O)(C(C)CO)N(C(C)CNC(=O)CCNc1ccncc1)CC C1(c2nnnn2C2CC2)(NC2CC2)CN(S(C)(=O)=O)CCC1C.CC1C(=O)N1 N1(CCC(C(=O)OCCO)NC(=O)Cc2cncnc2O)CC(C2CCCC2)C1 N1(C(CC(C(C)C)OCC)=O)CCN(C(=O)C(C)CC(C)(F)F)CC12CCC2 C12(C(N(C)CC3CCN(C(C4CN5CCN4CC5)=O)C3)=O)CCC(N=[N+]=[N-])C1C2 Cc1nnc2sc(C(=O)NCC3CCN(C(=O)C(C)CF)C34CC4)c(N)c2c1C C1(C(N2CC(SC)C(NC(C3(C#N)CCC3)=O)C2)=O)CCN(CP(C)(C)=O)CC1 N1(C(c2cccc(OCC)c2)=O)CCC(C)C(CNC(C2(CF)CC2)=O)C1.C(C)(=O)N C(=O)(C1=C(c2ccccc2)N(C)C(=O)N(C)C1c1coc([Si](C)(C)C)c1)OC c1(CC)cccnc1C(=O)NC1CCCCC1C(=O)NC(c1nc[nH]n1)CC C1(C(=O)NCCC2N(C(C(C)=C3CCCC3)=O)CCC2)CN(C)C(=O)CCO1 C1(CC(=O)NC2CCCCCC2CO)C2CCC(C2)N1C(c1ccn(C(F)F)n1)=O c1(C(=O)Nc2cccnc2O)cc(S(=O)(=O)N2CCOCC2)ccc1Cl C1(NC(C(CSC)O)=O)CCC12CN(C(=O)C(c1ccc(F)c(C)c1)=O)C2 N1(C(C(CC)NC(C)=O)=O)CC2(CC(NC(=O)C(O)c3cnc[nH]3)C2)C1 C=CCC(CC)C(=O)NC1CCN(C(c2snc(Cl)c2Cl)=O)C1CC N1(C(COCC(=C)C)=O)CCC(C2CCN(C(c3cc(CO)[nH]n3)=O)CC2)CC1 c1(C(N(CCCNC(C#CC(C)C)=O)C2CC2)=O)cc(=O)c2ccccc2o1 C#Cc1c[nH]nc1NC(=O)C(CCC)OCC.c12ccc(cc1)C(C)NC2=O Cc1cc(C(N2CCCC2C(=O)Nc2cccc(C)n2)=O)cc(Cl)n1 C1(C(C)(C)NC(C(C)N(CC(F)(F)F)C)=O)CCN(C(c2ccc(CO)s2)=O)C1 N1(C(COCCCCCC)=O)CCCC(C(C)(O)CNC(=O)C=CCF)C1 c1(CC)nc(=NC2CC(C)N(C(c3ccc(NCCCO)cc3)=O)C2)cc[nH]1 Cn1nc(C(=O)NCC(CO)NC(c2ccc(Cl)s2)=O)cc1C1CC1 S(=O)(=O)(c1cnc(OCC=C)cc1C)N(CCCN(C)C)CC1C2COCC12 S(=O)(=O)(c1c[nH]c(=NCCn2ccnn2)cc1C)N(C)Cc1cccc(C)c1 C1(OC(=O)CC2CC3C=CC2CC3)CCC2(CCCC2)C1 c1(CNC(C2CC(CNS(=O)(=O)C3CC3)C2)=O)ccc(Br)nc1 C(=O)(N=c1[nH][nH]c2ncc(Br)cc12)C1(C)CN(Cc2cccc(I)c2O)C1 c1(CC(N2CCC3CCN(C(c4cnn[nH]4)=O)CC32)=O)ccc(Cl)c([N+](=O)[O-])c1 Cc1nn(C)c(C)c1C(=O)NCC1(F)CN(C(c2cc(C3(C)CC3)on2)=O)C1 N1(C(CC=C=C)=O)CCC(NC(=O)C(C(C)O)NC(=O)C2CC2)C(CC)C1 C1(C(=O)Nc2c(C)nsc2)C2CN(C(=O)CC3CCN(C)CC3)CC12 N1(C(C(C)=C(CC)C)=O)CC2(COC(CNC(=O)CS(N)(=O)=O)C2)C1 c1(C(N2CCCC(NC(c3c(C)cns3)=O)C2C)=O)ccnc2c(F)cccc12 C1(CNC(C2(C)CCN(C(c3n(CC)nc(C)c3)=O)C2)=O)CN(C)CCN1C CC(O)C(F)(F)C(=O)NCCC1CN(C(=O)C(N)=O)CCCO1 N1(C(c2cn(CC(=O)OCC)nn2)=O)CC2(CCCC2NC(C2CC2(F)F)=O)C1 c1(C(=O)OC)cc(C(=O)NCC2CCN(C(c3cnccc3Cl)=O)CC2)c(C)[nH]1 C12=NC3=C(C(=NCCC(C)CN1C)N2)CCC3.C1(OC(C)C)CC(=O)N(C2CC2)C1 S(=O)(=O)(c1cccc([N+](=O)[O-])c1)NC1CCCN(Cc2c(C)ccc(Br)c2)C1 Cc1cnc2cc(-c3nc(Cc4ccccc4F)nn3CC3CC3C)ccn12 CC1CC(N(C)CCOCCO)CCN1C(c1ncccc1Cl)C(=O)N(C)C c1(CC(N2C(CN(C(c3nc(NC(C)=O)sc3)=O)C)CCC2)=O)cc(C)nn1C Cn1nc([N+](=O)[O-])c(Cl)c1C(=O)NCC(C1CCOC1)NC(=O)C(F)=CCCF c1(NCc2ccc(C)cn2)nccc(=NCC(F)C2CCC2)[nH]1 c1(-c2cn(CC3N(C(Cc4cc(CC)no4)=O)CC3)nn2)cccc(OC)c1Cl C=CCC(C)(C)C(=O)NC1CCC(NC(C2(N3CCOCC3=O)CC2)=O)C1 Cn1ccc(S(=O)(=O)N2CC(O)CC2C(N2CCSCC2)=O)n1 C1(C(N2CCC(N(C(=O)C(C)O)CC)CC2)=O)CCCC2C1C2(F)F c1(NC(=O)NCC2(C(N3CCC3)C)CCCO2)cccnc1C(F)(F)F C1(C(N2CC(c3onc(C)n3)C2)=O)NC(=O)OC1(C)C.c12ccn(c1)CNC2=O C1(C(=O)NC(CNC(c2c(O)nc(C)c(C)n2)=O)CO)CCc2cnn(C)c2C1 c1(CC)ncnc2c(OC(C)C)cccc12.C12(CCOCC1)N(C)C2 C12CCCCN1C(=O)CCCOC2.C(=O)(COC(F)F)NCC.C(CCO)OCCO Cc1nc(CCC(=O)NCC2(O)CN(C(c3cc(C(F)F)[nH]n3)=O)C2)oc1C c1(C(=O)NC2CN(C(Cc3cc(C)sc3C)=O)CC2F)cccc(C)c1Cl FC1COC2CN(c3ncnc4sccc34)CC12 c1(CNC(CN2CCC(C)(OC)C2)=O)ccc(C(=O)O)cc1C C1(CCNC(CCOC)=O)(C(=O)NCC2(N(C)C)CCCC2)CCCC1 C1(CCNC(=O)C=Cc2ccoc2)CC(F)(F)CN1C(=O)CC1CCCC1O C(=O)(CCC(C)(F)F)Nc1cc(C2CC2)no1.C1(OC)CN2CC1C2=O C1(C(=O)OC)CC(=O)N(C)C1c1cccc(Cl)c1.C12(C)CC1NC2=O C(=O)(C(C)(C)C(C)(F)F)N1C(CNC(CNC(CCC)=O)=O)CCC1 c1(N(CC(C)C)CCc2scc(C)c2)cnc2[nH]c(C(F)(F)F)nc2c1 c1(NC(C2COCC(C)O2)=O)ccc(Br)c2cccnc12 S(=O)(=O)(CCC(=O)NCC1(C)CCC(NC(=O)Cn2cnnc2O)C1)NC C(=O)(C(C)(C)CC(=O)OC)N1CCC(C(=O)NC(CN(C)C)CCO)(CC)C1 c1(C(N2CC(NC(=O)C(=Cc3c[nH]cn3)F)C(O)C2)=O)cc(Cl)nc(Cl)c1 c1(OC)ccc2nccc(C(=O)NC3(CO)CCN(C(C4C=CCC4)=O)C3)c2n1 C1(NC(CCP(C)(C)=O)=O)CCSC12CN(C(c1ccc(C(=O)CF)cc1)=O)C2 c1(C(=O)NC2CC(C)(NC(=O)CCCN3CCCC3)C2)cc(F)ccc1Cl Cc1cc(C(=O)NCC2(C)CN(C(=O)C(N)=O)C(C)(C)C2)c2c(O)nn(C)c2n1 c1(C(=O)NCC2N(C(C(C)=CC3CC3)=O)CC(O)C2)ccc(O)c(Br)c1 c1(C(=O)NC2CCN(C(CC=CC=C)=O)CC2C)ccn2cc(C)nc2c1 c1(C(N(C)CC2CCCN(C(=O)C3=CCCS3)C2)=O)sc2ncccc2c1Cl Cc1cnccc1CC(=O)NCC1(O)CCN(C(C2(C(=O)N(C)C(C)C)CC2)=O)C1 C1(C(=O)NCC2C(NC(c3c(CCC)n[nH]c3)=O)C2)CCOC2(CCC2)C1 CC(C)CC(O)CC(=O)NC1CCCCC1C(=O)NC1CCCC1(C)C C=CC1CN(C(=O)C(C)OC(C)(C)C)CC1NC(c1cccc(C)c1Cl)=O N1(C(CC(C)OC)=O)CCN(C2CCN(C(c3ccc(C(N)=O)[nH]3)=O)CC2)CC1 C1(C(=O)O)(C(N2C(c3n(CC=C)nnn3)CCCC2)=O)CCc2nc(C)ccc21 C1(CC)CCCC(NC(C2CCN(C(=O)NCCCN(C(=O)C(C)C)C)C2)=O)C1 C12COCC1NC(=O)C2.C1(CCCN(C)CCO)CCCO1.C(C)(C)(C)OCCO N1(C(C(=Cc2ccco2)C)=O)CCC(C2(NC(=O)CC34CC(C3)C4)CC2)C1 C1(NC(C=C(CC)C)=O)CC(CN(C(c2cnc(S)[nH]2)=O)CC)C1(C)C N(C1CCSc2ccc(Cl)cc21)C(C)C(=O)Nc1cccc(F)c1 c1(CC(=O)NC2C(CO)CCN(C(CCOCCOC)=O)C2)ccc2sccc2c1 C=Cn1ncc(C(=O)NCC(C)C(F)C(=O)NC2CCOC(C)C2)c1N c1(OC)ccc(C(=O)NC(c2ccccc2)C(C)NC(=O)CCCSC)s1 CC1CCCC=C1C(=O)N1CCCC1(C)CNC(C1CCCN1C)=O CC1CC(NC(=O)Cc2cncs2)CCN1C(=O)C(C)N1CCCC1 C12COCC1(NCC)c1nnnn1CC2.c1(CC)cc(Br)cs1 CC(CC(=O)NCCCN(C(=O)C(Cl)=CCl)C1CC1)C(C)(C)C Cc1cc(C(=O)NCC(C)N(C)C(c2cn(C)nc2C2CCOC2)=O)cnn1 Nc1ccnc(C(=O)NCC2CCCCC2NC(C2CCN(C3CC3)C2=O)=O)c1 C1(NC(c2c(NC(C)=O)c(Cl)ccc2)=O)CCN(S(=O)(=O)N2CCCCC2)CC1 C1(C(N2CC3C(Cn4cc(CN(CCOC)C)nn4)(C3)C2)=O)CCN(C)S1(=O)=O C1(C(=O)NC(C(=O)NC2(C#C)CCOC2)CC(F)F)CN2CCC1CC2 N(C1CCCc2nc(=N)[nH]cc21)C(=O)NC1CCN(CC(C)O)CC1 c1(C(C)C)ccc2c(c1)CN(C(CC(c1ccccc1)N(C(N)=O)CCO)=O)C2 c1(C(=O)NC2C(C)CN(C(=O)CS(N)(=O)=O)C2)cccc(N)c1Br c1(NC2(c3n(CC=C)nnn3)CC2(C)C)cccc2c1CCC2(C)C C(=O)(C1=NOC2(CCC2)C1)N(CC(C)CNC(=O)CO)C Cc1cc(C)c(C(N2CCC(Nc3nccc(C(C)C)n3)C(C)C2)=O)c(C)c1 Cc1nsc(N)c1C(N1CCC(O)(CNC(C2CCC2(C)C)=O)C1)=O N1(C(c2c(CC)nn[nH]2)=O)CCC(CNC(=O)C(C2CC(F)(F)C2)O)C(F)(F)C1 C1(C)(C(=O)OC)CCN(C(=O)Nc2cc(-c3ccccc3)sn2)C1.C1C(C)(C)CO1 C1(c2n(C3(C)CC3)nnn2)(NCC(CO)C(C)(C)C)CCCC(C2CCCC2)C1 C(=O)(C(C)(C)C(F)(F)F)NC1CC(CNC(C(C(C)C)CN(C)C)=O)C1 C1(OC)CCN(C(=NCCC2CN(C(=O)OC)C2)NCC2CCOC2)CC1 c1(NC(C2(F)CN(C(C3CCCCC3)=O)C2)=O)cc2cc(Br)cnc2s1 C1(C(=O)NC2COCCC2NC(=O)CCc2cc(C)no2)(NC(C)=O)CCCCC1 C1(NC(CCC2(C)CN(C(c3cc(Cl)c[nH]3)=O)C2)=O)CCCCCC1(C)C C1(C(=O)NCC2CN(C(C(n3ccc(C)n3)(C)C)=O)CC2O)CCC2(CCC2)O1 C1(CC(=O)NC2C(CC)CCC2)C(C)CCCN1Cc1ccc(Cl)cc1 c1(C(=O)Nc2c(NC)cncc2)ccc(F)cc1NC1CCN(C(C)(C)C)C1 C(=O)(C(C)C(C)NC(C1(C)CCCCO1)=O)NCc1ccn(C(C)C)n1 Cc1cc(C#N)cc(C)c1CNC(=O)N(CC(C)(C)O)C C(=O)(C1=CCC(NC(=O)C(C)=C2CCCC2)C1)NC(C#C)(CC)CC C1(N=c2ccn(-c3cccc(F)c3C)[nH]2)(c2n(C(CC)(C)C)nnn2)CSC1C Cc1ccc(C(=O)NCCC2CCC(NC(=O)C#CC3(C)COC3)C2)c(=O)n1C C#CCCCC(C)C(=O)N1CC2CC2(C(=O)NCCN2CC=CCC2)C1 c1(C(N2C(C)C(NC(=O)C=C3CCN(C)C3)CCC2)=O)cccc2c1CNC2=O C1(CNC(Cc2nc(=N)[nH][nH]2)=O)CC(O)CN1C(=O)C=CC1CC1.C1C(F)C1 C1(CNC(C2CC(OC)C2)=O)CC(C)(C)CN1C(=O)C(c1cnn(C)c1)C C1(C(=O)NC(c2nc(C)on2)C)CCCCN(C(=O)Cn2ncn(C)c2=O)C1 c1(C(=O)OC)ccc(O)c(C(=O)N(CCCNC(=O)C=CBr)C)c1 N1(C(CC2CC(C)C2)=O)CCC(C=CC(=O)NC2CCC3(CC2)N=N3)CC1 N1(C(c2csc(Br)n2)=O)CCOCC(CNC(C2(F)CC=CC2)=O)C1 C1(CNC(Cc2c(C)con2)=O)CCN(C(=O)C(F)(F)c2cncs2)CC1C c1(OC)cc(C)c(C(N2CCCC2CCNC(=O)C2=CCOC2)=O)c(C)c1 Cc1ccc(OC(C)C(=O)NCC2(F)CCC(NC(=O)CN(C)C(N)=O)C2)cc1 C12(C(=O)NCC)CCC(OCCC)(CC1)CC2=O CCC(CC)(C(=O)NCC(F)CNC(c1c[nH]ccc1=N)=O)c1ccc(Cl)cc1 C1(C(N(C)CCNC(c2ccc(CO)o2)=O)=O)CC(=O)CC12CCC2 c1(CCC(=O)N(CCN(C(C)C)C(C2(C(C)(C)C)CCCO2)=O)C)cncn1C C1(CC(=O)NCC(C)(C)OCCNC(CCc2ncn(C)c2)=O)CCCS(=O)(=O)C1 Cc1cccc(Br)c1C(C(=O)NCC(C)CO)NC(c1cc(CO)[nH]n1)=O CCC(C)(C#N)C(=O)N1CC(CN(C(=O)C=Cc2nc(C)c(C)[nH]2)C)C1 N1(C(c2nnc(C)s2)=O)CCCC(C)C1CNC(c1cc(C2CCC2)no1)=O CC(C)(C)C(CNC(c1c[nH]nc1C1CCC1)=O)NC(C1CCCSC1)=O c1(CNC2CCC(NC(c3c(F)cc(Cl)cc3F)=O)C2)cccc2occc12 CCC(C)CCCC(=O)N(CCC(=O)NC(C)CN(C)C)CC C1(OCC)CN(C(=O)C(CCC2CC2)SCC)CC1CNC(c1cc(C)on1)=O c1(NC(c2n(C)ncc2)=O)cnc2[nH]cc(-c3cnn(C4CCC4)c3)c2c1 c1(C(C(=O)N(CCN(C(C(F)=CC)=O)C)C)N(C(=O)COC)C)ccccc1 C1(C(=O)NC(C)Cn2cc(-c3cnn(C)c3C)nn2)CCOC12CCCC2 c1(CC)cc(N)c(C(=O)NCC(C)NC(=O)C(C)CC(C)(C)C)c(F)c1 Cc1ccc(CNC(=O)CCOCCCNC(c2cc(CCO)on2)=O)o1 c1(C(N(C2CCCN(C(C3C(C=C)C3)=O)CC2)C)=O)cnc2sc(C)cn2c1=O N1(C(C2(NC(c3cn(CC)nn3)=O)CC(F)(F)C2)=O)CC(C)=CC(C)C1 C=CC1CN(C(c2ccncc2OC)=O)CC1NC(=O)CCC(C)(C)OC c1(C(=O)NC(CN(C(C(C(C)C)OCC)=O)CC)C)ccc(OC)c2ccsc12 S(=O)(=O)(c1ccc(Br)c(Cl)c1)NC1COCCN(C(C2CC2F)=O)C1 C1(N(C(=O)CC2SC(=N)NC2=O)CC)CCN(C(=O)C(=O)N(CC(F)F)CC)CC1 C1(C(=O)NCCC2(CNC(c3c(C)cn(C)c3)=O)CC2)CC2CCC1CC2 c1(CC(=O)NC2CCN(CC3(OC(C)C)CC3)CC2)ccc(C(F)F)cc1 C=CC(C)(C)CC(=O)NCC(c1ccccc1)NC(C1CC1C(F)F)=O C(=O)(C1=C(C(C)F)N(CC2CCC2)C(=O)NC1c1ccn(C(C)C)c1)OCC c1(C(=O)NC2(CO)CCCN(C(C(C(=O)OC)(C)F)=O)C2)coc2c1COC2 c1(C2(C(=O)NCC(C(C)C)NC(c3c(C)snc3)=O)CCCC2)ccc(Cl)cc1 CC(C)CC(C(=O)NCC1CCCN1C(=O)C(O)(C1CC1)C1CC1)n1ccnc1 N(C1CN(C(C2CCC3CC23)=O)CCc2ccccc21)C(=O)CC1CCCCO1 c1(C(N2C(CN(C(COC(CC)C)=O)C)CCC2)=O)cc2ncccc2o1 c1(OC)c(Cl)nc(NC(C2CCCN(C(c3cc(C#N)ccc3O)=O)C2)=O)nc1Cl c1(SC)cnn(C)c1C(N1CCC(C2CCCN2C(c2ncccc2F)=O)C1)=O CC1(C)CNC(CC(N2CC(C)(C(N3CCOCC3)=O)C2)=O)C1 N1(C(C)Cc2ccccc2)CC2COCC2(C=O)C1.N1(C)CCOCC1CC#N c1(NC(C)Cc2ccc(Cl)cc2Cl)ccc2nnc(CCCO)n2c1 C12(CC(=O)NC3CC4C(C3)C4(F)F)CCC1CN(C(=O)C=CC(F)F)C2 c1(C(=O)NC2C(NC(C(C)CC(F)(F)F)=O)CCCC2)cc2c(s1)CC(C)(C)C2 Cc1ccnc(C(=O)N(C)CCOCCNC(=O)CCOC2CCCO2)n1 CCC(C)C(O)C(C)C(=O)N1CC(C)(C)CC1CCO C1(CNC(CN2C(C)CCC2)=O)CCN(C(=O)CCC2CCCN(C)C2)CC1 C1(C(=O)NCCOCC(C)C)(NC(c2ccc(=N)[nH]c2)=O)CCN(C)C1 c1(C(C(=O)NCC2(CO)CN(C(CCCOCCC)=O)C2)C)cccc(Cl)c1Cl N1(C(C(CC)Oc2ccccc2)=O)CC2CC1(CNC(=O)CCCOC(C)C)C2 N1(C(CCOCC(C)C)=O)CCCC(C(=O)NCC(=O)OCCOC)C1 c1(CC(=O)NC23CCCC(C(=O)Nc4ccccc4)(C2)C3)cc(F)c(Cl)cc1F N1(C(c2cc(C)c(Br)o2)=O)CC2CCCCC2(CNC(c2cn(C)cn2)=O)C1 N1(CC(C2CCN(C(c3ocnc3C3CC3)=O)CC2)F)CCCC12CCC2 N1(C(C2(Oc3ccccc3)CC2)=O)CC2(NC(C3CC(=C4CC4)C3)=O)CC1CO2 c1(OCCOC)ncccc1C(=O)N(c1cc[nH]n1)Cc1ccc(F)cc1 C12CCCCC1NC2=O.c1(C(N2CCC(CC=CC)C2)=O)ccc(OC)nc1 CC(C)CCCCC(=O)NCC1CC(CNC(=O)CC2CC2C)C1 c1(C(N2CCN(C(c3n(CC)nnc3)=O)C(C)C2C)=O)cnc2c(c1)nnn2C c1(CC)nnc2c(C(=O)NC3(CNC(c4scc(C)c4OC)=O)CC3)cccn12 Cc1cc2cccnc2nc1C(=O)NCC(CO)NC(C12CC(C1)C2)=O CCCC(CCC)CC(=O)NCC(O)CNC(C1Cc2cccc(F)c2O1)=O CN(C1CCOc2cc(F)ccc21)C(c1cc2c(C(F)(F)F)cncc2s1)=O C(=O)(C(F)(F)CC1CC1)NCC(CNC(C1CCOC1C(C)C)=O)OC c1(C(N(CC(CN(c2ncc(C)c(O)n2)C)O)C)=O)cnc([N+](=O)[O-])cc1C c1(CN2CCOCC(NC(c3c(C)ncn3C)=O)C2)c(Cl)ccc(Cl)c1Cl c1(OC)ccc(N)c(C(=O)NCC2C3CN(C(=O)CC4CC4)CC23)c1 C1(CNC(c2ncc(C)cn2)=O)C(C)CCCN1C(c1n[nH]cc1C)=O c1(NC(C2N(C(c3c(C)n(CCO)nc3)=O)CCOC2)=O)cccn2nccc12 n1(CCC(N2CCC(CNC(c3cc(O)no3)=O)CC2)=O)cnc2ccccc12 C(=O)(CC1=CCN(C(=O)CC(C)(C)CN(C)C)CC1)N(CC)Cc1occc1C C1(C(N(C)Cc2ncc[nH]2)=O)(CNC(c2cncn2C)=O)CC12CCC2 C(=O)(CC1=CCCCC1)NC(CC(=O)N(CC(CC)O)C1CC1)C(C)OC c1(C(=O)NCC(N(C)C(C2(CO)CCOCC2)=O)C2CC2)ccc(F)nc1F C(=O)(CC(C)(C)C#N)N1C(C(N2CCC2C)=O)(COC)C=CC1 C1(NC(c2ccnc(C)n2)=O)CCN(C(C23CC(CN2C2CC2)C3)=O)C(C)C1 N1(C(CN(CCC(C)C)C(=O)CC2CCCC(C)C2)=O)C2C=CCC1CC2 S(=O)(=O)(c1ccc(Br)cc1NC1CCN2CCCC12)NCC(CSC)OC C(CC(O)C(=O)NC1(N(C)C)CCCC1)NC(C(C)SC)=O C(C)(CO)(C(=O)NCCS(C)(=O)=O)NC(CSC)=O c1(C(=O)NC2CCN(C(CCC)=O)CC2O)cccc2occc12 c1(C(N2CCC(CC(=O)Nc3cccnc3)C2)=O)c(F)cncc1Br C(=O)(C(=O)N=S(C)(C)=O)N(CCCNC(C1(COC)C=CCC1)=O)C(C)C c1(OC(Cn2cc(-c3nccc(OC)n3)nn2)OC)ccc(Br)cc1C c1(C(=O)NCC2C(NC(C(CC)(C)O)=O)CC2)cc2cc(Cl)ccc2[nH]1 N1(C(C2CC=C(C)CC2)=O)CC(NC(=O)CCC=Cc2ccccc2)C2CC2C1 c1(C(C(N2CC(N(C(=O)C(C)C)CC)OCC2)=O)O)ccc(F)c(Cl)c1 C1(CC(=O)NCc2ccc(Br)cc2)COCCN1C(C1CCCC(O)C1)=O C1(NC(C2CCN(C(C(CC)O)=O)C2C)=O)CN(C)C(=O)C12CC2 C1(NC(=O)CCc2ncc[nH]2)CC2(CCN(C(C3CC4(CCCC4)CO3)=O)CC2)C1 N1(C(c2c(C)cn(C(C)C)c2)=O)CC2CCCC2(CNC(c2c[nH]c(=N)s2)=O)C1 c1(C(=O)NC2C(NC(C(Cn3ccc(C)n3)C)=O)C2)ccc(F)c(F)c1C N1(C(CC2N(C(C)C)CCC2)=O)CC2CN(C(C3CC4C=CC3C4)=O)CC2C1 C(C(CC)CC)N(C(=O)C(C)n1cccn1)CC=C(C)C Cc1cc(N)cnc1C(N1CCC(CNC(=O)CC2(C)CCCC2)C12CC2)=O N1(CC(C)C)CC(C(=O)NC2CCCCC2NC(=O)CCC2CCCC2)CC1=O c1(C(=O)NC(CC(C)NC(c2[nH]cc(C(=O)OC)c2)=O)C)c(F)cc(C)cc1Cl C1(C(=O)NCCN(C(C2CC2C2CCC2)=O)CC)CCCCC1(C)C c1(C(C)(C)C)cc(C(N2CCC(N3CCOC3=O)C2)C(=O)NCCCF)on1 n1(CC(N2CCN(C(c3nccc(C)c3)=O)CC2)=O)cnc2c1CCCC2 C1(C(=O)NCC2(CC#C)CCCN2C(=O)OC(C)(C)C)CCCCN1N=O c1(C(=O)NCC(C(C)C(C)C)NC(C2(C(C)C)CC2)=O)cnc2n(c1=O)CCS2 S(=O)(=O)(c1c(C)coc1C)Nc1cc(C)n(C)n1.C1CC(F)(F)Cn2cc(nn2)S1 N1(C(C)(C)CNC(c2ccc(Cl)s2)=O)CCN(C(c2cnc(S)[nH]2)=O)CC1 c1(C(=O)NCC(C)NC(c2c(OCC)nccc2)=O)nc(C)ccc1O OC1CCCC(N=c2[nH]c(=NCc3ccc(Cl)o3)[nH]c3c2CCC3)C1 Cc1cccc(CCNC(C23CC2CN(C(C2(CO)CCOC2)=O)C3)=O)n1 c1(OC)cc(CNc2cc(C)n(C(C)(C)C)n2)ccn1.N12CCC(CC1)C2=O c1(CNC(N2CC(OC)CC23CCC3)=O)cc(S(N)(=O)=O)c(C)o1 c1(-n2cc(C3CCNC3)nn2)ccc(Cl)cc1Cl.Cc1cc(OC(F)F)ncn1 C#CC1CCCN(C(=NCCCCN2CCCC2)NCc2ccccc2)C1 C=CCCCCCC(=O)NC1CC2CCC1N2C(c1nc(O)sc1C)=O c1(CC(Cn2ccnn2)NCCc2cscn2)ccccc1.C1(CC=O)CN(C)C1 C(=O)(C1=CC2CCCC12)N1CCCC(CCNC(C=Cc2cncc(C)c2)=O)C1 c1(C(C)C)ccccc1C(=O)N(C1(c2ccco2)CC1)C1CC1.NC=O C(=O)(CCCCCN=[N+]=[N-])NC1CC(C)(C(=O)NOC2CC3C(C2)C3(F)F)C1 C(=O)(C(CCN(C)C)NC(=O)CCNC(=O)CO)NCC(C)N(C)C c1(CNC(C(=O)NC(c2cn(CCCC)nc2C)C2CC2)=O)cc(C)nc(O)c1 C1(C(=O)NCCC(C)NC(CCN2CCN(CC)CC2)=O)C2CCCCCCC12 c1(OC)nc(=NCc2cccc(COC3CCCNC3)c2)[nH]cc1C N1(C(C(C2CC2)SC)=O)CCN(C(C)=O)CC1.c12cn(nn1)C2 C1(CN(C(COCc2ncc(C)o2)=O)C2CC2)CC1C1CCCCC1 Cc1nc(CCCNC(=O)CC2CCN(C(=O)Cc3sccc3C)C2)n[nH]1 Cc1cc(-n2cncn2)ccc1NC(=O)NCC(c1ccno1)C N1(C(CC=CC)=O)CCCC1CN(C(c1csc(-c2csc(C)n2)c1)=O)CC C(=O)(C(C)(C)C(=O)NCCF)NC1CC(C(N(C)C)=O)CC1O N12CCCC(C1)N(C(c1nccn1C)=O)CC2=O.CCCC(=O)NCC1CC1(C)C c1(C(=O)NCC(C)NC(=O)C(C)C(C)O)cccc2c1CCO2 C(c1ccc(F)c(Cl)c1)=CC(=O)NC(C1CCCC1)CNC(C(C)OCC#C)=O c1(C(c2nnnn2C2CCC2)N(CCCOC)CCO)ccccc1Br c1(SC)cccc(CC(=O)NCCC(C(C)C)NC(=O)C2=COCC2)c1 C1(NCCSC)CC2CC3CC(C2)CC1C3.C1(=O)C(C)(C2CC2)N1C c1(CC(C)C)cn(C2CN(C(=O)CC3CC(NS(C)(=O)=O)C3)C2)nn1 N1(C(CC2N(C(C(C(C)C)OC)=O)CC2)=O)CCC(O)(C(C)C)CC1 Cn1nc(CC(=O)NCC(CO)NC(c2cc(CCCO)on2)=O)cc1C1CC1 c1(C2(OCC)CC2)ccccc1C(N1CCN(C2CSC(N)C2=O)CC1)=O N1(C(c2scc(OC)c2)=O)CCC(C#N)(NC(C2CC=CCC2)=O)C1 c1(CNC(C(C2CC2)OC)=O)ocnc1C(=O)NCCC1C=CCC1 c1(NCCC(N)C2CC2)cccc(CCCC(F)(F)F)c1 Nc1nc(-c2cn(CCCC(=O)NCC(=O)O)nn2)ccc1[N+](=O)[O-] C1(C(C)(C)C)CN(C(C(=O)CCc2ccc(NC(C)(C)C)nc2)=O)CCC1CO N1(CC=CC(N2CC=CC(NC(=O)C=CC3CCCC3)C2)=O)CCCS1(=O)=O C1(NC(c2cnc(S)[nH]2)=O)CN(C(C2CC3CCC2C3)=O)CC12CCCC2 c1(NC(C2CC(c3cccc(F)c3)C2)=O)nnc2n1CCNC2 C1(CCCC)CCCCC1Nc1cccc(NC(=O)C2CC2)c1 c1(C(=O)NC(C2CCN(C(c3ncc(OC)nc3)=O)C2)C)cccc(C#N)c1 C1(NC(=O)NC(C2CC(=C)C2)C)COC2(CCOCC2)C1 C1(C(F)F)(OC)CC(N)(C(=O)NCC2(c3ccccc3C)CCC2)C1 Cc1nncn1NC(=O)C(C)N(C(=O)CC1CC=CCN1C)C C1(C(N2C(C)CC(CNC(=O)C=C3CCCCC3)C2)=O)CC2(CCC2O)C1 c1(CC(=O)NCC2N(C(COCCCC)=O)CCC2C)c(Cl)cccc1Cl CC1CC2CCCCC2N(C(c2cnc(C(F)F)s2)C(=O)NC2CCC2)C1 C#Cc1ccc(C(=O)NCC(CC)NC(=O)Cc2cc(C)ccc2Br)cc1C c12oc(cc1C)C(=O)NCC1(CC1)CNC2=O.C1C2COCC12.CC c1(C(=O)NCC2(C(=O)NCCc3ccccn3)CC2)cc(F)c(O)c(F)c1 CC1(C)CC(CNC(C2CCCCNC2=O)=O)N(C(C2(C)CCOC2)=O)C1 c1(C(C)(C)C(=O)NC2CC(NC(=O)Cn3nnc(C#N)n3)C2)ccc(Cl)cc1Cl Nc1c(C(=O)NC2CCC(NC(c3ccnc4[nH]ncc34)=O)C2)cc(F)cc1F c1(C(N2CC(N(C(CCNC(=O)NC)=O)CCO)C2)=O)ccc(C(C)=O)cc1F C(CC1=CCN(C(c2cc(Br)cc(F)c2F)=O)CC1)NC(C(C(C)O)C)=O C1(C(=O)NCC2C(NC(=O)CCCC(F)(F)F)CC2)CCc2nnc(O)cc2C1 C1(C(=O)NC(CCC)CCO)CC(C)CN(C(=O)CCCC(=O)C2CC2)C1 Cc1nc2cc(CNC3CC3C(=O)Nc3nc(Br)cnc3Cl)ccc2s1 C1(N(C(C(OCC)C2CC2)=O)C)CCCN(C(c2ccccc2SCC)=O)C1 c1(C(N2CC(O)(CN(C(c3c(CC)noc3)=O)C)C2)=O)c(N)cc(C)cc1F C1(C(=O)NCc2c(C)ccc(F)c2)N(C(C2CC2(F)Cl)=O)CCCC1(C)C C1(C2CC2)(CNC(c2ccn(O)c(=O)c2)=O)CCN(C(c2c[nH]ccc2=O)=O)C1 c1(NC(CNC(C(CCC)CCC)=O)C2CC2)ncnc2cc(C)[nH]c12 CN1C(=O)CCC1CC(N1CCCC1CN(C(c1cn[nH]c1)=O)C1CC1)=O C12(CNC(C(CC)Sc3ccccc3)=O)CCC(C1)N(C(c1cccnc1)=O)C2 c1(OC(CC)C)ccc(C(=O)NC2CCC(NC(c3ncccc3O)=O)C2)cc1 c1(CNC(C(CCF)NC(C2C(C)=CCS2)=O)=O)cccc(F)c1C C1(NC(C(C)N2CCC2)=O)CN(C(c2ccnc(C(F)(F)F)c2)=O)C(C)(C)C1 c1(-c2n(CC(CCC)O)ccn2)ccc(OC)c([N+](=O)[O-])c1 O=S(=O)(C1=CC(O)(I)C=C1)N(CCCO)CCNCc1ccc(O)cc1 c1(C(C)CC(=O)NCC(O)COC(F)(F)F)cccc2ccccc12 c1(CCC)nnc(S)n1CC(=O)NCC1CCN(C(=O)Cn2nnnc2C)CC1 C1(NC(NC(CC)CC)=NCCN(S(C)(=O)=O)C)COc2c(C)cccc2C1 C12(CNC(c3ccc(CO)s3)=O)CCC(CC1)N(C(C1CC3CCC(C1)C3)=O)C2 c1(OC)cc(N2CCC(C(C)(C)NC(c3ccc(C(=O)CF)cc3)=O)C2)ncn1 Cc1ccc(C2(C(N3CC(C)(NC(c4cnnn4C)=O)C3)=O)CCC2)cc1 CC(CCCCN=c1ccn2nccc2[nH]1)NC(=O)CN(C1CCC1)C C1(CNC(CC(C)(C)OC)=O)CC2CCC1N(C(c1ccnc(F)c1)=O)C2 C1(C(c2nnnn2CC(F)F)NCCc2ccon2)CCC2CC2C1 C1(C(N2CC(NC(c3cc(C4CCOCC4)on3)=O)C2)=O)(COC)CCNC1=O c1(NC(N(C2CCCCCC2(C)C)C)=O)nccn2c(I)ccc12 C(=O)(C1=NN(C)C(=O)CC1)NC1CCCC(CNC(C2(CC#C)CCC2)=O)C1 CN1CCC(CC(=O)NCC2CC(NC(=O)Cc3ccco3)C2)C1=O Cc1ccn(C(C)(C)C(=O)N(C2CCOCC2)CC(C)C)n1 Cc1cc(Br)cc(F)c1C(c1nnnn1C1COC1)NC1CS(=O)(=O)C(C)(C)C1 c1(C(N2CC(CC=C)(NC(=O)C#CC3CC3)C2)=O)cn2c(n1)CC(C)CC2 N1(C(=O)CC2CNCCOC2)CCC(C(F)F)(C(=O)O)CC1 c1(NC(c2cc(-c3ccc(C#C)cc3)[nH]n2)=O)c(C)cc(F)cc1[N+](=O)[O-] c1(NCC(C(CC)CC)O)ccc(S(=O)(=O)N2CCCC(CC(=O)OC)C2)cn1 C1(OC)CC2CN(CCc3nc(-c4ccc(C(=O)NC)nc4)no3)CC2C1 c1(C(N(C)CC2N(C(C(CSC)C)=O)CCCC2)=O)cc(C)cc(N)c1 C12(CNC(C(CCC)OCC)=O)CCCC1N(C(c1ccccc1Cl)=O)CCC2 N(C1CCc2cc(NCC=Cc3cc(F)c(OC)c(F)c3)ccc21)C(CC)=O N1(C(C(C)Oc2ccccn2)=O)C2CCCC1CN(C(c1ccsc1C#N)=O)C2 N1(C(CCSc2n(C)nnn2)=O)CCN(C(C2C=CCCC2)=O)C(CCO)C1 C#CCC(CC(F)F)OCC(=O)NC1CC(NC(C2CCC(O)CN2C)=O)C1 C1(CC)CCN(C(=O)C(C)N2CC(C)C2)C1C(=O)NC(CO)C(F)(F)F CC1(C)CN(C(c2nc(Cl)c(C#N)s2)=O)CCC1NC(C1CCC(F)(F)CC1)=O c1(C(=O)NC2CC(NC(C3CC(C)SCC3)=O)C2)ccc(S(=O)(=O)CCO)cc1 CCC(CC)CC(F)C(=O)NC1CC(=O)N(C2CN(C(c3ccnn3CC)=O)C2)C1 N1(C(Cn2n(C)c(C3CC3)c(C#N)c2=O)=O)CCOc2c(F)cccc2C1 n1(CC)c(C)cc(C(=O)NC(C(C)NC(=O)CCS(N)(=O)=O)C(C)C)c1C C(=O)(C1=COCCC1)N1C(C)CC(CNC(c2ccc(OCC(F)F)cn2)=O)C1 N1(C(COC)=O)CC2CCC2(CCNC(=O)CCP(C)(C)=O)C1 C(=O)(C(C(C)(C)C)OC(C)=O)NC(CC)CNC(=O)CC(C)(C)OC C12(NC(c3cnc(SC)s3)=O)CCCC1N(C(=O)C=Cc1ccn(C)c1)CCC2 C(=O)(CCC1=CCCCC1)NC1CC(N(C)C(C2CC2c2ccsc2)=O)C1 c1(CC(=O)NC2CCCC(n3cc(C(=O)O)nn3)C2)csc2cc(Br)ccc12 N1(C(C(C)(C)OC(C)C)=O)CCCN(C(c2scnc2C2CC2)=O)C(C)C1 C1(NC(c2scnc2Cl)=O)CCCC12CCN(C(c1sccc1C1CC1)=O)CC2 C1(C(=O)NC2(CNC(=O)CN3CC=CC3)CCC2)C2CCC=C3C(C2)C13 C1(C(=O)NC(c2cc(C(N3CCOCC3CC(N)=O)=O)on2)C)CCC(F)(F)C1 N1(C(C2(C(C)(C)OC)CC2)=O)CCC(N(C(=O)C(C2(O)CCCC2)F)CCO)C1 C(=O)(C(C)(CNC(c1cc(F)ccc1F)=O)CC)N(CC(CC)OC)C N1(C(C(C2C(C)C2)ONC(c2cc(C3CC3)[nH]n2)=O)=O)CCc2nccnc2C1 CCC(C)CC(=O)NCC(C1CC1)N(C(=O)CCC(=O)NCC1CC1)C N1(C(C(=Cc2cnc[nH]2)C)=O)CCOCC(NC(=O)CC2(C#N)CCCCC2)C1 C1(CC)CCCCC1C(=O)NCCn1ccc(C(=O)NCCS(N)(=O)=O)c1 c1(C(=O)NC23C(n4cc(CC(C)(C)O)nn4)CC(CC2)C3)cnc2ncccn12 C(C(=O)N1CCC(C(N2CC(N(C)C)C(C)C2)=O)O1)c1c(SC)cccn1 c1(N(CCC2CCN(C(c3c(C)cns3)=O)CC2)C)cc(=O)n2ccccc2n1 C1(C(=O)NCCCCNC(c2n(C)nc(C(F)(F)F)c2)=O)CC2CCC(C1)O2 c1(CC(N2C(CNC(C3CC3CF)=O)CCCCC2)=O)ccc2c(c1)OCCO2 C1(OC)CCC12CC(C(=O)NC1(CCNC(=O)C=CC(C)(C)C)CCC1)C2 CC(C)(CC(=O)NCC1CC1NC(C1CNC(=O)N1)=O)C(F)(F)F Cc1cc(-c2cn(CC(=O)NC(C)(CO)CC(F)F)nn2)nnc1O C1(c2nnnn2C2CC(F)(F)C2)(NCCc2c(C)cccc2)CCN(C)C1C c1(C(N2C(C(C)(C)C)C(C(=O)NCC(O)CF)CC2)=O)ccc2occc2c1 c1(C(=O)NCCCN(C(CC2CC(=C)C2)=O)C2CC2)cccc(C2CC2(F)F)c1 N1(C(C(Cn2cncn2)NC(c2c(C)nc(C)o2)=O)=O)CCC2(CNC(=O)O2)C1 c1(-c2cc(C)nn2C)nc2ccc(N(CC)Cc3ccc([N+](=O)[O-])cc3F)cc2s1 Nc1c(C(=O)NCC2CC(NC(C3(F)CC4(CCC4)C3)=O)C2)cccc1[N+](=O)[O-] c1(C(C)C)cnc(Cl)nc1N1CCC2CC2(NC(=O)C(C)OCC2CC2)CC1 N1(C(c2c(C)ccnn2)=O)CC(C(=O)NOCCCCN(C)C)CC1(C)C.C(=O)O CC(C)C(O)C(F)(F)C(=O)N(CC(CO)(CO)NC(=O)C=Cc1cccnc1)C C(=O)(CCCN=[N+]=[N-])NCC1C(CNC(C2N(C)CCC2)=O)C1 c1(C(=O)NCC2CCN(C(CCN(CC)CC)=O)CC2)cccn2cnnc12 C1(NC(C(C2CCOC2)OC(C)(C)C)=O)CC2C(NC(c3cc[nH]n3)=O)C2C1 C1(CNC(C(COC)(C)O)=O)CC2CCC(C1)N2C(c1c[nH]c(C(N)=O)c1)=O c1(CNC(CC2N(C(c3nc(C)n(C)c3)=O)CCCC2)=O)cccc(F)c1O C1(C(N2CCCCC(NC(Cc3nc(C)[nH]n3)=O)C2)=O)CCc2ncncc2C1 c1(C(=O)NC2CCC(C(=O)NCc3nc(COC)on3)C2)nc(O)sc1C N1(C(CCC(C)OC)=O)CCC(F)(CNC(C2CC2c2ccccc2C)=O)CC1 c1(C=O)ccc(C)nc1.N1(C(CCC)=O)C(C2CCCC2)CC1C N1(C(c2cc(CNC(C3(C)C(C)CCCC3)=O)oc2)=O)CCC2(C1)CN(C)C2 c1(C2CCN(C(COc3c(C)cccc3)=O)CC2)cccc2c1OCCO2 N1(C(=O)CC2CC(O)C2(C)C)CC(C)(C)OC(C)(C)C1.CC(C)C1(F)CNC1=O c1(C(NOCC(=C)Br)=O)cc(Br)ccc1OC1CCC1 CCC(CNC(c1nnsc1C)=O)(CC)C(=O)Nc1ccc2nonc2c1 c1(CS(=O)(=O)NC(C(C)OC2CC2)=O)ccc(Br)cc1 CC1COC(C(=O)NC(C)CN(C)C(c2cn(CC(F)(F)F)cn2)=O)C1 c12nccc(n1)N2.N1(C(N(c2ccccc2)C)=O)CC2C(CN=[N+]=[N-])C2C1 c1(NCC(n2ncc(C)c2)C)ccc2c(c1)CCC2 c1(C(=O)NCCN(c2ncnc3sccc23)CC)cnc(O)c2ncccc12 C(=O)(CCCC(C)O)NC1CC(CNC(COCc2cccc(OC)c2)=O)C1 Cc1ccc(C(=O)NCC2(O)CCN(C(=O)C(n3cc(C)cn3)C)CC2)c(C)c1 N1(C(C(C)SC)=O)C2CCC1C(CNC(=O)Cc1ccc(C)c(Br)c1)C2 c1(OC)ccc2ccc(CNC(c3ccccc3)CF)cc2c1 C(N=c1[nH]cnc(=N)[nH]1)C1C(NC(CCNc2c(OC)nccc2)=O)CCCC1 C1(C(=O)NCCOC(C)=O)CCN(C(=O)CC2(C)CCOC2)C1C(C)C CN1CCC(CCNC(C2C=CCN2C(C2CC=CC2)=O)=O)C1=O c1(C(N(C(C)CN(C(=O)CC2CCC2(F)F)C)C)=O)ccc2c(c1)CCCCN2 c1(C(N(C)CC2CCSCC2)=O)c(OC(C)(C)C)c(Cl)cc([N+](=O)[O-])c1Cl N1(C(C2(F)CCN(C(CN(C(C)C)C)=O)C2)=O)CCCC2CN(C)CC12 Cc1cc(O)nc(C)c1C(=O)NC1CN(C(=O)CC(C)CN(C)C)C(C)(C)C1 C1(NC(CC(C)N(C)C)=O)CN(C(=O)CCSc2ccc(F)cc2)C2(CCCC2)C1 C1(CNC(Cc2cc(CC)no2)=O)CCC(C)CN1C(C1(NC(C)=O)CCC1)=O c1(CN(C)CCOCCN(C(=O)CCCC2CCCC2)C)cc2n(n1)CCCC2 C1(CNC(c2ccc(CC3CC3)s2)=O)CC(F)(F)CN1C(C1C2CCCOC12)=O N1(C(c2c(C)cn(C(C)C)c2)=O)CCN(C(=O)Cc2c(Cl)cnn2C)C(C)C1 c1(NC(C2CN(C(c3cc(Br)nc(Br)c3)=O)CCO2)=O)cccc(F)c1F O(NC(=N)C1(C)CCOc2ccccc21)CCc1ccc(OCCCCC)cc1 c1(OCC)ncc(C(N2CCCC(C(C)(C)C)C2)C(=O)NCc2cccs2)cn1 c1(OC)cc(C(=O)NC2(C)CCN(C(=O)C(C3CCCO3)C3CC3)C2)ncn1 c1(C(=O)NCCCN(C)C(C2CC(F)C(=O)N2)=O)cc2sc(F)cc2[nH]1 c1(C(C)NCCC2CCCO2)ccc(I)cc1 c1(C2CC2c2ccccc2)ncc(F)cn1.c1(CC(=O)N2C(C)C2)ccsc1 c1(C(CNC(Cc2ccc(C)s2)=O)NC(C2C=CCC2)=O)ccccc1CO C(=O)(C(C)C(F)(F)F)NCC(CC(=O)N(CCC(=O)OC)C1CC1)C1CCC1 C=C(C)C(C)(O)C(=O)N1CCCC(F)(CNC(c2ccc(C)cc2Cl)=O)C1 C1(CC)CN(C(=O)CC(O)C(C)C)CCN1C(c1cnc(C)[nH]c1=N)=O c1(C(=O)NCCC2CCCN(C(c3nc(N(C)C)oc3)=O)C2)cccc(N)c1O c1(CC(C)C)cn(CCN(C(=O)C(C)c2ccsn2)C2CC2)nn1 c1(COC)nc(NCCCCOC(C)(C)C)cc(=NC2CC(CO)C2)[nH]1 C1(NC(CNC(C)=O)=O)CN(C(=O)Cn2nnnc2C(C)C)CC12CCOCC2 N12CCc3cc(ccc31)CNC2=O.C1(c2nn[nH]n2)(C(C)(F)F)CC(F)(F)C1 n1(CCC)nc(C)c(C(=O)NCCCn2cc(-c3ccc(F)c(F)c3)nn2)c1C Cc1cc(CNC(c2cc(CNC(=O)C(C)n3cnnn3)no2)=O)nc(C)c1 c1(CC)ccc(C(=O)NCC23CC2CN(C(=O)C2=CCCCC2)C3)c(O)c1 CCC(C)(C)C(O)C(=O)N1CC2CC(NC(=O)CCC(N)=O)C2C1 c1(C(N2CCC(N(C(C3CC(CC)OCC3)=O)C)CC2)=O)nccc2occc12 CC1(C)C(C(=O)NCC2CC3CC3C2)CCN1C(=O)CCCNC(N)=O c1(NC(N)=O)ccc(NC(=O)Nc2ccc(C3CCC3)nc2)cc1 C(CN=[N+]=[N-])(C(=O)N(C)Cc1c(C)noc1C)NC(c1ccc(OC)s1)=O C#Cc1ccc(C(=O)NCC(C(=O)NC2CC(=O)NC2=O)N(C)C)nc1 C1(C(=O)NCc2c(C)nn(C)c2C)COc2ccccc2CN1 C1(NC(C2(OCC)CCC2)=O)CN(C(c2cc(C)n(C)c2)=O)CC1N=[N+]=[N-] C(C)(C)(C(C)CC(=O)N1CCCC(O)C1)NC(C1C(C(C)C)CCC1)=O CC(C)C(C(=O)OC(C)(C)C)C(=O)NCC(C)NC(c1cc2n(c1)CCCC2)=O C1(N(C(=O)C(C2CCCC2)OC)CCNC(C(C)=CC)=O)CCCCC1 C(C(C)(C)CC(=O)NC(C(=O)N1CC(CC(F)C(=O)OC)C1)C1CC1)SC CC(C(F)C(=O)NC1CCN(C(c2cnn(C)c2N)=O)CCC1(F)F)C(F)(F)F c1(CC(=O)NC2CCN(C(=O)C(F)(F)c3cscn3)CC2O)ncc(F)cc1F c1(C(=O)NC(CC=C)CNC(=O)CCCn2ccnc2)cnn(CCC)c1Cl c1(C(=O)NC2CC3CN(C(CC(=C)C)=O)CC2C3)ccc2c(n1)CCC(C)C2 C(c1ccc(F)nc1)=CC(=O)NCC(C1CCCCC1)NC(C(C=CC)O)=O N1(Cc2c(C)cc(F)cc2)CCC2CC(C(=O)NCC(O)CO)C2C1 c1(SCC(=O)NC2(CF)CCN(C(C(C)=C(CC)C)=O)C2)nc2ccccc2s1 c1(C(=O)NC)cc2ncc(CC)cc2[nH]1.c12ccccc1NC(C#C)CNC2=O c1(C(=O)N(C2CCCOC2)CCO)n[nH]c2cccc(-c3ccc4[nH]ccc4c3)c12 N1(CCc2cn(CC)nc2)CCC(NC(=O)Cn2cc(Cl)cn2)CC1C N1(C(c2cc(OC)c(O)cc2)=O)CC2CCCCC2(CNC(c2cc[nH]n2)=O)C1 C(=O)(C1=NOC2(CCC2)C1)NC1C(CNC(c2c(S(N)(=O)=O)scc2)=O)CC1 C(=O)(C(C)(F)C(C)(C)F)NC(C(C)C)C(=O)NC1(C)CCCCCC1 N1(C(c2ccccc2N2CCC(O)CC2)=O)CCN2CCOCC2C1 N1(C(CN2CCC(C)C2)=O)C2CCCC1CC(CNC(=O)C1=NNC(=O)CC1)C2 c1(CC(=O)N(C2CCN(C(=O)C(C)NC(C)=O)C2)CC)ccc2c(c1)CC2 C1(c2ccc(OC)o2)CCCCCN1CC(c1cscc1Br)=O CCC(F)(C(=O)OC)C(=O)N1CCC(COC)(NC(c2ccc(Cl)nc2OC)=O)C1 C(=O)(C(C)C(C)c1ccc(F)cc1)NC(CNC(C1(CC)C=CCC1)=O)C(C)C CC1C=C(C(=O)NC(C)CN(C)C(c2csc(C3CCCC3)n2)=O)CC1 C1(CC)CN(C(c2ccnn2CC(F)(F)F)=O)CCC1NC(=O)COC(C)(C)C CC(CNC(c1cn(COC)nn1)=O)C(=O)NCCN(C1CCCC1)S(C)(=O)=O CC(C)C(C)(CN=c1[nH]ncs1)NC(c1ncc(C(F)F)cn1)=O C1(=O)C(CCC2CC2)N(C)CCC=CCO1.C(C)(C)(C)NCCC N1(C(c2ccc(NC(C)=O)o2)=O)CCN(C(=O)CCCF)C2(CCC2)C1 N1(C(C(C)CC2CCCCC2)=O)CCN(C(=O)Cc2cncnc2)CC12CC2 c1(CSC)nccc(C(=O)NC(CCN(C)C(C2CC(CC3CC3)C2)=O)C(C)C)n1 c1(CC(=O)NC(C2CN(C(C3CNC(=O)N3)=O)CCO2)C)ncc(O)cn1 c1(CCNC(C)(CCC#N)c2nnnn2C2COC2)nc2ncc(Br)cn2n1 N1(C(CSCCC(C)C)=O)CC2(CCOCC2)C1 C1(CCNC(=O)C=CCO)COCCN1C(c1ccnc(-c2ccncc2)c1)=O C(CN=[N+]=[N-])(C(=O)Nc1cnn(C(F)F)c1)NC(Cc1c(C)n[nH]c1)=O c1(C(N2CC(N(C)C(c3cccc(F)c3N)=O)C(F)C2)=O)cc2cccnc2s1 CC1CC(NC(C2CCCO2)=O)CCN1C(c1ccc(C(F)(F)F)c(O)c1)=O C(C)(C(=O)N1CCCCCO1)n1cc(NC(C(C)SC(C)C)=O)nn1 N1(C(c2n[nH]c3c2CSCC3)=O)CCC2(CC(CN)CO2)C1.C(C=O)=CC=CC C1(C(=O)NCCCC2(NC(=O)COc3cccc(F)c3)CC2)CCCC(F)C1 CCCCC1C(=O)Nc2c(c[nH]n2)C(=O)N1C.C1(NC(C)(C)C)CCN(C(N)=O)C1 N1(C(c2cc(CC)nn2C)=O)CCCN(CCNC(C2(C)CCCO2)=O)CC1 c1(C(=O)NC2CCN(C(CC(=O)Nc3nccs3)=O)CC2)n[nH]c2c1CCC2 c1(C(=O)NC2(CC(=O)NCc3nc(C)on3)CCC2)ccc2occc2c1O C1(N(C)CC)(C(=O)NC2C(NC(C=CC)=O)CC2)CCOCC1 c1(CCC(=O)NC(C)C(C)NC(c2cc(C#N)c[nH]2)=O)nnc(S)nc1O c1(C(=O)NCC(CC=C)NC(=O)C(C)=C2CC2)cccc2cnccc12 C(=O)(C(C)(C)c1nncn1C)NCCC(C)NC(=O)CCCNS(C)(=O)=O Cc1nsc(C(N2CCC(C(=O)NC3CCC4CCC34)C2)=O)c1N N1(C(C2OCCN(CC)C2)=O)CC(NC(c2ccnnc2S)=O)CC(F)C1 C(C)(CCC(=O)N1CCCC1CNC(c1cnc(C2CC2)o1)=O)OC Clc1cccc2c1OCC2NCc1ccc(CNc2ncccn2)cc1 C1(C(=O)NC(CCNC(c2cc(C)n(C(C)C)n2)=O)(C)C)CCCCC1(F)F c1(C(N(CCn2cc(CCN3CCOC3=O)nn2)CC)=O)cnc2[nH]cncc1-2 c1(NC(C)=O)c[nH]c(C)c1C(N1CC2C(CNC(=O)CC(F)F)C2C1)=O C1(C2CCC2)(C(=O)NC(CC(C)NC(c2c(C(C)C)ocn2)=O)C)CC1 N1(C(CCOCCOC)=O)CCN(C(=O)C2CCc3c[nH]nc32)CC(C)(C)C1 CC1(NC(=O)Cc2ccsc2)CCN(C(C2(C#N)CC2C(F)(F)F)=O)C1 N1(C(COCCC(C)C)=O)CCC2CN(C(c3ccc4c(n3)NCC4)=O)C2C1 C1(NC(C(COC)C)=O)CCN(C(C2CC2c2ccc(C)cc2)=O)CC1 N1(C(CC(C(C)C)C)=O)CC2(CCC(CNC(C34CC(CO)(C3)C4)=O)O2)C1 c1(NC(C2CCCCN2C(=O)NC2CN(C(=O)C3CC3)C2)=O)cccc(Cl)c1 C1(NC(Cc2c(C)n[nH]c2)=O)CCN(C(=O)C(O)CC2CCCC2)CC(O)C1 c1(C(=O)NCC2(NC(C3(O)CCOCC3)=O)CC3CCC2C3)ccn2nccc2n1 N1(C(CCCCOCC)=O)CCCCC12CN(C(=O)Cc1cc(C)on1)C2 Cn1c(C(=O)N(C2(C(=O)NC3(CCC4CCOCC4)CC3)CC2)C)ccc1C#N N1(C(CC=C)=O)CCCC(NC(C2CCCC(C(=O)OCC)CC2)=O)CC1 N1(C(C(N(C(c2cc(C)c(C)s2)=O)C)C2CC2)=O)CC(C)(C)C2COCC12 C1(N=[N+]=[N-])(C(N(CCC)CCO)=O)CCN(C(=O)C(F)CC2CCOC2)C1 c1(C(=O)NCC2CN(C(c3c(C)cc[nH]c3=N)=O)C2)ccnc2ccc(F)cc12 S(=O)(=O)(c1cn(CC(F)(F)F)nc1C1CCCC1)C(=O)Nc1c(C(=O)OC)ncs1 N1(C(C2C(CC)C2)=O)CC(CNC(=O)Cn2cc(Br)cn2)C2(CC2)C1 c1(OC)ncc(Br)c(C)c1C(N1CC2(CCC(NC(=O)Cc3ccn(C)n3)C2)C1)=O c1(CC(C)NC(C2COCC2NC(=O)CCCF)=O)ccncc1 c1(OC)cc(-c2nc(C3CCCC3)nn2C2CC3CCC2C3)ccc1OC N1(C(CCNC(CCOCCOCC)=O)=O)CCC(CO)CC1C C1(C)(CNC(c2n(CC)ncc2)=O)CCC(Nc2ncc(OC(C)C)cn2)CC1 c1(OCC(CNC=O)O)cc(F)cc(F)c1.N12CC=CC(C1)NCC2=O Cc1cc(=NC2C(C)CN(C(c3ccnc(CO)c3)=O)CC2C)[nH]c(C2CC2)n1 CC(C)CS(=O)(=O)CCC(=O)NC1CC1NC(c1ccc(=O)n(C)c1)=O N1(C(c2cc(COC)on2)=O)CCC2(NC(=O)C(F)CC(C)C)CCCCCC12 N12CCCC1COC2=O.C1(N(C2C3CC(C3)NC2=O)C)CCCCC1.CCCC N1(C(CN(CCOC)C)=O)CC(C(N2CC(Cn3ccnn3)C2)=O)C(F)(F)C1 C(=O)(C(F)CC(C)(C)NC(=O)CN1CSCC1=O)NCCN(C(C(C)C)C)C C1(CNC(C2CCCOCC2)=O)CC(O)CN1C(c1ccc(C(F)F)cn1)=O c1(C(C)C(=O)NCCCN(C(=O)Cc2ccc(=N)[nH]c2)C)cccc(O)c1 C=CCC(C)(C)C(=O)NCc1ncc(C(=O)O)s1 Cc1cc(C)c(C(=O)N(C2CC2)Cc2ccc(Br)cc2F)c(OC2CCOC2)n1 C1(CCNC(C(C)SC)=O)CC(F)(F)CN1C(c1cccc(C2CC2)n1)=O N1(CC(=O)NCC2(C)N(C(C(CC)C#N)=O)CCC2)c2ccccc2CS1(=O)=O CC1=C(C(=O)NC(CC(N)=O)C(=O)NCC(CC2CC2)CO)CCO1 Cc1nc(N2C3CCC2CN(C(c2ccn4cncc4c2)=O)C3)c2c[nH]nc2n1 C1(CNC(CC(=O)NCC)=O)CN(C(c2c(Br)noc2C)=O)CCO1 Cc1nc(C(N2CCCCC2CCNC(=O)CC2COC(=O)N2)=O)c(C)s1 C1(CC(=O)N(C2CCN(C(c3ccon3)=O)CC2)CC)CC2(CCC2)CCO1 c1(CCC(=O)NC(C2CCCN(C(C3CCOC3)=O)C2)C)cncnc1O c1(C(=O)NCCCN(C(CC2CC(CC)OCC2)=O)C)c(C)nn(C2CC2)c1Cl c1(OC)nn(C)cc1C(N1CCCC(C(C)NC(=O)C=CC2CCCCC2)C1)=O CC1CC2CCC(C(=O)NCC3C(C)CCCN3C(c3coc(Cl)c3)=O)CN2C1 N1(C(Cc2ncn(C)c2)=O)CCCC(CNC(=O)Cn2cc(C3CC3)cn2)CC1 c1(CC)nccnc1C(=O)N(C(C(=O)NCCCn1cnnn1)C1CC1)C Cc1cc(CNC(=O)C(C2CCCO2)NC(c2ccc(C)c(O)n2)=O)nc(C)c1 c1(C(=O)OC)ccc2cncc(Br)c2n1.C1(C(N(CCCOC)C)=O)CC1(C)C C1(C(=O)NC2CN(C(=O)C3CC3)C2)CCCC2(CC2)C1.C12(CCOC1)CC(=O)N2 CC(C)CC(C(=O)N1CC(C)(O)C1)NC(=O)CC1CCCC1O N1(C(Cc2c(C)cccc2)=O)CC(CNC(=O)C(C)C(C)(F)F)C2(CC2)C1 C1(CC(N2C(C3(NC(C(C)OCCC#C)=O)CC3)CCC2)=O)C(C)(C)C1(C)C C#Cc1cnc(C(N2CCC(C3CC3)C2C(=O)NOCC2CC2)=O)c(C)c1 CC(CC(C)(C)C)C(=O)N(CCC(=O)NC1CCN(CC2CC2)C1)CCO N1(C(C2(Cl)C(C)(C)C2)=O)CCN(C(=O)CN2CCN(C3CC3)CC2)C2(CCC2)C1 N1(C(CNC(=O)CN(C(c2cn[nH]c2)=O)C2CC2)=O)CCC(C2CCC2)C1 C1(C(=O)NCCC(C)CO)(CNC(C(C)OCCC#C)=O)CC=CC1 C(=O)(C1=NNC(=O)CC1)NCC(C1N(C(c2cc(C)nc(C)n2)=O)CCC1)(C)C N1(C(CCNC(CN(c2ccnn2C)C(=O)OC)=O)=O)CCCCC2CC12 c1(OC)ccc(C=CC(=O)NC(C)CNC(=O)COC(C)C)cc1OC c1(CN(C(C2CCCN2C(=O)C=Cc2cccs2)=O)C2CC2)ccccc1 Cc1csc(C=CC(N2CC(NC(c3ccn(C(F)F)n3)=O)C3CC23)=O)n1 Cc1ccc(C(=O)C(N2CCCC2CN(C)C)=O)cc1C.N12CCCC(C1)C2=O CC1CCN(C(=O)CC2(C#N)CCC2)CCN1C(c1cccc(C(F)F)c1Cl)=O c1(C2CN(CC3(c4c(C)cccc4)CCOCC3)C2)cc(Cl)ccc1Cl N1(C(C(=O)NC(CSC)=O)=O)CCN(C2CCC(Nc3cnn(C)n3)C2)CC1 CC(C)(C)CC(F)C(=O)NCC1(C(N2CC(C(=O)C3CC3)C2)=O)CCCCC1 N1(C(c2cc(OC)ns2)=O)C2CCC1CN(C(=O)C(C)(O)C1CCCCC1)C2 O=C1CCC(C(=O)NCCCOC2CCOCC2)C2(CCOCC2)N1 Cc1cc(C(=O)NC(C)(CNC(=O)Cc2ccc(F)cc2)C(C)C)c(C)o1 C1(C(=O)NCCCC(C)C)CCCC(NC(=O)C=CC2CCCN2C)CC1 N1(C(=O)C=Cc2cnccn2)CCN(C(=O)COCCCF)C(c2cn[nH]c2)C1 Cc1sc(=O)n(CC(N2CCC(NC(C3CCN(C)C3=O)=O)C(O)C2)=O)c1C CC(C)C(CN(C)C)C(=O)NC(C(=O)N(CC(C1CCCC1)O)C)C(C)C c1(NC(CC2(NC(C3=CC(=O)CC3)=O)CC2)=O)cncc2ccccc12 N1(c2nnc(C)s2)CCCC12CCN(C(C13CCC(C)(CO1)C3)=O)C2 C(CC(N)=O)(C(=O)NCCN1CC(OC)C1)NC(CC1CC(OC)C1)=O C#CC1(O)CCN(C(C2CC(=O)N(c3ccccc3C#N)C2)=O)CC1 CC1=C(C(=O)NC2CCC(CC(N3CC4(C3)CC4(F)F)=O)CC2)COCC1 C(=O)(CCCCN=[N+]=[N-])NC1(C)CCN(C(=O)C#CC2CC2)C1 C12(C(N(CCC)CCN(C(=O)C(COC)OC)CC)=O)CCCN(CC1)S2(=O)=O n1(C(CC)CC)nc(-c2ccc(Cl)nc2)nc1Cc1ncc(C)o1 c1(NCCC)ccc(C(=O)N(C)C(c2nc(C(C)C)no2)C)cc1F Cc1ccc(NC(C2CC3CCNCC23)=O)c(C(N)=O)c1 C(C(=O)NCC(C)(C)NC(=O)C(=Cc1c[nH]cn1)F)(C(C)C)SCC(C)C C(=O)(C(CC(C)C)C(N)=O)NC1CCC(NC(C2CC3(CC(=C)C3)C2)=O)CC1 C(=O)(C#CC1CCCCC1)NC(CN(C)C)C(N1CCC2(CCOC2=O)C1)=O C1(NC(CSCC=C)=O)CN(C(=O)CC(C)c2ccco2)CC2(CCC2)C1 C(=O)(C1=CC2CCCCCC12)N1CC(CNC(=O)CC2CC3(CCC3)C2)C1 c1(NCC(=O)NCCC(C)(C)NC(C(CC)C)=O)nccc(OC)n1 N1(C(CCC(C)N(C)C)=O)CC2(CO)CC1(C(N1CCC3CC13CO)=O)C2 N1(CC)CC(C(=O)NC2CC(NC(=O)C=CC(=O)N(C)C)C2)NC1=O c1(N(CC(=O)NC)C)nc2cc[nH]c2c(=NCc2c(SC)cnn2C)[nH]1 CC(C)C(C(=O)NCC1CC(F)(CNC(=O)C(n2cc(Cl)cn2)C)C1)N(C)C C(=O)(C#CC1(C)CCCO1)N1CCCC(N(C)C(c2ccc(C(N)=O)s2)=O)C1 C1(NC(CC=CCC)=O)CN(C(=O)CC2CCC(F)(F)CO2)CCC1O CCC(C(=O)OC)C(=O)NCc1csc(C(=O)NC2CC2c2cnn(C)c2)c1 N1(C(Cc2ccc(C)c(Cl)c2)=O)CC2CCC1C(NC(=O)CC1CCCOC1)C2 Cc1cnncc1C(=O)NC(CNC(=O)CCCNC(=O)C1CC1)CC(C)C CCCCCCCNC(=O)CCN(C(=O)CCc1conc1C)CCCO N1(C(CC(C=C)CCC)=O)CCN(C(c2cnc(O)c(OC)c2)=O)C2(CCC2)C1 CCC(C(C)(C)C)NC(=O)Cc1ccc(OC)nc1 C1(C(=O)NCCC23CC(CO2)C3)CC12CCN(C(c1ccc(CO)o1)=O)CC2 CSC=CC(=O)N1CCC(OCCNC(C2(F)CCC2)=O)C1 CCC(O)C(C)C(=O)N(CCCCCNC(=O)C(c1ccc(Cl)cc1)C)C CC1(NC(C2CCCCN(C(=O)CCCn3cncn3)C2)=O)CCCC1(F)F n1(CC(=O)N(C)CC2(NC(C=C(CC)C)=O)CC2)ccc2c(C)cccc12 Cc1cc2ncnc(N3CCC(NC(C4CC(O)C4)=O)C(C)C3)c2[nH]1 C1(CNC(CC2C(C)C(=O)CC2)=O)CCC2(CCC2)CO1 c1(C(=O)NC(C2CCCN2C(c2cc(C#N)ccn2)=O)C)ncc(Cl)cc1F N1(CC(N2CCC(C)C(CNC(C3(C)CCC3)=O)C2)=O)CCc2sccc2C1 c1(C(N2CCC(NC(C3CCC(CC)O3)=O)C2C)=O)cc(O)c2ccoc2c1 CCC1=NOC(C(=O)N(CCC(N2CCC(COC(C)=O)C2)=O)CC)C1 C(CCCN=[N+]=[N-])NC(C(C1CC(CNC(=O)OC(C)(C)C)C1)N(CC=C)C)=O Cc1ccc2ncc(C(=O)NC3CC4CCC3(NC(=O)C(F)C3CCC3)C4)n2c1 Cc1cc(=NCC2CCCC23CCC3)[nH]c(N2CCC(C(N)=O)CC2)n1 C(CN=c1[nH]cncc1Cl)N1CCCC(NC(C)=O)C1 c1(C(N(CC(C)NC(CCCOCC)=O)C)=O)cc(OC)ncc1F C1(C(=O)NC(C)CCCNC(=O)Cc2n[nH]c(=N)s2)CN2CCC1(C)CC2 C(CC(=O)N1CCN(C(c2cc(C=O)[nH]c2C)=O)CC1CO)(C(N)=O)NC(C)=O c1(CNC(C2CCCCC2)CC)ccc2c(c1)CCS2(=O)=O Cc1cnc2c(cnn2CC(N2CCCC(C)C2CC(N)=O)=O)c1 Cc1c(C(=O)NCCOC2CN(C(C3CCCOC3)=O)C2)cc(C2CC2)n1C.CO c1(OC)cnc(C)cc1NC(C1CN(Cc2sc(Br)nc2Br)C1)=O CCC(O)(CC(=O)NC1CC(C(=O)Nc2cnc(S)n2C)C1)c1ccccc1 c1(CC)c(C(=O)NCC2(C(F)F)CCN(C(c3cnsn3)=O)C2)cccc1F C=CC(F)(F)C(=O)N(C1CN(C(=O)C)C1)CC.c1(NC(=O)COCC)ccccc1 C=CCC(CC(=O)N1CCCC1(C)COC(C)=O)NC(=O)CS(=O)(=O)CC Cn1ccnc1CC(=O)NCC(C)(C)CNC(=O)CCc1ccsc1 c1(C(N2C(C)CCC(NC(=O)CC3C=CCC3)C2)=O)c2c(nn1C)CCC2 N#CC1CCC(CC(=O)NC2(CCNC(C3(C#N)CC=CC3)=O)CCC2)C1 Cc1nc2cc(C(=O)NC3CN(C(=O)CCCF)CC3(C)C)[nH]c2s1 c1(OC)cc2cnccc2cc1NC(=O)NCC1CCC2(CCCCC2)O1 C1(NC(Cc2ccc(OC)cc2)=O)CN(C(c2c[nH]nc2C2CC2)=O)CCC1C c1(C(c2nnnn2C(C)(C)CC)NC(C2CCCOC2)CC)nc(Cl)cs1 c1(C(=O)NC(CNC(c2cc(C)cc(O)n2)=O)CC(C)C)ccnc2[nH]nnc12 Cc1ccnc(C2CCN(C(=O)C(N3CCCC(NC(=O)CCN(C)C)C3)=O)C2)c1 c1(C(N2CC(C)(C(=O)NC(C)CCO)C2)=O)ccc(F)cc1Br N1(C(C2OCCN(C)C2)=O)CCCC2(C1)CN(C(c1cccc(O)c1)=O)CCO2 C(=O)(CCS(C)(=O)=O)C1C(CSC(F)F)NC(=O)C(CCSC)NCC1 N1(C(CC2CCC(=O)N2)=O)CCN(C(=O)C(F)(F)CCOC)CC2(CC2)C1 c1(C(=O)NC2CC(O)(CNC(CCC(C)N(C)C)=O)C2)cnc(N)c(N)c1 c1(OC)nccc(C(=O)NC2CC(CO)N(C(C3CC(C)CCO3)=O)C2)n1 C#CC(C)(C)C(=O)NC1CC(NC(c2n[nH]c(COC)c2C)=O)C1 c1(NC(c2ccc(Cl)cc2)=O)c(C(N2CCCC2C(=O)NC2CC2)=O)cccc1Cl c1(C(C(=O)NC2CCC(NC(C3CC=CC3)=O)CC2)O)ccc(Cl)c(F)c1 c1(-n2cc(CNC(n3ncc(C)c3)=O)nn2)ccc(SCc2cccc(F)n2)cc1 Cn1cnc2cccc(CNC3(c4nnnn4C4CCCCC4)CC4CC4C3)c12 C=C(Cl)C(C)(C)C(=O)N1CC(CC(C)NC(=O)COCc2ccccc2F)C1 CN1CCOC(C(N2CCCOC(CNC(C3COCC(C)(C)O3)=O)C2)=O)C1=O c1(CNC(CCCC#C)c2nnnn2C2CCOC2)c(F)cccc1Br C1(CN(C(=O)C(C2CCCCC2)F)C)CCCN1C(C1CCC(=O)C1)=O c1(C(N(CC(=O)NCC(=O)NCCO)CC)=O)sc(C)cc1C Cc1cc(F)sc1C(=O)NC(c1ccccc1)CNC(=O)C(C)NC(C)(C)C c1(C(=O)NCCCCNC(c2ccnc(C(F)(F)F)c2)=O)ccc([N+](=O)[O-])nc1 n1(CC(=O)NCC(C)N(C(c2c(CC)non2)=O)C)cccnc1=O CCCC(CCCS(C)(=O)=O)C(=O)OC1CCN(C2CCS(=O)CC2)C1 N1(C(C(CC)C(C)O)=O)CCC(C2(O)CC(NC(C3CC4(CC4)C3)=O)C2)CC1 CN1CCCC(C(C)(C)CNC(=O)C(C2CCC(F)(F)C2)O)C1 N1(C(CC(CC)C2CC2)=O)C2CCC1CC(N(C)C(c1cc(=O)c(C)c[nH]1)=O)C2 c1(C(=O)NC(C2CN(C(c3c(C)n(CCO)nc3)=O)C2)C)cccc(F)c1C C12(C(=O)Nc3c(OC)cc(CC(N4CCCC4)=O)cc3)CCC(F)(CC1)CC2 C1(CCCC)CN2CCN1C2=O.c1(N(C(=O)OC(C)(C)C)C)cnn(C)c1 Cc1ccc(CN2CCC(C(=O)Nc3ccc(I)c(C)c3)C(O)C2)c(Br)c1 C1(C(N(CC(C)NC(CCc2cc(C)[nH]n2)=O)C)=O)CCC(=O)N1C N1(C(CC(C)N(C)C)=O)CC(F)CC1C(=O)NCC1(C)CCC(=O)C1 Fc1cccc(-c2ncc(CN(c3ccc(Br)cn3)C3CC3)s2)c1 Cc1nc(CNC(=O)CC2CCC2)oc1C(=O)NOCCOC(C)C C=CC(C)(C)CC(=O)N1CCC(C)(CC(N2CCCC(F)(CO)C2)=O)C1 C(CC(C)CCNC(=O)C(O)c1ccsc1)NC(Cc1nc(C)[nH]n1)=O N1(C(C2CCN(C(C)=O)CC2)=O)CCC2(CC1)CCN(C(c1sncc1C)=O)C2 C=CC(CC)CC(=O)N1CC(CNC(c2cc(Cl)n[nH]2)=O)C(F)(F)C1 C1(C(=O)NCCC(C)NC(c2ccc(OCC)c(C)c2)=O)CN2CCN1C(C)C2 c1(C(=O)NCCC2(C)CCN(C(CC(=C=C)C)=O)C2)c(C)cccc1N C(=O)(C(=O)N=c1ccn(CC(F)F)[nH]1)NCc1ccccc1OCCOC S(=O)(=O)(c1ccc(Cl)c(N2CCOCC2)c1)NCC1C(c2cn(C)nc2)C1 C#CC1(NC(=O)COc2cncc(Cl)n2)CCN(OC(F)(F)F)C1 c1(CC(N2CCC(F)(CNC(=O)OC(C)(C)C)C2)=O)nc2ccccc2[nH]1 CCC(CCC(=O)NCCN1C(=O)CNC1=O)NC(c1cncc(Cl)c1)=O c1(C(=O)NCCN(C(=O)C(O)CN(C)C)CC)cc(C(C)C)ncc1Br C1(C(=O)N(CCCN(C)C(C2CN(C(C)C)C2)=O)C)CCCN1C1CCC1 c1(OC)ncc(F)cc1C(N1CCC(c2ccc(Br)cc2)(C(=O)O)C1)=O C#CCCCCC(=O)NCc1ccc(CCNC(=O)CC2CCC(C#N)C2)cc1 N1(C(COC(C)(C)C)=O)CCCC(CC(=O)NCC2CC(CF)C2)CC1 C#CCC(C)(C(=O)NCC1COC(=O)N1)NC(C1CCOC1)=O c1(OC)ccc(C)c(C(=O)NCC2C(C)CCN2C(=O)Cc2cccc(Cl)c2)c1 c1(C(=O)Nc2c(SC)cccc2)cc(C2=CCC(C)(C)CC2)c2[nH]ccc2c1 C=CC(F)(F)C(=O)NC1CCCN(C(=O)COCc2cccc(C)c2)C1 N1(C(c2cn(CC)nn2)=O)CCC2CN(C(=O)C(=CC3CCCC3)C)CCC2C1 c1(C(N2CCCC2)=O)ccc(F)cn1.C12CCCN(C1)CC(=O)NC2C N1(C(C(OC)OC)=O)CCC2(CC1)CC2(CNC(=O)C(C(F)(F)F)C(F)(F)F)CO c1(C(N2CCC(CC)C2C(=O)NC(C2CCOC2)CO)=O)cc(O)cc(F)c1 C(=O)(C1CCCn2ncnc21)OCCOCCN(C(C)=O)CC CC1(C)OCC2CC12C(=O)NCC1(O)CCCN(C(=O)CCN2CCCC2)C1 C1(C2CN(C(=O)CC3(c4cc[nH]n4)CC3)C2)(NC(C(c2cccnc2)C)=O)CC1 N1(C(CC(=O)OC)=O)CCN(C(c2cncc(SC)c2)=O)CC1C c1(C(=O)NC2C(NC(C3C(COC)CCC3)=O)CCC2)ccnc2c1ncn2C c1(C(=O)NC2CN(C(C3(OCC)CCOC3)=O)CC2C)ccc(OCC)nc1 C1(CNC(c2cc(SC)oc2)=O)COC(C)(C)CN1C(=O)CC1CCCN1C N1(CCC)CC(C(N2CCN(C3CCN(C(=O)C(C)CC)C3)CC2)=O)CC1=O C12(C(=O)NCCOCCC(C)C)C(NC(=O)CCS(N)(=O)=O)C3CC1C2C3 N1(C(CC(C)C(C)(C)C)=O)CCC2(CC1)CC(NC(=O)CCC1OCCO1)C2 n1(CCC)cc(C(=O)NCC(C)(C2CC2)NC(=O)CC2CC(CC)C2)nn1 C12(C(=O)NC(CCCC)CNC(c3sccc3CC)=O)CC(C)(C1)OC2(C)C c1(C(=O)NCCOCCN(C(=O)CC2CCC(=O)O2)C)cnn2c1NCCC2 CCCCC(C)(F)C(=O)N1CCC(N(C)C(C2CCCN2C=O)=O)CC1 N1(C(=O)Oc2nc(C)c(C)s2)CCC(NC(c2c(Br)cnn2C)=O)CCC1=O N1(CC(=O)Nc2ccccn2)CCC(CO)C1.CC1CNC(=O)CO1 C(=O)(C1CCCc2ccccc21)NC1CC(NC(c2cc(C#N)oc2)=O)C1 CCC(CC(=O)NCC1(NC(=O)Cc2ccn(C(F)F)n2)CC1)CC(F)(F)F N#CC1CCCC(C(N2CCC(O)(c3ccc(Br)cc3)C2)=O)CC1 n1(CCC(=O)NCCCN(C)C(C2CC=CC2)=O)cnc2sccc2c1=O CC1CN(C(=O)Cc2cncnc2)CCC1NC(C1C2(CC2)C12CC2)=O C1(CC(=O)NC2CC(=C)C2)CCN(C(=O)CNC(N)=O)C1(C)C C(=O)(CCCN1CCCC1)NCC(CC)NC(c1ncsc1C)=O C1(O)(CNC(c2n(C=C)ncc2)=O)CCCN(C(c2sccc2CN(C)C)=O)C1 Cc1ccccc1C(=O)NCC(O)CNC(c1ocnc1C)=O C1(CNC(=O)C2=CCC2)C2CCC(C2)N1C(=O)Cc1cccnc1O N1(C(CCNC(C#CC(C)(C)C)=O)=O)CCC2CCC(C1)N2C CC1CC(C(=O)N(C)CC2C(C)(C)C2(C)C)N(C(C2CCOCC2)=O)C1 N1(C(CN(C)CC)=O)C2CCC1CC(NC(C1(C)CC(C3CC3)=NO1)=O)C2 N1(C(C2(CF)CC(=C)C2)=O)CCOC2(CCCN(C(C3(C)CCSCC3)=O)C2)C1 c1(C(=O)NCCN(C(=O)Cc2cccc(Br)c2)CC)c(C)cc[nH]c1=N Cc1cc(C(N2CCC(C)(C(=O)NC3CC3CN(C)C)C2)=O)cnn1 N1(C(c2nc(C)oc2)=O)CCC2C(NC(c3cc(C(C)(C)C)oc3C)=O)C2CC1 N1(C(CCNC(C)=O)=O)CCC2(CCCC2C(=O)Nc2cnc(Cl)nc2)C1 C1(NC(CCc2onc(CC)n2)=O)CCCCC1CNC(c1c(Cl)n[nH]c1C)=O c1(CC)ccc(C(=O)NC(CCN(C)C(C2(F)CCOC2)=O)C(C)(C)C)c(C)n1 CCC(O)C(F)(F)C(=O)NC1CC2(C1)CC(C(=O)NCc1cc(=N)[nH]c(Cl)n1)C2 N1(C(C=CC)=O)CC2CN(C(c3ccc(C(F)(F)F)c(O)c3)=O)CC12 c1(C(=O)NCCC2CN(C(C3C(CCC)C3)=O)C2)ccc(C)n1C.C(C=C)=CCC N1(C(C23CC(C(=O)OC)(C2)C3)=O)CCC2(CC(NC(c3cc(C)n(C)n3)=O)CO2)C1 C1(Nc2nc(OC)cc(OC)n2)CCCCCN(C(C2CC(=O)NC2(C)C)=O)C1 C1(CC#C)(C(=O)NC(CNC(=O)CCn2cnnn2)C2CCC2)CCCCO1 C(CC#CC)(C(=O)Nc1conc1C)NC(c1n(CC#C)cnn1)=O C1(CCC)CN(C(C2CC(=C(F)F)C2)=O)CCN1C(C1CCN(C)C(=O)C1)=O N1(C(CC)CC)CC(C(=O)NCC=CCNC(C2OCCOC2C)=O)CC1=O C1(CN(C(CSCCN(C)C)=O)C)CCN(C(c2scnc2C(C)(C)C)=O)CC1 c1(C(N(CCNC(C2(COCC)CC2)=O)CCOCCO)=O)ncccc1N=[N+]=[N-].CS c1(C(=O)NCC2(C)CCN(C(C(CC#C)O)=O)C2)cc(S(N)(=O)=O)c(C)s1 C#CCC(O)C(=O)N1CCCC(N(C(=O)CCN2CCCCCC2)C)C1 C1(C(=O)NCc2nc(COC)sn2)CC2(CCC2)CN1C(=O)OC(C)(C)C C#Cc1ccc(C(=O)NC2CN(C(=O)C(O)C(F)F)CC2F)c(OC)c1 n1(C(C)C)nncc1C(N1CC(CNC(C2CCC(C(F)(F)F)O2)=O)C1)=O C(=O)(C1=COCCC1)N(CC(C)N(C)C(c1cc(Br)cc(Cl)c1)=O)C C12(CNC(CCCC3C(C)C3)=O)CC1CN(C(c1cnn(CC(F)(F)F)c1)=O)C2 c1(C(=O)NCCC(C)N(C(C2(CCCC)CC2)=O)C)cnn(CC)c1CC Cc1ncc(Br)c(C(N2CC=CC(NC(c3ccc(F)cc3F)=O)C2)=O)n1 c1(NCCCC2N(C(CCSCC)=O)CCC2)cc(C)c(C)o1 Cc1ccc(C)c(C(=O)NCC2(O)CCN(C(=O)NC(C)C)C2)c1 N1(C(=O)CC2CCCO2)CCCC1CCC1CCCN1C(c1cscn1)=O C1(C(=O)NCC(COC)(F)F)C(C)CCN1C(c1ccc(C#N)[nH]1)=O N(C1COc2c1ccc(Cl)c2Cl)CC(c1ccc(Br)cc1)C.C(CO)O c1(C(N2C(CC34CC(C3)C(=O)N4CC)CCC2)=O)cccnc1O.N(C)C S(=O)(=O)(C(C)CN=c1[nH]c(=NCc2cccn2C)[nH]c2c1CSC2)NC C1(C(=O)NCCCCCn2cc(C(C3CCCOC3)C)nn2)CCCCN1N=O C1(O)(CCNC(c2csc(Cl)c2)=O)CCN(C(C2CC(C(F)F)C2)=O)C1 c1(C(N2C(CNC(C(CCC)OC)=O)CC2)=O)n[nH]c2c1CCSC2 c1(OC)ccc(CCC(=O)NCC(C)(C)CNC(c2cncnc2C)=O)cc1F c1(C(=O)NC(C)CN(C(=O)C=CCCc2ccccc2)C)ccn(C)c(=O)c1O CCCCCS(=O)(=O)CC(=O)NCc1cn(C2CN(C3CN(C)CCO3)C2)nn1 c1(C(=O)NCC(C2CC2)SC)coc2c1CN(C(=O)C(C)(C)N=[N+]=[N-])C2 C1(C(N2CCC(CCN(C(C(OC)OCC)=O)C)CC2)=O)CCCC12CCC2 N1(C(=O)Cn2cnnc2O)CC2(CNC(C3CC34CC(F)(F)C4)=O)CC1CO2 C1(NC(C2(COC)CCC2)=O)(NC(=O)C(=O)NC2CC2)CC(O)C1 C1(CNC(c2cccnc2)=O)CCCCN(C(c2cc(Cl)c(Cl)s2)=O)C1 c1(C(N(CC(C)NC(=O)C(C)CSC)CC)=O)cccc(F)c1OC C1(CNC(=O)CC2CS(=O)(=O)C2)C2CN(C(c3ccnc(C4CC4)n3)=O)CC12 Cc1ccc2cc(C(=O)NC3CCCCN(C(=O)CC(C)F)C3)ccc2c1 N1(C(CCN(C(CCCC(CC)C)=O)CC2CC2)=O)CCc2nnnn2CC1 CCCCS(=O)(=O)NC1C2CN(C(c3scnc3C(F)(F)F)=O)CC12 N1(C(c2c(OC)ccc(O)c2)=O)CCN(C(=O)C(C)=C(C)C2CC2)CC(C)(F)C1 c1(OC(C)C)cc(C(=O)NCCCCNC(C2COC(C3CC3)C2)=O)ccn1 C1(O)(C(N2CCC(C(C(=O)NC3CC(OCC)C3)C)CC2)=O)CCOC1(C)C N1(C(CNC(=O)NC2CC2)=O)CC2CN(C(c3cnsc3C)=O)CC2(C)C1 CC1CN(C(=O)CCN(C2CCCCC2)C)CCC1CNC(=O)Cn1cnnc1 C(=O)(CCC(C)CN(C)C)NC1CC(CCC(=O)NC(C(=O)OC)C2CC2)C1 C(CC(=O)N1CC2(CNC(=O)CC3CCC3C)CCC1CC2)(C(F)(F)F)OC N1(C(C2CN(C(N(C)C)=O)C2)=O)CC=CC(NC(c2ccc(C3CCC3)cc2)=O)C1 CN1CCc2cc(C(=O)NCC3CN(C(=O)Cn4cnnc4O)CCO3)ccc21 N1(C(C(CC)CC)=O)C2CCC1CC(NC(=O)C(O)Cn1cncn1)C2 CC(N=c1nc(N(CCCF)C)c2c([nH]1)CCS2)c1cn[nH]c1 C(=O)(C1CCCc2nc[nH]c21)NC1CN(C(C(CC)(F)F)=O)CC1C C1(C(=O)NC2C(CNC(CCCC#C)=O)CC2)CC2(C1)CC(F)(F)C2 c1(C(=O)OC)nc(CC2(NC(=O)C(=O)NC(C)CC)CC2)c(Br)s1 N1(C(COCC)=O)CC2(CCCCC2)CCC1Nc1ccc(OC)cc1 C1(NC(C2CCN(C(=O)NC)CC2)=O)CCC2CC1CN2C(=O)COCCCF C12(C(N(CCCCC(=O)NC(CCOC)C)C)=O)CCC(C1)OC2C C1(CNC(C(C2CCCC2)OCC)=O)(NC(C2CCCO2)=O)CCCCC1 O=C(C1=CC2CCCCC12)NC1CC(CCNC(=O)C(O)CC2CC2)C1 Cc1ccnc(O)c1C(N1CC2CC(NC(=O)CC3CCS(=O)(=O)C3)C2C1)=O C1(NC(c2nc(OC)oc2)=O)CCCCN(CC2CC23CCOC3)C1 c1(CC(N2C(CNC(C(C)(C)N=[N+]=[N-])=O)CC3CC32)=O)nc2ncccn2n1 Cc1cc(CO)oc1C(=O)NCC1(O)CN(C(=O)CCC2CCCC(=O)N2)C1 C1(C(N(CC(C)(C)C(=O)NC2CC3CCCC3C2)C)=O)Cc2ccccc2C1 c1(N(CC)CC)nnc(-c2ccccc2F)n1CCCSC1CCSC1(C)C c1(C(=O)NCC2(NC(C(C)=C(CC)C)=O)CC2)c[nH]c2cc(F)c(F)cc2c1=O Cc1nc(C)n(O)c1C(=O)N(C)CC1CCCN1C(=O)Cc1cccc(F)c1 CON(C)S(=O)(=O)c1ccc(C(N2CCN(C(c3sccc3N)=O)CC2)=O)cc1 c1(OC)ccc2[nH]cc(C(=O)NC3CCC3NC(c3ccn(C(C)C)n3)=O)c2c1 N1(C(C(C)n2cccn2)=O)CCCC(NC(=O)CSCc2ccc(F)cc2)CC1 c1(NCC2CCN(CCOC)C2)nccc(=NCc2cc(F)cnc2Cl)[nH]1 N1(C(=O)NC(c2ccc(C)nc2)C2CC2)CCCC(C)C1CO N1(C(CC2CCN(C(c3ccc(OC)s3)=O)C2)=O)CCSCC1C(N)=O C1(C(=O)NC(C2CCC(C(=O)NCCF)O2)C)CCNC(=O)C1 C(CCC(CCC)NC(=O)CSCCCC)NC(CCC(=C)Cl)=O C1(N(C(c2cc(COC)no2)=O)C)CCN(C(=O)C=C=C(C)C)CC1 N1(C(COCCOC)=O)CCOCC(NC(C2(c3cc(C)cc(C)c3)CCC2)=O)C1 C1(C(=O)NCC2(CN(C(=O)Cc3cnn(C)c3)C)CC2)CCN2CCCCC2C1 C1(CNC(c2csc(C(F)F)n2)=O)CCCN1c1nc(C2CC2)ns1 C1(CC)CC(CC(=O)NC2CCN(c3nc(SC)ns3)C2)CCO1 N1(C(CC2N(CC)CCOC2)=O)CC2CCC(C1)N2C(=O)C(O)CN(C)C C#Cc1cccc(C(=O)NCC23CC(NC(C4CC4(F)F)=O)(C2)C3)c1Cl C(=O)(C1=CCN(C(c2ccc(C)c(C)c2)=O)CC1)NC(C1CCOC1)C#C Cc1cc(C(=O)NC2CC(C(=O)NC(CO)CCO)C2(C)C)n(C)n1 C(CS(=O)(=O)CC(=O)NCC(C)C(F)C(=O)N1CCOC(CF)C1)OC C(=O)(C1CCCc2ncnn21)NCC(CO)NC(c1c(SC)cccn1)=O C1(C(N2CC3CN(C(C=CC=CC)=O)C3C2)=O)CCc2ccccc2C1O c1(OC)ccccc1S(=O)(=O)NC1CCCN(C(c2ccc(O)cc2Cl)=O)C1 N1(CC(=O)N(CC=CC(=O)NC2CCC(OC)C2)C)CCC(C)CC1 C(=O)(C(C(C)C)N(C)C)N1C(CNC(CC2(CSC)CC2)=O)CCC1 C12(C(N3CC(NC(C4(CC)CCCCC4)=O)C(C)C3)=O)CCC(F)(CC1)CC2 c1(C2CCC(C(C)C)CC2)nc(C2=NOCC2)no1 CC1(C)CC2(CC(C(N3CCN(C(C45CC6CC4C5C6)=O)CC(O)C3)=O)C2)C1 C12(C(=O)NC(C)CN(CC(F)(F)F)C(=O)C=CC=CC=CC=N)CCOC1CCOC2 CC(C(=O)NCc1csc(C(=O)NC(C(N)=O)C(C)(C)C)c1)S(N)(=O)=O c1(CCC(=O)NC2C(C)N(C(c3sccc3F)=O)CC2)ccc(Cl)c(F)c1 C1(CNC(c2nc(C)oc2)=O)CC12CCN(C(=O)C(F)CC(C)(C)C)CC2 C(=O)(CCCCCF)N1CC(NC(CCC(C)C)=O)C(C(F)(F)F)CC1 c1(OC)ccc(Cl)cc1CC(=O)N(C)CC1CN(C(=O)C(C)CSC)CCO1 Cc1c(O)ccc(C(N2CCC(CNC(=O)C3=NOCC3)C2(C)C)=O)c1C N1(C2(CNc3nc(C)oc3)CC3(CSC3)C2)c2ccccc2Sc2ccccc21 c1(OC)cc2c(c(S(=O)(=O)N3CCC(c4cccc(C)c4)C3)c1)OCC2 c1(-c2cn(C(=O)O)nn2)cnccc1NC(c1coc(-c2ccc(Cl)cc2)n1)=O c1(C(N(C)CC2N(C(Cc3c(C)nc[nH]3)=O)CCCC2)=O)ccc(Br)cc1C#N CC(C)(C)CC(C(=O)NCC1CC1)N(CCC(N1CCOCC1=O)O)C c1(CC)c(C(=O)NCC2CCCC(NC(c3cc(C)on3)=O)C2)nnn1CC N1(CC)N=C(C(=O)N2CC(OC)C(NC(=O)C(C)CO)C2)CCC1=O CN1CCN(CC(C)(C)C(=O)N(C2CCC3CC23)C)CC1.C(=O)(CSC)OC C1(NC(C=CC(C)C)=O)CCCN(C(=O)Cc2cccc(Cl)c2F)CC1F c1(NCC(N2CC3C(NC(=O)C(C4CCCOC4)O)(C3)C2)=O)cc(Cl)cc(Cl)c1 Cc1cc(C(=O)NC2(CCNC(C3(F)CC3C)=O)CCC2)nn1C CC1(C)CC(C(=O)NCCCCCC2CC2)CN(C(=O)C=CC2CCCC2)C1 Cn1cc(C(=O)NC2CN(C(c3ccc(-c4cccs4)[nH]3)=O)C2)c(C(C)(C)C)n1 c1(OC(C)C)ccc(NC(c2cc(CNC(=O)COCCF)on2)=O)cn1 C1(CNC(CC2CCN(C)C2=O)=O)Cc2ccccc2CN1C(=O)Cn1cnnn1 CCC(CCCC(=O)N1CCS(=O)C(C)C1)NC(C1CCN(C)C(=O)C1)=O Cc1cccc(C(=O)NC(C)CC2CCN(C(c3c(C)ccn3C)=O)CC2)c1 N1(C(CCC=C=C)=O)CC(C)(C(=O)NCc2cscc2C)CC1(C)C N1(C(C2N(C(C(C)N(C(C)=O)C)=O)CCCCCC2)=O)CCC2(C=CCO2)CC1 c1(C(N2C(C)CC(NC(C3(COCC)CC3)=O)C2)=O)cncc(Br)c1C N1(S(=O)(=O)c2cccnc2NC2(CC3CC3)CC2)CCCC2(CCCCO2)CC1 N1(C(C(C)NC(CC)=O)=O)CCCC(C2CCCN(C(c3cccs3)=O)C2)C1 c1(NC(CSCC#C)=O)ccc(Cl)c(NC(=O)CCOC2CC2OC)c1N C1(C(=O)NCCn2c(C)nnn2)CC2CC1CC2NC(=O)OC(C)(C)C N#Cc1cc(F)ccc1CC(=O)NCC1(O)CN(C(c2cc(C3CC3)on2)=O)C1 Cc1n[nH]c2cnc(C(=O)NC3CN(C(=O)CSC(F)F)C4CC34)cc12 C1(N(C(=O)CCn2cnnn2)CC)CCN(C(=O)CN2CCOCC2)C1 C(C(=O)Nc1cn(C)nc1Br)(C(C)C)NC(CCc1onc(C)n1)=O C(=O)(CCC(=O)N1CC(NC(C2CN(C)C(=O)N2)=O)CC1CO)OC c1(C(N(CCCNC(=O)C(c2cncn2C)OC)CC)=O)nc(=N)cc[nH]1 C1(C(C)C)CN(C(=O)Cc2nccn2C)CCC1NC(=O)C(C)SC(F)(F)F C1(C2CCCN(C(=O)CCN3CCOC3=O)C2)(NC(=O)C#CC2CCCO2)CC1 C1(CNC(=O)Cc2ccco2)C2CN(C(=O)CCCF)CC12 N1(C(C2OCCC(C)C2)=O)CC2CCCC(C1)N2C(=O)CCCc1ccccc1 CCC(F)(F)C(=O)N1CCCC1CN(C)C(C1CCCCC1CC)=O C(=O)(C(C)(C)C(=O)NC1CCCC1CN(C)C(c1cnc(NC(C)=O)o1)=O)NC c1(C2(C(=O)NCC(CC)NC(C3(C)COC3)=O)CCCC2)c(F)cccc1F C1(C)(CC)CCN(Cc2nc[nH]c2C(F)(F)F)C1 O=C1OC(C(=O)N(C2CCCC2)CC2CC2)Cc2ccc(F)cc21 c1(CC)cc(C(N2CCC(CN(C)C(c3nccnc3Cl)=O)CC2)=O)c(C)nn1 C(CCC(C(=O)NCCc1cccc(O)c1)NC(=O)Cn1nc(C)oc1=O)OC C(CC(C(=O)NC(C)Cc1cnn(C)c1)NC(c1ncsc1C)=O)=CC c1(C(=O)NC(C2OCCN(C(C=C(CCC)C)=O)C2)C)ccc(Cl)c(C(=O)OC)c1 N1(C(CNC(=O)NC)=O)CCC(C2CCCN(C(C3CC4(C3)CC4F)=O)C2)C1 N#Cc1ccc(=NC2CCCCN(C(c3cnc(Cl)c(Cl)c3)=O)C2)[nH]n1 CC1(C)C(C(=O)NCC2CC(NC(C3(CO)CC3)=O)C2)CCS1(=O)=O C(=O)(C1=NOC2COCC12)N.c1(C(=O)NCO)cc2n(n1)CCO2.C12CCN(C1)C2=O c1(C(=O)NC2C(C)CN(C(c3cn(C)cn3)=O)C2)cc2[nH]ccc2s1 N1(CC(=O)NC(C(=O)NC(C)C(=O)NO)(C)C)C(=O)CNC1=O c1(C(=O)NC2CC3(C(NC(c4c(C)ccs4)=O)C3)C2)ccc(O)c(F)c1 c1(C(N2CC(C(C)NC(c3cncc(F)c3)=O)C2)=O)cc(N(C)C)ccc1F O=S(=O)(c1ccc(NCCC2CCCC(CO)C2)nc1)Nc1c(F)ccc(Cl)c1F C(=O)(C(C)C(C)S(C)(=O)=O)N1CCOCC(NC(C2(C)C(C)CCC2)=O)C1 CC(F)(F)C(C)(C)C(=O)NC1(C2CN(C(=O)CSC3CCOC3=O)C2)CC1 C(CCN=C(NCC1CCC1)N1CCC(C2CC2)CC1)N1C(C)CCC1 c1(C(=O)OC)cc(C(=O)NCC(c2ccncc2)NC(c2cccs2)=O)c[nH]1 C(=O)(C1=NOC2(CCC2)C1)NC1C(NC(C(C(C)(C)C)C2CCC2)=O)CCC1 C(CC1=CCN(C(=O)CN(C2CCCC2)C)CC1)NC(C(C)OCC)=O c1(CC)sc(C(=O)NCCN(C(=O)CC2OCCCO2)C(C)C)cc1Br C1(c2c([N+](=O)[O-])ccc(F)c2)CCCCN(N2CCCCC2Cc2cccnc2)C1 CC12CCCCC1CN2C(C1CN(C(C2CC2Cl)=O)CC12CC2)=O CCC(CCC(=O)N(CC(C1CCC1)OC)C)NC(c1nccs1)=O C(CCCN=[N+]=[N-])NC(C1CC(CCNC(C(C)(C)c2ccno2)=O)C1)=O c1(-c2n(C)ccc2)ccc(C(N2CC3CC2C3CNC(c2ccc[nH]2)=O)=O)cc1 CCC(C(=O)NCC1CC1NC(=O)C(N1CCOCC1)C1CCC1)OC c1(C(N2C(C(C)(C)CC(N3CC(C)(O)C3)=O)CCC2)=O)cc(O)nc(O)n1 N1(C(CC2CCC(C)O2)=O)CC2CC2(CNC(=O)CC(C)(C)C)C1 C1(C)(CNC(C2C(C)CCCC2)=O)CCN(C(c2cncn2C(F)(F)F)=O)CC1 N1(C(C(Cc2ccco2)NC(CC(CN(C)C)O)=O)=O)CCCCC(CO)C1 N1(C(C2ON=C(C)C2C)=O)CCC2CN(C(c3ccc4sncc4c3)=O)CC2C1 C1(=O)CC(C)CO1.C1(CC(=O)OCC)OCCC1C(F)(F)F c1(C(=O)NC(C(=O)N(CC(C2CCC2)OC)C)C2CCC2)ccnnc1C C(=O)(C(C)(C)C1=CCN(C(C2CC(F)CN2C)=O)C1)NCC(C(=O)NC)O c1(CCC(=O)NC2CCN(C(c3coc(Br)c3)=O)C2)ccsc1Br C(=O)(C(CNC(=O)CSC)CC1CCCC1)NCCN(CC)CC Cc1cccc2sc(N3CCC(CF)(NC(C4CCC5CC5C4)=O)C3)nc12 C1(F)(CNC(CN(C)CC)=O)COCCN(C(=O)CC(O)CC(C)C)C1 C(=O)(CC1=CCN(C(C2CC3CCC2O3)=O)CC1)NC1CCCN(C(CC)=O)C1 N1(C(c2ccc(NC(c3nnc4ccccn34)=O)cc2)=O)CCC2(CCOC2)C1 N1(C(CONCc2n(C)ncc2)=O)CCCC(C(F)(F)F)C1 N1(C(c2onc(CC)n2)=O)CC2CC(NC(C3CCCS3)=O)C2C1 Cc1c[nH]c(C(=O)NCCC(C)NC(c2cn[nH]c2)=O)c1C CCC(C)C(O)CC(=O)N1CC(C(N2CC(F)(F)CCC2C)=O)(SC)C1 N(C(=S)SC(Cc1ccccc1)C(=O)OC)(CCC#C)CCC#N c1(C(C)C)ccc(C(=O)NCCCN(C(=O)CC2CCCOC2)C2CC2)cn1 Cc1nn(C)c(C)c1OCC(=O)NC(C1CCN(C(=O)CCn2ccnn2)C1)C C(N=c1[nH]c(N2CC3CC2CN3CCC)nc2c1SCC2)c1cnn(C)c1Br C1(=O)C(C)(C)C(=O)NCCNC(=O)C(CO)CNC1=O.C(C)(C)(C)O.CN CS(=O)(=O)C1(C(N2CC(NC(=O)CCc3ccsc3)C(O)C2)=O)CCC1 c1(C(=O)NCCCNC(COC)C(C)C)cc(C)c(OC)cc1C C(=O)(CC(C)(C)CNC(c1cncn(C)c1=O)=O)NC(C=C)C1CC1 C(=O)(CCCCCCCC1CC1)N1C(C)C(NC(=O)Cc2ccsc2Cl)CCC1 CCCCC(O)C(C)C(=O)NCC1N(C(c2cc(OC)cnn2)=O)CCC1(C)C C1(C(N2CCC(NC(CC3CC(OCC)C3)=O)(CF)C2)=O)CCn2ncnc2C1 c1(C(N2C(CCC(=O)NCC(COC)(C)CO)CCCC2)=O)cnc(O)cc1C N1(C(c2nc(C(C)=O)sc2)=O)CC2CCC2(NC(C2Cc3nccn3C2)=O)C1 c1(C(=O)NCC2CCCN(C(C3(F)CCC3)=O)C2)ccc2nc(Br)nn2c1 c1(C(N2CCC(F)(C(N(C3CCCOC3)CC)=O)C2)=O)c(O)cccc1F N1(C(c2cnc(CC)[nH]2)=O)CC(CO)C2(CCN(c3nnc(CC)s3)CC2)C1 c1(NC2CCN(C(C(C)N(C(C)=O)C)=O)C2)ncnc2[nH]c(C)c(C)c12 C1(CNC(C2C(CCOC)C2)=O)CN(C(C2CC(C#N)C2)=O)CC1(F)CO c1(CCC)cc(N(c2ccnc(C)n2)C(=O)Cc2ccc(Br)cc2I)nc(Cl)c1 Nc1cc(F)cc(C(N2CCCC(CO)(NC(c3coc(Cl)c3)=O)C2)=O)c1N CCC(C(=O)NCCn1cc(CNC(C2CN(C3CCC3)C2)=O)nn1)C(C)O c1(C(N2CCC(C)(CC)CC2)=O)cc2cnccc2nc1C C(=O)(CC(C)(C)CNC(C1(F)CCCCCC1)=O)NC1CCCC(CC#N)C1 C(C(C)(C)CCNC(c1cnc(C2CCC2)o1)=O)NC(c1c(C(C)=O)csc1)=O C1(CC)CN(C(=O)C(F)(F)C(F)F)CCC1NC(=O)Cc1nc(C)c(C)s1 CN1CCC(CCNC(C2C3CC4C(C3)C24)=O)C1=O C(C1CN(C(C2CCCC(=O)N2)=O)CC1C(=O)NCC(C)NC(C)(C)C)=CC C(CCCC(=O)NCC1CCC1NC(c1cncn1C1CC1)=O)SC C#CCC(CC#C)C(=O)N1CC(CCCCNC(C2CC2(Cl)Cl)=O)C1 c1(NCC)nc(C)ccc1C.C12(C(=O)NCCCC=CC)CCN(C1)C(=O)C2.CC=C C(=O)(C(O)CN(C)C)NC(C)CCNC(=O)C=CCOCC(F)(F)F N1(C(C2C(OC)C2)=O)CC(CNC(=O)Cc2cc(F)ccc2C)OC(C)(C)C1 C1(C(=O)NCC2(O)CCCN(C(C3CN(C)C3)=O)CC2)Cc2ccccc2CO1 c1(CC)cccc(C(=O)NCCCC(CO)NC(C2CCC(N(C)C)C2)=O)n1 c1(C(N2CCOC(CNC(N)=O)C2)C(=O)NCC(=C)C)cccc(Cl)n1 Cc1c(C(=O)N(C)CCN(c2ccon2)C)c[nH]c2nccc1-2 C1(C(=O)OC)CCCC(C(=O)NCC(C)CNC(=O)C(C)Cc2cccnc2)C1 N1(C(=O)CC2CCC(O)C2)CCC2(CCCN2C(=O)CCOC2CC2)C1 C(c1c(C)noc1C)=CC(=O)NCCCN(C(C1(O)CCCC1)=O)CC c1(C(=O)NC(C(C)NC(C2C(C=C)C2)=O)(C)C)cc(Cl)c(Cl)cc1C C=CC1(C(=O)N(CC(C)(C)C#N)C)CCN(C(c2cc[nH]c2C)=O)C1 Cc1[nH]nc2c(C(=O)NC(C)CCCCNC(=O)CC(C)C(F)(F)F)cccc12 Cc1cc(C(=O)NCC2CCCCN2C(c2ncoc2CN)=O)c(C(F)(F)F)o1 CN(C)NC(=O)CCC(=O)NC1CCCC1NC(c1cc(C#N)cs1)=O Cc1cc(F)c(C(N2CCC(F)(Cc3nn[nH]n3)C2)=O)cc1F CS(=O)(=O)c1ccc(NCC2(O)CCCN(C(C3C4CCC3CC4)=O)C2)nc1 N1(C(CSCC)=O)CC(NC(=O)CCCc2sccc2C)CC(O)C1 C=CCC1C(=O)N2CCC(CC)(C2)C(=O)N1CC.c1(NC)cnccc1N(C)C N1(C(C2(C#C)CCC2)=O)CC2CCC(CNC(C3CC3(C)C(F)F)=O)C2C1 C1(C(=O)NC2C3CN(C(CCCCC)=O)CC32)CCc2nnc(O)n2C1 C1(C(N2CCCC(CCCCNC(C(C=CC)O)=O)C2)=O)CNc2ccnn2C1 C1(CC(=O)NCC(C)N(C(=O)C(C)(C)C#N)C)CCC(F)(F)CC1 Cc1cc[nH]c1C(=O)NCCOCCCN(C(=O)C(C)C1CCCO1)C Cn1cnn(CC(=O)NCC(O)CCNC(C2C=CCC2)=O)c1=O c1(C(N(CC(C)N(C)C(c2ccnc(S)c2)=O)C)=O)csc([N+](=O)[O-])c1 CCC(CNC(=O)C(=CCOC)C1CC1)(CC)NC(=O)COCC1CCCC1 CCCCC(C)CCC(=O)NCC(C)NC(c1cc(C)nn1C(CC)CC)=O c1(CC(N2CC(NC(CC(=O)NCC)=O)C(C)(C)C2)=O)c[nH]c2cc(F)ccc12 C1(NC(C2CC(OCC)C2)=O)(CF)CCN(C(c2cnn(C(C)C)c2C)=O)C1 c1(CC(=O)NC2(C)CCCN(C(C3CC(SC)C3)=O)C2)ccc2c(c1)CCC2 C(CN=c1[nH]ccc(=NCC(Cl)(Cl)Cl)[nH]1)C1CCCC(C)C1 N1(C(C(C)SC(C)C)=O)CCC1(C)CC(=O)NC1(C(O)CO)CC1 N1(c2c(C)ccc(C)n2)CCC(NC(c2snnc2C(C)C)=O)CC(C)(C)C1 CC(CC(F)(F)F)C(=O)NC1CCCCN(C(C2(C#N)CC2C(F)(F)F)=O)C1 C1(NC(C(CSC)OC)=O)CC2(C1)CC2C(=O)NCCC1CCCC1(C)C C1(CN(C(c2nc(C)sc2)=O)C)C2CN(C(c3cccc(OC(F)F)c3)=O)CC12 c1(OC)ccccc1N1CCC(NC(=O)CNCC2(C)CC2(F)F)C1 N1(C(C)=O)CCCCC1C(N1CCCCC1CN(C)C(C1(C)CCCC1)=O)=O N1(C(Cc2cn(C)nc2)=O)CC(NC(C2(CC(F)F)CCC2)=O)CC(O)C1 c1(C(=O)NC2CC(CC(=O)OC)C2)cnn(CCNC(C2(C)CCOC2)=O)c1 N1(C(CC(COC)C)=O)CCN(C(=O)Cc2ccsc2C)CCC1C N1(C(Cc2cc(C)[nH]n2)=O)CCC(C(=O)NCCc2c(C)noc2C)CC1C c1(C(=O)NCCCNC(=O)CCNC(C2CCC2)=O)c[nH]nc1Br c1(C(=O)NCCN(C(C2C3C4CCC(C4)C23)=O)CC)cc2cnccc2[nH]1 CC1CC(N(C(C2(C(=O)N(C)C)CC2)=O)CCC)CN(C(C2CCC(=O)N2C)=O)C1 C12(C(=O)NCC=CCNC(C3C=CC(OCC)C3)=O)CCCC(C)(C1)OC2 C1(C(=O)NCC(CC=C)NC(=O)CCCCn2ccnn2)CC2CCC(C1)C2 C1(CNC(C(C)OCOC)=O)CCCCN(C(C2C3CCCCCC23)=O)C1 c1(NC(=O)Cn2cc(CNC(=O)CCCCCF)nn2)cccc2cc(O)ccc12 CC1(C(=O)NCCC2CCC(F)(F)CC2)CCCN(Cc2ccc(F)nc2)C1 C(=O)(C(C)(F)C(C)(C)F)N1C(C(=O)NC(c2ccccc2F)C(C)C)COCC1 CC1CCCc2c(C(N3CCC(Cc4ccccc4F)CC3)=O)cnn21 c1(C(N2CCS(=NN)CC2)C(=O)NCC2(COC)CC2)sc2ccccc2c1Br C(=O)(C(CCS(C)=O)N(C)C)N1CCC(CNC(C=Cc2ncc(C)[nH]2)=O)C1 c1(NC(C(=O)N(CC(c2ccc(F)cc2)O)C)=O)cccc2nsnc12 C1(CC)CN(C(C2C=CCC2)=O)CCN1C(c1ccc(C(=O)OC(C)(C)C)o1)=O c1(CN2C(C)(C(N3CCC(Br)C3)=O)CC2)c(F)cc(Cl)cc1Br c1(CC(=O)NC2CCCCO2)ccc(Cl)s1.n12cc(nn1)C(N1CCOCC1)CN1CC2C1 CS(=O)(=O)c1ccc(NC(C2CC(n3cc(C(N4CCCC4)=O)nn3)C2)=O)nc1 c1(OC)ccc(Cl)cc1C(=O)NC(C)CNC(c1nnc(O)nc1O)=O C1(C(N2C(CNC(C(COC)C)=O)CC2)=O)CCC(NC(C)=O)CC1 C(=O)(C(C)(CNC(=O)Cn1cc(C)cn1)CC)NC(CC)C(C)(F)F N1(C(C2CCN(C(c3cnn[nH]3)=O)C2)=O)CCCCCC1CCO N1(c2cc(SC)ncn2)CCCC(CNC(c2ccc(C)cc2)=O)CC1 C(=O)(CCC(=O)NC(C)CN(C)C(C1CCCN1Cc1nnn(C)n1)=O)OCC C=CC(C)C(=O)N1CC(O)(CC(=O)N(CC(O)COCC)C)C1 c1(C(=O)NCC(C)NC(=O)Cc2cccs2)ccnc2ccc(O)cc12 N1(C(c2nc(OC)nc(O)c2)=O)C2CCC1CN(C(=O)CC1OCCCO1)CC2 Cc1cc(NC(=O)CC(C(F)F)NC(c2cc([N+](=O)[O-])n[nH]2)=O)cc(C)c1 CC(C)(C(=O)NC1(Cl)CCC1)SCc1ccccc1 C(=O)(CCCCC(C)(C)OC)N(C(CN(C(C(C)OCCOCC)=O)C)C)C N1(C(COCCOCC#C)=O)CCCC(CC(C)NC(C2(C)CCCCC2)=O)C1 c1(C(=O)NCC#CCNC(=O)C=CCN2CCCCC2)ccc2sc(O)nc2c1 N1(C(c2cncc(C)c2)=O)CCCC(C)C1CNC(=O)Cc1ccsc1C c1(CC)nn(C)c(Cl)c1C(=O)NCC(O)CCNC(c1coc(OC)n1)=O CC(C)C(O)C(=O)N1CCCCC1C(=O)NCc1ccc(CC(F)(F)F)cc1 N1(C(c2cccc(CC)n2)=O)CC2CCN(C(=O)C(C(C)O)N(C)C)C2C1 C1(C)(CC)CC(NC(=O)C2CC2)CN1C(C1(c2cccnc2Cl)CC1)=O C#CCC(C)(C(=O)N)NC(=O)CCNC1CC1C.N(C(C)=O)(CC)CC c1(C(N(CCN(C(C(CC)F)=O)C)C(C)C)=O)ccc2c(c1)C(=O)N(C)C2=O c1(CN2CCCC(CC(=O)Nc3cc(Br)cc(F)c3)C2)ccc([N+](=O)[O-])cc1 c1(C(C(=O)NCCC#N)N(CC(CCC)C)C)c(C)nn(C)c1C C12(NC(=O)OCc3c(C(N(C)C)=O)cccn3)CCCCC1CCC2 C1(CC(=O)NCCN(C(C(C)c2cc[nH]n2)=O)CCCN(C)C)CCCC1(F)F c1(C(N2C(C)CC(NC(C3(CF)CC3(F)F)=O)CC2)=O)cc2ccc(F)cc2o1 C1(C(=O)NCC2CCC2)CCC(C2CC2)N1C(c1cccc(=O)o1)=O C1(C)(C(N(CCCNC(c2ccc(C)s2)=O)C)=O)CCc2ccccc2C1 O=C1OC2(CCCN(C(C(=O)NCC(F)F)C3=NOC4CCCCC34)C2)CO1 c1(C(C(=O)NCCOCC)N(CCN(C)C)C2CC2)ccc(F)c(I)c1 N1(C(CCC(C)OCC)=O)CC(NC(=O)CC2CCC(C)(C)CC2)C2CC2C1 Cc1cc(NC(=O)NCC(c2ccco2)O)c(Br)nc1C C(=O)(C1=CCS(=O)(=O)C1)NCC1OCCN(C(c2cc(C#N)sc2)=O)C1 CC(C(=O)NCC(C1CC1)NC(=O)C(C)(C)c1cncs1)C1=CCCC1 c1(OC)ccc(C(C)(C)C)cc1SC.N12CCN(CC1)c1ccc(nc1)C2=O N1(C(CCSC)=O)CC2(CNC(=O)Cc3cc[nH]n3)CC1CO2 C1(CC=C)CCCN(C(c2coc(C(C)NC(c3c(C)n[nH]c3C)=O)n2)=O)C1 N1(C(CS(CC)=O)=O)CCC2(CCCCN(C(c3ccn4cncc4c3)=O)C2)C1 N1(C(CC2CCCN(C(COCCN(C)C)=O)C2)=O)CC2CCCC(C2)C1 C1(Nc2cccc(O)c2F)CCN(C(=O)C(=O)N(C=O)C2CC2)C(SCC2CC2)C1 CC1CN(C(c2ccsn2)=O)CCN1C(C1CC2C=CC1C2)=O c1(N(CCCOC)CC2CCCO2)ncnc(NCC2CCC(C)(C)O2)c1C C1(NC(C2(CS(N)(=O)=O)COC2)=O)CCCCN(C(C2CC23CCOC3)=O)C1 C(=O)(CCCCCC#N)N1CCC(C2N(C(c3c(CC)nc(C)o3)=O)CCCC2)C1 C(=O)(C(O)CC(C)(C)C)NCCC(C)NC(c1csnc1Br)=O C1(C(N2CCCC(F)C2)=O)CC2(CCN(S(=O)(=O)c3ccc(I)cc3)CC2)CO1 c1(CNC2CC3OC(=O)CC23)n[nH]c2c1CCSC2.c12ccc(cc1)OC(=O)N2 c1(CC)cccc(C(N2CCC(C)(CC(=O)NCCC3CC(=O)N(C)C3)C2)=O)n1 C(=O)(C1=CCCC1C)N1C(SC)CCC1.c1(C(=O)NCCNCC(C)O)ccc(Cl)cn1 C(=O)(CC(C)(C)CC(F)F)N(CCCCCC)CCNC(c1csnc1Cl)=O N1(C(c2c(C)snn2)=O)CC(CNC(c2n[nH]c3c2CSCC3)=O)N2CCC1C2 N1(C(c2ncc(OC)nc2)=O)CC(O)CCC1C(=O)NCCc1ccco1 Cc1c(C(=O)NCC(C)(C)CN(C)C(C2CCS(=O)(=O)N2)=O)ccn1C(C)C C1(C(N(C2CCCCC2O)CCC)=O)CC2(C1)CN(Cc1cccc(F)c1C)C2 C(=O)(C(C)(C)CC1CCOC1)N1CCC(C(C)(C)NC(CCN(CC)CC)=O)C1 CCC(CC)CC(F)C(=O)NC12CCC(C(=O)NC(c3ncc(C)s3)C)(CC1)C2 CCC(CC(=O)N(CCC(=O)N1CC2(CCC2)C1)OC)OC c12ccc(cn1)C1CC1C(=O)NCC1(CC1)CCNC2=O.c1(CC)cc(C)on1 CC1C(C)N(C(=O)N=Cc2cccc(-c3ccccc3)c2)CCS1=O CCC(C)CCCC(=O)NCCCNC(=O)CC1CC2CCC(C1)N2C C1(NC(C(C)C2CCC2)=O)CCN(C(=O)Cc2ccc(Cl)cn2)CC1F c1(C(=O)NCCC(=C)CNC(=O)C(O)C2CC2)cc(S(=O)(=O)C(C)C)ccc1Cl c1(C(N(CC(CC)NC(C2CCCCN2CC(F)F)=O)C)=O)c(C)n[nH]c1C N1(C(CS(CC)=O)=O)CCC(C2(NC(=O)CCC3CCCOC3)CC2)CC1 c1(Cc2cc(OC)cc(C)c2)cc(F)c(F)c(F)c1.c12cncc(c1)NC2=O c1(C(=O)NC2C(NC(CCCN(C)C)=O)CS(=O)(=O)C2)ccc2nc[nH]c2n1 c1(C(N2CC(OCCNC(=O)CCCc3ccsc3)C2)=O)cccc2c1CCOC2 c1(OCCC(=O)NCCO)ccccc1.C1(C(=O)CN)CCS1(=O)=O.C1CCO1 CC1(C)CC(CNC(=O)C(F)(F)c2cscn2)CN1C(c1ccsn1)=O N1(C(C(CC)OCC)=O)CCn2nc(CNC(c3sc(C)cc3Cl)=O)cc2C1 N1(C(C2=CCC(C)CC2)=O)CC2CC(NC(=O)CCC3CCOCC3)CC(C2)C1 C(=O)(CCCC(CC)CC)NCCN(C(C(CC#C)C)=O)CC1CC1 C1(C(N(CCCN(C(=O)CCCc2ccsc2)C)C)=O)CCc2nnnn2C1 N1(C(c2ccc(C)cn2)=O)CCC2CN(C(=O)Cn3cnnc3O)CC12 C(=O)(C1OCCn2ccnc21)NC1C2CN(C(c3cc(C)nc(C)n3)=O)C(C2)C1 c1(CN(C(=O)C(c2ccoc2)NCc2cncnc2)C)ccc2nccn2c1 C1(C(=O)Nc2cnc(F)nc2)(CC)CCN(C(c2cnn(C)c2Cl)=O)C1 c1(C(=O)NCC2N(C(CC=C)=O)CCC2)cnc(NCC)nc1 C(=O)(CCCn1cc(-c2cc[nH]n2)nn1)NC(N)=O.C1C(F)(F)N1 c1(N)ccc(C(=O)NCCC2(O)CN(C(c3coc(C(N)=O)c3)=O)C2)cc1F.C(N)=O CC1(C)CC(CNC(C2(C)CC=CCC2)=O)CN1C(=O)CC1CC(=O)NC(=O)C1 C#CC1(O)CC(C(N2CCCC2Cc2cn(CC3COCCO3)nn2)=O)C1 Cc1c(C(=O)NCc2cccc(C(=O)O)c2)nnn1C1CCCCC1O Cc1sc(C(=O)NCCCN(CCCNC(C2CCN(C)CC2)=O)C)c(C)c1C c1(C(N2CC(CCNC(C3(OC)CCOC3)=O)(OC)C2)=O)ccc(=N)[nH]n1 n1(CC)cc(Br)c(C(N2CCC(CCOC)(NC(C3CCN3C)=O)C2)=O)n1 C(=O)(C1c2ccccc2CN1C(c1cc2ccccc2nc1Br)=O)NC c1(OC)cc(C)c(C(=O)NCC#CCNC(c2nc(C)sc2Br)=O)cn1 C1(C(N2CC(CNC(C3(C#N)CCOCC3)=O)C2)=O)CN2CCCC2CO1 N1(C(c2ncc(CC)nc2)=O)CCN(C(=O)C(C)C(O)CCSC)CC(C)(F)C1 C1(C(N(CCN(C)Cc2cccc(Cl)c2)CC)=O)Cc2cc(F)ccc2O1 c1(NC(C2C(CC3(CC(C)C)CC3)C2)=O)[nH]c2ccc(C(=O)OC)cc2c1C N1(C(C(CCOC)NC(=O)C(C)Cn2ccnc2)=O)CCn2nc(C)cc2C1 N1(C(C2(C=C)CCC2)=O)CC(N(C(=O)C(CC)(CC)NC(C)=O)C)C2(CC2)C1 N1(C(c2ccn(C)c2)=O)CCCC2CCN(C(=O)C(C)(C)CC(F)F)CC12 Cc1ccc(SCC(=O)NCCC2CC(N(C)C)C2)cc1.C12(C)CCN(C1)C2=O N1(C(c2cnn(C)c2F)C(=O)NCC=C)CCc2sc(Cl)cc2C1 Cc1cc(Cl)c(C(=O)NCC2C=CCN2C(C2CCCNC2=O)=O)c(Cl)c1 C1(n2cc(-c3nccc(C)c3)nn2)CON(C(=O)CC2CC2c2ccccc2F)C1 c1(C(=O)NC(CN(C(C2CCCOCC2)=O)CC)C)cc(C)cc(OC)c1C CCCCCC(=O)NC(c1ccccc1F)CNC(c1nc(C(C)C)oc1C)=O N1(C(C(CC)C(C)C)=O)CCCN(C(c2cccc(NC(C)=O)c2)=O)C(C(C)C)C1 Cc1cc(C(N2CCN(C(c3sccc3Cl)=O)CC(C)C2)=O)c(F)cc1F N1(C(Cn2c(C(C)C)nnn2)=O)CC2CC(C1)CN(C(C1NC(=O)C3CC13)=O)C2 Cc1nn(C)c(Cl)c1CC(=O)NC1CN(C(C2CC2F)=O)CCC1C(F)(F)F N1(C(CC(c2cc(-c3ccncc3)[nH]n2)=O)=O)CCCCC1c1ccccc1Cl CCC(C(=O)OC)C(=O)N1CCCC(NC(=O)CN(CC(=O)NC(C)C)C)C1 c1(CC)cc(Br)cc(CC)c1NC(=O)CC(C)(C)CCSC N1(C(C(C(=O)OCC)OC)=O)CC2(CC(C(=O)N(CC(O)C(F)(F)F)C)CO2)C1 C#CCCCCCC(=O)N1CCCC1C=CC(=O)N(C1(c2cc[nH]n2)CC1)C C(C(=O)NCc1ocnc1C(=O)N(C)Cc1n[nH]c(C)n1)(C(C)C)SC CC(C)(O)C(C)(C)C(=O)NC1CCC(NC(c2n[nH]c3c2CSCC3)=O)CC1 C(=O)(C1=CCCC1(C)C)N1CCN(C(CCCC(=C)C)=O)C(CC(=O)NC)C1 Cc1cc([N+](=O)[O-])cc(C(=O)NCCCNC(=O)CC2NC(=O)NC2=O)c1Cl C1(CC(=O)NCC2=CCCOC2)CCC2CC2C1.C12CCN(C1)C2=O n1(C(CC)CC)nccc1C(=O)NCC(C1CCOC1)NC(=O)CCSC CCC(CC(=O)NC1CC2CC(C1)CN(C(c1cc(F)n[nH]1)=O)C2)C(C)(C)C C(=O)(CC(C)C(F)F)NCC1CCC(CC(=O)NC(c2cn(C)nn2)C)CC1 C=C(C)CCC(=O)NC1C2CCN(C(C3CC3c3ccccc3)=O)C12 C1(NC(C2C(CC)CN(C(C3(C#N)CCC3)=O)C2)=O)CCCC1C1CC1 N1(C(C2(CCCC)CC2)=O)CC(NC(C2CCC(=O)N2C)=O)C(C(F)F)C1 C1(CCNC(C(C)OCCC=C)=O)CCN(C(=O)COc2cccc(C)c2)CC1 C1(C(N2CCC(O)(C(=O)NCCCCC3(OC)CC3)C2)=O)CCS(=O)(=O)C1(C)C c1(OC(CCC)C)cc(OC)c(C)c(C(C)=O)c1.c1nnnn1C1(C)CC1 CN1C(=O)NCC1C(N1CC2C(CNC(c3cc(C4CC4)[nH]n3)=O)C2C1)=O c1(CCCNC(=O)Nc2c(CC)n(C(C)(C)C)nc2)ccc(F)c(F)c1F c1(C(=O)NC(C)C(=O)Nc2ccsc2)n[nH]c2c1COC2 N1(C(C(C)NC(C)=O)=O)CC2(CCN2C(c2cnc(O)c(F)c2)=O)C1 Cc1ccc2c(N(c3cc(Br)cs3)C)nc(N3CCC(C)C3)nc2c1 N1(C(c2nc(C)n(C)c2C)=O)CCC2(CCN(C(C3CC4(C3)CC4F)=O)CC2)C1 C(C)(c1cnccn1)=CC(=O)NC(C1N(C(c2cc(CC)on2)=O)CCCC1)C c1(C(N2CC(C)CC3CCCCC23)C(=O)NCCOC)ccc2c(c1)C=CC(C)(C)O2 c1(CNc2cncc(C(N3CC4(CCC4)C3)=O)c2)cc2ccccn2n1 C1(NC(c2cc(C)nnc2)=O)CC=C(C(=O)NC2CC(n3cncn3)C2)C1 Cc1cncc(CC(=O)NCC(O)CCNC(c2ccc(C(N)=O)cc2)=O)c1 N1(C(c2c(C)onc2)=O)CCCC2CN(c3nc(C4CC4)nc(Cl)c3C)CCC12 C#Cc1ccc(C(N2CCC(NC(c3nn(C)c(C)c3Cl)=O)C(C)C2)=O)cc1 N1(C(C(CC=C)C)=O)CC2CCC1C(NC(=O)CNC(c1cscn1)=O)C2 c1(OC)cc(C(=O)NCC2COCCN2C(=O)CC(O)C(C)C)cc(Br)c1 C(=O)(C1CCCn2ccnc21)N1CC(C)N(C(=O)C(C)OCCN(C)C)CC1 N1(C(C2(C)N(C(C)=O)CCC2)=O)CCN(C(C2CCCN2C)=O)CC1C c1(OC(C(=O)N(CCC(C)NC(=O)C=C(Cl)Cl)C)C)ccc(C(F)(F)F)cc1 C1(CC=C)(NC(c2ccc(CO)o2)=O)CCCN(C(=O)CC2(N3CCCC3)CC2)C1 N1(C(=O)Cc2c[nH]nc2O)CCC2CN(C(C3(c4ccno4)CC3)=O)CC2C1 CCC(C)C(O)CC(=O)NCC1(C(N2CC3CCCC2C3CO)=O)CCCO1 N1(CC(C)(C)Cn2cccn2)C(=O)CCN(c2ccn(CCO)n2)C1=O C(=O)(C(C)CC(=O)NC(C)CN(C)C(C1(C)C(C)(C)C1(C)C)=O)OC C(C(C)C)(C(O)C(=O)N1CCCCCC1c1noc(C2CC2)n1)OC C(CNC(=O)C(C)CC)(CC(F)(F)F)NC(c1c(CC)c[nH]c1)=O c1(NC(N(C(C2CCCC2)CO)C)=O)c(C#N)ccc(Cl)c1O CC(C)C(C)C(CNC(=O)Cc1csnn1)NC(c1cn(C2CCC2)nn1)=O Cc1c(Br)ccc(C(=O)NC(C)C(C(C)C)NC(C2CCC2)=O)c1F N1(C(Cc2n(C)ccn2)=O)CCCCC(CNC(C23CC(C(F)F)(CO2)C3)=O)C1 c1(C(=O)NCC(C)N(C(C(CC#C)C2CC2)=O)C)cc2n(n1)CCCC2=O N1(C(c2ccc(CSCCC)o2)=O)CCCCCC(NC(=O)CCS(C)=O)C1 C1(NC(COC2CC(NC(=O)C(O)C3CC3)C2)=O)CCC2CC12 CC1C(C)N(C(c2nncn2C)C(=O)NC(C)(C)C)CCS1(=O)=O C12(CC(=O)OC)CCC1CN(C(C1CCOCC1)=O)C2.c1(C(=O)N)cnc(C2CC2)cn1 N1(C(CCN(C)C(C2(F)CCOC2)=O)=O)CC(C(N)=O)C(C(N)=O)C1 c1(CC)onc(C(=O)NCC#CC(=O)N2CCC(COC)C2)c1C CC1(C)CCCC(CC(=O)N(CCCO)CC(F)F)O1 Cc1cccc(N2CCCC(C(=O)NCc3cc(C)[nH]n3)C2)c1 C(CCCC(=O)NC(CC)C(=O)NCCc1cccs1)OC N(C(=NCc1cccc(CC(N)=O)c1)NCc1cccs1)C(CC)C c1(OC)ccc(N(CCO)CCOC(c2ccc(Cl)cc2)CC=CBr)cc1 C1(O)(CCNC(c2c(CC(C)C)onc2)=O)CCN(C(c2csc(Cl)n2)=O)CC1 c1(CCC(N2CCC(N(C(Cc3cc(C)ns3)=O)C)C2)=O)cccc(N(C)C)c1 C=CCC(C)(C)C(=O)NC1CN(C(=O)C(C)Cc2c(C)nn(C)c2C)CC1OC Cc1oc([N+](=O)[O-])cc1C(=O)NC12CC1CN(C(C1CCC(=O)NC1)=O)C2 c1(C(=O)NC(CC=C)CNC(c2cnc(C)c(C)c2)=O)ccc(C#N)nc1C c1(CC(=O)NC2CCN(C(C3CSC3)=O)CC2F)ccc2ncsc2c1 C1(NC(COCCC(C)C)=O)CC(CNC(c2cc(F)ccc2Cl)=O)C12CCC2 c1(C(N2CCC(CCOC)(NC(CCOCC)=O)C2)=O)nncc2c1CCCC2 N1(C(CNC(=O)OCC)=O)CCCCC(N(C(=O)C(C)CCCSC)C)C1 C1(C)(C(=O)NC)CCCN(C(c2occc2Cl)C(=O)NCc2ccco2)C1 N1(C(C(CCC)N(C)C)=O)CCC2C(CCN2C(c2cc[nH]n2)=O)C1 n1(CC)cc(C2CC2C(=O)NCC(C)CNC(=O)COCCOC)cn1 C1(CNC(C(C)(O)C2CCC2)=O)CC2(CCN(C(C3CC(C#N)C3)=O)CC2)CO1 N1(C(C2(C)C(C)C2)=O)CCC(F)(F)C(CC(=O)OC(C)(C)C)C1 C1(=O)C(O)CN1.C1(N(C(C(C)OCC(C)OC)=O)CC)CNC1=O.OCC C(=O)(C(F)CC(C)(C)NC(=O)CN1CC=CC1)NCC(C)(C)CO c1(C(N2CCC3(C(NC(C(COC(C)C)(C)C)=O)C3)C2)=O)cccn2cncc12 N1(C(c2c(CSCC)cccc2)=O)CC(C)N(C(c2ccccc2)=O)CC1C C1(C(=O)NOOC=C)(Cc2cn(C)nc2C)CCCN1C(=O)C=CCO CCCC(C(=O)N1CCCC1CN(C(=O)C=Cc1ccc(CC)o1)C)NC(C)=O CC1CCC(=CC(=O)N(C(C)(C)CC(=O)NC(CCO)C2CCCC2)C)CC1 c1(C(N2C(CC(=O)NC3COCC3O)CC2)=O)ncc(Cl)cc1Cl C1(NC(c2c(C)n(C3CC3)cc2)=O)CCC(C)N(C(c2c[nH]cc(Cl)c2=O)=O)C1 C(=O)(CC(C)(C)C(=O)NCC1CN(C(c2cncc(OC)c2)=O)CCN1C)OC CCCC(C)(O)C(=O)NC(C)CC1CCN(C(C2CCNC2=O)=O)CC1 C1(CNC(C2CCCC(C(=O)OC)C2)=O)CN(C(=O)C=CC=C(Cl)Cl)CCN1C C12(CNC(C3C(C)OC(=O)N3)=O)CC(CO1)N(C(C1CC3(CC3)CO1)=O)C2 N1(C(C2N(C(CC(C=C)C)=O)CC(C)(C)C2)=O)CCOC(C(=C)C)C1 C1(C(N2CCC(CN(C(=O)CS(=O)CC)CC)CC2)=O)CC(=O)NC(CC(C)C)C1 c1(NC(C2N(Cc3cccc(C)c3)CCNC2)=O)cc(Cl)cc(Cl)c1Br C1(NC(=O)NCCS(CC)(=O)=O)CC(F)(F)CN1C(=O)OC(C)(C)C C=C(C)CC(C(=O)N1CCC(C)(CNC(C2CCCC23CC3)=O)C1)OC C1(NC(c2cc(OCC)no2)=O)COC2(C1)CN(C(=O)C(C)(C)C(=O)NC)C2 C1(NC(CCCC)=O)CC(C2CCN(C(c3c(C)cc(F)cc3C)=O)C2)C1 c1(C(=O)NC(C2CCCC2)CNC(c2c(C)n(C)nc2)=O)ccc(F)cc1Cl c1(C(c2ccccn2)NCCCO)cc(Br)cc2[nH]ncc12 c1(C(=O)NC(C(=O)NC(COC)CO)CC2CC2)c[nH]c(=O)cn1 N1(C(C(c2nc(C)sc2)=O)=O)CC2CCCC(NC(c3ncc(Cl)n3C)=O)C2C1 C1(C(=O)NCC2(C(N)=O)CN(C(c3c(CC)nns3)=O)C2)NC(=O)OC1C c1(C(=O)NCCCC2(NC(c3cc[nH]n3)=O)CC2)nnc2ccccc2c1O N1(C(c2c(CC)scc2)=O)CCCC(C)(NC(=O)CC2(CSC)CC2)C1 N1(C(C(Cc2ccco2)NC(C(C=C)OC)=O)=O)CCOC(CCO)C1 C1(C(=O)NC2(CC=CC(=O)NCc3cnc(C)[nH]3)CCC2)CN2CCN1CC2 c1(C(=O)OC)nc(=NCCN(C)C(c2cc3sccc3cn2)=O)c(C)c(C)[nH]1 N1(C(C2(c3ccco3)CCC2)=O)CC2CCC(C1)N(C(=O)Cc1ccsn1)C2 c1(C2(C(=O)NCCN(C(C3CCC4CC34)=O)CC)CCC2)cccc([N+](=O)[O-])c1 c1(CC(N2CCCC(NC(c3n[nH]cc3F)=O)C2)=O)c(Cl)cccc1Cl c1(C(=O)NC(CNC(C(C(=O)OCC)(C)F)=O)CC(C)C)cccc2c1CCC2 N1(C(CC)=O)CCN(C(C2CCCN2S(=O)(=O)CC)=O)CC1Cc1ccccc1 N(C1CCOc2c(C)cccc21)C(c1n(CC)nnn1)C1(C(C)C)CC1 Cc1cc(C(=O)NCC(C)(C)CNC(c2cc(O)n(C)n2)=O)cnn1 c1(OC)ccccc1CN1CC2C(CO)C2C1.C1(C(=O)O)CCCN1C(C1CCOC1)=O c1(NC(=O)NCCC2C(C)(C)OCC2)c(C(F)(F)F)nc2ccccn12 C=CCCCC(C(=O)NC1CC(NC(=O)CCC(=O)N(C)C)C(O)C1)N(C)C C1(NC(C2C(C)(Br)C2)=O)CCN(C(=O)C(=Cc2ccccc2)C#N)CC12CCC2 O=C1NCc2c(NC(=O)C(=O)NCCOC(=O)Nc3cccs3)cccc21 c1(NCC2CCN(CC)C2)[nH]c(=NCc2ccc(C)o2)nc2sccc12 CC1CC(NC(=O)NCCC23CC(CCO2)C3)CC(C)S1 c1(CN(C(=O)CC2CCC(C)(C)C2)C)cc(Cl)cc(Cl)c1 CC1CCC(NC(=O)Cc2cnoc2)CN1C(=O)CCOC1CC1 CC1CC(NC(=O)CC(C)(O)c2ccccc2)CN1C(C1(c2ccncc2)CC1)=O C=CC1(C(N2CC(NC(C3CN4CCC3CC4)=O)C(COC)C2)=O)CCOCC1 C1(=CC(N2C(CNC(C=CCOC)=O)CC2)=O)CCN(C)C1 CC(C)CC(C(=O)NC1C=CC(CNC(C2CCCC2C)=O)C1)C(N)=O c1(CC)ncnc(N2CCCC2C(=O)Nc2cnn(-c3ccc(Cl)cc3)c2)c1F C(=O)(C1CCCc2nncn21)N1C(C)(C)C(NC(=O)CC2CCCCC2)CC1 CC(CN=c1[nH]c(=N)[nH]c(=NCc2cccc(Cl)c2F)[nH]1)C(C)(F)F C(=O)(C(CC)CC(C)C)NCC(C(=O)NCCCOCC)CC1CCCC1 n1(CC2CCN(C(c3cc4cnn(C(C)C)c4s3)=O)C2)ccc2cc(Cl)ccc12 O=S(=O)(C=Cc1ccc(F)cc1)NC1CCC1CF c1(OC)cc(Cl)ccc1C(=O)NCC1(C(N)=O)CCCN(c2nnc(O)s2)C1 c1(OC(C)C(=O)NCC2C3CC2N(C(C2(N(C)C)CC2)=O)C3)ccccc1Cl O=C(C1=Cc2ccccc2C1)N1CC2CC1CCC2NC(C1CC(F)(CO)C1)=O c1(C(N2CC(C(=O)OC)C(F)(F)C2)C(=O)NCC(F)F)cc(Cl)c(F)c(Cl)c1 C1(CNC(CN(C)C)=O)CN(C(=O)CC2CN(C(N)=O)CCO2)CCN1C C1(CC(=O)NCC2(C)N(C(c3cncc(C)n3)=O)CCC2)CCCCC12CC2 c1(C(=O)NCCC2CCN(C(=O)Cn3ccnn3)C2)ccc(-c2cnn[nH]2)cc1 c1(N2CCCC(CNC(CCOCCN(C)C)=O)CC2)ccc([N+](=O)[O-])cn1 CC1(C2CC2)CCN(C(=O)C(c2cccs2)NC(=O)CCOCC(F)F)C1 S(=O)(=O)(c1ccc(C(=O)O)cc1)N1CC(C)N(Cc2cc(Br)cs2)CC1 C(=O)(C#CC1CCOC1)NC1CC2(CC(CNC(C3(C)N(C)CCC3)=O)C2)C1 N1(C(C2CC(OCC(C)C)C2)C(=O)NCCCC2CC2)CCOCC1 Cc1sc(Cl)nc1C(=O)NCC(C)(C1CCC1)NC(=O)CCCn1ccnn1 CC(CN)CC(=O)N(C)C.C1C(Cc2ccccc2O)C(=O)N1.C(C)(C)(C)OC=O c1(OC)cc(CC(=O)NCCCCN(C(=O)C#CC(C)(C)C)C)cc(OC)c1O CCC(C)(C)C(C)CC(=O)NCCN(C(=O)CC(C)C(F)F)CC1CC1 c1(C(=O)NC2CCCCN(C(=O)C=CC3CCCC3)C2)cnc(O)c2cncn12 C1(C(=O)NCC2(CNC(CN(C)C(N)=O)=O)CCC2)COc2cc(O)ccc2C1 c1(C(=O)NCCN(C(CC(C(F)(F)F)OC)=O)CC)cc2c(F)c(F)ccc2[nH]1 C1(NC(CC(C)C)=O)(CF)CCN(C(c2ccc(C(N)=O)cn2)=O)C1 CC(CCO)C(=O)NC(CNC(=O)Cc1nncn1C)CO C1(C(=O)NCC(=O)OC)CN(C(=O)C(F)C2CCOC2)C1 N1(C(CCSC)=O)CCC2(CC1)OC1(C)CC2(NC(C2CCCCC(=O)N2)=O)C1 C(=O)(C1=CCCCC1C)N1CCCC(C(=O)NCCn2cccn2)(CC)C1 C12(NC(CC)=O)CCN(C(=O)Cn3nc(C(F)F)cc3C3CC3)CC1C2 c1(C(N2CCC(N(C)CC)C2)C(=O)NCCSC)cc(Br)cc2cccnc12 c12cc(Cl)ccc1O2.N1(C(C2(OCC)CC2)=O)CC(C(N)=O)C(C(F)(F)F)C1 C1=CC(F)C(=O)NC(C(C)C)CNC(=O)CC1.C(C(=O)OC(C)(C)C)SC.C=O c1(NC(C2CCC(c3cnc(C)o3)CC2)=O)cc(Cl)ccc1O N1(C(C(n2ncc(C)c2)C)=O)CCCN(C(=O)CC(C)C)CCC1 c1(C(=O)NC(CN(C(c2c(CC)nns2)=O)C)C)cnc2c(ccn2C)c1 C(=O)(C(C#N)CC1CC1)NC(CC(C)OCC)c1nnnn1CCCNC1CC1 c1(C(c2cn(-c3cc(OC)ns3)nn2)C)nc(C2CN(C3CCOC3)C2)n(C)n1 C(=O)(C(F)C(F)(F)F)NCC(CNC(C1C(CN(C)C)C1)=O)(C)C c1(COC(c2ccc(N3CCOCC3=O)cc2)=O)ccc(S(=O)(=O)CCO)cc1 C1(CC(N2CC(COC)(NC(c3ccc(Br)o3)=O)C2)=O)CCCCN1C CC1(C)COCCC1C(=O)Nc1ccc(SC(F)(F)F)nc1 N1(C(Cc2c(C)nc(CC)nc2C)=O)CCN(C(=O)Cc2cnsc2)CCC1C CC1(C)CN(C(C23CCCC2C3)=O)CCC1C(N1CCC(CC(F)F)C1)=O c1(C(N2C(C(N(C)CC3(F)CCC3)=O)C(C)(C)CCC2)=O)ccc2cc[nH]c2n1 C(=O)(C1CCCc2nnn(C)c21)NCC1(CC(=O)NCC(c2cccs2)C)CC1 Cc1cc(C(=O)NCCN(C2CCCCCC2)C(C2CC2Cl)=O)[nH]c1C c1(C(=O)NCC23CCC2CN(C(C2CCS2(=O)=O)=O)C3)cc2cc(F)ccc2s1 C(=O)(C(C)(C)CNC(c1cc(C2CC2)no1)=O)NCCCC C1(NC(c2cn(CC)nc2)=O)CC(O)CN(C(=O)C(c2cncn2C)O)C1 C(=O)(CC(C)C(F)(F)F)NC1CC(NC(C(c2c(OC)ccc(F)c2)=O)=O)C1 C(=O)(C1=CC2CCCCC12)NCC1CCC(NC(CC(C=C)CC)=O)CC1 C12(CC)CCC(C(=O)NC3CC(CNC(c4cc(C(N)=O)c[nH]4)=O)C3)(CC1)CO2 CC1C(CC(=O)NOCCCCF)CCN1C(c1cnncc1O)=O C(C(C)(O)CC(=O)N1CCOCC(CNC(C2CC3(CSC3)C2)=O)C1)OC C1(CCCC(N2CC(CC=C)(NC(=O)Cc3nc(=N)[nH][nH]3)C2)=O)CCCC(=O)N1 C1(C(=O)NCCC2CN(C(=O)CC3CSC3)C2)CCOC1C1CC1 Cc1ccc2cc(C(N3CCC(N(C(=O)C(C)(C)C(C)C)C)CC3)=O)oc2c1 C1(C(=O)NCCCN(C(=O)C(C)CCOC)CC)CCC(N(C)C)CC1 c1(SC)cccc(CO)c1.c1(CCC(=O)NC(c2ccccc2)C)ccc(C(=O)N)[nH]1 Cc1cc(C#N)sc1C(=O)OCC(c1ccccn1)C C(=O)(C1=CCCCO1)N1CC(O)(CNC(c2nnc(C)s2)=O)C1 c1(C(=O)NCC2N(C(CS(CC)=O)=O)CCC2)ccc2cnnc(O)c2c1 N#Cc1cc(C(=O)NCC2(CO)CCCCCC2)ccc1Br N1(c2n(CC=C)c(C3CCOCC3)nn2)CN=C(N2CCOC(C)C2)NC1=O c1(C2C(CNC(C3CC3CNC(c3coc(Br)c3)=O)=O)C2)ccccc1Cl Cc1cc(NC(c2cc(Br)cn2C)c2nnnn2-c2ccccc2)cnc1Cl C1(C(=O)NCC(C)NC(C2CC=CCO2)=O)Cc2cc(F)cc(F)c2O1 CN1CC(C(=O)NC2COCC2NC(c2nonc2N)=O)NC1=O Cc1ccc(C=CC(=O)NCC(O)CCNC(=O)C(C)SCC(N)=O)o1 CCC(CCC(=O)NC1(CCNC(c2ccc(OC)c(F)c2)=O)CCCC1)OC c1(C(N2C(c3cccs3)CCC(C)C2)=O)n[nH]c2ccccc12 c1(CC)ccc(C(N2CC=C(CNC(=O)COC3(C)CCCC3)CC2)=O)c(F)c1 C1(C(=O)NC(C)CCNC(=O)CCCC2CCOCC2)CCC(C(F)(F)F)CC1 Cc1nc2c([nH]1)COC2=O.C1(NC(=O)OC(C)(C)C)CCCN1CC(C)C N1(C(c2cnc(-c3ccccc3F)s2)=O)CCC12CCSCC2 c1(CC)nc(C(=O)NCC(O)CCNC(=O)C(CCC)OCC)c(N)s1 c1(OCC)cc(CNCCC[Si](C)(C)C)cc(OC)c1C#N C1(CCOCC)(NC(=O)CO)CCN(C(=O)CCc2cccnc2)C1 c1(OC)ccc(C=CC(=O)NC(C)C(C)NC(=O)C=CS(C)=O)c(C)c1 CCC(C)C(=O)C(=O)N1CCC(C(N2CC(C)(CO)C2)=O)O1 N1(C(C(C(C)C)O)=O)CCC2CCC(NC(=O)CSc3ccc(Cl)cc3)C12 C1(CNC(C2N(C)C(=O)CC2)=O)CCN(C(c2cncc(F)c2)=O)C12CCC2 c1(C(N(C2CCC(NC(CC3C(C)CCO3)=O)CC2)C)=O)cc(F)cc(Cl)c1 CCCCCCC(CC)(CC)C(=O)N(C1CCC12CCNCC2)CCN(C)CCO N(C1CN(C(c2cccc(O)c2)=O)Cc2ccccc21)C(C(C)(O)C(F)(F)F)=O C1(NC(C(CC)CC)=O)COC2C(NC(c3nc(C)n(C)c3C)=O)COC12 C1(OC)CN(C(=O)C(C(C)C)NC(=O)CN2CSCC2=O)CC1(C)C C1(CNC(C2(C)CCCC2O)=O)(NC(=O)C#CC2CCC2)CCCCCC1 Cc1nnsc1C(=O)N(C(C)(C(=O)NC(CO)C1CC1)C1CC1)C C1(NC(C2(C)CCC(C)C2)=O)COC2(C1)CN(C(=O)Cc1c(Cl)cnn1C)C2 c1(C(=O)NC2CCCN(C(C(CC)(C)CC)=O)C2)cc(OC)c(S(N)(=O)=O)s1 C(=O)(CCCCC(=O)N1CCCC(NC(=O)CC2CC3CC3C2)C1C)OCC C1(NC(C2CC(OC)C2)=O)CCC(C(=O)NCc2ccc(C)o2)C1 C12(C(=O)NC)CC(Cc3ccccc3)(C1)OC2C.CC1C(=O)NCCNC(=O)N1 N1(C(CCN(C(CC(C)(C)C2CC2)=O)CCO)=O)CCOC2C(O)CC12 CC(C)CC(C)(CO)NC(C1CCCCN1C(C1OCC2CCCC12)=O)=O C1(CC(N2CC(CCCCNC(c3nc(C(C)C)oc3)=O)C2)=O)CCCCN1C c1(CC)nccnc1C(=O)NCc1cc(C(=O)N(CCCCC(C)C)C)on1 c1(C(=O)NC2CCN(C(=O)COc3ccsc3Cl)C2)cc(Cl)cc2ccncc12 C(CCCCCN(C1CCS(=O)(=O)C1)C)NC(C1(C(c2ncccn2)CC)CC1)=O N1(c2n(CCOC)c(C(c3ccco3)C)nn2)CC2CCCCC2C1C c1(C(C(=O)N(C2CCN(C(=O)CCN3CCCCC3)C2)C)O)ccc(Cl)c(F)c1 c1(NC)cnc(C(=O)NCC2CC(C)N(C(=O)CN3CCCNC3=O)C2)cn1 CC#CCC(C(=O)N1CCC=C(C)C1)NC(c1cc(C)cc(C)n1)=O C1(NC(C(F)=CCC)=O)CCCN(C(c2cccc(C(N)=O)c2O)=O)C1C c1(OC)nccc(C(N2CCC2C(=O)N(C)Cc2cnccc2C)=O)n1 CC(C)(C)C(O)C(=O)NCC12CC1CN(C(=O)Cc1nc[nH]n1)C2 C(CCCC(C)C)(C(=O)NCCCOC)N1CCN(C(CC)C)CC1 Cc1nc(CCC(N2CC(CNC(=O)CN3CCCCC3=O)C(O)C2)=O)oc1C c1(C(=O)NC2C=CCN(C(C3(C)CC3(F)F)=O)C2)cc2ccccn2c1 c1(C(=O)NCC2C(NC(c3nc(Br)c[nH]3)=O)C2)c(Cl)ccc2ncccc12 c1(C(N2CCN(C(CSc3nc(C)[nH]n3)=O)C3C2C3)=O)ccc2nccnc2c1 Cc1cc(NCCCN2CCN(C)CC2C)nc(N2CCC(CC(C)C)CC2)n1 N1(C(c2c(C)cn(C)c2)=O)CCCC(C)(C)C1CNC(=O)CC(C)c1ccco1 c1(C(=O)NCC2C(C)CCN(C(=O)C(N)=O)C2)ccc2sccc2c1 C1(F)(CNC(=O)COCC2CCCO2)CN(C(c2ncoc2C2CC2)=O)C1 c1(N2C(C)(C(=O)Nc3ccc(C(F)(F)F)c(F)c3)CC2)ncnc2c1CCCC2 N1(C(C(C)C2CC2)=O)CC(NC(=O)CCCc2nccs2)C2(CCOCC2)C1 c1(C(=O)NC(CCNC(c2nc(C)oc2)=O)C)c[nH]c2nccc(Cl)c12 C1(CCNC(c2n(CCCOC)nnn2)c2sccc2C)CCCCCC1 C1(C(=O)NC2CC(C)(C)N(C(=O)C=CBr)C2)CCCC2(CCC2)O1 N1(C(CC2(COC)CC2)=O)CCC(C)C(N(C(=O)CC(C)n2ccnc2)C)C1 N1(C(c2c(C)oc(CNC(C3CC(=O)NC(C)C3)=O)n2)=O)CC(C)CCCC1C C(c1ccccn1)=C(C)C(=O)NC(C)(C)CNC(c1ccnc(N(C)C)c1)=O n1(CC)ncc(Cl)c1C(N1CCCC(C(C)(O)CNC(=O)Cn2nccn2)C1)=O c1(SCCC(=O)NCC2(NC(C3(C)CC3Br)=O)CC2)ccccc1 C1(NC(Cc2ccc(OC)cc2OC)=O)CN(C(=O)C=CS(C)=O)C2(CCC2)C1 c1(CN(CC(C)C#N)C(N2C(COC)CCC2)=O)cccc(Cl)c1 N1(C(c2nc(CC)oc2)=O)CCC(CC)CC1C(=O)NCCOC(=N)O c1(C(=O)NC23CCN(C(c4cccc(Cl)c4O)=O)CC2C3)cccc2c1CCC2 N1(C(c2ccc(C)o2)=O)CC(O)CC1CNC(=O)CCc1ccc(C(F)F)cc1 C1(COC)CN(C(=NCCNS(=O)(=O)c2ccc(C)c(C)c2)NCC(C)C)CCO1 c1(NC(C2C(C)CN(C(C3CCCCO3)=O)C2)=O)cncc([N+](=O)[O-])c1 c1(CC(C(=O)NCC=CCNC(=O)C(O)Cc2cnc[nH]2)O)cc(Cl)cc(Cl)c1 c1(OC)cc(C(=O)NCC2CCCN2C(C2OCC2(C)C)=O)ccc1C(N)=O N1(C(c2cc(Br)nn2C)C(=O)NCCOC)CCC(S(C)(=O)=O)C1 CC1(C)CN(C(C2CC(F)(CO)C2)=O)C1C1CCN(C(C2C=CCC2)=O)CC1 N1(C(c2ccc(CC)s2)=O)CCN2C(=O)C(NC(=O)CCCC(=O)OC)CC2C1 n1(CC)nc(C)c(C(=O)NCC(C2CC2)N(C(=O)CC2CCC(C)(C)C2)C)c1Cl c1(C(C(N2CC(C(C)NC(c3ccns3)=O)OCC2)=O)O)cc(F)c(F)cc1F C1(C(N2CC3CC2C3)C(=O)NCCSC)CCC(CCC(C)C)CC1 C1(NC(c2sccc2C2CC2)=O)(CNC(=O)CC2CCC2)CCCC1 CC1OCCC1(C)C(=O)NCCNC(c1sccc1C(=O)Nc1ccccc1Cl)=O CC(C)C(C(=O)N1CCC2(CC2NC(C2C3CC4C(C3)C24)=O)C1)C(C)C CCC(CC)C(C(=O)NC(C)CC1CN(C(c2c[nH]nc2Cl)=O)C1)OC c1(C(C)=O)csc(C(=O)NCCCNC(C2CCN(CC(C)C)C2)=O)c1 C1(CC(=O)N(C2CC(NC(c3c(CCC)nco3)=O)C2)C)SC2=NCCN2C1=O N1(C(c2c(OC)cccc2)=O)CC(CNC(=O)C(C)N(C)C(C)=O)C2(CC2)C1 c1(NCC(c2ccc(C(C)C)cc2)C)nncc2ccccc12 Cn1cc(C(=O)NCC#CCNC(C23CCCCC2CCC3)=O)c(=O)n(C)c1=O C1(C)(C(=O)NCC(CC)NC(=O)C(O)Cc2cnc[nH]2)CCCCNC1=O C1(CNC(c2c(Cl)cc(C)s2)=O)CN(C(=O)CC2CC(=O)NC2=O)CCC1(F)F c1(C(=O)NC2C=CCN(C(C(C=C)O)=O)C2)c[nH]c2c(F)cccc2c1=O C(C)(C)(CCC(=O)N(C(CC(F)F)C(=O)NCC(C)CC(C)C)C)OC n1(C(F)(F)F)cncc1-c1nc(C23CCCC2C3)no1 c1(C(=O)NCC(CO)NC(C2C(F)(C(N)=O)C2)=O)cc(-c2ccncc2)[nH]n1 N1(C(=O)Cc2csnn2)CCC2CN(C(C3CCCC(F)(F)C3)=O)CC2C1 C(=O)(C1Cc2ccccc21)NCc1c(C(=O)NC2CCC(C(N)=O)C2)occ1 c1(C(N(CCCNC(C2CCCCC2)=O)C)=O)cnc2ccc(Cl)cn2c1=O C1(C(C)C)CN(C(C2CCS2(=O)=O)=O)CCN1C(=O)CCCc1cccs1 Cc1cc(C(=O)N(C(C(=O)NC2CC3(CCC3)C2O)C2CC2)C)c(O)nn1 C=CCC(C)(O)C(=O)NCc1ocnc1C(N1C2CSCC1C2)=O Cc1cccc(C(N2CC(NC(=O)CC=CCSc3ccccc3)C(C)C2)=O)c1 c1(CC)c(C(N2CCOC(CC(=O)NCc3nnn(C)n3)C2)=O)cnn1C C1(NC(CNC(COc2c(C)occc2=O)=O)=O)CC(C)CC(C)(C)C1 C1(C(N2CCC(CN(C(C=CSC)=O)C)C2)=O)CC2(CC2)CO1 Nc1cnccc1C(N1CCCC(NC(C2CC2c2ccncc2Cl)=O)C1)=O CC1(NC(c2ccc(O)nc2)=O)CCN(C(C2CCN2S(C)(=O)=O)=O)CC1 C1(CCNC(CCN(CCC)C)=O)CCN(C(c2snnc2CC)=O)C(C)C1 C(=O)(C(C)C(C)(C)C)N1C(C(=O)NCc2c(C)ccs2)C=CCC1 N1(C(C(CC)Oc2cccc(Br)c2Cl)=O)CCc2ccccc21 N1(C(COC2CC(NC(c3c(CC)cncc3)=O)C2)=O)CCOC(C)(C)C1 Cc1cnc2cc(C(=O)NC(CCNC(C3COC(=O)O3)=O)C(C)C)ccn12 C(=O)(N=c1cc[nH]c2cc[nH]c12)c1cc(=NCc2c(CC)c(F)c(Cl)cc2)[nH]cn1 c1(C(=O)NC(C2CCN(C(c3nn(C)cc3Cl)=O)C2)C)ncncc1F N1(C(C=C(CC)CC)=O)CC2CCC2(CCNC(c2cnc(C)cc2C)=O)C1 N1(C(c2c(C#C)c[nH]n2)=O)CCC2CCC12CNC(c1cccc(SC)c1)=O c1(C(N2C(C)C(C(=O)NOCC(O)C(C)(C)C)CC2)=O)cc2cccnn2c1 C#CCCCC(=O)NCC(CC)(CC)NC(=O)C(C)CC=CCC C1(C(N2CCC(F)(F)C2)=O)CN(C(=O)CCc2nncs2)C2(CCC2)C1 Cc1cc(C(=O)NC2CCCC23CCN(C(=O)C(C)(C)F)C3)c(N)c([N+](=O)[O-])c1 Cc1nc2c([nH]1)CC(C(=O)NCCOC1CCN(C(=O)C=CC(C)(C)C)C1)CC2 c1(C(=O)NCCC2CCN(C(c3cnc(C4CC4)s3)=O)C2)cnn2ccccc12 CN(C1CS(=O)(=O)c2ccccc21)S(=O)(=O)c1ccc(NCC(Cl)(Cl)Cl)c(F)c1 c1(OC)c(Cl)nc[nH]c1=NCC(C)NC(c1ccc(F)cc1)=O N1(C(C(F)=CC)=O)CCC(CCNC(=O)CCCCC#N)CC1C Cc1cc(=NCC2C=CCC2)[nH]c(NC(C)COC2CCC2)n1 Cc1cc(C(N2CCC(O)(CCNC(C3CC(C)(C)O3)=O)C2)=O)ccc1C1CC1 c1(C(N(CC(C)NC(C2(OC)CC2)=O)C2CC2)=O)c(Cl)cccc1Br C(CC(C(=O)N1CC2CCC1C2)NC(c1cnccn1)=O)N(C)C N1(CCOCC)CC2(CN(C(c3n[nH]c4ccc(O)cc34)=O)CCO2)C1 C(=O)(C1=CNC2=NCCC2=C1)NCC1(CNC(=O)C(F)C(F)(F)F)CC12CCC2 c1(N2CC3(CCN(Cc4cc(C)[nH]n4)CC3)C2)n[nH]c2ccc(C#N)cc12 C(C(=O)NC1(C)CC1)(C1=NOC2CCCCC12)N1CC(C)(C)C(F)(F)C1 C(=O)(C(C(C)(C)C)C1CCC1)N(C(C)C)CCN(C)C(C12CCC(C1)C2)=O N1(C(C(CNC(C(C)C(F)(F)F)=O)(C)C)=O)CCC(F)(F)C(O)C1 c1(C(N2CCCC(NC(C3CC4C(C)(C)C4C3)=O)C2)=O)ccc(Cl)c(Cl)c1N CC1CN(C(C2CC(=O)C2)=O)CCC1C(=O)NCC(C)(C)CC1CC1 C1(C(=O)NC2C(NC(CC(CC)(C)C)=O)CCC2)CCn2c(cnc2C)C1 C1(NC(COCCC=C)=O)C2CCN(C(c3cnc(C(C)C)nc3)=O)CCC12 c1(SC)ncc(C(=O)NCC2(O)CN(C(=O)CCC3CC3(F)F)C2)s1 C1(CC)CCC(C)N(C(c2ccnc(CNC(C3COCC3C(N)=O)=O)c2)=O)C1 CC1(c2ccccc2)NC(=O)N(c2ccccc2Sc2ccc(C(=O)O)cc2)C1=O Cc1cc(CNCc2csc(-c3ccccn3)n2)cnn1 C1(OC(=O)CC2CCC23CCC3)CCOC2(CCC2)C1 C12(CNC(CN(C)CC)=O)CC(CC(C3CCN(CC(F)F)CC3)=O)(CO1)C2 C1(C(=O)NC2CC(NC(C3CCC(CC)O3)=O)C2)CC2C=CC1C2 C(CCC(=O)NCC(Cc1ccccc1)NC(=O)CCC1CCOC1)=CC N1(C(C(CC(=O)OC)(C)C)=O)CC2COCCC2(NC(c2ccc(Cl)s2)=O)C1 CCC(CNC)CC(=O)NCC=CCNC(c1nc(-c2ccccc2)ccc1F)=O N1(C(C(C2CCN(C(c3ncon3)=O)CC2)C)=O)CC2CCCCCCC12 N12CC3CCC3(C1)CC2=O.N1(C(COC)=O)CC(OC(C)(C)C)CC1CO CC1CCN(C(c2cnc(C(C)(C)C)nc2)=O)CCN1C(=O)Cn1nccn1 c1(C(=O)NCCC2N(C(CC3C(=O)NC(=N)S3)=O)CCC2)cccc2cc[nH]c12 C12(NCN(C(=O)CCOC3CCCOC3)C)CCCCC1C2(F)F C1(NC(c2coc(Cl)c2)=O)CN(C(c2nccc3c[nH]nc23)=O)C2CCCCC12 c1(N2CCC(=O)NC(C)C2=O)nc(=NCCCNS(C)(=O)=O)[nH]c2c1cnn2C C(C(=O)NC1CN(C(=O)C(=O)NC2CC2)CC1C)(C(C)C)OCCCOC N1(C(C2(C(=O)NC)CC2)=O)CCC(F)(C(=O)NC2CN(C)C(=O)C2C)CC1 N1(CC(C)C)CCN(C(c2scc(Cl)c2Cl)C(=O)NCc2cccnc2)CC1 C(=O)(C1=NOC2(CCOC2)C1)NC(CC)CNC(=O)Cc1nc(C2CC2)cs1 c1(C(=O)NCCOCCCNC(C2OCC(C)C2)=O)c(F)ccc(F)c1O N1(C(c2c(OC)cncc2)=O)CC=C(CNC(C23COCC(C2)C3)=O)CC1 N1(C(C(COC)COC)=O)CC2CC1CN(C(c1ccn(C3CCCC3)n1)=O)C2 c1(C(N2CCC(N(C)C(c3ccccc3O)=O)C2)=O)[nH]nc2ncc(Br)cc12 c1(CC(C)(C)C)ccc(N2CCCC2c2nc(C3CC3)no2)cc1 N1(C(C(C)(C)C)=O)CC2(CCOCC2)CC1CNC(=O)C(F)(F)C(C)(C)O c1(NC2C(OC)COCC2)nc(C)cc(=NCCc2cn3c(n2)COCC3)[nH]1 N1(C(C2CCC2(F)F)=O)CCN(C(c2ccnc(N(C)C)c2)=O)CC1.CO c12cc[nH]c1C(=O)NC2.N12CCC(C1)C2=O.C(C(=O)OC)N(C)CC c1(C(N(CCNC(C2(C)CC(=C)C2)=O)C)=O)c(C)ccc(F)c1Br C=CC(CC)CC(=O)N1CCCC1CN(C(=O)CC1(N(C)C)CCCCC1)C C1(CNC(c2cc(CC)c(C)s2)=O)CC(NC(=O)CC(C)(C)O)C12CCC2 c1(CNC(C(=O)NCC2CN(c3ccc(C)cc3)C(=O)C2)=O)cc(C)nc(C)c1 c1(C(=O)NC2CN(C(C3(SCC)CC3)=O)C2)cnn(CCCF)c1 N1(C(CC(=O)NCC(COCC)C(C)C)=O)CCCC(F)(c2ccccc2)C1 C1(O)(COC(C)(C)C)CCCN(C(=O)Cn2occ(C(=O)OC(C)(C)C)c2=O)C1 C12(NC(C3(NC(c4cccc(F)c4)=O)CC(F)C3)=O)CCN(CC1)CC2 C1(C(N2CCC(O)(COC)C2)=O)(NC(C(C)SCCCC)=O)CCN(C)C1 C1(C(=O)NCCCN(C(c2cc(Cl)cs2)=O)CC)CCCCN1C(N)=O C1(NC(CSCC=C)=O)CCN(C(=O)C(C2CCCCCC2)OC)CCC1(F)F Cc1nc2c(C(=O)NC3CCCCC3CNC(c3n[nH]cc3Br)=O)cccc2o1 c1(C(N2C(C(C)C)CN(C(C3(C)CNC(=O)C3)=O)CC2)=O)onc2ccccc12 CC(C)CC(CN(C=O)C(c1c(F)cccc1F)C)CC(=O)O C(=O)(C(C)(C)S(C)(=O)=O)N(CCN(C(c1cc(OC(C)C)ncc1)=O)C)C N1(C(CCC2C(C)C2)=O)CCC(CF)(NC(c2cc(=N)[nH]n2C)=O)C1 CC#CCCC(=O)NCCCC1CN(C(C2(CN(C)C)CCCC2)=O)CCO1 c1(OCC(C)C)c(C(N2CCC(N(CCO)C(C3CC3C)=O)C2)=O)cccc1C c1(C(CC)C(=O)N2CCCC2CN(C)C(C2(CF)CCC2)=O)ccc(F)cc1 CC1(C)CC(C(=O)NC2CC2)CN1C(=O)CC1CC=CCC1 C(CO)(CCC)OCCC(=O)NC(C#C)CC1CCCO1.C12CN(C1)C(=O)C2 N1(C(CC2(C)CC2)=O)C(CNC(C23CC(C)(C2)OC3(C)C)=O)CC2CCCCC12 Cc1cc(C(N2CCNC(C(N3CCC(C(F)F)CC3)=O)C2)=O)nc(C)c1 C(=O)(C1=C(Cl)CCOC1)N1CC(C)CC(NC(c2c(C)sc(O)n2)=O)C1 c1(C(=O)NC2CCC(NC(C(C)NC(C)(C)C)=O)C2)ccc2cc(F)c(F)cc2n1 CCCCC(O)C(=O)NCCCC(C)(C)NC(=O)C(CN(C)C)C(C)C Cc1cc(C(=O)NC23CC(NC(C4CCNC4=O)=O)(C2)C3)cc(C)c1C#N CC1=C(c2ccc(C(=O)NCc3cc([N+](=O)[O-])ccc3Cl)s2)CCCC1 Cc1cccc(CNC(=O)C(CCC2CCC2)NC(=O)CCCn2cncn2)n1 c1(NC(=O)NCc2nn[nH]n2)ccc(=NCc2ccc(Br)cc2)[nH]c1 C1(NC(C2CCCCN2CC(F)F)=O)C2CN(C(c3csc(O)n3)=O)CC12 Cc1ccc(NC(=O)NC2C=CCC2)nc1 CC(CCCC(=O)NCCNC(C1(C#N)CC1(C)C)=O)c1ccccc1 [N-]=[N+]=NCCCCCCC(=O)NC1CC2(CCN(C(C34CC(F)(C3)C4)=O)C2)C1 c1(C(=O)OCC)c[nH]ccc1=N.c1(C2CCC2)ccc(F)cc1 C(=O)(CCC(CC1CCCC1)NCCCOCCN(C1CCC(C)CC1)C)OCC N1(C(C(CC)C(=O)OC)=O)CC2CC(C1)CN(C(C1C3(CC3)C13CC3)=O)C2 C12(C(=O)NC3CCC(NC(C4CN(C)C(=O)CC4)=O)CC3)CCC(C)(CC1)OC2 N1(C(c2ccccc2F)=O)CCN(C(=O)CCF)C(c2c(F)cncc2F)C1 C(=O)(C(C)P(C)(C)=O)NC1CC(NC(CCNC(COC)=O)=O)CC1O C1(NC(C(CSC)O)=O)CCN(C(=O)CNC(c2ccc(C)c(C)c2)=O)CC1O C1(C)(C(N2CC(CNC(C(CCSC)(C)C)=O)C(O)C2)=O)CC(C(C)(C)C)=NO1 C1(C(=O)NCC2CC(CC)C2)CCC(C)CN1C(c1ccc(C(N)=O)[nH]1)=O Cn1c(Cl)cnc1C(F)(F)C(=O)NCC1(NC(C2CCCCO2)=O)CCCCC1 C1(C)(C(=O)NC(C)CCN(C)C(c2cccc(=O)o2)=O)CC(C(C)(C)C)=NO1 C1(OC)CC(CNC(c2c(C)ccn2C)=O)N(C(=O)COc2cccc(Cl)c2)C1 N1(C(C(CC)N(C(=O)CC2CSCCO2)C)=O)CC(C2CCCC2)C1 c1(CC(=O)NC(C(CC)C)CC(=O)NC(C)C)c(C)nc2cc(O)nn2c1C c1(CC)c(C(=O)N(CCN(C(=O)CCOCCO)C2CC2)CC)nnn1C c1(-c2nn(C)c(C3CCCN(C(C4(F)CCOC4)=O)C3)n2)cc(F)cc(F)c1 C(=O)(C(=O)C(C)(C)C)NCC1C(C(CCNC(Cc2cc(C)on2)=O)(C)C)C1 C(=O)(C1c2c[nH]nc2CN1C(=O)CC1CC(C)(C)CO1)NC(CC(=O)OCC)C C1(NC=O)CCc2n[nH]cc2C1.N1(C23CC(CC)(C2)C3)CCC(F)(OC(C)(C)C)C1 c1(C(N2CCC(C3N(C(c4cc(C)ns4)=O)CCC3)C2)=O)cccc(C(N)=O)c1 N1(C(C(CC=C)NC(C)=O)=O)CCN(C(=O)C=C2CCC(C)C2)CC1CCO C1(NC(C#CC(C)(C)C)=O)COC2C(NC(=O)CCc3n[nH]c(=N)s3)COC12 N1(C(CNC(c2ccc(OC)cc2)=O)=O)C(CNC(=O)C(C)O)CC2COCC12 C(=O)(C1OC(=O)c2ccccc21)N(CC(C)(C)NC(c1ccc(OC)cn1)=O)C c1(C(CC)C)ccc(C(=O)NC(C)CCCNC(=O)CNc2nccs2)c(O)n1 N1(C(C(CCCC)NC(N)=O)=O)CCC(NC(C2CCCSC2)=O)C(CO)CC1 Cc1cc2c(cn1)C1(CCCCC1)C(C(=O)N(C)CCCCl)O2 C12(NC(C(C3CC3)SC)=O)CCCCCC1N(C(c1cc(C)cnc1N)=O)CC2 C1(C(=O)NCCCCN(C(c2cn(CC)nc2)=O)C)CCC2(CC2)C1 C1(CNC(C(C)(Cl)Cl)=O)CN(C(=O)CCNC(c2ccco2)=O)CC12CCC2 C(CC(=O)NCC(CC)NC(=O)CCC1CC1CC)OCCOCC C(=O)(C1=CCCCC1)N1CCC(C(C)C(=O)N(C2CCOCC2)CCF)CC1 c1(C(N2CCC(CCF)C2)=O)cc2scc(Br)c2[nH]1 C1(C(=O)NC(CN(C(C2SCCCS2)=O)CC)C)CN(C)C(=O)CCO1 c1(C(N2CCC(C)C2)C(=O)NC)nccn2nccc12.C12CCCCN1CCN2 N1(C(CC2ON=C(C)C2)=O)CCC(CC(C)NC(c2occc2F)=O)CC1 C(=O)(CCC(F)C(=O)NCc1nsc(N2CC(CCO)OC(C)(C)C2)n1)OC Cc1cc(C(N2CC3(CCN3C(=O)C(O)CN3CCCC3)C2)=O)c(S(N)(=O)=O)s1 C1(C(=O)NCCCCCNC(C(c2cncc(F)c2)C)=O)CCC(CO)CC1 C1(C(C(c2cccc(F)c2)CCCC2CC2)=O)CCC2(CCc3ccccc32)CC1 N1(C(C(C)(O)CN(C)C)=O)CC2(CCCN(C(=O)C(O)Cc3cnc[nH]3)C2)C1 Cc1c(C(=O)NCCOCCN(C)C(C2CCCC2O)=O)cccc1Br c1(CCNC(C(C2CCOC2)NC(C(C=CC)O)=O)=O)cccnc1F C1(C(N2CCN(C(=O)C3CC3)CC2)=O)CC12CCN(c1nnc3ccccn13)CC2 C1(NC(C(C)OCCOC)=O)CC2C(NC(c3cc(SC)c(C)o3)=O)C2C1 N1(C(=O)C=CCF)CC2C3CCC(C2C1)N(C(c1cc(O)cs1)=O)C3 CN1CCc2[nH]nc(C(=O)NCC34CCC(CC3)N4C(=O)C=CBr)c2C1 N1(C(C2(C(F)(F)F)CC(=C)C2)=O)CCC(CCOC)(NC(=O)C(=O)NCC)C1 CC(C)CC(C(=O)NC1CCN(C(c2csc(C(N)=O)n2)=O)C1(C)C)C(N)=O S(=O)(=O)(c1cccnc1OC(F)F)C(=O)OC(C(C(=O)OC)C)C CCCCCCCC(=O)NC(CC)CCCC(=O)NC(CC)C(C)CN(C)C c1(C(=O)NC2CN(C(COCC)=O)CC3(C2)CC3)ccc2c(c1)nnn2C Cc1n[nH]c(C)c1C(C)NC(=O)COCC(C)(C)NC(=O)CC(C)(F)F N1(C(C2CCCN(Cc3c(C)nns3)C2)=O)CCC2(CC1)CC(C)(O)C2 CC1(C(N2CC(NC(c3cc(N(C)C)ccn3)=O)C2)=O)CCC(=O)N1 S(=O)(=O)(c1csc(C(F)F)c1)NCC1CCCN(c2c(OC)cccc2)C1 C1(CN(C)C(C2CCSC2)=O)CCCC(NC(C2CC(O)C2)=O)C1 C1(NC(C(N2CCC3CCC23)(C)C)=O)CCCCCC1C(c1csc(=N)[nH]1)=O c1(C(=O)NCCN(C(c2cncc(N)n2)=O)CC)ccc(Br)c(F)c1F c1(C(N2CCC(C)C2c2cn(CC3(O)CCC3)nn2)=O)c(F)ccc(F)c1Cl c1(N(C)C)ccc(C(N2CC(n3cc(CCO)nn3)C(O)C2)=O)cc1F N12CCC3CCN(CC13)CCCN(N(C)C)c1cccc(c1)C(OC)C2.C(C)SC N1(C(CC(C)(F)F)=O)CCCC(C2CCCN(C(=O)CCc3cncs3)C2)C1 c1(C(=O)NC23CN(C(c4cccc(OC)c4)=O)C(C2)C3)c[nH]c2nccc-2c1 C1(CNC(C(CCC)(C)C)=O)CN(C)CCN(C(=O)CC2CC(C(C)(C)C)C2)C1 Cc1cc2[nH]c(C(=O)NCCC3CCCN3C(=O)CCc3ccco3)cc2s1 c1(CCC)ccc(CC(=O)NC2CCC(Nc3nccc(OC(C)C)n3)C2)cc1 C(CCCCCCSc1cnn(C(C)C)c1)NC(N(C)Cc1cnc(C)s1)=O N1(CCCNC(C2(C)CC(=C)C2)=O)CCN(C(C2CC3CCC3C2)=O)CC1 C1(NC(C2CCN(CC)C2)=O)CC2CC(NC(C3(CC)CCC3)=O)C2C1.CCO N1(C(c2c(C)cc(F)c(Cl)c2)=O)CCC2(CC1)CCN(C(C13CC(C)C1C3)=O)C2 N#Cc1c(NC(=O)CCCCC2CCSS2)cc(Br)cc1F.c12ccc([nH]1)NC2 C(=O)(C1=CCCN(C(C2(C)CCC(=O)C2)=O)C1)NC1CN(C)C(C)(C)C1 N1(C(C(C(C)(C)C)=O)=O)CC2CC(C(=O)NC3(C4CC4)CC3)C(C2)C1 C=CC1(O)CN(C(=O)CCN(C(=O)C=CC2(C)COC2)C(C)C)C1 c1(CNC(=O)NC2CCC(NC(C(N3CCCCC3)C)=O)C2)ccc(F)cc1 CC1OCCCC1C(=O)NC1CC(NC(c2cc(N3CCCCC3)ncn2)=O)C1 c1(C(N2CCC(C(=O)NCC)CC2)C(=O)NCCCCCC)nn(C)c(Cl)c1Br c1(CN2C(CCC)CN(C(=O)C(C)C)CC2)ccc2n[nH]c(C)c2c1 CCC(C(=O)NC1(CCNC(=O)Cc2ccccc2)CCCC1)n1nccc1C C(=O)(C1=NN(C)C(=O)CC1)N1CC(C(C)NC(c2ccc(Cl)cc2)=O)OCC1 c1(NC(C2(CCCC)CC2)=O)ccc(NCc2cn(C(C)C)nn2)cc1 c1(C(=O)OC)cncc(C#CCNC2CCC(n3cc(C4(C)CC4)nn3)C2)c1 CCC(C(=O)NC1(CNC(=O)C(O)CC2CC2)CC1)C(C)O CCC(CC)CCC(=O)N(C(C)CCNC(c1cc(C(F)F)ccn1)=O)C c1(CC(=O)NCCCCN(C)C(C2(C)CC(F)C2)=O)cc(F)ccc1F C1(NC(CC(CC)NC(c2c[nH]ccc2=O)=O)=O)CCc2nncn2C1 CCC(C)CCCCC(=O)NCC1(C)CC(F)(F)CN1C(c1cscc1OC)=O C(=O)(C(CC)C(C)(C)CC)NC1C(C(N2CC3(CC(=C)C3)C2)=O)C1(C)C c1(CC(=O)NCC2CC2NC(=O)COC(F)F)ccsc1Cl CCC(C)C(O)CC(=O)N1CCCC1(C)C(=O)NCCNC(=O)N(C)C(C)C N1(C(CCN(CC#C)C(c2ccc(C#C)cc2)=O)=O)CCc2ncsc2C1 N1(C(C(COC)O)=O)CCC2(CC(NC(C3CCC(C4CCC4)CC3)=O)C2)C1 c1(CC(N2C3CC(CNC(=O)CCc4cnn[nH]4)C2CC3)=O)ccc2nc[nH]c2c1 c1(NCc2c3cc(C)[nH]c3ccc2)nc(=NCC2(C)CCCO2)[nH]c2c1CCC2 C(=O)(C(O)CC(N)=O)NCC(C)NC(c1cc(-n2ccnc2O)ccc1Cl)=O C1(c2nnnn2CCOC)(NCc2cnn(CC)n2)CCSC1C c1(CC(=O)N(C2CN(C(C34CCC3C4)=O)C2)C)ccc(F)cn1 C1(C(N(N(CCCN)C)C)=O)CCN(C)C1=O.C1(C=O)CCOCC1 N(C(=NCCCCl)NCc1c(F)cc(F)c(F)c1F)CC(C)(C)C(F)F N1(C(C)C)CCCC(C(N2CCCCC2C(=O)N(CCO)CCN(C)C)=O)C1 c1(C(N(C2CCN(C(C(CC)CC3CCCC3)=O)C2)C)=O)cn2cccnc2n1 N1(C(CC(C=C)(C)O)=O)CCC2(CC1)CN(C(C1(CN(C)C)CC1)=O)CC(C)O2 N1(C(c2c(C)cncc2)=O)CCN(C(C2CCC(=O)N2C2CC2)=O)C(CCO)C1 C1(C(C(=O)NCCN(C2CCOCC2)C2CCCC2)N(C)C)CCCOCC1 C1(CN)CCN(C(C2(SC)CCC2)=O)CC1C.n1(CCC)ncc(C(=O)N)c1C C1(CC#C)(C(=O)NCC#CCNC(C2CCCN2CCC(F)(F)F)=O)CCCO1 C1(NC(c2n(CC)nc(C3CC3)c2)=O)CC2CN(C(=O)C#CC(C)C)CC12 N1(C(CCC)=O)CCC(c2nc(CSC)nn2CC(F)(F)F)CC1 O=C(CCCF)NCc1cc[nH]c1C(=O)NC(Cc1ccco1)CO C#CCC(C)(C)C(=O)NCC1CN(C(=O)CCCCOC)CC1N(C)C C=C1CN2C(=O)CCC2(C(N2CCC(C)(NC(c3cn(CCO)nn3)=O)C2)=O)C1 N1(C(C(CC)c2ccccc2)=O)CC(NC(=O)CN2CCC(=O)NC2=O)C2CC2C1 N1(C(C(CC)C#N)=O)CC2(CCN2C(c2ccc(C(C)(C)C)cc2)=O)C1 C1(C(=O)NC2C(C)C2C)(NC(c2cc(CO)on2)=O)CCC(C)(C)C1 c1(CN(C(=O)NCC(COC)C(C)C)C)c(C)cccc1F N1(C(C(C(C)C)OC(=O)CC2CCCN(S(C)(=O)=O)C2)=O)CCCCCCC1=O C1(N(C)C(C2CCN(C(c3ccc(Cl)cc3)=O)C2)=O)C2CCC1(C)C2(C)C CCCC(C(=O)OC)C(=O)NCC#CCNC(=O)C(c1ccn(C)n1)C C(CCC(=O)NOC1CCOC1)(C(C)C)NC(CC(CC)COC)=O C12(C(=O)NCC(C)NC(C3(O)CC(C)(C)C3)=O)CCC(C)(CC1)CO2 CCC(C)CC(C)C(=O)NC(C)(CNC(c1ccc2ccnn2c1)=O)C1CC1 N1(C(c2nn(C)c(Cl)c2)=O)CC2=C(C1)CN(C(c1ccnc(C3CC3)c1)=O)C2 N1(C(c2cc(CSC)c(F)cc2)=O)CC(C)C(NC(C2(C)COC2)=O)C(C)C1 N1(C(c2cccc(OCC)c2)C(=O)NCCCSC)CC(C)c2ncccc21 N1(CCCC)CCCC(N(C)C(c2cc(C)c(Cl)s2)=O)CC1 c1(C(=O)NCCN(CC(C)O)C(c2ccc(Cl)s2)=O)ccc(C(C)(F)F)cn1 Cc1ncc(C(N2CC(NC(C34CCCCC3C4)=O)C(CC3CC3)C2)=O)cc1N N1(c2nc(C)cc(C)n2)CC2CCCC(NC(=O)C(N3CCCCC3=O)C)C2C1 c1(N(C(=O)CC2COCC(C)(C)O2)CC)cc(CC2CCCN2C(N)=O)nc(Cl)n1 N1(C(CS(CC)(=O)=O)=O)CCC2C(CCCN2C(=O)CCP(C)(C)=O)C1 C(C)(CCC(=O)NC1(C2CCCCN2C(c2n[nH]c(C)n2)=O)CC1)SC n1(C(C)C)nc(C(F)(F)F)cc1C(=O)NCCNC(C1C2CCC(=O)C12)=O C(=O)(C(C)(C)CS(C)(=O)=O)NCC(C(C)C)NC(=O)C(c1ccc(F)c(F)c1)C N1(C(C2(NC(c3cccs3)=O)CCOC2)=O)CCCN(C(C23COCC2C3)=O)CC1 C1(NC(C2CC(SC)C2)=O)CN(C(c2cc(CO)n(C)n2)=O)C2(CCOCC2)C1 c1(C(=O)NC2CCC(C)N(C(C3CC3(Cl)Cl)=O)C2)cccc(N=[N+]=[N-])c1 C(=O)(CCCC(F)(F)CO)NC(CCN(C)C(c1cccc[n+]1[O-])=O)C(C)(C)C C(C)(CCC#N)(c1nnnn1C1CCC1)CCOCC(=O)NC(C)C C1(CC)CC(F)CN(c2ncncc2I)C1.c12sc(C)cc1N(N1CCCC1)C2=O C1(C(=O)NCC2=CC(=O)N2C)(CC)COC1.C(C(=O)NC1CC1)=C.C1CC1 c1(C(=O)NC(COC)C(=O)N(CC(C)(C)C#N)C)cc(C)c(C)cn1 Cc1ccc(NCC2(Br)CC2)cc1-n1nnnc1C(c1cc(F)cc(Cl)c1)NC C12(C(=O)OC)CCC(NC(C)CC(O)c3cccs3)(CC1)CC2 Cc1ccc(CC(N2CCCC2(C)C(N2CCOC(C#N)C2)=O)=O)cc1[N+](=O)[O-] c1(N2CCCC(CSC)C2)ncc(S(=O)(=O)NC2CCSCC2)cc1Cl CCCC(C)C(=O)N1CC(O)CC1CO.c1(N2C(=O)C2)ccc(C(C)=O)cn1 Cc1c(NCc2ccc(-c3cc[nH]n3)cc2)ncnc1NC1CCOC1C C1(CNC(CCOC(C)C)=O)OCCC1C(=O)N(C1CC1)Cc1cncs1 N1(C(c2c(C)oc(CNC(=O)C(C)CC3CC3)n2)=O)CC[Si](C)(C)CC1 N1(C(CN2CC(CC)C2)=O)CCC2(CCN(C(C3(F)CC3C)=O)CC2)C(C)C1 c1(C(=O)NCCC(C)N(C(C2=CC(C)CC2)=O)C)ccc2oc(O)nc2c1 C(=O)(C(C)CC(C)(C)C)N(C)CC1OCCN(C(CCc2c(C)noc2Cl)=O)C1 O=C1NC2CCCC1CN(CC(=O)NCc1ccc(-c3ccccc3Cl)nc1)C2 CC1(C)CCCN(C(c2cc(C3CC3)on2)=O)C1C(N1CC2CCC(O)C2C1)=O Nc1cc(Cl)ccc1C(N1CC=CC(NC(C2CC(C3CC3)=NO2)=O)C1)=O C=CCCC(F)(F)C(=O)NC1CCCCCN(C(c2cc(C(C)C)oc2C)=O)C1 N1(C(c2nc(Br)c[nH]2)=O)CCN(C2CCN(C(C3CCOC3)=O)C2)CC1 C(=O)(CCC(C)C)N1CCC(C(C(=O)NC(c2cncc(C)c2)CC)F)C1 c1(CCCC(=O)N2CC(OCCN(C(c3n(C)ncc3)=O)CC)C2)cccc(F)c1 N1(C(C2CC(=C)C2)=O)CCC(C(N2CCCCC2C(=O)NC)=O)(CC)C1 C1(NC(c2ccncc2O)=O)CC2CCC(C1)N2C(C1CC2CCC(C1)C2F)=O Cc1cc(NC(=O)CCN(C)CCO)ccc1NC(c1cncnc1C(C)C)=O C(=O)(CCCC(C)(F)F)NCCC1CCCN(C(CCC(=C)Br)=O)C1 C=C(CNC(C1C2COCC12)=O)CCNC(=O)C(C)Sc1ccccn1 Cc1cc(C#N)cc(C)c1CC(N1CCCCC1CNC(=O)Cc1ccoc1)=O N1(C(CCC)=O)CCC2CN(C(=O)OC(C)(C)C)CCC12.C(CCN(C)CC)N c1(C(=O)NCC(Cc2ccccc2)NC(C=CC(=O)OCCCC)=O)csc(C)c1 c1(C(=O)NC2CC(C(C(=O)N(CCC(C)O)C)F)C2)ccncc1Cl C(CCNC(=O)CN(c1ccncc1)C)(C(C)C)NC(C1N(C(C)C)CCC1)=O C(C)(c1ccc(F)cc1F)=CC(=O)NC1(C(F)F)CC(NC(C(C#C)(C)C)=O)C1 c1(Nc2c(C)c(NC(C)CS(C)(=O)=O)ncn2)cnn2c1OCCC2 C(CN=C(NCCF)NC1CCCC(c2cccnc2)C1)C1(CO)CCOCC1 c1(OC)cccc(C)c1C(N1CC(CNC(c2cc(C)sn2)=O)C(C)C1)=O CC(C)CC(C)(CNC(=O)CC1CC12CC2)NC(c1c[nH]nc1CN(C)C)=O N1(C(CN(C(C)=O)C)=O)CCOC2(CCN(C(c3nccc(C)n3)=O)C2)C1 CC1(C#CC(=O)NCC(C)(C2CCC2)NC(=O)CCOC2CC2)CC1 C1(OC)CCN(C(=O)C(CNC(c2ccc(O)nn2)=O)CC2CC2)CC1(C)C C12(CC)CCC(C(N3CCCN(C(=O)CSCCN(C)C)CC3C)=O)(CC1)CO2 c1(C(N(CC(C)NC(C2C3CC(F)(F)CC23)=O)CC)=O)cc(Cl)cc(Cl)c1O N1(C(C(C(C)C)CN(C)C)=O)CCC(CNC(=O)CS(=O)(=O)CCO)C(F)(F)C1 NS(=O)(=O)c1cc(C(N2CCCC(Cn3cc(-c4cn[nH]c4)nn3)C2)=O)cc(Br)c1 Cc1ccccc1C(C(F)(F)CBr)NC(N1CCCC1Cn1ccnc1)=O Cc1ccn(CC(=O)NCC2C=CC(NC(=O)C(C#N)C(C)C)C2)c(=O)c1 N1(C(CSC)=O)CCCC(Cc2cn(CC(CSc3ncccn3)(C)C)nn2)C1 C(c1cnc2ccccc2c1)=CC(=O)NCC(CC)NC(=O)C(C)(C)c1cscn1 C1(C(=O)OC)CC(C)N1C(=O)C(C1CC1)NC(c1cn(C(C)C)cn1)=O c1(C(N2CC3C(Cn4cc(-c5cn(C)nc5)nn4)(CC3)C2)=O)n[nH]c2c1CCOC2 c1(N2C(C)C(NC(C3CCCN3CC(F)(F)F)=O)CCC2)ccc([N+](=O)[O-])cc1 Cn1oc(C(=O)NCC2(CCNC(C3CC34CCOC4)=O)CC2)cc1=O c1(N(C2COC2)C(C2CC(OCCO)C2)C)cnc(OCF)o1 C1(C(=O)NCC(C(C)C)NC(c2ccncc2O)=O)C2CCN(CC2)S1(=O)=O Cn1cc(CNC(c2scnc2Br)c2nnnn2-c2ccccc2Br)c(I)n1 CCC(C)(COC)C(=O)NCCC1(O)CCCN(C(=O)CCc2ccon2)C1 c1(C(N2CCC(C(C)C#N)CC2)C(=O)NCCOC)ccc2nc(C)[nH]c2c1 N1(C(c2ccn(CCOC)n2)=O)CC2CCC(CNC(=O)CCN(C)C)C2C1 CC(C)C(C(=O)NC1CCN(C(C2CSCC(=O)N2)=O)C1)n1ccnc1 N1(C(C(C=C)C)=O)CCOC(CCNC(=O)Cc2c(C)cnn2C)C1 C12(CNC(C(N3CCN(C)CC3)C)=O)CCC(CN(C(=O)COCC3CC3)C1)C2 C12CC13CCN(CC3)C(=O)COC2=O.c1(C2C(C(C)(F)F)C2)ccccc1 c1(C(=O)NCC2CC(NC(c3ccc(C(N)=O)[nH]3)=O)C2)ccc2cnccc2n1 C1(CCNC(CC(=C)C)=O)CN(C(c2ccc(C)c(Br)c2)=O)CC(C)O1 CC(C)CC(F)(F)C(=O)NCCN(C(c1cc2n(c1)CCCC2)=O)C(C)C C(=O)(C(C)(C)C(N)=O)NC.c1(C(C)C)ncsc1C(=O)NCCC(C)N C(CCN=c1[nH]c2ncc(Cl)cc2s1)N(C(C(CC=C)C)=O)CC1CCCC1 N1(C(c2cnccc2OC)=O)CCCC(C(C(=O)O)OC)(C(F)(F)F)C1 C1(Nc2nc(C)nc(Cl)c2)CC2CC(C1)N(C(=O)C#CC1CC1)C2 C1(C(=O)NCC(C)NC(C2(C)CSC2)=O)CCc2nncn2CC1 c1(C(=O)NCC2(C)CCC(C)CC2)ccc(S(N)(=O)=O)c(Cl)c1 C1(NC(C2(C)C=CCCC2)=O)(CNC(c2cn[nH]c2)=O)CCC(F)(F)CC1 N1(C(C(CCC)O)=O)CCCC2CN(c3nc(C(F)F)nc(=N)[nH]3)CCC12 CC1=NOC2(C1)CC(C(=O)NCC1C(C)CCN1C(n1ncc(C#N)c1N)=O)C2 c1(CC(=O)NC)cc2cc(C(=O)OCCC(C)(C)C#N)ccc2[nH]1 C1(CNC(=O)C=CC=C(Cl)Cl)CC2CCC1N(C(=O)CCc1cccs1)C2 c1(OC)ccccc1C(C(=O)NCC1(NC(c2nn[nH]c2Cl)=O)CCOC1)OC c1(CC(=O)NCCCNC(c2c(C)n(C(C)C)nn2)=O)cn2c(C)cncc2n1 N1(C(c2c(SCC)cccc2)=O)CCCN(C(=O)C(F)C(C)(C)O)C(C)C1 C=CCCCCCCC(=O)NCCC1CC(NC(=O)C(C2(O)CCCC2)F)C1 C1(C(=O)NCC2CC(C(=O)NC3(CCCF)CC3)CO2)CC2(C1)CC2(F)F C(=O)(C(C(C)(C)C)OC(C)=O)NC1CN(C(CNC(=O)OCC)=O)C1(C)C C=CC1(C(=O)N=c2ccn(CC)[nH]2)CCN(C(c2cccnc2)=O)CC1 c1(C(N(C(CC(N2CC(CCC)OCC2)=O)(C)C)C)=O)cc(=O)n(C)cn1 CC1CC2(CCN(C(C3CNC(=O)CN3C(=O)CCCn3ccnn3)=O)C2)CO1 c1(C(=O)NC(CCOC)CNC(c2cscn2)=O)cc(COC)oc1C CC1C(NC(c2cnn(C)c2N(C)C)=O)CCCN1C(=O)C(C)Sc1ccccc1 c1(N2CCC(CC=C)C2)nc(=NCC2Cc3ccccc32)[nH]c2cccnc12 C1(N(C)C(c2ncsc2C(F)(F)F)=O)CCCN(C(=O)C(c2ccccn2)O)C1 c1(C(C(N2CC(C)(NC(c3cn(C)c(O)n3)=O)C2)=O)OC)cc(F)ccc1F N1(C(C(C)(C)SC)=O)CC2CCCCC2(CN=c2nc(C)[nH]s2)C1 C(C(COC)C(=O)NCCCCCCN(C(=O)CC1SC(=N)NC1=O)C)OC c1(C(N2CCC(C3CCCN3C(=O)Cc3cc[nH]n3)C2)=O)ccc(O)c(F)c1 CC1CCCN(C(=O)C(=O)NCCNC(c2nc(Cc3cn[nH]c3)no2)=O)C1 CC1CCN(C(=O)CCCCC2CC2)CC1NC(=O)Cc1cnoc1 CON1CCC(C(=O)NC(C)CCCCNC(c2ccc(C#N)cn2)=O)CC1 c1(OC)cccc(C(=O)N(C)CC2(C)CCCC2NC(C2CCOC2)=O)c1F C1(C#N)(C(=O)N)CCCOC1.c1(CC(=O)NC(COC)(C)C)nncn1C(C)C C1(CCCNC(C(C)SCCCC)=O)CCCN1C(=O)C(C)n1ccnc1 C1(OCC)CCC(C(=O)N(C(CNC(=O)C(c2ccnn2C)C)C2CC2)C)CC1 CC(CNC(c1cncn1C1CC1)=O)CC(=O)N1CCC(C)(CO)C1 C(=O)(C1=C(C)OCCS1)N1CCN(C(CCSCCCC)=O)CC1CCC C#CCC(C(=O)NCc1ccn(C2CC2)n1)NC(=O)CC1CCCNC1=O N1(C(c2c(C(C)C)onc2)=O)CCC(N(C(=O)CSc2cnn(C)c2)C)C(C)C1 N1(C(C2(OCC(=O)NCC)CCC2)=O)CC2CC(O)C1C2NC(=O)CC(C)C C1(CNC(CC2C(CNC(CCCOC(C)=O)=O)C2)=O)CCOC1(C)C CC1COc2c(C(N3CCC(F)(CNC(C4CCC4)=O)C3)=O)cnn2C1 C1(NC(C2N(C(c3ncn(CC)c3)=O)CC=CC2)=O)CC=C(C(C)C)CC1 N1(C(c2ccc(CC)cc2)=O)CCC2CC1CN(CC#CCN(C)C)C2 C=CC(C)(O)CC(=O)NCCOCC(=O)N(C1CC(SC)C1)C CN1CC(F)CC1C(=O)NCCC1CCCN1C(=O)C=Cc1ccccc1 c1(C(=O)NCCC(C)N(C(CCc2scc(C)n2)=O)C)cnc2sccn12 Cc1nc(NC(C2CSCCN2Cc2ccc(O)c(I)c2)=O)c(C#N)n1C O=C(CC1=CCCCC1)NC1CC(CCNC(C2CCCCC2C2CC2)=O)C1 CCCCC(C(=O)N1CC(C(N)=O)(N(C)C)C1)NC(=O)C(C(=O)OCC)OC C(=O)(C1=COc2ccccc2O1)NC1CC(NC(CCNC(=O)NC)=O)C1 c1(OCCC(=O)NCC2C(NC(C(CC)OCC)=O)COC2)ccc(C)c(C)c1 Cc1ccc(C#N)cc1C(=O)NC1C2CC(NC(C3CC4CCC4C3)=O)CC12 c1(C(=O)NC(C(=O)N(C)CC)C)cc(CNC(=O)C=Cc2cncs2)no1 C=CCC(C)(C)CC(=O)N1CCC(C2CCCN2Cc2ccc(CCC)s2)C1 CC1(C#CC(=O)NC2CC3(C(=O)NCCS(N)(=O)=O)COC2C3)CCCO1 C1(Cl)(C(N2CC(C(N)=O)(CNC(C3CCCC3F)=O)C2)=O)CC12CCC2 c1(C(=O)NC(C)CNC(c2csc(-c3nc[nH]n3)n2)=O)cnc(Cl)c(N)c1 c1(C(=O)NC2CC3CN(C(Cn4c(C)cnn4)=O)CC32)ccnc2c1CC(=O)N2 c1(CNC(C(CC#C)(C)C)=O)nc2c(s1)CN(C(c1cccn1CC)=O)CC2 CC1CC(C(=O)NCC2CN(C(=O)CCCNC(=O)C3CC3)C2)CO1 C1(NC(c2cn(CC)nn2)=O)(CNC(=O)CSc2n[nH]c(O)n2)CCCCC1C CC(=O)CC(C)(C)CC(=O)NC(CNC(c1ccc(Cl)cc1C)=O)C1CC1 C1(N(C(=O)C=Cc2cccs2)CCC)CCN(C(C2C(C=CC)C2(C)C)=O)CC1 c1(OC)ccc(C=CC(N2CCC(NC(=O)Nc3c(F)cccc3I)C2)=O)cc1 C1(CCNC(c2[nH]cc(C(N)=O)c2)=O)CCCCN1C(=O)Cc1cccc(Cl)n1 N1(C(CN(CCC)C)=O)CCC2(CC1)CC(C)N(C(C1CC3CCC3C1)=O)C2 N1(C(CC=C(C)C)=O)CCC(NC(C2CCCN2C2CCCC2)=O)CC1C c1(OC)c(Br)cc(CNC(=O)CC2CCN(c3nccc(C)n3)CC2)cc1Br CC1CCC(C(=O)NCC2(C3CC3)CC2)CN1C(C1(C(N)=O)CC1)=O N1(C(CCCOCC=C)=O)CCC(NC(C2OCC23CCC3)=O)C12CCC2 C1(C(N(C(CN(C(c2cncc(OC)n2)=O)C)C)C)=O)CC2C(C1)C2(F)F CC#CC1CCN(C(C2(C3CCCN3C(=O)Cc3cnccn3)CC2)=O)C1 Cc1nc2c(o1)CCN(C(C1CCC(C)C1)=O)C2 C1(N(CC#C)C(C2CCC(=O)N2C)=O)CCN(C(c2cccnc2NC)=O)CC1 C1(CNC(c2c(C)nc(CCC)o2)=O)CN(C(=O)CC2CCCSC2)CCN1C N1(C(C=C(C)C2CC2)=O)C2CCC(C2)C1NC(=O)OC1(C(=O)N(C)C)CC1 c1(C(=O)NC2C=CC(CC(N3C(C(=O)OC)C(C)CC3)=O)C2)cc2cccnn2c1 c1(C(N(C)CC2(NC(=O)C(CO)C(C)(C)C)CC2)=O)cccc2ccoc12 C(=O)(C1=NNC(=O)CC1)NC1C2CN(C(c3cc(CC)c(OC)cc3)=O)CC21 N1(Cc2cccc(OC)c2)CCC(O)C(C(=O)Nc2cc(OC)ccc2I)C1 N1(C(C2(OC)CS(=O)(=O)C2)=O)CCCN(C(c2ccc(F)c(C)c2)=O)CC1 C1(C(CC)NC2CCNC(C)(C)C2)Cc2ccccc2C1C c1(C(=O)OC)ccc(CNC(C2CC2NCC2CC2(Cl)Cl)=O)nc1 C1(NC(C(C)OC(C)=O)=O)C2CC3C1C3C2C(=O)NCc1nc(C)c(C)[nH]1 c1(OCCNC(=O)NC(c2ncccn2)CC)ccccc1O N1(C(=O)COCC2CCC2)CC(O)CC1C(=O)NC1C2CCC1CC2 C(=O)(C(C)(C)CN(C)C(C1CCCCO1)=O)N(C)Cc1c(C)nco1 c1(C(=O)NCc2ccc3occc3c2)n[nH]c2ccc(-c3ccnc(F)c3)cc12 CC1(C)CCC2(C1)C(=O)CC(=O)N2.c1(COCC2CCC2)nc(C2CC2)n[nH]1 CN1CCCCC(C(=O)NCC2CC3CCC2N3C(C2CCCCN2C)=O)C1=O N1(C(C)(C)C)CCCC1C(=O)NCCNC(=O)CC1CC1 c1(C(=O)NCC#CCNC(C2(C)CCNC2=O)=O)n[nH]c2c1CCC2 CC(C)(C#Cc1cn(Cc2csc(Br)c2)nn1)NC(=O)CC1CCCCC12CC2 N1(C(C(C)(C)OC)=O)CCC(C2CN(C(=O)C(CO)C(F)(F)F)C2)CC1 CCCCCCC(=O)NC(CCCOC)C(=O)N(C1CCC1)C1CCC1 C(=O)(C(C)(C)C(=O)OC(C)(C)C)NCC(C(=O)NCC1ON=C(C)C1)C N1(C(C2CC(=C3CC3)C2)=O)CC(O)(C(F)C(=O)NC2C(O)CC2O)C1 C1(NC(c2cc(OC)no2)=O)C(C)CCN(C(c2cc(C3CC3)no2)=O)C1C N1(C(C2(COCC)CC2)=O)CC2CC(C1)CN(C(c1coc(O)n1)=O)C2 n1(Cc2ccc(C(=O)NCC3CCC(C)NC3)cc2)cnc2ccccc12 N1(C(CN(C)CCO)=O)CC(N(C)C(C2CCCC(=O)N2)=O)C(F)C1 c1(Nc2[nH]c(=NCc3ccncc3C#N)cc(C)n2)ccn2c1CS(=O)(=O)CC2 N1(C(C(C)SC(C)C)=O)CCC(NC(=O)C(F)(F)CN2CCOCC2)C1C N1(c2cc(F)nc(I)n2)CC2C3CCC(CC3)C2C1 c1(OCCC)cc(NCC2(CNC(c3ccc([N+](=O)[O-])o3)=O)CC2)nc(C)n1 N1(C(CCCNS(C)(=O)=O)=O)CCOCC1CNC(=O)C(c1ccccc1)C1CC1 c1(CC)cc(N)c(C(=O)NCC(C)(O)CNC(c2cn[nH]c2)=O)cc1F C1(Cl)(NC(COC(CSC(C)C)=O)=O)CC1C(C)=O C1(C(C)(C)NC(C#C)=O)CCN(C(=O)CC2CCCN2Cc2ccsc2)CC1 c1(C(=O)NCC(CNC(CCCCC#C)=O)(C)C)cc(C)c(OC(F)F)c(C)c1 CC(=O)CCCC(C)C(=O)NCC1(C)CCN(C(C2CCN(C(N)=O)CC2)=O)C1 C1(NC(c2cc(C)c(Cl)s2)=O)CN(C(c2ccc(C#N)c(C)n2)=O)CC1N=[N+]=[N-] C(=O)(CCC(F)F)NC1CC(CNC(CC=CCC)=O)C1 Cc1ccc(N2C(=O)CCC2C(=O)NC2CC2NC(c2ccncc2Cl)=O)cc1 CC1(CNC(c2cccc(CN=[N+]=[N-])c2)=O)CCN(C(C2CCCC3CC23)=O)C1 Cc1scnc1C(=O)N(CCCNC(C1(Br)CC1)=O)C N1(C(N(c2ccccc2)CC)=O)CCC(C)CC1CSC1CCC1 C=CCCCCCC(=O)N1CCC(NC(=O)CCCN2CCCC2)CC1 C#Cc1cc(C(=O)N(C2C3CN(C(c4cnco4)=O)CC23)C)cc(F)c1 N1(C(c2c(C#N)scc2)=O)CCC2CC2(NC(=O)C2=COCCO2)CC1 CC1CN(C(=O)CC2(NC(=O)C=C3CCCCC3)CC2)c2cccnc21 C(=O)(C(C)S(C)(=O)=O)NC(CC(C)C)CNC(=O)C(C)Oc1ccccc1 c1(C(=O)NCC2(CNC(C(C(C)C)CN(C)C)=O)CCC2)cccc2c1COC2 N1(CC(C)OC)CCOC(C)(CNC(C2CCCSC2C)=O)C1 C1(CNC(c2cc(C3CCC3)on2)=O)CCCN(C(=O)C=CC2CC2)C1 C1(C(N2CCCCC(CO)C2)=O)CCN(C(c2ccc(CO)nc2)=O)C12CC2 CC1(C)CCC(O)(C(=O)NC2CC(CNC(=O)CSc3nc[nH]n3)C2)CC1 N1(C(CC(C)(C)OC)=O)C(CNC(=O)C(C)(C)C(C)(F)F)CC2COCC12 C1(CNC(Cc2c(C(C)C)cccc2)=O)COC(C)(C)CN1C(=O)C=CC1CC1 CN1C(=O)CCC1C(=O)Nc1n[nH]cc1NC(=O)C(C1CCCCC1)O C1(C(NNC(C2C(N)C(O)CC2)=O)=O)CCn2c(O)nnc2C1 C(=O)(CS(=O)(=O)C(C)(C)C)N1CCCC(N(C(=O)CC2C=CCC2)C)CC1 c1(CCNC(=O)NC2CN(C(=O)OC(C)(C)C)CC2O)c[nH]c2cnc(Cl)cc12 N1(C(C(C)O)=O)CCC2CN(C(c3c(F)c(F)ccc3F)=O)CC2C1 C#Cc1ccc(C(=O)N(C2CN(C(c3csc(CC)n3)=O)CCC2C)C)cc1C C1(C)(C(=O)NCC=CCCOC)CCN1C(=O)CCOC(C)C CN1CCC(C(N2CC(N(C)C(c3cscn3)=O)C(C)(C)C2)=O)S1(=O)=O C(=O)(C(CCc1cnn(C)c1)N(c1cccnn1)C)NCCOCC C12(CCC)CCN(CC1)C2=O.c1(CNC(c2ccccc2)=O)cccc(CO)n1 c1(C(=O)OC)cc(C(=O)NC2CC23CC(NC(=O)CS(C)(=O)=O)C3)cc(F)c1 C1(C2N(C(CNC=O)=O)CCC2)CCCN(C(c2ccc(O)nc2)=O)C1 N1(C(C2CCC(C(N)=O)CC2)=O)CC(C2CN(C(=O)C(F)n3cccn3)C2)C1 CC1CC(CNC(C2CCN(C)C2)=O)CN(C(=O)C=CCN2CCCC2)C1 c1(C(N(C2CNC(c3n[nH]c(=N)[nH]3)C2CC(CC)CF)C)=O)csc(C2CC2)n1 c1(C(N2CC(C=C)C(NC(=O)CCCC#N)C2)=O)c(C)cc(C)oc1=O CC(CNC(c1ccn(CC(F)F)n1)=O)(CO)NC(C1CS(=O)(=O)C1)=O CCCCC(O)CC(=O)NC1CCCCN(C(=O)CSc2nc[nH]n2)C1 CCCCC(O)C(=O)N1CCC(COC)(NC(c2cc(O)nc(N(C)C)n2)=O)C1 c1(C(N2CCCC2)=O)nnn2c1CN(C(c1nc3ccc(C)cc3[nH]1)=O)CC2.CN N#CC1(C(N2CC3CC3(CNC(=O)CCC3CCC3)C2)=O)CCCOC1 c1(C(=O)NCC2(CNC(CN(C)S(N)(=O)=O)=O)CC23CCC3)cc2ccsc2n1C N1(C(CSSC)=O)CCC2(CCCN2C(=O)Cc2cnccn2)C1 c1(C(=O)NCC(N(C(C(C)SC(F)(F)F)=O)C)C2CC2)sccc1S(N)(=O)=O C1(C(=O)NC(C)CCCCNC(c2cc(Cl)cs2)=O)(CF)CC2(CCC2)C1 C(=O)(C1=CC2CCC(C1)C2)N1CCC(C(=O)NC2CCC(OCC)CC2)C1(C)C c1(OC)ccccc1C(CCNC(=O)CCn1ccc(=N)[nH]1)OC(C)=O N1(C(C2(C(C)C)CC2)=O)CC2CCC(CNC(=O)C(C)(C)C(N)=O)(C2)C1 CCCCCC(O)CC(=O)N1CC(CCNC(C2OC3CCC2C3)=O)OC(C)C1 N1(Cc2c(CC)cccc2)CC2(CN(C(c3ccc(C)nc3)=O)CC2CO)C1 N1(C(C23CC(C(C)C)(C2)C3)=O)CC2CN(C(C3CC3C#N)=O)CC2C1 c1(CN(C(C)C)CC2CCCCO2)cc2c(s1)CCC(C(C)C)C2 C(C(=O)NC(c1cccnc1O)C)(C(C)(C)C)NC(C(COC(C)=O)C)=O N1(C(Cc2c(C)cccc2)=O)CCC2CCCN(C(=O)CN(S(C)(=O)=O)C)C2C1 CCC(C(=O)NC1(CCO)CN(C(c2cc(Cl)c[nH]2)=O)C1)n1cccn1 CC(CC(=O)N1CC2CC2(NC(c2cnc(C3CC3)nc2)=O)C1)P(C)(C)=O CP1(=O)CCN(NC(=O)Nc2c(-n3ccnc3)cccc2Cl)CC1 C1(CNC(CCc2onc(C)n2)=O)CCN(C(c2[nH]ccc2CN(C)C)=O)C(C)C1 CS(=O)(=O)C1CN(CCF)CC1NS(=O)(=O)CC1CCC(F)(F)CC1 c1(CC)c(C(=O)NCC(O)C(C)(C)C)ccn1C.c12nocc1C(=O)N(C)C2C C(CCCCCC(=O)NC1CCCS(=O)(=O)C1)n1cc(C(CC)(C)O)nn1 C1(CC2CC(=O)NC2)CN(N2CCC(C(O)C(F)(F)F)CC2)C1 Cc1ccc(S(=O)(=O)N(c2ccc(F)c(Br)c2)CC2CCN(C)CC2)cc1C C1(NC(=O)Cc2ccc(Cl)s2)C2CC(O)C1N(C(c1ccnc(C3CC3)n1)=O)C2 c1(C(N2CCOC3C(O)CC23)C(=O)NC)cccc2c1CCO2 C1(C(=O)NC2CCN(C(C3CC(C)(CC)C3)=O)C2C2CC2)CCc2c[nH]nc2C1 N1(C(C(CSC)O)=O)CC2CCC1C(CNC(c1sc(C(F)(F)F)nc1C)=O)C2 C1(C2CC2)(C(=O)NC(C)C(C)NC(=O)CN(C)C(c2ccoc2)=O)CC=CC1 N1(C(CC2CCC(CC)O2)=O)CC2CC(CNc3cc4nncn4cn3)CC1C2 C(=O)(C(F)(F)CC)NCC(C)N(C(C1C(CC)C1)=O)C CC(C)CC(O)C(=O)NC1CN(C(=O)Cc2cc(C3CC3)no2)CCC1F C1(C(=O)NCC2C(NC(CCC#C)=O)COC2)COCCC1(F)F c1(C(=O)NC2CCN(C(c3c(C)snc3)=O)C(C)C2)c(F)ccc(N)c1F Cc1cccc(C(N2CCCCC2CCN(C(=O)CC(C)(F)F)C)=O)n1 c1(C(N2CC(N(C(CCC=C)=O)C)C3(C2)CC3)=O)ccc(O)c(C)c1C N1(C(c2n[nH]c(CC)c2C)=O)CC(NC(=O)CN2CCC(C)CC2)CC1(C)CC N1(C(c2ccc(CC)[nH]2)=O)CCC2CCN(C(c3coc(C(F)(F)F)c3)=O)C2C1 C1(N(CCC)C)CCN(C(=O)CCN(C(C2(CC)CCOC2)=O)C(C)C)CC1 c1(OCC)cccc2c1OCC(C(=O)NC(C)C(C)NC(=O)CN(C)C(N)=O)C2 C12(C(=O)NC(CN(C(C=NOC)=O)C)C)CC=CCN1CCC2 C1(CNC2(c3n(CCCC)nnn3)CCOC2)CC2(CCC2)C1 Cc1cn(CC(=O)NC23CCC(CN(C(=O)CC(C)F)C2)C3)c2ccccc12 N=c1[nH][nH]cc1C(=O)NC1CC(CCNC(c2[nH]nnc2C2CC2)=O)C1 CC(C)CCCCCC(=O)NC(C)CCCNC(=O)Cc1ccccc1CC#N c1(C(=O)NC2(COC)CCN(C(=O)C(C)=C3CC3)CC2)n[nH]c2c1CC(C)CC2 C1(C(=O)NC(CNC(C2(CCC=C)CC2)=O)(C)CO)CC2CC1CO2 c1(C(N(CCN(C(C2(C(=O)OCC)CCO2)=O)C)C)=O)ccnc(Br)c1N c1(OCC)cc(OC)cc(C(N2C3CN(Cc4cc(Cl)cc(I)c4)CC23)=O)c1 CCC(C)C(C(=O)NC1CCC(CO)CC1)N(C(=O)C=CCF)C C12(n3cc(CN(C(C(C)Cc4ccco4)=O)C)nn3)CCC(NC(N)=O)(CC1)C2 N1(C(C(CCCC)O)=O)CC2CCCC(C1)N2C(c1scnc1CC)=O C1(OC)CCCN(CCC(=O)N(C2CCCC2O)C)C1 C(=O)(CC1=CCCCC1)N1CCCC(CCNC(=O)Cc2ccsc2Cl)C1 C(=O)(C(CC)C(=O)OC)N1CC(CCC=C)(C(=O)NC(c2nccn2CCC)C)C1 c1(-n2ncc(C(N3CCC(c4cn(C5CCC5F)nn4)C3)=O)c2)ccccc1F CCCCCCCC(=O)N(C)CC1CCCCN1C(c1cnc(C)c(C#N)c1)=O C1(C)CCN(C(=O)CCc2cnn[nH]2)CC1.C(CC(=O)NC1CCC1C=O)=CC N1(C(C(Cc2cc[nH]n2)NC(c2ccc(COC)o2)=O)=O)CC(CO)C1(C)C C1(NC(=O)CC2CC2)CC2(C1)CC(C(=O)N)C2.C(C(O)C(F)(F)F)CCC1CC1 C=CC(F)(F)C(=O)N1CC(O)(CN(C)C(c2c(SCCNC(=O)CC)occ2)=O)C1 O=C1CCCCC(C(=O)NC(CC2CCC2)C(=O)NC2(C(F)(F)F)CCC2)C1 c1(C(=O)NC2C(NC(c3cnc(C)nc3)=O)CCC2)cc(C)c(F)cc1Cl Cc1sc(C(=O)NCc2ccn(CC3CC3)n2)c(C)c1C N1(C(c2cncc(F)c2)=O)CC2CN(C(C34CC=CC(C3)OC4)=O)CC2C1 c1(CCNC(c2n(CC=C)nnn2)c2sccc2C(C)C)ccc2c(c1)CCO2 Cc1ccc(CNC(=NCCC2CNC2)NC(C)C)cc1Br.C(=O)(C1CC1)N CCCCC(C(=O)NCC(C)(C)CNC(=O)C(CCC)N(C)C)NC(N)=O C1(CNC(C(C(C)C)F)=O)CC2(CCN(C(C3C4C5CCC(C5)C34)=O)C2)CO1 CC1Cc2cc(CC(C(=O)NCCCCC(C)(C)SC)N(C)C)ccc2O1 Nc1ncccc1C(=O)NCCn1cc(CNC(c2coc(C3CC3)n2)=O)nn1 C(=O)(CCCC(=O)N1CCOC(C(C)NC(C2CCCC2F)=O)C1)NC(C)C Cc1cc(NC(c2ccccc2C)=O)n(C(C)C)n1.C12CC(C1)NC2=O C(C(=O)NC)(C(C)(C)C)SCCCC.N1CC(CC(=O)OC)CC1CO S(=O)(=O)(c1ccc(NCCc2cnccc2Cl)nc1)NCC(CCCCC)(C)C c1(C(N2CC3C(C(=O)NC(CC)C(=O)NC)(C3)C2)=O)cc(C#N)cn1C N1(C(CC(C)(C)O)=O)CCN(C(=O)C(C)(O)c2ccccc2)CC1c1cn[nH]c1 c1(C(N(CC(O)CNC(=O)CC2(CO)CC2)C)=O)cc(Br)c2nccnc2c1 C1(c2nc(CNC(C3ON=C(C)C3)=O)[nH]n2)CCN(C(=O)C2=CCC2)CC1 c1(-n2c(C(=O)NCC(C3CCCC3)OC)cnn2)cccc(Br)c1 N1(C(CC=C=C)=O)CCCC(NC(=O)CCc2cnn[nH]2)C1 c1(C(=O)NC(CC)CN(C(=O)Cn2cc(C#N)cn2)CC)c(C)nn(C)c1C C(C(O)C(F)(F)F)N(C=O)C(=O)N(c1ccccc1)c1ccoc1 CCN(NC(=O)NCC(C)C(F)(F)F)c1nc[nH]n1 N1(C(COC)=O)CC2CCN(C(c3ccc(F)cc3OC(F)F)=O)C2C1 C(=O)(C1=NN(C)C(=O)CC1)N1C(CC)C(NC(=O)C(O)CC(C)C)CC1 N1(C(c2ccc(C(C)=O)o2)=O)CCC2(CCN(C(=O)C(=O)C(F)(F)F)C2)C1 c1(C(N2CCC(N(C(=O)CCc3nncn3C)C)C2)=O)ccc2oc(=O)oc2c1 c1(C(=O)NCC2N(C(C(C)C)=O)C3C(C2)C3)nc2c(Br)cccn2n1 N1(C(C(C)(N(C)C(C2CCC(O)CC2)=O)C2CC2)=O)CCOC(C2(C)N=N2)C1 CCC(C)(C)C(O)CC(=O)N1CC2(CO)CC1(C(N1CCCCCC1)=O)C2 CC(C(C)(C)C(=O)NCCCC(N)=O)NC(=O)CN1CC(=O)NC1=O C1(NC(CC=C(C)C)=O)CC(CNC(c2cncc(C(F)(F)F)n2)=O)C12CCC2 c1(C(=O)NC2(CNC(C3C(CC)CCC3)=O)CC2)ccccc1Cl CC(C)C(C(=O)NCC1(O)CN(C(=O)C(c2ccc(Cl)cc2)C)C1)C(C)C c1(C(=O)NC(CC)(C)CNC(C2CCCC2)=O)cc(C)c(N)cn1 C1(CNC(C(CSC)O)=O)CC2(CCN(C(c3cn4c(n3)CCCC4)=O)C2)CO1 c1(C(NC(C2(COC)CC(=C)C2)=O)C(C)C)cccc2nc[nH]c12 N1(C(C(COC)C)=O)CCC2CCN(C(c3cc(O)n(CC)n3)=O)C2C1 c1(C(=O)NC2CC(O)(CNC(=O)CC3(CO)CC3)C2)ccc(=O)n2c1CCC2 c1(CC(=O)N(C2CCN(Cc3cncnc3)CC2)CC)ccc(C(F)(F)F)cn1 Cc1cc(=NCC2CC2C2CCCC2)[nH]c(=NCc2csc(Cl)c2)[nH]1 C1(N(C(C(=O)NC(CC)C)c2nccs2)C)CCCCC1O N1(C(c2nc(OCC)sn2)=O)CCC2C(NC(C3CC(SC)C3)=O)CC12 C(=O)(C(CC(F)F)N(C(=O)C(CC)OC)C)NC1(CC=C)CCCC1 N1(C(C(C(C)C)CNC(c2c(C#N)ncn2C)=O)=O)CCCC2(CCCO2)C1 C(=O)(CCCCCNC(c1ccc(OC)s1)=O)NC(CCC)C(=O)N(C)C CCS(=O)(=O)CC(=O)N1CC(F)(C(=O)NC(CC(=O)N(C)C)CO)C1 c1(C(N(C(C)C(=O)NCc2ccns2)CCC)=O)cn(C)nc1OCC C(=O)(C(=O)C(F)(F)F)N1CC(CC(C)NC(CC2C(CC)C2)=O)C1 C(CC(C(=O)NCC(C)CNC(c1ccc[nH]1)=O)N(C)C)SC Cn1ccn2cc(C(=O)NCC34CCC3CN(C(=O)C#CC3CC3)C4)nc2c1=O O=C(C1=CCCSC1)NCC1(NC(c2ccc(Cl)cc2)=O)CCOCC1 C(=O)(C(C)CCC(C)(C)C)NC(C(n1cc(C(O)CSc2ccccc2)nn1)C)=O C1(CNC(C=C(C)C)=O)CC(NC(=O)CN(C(C2CCCCC2)=O)C2CC2)C1(C)C c1(CCC)nc(-c2ccc(-c3cccc(Cl)c3)nn2)n(CC2CCCCO2)n1 C12(NC(c3cnc(CC)s3)=O)CCCC1N(C(=O)CCC=CC(C)C)CCC2 C=CC(C)(CC)C(=O)NCC1CCN1C(=O)CC1(C#N)COC1 c1(OC)ccc(F)c(C(=O)NC2CC2NC(c2c(C)ccnc2O)=O)c1 CN1CC2CCC(NC(=O)CCCOc3ccccc3[N+](=O)[O-])C2CC1 C1(CC(=O)NC2C(OC)CN(C(c3cc(C)nn3C)=O)C2)CCCC(C)(C)CC1 C1(C)(CC)CC(NC(c2cn[nH]c2)=O)CN1C(=O)CSc1ccc(F)cc1 C#CC1CCN(C(=O)COC2CCN(C(c3ccc(C)cc3)=O)C2)C1 C1(C(=O)OC)CC(C(F)(F)F)CCN1S(=O)(=O)N1CCCC(O)C1 CN1CCN(CC(=O)NCC2CCN2C(C2(O)CCSCC2)=O)CC1 N1(C(CC2CCC(C)C2)=O)CC2CN(C(C34CCCC3C4(F)F)=O)CC2C1 c1(C(N2CC(C3CN(C(CC(C)O)=O)C3)C2)=O)cc2n(n1)CCCC2O C(CNC(=O)C(=O)N(CC(F)F)C1CC1)(C(F)(F)F)OC C(=O)(C1=CCCOCC1)NC(CNC(C=Cc1nnc(C(C)C)o1)=O)(C)C S(=O)(=O)(c1ccc(CC(=O)NC2CN(C(C3OCCC3C)=O)CC2O)cc1)NC C1(CC)(NC(=O)CCS(N)(=O)=O)CCN(C(=O)CN(C)S(N)(=O)=O)CC1 CCC(C(=O)OC)C(=O)NCC12CC1CN(C(c1cc(C(F)F)no1)=O)C2 C1(N(C(C(C)SC)=O)C)CCCN(C(C2CC2c2cn[nH]c2)=O)CC1 c1(OC)n[nH]c(C(=O)NC(C)CN2CCN(C(=O)C(C)OC)CC2)c1Cl c1(C(N2CCCC(CC(=O)NC(C3CC3)C3CC3)C2)=O)ccc(F)c(O)c1 c1(CC#N)ccc(C(=O)NC2C3CN(C(C4CCC(=O)N4C)=O)CC23)cc1 C1(NC(c2scnc2C(F)(F)F)=O)CCN(C(C2CC3(C2)CC3F)=O)CC1 C(C(C(=O)N1CCN(C(=O)C(c2ccccc2F)C)C(C)C1)C(F)(F)F)OC C1(NC(c2cc(C(C)C)no2)=O)CCCCCN(C(=O)NCC2CC2)C1 C1(NC(=O)Cc2ccon2)CN(C(=O)CCC2CC2)CC2(CCOCC2)C1 CCCC(C)CCNC(=O)C(c1ccco1)NC(C1OC2CCC1C2)=O c1(C(=O)NCC(C)CNC(=O)CC2CC3(CCC3)C2)cc(Cl)c2n[nH]cc2c1 CN=C(NC1CCCC1)N1CCN(C(c2ccn(C(C)C)n2)C)CC1 C1(NC(CCn2c(C)ncc2)=O)CCCC12CN(C(=O)C(C(C)C)N(C)C)C2 N1(C(=O)NCc2cccc(F)c2)CCC(C)C(F)(F)CC1.Cc1ccc2c(c1)C2 C1(C(=O)NCC=C2CCN(C(CSC)=O)CC2)Cc2nccn2C1 N1(C(c2coc(Nc3cccc(SC)c3)c2)=O)CCNC(=O)c2c(Br)cccc21 C(=O)(C1=NNC(=O)CC1)NCC1C(C)(C)N(C(=O)CC2CCC3CC3C2)CC1 C(=O)(C1=C(NCCN(CCC)C(C)C)CCC1)NC(C12CCC(CO1)C2)=O c1(NC)cncc(C(=O)NCC2CC(NC(c3cncc(C)n3)=O)C2(C)C)c1 c1(C(C)C)ccc(O)c(C(=O)NC(C)C(C)NC(=O)C2=CCCSC2)c1 c1(CC(n2nc(C(N3C4CN(C(C)=O)CC34)=O)cc2C)C)ccc2c(c1)OCO2 c1(N(CC(=C)Br)C)nc(N2CC(C(N)=O)C3(CC3)C2)c2c(n1)CCCCC2 C(=O)(CCC(=O)N(C)C)N1C(C2(O)CN(C(C(C)(C3(C)CC3)OC)=O)C2)CCC1 C1(C(N2C(C(C)NC(C3CC(OC)(OC)C3)=O)CCC2)=O)CC2(CC2)CO1 N1(C(c2nn(CC)c(C)c2)=O)CCC2CC(NC(=O)C#CC3CC3)CCC2C1 C(CCCCCNC(=O)CN1CCCS1(=O)=O)N(C(=O)C1=CCCS1)C C1(NC(=O)NCC(C)OC(F)F)CC2(CNC2)S(=O)(=O)C1 C=CC(C)C(C)C(=O)N(CCCNC(c1cc(OC)ccc1NC)=O)CCO c1(OC)csc(C(N2CC(CNC(=O)Cn3ncc(Br)n3)CC2C)=O)c1OC Cc1ncc2c(n1)CCC(C(N1CCCC1(C)CNC(=O)Cc1cnsc1)=O)C2 C(=O)(C(O)CC(C)(C)C)N1CCN(C(CNC(c2c(CC)n(C)nc2)=O)C)CC1 C(=O)(C(C)(C)CNC(=O)CC1CC1CNC(=O)C(N1CCCCC1=O)C)NCC c1(NC(C2C(CNC(CCCCN(C)C)=O)CCC2)=O)ccc2c(c1)OCO2 c1(C(=O)Nc2nc(C)c(C(=O)NCC3(F)CCC3)s2)cc(Br)ccc1Cl C(=O)(CC(C(F)(F)F)n1ccnc1)NC1CC(C)CN(C(=O)Cc2cc[nH]n2)C1 c1(NC(C(C)Nc2c(C)n(C)nc2)=O)ccnc2cc(Cl)ccc12 C(=O)(C(CCS(C)=O)N(c1c(Cl)cccc1Cl)C)NC1CN(CCOC(C)C)C1 N1(C(c2ccc(CC)cc2)=O)CC2(CC2)CC1CC(=O)NCc1cc(C)ns1 c1(CNC(=O)N(c2ccccc2)CCSc2nc[nH]n2)ccc2c(c1)COC2=O N1(C(CC(C)NC(c2cc(O)cs2)=O)=O)CCC(O)(Cn2ccnn2)CC1 C(N=c1[nH]c2c(c(=NCC3(CN(C)C)CC3)[nH]1)CCC2)c1c(O)nnc(C)c1C CC1(C(N2CCC(n3cc(C(C)(C)O)nn3)C2)=O)CCCCCC1 C(=O)(C(CNC(C1CCCN1C(C)=O)=O)C(C)(C)C)N1CCN(C(C#C)C)CC1 CC1CCN(C(c2ncccc2Br)=O)C1CNC(=O)C(C)(C)c1cnsc1 CCC(C(C)O)NC(=O)C(C)(C1CCC1)NC(C1CC(=C2CC2)C1)=O C#CCCCCCC(=O)N1CCC2(NC(=O)CC(C)(O)C3CC3)CCCC12 Cn1ccc2sc(C(=O)NC3(C)CCCN(C(c4ccnn4C4CC4)=O)C3)cc12 c1(OC)ccc(NC(=O)C(N2CCC(C)(C(C)C)C2)C2CC2)c(C)c1 CCCC(C(C)CC)(c1nnnn1CC1CC1)NCc1cccc(OC)n1 c1(C(=O)NCC2(OC)CCN(C(C3C(=C)C3)=O)C2)ccc2c(c1)NC(=O)C2 C1(O)(CNC(C(CC2CCC2)NC(C(C)Cc2cnco2)=O)=O)CCOCC1 CCCC(CNC(c1cn(CCO)nn1)=O)C(=O)N(C)CCN1CCCC1=O CC1CC(NC(C2(N(C)C)CC2)=O)CN1C(c1cccc(N2CCCC2)c1)=O N1(C(COCCOCC)=O)CCC(C(=O)NC2CCOC2C2CC2)C(O)C1 C1(NC(c2ccc(CNC(C(CSC)C)=O)s2)=O)CCOC1(C)C c1(CC)ccc(NC2(c3n(C4(Oc5ccccn5)CC4)nnn3)CCOC2C)cc1 Cc1ccn2cc(C(=O)NC3CC4CCC3N4C(C3C(C)(C)C3(F)F)=O)nc2c1 c1(CC)cc(=NC(=O)C(N)Cc2c(OC)coc2C(F)(F)F)[nH]n1C C1(C(=O)Nc2c(C)nc(O)s2)CCc2cnccc2C1 C1(C(N2C(CNC(C(COC)(C)C)=O)COCC2)=O)CCC2(CC1)CC(O)C2 C1(Nc2cccc(C(N(c3cccc(Cl)c3N)CC)=O)c2)CN2CCN1CC2C CCC(C)(C)C(C(=O)N1CCC(NC(=O)C(C)(C)c2ccns2)CC1)OC c1(CNC(C(N2C(C#C)CCC2)C2CCC3(CC3)C2)=O)cc2cc(F)ccc2o1 C1(CNC(CC(CC)C)=O)C2CCC1CN(C(c1cccc(OC)c1F)=O)C2 N1(C(c2cc(C(=O)OC)on2)=O)CCOC(CC(=O)N(C)Cc2cncn2C)C1 N1(C(C2(C#C)CC2)=O)CC2COCCC2(NC(=O)Cc2sccc2C)C1 c1(OC)cccc2[nH]c(C(=O)NC3CCN(Cc4cnc(Cl)c(Cl)c4)C3)cc12 C(=O)(C1=CCCN(C(C2CCCCCC2)=O)C1)N1CCCC(CC(C)C)C1 c1(OC)cccc2c1C(C(=O)NC(C)Cc1ccc(-c3ccccc3)cc1)CC2 c1(C(=O)NCC(C(C)C)NC(=O)Cc2cnccc2Cl)cnc2n1CCCCC2 C(C)(CCC#N)(c1n(C(C)(C)C)nnn1)NC(c1ccco1)C C1(C(=O)NCCCN(C(=O)CC2CCCCC2F)CCC)CC2CCC1CC2 C(=O)(CCC(C)(C)F)NCCCC(CO)NC(c1nn(C)c(CO)c1)=O Cc1[nH]nc2c1CCC(C(=O)NC1CCCCCN(C(c3nc(Cl)cs3)=O)C1)C2 C(=O)(C1=CC2(CN(C(=O)Cc3nc(=N)[nH][nH]3)C2)OC1)NCc1ccc(OC)cn1 c1(O)ccc(C)cc1.C1(CC)CNC(C(N2CC(C(F)(F)F)(CO)C2)=O)C1 c1(C(C)NC(c2cnnn2C)c2nnnn2CCCF)ccc(C)s1 C1(CCNC(C=COCC)=O)CCCN(C(=O)C(O)C(C)(C)C)CC1 c1(NC(C(c2ccc(N)cn2)C)=O)cc(N(C)C)ncn1.C12CCCN1C2 C(=O)(C(C)(O)C(F)(F)F)N1C2CC(CNC(CCN(CC(F)(F)F)C)=O)C(C2)C1 C(=O)(CCS(=O)(=O)N(C)C)N(C)CC1CCN(C(c2cc(CC)n(C)n2)=O)C1 C1(CC)CN(C(C2CC(O)C2)=O)CC1NC(C1CC=CCC1)=O C1(CNC(CCSCCCC)=O)CN(C(=O)Cn2ccc(C)n2)C2(CCC2)C1 c1(CCC)onc(C)c1C(=O)NC1CCCC(CNC(c2ccc(C)n2C)=O)C1 CCCCCC(C)(CC)C(=O)N=S1(=O)CCC2(CC1)CN(C(=O)CCF)CCO2 CC(C)C(C)CC(=O)NC1CC2(C1)CC(NC(c1ccccc1OCC#N)=O)C2 C(=O)(C(C)N=[N+]=[N-])NC1CC(CO)(CO)C1.c12nc(co1)C(=O)NC2C CC(C)CC(F)C(=O)N1CCN(C)C(CNC(C2(COC(C)C)CC2)=O)C1 c1(C(=O)NC2CN(C(C(CCC)(C)C)=O)CC(O)C2)cccn2nnnc12 c1(C(C)C)c[nH]nc1C(=O)NC1CCC1NC(=O)CCC1CCCCC1 C1(CC)C(=O)CCC1NCCCc1cccnc1O c1(CN(C(C2=CCCC2C)=O)C)cc2c(nc1O)CCN(C)C2=O N1(C(c2c(CC)[nH]cc2)=O)CC2CCOCC2(NC(=O)COCC2CC2)C1 c1(C(N(CCOC)C)=O)cc(OC)c(OC)cc1Br.N1(CC=O)CCC1C C1(C(=O)NCC(C)(C)NC(=O)CC2CCCC(CC3CC3)O2)CCCCC1O C1(COC)(NC(C2C=CCCC2)=O)CCN(C(=O)CC2CCCC2O)CC1 c1(C(=O)NCC(C)N(C(c2cc(OC)cc(F)c2)=O)C)cc2n(c(=O)c1)CCS2 C1(C)(CNC(CNC(=O)OC)=O)CCN(C(=O)CCCCc2ccccc2)C1 C1(C=O)CCCC2(CCC2)C1.N1(C(CCN(C(N)=O)C2CC2)=O)C2CCC(C2)C1C=O N1(C(c2n[nH]c(C)c2I)=O)CCCN(C(=O)Cn2cnnc2O)CC1CO c1(NCC(=O)NCCN(S(CC)(=O)=O)C2CC2)ccc(SC(F)F)nc1 C=C(C)CN=C(NCC(F)F)N1CCN2C(=O)NCC2C1 N1(C(C(C=CC)O)=O)CC(NC(C23CC(C#N)(C2)C3)=O)C(CO)C1 N1(C(c2c(Cl)cn(CC#C)n2)=O)CC(C)OC(C)C1 CC1CC=CCC1C(=O)NCCC1CCCN(C(=O)C=C2CCCCC2)C1 C=C=CC(C)C(=O)N1CCCC(NC(=O)C(C)SCC)C1 N1(C(C(Cc2c(C)noc2C)C)=O)CC2CCCC2(NC(=O)C(C)C#N)C1 N1(C(C)=O)CCc2cc(C(=O)NC3CCCCN(C(C)CN(C)C)C3)ccc21 C1(NC(C2C(C)=C2)=O)CCN(C(c2cc(Cl)nnc2Cl)=O)C(C)C1 C(=O)(CS(=O)(=O)C(C)(C)C)N1CCCC(C(C)(O)CNC(=O)Cn2cnnn2)C1 c1(CC(N2CCCC3(N(C)C)C(C2)C3)=O)cc2ccccc2cc1N N1(C(C(C)NC(CCNCCCN(C)C)=O)=O)CC2CC1(c1ccco1)CO2 Cc1cc(OCC(C)NC(N2CCC(C)C(N(C)C)C2)=O)ccc1Cl C(c1cncnc1O)=CC(=O)NC1(CO)CCN(C(CCc2[nH]c(=N)sc2)=O)C1 CC1(C)CCN(C(c2c[nH]nc2-c2ccccc2)=O)CC1NC(=O)C=CC1CCC1 C1(CCNC(C(C)SCCOCC)=O)CCN(C(=O)C=CCO)CC1(F)F N1(C(=O)Nc2cncc(-n3cc(-c4ncc(C)cn4)nn3)c2)CC(C)N(C)C(C)C1 C(=O)(C(O)CCNC(C1CC(O)C(F)C1)=O)NC1C(OC)C(O)C1 CC1ON=C(C(=O)NCC2CCN(C(c3cn(CC(F)F)cn3)=O)C23CC3)C1C CCC(C)C(=O)C(=O)NCc1cc(C(N2CCSCC2C)=O)on1 C1(C(=O)NC)CCN(C(=O)C(CNCC(C)=CC(N2CCCC2)=O)N(C)C)CC1O CCCCC(O)C(C)C(=O)NCC(CNC(c1cc2ccnn2cn1)=O)CO c1(C(=O)NCC(CC(C)C)NC(c2n(C(C)C)cnc2)=O)ncnc2ccsc12 N1(C(CCCCSC)=O)C2COCC1CC(NC(=O)CC1CCCCN1C)C2 c1(NC2CC(N(C(=O)C(C)(F)F)C(C)C)C2)ccccc1N1CCCC1 C1(C)(CNC(c2n(CC=C)ccc2)=O)CCN(C(=O)CC2CCCN2C)C1 CCC(CC(=O)NCc1ccoc1C(=O)N(C1CCCC(C)C1C)C)C1CCC1 C(CC(C)C)(C=O)NC(C(C)NCCC(=O)NCCOC)=O.C(C)(C)S C1(S(C)(=O)=O)(C(N2C(CNC(c3cc(C(=O)OC)sc3C)=O)CC2)=O)CCCC1 C=CCCC(C(=O)N1CC(C(=O)OC)C(C)C1)NC(c1conc1CC)=O C(c1ccc(F)c2ccccc12)=CC(=O)NC1CC(S(=O)(=O)CCO)C1 CC(C(=O)N(C1CN(C(c2cn(C)nn2)=O)CC1(C)C)C)C(C)(F)F CC1CCC(NC(=O)C(C)CC(F)F)CN1C(=O)C=CCOc1ccsc1 c1(C(=O)NCC(CNC(=O)CC2C=CCC2)O)conc1-c1ccccc1 C(=O)(CC(F)(F)C(F)(F)Br)N(CC(C)C)CCNc1cocn1 N1(c2c(C)cnc(C)n2)CC(CNC(C2(O)CCCCCC2)=O)OC(C)(C)C1 c1(C(=O)NC2CCC(CNC(c3scc(OC)c3)=O)C2)c(CO)noc1C c1(CCN2CCC(C(=O)Nc3c(C)scc3)CC2)c(F)cccc1F.C1COO1 c1(NC2C(CC3(F)CN(C(c4ccccc4-n4ccnc4)=O)C3)C2)ccc(Cl)c(Br)c1 c1(C(=O)NC(C)(C)CNC(=O)CCC(N)=O)nc2cccnn2c1Br N1(C(C(CC)COC)=O)CCC(NC(c2sc(C(C)C)nc2C)=O)C(F)(F)CC1 C(c1ccncn1)=CC(=O)NCC1C(NC(C2(CCOC)CCCC2)=O)CCC1 c1(OC)ccc(F)cc1CC(=O)NCC1(NC(=O)CN(C2CCCC2)C)CC1 N1(C(C=C(C)C)=O)CCCC2CN(C(C3Cc4ccc(C)cc4C3)=O)CCC12 c1(CC)cc(F)ccc1NC(C12CC1CN(C(c1cnccc1Cl)=O)C2)=O C(=O)(C(C)CC(C)(C)C)N1CCC(C)(NC(c2c(C)nc(CC3CC3)o2)=O)C1 c1(CC(=O)NC2C(NC(C=CC=CCC)=O)C2)cccc(CCC)c1 c1(CC)c[nH]nc1C(N1CC=CC1C(=O)NCCNC(C1CCC1)=O)=O C1(CNC(c2cn(C3CCOC3)cn2)=O)CCCCCN1C(=O)Cc1cnns1 CC(C)(C(=O)O)C(c1ccccc1)NC(=O)CS(=O)(=O)c1cccs1 C1(CNC(CCOC(C)=O)=O)CC2CCC1N(C(c1ccc(=O)n(C)n1)=O)C2 N1(Cc2c(CC)noc2C)CC2CCN(C(c3cccc(F)n3)=O)C2C1 c1(CC)ccc(C(=O)NCCC2CCCN(C(C3(C)COC(=O)C3)=O)C2)cc1N c1(CC)nsc(N(CC(C)(C)NC(c2cc(C3CCCN3C)[nH]n2)=O)C)n1 C1(NC(C(C)C(C)(F)F)=O)CC1C1CCN(C(=O)CC(F)(F)Cl)CC1 c1(C(=O)NCCN(C(=O)CCOc2cccnc2)CCOC)cc(Cl)nnc1O N1(C(C(C)=CC2CC2)=O)CCCC2(CCCN2C(=O)CCc2ccc[nH]2)C1 N1(C(c2c(C)[nH]c(C#N)c2)=O)CCC2CN(C(c3ccn(C(F)F)n3)=O)CC2C1 C1(CCNS(CC=C)(=O)=O)CCCN(C(c2c(C)cnn2-c2ccc(F)cc2)=O)C1 N1(C(C(C)NCCC)=O)CCC2C(C(N)=O)C2C1.c1(C=O)cc(=N)[nH][nH]1 c1(CC)ncc(C(=O)NCCCNC(c2cc(CC)nc3ocnc23)=O)c(O)n1 C12=C3C(=NC=N3)NC(=NC(C)C3(CCOCC3)N1)N2.C1(C(=O)OC)C2COCC12 c1(OC)cc(Cl)cc(C)c1C(N1CCOC(C(C)NC(=O)Cn2cccc2)C1)=O N1(C(C2C(C)OCC2)=O)CC(C)(C)OC2(C1)CN(C(C1CCSCC1)=O)C2 C1(NC(C(C)NC(N)=O)=O)C2CC3C(C2)C13C(=O)N(C)Cc1cccc(O)c1 C1(C(=O)NC2C3CC2N(C(=O)COCC2CCOC2)C3)CC1C1CCOCC1 CC1COC(C)(C)CN1C(=O)C(Cc1ccco1)NC(=O)Cn1[nH]cnc1=N C(C(CC1CCCC1)C(=O)N(C1(C)CC1)C)NC(C(C=C)C)=O N1(C(C2(CC)CC2)=O)CCC2(CCC(NC(c3cnc(C4CC4)c(C)c3)=O)C2)C1 Cc1ccc2c(c1)CC(C(=O)NCCCNC(c1cccc(P(C)(C)=O)n1)=O)O2 C1(N(C(=O)CC(C)(C2CCC2)OC2CC2)C)CCCN(C(=O)COc2ccsn2)C1 C1(CC(=O)NC)CN(C(=O)Cn2cccn2)CCN1C(c1cocn1)=O N1(C(C(=O)NCC)=O)CCC2(CC1)CC2C(=O)NC1CC(OC(F)(F)F)C1 C(=O)(C(O)CC(F)(F)F)NCCCNC(=O)COc1ccc(F)c(Cl)c1 N1(C(C2C(CCC)C2)=O)CC2CCCC(N(C)C(C3CC=CC3)=O)C2C1 Cc1c(C(N2CCC(CN(C)C(C34CC(C3)C4)=O)C2)=O)cnn1C(C)C(C)C Cc1cc(O)nnc1C(=O)NC1CN(C(c2coc(Cl)c2)=O)CCC1C(F)(F)F c1(Sc2ccc(C(N3C(CCC)C=CC3)=O)cn2)ccc(OC)cc1C C1(CN(C)C(C2CC3CCN(c4cccc(C#N)n4)CC23)=O)CCn2cncc2C1 N1(C(C(C)Cn2cccn2)=O)CCC(NC(c2ncc[nH]2)=O)CC1C C#CC1(C(=O)NCC2CCC(C(=O)NCCn3cncn3)O2)CCCCC1 N1(C(=O)Cn2cccc2)CC2(CNC(c3ccn(C4CCC4)n3)=O)CCC1CC2 C1(CC)CN(C(c2coc(CNC(c3cnc(OC)s3)=O)n2)=O)CC(=O)N1 N1(C(c2scc(C)c2Cl)=O)CC(CNC(c2cc[nH]n2)=O)OC2COCC12 c1(OC)c(C(N2CCC(O)(CCNC(=O)CC3CCCO3)C2)=O)ccc(Cl)c1Cl C1(C(=O)OC)CCC(CSc2ccccc2)N1C(c1cnc(Br)s1)=O CON1CCC(CC(=O)NCC2CC2CNC(=O)C=Cc2ccccc2C)CC1 N1(C(c2c(N(C)C)cccn2)=O)CC2CC(NC(c3sccc3F)=O)C1C2 CCCCCC(O)C(C)C(=O)NCC(CC)NC(C1Cc2ccccc2N1C)=O C1(C(=O)NCCC2(OC)CN(C(C=C(CC)C)=O)C2)COC2(C(=O)OC)CC1C2 CCC(C)(CNC(=O)CC1CCCC1)NC(=O)CC1C=CCCC1 c1(NC(C2C(N(C(C(C)C)=O)C(=O)OC(C)(C)C)CC2)=O)ccc(C(N)=O)s1 C1(CNC(c2cc(C(=O)OC)sc2)=O)CC(OC)CN1C(c1c(C)cnn1C)=O CC12CCC(C(N3CCCC(NC(=O)CC(F)(F)C(F)F)CC3)=O)(CC1)OC2 c1(CC(=O)NC(CC=C)CNC(C2CC23CCC3)=O)ccnc(C(F)(F)F)c1 CC(O)(C(=O)N1CC2CC(NC(=O)CN3C(=O)CCC3=O)C1C2)C(F)(F)F c1(OC)ccccc1Oc1ccccc1CNC1(CNC(=O)COC)CCC1 C=C=CCC(=O)NCCCOCCNC(=O)CCCc1ccccn1 O=C1CCCC(CC(N2CC=CC(NC(=O)CCCc3cnccn3)C2)=O)C1 C1(C(N(C)Cc2ccc(C)cn2)=O)CCC(O)CN1C(C1CCCN1C(C)C)=O C(=O)(CCCCC(F)F)N1CC(NC(COCC(=O)NC)=O)C(C)(C)C1 C#CCC(C)(C(=O)NCCCC1C=NNC1=O)NC(=O)C(COC)COC CC(C)CCCCCC(=O)NCCCCNC(=O)CC1C=CCCC1 C(=O)(C#CC1CCCO1)N(C(C)CN(C)C(c1cnc(C2CC2)s1)=O)C CC(C(=O)NCc1nc(C(=O)Nc2cnn(CCF)c2)co1)C(C)(C)C C1(C)(C(=O)NCCC(C)(OC)SC)CCN(C(=O)CC2(O)CCCOC2)CC1 C(=O)(C(F)C(F)(F)F)NC1(CCCNC(C(C2CC2)OC)=O)CC1 CC1CCC(C(N2CC(NC(=O)CSC(F)F)C2)=O)CN1C(=O)C=Cc1ccco1 C(=O)(C1=CC(O)CCC1)N1CC(NC(c2c(C)nc(O)cc2)=O)C(C(F)(F)F)C1 C1(OCC)CCCCN(c2nnnn2CC)CC1.C123CCC(CC1)(OC2)CNC3=O CCC(CNC(=O)C(C)C#N)(CC)NC(c1cc(C2(C)CC2)n[nH]1)=O N1(C(C(C)=CC2CC2)=O)CCC(O)(C(C)NC(=O)CCC2CCC(O)CC2)C1 CCC1=NOC(C(N2CC=CCC2C(=O)NCC2(F)CCOCC2)=O)C1 C1(CCCNC(=O)NCC2CCC(CN(C)S(N)(=O)=O)CC2)CCCCNC1=O c1(CC(=O)NC2C(OC)COC2)ccc(O)c(C)c1 C1(NC(c2cc(CC)oc2C)=O)CCN(C(c2sc(N(C)C)nc2C)=O)CC1F C=CCCCC(=O)NCC1CN(C(c2ccc(CC)cn2)=O)C2CC12 C1(C(N2CCCCC2CC2CC2)=O)CC2(C1)CN(C(c1nn[nH]c1C(F)(F)F)=O)C2 C#CCCCCC(=O)N1CC(NC(=O)CSc2nncn2C)C2CC2C1 C(=O)(C1=NNC(C(F)(F)F)C1)N1C(CCNC(=O)COCCF)CCC1 c1(C(N(CC(F)(F)F)C(CN(C2CC2)CC)=O)=O)ccccc1 C1(CNC(C2CCN(C(C)=O)CC2)=O)C2CCCC1N(C(c1cc[nH]c1CO)=O)C2 C12(CC(=O)NCCN(C(=O)CCC3CC3(F)F)C)CCC(CC1)CC2 N1(C(c2c(C)nccc2)=O)CCC2CN(C(c3ccccn3)=O)CC12 n1(CC)nnc(C(N2CCC(C3OCC3(F)F)C2)=O)c1C Cc1oc(CNC(c2cc(CN(C)C)on2)=O)nc1C(=O)NC1CS(=O)(=O)C1 C#CC1CN(C(C2CCN(C(=O)Cn3cnnc3)CC2O)=O)CCN1C c12ncoc1CNC2=O.CCCCCN(CCCN(CC)CCO)C.CC N1(C(C2(NC(C(CC=CC)CC)=O)CC2C)=O)CC2C=CCC(C2)C1 Cc1cc(C(=O)NC2CN(C(=O)Cn3c(C)csc3=O)CCC2C)nc(O)n1 c1(NC2C(CNC(c3ncn(C)c(=O)c3)=O)CCCC2)cccc(N=[N+]=[N-])c1 c1(CN2CCN(C(C(CC=C)C)=O)C(c3nccn3C)C2)nc2ccccc2[nH]1 C(CNC(=O)CN1CCC(C)C1)(CC)(CC)NC(c1cc(C(C)=O)n(C)n1)=O c1(C(N(CCC)CCNC(=O)CCn2cccn2)=O)csc(C(C)(C)C)c1 C1(N(C(c2c(C)n(CCO)cc2)=O)C)CN(C(c2cc(Cl)ccn2)=O)CC1(C)C C1(NC(C(CCO)N(C)C)=O)CC2CCC1(NC(=O)C(C1(O)CCCC1)F)C2 c1(C(N2CC(N(C)C(c3cc([N+](=O)[O-])c[nH]3)=O)C2)=O)ncc2ccccc2c1O C1(C(=O)NC2CC(C)(NC(=O)C(C3(O)CCCC3)F)C2)CN(S(N)(=O)=O)C1 Cc1ccc(C)c(-c2ncccc2NC(=O)CCNC(C23CCN(CC2)C3)=O)c1 Cn1nc2c(c1NC(C1C3CCC(C3)C1NC(c1cncnc1)=O)=O)CCCC2 C(=O)(C(CO)C(C)(C)C)NC1(CNC(c2c(C)nc(CCC)o2)=O)CCC1 C1(C(N(CC(C)OC)C)=O)CCN(C(=O)Cc2ccc(C(C)C)cc2)CC1O C1(C(N2CC(C(=O)NOCCCOC)C3CC23)=O)C2(CC2)C12CC2 c1(C(=O)NC(CC)CNC(c2ccc(C)nn2)=O)oc2c(OC)cccc2c1C N1(C(CSCC)=O)CC(CNC(=O)CC2CCCC2C)(COC)C1 c1(C(=O)NCC2N(C(C(CCC)C#N)=O)CC(C)(C)C2)cc([N+](=O)[O-])cnc1C C(c1cc[nH]c1)=CC(=O)CC=CC(=O)NCC1(C(=O)OC)CC1C c1(CNC(C(COC)Cl)=O)cccc2c1CCN(c1nncs1)C2 CC(F)(F)C(C)(C)CNC(=O)C(CC1CCOCC1)NC(C1CC1Cl)=O c1(C(=O)NCCCC2N(C(C(CC)N(C)C)=O)CCC2)noc2c1CCCC2 c1(N2CC(NC(c3cccc(I)c3)=O)C(F)(F)C2)ncnc2cc(Br)sc12 N1(C(CCOCC)=O)CC(CNC(C2CC3CCC3C2)=O)C2(CC2)C1 N1(C(CSCCOC)=O)CCC2(CC1)OCCC2NC(c1ccon1)=O N1(C(c2c(C)nn[nH]2)=O)CCC2(CC2C(N2CC(O)C(O)C2)=O)C1 C(C(=O)N=c1cccn[nH]1)N1CCN(S(C(C)C)(=O)=O)C2(C1)CC2 N1(C(C(n2ncc(C)c2)C)=O)CC(F)CC1CN(C(=O)C(O)C1CCC1)C C(=O)(C(O)CC(C)C)NC1CN(C(c2cn(CCC)nn2)=O)CC1F c1(CN2CC(NC(=O)NC3(C=C)CCOCC3)C(F)(F)C2)cc(Cl)cc(Cl)c1Cl c1(C(N2CCOCC2n2cc(C(CC(N)=O)N(C)C)nn2)=O)ccc2c(c1)COC2 c1(OC)ccc2c(c1)CCC2NC(=O)CC1CC2CC1N(C(=O)OC(C)(C)C)C2 C12(C(=O)NCc3nnc(C)o3)CCC(CC1)N(C(=O)CC(=O)N(C)C)C2 c1(OC)cccc(C(c2ccccc2)(C)NC(=O)NC2CC(C#N)C2)c1 c1(C(=O)OC)ccc(O)nc1NC(C1CCN(C(=O)Cc2cc(C)no2)C(C)C1)=O N1(C(C(CNC(C2N(CC)CC2)=O)CC2CC2)=O)CC2CC3CC2C1C3 Cc1cccc(Cl)c1CNC1C=CCN(C(=O)C(C2CCCCC2)C)C1 c1(CNC(C2CCC(C)C(C)C2)=O)nc2c(s1)CN(C(=O)CC1(CO)CC1)CC2 N(C)(S(=O)(=O)N1CCNC(C2CCC2)C1)OCC#C C1(C(N2C(C(N3CC4CCC3C4)=O)C=CC2)=O)CC2C=CC1CC2 C1(OC)CC(CCNC(C2CCC(F)CC2)=O)N(C(c2n[nH]c(C)n2)=O)C1 c12cc(OC)c(nc1C)oc2=O.C1(N(CCCC)CC(N)=O)CCS(=O)(=O)C1 N1(C(c2cc3c(s2)CCC3)C(=O)NCCSC)Cc2c[nH]nc2C(C)C1 N1(C(C2CC(C)(C(C)C)C2)=O)CCC2(CCCN2C(=O)C(=O)N=S(C)(C)=O)CC1 c1(C(=O)NCC2C(CNC(CCOCCCOC)=O)C2(F)F)c(C)n[nH]c1C c1(C(N(CCCCNC(c2ccc(C3CCCCC3)s2)=O)C)=O)ccc(O)nn1 Cc1cc(C(=O)NCCCOCC2CC2NC(=O)Cc2ccncc2Cl)cnc1C C#Cc1ccc(C(=O)NC2C3CC4C2C4C3C(=O)NC(c2nccs2)C)cc1 c1(C(N2CC(CNC(C3CC4C=CC3CC4)=O)OCC2)=O)ccc(O)c(O)c1 N1(C(C2CC(=O)NCC2)=O)CCC2C1CCN2C(c1cnc2cccnn12)=O C1(NC2CCCOC2)CC(C(=O)O)CN(CCCC(=O)OC)C1 N=c1ccn(CCOc2ccccc2CO)c(O)n1 N1(C(C2(CCOC)CC2)=O)CCC2CN(C(c3ccc(Cl)nc3)=O)CCC2C1 C(=O)(C(F)C(C)CC(C)(C)C)N1CCC(OCCNC(CCCOCCOC)=O)C1 c1(N)ccccc1OC.C(=O)(CCCNCc1ccoc1)NCC(COC)O CC1(C)CC2(CC(NC(=O)C(CC3CCOCC3)NC(=O)Cc3ccsn3)C2)C1 N1(C(c2c(C(C)C)n[nH]c2)=O)CC2COCC2(C(=O)NC2CN3CCCC2C3)C1 Nc1c(C(N2CCC(C(F)C(=O)NC3CC(O)C3)C2)=O)cccc1F C1(N2c3nc([nH]c(=N)n3)N3CCN(CC3)CC2)CS(=O)(=O)CC(=O)N1.CCOC c1(C(=O)NC(C2CCN(C(C3CCC(SCC)CC3)=O)C2)C)cc(O)ccc1F Cc1nc(O)c(C(=O)NC2CCCCCN(C(=O)CC3C=CCC3)C2)nc1C c1(CC)c(C(=O)NC2CCN(C(=O)COC(F)(F)F)CC2)csc1C N1(C(CCC#C)=O)C(C=O)CCC12CC2.c1(N)cccc(SC)c1 Cc1nc(C(=O)NCC(C)(C)NC(=O)CC(C)C(F)F)ccc1C#N C1(OCC)(COCC(C)NC(N2CC(C)(Cc3cn(CC)nn3)C2)=O)CCOCC1 C12CCN(CC1)C(=O)N2C.C1(CC(=O)N(C)CCN(C)C)(OC(C)C)CC1 c1(O)cccc(CCCN(CC(N)=O)C2CC2)c1.c1(OC(=O)N)ccccc1F Cc1oc(S(=O)(=O)NC2CC2)cc1C(=O)NC1(NC(C23CC(C)C2C3)=O)CC1 C(C)(CCC(=O)NC1CC(O)(CNC(C2CCCC2OC)=O)C1)SC c1(CNC(C2(C)CC(C)OCC2)=O)cc2n(n1)CCN(C(c1ncn(C)n1)=O)C2 Cn1cc(C(C(=O)NC2CNC(=O)C2)NC(=O)CCC2CC2(F)F)nn1 CC(C)C(C(=O)N(CC(O)CNC(=O)CC1(O)CC1)C)NC(c1ccccc1)=O C1(OC)CN(Cc2cscc2Br)C2(CCC2)C1 c1(NC(C)=O)cccc2c1OCCC2Nc1ccc(S(=O)(=O)N2CCCC2)cn1 c1(C(=O)NC2C3CCN(C(CC(CCC)O)=O)C32)cc(C#N)ccc1N c1(CC(=O)NCC2C(NC(=O)COCC3CCCOC3)C2)cccc2nsnc12 Cc1ncnc2c1CC(C(=O)NC1(C3CN(C(=O)CC(C)(F)F)C3)CC1)CC2 c1(C(=O)NC2CCC(N(C(=O)CCC3(C#N)CCC3)C)C2)ccc(F)c(F)c1 C(=O)(C1=NOC2COCC12)NCC(CNC(c1c(C)oc(C2CC2)n1)=O)C Cc1cc(C(N2CC(NC(C3C4C=CSC34)=O)C(F)(F)C2)=O)cnc1F c1(CCN=C(NC(c2ccsn2)C)NC2CCC2)c[nH]c2cc(F)c(F)cc12 N(C(=NCC1CCC1)N1CCC(O)C1)CC1C(C)(C)CCCC1N C(=O)(CC(C)C(=O)C1CC1)OCC.C1(C(=O)N(CC2CC2)CC)(C)CCCCC1 C1(C(N(C2CN(C(c3ncccc3Cl)=O)CC2(C)C)C)=O)CCCCCS1(=O)=O C=CC(C)(C)CC(=O)NCc1csc(CNC(=O)CCCOCCC)n1 N1(C(CCN(CC)CC)=O)CC2(CCCC(CNC(=O)C(C)(C)CC3CC3)O2)C1 N1(C(CCN(C)CCO)=O)CCC2(C1)CN(C(C1(O)CCOC1(C)C)=O)C2 C(=O)(C(C(C)(C)C)C1CCCC1)NC1CCN(C(c2c(C)ccnn2)=O)C1 N(C1CCCn2ccnc21)C(C1N(C(Cc2c(C)scc2)=O)CCC1C1CC1)=O c1(C(C(=O)OC)N(CC(CC(C)C)OC)C(CC)CC)ccc2c(c1)CCC2 C1(C)(CC)C=C(C(=O)NCC2CCN(C(=O)Cc3csc(C(C)C)n3)CC2C)C1 C12(C(=O)NC(C3CC3C(N3CCC4CC34)=O)C)CC(C#N)(C1)C2 N1(CCC(C)CC(=O)O)CCc2c(ccnc2Cl)C1 c1(NC(c2c(C(C)C)cc(F)cc2)=O)ncc(CO)cc1Br N1(C(C2N(C(C)=O)CCC2)=O)CN(C(=O)Cc2cscn2)CC1CO C1(CC)CN(C(c2ccc(Cl)o2)=O)CCN1C(c1ccc(C#N)s1)=O c1(OC)ccc(C(N2CCC(O)C(C(=O)NCc3ccnc(C)c3)C2)=O)c(Cl)c1 c1(NC(c2ncoc2CNC(C2CC23CCC3)=O)=O)ccc2nncn2c1 N1(C(C(C)C)=O)CCC2(CC1)CC(NC(=O)C(C)Cn1cnc(C#N)n1)CCO2 c1(NCCn2c(C(C)C)nnc2)ccc(S(=O)(=O)NCCCN2CCCC2)cn1 C(=O)(C(C)(C)C(C)(C)C)NC(CC1CN(C(C2(C)ON=C(C)C2)=O)C1)C C#Cc1ccc(C(=O)NC2CC3(C(N4CCCCC(N(C)C)C4)=O)COC2C3)cc1 c1(C(=O)NCC2CC2CNCC=CCCO)cc(Cl)c(Br)cn1 c1(OC)ccc(NC(=O)NC2C3CC4C(C3)C24)c(Cl)n1.C12(C)CCCN(C1)C2=O C(=O)(CCC1=NNC(=O)CC1)NCC1C(C)CCN(C(C2(F)CC2)=O)C1 C(CC(=O)NC(C)(C)CC(C)(C)C)(C(F)(F)F)NC(CC1CC(=C)C1)=O CC(CC(C)(C)C)C(=O)N1CCN(C(c2coc(C(F)(F)F)c2)=O)CC1 c1(C(C)O)ccc(CNC2(C)CCN(C(C3CN(C4CCC4)C3)=O)C2)cc1 c1(N(CC(CCC)C)C)nc(=NCc2cc(C)cc(Cl)n2)[nH]c2c(F)cc(F)cc12 CCC(C)CCC(=O)N1CC(C(=O)NCc2cnn(CCF)c2)CCC1C CN1CC=C(C(=O)NCC(C)(O)CNC(=O)C(C(C)(C)C)NC(C2CC2)=O)C1 N1(C(c2cn(C3CCCC3)nn2)C(=O)NCCCF)CCCCC12CC2 c1(C(n2cc(CNC(c3cnn(C(C)C)c3)C)nn2)C)nc2ccccc2s1 C(=O)(C1CCCc2nc[nH]c21)N1CC2C(CNC(C=CCOC)=O)C2C1 c1(C(=O)NC2CC(CCNC(=O)C(F)CC3CCC3)C2)cnn2ncccc12 N1(C(CC(C)F)=O)CC2CCCN(C(c3ncnc4c3ccn4C3CC3)=O)C2C1 N1(C(c2c(C)cncc2)=O)CCCC(CCNC(C2CC3C(C2)C3(F)F)=O)CC1 C(=O)(CS(=O)(=O)CCNCC1CN2CCC1CC2)NC(CCOCC)C(=O)NC C1(CC(=O)N(C)CC2CN(C)CCO2)CC2(C1)CN(C(C1CCCCC1(C)C)=O)C2 c1(C(C(=O)NCC(CNC(c2scc(C)c2C)=O)(C)C)O)cccc([N+](=O)[O-])c1 N1(C(C=COCC)=O)CCC(C)(C)C(NC(=O)CCCCCc2ccccc2)C1 Cc1cc2[nH]c(C(=O)NC3CC3CNC(=O)C=Cc3ccccc3C#N)cc2o1 Cn1ccc(C(=O)NC2CCCC2(C)NC(c2cc(Cl)ccn2)=O)cc1=O C1(NC(C(CSC)C)=O)CN(C(=O)CC(C)(C)O)C2(CCCCC2)C1 c1(C(N(CCNC(C(C)OC)=O)C(C)C)=O)ccc2c(c1)CC(C)O2 c1(C(=O)NCC(CC)N(C)C(C2CCC(C(C)(C)C)O2)=O)csc(C)c1C c1(OC)ccc(Cl)c(C(c2nnnn2C2CC2)NC(C)CC2CCOCC2)c1Cl c1(C(=O)NC(CN(C(Cc2c(F)ccc(SC)c2)=O)C)C)cccc2nn[nH]c12 C1(CNc2c(C)c(N3CCC=C(Br)C3)ncn2)CCCC2(CNC2)O1 N1(C(C(C)Cc2ccco2)=O)CCCC(O)(CCNC(=O)CCC#N)C1 C(CC(C)(C)C)(C(=O)NCC1(SC)CC1)NC(C(CCCC)O)=O C12(C(N(CC(CN(C)C)O)C)=O)CCCC1N(C(C1CC(CF)C1)=O)CC2 C1(CC)(NC(=O)CCC=C(C)C)CCN(C(=O)CC2CCS(=O)(=O)C2)CC1 N1(C(CCC(=O)NC)=O)CCC2CCCC12CNC(c1ncc(OC)cn1)=O C1(CC(N2C(COC)CC2)=O)CC(O)CN1C(=O)CC1CCCC(=O)C1 C(C(CC(=O)N(C1(CCC)CC1)C)OC)NC(C1(CC)CCC1)=O c1(N(C(c2c(C)n(C)nc2C(F)F)=O)C(C)C)cc(C#N)ccc1[N+](=O)[O-] c1(C(N(CC(O)CN(C)C(C2(C(F)(F)F)CCCC2)=O)C)=O)cc(CO)n(C)n1 C1(C(=O)NCCc2onc(C)n2)CCCCN(C(=O)CCS(C)(=O)=O)C1 CC(C)CC(CNC(c1ccoc1Br)=O)NC(=O)C(C)Cn1ccnc1 c1(C(=O)NC(CC=CC)C(=O)NCCn2ccnc2C)nccc(C)c1N N1(C(COc2cccc(CC)c2)=O)CC2OCC(NC(=O)C(C)C(O)CC)C2C1 c1(C(=O)NCC(CC=C)NC(=O)C(C)CC=C)ccc(Br)cc1 n1(CC)cc(C(=O)NC2(CCNC(=O)CCC3CCCN3C)CC2)c(C)n1 c1(OC)nc(Cl)cc(=NCCCC2CCCCO2)[nH]1 C(=O)(CCCC(=O)NCC(O)CNC(=O)C1CC1)N(C(c1c(C)cccc1)C)C C(CC(C(=O)NC(CN(C)C)C(C)C)NC(=O)Cc1cnnn1C)OC c1(CNC(C(C(C)O)NC(C2CCS(=O)(=O)C2)=O)=O)c(F)cc(Cl)c(F)c1F C(=O)(C1=C2CCCN=C2NN1)NC1C(NC(=O)C=CC(F)(F)F)CCOC1 c1(OC)cn(CC(=O)NC(C)(C)CNC(C2ON=C(C)C2C)=O)c(C)cc1=O C1(F)(CNC(=O)COc2ccccn2)CCCN(C(c2cc(O)ccc2O)=O)C1 c1(C(=O)NCC2CCN(C(C=CC)=O)CCC2(F)F)coc2cc(F)cc(F)c12 N1(C(c2cc(C(C)=O)on2)=O)CC(NC(=O)C(c2cccnc2)C)C2(CC2)C1 c1(CC)ccc(F)c(C(=O)NCC(CNC(=O)CCC(C)C#N)S(C)(=O)=O)c1F c1(NC(C2CCC(NCc3ncn(C)c3)C2)=O)cc(F)c(Cl)cc1Cl C1(CNC(C2CCOC2)=O)CC2(CCN(C(c3c(F)cccc3F)=O)C2)CO1 c1(C(N2CC(C3CN(C(C4CC(OC)C4)=O)C3)C2)=O)cc(F)cc2nn(C)cc12 O=S(=O)(c1[nH]c(=NCC2CCCC2(F)F)ccc1Br)NCc1ccc(F)cc1 C1(NC(c2nc[nH]c2C(F)(F)F)=O)CCOCC1NC(C1CCOCC1)=O C(=O)(C1=CCCOCC1)N1CCCN(C(C2C(C#N)C2)=O)CC1 C1(CC(=O)NCCn2c(C)nnc2)CCCCN1C(=O)CN1C(C)CCC1C c1(CCC(=O)N(CC)Cc2ccc(CN3CCOCC3)o2)nnc(O)nc1O O=C1CC(OCC(N2CCC2C(=O)NC2CCOC2=O)=O)C(=O)N1 N1(CC(=O)NCC(C2CCCC2)C)CCN(C(=O)CCc2nncs2)CC1 c1(C(=O)Nc2c(OCC(C)C)ccc(Br)c2)ccc2occc2n1 C(=O)(C#CC(C)(C)C)N1CCCC(CCNC(c2c(CCC)n(CC)nn2)=O)C1 C1(C(N2CC(C)(CC)C2)=O)N(C(=O)C(C)N2CCCC2)CC12CCCC2 C1(NC(C(=Cc2ccco2)C)=O)C2CC(O)C1N(C(c1cnnc(O)c1)=O)C2 CC1CCC(O)(C(=O)NC(C)(C)CCCNC(=O)CN(C)C(=O)C2CC2)CC1 C1(NC(C(CC)SC)=O)CC2CN(C(=O)C(C3CCOCC3)F)CC12 CC(C)(C)CC(=O)NCCCC1CCCN1C(=O)C(F)(Cl)c1ccccc1 N1(CCC=C)CCC(C(=O)NCC(C2CCC2)NC(c2sccc2CC)=O)CC1 c1(C(N2CC3CC(NC(c4c(C(C)C)n[nH]c4)=O)C3C2)=O)ccc([N+](=O)[O-])n1C C1(C)(C(=O)NCCCC2N(C(c3cc(OC)n(C)n3)=O)CCC2)CCCC1(F)F n1(C(C)C)cc(C(=O)NC2CN(C(=O)C(C)N(C)C)CC23CC3)c(O)nc1=O C#CCC(C)(C)CNC(=O)CC(C1CC1)NC(=O)CC1COC(=O)C1 CC1(C)CN(C(C2(C(F)(F)F)CC=CC2)=O)CC1CNC1CS(=O)(=O)CC1O C1(CNC(c2nc(OCC)oc2)=O)CC(C)N(C(c2cnn(CC)n2)=O)C1 c1(C=O)cccc2nn(C)cc12.c1(CCC)ccc(SCC)cc1.C12CCN(C1)N2C N#CC1(C(=O)NCCCN(C(C2CNC(=O)C2)=O)C2CC2)CC=CC1 c1(C(N2C3(CN(C(c4cccc(C(=O)OC)c4)=O)C3)CC2)=O)cc2sc(C)cc2[nH]1 Cn1cc(C(N2CCC(CF)(NC(=O)CC3(C#N)CCC3)C2)=O)c2ccccc12 N1(C(c2nc(CC)sc2)=O)CC2(CC(NC(C3CC(C)C3)=O)C2)C1 [N-]=[N+]=NCC(F)CCNC(=O)C=CCNC(C1(n2nccn2)CC1)=O C(=O)(CCCCC(F)(F)F)NCC12OCC(NC(c3nccc(C)n3)=O)C(C1)C2 C1(NC(C(C(C)C)C#N)=O)CN(C(C2CC3(C2)CC(O)C3)=O)C2(CCC2)C1 CC(=O)CC(C(=O)O)NC(=O)CCNC(c1ccc(C)cc1)=O c1(COC)nn(CC(=O)N(C(C#N)C2CCC2)CC2CCOCC2)c(=O)o1 C1(C(N2CCC(NC(C=CCC)=O)(CF)C2)=O)Cn2c(C)nnc2CN1C c1(C(N2CC(N(C(=O)CC(OC)OC)CCC)C2)=O)cc2occc2[nH]1 C1(NC(C2CC(=C)C2)=O)CN(C(C2(C(=O)OC)CC2)=O)CC(C)(C)C1 C1(CNC(C2CC(OC)C2)=O)CC(F)(CNC(=O)CCOc2ccncc2)C1 N1(C(c2ccc(OCCC)cc2)=O)Cc2[nH]nc(-c3cccc(F)c3OC)c2C1 N1(C(C)=O)CCC(C)(C(=O)NC(CNC(C2(C)CCN(C)C2)=O)C2CCC2)C1 N1(C(c2c(CCC)nsc2N)=O)CC(C)C(N=c2ccc(C#N)n[nH]2)C(C)C1 N1(C(c2c(C)nsc2)=O)CCCC(CCNC(C2CC3CCC2C3)=O)C1 c1(CN2C(C(N3CC(CN(C)C)OCC3)=O)C=CC2)c([N+](=O)[O-])ccc(Cl)c1Cl CP(C)(=O)c1cnc(C(=O)NCc2cn(CCO)nn2)nc1 N1(C(CC(=O)NCC)=O)CCCC(N(C)C(c2ccc(C(N)=O)[nH]2)=O)C1 Nc1ccc(O)c(C(N2CCC(OCCNC(C3CCOC3)=O)C2)=O)c1 N1(C(=O)OC(C)(C)C)CC2CC(F)C1C2C(=O)NCc1ccco1 C1(C(=O)NCC2N(C(C=CC=CCC)=O)CC(F)C2)CC2CCC(C1)C2O C(C(O)CC(=O)NCC1=NOC(C)C1)NC(c1cn(CC=C)nn1)=O c1(OC)cc(C(=O)NC23CC(C(N4CC(C)SC(C)C4)=O)(C2)C3)c(Br)cn1 N1(C(C(CCSC)OC)=O)CCC2(CCCN(C(c3ccc(CO)s3)=O)C2)CC1 Cc1cc(CNC(=O)C(Cc2ccoc2)NC(c2nnsc2N)=O)c(C)s1 n1(CC)nc(C(=O)NCc2cnn(C)c2C(=O)NOCC(C)(C)O)c(C)n1 N1(c2nnc(C)s2)CCC2(CC1)CCN(C(=O)CCOc1ccc(Cl)cc1)CC2 S(=O)(=O)(c1ccc(C(=O)NC2CCC2CNC(=O)C(F)n2cccn2)s1)NCC C1(C(=O)NCC(CC=C)(C)CO)CN(C(=O)CCCCCF)CC(C)(C)C1 c1(C(=O)NCC23CC2CN(C(=O)Cc2cscn2)C3)cccc(I)c1Cl C(=O)(C(COC)CC(C)C)NCC(CC=C)NC(c1nscc1Br)=O N#Cc1cccc(NC(C2(NC(C3CC3c3cccs3)=O)CCCC2)=O)c1 C(C(F)(C(=O)N(c1ccsc1)C)C(C)C)NC(C(C1CC1)OC)=O C12CCCN(C1)C(=O)COCC(=O)N1CCC(C1)O2.C(=O)(CSNCCC)NC.CC C1(NC(COCCSC)=O)CC2CCC(C1C)N2C(=O)C(CC(C)C)CC(C)C N1(C(c2n(CC#C)ccc2)=O)CC2CC2(C(=O)NC(C)CCC2CC2)C1 CCCC(O)(CCC)CC(=O)N(C)CCNC(c1ccn(C2CC2)n1)=O C1(NC(=O)CC2COCCO2)CN(Cc2ccc(F)nc2F)CCC1(F)F c1(N(C(=O)CSc2nn[nH]n2)C(c2ccc(Cl)cc2)C)cccc(F)c1N C(N=c1[nH]c(Cl)ncc1F)C1CCC(NC(c2c(C)oc(-c3ccccc3)c2)=O)C1 c1(C(N2C(C(C)NC(c3c(C)nsc3C)=O)CCCC2)=O)ccc(N)c(F)c1 N(C(=NCCCCl)N1CCC(C2CCC2)C1)C(=O)C1Cc2ccccc21 CC1CC(NC(=O)Cn2cccn2)CCN1C(=O)CCc1cc(F)ccc1F c1(CC(=O)NCCC(CNC(C2(C)CCCC2O)=O)OC)ccc(C(N)=O)nc1 n1(CC(=O)NCC(CNC(C(C)(F)c2ccccc2)=O)F)nc(O)ccc1=O Cc1cc(C(=O)NCC(C)(C)CNC(C2(C)CC2(F)F)=O)cc(C)c1O c1(C(N2CC3CN(C(CSCCOC)=O)C3CC2)=O)cnc2c(c1)N(C)CCO2 N1(C(C2OCCN(C)C2)=O)CCC(NC(c2cn[nH]c2)=O)C12CC2 C1(C(=O)NC(C(=O)NCC(COC)O)CC2CCC2)C2CCCC(=O)C12 N1(CC(=O)N(CCN(C(=O)CC#N)CC)CC)C(=O)NC2(CCCC2)C1=O C(CS(=O)(=O)C(C)(C)C)NC(c1cnc(COC)[nH]1)c1nnnn1C1CC1 C1(CNC(=O)C2=CCCO2)C2CCCC1N(C(c1cnc3ccoc3c1)=O)C2 C1(n2cc(CCCOC)nn2)CN(C(=O)CNC(=O)CC2CCOCC2)CC1C C=C=CCCN=c1nc(N2CCOC(CC)CC2)c2c([nH]1)CCC2 C1(F)(N(C)CC)CCN(C(c2ccc(C(=O)OC)o2)C(=O)NC)C1 N1(c2nnc(CC(C)C)s2)CC2CC(NC(C3CCNC3=O)=O)CC2C1 c1(C(=O)NCC(C(C)C)NC(c2cc(OC)ns2)=O)ccc(CCF)cc1 c1(CC(=O)N(CC(O)CNC(=O)C(C)(C)S(C)(=O)=O)C)ccc2c(c1)CCCO2 Brc1cccc(CNCC2c3cn2nn3)c1.C1(C)CCCOC1.C1CC1 C(=O)(C(F)(F)C(C)(C)O)NC1CCN(C(c2ccc(C)cc2Cl)=O)CC1F CCC(CC(=O)NC1(C)CC(NC(=O)CCN2CCCCC2)C1)OC CC1(C)CCCC(C(=O)NCCOCCNC(=O)CCCC#N)C1 c1(C(N2CC(C(C)NC(=O)CNC(c3nccs3)=O)C2)=O)cccc[n+]1[O-] CC(C)CS(=O)(=O)CC(=O)N1CCOC(CNC(C2CC2(F)F)=O)C1 C(C)(C(C(=O)NC(C)C(C)(C)NC(=O)C=C(C1CC1)C1CC1)N(C)C)OC c1(N(C)Cc2nn(C)nc2Br)nc(N2CC3CC3C2)nc2sccc12 c1(N2CCC(CN(CC)CC)C2)nc(=NCC2(C)CCN(C)C2)[nH]c2c1CCC2 CC1CN(C(=O)CCn2ccnn2)CCCN1C(c1ccc2nn[nH]c2c1)=O c1(C(N(CC(=O)NC2CCC3(CC3)C2)CCC)=O)cc(CO)c(C)o1 N1(C(CSCC)=O)CCC2(NC(c3nc(C)nn3C)=O)CCCC12 Cc1cscc1C(=O)NC(CC1CCC1)C(=O)NCC1(CO)CC=CC1 c1(C(N(C(C)C(=O)NC(C(O)CO)C2CC2)CCC)=O)c[nH]c(C#N)c1 c1(COC)ccncc1NC(c1cc(C)on1)c1nnnn1C1CCCCC1 c1(OC)ncnc(C(N2CC3CC(CNC(c4cc(CO)on4)=O)C3C2)=O)c1F C1(CNC(c2cn(CC=C)nc2)=O)COCCN(C(c2cc(C#N)no2)=O)C1 c1(C(=O)NC(C2OCCN(C(c3ccc(C)nn3)=O)C2)C)cnc(C)cc1C c1(C(=O)NCCC(C)NC(C2C(C)C2C)=O)nn(C)c2c(=O)[nH]cnc12 c1(C(=O)NCC2(NC(C)=O)CC2)c(F)ccc([N+](=O)[O-])c1Cl.N12CCCC1C2=O C(CNC(=O)CC1(OC)CCC1)(C(=O)NCCC1CCOC1)OC C(=O)(C(C)(CNC(=O)C=CCF)CC)NCCC(CC)C C(=O)(CC1OCCc2sccc21)NC1C(C)N(C(=O)C=CC(C)(C)C)CCC1 C=C1CCN(C(C2CCC(C)(C)CC2)=O)C(C(=O)NC(C2CCCCC2)C)C1 c1(CCNC(CC)=O)ocnc1CNC(=O)C(c1cnn(C)c1)NC(C)=O C1(C(N2CCC(OCC#C)CC2)=O)CN(C(C2(COC)CC(=O)C2)=O)CC1(C)C C1(C(N2CC(NC(N)=O)C2)=O)CCCC1NC(=O)CNc1ccccn1 CC1CC(C(=O)NC2CC(CCNC(=O)CC3NC(=O)NC3=O)C2)CN1C C(=O)(C(C)CN(C(c1ncccn1)C(=O)NCCN1CCOCC1)C)OCC c1(CCC)cc(C(=O)NCCN(C(=O)CC(C)COC)CC2CCCC2)ccn1 CC1CN(C(c2cc(O)ncn2)=O)CC(C)N1C(=O)C(C)(C)Cc1cnn[nH]1 C(C(CNC(C1CCCC(C)(C)O1)=O)S(C)(=O)=O)NC(C1(CC)CC1)=O C1(NC(C2CC(C)N(C)C2)=O)CC2CCC1CN2C(c1cnc(N)cn1)=O c1(C(N2CC(C)(C(=O)NC(CCC)C)C2)=O)ccc(CO)cn1 C(=O)(CC(C)C(F)F)NC(CN(C(CCCN(C(=O)OCC)C)=O)CC)CC C(=O)(C(F)(F)C(O)C1CC1)N1CCC(CCC(=O)Nc2c(C)nccc2)C1 c1(C2(C(=O)OC)CC2)ccc(C(=O)N(C2CCCC2)C(CC2(C#N)CC2)=O)cc1 c1(C(N2CC(OC)C(NC(=O)C(c3cnccc3C)O)C2)=O)ccc(F)c(Cl)c1 N1(C(C(COC)C)=O)CCC2CCN(C(C3CCN(C)C(=O)C3)=O)CC2C1 N1(C(CS(CC)=O)=O)CCC(C(=O)N(CC(O)COC)C)C1(C)C c1(CCC(=O)NCCN(C)C(C2CCC(CC3CC3)C2)=O)cccc(F)c1Br c1(C(=O)NCC(CC=C)NC(c2ccsc2C(F)(F)F)=O)cc2n(c1)CCC2 Cc1c(C(=O)OC2CCOC(C)(C)C2)[nH]c2cc(Cl)ccc12 N1(C(c2ccc(C)o2)=O)CC(C)CN(C(=O)CCc2nc(C)no2)CC1C N1(C(C(CCC)CC)=O)CCOC2CCN(C(c3ccc(Br)o3)=O)CC12 C1(NC(Cc2ccc(OC)cc2)=O)CCN(C(C2CCCCN2N=O)=O)C12CC2 c1(COC)nc(=NC2CCCCC2NC(C2CCN2C2CCCC2)=O)s[nH]1 c1(C(=O)NC2CC3CC(C2)N(c2nncs2)C3)ccc2ncc(=O)[nH]c2c1 c1(C(N(CCC(C)NC(C2(O)CCC2)=O)C)=O)ccc2nc(O)cn2c1 C(=O)(C(C(C)C)N1CCCC1=O)NC1CC(CCNC(C2(C)CC(=C)C2)=O)C1 C1(CC)CCCCC1C(=O)NCC(CO)NC(c1coc(C(F)(F)F)n1)=O C(c1cccc(Cl)c1)=C(C)C(=O)NCC(C1CC1)N(C)C(c1cc(C)nn1C)=O C1(CC(=O)NCC(O)CN(C(=O)CC(C)F)C)(CC)CCOCC1 c1(C(N2CC3C(CNC(Cc4cc(C)on4)=O)(C3)C2)=O)ccc(Cl)c(F)c1 C=CCCN=C(NCc1cccc(C)c1)N1CCC(C)(C(N)=O)C1 N1(C(c2nc(CC)oc2)=O)CC(CNC(c2ccccc2F)=O)CC1C C(C(=O)N(CCC(=O)N(C(C)C(C)SC1CC1)C)CCO)(C(C)C)OCC c1(C(=O)NCc2cncc(C(=O)NCC(C(C)C)CO)c2)cnn(C)c1C#N C1(C(C2CC2)NC(CCOC(C)C)=O)CCN(C(=O)C(O)CC2CC2)C1 N1(C(c2c(C)nsc2C)=O)CCC2(CC1)CC2CNC(=O)CC(=O)NCC1CC1 C1(CNC(C(C)O)=O)CN(C(c2ncc(OCC3CC3)cc2F)=O)CC(C)(C)O1 N1(CC)C(C)CN(C(c2cc(CCNC(C3CCNC(=O)C3)=O)on2)=O)CC1C N(C(=NCCC(C)O)NCC1CCCO1)CC(C)(C)OC Cc1cccc(OCC(=O)NC(C)CCCCNC(=O)CC2CNC(=O)C2)c1F C(CC(C(=O)NC(C)C(=O)NCCOC)NC(c1ccoc1C)=O)OC c1(C(N(CCCCNC(Cc2cc(C)nc(O)c2)=O)C)=O)cc(C#N)ccc1F C(C(=O)NCC(C)(C(C)C)NC(=O)C1=CCCC1)(C(C)C)OCC N1(CCCCOCC#C)CC2CCCN(C(c3nc(OC)cc(OC)n3)=O)C2C1 c1(CC(=O)NCC2CCCN(C(C3(C)CCCCO3)=O)C2)cc2ccccc2s1 C(=O)(C1=NOC(C(C)(C)C)C1)N(C1CCCN(C(c2c(CC)con2)=O)C1)CC C1(=O)N2CC(CO2)N1.c1(-c2cn(CC(=O)NCC)nn2)ccc(OC)nn1 CCCCC(F)(F)C(=O)N1CCC(N(C)C(c2ccc(CSC)o2)=O)C(C)C1 C(=O)(CCCC(C)(C)CC)NC1CCCN(C(C(c2ccccc2)OC)=O)C1 C12(NC(CN(C(C(N3CCC(OC(F)F)C3)=O)C3CCC3)C)=O)CCCC1OCC2 CC(C)C#CC(=O)NCC(C1CC1)NC(=O)CCCOc1ccccc1Br C#Cc1ccc(C(=O)NC2(CC=C)CCN(C(c3coc(C(F)F)c3)=O)C2)nc1 N1(C(c2ccc(OC)cc2F)=O)CCC(C)(C)C(NC(C2CCOC2C)=O)C1 c1(C(=O)NC(C2CCOC2)CNC(CC2CC(=C)C2)=O)cc(C(=O)OC)n(C)c1 N1(C(C(COC)C(F)(F)F)=O)CCC2C(=O)OCC12C c1(OCC)cccc(NC(C2CCN(CCc3cc(CC)[nH]n3)CC2)=O)c1 N1(C(C(C)SCC(C)C)=O)CCn2c(CNC(C3(C#N)CC=CC3)=O)nnc2C1 N(C1CCCc2nc(C)[nH]c21)Cc1ccc(OCC=C)cc1C CN1CC(O)CCC1C(N1CCN(C(=O)CCc2ncnn2C)C(CO)C1)=O C1(C)(NC(c2c(C)cco2)=O)CCN(C(C2CCCC2c2nc(S)n[nH]2)=O)CC1 C1(NC(C(C)N(C(C2(CC=C)CCOC2)=O)CC)=O)CC(=O)N(CC2CC2)C1 CC1=C(C(=O)N2CC3CC2CCC3NC(c2coc(C)n2)=O)CCCO1 c1(C(N2C3(CNC(CC4C(C)CCC4)=O)CC(C2)C3)=O)cc(N)cc(O)c1 c1(C(N2CCC(CNC(C3(C)CCOCC3)=O)C2)=O)ccc2c(c1)CC(=O)N2 C(C)(CCC(=O)NC1CCC(CC(=O)NCc2nnc(O)n2C)C1)OCC Cc1ccccc1C=CC(N1CCN(C(c2cccn2C)=O)C(C)C1)=O C#CCC(CC(=O)NCCCO)NC(=O)CCCCCSC c1(OC)cc(NC(C2CCOCCN2C(C2CCC2C#N)=O)=O)cc(F)c1 C1(C)(CC)CCN(C(C2(CNC(c3cnc(C)cn3)=O)CC=CC2)=O)CC1 c1(C(C(=O)NCC2CCOC2)N(C2CC2)CC)cc(F)ncc1F c1(C(N(C)CC2CN(C(C3(SC)CCC3)=O)C2)=O)cc2nn[nH]c2cc1F C1(OCC(=O)NCC(n2cncn2)C)CCN(C(c2cnc(C3CC3)s2)=O)CC1 c1(OCCCCCC)ccc(-c2csc(CN3CCC(C(C)(F)F)CC3)c2)cc1 C#CC1(C(=O)N2CC=CCO2)CCN(C(=O)CSC(F)F)CC1 CC(C)(CS(C)(=O)=O)NC(=O)CCCc1ccc(F)c(F)c1 n1(CC)cc(C(=O)NCC(c2ccccc2)NC(c2csnc2C)=O)c(C2CC2)n1 C1(NC(C2(CC=C)CCOC2)=O)C=CCC(C(=O)NC2CCCSC2)C1 C(C1Cc2ccccc21)N(c1ncc(C#C)cn1)C.c12ccccc1CNC2=O c1(NC(C2=CCN(C(CC3CC(=O)NC3=O)=O)C2)=O)cccc2c1CCC2 c1(C(N2C3CN(Cc4ccc(C(F)F)cc4)CC23)=O)cc(F)c(Br)c(F)c1 C1(CC)CN(C(c2nocc2Br)=O)CCN1C(c1[nH]cnc1CC)=O n1(CCC(=O)NC2C(CNC(COCCCCCC)=O)CCC2)ccccc1=O C1(C)(C(=O)NCCN(C2CCCC2)C(c2ccc(SC)o2)=O)CC2CC2C1 Cc1ccc(F)cc1C(=O)NC1CC(NC(C2CCC3CC23)=O)CC1O c1(C(=O)NCC2CCCN(C(CCCCC)=O)C2)cnn2c(Cl)cccc12 C1(C)(C(=O)NC23CC(CNC(C(c4ccn(C)n4)C)=O)(C2)C3)CCCN(C)C1 c1(OCC)ccc(O)c(CNC(c2ccc(C#N)cn2)CCc2ccccc2)c1 N1(C(C(C)=C(C)C)=O)CCC2(C1)CN(C(C1CC3CCC1O3)=O)C2 C1(OC)CC2CC(C(N3CCN(CCCNC(=O)C#CC4CC4)CC3)=O)CC12 c1(C(N2C(C)C(NC(=O)CC3(N(C)C)CC3)CC2)=O)cnn2c1S(=O)(=O)NCC2 O=S(=O)(c1c[nH]ccc1=NCC1CCC12CCOCC2)NCCc1nncs1 N1(CC(=O)NCC(C2CCCCC2)NC(CCS(C)=O)=O)C(=O)CC(C)(C)C1=O N1(C(c2ncc(CC)s2)=O)CC2CC1CN2Cc1c(C)nn(CC)c1C C1(NC(=O)Cc2cncc(F)c2)CC2(CCCCN2C(=O)CC2C=CCC2)C1 Cc1ccc(F)c(C(=O)NC(C2CCCN2C(=O)CCCc2sccc2C)C)c1 O=C(CCCC(F)(F)F)NC1(CNC(=O)C(O)C2CCCC2)CCOCC1 c1(C(N(CCNC(C2CC2OC(C)(C)C)=O)CC)=O)c(F)ccc(N)c1F C(C)(C)(CC(F)C(=O)NCc1cnc(C)n1CC)NC(C(C(CC)O)C)=O c1(C(N2CCN(C(CC(C=C)CC)=O)CC2C)=O)cc2ccccc2[nH]1 C(=O)(CS(N)(=O)=O)N(CC(C)O)CCNC(=O)CCN(C)CCc1ccccc1 c1(OC)cccc(C2(C(=O)NCC3CN(Cc4ccc(=N)[nH]c4)C3)CC2)c1F C(C1C(C(=O)NC2CCN(C(=O)CNS(=O)(=O)CCCC)C2)C1(C)C)=C(C)C Cc1ccn(C(C)C(=O)NC(C)CCCNC(=O)C(O)Cc2cnc[nH]2)n1 c1(C(C(=O)NC(C)CCNC(=O)COCC(F)(F)F)(F)F)nc2ccccc2s1 CC1(C)C(NC(=O)CN(c2ccncc2)CCO)CCN1C(C1COCCO1)=O Cc1ccc(C(=O)NC2(CCNC(=O)CCNC(=O)CO)CCCC2)c(=O)n1C CC1CCn2cc(C(N3CCC(c4nnc5ccccn45)CC3)=O)nc2C1 C(=O)(CCCCC(=O)c1ccccc1)NCC1N(C(CCCOC)=O)CC(O)C1 CC(CS(C)(=O)=O)C(=O)N1CC2CCN(C(=O)CC3CCCCCCC3)C2C1 N1(C(C2C(OC)C2)=O)CC2CCCC2(NC(C23CC(CF)(CO2)C3)=O)C1 c1(C(=O)NCC(=O)NC(C)CC(C)NC(c2cnnn2C)=O)ccc([N+](=O)[O-])cc1 CC1CN(C(=O)C(c2ccc(F)cc2)=O)CC1NC(=O)CC1CCC(=O)N1 C1(CNC(C(CC)(C)CC)=O)CN(C(=O)CC2(C(F)F)CC2)C2CCN1C2 CCC(C(=O)NC1CCC(CCNC(=O)COc2ccon2)C1)SC CC1(C)CCN(C(C2CCCC2NC(c2ccc(OC(F)(F)F)cn2)=O)=O)CC1 C1(F)(CNC(CC(C)OC)=O)CCC(CNC(=O)Cn2nccn2)C1 C1(NC(CCCC#CC)=O)COC2CN(C(C3C=CCC3)=O)CC12 CCC(O)C(F)(F)C(=O)NCC1CN(C(c2ncccc2Cl)=O)CC1(F)F C1(CC=C)(C(=O)NC(c2csnn2)C)CN(C(=O)CCC2CC2(C)C)C1 C1(CC(=O)NC(C2CCCC2)CNC(C=C(C)C(C)C)=O)COCCN1C N1(C(C(C)CC2CC2)=O)CCC(C(C)(O)CNC(C2SCCS2)=O)CC1 CC(C)CC(C)C(=O)NCC(C)(C)CNC(C1CN(C(N)=O)C1)=O C12(C)CCN(CC1)C(=O)Cn1cc(nn1)C2.C1(=CC(=O)OC(C)(C)C)CCOCC1 C1(CC(=O)NC(CCC)(C)CC)C2CCC(C2)N1C(=O)C=C=C(C)C CN=c1cc(C(=O)NCCCC(C)NC(=O)CCCc2cc(C)no2)cc[nH]1 c1(C(N2C(CNC(CCC=C=C)=O)CC(O)C2)=O)cc(C)c2nc(C)cn2c1 c1(CC(=O)NC2(C)CN(C(C3CC4(CSC4)C3)=O)C2)ccc2ccccc2c1 C1(CNC(c2nc(C)n(C)n2)=O)CN(C(=O)C(C)O)C2(CCC2)C1 CC(C)(CNC(C1COCCC1NC(c1cc(C2CC2)no1)=O)=O)CC(F)F C1(C(N(CC(C)O)CCNC(c2c(C)con2)=O)=O)CSC(c2ccccc2)=N1 C1(NC(=O)OC(C)(C)C)CCCOC1CC(=O)NC1(CC(N)=O)CCOC1 c1(C(=O)NCC(C(=O)N(CCOC)CCO)OC)cc(CSC)n(C)n1 C1(CNC(CN(C=O)C2CC2)=O)CN(C(c2ncncc2F)=O)CC12CC2.C(=O)OC c1(C(=O)NC2CC(CCNC(C3N(C=O)CCC3)=O)C2)cc2ccccc2o1 C(=O)(C(F)(F)C(F)(F)C(F)(F)F)NC(C1OCCN(C(C=C(C)C(C)C)=O)C1)C c1(C(N2C(CNC(=O)C(F)(F)c3cnccn3)CCC2)=O)ncc(F)cc1F N1(C(C=C(CCC)C)=O)CC(O)(CN(C(=O)Cc2cn(CC)nn2)CC)C1 C1(NC(c2ccc[nH]2)=O)CCN(C(c2cnn(-c3ccccn3)c2)=O)C12CCC2 C1(C(=O)OCc2c(OCCC)cccc2)CC(=O)NC1(C)C CC(CNC(C1CCCC(CF)C1)=O)CN=[N+]=[N-] N1(C(c2c(C)cco2)=O)CCC2(CC2C(=O)Nc2cc(O)ccc2C)C1 N1(C2CCN(C(C3C(C)(Br)C3)=O)C2)CCN(Cc2ccc(C(F)(F)F)s2)CC1 C1(O)(CCNC(C=CC(C)N(C)C)=O)CCN(C(=O)CC(C)N(C)C)CC1 C1(NC(C(C)n2ccnc2)=O)CCC2CC1CN2C(C12CCCC1CCC2)=O c1(C(N(CC(C)NC(c2ccc[nH]2)=O)CC)=O)cccc(OCCOC)c1 N12CCCCC1C1CCCN1CC2=O.c1(CN(CCC#N)C(C)C)ccccc1 N1(C(c2ccc(F)s2)=O)CCOC2CN(C(C3(F)CC3)=O)CC12 C12(C(N3CC(CNC(C(C4CCC4)OCC)=O)C3)=O)CCC(O)(CC1)CC2 C1(CCOC)CN(C(c2coc(Br)n2)=O)CCN1C(=O)CCS(N)(=O)=O c1(OC)ccc(CN2CCC3(CCC3)C2)cc1NC(=O)Cc1ccoc1 C(=O)(CCC(=O)NCC1CC(NC(c2cc(Cl)n(C)n2)=O)C(O)C1)OCC c1(C(=O)NCC2(C(N)=O)CN(C(CSC)=O)C2)cn(C)cc1C(F)(F)F N1(C(c2ccc(C(F)F)cc2)C)CCCC(C(N2CCCC(N)C2)=O)CC1 Cc1ccc(Cl)c(C(C(=O)NC2COC2)N(C)CC2CC2)c1 N1(C(c2nc(CC)oc2)=O)CCC(N2CCNC(=O)C2C)C(C)CC1 CC1OC2CCC1(C(=O)NCC(C)CNC(=O)CSC1CC1)C2 C1(N(C(CSCCOC)=O)C)CCCC(NC(C2CNC(=O)C2)=O)C1 c1(C(=O)NC2CC(C(C(=O)N(C3CCCCC3)CC)F)C2)nnc(O)nc1O C12(C(=O)NC3(C(N)=O)CC3)CCC(F)(CC1)C2.C1(C(C)(C)C)CN2CC1C2=O c1(OC(C)C)cccc(C(=O)NC(C2CCN(C(=O)C(C)N(C)C)C2)C)c1Cl N1(C(C(C)N=[N+]=[N-])=O)CCC(C(=O)Nn2cncn2)C(O)C1 CC1(OCC(=O)NCC(C2CCC2)NC(C2CC2CF)=O)CCOCC1 CC(CCCCNC(=O)C=Cc1cn(C)nn1)NC(=O)C(c1ccc(Cl)cc1)=O C1(C(=O)NCCCCC(C)NC(CCC(=C)C)=O)CN2CCCC2CO1 C1(CNC(CC(CN(C)C)O)=O)CC(C(=O)NCC(O)C(N)=O)=NO1 C1(CNC(COCCOC)=O)CC(F)(F)CN1C(c1cc(C(C)C)ccc1C)=O CCC(CC)(CCNC(=O)CC1CC=CCC1)NC(C1(C)CCCN1C(C)=O)=O C1(NC(=O)C=CCC2(NC(=O)CCc3cnoc3)CCC2)Cc2ccccc2C1 N1(C(CSC(C)C)=O)CCCC(C2CCN(C(c3cccc4sccc34)=O)C2)C1 Cc1cccc(C#CCO)c1NC(=O)C(C)C(C)CN CCN=c1[nH]c(C(=O)NC2CN(C(=O)CC=C(Cl)Cl)C(C)(C)C2)cs1 c1(C(C)OCC)noc(CCC(=O)N(CC(O)CNC(C2(Cl)CC2(F)F)=O)C)n1 c1(CCCC)nc(C)c(CC(=O)N(C2CCN(c3nnc(CC)s3)C2)C)s1 c1(OC2(C)CN(C(=O)C(C)(C)O)C2)ccc(F)cc1F.C1(C(=O)NC)(NC=O)CC1 c1(CC)nocc1C(N1CC(C(C)NC(c2cc(CO)[nH]n2)=O)C1)=O C1(C(NOC(CC(=O)NCCC(C)O)=O)=O)(C2CC2)CCCO1 N1(C(C(C(C)C)SCC)=O)CC(CC(N2CC(N(CC(C)C)C)C2)=O)C2(CC2)C1 c1(OC)cc(C(=O)N(CCCNC(C2CCCCC2C)=O)C(C)C)cnc1O CC1CCc2c(C(=O)NC3CCC(NC(=O)CC4COC(=O)C4)C3)csc2C1 c1(C(C(N2CC(OC)C(F)C2)=O)NC(=O)C2CC2)ccc(Br)c(Cl)c1F c1(C(COc2ccc(C(=O)OC)c(C)c2)=O)ccc2c(c1)c(C)c(C)n2C=C(C)C N1(C(c2c(C)nc3sccn32)=O)CCC2(CC1)CC(NC(C13CC(C1)C3)=O)CO2 C1(NC(c2c(CC(C)(C)C)cccc2)=O)CC2CC1N(C(c1cncs1)=O)C2 C=C(Cl)CC(C(=O)NC(CC1CC1)C1CC1)NC(c1nnc(O)nc1O)=O c1(C(=O)OC)nc(=NC2CN(C(=O)NCC3CC(C)CC(C)C3)C2)cc[nH]1 c1(C(N(CC(C)O)CCNC(C(CC)NC(N)=O)=O)=O)cnn2c1NCCC2 C1(C(N2C(C)CCCC2C(N2CCOCC2)=O)=O)Cc2cccnc2C1 c1(C(C(=O)NCCSC)N(C2CC2)CC)ccc(C(C)(C)C)cc1 N1(C(Cc2cccc(C)c2F)=O)CCCC12CCN(C(=O)CN(C)CCO)CC2 N1(S(C(C)C)(=O)=O)CC2(CCC(NC(c3cc(Br)cnc3O)=O)CC2)C1 N1(C(C(CC(F)F)NC(c2c(C)csn2)=O)=O)CCCCN(C)CC1 C1(C)(CNC(c2cc(COC)sc2)=O)CCCN1C(c1c[nH]nc1C)=O c1(C(C)NC(c2csnc2C)C(=O)NCCCF)cccnc1OC(F)F Cc1nn(CC(=O)NC2COCC2NC(C2CCC(C)(C)O2)=O)c(=O)n1C C1(C(=O)NC(CC)C(C)O)CC=CCN1C(C1CCCC1F)=O c1(OC)ccc(F)c(C(N2CCCN(C(c3cnn(C)c3)=O)CCC2)=O)c1N c1(CN(CCN2CCCCC2)CC2CCN(C)C2)c[nH]c2nccc-2c1 C#CCCC(C(=O)NCC1(O)CCCC1(C)C)NC(=O)CCCCC CCCCC(CC)C(=O)NC1(CO)CCN(C(=O)Cc2nc[nH]n2)C1 c1(C(=O)NCC2N(C(C=CC(C)(C)C)=O)CC2)cc(-c2ccco2)on1 N1(C(C(CC)SCC)=O)CCN(C(c2cccc(C#N)c2)=O)CC1C1CCCC1 c1(C(N2CC3C(NC(c4ncccc4F)=O)(C3)C2)=O)cc2c(Cl)nccc2o1 N1(C(C=Cc2n(C)cnc2)=O)CC2(CCCCN(C(c3cccnn3)=O)C2)C1 c1(-n2ncc(C(=O)NC(C)CNC(C3(CO)CC3)=O)c2)ccc(Br)cc1 Cc1c(C(=O)NCCCCNC(C2(C)CCC(C)(C)CC2)=O)nn2ccccc12 Cc1ccc(F)c(C(=O)N(C(C)CNC(=O)C(C)(C)CN2CCOCC2)C)n1 C(=O)(C1=CS(=O)CCC1)NCC(N1C(C)CCN(C(=O)CC(C)(C)C)CC1)=O c1(NC2C(CC=C)C(O)C2)ccnc(OC)c1Br C(=O)(C(C)(C)CNC(c1nc(Br)sc1Br)=O)NCC N1(C(c2ccn(C)c2)=O)C2CCC1CC(C(N1CCCC(OCC(N)=O)C1)=O)C2 CC1CC2CN(C(=O)CC(C)(C)F)CC2N1C(c1cccc2ccncc12)=O C1(CC(=O)NC2(C(=O)OCC)CC2)CN(C(=O)Cn2nccn2)C(C)(C)C1 Cc1cc[nH]c1C(N1CCC(N(C)C(c2csc(CC(F)(F)F)n2)=O)C1)=O C=CC1COCCN1C(C1CC(F)CN1C(c1ncccc1N)=O)=O N1(C(CCSC)=O)CCC(NC(=O)CCCn2nc(C)nc2C)C(OC)C1 C1(C(N(C2CCN(CC3CC3C3CC3C)CC2)CC#C)=O)C2CCCCCCC12 CCCCCCCCNC(C1C2CCC(C2)N1C(c1cc(CO)ccc1Cl)=O)=O Cc1c(C(=O)NCC23CC2CN(C(=O)CC2(C)CC2)C3)noc1-c1ccccc1 c1(C(=O)NCCCCC=C)cc2ccc(-c3cc(C)cnc3OCC)cc2o1 C1(NC(C2CC2C2CC2)=O)CC12CCN(C(c1cnn(-c3ccccc3)c1)=O)C2 C(=O)(C(CNC(C1CC1Cl)=O)N(C)C)NCCCOC C(=O)(N=c1ccn(CCN(C)C)[nH]1)C12CC(c3ccc(CCC)cc3)(C1)C2 C(CC1c2ccccc2CCN1c1nnn(C)c1N)NC(CCC=C)=O c1(CC)ncncc1C(=O)NC1CC2(C1)CC2C(=O)NCc1cc(C(N)=O)co1 N#Cc1cccc(C2(C(=O)NCC(O)CNC(=O)CCCC3(CO)CC3)CC2)c1 N1(C(CCC(C)NC(c2cc(=O)n(C)cn2)=O)=O)CC2CC1C(F)(F)C2 C1(C(=O)NCCCn2c(C)ncc2)CC(O)CN1C(c1ccco1)=O C(=O)(C(F)(F)C(N)=O)NC1CCC(CC(=O)Nc2ccc(COCC)cc2)CC1 c1(C(N2CCCC(F)(CNC(C(CO)N(C)C)=O)C2)=O)cc2ncccc2s1 c1(C(=O)NCC(C)NC(C2OCCOC2(C)C)=O)n[nH]c2c1COc1ccccc1-2 C1(CC(=O)NCc2ccncc2N2CCOCC2)CCc2ccccc2N1 C(C(=O)N1CCC(NC(=O)CC2CCC2(C)C)CC1)(C(C)C)NC(=O)OC c1(N(C)C)ccc(C(=O)NC2CC(C)(NCC=CC(F)(F)F)C2)nc1 c1(C(N2CCC(C(C)NC(c3ccc(O)nc3)=O)C2)=O)ccc(O)nc1Cl C#CCC(C)(C)C(=O)N1CCCC1CN(C(=O)Cc1cccc(C(C)(C)C)c1)C C(C(C)(C)CC(=O)NC1C(C(=O)OCC)C1(C)C)NCCCN(C)C(C)C c1(C(=O)NCC2C3N(C(C(C)SCCCC)=O)C(CC3)C2)cc(N)c(O)c(F)c1 c1(C(N2CCC(C#N)C2)C(=O)OC)nc(Br)ccc1F.C(C(F)F)OCC C1(O)(C(=O)NC2CN(C(CC3C(C)(C)CCO3)=O)C2)Cc2ccccc2C1 CC(C)C(C(=O)N1CC(NC(c2ccc(CSC(F)F)o2)=O)C1)c1cnn(C)c1 C1(C(=O)NCCC2CC(C)N(C(=O)CCOC3CC3)CC2)CCC2(CCC2)CC1 c1(C(CC)NC(C2(CNC(=O)CC(=O)OC)CC2)=O)ccc2nccnc2n1 C(CCCCC(=O)NC1(CN(C)C(C2(C)CCCC2C)=O)CC1)=CC c1(NC(C(C)C)CNC(c2cc(C(C)(C)C)no2)=O)cc(=O)n2ccccc2n1 c1(SC)ccc(CCC(=O)NC2CC(C)(CNC(c3cccnc3)=O)C2)cc1 C(=O)(CCC(C(C)C)NC(C12CCC(C1)C2)=O)N1CCC(C#C)CC1 n1(CCOC)nccc1C(=O)NC(CNC(=O)CSc1ccccn1)C(C)C C(=O)(C1=CCCSC1)N1CCC(CCNC(C(C(C)C)SC)=O)C1 c1(C(N2CCCC(O)(CCNC(C(CCC)(C)C)=O)C2)=O)cccc2occc12 c1(C(=O)OCC)cc(Br)ccc1N(C)Cc1sc(C)cc1C c1(NC(C2CN(C(c3cccc(C)c3)=O)C2)C)cc(Cl)nc(CC(C)C)n1 C1(CC)(NC(=O)C(c2ccoc2)NC(=O)Cc2cc(C)[nH]n2)CC2CCC1C2 C(C(C)C(C)(C)C)N(C(C(CSCC)NC(c1cnsn1)=O)=O)C C1(C(=O)NC(CNC(CC(=O)OCC)=O)(C)C2CCC2)CCC2CC1C2(C)C N(C(=NCCCF)NCC1(C2CC2)CCC1)Cc1c(OC)nccc1 c1(OC(C)C)cccc(-c2nc(C3CNCC3C)no2)c1 CC(CC(=O)N1CCC(C)(NC(c2ccc3c(c2)CC3)=O)C1)CC(C)(C)C c1(C(C(=O)NCCN(C(c2c(CC)csc2)=O)CCOC)C)cccc(Cl)c1 CC(C)(CC(F)(F)F)C(=O)NC1COCCC1NC(=O)CN1CCCOC1=O C(C)(C(=O)N1CCC(N(C(=O)Cn2nnnc2C2CC2)CCO)C1)(C(C)C)OC N1(C(C2(OC)CCC2)=O)CCCC(CNC(=O)C(CO)c2ccccc2)CC1 c1(C(N2CC(C=C)OCC2)C(=O)NC2CCCC2)cccn2ccnc12 O=C(CCCn1cc(-c2cccn2C2CCCC2)nn1)NCS(=O)(=O)N1CCCC1 C1(CC=C)(NC(C2CC(CNC(=O)COC3CC(F)(F)C3)C2)=O)CC=CC1 C1(OC)CC(C(N2CC=CC(NC(C3CC=CCO3)=O)C2)=O)CC1OC N1(C(c2ccnc(C)n2)=O)CC2CCCC2(NC(=O)CC2CCC(C)(C)O2)C1 C(=O)(C(C)(C)CN(C)C)NC1(CN(C(C2CCC(CCCC)C2)=O)C)CC1 C12CN(CC1C)C2=O.c1(OCC=C)ccc(C(=O)OC)cc1 C1(NC(=O)COC2CCOC2)C2CCCCC12.C1(OC)CC2N(C1)C2=O c1(C(N2CC3C(CNC(C(C4CCCC4)OC)=O)(C3)C2)=O)cc(C)cc(F)c1 c1(NC(CC)C(=O)NCC2COCCN2C(=O)Cc2cc[nH]n2)ccccc1F c1(C(N2C(C)CC(CNC(=O)C#CC3CC3)C2)=O)ncc2ccccc2c1O N1(C(C(C)C(=O)N2CCOCC2)=O)C2CCC1CN(C(C1(CF)CC1)=O)C2 c1(C(=O)NC2C(N(C)C)COC2)cc(OC)ccn1.C1=CC(=O)NC(C)(C)C1 C(c1ccc(F)cc1)=CCC(=O)NCC1C=CC(NC(=O)C2=CCCOC2)C1 c1(C(=O)NC2CN(C(c3c(C)cccn3)=O)CC2C)cccc2c1CCC2=O c1(CNC)ccc2c(c1)CN(S(=O)(=O)C1CCOC(C(F)(F)F)CC1)CC2 Cc1nc(NCC2(O)CN(C(=O)CCc3cc(C)on3)C2)c2cnn(C)c2n1 N1(C(c2cc(C(N)=O)ncc2)=O)CCN(C(=O)CC2CNC(=O)O2)CC1C(F)F c1(C(N2CCCN(C(Cc3cnc(C)s3)=O)C(C)C2)=O)cc([N+](=O)[O-])cnc1N c1(CC(CNC(CCN(CCC)C)=O)N(C(=O)CC(=O)N(C)C)C)ccccc1 Cc1cc(CN2CCC(N(C(C)C)C(c3nnc(N(C)C)o3)=O)CC2)cc(C)c1 c1(C(=O)NCCC(C)NC(CCSCC)=O)cc(C)ccc1[N+](=O)[O-] C1(C(OC)OC)CCC(CN2C=NC(CC(=O)N)C2)CC1.C(C)(C)(C)OC(=O)N c1(C(=O)NC2CCCN(C(C3(C)CC(C)OCC3)=O)CC2)ccc2c(c1)CCC2 N1(C(c2n(CC=C)nnn2)NC(C)C(=O)NCCC)CCOCC1=O C1(NC(c2n(C)nnc2)=O)CCCN(C(=O)Cc2ccc(Cl)cc2Br)CC1 CCCCC(CNCc1nc(-c2cccc(C#N)c2)cs1)CC C1(C(C)NC(=O)C=C(Cl)Cl)CCCCN1C(c1cccc(F)c1)=O C(=O)(CCCCC#N)N1CCC(C(=O)NOCC(=C)Cl)(CC#C)C1 c1(C(=O)NCC(C)NC(c2cc(O)cc(Cl)c2)=O)cc2sccc2n1C C(C)(CC(=O)NCCCCN(C)C(c1cn(C(C)(C)C)cn1)=O)SC C1(CNC(c2ccc(C)s2)=O)CN(C(=O)CC2(O)CCCC2)C(C)(C)C1 CC(C)C(F)C(=O)NC1CCC(CNC(c2ccccc2Br)=O)CC1 c1(CC(=O)Nc2scc(C(=O)NC(C(C)O)CO)n2)cc(F)ccc1F c1(N(C2CCN(C)C(=O)C2)C(N(CCC)CC2CC2)=O)ccc(C)c(C)n1 C1(OC)CC2(C1)CC2NC(N1CCC(NC(=O)CCOC(C)=O)C1)=O C1(NC(=O)Cn2nnc(=O)[nH]2)CN(C(c2coc(Br)n2)=O)CC12CCOCC2 c1(C(=O)NCC2(NC(c3onc(C)c3C)=O)CCCC2)c2c(c[nH]c1=N)CCC2 C(=O)(C(C(C)(C)C)n1ccnn1)NC1CN(C(C2(C)CCCO2)=O)C1 N1(C(C(CC)C#N)=O)CCCC(N(C(=O)C=Cc2cccs2)C)CC1 CN1CCCCC1C(N1CCC(O)(C(C)CNC(C2(CO)CC(F)(F)C2)=O)C1)=O C(=O)(N1OC2CCC1C2)C1(F)CCCN(C(C(COC)C)=O)C1 c1(NC(C2C(F)CCN(C(CCOC)=O)C2)=O)ccc2occc2c1O CC1COCC(CC(=O)N(CC(CO)(CO)NC(=O)COC2CC2)C)O1 N1(C(CN(C(C)=O)CC)=O)CSCC1C(=O)NC1CN(C(=O)COC)C1 C#CCC(C(=O)N(C)CC1(F)CCC1)NC(=O)Cn1ccccc1=O C12(C(N(CCSC)C)=O)CC1CN(C(C1COCC1(C)C)=O)C2 C(=O)(C(C(C)(C)C)OC)N1CC(CN(C(c2c(OC)scc2)=O)C)OCC1 N1(C(C(C(C)n2cccn2)C)=O)CC2CC1CCC2NC(C1CCC(=O)N1)=O n1(CC(=O)NCC2(C(N)=O)CN(C(CNC(CCC)=O)=O)C2)ccccc1=O N1(C(C(C)CC(C)(C)C)=O)C2CCCC1CN(C(=O)C=CCN1CCCC1)C2 N1(C(C(OC)OC)=O)CCN(C(=O)C(c2cncn2C)O)CC1c1ccncc1 CCCC(C(=O)NC1CCN(C(=O)C(C(C)O)N(C)C)CC1)NC(N)=O C(=O)(C1=CCCCC1)N1CCCC(C(C)NC(c2nc(Cl)c(Cl)s2)=O)C1 Cc1ccc(N)c(C(=O)NC2(N(C(=O)C(c3cccnc3)C)C)CC2)c1F C(=O)(CCC(=O)N(CCN(C)C)Cc1n(CC)ccn1)N1C(CC2CC2)CCC1 C1(NCc2c(CC)cccc2)CN(C(C2CCS(=O)(=O)C2)=O)CCC1F C(=O)(C(=O)N=S(C)(C)=O)NC(CC(C)C)CNC(C1(N(C)C)CC1)=O c1(CN2C3C(C(=O)NC(c4nn[nH]n4)C)C(C3)C2)ccc(F)c(O)c1 C(=O)(C1=CCS(=O)(=O)C1)N(CC(O)CNC(c1ccccc1-c1nc[nH]n1)=O)C C1(C(N2CC(C(C)NC(c3ccc(C(C)C)cn3)=O)C2)=O)CCC(C#N)CC1 C1(CNC(C(C)(C)OC)=O)CC2(CCOCC2)CN1C(c1cnc(C)n1C)=O C1(C(=O)NCCC(C)C2CC2)N(C(c2ncn3ccccc23)=O)CCCC1(C)C CC1(O)CCN(Cc2[nH]c(-c3ccccc3)nc2Cl)CC1(O)c1ccccc1 c1(C(N2CCN(C(C3CC3F)=O)C(CC(F)F)C2)=O)cn2ncccc2n1 C(CC(=O)N1CC(CNC(=O)C(C2CC2)SC)C1)NC(=O)OC N1(C(c2c(C)[nH]c(C(C)(C)C)c2)=O)CC2CCC1CN2C(C1CC1(F)F)=O c1(-c2onc(C)n2)ccc(NC(=O)NCC(C(F)F)N2CCCC2)cc1 c1(C(N(CCCN(C(C(C)c2ccco2)=O)C)C)=O)ncn(-c2ccccc2)n1 CCC(C(O)C(C)C)NC(C1C2CC3C(C2NC(=O)CCc2ccnn2C)C13)=O c1(C(C)(CO)NC(=O)CC2CC3CCC2O3)ccccc1Cl C1(C(=O)NC(Cc2c(C)noc2C)C)CN(C(c2ccncc2)=O)CCC1O C(=O)(C1=CCN(C(C2CC3C=CC2CC3)=O)CC1)N(C1CCOC1=O)C c1(NC2CC=C(C)CC2)ccc(S(=O)(=O)N2CCc3ccccc3C2)cc1Br C1(CNC(CNC(c2c(C)occ2)=O)=O)CCCCCN1C(C1CC(C#N)C1)=O N1(C(C(C)=C(CC)C)=O)CC2CCCC(C1)N2C(c1c(Cl)noc1C)=O N1(C(Cc2cc(C)c(Cl)cc2)=O)CC(CNC(=O)C2=NNC(=O)C2)C2(CCC2)C1 C1(C(N(CC(CC)NC(C2CC(=C)C2)=O)CC)=O)CC(c2ccccc2)=NO1 C1(C(N2CCC(c3cn[nH]c3)CC2)=O)(OC)CCN(Cc2cccc(O)n2)CC1 N1(C(C=CC(C)NC(CC(CC)C2CCC2)=O)=O)CCC(C2(O)CC2)CC1 C1(CNC(c2ccc(CC)cc2)=O)CC(NC(c2ncccc2O)=O)C12CCC2 C(c1ccco1)=C(C)C(=O)NC1(CO)CCCC1.N12CC(C)(C1)C(=O)NO2 N1(C(c2ccnc(C)c2N)=O)CC2CCC1CN2C(C1CC2(CCC2)CO1)=O N1(CCC(=O)NCC2CCN(C(c3c(C(C)C)n[nH]c3)=O)C2)CCP(C)(=O)CC1 N1(C(c2cc(C(C)C)nn2C)=O)CC(NC(C2CC2(C)Br)=O)C2(CCOCC2)C1 N1(C(CN2C(C)CC2)=O)CCCOC(CCNC(=O)CN2C(=O)CNC2=O)C1 CC(C1CC1)=C(F)C(=O)NCC(O)CNC(C1CC(OC(F)(F)F)C1)=O N1(C(CN(CCC)C(C2CCN(C3CC3)C2)=O)=O)CC2(CCCN2C)C1 C(CCCC)(CC(=O)N1CCCC(CC=CC)C1)NC(CCC#C)=O c1(OCC(=O)NC2CC(NC(=O)CC3CSCCS3)C2)ccc2cnccc2c1 c1(C(N2CC3(CCC3)C2)=O)ccc(-c2ccc3c(c2)C(=O)NC3)c2c1OCO2 C(C(C)NC(=O)C=CCNC(C1CC1F)=O)N(C(C)C)C n1(CC)nc(C)cc1C(N1CCOCC1CNC(C1(CO)CC(F)(F)C1)=O)=O CC12OCC(CO1)NC(C1(NC(=O)C(=O)Nc3ccc(F)c(Cl)c3)CC1)C2 c1(C(=O)NCC(C(C)(C)C)NC(CC2(COC)CC2)=O)ccc(Br)c(N)n1 N1(C(C(C(C)(C)C)SC)=O)C2CCC1CN(C(c1cnccc1Cl)=O)C2 C1(NC(=O)CC2CC(F)(F)C2)CCC2(CCN(C(=O)C(O)C3CC3)C2)C1 c1(C(N2CC3C(CNC(c4cnn(CCO)c4)=O)C3C2)=O)cccc2[nH]ccc12 C1(F)(CNC(CSCCOC)=O)CCC(NC(=O)C(c2cccc(C)c2)C)C1 Cc1cccc(CC(=O)NC(C)(CNC(C2C(C)C2(F)F)=O)C(C)C)c1Cl C(c1ccc(C)cc1)=CC(=O)NCC1N(C(C(C)OCCCC)=O)CC(OC)C1 C1(C(=O)NC2C(CNC(CSC)=O)CC2)CN2CCN1C(C)C2 N1(C(CC(CC)C)=O)CCC(CC(N)=O)(NC(C2CCCS(=O)(=O)N2)=O)CC1 N1(C(C2N(C(c3c(CC)cco3)=O)CCC2C)=O)CC2CC3CC2C1C3 c1(C(N)=O)ccc(C=CC(=O)NC2CC(NC(C3C4CCC3CC4)=O)C2)o1 Cc1ccc2cc(S(=O)(=O)N3CC(S)CC3(C)C)ccc2c1 c1(C(=O)NCC2CC(C)(C)N(C(=O)C3=NOCC3)C2)cc(F)cc([N+](=O)[O-])c1N C1(C(=O)NC(C(=O)NCC2CCC(C)(C)C2)Cc2ccoc2)CCCCC(=O)N1 c1(C(N2CCC(O)(C(C)NC(C3CC(OC)C3)=O)C2)=O)n[nH]c2c1CC(C)CC2 CC(C)(CC(=O)NCC(C(F)(F)F)N1CCN(C(C2CSC2)=O)CC1)C1CC1 C1(C(C)NC(C2(F)C(C)C2)=O)CCN(C(C2(c3ccccc3)CC2(F)F)=O)CC1 c1(CN(C(C)C)C(=O)NC2CN(C)C3(CCCC3)C2)ccc2c(n1)NCCC2 c12cccc(c1O)OC(=O)c1ccccc1-2.N1(CCC)CCC2(CC2)C1 Cc1ccc(C=CC(N2CC(NC(=O)C3=CCOCC3)C3CCCC23)=O)c(C)c1 C1(CC(=O)N(CC(C)NC(c2n(CCCC)ncc2)=O)CC)COCC1(C)C N1(C(C2CCCN(S(C)(=O)=O)C2)=O)CCC(C)CC1CNC(=O)CC(F)(F)F C1(NC(Cc2ccc(C)nc2)=O)CCCC12CCN(C(=O)CSCC(N)=O)CC2 c1(CC)ccc(C(=O)NCCOCCCNC(C2CC3CCC2O3)=O)cc1 C1(C(=O)NC2C(CC)N(C(c3cc(C)c(F)cn3)=O)CC2)CC12CCOCC2 C1(C(N2CC(NC(C(C)CC3CCC3)=O)C2)=O)CCN(c2cccc(Cl)c2)C1=O Cc1ccn2ncc(C(=O)NC(C)CCNC(C3(NC(N)=O)CCCC3)=O)c2c1 C1(CC(=O)NCCC2N(C(c3c[nH]c(=N)s3)=O)CCC2)(N(C)C)CCCCC1 C1(NC(c2c(CNC(c3scc(C)c3)=O)noc2)=O)CCCCCC1C(N)=O c1(C(=O)Oc2c(Br)ccc(C)c2)cc(F)cc2ccoc12 c1(C(=O)NCC(CC)NC(=O)OCC)ccc(CC)nc1O.C1C(=O)N1C Cc1ncnc(C)c1CC(N1CCN(C(=O)CC2CCC3(CC2)CC3)CC1C)=O N1(CC2(CO)CCC(C)C2)C(=O)CN(CCCc2ccc(F)c(Br)c2)C1=O c1(OC)nccc(I)c1C(N1CCNC(NCCN2CC(C)OC(C)C2)C1)=O C1(C(N2CC(OCCNC(c3ccn(CCC)n3)=O)C2)=O)C2CCCCCC12 c1(C(=O)NC2(C(N3CCC(C#C)(O)C3)=O)CCN(C)C2)cc2cccnc2[nH]1 Cc1ccn(CC(=O)N(CCCCNC(=O)Cc2nc[nH]n2)C)n1 Cn1cccc1CCC(=O)N(C1(C(N2CC(N3CCC3)C2)=O)CCCC1)C1CC1 C1(C(=O)NCC2(F)CC(NC(C3(CC#C)CC=CCC3)=O)C2)COC(C)(C)CO1 C#Cc1ccc(C(=O)N(C2CCN(C(=O)C(C)=C3CCCC3)C2)C)c(F)c1 C1(CNC(c2cccc(OC)c2O)=O)CC2CCCC2N1C(=O)Cc1cccs1 C=CCC(C)(CC)C(=O)N1CCCC(O)(CNC(C2CC3(C2)CC2(CC2)C3)=O)C1 N1(C(C2CCN(C(=O)NC)C2)=O)CCN(C(=O)COCCCOC)C(CCO)C1 C1(C(=O)NC(C)(C)CNC(c2cc3ccccc3o2)=O)CCc2ncccc2C1 C1(C(=O)NCC(c2ccc(Cl)cc2)NC(C=C(CC)CC)=O)CCCC(CF)C1 C(=O)(C(C)(C)C(N)=O)NCCN(C(c1cnn(CC(C)C)c1Br)=O)C n1(CC(=O)N(CCCNC(C(N)=O)=O)C2CC2)cc(Br)c(O)nc1=O C(CNC(C1(n2cncn2)CC1)=O)(CC(F)(F)F)NC(C(C)n1cccc1)=O C=CCCCCC(C(=O)NCc1ccccc1)N1C2C=CCC1CCC2 C1(C(=O)NCc2cccs2)CCCN(C(=O)CC2(CC(F)F)CC2)C1 N1(S(C)(=O)=O)CCOCC1C(=O)N(C(C1CCCN1C(=O)CNCC(F)F)(C)C)CC C1(C(=O)NCCN(CCC)CC)CCCCCCN1C(C1(CO)CCOC1)=O c1(C(=O)NC2C3CN(C(CCS(C)=O)=O)C2C3)cncc2ccccc12 CCC(C)C(O)C(=O)NC1CC(C)(CNC(=O)C(F)(F)C=Cc2ccccc2)C1 CC1CCCCN(C(=O)C=CC(C)(C)NC(=O)CC2(O)CCC2)C1 N1(C(c2c(C)cccc2)=O)CC(C)N(C(=O)Cc2cccnc2Cl)CC1C CCCC(CC(=O)NCc1nocc1CC)NC(=O)C(C)(C)C(=O)N(C)C Cc1cc(F)ccc1C(=O)NC1COCC1CNC(=O)C(C)SC(F)(F)F CCCC(CC)CC(=O)N1CCC(F)(F)C(CNC(=O)CCCC(C)CC)C1 c1(OCC2CC2(Cl)Cl)cccc(F)c1.CC1C2CC1NC(=O)N2 N1(C(C(C(C)C)F)=O)CCN(C(c2cc(C3CCC3)on2)=O)CC1C1CCCC1 Cc1ccn(C)c1C(=O)NCC(C1CC1)NC(=O)C(C)CF c1(OC)nsc(OC)c1CN1CCCC1Nc1nccc(C)n1 C12(C(N3CC(NC(c4cnn(CCF)c4)=O)C3)=O)CCN(CC1)C2 N1(C(c2nc(C3CC3)cs2)=O)CCc2c(F)ccc(Br)c2C1 C(=O)(C(C)C(F)(F)F)N1C(CNC(c2cc(C)c(C)s2)=O)CCC1.n12cc(nn1)C2 N1(C(C(C)NS(C)(=O)=O)=O)CCCC2(NC(=O)C=Cc3cccn3C)CC2C1 C12(C(=O)NC(c3ccccc3)C(C)NC(=O)CO)CC(C1)C(C(F)(F)F)O2 N1(C(C=CCCC)=O)CCCC2(NC(c3cn(C)nc3-c3nccs3)=O)CC2C1 C1(C(N2C(C(C)NC(CCSCCCC)=O)CCC2)=O)COCCN1C=O CC1CCCCC1(CNC(=O)C=Cc1ccncc1)NC(=O)CCc1cc[nH]n1 CCC(F)(F)C(C)(C)C(=O)NC1CCCCC1CNC(c1occ2c1CCC2)=O N1(C(C=C2CCC(C)C2)=O)CC2CCCC1C2CNC(=O)CCc1ccnn1C C1(C(N2CC(NC(C(C(C)(C)C)(C)O)=O)C2)=O)Cc2ccccc2CO1 CN1CCC(c2nc(-c3ccc(OCCF)cn3)nn2CC2CCCO2)C(O)C1 c1(C(=O)NCC2(CNC(c3ccncc3O)=O)CC23CCC3)cc2n(n1)CCO2 c1(C(C(=O)NCCC(C)NC(=O)C(C)(C)CF)O)ccc(F)c(Cl)c1 c1(C(=O)NCCC2(O)CN(C(C3C4CCCC34)=O)C2)cncc(O)c1 c1(C(=O)NC2CN(C(CCOCC=C)=O)C2)cncc(SC)c1 c1(C2CCN(Cc3nc(C(=O)OCC)c(C)s3)C2)ccnc2ccccc12 Cc1cc(CCC(=O)NCC(c2ccccc2)OC(=N)O)cc(C)n1.C1C(=O)N1 C1(c2ccccc2)(NC(C(C=CC)O)=O)CCN(C(=O)CS(N)(=O)=O)C1 N1(C(C2C3N(C(C(c4ccn(C)n4)C)=O)C(CC3)C2)=O)CCCCC(C)(F)C1 c1(C2C(C(=O)OCc3c(NC(C)(C)C)n[nH]c3)C2)ccc(Cl)c(Cl)c1 c1(C(=O)NCC2C3CN(C(C(CC)(CC)CO)=O)CC32)cc(=O)n2ccsc2n1 c1(C(N2C(CN(C(CC=C=C)=O)C3CC3)CCC2)=O)cccc(-n2cccn2)c1 c1(C(=O)NCC(CCNC(C2CC(=C)C2)=O)OCCOC)ccc([N+](=O)[O-])cn1 c1(C(C)(C)C(=O)NC2CCC(NC(C3CS(=O)(=O)C3)=O)C2)ccc2ccoc2c1 Fc1cc(CSCC2CC23CCOCC3)cc(Cl)c1 c1(C(N2C(CN(C(=O)CC3CC4(CC4)C3)C)CCC2)=O)ccc2cnnn2c1 C(CCC(C)(C)C)(c1nnnn1CC1CC1)NCc1cnn(CC)c1C c1(OC)ccc2c(C(=O)NC3CCN(C(=O)C=C(C)C)C3C)csc2c1 Cc1cc(=NC(C)C2CN(C(c3nccc4[nH]ccc34)=O)CCO2)[nH]c(C)n1 c1(NC(N2CCC(C)(C)C(c3ccccc3)C2)=O)c[nH]c2ccc(F)cc12 C(=O)(CC(C)(C)C1CC1)N(C1CCN(C(c2ncoc2C2CCCO2)=O)C1)CC C1(COC)(CNC(=O)CN2CCC(C)C2)CCN(C(=O)C(CO)OC)C1 C(=O)(C#CC1(CC)COC1)NC(CC#CC)C(=O)NC1CCC(=O)NC1C n1(CC)cnc2c(NCCCC3CC3)nc(N(CCC(C)O)C)nc12 N1(C(C2N(C)CCC2)=O)CCN(C(CNC(c2cn(C)cn2)=O)C(F)(F)F)CC1 C(C(C)(C)C(=O)NC(c1nnc(C)o1)C)NC(C=C(C)C(C)C)=O CCC(C)C(C(=O)N(C1CCCCC1)CCNC(=O)CCNS(C)(=O)=O)OC C(=O)(C(O)CC(N)=O)NC(CNC(c1n(CC)nc(C(F)(F)F)c1)=O)C1CC1 CCCC(CNC(c1cc(OC)n(C)n1)=O)C(=O)NCCOC(C)=O N1(C(Cn2ccc(C)c2)=O)CC(O)CC1CNC(c1cc(Br)n(C)c1)=O CN1CCN(C(c2cncc(O)c2)=O)C(C(=O)NC2CCN(C3CC3)C2)C1 c1(C(=O)NC(CCNC(C2(CC)CNC(=O)C2)=O)C)ccc2ncc(=O)[nH]c2c1 C1(C(=O)NC2(C(CCNC(COC(C)C)=O)=O)CC2)COCC1C(F)(F)F c1(N(CCCNC(=O)N(C)C)C(c2cccc(C)n2)=O)nc(Cl)c2c(n1)COC2 C1(C(=O)NCC2CC(OC)C2)CC12CCN(C(C1CCN(C(C)C)CC1)=O)C2 N1(C(C(CNC(=O)CCc2ccsc2)N(C)C)=O)CCCC(C2CC2)CC1 Cc1cc2[nH]c(CNC(c3cc(Cl)ccn3)c3nnnn3C)cc2s1 C1(CC)C(C(=O)NCCSC(C)C)CCCN1C(C1(C)CCC(=O)NC1)=O N1(C(C(CC#C)C2CC2)=O)CC(C(=O)N(C)C(c2ccccc2)C)C(F)(F)C1 N1(C(C2CC(OCC)C2)=O)CC(C2(NC(c3ncccn3)=O)CC2)C1 c1(C(=O)NCC2N(C(CCSCCCC)=O)CC(C)(C)C2)[nH]nc2ncccc12 Cc1c(C(N2CCC(C(C)NC(=O)Cc3cccc(O)c3)C2)=O)c(Cl)nn1C Cc1cc2c(NC3CCN(C(c4cnccc4C(F)(F)F)=O)CC3)ncnc2[nH]1 C1(CN(C(=O)CSC(C)(C)C)C)CCCN(C(C2CC2c2cccc(Cl)c2)=O)C1 C1(NC(CC)=O)COC2(CCCN(C(c3cc4cc(Cl)ncc4[nH]3)=O)C2)C1 O=C(CC1=CCOCC1)NCC(C1CCOC1)NC(c1cnc(O)nc1O)=O Cc1ccc(N)c(C(=O)NCC2(CNC(C3(C)CC3F)=O)CC2)c1F C1(C(=O)NCC2N(C(Cc3nn(C)c(Cl)c3)=O)CC2)CCc2ccnn2C1 Cc1cn2cc(C(=O)NC3CCCCC3NC(C3C(C4CC4)C3(F)F)=O)nc2s1 C12(CNC(C(C)(C)C3CCOC3)=O)CC1CN(C(=O)Cc1cc[nH]c1)C2 C(CC1CCc2ccc3c(c21)CCO3)NC(=O)NC1(NC(CCCC(C)=O)=O)CC1 c1(OC)ccccc1C(N1CC(OCC(=O)OCCN(C)C)C(OC)C1)=O c1(OC)ncc(Br)c(=NC(=O)C2CN(Cc3cccc(I)c3F)CCO2)[nH]1 C1(C(=O)NC2(CCCOC)CC2)CC(C)(NC(c2cnn[nH]2)=O)C1 N1(C(C2(COC)CCCO2)=O)CCC(CO)(NC(=O)C(F)(F)C2(OC)CCC2)CC1 C1(CNC(c2n(C)ccc2)=O)C2CN(C(=O)CCNC(=O)OC(C)(C)C)CC12 C(CCCCC(=O)NCC12CCC(F)(CC1)C2)N(C(=O)C(O)C1CC1)C Cc1cn2c(CC(=O)NC34CCC(NC(=O)CCCN(C)N=O)(CC3)C4)csc2n1 c1(C(=O)OC(C)Cc2ccccc2Br)cncc(C(F)F)c1 C=C=CCCC(=O)N1CCC(N(C(=O)CSC(F)(F)F)C)C1 N1(C(C=C(C)C(C)(C)C)=O)CC(CNC(c2cnc(C)s2)=O)C2(CCC2)C1 Cc1nc(O)c(C(=O)NCC2CCCCN(C(C3(CF)CC3(F)F)=O)C2)nc1C N1(C(CCCCN(C)C)=O)CC2CC(C(=O)OC(=O)C(F)(F)F)C(C2)C1 N1(C(C=CC(C)(C)C)=O)C(CNC(C2(C)CNC(=O)C2)=O)CC2CCCC12 N1(C(C2CCC(=O)N2C2CC2)=O)CCC2CCN(C(=O)COCCOCCO)CC12 O=C(N=c1ccnc2[nH][nH]cc1-2)C1CCCN1S(=O)(=O)c1ccc(Br)cc1F c1(C(=O)NCC2CN(C(C)=O)C(C)C2)cnc2c(c1)N(C)CCO2 c1(C(=O)NC2C(C(=O)NCC(CC)(C)COC)OCC2)cc(C)ccc1F C1(C(=O)NCC2CCCCCN2C(c2ccc(Cl)cc2)=O)(OC)CCC12CCC2 Cc1cccc(OC(C)C(=O)NC(C)CN(C)C(c2cc(C(C)C)[nH]n2)=O)c1 CC1(NC(c2csc(C3CC3)n2)=O)CCCN(C(C2CC3CC3C2)=O)C1 C(C(CC(C)C)C(=O)NCCNC(=O)OC)NC(C(CC=CC)C)=O Cn1nc(C(=O)OCc2c[nH]c3ncccc23)c2c(c1=O)CCN(OC(F)F)C2 C1(C#N)(CC(=O)N(CC(C)NC(=O)C(C)O)C)CC1 CCCCC(O)C(=O)OC(CSc1ccc(Cl)cc1)CNCC C1(C(=O)Nc2ccccc2)CCC(NC(c2ccn(C3CCCCO3)n2)=O)C1 C(C(C)(C)CC(=O)NC1(C)CCCC1O)NC(C1OCCN(C)C1)=O C(=O)(CS(=O)(=O)C1CC1)NC(C)CC1CN(C(=O)CCS(C)(=O)=O)C1 N1(C(Cn2c(C)ncc2)=O)C(C(N2CCC2C(N)=O)=O)CCC1C CC1CCC(CC(=O)NC2C3CC2N(C(=O)CN(CC(C)(C)C)C)C3)CC1C C1(C(N(C(C)C(N2CCC23CCC3)=O)CCC)=O)CCCC2(CC2)C1 N1(C(c2c(NC(C3(C)CCCC3)=O)cncc2)=O)CCCC(F)(F)CC1 CCCCC(CC)CC(=O)NC(c1ccccc1CC)CNC(C1(O)CCCC1)=O C1(CNC(C(C2CC2)OCC)=O)CC2(CC2)CN1c1ccnc(C)n1 c1(CNC(CC(=O)OCC)Cc2cccs2)cc([N+](=O)[O-])ccc1C C1(NCC2CCC(C)(CC)O2)CC2(C1)C(C(=O)O)C2(F)F C(=O)(C1=NOCC1)NCC1(COC)CN(C(C2CC(OC)C2)=O)C1 C1(C(=O)NCCn2c(CC)ncc2)CCCN(C(C2COCOC2)=O)C1C c1(C(N(C2CC(NC(C34CCC3C4)=O)C2)C)=O)c2ccccc2cc2ccccc12 C(=O)(C(CCC1CC1)NC(c1cscc1Cl)=O)NC1CCN(CCOC)C1 c1(C(C(=O)NCC(C)NC(=O)C(CO)NC(N)=O)(F)F)cc(Cl)ccc1Cl c1(-c2c(C(=O)NCCN(C(=O)C=CCOC)CC)nco2)ccc(C)cc1 c1(CC)c(C)noc1NC(c1nc(CNC)cs1)=O C(=O)(CCCCN1CCOCC1)NCC(C1CC1)NC(=O)CNC(=O)C1CC1 C1(NC(C2N(C(c3nc(C)sc3)=O)CC(=O)NC2)=O)CCOCC12CCC2 c1(CCNC(=O)NCCC2CCCSC2)cccc2[nH]ccc12 c1(CC(=O)NC2CCCN(C(CC3CCC(=O)NC3)=O)C2)cc(F)ccc1Cl N1(C(COCc2c(C)ncs2)=O)CC(C2(NC(=O)C(C)CN(C)C)CC2)C1 c1(NC(C2CC(NC(c3ccc(SC)cc3Br)=O)C2)=O)cnccc1[N+](=O)[O-] c1(-c2cn(C(C(=O)NC(c3nncs3)C)C)nn2)ccc(Cl)cc1Cl C(=O)(C(C)(C)C(F)(F)CC)N1CCC(C(C)NC(CC(CC)OC)=O)CC1 C1(NC(c2n(C)nc(C3CC3)c2)=O)CCC(C)(NC(=O)CC2CCCCO2)CC1 C1(c2nnnn2C)(Nc2cnn(C(C)C)c2)COCCOC1.CCC(C)C(C)C C=CC1(C(=O)NC2CCCC(N(C(=O)C=CC3(C)COC3)C)C2)CCOCC1 Cn1c(=O)c2[nH]c(=NCc3ccc4c(n3)CCC4=O)[nH]c2n(C)c1=O CCCC(C(=O)N1CCC1c1nnc(-c2ccc(F)cc2)s1)C(=O)O N1(CCC(=O)NCC2CCCC2NC(C2CC2(F)F)=O)CCCS1(=O)=O C12(C(N3C(CNC(c4n(C=C)ncc4)=O)CCCCC3)=O)C3C4C1C1C2C3C41C C(C)(CCCNC(C1(CO)CCOC1)=O)NC(C1CC(=C)C1)=O c1(C(=O)NCCCCCN(C)C(c2c[nH]cc(Cl)c2=O)=O)ccn2nnnc2c1 C1(CNC(Cn2c(C)ccn2)=O)CC(C(C)C)CCN1C(C1CC(N(C)C)C1)=O N1(C(=O)Cc2cn[nH]c2)CCOCCC1C(=O)NC12CCC(C1)C(O)C2O C1(C(=O)N(C(=O)Cc2ccccn2)CCl)CCCN(C(=O)CC2CCCNC2=O)C1 C1(C(=O)OC)CCCN(C(C2(N(C)C)CCC2)=O)CC1 Cc1cc(=NCC(C)(C)CC(F)(F)F)[nH]c(N(C)CCOCCO)n1 C1(OC)(CNC(c2ccnnc2C)=O)CCN(C(C2CC2C(F)(F)F)=O)C1 Cc1cc(C(=O)NCCN(C(C2CC3C=CC2O3)=O)CC2CC2)ncn1 N1(C(C=CCCC)=O)CC(NC(c2cc(-c3cnn(C)c3)[nH]n2)=O)C(C2CC2)C1 C1(C(N2CCC(N(C)C(c3ccnnc3O)=O)C2)=O)CC2(COC(=O)N2)C1 c1(OC)ccc(C)cc1OCC(N1CCC(CCO)(C(=O)NCCOC)C1)=O c1(CCN(c2nnc(-c3ccc[nH]3)n2CC2CCCCO2)C)ccc(F)c(F)c1 c1(C(C)(C)CN2CCC(C(C3CCCNC3)O)CC2)ccc(F)cn1 C(C(C(CC)CC)OC)NC(C(C1CCC(C(F)(F)F)CC1)CC)=O c1(C(N(C2CN(C(C(C)NC(=O)OC(C)(C)C)=O)C2)C)=O)cnc(C(=O)O)nc1 C1(C(=O)NC2(CN(C)C(c3cnnc(O)c3)=O)CC2)CC2(CCCO2)C1 Cc1ccc(C)c(C(N2CCCCCC2CNC(C2CC(=C3CCC3)C2)=O)=O)n1 c1(C(=O)NC2CCN(C(=O)CCC3CCC3)CC2CO)ccc2nn[nH]c2c1F N1(C(C2C3CCC(N(C(c4ncc(C)cc4F)=O)C2)C3)=O)Cc2ccncc2C1 N1(C(C)C(=O)NCC(C2CC2)N(C)C(c2nn[nH]c2Cl)=O)C(=O)CCC1=O C1(C(N2CCCC2CS(N)(=O)=O)=O)NC2CC1CC2O N1(C(CCc2ccc(N)cn2)=O)CC2OCCN(C(c3cnco3)=O)C2C1 C=C(C)C(C)(C)C(=O)N1CCCC(C)(NC(c2ccc(C(F)(F)F)cn2)=O)C1 Cc1cc(C#N)c[nH]c1=NC1CC(F)(C(=O)Nc2cccc(Cl)c2)C1 C(c1cc(F)cc(F)c1)=CC(N1C(C)CC(NC(C2C3CCC2CC3)=O)CC1)=O C(=O)(C(C#N)C(C)(C)C)N(C1CN(C(c2ccn3nccc3c2)=O)CC1(C)C)C c1(C(C)=O)ccc(F)cc1F.C(=O)(CCCCCSC)N1CC23CC(C2)(C3)C1 C#Cc1cc(F)c(C(N2CC3CN(C(=O)CC4CCCOC4)CC3C2)=O)cc1F c1(C(=O)NC2C(CC)CN(C(c3nsnc3O)=O)CC2)cnc2c(Cl)cccn12 C1(OCC(=O)NC(C2CCCC2)CNC(COCCCC)=O)CC1(C)C C1(CC)(CNCc2ccc(F)c(N)c2)Cc2ccccc2C1 c1(C(=O)NC2CC(C)(NC(C(C)n3ccnc3)=O)C2)cnc2[nH]ccc2n1 c1(OC)ccn2c(C(=O)NCC3CCN3C(=O)Cc3ccc(N)cc3)cnc2c1 C=CC(C)(C)C(=O)NC1C(C(=O)NOCC(C)O)CC1O C1(NC(C2CN(C(=O)NC)C2)=O)CC(CNC(=O)CC2CSCCO2)C12CCC2 C1(C(N2C(C)(CNC(C3CCC(=O)N3)=O)CCC2)=O)CCC(=O)N(C2CC2)C1 CC1(CO)CC2(CCN2C(C2N(C(c3c[nH]c(=O)cn3)=O)CC23CCCC3)=O)C1 C1(C(=O)NCCCCCNC(=O)C(O)C(C)C)(OCCCC(C)C)CCOCC1 CC1CN(C(=O)CCN(C(C2(CO)CCCO2)=O)CC2CC2)CCN1CCO c1(-c2c(OC)nccc2)cc(C(=O)NCc2cnc(C)[nH]2)cc2[nH]ccc12 N1(C(c2c(C)ccnc2)=O)CCC(O)C(NC(=O)C(C)Oc2cccc(Br)c2)C1 C1(CNC(C2CCOC2CNC(C(C)NC(CC)(C)C)=O)=O)CCC(CC)CC1 Cc1cc(F)c(C(=O)OCc2cc(Br)cs2)c(F)c1 C(C)(C(=O)NCC(C)OC)(CCOC)NC(CC=C)=O CCC(C)(C)C(=O)N1CCCC(N(C(=O)COCCF)Cc2cccc(C)c2)C1 CC1OC(C)C(C)C1C(=O)NCC1(F)CCN(C(C2CCC(=O)O2)=O)CC1 c1(N(CC(F)F)CCC)nccc(N(C)CC2CCOC2C)n1 C(CN=c1[nH]c(N2CCC(F)(CF)C2)nc2c1COC2)(CC(C)(C)C)OCC C(=O)(CCCN(C)N=O)NC(CCC)CCCNC(=O)Cc1ccc(SC)cc1 C(CN=C(NCC(c1ccc(Cl)cc1)SC)N1CCCCCCC1)OCC CC1(C)CC(O)CN(c2nnc(CN3CCCS3(=O)=O)n2CCc2ccsc2)C1 N1(C(c2cc(C)ns2)=O)CCN(C(C2CCCN(C)C2)=O)C(c2cn[nH]c2)C1 N1(C(CC2(NC(C(C)NC=O)=O)CCC2)=O)CC2COC(=O)C2C1 N(C1CCc2cc(CNC(C3CCC3)=O)ccc21)C(C(C)Cc1cnn(C)c1)=O N1(C(C(C)N(C(C2(C#C)CCCC2)=O)CC)=O)CC(C)(C)CCC1C Cn1nnc2cc(C(=O)NC3CN(C(C4CNC(=O)C4)=O)CC34CC4)ccc12 Cc1cnc(C(N2CC(C(F)(F)F)CCC2C)C(=O)NC(C)C)cc1Br C1(CC(=O)NCC(C#C)OC)CCCCN1C(c1cn(C2CC2)nc1C)=O c1(OC)cc(CCC(=O)NCCCCNC(=O)CCc2nc(C(C)C)no2)on1 CN=c1[nH]cc(C(=O)NCCc2n[nH]cc2C(=O)NCC2(C)C=CCCC2)s1 n1(CC(=O)NCc2c(CNC(C=CS(C)=O)=O)cccc2)cc([N+](=O)[O-])ccc1=O C1(CCC(=O)C2(CN(C(c3n(CC#C)ccc3)=O)C)CC2)CCCCN1C.CCN CC(C)(C)CC(C)(C)CNC(=O)C(C1(C)CC1)NC(=O)Cc1cn[nH]c1 c1(C(CC)N(C(c2ccc(Cl)s2)CC)C2(C)CC2)nnnn1C1(C)CC1 C(=O)(C1=C(C)OCCC1)N1CC(O)CC(NC(c2c(C(=O)OC)cccc2)=O)C1 c1(C(=O)NCC2N(C(CC3(CC(=O)OC)CC3)=O)CC2)csc(-c2cnc[nH]2)n1 N1(C(C2(NC(c3ccc[nH]3)=O)C(C)CCC2)=O)CCC2C(C(N)=O)C2C1 N1(C(c2c(C)noc2C(C)C)=O)CCC(NC(c2cnc(S)nc2)=O)C(F)C1 CCC(C)CC(C(=O)NCc1cccc(F)c1F)NC(=O)CCSC C(=O)(C1=CCCN(C(c2ccc(O)nc2C)=O)C1)NCCSCC#C Cc1c(C(N2CCC(N(C)C(C3CCCSC3)=O)C2)=O)oc2c(F)cccc12 C(C1=NOC2CCCC12)NC(C1C(C)N(C(c2ns[nH]c2=O)=O)CC1)=O Cc1nccc(C(=O)N(CC(C)(C)C(=O)NC2COCC2C(N)=O)C)n1 C1(C)(CNC(C(C)=C2CC2)=O)COCCN(C(c2ccc(OCCF)cc2)=O)C1 N1(C(C2CN(S(C)(=O)=O)C2)=O)CC(NC(c2csc(C(F)F)n2)=O)CC12CCC2 C1(C(N(C)CC2CN(c3nc(CC)c(C)cn3)C2)=O)CCOCC12CCC2 c1(N)cnn2c1CCC2.N1(C(CC2ON=C(C)C2)=O)CC(C(N)=O)C(C)C1.C1C(=O)N1 c1(CC)c(C(=O)NCCCN(C2CCCC2)C(c2cc(C3CC3)sn2)=O)cnn1C c1(N(CC=C)C(=O)NC(CC#CC)OC(C)(C)C)ccc(Br)cc1 C1(C)(NC(C(C2CCC2)OCC)=O)CCN(C(=O)C=C(C)C2CC2)C1 C(C)(CNC(C1CC1c1ccnn1C)=O)(C(C)C)NC(C=C(CCC)C)=O CC12CC(NC(=O)C(=O)NC3CCCCC3)(C1)C(C)(C)O2.N12CC3C(C3C1)C2=O N1(C(CN(CC)CC)=O)CCCC(NC(C2CCCCCC2)=O)C1 c1(-c2c(C)ccs2)nc(C2CSC2)nn1CCC(C)C N1(C(C=CSC)=O)CCC(C)(CCNC(C2CCCOCC2)=O)C1 N1(C(CCCCCNC(c2cn(CC)nc2C)=O)=O)CC2CC(OC)C(C2)C1 c1(C(N(CCOCCO)CC)=O)cnc2[nH]cc(-c3cccc(F)c3SC)c2c1 N1(C(C=CC)=O)CCCCC1C1CCCN(C(c2cccc(=O)o2)=O)C1 N1(C(=O)NCC2(CC3CCC3)CCCO2)CCN(C2CCC2)CC1 N(C(=NCCC(=O)Nc1ccccn1)N1CCC(NCC2CCCC2)C1)C(C=C)C C1(F)(C(=O)NC2(COC)CCCO2)CCN(C(=O)C(C)(C)CCOC)CC1 c1(C(=O)NC2C(NC(C3C(C)=CCS3)=O)CC2)sc(C#N)cc1Cl N1(C(C(CCC)NC(c2nn[nH]c2CC)=O)=O)CC2CCCC(C1)N2C(C)=O C(=O)(C(C)(C)CF)NC1CCC(CC(=O)N(CCN(C)C)C2CC2)C1 C1(C(=O)NC(C)CN(C(C)C(=O)NCC(F)(F)F)C(C)C)CCOC2(CCCC2)C1 C#Cc1ccc(C(=O)NCC(c2ccccc2)CNC(C2CC2CC)=O)c(C)c1 N1(C(C(CC)C)=O)CCC(O)(C(=O)NCc2cn(C)nc2C)C1 C1(C(N2CCC(=CCC)C2)=O)CCCCCN1C(=O)CNC(=O)C1CC1 CC(C(=O)OCc1cccc(F)c1N)C(F)(F)F N1(C(c2c(C)c(Cl)ccc2)=O)CC23CCCC2(C1)CN(C(C1CCC(=O)C1)=O)C3 N1(CCOC)CC(C(=O)NCC(C(C)(C)C)NC(c2cnccn2)=O)CC1=O c1(C(=O)NCCCCN2CCN(C)C(F)(F)C2)c[nH]c(=NCCO)cn1 N1(C(C2N(C)CCCCC2)=O)CCC(C(=O)NCc2ncc[nH]c2=O)CC1(C)C C1(O)(CC(N2CCC(NC(C(C)Cn3ccnc3)=O)C2)=O)CCOCC1 C(=O)(C#CC1CCOC1)NCCOC1CCN(C(c2cccc(N)n2)=O)CC1 Cc1[nH]c(=NCC2CCCC2NC(c2cc3c(Cl)nccc3o2)=O)ccc1[N+](=O)[O-] c1(C(=O)NCC(C2CC2)NC(C(CC=CC)CC)=O)cc2c(C)n[nH]c2cn1 C12(NC(C3ON=C(C(C)(C)C)C3)=O)CCOCC1CN(C(c1cscn1)=O)C2 CSC1=C(C(=O)N2CCCC2(C)CNC(=O)CCc2ccc(F)cc2)CCCC1 N1(C(C2OCCC(NC(C3C(C)OCCC3)=O)C2)=O)CC2CSCC2C1 c1(CC(=O)NCC(CNC(CCC=CCC=C)=O)CO)n[nH]c2ccccc12 c1(C(CC(=O)NCCC(C)NC(c2cnn(C)c2C2CC2)=O)C)ccc(F)cc1 c1(C(=O)NCC(C)(CNC(=O)CC2CCC(=O)C2)OC)cc(C)sc1C N#Cc1cc(C(N2CC3CC(C2)C3(F)F)=O)c(O)cc1N c1(NCc2cc(C)no2)cc(C)c(S(=O)(=O)NCC(N2CCCC2)C)cn1 C1(C(=O)NCC(CNC(CCCOCC=C)=O)C)CC(F)(F)CO1 N1(C(C2CCC(CC)C2)=O)CCC2(CC1)CC2C(=O)NCC(CC)(CC)OC CC1Cc2cc(CC(=O)NCC3CC(NC(=O)C(F)(F)CO)C3)ccc2O1 N1(C(c2scc(C)c2)=O)CC(C(N2CCC2C(C)O)=O)C2(CC2)C1 Cc1ccc2c(C(=O)NC3CN(C(C4COC(=O)O4)=O)CC(C)(C)C3)c[nH]c2c1 c1(CNC(C(C2CC2)NC(CC2(COC)CC2)=O)=O)ccc(C)c(C)c1 N1(C(C=Cc2cn(C)nc2)=O)CC(C(F)(F)F)OCC1CNC(C1CC(O)C1)=O N1(C(CCN(C)CC)=O)CCC(O)(C(C)NC(=O)COc2cc(C)on2)CC1 c1(OC)ccc(Br)cc1CC(N1CCC(NC(=O)CCNC(C)C)C2CC12)=O c1(C(=O)NC2CC(N(C(c3c(C)nc(CCC)o3)=O)C)C2)cncc2[nH]ccc12 C(=O)(C(CC=CCl)c1ccccc1)NCCN(C(=O)Cc1nonc1C)CC C(=O)(CCCC(C)NC(C1CCC2CC12)=O)NCC(C(C)C)(C)C N1(C(c2c(C)c(F)ccc2)C(=O)NC2CCC2)CC(S(C)(=O)=O)CC1C(=O)OC Cc1cn2c(n1)C(C(=O)NC(C)CCNC(=O)Cc1cccnc1)CCC2 C(=O)(C(C)(C)C(N)=O)N1CC(OC)C(C(N2CCC(C)(C(=O)OC)C2)=O)C1 c1(C(N(C)CC2(O)CN(C(C3COCCN3C)=O)C2)=O)c(F)ccc(F)c1N c1(C(N(CC(C)NC(c2cc(F)cc(F)c2)=O)CC)=O)cncc2n[nH]cc12 N1(CC(=O)N(C(c2ccccn2)C)CC=C(F)C(=O)NC2CCC2)CC2CC2C1 C1(C(C)C)C(NC(=O)C(O)C(C)C)CCN1C(=O)COCCc1ccsc1 C1(CNC(C2CC(=C)C2)=O)CC(F)(CNC(=O)C(=O)NCC(F)(F)F)C1 c1(OCC=C)ccc(C(=O)NCC2CN(Cc3ccsc3Br)CC2O)cc1 C1(C(=O)NC(CC=C)CNC(C2(C)CCCCO2)=O)CCC2(CCCC2)CC1 C(=O)(C(C)(C)CCNC(C1CC2(CCO1)CC2)=O)NCc1cn(C)nc1 C(C)(CCCCNC(=O)Cn1nnc(C2CC2)n1)NC(c1n(C(C)C)ccn1)=O c1(C(=O)NC(C2CCCN(C(=O)Cc3ccccc3)C2)C)c(F)cc(O)cc1F C1(N(C(=O)Cn2cccn2)C(c2ccc(F)cc2O)C)CCC2(CC1)CNC2 C1(CNC(CC(C)CCC)=O)CC2(C1)CN(C(=O)CCC1CC(OC)C1)C2 CC1CCN(C(=O)C(=O)Nc2ccccc2SC2CC2)CC1c1nccn1C Cc1c(S(=O)(=O)N2CC(C)(N)C2)sc2c(F)cccc12 Cc1ncnc(C)c1CC(=O)NCC(CO)NC(c1ccc(F)c(Br)c1)=O c1(C(=O)Oc2cnc(C(C)OC)nc2O)cc(C)c(CO)cn1.c12cn(nn1)C2 C1(N(C)C)CN(C(C2C(C)(C)C2(F)F)=O)CC1CNC(=O)Cc1cnsc1 C1(NC(C2(C)CN(C(COCCCC)=O)C2)=O)CC2CC1OC(=O)N2 N1(C(C(C)NS(CCCC)(=O)=O)=O)CCN(C(=O)CC2(C)CCC2)CC(C)(F)C1 N1(C(C2C(C)(C)COCC2)=O)CC(CNC(=O)C2=COCC2)OC2(CCC2)C1 N1(C(C2C(C(=O)OC)CCC2)=O)CCC(CO)C(NC(c2scc(C)c2C)=O)C1 C(C1(O)CCc2ccccc21)N(C)C(C1CCCN1S(C)(=O)=O)=O c1(C(=O)NCc2cccc(-c3c(C)nn(C)c3)c2)cc2cc(F)ccc2[nH]1 c1(C(=O)NCC(C)CN(C(=O)CNC=O)C)sccc1SC(F)F c1(C(=O)NC23CC(NC(c4cc(OC)no4)=O)(C2)C3)cc(Cl)cc(Cl)c1F C1(CN(C(C2N(CC)CC2)=O)C)COCCN1C(c1nc(C)sc1C)=O C1(NC(CCOCC)=O)C(CNC(c2cccc(Cl)c2O)=O)CCC12CCC2 N1(c2nnc(C#N)s2)CCN(C(C23COC(CF)(C2)C3)=O)CC(O)C1 c1(N2CCCC(C(=O)OC)C2)nc(C)cc(=NC2CN(OC)CC23CCC3)[nH]1 N(C(=NCCCF)N1CCC(C2CCC2)C1)Cc1scc(C)n1 c1(C(CC)=O)ccc(C(C)(C)NCCN(CCN(C)C)Cc2ccccn2)cc1 CC1CCN(C(=O)CC(C)(C)O)CC1CC(=O)NCc1nnc(O)o1 c1(C(N2C(CNC(C(CC=C)NC(C)=O)=O)CC(O)C2)=O)cc2c(cn1)CCCC2 C1(C)(C(=O)NC(CC(C)C)CNC(=O)CCc2cnn(C)c2)CCS(=O)(=O)CC1 Cc1cc2ccc(C(=O)NC3CN(C(c4cc(Cl)c5n[nH]cc5c4)=O)C3)cc2o1 N12CCC(CC1C)C2=O.c1(-n2cc(C)nc2)cc2sccc2[nH]1.C12CCN(C1)C2 C=CCCC(C)(C)C(=O)NC1CCCC(NC(=O)C(C)OCC(F)(F)F)C1 C(c1c(Cl)nc2ccc(Br)cn12)=CC(N1C2CCCCC1CC2)=O Cc1cccn2cc(CC(=O)NCC3(C)CC3Br)nc12 O=C(O)CCCC(=O)NCCc1ccc(Cl)c(Cl)c1 C(=O)(C(CNC(C1CCCCNC1=O)=O)CCC)NCC1CCN(CC=C)C1 N1(CCNC(CCN2CC(C)(C)C2)=O)CCN(C(C2(C)C=CCC2)=O)CC1 CC1CCCC1(C(=O)N(C)Cc1nc[nH]n1)NC(c1cccc(C2CC2)c1)=O n1(CCC)ncc(C(=O)NCCC2(O)CN(C(c3cccc[n+]3[O-])=O)C2)c1Cl Cc1nccnc1-n1cc(C(C2CCCN(C3CCC3)C2)O)nn1 c1(C(N2CCC(C3N(C(C(CC)F)=O)CCC3)C2)=O)ccnc(C2CC2)n1 CCC(C)C(O)CC(=O)NC(C)(CNC(C1(SC)CCC1)=O)Cn1cccn1 N1(C(C(C)(F)CC2CCCC2)=O)CC(C2(OCCNC(=O)C(Cl)=CCl)CC2)C1.C(CS)O C=C1CC2(C1)CC(C(=O)NC1CN(C(C3(SC)CCC3)=O)CCC1CO)C2 c1(-c2cn(CC(=O)N(C)Cc3c(C)nc(C)o3)nn2)c[nH]c2nccc-2c1 c1(CC)nc2c(C(N3CCCC3(C)CNC(=O)CS(C)(=O)=O)=O)ccnc2[nH]1 C1(C(C)C)C(=O)N2CC(C2)O1.N1(C(COCC)=O)CCNC(=O)C1 CCC(O)C(F)(F)C(=O)NCCCN(CCO)C(c1cc(C(=O)OC)ccn1)=O c1(C(CC(=O)NCC2CCN(C(c3c(C)ncs3)=O)C2)C)c(C)n[nH]c1C N1(C(CCCN(C)C)=O)CCCC(C2CN(C(=O)CC3CSC3)C2)C1 N#Cc1cccc(CCC(=O)NCc2nc(C3(Cl)CC3)cs2)n1 C1(N(C(CCN(C(c2cscn2)=O)CC)=O)C)CCCCCCC1 CC1(C(=O)NCCN2CCCC2)CC(O)CN1C(=O)Cc1cccc(O)c1 CC1(C)OCC(c2cn(CC(F)Br)nn2)O1.C1(N2C3CC(C3)C2=O)CCCC1O c1(C(=O)NCC2CCN(C(CCCCSC)=O)CC2)cccc(C(C)C)c1O C1(C(=O)NCCCCC2CCCO2)COC2(C1)CN(C(C1CC3CCC3C1)=O)C2 C1(C(=O)OC)CCOC1C(=O)NCc1coc(CNC2(C3CC3)CCCC2)n1 C1(C(=O)NCCn2c(C(=O)OCC)cnc2)C2CC1N(C(=O)C=C1CCOCC1)C2 c1(OC)ccc(C(C)C)cc1CN1CC2C(C(N3CC(C)(O)C3)=O)C2C1 C(=O)(CC(C)(C)CC(=O)NCC(C)(CC(C)C)NC(=O)C(C)N1CCC1)OCC N1(C(c2c(C)[nH]cc2)=O)CCC(C)C(NC(=O)CC=Cc2ccc(Br)cc2)C1 c1(C(C)C)n[nH]c(=NCC(C)CNC(C2CC3(CC(=O)N3)C2)=O)o1 c1(C(CCNC2CN(C(=O)C(C)(C)C3CCC3)C2)OC2C(OC)C2)ccccc1 C#Cc1cc(NC(C2CCOCCN2C(c2cc(OC)n[nH]2)=O)=O)cc(F)c1 CC(C(=O)NCC1CCCCCN1C(c1c[nH]nc1F)=O)S(N)(=O)=O c1(CC(N2CC(CC)N(C(C3CC3C(C)C)=O)CC2)=O)ncn2c1CCCC2 C(=O)(C1=CS(=O)(=O)CCC1)NCC(C)(C)NC(=O)C(C)(C)c1cccs1 C(=O)(CC(C)(C)COC(C)C)NCC(C)(C)NC(C(C=C)c1ccccc1)=O c1(CC)ccc(C(N2CC(C)C2C(=O)NC(C)Cc2cn[nH]c2)=O)cn1 CC(C)CCC(O)C(=O)N(C)CCOCCCN(C)C(c1ccc[n+]([O-])c1)=O c1(C(=O)NCC2N(C(C(F)OC)=O)CC(F)C2)cc2cccnc2cc1F C1(C(N(C(CC(=O)NC)C)C)=O)(CF)CCN(C(C2CCCCO2)=O)C1 Cc1ccc(F)c(C(=O)NCC(C2CCCC(C)C2)=O)c1 C(=O)(C(C)CN(C(=O)CCCN(C)C(C1CCCN1C)=O)C)OC CCCCC(COC)NC(=O)CCN(C(=O)CCc1ccn(C)c1)CCO c1(C(=O)NCC2CC(NC(C34C(C)OC(CO)(C3)C4)=O)C2)cc(Br)c(F)cc1N c1(OC)cc(F)cc(C(=O)NCC2CCN(C(c3c(Cl)cnn3C)=O)CC2C)c1N C1(NC(C(C)OCC(C)C)=O)CC1C1CCCN(C(=O)COCC2CC2)C1 Cc1ccn(CC(=O)NC2CN(C(c3cccnc3)=O)C2)c(=O)c1 N1(C(CCN(C(=O)C(C(C)C)NC=O)CC)=O)CCOC2COCC12 C1(NC(C(C)c2ccco2)=O)CCCCN(C(=O)CN2CCC(F)CC2)C1 CCCCCCCCC(=O)N1CC(CNC(C2(CCOC)CC2)=O)C2(CCC2)C1 c1(C(=O)OCC)cc(F)cc(S(=O)(=O)NCCCCCCC(C)C)c1 CCCC(C(O)C(=O)N(CCCO)CC)NC(c1cc(C)nnc1C)=O Cc1nocc1C(=O)NCC(F)CNC(C1C=CCCC1)=O N1(C(c2c(CCC)n[nH]c2)=O)CC2CCN(C(c3ccc(C(C)C)nc3)=O)C2C1 CC1(C)CN(C(=O)COc2ccsn2)CC1NC(c1cn(C2CC2)nn1)=O c1(C(=O)NC(CNC(=O)C2=CCCS2)C2CCC2)nccc2cccnc12 C1(NC(c2c(C(C)C)ocn2)=O)COC2(C1)CN(C(=O)COCC1CCOC1)C2 N1(C(c2cccc(CC)n2)=O)CC2(C)CN(C(=O)CCCC(N)=O)CC2(C)C1 C1(NC(c2n(CCSC)nnn2)c2nc(CC(F)(F)F)no2)CC(C)(C)C12CC2 c1(CNC(C2(c3nccs3)CCOCC2)=O)nc2n(n1)CC1(CC2)OCCO1 n1(C(c2c(C(C)=O)cccn2)=O)ccc(=NC(=O)C2CNC(=O)C23CC3)[nH]1 c1(C(N2C(CN(C(CCC(=O)NCC)=O)C)COCC2)=O)cc(Cl)c(F)cc1Cl C1(C(=O)NC(C2(O)CCN(C(c3scnc3C(F)F)=O)C2)C)CCC2CC2CC1 CCC(CC(=O)NCC(C)CNC(c1cn2ncccc2n1)=O)C(C)(C)C C(=O)(C(CC(F)F)C1CCC1)N1C(C2(C(=O)OC)CC2)CCC1.c1(OC)ccc(S)nc1 C1(CC)CN(C(c2cnc(F)c(C)c2)=O)CCN1C(=O)Cc1ccccc1F c1(C(N2C(CNC(C(C(C)C)=O)=O)CC2)=O)ccc(F)cc1C(N)=O N1(C(CNS(CC)(=O)=O)=O)CCC(C2CCOCC2)(CNC(=O)C(C)(C)CF)C1 C(CSC)(C(=O)NCCOC1CN(C(c2ccn(CC(F)F)n2)=O)C1)OC C(=O)(C(CO)C(F)(F)F)NCCn1ccc(C(=O)NC(C(C)F)C)c1 C1(CNC(c2cccc(N)c2)=O)CCN(C(C2CC3CCC2C3)=O)C12CC2 c1(C(N2CC(O)(CCNC(c3ccncn3)=O)C2)=O)c[nH]c2nccc(Cl)c12 C(c1ccccn1)=CC(=O)NC1(CCNC(C2C(C(C)(F)F)C2)=O)CCC1 c1(C(=O)NC(C)CN2Cc3ccccc3C2=O)ccc2c(c1)CCCC2=O N1(CCC(C=C)(C)C(=O)OC)CCCC(N=c2[nH]nc(-c3ccccc3)o2)C1 C(=O)(C1CCCc2nc[nH]c21)NCC(CN(C(C1C2CCC12)=O)CC)(C)C c1(NC(COC(=O)NCCCC)=O)ccc(CNC(=O)Cc2nccn2C)nc1 C=C1CCN(C(=O)CC(COC)COC)C(C(=O)NCC2CCN(CC)C2)C1 C(=O)(CCCCC(F)(F)F)NCCCN(C(=O)Cc1ccc(Cl)cn1)C C1(COC)(NC(=O)C(C)O)CCN(C(=O)Cc2csc(C3CCCOC3)n2)CC1 C1(C(C(=O)NCC(CCC)NC(=O)CCOCCOC)O)CCCCCC1 C12(NC3CN(C(=O)NCc4cc(C(=O)OCC)[nH]n4)C3)CCC(CC1)OC2 S(=O)(=O)(c1ccc(C#N)cc1)NC(C(C)C)C(C)NC(=O)CNc1scnc1Cl N1(C(C2C3CCC2CC3)=O)CCCC(C2CCCN(C(c3cnc(O)o3)=O)C2)C1 C(C(C)(C)C(=O)NC1CN(C(=O)C(c2ccc(C)cc2)F)CC1SC)SCC c1(C(C(=O)NCCCSC)N(C(C#C)C2CCC2)C)ccc(C#N)cc1 Cc1cc(-n2cc(CC(C(C)C3CCCC3)NC(=O)C(C)C#N)nn2)cnc1Br c1(C(N2CC(CNC(c3ccc(Br)cn3)=O)OCC2)=O)cc(Br)nc(Br)c1 c1(C(N2CC(CCNC(C(C)NC(C3CCCC3)=O)=O)C2)=O)cc2n(n1)CCO2 c1(OC)ccccc1CN(C1CCOC(C)C1)C1CCNCC1 C1(NC(C(C)(C)CF)=O)CC2CN(C(c3c(Cl)ccc(F)c3N)=O)CC2C1 N1(C(c2[nH]cc(C)c2)=O)CC(NC(C2CN(C(C)C)C2)=O)CC(C)(C)C1 c1(C(=O)NCCC2(NC(=O)Cn3cnnc3O)CC2)ccc(-n2ccnc2)cc1 C(=O)(CP(=O)(C(C)C)C(C)C)N1CCC(C(C)NC(C2CCC(CC)O2)=O)CC1 n1(C(c2nn(CC=C)c(C=Cc3c(C)noc3C)c2)C)c(=O)oc2ccccc12 C1(NC(C(C)=CC=C)=O)COCCC1C(N1CCC(CCCO)C1)=O C1(C#N)(C(N(C(C)C(=O)NCCc2cscn2)CC)=O)CCCO1 CCC(O)CC(=O)N1CCOCC1CN(C(=O)C(c1cnccn1)C)C N1(C(c2c(C)occ2C(F)(F)F)=O)CC(NC(c2cnn(C)c2)=O)CC(O)C1 C=CC1(C(N2CC(CC(F)C(=O)NCCC(C)(O)C3CCC3)C2)=O)CCCCC1 C12(C(=O)NCC3N(C(=O)CC4CCCC4)CC(O)C3)CC(CO)(C1)OC21COC1 C1(CNC(C(C(C)C)NC(N)=O)=O)CN(C(=O)CCc2nc[nH]n2)CCN1C N1(C(C(=O)NCC2CC2)=O)CC(O)CC1CNC(C1(F)CCCOC1)=O c12ccc(cn1)NCC1CC1C(=O)NCC(CCN)NC(=O)C2.CN(C)C(N)=O N1(C(c2c(OCCCC)cc(OC)cc2)=O)CCN(C2CCCC2)CC(C)C1 C1(CC)CN(C)C(=O)CN1C(=O)COC1CC(N(C(=O)Cc2nccn2C)C)C1 Cc1nc(N2CCC(NC(=O)Cn3cc(F)ccc3=O)C(F)C2)c2ccsc2n1 c1(C(=O)NCC2(O)CN(C(C3C(F)(F)C34CCC4)=O)C2)ccc2c(c1)NCCC2 CC1OC(C)(C)OC1(C)C(=O)NCC(C)(C)NC(=O)Cc1ccc2c[nH]nc2c1 c1(SC)ccc(O)c(C(N2CC(CNC(c3ccc(C(C)=O)nn3)=O)C2)=O)c1 C(=O)(CCS(N)(=O)=O)N1C(CC)C(C(=O)N(C(C)C)Cc2ccco2)CC1 c1(OC)ccccc1C(=O)NCc1cc(=N)[nH]o1 N1(C(CNc2c(C)cccc2C)=O)CC2(CCCC2NC(=O)Cn2ccnn2)C1 N1(C(CCC2CCN(C)CC2)=O)CCOCC(F)(CNC(=O)CSC(F)(F)F)C1 C1(C#N)(C(=O)NCC(C2CCN(C(COCC(C)(C)C)=O)CC2)F)CC12CCC2 N1(CC(=O)NC2CC(F)(CNC(CS(=O)(=O)NC)=O)C2)C(C)=CC(C)=NS1(=O)=O c1(C(=O)N(CC(C)(c2ncc[nH]2)NC(=O)C=CC2CC2)COC)cncc(C2CC2)c1 c1(C(=O)NCC(CC)NC(C2(CC)CCCC2)=O)cnn(CC(F)(F)F)c1C c1(C(=O)OCC2(CC)CCCOC2)ccccc1S(=O)(=O)C(F)(F)F C(C1=C(C)CCC1)NC(c1nn(C)cc1C)c1n(CCCC)nnn1 C1(F)(C(N2CC(C(=O)O)(CNC(C3CCC(O)C3)=O)C2)=O)CCOC1 c1(NC2CC(NC(CCCCC#C)=O)C2(C)C)ncnc2c1ncn2C C(C(C)(C)CO)NC(C(c1cn(CC(=O)O)nn1)C)=O CCCCN(C(=O)CC1CCN1C(C1(CSC)CC1)=O)C C1(C(C)(C)C)(CNC(CSCC(=O)OC)=O)CCN(C(=O)C(C)n2cnnn2)C1 N1(C(C(C=C)(F)F)=O)CCC(C2(NC(=O)C(c3cncc(F)c3)C)CCC2)CC1 CC1(C(=O)NCC2(C)CCCN(C(=O)CC#N)C2)CCCCCCC1 Cc1cc(Cl)cc(C(N2CC(C)(NC(=O)CCNC(C3CCCO3)=O)C2)=O)c1O CC(CCC(=O)NCC1(O)CN(C(c2ccccc2C(F)F)=O)C1)S(C)(=O)=O c1(CC)ncncc1C(=O)NC1(C)CCN(C(C2(C#N)CC2)=O)C1 c1(C(C)OC)nc(C(c2cccnc2)C)n(-c2cccc(C(F)(F)F)c2)n1 c1(C(=O)NCC(CCOC)NC(C2CCN(C)C(C)C2)=O)ccc2c(c1)CC2 c1(-c2cn(C(C(=O)NC(c3ncc(C)s3)C)C)nn2)cnn(C)c1C c1(CC)cc(C(=O)NC2CC(C)(C(=O)C(C)N(C)C)C2)c2c(c1)CCO2 N1(C(CCOCC)=O)CC(NC(=O)C(CC)Oc2ccc(F)cc2)C2(CC2)C1 Cc1ccc(O)c(C(N2CCC=CC2C(N2CC(OC(C)C)C2)=O)=O)c1 C1(C(N2CC3C(CC)(C3)C2)=O)CCC2(CC2)N1C(=O)C(c1cnn(C)c1)C c1(NC(C=CC=CC)=O)ccc(-c2ccc(Cl)s2)nc1 c1(CC)ccc(C(=O)NC(C(=O)NCC2(CO)CCC2)C2(C)CC2)o1 c1(C(C(=O)NC(COC)(C)CO)OC)cccc(C(F)(F)F)c1 c1(C(N2CC(F)CC(NC(CN(C(COC)=O)C)=O)C2)=O)c(Cl)ccc(C)c1N c1(CC(=O)NCC2N(C(c3ccn(C(C)C)n3)=O)CCC2)ncn2c1CCCC2 C1(CC)(CNC(c2cc(CNC(C3CC3(Cl)Cl)=O)ccn2)=O)CCCCO1 Cc1cc(Cl)ccc1OCC(=O)NC(C)CCNC(c1ccc(N)c(Cl)c1)=O c1(C(CNC(C2CCN2Cc2ccncc2)=O)O)ccc(OC(F)F)cc1 C(C(F)(C(=O)NCC#CCN(C)C)C(C)C)NC(COCCN(C)C)=O c1(N(C)C)cccc(C(=O)NC2CCCN2C(=O)CS(C)(=O)=O)c1.c12cn(nn1)C2 C(C1CN(C(=O)C(C)C2CCC2)CC1C(N1CCC(O)(COC)C1)=O)=CC N1(C(CNC(C)=O)=O)CCN(C(c2ccc(C(=O)OC(C)(C)C)cc2)=O)CC1C CCCCC(CN(C(=O)C(C)N(C(c1ccc(F)s1)=O)CC)C)CC C(=O)(CC(C)P(C)(C)=O)N(CCC(N1CCCC(CC)CC1)=O)CC(C)C C12(CCCCC1)C(=O)N2C1CC1.C(C=O)=CC=CC.C(CC#N)NC c1(C(=O)NCC(CC=C)NC(=O)C(C)OCCC(C)C)cc(SC)cc(F)c1 c1(C(N2C(C)CCC(NC(CCCCCC=C)=O)C2)=O)cnc2cc(C)[nH]c2c1 C1(c2n(CCCCS(C)(=O)=O)nc(CN3CCOCC3)n2)CCc2nnnn2C1 N1(C(C2C(C=C)OCC2)=O)CCCC(C)C1CNC(C1(c2ccno2)CC1)=O C(=O)(CCCCNC(=O)C(C)(C)C1(O)CCOC1)NCCOC C1(NC(c2cnc(C)o2)=O)CC2CCC(C1)N2c1ncnc2[nH]cnc12 CC1CN(C(=O)Cc2cccc(Cl)c2)CC1CNC(c1cnn(C(F)F)c1)=O c1(C2(C(=O)NCC3(F)CC(NC(C4OCCO4)=O)C3)CCC2)c(F)cccc1Cl c1(C(=O)NC(CCC)CCCNC(c2cc(=O)cc[nH]2)=O)ccc([N+](=O)[O-])n1C CC(C#N)CCC(=O)NCC(C1CC1)N(C)C(c1cn(C2CCCC2)nn1)=O C1(CC)CN(C(=O)C(C)(C)c2cscn2)CCN1C(c1cn(CCO)nn1)=O C12(C(=O)NCc3ccc(CC)cn3)CCCC1CCN2C(c1sncc1C)=O C1(NC(C2CC(C)(O)C2)=O)C2CC(O)C1N(C(=O)C(Cl)=CCl)C2 C1(C(=O)Nc2c(C)nn(C)n2)CS(=O)(=O)CC12CC2 C(=O)(CC(C(C)CC)NC(=O)CC1(OC)CCOCC1)NCCC=CC=C C#CC(CC(C)(C)C)NC(=O)C=CCN(C)C(C1CCC2(CC1)CC2)=O c1(-c2onc(CNC(=O)C(=O)NC3CCCO3)n2)cccc([N+](=O)[O-])c1 C1(C=O)C2CC2CN1C(=O)C#CC(=O)O c1(CC)oc(C)cc1C(=O)N(CCCCC(=O)NC1(CF)CCCC1)C N1(C(c2c(OC)nccc2)=O)CCC2CN(C(C3CN(C)CCO3)=O)CCC12 C1(C(N2CCC(OCC)C2)=O)C2CCN(C(C3OCCC3(C)C)=O)CC12 C12(NC(c3c(CNC(C(CCC)OCC)=O)ocn3)=O)CCCN(CCC1)C2 c1(C(C)C)cccc(F)c1C(=O)NCC1CC(NC(c2cnc(C3CC3)s2)=O)C1 CC1CCCC(C(=O)NC2CCC(N(C)C(c3nccnc3N)=O)CC2)CC1 Cc1oc(Br)cc1C(N1CC=CC1CNC(=O)C=CCOC1CCOCC1)=O N1(C(c2cccc(OC)n2)C(=O)NCC=C)CCC2C(C1)C2(F)F C(CCCCCC(=O)N1CC(O)C(O)C1)NC(C(C)(C)c1ccno1)=O c1(OC)ncc(CN2CCC(C)(NC(=O)CN3CCOCC3)C2)cn1 N1(C(CNC(C2CCC2)=O)=O)CCCC1C(=O)NCC(CO)C1CCC1 c1(C(C)(C)NC(c2n(CCC)nnn2)C2CC=CC2)cnn2cc(Br)cnc12 N1(C(c2c(C)nc(CCC)o2)=O)CC(NC(c2sc(SC)cc2C)=O)CCC1C c1(CN2CCC(C(N(C(C)C)CC)=O)C2)ccc(-c2cccc(CO)c2)cn1 c1(C(=O)NC2(CNC(c3cc(CN(C)C)on3)=O)CCC2)cn2c(n1)CCCC2 N1(C(C(C)OCC2CC2)=O)CCCC(C2CN(C(c3ccc(O)nc3Cl)=O)C2)C1 c1(CN2CC3(CN(C(C4C(C)C4)=O)C3)C2)n[nH]c2cc(Br)cc(F)c12 CN1N=C(CC(=O)NC2(CO)CCCN(C(C3CCC(C)(C)OC3)=O)C2)CC1=O C1(CNC(C23C(C)OC(C)(C2)C3)=O)N(C(c2cc(Cl)sc2Cl)=O)CCCC1(C)C C(=O)(C(O)C1=CCCCC1)NCC1N(C(C(=O)NC(C)C2CC2)C)CCC1 CC1CN(C(C2CN(C(N)=O)C2)=O)CC(C)N(C(=O)Cc2cccc(F)c2O)C1 c1(C(=O)NC2CN(C(C(CC#C)O)=O)CC23CCC3)ccc(=O)n2c1COCC2 CC(C)C(C(=O)N(C1CCN(C(c2cn(C)cn2)=O)C1)CCO)c1cnn(C)c1 Cc1ccccc1-c1cccc(C(C2CCCC2)NCCCCCCl)c1 C(=O)(C(C)C(C)COC)NCCCN(C(c1cncc(N)c1C(F)(F)F)=O)CC C1(NC(C=C(C)C)=O)CC(C)(NSS(C)(=O)=O)C1.C1(=O)C(O)CN1 C1(CNC(C(COC)C)=O)CCC2(CCC2)CN1C(=O)C=C1CN2CCC1CC2 C=CCC(C(=O)N1CCC(CCNC(c2c(N)cc(Cl)nc2Cl)=O)C1)C(C)C C1(CNC(CC2(NC(c3c(C)snc3)=O)CC2)=O)CCC(=O)NC1C C1(C(=O)OCC)CCC(C(=O)Oc2nnc(COC)s2)CN1 CC(C)CC(C(=O)N1CCC1CNC(C1NC(=O)CCC1C)=O)N(C)C N1(C(Cc2c(C)nc(C)s2)=O)CC2CC(NC(c3c(C)nsc3C)=O)CC2C1 N1(C(CSCC)=O)CC(CCNC(c2cnc(SC)nc2)=O)C(C)C1 C1(C(=O)NC2(C)CC(F)(F)C2)CCOCCN1C(C1CCC(F)(F)C1)=O C(C)(C(=O)NCC1CCCC1N(C)C)(C1CCC1)NC(C(C)=CC(C)(C)C)=O C1(NC(C2(C=C)CCN(C(=O)C(C3CCCC3)OC)C2)=O)CCC2(CCCC2)C1 N1(C(C2(CC(C)C)CC2)=O)Cc2nccn2CC(NC(=O)CN2CCC(C)(O)C2)C1 N1(C(C)=O)CC2CN(C(C3CC(=O)N(C(C)C)C3)=O)CC2C1 Cc1oc(S(=O)(=O)N(C)C)cc1C(N1CC(C2CCCC2=O)C1)=O.C(=O)O N1(C(c2cncc(CC)c2)=O)CCN(Cc2cc(C)cc(C)c2)C(SC)C1 c1(C(=O)NC2C(CNC(CCP(C)(C)=O)=O)CC2)cc(F)c(F)cc1Br c1(C(N(CCN(C(c2cccc(F)c2)=O)CC)CC)=O)cc2sc(C)nc2[nH]1 c1(C(=O)NC2C(C)CN(C(=O)Cc3nncs3)CC2)cnn2ccncc12 c1(NC(C(CCOCCO)NC(CSCC)=O)=O)ccc(CC)c(F)c1 N1(C(c2c(CC)cno2)=O)CCC(C)(C)C(C(N2CCC(CF)C2)=O)C1 c1(C(=O)NC23CC(CNC(CCC(=O)NCCC)=O)(OC2)C3)[nH]cc2c1CCC2 N1(C(CCC2(C)CC2)=O)CCOC2(CC2)C1.C(=O)CC1CCC1 C1(NC(CCCCSC)=O)CC1C1CCCN(C(c2nn(C)cc2SC)=O)C1 N1(C(C)C)CCCN(C(=O)CC2CC3(CC3)CN2C(=O)C=Cc2nccs2)CC1 C#Cc1cc(C(=O)NCC2CCN(C(C3(F)CCC3)=O)CC2C)cc(Br)c1 CC(C)(C)C(C(=O)N1CCC(N2CCNC(=O)C2)CC1)NC(C12CC3CC1C2C3O)=O c1(C(N2CCCC(N(C)C(c3cnn(C)c3Cl)=O)C2)=O)cc2cccnc2o1 C1(C(NOCC(C)C)=O)CCCCC1(C)CCNC(=O)C=CCN1CCC1 C1(CN(C(c2[nH]cc(CC)c2)=O)C)CN(C(=O)CC(C)O)CCO1 c1(CNC(C(C)NC2C3=NOC23)=O)cc(-c2ccccc2)nn1C c1(OC)cccc([N+](=O)[O-])c1C(N1CC(O)(CNC(c2ccc(F)cn2)=O)C1)=O N1(C(C2C(C)C(=O)C2)=O)CCOCC1CNC(c1ccn(C(F)F)n1)=O CC1(C)CCN(C(=O)CC2CCCC23CC3)CC1CNC(C1(F)CC1)=O CC(C(N)C(=O)NCCC1(C#N)CCCC1)c1ccccc1 C1(CC)CN(C(=O)C(C)CNC(=O)Cc2cc(C)no2)CCC1NC(C)=O N1(CC(=O)NCCC(C)(C)NC(=O)C=CC(=O)N2CCC2)CCCCC1=O N1(CC(COC)S(=O)(=O)OC)CCC(=O)N(Cc2cc(Cl)cc(OC)c2O)C1=O N#CC1CCCCC1NC(=O)CNC(=O)CN1CC=CC1 Cc1nsc(C(N2CCCC(CC(=O)NCc3ccnn3C)C2)=O)c1N c1(NC(C2CN(c3cc(CC4CC4)ncn3)CCS2)=O)ccc(F)c(C(=O)O)c1 Cc1c(C(N2CC(N(C)C(C)C3CC3)CC2C)=O)nc2ccccn12 C1(CNC(COC)=O)CC2(CCN(C(c3c[nH]nc3OC)=O)CC2)CO1 N1(C(c2cc(C(C)C)no2)=O)CCCC(CO)(NC(=O)CCC2CCCO2)C1 c1(-c2n(-c3ccc(COCC)cc3)nc(C3CC3C)n2)ccc2c(c1)NC(=O)CO2 n12c(N3c4cc(no4)C3)nnc1C1CC1C2.C(C)(C)(C)OCC.C1(CC2CC2)CCC1 N1(C(c2c(CC)[nH]c(=N)s2)=O)CCC2(CCC2NC(C2CC(C)N(C)C2)=O)CC1 C(C(=O)NC1CCCN(CCNC(=O)C2CC2)C1)(C(C)C)SC.C1(S)CC1 C(=O)(N=c1ccn(C(C)(C)C)[nH]1)C1CCCN(C(C(C)C2CCC2)=O)CC1 C1(N(C(C2(C(=O)OCC)CC=CC2)=O)C)CCN(C(C2(C)CCCCO2)=O)CC1 C(=O)(CCCCCCCBr)N1CCCC(CN(C)Cc2cc(F)c(F)cc2Cl)C1 C(c1c(C)noc1C)=CC(N1CCN(C(CCCNC)=O)CC1)=O CC(C)C(O)C(C)C(=O)N1CCC(C(=O)NCC(=O)N(C)C)(OCCO)C1 CCCN=C(NCC(C)CN(C)C(C)C)N1CCC(C(F)F)C1 N1(C(CCC(=C)Cl)=O)CCCCN(C(=O)CCCCC2CCCCC2OC)CC1 N1(CCNC(C(C)OCC)=O)CCN(C(=O)Nc2c[nH]nc2-c2cccs2)CC1 CCCCCC(C(=O)NC(C)(C)CC)N1CCN(c2cccc(Cl)c2C)CC1 c1(C(=O)NC(CNC(c2cc(C(F)(F)F)on2)=O)CO)ccc(Cl)nc1O C1(CNC(C2(c3nccs3)CCCCC2)=O)CCCN(C(c2ccncc2)=O)C1 N1(C(CC2(OC)CN(C(C3C(OC)C3)=O)C2)=O)CCCN(CC(C)O)CC1 c1(C(C)C)nc(=NC2CC(CCN(C(c3cc4ccncc4s3)=O)C3CC3)C2)s[nH]1 N1(C(CCNC(C)=O)=O)CCN(C(C2OCCOC2C)=O)C(CC(F)(F)F)C1 N1(C(c2[nH]cc(C(C)C)c2)=O)CC2CCC(CNC(C3(C(=O)N(C)C)CC3)=O)(C2)C1 C1(CC(F)F)(COC)CCN(C(=O)Nc2ccc(C3CCCOC3)cc2)CC1 c1(C(=O)NC(CC=CC(=O)NC(C)CC(F)(F)F)(C)C)cc2cccnc2[nH]1 c1(NC(C2N(C(Cc3cnc(C)s3)=O)CC2)=O)cc(Br)ccc1[N+](=O)[O-] c1(NC(N2CCC(CC(=O)NCC(=C)C)CC2)=O)ccc(N(C)C)c(F)c1 N1(C(c2cnc(C3CC3)s2)=O)CCCS1(=O)=O.c12cn(nn1)CC1CN(C1)C2 c1(N2CC(C)C(NC(c3cccnc3N)=O)C2)nc2ncc(Cl)cc2o1 c1(C(N2C(CC(=O)N(C(C)C(C)C)SCC)CC2)=O)cc2n(n1)CCO2 N1(C(CC=C=C)=O)CCCC(CN(C(=O)CC2CCOC2)C)CC1 c1(C(N2CCC(C)(CC(=O)NC3CCC(C)(O)CC3)C2)=O)ccc2[nH]ccc2c1 C1(NC(CC=C=C)=O)CCC2(CC1)CN(C(=O)Cc1n[nH]c3ccccc13)C2 CCCC(CCC)CC(=O)N1CCCCC1CCCNC(C12CC(OC)C1C2)=O N1(C(CNc2ccc(OC)cc2)=O)CCCC(N)(CO)C1 CC1CCCN(Cc2ccccc2NC(=O)COCc2ccccc2)C1 C(C(=O)N(CCC(=O)NCC(C)(C)OCC1CC1)C)(OC)OC C1(C(N(C(C)C(C)(C)C)C)=O)(CF)CCN(C(=O)Cc2ccc[nH]2)C1 c1(CCNC(C(C)n2cnnn2)=O)ocnc1CNC(=O)Cc1ccco1 c1(NCC2CCN(C(c3c(C)cc(Br)cn3)=O)CC2)ncc(S(=O)(=O)O)cc1Br C1(Cn2c(N3C(C)CSCC3)nnc2C2CCC2)CCCCC1(F)F Cc1sc(Br)nc1CC(=O)NC1CC(NC(=O)COCCF)C1 C1(CNC(Cc2n(C)nnc2)=O)CN(C(C2(C)CCOC2)=O)CC12CCC2 N1(C(C2CC(OC)C2)=O)CC2(COC(CNC(c3cn(C)cn3)=O)C2)C1 O=C(CS(=O)(=O)c1ccc(Cl)cc1)NCC1(O)CN(C(=O)C=CC(F)(F)F)C1 C1(C(CC)CC)CCC(NC(C(=O)NCCCOC)=O)CC1 C(CNC(C1(CO)CCOCC1)=O)(C(C)C(C)C)NC(c1cc(COC)no1)=O c1(C(=O)NCC2(NC(C3CN(C)C3)=O)CC2)coc2c1CCCC2 C(=O)(C(C(C)(C)C)N(C)C)N1C(C(CNC(c2ccc(C)o2)=O)(C)C)CCC1 CCC(C(C)C)C(=O)N1CC2CC(NC(c3ccc(C(=O)OC)cc3)=O)C1C2 C#Cc1ccc(C(=O)NC23CCC(C(=O)NC4(CCC)CCOC4)(CC2)C3)nc1 Cc1cnc(C(C)NC(=O)C(C2CCOC2)NC(=O)Cc2ccc[nH]2)s1 C(C(CC1CCCC1)C(=O)NC(c1ccns1)C)NC(CCCC)=O c1(C(=O)NCC23CC2CN(C(=O)C(F)F)C3)cc(O)ncn1 N1(C(CN(C2CCC2)C)=O)CCCC(NC(c2cocc2C(N)=O)=O)C1 c1(CC(C(=O)OC(C)(C)C)OC(=O)NCCOCC=C)cc(Br)ccc1[N+](=O)[O-] C#CCCCCC(=O)NCC1CN(C(=O)C=CC(F)F)CCC1C N1(C(C2(C)N(C)CCC2)=O)CC(C2CN(C(=O)CN3CC4CC4C3)C2)C1 CC(C)CCC(=O)N1CCCC(NC(=O)CC2CCCC2)C1 C1(C(N2C(CC(=O)NCC3(OC)CCC3)CC2)=O)(CO)CCCO1 c1(OC)ccc(C(N2CC3(CCC3)C2C2CCOCC2)=O)nc1N c1(N2CCCC(OCCOC)C2)nc(=NC2CC(OC(C)C)C2)[nH]c2c1CCC2 C1(NC(C2C(OCC)C2)=O)CC(O)CN(C(c2ccc(Cl)cc2)=O)C1 N1(C(COCCCCC=C)=O)CC(C)N(C(=O)CCCC(C)C)CC1C CC1(C)CCCC1(C)NC(C1CN(C(c2ccnc(O)c2)=O)CCO1)=O c1(NC(=O)CC2CCN(C(c3cnc(Cl)cn3)=O)C2)cc(F)c(Cl)c(Br)c1 c1(Cn2cc(C3(O)CN(C(=O)CCCCC4CC4)C3)nn2)cc(Cl)ccc1Cl Cn1ccc(C(F)=C2CCOCC2)n1 c1(OCCC(=O)NC(CN(C(C2C(CCC)C2)=O)C2CC2)CC)ccncc1 C1(NC(=O)CC2CCOC2)CCCC2CN(C(c3ccc(O)c(Cl)c3)=O)CC12 c1(NC(CSC)C)ccc(S(=O)(=O)NCC2CCOC3(CCC3)C2)c(Cl)c1 c1(OCC2C(c3ccc(C)cc3)C2)cc(F)ccc1C C(c1cc2ccccc2o1)=CC(=O)NC1CC(NC(c2n(C)ccc2)=O)C1 C1(C)(NC(C)=O)CCN(C(=O)CC2CN(C(=O)COCCCN=[N+]=[N-])C2)C1 N1(C(c2c(OC)csc2)=O)CC(NC(C2CC23CCOCC3)=O)CC(F)(F)C1 c1(N2CCCC(CN(C(c3c(CC)occ3C)=O)C)C2)nc(OC)c(F)c(C)n1 N1(C(C(CO)N(C)C)=O)CCC(C)(CC(=O)NCCN2CCOCC2)C1 c1(CN2C(C)CN(C(Cc3c(C)cc(Cl)cc3)=O)CC2)ccccc1N=[N+]=[N-] C=CCC(C(=O)N1CCC(F)(F)C(CNC(=O)Cc2cnoc2)C1)C(C)(C)C C(=O)(CC(CCCC)NC(=O)CCc1cncnc1)N1CCCC(C#C)C1 CCCCCC(O)CC(=O)N1CCN(C(C2CN(C(C)C)C2)=O)CC1C(F)F CC1(C)CCC(NC(c2coc(Cl)c2)=O)C(CNC(=O)CC(F)(F)F)C1 c1(C(=O)N)cc(OC)nn1C.c1(C(CC)NC(=O)CC2CC2C)noc(C)n1 c1(OCCC#C)ccc(C(=O)NCC(CC2CC2)CO)cc1 C=CCC(C(=O)OCC)NC(=O)CCN(CC=C)C(C1C2CCCC12)=O N1(C(c2ccc(COC)o2)=O)CCC(NC(C2CCN(C)C(=O)C2)=O)C(C)(C)C1 Cc1cc(C(=O)NC2CC2CNC(=O)C(C(C)C)N2CCCCC2)c(O)nc1C CC1CN(C(c2ccccc2Br)=O)CCN1c1ncncc1I C1(NC(c2nn(C)c(CO)c2)=O)CCN(C(=O)C=Cc2cncs2)CC1(C)C C(=O)(CC(C)C(C)(C)NC(c1ccn2cccc2c1)=O)OCC c1(C(N2CCCC(C)(CNC(c3cnc(C)[nH]3)=O)C2)=O)ccnc2ccccc12 N1(C(CNS(CC)(=O)=O)=O)CCN(C(=O)C(c2cccc(Cl)c2)(C)O)CCC1C c1(CC(=O)NC(C2CCCN2C(=O)C(F)n2ccnc2)C)ccc2nn[nH]c2c1 c1(N(CC=C2CCN(c3ncncc3C#N)C2)C(=O)OC)ccccc1[N+](=O)[O-] N1(C(c2cc(Cl)ccc2F)C(=O)NC)CCCc2cc(C(C)(C)C)ccc21 C#CCC(CC(=O)N1CCC(C)(COC)C1)NC(=O)C(CC(C)C)N(C)C C1(CNC(=O)CN2CC3CC3C2)CN(C(=O)CN2C(=O)CNC2=O)CC1O N1(C(C2CCN(C)CC2)=O)CCC2(CCN(C(C3(C)CC=CCO3)=O)C2)C1 Cc1cc(NC(C2(C)CCN2Cc2ccc3n[nH]cc3c2)=O)c(F)cc1F c1(OC)cccc(NC(C2(C)CCCN2C(c2ccnnc2)=O)=O)c1O N1(C(C2C(OCC)C2)=O)CCC(C(C)C(=O)NC(c2cc[nH]n2)(C)C)C1 c1(OC)ccc(C(O)C(N2CC(NC(c3ccccc3F)=O)C(C)C2)=O)cc1 c1(C(N(C2(C#N)CC(C)C2)Cc2cccc(OC)n2)=O)cccc([N+](=O)[O-])c1 c1(C(=O)NCC2N(C(CC(=C)C)=O)CC(C)(C)C2)cc2c(o1)CCCC2 N1(C(CCCCOCC)=O)CCC2(CCCN2C(=O)CC2NC(=O)NC2=O)CC1 c1(C(=O)NCCC2CC(NC(C3(OC)CCC3)=O)C2)cnc(C)nc1 C1(CNC(C(CC)NC(N)=O)=O)CN(C(c2ccc(OC)nn2)=O)CC(C)(C)C1 c1(C(=O)NC(CC2CN(C(c3c(C)onc3CO)=O)C2)C)cnc(O)c(F)c1 c1(C(c2noc(-c3cc(C4CC4)[nH]n3)n2)(C)C)ccc(C(F)F)cc1 N1(C(C23CC(C)(OCC2)C3)=O)CCCC(C2CN(C(C34COCC3C4)=O)C2)C1 OCCS(=O)(=O)NNC(=O)C12CC1CCC2(F)F.c1(CN)ccccc1 Cc1cn2nc(C(=O)NCCCC(C)NC(C34CC(C3)C4)=O)cc2c(=O)[nH]1 c1(C(C(=O)NC(CNC(CN(CCC)C)=O)CN(C)C)O)cccnc1 C1(C2(O)CCOCC2)(C(N2CC3CCN(C(=O)C4=C(Cl)CCCC4)C3C2)=O)CC1 C1(CNC(CCCN(C)C)=O)CN(C(c2c[nH]nc2C2CCCCC2)=O)CCO1 c1(C(=O)NC2C(CNC(C=CC(C)C)=O)CC2)cc(C(C)(C)C)n(C)n1 C1(C(N2CC(C(C(=O)NCC(O)CSC)OC)C2)=O)CCOC1(C)C n1(CC(C(=O)NC2(CF)CCN(C(C(C#C)(C)C)=O)C2)C)ccc2ccccc12 C1(CNC(COCC)=O)CC(OC)CN1C(C1(n2nccn2)CC1)=O N1(C(Cn2cc(CCC(C)(C)O)nn2)=O)CCCC(Oc2ncc(Br)cc2)C1 C(=O)(C(CC#N)c1ccccc1)NCCN(C(C)C)C(c1cnoc1C(C)C)=O N1(C(C(C)N(C(=O)C=Cc2cnn(C)c2)C)=O)CCC2CCN(C)CC12 O(NC(=O)CC(C)COC)CC(N1CCCC(COC)C1)=O CC1(C)CC2(CC(C(=O)N(C3CCN(C(=O)C(C)(C)O)CC3)CC(F)(F)F)C2)C1 Cc1cc(Cl)n[nH]c1=NC(=O)C1(F)CN(C(c2cc(Cl)cc(Cl)c2Cl)=O)C1 CC(C)(C#CC(=O)Nc1cccc(F)c1O)CNC(C1CCCC1O)=O C1(c2n(CCC)nnn2)(NCc2cn(C3CC3)nn2)CCC(CC)C1 N1(C(c2cccc(C)c2Cl)C(=O)Nc2ccccc2C)CCC(O)C(C)(C)C1 N1(C2CCN(C(c3csnc3Br)C(=O)NC3COC3)CC2)CCC(F)(F)CC1 c1(NC(C2(C)C(C(=O)OC)C2)=O)cc(Cl)ccc1OC.C12CC(OC)CN1C2=O C#Cc1cccc(C(N2CC3(C2)CN(C(C2CC2c2ccoc2C)=O)C3)=O)c1F C1(NC(c2c(C)csc2)=O)CS(=O)(=O)CC1NC(c1c(C(F)(F)F)coc1C)=O N1(C(CCN2C(C)CCCC2)=O)CC(C2(NC(C3CC(n4cccn4)C3)=O)CC2)C1 C1(C(=O)NCc2c(C(=O)NCC(CC)C)n[nH]c2)CN(C)CC(C)O1 C1(c2n(C(C)C)nnn2)(Nc2ccc(F)c(Cl)c2)CN(C)CC1C c1(C(=O)NCC2(O)CCCN(C(CC3(COC)CC3)=O)C2)ccc2occc2c1 CC1(C#CC(=O)NCC2CCCCC2NC(C2CCCC3C2C3(F)F)=O)COC1 C=CCCCCC(=O)NCC1CN(C(c2c(C3CCC3)cnn2C)=O)C1 Cc1nn(CC(=O)NCC(C)(C)CN(C(=O)CCN2CCOC2=O)C)c(=O)o1 c1(C(N2CCC3C(CCN3Cc3cc(Br)cc(I)c3)C2)=O)ccc(I)c([N+](=O)[O-])c1 N(C1CCC(NC(=O)CC(C)(C)O)c2ccccc21)C(CC=C=C)=O c1(CN(C2CCCC2)CC(C)C)c(F)ccc(C#N)c1F C1(NC(c2c(COC)cc[nH]2)=O)COC2C(NC(=O)CN(C)C(C)=O)COC12 N1(C(CC(C)=C(C)C)=O)C(CC(=O)NCC2(C)CCCC2)C2CCCC12 N12CCCCC(C1)CC2=O.C1(NC(C=C(C)C2CC2)=O)COCC1CN(C)C CS(=O)CCC(=O)NC12CC(CNC(c3ncoc3-c3cccc(F)c3)=O)(C1)C2 C1(NC(CS(=O)(=O)NC)=O)CN(C(=O)CC2CCC3CC3C2)CCC1(F)F Cc1ccc(CC(=O)NCC2(C(N3CCN(C)C(C(C)C)C3)=O)CCC2)cc1O C1(CC(=O)NC(C2CC2C(N2CC(C3CCCO3)C2)=O)C2CC2)CC(F)(F)C1 CCCC(C)C(=O)N(C(C)(C(N1CCC(C)(CO)C1)=O)C1CC1)C N1(C(c2cnc(CC)s2)=O)CCCC(NC(c2cc(C)c(C)o2)=O)CC1 N12CCOCC(C1)NC(=O)CCC2=O.c1(CC(=O)NCC)cc(Br)ccc1C Cc1ccnnc1C(=O)NC1CCOCC1C(=O)NCc1c(C)coc1C N1(C(CCCc2onc(C)n2)=O)CC2CCCC(NC(C3CCNC3=O)=O)C2C1 CC1(NC(=O)CC2(C3CC3)CC2)CC(NC(=O)C(O)C2CCCC2)C1 C1(NC(C2(COC)CCC2)=O)CCN(C(c2ccc(C3CC3)nc2O)=O)CC1F C1(C)C(C)(C)C(=O)N1.C(C)(CCC(=O)N(CC(=O)NC)CC1CC1)OCC Cc1ccccc1N1CC1C(=O)NC(C)(CNC(c1ccnnc1)=O)C1CC1 C1(OC(C)C)CC(NCCCc2ccccc2)C1(C)C c1(CC(N2C(C)CC(NC(CCOCCC)=O)C2)=O)c(Cl)cccc1Br C1(C(N2C(COC(CC3(C(=O)OCC)CCC3)=O)CCC2)=O)CCCN(C)C1 c1(C(=O)NC(C2(O)CN(C(C3COCCN3C)=O)C2)C)cc2cc(F)ccc2o1 C1(CNC(c2c(C)cc(C)s2)=O)CC2CCC1N2C(c1cc(CO)on1)=O c1(N(CCCN(C(C2CC2Cl)=O)CC)C)ccnc(C2CCC2)n1 N1(C(c2ccn(C)c2)=O)CCN(C(c2cccs2)=O)CC1CO Cc1cc(CC(=O)NCCC2C(C)CCCN2C(c2cscc2C)=O)ccc1F C1(CC(=O)N(C2CCCOC2)CC)(OC)CN(C(C23CCC(C2)C3)=O)C1 C1(CNC(C2CCN(C(C(CCC)OC)=O)C2)=O)CCCN(C)C1=O c1(OCC)nccc(C(=O)CNC(N2CCC(C)C(c3ccc(O)cc3)C2)=O)c1Br c1(C(=O)NC2CC(CCNC(=O)CN3CCOC3=O)C2)cnncc1O Cc1cc(C(=O)Nc2cccc(C#N)n2)nc2ccc(I)cc12 C1(C2C(C(=O)NC3(CCNC(=O)OC(C)(C)C)CC3)CCC2)(CC2CC2)CCOCC1 C#Cc1ccc(OCC(N2CC(NC(=O)CC3CCC3)CC2COC)=O)cc1 c1(C(=O)NCCCN(C(=O)CCCn2cccc2)C)cccc2oc(=N)[nH]c12 CN1CCc2c(CNCc3csc(=N)[nH]3)cccc21 C1(NC(C(C)N(C(=O)C(F)OC(F)(F)F)CCC)=O)CCCCC12CC2 C12(CC)CN(C(C3CC(C)OC3=O)=O)C(CNC(=O)C(C)(C)C)(C1)C2 C1(C(=O)NC(C2CCOC2)C#C)CC2(C1)CN(C(=O)C(C)(C)c1cccs1)C2 C(=O)(C1=CS(=O)CCC1)N1C(CCNC(c2ccc(C)nc2N)=O)COCC1 C1(NC(c2nc(COC)oc2)=O)CC2(C1)CC2C(=O)NC1CC12CCC2 C12(NC(CCC=C)=O)CC(CO)(C1)OC21CN(C(=O)C(C(=O)OC)OC)C1 c1(C(=O)NC23C(CN(C(CS(CC)=O)=O)C2)C3)ccc2ncncc2c1 C1(NC(C2CCCC(O)C2)=O)CCCC12CN(C(=O)CO)C2 C(C1(C)COC1)=CC(=O)NC1(CN(C(=O)Cn2ccc(Br)n2)C)CC1 c1(CNC(c2ccco2)=O)ccccc1-c1csc(C(=O)NCCCCCO)c1 c1(CC2N(Cc3c(C)nc(C4CCCO4)s3)CCC2)cccc(F)c1Cl CCCC(C#N)C(=O)NCC1CCN(C(=O)Cn2cnc([N+](=O)[O-])c2)C(C)C1 c1(C(=O)NC(C(C(C)C)NC(C(C)NC(=O)OC)=O)C)cc2c(s1)CCCCC2 c1(C(=O)NCCC(C)CCNC(C2CCC(C#N)CC2)=O)ccc2cncn2c1 C1(C(N(C2CCCN(C(c3c(C)coc3)=O)C2)C)=O)CCCc2ccccc2C1 C1(OC)(CNC(=O)CC2CC2c2cnn(C)c2)CN(C(=O)CSc2nccn2C)C1 Cc1nc(N2C(NC(=O)Nc3cc(Br)cc(C#N)c3)CC3CC23)c2c(n1)CCC2 CCC(CC)CCC(=O)N1CC2(C1)CN(C(c1cncnc1)=O)C2 C1(n2cc(-c3cn(C)nc3)nn2)CC2CCC1(NC(c1nscc1Br)=O)C2 N1(C(C(CC(C)C)OC)=O)CCCN(C(c2cncc(C)n2)=O)C(C(C)C)C1 N1(C(C(CC#C)O)=O)CCCC(NC(c2ccc(-c3nnc(C)o3)cc2)=O)C1C C(CC(C)C)(C(=O)N1CCC=C(F)C1)N(C(C(C1CCC1)OCC)=O)C C1(CN(CCCCCO)C(c2ccc(CC)[nH]2)=O)CN(C(C)C)CCO1 c1(NCC(Br)=C(C)C)nc(=NCC2CCC3(CCC3)O2)[nH]c2c(C)nn(C)c12 C(C)(CO)(CC(C)C)NC(c1cc(CNC(c2c(OCC)ccs2)=O)ncc1)=O Cc1ccc(C2CC2)cc1C(N1CCN(C(=O)Cc2c(C)cnn2C)C2CC12)=O CC(C)CCCCCC(=O)NC1CCOCC1NC(c1cc2cccnc2[nH]1)=O c1(C(C)=O)cc(C(=O)NCCCNC(=O)C(C)NC(C2CCCCC2)=O)co1 C1(N(C)C(c2cc(=O)cc[nH]2)=O)CCCCN(C(=O)C(CN)c2ccccc2)C1 O=C1CC(NC(c2coc(CNC(=O)CC3CCCCO3)n2)=O)CC(=O)N1 CCC(CO)CCNC(=O)CC(C)NC(=O)C(c1ccnn1C)C c1(C(C)=O)ncnc2ncn(C3CCN(c4ccc(I)cc4Br)CC3)c12 c1(C(CC(=O)NC(CNC(CN(CCOC)C)=O)C(C)C)C)ccc(F)cc1F C#CCC(C)(CC)C(=O)N(CC(C)NC(=O)C=Cc1ccc(Br)cc1F)C C1(C(N2C(C(C)NC(c3c(COC)ccs3)=O)CCC2)=O)C2CCCCC12 c1(C(=O)NCC(CNC(CC2C(C)(C)CCC2)=O)F)cc(Cl)c2n[nH]cc2c1 N1(C(c2ccc(C(C)C)s2)=O)CCC2(NC(c3nc(Cl)sc3Cl)=O)CC2C1 C1(CN(C)C(C2CC2(C)C)=O)CCCN(C(=O)Cc2ccn(C(F)F)n2)C1 C1(C)(NC(c2nc(C)n(-c3nc[nH]n3)n2)=O)CCCN(C(C2OCC2(C)C)=O)C1 N12CC3CCCC3(C1)N(C(C)C)C2=O.c1(O)cccc(C)c1.C(C(O)CCCCN)CC O=C(CCCCCn1cc(C2CCCCC2)nn1)N(CC(F)F)CC1CCCSC1 C1(C)(CCC)CCCN(C(=O)C(C)C(C)NC(c2ccccc2O)=O)C1 N1(C(C2CC(OCC)C2)=O)CC(C(N2CCC(C(C)(C)C)C2)=O)C2(CC2)C1 C(CC1=CCCCC1)N(C(CCNC(CCCC=C)=O)=O)C(C)C CC1=CCC(C(=O)NC(C)(C)CCNC(=O)CNc2ccc(C(N)=O)cn2)CC1 C(c1ccc(F)cc1)=C(C(C(=O)NCC)N1CC(C)(C)C1C1CC1)C S(=O)(=O)(c1cccc(Cl)c1)Nc1c(C)cc(C2CCCN2C(=O)CN)cn1 c1(C(N2CCCN(C(C(CCC)(C)CC)=O)CC2)=O)cnc2c(c1)CCCC2 c1(C(N2C(C(C)NC(C(CCSC)O)=O)CCC2)=O)cc2n(n1)CCCNC2=O C12(C(=O)OCC)CC(C1)C(Nc1cncc(Cl)c1C(=O)O)CO2 C(=O)(CC(C)(C(F)F)N(C)C)N(C1CCN(C(CC(CC)C(F)F)=O)CC1)C C=C(Cl)C(C)(C)C(=O)N1CCCN(C(=O)C=C2CCC2)CC1 CC1CCCC1CC(=O)N(C)CCOCCCNC(=O)C=Cc1ccoc1 S(=O)(=O)(c1cccc(F)c1)NCC(=O)NCC(CCNC(CC1C(OC)CC1)=O)O c1(OC)c(C(=O)NC2CCC(CO)C2)ncnc1Cl C#CCC(C(=O)NCc1cccc(O)n1)NC(c1cnn(C)c1C)=O c1(C(=O)NC(C)CNC(=O)CC(=O)N(C)C)cc(Cl)c(F)c([N+](=O)[O-])c1N Cc1ccc(Cl)c(OC(C)C(=O)NC2(CCOC)CCN(C(=O)C(C)(C)O)C2)c1 C(C1CCCCC1)=C(C(=O)NCC(C)(C)OCCNC(C1CC(F)(CC)C1)=O)F C12CCCN(C1)C2.CC(CC(=O)N(C)Cc1ccc(C(=O)O)s1)n1cccn1 C1(NC(C(CC)OCC)=O)CCC2(CC1)CCN(C(=O)COCCCF)C2 C1(NC(c2c(Br)n[nH]c2C)c2n(CCC)nnn2)CCn2ncnc2C1 C=CC(C)(CC)C(=O)NC1C2CCN(C(c3ncccc3Cl)=O)CC12 c1(CCC(=O)NCC(C)NC(C(C)(C)OCC)=O)nc2ccccc2[nH]1 c1(CCCNC(=O)C(N2CC(CCO)C(O)C2)=O)ccc(O)cc1 n1(CC)nc(C(N2CC(C(C)NC(C3CCC(=O)N3C(C)C)=O)C2)=O)ccc1=O c1(C(=O)NC2CCC(CCNC(C(C)(C)OC)=O)C2)cn(CC2CC2)nc1C CCC(CC)CCCC(=O)NOC(CC(C)C)C(=O)N1CC(C)(OC)C1 C#CCCCCCCCC(=O)NCC1(CO)CCN(C(=O)CN2CC3CC3C2)CC1 C(=O)(C(F)C(=O)CC)OCc1cn(-c2cncc(Sc3ccc(N)cc3)c2)nn1 c1(C(=O)NCCC(C)CCNC(C2CC23CC3)=O)cc2ccncc2o1 c1(OC)ccc([N+](=O)[O-])cc1S(=O)(=O)N(C)Cc1cc(Cl)cc(Br)c1 C(C(CC1CC1)C(=O)N1CCC(OCC(N)=O)C1)CNC(Cc1ccn(C)c1)=O N(C1CCc2cc(CNC(c3cnnn3C3CC3)=O)ccc21)C(CCOCC)=O C(=O)(N=c1[nH][nH]c2cc(C#N)ccc12)C1CCC(NC(COCCOC)=O)CO1 CC1C(NC(C2CC2C(F)F)=O)CCCN1C(c1cc(C(F)(F)F)cnc1O)=O c1(C2C(C(=O)NCC(C)NC(C3CN4CCN3C(C)C4)=O)C2)coc2ccccc12 N1(C(CN(CC)CC)=O)CCC(N(C(=O)C(O)CCn2cncn2)NC)CC1 C=CCCN=C(NCc1ncccn1)N1CCc2c(Br)cc(C)cc2C1 N1(C(CC2(C=C)CN(C(=O)C(O)C3CCC3)C2)=O)CCS(=N)(=O)CC1 c1cc(F)c(F)cc1O.C1(OCCCC(=O)NC)CCC(C(=O)NC(C)=O)CC1 C(=O)(C1=CS(=O)(=O)CCC1)N1C(COC)CN(C(c2ccsc2Cl)=O)C1 CC1(C)CC(CNC(=O)COc2ccccc2)N(C(C2CC(F)C2)=O)C1 C#CCC(CC(F)(F)F)C(=O)N1CCC(C(=O)NC2CCCS2(=O)=O)CC1 C12(C(=O)NC(CC=C)(C)C)CC(CN1C(=O)Cc1csc(C)n1)C2 C1(C(C)NC(CSCCOC)=O)CCN(C(=O)Cc2cnn(C)c2)CC1 C(CCC)(C(=O)NCC(c1ccc(F)cc1)NC(C1CS(=O)(=O)C1)=O)=CCC C1(NC(C(C)OCC)=O)CC2CC(C1)N(C(=O)Cc1noc3ccccc13)C2 Cn1cc2c(n1)CCCC2C(=O)N1CC(O)(CNC(=O)CC2(C#N)CC2)C1 c1(CNC(NCC(C)SC)=NCCCN(C)C)cc(C)c2ncccc2c1C c1(C(=O)NC2CCC(F)(CNC(C3(COC)CC3)=O)C2)ccc(C)c(Br)n1 N1(C(c2ccncc2F)=O)CCCC(C2CCN(c3ccn4nccc4n3)C2)C1 C(N=c1ccnc(C#N)[nH]1)C1CC(C)N(C(=O)C(C2CCOCC2)F)C1 Cc1n[nH]c(C)c1CC(=O)NC1CCC(CCNC(c2cn(C)nc2Cl)=O)C1 c1(C(=O)NC(C(=O)NC(C)Cc2ccco2)C2CCCO2)ccccn1 C(=O)(C(C)CCC(C)(C)C)NC1(C(=O)NCC(COCC)O)CCSC1 Cc1ccc(C(c2ccccn2)NC(=O)C(=O)NC23CCN(C2)S(=O)(=O)C3)c(C)c1 N1(C(C2C(CCC)CCC2)=O)CC2(C1)CN(C(=O)C(C1CCOCC1)C)C2 C1(C(=O)NCC(C)NC(C(C2CC(F)(F)C2)OCC)=O)CCC(=C2CCC2)CC1 c1(C(N2C3CN(Cc4c(Cl)cccc4I)CC23)=O)cc(F)c([N+](=O)[O-])cc1F c1(NC(Cc2nc(NC(C(CC)C)=O)sc2)=O)ccc(Cl)c(C#N)c1 N1(C(C(c2c(C)cccc2Br)NC(C2CCCOC2)=O)=O)CC(C)(C)C12CCC2 O=C(CCCCN1CCCC1)NC1CC(CC2(C(F)(F)F)CC(O)C2)C1 c1(C(=O)NCCNC(C23OCCCC2C3(F)F)=O)cccc2c1OCCC2 C1(CNC(c2ccc3cc[nH]c3n2)=O)C(C2CC2)CCN1C(=O)C=C1CCC1 N1(C(c2c(CCCC)ocn2)=O)CCC(CNC(c2cc(C)c(C)s2)=O)C(O)C1 c1(C(N2CC(C)OCC2)=O)noc2c1CN(C(=O)CCc1cc(F)ccn1)CC2 CCCC(C)(C)C(=O)NC(C)C(C(C)C)NC(c1cn(C)c(C)n1)=O C(C1CCOCC1)=CC(N)=O.C12(F)CC(C1)CNC(=O)NC2.n12ccnc1C2 C12(NC(COC(CC)(C)C)=O)COC(C1)C(NC(C1(n3cc(Cl)cn3)CC1)=O)C2 C1(C)(NC(C(C)Cn2ccnc2)=O)CCCN(C(c2ccc(O)cc2)=O)C1 N1(C(C(CC)OCC)=O)CC2CCCC2(NC(=O)CSc2ccccn2)C1 C1(NC(=O)CCCc2cccs2)(CO)CCN(C(C2CC(n3cnnc3)C2)=O)C1 CC#CCCC(=O)N1CCC(CN(C(=O)C(C(C)C)N2CCCC2=O)C)CC1 N1(C(c2cnn(CC)c2C)C(=O)NCCOCCOC)C2CCC1CN(C)CC2 c1(CCC(=O)N(C(CN(C(C2(CCC)CC2)=O)C)C)C)cccnc1C c1(C(=O)NCC2(O)CC(NC(c3c(C)coc3C)=O)C2)ncn2c1CCCCC2 c1(C(=O)NCC(N(C(c2c(C)ccs2)=O)C)C2CC2)cccc(C2CCOC2)c1 C(=O)(C#CC1(C)CCCO1)NC1(CNC(C=CC(CC)C)=O)CCCCCC1 c1(Cc2scc(C(=O)NCC(C(C)C)NC(C3(CF)CC3)=O)c2)ccccc1F N1(C(c2c(CC)nn[nH]2)=O)CCN(C(=O)Cc2cccn2C)CC1C(F)F c1(CC)n[nH]cc1C(=O)NCC1(CCNC(c2cc(C(F)F)cs2)=O)CC1 N(C=CC(=O)C(F)(F)F)C(C12C(CN(C(c3cc4cc[nH]c4cn3)=O)C1)C2)=O C(CN=c1ccc(Br)c(S(=O)(=O)N(CCCC)C)[nH]1)SCCS(=O)(=O)CCCC CCC(F)(F)C(C)(C)C(=O)N1CC(NC(=O)C(C)(C)CCSC)C(C)C1 C(C)(CO)(C(=O)NCC(C(C)(C)C)NC(=O)CCSC(C1CCCO1)C)OC C1(NC(C(c2ccnn2C)C)=O)CN(C(=O)C=C2CCCCC2(C)C)CCC1O C1(N(C(c2ccc(C)cc2)=O)C)CN(C(c2onc(C)c2C)=O)CC12CC2 c1(C(=O)NCC(C)NC(=O)CCCn2ccnn2)c(C(F)(F)F)sc2c1CCC2 C1(C(=O)NC2(C)CN(C(C(Cc3c(C)nc[nH]3)O)=O)C2)CCc2n[nH]c(C)c2C1 N1(C(=O)C(C2CC2Cl)=O)CC2(C1)CN(C(C13CCCN(CC1)C3)=O)C2 N1(CCCC=C)CC2OCCN(C(=O)CCc3ccc(OC)cc3Br)C2C1 CCC(C)C(C(=O)NCC=C(Cl)Cl)N(C(=O)Cc1cc(C)on1)C c1(CC)cc(OC)ccc1C(=O)NC(C)C(C)NC(=O)CCCCN(C)C(C)C N1(C(c2cnc(OC)c(Cl)c2)=O)CCOCC(F)(CNC(c2cnco2)=O)C1 C1(NC(CC2CC(=C)C2)=O)CN(C(c2cc(C(=O)OCC)[nH]n2)=O)CC1OC C#CCC(C)C(=O)NC(C1CCCC1)CNC(c1ccc(C(F)(F)F)s1)=O c1(OC)nccc(C(=O)NC(C)CNC(=O)C(C)(C)C2(O)CCC2)n1 C(C(COC)C(=O)NC1(c2ccccc2)CCN(C(c2cc[nH]c2)=O)C1)OC c1(CSCCNC(N(C)Cc2c(C)noc2C)=O)cccc(F)c1F C1(NC(c2nc(C(C)(C)C)oc2)=O)CC12CCN(C(=O)Cc1cccnc1)CC2 c1(C(N2CCCC2CNC(C(C=C)(C)O)=O)=O)ccc(C(=O)OCC)cc1O C1(NC(=O)NCCCc2nc(C)c(C)[nH]2)CCN(C(=O)OC(C)(C)C)CC1O CN1C(=O)CSC1=CC(=O)NC1CCCN(c2ccnc(Cl)n2)C1C C1(C(=O)NCC2C(CNC(c3c[nH]cc3C3CC3)=O)C2)CC1C1CCCC1 N1(C(C2C(C)C2)=O)CCN(C(c2cc(C3CC3)ccc2F)=O)C2(CC2)C1 N1(C(C2C3(CCC3)C23CCC3)C(=O)NCCCSC)CCCC2(CC1)CC2 N=C1NC(=O)C(CC(N2CC3CC3(CNC(C3CNC(=O)C3)=O)C2)=O)S1 C1(C(N2CC(CCO)(NC(=O)CC3COCCO3)C2)=O)(COC)C=CCC1 c1(CCNC(C2C(CNC(=O)C(O)Cn3cncn3)C2(C)C)=O)cccc(O)n1 Cc1nn(CCO)c2ncc(C(N3CC4COCC4(CO)C3)=O)cc12 Cc1ccc(C(=O)NCC(C2CCN(C(c3ccnnc3C)=O)CC2)C)cc1 C12(NC(c3scc(C(N)=O)c3)=O)CCN(C(c3cnc(Cl)s3)=O)CC1C2 C1(C(N2CCCC(N(C(=O)CSc3ccccn3)C)C2)=O)CCC(C)(C)OC1 CCCC(C(=O)NC1CC(OC)CN(C(=O)C=C(Cl)Cl)C1)OC CCCC(C)(C)CC(=O)N1CCN(C(c2cc(CSC)[nH]n2)=O)C(CCOC)C1 C(=O)(CCCCN=[N+]=[N-])NCCC(C(=O)NCC1CCC(=O)O1)N(C)C c1(C(N2CC(Cc3cn(CC(F)(F)F)nn3)C2)=O)ccc(Br)nc1F N1(C(C(C=C)O)=O)CC2(CCN(C(c3cnc(C)nc3C3CC3)=O)CC2)C1 N1(C(c2c(C)oc(Cl)n2)=O)CC(NC(=O)CC2CCC(F)(F)C2)C2CCCCC12 N1(C(c2c(C)cnnc2)=O)CCOC(C)(CNC(=O)CCCc2cccs2)C1 C1(C(=O)NCc2ccn(-c3ccccc3)n2)CCOC2(CCS(=O)(=O)C2)C1 C1(CC#C)(C(=O)Nc2cnn(CCF)c2)CCN(C(C2CCC3(CC3)C2)=O)C1 C(CC(F)(F)Cl)NC(CCN(C(=O)C(F)=CC)CC=C)=O c1(C(=O)NCC(C)NC(C2CCC3(CC3)C2)=O)cc(=O)n(-c2ccc(F)cc2)[nH]1 C1(CNC(C(N2CC(C)C2)C)=O)CN(C)CCN1C(c1ccc(C2CC2)cc1)=O c1(C(=O)NCC2(F)CCC2)cc2n(n1)CCCN(C(=O)CC1(O)CCC1)C2 C=C(C)CC(C)C(=O)N1CCCC(C2CCCN2C(c2cc(C)c(O)nn2)=O)C1 Cc1cc(C(=O)NCC2(CNC(=O)C(C)(C)N(S(C)(=O)=O)C)CC2)ncc1Cl N1(C(CCc2c(C)n(C)nc2)=O)CCC2C1CCCN2C(=O)CN1CCOCC1 N1(C(c2c(C)n[nH]c2C)=O)CCCOC(CNC(c2ccc(C3CC3)cc2)=O)C1 C1(C)(CC)C=C(C(=O)N2CCCC2CNC(C2CC3CCC3C2)=O)C1 C1(NC)(CO)CCN(C(C)=O)C1.C1(=O)C(C2CCOC2)CN1 CC1CN(C(=O)C=CC2CCC2)CC(C(=O)N(CCCC2CCOC2=O)C2CC2)O1 c1(C(N2CC(CNC(C3C(OC)C3)=O)OCC2)=O)ccn2cncc2c1 Cc1ccc(C(=O)NC2CC(NCc3cnc4ncccn34)C2)cc1[N+](=O)[O-] N1(NCC2N(CCC)CCC2)CCCC(O)(CC)CC1 N(C1CCCc2c[nH]nc21)C(C(C)CNC(=O)CCc1cn[nH]c1)=O C12(CNC(c3cn(CCCOC)nc3)=O)CCC1CCN2C(=O)C1=CCOC1 C1(C(N2CC(F)(C(=O)OC)C2)=O)CCC(C)(NC(=O)C(C)OCCN(C)C)CC1 Cc1cccc(N)c1C(=O)NC1CC(F)CN(C(C2CC2CF)=O)C1 C(CN=c1[nH]c(Cl)nc2c1CS(=O)(=O)C2)c1c(C)ccc(OC)c1 c1(-n2cc(-c3cnc(C(C(c4ccccc4)C)=O)s3)nn2)ccc2[nH]ncc2c1 C(C)(C)(CCC(=O)NC(C(=O)NCC(=O)N(C)O)C1CCC1)OC C(=O)(C(F)(F)CC(C)C)NC1C(CC)CN(C(=O)Cc2ccc(C)s2)CC1 C1(C(=O)NCC(C)(C)NC(c2csc(C(C)C)n2)=O)(OC)CCCCC1C C(=O)(n1c(NCCSC)cc(=O)cc1C)OC(C)(C)C.N1CCOC(C)(C)C1C C1(NC(C(c2ccccc2)OCC)=O)CN(C(=O)C(F)C(CC)CC)CC(C)(C)C1 C(=O)(C1=CS(=O)(=O)CCC1)NC(C)CCNC(C1(CC2CC2)CCCO1)=O CC1CCC(C(=O)NCC2CC(F)CN2C(c2coc(CO)c2)=O)CC1 c1(C(=O)NC(C)CCN(C)C(C2CN(C3CCC3)C2)=O)csc(=NC2CC2)[nH]1 CCC(CC)C(C(=O)NC(CCN(C)C(c1cc(C)c(Cl)cn1)=O)C(C)C)OC c1(CC(=O)NCCCCCN(C(=O)CN(C)C2CC2)C)ccc2c(cnn2C)c1 c1(C(=O)NCCCN2CCC(NC(CC=C=C)=O)C2)csc(=NC)[nH]1 C1(N(C(c2c(C)n(C3CC3)cc2)=O)C)CCN(C(C2(F)CCOC2)=O)CC12CC2 C1(NC(c2nccc(CC)c2)=O)CCCN(C(C2CC(C(C)=O)C2(C)C)=O)CC1 c1(CC)cccc(NC(=O)C(=O)NC2CN(C(=O)OCCOC(C)(C)C)C2)c1 c1(NC(C2N(C(CC#N)=O)C3C(C2)C3)=O)ncccc1Sc1cccs1 N1(C(c2c(C)cns2)=O)CC2CC(C1)CN(C(c1nccc3ccncc13)=O)C2 c1(C(=O)NC2C(C)(C)N(C(c3cc(Cl)cs3)=O)CC2)occ2c1CCOC2 C1(CCCC(=O)NCC(C)NC(=O)CS(=O)(=O)N(C)C)CCC(C)C1(C)C c1(CSC)cc(C)ccc1C(=O)NCC1(O)CN(C(c2cc(O)ccc2Cl)=O)C1 C1(CC)CCN(C(=O)Cc2cc[nH]n2)C1C(N1CCC(OCC(N)=O)C1)=O C(=O)(C(C)(C)c1ccn(C)n1)NCC(CNC(c1cc(C(C)C)no1)=O)OC C1(NC(C(CC=C)C)=O)CC2CCC(C1F)N2C(c1cnc(N(C)C)c(Cl)c1)=O c1(CC(N2CCN(c3ccc(C)cc3)CC2C)=O)cc(F)cc(F)c1Br Cn1ncc2ncnc(N3CC(C(=O)NCc4ncc(C(F)(F)F)[nH]4)C3)c12 CCC(O)C(C)(C)C(=O)N1CCN(C2CN(C(=O)CCCN=[N+]=[N-])C2)CC1 c1(C(=O)NCCNC(C(C)OCC2CC2)=O)nc(Cl)ccc1OC(C)(C)C C1(NC(C=C(C)C(C)(C)C)=O)CC2CN(C(=O)CS(=O)(=O)C(C)C)CC2C1 N1(C(CCc2nc(C)c(C)[nH]2)=O)CCN(C(=O)CC2CCOC2)C2(CC2)C1 C1(C(N(CCC(=O)NCC2C3CCCCC23)CC=C)=O)C2(CC2)C12CC2 N(C1CCCc2c1cnn2CCO)CCCSC C1(C(N2CC(CNC(CCSC)=O)C(C(F)(F)F)C2)=O)CCCC2(CCC2)C1 C(=O)(C(C)CC(=O)NC1(C(=O)NCC2(F)CCCCC2)CC1(C)C)OC N1(C=O)CCSCC1.c1(C(N(CCNCC=C(C)C)CC)=O)ccco1 C(=O)(CCC(O)C(C)(C)C)N1CC2(CN(C(C3CCN(C)C(=O)C3)=O)C2)C1 c1(C(N2C(C)C(C(=O)NC3(C(F)(F)F)CC3)CC2)=O)ccc2cc[nH]c2n1 C1(C(=O)NCC#CC)CC12CC(NC(c1ccncc1NC)=O)C2 C12(CNC(=O)Cc3cccs3)COCCN1CCN(C(C1CC1F)=O)C2 C1(CNC(=O)C=CCF)CN(CC(=O)N(CC)Cc2ccccc2)CCO1 c1(C(=O)NC(CCNC(c2c(C(C)C)n[nH]c2)=O)C)cc[nH]c2nccc1-2 Cn1cc(C#N)cc1C(=O)NC(C(=O)NCCSCCO)C(C)(C)C Cc1ccc(Br)c(NC(C2CC23CN(C(=O)Cn2cc(Br)cn2)C3)=O)n1 c1(CNC(C(CNC(C(CCC)C)=O)OC)=O)cc(C)cc(C)c1 C(=O)(C1=CCCCO1)N1C(C(=O)NC(C)C)C(C)(C)C1 C(=O)(C1=CC2CC(C1)CC2O)NC12CC(CNC(c3c(CC)noc3)=O)(OC1)C2 N1(C(CCCCC)=O)CC(C2CN(C(c3c(Br)c(C)nn3C)=O)C2)C1 c1(C(=O)NC(C2CN(C(=O)C(C(C)(C)C)NS(C)(=O)=O)C2)C)ccc2ccsc2c1 c1(CCC(=O)N(C)CC2(CNC(C3CCC(O)CC3)=O)CC2)cncnc1O C1(NC(CCN(CC#C)C(c2coc(C(C)C)n2)=O)=O)CCCC12CC2 Cc1nc2c(F)cccc2cc1C(=O)NCCN(C(c1ccon1)=O)CC1CC1 c1(N(C)CCC2(C)OCCO2)ccc(S(C)(=O)=O)nn1 c1(C(=O)NCC(CC=C)NC(c2csc(C(F)(F)F)c2)=O)c(C)coc1C CCCN=C(NCc1ccsc1S(C)(=O)=O)N1CCC(C(=O)OC)(C(C)C)C1 c1(C(=O)NCC(CN(C(CCCOC)=O)C)C)cnc(C)nc1 C1(C(=O)NCCN(CCCC)CCCC)CCC(NC(C2CCCC2)=O)CC1 c1(C2(C(N3C(CNC(CCC4CCN(C)C4)=O)CC3)=O)CCC2)ccccc1Cl C1(C(=O)NCc2c(C)noc2C(F)(F)F)CCC(C)CN1C(=O)Cc1cccs1 CC(C)CC(Cc1cn(C)nn1)C=O.C12(C(=O)O)CC(NC(=O)NC3CC3)(C1)C2 C1(CC(=O)NC(CNC(COC)=O)(C)CSC)CC2(CC2)CO1 N1(C(C(C)OCC#C)=O)CCC(NC(c2occc2-c2ccccc2)=O)C1C C(=O)(CCCS(N)(=O)=O)N1C(CNC(=O)NC2CCC(C)CC2)C=CC1 N1(C(c2c(CC)ccs2)=O)CCN(C(C2CCCS2(=O)=O)=O)C(CC)C1 c1(C(N2C(C(C)NC(c3c(SC)n(C)nc3)=O)CCCC2)=O)ccc(O)c(Cl)n1 c1(CCN=C(NC(C=C)C)NC2CC23CC(C)(C)C3)cccc2cc[nH]c12 CC(C)CCCCC(=O)NC1CC2CC1N(C(=O)CS(=O)(=O)C1CC1)C2 c12cc(c3cc[nH]c3c1)C(=O)NNC2=O.C(C)(CNC(=O)OC(C)(C)C)OC Cc1cn(C(C)C)cc1C(=O)NC1C2CN(C(C3(C(=O)N(C)C)CC3)=O)CC12 C(=O)(C#CC(C)(C)CNC(=O)CC1(C)CCOCC1)Nc1ccc(OC)c(C)c1 c1(CNC2CN(C(CC(C)O)=O)CC23CC3)n[nH]c2ccc(Br)cc12 Cc1nc(N(C2CNCC2O)C(C2CCCN2C)=O)c2cc(Br)ccc2n1 C(=O)(C(=O)CC(C)C)N1CCC(CC=C)(C(N2CC(O)(C(N)=O)C2)=O)C1 C=CC(CC)CC(=O)N(C1CCN(CC(=O)NCC(C)(C)CCOC)C1)C1CC1 N1(C(C2CCN(C(C)=O)CC2)=O)CCC2C(C1)CN2C(=O)C(C)c1ccsn1 Cc1c(C(N2CCCC(C)C2CNC(=O)Cc2cn[nH]c2)=O)sc2ccccc12 N1(C(c2[nH]ccc(=N)n2)=O)CCCCC(NC(c2cc(F)ccc2Cl)=O)C1 c1(OC(C(=O)NCC(C)CNC(C2CCC3(CC3)C2)=O)C)ccc(Cl)cc1Cl N1(CC(=O)N(C(C)C)C)CC(NC(C2CCCC2(C)C)=O)CCC1C C1(OC)CC2CCC1CC2C(N1CC(NC(C2CC(SC)C2)=O)CC2(CC2)C1)=O n1(CC=C)nnnc1C(c1cnc(C(C)C)[nH]1)NC(C1CCOCC1)C N1(C(C2N(C)C(=O)CC2)=O)CCOC2CCN(C(C3(F)CC4(CCC4)C3)=O)CC12 N1(C(C=C(C)C(F)F)=O)CCC2CN(C(C3CC=CC3)=O)CCC2C1 C(=O)(C1=CC2(CCN(C(c3nc[nH]n3)=O)C2)C1)NCCC(CCC)C1CC1 C1(C(C=CC(=O)NC2(CNC(C(C)(C)n3cccn3)=O)CC2)=O)CCS(=O)(=O)C1 CC1=C(C(=O)NC(CNC(C2CCS2(=O)=O)=O)C2CC2)CC1 C1(NC(CSC)=O)(CNC(c2nnc(C)s2)=O)CCOCC1 N1(C(=O)CCCCC2CCCCC2)CC2CC(NC(=O)C(F)(F)C(F)(F)F)CC2C1 CCCCC(C)(F)C(=O)N1CCC(C)(CNC(=O)C(C)(CC)OC)CC1 C1(NC(CC=CC)=O)CC(O)CN(C(c2ncncc2Cl)=O)C1 c1(C(=O)NCC(CC)NC(C2CN(c3nncs3)C2)=O)ccc2ncsc2c1 c1(CNC2C(C(=O)NC(C)C(N)=O)C2)c(F)ccc(F)c1O C=CCCC(C(=O)NCCc1scnc1C)NC(c1ccc(OC)o1)=O n1(CC)nc(C(N2CC(F)CC2CNC(c2cnsc2C)=O)=O)c(Br)n1 c1(OCC)cc(N)c(Cl)cc1C(=O)NCC=CCNC(C1(F)CCOCC1)=O C(c1cncc(OC)c1)=CC(=O)NC(CCOCC)CO N(C(=NCCC(C)=O)NCCC12CCC(CC1)CC2)C1C(OC)CCC1 C1(C(=O)NC(C(C)C)CCN(C)C(C2(Cl)CC2)=O)CCc2ncncc2C1 c1(C(=O)NC(CC)CNC(C2CCN(CC3CCC3)C2)=O)ccc(C)c(C)n1 CC(CCC(=O)NCCC12CCCC1C2)NC(=O)C=Cc1cccnc1 Cc1ccc(C2C(C(=O)O)C2)c(C)c1.C1(=O)CN1C C1(SCCCF)CCN(C(c2cc(C)c(Br)s2)C(=O)N(C)C)C2(CC2)C1 C12(NC(C3CC3(F)F)=O)CCC(C(N3CC4C(C3)C4(F)F)=O)(CC1)C2 CC1COCCC1C(=O)NCC1(C(C)(C)O)CN(C(c2cnn(C3CC3)c2Cl)=O)C1 C1(OC)CCC(C(=O)NCC2CN(C(C3(C)CC4(CC4)C3)=O)C2)CC1 Cc1cc(C#N)cnc1C(=O)NC1CS(=O)(=O)CC1NC(c1ccc(Cl)o1)=O Cc1nc(=NC(=O)CCOc2cccc(Cl)c2)o[nH]1.C1C(=O)N1C(C)C C(=O)(C(C)(C)CN(C)C(=O)CC)N.C1(C)(OC)CNC(=O)C12CC2.C(C)(C)(C)O C(C)(C)(CC(F)(F)F)NC(CC)CC(=O)N(C(C)C(=O)NC1CC1)CC C=CC1CN(C(=O)CCOCCNC(c2cccn2CC)=O)CC1O CCC(C)C(C)C(=O)NCC(C1CCN(C(=O)C=CI)CC1)O CC(CC(N)=O)C(=O)NC(C)(C)CNC(c1cnccc1-c1cc[nH]n1)=O CC1CCN(C(c2cscc2C#N)=O)CC1CNC(c1cncnc1)=O Cn1nc2c(c1C(=O)NC1CC(C)(NC(c3cnn(C(C)(C)C)c3)=O)C1)CCC2 CC1(C)CCC(C(N2CCN(CC3(NC(C4CCC(=O)O4)=O)CC3)CC2)=O)CO1 C=CCC(F)(F)C(=O)NC1CC2CN(C(=O)CCCOCC=C)CC12 N1(C(C(C)NC(=O)NC)=O)CCC(CNC(c2n[nH]cc2[N+](=O)[O-])=O)(OC)CC1 c1(Cc2nc(C)nn2-c2cnnn2C)cn(CCO)c(=O)nc1O c1(OCC)ccc(C)c(C(N2CC(N3CCC(F)(F)CC3)C(O)C2)=O)c1 N1(C(C(C)=CC2CC2)=O)CC(CNC(=O)C#CC2CC2)C2(CCC2)C1 C(=O)(C(C(C)(C)C)OC(C)(C)C)NC1CCC(c2cn(C(CC=C)(C)C)nn2)C1 CN1N=C(CC(=O)NCC23CC2CN(C(C2(C(F)F)CCC2)=O)C3)CC1=O c1(C(N2C3CC(CNC(C4(NC(C)=O)CCC4)=O)C2CC3)=O)cc2occc2n1C C12(C)CN(CCO1)C(=O)CCc1ccc(cc1)C(=O)NC2.C1(CSC)(CO)CC1 C12(NC(=O)Cc3nncs3)CCCC1N(C(c1ncc(C(C)(C)C)o1)=O)CCC2 Cc1cnc(N2CCCC2CNC(c2c(C(F)(F)F)cccc2F)=O)nc1C C(=O)(C(C1CCCC1)NC(C)=O)NCCN(C(=O)CC1(C(F)(F)F)CC1)CCC N1(C)CCN(C(C2CCC2)C)CC1.c1(N)nn[nH]c1C1CC1 C(=O)(C1=CC2C=CC(C1)C2)NCCN(C(c1ccc(C)c(O)c1)=O)C CC(C(=O)NCC1CN(C(=O)CCc2ccco2)CCO1)C(F)F C12(c3cn(CCCC(=O)OC)nn3)CCC(C(=O)O)(CC1)C2 n1(CC)ccc(CC(N2CC(C)C2C(=O)NCC(CSC)OC)=O)n1 C(=O)(CC1OCc2ccccc21)N(C(CCNC(c1cn(C(C)C)nc1)=O)C)C C1(CCC(=O)NCCN(C2CCCCC2)C(C(C)SCC)=O)CCCCN1C N1(C(CCc2ccc(C)o2)=O)CCCC(NC(c2ccsn2)=O)C1 C12(CNC(C(C)N(C(C)=O)C)=O)CN(C(C3CC(N(C)C)C3)=O)CC1CCO2 C1(C(N)=O)C=CCN1C(=O)CNCc1c(C(=O)NC(C2CCCO2)=O)cco1 C1(C(N2CC(C)C(CCNC(=O)Cn3cnnn3)C2)=O)CC(C)(C)OC1(C)C c1(C(=O)NCC(=C2CN(C(C3C(OCC)C3)=O)C2)F)ccnn1C1CCC1 C=CC(C)CC(=O)N1CC2CC2C1C(=O)NC1CCN(CCCO)C1 N1(C(C2(CCC=C)CCN(C(=O)C=CCO)CC2)=O)CCn2ncnc2C1 N1(C(C2C(CN)CC2)=O)CC(O)C(C#N)C1 c1(C(=O)NC23C(CN(C(CCC=C)=O)C2)CC3)coc(=O)c2ccccc12 C12(C(=O)NC(CC=C)CNC(=O)CC3(C(F)(F)F)CC3)CCCN(CCC1)C2 C#Cc1cnc(C(N2CCC(CC(=O)NOC3CCCCC3)CC2)=O)c(C)c1 C1(N(C)C(c2ccc(F)cc2)=O)CN(C(C2CN3CCN2CC3)=O)CC1(C)C.CCS C1(C(=O)NCC(CC)(C)O)(CC)CCCN1C(c1cnsc1)=O c1(N(C)CC2CCN(C(c3ncn(CC)n3)=O)C2)ncnc2c1SCCC2 c1(C(N2CC(F)(CNC(c3csc(Br)n3)=O)C2)=O)cnc2c(c1)CNC2=O c1(C(N2CCN(C(CCC3(C)CC3)=O)C(C(C)(C)C)C2)=O)cnc2ccnn2c1 C#CC1CN(C(=O)CSc2cn[nH]c2)CCN1C(C1CC(C2CC2)=NO1)=O c1(C(C)(C)C)nccc(C(=O)NC2(CNC(=O)Cc3cnoc3)CCCC2)n1 CCC(CC(=O)N1CC(CC(=O)NCc2ccn(CC)n2)C(C)C1)C(C)C S(=O)(=O)(c1cccnc1)N1CC(CC(N2CCCC(N3CCCC3=O)C2)=O)C1 c1(C(=O)OC)cc2n(n1)CCN(CC1CCNC1C(C)C)C2 C1(OC)CN(C(c2cccc(SC)c2)=O)CC1NC(c1nsnc1O)=O c1(C(=O)NC2(CNC(C(C)N(CC)CC)=O)CCC2)cccc2ccnn12 CC1=NN(C)C(=O)C1CC(=O)NC1CCN(C(=O)CC2CC(C(C)C)C2)C12CC2 C#CCC(C(=O)NCC1=NOC(C)C1)NC(=O)CC1CCOC1(C)C C1(CC=C)CC(O)CC(CC(=O)NC2CCN(C(c3ccc(CC)[nH]3)=O)C2)O1 N1(C(COCCNC(C(C)N(C)C)=O)=O)CC2CCC(C1)C(=O)O2 c1(C(=O)Nc2n[nH]c3c2CN(C(=O)C#CC2CC2)C3)cc(O)nc2ccccc12 c1(C(=O)NC2C(N(C(COCCCC)=O)CC)CCCC2)c(OC)ccnc1F C1(C(=O)NCCCN(CCCCNC(C2CCC(C)O2)=O)C)CC(=O)N(C)C1 N1(CCNC(CCCOC)=O)CCN(C(C)C)CC1.C1(=O)CCCN1 C1(C)(C(N(CC(=O)NC2CC(CC(C)(C)C)C2)CCOC)=O)CSC1 c1(N2CCC(NC(CC)=O)C2)nc2c(c(=NCc3csc(=N)[nH]3)[nH]1)CSC2 CC(CC(=O)NC1(C(=O)NCCc2cccnc2O)CCN(C)C1)C(F)F C1(NC(C2CCC(C)O2)=O)C2CC3C(C2)C13C(=O)NC1CC(O)C(F)C1 c1(N(CC(C2CCC2)OCC)CCNC=O)ccnc(CC)n1.c1(O)ccccc1 c1(C(N2CC(CC(C)NC(C(CCCOC)C)=O)C2)=O)nccc(Br)c1O c1(CC(=O)NCC(C2CCC2)NC(C(C2CCC2)OCC)=O)ccn(C)n1 C12(C(=O)NC(CC)(C)C)CC1CN(CC(Cl)=CCl)C2 Cc1cc(=O)n(C)nc1C(N1CCN(C(=O)CCc2nccn2C)C(CO)C1)=O N1(C(c2c(-c3ccc(C(=O)OC(C)(C)C)nc3)ncs2)=O)CC2COCC2C1 c1(C(N2CCC(OC(C(C)C)=O)C2)=O)c(C(n2cc(Cl)cn2)C2CC2)cccc1F S(=O)(=O)(c1ccc(=NCC(C)N(c2ccc([N+](=O)[O-])cn2)C)[nH]c1)N(C)CC C(=O)(C(C)(C)C1=CCSCC1)N1CC(CC(C)NC(=O)C(F)C(C)(C)O)C1 N1(C(C2(CCC)COC2)=O)CCC(C)C(NC(=O)C=Cc2ccc(CC)s2)C1 CCC(C)CCC(=O)NCC(C)(CO)NC(=O)CCc1cc(Cl)no1 C=CCCC(C)C(C(=O)NCCCC)N(C)Cc1nc(C)cs1 N1(C(COCCC=C)=O)CCC(F)(F)C(C(=O)NCCN(S(C)(=O)=O)CCC)C1 N1(C(c2nc(C(C)C)oc2)=O)CCCC(NC(=O)CCc2cccn2C)C1 c1(C(N2C(C(=O)NC(C=C)(C)C)C=CC2)=O)cc2ncccc2[nH]1 CC1Oc2ccc(-c3nc(-c4ccc(Cl)cc4)nn3-c3cccc(Br)c3)cc2C1C c1(C(N(CC(CC)NC(=O)C(=O)C(C)(C)C)CC)=O)cccc(C#N)c1F C#CC1(C(=O)NC2CCC(=O)N(CC)C2)CCN(C(=O)CCCn2ccnn2)C1 c1(C(N2CCN(C(C(COC)OC)=O)CC2C2CCC2)=O)cnc2cccc(C)n12 Cc1ccc([N+](=O)[O-])cc1C(N1CC2CC1CC2NC(c1ccco1)=O)=O Cn1nc(C(=O)NCC(O)CCNC(c2cc[nH]c2)=O)c(Cl)c1C(F)(F)F C(C(C)N=c1cc(C)[nH]c(=NCCCC(=O)OC(C)C)[nH]1)c1ccc(OC)cc1 C1(CNC(c2cc(C)n(C(C)C)n2)=O)CCN(C(C2CCCCC2O)=O)C1(C)C C(=O)(C1CC(=O)Nc2ncccc21)NC1(CNC(C(COC)(C)C)=O)CCOC1 C(=O)(C(C)C(C)S(C)(=O)=O)N(CC=CCNC(C1(CCC)CC1)=O)CC c1(C(=O)OC)cc(=NC(=O)C2CCN(Cc3cc(Br)c(F)cc3O)C2C)[nH][nH]1 c1(C(=O)NC(CCOC)CNC(C2CC(OC)C(OC)C2)=O)cc(F)c(N)cc1F C(=O)(C1=CC2CCCCC12)NCC1(F)CCCN(C(CSCC)=O)C1 Cc1cccc2c1c(CN1CC(F)(F)CC1C(=O)NCCCO)cn2C C1(C)(C(=O)NC(c2c(C)ncs2)C)CCCN(C(c2ccc(C(N)=O)[nH]2)=O)C1 N1(C(c2ccc(CNC(c3ccc(C(C)C)o3)=O)s2)=O)CCCC(F)(F)CC1 C#CCCN=C(NCCc1ccccc1OC)N1CCN2C(=O)CCC2C1 CC1CCN(c2nnc(CO)s2)CC1NC(c1cccc(Cl)c1Cl)=O C1(C(=O)NC2(C(=O)NCCC(C=C)C)CC2(C)C)COCCN1C C(c1cccc(F)c1F)=CC(=O)NC1CCC(NC(c2c(C)scn2)=O)CC1 c1(C(=O)OC)ccc(CCC(=O)NC(CNC(c2cn(C)nn2)=O)C2CC2)cc1 CC1=C(C(=O)NCC2=CCN(C(c3ncc(C(F)(F)F)cc3N)=O)CC2)CCO1 C(=O)(C1=CCCOC1)NCC(C1CCCN(C(CCN(CC)CC)=O)C1)(C)O CC1CC(NC(=O)CCF)CCN1C(c1cnn(Cc2ccccc2)c1)=O C(=O)(CCCN(C)N=O)NCC(CC(=O)NCC(=O)NC(COC)C)C N1(C(C(CC)(C)CNC(c2c[nH]c(C(N)=O)c2)=O)=O)CCCOC(C)(C)C1 C1(NC(Cc2cccc(C)c2)=O)CCN(C2CC2CC(C)(C)C)CC1C(N)=O CC(C)CCCCC(=O)N1CCCC(O)(CCNC(C2CC3(C2)CC(C)C3)=O)C1 c1(OC)cc(C(N2CCOC(CNC(=O)C(C)(C)CSC)C2)=O)ccc1O C(=O)(C(C)(C)CN(C(=O)CC(=O)N(C)C)C)NCc1n(C(C)C)ccn1 N1(C(CC2(C=C)CCC2)=O)CC(NC(c2nnc(C)s2)=O)C2CCCC12 Cc1nc(C(N2CCC(C)C2CNC(=O)CS(N)(=O)=O)=O)n(C)n1 C(=O)(C(C)(CO)NC(c1scnc1Cl)=O)N(C)CC1(C#N)CC1 N1(C(C#CC(C)(C)C)=O)CCCC2CN(C(=O)C(C)(C)CC#N)CCC12 c1(C(=O)OC)ccc(F)c(C(N2CCCC(CO)(NC(=O)C(C)C3CC3)C2)=O)c1 C(=O)(C(C)(C)C(=O)OC)OC(CC(=O)N1CC(CC(=O)OCC)C1)(C)C C=CCCC(C)(C)C(=O)NCCCC1CCCCN1C(c1[nH]c(C)nc1C)=O N1(C(C2CCC(=O)O2)=O)CCOC(C(=O)NCCCc2cn[nH]c2)CC1 CCC(CCC(F)(F)F)(N=c1ccc(Br)c(S(=O)(=O)N2CCCSCC2C)[nH]1)N(C)C CC(CCCNC(=O)C(C)OCc1ccccc1)NC(c1csc(C2CC2)n1)=O C1(C(=O)NC(C=C)(C)C)CN(C(C2CC2O)=O)CC1F.C(C)(C)(C)OC(C)=O c1(CN(C2CC2)CC)c[nH]c2c(Cl)cc(F)cc12 S(=O)(=O)(c1cnn2ccc(=NCCC(F)F)[nH]c12)N1CCC(C=C)C1 c1(CC)ccc2c(c1)CN(C(=O)C1=CCOC1)CC2 N1(C(C2N(CC)CC2)=O)CCC(C)(CC(=O)NCC(C2CC2)OC)C1 c1(CC(C2CCN(C(c3c(OC)ccc(F)c3)=O)CC2)=O)c[nH]c2ncc(F)cc12 Cc1ccc(C(N2CCN(C(=O)COC3CC3)C3CCCC23)=O)c2c1CCCN2 c1(C(=O)N(c2ncc3[nH]ccc3n2)C2C3CNCC23)cc([N+](=O)[O-])ccc1F N1(C(CCCCSC)=O)CCC2CCN(C(c3scnc3C)=O)CC2C1 C1(CO)CCN(c2ccccc2)CCC1C.N12CCN(CC1)C(=O)CC2 C#Cc1ccccc1CNC(=O)CNC1CCC(C=CC(=O)NC)C1(C)C CC(C)(CNC(c1ccc(C(F)F)o1)=O)CCNC(=O)C=CC1CC1 c1(CN2CC3C(NC(C4CC(=C)C4)=O)C3C2)cc2cccc(Br)c2[nH]1 C(C(F)F)(C(C)(C)C)N(C(=O)C=CCn1cc(-c2ncccc2F)nn1)C C1(CNC(c2cc3ccccn3c2)=O)CCCC2CN(C(c3cncs3)=O)CC12 C1(F)(CNC(C2C(CC)CCO2)=O)CCN(C(=O)C(N2CCC(O)CC2)C)CC1 N1(C(C(C)(C)SC)=O)CCN(CC2CN(C(c3nsnc3O)=O)C2)CC1 N1(C(C2CN3CCC2CC3)=O)CCC2(CC1)CCN(C(C1(C3CC3)CC1)=O)CC2 N1(C(CCCCCCC)=O)CCOC2(C1)CN(C(=O)C(C)Cc1ccncc1)C2 C(C(C(=O)NCCN1C(=O)CNC1=O)C(C)(C)C)NC(c1n(C=C)ncc1)=O c1(NC(=O)OC)cc(C)nnc1N1CCC(N(C(=O)C(C)NC(C)=O)C)C1 c1(OC)c(C)cc(C(=O)NC(CNC(C2CCCC3(CCC3)O2)=O)CO)cc1C O=C(CCCn1ccnn1)NC1CC(NC(c2csc(C(C3CCCC3)=O)n2)=O)C1 CC(Cn1cnnc1)N=c1nc(N2CCCN(C)C(=O)C2)c2c([nH]1)CCCCC2 CC(C)(C)C(C(=O)NC1CCCC(O)C1O)NC(c1nc[nH]n1)=O Cc1ccc(CC(N2CCC(N(C)C(c3n[nH]cc3Cl)=O)C2)=O)cc1C CS(=O)(=NC(=O)c1ccc(NC(N)=O)o1)C1CC(CN2CCOCC2)C1 Cc1cc(C(N2CC3CCC2CN3C(C2(C#N)CC(C)C2)=O)=O)c(C)nc1C N1(C(c2c(NC)cccc2)=O)C2CCC(C2)C1C(N1CC(n2cnnc2)C1)=O Cc1cc(C(=O)NC2(CNC(c3[nH]c(O)nc3C)=O)CCC2)ccc1Cl Cc1ccc(C(=O)NC(C2CCCN2C(C2CC3C=CC2C3)=O)C)c(C(C)C)n1 C=CCC(CC(=O)NCC1(C=C)CCCC1)NC(=O)C(c1ccn(C)c1)C c1(CCNC(C2COCCOC2)=O)cccc(F)c1Br c1(N(C(C2CCC2)C)C)nnc(C2CCCC2)n1CCOCC.C1(CO)CCC1 CC(C)CC(C)C(=O)NC(C)(CNC(c1c[nH]cc(Br)c1=O)=O)C1CCC1 C1(NC(CNC(CC(C)(C)C)=O)=O)CCCC12CCN(C(=O)Cc1cccs1)C2 C=CC(CC)C(=O)N1CCC(C(=O)N(CC(O)C2CC2)C)(CC)C1 c1(C(N2C(C)(C(N(C)CC3CC(=C)C3)=O)C=CC2)=O)ccc2cc[nH]c2n1 c1(-c2cccc(COCC(C)NC(C)=O)c2)ccc2c(c1)NC(=O)C2 N1(C(C2(C#C)CN(C(c3ccc(N)cc3)=O)C2)=O)CCOC(C)C1CC N1(C(c2cc(C)oc2)=O)CCC2CN(C(=O)Cc3c(O)ncnc3O)CCC2C1 C(=O)(C1=COCCO1)NC(c1ccccc1C(F)(F)F)C(=O)OC CC(C)C(CCNC(C1(C)CCOCC1)=O)NC(=O)C(C)NC(C)(C)C c1(C(C)C)nocc1C(=O)N(C)CCNC(C1CC2CC2C1)=O C(=O)(C1=Cc2ccccc2C1O)NC1CC(NC(C2CC(=C)C2)=O)CC1O n1(CCNC(=O)NC2CCC2c2ccccc2)cnccc1=O c1(N2CCCCC(C(N)=O)C2)ncccc1S(=O)(=O)N1CCC(n2cncn2)C1 N1(C(CCC#C)=O)CC2CCC1C(NC(c1cc(N(CC)CC)ccc1O)=O)C2 C1(NC(c2cnc(C(C)(C)C)s2)=O)CCCC(NC(=O)C(C)(C)NC(C)=O)C1.[SH](C)(=O)=O N1(C(=O)CCn2ccccc2=O)CCN(C(c2cnn3cc[nH]c23)=O)CC(O)C1 C1(C2OCCO2)COC(CSC)C1.N12CC(C1)CC2=O.C(CNC=O)O.CCOC c1(SCC(CC)NC(=O)C(=O)Nc2c(OC)noc2C)ccc(F)cc1 CC1=CC(C)=NS(=O)(=O)N1CC(=O)N(C1CC(NC(c2c(C)ncn2C)=O)C1)C C1(NC(c2c(C)coc2C)=O)CN(C(=O)C(C)n2cncn2)C2(CCCC2)C1 C1(CCC)CN(C(c2ccncc2)=O)CC1C(=O)N(C)CCn1ccnc1 N1(C(C(C)C#N)=O)CC(C(=O)NCc2ccc(F)cn2)CCC1(C)C C1(NC(C2C(=C)CC2)=O)C2CN(C(C3C4(CC4)C34CC4)=O)CC12 C=CC(O)C(=O)NC1CCCC1C(=O)NCC1(O)CCCC1 C(C(C)(C)C(C)(F)F)NC(C1N(C(=O)C(C)CCSC)CCC(CC)C1)=O CCCC(C)CC(=O)NCCCCN(CCCNC(=O)Cc1cccn1C)C O=C(N=c1ccn(CCO)[nH]1)c1cc(CCNC(c2cc(Cl)c[nH]2)=O)on1 C1(C(N2C(CCCNC(C(C)S(C)(=O)=O)=O)CCCC2)=O)CC2(C1)CC(F)(F)C2 Cc1nn(CC(=O)N(C2CCCC(NC(c3ccc(=O)oc3)=O)C2)C)c(C)c1Cl C1(CNC(c2n[nH]c3c2CCC3)=O)CN(C(C2CCCCO2)=O)C2COCC2O1 N1(C(C2(OC)CCCOC2)=O)Cc2[nH]nc(C(=O)N(C)CCF)c2C1 N1(C(c2cc(OCC)ncc2)=O)CCC2CCN(C(=O)Cc3ccsn3)C2C1 C1(NC(C2CN(C(c3c(CC)nn(C)c3)=O)C2(C)C)=O)C(O)C2CCOC12 c1(C(N2CCC=CC2C(=O)OC)C(=O)NCC=C)ncccc1Cl N1(C(C(C)SC(C)C)=O)Cc2[nH]nc(C(N3CCC(C)C3C(N)=O)=O)c2C1 N1(C(CCC(C)OC)=O)CCN(C(c2cccnc2)=O)CC1CCN(C)C C1(OC)CN(C)CC1N=c1[nH]c(=NCCCc2cccnc2)[nH]c2c1COC2 C1(CC(=O)NC(C(C)O)(C)C)C=CCN(C(C2CC(=C3CC3)C2)=O)C1 C1(C(=O)NC(CC=C)(C)C)CCCN(C(C2(N(C)C)CCCC2)=O)C1 C1(C(=O)Nc2cnccc2C)(NC(CCSCC)=O)CC1(C)C C12(NC(C3C(C)(CC)C3)=O)CC(CO)(C1)OC21CN(C(=O)C(=O)NCC(F)F)C1 c1(C(=O)NC2COCCN(C(CC(CC)(F)F)=O)C2)ccc([N+](=O)[O-])n1C C1(CC(=O)NC(C(=O)N2CC(c3ccccc3)C2)c2ccoc2)NC(=O)NC1=O CC1CCN(C(c2c(Br)ncn2C)C(=O)Nc2ccccc2)CCS1(=O)=O C(CC(C)C(=O)N1CCC(C(=O)N(CCC(N)=O)C)C1C)OC c1(C(N(C)CC2N(C(C(=O)NC(C)C)=O)CCCC2)=O)nc[nH]c2ncnc1-2 Cc1ccc(C(=O)NC2CC(C(=O)NC3CCCC(F)C3)C2)nc1 C(=O)(C(CCC(N)=O)N(C)C)NCC1N(C(Cn2c(C)csc2=O)=O)CCN(C)C1 c1(NCC2CCN(C(c3ccc(C)cn3)=O)C2(C)C)c([N+](=O)[O-])cnn1C N1(C(c2ccc(C=C)cc2)=O)CCC(NC(=O)C(N2CCCCC2)C)C(C)(C)C1 C1(C(=O)OCC)(NCc2ccon2)CC(C)(c2nnnn2C(C)C(=O)OC)C1 C1(NC(c2c(CC)ocn2)=O)CCN(CCNC(=O)C(C)(C)C)CC1C N1(C(c2cncc(OC)n2)=O)CCOCC(NC(C2(SC)CCCC2)=O)C1 C1(CNC(C2(COC)CCC2)=O)CCC(CN(C)C(C2SCC=C2C)=O)CC1 N12CC=CC1C(=O)NC=CC=CC2=O.C1(C(C)(C)C)(CO)CCCO1 C1(C(N2CCC(NC(C(C)NC(C)=O)=O)C2)=O)C2CC1(c1ccccc1)CO2 C(=O)(CC1OCCc2sccc21)NCCCN(C(CCC(=C)C)=O)C c1(OCC)c(CC(=O)NC2CC(N(C)C(C3CCCC(C)O3)=O)C2)cccc1Cl C(=O)(CCCC(=O)N1CC(NC(=O)Cn2ccnc2C(C)C)CC1C)NCC c1(SC)cscc1CNC(c1nnnn1C(C)(C)C)(C1CCOCC1)C C1(CNC(c2ccccc2)=O)C2CCCC1N(C(c1cc(Cl)n[nH]1)=O)C2 c1(OC)ccnc(NC2C3CN(C(c4nnn(C)c4C)=O)CC23)n1 c1(C(N2C3C(NC(c4c(C)scc4)=O)CC(CC3)C2)=O)ccc2c(c1)C(=O)NC2 Cc1sc(Cl)c(C(=O)NC2CCC2NC(C2(n3nccn3)CC2)=O)c1C Cc1cc(O)c(F)cc1NC(C1CN(C(c2[nH]ccc(=O)c2C)=O)C2(CCC2)C1)=O c1(C(=O)NCC2CC(F)CN2C(c2cc(F)n[nH]2)=O)cnc2c(c1)CNC2=O c1(N2CCC(NC(CNC(CC(C)C3CC3)=O)=O)C2)nccc(CO)n1 C1(NC(c2c(C)onc2-c2cccnc2)=O)CCC(C)N(C(C23CC(C2)C3)=O)C1 CCC(C)(C)C(C)CC(=O)NCC1C=CCN1C(=O)CSc1ccc(OC)cc1 c1(-n2c(-c3cnc4sccn34)nc(C(C)SCC)n2)ccc(F)c2ccsc12 CC1CC(NC(=O)CC(C)(C2CCC2)N(C)C)CN(C(C2CC(C)(O)C2)=O)C1 N1(C(C2N(C)CC2)=O)CC=C(C(=O)NC23CCCC2OCC3)C1 Cc1ccc(C=CC(N2CCC(NC(=O)C3=CCCOC3)C2C(C)C)=O)cc1C N1(C(C2C(C)COCC2)=O)CCS(=O)(=O)N2CCOCC12 CC1=C(C(=O)NCC2(C)CCN(C(=O)CCc3ccccc3)C2)C(=O)OC1(C)C CCC(O)C(C)C(=O)NCC1(NC(c2cc(C3CCC3)no2)=O)CCCCC1C c1(OC(C(=O)NCCN(C(C(C)OCc2nncn2C)=O)C)C)ccc(C)cc1 c1(N2CCN(C(C(C)Oc3ccccc3)=O)CC(O)C2)nc2ccc(F)cc2s1 C#Cc1ccc(C(N2CC(CNC(=O)CC3CCC(=O)NC3=O)C(C)C2)=O)cc1 c1(C(N(CCCN(C)C)CCNC(C(CC)OC)=O)=O)ccc(C(N)=O)cc1 CC#CCC(CO)NC(=O)CN(C(=O)C(C)CC1CC1)C1CCC1 Cc1c(N)ccc(C(N2CCOC(CNC(=O)CCC3(C)CC3)C2)=O)c1Cl c1(C(N(C(C)CN(C)C(C2(O)CC2(C)C)=O)C)=O)cnn2cccnc12 C(N=C(NC1CC1)N1CC(C)CC(C)C1)c1cc2ccc(CC)cc2cc1 CC1(C)CC(n2ccnc2-c2cccc(C(F)(F)F)n2)C(=O)N1 C1(OC)CCN(C(c2nonc2N)=O)C(C)C1.C12CC(C1)CC(=O)N2 c1(CC(=O)NCCN(C(=O)CNC(=O)CC(C)(C)C)CC)ccc(O)nc1 c1(CC)ccc(O)c(C(=O)Nc2cccc(C)c2Oc2cc(C(N)=O)n(C)c2)c1 Cc1cc(N)cc(C(N2CCCC(NC(C3CN(C)C(=O)N3)=O)C2)=O)c1F c1(C(C)OC)nc(-c2ccc(C(F)(F)F)nc2)n(CC(C)C)n1.C1(C)CC1 c1(N2CCC(n3ccnc3)C2)nccc(=NCc2nnnn2C)[nH]1.C12CC(C1)NC2 C1(NC(C(CC)CCOC)=O)CC2CCC(C1)N2C(=O)Cc1ccccc1O c1(OC)cc(Cl)ccc1C(=O)NCCCN(C(=O)C(F)(F)CC1CC1)C1CC1 CC1=C(C)CC(C)(NC(=O)C(Cc2ccco2)NC(c2ccc(F)s2)=O)CC1 c1(OC)cc(NC(=O)NCCc2ccc(Cl)c(OC)c2)ccc1C O=C1NC(=O)C(c2cn(C(Cc3ccccc3)C(=O)N3CC4CC4C3)nn2)N1 C1(C)(NC(C(CCC)NC(=O)COCCCN(C)C)=O)CCCC(C)(C)C1 CCS(=O)(=O)C=CC(=O)N1CCC(NC(C2CCOCC2(C)C)=O)C(OC)C1 CCC(CC)CN=c1[nH]c(=NCC2(C)CC3CC3C2)c2cccc(F)c2[nH]1 CCC(CCC(=O)NC1(C)CCOC1)NC(=O)CCOCC(C)C C1(CC=C)(NC(=O)C=CC(C)=O)CCCN(c2ncc(OCC)cn2)C1 c1(CNC(=O)NC2CC3(C2)CC32CCC2)cccc2ccccc12 C1(CCC)(NC(c2ccc(COC)cc2)=O)CCCN(C(=O)CC2=CCCC2)C1 C1(CC)CN(C(C23CCC(C2)C3)=O)CCC1NC(=O)Cc1cnsc1 C(=O)(CC(C)C(C)C)NCC(C(=O)N(CC(C)C#N)CC)CC1CCCC1 C1(C(=O)NC2C(OC)CN(C(=O)C(C)(C)CN(C)C)C2)CC2CCC1C21CC1 Cc1ccc2c(c1C)CCCN2CC(=O)NC1(CC(F)F)CCC1 c1(C(CC(=O)NC2C(NC(CC(CC)C)=O)CC2)C)ccc(F)c(F)c1 Cc1ncc(C(=O)NCC2CC3CCC2N3C(=O)CCC2CC2(F)F)c(C)n1 c1(C(=O)NCCC(C(C)C)NC(=O)CC(O)C2CCCC2)nccc2occc12 c1(C(N(C2CCCN(C(=O)CCC(C)SC)CC2)CC)=O)cn2cc(C)sc2n1 C(=O)(C1=CCCCC1C)NC1CC2CC(NC(c3c[nH]cc(C)c3=O)=O)CC21 C1(C(=O)NCCS(CC)=O)CCCCN1C(=O)Cc1cncnc1 c1(C(=O)NC2CC(NC(C3CCOC3)=O)C23CCC3)ccc2[nH]ccc2c1 C1(C(NOCC=CC)=O)CCCC(NC(=O)C(C)NC2CC2)C1 c1(CC)ccc(C(=O)NCCCCCCN(C)C(C2(C#N)CCCO2)=O)cc1Cl C(=O)(CC(C)(C)C(F)F)N(C1CCCN(C(C2COC(=O)O2)=O)CC1)CC C(=O)(C1=C(C)OCC1)N(C)CC1N(C(c2ccc(CC)nc2)=O)CCCC1 CCCCC(C(=O)C(C(=O)NC)=NOC(C)CNCCCOCCCN)N(C)C C#CCC(C)(CC)C(=O)N1CCC(CNC(c2cccc(F)c2C)=O)C(F)(F)C1 c1(C(=O)NCC(CC)NC(=O)C(C)(C)C(N)=O)oc2c(Cl)cccc2c1C C1(C)(C)CCC(=O)NC(N(CCC)C)CCCCC1 C1(NC(c2ccc(Cl)cc2)=O)CC2CC(NC(C3(CO)CCCO3)=O)C2C1 Cc1ccc(C)c(C(=O)NCC2CC2NC(c2cnc(O)c(F)c2)=O)c1O C(CO)(C(C)(C)C)NC(c1nnnn1CCC1(C)CC1)(COC(C)C)C C1(NC(c2c(C)nc(O)[nH]2)=O)CN(C(C2CC2C)=O)C2(CCCC2)C1 Cc1cc(C(=O)NCC2(O)CCCN(C(=O)CN3CCC3C)C2)nnc1O N1(C(C(CC=C)OC)=O)CCn2ncc(CN(C(=O)CCS(N)(=O)=O)C)c2C1 C1(CC(N2CCCCC2C2CCN(C(C3CCSC3)=O)C2)=O)(COC)CCOCC1 N1(C(C(CCSC)OC)=O)CC2CCN(C(c3sc(F)cc3Cl)=O)CC2C1 O=C(CC1=CCOCC1)NC1CCCCC1NC(=O)C(F)(F)CC1CCCO1 S(=O)(=O)(c1cccs1)NC(C(CCSC)N(C)C1CC1)=O C(CC(C(=O)N1CCCNCC1)NC(=O)CN)OC C1(F)(C(N2CC(C(=O)OCC)C2)=O)CCCN(C(=O)CC2CCC(=O)C2)C1 N1(CC=C)CCN(C(C)CC(=O)Nc2cccc(-c3nnco3)c2)C(C)C1=O C1(NC(CC(c2c(C)n[nH]c2C)C)=O)COCCN(C(=O)C=Cc2ccccc2)C1 CC1OC2(CO)CC1(C(=O)N(C)CCNC(C1CCCN(CC(F)(F)F)C1)=O)C2 N1(C(C(C)O)=O)CCOCC1CCNC(=O)CSc1ccccn1 c1(C(=O)NCCN(CCC)C(C2CC2C#N)=O)nnn(CC)c1C(F)(F)F c1(C(=O)NC(CC)(CC)C(N)=O)n[nH]c2c1CN(C(c1cncc(NC)c1)=O)C2 Cc1c(Cl)cnn1CC(=O)N(CCCNC(=O)Cc1cnc[nH]1)C C1(C2CCN(C(C3CC3F)=O)CC2)(NC(c2ncccc2Br)=O)CCC1 C1(C(N(C2CCC2)CCN(C)C)=O)CC(NC(=O)CCOC2COC2)C1 CC(C)(O)C(F)C(=O)N(C1CCN(C(=O)CC2CC3(CCC3)CO2)CC1)CCO C(=O)(CCCN=[N+]=[N-])NCCCC(=O)NC(C)CC1(O)CCC1 N1(C(C(C(C)(C)C)=O)=O)CCC2(CC1)CCN(C(C1CCC(C(=O)N(C)C)C1)=O)C2 c1(CC)cnsc1C(=O)NC1COCC1n1cc(C(=O)OC)nn1 c1(C(=O)NC23CC(CNC(C=C4CCC(C)C4)=O)(C2)OC3C)cnc2cccnn12 CN1CCN(C)CC(C(N2CCN(C(c3ccc(F)cc3)=O)C(C(F)F)C2)=O)C1 C1(C(C)NC(=O)CCOCc2ccccc2)CN(C(c2cc(O)no2)=O)CCO1 CCC(C(=O)NCC1CCN1C(c1cc(C(C)=O)no1)=O)Oc1ccccc1 c1(C(=O)NCC2(CCN(C(C)C(=O)O)CC)CC2)c[nH]nc1-c1ccoc1 Cc1ccn2c(=O)c(NC(=O)NCC3(CO)CC(C)(C)C3)cnc2c1 CCS(=O)CC(=O)N(CC(O)CN(C)C(c1cc(Cl)ns1)=O)C N1(C(C2(COC)CC2)=O)C2CCC(C2)C1C(=O)Nc1ccc(O)c(Cl)c1 N1(C(C2CNC(=O)N2)=O)CCC(NC(c2ccncc2C(F)F)=O)C(F)C1 CCCCC(c1nnnn1Cc1cccs1)NC(C1CCCO1)Cn1cc(C)cn1 C1(CCC)(C(=O)NCCCNC(C2CN(S(=O)(=O)CC)C2)=O)CCC1 C1(NC(CCCC#C)=O)CC2CCC(C1)N2CC1CCC(C)C1 CC1CCCCN1CCNC(=O)C(C)(C)c1sccc1Cl.C(C)(=O)O C1(CCC)(NC(=O)C(=O)CC)CCCN(C(=O)CCCCCOC)C1 N1(C(CCCCC=C)=O)CC(CNC(c2cnc(C)[nH]2)=O)CC12CCOCC2 N1(CCC(=O)N(CC(C)(C)NC(C(C2CCOC2)OC)=O)C)CCOCC1=O C1(C(=O)NCCCCC#CC)CN(C(=O)C(C)OCCCC)CCC1(C)C c1(C(N(CCCN(C)C(C2CCCC2C(N)=O)=O)C)=O)cc(F)cc2nc[nH]c12 C(=O)(C1CCc2cccnc21)N1CC2C(NC(C=Cc3c(C)cccn3)=O)C2C1 CC(C)(F)CN=c1[nH]c2c(c(=NCc3ccc(Cl)o3)[nH]1)CCCC2 CCC(CC(=O)N1CCN(CC(O)CO)CC1)NC(=O)CC1CCC1 c1(OC)ccc2c(=NCC=CBr)[nH]c(=NCc3ccc(=N)[nH]c3)[nH]c2c1 CC1(C)CC(CC(=O)NC23CC2CN(C(=O)CCCCc2cnn[nH]2)C3)C(=O)O1 C(=O)(C1=NN(CCO)C(=O)CC1)NCC1(C)N(C(CCC=C(C)C)=O)CCC1 n1(CC(=O)N(CCNC(=O)CCC2CCCC(O)C2)C2CC2)ncc2ccccc12 C(=O)(CCC(=O)N1CC(O)(C(C)NC(=O)C(c2ccc(C)cc2)(C)C)C1)NC C(=O)(C(C)(C)S(=O)(=O)C1CC1)NC(CCCC)CNC(c1onc(C)c1C)=O C1(CCNC(COCCCCC)=O)COCCN1C(=O)C(N1CCC(C)C1)=O c1(C(C)C)cc(C(=O)NCC(C)NC(c2ccncc2Cl)=O)cc(F)c1 C1(NC(C(C)(C)CF)=O)CC(F)CN(C(c2c[nH]ccc2=N)=O)C1 CS(=O)(=O)c1ccc(C(=O)Nc2ccc(-n3cccc3)c(Cl)n2)cc1 C(=O)(C(O)C(C)CC)N(CCCCCNC(CCCCC)=O)C(C)C C1(C(N(C)CC2CCC(=O)NC2)=O)CN(C(c2ccncc2Br)=O)CCC1O C=CCCCC(C)(c1nnnn1C(C)C(=O)OC)NC(C1CC1)C1CC1 Cc1cc(OC(C)C)ncc1S(=O)(=O)NC1(C(=O)NC(C)C)CCCOC1 c1(C(N2CCCC2N(CC(F)(F)F)C)C(=O)NCCCC)cc(Cl)cc(Br)c1F c1(C(=O)NC2C(NC(C(CCC)OC)=O)C2)cc(C(=O)OC)cc([N+](=O)[O-])c1 N1(CC(=O)NCC2(NC(c3c(C)[nH]cc3)=O)CCCC2)C(C)=CC(C)=NS1(=O)=O C1(NC(Cc2cn(CN(C)C(c3cnccn3)=O)nc2)=O)CCC(CO)CC1 CS(=O)C=CC(=O)N(C1CCCN(C(c2ccc(Cn3cc(Cl)cn3)o2)=O)C1)C N1(CCN(CC=C)CC)CC(=O)N(CC(C)F)C1=O N1(C(C(CC)(C)C)=O)CCC(NC(c2ccc(F)c(Br)c2)=O)C(C)C1 C(=O)(C(CC(C)C)C(C)C)N1CCC(O)(CN(C(C2(SC)CC2)=O)C)C1 c1(C(C)C)ccoc1C(=O)N(C)CCOCCC(=O)NC(c1cnsc1)C C1(NC(C(n2cc(C)nc2)(C)C)=O)COCCC1NC(=O)Cc1cnn(C)c1 C1(C(=O)NC23CC(CC)(C2)C3)CC2CCC(C1)N2C(=O)OC(C)(C)C CCCS(=O)(=O)C(C)C(=O)NC1CCN(CCNC(c2cc(C)oc2C)=O)CC1 N1(C(c2c(CC)cno2)=O)CCC(NC(=O)CN2CCOCC2)C(C)C1 c1(OC)ccc2oc(C(N3CCC(NC(=O)C=C4CC4)C(C)C3)=O)c(C)c2c1 C(C(=O)NC1CC(CNC(C2(C)CCN(C(C)=O)C2)=O)C1)(C(C)C)SC c1(NC(C2(O)CCN(C(CC(=C)C)=O)CC2)C)ncnc2sc(C)c(C)c12 c1(COC)c(C(=O)N(C(C)CCNC(C2CC3(CC3)CO2)=O)C)cnn1C Cc1cc(C(N2CCC(OC(F)(F)F)C2)=O)ccc1C(=O)Nc1n[nH]c(C)c1C c1(OC)ccc(OC(C)(C)C)cn1.C1(NCCN(C)CCSC)CCN(C=O)C1 c1(C(=O)NC(C)CCNC(=O)CCCC(F)(F)F)cncc(N=[N+]=[N-])c1 C1(CCC)CN(C(c2cc(C)nn2-c2ccccn2)=O)CCN1C(=O)C(Cl)=CCl c1(-c2ccc(C(=O)NC)cc2)ccn2nc(C(=O)NC(CO)C(C)O)cc2c1 n1(CC(=O)NC(C)(C)CNC(=O)CCC2CC2(Cl)Cl)cc(CO)nn1.S(=O)(=O)(C1CC1)N CCCCC(F)C(=O)N1CCSCC1C(=O)NCC1CCOC1 N1(C(C=C(C)C2CC2)=O)CC(NC(c2n[nH]c(C)c2C(F)(F)F)=O)C(F)C1 C#CCCCCCCC(=O)N1CC(NC(c2ccn(CCC(F)(F)F)n2)=O)C(O)C1 C1(CC)CCN(C(C2CN(C(C3(n4cccn4)CC3)=O)CCS2)=O)C1C N1(C(C(CC)COC)=O)CCN(C(CC)=O)CC1C(C)(C)C.c1c(C)ccn1C C(C)(C(C)(C)C(=O)NC1CC(CN(C)C)C1)NC(C(C(C)O)N(C)C)=O C1(NC(CCC(C)=O)=O)CC(NC(=O)C=Cc2nc(C)cs2)C12CCC2 c1(CCC(=O)NCC2CCN(C(=O)Cn3ccc(C4CC4)n3)C2)ccc(F)cc1 C1(CC(=O)NC(C)C(C)NC(c2cnc[nH]c2=N)=O)CCS(=O)(=O)CC1 N1(C(C2(CNC(Cc3c(C)nsc3)=O)CC(F)(F)C2)=O)CC(C)OC(C)C1 c1(C(C)OCC)nc(C)c(C(N2CCC(C)(NC(c3snnc3CC)=O)C2)=O)s1 c1(N2CC(OC)C3(C2)CCCC3)nc(=NCCc2cccs2)[nH]c2ncn(C)c12 N1(C(c2cncc(C)c2C)=O)CCC(NC(C2CCC2)=O)C(CO)CC1 O=C(C#Cc1ccccc1)N(c1ncnc2sccc12)C1CCC(N)C1 c1(C(=O)NCCCN(C(c2c(C)n(CCO)nc2)=O)C(C)C)cnn2c1CCC2 Cc1cccc(C(N2CCOC(C(=O)NC3CC4C=CC3CC4)C2)=O)c1O N1(C(CC2(C)CC2)=O)CCC(F)(F)C(CNC(=O)CCCc2ccccc2)C1 C12CCc3nc(C)nc(c3C1)C(=O)N2.c1(OC)cc(SC)c(OC)cc1N(C)C CCC(CC(=O)NCCCCCN(C(=O)C=CC1CCCN1C)C)SC Cc1nc(N(CC(C)NC(=O)CC(C)c2ccco2)C)c2scc(C)c2n1 c1(C2C(C(=O)NC(COCC(C(=O)OC)C)C3CC3)C2)c(F)cccc1Cl O=C1CC(NC(C2CC(O)CCN2C(C2C3CCC(F)(F)C23)=O)=O)CC(=O)N1 C1(C(=O)NCC(C(=O)NCC(CC)(C)Cl)C)C2CC3C(C2)C13 c1(COC2CC(OCC)C2(C)C(CN)OC)cc2ccccn2n1.C(=O)OCCC C(CC(=O)NCC1CC1CO)(C(F)(F)F)NC(CCC(C)(C)O)=O Cc1nc(N)c(CC(=O)NCC(CNC(C2CC2(C)C)=O)CO)c(O)n1 c1(C(=O)NCC=CCC(=O)NCCSCC)cnc(C(C)C)o1 N1(C(c2nccc(C)n2)=O)CCC(NC(=O)C(CCS(C)=O)N(C)C)C(C)(C)C1 C1(CNC(C2(CC)CC2)=O)CN(C(=O)C(F)C(F)(F)F)C2COCC2O1 N1(C(C(CCNC(C)=O)O)=O)CCN(C(=O)OC(C)(C)C)C2CCC12 C1(NC2(c3n(CCCC)nnn3)CN(C(C)=O)C2)CCCC(CO)C1 c1(C(C)(C)N(C(=O)NC(CC)COC)C)ccccc1Br.C1(N)CCC1 C1(C2(O)CN(C(=O)C(CC(C)C)NC(N)=O)C2)(CNC(=O)NC(C(C)C)=O)CC1 C(C(C)C(=O)N1CC(C(C)O)C1)NC(CC)=O.C1C(=O)N1C1CC1 C(=O)(C(C)(C)CC(C)C)NC1C=CC(CC(N2C(CCCC)CCC2)=O)C1 Cc1ccc2c(c1)N(C(=O)C(=O)NC1(c3ccccc3F)CCC1)CCNC2 c1(C(=O)NC(C(C)C)CCN(C(=O)Cc2cccc(F)c2)C)c(F)cccc1F C1(C(=O)NCC(CCNC(C2(CC)CC2)=O)(C)C)CC(Cc2ccccc2)=NO1 C1(NC(C(C)Cc2ccccc2)=O)CCC(C)N(C(c2cn3ccsc3n2)=O)C1 Cc1c(F)ccc(Br)c1C(=O)NCC(F)CNC(c1nc(=N)[nH][nH]1)=O C(=O)(C(C)(C)CCCc1ccccc1)NC1C2(CC(NC(CSCC)=O)C2)C1 C(=O)(CCCCCC(=O)NCC(C)NC(C1(C)CC1(F)F)=O)OC C(=O)(CCCCC(C)(C)C)N1CCC(CNC(CCCC#C)=O)C(F)(F)C1 C1(NC(c2ccc(C)nc2)=O)CN(C(c2cc(C)cc(O)c2)=O)C2CCCC12 c1(N2CCCC(CC=C)(NC(=O)C(C)OCC)C2)ncnc2[nH]ccc12 c1(C(=O)NCC(CO)NC(c2cc(CCC)[nH]n2)=O)cc2n(c1)CCCNC2=O N1(C(C2CCC(=O)O2)=O)CC2CCCC1C2CNC(c1c(Cl)n[nH]c1C1CC1)=O C1(C(=O)Nc2csc(-c3ccoc3)n2)CCCN1C(=O)Cc1cccs1 N1(CC23CCCC2C3(F)F)C(=O)CN(c2c(C)oc(-c3ccccc3)n2)C1=O c1(C(CNC(C2COC3(CCC3)C2)=O)O)c(F)cc(F)cc1F N(C1CN(C(c2ccc3c(c2)CC3)=O)Cc2ccccc21)C(CCOCC#C)=O C1(NC(C=CC)=O)CCCCN(C(=O)CSc2ccc(F)cc2)CC1 Cc1cccc(C(N2CCOC(CN(C(=O)C(C)OCC3CC3)C)C2)=O)c1C C1(C(=O)NC2C(NC(=O)CCOC3COC3)C2)C2CC3C(C2=O)C13 Cn1cc(C(=O)NC2CC(NC(=O)CCC3CCCC(=O)N3)CC2O)ncc1=O N1(C(=O)C(F)C2CCC2)CCN(C(C2CCc3n[nH]cc3C2)=O)CC(O)C1 N1(C(c2ccn(CC)c2C)=O)CCN(C(c2ncncc2C)=O)C(CCOC)C1 C1(C(=O)NCC2(OC)CN(C(C(F)=CCC)=O)C2)CCS(=O)(=O)C(C)C1 N1(Cc2cnc(C)s2)CC(NC(=O)CSc2ccccn2)C(C#N)C1 c1(C(C)NC(C2N(C(C(C)C)=O)CSC2)=O)ccc(F)cc1 Cn1cnc(NCC2(CNC(=O)CC3CCC(C)(C)CC3)CCCC2)cc1=O C(=O)(C(C(C)(C)C)N1CCNC1=O)NCC#CCNC(C(n1ccc(C)n1)C)=O C1(CCOC)(NC(c2[nH]ccc2C)=O)CCN(C(=O)C(C)N(C)C)C1 c1(C(=O)NCCOCC#C)ccc(C(c2nnnn2C)NC)o1 c1(CC(=O)N(C2CCN(CCOC)C2)CCC)nccc2ccccc12 CC(C)CC(CNC(=O)C(C)(O)C1CCC1)NC(=O)CSc1ccc(F)cc1 c1(C(c2nnnn2C2(C)CC2)NCc2ccc(C)cc2)c(C)cccc1F c1(NC(c2c(C)scc2)=O)ccc(NC(c2csc(Br)c2)=O)cn1 CC1CCCC=C1C(=O)N(C)CC1CCCN(C(=O)C(F)(F)c2cscn2)C1 C1(CNC(C=CS(C)=O)=O)(NC(c2cnn(C3CCCC3)c2)=O)CCCCCC1 c1(C(=O)NCCC(=C)CNC(=O)Cc2ccc(Cl)c(F)c2)cc(O)nc(OC)n1 N1(C(c2c(C)snn2)=O)CCOC2(C1)CN(C(=O)CCC1CCCC1)C2 C1(NC(=O)NC(CSC)(C)C)CCCC(F)C1 CCC(CCC(=O)N1CC(O)CC1CNC(=O)CCCC1CCCO1)OC N1(C(Cn2ccc(C)n2)=O)CCCC(C)(NC(=O)CSCc2ccccc2C)C1 N1(C(C2C(CCC)C2)=O)CCC(NC(=O)C(=O)N(C)C)C(F)(F)CC1 c1(C(=O)NC2CCCC(N(C(CC=C=C)=O)C)C2)cn2c(n1)CCCC2 C1(C(=O)NCC2C(NC(C3CC3(Cl)Cl)=O)COC2)CCC(F)(F)CC1 N1(CC)CCC(Cc2nc(C(=O)Nn3cncn3)sc2)C1 CC1(C)C2CC1CNC2=O.c1(CC(=O)NCC(F)F)n[nH]c(=N)s1.C1(=O)CO1 c1(C(C(=O)NCCN(C(C2CCCN2C2CC2)=O)CC)O)cnn(C)c1 c1(Cc2nc(C(C)(C)NC(C)=O)sc2)cccc(S(=O)(=O)C(C)C)c1 C#CCC(C(=O)NCC(C)(N)CSC)N(C(=O)C(CC)N(C)C)CC C(=O)(C1=NOC2(CCC2)C1)NC1CC(C)CN(C(c2cccn3nnnc23)=O)C1 N1(C(=O)OC(C)(C)C)CC(CC2C3CCCCC23)CC2CCCCC12 C(=O)(CCCCC(=O)OC)NCC1(CC(=O)OC)CC1.C1(=O)C(C(C)C)CC(=O)N1 CC(CS(C)(=O)=O)C(=O)NCCC1CCCN(C(=O)C2=CC3CCCC23)C1 CC1CC2(CCN(C(c3cncc(CO)c3)=O)CC2)CN1C(=O)C1=CCC1 C(CN=c1cc(Cl)c(O)n[nH]1)(N(C(C(CCSC)O)=O)C)C1CC1 N1(C(C2(OCC)CCCC2)=O)CCC2(CC1)COC(CNC(=O)C#CC1CC1)C2 N(C1CCCn2cnnc21)C(CC1(C)N(C(C2(COC)CC2)=O)CC1)=O c1(C(=O)NCCC2CCN(C(=O)CCC(F)F)C2)ncc(Cl)cc1Cl c1(C(=O)NCC2N(C(C3ON=C(CC)C3)=O)CCC2)noc2cc(F)ccc12 C12(NC(c3cn[nH]c3)=O)CCCN(c3nncs3)CC1C2.C1(C(=O)N)(CC)CCCCC1 C1(c2n(CC)nnn2)(NCCc2n[nH]cc2Br)CCOC(CCOC)C1 Cc1ccc2nonc2c1C(=O)NC(C)CCNC(=O)CCCc1n[nH]c(=N)s1 CC(c1ccc(OC(F)F)cc1)=CCNC(=O)NCC1(CN(C)C)CCCC1 c1(C(=O)NCCN(C(C2(CC#C)CCOC2)=O)CC2CC2)cc(Cl)cnc1OC c1(CC(CNC(CN(C(C)=O)C)=O)C(=O)O)c[nH]c2ncccc12 C(=O)(CCCCCS(N)(=O)=O)NCC1CCCC(NC(C2(C)C=CCC2)=O)C1 C1(C)(C(=O)NC(c2nc(C(=O)NC(c3ncc[nH]3)CO)co2)C)SCCCS1 CC(C)(CCC#N)C(=O)N1CC=C(CCNC(=O)CC2CN3CCC2CC3)CC1 C(=O)(C1CCCn2cnnc21)NCCN(c1ccccc1)C(C(C)C1CC1)=O C1(C(=O)NCC2N(c3nnn(C)n3)CCC2)CCC(=C(F)F)CC1 c1(C(N2CCCC3(CCNC3)C2)=O)ncnc2c1oc1ccccc21 C#Cc1ccc(C(=O)NCCN(CCC(C)O)C(C2(C)CCCS2(=O)=O)=O)cc1Cl C1(CC(=O)NCCN(C)C)CCCC(N)C1 c1(CNC(C2(CC=C)CC2)=O)ccoc1C(=O)NC1CCN(C(C)C)C1 c1(C(=O)NC2(C3CCCN3C(=O)NC)CCC2)ccc(OC2CC2)cc1 C(=O)(CCC(C)(C)OC)NC(CNC(CC1CC(=C)C1)=O)C1CCC1 C1(C)(CC)CC(NC(=O)CCNC(C)=O)CN1C(c1ncnc(C)c1C)=O CC1CC(N(C(=O)CCCN(C)C(c2csc(Cl)c2)=O)C)CC(C)C1 N1(C(c2ncc(OC)nc2)=O)CC(F)(F)CC1CNC(C12CCC(F)(CC1)C2)=O CC(C)(Cc1nn[nH]n1)NC(=O)Nc1sc(CC2CC2)nc1C(F)(F)F Cc1cccc(O)c1C(=O)N(C(C)(C(=O)NCC(C1CCOC1)C)C1CC1)C Cc1c(F)ccc(C(=O)NCCC2CCN(C(=O)Cc3cc[nH]n3)C2)c1N N1(C(c2c(C)nncc2)=O)CCC(C2CCN(C(C3(F)CC3C)=O)C2)CC1 c1(C(C)NCC2C(CCC)C2)cnn(-c2ccccc2)c1F c1(-n2cc(C3CN(C(C(c4ccoc4)N(C)C)=O)C3)nn2)ncc(Br)cn1 C1(C)(C(=O)NC2C3CC(NC(c4n(C)cnc4)=O)CC32)COC(C)(C)CO1 N(C(=NCCCCl)NCC1CCCC1O)Cc1cc(N(C)C)ncc1 N1(CC(CN(c2cccc(OCCO)c2)C)O)CCC(CO)C(O)C1 c1(CCC(N2CCC(OCCNC(c3ccncc3Cl)=O)C2)=O)cccc(O)c1 N1(C(C(C)CF)=O)CCC(NC(=O)C(O)C2CCCC2)CC1 C(CC(CO)C(C)C)NC(c1cc(CNC(C#CC(C)C)=O)sc1)=O N1(C(C)=O)CCOCC1C(N1CC(CNC(=O)C(F)(F)C2CC2)C(O)C1)=O N(CP(C)(C)=O)(C(=O)OC(C)(C)C)CC1CC1c1cccc(OC(F)(F)F)c1 C1(NC(C=C(CC)C)=O)CC2CCC1(CNC(c1nc(C)n(-c3nc[nH]n3)n1)=O)C2 C(=O)(NN1CCCC1C(=O)NCC1(C)CCC(=O)N1)c1nc(CC)sc1 c1(C(=O)NCC(CNC(c2c(C#C)c[nH]n2)=O)(C)C)c[nH]c(=N)nc1C(F)(F)F C1(NC(=O)CCc2cccnc2F)CC2CCC(C1)N2C(=O)Cn1ccnn1 C12(CCCCC1)C(=O)N2.C1(O)(C(N(CC#CC)C2CC2)=O)CCN(C(C)=O)C1 N1(C(c2cc(C(=O)OC)n(C)n2)C(=O)NCC(F)F)CCC2CCN(C)CC12 C(=O)(C1=CCCCO1)NC1CN(C(CCOc2ccc(C(N)=O)cc2)=O)C2C1C2 C1(C(C)C)CN(C(=O)Nc2ccc(C(=O)NC(C)C)cn2)CCO1 c1(CC)noc(CC)c1CC(=O)NCCC(C)(C)NC(c1csc(CSC)n1)=O C(=O)(C#CC(C)(C)C)N(C1CCCN(C(c2ccc(NS(C)(=O)=O)nc2)=O)C1)C C1(NC(C2(N(C(=O)C3CC3)C)CCOC2)=O)CCc2c[nH]nc2C1 c1(C(N2CCN(CC(N3CCC(C#C)CC3)=O)CC2)=O)cccc2c1CCC2 N12CCN(CC1)c1ccnc(n1)C2=O.n1(C(COCC)C)cc(C(C)=O)nn1 C1(CNC(CN(c2ncccn2)C)=O)CN(C(c2cncn2C)=O)C(C)(C)C1 N1(CC(=O)NCC)CCCOC(CN2CC(=O)N(CC)C2=O)C1.C(C)(C)(C)OC=O C(=O)(C1CCCn2c(Br)cnc21)N1CCCN(C(C(C(C)C)(C)O)=O)CC1 c1(C(=O)NC(CNC(c2nc(COCC)oc2)=O)CC)n[nH]c2c1CC(C)CC2 c1(C(N(C2CCN(C(=O)C(F)(F)c3cscn3)C2)C)=O)ccn(O)c(=O)c1 C(=O)(C1=CCCC1(C)C)NC(CCCC)CNC(=O)CCNc1ncccn1 C1(C(=O)NCCOCC(C)C)N(C(=O)COCC(F)F)CC12CCCC2 CCC(CC)(CCNC(C1CN(C)CCO1)=O)NC(=O)CCCc1ccsc1 CCCC(CNC(c1ccnnc1C)=O)C(=O)NCCOC1CCOC1 CC1(C)C(NC(=O)CC2CC(=O)NC(=O)C2)CCN1C(c1cncc(CO)c1)=O C1(NC(C=CC)=O)CCN(C(c2cc(CCO)on2)=O)C1C1CC1 C1(O)(CN(C(C(C)CC2CC2)=O)C)CCN(C(c2ccon2)=O)CC1 Cn1cc2c(n1)CC(C(=O)NC(CNC(c1csc(=N)[nH]1)=O)CO)NC2=O C#CC1CN(C(=O)CC2CCS(=O)(=O)CC2)CCN1C(=O)C(COC)N(C)C c1(C(=O)NCC(CN(C(C2CC3CCC2O3)=O)CC)(C)C)nc(O)nc(O)c1N c1(NC(=O)CC2CN(C(c3ccc(O)nc3)=O)C2)nccc(Cl)c1I c1(Sc2ccc(Oc3ccccc3)s2)ccnc(Cl)c1F.C12CCCN1C2=O c1(CC(N2C(CN(C(C3(COCC)CC3)=O)C)CCC2)=O)cnn(C)c1C C1(C(=O)NCc2n(C)ccc2)CCC(NCC2CCC(O)CC2)CC1 c1(NC(c2n(CCC)nnn2)(c2ccccc2)C)ccc(NC(=O)COC)cc1 C(=O)(C1Cc2ccc(Cl)cc21)N1CCN(C(Cc2c(C)nn(C)c2Cl)=O)CC1 CC(C)(C(=O)N1CCC(C2CCCN2C(C2CCCC2)=O)C1)C(F)(F)F N1(C(c2cn(C)c(OCC(F)(F)F)c2)=O)CCc2nc[nH]c2C1c1ccc(Br)cc1 C1(C(N2CCC(CCNC(c3cc(C(N)=O)[nH]n3)=O)C2)=O)CCC2C1C2(F)F N1(C(C(C(C)C)O)=O)CCN(C(=O)CCCC(F)F)C(C)C1 N1(C(c2c(C)n(C3CCOC3)nn2)=O)C2CCC1CN(C(=O)CC1(C)CC1)C2 C1(C)(C(=O)NCC(CC(C)C)OC)CC(O)CN1C(C1CC2(CC2)C1)=O C1(C(=O)NCC(C)(CO)CO)CCCN1NC(=O)c1coc(CO)c1 C1(C(=O)NCCC(C)F)COCCN(C(=O)C2=CCCC2C)C1 N1(CC(=O)N(CCC)Cc2ccc(Cl)cc2)CCN(CCC)CC1.C1(=O)C(C)N1 c1(C(C)C)nn(C)cc1C(=O)NCC(C1CCCC1)NC(=O)CCn1cncn1 C1(C(N(C(C(=O)NCC(C)(C)SC2CC2)C2(O)CCC2)C)=O)CCCSC1 Cc1cc(C(=O)NC(C)(CO)C(=O)N2CC(F)(CF)C2)oc1C N1(C(C(c2n(C)ccn2)(F)F)=O)CCOC(CNC(=O)CCSC2CC2)C1 C(=O)(CCC(C)(F)F)N1CCC(C(N2CC(CSC)C2)=O)(CF)C1 c1(OC(C)C)cncc(C(=O)NC2CC2CNC(C2CC3CCC2O3)=O)c1 C1(C(=O)NCC2CCC(F)(CNC(C3C(=C)CC3)=O)CC2)CC2(CC(C)=NO2)C1 C1(CNC(C2(C(F)F)CCCO2)=O)CCN(C(C23CC(CC(F)(F)F)C2C3)=O)C1 c1(C(=O)NCC(=O)NCC2(NC(=O)CSCC3CC3)CCOC2)ccc(F)cc1 N1(C(C(CC)CC)=O)CCCC2(C1)CN(C(C1(c3ccccc3)CC1C)=O)C2 N1(C(C(CN(C)C)NC(C2CC2c2ccccc2)=O)=O)CCOc2ccccc21 c1(N(C(C2(N3CCC3)CCC2)=O)CC)cc(Cl)ccc1[N+](=O)[O-] C=CC1CN(C(c2cc(C)ccc2OCCC)=O)CC1NC(=O)C(C)(C)CO C1(CCNC(=O)C(C)OC)(NC(S(CCC)(=O)=O)=O)CCOCC1 N1(C(c2ccc(C)[nH]2)=O)CCC(C)C(NC(C2(CN(C)C)CCCC2)=O)C1 C1(C(=O)NCC2(C)CCCN2C(c2cnccn2)=O)CCn2nncc2C1 N1(C(Cn2cc(C(=O)NC)nn2)=O)CCN(C(=O)C2=NOC(C)C2)C(CF)C1 C(CN=C(NCc1ccc(F)cc1)N(C)CN1CCCCC1)SC C(=O)(C1=CC2(CCN(C(=O)C(F)CCC)C2)C1)NC(CCCC)CC CC(C)CCC(O)C(=O)N1CCCCC(CCC(=O)NCCN(C)C2CC2)C1 C1(O)(CCNC(c2ccn(C3CC3(F)F)n2)=O)CN(C(C23COCC2C3)=O)C1 N1(CCCOC)CCCC(C)CC1.c1(NC(C2CNC(=O)O2)=O)cccc(Cl)c1 Cc1cc(C)c(C(=O)NCC2CC3CCC(C2)N3C(=O)CCCF)cc1Br c1(COC)c(C)nc2cc(Cl)ccn12.C1(C(C)(C)C(=O)OC)C2CC(C2)C(=O)N1 C(=O)(C1OC(=O)c2ccccc21)NC(CNC(CC1(C=C)CC1)=O)C N1(C(CCC2C(C)(C)C2)=O)CCOC(CNC(c2ccoc2Br)=O)C1 C(=O)(C1CCC(=O)c2cccn21)N1CCCCC(CNC(COCC=C)=O)CC1 N1(C(=O)Nc2ccc(C)cc2)CCN(c2nnc(C(=O)NC)n2CCNC)CC1C N1(C(c2oc(C)c(CO)c2)=O)CC(CNC(=O)C(F)C2CCOC2)CCC1C N1(C(C(CC)NC(C)=O)=O)CCOCC(CNC(C2(C)CCOC(C)C2)=O)C1 N1(C(CSC)=O)CCCC(C2CCN(C(c3nc(C)n(C4CC4)c3C)=O)CC2)C1 CC1CCN(C(=O)C(c2cnccn2)C)CCN1C(c1ccc(=O)oc1)=O c1(C(=O)NCC(=C)CCNC(C2COCC(C)O2)=O)c(Cl)ccc(F)c1C c1(OCC=C)ccc(CNc2cccc(N3CCOCC3=O)c2)cc1Cl C1(NC(C2=CCN(C)C2)=O)COC2C(NC(=O)CC3CC34CC4)COC12 C1(C(=O)NCCNC(C2C(COC)C2)=O)CC(C(C)C)=NO1.c1(S)ccc(F)cc1 c1(C(=O)NCCCNC(c2csnc2Br)=O)ccc2c(c1)OCO2 C12(CNC(CNC(CC(C)C)=O)=O)CCCC1N(C(=O)Cc1ccsc1)CCC2 Cc1ccc2sc(N(C)CCNC(=O)CC3CCCC3OC(C)(C)C)nc2c1 CCC(F)C(=O)NCC(O)CN(C)C(c1cnn(C(F)(F)F)c1)=O C1(C(=O)NCC2N(C(CCc3n(C)cnn3)=O)CCOC2)CCCC(C)(C)C1 c1(CC)sccc1C(=O)NC(C)(CNC(=O)CCNC(=O)COC)CC C1(C(N2CC(O)(C(C)NC(C(C)NC(CC)=O)=O)C2)=O)CC2CCC1C2 O=S(=O)(c1ccc(OC(F)(F)F)c(Cl)c1)NCCCc1ccc(F)cc1F C=C1CC2(C1)CC(C(N1CCOCC(NC(=O)C(c3ccc(C)s3)C)C1)=O)C2 CC1(C)CCCN(C(=O)CN2CCOCC2)C1CNC(=O)CCCc1nccs1 C1(C(=O)NCc2oc(C(N(C)Cc3c(C)nco3)=O)c(C)n2)CC(C2CC2)=NO1 C1(CNC(C(C)=C(CC)C)=O)CN(C(=O)C=CCN(C)C)C2(CCOCC2)C1 c1(C(N2CC3(CN(C(C(C(COC)C)C)=O)C3)C2)=O)ccc2ccncc2n1 c1(C(=O)NC(C)CNC(=O)C(C)(C)C2CC2)ccnc(N2CCN(C)CC2)n1 c1(C(=O)NC(CCC)(C)CO)nc(C)c(C)cc1N C1(CNC(CCN(C(CCC)C)C)=O)CC12CCN(C(c1ccsc1CC)=O)CC2 Nc1cc(F)cc(C(=O)NCC2CCC(NC(c3c[nH]nc3[N+](=O)[O-])=O)C2)c1N c1(OCCC)cccnc1C(=O)NCC#CCNC(=O)CCC1CCCC(O)C1 N1(C(CN(CCCCCC)C)=O)CCC2CCN(C(=O)Cc3nc(C)cs3)CC12 CC(CC(C)C(F)F)NC(C1CC(C)CCN1C(=O)CC1CCCC(C)O1)=O C(c1ncccc1C)=CC(N1CCC(C(C)NC(c2c(COC)cco2)=O)C1)=O c1(CCC(N2C(C(C)(C)CNC(C3CCO3)=O)CCC2)=O)ccc(F)cc1 c1(C(N(CC(CNC(Cc2cc(C)on2)=O)(C)C)C)=O)cccc([N+](=O)[O-])c1Cl N1(S(C)(=O)=O)CCC(c2nc(-c3cnncc3C)n(CCF)n2)CC1.C1(CC)CCC1 N1(C(CCC(C)OC)=O)CCCCC(C(=O)NC(CO)CCC2CC2)C1 N1(C(C(CCC)Cl)=O)CCC2(CCCCC2NC(=O)CSCC(N)=O)C1 O=C(CCC(F)(F)F)N(CCCCC1CN(C(=O)CC2(N3CCCC3)CC2)C1)CC c1(C(=O)NCC(CC)NC(c2ccc(F)c(O)c2F)=O)cc(C)sc1S(N)(=O)=O c1(CC(=O)N)cccc(OC(F)(F)F)c1.C12CC1C(=O)NC1CC1NC2.CCO c1(C(=O)NCC2(F)CN(C(C(C)(C)c3ccccn3)=O)C2)ccc(N)cc1Cl c1(-c2ccn(CCSC3(F)CCN(C(=O)OC(C)(C)C)C3)n2)cc(F)ccc1F CCC(C#N)C(=O)N1CC(O)(CC(=O)N(CC(F)F)C2CC2)C1 c1(C(=O)NCC(C2CCC2)NC(C2C=CCC2)=O)cccc(CF)c1 c1(C(N2CC(F)(CNC(c3ccc(F)cc3)=O)C2)=O)sc2cccnc2c1Cl C(=O)(CCC(N)C(=O)O)OC.c1(CC)noc2c1C2.N12CCC(CC1)C2 C1(C)(C(=O)NCCN(C(CNC(C(CC)CC)=O)=O)CC)OC(C)(C)OC1C C#CCCCCCCC(=O)N1CCC(C(N2CCC(CCOC)C2)=O)C1C(C)C c1(OC)cc(C(N2CC(O)(CNC(c3c(C)ccnc3O)=O)C2)=O)nc(C)c1 c1(C(=O)NC(CCNC(C23C(C(C)=O)(CCC2)C3)=O)(C)C)ccc(O)c(C)c1C c1(C(=O)NCC2(F)CC(NC(C(C)n3cncn3)=O)C2)ccc2c(c1)nnn2C c1(CC)cc(NC(c2nnnn2C2CCOC2)CC2CCC2)ccc1C c1(OC)cc(C(N2CC(NC(c3nc(=N)cc[nH]3)=O)CCC2C)=O)cc(C)n1 C1(CNC(=O)C=CCOC2CC2)CN(C(c2ccnn2C(F)F)=O)CC1(F)CC#N c1(C(N2CC3(C2)CC(F)(F)C3)=O)cc2cc(Br)ccc2s1 C1(NC(C(Cn2ccc(C)n2)C)=O)CCN(C(c2cc(Br)c[nH]2)=O)CC1O C(=O)(CC(C)(C)CCOC)NC1C2CC(CNC(CN(CCOC)C)=O)CC1CC2 C1(C(=O)NC(C#C)CC)CCN(C(=O)Cc2cccc(O)c2)C(C)(C)C1 N12CC(C)(C)C1C2.Cc1cnn(CCC(=O)Nc2cccnc2)c1 C1(OC)CN(C(=O)C(N2CCOCC2c2cn(C(C)C)nn2)C)C1(C)C C1(C(=O)NC(C(C)C)CC(N2CCCC(C)(C)C2)=O)CC2(C1)CC2(F)F c1(C(N2CC(C)CC(NC(c3c(CC)nc(C)[nH]3)=O)C2)=O)ccn2c1CCCC2 N1(C(CSCC)=O)CC2CC(NC(C3(c4ccccc4)CCC(=O)NC3)=O)C2C1 n1(CC(C(N2CCCC(N(C(C(C(C)C)O)=O)C)C2)=O)C)ncc2c1CCCC2 c1(N(C)C)cc(C(=O)NC2CCCC(NC(c3nsnc3O)=O)C2)cc(Cl)n1 c1(C(N)=O)nc(CC(=O)NCC(=O)NCC(O)CNC(=O)Cn2cn[nH]c2=N)cs1 N1(C(c2c(CC)ncs2)=O)CC2CCCC(N(C(=O)C(C)=C3CCCC3)C)C2C1 C12(C(N3CC(C)(CC)C3)=O)CC(CO1)N(C(=O)CC1CSCCO1)C2 Cc1ccc(CC(C)C(=O)N2CC(NC(=O)C=Cc3nc(C)co3)C2)cc1 N1(C(c2c(C)cccc2)=O)CC(NC(=O)C=CC(C)C)C(C2CC2)C1 C1(C(=O)NC(CC(C)C)CNC(C2CCCCCC2)=O)CC2CCC1CC2(F)F N1(C(c2[nH]c(=NC)sc2)=O)CC2CCC(C1)N2C(=O)C=CC1CCCC1 C1(CC)CN(C(=O)NC2(n3cc(Br)nn3)CC2)CCCO1 N#CC1=C(C(=O)NC2CN(C(C3CCCCC3O)=O)CC2N=[N+]=[N-])CCC1 Cc1cc(C)n(CC(N2CC(C)N(C(=O)CCS(N)(=O)=O)CC2C)=O)c(=O)n1 C=CC(C)(O)C(=O)N1CC2CC2(NC(=O)C=CC(C)(C)C)C1 Cc1ccc(NC(C2CCCN(C(=O)C(n3ccc(C)n3)C)C2C)=O)cc1C CS(=O)CCC(=O)NCC1COCC1NC(=O)C=Cc1cc(C(N)=O)co1 CCCCCCCNC(C1(N(C(=O)C(O)CC2CCCC2)CC)CC1)=O c1(C(C)=O)ccc(Cl)c(C(=O)O)c1.c1(CC(N2CCC(C)C2)=O)cn(C)nc1C C1(NC(=O)COc2ccccc2)C2CC1N(C(=O)CN1CCOCC1)C2 C1(N(CCC)CC)CN(C(=O)CCNC(=O)COC(C2(OCC)CC2)=O)C1 c1(C(=O)NCCC(C)N(C)C(c2cc(Cl)ccn2)=O)ccncc1F c1(CN2CC(O)(CCNC(C(c3c(C)n[nH]c3C)C)=O)C2)ncnc2c1CCC2 C1(NC(c2ccc(C)c(C)n2)=O)CN(C(=O)C(C)Cc2ccco2)CC(F)(F)C1 N1(C(CCC2C(C)C2)=O)CCOC2CCN(C(=O)C=C3CCSCC3)CC12 N12CCN(CC1)C(=O)C(C)CC2.Cc1nccn1CC(=O)N(C(=O)C(C)C)C C1(F)(CC)CCN(C(C2CCC(CNC(=O)CCCN3CCCC3)O2)=O)C1 N1(C(=O)OC)CCN(C(=O)C2CC2)CC1.n1(C(CO)C)cc(C)nn1 C1(N(C(C2C(C)CCO2)=O)C)CN(C(=O)CC2(C(F)(F)F)CCC2)CC1O CC(C(=O)NCC(C(=O)N1CCC(CC(C)(C)C)C1)N(C)C)C(C)(C)C c1(CN(C(C(CC)OC)=O)C)cccc(C2CCC2)c1 N1(CCNc2nc(C)nc(N3CCCCC3)c2)CCCNC(=O)C(F)(F)C1 c1(C(N2CCC(C(C)NC(=O)CC3CCSCC3)C2)=O)ccc2c(c1)OCCO2 c1(C(NCC(N2CC(CC)C(O)C2)=O)=O)cc(C)ccc1OC c1(C(C)(F)F)cc(C(=O)NCC(C)(C)CNC(=O)CC(C)n2cccn2)[nH]n1 c1(C(=O)NCCN(C(c2nc(C)n(C)c2)=O)C2CC2)cc2c(C)nn(C)c2s1 N1(C(C(C)OCC)=O)CC2CC(C(=O)NCC3CC3C(F)(F)F)(C2)C1 c1(C(=O)NCC(C)N(C)C(C2(F)CCCN(C)C2)=O)cncc2c[nH]nc12 N1(C(c2c(C)nc(CC)o2)=O)CC(N(C)C(C2CC2c2ccsc2)=O)C(C)(C)C1 C1(C2CCOCC2)(C(=O)NCC2CC(F)(CNC(CCC(=O)NC)=O)C2)CC1(F)F n1(CC(=O)N(CCCNC(C(C)N2CCCC2)=O)C)cc(F)ccc1=O C(C(C)(C)C#CC(=O)NCC1CCCN(C)C1=O)NC(CC=C)=O c1(CNN2C(CCC(N3CC4CC3CS4=O)=O)CCC2)cccc2c1OCCO2 C1(NC(C2(C)CCC2)=O)COC2(CCCN(C(=O)CC3CC(F)(F)C3)C2)C1 C1(NC(Cc2n(C)ncc2)=O)CCCCC1NC(=O)Cc1cnc[nH]1 C=CCC(C(=O)NC(C)(C)CCNC(C1CC2CCC2C1)=O)NC(C)=O C1(CC(NOCC2CC(=C)C2)=O)CCCCN1C(=O)C(n1ccnc1C)C N1(C(C2C(CC)OCC2)=O)CCC(CCNC(=O)C(F)(F)c2cnn(C)c2)CC1 C1(C(N2C(C)CC(CC(=O)NCCC(C)CO)C2)=O)CC12CCOCC2 CC(Cc1cnco1)C(=O)NCCCC(C)NC(=O)NCc1ccccc1 C1(CNC(C2CC=CCC2)=O)CCN(C(c2cc(O)ccc2N)=O)C12CCC2 C1(NC(c2ccc(CC)nc2)=O)C2CCN(C(=O)C(C)N3CCCC3)CC12 c1(C(=O)OC)cnc(NC2CCNCC2F)nc1 O=C1CCC2(C(=O)NCCCNC(c3ccc4occc4n3)=O)CCCCC2N1 C(c1ncc(-n2cc(CC(C(=O)O)c3ccccc3)nn2)cn1)=CC(C)C C1(C(C(c2cc(OC(F)(F)F)cc(Br)c2)C#N)=O)Cc2ccccc2NC1=O C(=O)(C(C(C)(C)C)N(C)C)N1CC2C(CNC(c3c(C)ccs3)=O)(C2)C1 Nc1c(C(=O)NCC(CO)NC(c2cnn3cnnc3c2)=O)ccc(Br)c1F CC(C(C)(C)C(=O)NC1(C2CC2)CCC1)NC(c1cnc2n1CCC2)=O C(=O)(CC(C)(C)CN(C)C)NCC(C)N(N(c1ccc[n+]([O-])c1)CCO)C N1(C(COCCCOC)=O)CC2(CC(C(N3CC(OCCO)C3)=O)CO2)C1 C1(OC)CN(C(=O)Cc2cc(Cl)c(Cl)s2)CC1c1cn(CC2CCCO2)nn1 c1(C(=O)NCc2c(C(N3CCC(C(=O)OCC)C3)=O)n[nH]c2)c(C#N)cnn1C Cn1nc(C(c2conc2C2CC2)N(C2CCCCC2)CCF)c2c1CCSC2 C(c1cncs1)=CC(=O)NC(CC1CCOCC1)C(=O)NCCC1CCCCC1 C1(CNC(CCN(S(C)(=O)=O)C)=O)C2CCC(C2)N1C(=O)C1=NOCC1 Cn1c(=O)n(CC(=O)NC2C=CCN(c3cc(=O)n(C)c(O)n3)C2)c2c1CCC2 N1(Cc2ccc(CNC3(C)CC(NC(=O)OC(C)(C)C)C3)o2)CCN(C)C(=O)C1 N1(C(c2c(Cl)ccc(C)c2Cl)=O)CC2COCC(C1)N2C(C1CCC(C)O1)=O N1(C(=O)OC(C)(C)C)CC(CC(=O)O)C2(CCCOC2)C1.c12ccc(nc1)CN2 N1(C(c2onc(CC)n2)=O)CCC(NC(c2cnc(Cl)cn2)=O)C12CCC2 N1(CCC(=O)N(C2CCN(C(=O)COCc3ccncc3)C2)C)CCC(O)CC1 CCCC(CC)C(=O)N1CCC(C(N2CC=CC2C(=O)N(C)C)=O)C(C)C1 CC1(CCC(N2CC3(CCC3)C2)=O)CCCN1C(=O)CN1CCCC1 C1(CC(=O)N(CC(=O)NCCN(C(C(C)C)CO)C)C2CC2)CCC(=O)NC1 N1(C(c2ccon2)=O)CC(C(=O)NCCOCc2ccccc2)C(F)(F)C1 C12(N(C3CN(C(C)=O)CC3(C)C)C(c3nc(F)ccc3Cl)=O)CCC(=O)N1CCS2 c1(C(=O)NC(C2(NC(C3CC=CCO3)=O)CC2)C)nc(-c2ccccc2)oc1C C1(C(=O)NCC2CCC(NC(CC(=C)C)=O)CC2)CCn2c(C)nnc2C1 N1(C(=O)CCc2ccsc2)CCC2CCN(C(C3CC(=O)N(C4CC4)C3)=O)C2C1 C1(CNC(=O)C2CC2)CCCC12CCN(C(C1(CO)CCCCC1)=O)CC2 c1(C(=O)NC(CC)(CNC(C2CC2(Cl)Cl)=O)CC)noc2c1COCC2 N1(C(c2ccn(CC)n2)=O)CC(NC(c2ccn(CC#N)n2)=O)C2(CC2)C1 CC1(NC(=O)C(CCC2CC2)NC(=O)CCc2nncs2)CC2CCC1C2 C(N=c1nc2scnc2c(NCC2(CO)CC2)[nH]1)C1CC(C)S(=O)(=O)C(C)C1 N1(C(C(COC)COC)=O)CC2CCOC2(CNC(c2cn(C)c(=O)cn2)=O)C1 C1(C(=O)NCCCCN(C)C(c2cn(CC3CCOC3)nn2)=O)COC2(CCC2)C1 C1(NC(=O)CN2CCOCC2)CN(C(c2cc(Cl)sc2Cl)=O)CCC1F C(=O)(C(F)C(C)CNC(=O)COCCC)NC1(CC=C)CCC1 c1(C(N2CCC(NC(CNC(=O)NC)=O)CC2C2CC2)=O)nnc2ccccn12 C1(C(=O)NCC(C)=CC(N2CCC(c3cc[nH]n3)C2)=O)CCCC1C1CC1 c1(C(N2C(CN(C(=O)CC3CCCC3(F)F)CC)CCC2)=O)cnn(C(C)C)c1F c1(C(C)C)cc(Br)sc1NC(N1CCCC1c1ccc(Cl)nc1)=O c1(NC(C2CC3(CC(OC)C3)C2)=O)ncnc2c1CCC2 c1(C(c2n(CC=C)nnn2)NCCc2ccncc2C)ccccc1CC CCCC(C)(O)CC(=O)NC1CN(C(=O)C(C)=C(C)CC)CC1CO C#CCCN=C(NCC1CCN(C2CC2)C1)NCC1(C2CC2)CC1 C(=O)(CCC1=NNC(=O)CC1)NC1CC(NC(c2c(C)ncnc2)=O)C(O)C1 C1(CC)CN(C)CCCN1C(c1c(Cl)sc(Cl)c1Cl)C(=O)NCCN1CCOCC1 c1(-c2c(OC(C)C)cncc2)ccn2cc(C(=O)NCC(O)C(F)(F)F)nc2c1 CC(=NO)C1CC(C(=O)NC2(CO)CN(C(=O)CC3CC4(CC4)CO3)C2)C1(C)C Cc1cc(=NCC(C)CNC(c2[nH]cnc2C)=O)[nH]c(C(F)(F)F)n1 C1(OCCC)CCN(c2nnc(C3CCCCO3)n2CC2COCCN2C)CC1 CC1=CC(C)CN(C(=O)C(O)CCCNC(c2c[nH]c(=N)c(C)c2)=O)C1 c1(CC)cccc(NC(=O)CONC(=O)Cc2ccon2)n1 CC(C)CC(C)CC(C)C(=O)NC1CN(C(C2CC(=O)CO2)=O)C1 c1(C(C)C)ccc(C(=O)NC2CN(C(C3CCN(CC(F)F)CC3)=O)C2)c(F)c1 CCC(CC)(CC)C(=O)N1CCCC(C)(NC(=O)C(n2ccnc2C)C)C1 CCC(C)C(C(=O)NCC(c1nncn1C)C)N(C)C.c1c(=O)n1 C1(NC(C(C)c2cc[nH]n2)=O)C2CC3C1C3C2C(N1CC(C)(CO)CC1(C)C)=O C1(C)(NC(CCc2cc(C)on2)=O)CCN(C(=O)C(C)NS(C)(=O)=O)C1 c1(OC)cc(SC)ncn1.N12CC(C(=O)N(CC(C)C)C)(C1)NCC2=O N1(C(c2ccc(F)nc2)=O)CCOC2(CCN(C(=O)C(F)(F)CC3CCCO3)C2)C1 C1(O)(C(N2CC(NC(c3coc(-c4ccccc4)n3)=O)C2)=O)CCSCC1 N1(C(C(C(C)C)SC)=O)C2CCC1C(C)C(NC(c1cc(C3CC3)no1)=O)C2 N1(C(C(CNC(COCCCOC)=O)(C)CC)=O)CCCCC(N(C)C)C1 c1(C(N2CCN(C(C3C(C)(CC)C3)=O)C(CO)C2)=O)n[nH]c2c(C)cccc12 N1(C(CC=CC)=O)CC2CC2(C(=O)NC2(CCCCO)CC2)C1 C1(NC(CCSC)=O)Cc2ccccc2CN1c1cc(F)cc(F)c1[N+](=O)[O-] c1(C(c2nnnn2C)NC2(CC)CCC2)ccccc1C(=O)N(C)C CC(C)C(C)(CNC(c1coc(C2CC2)n1)=O)NC(c1conc1C1CCC1)=O c1(-c2scc(C)n2)ccc(CN2CC(CO)CC2C)cc1.c12ccc(cc1)o2 C1(NC(C(C(CC)C)N(C)C(c2ccn(CCF)n2)=O)=O)CCCCC12CCC2 c1(C(=O)NC2CC(CNC(CC=C=C)=O)C2)cn(CC(C)C)nc1C(=O)OC N1(C(Cc2c(C)ccs2)=O)CCCCCC1CNC(C1CSCC(=O)N1)=O N1(C(C2CCN(C(=O)CC3CCOCC3)CC2F)=O)CC(F)(F)C(F)(F)C1 c1(C(N2CCC(C)(NC(CCC(=C)Br)=O)C2)=O)ncc(F)c(OC)n1 c1(CC(=O)NC(C(CO)NC(C(CC)n2ccnc2)=O)C)ccc2c(c1)CCO2 C1(NC(=O)C=Cc2cnc[nH]2)CCC(NC(c2ccncc2C2CC2)=O)CC1 c1(OCC)ccc(NC(=O)C(N2CC(O)C(O)C2)=O)cc1S(N)(=O)=O c1(CN2CCN(C(Cn3ncc(C(=O)OC)c3)=O)C3C2C3)cccc2scnc12 C(=O)(CC1=NNC(=O)C1)NC12C(NC(C3(C(=O)OC)CCCCC3)=O)CC(CC1)C2 c1(COC)cc(C(C(=O)NC2(CSC)CCC2)N(C)CCF)cc([N+](=O)[O-])c1 c12nc(C)c(o1)C(=O)NC2.c1(CC(=O)OC)c(C)cnn1C.C12CC1CNCC2 c1(CN(C23CCCC2OCC3)C)ccc([N+](=O)[O-])cc1Cl c1(Cn2cc(C3CN(C(c4c(CC)cncc4)=O)C3)nn2)scc2c1OCCO2 Cc1cc(C(F)(F)F)ccc1C(=O)NCCOCCOCCNC(N)=O c1(COC)nc(N)cc(Cl)n1.N12CCC(C1)CCN(C)C(=O)OCC2.C(C)(C)(C)OC c1(CNC(C(N2C(C=C)CCCC2)=O)=O)cc(C)c(Br)cn1 N1(C(CC(CNC(C=CCN(C)CC)=O)O)=O)C2CCC1CC(=O)NC2 Cc1cc(C(=O)NCC2(O)CCCN(C(=O)Cc3ccsc3)C2)c2occc2c1 C12(C(=O)NCC3(NC(C4(O)CCSC4)=O)CCCC3)CCC(O1)c1ccccc12 C(=O)(NNC(=O)C1CCCCN1CC1CCCCC1)C1C(OCC)C1 c1(OC)ccc(Br)c(C(=O)NCc2cc3n(n2)CCO3)c1F C(=O)(C(C(C)(C)C)NC(c1cnns1)=O)NC(C)CC1CCCC1 C(=O)(CC(C)C(=O)N1C2CCC1C(C(=O)Nc1c(C)c(C)nn1C)C2)OCC N1(C(CCSCCC)=O)CCC(CNC(=O)CCNS(C)(=O)=O)(OC)C1 C1(C(=O)N(C2CC2)CC2(CC(N3CCCC3c3nc[nH]n3)=O)CC2)C2CCCCC12 Cc1cc(C(N2CC3CC3(C(=O)Nc3cc(Br)nc(Br)c3)C2)=O)cc(C#N)c1 N1(C(C(C)NC(=O)C2CC2)=O)CC(NC(=O)C(C)(O)C(C)C)CCC1C C(=O)(CS(=O)(=O)C(C)(C)C)NCC1C(NC(CCc2ccc(OC)c(F)c2)=O)C1 N1(C(CCc2cn(C)nc2)=O)CCC(O)C1C(=O)NC1(C)CCCC1C C=Cn1nncc1C(=O)N(C1CCN(C(c2ccc(C(C)=O)cn2)=O)CC1)C c1(NC(C2CC2C(=O)Nc2cc(O)ccn2)=O)cc(Br)ncc1[N+](=O)[O-] N1(C(c2cnc(CC)o2)=O)CC2CN(C(=O)C(C3CC3)SC)CC2(C)C1 C(CC(O)CNC(C1CNC(=O)N1)=O)NC(C(c1ccncc1)C)=O c1(CN(C)C(C2(C(=O)O)CCCOC2)=O)coc2c(F)cc(F)cc12 C=C(C)C1CN(C(C2CCCN(C(C3(F)CCCC3)=O)CC2)=O)CCO1 C1(O)(CCNC(C2(CC#C)CCOC2)=O)CCCN(C(c2nc(Cl)sc2Cl)=O)C1 C(=O)(C1=CCCS1)NCC1C(C(=O)NCCNC(=O)OC)CCC1 N1(C(CNC(C(CC)C)=O)=O)CC2(CCCN(C(c3n[nH]cc3F)=O)C2)C1 Cc1cc(C(=O)NC(CNC(=O)C(C2CCCCCC2)F)C2CC2)ncc1F c1(OC)ccc(Cl)c(C(=O)NC2CCCN(C(=O)Cc3ccc(Br)cc3)CC2)c1 Cc1cc(Br)c(NC(C2CC3(C2)CN(C(=O)C(C)c2cccs2)C3)=O)cc1C C(=O)(C(C1=Cc2ccccc2OC1)N1CCCCc2ccc(Cl)cc21)NCC(C)C N1(C(C2(CNC(Cc3nc(C)oc3)=O)CC2)=O)CCn2cnnc2C1 c1(NC(=O)CC2(C(N3CCCC3)=O)CC2)cccc2cccc(Cl)c12 N1(C(c2c[nH]c(=NC)s2)=O)CC(NC(c2ccc(F)c(C)c2N)=O)CC(C)(C)C1 C1(NC(C(CCOC)C)=O)CN(C(=O)CCCc2nc(C(C)C)no2)CCC1C c1(CCCC)cc(C(=O)NCC2CCCN2C(=O)CN(C)C2CC2)c(C)o1 N1(C(c2cnns2)=O)CC=CC1Cn1cc(-c2c[nH]nc2F)nn1 C(=O)(C1=C(C)CCCC1)N1CCOCC(NC(C(CC=CC)C)=O)C1 n1(CC)nc(C(=O)NC(C)C(C)NC(=O)C=Cc2cn(C)nn2)c2c1CCOC2 C1(CNC(c2ccc(OC)s2)=O)CC2(CCOCC2)CN1C(=O)C(O)P(C)(C)=O c1(N(C)CCN)ccc2c(ccn2C(F)F)c1.Cc1nc(CC=O)co1 c1(C(N2CCC(NC(c3c(C)cn(C)c3)=O)C(CO)C2)=O)cccn2nccc12 c1(C(N2CC=CC(NC(C3C=CC=CC=C3)=O)C2)=O)cc(C2CC2)nc(Cl)c1 C1(C(=O)NCC(c2cnn(C)c2)C)N(C(c2ncccc2O)=O)CCCC1(C)C c1(N(C)C)cnc(CNC(=O)C(N2CCOC(C3(C4CCCC4)CC3)C2)=O)nc1 C1(C(N2CCC(C)(CNC(c3cc(Cl)c[nH]3)=O)C2)=O)CCOC2(CCCC2)C1 C1(Cl)(C(N2CC(CC=C)(C(N3CCC3CC)=O)C2)=O)CCCCC1 c1(S)cc(F)ccc1F.O=CC(F)NCCCNC(C1C(C(=O)NCCOC)C1)=O c1(C(=O)NC2C(NC(C=C(C)C(F)(F)F)=O)CCCCC2)cnc(C)c(C#N)c1 C(=O)(CCCS(C)(=O)=O)NCC1C(NC(CCn2ncc(C)c2)=O)CC1 N1(C(C2(OC)CCS(=O)(=O)C2)=O)CC2CCCC(C1)N2C(C1CCC(C)(C)O1)=O c1(C(=O)NC(C2CN(C(=O)C(c3ccccc3)N(C)C)C2)C)[nH]nnc1C1CC1 C1(NC(C(CC=C)C)=O)CC2CC1N(C(c1c[nH]nc1-c1ccsc1)=O)C2 N1(C(C(=O)NCc2c(Br)ccc(C)n2)=O)CCC2(CC(C(F)F)=NO2)C1 c1(CC)ncsc1C(=O)NCC1CCCC1NC(=O)C(Cc1ccccc1)C1CC1 CC(CCCNC(c1cnc(Cl)[nH]1)=O)NC(C1CN(C(=O)C2CC2)C1)=O C(CC1CCC1)(C(=O)NC1CCC(NC(C2CC(F)(F)C2)=O)C1)OC C1(n2cc(-c3c(C)cn(C)n3)nn2)CCCN(C(C2CCC2)=O)CC1 Cc1cc(=O)c(C(N2CC=CC2CNC(=O)C(n2cc(Cl)cn2)C)=O)cn1C C1(C(N2CCC(CCCCNC(CC(CC)C)=O)CC2)=O)CC2(C1)CS(=O)(=O)C2 C(CC(C(=O)NC1CN(C(C)=O)C1)NC(c1ccc(OC(C)C)cn1)=O)OC Cc1cc(N)c(C(=O)NCC(F)CNC(C2CCC3CC2CO3)=O)c(F)c1 C12CCN(C1)C(=O)C(C1CCC1)CNC(=O)C2.CC(C)C(O)C1CCC1 c1(N2CC(C(=O)Nc3cccc(F)c3I)C(F)(F)CC2)ncnn2cc(Br)cc12 CN1CC(O)CCC1C(N1CC(CC(=O)NCc2nccs2)C2(CC2)C1)=O c1(CC(=O)N(CCC(C)NC(=O)CSCC(F)(F)F)C)cc[nH]c(=N)c1 C1(Nc2c(C(=O)NCC(C(C)C)NC(CC)=O)ccnc2)CCC2(CC1)CC2 C(=O)(CCCCCCS(N)(=O)=O)N1CC(N(C)C(C2(C3CCC3)CC2(F)F)=O)C1 C1(C(N2CCCC(CN(C(=O)C(N)=O)C)C2)=O)CCC2(COC2)OC1 C1(CC(C)NC(=O)C2CC2)CC2CCC(C1)N2C(=O)C=Cc1ccccc1 c1(CC)c(C(=O)NC2CCC(NC(=O)C(C)P(C)(C)=O)C2)[nH]c2ccccc12 C1(C(=O)NCCCc2c(C)n[nH]c2)CC(O)CN(C(C2(C3(O)CCC3)CC2)=O)C1 C(=O)(C(CNC(=O)CC(C)(C)N(C)C)C(C)C)NCC(C)(C)OC N1(C(c2c(CC)ocn2)=O)CCCC(CN(C(=O)CCOc2ccccc2)C)C1 C1(C(=O)OC)CS(=O)(=O)CN(C(C2CC=CC(C(=O)CCO)C2)=O)C1 C(=O)(C1COc2ccc(F)cc21)NCCCN(C(c1[nH]cc(OC)c(=O)c1)=O)C c1(OCC)cc(C(=O)NCC2(O)CN(C(=O)C(F)=C(C)C)C2)oc(=O)c1 C#Cc1ccc(OCC(=O)NCC2C3CN(C(=O)C(C)(O)COC)CC23)cc1 Nc1cccn(CC(=O)NC2CC(NC(C3(CO)CCCCC3)=O)C(O)C2)c1=O c1(C(=O)NC2CN(C(Cc3cc(C(C)C)no3)=O)CC2F)ccc(S(C)(=O)=O)s1 C1(C(N2CCCN(CCNC(c3cc(Cl)ns3)=O)CC2)=O)CCC2(CCC2)O1 c1(CC)nc(-n2cccc2)sc1C(=O)NCC(O)CNC(c1scnc1CC)=O CC(=C(Br)Br)NC(CCCl)c1nnnn1CSc1ccccc1 C(=O)(C1=CCC(C)CC1)N1CCC(CCOC)(NC(=O)C=CC2CCOC2)CC1 Cc1nc(C(N2CCC3(CCCN3C(C3CCCN3C)=O)C2)=O)c2n1CCCC2 c1(OCC)ccc2[nH]c(C(=O)O)cc2n1.c12ccc(cc1)CNC(=O)C(=O)NC2 C1(C(=O)NC2(C(N(C3CC3(C)C)C)=O)CCC2)CCC(=O)C1 CCCC(C)(C)C(=O)N1CC(C2CN(C(C3(C)CC=CC3)=O)CC(C)O2)C1 c1(NC(C(=O)OC)(CSC)OC)ccnc2nc(C)nn12 NC(=O)CCC(=O)NCC(CNC(c1cccc(OCC(F)(F)F)n1)=O)CO N1(C(CC2CCC(C)O2)=O)CCOC2(C1)CN(C(c1cn3c(n1)SCC3)=O)C2 C#CC1(O)CCN(CC(=O)NC(C)C(C)NC(c2ncoc2Br)=O)CC1 N1(C(C(C)=C2CC2)=O)CC2CCCC(CNC(=O)C3=CCCCC3C)(C2)C1 CC1=C(C(=O)N2CCC2)CCC1.C(=O)(CCC(F)F)NC(C1CC(OC)C1)(C)C c1(C(=O)NCCC2(NC(C(C)OCC(C)C)=O)CCC2)c(F)ccc(Cl)c1N C1(C(N(CCCCNC(C2CN(C)C(=O)N2)=O)C)=O)CCc2c(cnn2C)C1 CCC(C)(C)C(=O)NCCCN(C(=O)CN1C(C)CCC1C)C c1(C(N(C(C)C(=O)NC)CC)=O)c[nH]c(C=O)c1.C1(CC2CC2)C(=O)N1 N(C(=NCc1cnnn1C)N1CCN(Cc2cc(C)on2)CC1)C(CC)C(F)F C1(O)(CN(C(C=C(COC)C)=O)C)CN(C(c2csc(C(C)C)n2)=O)C1 N1(CCCC)C(=O)NC(c2cnc(C(=O)NC)s2)C(C(=O)OC)=C1C(=O)OC C(=O)(C(C)CC(C)(C)C)NCC(C)(C)NC(CC(C)c1cnn(C)c1)=O C#CCCCC(C)C(=O)NC1CC2CC1N(C(=O)Cc1ccc(C)nc1)C2 O=C(CC1=CCOCC1)NC1CCC(C(=O)NC2CN(CC(F)F)C2)C1 N1(C(CC=CCC)=O)CCC(C2CC2)C1CNC(=O)CCc1cnc(C)o1 CCCC(CCC)C(=O)N1CCOC(C(C)NC(c2ccc(N)c(Cl)c2)=O)C1 O(NC(=O)C(C)(CSC)NC(=O)CC(C)C1CC1)CCCC.OC N1(C(C2C(CNC(Cc3cn(CC)nc3)=O)CC2)=O)CCC2C(O)CC12 C=C(C(=O)NC1CCCC1CNC(c1cccc(Cl)c1F)=O)C(F)(F)F C1(CN(C(C2C(OC)CC2)=O)C)CC(F)CN1C(c1cnc(Br)s1)=O CC(C)C(C(=O)N(C)Cc1cncs1)NC(=O)C(C)Cn1ccnc1 N1(C(C=CC)=O)CC(C=C)(CC(=O)NC(CC)C(=O)NC(C)(C)C)C1 C(=O)(CC(O)C(Cl)(Cl)Cl)NCCCC(C)(C)NC(C(CC)COC)=O C1(C(=O)NCC#C)CC(C)(C)CCN1C(=O)C(N1CCOCC1)C C(N=c1cc(C)nc(Cl)[nH]1)C1CCC(NC(c2c(OC)cccc2F)=O)C1 C(CCC(C)C(=O)NCC1CN(C(=O)CC2CC(N(C)C(C)C)C2)C1)OC Cc1ccc2sc(C(=O)NC3CC4CC3N(C(C3(C)COC(=O)C3)=O)C4)cc2c1 c1(CCC)noc(CCCC(=O)NC(C2CCN(C(=O)CC3CC(F)C3)C2)C)n1 C1(NC(CC(C)(C)O)=O)CCCC12CCN(C(=O)C=CC1CCCCC1)C2 c1(-c2cn(CC(=O)NCC3N(CC(CCC)C)CC3)nn2)ccc(F)nc1 C(=O)(C1=CCCOC1)NCCCCCCNC(C(c1ccn(C)n1)(C)C)=O C(C(=O)N1CC(CCNC(=O)CC(O)C2CCC2)C1)(C(C)C)NC(COC)=O C(CCC(C(=O)NC1(C2CC2)CCCC1)OC)OC.C1COCCN1CCO c1(N(C)C)ccc(C(N2CCC2CN(C(=O)CCCC(F)F)C2CC2)=O)cc1F C(=O)(C1=CCC(C)CC1)NC1(c2nc(C)[nH]n2)CC1.N12CC(O)CC1C2=O c1(C(N2CC(CN(c3ncc(C4CC4)s3)C)OCC2)=O)c(N(C)C)cccc1C Cc1ccccc1-n1cc(C(N2CCC(N(C)C(c3ccc(C)s3)=O)C2)C)cn1 CCC(CCC(=O)N(CC(O)(CC)CC)C)NC(c1ccc(O)cn1)=O N1(C(C(c2nc(C)sc2)=O)=O)CCC(C(F)(F)F)C(NC(c2cocn2)=O)C1 CC#CCCC(=O)NCC(CNC(=O)COC1(C)CCC1)OC c1(CCC)ncoc1C(=O)N(CCCCCNC(=O)C(O)CN1CCCC1)C N1C(=NCc2ccc3nc(O)oc3c2)N2CCC(C2)C1.CC(C)N(C)C C(=O)(CC(CC)CCCC)N1CC2C(CNC(CCCCCC)=O)(C2)C1 C1(C(=O)NCC2C(C)(C)CN(C(C3CC(CF)C3)=O)C2)C2CCC3C(C2)CC13 Cc1cc(C(=O)NNC(=O)c2cc(O)cs2)c(C)n1CCC#N c1(C(=O)NC2CC(NC(c3cncc(O)c3)=O)C2)c(F)c(F)cc(F)c1F N1(C(CSCCOC)=O)CCCC1(C)CNC(C1CCCC12CC2)=O C(=O)(C(CO)N(C)C)N.CCCCCOCCC(=O)NCC(C)(C1CC1)NC(=O)C(C)C c1(OC)ncc(I)cc1CN1CCSCC1C(=O)Nc1ccc(Cl)c(C(N)=O)c1 Cc1cccn2ncc(C(=O)NC3CCCC3c3ccccc3)c12 CC1=CN=C2N=C2C=C(C)N(CC(=O)NOCCCCC(C)C)C(=O)C=N1.C1CS1 C1(CNC(C2CC2c2ccsc2)=O)CC2CCC(C1)N2C(C1C2CCCC12)=O CC1(C(=O)NCCCN(C(c2cscc2C2CC2)=O)C2CC2)CCCC1O CC1(C)CCCN(C(=O)CCn2cccn2)C1C(=O)NCC1=CCCC1 C1(NC(C2(OC)CC(C)C2)=O)CCC2(CCN(C(c3cc(C(C)C)no3)=O)C2)C1 Nc1cc(C(=O)NCC2CCC3(CC3)C2)cc(F)c1 C1(C(=O)NCC2(F)CCN(C(C3C4(CC(OCC)C4)C3)=O)C2)CC(=O)NC(=O)N1 C1(C(=O)OC)N(C(c2ccc(C3CC3)o2)C(=O)NC2CC2)CC12CCCCC2 N(C1CCc2cccnc21)Cc1cn(Cc2c(C(=O)O)[nH]c3c(Br)cccc32)nn1 c1(C(N2CCC(C(=O)Nc3c(C)cnc(F)c3)C2)=O)ccc(Br)c(O)c1Br C1(Sc2c(C(=O)OC)scc2)CCN(N(C)C(C23CCCCC2C3)=O)CC1 C1(OCC)CC2(C1)CC2C(N1CC(O)(C2CCCN2C(c2coc(C)n2)=O)C1)=O C1(NC(C(=Cc2ccco2)C)=O)CN(C(C2CC(C)(C)CN2C)=O)CCC1CO N1(C(c2n(CC)ccc2)=O)CCC2CN(C(=O)C=Cc3ncco3)C2C1 C1(N(C(c2ncn(CC)n2)=O)C)CCC2CN(C(=O)CCCN(C)C(C)C)CC12 N1(C(C=CSC)=O)CC(NC(=O)C(C)N2CCC2)Cc2ccccc21 C1(NC(CC2(C)CC2(Cl)Cl)=O)CCN(C(C2SCCCS2)=O)CCC1CO c1(-c2cc(NC3CNCC3F)ccc2)cccc2c1OCO2 C(=O)(NNc1ccc(Cl)c(C)n1)c1ccc(-n2ccc(C)n2)c(F)c1 c1(C(=O)NCC2C(CC=O)C2)ccc(S(C)(=O)=O)o1.CC(O)C1C(=O)N1.C(N)(=O)O c1(NC(C)=O)c(COC)occc1=O.C1(C(C)N)CCCCN1C(=O)COCCF C(=O)(CC1=NNC(=O)C1)NC(CN(C(C(c1c(C)n[nH]c1C)C)=O)C)C n1(CC(N2CCC(NC(C)=O)CC2)=O)ncc2cc(C3=CCN(C)CC3)cnc12 N1(C(CC(COC)NC(=O)CS(N)(=O)=O)=O)CCC(C)(C2CC2)CC1 Cc1ccc2[nH]c(C(=O)NC3CCC4CC3CN4C(C3CC3C)=O)cc2c1C CCCC(C(O)C(=O)N1CCOCC1C(C)O)NC(C1(C(F)(F)F)CC1)=O c1(CC)ccc(C(C)C(=O)NCC(C)NC(C)C2CC2)cc1 c1(C(=O)NC(CCN(C(CCCC)=O)C)C(C)C)cccc2[nH]cc(Cl)c12 O=[N+]([O-])c1cc(Cl)c(Cl)cc1S(=O)(=O)NCC(F)F.c12ccc(cc1)N(CCO)C2 N12CCOCCC1C2=O.O=C(C#CC1CC1)N1CCC1CC1CC1 C1(CCN(C(COCC#C)=O)C)CCCCN1C(=O)CC1CCC(C)CO1 C(=O)(C1CCc2ccccc21)NC1C(C(N(C(C)(C)C)CC2(O)CC2)=O)C1 c1(C(=O)OC)cccnc1NC(=O)NC1CCNC(=O)C1 N1(C(COCCC=C)=O)CCCC(C)(C(=O)NCCNc2cnncc2C)C1 C1(NC(C(C(CC)O)C)=O)CCCC12CN(c1nnc(CC(C)C)s1)C2 N(C(=NCCN(C)C1CC1)NCC1CC2CCC1O2)CC(C=C)(C)C C1(N(C)C(C2CC(F)(F)C2)=O)CCCN(C(c2cc[nH]n2)=O)C1 N1(C(C2(CF)CCN(C(c3cc(C)cc(C)c3)=O)C2)=O)CC2CCCCC2C1C C1(NC(C(=O)NCCOCCCC)=O)CCN(C(c2ccccn2)=O)C(C2CC2)C1 N#Cc1ccc(CN2CC(C(=O)NCC(=O)Cc3cccs3)CC(F)C2)c(Br)c1 c1ccc(C=O)cn1.C(CC(=O)N(C1CC(OCC)C1)CC)SCC c1(C(=O)OCC)cc(NC(C2CC(NC(c3c[nH]c(=NC)o3)=O)C2)=O)ccc1I c1(C(N2CCCC(F)(CNC(=O)CCOCC3CC3)C2)=O)c(F)ccc(F)c1F n1(CC(=O)OCC)cc(Cl)c(C(=O)NCC(C2CC2)NC(=O)C(O)C2CCCC2)n1 C1(NC(c2c(CC)nco2)=O)CC2CCC1CC2NC(=O)CCc1ncnn1C C1(CC=C)(NC(=O)C(c2ccccc2C)C)CCN(C(c2cc[nH]n2)=O)C1 O=C(C#CC1CCOCC1)NCC12CCC1CCN2C(c1ccc([N+](=O)[O-])o1)=O c1(C(=O)NC23CC(CNC(C(C)CF)=O)(C2)OC3C)cccn2nccc12 c1(COC)ccc(C(=O)NC2CCC(NC(C3CCNC(=O)C3)=O)C2)cc1F c1(C(=O)NC)ccc(C(=O)N(CC(O)CN(C)C(c2nnc(C)s2)=O)C)cn1 c1(C(=O)NC2C3(CC(NC(C(C(CC)(C)C)O)=O)C3)C2)c(N)sc2c1CCSC2 C1(NC(C(CC)n2ccnc2)=O)CCC(C)N(C(c2ccc(Br)cc2)=O)C1 C1(C(N2C(C(C)NC(C3(C(C)C)CC3)=O)CCC2)=O)CCCCN1C N1(C(CC(CC2CC2)NC(Cc2cc(C)on2)=O)=O)C2CCCC1CN(C)C2 C1(C(=O)OCC)(C(=O)NC(C(C)N(C(=O)Cc2cn[nH]c2)CC)C)CCC1 N1(C(C2N=C(C)SC2)=O)CCC2CCN(C(=O)CCC(=O)C(C)(C)C)CC2C1 C1(C(N2CC(OCCOC)C2)=O)CC(C)N1C(C1CC2CC2C1)=O C1(NC(CC2(C)CCOC2)=O)CC(CO)N(C(C2COCC2C(N)=O)=O)C1 C(=O)(CC1(O)CCOc2ccccc21)NCC(C)NC(CCCC#C)=O C1(CCN(C)C(c2ccnc(O)c2)=O)CCCCN1C(=O)CC1CCC1(F)F C=CCC(C)(C)C(=O)N1CC=C(CNC(=O)C(C)(Cc2ccccc2)CC)CC1 C1(NC(=O)CC2(CO)CC2)CC2(CCCN(C(c3csc(Cl)c3)=O)C2)C1 C1(NC(C(=Cc2cnc[nH]2)C)=O)CC(C)N(C(=O)CN(C)C)C1 Nc1ccc(C(N2CCCC(c3cc(O)n[nH]3)C2)=O)c(F)c1 C(=O)(C(O)CCCC)NCC1CN(C(c2ccc(CCCCCC)o2)=O)CC1C c1(NCc2c(C)ccc(SCC)c2)cn2c(C)cc(C)nc2n1 C=CCC(C)C(=O)NCc1ccc(CNC(c2cc(C(F)(F)F)ncn2)=O)cc1 C1(C(=O)NC2CN(C(=O)C3=CCSC3)CC23CC3)CC(c2ccc(F)cc2)=NO1 C(C)(CCN=c1ncc(C(F)F)c[nH]1)NC(C1CCC(=C)CC1)=O C=C(C)C1CN(c2cc(NCc3nc(=N)s[nH]3)nc(C)n2)CCO1 C1(CN(C=O)Cc2cc(Br)ccc2OCCO)CN2CCCCC2CO1 c1(C(=O)NCCC(C)NC(Cc2ccc(CCC)cc2)=O)cnn2c1N(C)CC2 N1(C(C(C)O)=O)CC2CC1C2NC(c1cccc(C2CC2)c1)=O c1(CN2C(CC(=O)NCC3(CC(=O)O)CCC3)COCC2)ccc(Cl)cc1O CCCCC(C(=O)N1CCCC(F)(CO)C1)NC(=O)C=Cc1nccs1 C(=O)(C1SCCc2ccccc21)NC1CN(c2nc(CC)c(C)s2)C(C)CC1 C(=O)(C1=CC2(CN(C(C3C4CCCCCC34)=O)C2)OC1)NC1CCC(C)(C)CC1 c1(C(=O)NCC2CC3CCC2N3C(C2CC2c2ccco2)=O)cc2cccnn2c1 C1(C(N(CC(CN(C(=O)CC(O)C2CC2)C)O)C)=O)CS(=O)(=O)CC(=O)N1 C1(C(=O)NCC(CN(C)C(C23CCC2C3)=O)O)CCOCC1 c1(C(=O)OCc2nc(CC)oc2)ccc([N+](=O)[O-])cc1Cl C=C=CC(C)C(=O)NC(c1nocc1C(=O)NCCc1cc(CC)no1)C C1(C(=O)NCC(CC)(C)Cl)CC(O)CN1C(c1nccnc1C)=O O=C(CCCc1ccco1)NC(C(=O)NCC1(C(=O)O)CCCC1)c1ccoc1 N1(C(c2n(C(C)C)ccc2)=O)CCC2(NC(=O)CCOC3CC(F)(F)C3)CC2C1 c1(C(CC)(C)C)n[nH]c(=NCC2CC(C)N(C(=O)CN(C)C)C2)o1 N1(C(C(c2ccccc2)OC(C)=O)=O)CCCN(C(c2cc(C)n(C)c2)=O)CC1 C(=O)(CCCC(C)C)NC(C(CCc1ccccc1)NC(CCC)=O)C C(CCC(N)=O)(C(=O)N1CCC(C)(Cc2cnn(C)c2)C1)NC(=O)OC(C)(C)C Cc1cccc(O)c1C(=O)NCCc1ccc(CNC(C2(CO)CCC2)=O)cc1 c1(CC(=O)NCC(C2CC(F)C2)NC(C)=O)ccc(N2CCOCC2)cc1F C1(C(=O)NC2CC(O)(CNC(c3ccc(F)s3)=O)C2)CCc2nnc(O)cc2C1 C12(NC(C3(OCC)CCCC3)=O)CC1CN(C(C1CCC(=O)N1C)=O)C2 c1(C(N2C(CNC(C(F)=CC)=O)CC(OC)C2)=O)ccnc2c1ncn2C c1(C(N2CCC(CNC(=O)COc3ccc(F)nc3)C2)=O)c(Cl)cncc1Cl C(C=O)(C(C)C)SCC.N12CCC(CC)(C1)C2=O.C1(NC)CN(C)C1 C1(CC(=O)NCC(CC)NC(=O)C(O)Cc2cccc(Cl)c2)CC2(CCC2)C1 c1(C(=O)NC2CN(C(C3(C)C(C)CCCC3)=O)C2)csc2c1CCC(C)(C)C2 c1(C(N2C(C)CC(NC(c3cnc(S)nc3)=O)CC2)=O)nccc2c1NCCC2 C1(C(=O)O)(NC(C2CC2C2CCCO2)=O)CCS(=O)(=O)CC1 c1(CNC(C(CC)NC(=O)C=CC2CCC2)=O)cncc(C)c1 c1(C(=O)NC2CN(C(c3cc(C)c(C)[nH]3)=O)C(C)CC2)n[nH]c2c1NCCC2 c1(NC(CCC2N(C(c3c(C)cco3)=O)CCC2)=O)cc(C(N)=O)ccn1 N1(C(CC(CNC(C(C=C)(C)C)=O)C2CCC2)=O)CC2(CNC(=O)OC2)C1 c1(C(=O)NCC(C)N(C(C(CCC)OCC)=O)C)c(OCC2CC2)cccc1Cl C(C(=O)Nc1ccc(F)cc1)(C(C)C)N1C(C=C)CC1 C1(C(N(CC(C)SC)C)=O)CN(C(=O)CC2C=NN(C)C2=O)CC(C)(C)C1.C(C)(=O)O CC1CN(Cc2coc(C3CCOCC3)n2)CCN1C(=O)C(=O)NCC(F)F CS(=O)(=O)c1ccccc1CN1CCCC(C(=O)NCc2c(Cl)cccc2Cl)C1 c1(OC)cc(F)c(F)cc1C(N1CC2CC1CN2C(c1cc(C#N)c[nH]1)=O)=O Cc1cccc2c(C(N3CC(NC(c4cc(=N)[nH]c(Cl)n4)=O)C(C)C3)=O)n[nH]c12 N1(C(C=CC(C)C)=O)CCN(C)CC1CNC(c1[nH]c(=N)sc1C(F)(F)F)=O N1(C(C(CC)(C)O)=O)CCC(C)(Nc2ncc(C)cn2)CC1 Cc1cc(CC(=O)NCC2(C)CCN(C(C3C4(CC4)C34CC4)=O)C2)ccc1F Cc1cc(C)nc(N2CCCC(NC(=O)CCn3cccnc3=O)C2)n1 c1(C(=O)NCCN(C(C(C(=O)OC)(C)F)=O)C)ccc(O)c(C)c1C Cc1csc(C(=O)NC(c2ccc(C(N3CC(F)(F)C3)=O)cc2)C)c1C c1(OC)ccc(CC(=O)NCCN(CC(C)O)C(=O)Cc2ccoc2C)cc1F N1(C(C(CCC)CC2CCCC2)=O)CC2(CCN(C(C3(CF)CC3)=O)CC2)C1 CC(C)C(C(=O)NCC1C2CC1N(C(=O)CC(C)C1CCCO1)C2)n1cnnc1 C1(CC(=O)N(CC(=O)NC2CC2)C)C2CN(C(=O)CC(C)(F)F)CC12 Nc1cc(Cl)cc(Cl)c1C(=O)NC1CCC1NC(=O)C=C1CCSCC1 C1(C(C(=O)N(CCCO)CC)C)CCN(CCCn2ccc(SC)n2)C1 c1(CC)nc(C)[nH]c1C(N1CCC(=CCNC(=O)C=C=C(C)C)CC1)=O n1(CC=C)nnnc1C(c1ccoc1C)NC(C)COCC C1(NC(c2c(C)snc2)=O)CC2C(NC(=O)CC3CCCN(C)C3)C2C1 Cc1cnc2c(cnn2CC(=O)NC2CCN(C(=O)CNc3cnn(C)c3)C2)c1 N1(Cc2ncc(C#N)cn2)CCC2(CC(C(=O)N=c3occ(Br)[nH]3)=NO2)C1 N1(C(C2(c3n(C)ccn3)CC2)=O)CCN(C(=O)COC2C3CCCC23)CC1 c1(C(=O)NC2CN(C(=O)CC3CC4CCC3C4)CC2O)c(Br)ccc2cccnc12 c1(CC)oc(C)cc1C(=O)NC(CN(C(C1(C(F)(F)CC)CC1)=O)CC)CC c1(OCC=C)ccc(C(=O)NNC(=O)c2ccc(N(C)C)cc2)cc1[N+](=O)[O-] Cc1nc(CC(N2CCC(O)(CNC(=O)CCCc3nncn3C)C2)=O)c(C)s1 C1(C(=O)NCC2(OC)CN(C(=O)CCOC(C)C)C2)CCCC1P(C)(C)=O C(=O)(C1CCc2c[nH]nc21)NCC(CNC(c1n(C)nc(O)c1)=O)CO CCC(C)(C)C(=O)C(=O)N1CCC(C(=O)NC2CCN(C(C)=O)C2)C1 C#Cc1cccc(CNC(=O)C(C2CCN(C(=O)C(C)n3cncn3)C2)F)c1 CC1(O)CCN(C(C23COC(C2)C(NC(=O)CC(O)CNC)C3)=O)CC1 N1(C(c2c(CC)cno2)=O)CC(NC(=O)COC(F)(F)F)CCC1C C(=O)(C(C(=O)OC(C)(C)C)C(C)C)NCC(C)N(C(c1c(CC)cno1)=O)C Cc1cc(=NC(=O)C(=O)N2CCCCC(N(C)C(c3cc(Cl)cn3C)=O)C2)[nH]o1 c1(C(N2CCC(C3CCC3)C2)C(=O)NCCOCC)cnc2cnccn12 C1(CNC(C(=O)Nc2ccc(CCN)s2)=O)CCCC12CC2 C12(C(=O)NC3CCCN(C(c4c(C)onc4)=O)C3)CC3CC1C2C3(F)F c1(C(=O)NCC(CC)NC(C2CC(F)(CO)C2)=O)cncc(F)n1 S(=O)(=O)(c1cccc(C(=O)NCc2ccc(S(N)(=O)=O)o2)c1)NCCOC N1(C(c2c(C)cc[nH]2)=O)CC2OCC(NC(c3cccn4nccc34)=O)C2C1 C1(C)(CC)C=C(C(=O)N2CCCC(CNC(c3cc(COC)ccc3Cl)=O)C2)C1 CC1=C(C)CC(C)(C(N2CC(CNC(=O)CP(C)(C)=O)C(C)(C)C2)=O)CC1 N1(C(C2CCC(N(C(=O)CN3CCS(=O)CC3)C)C2)=O)CC2(CCN2C)C1 C=C(Cl)CC(C(=O)NCc1nc(C)nn1C)NC(c1cc(C)nnc1C)=O CC(C)C(C(=O)N(CCC(C)NC(C1CC(C2CCC2)C1)=O)C)C(C)C c1(CC)cc(Cl)ccc1C(=O)NC1CCC(CNC(=O)CCC(N)=O)C1 c1(C(N2CCCC(C(C)NC(CC=CCCCCC)=O)C2)=O)ccc(C)c(C)n1 C1(CNC(C(=Cc2ccco2)C)=O)COCCN(C(=O)C(F)CC2CCCC2)C1 Cc1ccc(C(=O)NCC(C)CNC(c2cnccn2)=O)c(F)c1 C=C1Cn2c(C(N3CCCC3CNC(=O)CC(F)(F)CC)=O)nnc2S1 c1(C(N2C(C(C)C)CN(C(=O)CC3CSCCS3)CC2)=O)ccc2nnnn2c1 c1(C(N(C2CCCN(C(C3(CF)CC3)=O)C2)CC)=O)sc(C)cc1Cl N1(C(C=NOC)=O)CCCC2CN(C(C3(C(F)F)CCCO3)=O)CCC12 Cc1cccc2cc(C(=O)NC3CCN(C(=O)CC4CCOC4)C(C)C3)[nH]c12 N1(C(CCc2n(C)cnn2)=O)C2CCC1CN(C(c1cc(C(F)F)n(C)n1)=O)C2 C1(C(=O)NC2(CCCC)CC2)CCCCC1CNC(C1(C)CNC(=O)C1)=O C1(CC(N2CCC(F)(CF)C2)=O)CCCN(C(C2CCCCS2)=O)C1 C#CC1CC2(CC2)CN1C(c1ccnc(CNC(=O)C(C)(C)CC(F)F)c1)=O CC1CC(C(=O)NCCC2CCCN2C(c2cnc(-c3cnccn3)s2)=O)=NO1 N1(C(C(=O)OCC)=O)C2CC1CN(C(c1sc(C)nc1C(C)(C)C)=O)C2 N1(C(CCOCC#C)=O)CCCC(O)(CCNC(=O)CC(C)(O)C=C)C1 c1(C(N2C(CC(N3C(C(N)=O)CCC3)=O)CC2)=O)ccnc2cc[nH]c12 C1(CC(=O)NCCCCC#CC)C2CCC(C2)N1C(c1cc(C)nn1C)=O C1(OC)C(N=c2[nH]c(=NC3CC(SCCO)C3)[nH]c3c2COC3)CC1(C)C C1(CCC)CN(C(C2CCNC2=O)=O)CCN1C(=O)C(C)=CCOCC1CCC1 C1(CCCC)CN(C(=O)C(C)CSC)CCN1C(c1nn(C)cc1C)=O CC1=C(C(=O)N2CCC(NC(c3cc(C)on3)=O)CC(C)(C)C2)C(C)(C)CCC1 C#Cc1cc(F)c(C(=O)NC2CC3(C2)CC3NC(c2cccc(C)n2)=O)c(F)c1 N1(C(C(CSC)O)=O)CCCC2CN(C(=O)CN(C)CCc3ccccc3)CC12 c1(C(N2CCC(CNC(c3cccc(C(C)C)n3)=O)C2)=O)ccc(N)c(F)c1 c1(CCC)ccc(C)c(CN(C(C)CNC(c2cscc2OCC)=O)C)c1 C1(C(=O)NCC(C(=O)OCC)(C)C)C2CCCC2CN1C(=O)CN(C)C(=O)OC C1(CNC(c2[nH]cc(C)c2)=O)CCCCCN1C(=O)CCc1nc(C(C)C)no1 Cc1ccc(C(=O)NCC2(F)CCN(C(=O)C(C3CCCCC3)C)C2)nn1 c1(CSC)cc(C(=O)NC(C)CNC(C23CC4CC2C3C4O)=O)ccc1F Cc1cc(Br)cnc1C(=O)N(C)CC1CCCN1C(=O)C(O)C1CCCC1 C1(OC)CCCN(C(=O)CC(C(C)C)NC(=O)CC=C(C)C)CC1 C1(NC(c2cc(CC)nn2C)=O)CC2CN(C(=O)CC(C)c3ccncc3)CC12 C(=O)(N=c1ccn(C(C)(C)C)[nH]1)C1(C)N(C(COCC(=O)NC)=O)CCC1 CN1CCN(C2CC(CCNC(=O)C(C3(C(=O)OCC)CCC4CC34)Br)C2)CC1 O=C1N(C2CC2)CCCC12CCCN2C(c1cn2cc(F)ccc2n1)=O C(C(CC(F)(F)F)NC(c1ccnn1C1CC1)=O)NC(c1c(C(C)C)[nH]cc1)=O C1(C(N2CCCC(C(=O)NCC3CN(C(=O)NC)C3)C2)=O)(CC)CCNC1=O c1(NCC(CCCCC)O)ncc(C)cc1S(=O)(=O)N1CC2CC2(CO)C1 Cc1cc(C(=O)NC23COCC2CN(C(c2cc[nH]c2)=O)C3)c(C)nc1C c1(C(N2C(CO)CC(NC(CCNS(CC)(=O)=O)=O)C2)=O)cc2ccsc2n1C N1(C(c2c(CC)cc[nH]2)=O)C2CCC(C2)C1CC(=O)NCC1(F)CCC1 CCC(CCCC(=O)NCCCOCC(F)F)NC(=O)C=C1CN2CCC1CC2 c1(C(N2CCC(CNC(C(C)n3cnnn3)=O)C23CC3)=O)cn2ccncc2n1 C(C(C)CC(=O)NCC1(NC(c2cnccn2)=O)CCOC1)OC c1(OC)ccccc1OCOCC(=O)NCC1(NC(=O)C(C)CO)CC1 N1(CC)N=C(C(=O)N2CCCC(C)C2CNC(=O)CCCCC(C)C)CCC1=O c1(NC(C)=O)cccc(Cl)c1C.c1(C2C(=O)N2CCN(CC)CC)cc(Cl)cs1 c1(C(N2CCCC(NC(C(CCC)C)=O)(CO)C2)=O)cc2c(cn1)OCCO2 C12(C(N3CCC(NC(c4c(C)csc4)=O)C(CO)C3)=O)CC(C)(C1)OC2(C)C c1(CC(=O)NCC2C(C)CN(C(=O)C=CCO)C2)noc2cc(Br)ccc12 Cc1cccc(C2(C(=O)NCC(CO)NC(c3cccnn3)=O)CCC2)c1 c1(Cn2cc(C(N3CC(CN)C(O)C3)=O)nn2)nnc2n1CCC2 CONC(=O)CNC(c1coc(CNC(=O)CN2CC3CC3C2)c1)=O c1(C(N(CCC(O)CO)C)=O)ccc(C(C)(C)C)cc1 C(C)(C)(CCC(=O)NCc1ncc(CO)[nH]1)NC(c1c(C)non1)=O c1(-c2nc(N(CC)Cc3occc(=O)c3OC)sc2)ccc2c(c1)CCCC2=O CC1CN(C(=O)Cc2cnco2)CC1CNC(c1ccc(OC(F)(F)F)cn1)=O c1(Cc2cnc(NC(c3c(C)csc3Cl)=O)s2)cc(F)cc(C#N)c1 Cn1c(=O)c(NCc2c[nH]c3nccc(Br)c23)nc2ccccc12 C1(N(C2CCOC2)C(N2CCC(=CCC)C2)=O)CCCC(OC)C1 CC(CCc1ccc(F)cc1)C(=O)NCC1CC1CNC(c1c[nH]c(=N)o1)=O c1(C(=O)NC2(CC)CCCN(C(=O)CCC(C)(F)F)C2)ccc2nc[nH]c2n1 CC1CCCC1(C)CCN1CCN(c2ccc(OCN)cc2)CC1 c1(CN2CC(C(N(CCCC)CCCC)=O)SCC2)cc(C)cc(C)n1 N1(C(C(N2CCOCC2)C)=O)CC(CNC(c2nn(C)cc2N)=O)CC12CCC2 N1(C(C(CSC)O)=O)CC(NC(c2ccc[nH]2)=O)C(CC(C)(C)C)C1 C=CC1CCCCN1C(=O)C(CC=C)NC(=O)C=Cc1ccnn1C N1(C(CC=C)=O)CCC(NC(=O)Cc2ccc(Br)nc2)C2(CCC2)C1 C(=O)(C1=NOC(CNC(c2cn(C)ccc2=O)=O)C1)N1CC(O)(C(=O)OCC)C1 C1(NC(c2nc(CC)[nH]n2)=O)CCC2(CC1)CN(C(c1nc(O)c(C)s1)=O)C2 c1(C(N2CC(S)OCC2)=O)cc(S(=O)(=O)NS(C)(=O)=O)cs1.CO C(=O)(C(C)(C)C(C)C)NCC(CNC(c1nn(C(CC)C)c(C)c1)=O)(C)OC c1(C(N2C(CNC(C(C=C)(C)C)=O)C(C)(C)CC2)=O)ccc2c(c1)CCN(C)C2 c1(CCNC(CCOCCN(C(C(C)n2cnnn2)=O)C)=O)ccccn1 C=CCC(C)(C)CC(=O)NC1CCCC1CNC(=O)COC(C)(C)C N1(Cc2csnn2)CCC(O)CC1.C123CC(C1C2)n1cc(nn1)CNC3=O N1(C(CCC=C=C)=O)CC(CNC(=O)CC2CCC(=O)NC2)C2(CCOCC2)C1 N1(C(CNC(C)=O)=O)CCC2CN(C(=O)COc3ccc(F)c(F)c3)CC2C1 N1(C(C2OCC(C)(C)C2)=O)CC(C(=O)NOCc2cncc(C#N)c2)C2(CCC2)C1 N1(C(C2CCC(C(=O)OC)CC2)=O)CCC(C)C(NC(=O)Cc2nnc(C)s2)C1 CC1CC(NC(C2(C)CC(C)(C)C2)=O)CCN1C(=O)CC=CC(C)(C)C S(=O)(=O)(CC(=O)N(CCC(C(C)C)NC(c1cc(SC)c(C)o1)=O)C)NCC N1(C(CCc2cnc(C)o2)=O)CC(O)CC1CNC(=O)CCN1CCCCC1 N1(C(C(CNC(C2(O)CCOC2)=O)N(C)C)=O)CCn2ncnc2C1 C(=O)(N=c1cc(Br)n(C)[nH]1)C(C(C)(C)NC(CS(Cc1cn(C)nc1)(=O)=O)=O)C Cc1ccc(O)nc1NC(=O)CSCCNC(C1CC(=O)C1(C)C)=O C(=O)(CC1=NNC(=O)C1)NCC1(N2CC(NC(=O)OC(C)(C)C)C2)CCOCC1 S(=O)(=O)(c1ccccc1)N(CC(N1CCC(N(C(=O)C2=CCC2)CC)C1)=O)CC N1(C(C(CCCOC)C)=O)CCCN(C(=O)C(F)(F)CN2CCCC2)CC1C N1(C(c2c(CCC)occ2)=O)CCC(C2(NC(c3cncc(CC)c3)=O)CC2)C1 C(=O)(CCCCCC(C)C)N1CCCC(NC(c2n(CC)nc(C)c2)=O)CC1 Cc1nc2ccccn2c1C(=O)N(C)CC1(CNC(=O)C(C)C(C)C)CC1 CN1N=C(C(=O)NC2CCC(C(=O)NCC(=O)N3CCCO3)C2)CCC1=O c1(OC)cccc(CCC(=O)NCCSCC2CNCCO2)c1OC(C)C(=O)O c1(C(=O)NC(C2CN(C(C3(c4ccccc4)CC3)=O)C2)C)ccc(C(C)(C)C)[nH]1 n1(CC)nc(C)c(C(N2CC(O)(CN(C(=O)CC3(C#N)CC3)C)C2)=O)c1Cl C(=O)(CCCc1ccsc1)NCCC1(C(N(C)CC2CCOC2)=O)CCC1 CCCCCCC(C)CNC(=O)C(CC(C)C)N1CCCCC1=O C1(CCNC(=O)Cc2cnccn2)COCCN1C(=O)Cc1cncs1 C1(CC)CCCN(C(c2ccnn2C)C(=O)NCc2ccco2)CC1 n1(CC)nc(C2CC2)cc1C(=O)N(CCNC(C)=O)CCOC.C1(C)CCCCO1 C1(C(=O)NC2CN(C(C3CCC(C)CC3)=O)CC2O)CCCC2(CC2)C1 c1(C(N(CC(O)CN(C)C(c2ccc(Cl)o2)=O)C)=O)csc(=O)[nH]1 C1(C(F)(F)F)(OC)CC(C(N2CC(O)(CN(C(=O)Cc3nnc(O)s3)C)C2)=O)C1 CON(CCO)C(=O)COC1CN(C(=O)C=C(C2CC2)C2CC2)C1 C(CCCC(CO)NC(C12CCC1CC2)=O)NC(C1CCN(C)CC1)=O c1(C(N2CC(O)(CNC(C3CCn4cncc4C3)=O)C2)=O)ccc(F)c(F)c1F N1(C(CC)=O)CCN(C(=O)C(C(C)C)NC(=O)C2CC2)C2CCC12 c1(C(C)=O)ccc(SC(C)C(=O)NCc2ccc(Cl)cn2)cc1 C#Cc1cn(C)nc1C(N1CCC(CCC(N2CC(F)(COC(C)=O)C2)=O)C1)=O C1(N2CCN(C(COCCCC)=O)CC2)CCN(CC(C)OCCCC)CC1O C(=O)(C1(C)CCCc2ccccc21)NCC(CC)(C)NC(=O)C#CC(C)(C)O C1(NC(C2CC3CCC3C2)=O)CCN(C(=O)CC2CCC2(F)F)CC1 c1(CNC(C)=O)cccn(CC)c1=O.Cc1ccsc1CC(=O)NOCCCO CC(C)(C#N)CCCC(=O)N1CCC(NC(=O)C=C(Br)Br)C1 Cc1ccn(C(C)(C)C(=O)NCC2(F)CC(NC(=O)C(N3CCNC3=O)C)C2)n1 CCC(CC)C(C)C(=O)NCc1ncoc1CCNC(c1cnc2sccn12)=O c1(C(=O)NCc2c(CCNC(C(CC)OC)=O)ocn2)nnc(O)cc1O C1(NC(C(c2cncnc2)C)=O)CCCC(C(=O)NC2(C(C)O)CC2)C1 c1(CC2CCOC2)nnc(C2CC2)n1-c1cccs1.O=CCCNC(=O)CCF N1(C(C2C(OCC)C2)=O)CCC(C2CCCN(C(=O)CC(C)=C(C)C)CC2)CC1 c1(C(=O)NCC=C)ccc(-c2ccnc(N3CCN(C)CC3)c2)c(C(F)(F)F)c1 CC1(C)CCC(NC(c2ccc(O)nc2)=O)c2ccoc21 N1(C(CCC2(C)CC2)=O)CCC(CNC(=O)Cc2nc([N+](=O)[O-])n[nH]2)C12CCC2 N1(C(c2c(OC)ccs2)=O)CCC(O)C(C(=O)OC(C)(C)C)C1.N12CC(F)(C1)C2=O c1(C(=O)NC2N(Cc3n[nH]c(C)c3C)CCC2)cc(Cl)c([N+](=O)[O-])[nH]1 c1(C(N2C(CNC(c3c(OC)n[nH]c3)=O)C=CC2)=O)ccc(C)c(CO)c1 c1(NC(CC2N(C(c3nc(C(C)C)sc3)=O)CCC2)=O)ncc(Cl)nc1Br C1(COC)(NC(c2ccnn2CC(C)C)=O)CCCN(C(=O)C(C)(F)F)C1 CCCCCC(O)CC(=O)NC(C)CCCNC(c1cc(F)cc(Cl)c1)=O c1(C(N2CC(NC(c3cncs3)=O)CC3(C2)CC3)=O)cc(F)c(F)c(O)c1F C1(CNC(=O)C=Cc2ccco2)CC2CCC(C1)N2C(=O)CCC(F)F c1(C(N(C(CNC(C2(CC#C)CCOC2)=O)C2CC2)C)=O)cc2nnn(C)c2s1 C1(C)(C(=O)NCCCOCCOCCNC(c2nc(CC)sc2)=O)CCCCC1C C1(C2CC2)(NC(CC(=C)Br)=O)CCN(C(=O)Cc2ccc(Cl)cc2)C1 c1(C(N(c2c(OCC(C)=O)cccc2)C)=O)ncn2c1CCCC2 Cc1nocc1NC(=O)CC1CCN(C(C2CC2(C)C(F)F)=O)C1 c1(C(=O)NC2CC3CCC2N3C(=O)CN2CSCCSC2)cc2cccnn2n1 c1(CNC(C2CN(C3CN(C(CC)=O)C3)C(=O)C2)=O)csc2cncn12 Cn1nc2c(c1C(=O)NCC(C)(C1CC1)NC(=O)COC1CCCC1)CSCC2 C(=O)(C1=CCCOC1)NC(CN1CCN(C(C2C(OCC)C2)=O)CC1)(C)C C1(CCC)CN(C(c2ccc(Cl)o2)=O)CCN1C(=O)CCC1(C#N)CCC1 N1(c2cc(OC)ncn2)CCC2CN(C(c3c(F)ccc(C)c3Br)=O)CCC2C1 N1(C(CNS(C)(=O)=O)=O)CCC2(COC(CNC(=O)CN3CC4CCC3C4)C2)C1 C1(NC(C(c2ccccc2)NC(N)=O)=O)CCOCC1NC(=O)CCSC1CC1 c1(CNC(C2CC(CN(C)C)OCC2)=O)cn(CC2CC2)c(=O)nc1O C1(NC(C(C)NS(CCC)(=O)=O)=O)C2CCN(C(=O)CNC(=O)OCC)C2C1(C)C Cc1sc(C(N2CCCC2C(C)NC(=O)CC(C)F)=O)nc1O c1(CC(N2CCN(C(C(CC)F)=O)C(C3CC3)C2)=O)cccc2nonc12 N1(C2CC(OC(c3sccc3Cl)=O)C2)C(=O)NC2(CCc3ccccc3C2)C1=O c1(C(=O)NC(C(=O)NC(c2n(CC)ncc2)C)CC2CC2)cccc2[nH]ccc12 C1(C(=O)NCCCCCn2cc(-c3c(C)cncn3)nn2)CC(=O)NC1(C)C C1(C(=O)NCC2(CC(C)C)CC2)CCC(C)(C)N(C(C2CCCN2C=O)=O)C1 CCC(C)C(C(=O)N1CCCC1)NC(=O)Cn1nnc(=N)[nH]1 c1(C(=O)NCCC2CN(C(=O)C(F)C3CCCC3)C2)ccc(OC(F)(F)F)nc1 N1(C(c2cc(C)on2)=O)CCCC12CCCN(C(c1cc(Cl)cn1C)=O)C2 C(c1c(Cl)cccc1Cl)=CC(=O)NCC(C)N(C)C(c1ccc2ncoc2c1)=O CCC(C(=O)N1CCC(C(C)NC(c2cccn2C2CCCC2)=O)C1)OC C1(CCC(=O)NCC2C(C(=O)OC)C2)CCCN(C(=O)CC2CC2CO)C1 C1(CC#C)(C(=O)N(C)Cc2cnn(C)c2)CCN(C(c2cc(Cl)no2)=O)C1 C(CCCCN(C)C(c1ccn(CC)n1)=O)NC(C=CC(=O)OCC)=O CC1=C(C)CC(C(=O)NC(C2CCCN2C(c2nn(C)c(C)c2Cl)=O)(C)C)CC1 C1(NC(c2cc(C(F)(F)F)ncc2Br)c2n(C)nnn2)CCCC12CCOCC2 n1(CC)nc(C)c(C(=O)Nn2cnnc2)c1C c1(Nc2nc(C3C(C)C3)nc(N3CCCC(F)(F)C3)c2)cc(O)ccc1Cl c1(CC)ccccc1C(=O)NCCC1(NC(c2ccccc2OC)=O)CC1 CCC(CC(=O)N(C)CC1(O)CCN(C(=O)CC2(C#N)CCCCC2)C1)C(C)C C1(S(C)(=O)=O)(C(N2C3CC(CNC(C(C(C)O)C)=O)C2CC3)=O)CCOCC1 C1(C(N(CCNC(c2cc(COC)on2)=O)CCOCCO)=O)C2COCC12 N1(C(c2c(C)cnn2C)=O)CCCN(C(C2CC2C)=O)C(c2ccccc2)C1 c1(C(N(C2CCN(C(=O)C(C)CO)CC2)CC)=O)noc2ccc(Cl)cc12 N1(C(C#CC(C)C)=O)CC=C(C(C)(C)C(=O)N(CCC(=O)NC2CC2)C)C1 c1(C(=O)NCC2CCN(C(CNC(CNC(C)=O)=O)=O)C2)cc(Cl)c(F)c(Cl)c1 c1(NCC(CCC)OC)cc(Br)ccc1S(=O)(=O)NC(c1cc(C)cc(C)n1)=O CN=C(NCc1cc(OC)cc(C(N)=O)c1)N1CCC2(CCN(C)C2)C1 C12(NCc3scc(C(C)C)n3)CCC(C(=O)Nc3nccc(Br)c3Cl)(CC1)CC2 c1(N2CC(C)C(NC(=O)CC3CCCC3(F)F)CC2)ncnc2sc3c(c12)CCC3 C(C(C)(C)CNC(=O)C(C)NC=O)N(C(C1(COC)CC1C)=O)C CCC(C)C(C(=O)N1CCC1Cn1cc(-c2ccc(OC)c(N)c2)nn1)N(C)C C1(C(N2CC3C(NC(=O)COCc4ccccc4)(C3)C2)=O)CCCCCCC1 C1(C(=O)NCC2CCC(CC)O2)CCCCN1C(=O)C(CC)OC CCCCCC(C)(c1nnnn1C1(C)CC1)NC(c1cc(Cl)cs1)C Cc1nn2c(c1C(=O)NCC1(C)CC(NC(=O)C(=O)N(C)C)C1)CCCC2C n1(CC(=O)NCC2CC(F)CN2C(c2cnsc2)=O)cccnc1=O N1(C(c2cc(C)ns2)=O)CC(C(=O)NCc2nonc2C)C2(CCC2)C1 c1(C(=O)NCC2CN(C(C3C(C(=O)OCC)CC3)=O)CC2C)nnc(O)nc1O CC1CN(C(=O)COC(C)(C)C)CC(C)C1NC(c1ccc(S(C)(=O)=O)o1)=O C(CC(C)(C)CC(=O)NC(CNC(=O)CC1(O)CCN(C)CC1)CO)OC c1(NC)ccccc1C(=O)N(C(C)CC(=O)N1CCC1)C CC1=C(C)CC(C(=O)NC(C)CNC(c2cn(C)[nH]c2=N)=O)CC1 C12(C(=O)NC3CCN(C(c4cccn4C4CC4)=O)C3)CC3CC(CC(C3)O1)C2 C12(NC(CCC(C)(C)F)=O)CCN(C(=O)Cc3coc(C(F)F)n3)CCC1C2 C(C)(C)(CCC(=O)NC1CC(CNC(C2CCO2)=O)C1)OC C1(NC(c2nc(C)sc2)=O)CCCN(C(C23C=CC(CC2)C3)=O)CC1 C1(CCNC(C2C=CCC2)=O)CCN(C(c2cnsn2)=O)CC1 CN1CCC2(CCN(C(=O)NCC3CCCCN3c3ccncc3)C2)C1 c1(C(N2C(CNC(C(CCC)c3ccccc3)=O)CC2)=O)nc(O)[nH]c(=O)n1 N1(C(C=CC(CC)C)=O)CCCC(NC(c2cnc(C)c(Cl)c2)=O)C1C CC1(C)CC(CNC(c2cnoc2C2CCOCC2)=O)CN(C(=O)C(N)=O)C1 C1(NC(c2cc[nH]n2)=O)CN(C(C2(c3ccccc3)CC(O)C2)=O)CC1C1CC1 Cc1ccc2c(CN3CC(CNC(=O)NC(C)(C)C)C(C(F)(F)C)C3)coc2c1 c1(C(=O)NCC(CNC(Cc2c(C)cc(C)s2)=O)F)cnn2ccc(O)nc12 CCC(C)(C(=O)NCC1(O)CCN(C(=O)Cc2ccc(F)cn2)C1)C(N)=O C1(C(=O)NC(c2ccc(OC)cc2)CC)CC2COCC(C1)C2N c1(C(N2C(C(C)NC(c3c(CCC)n[nH]c3)=O)CCC2)=O)ccc(C)c(F)c1 c1(CCC=CC(=O)NCC(CNC(=O)C=Cc2nccs2)OC)ccccc1 C(=O)(C(C)(C)C(=O)NC(CNC(c1ncsc1Br)=O)C1CC1)NC c1(SCCOCCNC(N(C)C)=O)ccnn1C(C)(C)C c1(C(=O)OCCCC(N2C(c3c(C)nn[nH]3)CCC2)=O)nc(S(C)(=O)=O)ccc1Cl N1(C(CC2(C)N(C(C(C(C)C)O)=O)CC2)=O)CCOC2(CCC2)C1 c1(COC=CC(C2CC2)NCC(C)(C2CC2)C2CC2)ccc(C(F)(F)F)cc1 C(=O)(CC=C(Cl)Cl)N(C(C)(C)C)CC(C1CCCC1)C.C(C(=O)C)S Cn1cc(C=CC(=O)NCCC(O)CNC(=O)Cc2cccc(Br)c2)nn1 Cc1sc(Cl)c(C(N2CC(Oc3ccccc3)C2)=O)c1C.N12CCCC(C1)C2=O N1(C(=O)OC(C)(C)C)CC(CNC(c2ccc(Br)cc2F)=O)CC1(C)C C1(NC(C2CC(C)(C(=O)O)C2)=O)(NC(C(c2ccccc2)C)=O)CCN(C)C1 c1(NCC2(C)CCCCC2O)ccc2c(c1)OCC1(CC2)OCCO1 C1(CNC(C2CC3CCC2CC3)=O)CC(C)CCN1CC.c12cc([nH]n1)C(=O)N2 C(C)(CO)(C(=O)N(C1(CC(N2CCOCC2C)=O)CC1)C)OC c1(C(=O)NCC2C(NC(Cc3cc(C)sc3)=O)CCC2)c(C(C)C)cccc1C c1(C(N2CC=CC(NC(c3cnn(C)c3F)=O)C2)=O)cc2nccnc2cc1F N1(C(c2cccc(CC)c2N)=O)CC2CCC(NC(=O)C#CC3(C)CC3)(C2)C1 N1(C(c2c(CC)nn[nH]2)=O)CCOC(C(C)NC(C2(C(F)F)CCCC2)=O)C1 C1(CNC(=O)Cn2cc(Cl)cn2)CN(C(=O)Cc2ccsn2)C2CC12 CC1=CCCN(C(C2CC(C)N2C(c2nccn2C)=O)=O)C1 CC(C)CC(CNC(=O)C(C)C(C)C)C(=O)NC(C(C)(C)CO)C1CC1 c1(C(N2CCCC(C)(NC(c3ccoc3I)=O)C2)=O)ccc(F)c(N)c1F C(=O)(CC(O)c1ccccc1)N(CC(C)NC(=O)CCOCC(F)(F)F)C c1(C(=O)NCC(CNC(c2c(CC)ncnc2)=O)O)cnc2cccnn12 N1(C(CC2CCCN(C(=O)CN3CC4CCC3C4)CC2)=O)CCCC12CCOC2 C1(CNC(CCC(=O)NCC=C)=O)CC(CNC(=O)CN2CCOCC2)CCO1 C(=O)(C1=CC2C=CC1C2)N(C(C(=O)N(C(CC(CC)C)C)C)C)C N1(C(c2cc(C#N)[nH]c2)=O)C2CC=C(C(=O)N3CCCC3C(N)=O)C1CC2 CCC(C(=O)NCC#CCNC(C1CC(F)C1)=O)OC1CCCC1.C(C)CC(C)C N1(C(C(C)(C)CC#N)=O)CC2(CCC(CNC(=O)CC3C=CCCC3)O2)C1 CCC(C)C(C(=O)N1CCC1C(=O)NCc1ccc(C)nc1O)NC(C)=O.C(=O)OC CCN(C)NC(=O)Cn1cc(CNC(C2CN(C3CCCCC3)C2)=O)nn1 C1(C#CC(=O)N2CCSCC2CCNC(c2cncc(F)n2)=O)(CC)COC1 Cc1ccc(C(N2CC(C)(C)CC2CNC(=O)C(C)n2ccnn2)=O)c(F)c1 c1(CN(C2CCCN(C(c3c(C)nccc3)=O)C2)C)ccc(Cl)cc1O N1(C(c2n(CC)ncc2C)=O)CCC2(C=C(C(=O)Nc3ccc(F)nc3C)C2)C1 c1(OC)ccc(C(N2CCC(NC(=O)C(C)CC(C)(F)F)C2C)=O)c2sccc12 c1(N(C(C(=O)OC)C2CC2C)C(=O)CCC2CC2)ccc(O)c(OC)c1 C1(NC(CNC(N)=O)=O)CC(NC(C2CCCC2CF)=O)C(O)C1 C#Cc1ccc(NC(C2CC23CCN(C(c2cnn(CC)c2C)=O)C3)=O)cn1 C(CC(C)C)(C(=O)NC(CCC)CCCC)NC(C(CCCC)O)=O N1(C(C2(C(=O)OC)CCCC2)=O)CC2CC2(C(N2CCNC(=O)C2)=O)C1 C1(C(=O)NC(C)Cc2nccn2C)COCC1C1CC1 N1(C(C(n2c(C)nc(C)n2)C)=O)CCC(C)(C)C1C(=O)NOCC1CCCCC1 C1(NC(COCCC#C)=O)CN(C(=O)CCC2CC2(C)C)C2(CCOCC2)C1 C(=O)(C1CCc2cc(OC)ccc21)N1C(CCC(=O)NCCCOC)CC1 CC1(C)Cc2[nH]nc(C(=O)Nc3ccc(=O)n(CCF)c3)c2C1 C1(NC(=O)CN(C(=O)CCC2CCC2)CC2CC2)CCCC(CO)CC1 CC(C)CC(CNC(c1ncccc1Br)=O)NC(C1CCCSS1)=O C(=O)(C1=CCCCC1C)N(C1CCCC1)CCCNC(=O)C1=CSCS1 c1(OC)ccc(C#N)c(NC(c2cc(-c3cnn(CCN(C)C)c3)[nH]n2)=O)c1 Cc1ccc(C(=O)NCc2ccc(CC(C)NC(c3cnn[nH]3)=O)cc2)nc1C N1(C(C(C)OCCOC)=O)CC2CCC(N(C(=O)Cc3cncs3)C)C2C1 C1(CC)C(=O)NCCN1C(=O)Cc1cn(C(C)(C)C(=O)O)nn1 O=NN1CCCC1C(=O)NCCC1CC(NC(C23CC(C#N)(C2)C3)=O)C1 Cc1noc(C)c1C(C)CC(=O)NC1CCN(C(=O)C(n2cc(Cl)cn2)C)C1 C1(C(=O)NC(CC=C)CNC(C2(C(=O)OCC)CCCC2)=O)CC(=O)N(O)C1 N1(CC2CCC(C)O2)CCSC(C(=O)Nc2ccnc(Cc3ccccc3)n2)C1 N1(C(C2(CC#N)COC2)=O)C2CCCC1CN(C(=O)Cn1cccn1)C2 N1(C(CSCC=C)=O)CC(O)CC1CNC(=O)C(c1ccccc1Cl)O c1(N2CC3N(Cc4cccc(F)c4Cl)C(C3)C2)ncnn2ccc(Br)c12 n1(C(CC)C)ncc2cc(C(=O)NC3CN(C(c4cnsn4)=O)CC3F)cnc12 c1(C(N2CC(NC(c3c(C)cccc3F)=O)C3C2C3)=O)c(Cl)ccc(F)c1N C(=O)(C1=CCCSC1)N1CCC(N(C(=O)CCCOC(C)=O)CC)C1 CCC(CC)CC(=O)N1CC2CC(NC(=O)Cc3cc(F)ccc3C)C1C2 CC1=CCN(CCNC(=O)CCCCN(C(=O)CC2CCOC2(C)C)C)CC1 N1(C(C2C(OCC)CCCC2)=O)CC2CCC1C2C(=O)NC1(C)CCC(=O)NC1 Cc1ccc(Br)c(CC(=O)NCCOCCCNC(c2cc(C)on2)=O)c1 c1(C(N(C2CCN(C(C(CC#C)C)=O)C2)C)=O)ncc(C(=O)OC)cc1Cl C(=O)(CC(C)C(C)C)N1C(CCNC(c2nc(C)n(C)c2)=O)CCCC1 C1(NC(c2c(C)nn(C(C)(C)C)c2N)=O)CCc2nnnn2CC1 c1(C(=O)NC2C(NC(c3cc(COC)no3)=O)C2)cnc([N+](=O)[O-])n1C CC1CC(c2cn(C3CCOC3)nn2)CCN1C(c1c(C(=O)OC(C)(C)C)occ1)=O N1(C(c2cncc(N)n2)=O)CCCCC(CNC(c2cc(Cl)sc2Cl)=O)C1 C=CCC(CNC(=O)Cc1ccc(Br)cc1)C(=O)NCCSCCOC C1(C(C)NC(c2nc(OC)oc2)=O)CN(C(C2C(C)C2C)=O)CCO1 c1(CSC)ns[nH]c1=O.c1(C2CNC(=O)C3(CCC3)C(=O)OC2=O)ccccc1 Cc1cc(I)ccc1C(=O)Nc1cccc(NC(c2c(Cl)ccnc2Cl)=O)c1 c1(NC(CCC)C(C)(C)C)ncccc1S(=O)(=O)NCc1cnsc1 C1(CC=C)CC2CC(O1)CC(=O)N2.C1(C(=O)OC)COC(CC(C)C)C1 Cc1ccc(CC(=O)NC2CC23CCN(C(C2CCC(C)C2)=O)C3)cc1F N1(C(=O)C=CC(c2ccccc2)=O)CCCN(C(C2(F)CCCC2)=O)CCC1 C1(SCC(CCCCCCO)=O)CCC2(CCCC2)O1.OC C(C(=O)NC1(CC(C)C)CCN(C(=O)C=Cc2nc(C)co2)C1)(C(C)C)OCC C1(CNC(C2(COC)COC2)=O)CC2(C1)CN(C(c1nc(OC)ccc1C)=O)C2 N1(C(CCCOC)=O)CCCCCC1CNC(c1cccc(-c2nccs2)c1)=O Cc1cnc(NC(C)CC(C)NC(c2nn(C)c(C)c2N)=O)nc1S(C)(=O)=O C1(c2sc3cc(C)sc3n2)CC2(CCN(C(=O)NCC3(C)COC3)CC2)C1 Cc1ccc(C(C)NC(c2cn(CCNC(C3CCCC4CC34)=O)nn2)=O)cc1 CC(F)CC(=O)NCCCN(C(=O)CCC1CCCN1CC1CCCC1)CCO C1(C(=O)NCCC2(OCC)CCC2)CCN(C(C2CC2F)=O)CC1 Cc1cccc2sc(C(=O)NC3CCC4CC3CN4C(=O)CCCC#N)c(Cl)c12 c1(C(N2CCCC(C(F)(F)F)CC2)C(=O)NCCCC)sc(Br)c(C)c1C C1(CNC(c2n(C(C)C)ncn2)=O)COCCN1C(=O)CCOCCN(C)C Cn1ccc(=NC(=O)c2ccnc(CNCc3cccc(O)c3)c2)[nH]1 n1(CC(N2CCC(CNC(C3CCCN(CC)C3)=O)C2)=O)cc2ccccc2n1 N1(C(CC2(OCC)CCC2)=O)CC2CCC1C(CO)C2.c12cnnc(c1)C(=O)N2 C=CCC(C(=O)N1CC2(CC(CC(=O)NCC3CCOC3=O)C2)C1)C(C)C N(C)(CP(C)(C)=O)C(CC1C=CC(NC(CCc2cnc(C)o2)=O)C1)=O C(=O)(CCC(C)(C)C#N)NC1C(C)CN(C(c2c[nH]ccc2=O)=O)CC1 C(=O)(C1=COCCO1)N1C(C)CC(CNC(c2cnccc2Cl)=O)C1 c1(C(=O)NC(CCCNC(C(CCSC)OC)=O)C)nc(C)c(C)nc1O CC1CN(C(=O)CCc2nccn2C)CCCN1C(c1cnc2[nH]cncc1-2)=O N1(C(CN(C(C)C)C)=O)CC2CCC1C(NC(c1c(Cl)ccc3n[nH]cc13)=O)C2 C1(CNC(CCOC)=O)(CO)CCN(C(C2CCCN2C2CC2)=O)C1 C12(CNC(C(CC)(C)C)=O)CCCC1CCN2C(c1ccc(C(N)=O)o1)=O c1(CC)cc(C(=O)NC2CCC(NC(=O)CC3CC3CC)C2)ccc1F c1(CC(=O)NCC(CC=C)NC(=O)C(CO)N(C)C)cnc(C(F)(F)F)cn1 C12(C(N(CC#C)CC3CCC3)=O)CCC(NC(=O)Cc3ccccc3F)(CC1)C2 O(N1CCC(N=c2cc(C)[nH]c(=NCC3CCC(C)C(=O)N3)[nH]2)CC1)CC N1(Cc2n(CCOC)nnn2)CCC(O)C(C(=O)NC(C)Cc2ccccc2F)C1 c1(OC)cccc(C(=O)N(CCNC(=O)C=C2CCC(C)C2)C(C)C)c1 C1(C(=O)NCC(C(C)C)NC(=O)CCCC#N)CC12CCOCC2 Cc1nc(C=CC(N2CCCC2CNC(C2CC(C)(O)C2)=O)=O)[nH]c1C C(CC(C)(C)CC(=O)NC1C=CC(CC(N2CC3CCC3C2)=O)C1)OC C(C(CC1CCCC1)C(=O)N(C)CC1CCOC1)NC(CN(CC)CC)=O Cc1ccc2oc(N3CC(C)(C)CCC3CNC(=O)C(C(C)C)N(C)C)nc2c1 CC1=C(C(=O)NCCCN(C(=O)CC2CCOCC2(C)C)C)CCCC1 N1(C(CC2CC(C)C2)=O)CC2CC(O)C1C2N(C(=O)CN1CCCCC1)C1CCC1 CCCC(C#N)C(=O)N1CCN(C(CNC(c2cc(C)c(C)o2)=O)C(F)F)CC1 C(=O)(C1=CCN(C(c2cccc(F)c2N)=O)C1)Nc1ccc(CC)nc1 c1(C(=O)NC(CN(C(=O)C(C)CC2CC2)CC)C)ccc(OC)cc1Br N1(C(c2c(C)ocn2)=O)CC2CC2(NC(c2ccc(SC(F)(F)F)o2)=O)C1 c1(C(N(CC(C(=O)Nc2cn(CC#C)nc2)C)C(C)C)=O)cc(C#C)ccn1 N1(C(c2nc(COC)oc2)=O)CCCC(CCNC(C2CC3(CC3)C2)=O)CC1 N1(C(c2nc(CC)sc2)=O)CCC(C)C(N(C(=O)CCc2cncc(F)c2)C)C1 S(=O)(=O)(c1cccnc1NCc1cnsc1)NC1OCCN(CC)C1 N1(C(c2c(OC)n[nH]c2)=O)CCCCC1C1(NC(=O)COC2CCC2)CCC1 Cc1nc2cc(Br)cc(C(=O)NCc3ccc(S(N)(=O)=O)cc3)c2o1 c1(C2CCCN(C(C(=O)NC3C(N)CCC3O)=O)C2)c(Cl)cccc1Cl N1(C(CC2CC(C)C2)=O)CC2CCC2(CNC(=O)CCCNC(=O)C2CC2)C1 c1(C(=O)NC2C(OC)CN(C(=O)C(F)C3CCC3)C2)cc2cccc(F)c2s1 C(=O)(C(c1cccs1)=CC(C)C)N1CC(CNC(C)=O)C1.N12CCC(C13CC3)C2=O N1(C(c2cc(COC)sc2)=O)C2CCC1CN(C(C1CC(O)CN1C)=O)C2 CC1(O)CON(C(=O)CC(CNC(C2(NC(N)=O)CC2)=O)C2CCC2)C1 c1(C(=O)NC(c2ccccc2F)CNC(c2ccc(C)s2)=O)cncc(N)c1 CC(C)(CC(=O)NC1CN(C(C2CCN(C(N)=O)CC2)=O)C2CC12)n1cnnn1 C(=O)(C(F)(F)C(F)(F)C(F)(F)F)N1CC2CCN(C(c3cn(C)nn3)=O)CC2C1 c1(OC)cc(NC(C2C3CC2N(Cc2sccc2Cl)C3)=O)cc(F)c1 C(=O)(CCCCC(C)C)NCCC(CNC(=O)COc1cncc(C)n1)OC C1(CC)C(C(=O)NCCN(C)CCF)CCCN1C(c1cc(C2CC2)no1)=O N1(C(C2CC(COC)C2)=O)CC2CC2(C(=O)OC)C1.C12(CC1)C(=O)NC2 CC(C)(C)C(C)(C)C(=O)N1CCOC(CCCNC(=O)CO)C1 Cc1cc(C)c(S(=O)(=O)N2CCC(c3ccc(F)cc3Cl)CC2)cc1[N+](=O)[O-] c1(OC(C)C)ncccc1C(=O)NCC(C)(O)CNC(c1nc(Cl)c(Cl)s1)=O N1(C(CC2CN(C(CCOCCOC)=O)C(C)C2)=O)CCSC2(CCC2)C1 C12(C(=O)NC3(CO)CCCN(C(c4ccc(C)cc4C)=O)C3)C3C4C1C1C2C3C41C CC(C)CC(C)C(=O)NCC1(O)CC(C(=O)NCC(O)C2CC2)C1 C1(CNC(=O)Cc2ccsn2)C2CN(C(=O)CSc3cccc(Cl)c3)CC12 Cc1cnc(NC2(C(N3CCC(N4CCN(C(N)=O)CC4)CC3)=O)CC2)c(F)c1 c1(N(C(=O)CC2CCCN2C(c2n[nH]c(C3CC3)n2)=O)CCC)ccc(C#N)cc1 N1(Cc2ccc(C(C)C)cc2)CC2C(C1C(N1CC(=O)NC(C)C1)=O)C2(C)C C1(CN(C(C2CCCCO2)=O)CC)CN(C(=O)CCc2cccnc2)C(C)(C)C1 c1(C(N(CC(=O)N(CCOC)CC2CC2)C2CC2)=O)cccc(F)n1 C(CNC(=O)CN1CC2C=CC1C2)(CC(F)(F)F)NC(c1c(C(C)C)cco1)=O N1(C(COC)=O)CC(NC(=O)CC(C)(C2CCC2)N(C)C)C2(CC2)C1 N1(C(C=Cc2n(C)ccc2)=O)CC2CC(NC(c3cnc(C(N)=O)nc3)=O)C2C1 CCCS(=O)(=O)CC(=O)NCC12CN(C(c3cc[nH]n3)=O)CC1CS(=O)(=O)C2 N1(C(C2C(C)=C2)=O)CCOC(C(C)NC(C2CC3C=CC2C3)=O)C1 C12(CCNC(c3csc(Cl)c3)=O)CCC1CN(C(=O)Cc1csnn1)C2 c1(C(C)C)cc(N(CC(C)NC(c2occc2-c2ccccc2)=O)C)ncn1 CC1CCSCCN1C(C1COCC1NC(C1(C(C)C#N)CCC1)=O)=O c1(CC)oc(C)cc1C(=O)NCCCCC(C)NC(c1ccnn1C(C)CC)=O C1(C(=O)NCC(=O)NCC=CCNC(C2CC=CCC2)=O)(CC)CCC1 N1(C(C(C)NC(=O)OCC)=O)CCCC(NC(=O)CCSc2ccccn2)CC1 c1(N2CC3(OCC(NC(c4ccc(F)cc4Cl)=O)C3)C2)c(Br)cccc1[N+](=O)[O-] C#Cc1cccc(C(=O)NCCC(=O)NC(CN(C)C)CO)c1 C1(CC)(CC)CC(NC(c2nnc(S)n2C)=O)CN1C(=O)CC1CC1(C)C n1(CC(=O)NCC(CNC(=O)C(O)Cn2cncn2)OC)c(C)c(C)sc1=O C(=O)(CC(=O)NC)NCCOCC#C.C1(OCCCNC)CC1C(=O)OCC n1(CC(C)O)cc(C(=O)NC23CC2CN(C(c2cc(C)co2)=O)C3)ccc1=O CC1CCN(C(C2CC2c2ccccn2)=O)CCN1C(c1cnn(C2CC2)c1)=O C1(CNC(=O)NC(c2ccccc2Br)CC)(OC)CCC(C)C1 N1(C(C2C(C#N)C2)=O)CCOCC(CNC(C2(c3ccc(Br)cc3)CC2)=O)C1 O=C1CCC(CC(N2CCCC(CCCCNC(C3(CCF)CC3)=O)C2)=O)CN1 c1(C(=O)NC2C(NC(C3N(C(C)=O)CC(O)C3)=O)CC2)cc2n(c1)CCSC2 N1(C(c2ccc(Cl)s2)C(=O)NCC2CC2)CCCCC1c1ccccn1 CN1CCC(C(=O)NCCNC(=O)CC2CCC3CC23)(NC(=O)OC(C)(C)C)C1 N1(C(C(c2ccc(C)cn2)(F)F)=O)CC(C2(NC(c3nonc3N)=O)CC2)C1 c1(C2(C(=O)NCCNC(C(C)OCC)=O)CCCC2)cccc(Cl)c1.C(COC)=C c1(C(=O)NC2(c3nn[nH]n3)C(CCC(C)C)CCC2)cccc(C(N)=O)c1 CC12CN(CCC(N)C3CC3)CC1C1C=CC2C1 N1(C(C)=O)CCCCC1C(N1CCC(C(=O)NCCC2CC2C)CC1)=O c1(OCC=C)ccc(C(=O)NCC(CO)NC(=O)C(C(C)C)SC(C)(C)C)cc1 C1(C(=O)NC2C3OCC(NC(=O)CC(F)F)C3OC2)CC(C2CCOCC2)=NO1 C(=O)(CC1=NNC(=O)C1)NCC(OC)NC(=O)CC1CC(N(C)C)C1 CCCC#CC(C)(C)NC(=O)C(C)N(C(=O)C(C)N1CC(C)C1)C C(=O)(CS(=O)(=O)CCOC)N(C1(CC(=O)N(CC=C)CCC)CC1)C c1(C(N(CCCN(C(c2nc(OC)oc2)=O)C)C)=O)ccc(CO)c(Cl)c1 C1(NC(N2C(C)Cc3cc(Br)cnc32)=O)CC(c2ccncc2)=NO1 c1(C(=O)OC)ccccc1C(=O)N(CCO)CCN(C)C C1(CNC(CN(C2CC(C#N)C2)C(C(c2ccccc2)C)=O)=O)CC12CCOCC2 C1(C(=O)NCC(CN(C(c2cc(Cl)c[nH]2)=O)CC)(C)C)C(F)(F)C12CCC2 N1(C(Cc2ccc(OC)cn2)=O)CCC(C)(C)C(CNC(=O)C(O)C(F)F)C1 O(NC(=O)CC(C)(F)F)CC(=O)NCC1(CCC#C)CC1 n1(CC)ncc(Cl)c1C(=O)NC1CC(F)(CNC(=O)C(c2ccc(Cl)s2)=O)C1 c1(-c2c(CN3CC(C(=O)O)CC(F)(F)C3)cccn2)ccc([N+](=O)[O-])cc1F c1(C(N2CCN(C(C(CSC)OC)=O)CC2C)=O)ccc2c(c1)nnn2CCO c1(C(=O)NC(CO)C(=O)NC2CC(O)C2)ccc2[nH]ccc2c1 c1(OC)cncnc1C(N1CCC(C)(C(=O)NC(C(O)CO)C2CC2)C1)=O c1(C(C(N2CC(CNC(c3n[nH]c(C)c3C)=O)C(O)C2)=O)C)cccc(C#N)c1 c1(C(=O)NCC(C)CNC(=O)C(C)(C)c2ccno2)ccc2nccn2c1 C1(CNC(C(C)Cc2cccc(Cl)c2)=O)CC2CCC1N2C(=O)CCCCN(C)C c1(C(CNC(CC2CCC(=O)N2)=O)NC(C2CCCC2)=O)ccccc1F c1(C(=O)OCC)cccc2[nH]nc(C(=O)NCC(C)NC(=O)COC)c12.C1CCC1 c1(CC(=O)NC2CN(C(c3cc(Br)no3)=O)C2)ncc(F)cc1F N1(C(CSCCCC)=O)CCC(C(=O)NCC2CC2)C12CC2 Cn1cnc2ccc(C(N3CCCCC(CNC(=O)C(O)CC(N)=O)C3)=O)nc12 CCCCCC(F)C(=O)NCCNC(c1cc(O)ccc1F)=O C(=O)(CN=S(C)(C)=O)NCC(c1c(CC)cccc1)NC(C1CC1CC)=O C12(NC(C3C(C)CN(C)C3)=O)CCC(CC1)N(C(c1cc(Cl)no1)=O)C2 C1(CC)CN(C(C2CCCCC2O)=O)CC1C(=O)NCCN(C(C)C)C1CC1 c1(C(=O)NCC2(NC(c3ccncc3Br)=O)CCC2)cc2cccnc2cn1 N1(C(CC(CCC)O)=O)CC2CC(C1)N(C(C1CCN(C)C(=O)C1)=O)C2 c1(C(=O)NC(CNC(COCCOCC)=O)CC)c2n(c(=O)n1C)CCCC2 Cc1cnc(C(N2CCC(NC(c3onc(C)c3C(F)(F)F)=O)C2)=O)cc1C CC(C)CC(c1nnnn1C1CCCCC1)NCc1csc(C2CC2)n1 N1(C(Cc2cccc(C#C)c2)=O)CCC(F)(F)C(CNC(c2sc(C)cc2Cl)=O)C1 N1(C(c2c(CC)nccn2)=O)CCC2C(CCCN2C(=O)C(C)CSC)C1 C1(N(C(CCCN(C)C)=O)C)CC2CCC(C1)N2C(c1n[nH]cc1C1CCC1)=O c1(C(=O)NCC2C(CNC(C(C)CC3CCCC3)=O)C2)ccc(C(F)(F)F)nc1 CC(C)CC(=O)C(=O)N1CC2C(NC(=O)COc3ccsn3)C2C1 CCC(C)C(O)C(C)C(=O)NC(COC)CC(=O)NC(c1nc(C)cs1)C C(=O)(C(F)(F)C(F)(F)F)N1CCCC(CNC(C(C)(c2ccccc2)OC)=O)C1 c1(C(=O)NCC(CCCC)NC(=O)C(O)CCSC)cc2cc(Cl)sc2[nH]1 C(=O)(CCCCCCN(C)C(C)C)N(CC(=O)N(C(CC)C)CC)C(C)C CC(CC(=O)N1CCCC(C)(CNC(=O)CC2CC3CCC2O3)C1)P(C)(C)=O Cc1cc(F)ccc1COCC(=O)N(C1CCCN(C(C2CC2F)=O)CC1)C C#Cc1ccc(C(N2CC(F)(F)CC2CNC(=O)C(C)CCCOC)=O)nc1 C#Cc1ccc(F)c(C(=O)N(CC(C)NC(=O)CC2CC2(Cl)Cl)CC)c1 c1(CN2C(C)(C(=O)Nc3cc(C)sc3C)CC2)ccc(Br)nc1Br CC(C)(C)C(C(=O)NCCC12CC(CCO1)C2)NC(C1CC(F)(CF)C1)=O c1(NC(N(C)C)=O)cn(C)c2ncc(-c3ccc4sccc4c3)cc12 c1(C(C(=O)NCC(C)NC(c2cnsc2)=O)OCC2CCCO2)ccc(F)cc1 N1(C(C(N2CCSCC2)C)=O)CCC(CO)(CNC(=O)CN2CCOCC2=O)C1 Cc1ccc(SCC(N2CC3CCC3(NC(=O)C(O)C3CC3)C2)=O)c(C)c1 C12(C3CN(C(C(C4CC4)SC)=O)C3)COC(C1)C(O)C2.C1(=O)C(C)OCC(=O)O1 Cc1cc(=NCCCC(C)(C)NC(=O)C(C)Cc2ccccc2)[nH]c(CC2CC2)n1 CCC(CC)C(=O)NC(C)CCNC(=O)C(CC)OCC(=O)N(CCCSC)C CC(C)C(C(=O)NCC1CC1CC(=O)N(C1CC2CC2C1)C)C(C)C c1(C(=O)NCC(CO)NC(c2cccc(C(C)C)c2)=O)cc(Cl)cc2c1OCC2 n1(CC)nc(Cn2ccnc2)nc1-c1cccc(COCC2CC2)c1 CC(N=c1nc(N2CC(=O)NC(C)(C)C2)c2ncccc2[nH]1)c1ccoc1 C1(NC(N(C2CC2)Cc2ccc(C)s2)=O)CCC2(CCCCC2)O1 C1(NC2(COC)CCCOC2)CC2(CCCCCC2)C1 c1(OC)ccc(CN(C)Cc2ccc(CC3CCC(C)CC3)o2)c(OC)n1 CCC(C(=O)NCCOCCNC(=O)Cc1c(C)nn(C)c1Cl)C(C)(C)CC C(=O)(C(C)(C)N=[N+]=[N-])NCc1c(C(=O)NCCc2nc(C)[nH]n2)occ1 C1(C(=O)NCCn2ncc(C(=O)NC3CC(CF)C3)c2)CCC(n2ccnn2)C1 C(=O)(CC1=CCCC1)NCCC1CCCN(C(CCCc2n(C)cnn2)=O)C1 N1(C(C2C3(CC(OCC)C3)C2)=O)CC(NC(C2CC3CC3C2)=O)CC2(CC2)C1 C1(CNC(C(C)CC(F)(F)F)=O)CCCC2(CN(C(=O)CC3CC(C)(C)C3)C2)O1 CCCCC(O)C(C)C(=O)NCC(C)=CC(=O)NC(c1cnc(C)s1)C Cc1ccc(F)c(C(=O)NCC2(NC(=O)C(C)Oc3ccc(F)cc3)CC2)c1Cl c1(C(=O)NC(CC)CN(C(=O)CC2CC2)C)ccc(N(C)C)cc1OC CC(=O)CCCC(=O)NC(C)(CNC(=O)CCCc1nncn1C)CO CCCC(F)C(=O)N1CCC2CC12C(=O)NCc1cc(C#N)c[nH]1 c1(CC(=O)NC(c2nocc2C(=O)NCC2(C(N)=O)CC2)C)cncnc1O CC(C)C(O)C(F)(F)C(=O)N(CCNC(C1CCCCC(=O)N1)=O)C1CC1 C1(CN(C(COC(CC)CC)=O)C)CCCN(C(=O)CCCC2(NC)CCC2)C1 c1(C(CC)NC(=O)NC2CC(C)(C(F)(F)F)C2)cccc(Cl)c1 C(=O)(CCP(C)(C)=O)NCC1(O)CCN(C(C(C)O)=O)C1.c12cn(nn1)CN2 C(c1cc(F)cc(F)c1)=CC(=O)NCC1C(C)CCN1C(=O)Cc1ccc(Cl)s1 C(N=c1cc[nH]cc1[N+](=O)[O-])SCCNC(C1CC(C)(C)OC1)=O c1(C(C)OC)nc(C)c(S(=O)(=O)N2CCCCC2C(=O)OC)s1 Cc1ccc(C(=O)N(C2CCN(C(=O)CCc3ccccc3Cl)CC2)C)nn1 C(N=c1ccn2nccc2[nH]1)C1CCCN(Cc2c(OC)cccc2F)C1 c12ccc([N+](=O)[O-])c(c1)C(=O)N1CCN2CC1.c1ccc(S(N)(=O)=O)cc1.CO c1(C(N2CC(C)(C)C(C(=O)NCC3CC34CC4)C2)=O)c[nH]c2cnccc12 N1(C(C(CC)OC)=O)CCCCC(C(=O)NC2CC2(C)C)C1 C1(NC(c2on(C)c(=O)c2)=O)COC2(C1)CN(C(c1cc(Cl)cc(Cl)c1)=O)C2 C(=O)(C1CCc2ccc(C)cc21)NC(CC)CNC(c1cc(F)c(F)c(F)c1)=O Cc1nc(C(N2CCOC3(CCC3)C2)=O)c2ccnc-2[nH]1 c1(CC(=O)NC2CC2)cccc(Nc2ccns2)c1 C(=O)(C1CCc2c[nH]nc21)N1CCC2(C(NC(c3n(C)c(S)nc3)=O)C2)C1 C(=O)(C(C)(C)CC(F)F)N(CCC1N(C(C(C)=C2CC2)=O)CCCC1)C C1(CNC(C2CCOC2)=O)CCN(C(C2CC(C(F)F)C2)=O)C12CCC2 c1(C(=O)NCC(CNC(CSCCC)=O)F)cnn(CCF)c1 C1(C2(NC(CC(=C)Br)=O)CC2)CCCCN1C(c1ccccc1SC)=O c1(C(=O)NCCCOCCN(C(CC2N(CC)CCC2)=O)C)ccc(C)n1C c1(OC)cc(Cl)ccc1CC(N1C(C(=O)NC2CC(F)(F)C2)CC2CC12)=O N(C1CCCc2ccoc21)C(C1CC(C)N1C(=O)CCc1ccc[nH]1)=O C1(CC)CCN(C(C2CCCCS2)=O)C1CNC(c1cccc(OC)c1)=O c1(C(=O)OC)cc(CN2CC(O)CC2C(=O)O)c(C(F)F)cn1 Cc1cnc2nc(C(=O)NCC3CC3CNC(c3cc[nH]c3C3CC3)=O)nn2c1 N1(CC)CCOCC1CC(=O)NCC=CCNC(C1CCCC(C2CC2)O1)=O.OC N1(c2ncc(C)cn2)CCOCC(NC(=O)C(C2CCCCCC2)N(C)C)C1 c1(C(CNC(=O)C=CC(N2CCOCC2)=O)NC(C2C(C)C2)=O)ccccc1F N1(C(CC(C)CF)=O)CCCC(C)(NC(=O)C=Cc2cccc(Cl)c2)C1 c1(C(=O)NCCN(C(C2CC2(F)F)=O)CC2CCCC2)ccccc1C#CC1CC1 C1(CNC(c2cc(CCC)[nH]n2)=O)CCCC(NC(C2(Br)CC2)=O)C1 C1(C(=O)NC2CN(C(c3cc[nH]c3)=O)CCC23CCC3)CS(=O)(=O)CC12CCC2 c1(OC)ccc(C)cc1C(N1CC(O)(CNC(c2cc(C)ccc2O)=O)C1)=O CCC(C)(CNC(=O)CC12CCCC1C2)NC(c1[nH]nnc1C)=O C12(CNC(=O)C=Cc3cocn3)CCC1CN(C(=O)COc1ccc(F)nc1)C2 S(=O)(=O)(CC(=O)N1CCC(F)(CNC(=O)CCc2ccccc2OC)C1)NCC Cc1nc(N2CC(O)(CCNC(c3ccc(C(N)=O)o3)=O)C2)cc(C(C)C)n1 Cc1cn2cc(C(N3CCC(C)(NC(c4cc5n(n4)CCCC5)=O)C3)=O)nc2s1 C1(C)(CC)CC(NC(=O)C2=CCCC2)CN1C(=O)CN1CCSCC1 c1(C(=O)NC(CNC(c2ccn(C)c2)=O)C2CCC2)ccc(OC2CCC2)cc1 CCCCCCCCN(C(=O)C(=O)NC(C)CCc1ccc(OC)c(OC)c1)C c1(CC)cc(C(N2CCCC(CCNC(C3CCC(=O)N3)=O)CC2)=O)ccc1F CCCCCC(O)C(C)C(=O)N1CC(O)(CNC(c2cc3ccccc3o2)=O)C1 c1(CC(=O)NC(C2CCN(C(=O)CO)CC2)CO)ccc2scnc2c1 C(=O)(C(O)C(F)(F)F)N1CCC(CNC(c2ccc(CC(C)C)s2)=O)C1 C1(C(=O)NCCN(CCC)C(C2(SC)CC2)=O)CCCC(CC)C1 c1(SCC(N2C(c3cn(CCOC)nn3)CC2)=O)nc2ccccc2o1 c1(C(=O)NC(CNC(C(C)NC(=O)NC)=O)C(C)C)cc2ccccc2oc1=O C=CC1(C(=O)NCC2CCCCCO2)CCN(C(c2cncc(Cl)c2)=O)CC1 CC1(C)CN(C(=O)C=CC2CCOCC2)CC(CNC(=O)C(C)(C)CF)O1 c1(OCC)cc(C(C(=O)NC(C)(C)C)N(C)C(C2CC2)C2CC2)cc(Cl)c1 C(=O)(C(CC(C)C)C(N)=O)NC1CCC(C(N2CC=C(C)CC2)=O)CC1 C1(O)(NC(=O)CSCC2CCCO2)CCN(C(=O)C=CC(S(=O)(=O)C2CC2)=O)C1 N#Cc1cnccc1COC(=O)C=Cc1cccc(-c2ccc(Cl)cc2)c1 O=C1NC(C(=O)NCC(c2ccccc2)NC(C2CC2C(F)(F)F)=O)CCO1 C(S(=O)(=O)CCNC(c1cccnc1)=O)c1cn(CC=CCC(C)C)nn1 c1(OC)ccccc1C(CCNC(C)C(C1CCCCC1)C)OC C1(CNC(C(CO)OC)=O)CCC(CNC(C2(C)CC=CCC2)=O)CC1 C#CC1(C(N2CCC(CC(F)F)C2)=O)CCN(C(=O)CCc2cnoc2)C1 N1(c2nnc(OCC)s2)CCC2(CCN(C(c3ccc([N+](=O)[O-])cc3O)=O)C2)C1 C1(C)(NC(c2cccc(OC)c2)=O)CCC(NC(=O)Cc2ccccn2)CC1 c1(-c2c(C3(C(=O)NC)CC3)cccc2)cc(OC(C)C)c(F)c(F)c1 c1(CC)cc(C(N2CC(OCCNC(C3CC(C#N)C3)=O)C2)=O)c(C)o1 c1(C(N(CCCN(C(=O)C(C)(C)c2ccccn2)C)C)=O)cnn(C)c1N c1(C(=O)NC(CCN(C(CC(=C)C)=O)C)C)cccc(C)c1Cl c1(C(=O)NC(C)C(=O)NCCC2(C#N)CCC2)sccc1Cl N1(C(CNC(=O)NC)=O)CCC(C2CCCN(C(c3cccn3C(C)C)=O)C2)C1 Cc1ccc(C#N)c(C)c1Cc1noc(C2CCc3cn(C)nc3C2)n1 c1(OCC)cc(CCC(=O)NCCCCCNC(=O)Cc2ccc(C)s2)on1 N1(CCC=CCC)CCCC(NC(=O)CC(C)OC(C)=O)CC1 N1(C(CCC=CCC=C)=O)CCC(CNC(c2scc(C)c2Cl)=O)(OC)CC1 CC1(C)NC(=O)CC1C(=O)NCC1(O)CCN(C(c2ccncc2N)=O)CC1 C1(NC(=O)C=Cc2cccs2)CC2CC(NC(C34C=CC(CC3)C4)=O)CC12 N1(C(C2=NOC(C)(C)C2)=O)CCC2(CC1)CN(C(=O)C(C1CCCCC1)F)C2 C1(C2(O)CCOCC2)(C(=O)NCCC2CN(C(c3cnsc3)=O)CCO2)CC1 c1(C(=O)NCC(CCNC(C(C)OCC)=O)O)ccnc2ccncc12 C(=O)(CCCC(=O)NCCCNC(c1c(C(=O)OC)con1)=O)NCCO S(=O)(=O)(c1ccc(C(=O)N(CCC(C)NC(=O)C(O)CCSC)C)cc1)NC N1(C(C(CCC)OC)=O)CCCC(F)(C(=O)NCCN=[N+]=[N-])C1 c1(C(=O)NCC(CNC(=O)CC2COC(=O)C2)OC)ccc(F)c(F)c1 N1(C(C2N(CC(C)C)CCC2)=O)CCC(O)(CNC(=O)CCc2ccoc2)CC1 c1(C(N(CC(C)NC(=O)CCc2ncnn2C)C)=O)cnn2c1OCC(C)(C)C2 N1(C(C2(C(C)C)CCCO2)=O)CC2CC1CN2C(=O)CNS(C)(=O)=O C1(C(=O)N(CC(C)C(C)C)C)(CC)CCCN(C(c2ccc(C(C)C)o2)=O)C1 c1(C(=O)NC2C(CNC(c3n(C)ccc3)=O)CCC2)c(C(F)(F)F)cccc1O c1(C(=O)NC23CC(CNC(C4CC4[N+](=O)[O-])=O)(C2)C3)nccc(Cl)c1F N1(CCCOC)CCN(C(=O)CN2CCC(O)CC2)CC1.C12(CCOC1)C(=O)N2 Cn1nncc1CC(=O)NCC1(CCn2cc(C(C)(C)OC(=N)O)nn2)CC1 N1(C(Cn2cc(-c3cnn(C)c3I)nn2)=O)CCC(Cc2cscn2)C(F)(F)C1 CC1(CNC(=O)CC(C2CCC2)C2CCC2)CCC(NC(C2CNC(=O)O2)=O)C1 Cc1ccc([N+](=O)[O-])c(C(=O)NC2CN(C(C3CC4CCC4C3)=O)CC2O)c1C N1(C(c2cnc(S)[nH]2)=O)CC2CCC(C1)N2C(c1ccc(Cl)cn1)=O C1(NCC2(CC)CCC2)CCC2(CC1)CN(C(c1c(F)cccc1Br)=O)C2 C12(NC(C3(CNC(c4cnn5c4CCC5)=O)CC(=C)C3)=O)CCC(C1)C(O)C2O C1(N(C(=O)CC2CN(C(c3csc(O)n3)=O)CCO2)C)CCN(CC2CC2)CC1 N1(C(C2(CCOC)CCC2)=O)CCC(C2CCCN(CCS(C)(=O)=O)C2)CC1.CCS Cc1cccc2nc(SCC(N3CC(C)N(C(=O)CCC4CC4)CC3C)=O)[nH]c12 C1(C)(COC)CCCN(C(C2CCN(C(=O)CC3(C)CCCC3)C2)=O)C1 C(=O)(C(O)CCCNC(c1cnc(O)nc1)=O)N1C(CN(C)C)CCC1 C1(NC(=O)NC(Cc2ccc(C)cc2)(C)C)Cc2cccnc2C1 CC1(C)C(CNC(C2CCCO2)=O)CCN1c1ncc(C(F)F)cn1 N1(C(CCNC(COC)=O)=O)CC(NC(C2CC23CCCC3)=O)C(C)(C)C1 N1(C(C=C(CCC)C)=O)CC2CN(C(C3(COC)CC=CCC3)=O)CC2C1 N=c1[nH]c2ccc(C(N3CCC(CNC(=O)CCC(F)(F)F)C34CC4)=O)cc2[nH]1 N1(C(C#CC(C)(C)C)=O)CC23CCCCC2(C1)CN(C(C1CC(C#N)C1)=O)C3 N1(S(CC)(=O)=O)CCC2CCC(C1)N2C(=O)Nc1cncc(SC)c1 CC1CCCC(CC(=O)NC2CC(C)(OC(=O)NC(C)(C)C)C2)C1 N1(C(c2cnc(C(C)C)o2)=O)CCC2(CCC(NC(=O)CC3(CO)CC3)CC2)C1 C1(C(=O)NCC2(C(C)NC(=O)Cc3cnn(C)c3)CC2)CN(C)CC1(F)F c1(C(N(CCC)CC2CC2)=O)c(C(=O)NC)noc1C.c12nsc(n1)OCCN2 Cc1nc(N(C)C)sc1C(=O)NC1CC(CCNC(=O)C=CCF)C1 c1(C(C)NC(C2(O)CN(Cc3c(C)nc[nH]3)C2)=O)cccc(Br)c1 N1(c2c(OC)cc(Br)cc2)Cc2ccc(NC(=O)C(O)C(C)C)cc2C1 c1(C(N2CC(O)(C(C)NC(CC=CCC)=O)C2)=O)cccc(C)c1Br C1(NC(c2c(C(C)NC(c3c(C(=O)OC)csc3)=O)noc2)=O)CCS(=O)(=O)C1 c1(CNCC2CN(C(CC3C(C)CCC3)=O)C2)ccc(SCc2nc[nH]n2)cc1 N1(C(C(CC)COC)=O)C2CCC1C(C(N1CCC=CC1C(=O)OC)=O)C2 c1(OC2(C(=O)NOCCO)CCOC2)ccc(O)cc1.C1(=O)C#CCN1 C12(NC(c3c(CC)n[nH]c3)=O)CCC(C(=O)NC(C(F)(F)F)C3CCC3)(CC1)C2 C=C(C)CCC(=O)N1CCC(C(C)NC(=O)CS(C)(=O)=O)C1 C(=O)(C(C(C)NC(C1CCCC1O)=O)C(C)C)NCc1nccc(C)n1 c1(C=O)c(Cl)nc2ccccn12.n1(CC(C)NC)cc(CN2CC3CC3C2)nn1 C1(C(=O)OCC)CC2(CCC(CN(C)CC#N)O2)C1.c12cccc(n1)C2 CC1CN(C(=O)CC2CC3(CC3)CO2)CC1NC(c1cnc(O)s1)=O c1(CC(=O)NCCOCCCNC(c2cc(OCC)n[nH]2)=O)ccccc1C c1(C(=O)NC2(C)CC(NC(c3ccc(C(N)=O)s3)=O)C2)nccc(Cl)c1O CCCCCC(C)(C)C(=O)N(CC(C)(C)NC(C1CCCN(C(C)=O)C1)=O)C c1(C(=O)NCCCCC(C)NC(=O)C(F)C2CC2)cc(F)ccc1-n1cccn1 CC(C)C(F)(CNC(=O)CN1CCOC1=O)C(=O)NCc1cccc(O)c1 N1(C(C2CCCCC2)=O)CCC2(CC1)C(NC(C1CC(O)C1)=O)CS2(=O)=O C1(CNC(COC(C)(C)C)=O)CCCC1NC(=O)CCCc1ccsc1 C12(C(=O)NC(CN(C3CC3)CC)C)CCCN1CC(OC)C2.c1(C(=O)O)coc(C)n1 C1(CNC(CC2(NC(CNC(COC)=O)=O)CC2)=O)CNC(=O)CO1 Cc1cccc(OCCCCNC(=O)CONC(=O)OC2CC3CC3C2)c1 N1(C(C2(CC)CCC(O)CC2)=O)CC=CCC12CCC2 c1(C(=O)NC(CC(C)NC(COCCOCC)=O)C)cccn2c(C)cnc12 c1(C(CNC(C#C)CC2CC2)NC(=O)OC(C)(C)C)nnnn1C1CCC1 C1(OCCC(=O)CC(C)N)CCCCC1.C(=O)(CCN(C(=O)CC(C)(C)C)C)OCC c1(C(N2CCC(CNC(C(C)N(C(C)=O)C)=O)C2)=O)cc2c(nn1)CCCO2 c1(C(N2CC(NC(C(C=CCCC)O)=O)C(C(F)F)C2)=O)c(F)ccc(F)c1Cl N1(C(C2CCN(C(c3cc(N)c(Cl)nc3)=O)CC2)=O)CCC12CCOCC2 C(=O)(CCCCNC(=O)C(C1CCCO1)NC(=O)C(c1ccccc1)C)OCC N1(CCC(=O)NC)CCC(F)(C(=O)NCC23CCC(CC2)OC3)CC1 c1(C(N2CC3CN(C(=O)COCc4ccccc4)C3C2)=O)c(O)cc(F)cc1F c1(CN(C(C(CC(C)C)C)=O)C)cnn2c1CN(C(c1coc(Br)c1)=O)CC2 CCS(=O)CC(=O)NCC1(C(=O)NCCn2ccc(C(N)=O)n2)CCC1 Cc1ccc(Cl)cc1C(=O)NCC1CN(C(=O)CC=CC(C)(C)C)C(C)CO1 C1(C(C(=O)OC)C)CCCN1N1CC(C)(OC)C(C(=O)O)C1 CCCC(CCCNC(=O)Cc1ccsc1)NC(=O)C=CCOCCOCCO C(=O)(C(C(C)(C)C)c1cc[nH]n1)NCC(C)N(C(=O)CO)C C#Cc1ccc(Br)c(C(=O)NCCC2(O)CN(C(c3c[nH]nc3F)=O)C2)c1 N1(C(c2c(Cl)cnc(C)n2)=O)CC2OCC(NC(C3(CC(F)F)CC3)=O)C2C1 c1(C(=O)NC2CC(O)(CNC(C3CCC3(F)F)=O)C2)ccc(F)cc1Br c1(CNC(N2CCC(C(=O)Nc3ncc(OC)nc3)CC2)=O)ccc(F)c(Cl)c1 c1(C(=O)NCCC2(O)CN(C(C3OCCN(C)C3)=O)C2)ncnc(O)c1F O=C(CCCN1CCCC1)NCCC1(O)CN(C(=O)CC2CCC(=O)O2)C1 Cc1noc(C)c1C(C)C(=O)N(C)CC1C2CN(C(=O)COCC(F)F)CC12 c12cncc(c1)CNC(=O)C2.C(c1cn(C)cn1)=CC(=O)Nc1cn(CC)nn1 C1(C(=O)NCCSn2cnnn2)CC(OCCOC)CN1.C1=CCNC1=O C(=O)(C#CC1CCCOC1)NCC(C(C)C)NC(C1CC(=C)C1)=O N1(C(c2c(C)noc2)=O)CCOC2CCN(C(c3ccc4[nH]ccc4n3)=O)CC12 N1(C(C(C)OCCCC)=O)CC(NC(c2cc(CO)[nH]n2)=O)CC12CCCCC2 CC(C)CC(CNC(=O)C(C1CCOCC1)F)C(=O)N(CCC(N)=O)C c1(N(C)Cc2cccc(F)c2)nc2ccsc2c(=NCCNS(C)(=O)=O)[nH]1 C1(C(=O)OC)COCCN1C=O.C(=O)(CC1CN1CC)N(C)CC Nc1c(C(=O)NC2COCC2CNC(C2OCCC2C(C)C)=O)cc(Cl)cc1Cl C(c1cscn1)=CC(=O)NCC1(CN(C(C(C)=CC2CC2)=O)C)CC1 N1(C(C2(CCNC(c3n(C(C)C)cnc3)=O)CC2)=O)CCC(O)CC1C C1(NC(C(CC)COC)=O)CC2CCC1CC2NC(=O)COC1CC(F)(F)C1 C1(CNC(C(CCC)(C)C)=O)CC2CCCCC2N1C(=O)CCc1ncc(F)cn1 N1(C(CN(CCC)C(C2CC3CCC2CC3)=O)=O)Cc2c[nH]nc2C(C)C1 C(C(=O)N1CC(NC(=O)CN2CCOCC2=O)C(O)C1)(C(F)(F)F)OC(C)=O c1(C(N2CC(C)(C)OC(C)(C)C2)C(=O)NC)cc2c(Br)cccc2s1 c1(SCc2c(C)scc2)c(OC(F)F)cccc1Cl c1(CN(CCN(C(=O)CCc2cncn2C)C(C)C)C)ccc(C2CC2)c(F)c1 C12(NC(=O)Cc3ccccc3)CCOCC1CN(C(=O)CCC1OCCO1)C2 CC1CCCC1(C)C(=O)NCC1CC(NC(c2ccc(C3(C)CC3)cc2)=O)C1 C=CCC(C(=O)NC(C)CNC(=O)CCC(=O)Nc1c(F)cccc1F)C(C)C c12ccc(O)c(c1)OC2.C1(C(=O)OC2CCCCC2)CCCCC(=O)C1 C(=O)(C#CC(C)(C)C)NCC1CC(NC(c2cc(C(=O)OCC)sc2)=O)C1 CC(=O)C(C)(C)CC(=O)N1CC2COCC2(C(N2CCOC(CC(N)=O)C2)=O)C1 C1(NC(=O)CNC(N)=O)CC2(C(N3CCC(CCO)CC3)=O)COC1C2 Cc1ccc(CC(=O)NCC(O)CNC(C2(C)COCCO2)=O)c(Cl)c1 Cc1cc(C(=O)NCCC2CC(NC(C3(C#N)CC4(CC4)C3)=O)C2)nnc1C CC(CC(F)(F)F)C(=O)N1CCN(C(=O)C2=CCSC2)CC1CC(F)F c1(C(=O)NC(CCNC(c2cc(C(CC)C)no2)=O)C)cc(NC)ccc1F C1(NC(CS(N)(=O)=O)=O)C2CCCC1CC(NC(c1cc(=O)cc(Cl)[nH]1)=O)C2 C1(CNC(CC(=O)N(C)C)=O)CCN(C(=O)CCCN2C(=O)CNC2=O)CC1 CC1CCC(OCC(=O)NC2CCN(C(C3CCCN3S(C)(=O)=O)=O)C2)CC1 N1(C(c2csc(Cl)n2)=O)CC2CN(C(c3ncccc3C(F)F)=O)CCC2(CO)C1 CON1CCC(C(=O)NC2(CC(=O)NCC3CCSC3)CC2)CC1 Cc1nc(C=CC(N2CC(NC(c3ccncc3)=O)C(O)C2)=O)[nH]c1C N1(C(CC(CC)OC)=O)CC2CC(NC(C3CCN(C(=O)N(C)C)CC3)=O)C1C2 N1(C(c2cc(C3(C)CCC3)no2)=O)CCC2CN(C(=O)CCC(C)C)CCC12 C=C(Cl)CC(C(=O)NC(CC1CC1)CC1CC1)NC(c1cnc2n1CCC2)=O C1(CNC(C=Cc2nnn(C)n2)=O)CCN(C(C2CCCN2C2CC2)=O)C1(C)C N1(C(C(CC)C)=O)CC2CC(C1)N(C(C1CN(Cc3ccccc3)CCO1)=O)C2 c1(CC)ccc(C(=O)NCC(CC)NC(c2ccn(C)c2)=O)s1 N1(C(C#C)=O)CCC2(CCCC2C(=O)Nc2ccc(F)cc2C)C1 c1(CNC(C(=O)Nc2c(C)nn(C)c2)=O)ccc(Br)cc1I C(=O)(C1=NOC2COCC12)NC1C(NC(=O)C2=CSCCO2)COC1 c1(CC)nc(C)oc1C(=O)NCCOCCC(=O)N(C)Cc1occc1C CC(CCc1ccccc1)CC(=O)N1CCCC1CCNC(=O)C(=O)N(C)C C(C1=NOC2CCCC12)NC(C1(C)CCCN(C(c2cc(Cl)cs2)=O)C1)=O C1(NC(C(=O)N(C)C)=O)CCCC(NC(=O)CSc2ccccc2Cl)CC1 c1(C(C)NC(c2nnnn2CSc2ccccc2)C2CCOC2)nccc(Cl)c1F c1(CC)cccnc1C(=O)NCC(C1CCCCN1C(C1CCCC(C)C1)=O)(C)C c1(C(=O)NC2C3(CCC(NC(C(N)=O)=O)CC3)C2)c[nH]c2nc(F)ccc12 C#Cc1ccc(C(=O)N(C)CC2CC(F)CN2C(C2CN(CC)CCO2)=O)cc1 C1(CC)C(=O)N(C)CCN1C(C1C(CNC(c2ccc(OC)o2)=O)C1(C)C)=O Cn1ccc2c(-c3noc(CC4CCCCS4)n3)ncnc12 C1(CC(N2CC3CCC3(NC(=O)COC(F)(F)C(F)(F)F)C2)=O)CCC(F)(F)CC1 c1(C(N(C2CN(C(c3cc[nH]n3)=O)C2)C)=O)ccc2nnc(O)n2c1 N1(C(C(C)CF)=O)CCC(CO)(CNC(=O)C(C)CSCc2ccccc2)CC1 c1(CC2CC2C(N2CC(NC(C3(n4ccnn4)CC3)=O)C2)=O)ncc(CO)s1 CN1C(=O)CCCC1C(N1CCCC1Cn1cc(Cn2ccnc2)nn1)=O CC1CC2(CC(C(N3CC4CC(N(C(=O)Cc5cocn5)C)C3C4)=O)C2)C1 N1(C(C(COC)C(F)(F)F)=O)CCc2sccc2C1CNC(=O)CCCC(C)C CCCCCCC(C(=O)NC1CCCCC1C(=O)OC(C1(Cl)CC1)=O)NC(C)=O C#CCCCCCC(=O)NC1(C)CCN(C(=O)CSc2cc(C)ccc2C)C1 c1(CC)cc(Cl)ccc1C(N1CCC(NC(C2(OC)CCC2)=O)C1(C)C)=O n1(C(C)C)ccc(C(=O)NC(C)(C)CNC(=O)CCCC2CCOCC2)n1 CN1C(=O)CCC1C(N1CC(NC(=O)CCc2nccn2C)C(C(F)(F)F)C1)=O c1(C(=O)OCc2ccc(-c3cn(C)nc3)o2)cncc(OC(F)F)c1 Cn1cnc2cccc(C(=O)NC3CCC3NC(c3cnc(S)n3C)=O)c12 C1(CCC)(NC(C2C3(CC3)C23CC3)=O)CCCN(C(=O)Cc2cnns2)C1 CC(O)(CNC(=O)CCc1cnccn1)CNC(=O)CCC1CCCO1 N1(C(c2c(C)n(C)c(C(C)C)c2)=O)CCCC12CCN(C(c1ccoc1)=O)C2 C(C)(CCC(=O)NC1CCN(C)C1C)NC(C1C(CC)CCO1)=O C#Cc1ccc(C(=O)N(C2CCN(C(=O)OC(C)(C)C)C(=N)N2)CC)nc1C C1(NC(C(CCC)NC(N)=O)=O)CC2CC(NC(c3ccoc3CC)=O)C2C1 C1(C(=O)NCC2CC2NC(C2CCOC2)=O)(OC(C)C)CCC1 C12(CNC(CCNC(C)=O)=O)CCC1CN(C(c1cc3[nH]ccc3s1)=O)C2 c1(C(=O)NC(CCCC)CNC(c2ccncc2F)=O)cccc2c1COC2 c1(C(=O)NCCN(C2CC2(F)Cl)C(=O)C2CC2)cnoc1-c1ccccc1 C1(NC(CCSCCC)=O)CN(C(c2c[nH]cc2CC)=O)CCC12CCC2 C1(OCCNC(CCC=CC)=O)CCN(C(=O)CC(c2cccs2)C2CC2)CC1 C(=O)(CC(C)CC(=O)NC1CN(C(=O)C#CC(=O)N(C)C)CC12CC2)OC C1(NC(c2c(C)cno2)=O)CCN(C(c2csc(CC(C)C)n2)=O)C1C(C)C Cc1nn(-c2ccc(F)cc2)c(CNCc2nocc2C2CCC2)c1Br C(C(C)(C(C)C)NC(=O)CP(C)(C)=O)NC(CC1CC(NC(C)=O)C1)=O N1(C(C2C(COC)CC2)=O)CC=CC1(C)C(=O)NCCCNS(N)(=O)=O c1(CN2CCCC(NC(Cc3n(C)cnc3)=O)CC2)c2cc(Br)ccc2nn1C C1(C)(C(N(CCCNC(=O)CCCc2ncco2)C)=O)CCCCC1(F)F c1(CC(=O)NCC23CC(CNC(=O)Cc4ccc(Cl)cn4)(C2)C3)cccnc1O N1(Cc2ccc(CC)o2)CCN(C(=O)CN(c2ncnc(=N)[nH]2)C)CC1 N1(C(C2CC(OC)C2)=O)Cc2nccn2CC(NC(C2CCC2(C)C)=O)C1 c1(CC(C(=O)N(C)Cc2cnco2)NC(=O)CCc2cnccn2)cnn(C)c1O c1(C(C)C)nc2cc(n1)N1CCC(C1)CN2C.c1(SC(C)C)nccn1C c1(C(=O)NCC2(CNC(C3(C(F)F)CC(=C)C3)=O)CC2)ccc(Cl)c(S(N)(=O)=O)c1 C1(C(=O)NC(c2nc(-c3ccncc3)no2)C(C)C)CC2CCC(C1)C2(F)F N1(C(c2c(COC)cccc2)=O)CCCN(C(C2CC(=O)N(OC)C2)=O)CCC1 c1(COC(C(C)Cc2cccnc2)=O)ccccc1-c1cncnc1 N1CCCNCC1.c1(-n2cc(C3(C)CC3(Cl)Cl)nn2)ccc(F)cc1 c1(C(C)CNC(=O)C(=O)N(CC(C2CCCCC2)F)C)ccc(Cl)cc1 Cc1cc(C)n2nc(C(=O)NCCC3CCN(C(C4CCCS4)=O)C3)nc2n1 c1(NC(C2N(Cc3ccc(NC=O)cc3)CCSC2)=O)ccnc2ncnn12 c1(CC(=O)NC(CC(C)NC(C2CC2)=O)C)ccncc1Cl.c1(C)cnc[nH]1 c1(C(=O)OC)cncc(S(=O)(=O)NC(c2ccc(Br)cc2F)(C)C)c1 CCC(C)C(C)C(=O)OCC(=O)N(C1CC(F)(F)C1)C1(CS(C)(=O)=O)COC1 C1(=O)CCN(OC)C(=O)C(CO)N1.CCC(CC)n1ccnc1 C=C(C)C(C)(C)C(=O)NC1CCC(C(=O)NCC(O)C(N)=O)C1 N1(C(C2(CC)CCN(C(c3cc(C)c[nH]3)=O)C2)=O)CCCC(C)(C)C1C c1(C(=O)NC2CC(C)N(C(=O)C(N)=O)C2)cc([N+](=O)[O-])c(F)cc1N C1(CCOC)CN(C(C2CC2C(N)=O)=O)CCN1C(=O)Cc1ccco1 C1(NC(C2OC3CCC2C3)=O)CCC(NC(C2C(Cl)(Cl)C23CC3)=O)CC1 c1(OC)ccc(C(C)C(=O)NCc2cnn(C)c2CNC(=O)C(C)O)cc1 N1(C(CN(C(Cc2c(C)ccs2)=O)C)=O)CCN(C(c2nnn(C)n2)=O)CC1C Cc1nnc2n1C(C(=O)NCC(C1CC1)NC(c1ccn3cncc3c1)=O)CC2 n1(CC)nc(C(=O)NCC2C3CC3CN2C(C2CC2F)=O)ccc1=O C1(NC(c2c(C)snc2)=O)CCN(C(=O)C(C)CC(C)C)CC(C)(C)C1 N1(C(C(C)NC(=O)C=Cc2ccccc2)=O)CCCN(C(=O)CSCC(N)=O)CCC1 C=CC1(CNC(=O)C(CC)NC(c2nc(Cl)cs2)=O)CCC1 Cc1cc(NC(C23CC2CN(C(=O)C#CC2CC2)C3)=O)cnc1C C1(CC)(CC)CN(C(=O)CC(C2CC2)NC(=O)CCC2CCC(=O)C2)CCO1 c1(C(N2C(C(=O)NCCOc3cccnc3)CC(OC)C2)=O)ccc(O)cc1Cl C(=O)(C(C)(C)CC(C)(C)C)NCC(C)N(C(CCOC(C)C)=O)C CN=c1nc(C(=O)NCC2CCCN2C(=O)CN2CCC(C)(C)C2)cc(C)[nH]1 C=Cc1cncc(C(=O)NC2(CCC(N3CC4CC(C)(C)C3C4)=O)CCC2)c1 N1(C(c2ccc(C(OC)OC)o2)=O)CCC(F)(CNC(=O)Cn2c(C)csc2=O)C1 C1(NC(CCc2onc(C(C)OC)n2)=O)CN(C(c2[nH]c(C)nc2C)=O)CC1C c1(OCC)ccnc(NCC(N2CCC(C)(NC(C3CCCSC3)=O)C2)=O)n1 C12(C(N3CCCN(C(CC4OCC(C)OC4)=O)CC3)=O)CCC(N=[N+]=[N-])C1C2 Cc1ncc(Cl)cc1OCc1nc(C(C)C)n(-c2cccc(Br)c2)n1 Oc1ccc(-c2ccc(-c3nccn3C3CCNC3)nc2)cc1F C#CC1CCC(NC(c2ccc(CNC(c3ccc(C(N)=O)[nH]3)=O)nc2)=O)C1 c1(COC)cc(C(=O)NCCC(C)(C)CNC(=O)C(C)OC)ccc1OC1CC1 C1(C(=O)NC(CCCC)COC)CC(F)CCN1C(c1cc(C2CC2)[nH]n1)=O c1(OC)cc2nn[nH]c2cc1C(=O)NC1CC(NC(=O)CCC(C)(C)C)C1 Cc1nc2c(C(N3CC(NC(c4cn(C)c(C)n4)=O)CC3CO)=O)cccc2o1 Cc1c[nH]c(C(N2CCCC2(C)CNC(c2cnn(C(F)F)c2)=O)=O)c1C c1(OC)c(C)cc(NC(=O)CC2(O)CCN(C(c3ccc(C)o3)=O)CC2)cc1C N1(C(C(CSC)O)=O)CC2(CCC2)CC1C(N1CCc2sccc2C1)=O CC1(F)CN(C(c2ncn(C(C)(C)C)n2)=O)CCN(C(C2(C)CC2(F)Cl)=O)C1 c1(C(=O)NCC2(C)CCCN(C(c3cc(CO)on3)=O)C2)ccc2ncnn2c1 N=c1[nH][nH]c2ccc(C(N3CCCCC(NC(c4ccc(S)cc4)=O)C3)=O)cc12 C1(O)(C(=O)NCC2(CC)CCCC2)Cc2ccccc2C1.N12CC3(CC1C3)C2=O N1(C(C2OCCN(S(C)(=O)=O)C2)=O)Cc2ccccc2-c2ccccc21 n1(CCN=C(NC2C(C)C2)NCc2csc(Br)c2)ccc2c(F)cccc12 c1(C(=O)OCC2CC(c3ccccc3)C2)cc(=O)cc[nH]1 Cc1ccnc(C(=O)NCC2(C(F)F)CCN(C(C3(C)CC3C)=O)C2)c1N C1(NC(CC2(C)CN(C(C=CC=CC)=O)C2)=O)C=CC(C)(C)CC1 CC1C(NC(c2snnc2C2CC2)=O)CCCN1C(c1cc(C2CC2)on1)=O C(CN=C(NCc1ccnn1C)N(C)Cc1ccsc1CC)CC Cc1sc(C(=O)NCCCNC(=O)C(c2cccc(Cl)c2)N(C)C)c(C)c1C CCCN=c1[nH]c(=NC2CCCCN(C)C2)[nH]c2ccc(OC(F)(F)F)cc12 C1(C(=O)NC2C(NC(c3n[nH]c(CC)c3C)=O)COCC2)CC2OC1C1CC21 N1(C(Cc2cn(C)nn2)=O)CC2CCCC(NC(c3cnc4sccn34)=O)C2C1 c1(C(=O)NC2(C)CC(NC(C3COCC(C)O3)=O)C2)ccc2nccnc2n1 Cc1nc(CNC(=O)C(CN(C)C)NC(=O)CC23CCCC2C3)sc1C c1(C(=O)NCC(C2CC2)NC(C(C)(C)OCC)=O)cc2c(F)ccc(F)c2s1 n1(CC(=O)NCCC2CN(C(C3(Cl)CC3)=O)CCO2)ccc2ccccc12 CC1CC(C)(C(=O)NC(CCN(C)C(c2ccoc2)=O)c2cccs2)C1 N1(C(c2c(C)nns2)=O)CCCC2(CCN2C(C2CCC(O)C2)=O)C1 C(=O)(C(F)C(F)(F)F)NCC(c1ccccc1CC)NC(CCOCCC)=O CCCCCC(O)C(=O)NCc1ncccc1C(N1CC=CC(OC)C1)=O N1(CCC)CCCC1C(=O)NC(C)CCNC(c1cnoc1C1CC1)=O C(C(C)CC(=O)NCCCC(C)NC(=O)CSCC(c1ccccc1)=O)OC C1(C(=O)NCC2N(C(C=CC(C)=O)=O)CC(F)(F)C2)CCOC2(CCCC2)C1 CC(C)CS(=O)(=O)CCC(=O)N1CCC(C(C)NC(=O)CC(C)(F)F)C1 N1(C(COC(C)=O)=O)CC2C(NC(c3ccc(CF)cc3)=O)C2C1 c1(OC)ccccc1C=CC(=O)NCC1CC(NC(c2ncccc2CO)=O)C1 Cn1ncc2c(=O)n(C(=O)N3CCn4nccc4C3)c(C(F)F)nc12 N1(C(COCCC(C)(C)CO)=O)CC2CCC(O)CC2C1 c1(C(N2CCCC(CNC(C3C(OCC)C3)=O)C2)=O)cc(C)ccc1F c1(C(=O)NCCc2ccsc2)n[nH]c2c1CN(C(C1CC1Cl)=O)C2 O=S(=O)(c1ccc(NC(c2ccccc2)CO)c(Cl)c1)N1CCC=C(F)C1 CC(C(=O)NCCCN1CCC1)NC(=O)C(C)n1cncn1 C1(C(=O)NC(CNC(c2cc(=NC)[nH]cc2)=O)COC)CC(C)(C)OC1(C)C C12(NCCc3nc(C(C)C)sc3)CCCCC1C2Br C1(CC(=O)N(CCC)CCC(=O)COCCCCC)CCCC1C.N CCCCC(C)C(=O)N1CC(NC(=O)CCCN(C)C(=O)OC)C2(CC2)C1 N1(C(C(N(C)O)=O)=O)CCC(O)(CNC(=O)C(F)OC(F)(F)F)CC1 C1(CNC(C(n2ncc(C)c2)C)=O)CCCN(Cc2cc(C)n(C)n2)C1 c1(CC)cc(C(=O)NCC2(O)CC(NC(=O)CCC3CC(F)(F)C3)C2)c(C)nn1 c1(CC(=O)NCCCN(C(c2c(C)n(C)cn2)=O)C(C)C)csc2nccn12 CC(C)(C#N)CC(=O)NCC1(C)CN(C(c2cc(C3CC3)no2)=O)CCO1 c1(CNC(C(=O)NCC(CNC(C=C(C)C(C)C)=O)C)=O)ccc(F)cc1 N1(C(C=CCC)=O)CCCC(F)(CNC(c2n(CC(=O)NC)cnc2C)=O)C1 c1(CN(C(CCCOC)=O)C)cnn2c1CN(C(=O)C(C)S(N)(=O)=O)CC2 c1(CCCCC(=O)NCCN(C(C2(F)CC2)=O)C2CC2)nc2ccccc2s1 C1(NC(c2occ(C(=O)OC)n2)(C)CC)CC2OC(=O)CC12 Cc1cn2c(C=CC(=O)Nc3cnc(C#N)cn3)c(C)nc2s1 C=C(C)CC(C(=O)NCCOCC(C)(C)O)NC(c1cc(C(C)C)no1)=O CCC(CC(=O)NCC1(F)CC(NC(=O)Cc2ccc(F)cc2)C1)C(C)(C)C C1(CC(N2CC(CSC)C2)=O)CC(F)CN1C(C1CC12CC2)=O c1(C(=O)NCC2(O)CC(NC(c3cc(CCC)on3)=O)C2)n[nH]c2c1CSCC2 C(=O)(C1=CN(C)S(=O)(=O)N=C1C)N1CC(CC)(NC(C2CS(=O)(=O)C2(C)C)=O)C1 c1(C(N2CCC(OCC(=O)OC)C2)=O)cc(C#N)ccc1O C#Cc1cc(C(N2CCC(C)c3ccccc32)C(=O)NC)cc(C#C)c1 C(=O)(C(CN=[N+]=[N-])NC(c1ccc(C(C)C)o1)=O)NC1(C(=O)OC)CC(C)(C)C1 N1(C(c2ccn(C(C)(C)C)n2)=O)CCC(CO)CC12CC2 c1(CC(N2CC3(CN(C(c4ccc(C)cc4)=O)C3)C2)=O)cc(C)c(Cl)c(C)c1 C(CN=c1[nH]ccc(=NC2CC2c2ccc(C)c(C)c2)[nH]1)n1c(C)cc(C)n1 N1(C(C2(NC(C3C(C)CC3)=O)CC(O)C2)=O)CCCCCC1 c1(C(=O)NCC(CC)(C)NC(=O)C(C)=CC(C)(C)C)ccc(C)c(F)c1 N1(C(CSCC)=O)CCCC2(CNC(=O)C=C3CCC(C)CC3)CCCC12 Nc1ccccc1CCCC(=O)N1CC(F)(CNC(C2CCC(O)CC2)=O)C1 c1(C(N2C(CC)C(NC(c3cnncc3C(F)F)=O)CC2)=O)ccc(Cl)cc1O C=CCC(CNC(=O)C#CCNC1CSCN1C(C)=O)NC(=O)C1CC1 N1(C(CN(C(=O)OCC)C)=O)CCCC(CCC(=O)NCC(O)CC)C1 C(=O)(C1=NN(C)C(=O)CC1)NCC1(O)CCN(C(C=C2CCC(C)C2)=O)C1 C1(C(=O)NCC2OCC(CNC(CCC#C)=O)C2)CC2(C1)CC(C)(C)C2 N1(C(c2ccc(NC3CCC3)cc2)=O)CC(CO)CC(N=c2[nH]c(Cl)ncc2Br)C1 C1(C(=O)OC)(NC(C2CC(N(C)C)C2)=O)CCN(C(=O)C(C)Cc2ccco2)C1 c1(OC)ccc(C(=O)NCc2cc3ccccn3c2)c(Br)c1F N1(C(c2nc(C)oc2)=O)CC2CCCC1C2CNC(=O)CCOCC(F)F c1(C2C(C(N(CCC)CCNC(=O)CN(C)C(N)=O)=O)C2)nnnn1CC(C)C C1(C(N2CC(C)(CC=C)C2)=O)CCCCC1(C)NC(C1CCC1)=O CN1CCC(C)(C(=O)NCC23CC2CN(C(=O)CC2CSCCO2)C3)CC1 C(=O)(C(C)(C)C(N)=O)NCc1ccc(C(C)NC(c2[nH]cc(CC)c2)=O)cc1 C=CC(CC)C(=O)NC(CO)C(C)NC(c1cnn(CC)c1CC)=O N1(C(COCCSC)=O)C(C)CC2CN(C(=O)CCn3cccc3)CC12 c1(CC(C)C)ccn2ncc(S(=O)(=O)N(C3CCC3(C)C)CC3CCC3)c2n1 c1(C(N2CCCC(N(C(=O)CCC3(C)CC3)CC)C2)=O)c(F)ccc(C#N)c1F c1(C(=O)NC2CC(CCNC(c3n(C)c(O)nc3)=O)C2)cccn2nnnc12 C1(F)(CNC(C(c2ccc(F)cc2)OC)=O)CCN(C(=O)CC2CCC(=O)N2)C1 C(CNC(c1cccc(COC)c1)=O)(C(C)(C)C)NC(c1c(CCC)nns1)=O c1(C(=O)NC2C(NC(C=CC(CC)=CC)=O)C2)ccn(C2C(C(C)=O)C2(C)C)n1 c1(NC(C2CC(NC(CC(CC)O)=O)C2)=O)ccc(C)c(C#N)c1 Cc1cc(F)c(C(N2CCC3CCC23CNC(=O)C=CC(F)(F)F)=O)cc1F O=C(CCCCCCNC(=O)CC1CCCOC1)NCc1cccc(F)n1 C1(NC(c2ccnn2CCF)=O)CCCCC1CNC(C1CCCO1)=O CC1(C)C(NC(c2ccc(F)c(C(F)F)c2)=O)CCN1C(C1CC2(CCC2)C1)=O C1(CNC(CC=C=C)=O)CCN(C(C2(COCC)CC=CC2)=O)CC1C Cc1nc(F)ccc1CN1CC(O)C(F)C1.c1(CN)cc(Cl)ccc1C=O C1(C(=O)NCC2(CNC(c3cccc(SC)n3)=O)CC2)CCn2c(cnc2C)C1 N1(C(C(C(=O)OC)C)=O)CCCN(C(=O)Cc2ccc(F)c(Cl)c2)C(C)C1 c1(OC)cc(C(=O)NCC2COCCN2C(c2c[nH]cc2C)=O)cc(C2CC2)c1 C1(NC(CC(CC)C)=O)CC2CC(NC(c3cc(CO)[nH]n3)=O)C1C2 CN1CCC2(c3nnc(O)n3C)CCCCC2(C2CCC2)C1 C1(CCNC(C2CS(=O)(=O)C2)=O)CCN(C(=O)CC23CCC(CC2)C3)CC1 C1(NC(CSCCCC)=O)C(C)CN(C(c2occc2CC)=O)CC1C C1(C2CC2)(OC)CN(C(=O)C(C)(C2CCC2)NC(c2ccn(C(C)C)n2)=O)C1 Cc1nn(C)c2cc(NC(=O)CC3CCC(C)C3)ccc12 C(C1C(C(=O)N(CC(C)N(C(=O)CCSC(F)(F)F)C)C)C1(C)C)=C(C)C N1(C(C2CCOCC2)=O)CCN(C(C23CC(O)C2C3)=O)CC1CO N1(C(C2C(CCC)C2)=O)CCOC2CN(C(=O)C(C(C)C)n3cc(C)cn3)CC12 C=CCC(C(=O)N1CCC(C(C)(C)C)C1)NC(c1ccc(OCC)nc1)=O c1(OCC(N2CCC(N(C)C(C3CCC(F)C3)=O)C2)=O)ccc(F)c(Cl)c1 c1(OC(C)(C)C)ccc(C(N2CC(NC(=O)C=C3CCCCC3)C3CC23)=O)cc1 C12(NC(C(C)OCC)=O)CC(C)(C1)OC21CCN(C(C2CCC(F)(F)C2)=O)CC1 c1(OC)ccc2c(c1)CCCC2C(=O)NC12CC(NC(=O)CO)(C1)C2 c1(C(=O)NCC(=CC(=O)NCC#C)C)nnsc1N c1(C(=O)NC2CCC(C)(CNC(C3(SCC)CC3)=O)C2)cc2c(cc1N)OCO2 c1(CNC(c2nc(CNC(C=C(C)C(C)C)=O)oc2C)=O)cncc(C#N)c1 N#Cc1ccc(Cl)c(C(N2CCC3(CNC(c4cscn4)=O)CCCC23)=O)c1 CC(C)C(C)(CNC(=O)CCCN1C(=O)CNC1=O)NC(C1CC=CC1)=O C(=O)(C(C)(C)CC(F)F)NC(CN(c1cccc(C)c1C)C(C)=O)CC N1(C(=O)OCC)CCCC(C(=O)NC23CC(NC(=O)CCCN(C)C(C)=O)(C2)C3)C1 c1(C(N2CC3CN(Cc4c(Br)cn(C)n4)C3C2)=O)ccc2c(c1)CCO2 C(=O)(C(F)(F)F)NCC(=O)NC1CCN(C(=O)C(O)c2ccco2)C1 Cc1ncnc(C(=O)NCC2(F)CN(C(=O)C(c3ccccc3)F)C2)c1C Cc1cccc2[nH]cc(CC(N3CCC(C)C(NC(=O)C(F)F)C3C)=O)c12 C=CCCCC(C(=O)NCC1CCCO1)N1CC(F)(F)CC1CC(=O)OC Cc1cc(C(=O)NCC2(F)CC(NC(=O)CCC(C)CN(C)C)C2)c(O)nc1C c1(CNC(=O)CO)ccc(C2CCCN2)c(F)c1 c1(OCC)ccc(Cl)cc1CC(=O)NCCCCN(C(=O)CCC(=O)NCC)C C1(=O)C(CC2CCC2)N1C1CC1.C(=O)(CCNC(C)=O)NCC#CC C1(C(N2CCCC(COC)C2)=O)CC2C=CC1N(C(c1cnc(=N)[nH]c1)=O)C2 N1(C(c2csc(C(F)(F)F)n2)=O)CC2(CCN2C(c2ncccc2Cl)=O)C1 C(=O)(CCCN=[N+]=[N-])NCCN1CCNC(=O)C1.CC12CC(C1)C(=O)N2 N1(C(C=CCCC)=O)CCN(C(C2OCC2(C)C)=O)CC1c1ccc(F)cc1 N1(C(c2[nH]c(=N)sc2)=O)CCCC(C2CC2NC(c2nc(C(C)C)ncc2Cl)=O)C1 C1(C(N2CC(C(N(C)CC34CCC(CC3)CC4)=O)OCC2)=O)CC2(CCC2)CO1 c1(CC)cc(C)nc(N(C)CC2CCCCN2C(C2CC(=O)N(OC)C2)=O)n1 N1(C(C2(C)CC=CC2)=O)CCCC(CO)(NC(c2ccnc(O)c2)=O)C1 c1(C(=O)NC(CCNC(C=C(C)C(C)C)=O)(C)C)ccc2cnoc2c1 c1(C(N2CC(CNC(C3CCC(=C)CC3)=O)C(C)C2)=O)ccc2[nH]ccc2c1 C(=O)(C(C)(C)C(C)(F)F)N1CCN(C)CC1CNC(C1(CCO)CC1)=O c1(CN(CCC(=O)Oc2ccc(C)cc2F)CC)cccc(OC(C)(C)C)c1C C1(C(=O)OC)(NCCC(O)CN)CC=CCC1 N1(C(C(CCC)=CCC)=O)CC(NC(C2CCC3(CC3)C2)=O)CC12CCCC2 C1(C(C)NC(=O)CC2CC=CC2)CCN(C(c2cccn2C)=O)CC1 c1(OC)ccccc1OC1CN(C(=O)CC2(N)CCSC2)C1 N1(C(C2CC(C)(CC)C2)=O)CCC(CC(=O)NCc2ccc(C)cc2C)C12CC2 Cc1ccc(C(N2CCOCC2CCNC(=O)C(O)C(C)C)=O)c(=O)n1C C1(C(CC(C)C)N(C)C)CCC(C)CC1CCC(C)C C(=O)(C1=CC2CCCCCC12)N(C)CC1COCCN1C(c1occc1Br)=O C(=O)(CC(C)C(F)(F)F)NC1C(CNC(c2c(-c3ccc(C)o3)onc2)=O)CC1 c1(CN2CC(C(=O)NCCC(C)C)C(F)(F)CC2)cccc2cccnc12 CS(=O)(=O)c1ccc(C(O)Cn2cc(Cc3cccc(C(F)(F)F)c3)nn2)cc1 C1(N(C)C(c2ccc(C(F)F)o2)=O)CCC(NC(=O)NC(C)(C)C)CC1 N1(C(C(=O)N(C)C)=O)Cc2nccn2CC(NC(C2(F)CCC(F)(F)CC2)=O)C1 CN1CC(C)(NC(CCCN2CCC(NC(=O)CC(C)(C)O)CC2)=O)CCC1=O c1(C(=O)OC)cc(C)cnc1NC1CN(C(=O)C(C)(C)C(C)C)CC1C C1(NC(C(CC)Sc2nc(=N)[nH][nH]2)=O)CN(C(C2(N(C)C)CCC2)=O)CC1C c1(C(=O)NCC2OCCN(C(Cc3cncc(C)c3)=O)C2)cccn2ccnc12 N1(C(C(=O)N(C)C)=O)CCC2(CCCCC2NC(=O)CC(C)(O)C(F)(F)F)C1 N1(C(CNC(CCCC)=O)=O)CCN(C(=O)CC2(n3cncn3)CC2)C(CO)C1 c1(C(CNC(c2ccc(-n3c(C)cc(C)n3)cc2)=O)F)cccc(F)c1F c1(C(N(CCNC(c2cnccc2Cl)=O)CC)=O)cn2ncnc2nc1C C1(c2cn(CCOCC(C)C)nn2)COCCN1C(c1ncn(C)n1)=O C(=O)(C1=CC2CCC=CCCC12)NC1CN(C2CN(CCC)C2)C(=O)C1 N1(C(C2(C(=O)OCC)CC2)=O)CCC(F)C(NC(=O)CCOCC(F)(F)F)C1 C1(NC(c2cc(C3CC3)[nH]n2)=O)CCCC2CN(C(C3CCCCS3)=O)CC12 c1(NC(N2CC3(CN(C(c4c(C)cc(F)cc4)=O)C3)C2)=O)cc(C)cc(C)c1C CC1CN(C(c2cncn2CC(F)(F)F)=O)CC1NC(c1cn(CCF)nn1)=O C12(NC(CC(COC)(C)C)=O)CCN(C(C3CC(C)(C)C3)=O)CCC1C2 C=CCC(CC(F)F)C(=O)N(C)CC1(O)CCCN(C(=O)CCC(C)CC)C1 N1(C(C2(C#N)CC3CC3C2)=O)CC(NC(c2cnc(O)s2)=O)CC(F)(F)C1 Nc1ccc(S(=O)(=O)NCCCC(=O)NC(C2CCCCN2)C2CCC2)cc1 N1(C(C(CC)(O)c2nn[nH]n2)=O)CC(NC(=O)CCC2CCOC2)CC(F)C1 C1(C(=O)NCCNC(=O)CC2CCCNC(=O)C2)CCC(C2CCC2)CC1 c1(C(N2CCOC(C(C)C)C2)C(=O)NCCCC)ccc(COCC)cc1Br C(c1cn[nH]c1)=CC(N1CCCC1CC1(C(=O)NOCC2CC2)CC1)=O CC1Cc2cccc(O)c2N(C(c2ccc3ccccc3c2)=O)C1 c1(CC)ccc(CN(C(=O)NCCC(C)Oc2ccccc2)C(C)C)o1 C1(CNC(CCS(C)=O)=O)CCN(C(=O)CSCc2cccs2)C12CC2 C12CCN(C1)C(=O)CCOC2=O.c1(CN(C(C(C)SC(F)(F)F)=O)C)ccccc1 n1(CC)ncc(Cl)c1C(=O)NCC(F)CNC(C1CC(CF)C1)=O C1(NC(c2c(-c3cn(C)nc3)[nH]cn2)=O)CN(C(=O)C2=CCCOC2)C2(CCC2)C1 Cc1noc(Cl)c1CC(=O)N(C)CC1CCCC(NC(=O)CC2CCOCC2)C1 CCCC(CCNC(C1OCCC1CNC(c1occc1C(C)C)=O)=O)CCC N1(C(c2c(C)cccc2C)C(=O)NC(C)(C)C)CCSC2(CCCCC2)C1 CC1CCOC(C(N2CCC2CNC(c2ccc(Cc3nc[nH]n3)cc2)=O)=O)C1 C1(C(=O)NCC2CN(C(CCn3c(C)ncc3)=O)CC2C)CCc2nn[nH]c2C1 c1(C(C(=O)NC(C)C)N(CC(F)F)CCC)nscc1Br CC(C)(C(=O)NCC(O)(C(F)(F)F)c1ccccc1)C(=O)N1CCC1CF Cc1c(Cl)ccc2[nH]c(C(N3CCCN(C(C4CCOC4)=O)C(C)C3)=O)cc12 N1(C(CC=CC=C)=O)C2CCC1CC(CNC(c1cc(O)nc(Cl)c1)=O)C2 c1(C(=O)NCC2N(C(c3cncc(-c4ccncc4)c3)=O)CC2)cccc(O)n1 c1(N2C(C)CCC(NC(=O)C(C)(C)O)C2)nc2cccc(Br)c2o1 C(=O)(C1CCC(=O)c2ccccc21)N(CC(C)(C)NC(Cc1scc(C)n1)=O)C CC(CC(=O)NCCCCC(=O)N1CC(C)C(O)C1)C(F)F c1(C(=O)NCC2C(NC(c3cnsn3)=O)COC2)cncc2c1CCC2 CCC(F)(F)C(=O)NCCC1CCN(C(c2ccnc(OCCOC)c2)=O)C1 Cc1cc(N(C(C)CNC(=O)C(C)C(C)S(C)(=O)=O)C)n2ncnc2n1 CCCCC(C(=O)N1CCC(F)(CNC(c2c(C)cccc2O)=O)CC1)C(C)C S(=O)(=O)(c1ccc2c(c1)C(=O)NC2=O)N(C(C#C)C1CCC1)C c1(C(N2CCCCCC2COC)C(=O)NCCOCC)cnc2ccccn12 C1(CCC=O)COCCN1C(=O)C(C)C.Cc1nc(COC)cs1 N1(C(Cc2c(C)non2)=O)C2CCC1C(NC(c1scc(Cl)c1Cl)=O)C2 C=CC(C)(CCOC)C(=O)NC1CCCN(C(c2cnc(CC3CC3)s2)=O)C1C CCCCC(C)C(=O)NC1CC(OCC(=O)NCCC2CCCC2O)C1 c1(N(CC(=O)NCCC2CCN(C(C3CCCN3C)=O)C2)C)ccc(Cl)cc1 c12ccc3c(c1)OCCN3C(=O)OC2=O.c1(OCC(=O)OC)ccc(C)c(C)c1 Cc1ccc(C(=O)NC2COCCN(C(c3cn(C)nc3C)=O)C2)c(I)c1 O=C(C1CCCCCc2ccccc21)NC1C2CN(C(c3cnn[nH]3)=O)CC12 Nc1c(F)cc(C(N2CCN(C3CCN(C(C4CSC4)=O)CC3)CC2)=O)cc1F c1(NC2CCN(C(=O)OCC)CC2OC)ccc2ncc(Br)cc2c1 CC1CCN(C(c2ccc(N)cc2)=O)CC1NC(=O)CCNC(C1SCCS1)=O CCC(C(=O)NCC(C)(O)CNC(c1cn(C)[nH]c1=N)=O)C(C)(F)F N1(C(=O)C#CC2CC2)CC2(CNC(C3(CCN4CCCCC4)CC3)=O)CC1CO2 N1(c2ccnc(COC)n2)CCn2ncc(CN(C(=O)C(C)(C)CF)C)c2C1 Cc1cnn(CC(N2CCC(C3CCCN3C(=O)CC3CCCSC3)C2)=O)c1 c1(C(=O)NCC(C)NC(=O)CC2COCC(C)(C)O2)c2c(nn1C)CCSC2 N1(C(C2CCCO2)=O)CCC2(c3nn[nH]n3)CC2C1.C(CO)C(=O)O C(=O)(C(Cc1cnc[nH]1)NC(=O)CC(C)F)NC(c1cnnn1C)C c1(C(=O)NCC2(NC(CN3CC(C)C3)=O)CCC2)cnc2c(ccn2C)c1 c1(N(c2ccc(O)c(O)c2)C2CCCN(C(C3(SC)CC3)=O)C2)ccc(C#N)nc1 C1(O)(CCOC(C(Cc2ccccn2)NC(=O)OC(C)(C)C)=O)CCCN(C)C1 c1(C(=O)NCC2(C)CC(NC(c3c(OC)ccs3)=O)C2)cccc(C2CC2)n1 C1(C(=O)NC(CCC)c2ccco2)(NC(=O)Cc2cncn2C)CC1(C)C N1(C(C2CCCN(C)C2)=O)CCC(F)(C(N2CCCC(CC3CC3)C2)=O)CC1 N1(C(C(CCC)NC(C)=O)=O)CCN(C(=O)CC2=CCCC2)C(c2ccccn2)C1 C1(C(=O)N)C2CCC(C2)C1NC(c1cc(Cl)n(CC2CC2)n1)=O.C1(SC)(CN)CCC1 C1(CC)CCCCCCN1C(C1CCN(CC(N2CCCC(C)C2)=O)C1)=O C1(NC(c2ccc(C)nn2)=O)C2CC1CN(C(=O)C(F)(F)c1ccccn1)C2 c1(C(N2CCC(C)(NC(CCN(S(C)(=O)=O)C)=O)C2)=O)nc(Cl)ccc1N Cc1[nH]c(C(=O)Nc2ccnc(Cl)c2I)c(C)c1C(N1CCC(F)(F)CC1)=O N1(C(c2c(CC)n(C)nc2)=O)C2CCC1CC(NC(C1CCN(CC)C1)=O)C2 C1(CNC(c2cccc(C(C)C)c2)=O)(NC(c2cscn2)=O)CCCCC1C c1(C(=O)NCC(C)N(C(C(CC)O)=O)CC)cccc(-n2ccnc2O)c1 Cc1[nH]nc2c1CCC(CNC(=O)NC(c1ccccc1Br)CCO)C2 c1(CCNC(C2(NC(=O)CCc3ccoc3)C(C)(C)C2)=O)ccc(O)nc1 C1(C(=O)NC(CCC=C)C2CC2)CC12CCN(C(=O)CCNc1ccccn1)CC2 Cc1nsc(C(=O)N(C2CCN(C(=O)Cn3nccn3)C2)C)c1Br C1(NC(CC=C=C)=O)CC(NC(c2cnc3[nH]cncc2-3)=O)C12CCOCC2 c1(C(=O)NCCC(C)N(C(C(C=C)O)=O)C)cnc2ccccc2c1 Cc1nc(C(=O)NC(C)C(=O)N(C2CC(C)C2)C)ccc1C#N c1(OC)cccc(S(=O)(=O)N2CC3C(C2)N3c2ccnc(C)n2)c1 c1(CCSCC(=O)OC)ccncn1.C12(CCCO1)C(=O)N1CC(C1)OC2 N1(C(c2c(C)scc2)=O)CC(NC(=O)CC2CCSCC2)C(O)C1 N1(C(C)=O)CCCCC1C(=O)NC1CCC(CNC(c2cc(CCO)on2)=O)C1 c1(OC)cncc(C(=O)N(CC(=O)NCCC2CC(C)(C)C2)CC(C)C)c1 Cc1ccc2occ(C(=O)NC3CCCN(C(=O)C#CC4CCCO4)CC3)c2c1 C1(NC(Cc2c(C)non2)=O)CC(O)CN(C(=O)Cc2ccc(F)cc2)C1 c1(NC(=O)COCCCN(C)C)cccc2c1CCO2.Cn1nnc2c1CNC2 CCCC(CCCNC(=O)C=Cc1ccsc1)NC(=O)CS(=O)(=O)NC c1(C(=O)NC23CC(NC(C=COCC)=O)(C2)C3)cnn2cnc(Cl)cc12 N1(C(CC(=O)NCC)=O)CC(C(=O)NC(CC)C(C)O)C(C2CC2)C1 N1(C(c2cc(C(C)=O)on2)=O)CC(F)CC1CNC(=O)CC(C)(C)N(C)C C1(COC)CN(C(c2csc(O)n2)=O)CCN1C(=O)C1=CCCSC1 Cc1cc(=NCC2(c3ccc(F)c(F)c3)CCC2)nc(-c2ccccn2)[nH]1 C(=O)(CCC(=O)NN(C)C)NCC(CC=C)NC(c1cc(CO)ccn1)=O C(CC(C(C)(C)C)NC(C1(CCF)CC1)=O)N(C(CC1C=NN(C)C1=O)=O)C CC1CCC(CNC(c2ccc(C(N)=O)cc2)=O)CN1C(c1n[nH]c(=N)s1)=O C1(NC(c2n[nH]c3c2CC2CC32)=O)CCCCN(C(c2cccs2)=O)CC1 C1(C(=O)NCC2N(C)CCC2)C2CCC(C2)C1NC(c1ccoc1)=O N1(C(=O)Cc2cc3ccccc3o2)CCN(C(c2ccsn2)=O)C2(CCC2)C1 C#CCCCC(=O)NCCc1ccc(CNC(C2C3CN(C)CC23)=O)cc1 Cc1cc(=NC(=O)CC2(C)CCCN2C(c2nc(O)sc2C)=O)[nH]n1CCO CC1=NN(C)C(=O)C1CC(=O)N(CC(O)CN(C)C(c1ccnnc1)=O)C C#CC1(C(N2CCC(CC3CC3)C2)=O)CCN(C(=O)CN2CC=CC2)C1 CC1C(NC(C2CC3(CC3)CO2)=O)CCN1C(=O)CC1(C)CC1 c1(N2CC(C)(C(C)NC(=O)C3=COCCC3)C2)nccc(S(C)(=O)=O)n1 C(=O)(CC(C)(C)CN(C)C)NCC(CC(C)C)NC(c1c(F)cncc1F)=O c1(C(C)C)cccc(C(=O)NC(CNC(=O)CC2CCC23CC3)C(C)C)c1F C(=O)(C1=CCCCCC1)N(C1CN(C(c2coc3c2CCCC3)=O)CC1(C)C)C C1(C2(CN(C(=O)NCc3c(OC)cc(Cl)cc3)C)CC2)CCC2(CCCC2)CC1 c1(NCC(=O)NC2CN(C(C3CC(CCC)C3)=O)C(C)CC2)cccc(C#N)c1 C1(NC(C2(OC)CCCC2)=O)CC(CO)N(C(=O)CCCn2cnc(C#N)n2)C1 C1(NC(CC2(COC)CCCC2)=O)CC2CCC1N(c1ncc(C)c(O)n1)C2 c1(NC(C)C(F)(F)F)cncc(C(=O)NCCC2CCCC2)c1 C1(C(=O)NCC2CCCCN(c3ncnc(CO)c3F)C2)CCCCC12CCC2 C12CCCC(C1)C2.C1(CN)COC(=O)O1.C1(=O)CO1 c1(CC)cncc(Cl)c1C.C12CCC(O1)C(=O)N(C)CC(C)CNC2=O S(=O)(=O)(C1CCCCC1)N1C(C(=O)NC(c2cccnc2)CC)CC1 C=CCC(CC)NC(=O)CNC(=O)CNC(=O)CCC=C c1(NC(=O)CN2CCN(C(C3CC3C(CCC)=O)=O)CC2)c(C)cc(Br)cc1Cl C1(NC(C2(NC(Cc3cn(CC)nc3)=O)CC(F)C2)=O)CCN(C)CC1C#N O=C1NC(=O)C(CCNC(C2CCCN(C(c3ccnc(Cl)c3)=O)C2)=O)N1 CCCC(C(=O)Nc1cc(N(C)C)nc(NCC2CSC3CCCC23)n1)C(C)C C1(NCC2N(C(=O)OC(C)(C)C)CCCC2)COc2ccc(O)cc2O1 Cc1nc(C2CCC2)sc1CC(=O)NC1CC1CNC(C1OCCCO1)=O N1(C(=O)CSc2ccccn2)CC(NCc2ccc(Cl)c(O)c2)C2(CC2)C1 c1(C(=O)NCCC(C)NC(c2cc(N(C)C)ccn2)=O)cc(F)n(C)n1 CCC(C(=O)NCC1CC1CC(=O)NC1CC1C1CC1)C(C)(C)CC C1(NC(C(c2ccc(F)cc2)(C)C)=O)CCCN(C(=O)Cc2cc[nH]n2)CC1 c1(C(C)=O)ccc(C(=O)N(C(C)C(=O)N(C)Cc2nc(C)cs2)C)o1 c1(C(=O)OC)ccc(NC(C23CC2CN(C(=O)C=CC(C)C)C3)=O)c(I)c1 C1(NC(CCCC#C)=O)CC2CCC(C1)N2C(=O)CC1CCOCC1(C)C C1(C(=O)NCC#C)CN(C(C2(C(=O)[SH](c3cc(C)ns3)C3CCCO3)CC2)=O)CCO1 C1(NC(C2CC2CF)=O)CCC2(CCCN2C(c2ccc3cc[nH]c3n2)=O)CC1 c1(CNC(C2CCCCO2)C)cc(Br)cc(Cl)c1O C1(C(=O)NC(c2cncs2)C)CC2CC2N1Cc1cccc(OCCCl)c1 C1(C(N2CC(CN(C(COCCCCCC)=O)C)C2)=O)CN(C)CCO1 c1(C(=O)NCC2(OC)CCN(C(c3ccoc3)=O)CC2)ccn2c(C)cnc2c1 N1(C(=O)Nc2cc(C)cc(Br)c2)CC2(CCCC2)OCC1C C(c1ccc[nH]1)=CC(=O)N(C1CC(NC(C23CCCC2C3)=O)C1)C C=C(C)CCC(C)NC(=O)CC1(N(C(=O)C(C)COCC)C)CC1 N1(C(c2n(C)ncc2)=O)CCN(C(C2CCCCN2C(=O)CCS(C)=O)=O)CC1 N(C(=NCCF)NC1CCN(S(C)(=O)=O)C1)CC(CC)N(C)C C1(NC(CCC=C)=O)(CO)CCN(C(c2cn(Cc3cccs3)nn2)=O)CC1 CC(CSn1cnc(C2CC2(Cl)Cl)c1)C(=O)OC1(C(=O)OC(C)(C)C)CC1C N1(CC)CCC(NC(=O)C(O)CSC)C1=O c1(-c2c(C(=O)Nc3c(I)ccc(C#N)c3)ncnc2)cc2cc(Cl)ccc2[nH]1 C1(NC(COCC)=O)CCC2(CC1)CC2NC(=O)C=Cc1cscn1 C(=O)(C1CCc2ccccc21)NC1CC(NC(c2n[nH]c3c2CN(C)CC3)=O)C1 N1(C(c2scc(COC)c2)=O)CCN(C(C2CCC3CC23)=O)CC1CCO C12(NC(CC3CC(SC)C3)=O)CC1CN(C(=O)Cc1sc(O)nc1O)C2 c1(CS(C)=O)cccc(C(=O)NCCC2CCCN2C(C2CNC(=O)N2)=O)c1 C1(C(N2CCC(Br)C2)=O)CCc2nc(-c3ccc4n[nH]cc4c3)sc2C1 N1(C(=O)CCC2CCC(O)CC2)CC2CCC(C1)N2CCCc1cccs1 c1(C(N2CCN(C(C=CC)=O)CC3(C2)CC3)=O)ccc2ccnc(O)c2n1 c1(C(N2C(C(C)NC(C3CCSC3)=O)CCC2)=O)cc2ncccc2cc1Cl C1(NC(C(CCCC)ON=C(C)C)=O)CN(C(=O)C#CCSC)CC2CCCC12 c1(N2CC(C(N3CCOCC3)=O)OCC2)ncnc2sc(I)cc12 c1(C(=O)N(c2ccccc2)CC2CCCC23CC3)cc(C(F)(F)F)cc(Cl)n1 CC1=C(C(=O)N2C3CCCC2CC(CNC(=O)C(O)C(F)F)C3)CCC(C)(C)C1 CCCCC(C(=O)NCCc1ncccc1F)NC(=O)C(F)CC1CCOC1 Cc1cnc(F)c(OCC(N2CCC(N(C(=O)C(C)(F)c3ccon3)C)C2)=O)c1 c1(OCC)ccnc(N2CC(C(C)NC(C3CC3(C)Br)=O)C2)n1 C1(N(C(CCC)=O)C)CN(C(=O)CCC2OCCO2)CC1O CC1=C(C(=O)N2CCOCC2CCNC(=O)CSc2nccn2C)CCC1 C(=O)(C1=CCC2CCC1N2C(c1ccc(CO)s1)=O)Nc1c(OC)c(F)ccc1 C1(N(C(CCC=C)=O)C2CC2)COCCC1C(=O)N(C)OCCCC N1(C(C23CC(c4cn(-c5nccs5)nn4)(CO2)C3)=O)CCC(C)CCC1COC N1(C(C2C(COCC)(COC)C2)=O)CC2C3CCC(C2C1)N(C(c1cnsc1)=O)C3 N1(C(C(CC)NC(N)=O)=O)CC2CCCC(NC(=O)CC3=NN(C)C(=O)C3)C2C1 N1(C(c2c(C)occ2)=O)CCC(C)(C)C(C(N2CC3(CCCCC3)C2)=O)C1 CC1=CC(C)C(CNC(=O)NC2CC(N3CCOCC3)C2)CC1 c1(C(N(C(C)CNC(=O)C(C(C)C)N(C)C)CC)=O)cccc2nonc12 c1(C(=O)NCC(CNC(COc2ccc(C)cc2)=O)O)cc(N)nc(Cl)c1 C1(CNC(CCN(C)CC)=O)CCN(C(=O)CC2(O)CCC2)CC1C N1(C(C(C=C)(C)C)=O)CCOCC(C(N2CCC(C)(O)C2)=O)C1 C(N=c1cccc(S(=O)(=O)NC2CC3C=CC2CC3)[nH]1)c1cc(C(C)(C)C)no1 c1(C(N2CCCC(NC(c3n(CC)nc(C)c3)=O)C2)=O)cc2ccccc2o1 C1(CNC(COC)=O)CCN(C(c2cccc(C)c2O)=O)CC1C C(=O)(CC(C)CC(C)C)N(CCNC(c1cncc(C(N)=O)c1)=O)CC C1(CCCNC(C=C(C)C(C)(C)C)=O)CCCCN1C(=O)C=CC1CCCC1 N1(C(c2cnc(OC)s2)=O)CCC2(CCN(C(c3cc(Cl)c[nH]3)=O)C2)C1 c1(NC(C2(c3cccc(-c4ccc(C)nn4)c3)CC2)=O)cc(Br)c([N+](=O)[O-])cn1 N1(C(c2nc(C)oc2)=O)CC(CNC(=O)COCc2ccnn2C)C2(CC2)C1 C(CC1=CCN(C(c2cn(C(F)F)cn2)=O)CC1)NC(C(CCCC)O)=O N1(CC(C)(C)NC(c2c(C)ncs2)=O)CCN(C(C2COC2)=O)CC1 N1(C(C(F)=CC)=O)CC2(C1)C(NC(c1cc3cccnn3n1)=O)CCS2(=O)=O n1(CC(=O)N(C2CCCN(C(=O)COC)C2)C2CCOC2)ccc(=O)cc1C C1(C(N2CC(NC(COCC(N3CCC(N(C)C)C3)=O)=O)C2)=O)(CC)CCCO1 C(C(=O)N(C1CN(C(=O)CC2CC=CCC2)C1)C)(C(C)C)c1cnc(C)s1 C1(C(N2C3(C(=O)NC(C4CCCC4)CC)CC(CO)(C2)C3)=O)CCS(=O)(=O)C(C)C1 O=C(CS(=O)(=O)CCO)NCCCN(C(C1CCCC1)=O)Cc1ccncc1 C(C(=O)Nc1ccc(Cl)cc1F)(C1=CCCSC1)N(CCC)CC1CCOC1 N1(C(C(C(C)C)SC)=O)CC(C2CN(C(c3cccc(N)c3C)=O)C2)C1 C(=O)(CCS(=O)(=O)N(C)C)N1CC(NC(CC)=O)C(c2ccnn2C)C1 c1(C(=O)NC(CCNC(C(C)Cn2cccn2)=O)C)cc(Br)cnc1O O=C1Nc2c(C(N3CC4CN(C(C5(F)CCC5)=O)C4C3)=O)cccc2C1=O N1(CC(=O)NCCOC(F)F)C2C=CCC1CC2 C(=O)(C(O)CC(F)(F)F)N1C(CN(C(C(CC=C)(F)F)=O)C2CC2)CCC1 C#Cc1ccc(C(=O)NC(C)(C)C=CC(N2CCC2C2CCCC2)=O)nc1 c1(NCC(CC)O)ccc(S(=O)(=O)NCC2CCOC3(CCCCC3)C2)cc1Br N1(C(c2ccc(C#N)o2)=O)CCC(CNC(=O)CC(F)(F)C(F)F)C(F)(F)CC1 c1(C(N(CCNC(c2cnc[nH]2)=O)C2CC2)=O)csc(S)n1 c1(OC)nc(C(=O)N(C2CCOCC2)CCCO)cc(O)n1 Cc1cnc(Cl)c(C(=O)NCC2CN(C(c3ccc(C#N)o3)=O)CCCO2)c1 C1(N(C(=O)CSC2CC2)C)CCC2CN(C(c3cc4scnc4[nH]3)=O)CC12 C1(C)(CC)C=C(C(=O)N2CC(C)CC2C)C1.C(=O)CC(C)(C)O Cc1ccc(C(N2CC3CC3(NC(C3CC(C#N)C3)=O)C2)=O)nn1 Cc1noc(C)c1CC(N1CCC(C(C)(C)NC(C2COCCO2)=O)C1)=O c1(N2CCCC(C3C(NC(C4N(CC)CCC4)=O)C3)C2)cc(S(C)(=O)=O)ncn1 Cc1ncn(C)c(=O)c1C(=O)N(CC(C)CNC(C12COC(CCO1)C2)=O)C C(=O)(C(C)CC(F)(F)F)N1CCC(CNC(C(CCC)(C)O)=O)CC1 C1(NS(=O)(=O)c2scc(Br)c2Br)Cc2[nH]c(=O)c3ccccc3c2C1 C1(CC(N2CC3C(NC(=O)Cn4cnnc4O)C3C2)=O)CCC2(CCC2)O1 c1(C(=O)NCC=CCc2ncco2)ccc(OCC(F)F)cc1.C12(CC1)C(=O)N2 CCCC(C)(CC)C(=O)N1CCC(O)(C(C)NC(=O)COC)C1 C(CC(C)(C)C)(C(=O)N(C(C)C(=O)N(C1CN(C)C1)C)C)OC Cc1cc(C(N2CCCC2C(C)(C)C(N2CCNCC2C(C)C)=O)=O)nc(C)c1 C(=O)(C1c2ccccc2C2CC1C2)N1C(CC)CN(C(=O)CC(C)SC)CC1 N1(CCOCCC(=O)Nc2ccccc2)CCc2nc(O)ccc2C1 CN(C)NC(=O)CCC(=O)NCC1CCCN(C(=O)CCc2ncco2)C1 C=CCCC(C(=O)NCCCc1ccc(C)cc1)C(C1(C)CCC1)OC C1(C(=O)NCC(O)COc2ccccc2F)CCCC(C(=O)O)C1 N1(C(CCCC2(C)N=N2)=O)CCC(C(C)C(=O)NCCCC2(C#N)CC2)CC1 C(C)(CC(=O)N1CCC1CC(=O)N(CC(C)CO)C)=C(C)C c1(C(=O)NCCCCCNC(c2cc(CC)sn2)=O)cc(C)nn1C(CC)CC c1(C(=O)NCC2CN(C(CSC)=O)C3C2C3)c[nH]c2c(C)cccc2c1=O C(CS(=O)(=O)N(C(CC(N)=O)c1ccsc1)C)(C1C(CC)C1)OC O=C(C1CCCn2cnnc21)NC1CC(NC(C2CCCCNC2=O)=O)C(O)C1 C12(NC(C(CC)O)=O)CC(CNC(c3cnc(S)[nH]3)=O)(C1)OC21CCC1 N1(CC(=O)N(CCNC(CN(C(=O)OC)C)=O)C2CC2)CCCS1(=O)=O c1(C(=O)NCC2CC2CNC(C2(SC)CC2)=O)ccc2cc(OC)ccc2c1.CS C1(C2CC2)(C(=O)OC)CN(C(=O)CC(NC(=O)Cc2cnn(CC3CC3)c2)SC)C1 C1(C)(C(N(CCCC)C)=O)CCCN(Cc2cccc(CC(=O)O)c2)C1 CC1CCN(CC(=O)N(CCCOc2ccccc2)CCO)CC1 c1(OC)cccc2c1N(C(C1NCC13CCOCC3)=O)CC2 c1(OC(C)=O)ccc(F)c(C(N2CC(F)(CNC(=O)C(O)C(C)(C)C)C2)=O)c1 Cc1cccc2oc(NC(c3cnc(C4CCN(C(=O)CC5CC5)CC4)s3)=O)cc12 c1(CC2CN(C(C(C)OC(C)=O)=O)C2)cnc(C2CN(C(C)=O)C2)o1 c1(OC)cc(Cl)ccc1C(=O)NCCN(C)C(C1CCCCN1C(N)=O)=O N(C)(C1CN(C(=O)CCCCSC)CCc2ccccc21)C(C1(CC)CCC1)=O c1(NC(=O)NC2C(CC=C)C(O)C2)cccc(P(C)(C)=O)c1 c1(CC)cc(C(N2CC(F)(C(=O)NCC(C)(C)CCOC)C2)=O)c(C)o1 c1(C(=O)NC(C2CCN(C(=O)CCc3ccoc3)C2)C)cnc2[nH]nnc2c1 c1(NC(C(N2CC(CCC)OCC2)=O)=O)cc(C)ccc1SCC#N C1(N(C(=O)CSCC2CCCO2)C)CCN(C(c2cscc2Cl)=O)CC1 C(C1CCC(=O)c2ccccc21)N1CC(=O)OCC12CCC2 c1(C(=O)NCCN(C(c2ccnn2C2CC2(F)F)=O)CC)cccc2c1OCC2 C(C(CO)(C(C)C)NC(c1ncccc1Br)=O)NC(C1C(C(=O)OC)C1)=O c1(CN(C)C)ccc(Br)c(C(N(c2ccccc2)C(C(C)C)=O)=O)c1 N1(C(=O)CC2CCCC2)CC2(C1)CN(C(C1CCC(=O)NC1)=O)CC2CO N1(C(C2(C)CN(S(c3c(C)n[nH]c3C)(=O)=O)C2)=O)CCCC2(C1)OCC1CC21 C1(C(=O)NC(CC)CCc2ccco2)(CF)CCN(C(c2cc(C)no2)=O)C1 CC(CC(C)NC(c1ccnn1-c1ccccc1)=O)NC(=O)CCC1CCOC1 C1(C(N2CCC(CCC(=O)NC3CCCC(SC)C3)C2)=O)CC2CC(=O)C1O2 C(N=c1[nH]c(=NCc2cc(Cl)cc3c2OCC3)[nH]c2c1SCC2)C1OCC(C)C1 C1(C(=O)NCC2N(C(COC(C)=O)=O)CC=C2)CCn2c(C)cnc2C1 N1(C(C(CCC)F)=O)CC2CC(C1)CN(C(=O)COCCC(C)C)C2 c1(SC)c(C(=O)N(C2CC(NC(c3snc(Cl)c3Cl)=O)C2)C)cnn1C c1(CC(=O)NCC2C(NC(C3CC(OC)(OC)C3)=O)C2)ccc2c(c1)OCCO2 C1(C)(NC(C2CN(S(CC)(=O)=O)C2)=O)CCN(C(C2(OC)CCSC2)=O)CC1 Cc1cc(N(C(C)CCNC(c2ccc(F)cc2C)=O)C)nc(CO)n1 C(=O)(C(CCS(C)(=O)=O)N(C(=O)C(C)(C)N1CCCC1)C(=O)CCCSC(C)(C)C)OC c1(CN(C(c2ccnc(OC)n2)C(=O)NCC2(OC)CC2)C)nnc2n1CCC2 c1(C(=O)NC2(C)CCN(C(C3COC(C)(C)C3)=O)C2)ccc2c(c1)CCC2=O CC1CC(C(=O)NCC23CC(NC(c4coc(C(F)F)n4)=O)(C2)C3)CN1C c1(-n2cc(CNC(C3CCC(C(=O)O)NC3=O)=O)nn2)cccc2ncccc12 C#Cc1ccc(C(=O)NC2CCN(C(=O)CC3CC4CC4C3)C2(C)C)cc1 N1(C(CSCC#C)=O)CC2CC(C1)CN(C(=O)CCCCCC(C)C)C2 N1(C(c2cnc(CCCC)s2)=O)CC2(C1)CN(C(c1ccnnc1)=O)CC2CO n1(CC(=O)NCCCCNC(C2OCC(C)C2)=O)cc(P(C)(C)=O)cn1 CC(C)C(C(=O)N1CCOC(CC(=O)N(CC(O)CO)C)C1)C(C)C c12cc(=O)c(c[nH]1)NC2=O.C1(NC(C)=O)CC(CNC(C2(SC)CC2)=O)C1 Cc1cc(C(=O)NCCCCNC(C2(C)CNC(=O)C2)=O)cc2ccoc12 C(=O)(CCCC(C(=O)N(C)C(C)C)N(CC(=O)NC1CCCC1)C)OC C1(CC(=O)NC(C)C)CCCN(C(C2CC(=O)N(C3CCC3)C2)=O)C1 C#Cc1cccc(CC(=O)NC2COCCC2C(N2CCC(C(F)(F)F)C2)=O)c1 C(=O)(C(C)(C(C)C)NC(C)=O)NCC(CC=C)NC(=O)CCc1cn(C)nc1C C1(C(N(C)CCNC(C2(C(=O)OC(C)(C)C)CC2(C)C)=O)=O)CCCC(=O)N1 Cc1cnc2c(C(N3CC(NC(=O)CC4CCCC4)CC(O)C3)=O)cnn2c1 c1(OC)ccnc(CN2CCN(CCCNC(c3cncc(O)c3)=O)CC2)c1 C(=O)(C(CC(F)F)C1CCC1)NC1CCC(NC(CSCCOC)=O)CC1 C12(C(=O)NCc3ncnc(CC)n3)CC(C1)C(NC(=O)OC(C)(C)C)CO2 N1(C(c2c(N)c(Cl)ccc2)=O)CC2(CCC(CNC(=O)CCc3cnn[nH]3)O2)C1 CCC(C)CC(C)C(=O)NCCNC(C12CCC(F)(CC1)C2)=O C=C(C)C1OCCCC1C(=O)N(CC)CC1CN(C(=O)CCCN2CCCC2)C1 N1(C(c2c(C)ccnn2)=O)C2CC1CN(C(=O)CCN1CCOCC1)C2 Cc1c[nH]cc(C(=O)NC(C2CCN(C(=O)CSCC(F)(F)F)C2)(C)C)c1=O N1(C(CCCc2cc(C)no2)=O)CCC2OCCN(C(c3csnc3C)=O)C2C1 Cc1cccc(C)c1CN(CCNC(C1CN(C)C1)=O)C1CC1 N12CC(C)(C)CCC1COC(=O)C2.C(=O)(C1=CCCO1)Nc1c(C=O)scc1 N1(C(CC(=O)NCC)=O)CCC(C2CCN(C(=O)Cc3sc(C)nc3C)CC2)C1 C1(CC)CC(c2ccc(C)cc2)CCN1C(=O)CC12COCC(C1)C2 c1(C(N2CC(NC(c3c(C)cccc3)=O)C(CC3CC3)C2)=O)ncnc(O)c1F N1(C(C2CCC(CC)O2)=O)CC2(CCN(C(c3ccc([N+](=O)[O-])[nH]3)=O)C2)C1 c1(C(=O)NCCN(C(C2C(C)(C)C2(C)C)=O)CC)cc(Cl)ccc1-n1cccc1 c1(C(N2CCC(N(C(=O)C(F)OC)CC)C2)=O)ccnc(C)c1C C(CC1=CCN(C(=O)CSC2CC2)CC1)NC(c1c(NC)ccc(Cl)c1)=O N1(C(c2cc(CC)on2)=O)CCOC2(C1)CN(C(C1(S(C)(=O)=O)CCCC1)=O)C2 C(CCCC(CO)NC(=O)C(C)OCc1ccccc1)NC(CS(CC)=O)=O CC(C(=O)N1CC(CNC(=O)CCc2cnn[nH]2)C1)c1ccco1 C(C(O)C(F)(F)c1ccccc1)NC(c1ncn(CCF)n1)=O C1(C(=O)NCC(C)(C2CCC2)NC(C(C=C=C)C)=O)CCOC2(CCOCC2)C1 N1(C(c2cnc(Cl)s2)=O)CCN(C(c2cc(O)ccc2F)=O)C(CC(F)F)C1 Cc1cc2ncc(C(N3CCC4(CC(NC(=O)C(F)C5CCC5)C4)C3)=O)cn2n1 C1(C(=O)NCC(=C2CN(C(CCCOCCC)=O)C2)F)(CCF)CCOCC1 C1(C(=O)NC2N(S(C)(=O)=O)CC2)CC2(C1)CN(C(=O)COC1CCCOC1)C2 C(=O)(C1=CCCN(S(=O)(=O)c2cn[nH]c2)C1)Nc1c(CC)cnc(Br)c1 N1(C(c2cc(CC)on2)=O)CCN(C(C2CCN2CC)=O)CC1CC Cc1nc(-c2ccccc2)nc(O)c1CC(=O)NC1CCC1F C1(CNC(C(C=CCCC)O)=O)CC(NC(c2ccc(CC)cc2)=O)CCO1 C1(C)CN(C(=O)CC#N)C(C)(C)C1.c1(CCN(CC(=O)N)C)ccccc1 C1(C(N(CCO)CC)=O)CC(C)(C)CCN1C(=O)C(c1cncnc1)C C(=O)(C(O)CCNC(=O)CCNC(=O)OC)NC(CC)C CC1=C(C)C(NC(N2CC(c3cccc([N+](=O)[O-])c3)(O)C2)=O)CCC1 C1(CNC(c2cc3ccsc3s2)=O)CC2CN(C(C3(C(F)F)CC3)=O)CC12 c1(CC)conc1C(=O)NCC1CCCC1NC(C1(c2ncco2)CCC1)=O N1(C(Cc2nc(C)sc2)=O)C2CCCC1CN(C(C1CCCC(F)(F)CC1)=O)C2 C1(C(N2CCCC(N(C(c3ncn(C)n3)=O)CC)C2)=O)CCCCC(=O)N1 CP1(=O)CCN(CC(=O)NC2CN(C(C3CCC(C(F)(F)F)N3C3CC3)=O)C2)CC1 c1(C(C(N2CC(NC(C3CC3CF)=O)(CO)C2)=O)O)cccc(F)c1 S(=O)(=O)(CC(=O)N(C1CCN(CC(C)C)C1)CC(C)C)NC(CSCCOC)=O c1(C(=O)NCC(C)NC(c2cn(CCOC)nc2)=O)cncc(N2CCCC2)c1 C(=O)(C1=C(CN2CC=C(c3ccccc3)CC2)NC(=O)NC1C)OCC C1(C(NOCCCC)=O)CN(C(C2(C)CC2(F)F)=O)CC1C(C)C C1(C)(CC)CC(NC(=O)Cc2cc(Cl)ccc2OC)CN1C(=O)C(C)(F)F N1(C(c2c(CNC)ncs2)=O)CCC(O)(CNC(=O)CC2CCCC(OC)C2)CC1 c1(C(N(CC(CNC(Cc2ccc(CC)cc2)=O)O)C)=O)ccc2nn[nH]c2c1 c1(OC)cccc(OC)c1C(=O)NCC1CCC(NC(=O)C=C(Cl)Cl)CC1 O=C(CC1COc2ccccc21)Nc1nc2c(s1)CCCC2.c12ccc(cc1)CN2 c1(C(N2C(CN(C(C(C)Sc3ccccn3)=O)C)CCC2)=O)ccc(F)c(N)c1 C1(C(N2CC(O)(CNC(CCc3cc(C)n(C)n3)=O)C2)=O)CCn2cnnc2C1 C1(C(=O)NCC2CC3(CC(NC(CC(C)(F)F)=O)C3)C2)CCC2C(C1)C2(F)F N1(C(C2C3C4CCC(C4)C23)=O)CCC2CN(C(=O)CC3CCCOCC3)C2C1 N1(C(CC(CC)OC)=O)CC(CNC(=O)CC2=CCCC2)C2(CC2)C1 C1(C(=O)NC2C=CCCCC2)CC2(CC2)CN1C(c1cc(O)cs1)=O C1(NC(c2csnc2Cl)=O)CC(C(=O)NC2CC3CCC2O3)C12CCC2 N1(C(C(N)Cc2ncccc2Br)=O)CC2CCC1C2N C(=O)(CCC(C)(F)F)N1CC(C(C(=O)N(C)Cc2cncnc2)O)C1 C=CCC(C)(C)C(=O)N(CC1CN(C(=O)CCOC(C)CCCC)CCO1)CC c1(NC(=O)Nc2ccc(C)c(C)c2)cnc2c(Br)c(C)ccc2c1 C(N=c1[nH]c(=NCCSC2CCCC2)c2ccccc2[nH]1)c1c(C)c(F)c(F)cc1 C1(F)(c2cn(CCCC)nn2)CCN(C(=O)Cc2ccc(C)c(I)c2)CC1 C1(S(N)(=O)=O)(CC(=O)NCC(C2CCCCC2)NC(COCCOC)=O)CCC1 c12nn(C)c(Cl)c1C(N1CCOCC(C(C)C)C1)C(=O)NCC2.CN N1(CC(c2ccccc2)C)CC(=O)N(CC2CN(CCCN(C)C)CCO2)C1=O CCC(C)C(O)C(C)C(=O)NCC(C)(C)CCNC(=O)Cc1cccc(O)c1F Cc1nc(Cl)nc(N2CCC(N3CCN(C(C4CCCN4C)=O)CC3)CC2)c1Cl CC(CN(C)C)C(=O)N(C)CCOCCN(C)C(c1coc(C(C)(C)C)n1)=O c1(C(=O)NCC(CN(C)C(C2CNC(=O)N2C)=O)(C)C)ccccc1C(F)(F)F c1(C(N(C(C)CNC(C2CCC(CC)O2)=O)CC)=O)ccc2n[nH]cc2c1F c1(C(=O)NCC(C2(O)CN(C(C(C)=C3CCC3)=O)C2)(C)C)nc(C)ccc1F c1(OC)csc(C(N2CCN(C(C3(CCF)CCC3)=O)CC2)=O)c1OC C1(CNC(C(CC)F)=O)CN(C(C2(CSC)CCOCC2)=O)CC(C)(C)O1 n1(CC)nc(C(=O)NC2(CNC(=O)C(O)CC3CCCC3)CCCCC2)cc1O C1(NC(C(C)(C)N(C(C)=O)C)=O)CC2(C1)CC(C(=O)NC1C3CCCCCC13)C2 N1(C(C2C=CCN(C(C(C)OCCCC)=O)C2)=O)CC(CO)C2(CC2)C1 c1(C(=O)NCC2(F)CCCN(C(CCC(C)=O)=O)C2)cccc2c1nc(O)n2C N1(C(C=Cc2c(C)ccs2)=O)CCN(C(=O)Cn2nccc2C)CC1CC(F)F N1(C(CCc2c(C)cccc2)=O)CCN(C(=O)CCc2cnn(C)c2)C(C#N)C1 Cc1cncc(C)c1C(=O)NC1CCCC1NC(=O)CC(F)(F)F C1(C(C(=O)NCCCSCC)F)CCN(C(c2coc(C3CC3)n2)=O)C1 C=CC1(C(=O)NC2CN(C(=O)C(C)CC3CCCC3)CC2C)CCOCC1 CCCC(c1ccco1)NC(=O)CCN(C(=O)C(=O)NC(C)C)C1CC1 C=C1CC(C)(C(=O)NC(C)C(C)NC(=O)CCOCCCNC(C)=O)C1 c1(COC)csc(C(=O)N(CCCCNC(=O)CCc2nc(C)cs2)C)c1 C1(NC(C(C)(C)CC2CC2)=O)CCOC12CCN(C(C1CC13CCC3)=O)CC2 C(=O)(CCN=c1[nH]cco1)N1CC(O)(CNC(c2cnc(CC(C)C)[nH]2)=O)C1 c1(C(=O)NC(C)C(=O)O)[nH]nc2ccc(-c3coc(C(=O)O)c3)cc12 c1(CNC(C(C)OCCCNC(COC(CC)C)=O)=O)cnc(C)o1 C1(C)(C(=O)NC)CCCN(Cc2ccc(-c3ccc(C)c(OC(F)(F)F)c3)s2)C1 CC1CN(C(c2cscc2C(F)(F)F)=O)CC1NC(=O)C(C)(C)c1cnn(C)c1 CC(CCC(F)(F)F)NC(=O)C(C)N(C(=O)CC1CCCC1)C Cc1c(C(=O)NCCCN(C(=O)C(C)N2CC(C)C2)C(C)C)[nH]c2c(C)cccc12 N1(C(C(C)S(N)(=O)=O)=O)CC(C)CN(C(C2CCCC(C)(C)C2)=O)CC1C N1(C(C)C)CCCC(CC(=O)NC2CCCC(NC(=O)Cc3ncc(Cl)s3)C2)C1 C1(CCOCCO)C(=O)N1.C(CC(=O)NC)(NC(C)=O)NCCC1CC(O)C1 c1(C(=O)NC2C3CN(C(CSCc4ccc(C)cc4)=O)CC32)ccc(F)c(C)n1 Cc1n[nH]c(C)c1SCC(N1CC(CNC(=O)CSCC(C)C)C(C)C1)=O C(=O)(C(CN(C)C)C(C)C)NC1(C)CN(C=O)C1.C1(CC#C)(N)CCOC1 c1(C(=O)NC2CCCC(NCC(F)(F)F)C2)c(OC(F)F)cccc1Cl C(=O)(CC(C)C(F)F)NC.C1(C=O)(CNC(CN(C2CC2)CC)=O)CCCC1 CCCC(C)(CC)C(=O)N1CCCOC(CCNC(=O)CS(C)(=O)=O)C1 C(=O)(CC(C)C(=O)OC)N1CCC(C(=O)NCC2(COC)CC2)C1 C1(NC(CCCC)=O)CN(C(=O)C(C)Cc2ccccc2Cl)CC1O C1(CC(=O)NCC(C(=O)NC)O)N(C(=O)CN2CCNC(=O)C2)CCC1(C)C c1(OC)ccccc1C(C)C(=O)NCCCCCCNC(C1(C)CC(F)C1)=O N(C(=NCCc1ccc(F)cc1)NCc1cccs1)CC1C(OCC)C1 Cc1ccc(Cl)c(CNC(c2nc(Cl)sc2Cl)c2nnnn2C(C)C)c1 N1(C(c2ccc(CO)o2)C(=O)NCC=C)CCCCC1c1nc(C)no1 C1(CC)C(NC(=O)CCc2ncccn2)CCCN1C(c1ccc(Cl)cn1)=O CCC(O)(CC)CCNC(C1CCN(c2ncnc(OC)c2C)CC1)=O CC(C)(C(=O)NC1CC(O)(CNC(c2ccc[nH]2)=O)C1)Oc1ccccc1 c1(C(N2CCN(C(C(CCC)CCC)=O)CC2C)=O)ccc2c(C#N)c[nH]c2c1 C(C)(C)(CCC(=O)NC1CC(F)(F)C1(C)C)NC(c1n(CCC)ccc1)=O CC1CCC(O)(C(=O)NCC2CCN2C(C2CCC(C)(C)C2)=O)CC1 C(N=c1cc(C)[nH]c(=NCc2cnc(O)[nH]2)[nH]1)CC(C(=O)OC)F c1(C(=O)NCC2(O)CN(C(C3(C#C)CC3)=O)C2)[nH]nc2ncc(Br)cc12 N1(C(CCCSC)=O)CCC(C(F)(F)F)C(NC(c2cc(C(N)=O)no2)=O)C1 C1(C(=O)NC(C2CN(C(C(=O)NC(C)C)=O)C2)C)CC(c2cccc(F)c2)=NO1 N1(C(C(CC)C)=O)CCN(C(c2cc(C)n(C)c2)=O)CC(C)(F)C1 c1(N2CC(C)c3c(cccc3)CC2)nc(=NCc2ccc(Br)s2)[nH]c2c1COC2 c1(C2(C)OCCO2)cccc(C(=O)NC2CCC(NC(=O)C(F)=C3CCC3)C2)c1 C(CCCC(=O)NCCCN(C(=O)C(CC(C)C)N(C)C)CCSC)(OC)OC N1(C(C(=O)NCCOCC)c2nnc[nH]2)CCC(C#N)(C(C)(C)C)CC1 C(=O)(C1=CCN(C(=O)C2=NOC(C)C2C)CC1)N(C1CCOC1)CC#C N1(C(CNC(CNC(C)=O)=O)=O)CCC(CO)(NC(c2n[nH]c(C)c2C)=O)C1 c1(OC)cc(F)c(CC(=O)Nc2ccc(OC)c(F)c2)cc1F c1(C(C2CCOCC2)CNC(c2cc(C)no2)=O)cnc(C(F)(F)F)nc1 N1(C(COCC=C)=O)CCCCC(Cn2c(C3CC3)nnc2-c2ccccc2)C1 C1(C(N(CC#C)CC2CC2C)=O)CCN(C(=O)CCCN(C)C(C)C)CC1 c1(N(C(N2CC(c3cccc(OC)c3)OCC2)=O)C)cnn(C2CNC2)c(=O)c1 C1(O)(CNC(CCSCCCC)=O)CCCN(C(c2cncn(C)c2=O)=O)C1 CC(C)(C(=O)NNC(=O)C(C)(C)CCCCNC(C12CC(C1)C(C)(C)O2)=O)C(N)=O C1(C(=O)NC(C(C)(C)NC(CCc2cnc(C)o2)=O)C)CC2OC1C1CC21 C(=O)(C(CCc1ccccc1)OC)NC(CC=C)CNC(c1nnsc1SC)=O O(NC(=O)C1=CC2(CCN(C(=O)C=CC(C)(C)C)C2)C1)CC(C(C)C)O C(=O)(CC(CC)CC(F)(F)F)N1CC2C(CNC(C(CC)(C)CC)=O)(C2)C1 C1(CC=C)(NC(=O)CC2C=CS(=O)(=O)C2)CCN(C(c2ccc(F)cc2)=O)CC1 Cc1cc(C(=O)NC2CCN(C(=O)COCC(C)(C)C)C2C)nc(C)c1 N1(C(C(C)=C2CCCC2)=O)CC2CCC1CN(C(=O)CN1CCCNS1(=O)=O)C2 c1(C(=O)NC2C3CN(C(C4=C(C)OCC4)=O)CC2CC3)cc2cc(Br)ccn2n1 c1(NC)cncc(NC(=O)CC2CN(C(=O)C(C)(C)SC)CC2C)c1 N1(Cc2ccc(CN(C)C)cc2F)CCC2(CCCN2C(=O)CCCCCl)CC1 C1(C(=O)NC(C2N(C(CNC(=O)NC)=O)CCC2)C)CCn2ncnc2C1 CC(C)C(F)(CNC(=O)CN1CCN(C)CC1)C(=O)N1CCC1CO C1(O)(CNC(c2sc(C)c(O)n2)=O)CC2CCC(C1)N2C(C1(C)CCCOC1)=O CCCCCN(CCC(=O)NCC(CO)NC(=O)C(C)OC(C)=O)C c1(C(=O)NCCC2(NC(CC(CC)OC)=O)CCC2)cc(Cl)c2c(c1)OCCO2 c1(NC)ccc(F)cc1C(=O)NC1CC(CC(=O)NCC2(C(O)C(F)(F)F)CC2)C1 c1(C(C)=O)cccc(NC(C(C)Cc2nnnn2C)C2CCCC2)c1.c1ccccn1 N1(C(c2c(C)nccc2)=O)CC(C)(C)OCC1CNC(C1(C2(O)CCC2)CC1)=O C1(C)(C(=O)NCCN(C(=O)COCC2CCCCO2)CC)CCN(C)C1 C12(CNC(C(C3CCC3)OC)=O)CCCC1N(c1ncc(F)cn1)CCC2 C1(CNC(=O)CCc2cnc(C3CC3)o2)CC2CC2N1C(C1CCC(F)CC1)=O c1(C(C)C)nc(NCc2csc(CN(C)C)n2)cc(N2CCC(Cl)=C(Cl)C2)n1 C(=O)(C(CC(C)C)C(C)C)NC1(CC)CCN(C(=O)CC(C)c2ccco2)CC1 c1(OC)ccnc(C(=O)NC2CC(CNC(C3(C)CC3(Cl)Cl)=O)C2)c1N N1(C(C2(C)COC2)=O)CCCC(C(N2CCN(c3ncccn3)CC2)=O)C1 N1(CCNC(Cc2cn(C)nc2)=O)CCN(C(=O)CC2CCC2(C)C)CC1 N1(C(CC2(C)CCC2)=O)CCC2(CCN(C(C3CCn4c(O)nnc4C3)=O)C2)C1 CCCC(C(O)C(=O)N(C)Cc1cccc(C)c1)NC(=O)CCCOC(C)C N1(CCNS(CC)(=O)=O)CCN(C(=O)Nc2cc(C)ncc2Cl)C(C)C1 c1(C(=O)NCC2(C(N3CC(C(N)=O)C(C)C3)=O)CC(=C)C2)cc(C)c(C)nn1 c1(C(N(C2CCC2)CC#C)=O)ccn(CCNC(=O)CCn2ccnc2)c1 C1(C)C(=O)N1.C1(C(=O)NC)(C(=O)NCC2CC2NC(=O)C2CC2)CC1 c1(N2CCCN(C)CC(C)C2)cccc(S(=O)(=O)N2CC3CCOC3C2)n1 CC12CN(C(=O)CC3CC4CC4C3)CC1(C)CN(C(=O)C1CCCc3scnc31)C2 Cc1nc2cc(C(N3CC=CC(NC(=O)C(C)(C)CN(C)C)C3)=O)c(F)cc2[nH]1 Cn1cc2c(C(=O)NCCC(O)CNC(c3cccc(F)c3O)=O)cccc2n1 CC1(C)CC(C)(C(=O)NC2CCC(CNC(c3cnc(C4CC4)o3)=O)C2)C1 N1(C(CCc2cc(C)no2)=O)CCCC(CNC(C2(CO)CC2)=O)CC1 C(C(C(=O)N(C(C)C(C)C)C)NC(=O)C(C)=CC)OCC c1(C(=O)OCC(c2ccccc2)CC)ncc2scc(Br)c2n1 c1(C(N2C(COC)CN(C(C3CC3F)=O)CC2)=O)c[nH]c(C)c(Cl)c1=O N1(C(c2nnn(C)c2N)=O)CCC(NC(c2ccc(F)c(O)c2)=O)CC(O)C1 N1(C(=O)OC(C)(C)C)CC2(CC2)CC1CNC(C(C1CC2(CCC2)C1)C(=O)O)=O N1(C(C(c2ccccc2)N(C)C)=O)CCC(CF)(NC(c2ccc(CO)o2)=O)C1 C(C(CCC)CC(C)C)NC(C(CCOC)NC(CC=CC)=O)=O C(CC(O)C(=O)N1C(C(=O)NCC2CCN(C)CC2)CCC1C)SC c1(OC)c(-n2cc(C(c3nnnn3C)Nc3ccc(Br)c(Cl)c3)nn2)cccc1F N1(C(C=CC)=O)CC(C(C)(C)O)(CNC(c2ccn(-c3ccccc3)n2)=O)C1 c1(CN2C(C(=O)Nc3cc(OC)ncn3)CC2)ccc(F)c(F)c1Br N1(C(CC2(C)CC2)=O)CCCC(NC(=O)CCc2ccc(Cl)nc2)C(F)C1 CN1C(=O)CCC(NC(C2COCCN(C(c3cc4n(n3)CCO4)=O)C2)=O)C1=O C1(C(N)=O)CN(C(C2(n3cnnn3)CCCCC2)=O)CCC1C(=O)O Cc1nc(C)cc(O)n1.c1(C(c2nnnn2CCOCC2CC2)N)cccc(Cl)c1Cl c1(N2CC(O)CC(OC)C2)cc(C)c(S(=O)(=O)N2CCCN3CCCCC3C2)cn1 N1(C(C2CCS(=O)(=O)N2)=O)CCC(F)(F)C(CNC(C2(C3CCC3)CC2)=O)C1 C1(NC(c2ccccc2Cl)=O)COCCN(C(c2cc(Cl)ncc2F)=O)C1 N1(C(=O)CCn2cnnn2)CCC2CCC(C1)N2C(=O)C=CCOC1CCOCC1 C(=O)(C(CC(F)F)NC(=O)CCCn1ccnn1)NCC(CC)CO N1(C(c2c(CC)ccs2)=O)CCCCC1CCC(=O)NCC(Cl)Cl C1(N(C(C(C(C)C)NC(C)=O)=O)C)CCCN(C(c2cncc(C)n2)=O)CC1 Cc1ccc(SCC(=O)NC2CCCC2NC(C2CCCC2(F)F)=O)c(C)c1 C=CCC(F)(F)C(=O)N(CC(CO)(CO)NC(=O)CCC=Cc1ccccc1)C c1(C(=O)NC(C2CCCN2C(c2c[nH]c(C#N)c2)=O)C)cc2c(s1)CCCCCC2 C12(NC(=O)CSCc3ccc(Cl)cc3)CCN(C(c3coc(O)n3)=O)CC1C2 n1(CC(=O)O)c(O)nc2ccc(C(=O)N(C3CCCCC3)C3CC3)cc12 C=C(C)C(O)CC(=O)N(C1CCCN(C(=O)CNC(=O)CC(F)(F)F)C1)CCO N1(C(CNC(c2cnc(C)[nH]2)=O)=O)CC2(CC2)CC1C(=O)NCc1cccnc1 C1(NC(C=Cc2ncc(C)[nH]2)=O)CC(O)CN(C(=O)CCc2ccc(F)cc2)C1 N1(C(C(C)OCCC=C)=O)CCN(C(c2nc(C)c(N)s2)=O)C(C)C1 c1(C(=O)Nc2cc(Cl)ncn2)cc(F)ncc1NCC1CCCO1 CC1CC(C)CN(CCN2CC(c3nn[nH]n3)CCC2=O)C1 c1(C(=O)OCc2c(C(=O)OC)cc[nH]2)ccc(-n2ccc(C(=O)OC)n2)cc1 C1(C(N(C(C#C)C2CC2)C)=O)CCN(C(=O)Cc2ccc(F)cc2)CC1(C)C N1(C(c2c(C)ccnc2)=O)CC(NC(C2(CN(C)C)CC2)=O)C2(CCOCC2)C1 CCC(CC(F)(F)F)C(=O)NC1CC(NC(c2cc3nc(=O)ccn3[nH]2)=O)C1 C(CCCCCC(C)C)NC(c1cc(CNC(C(C=C)OC)=O)on1)=O N1(C(c2c(C)ccnc2F)=O)CC2(CCC(C(N3CC(O)CC3C(N)=O)=O)O2)C1 N1(C(C=CC(CC)C)=O)CCN(C(=O)C=CCOC)C(c2ccc(OC)cc2)C1 CCC(CC(=O)N(c1ccccc1F)CCO)NC(=O)C(C)(C)OC(C)C N1(C(C2(F)C(C)C2)=O)CCCC2(CCN(C(=O)CC(C)(C)CC(F)F)C2)C1 C1(NC(C=CCCC)=O)CCC(C)(CNC(c2cc(C)oc2C)=O)CC1 c1(C(N2CCC(CN(C(=O)CC3CCN(C)C3=O)C)C2)=O)ccc2scnc2c1 C1(C(=O)NC2CCC3CC23)(CN(C)C)CCN(C(c2c[nH]nc2C2CC2)=O)C1 n1(CC(=O)NC(C2N(C(CSCCN(C)C)=O)CCOC2)C)cc(F)ccc1=O S(=O)(=O)(c1ccc(N(C)CC2(CO)CC2)c(Cl)c1)NC1C2N(C)C(CCC2)C1 Cc1cn2cc(C(N3CCN(C(=O)C(F)CC4CCC4)CC3)=O)sc2n1 C12(C(=O)NC(C(C)NC(C3CC=CCO3)=O)C)CC3CC(F)(C1)CC(F)(C3)C2 C(CCCCC(=O)NC1CCCN(C(N)=O)C1)NC(c1cc(C)nn1C)=O Cn1nc(C(=O)NC2(CCNC(C3CC4CC4C3)=O)CCC2)c(Cl)c1Cl C(CO)(C(F)(F)F)NC(CC1CCC(NC(C(C)OCC2CC2)=O)C1)=O C=CCCCC(C)C(c1nnnn1CCCOC)N(CC(C)(C)COC)C1CC1 N1(C(c2nc(OC)oc2)=O)CCC2CN(C(c3cc4cnccc4[nH]3)=O)CC2C1 N1(C(C=CC(CC)=CC)=O)CCOCC1CCNC(=O)CCc1cc(C)no1 C(=O)(CC1OCc2cc(F)ccc21)Nc1nn2c(=O)cc(C)nc2s1 N1(C(C(CC(=O)OC)(C)C)=O)CC2(C1)CN(C(C1C=CCCC1)=O)CCO2 C1(COC)SC2=CCOC2CN1CC(=O)NCCc1cc(Cl)ccc1OC c1(C(=O)NCC2(NC(CCCSC)=O)CC2)cncc(Sc2ccccc2)c1 N1(C(c2cnn(CC)c2F)=O)CC(NC(C2CC3(CCC3OC)C2)=O)C2(CC2)C1 c1(C(C)NC(=O)C(C)(C)Nc2ccccn2)ccc(C#N)cc1 CCC(C(=O)N1CCC(CO)(NC(c2cc(C(F)F)n(C)n2)=O)CC1)C(F)(F)F C(C1c2ccccc2CCN1C(c1cnc(F)c(Cl)c1)=O)NC(c1cc(C)no1)=O C1(CNC(C23CC2CNC3=O)=O)CN(C(CC2(CC)CCC2)=O)CC1OC c1(C(=O)NCC2N(C(c3cnc(COC)s3)=O)CC2)ccc(NC(C)=O)c(F)c1 c1(CCC(=O)NCCCCCc2onc(C(C)(C)C)n2)cccc(Br)c1 N1(C(c2[nH]c(=N)sc2)=O)CC2(C1)CN(C(=O)CCOCC1CCCO1)C2 C1(n2cc(C3N(C(C4C(c5onc(CC)n5)C4)=O)CC3)nn2)C(=O)OCC1(C)C Cn1nnc2cc(C(=O)NC3CCN(C(C4C5CCC45)=O)CC3)cnc12 CCC(C#N)(CC)C(=O)N1C2CCC(C2)C1CNC(C1C(C)C1(F)F)=O N1(C(C(CC)SC)=O)CC(NC(c2cc(Cl)c(Br)[nH]2)=O)C(C)C1 c1(C(N(C2CCN(C(C3CCCC3O)=O)C2)CCC)=O)sc2cncn2c1C c1(CNC(CCCOCCC)=O)nc2c(s1)CCN(C(c1cncnc1)=O)C2 C1(C(=O)NCC2CN(C(CN(C3CCCCCC3)C)=O)C2)CC1C1(C)COC1 c1(N(C2CC2)CC2N(C(=O)OC(C)(C)C)CCC2)cc2sccc2s1 c1(N2CCC(CCOC)C2)nc2c(c(=NC3CCC4(CC3)CSC4)[nH]1)CCCC2 c1(C(C)(C)N(C(=O)C(C)NCC2CCCO2)CC(C)C)n[nH]c(CO)n1 N1(C(C=CCN(CC)CC)=O)CCCCC1C(=O)NCCCCC1CCCC1 N1(C(C2CC2C(F)(F)F)=O)CC(C(=O)NC2CC23CCCC3)C2(CC2)C1 CC(CNC(=O)C=CCN(C(=O)C(C)n1cncn1)C)CO c1(C(=O)NC(C)(CNC(=O)C(O)C2CC2)CO)cc(F)ccc1F C1(NC(C(c2ccccc2)OCC)=O)CCN(C(C2C=CC=CC=C2)=O)C(C)C1 CCCCCC(F)C(=O)NC1CC(CNC(=O)C(n2ccc(C)n2)C)CC1O N1(C(=O)NCCCC)CCCC(C(=O)NCC(C)C(C)(C)C)CC1 c1(NC(N2CCCCCC2Cc2ccc(F)cc2)=O)ccc2nnnn2c1 C=CCC(C)(C(=O)NCC1CC(C)N(C(c2nn(C)c(Cl)c2Cl)=O)C1)N(C)C C12(NC(C(CSC)OC)=O)CC(CNC(c3c(F)cccc3F)=O)(C1)OC2(C)C c1(CN(C(Cc2ccc(C)s2)=O)C)ccc(CNC(=O)C=C2CC2)cc1 c1(C(C)C)ccc(C(C)C(=O)NC2C=CC(CNC(c3ccccc3)=O)C2)cc1 c1(OCC)ccnc2sc(C(=O)OC)cc12.C12CN(CCO1)C(=O)C(C)OC2C c1(SC)nc2ncnc(N3CCCC(CNC(C4(C)CCC4)=O)C3)c2s1 Cc1cc(N)cnc1C(=O)NCC1CCN(C(C2(C)CSC2)=O)CC1O c1(CNC(C2N(C(C=C=C(C)C)=O)CCSC2)=O)ccc(C)cc1F CC1CCC2(CC2)N(C(c2ncn(C)n2)C(=O)NC2(C)CC2)C1 N1(C(CCCCSC)=O)CCCC(NC(=O)Cc2ccc(F)cn2)C(F)C1 CCC1=NOC(C(=O)NC(C)CCCNC(=O)C(N2CCCCC2=O)C)C1 CC1CC(CNC(c2csc(C3CC3)n2)=O)CN1C(c1cnc(O)n1C)=O CC1(C)CC(CC(=O)NC2(CO)CCN(C(c3c[nH]ccc3=N)=O)CC2)CCO1 Cc1ncc([N+](=O)[O-])cc1C(N1CC(C)(NC(=O)C=C2CCOCC2)C1)=O c1(C(=O)NC2CCCN(C(C3CC(C)N(C)C3)=O)C2)c[nH]c(=O)c2ccncc12 c1(CN2C(C(N3CCCC(O)C3)=O)C=CC2)c(Cl)cccc1Br c1(C(N2CC(C(C(=O)N(C)CCn3ccnc3)O)C2)=O)cc[n+]([O-])cc1 CC(C)CC(C)CC(=O)NCC1CCCN1C(c1cc(CCCO)on1)=O C1(NC(CCNC(N)=O)=O)CCCN(C(c2cc(Cl)ccc2N)=O)CC1 C#CCC(C)C(=O)N1CC(NC(=O)CSc2ccccc2OC)C(O)C1 c1(NC(=O)NC(CNC(C2C(=C)C2)=O)(C)Cn2cccn2)cn2ccsc2n1 N1(C(C=CCCC(C)C)=O)CC(C)(CNC(C2CN(S(C)(=O)=O)C2)=O)CC1(C)C c1(C(=O)NC(CCC(N2CCC(CC)(CO)CC2)=O)(C)C)cncc2[nH]ccc12 C12CCC3(CN(C3)C(=O)CC(=O)N1)O2.c1(C(=O)OC)cnc(OC)c(Br)c1 N1(C(c2ccn(C)c2)=O)CCC2(C(N3CCCC(C)(C#N)C3)=O)CCCC12 C1(NC(c2c(OC)scc2)=O)CN(C(c2cn(CC(N)=O)nn2)=O)C(C)(CO)C1 c1(C(N2C(CCCNC(C3N(CC)CC3)=O)CCCC2)=O)cccc(N)c1O c1(C(=O)NC2CC3CN(C(CCOCCN(C)C)=O)CC32)ccnc2[nH]nnc12 N1(C(c2c(OC)c(=O)cco2)=O)CCN(c2ncnc(=N)[nH]2)CC(O)C1 CN1CCCC(C(C)(C)C(N2CCC(NC(C3CC(O)C3)=O)CC2)=O)C1 C(C(C)(O)CC(=O)N1CCN(CC(=O)NC2CCC(C(C)C)CC2)CC1)OC C1(NC(C2N(C(CNC=O)=O)CCC2)=O)Cc2cc(Cl)ccc2O1 N1(CCNCc2nccc(OC(C)C)c2)CCOC2(CCCCC2)C1 C(=O)(C1=NOC2CN(C(=O)CC(C)(C)F)CC12)OCC c1(C(N(CC(C)(C)CNC(=O)CC2=CCCC2)C)=O)cncc(P(C)(C)=O)c1 c1(OC)cc(C)c(Cl)cc1COC(=O)C(F)(F)C1(OC)CCCC1 N1(C(CNC(C(CC)C)=O)=O)CC2CCCC(C(=O)Nc3oncc3C)(C2)C1 N1(C(C)=O)CC(NC(=O)COc2ccsc2Cl)C(O)C1 n1(C2(N(CCOC)C(c3cc[nH]c3)=O)CC2)cc(C2CCCC2O)nn1 C#CC1(O)CCN(C(C)C(=O)NCC(C)N(C)C(c2scnc2C)=O)CC1 N1(C(CN(C)C)=O)CCC(C(=O)N(C2CC2(C)C)C)CC1(C)C c1(C(N2C(C)CC(CNC(C(C(CC)C)OC)=O)C2)=O)cc(F)cc2nn[nH]c12 CC1Oc2c(C(N3CC(C)(NC(c4cc[nH]n4)=O)C3)=O)cccc2NC1=O c1(C(=O)NCC(CC(C)C)NC(c2n(CC)nnc2C)=O)cnc(C)nc1C C(=O)(C(CC(C)C)C(C)C)N1C(c2onc(CN3C4CC(=C)C(C4)C3)n2)COCC1 CC(CC(=O)NC(C)(C)CC=CC(=O)NC1CCCC(C)(C)C1)CC(C)(C)C c1(NC(C(CC2CCOCC2)NC(C(CCCC)F)=O)=O)cc(C)cn(C)c1=O N1(C(c2c(OC)ccnc2)=O)CC2CC3CC2C1C3Nc1cc(=O)n(C)cn1 Cc1cc(C(=O)NCC2CCC(NC(c3ocnc3C)=O)CC2)cc([N+](=O)[O-])c1 c1(C(N(C2C3CN(C(CC(C=C)C)=O)CC32)C)=O)cccc(=S)n1O C1(C(=O)NC(C(=O)N(CCCCCC)C(C)C)CC2CC2)CCc2n[nH]cc2C1C Cc1cc(C(N2CC3=C(C2)CN(C(C2(CO)CCCO2)=O)C3)=O)cc(N)c1O N1(CC)CCCCC1C(=O)NCC(O)CN(C(=O)C(=Cc1c[nH]cn1)F)C N1(C(C(C)C2CC2)=O)CCN(c2ccc(C(=O)NCc3cccc(F)c3)cn2)CC1 N1(C(CC2(OCC)CCC2)=O)CC(NC(C2(CC#N)COC2)=O)C2(CCC2)C1 C1(C(=O)NC(CC=C)CC)COCCN(C(=O)C(C)=CC2CC2)C1 NS(=O)(=O)c1cc(C(=O)NC(C)(CNC(C2(F)CCCC2)=O)C2CCC2)cs1 c1(CCC(N2CC(C)(NC(c3cncs3)=O)C2)=O)cccc(C#N)c1 N1(C(=O)C(F)F)CCC(F)(F)C(NCc2cc(F)cc(F)c2Cl)C1 c1(C(N2CCC(O)(CCNC(C3CC(=C)C3)=O)C2)=O)ccc2ccncc2n1 Cc1ccccc1OCCCC(=O)NCC1(CNC(=O)CCC=CBr)CC1 C1(C)(C(=O)N(C)C)CCCC1.C12(CC1)C(=O)NCCN(C)C2=O Cc1scnc1NC1CN(C(=O)C(C)(C)Sc2ccccc2)C1 C1(NC(CCCCCOCC)=O)CCN(C(=O)Cc2csnn2)C12CCC2 C(CC(C)(C)C(=O)N1CCC(O)(C(C)NC(=O)CCSC(F)(F)F)CC1)OC N1(C(c2c(CC)n(CC)nc2)=O)C2CCC1CC(CNC(=O)C(C)SC)C2 c1(C(=O)NC2CCN(C(COC3(C)CCC3)=O)CC2O)nc2c(s1)COCC2 CCC(=O)CCC(=O)NCC1CCCCC1C(=O)NCCSCCCO c1(NCC(=O)NC(CCCC)CNC(=O)CC2CC=CCN2C)c(C)cccc1Cl c1(CC(=O)NCC(C2CC2)OCC)ccc(OC)c(F)c1.N12CCC(C1)C2=O C(=O)(C(F)C(C)(F)F)NCC(N1CCN(C(C2CCOC2C(C)C)=O)CC1)C C(CC(N)=O)(C(=O)NCC1(C)CNC(=O)O1)NC(CSC(C)C)=O C1(NC(CC2CCCN(C)C2)=O)CCCCCC1C(N1CCC1CO)=O C1(NC(C(F)OC)=O)CCN(C(=O)CSCC2CCCO2)C12CCC2 N1(C(c2cn(CC=C)nc2)=O)CCC(CNC(C2CCC2C(F)F)=O)C12CC2 c1(NC(C(COC(C)C)NC(C(CC)NC(N)=O)=O)=O)cc(C)ccc1C C1(NC(C(C)C#N)=O)CCN(C(c2ccnn2CC(F)F)=O)C(C)C1 C(=O)(C#CC1(C)CCCO1)N1CC(C2(NC(c3ccc(C(=O)OC)[nH]3)=O)CC2)C1 C=CCC(C)(C)C(=O)N(CC(=O)NCC(C)(C)C(F)(F)F)C CC1CN(C(c2cccnc2)=O)CC1(C)CNC(=O)CSCc1ccccc1Cl C1(N=[N+]=[N-])(C(=O)OCC)CCN(C(c2cnccc2Br)=O)C1 C#CC1(C(=O)NC(C)CC2CCOC2)CCN(C(c2ccc(C)cc2)=O)CC1 C1(NC(CCC#C)=O)C2CC3CN(C(C4CCC5(CCCC5)CC4)=O)C1C3C2 c1(C(=O)NCC(CN(C(C(C)SCC)=O)C)O)ncc(Br)cc1C N1(C(COCC=C)=O)CCC(C2CCN(C(c3cnc(C)nc3C)=O)C2)C1 c1(C(C)=O)ncc(C(=O)NCC2CC2NC(=O)C(N2CCCC2)C2CC2)s1 N1(C(C2CC(NC(C(F)=CCC)=O)C2)=O)CCC1C=C C1(CC(N2CCC(F)(CNC(=O)CCOCC(F)F)C2)=O)CN2CCN1CC2 C1(N(C)C(C2CCCN2S(C)(=O)=O)=O)CCC(NC(=O)CSCC(F)(F)F)CC1 c1(SCCC(=O)NCC2CC(NC(CSSC)=O)C2)ccc(F)cc1F N1(c2cc(C(=O)OC(C)(C)C)[nH]n2)CCN(C=O)CC1.C1(C)(S)CCCCC1 c1(CCC(=O)NCC=CCNC(C2OC3CCC2C3)=O)cccc2c1OCCO2 c1(NC(=O)CCC(C)OC)n[nH]c(=NCc2ccc(SCC3CC3)c(F)c2)o1 C1(C(C)(C)CNC(C2CC2C(C)(F)F)=O)CN(C(=O)C(N)=O)CCO1 Cc1cc(C(N2CCCCC2CCCNC(=O)C=Cc2cscn2)=O)c[nH]c1=N c1(CCN(C)CC)nnc(C2=NOCC2)n1CCCCc1ccc(O)cc1 Cc1cc(CC(N2CC(CN(C(=O)C(c3cccc(F)c3)(C)C)C)C2)=O)n(C)n1 C1(C(N(CCCCN(C(C2ON=C(CC)C2)=O)C)C)=O)CC2(CCOCC2)CO1 c1(C(=O)NC2CN(C(C(CSC)C)=O)CC2O)ccc(S(=O)(=O)N2CCCC2)o1 C(=O)(C(C#N)=CCl)NCc1ccc(C(=O)NCCCC(=O)OC(C)(C)C)o1 C(=O)(C(O)C(CCC)C(=O)NOCC(C)C)N(CCSCC#C)C1CC1 c1(C(=O)NCC2(NC(c3cc[nH]n3)=O)CC2)ccc2c(n1)CCCN2 C1(CNC(C(CC)C)=O)CC12CCN(C(c1sc(Cl)cc1Cl)=O)CC2 C1(C(N2CCC(C(C)NC(c3cnco3)=O)C2)=O)CC12CCOc1ccccc12 N1(C(c2c(COC)nc(C)nc2)=O)CC(C)CN(C(c2ccoc2Br)=O)C(C)C1 N1(C(CCC(C)OC)=O)CCN(C(c2nc(Cl)c(Cl)s2)=O)CCC1C C1(C(=O)NC(CCSC)C(=O)O)CCCN(C(c2n[nH]cc2Cl)=O)CC1 c1(SC)cccc(CC(=O)NCCCCNC(=O)C(F)(F)c2ccccc2)c1 Cc1cc(C(=O)NC2(CCNC(c3nnc(S)n3C)=O)CC2)ccc1Br C(CC(C(=O)N1CCCC(CCNC(=O)C2=C(C)CC2)C1)OC)OC C(=O)(C1=NOC2(CCC2)C1)NCCCCCCC(=O)Nc1ccc(CC)nc1 CCCCC(CC(=O)NC1(CO)CCCCC1)NC(C1CCC(OCC)CC1)=O C1(NC(c2cc(CC)no2)=O)CCN(C(C2CC3(CC3)C2)=O)C12CC2 N1(C(COCCOCC#C)=O)CCCC(NC(C2CCN(C)C2=O)=O)C1C CC(C)C1=NOC(C)(C(=O)NCCCCNC(=O)CCc2ccn(C)c2)C1 c1(-c2cn(CC(=O)NCCOCC(=O)O)nn2)cc(F)ccc1F C1(NC(c2n(C)nnc2)=O)C2CCCCN(C(c3cncc4[nH]ccc34)=O)C12 c1(C(=O)NC(C(C)NC(c2c(COC)cc[nH]2)=O)CO)ccnnc1C C#CCC(C(=O)NCCC(C)NC(C1CC(N(C)C)C1)=O)C1CC1 C1(CC(=O)NCC(C(C)C)NC(c2cc(CO)[nH]n2)=O)NC(=O)NC1=O S(=O)(=O)(CC(=O)NCC(C(C)(C)C)NC(=O)CC1CCCCN1C)NC C(C(=O)N1CCC(C(N)=O)O1)c1cn(C2CCN(C(c3cn(C)nc3)=O)C2)nc1 N1(C(c2c(C)nco2)=O)CCC2CN(C(=O)C(=O)Nc3ncc[nH]3)CCC2C1 C12(C(N3CCC(C)(CO)C3)=O)COCC1CN(C(C13CSCC1C3)=O)C2 n1(C(C)C(=O)NCC2CCN(C(C34CC(O)C3C4)=O)C2)c(=O)oc2ccccc12 Cc1ccc(C(=O)N(C2CCN(C(=O)C(F)C3CCC3)C2)C)c(O)n1 c1(CC)nnc2n1CCCC2C(=O)N1CCN(C(C2CC(O)C2)=O)CC(C)(C)C1 CC(C(C)C(=O)NC(c1nc(=O)o[nH]1)C)NC(=O)C=Cc1cnccn1 c1(OC(C)C)ccccc1C(=O)NCC1CN(C(C2CCCSC2)=O)C1 C(c1cccc2ccccc12)=CC(=O)NC1CCCC(N(C(CCSC)=O)C)C1 c1(C(=O)NCC2CC2NC(c2ccnn2CC(F)F)=O)cc(F)c(F)cc1F CC(CO)C(=O)NCCC(C)(C)NC(=O)CCc1nnc(C2CC2)o1 c1(CNC(=O)CCc2ccoc2)ncccc1C(=O)NCC(=O)NC1CC1 C1(NC(c2ccc(C)cc2)=O)CCN(C(c2nc(O)[nH]c(=O)n2)=O)CC1C N1(CCNC(=NCC)NCC(=O)OC)CCCC2CN(CC)CCC12 c1(NC(c2nc(-c3c(OC4CC4)ccc(C)c3)sc2)=O)cccc(F)c1[N+](=O)[O-] C1(CC(=O)N(CCC)CCNC(=O)C(C)Cc2cnco2)CCCC(=O)C1 Cc1ccn(CC(=O)NC2CC(NC(=O)CSCCC(F)(F)F)C2)n1 N1(C(c2cnc(C)nc2)=O)CCC(C)(C)C(CNC(=O)CNC(=O)C(C)(C)C)C1 NS(=O)(=O)CC(=O)NCC#CCNC(=O)C(C1(O)CCCCC1)(F)F c1(C(=O)NCCC2CC(NC(c3c(C)cnnc3O)=O)C2)cc2c(s1)COCC2 C1(c2nc(C(c3cccc([N+](=O)[O-])c3)OC)on2)CCC2CCCCC2C1 c1(C(N(C(CN(C(C(c2c(C)cccc2)C)=O)C)C)C)=O)ccc2snnc2c1 CCC(C(=O)N1CCCC1C(C)NC(c1cnc(C2CC2)s1)=O)c1ccccc1 CCCCC(C(=O)NC(C)CN1CCCC1)NC(c1ccc(=N)[nH]n1)=O C(=O)(CCCC(F)(F)F)N1CCC(C(=O)Nc2cncc(C)c2)C(C)C1 c1(CCNC(=O)Nc2c(C)n(C(C)C(C)(C)O)nc2)cccc2c1OCCO2 CC1(C2CC2)CCN(C(=O)C(Cn2cncn2)NC(c2ccoc2)=O)C1 Cc1cc(Cl)cc(C)c1OCC(N1CCOC(CCNC(C2(C)CC2C)=O)C1)=O N1(C(C)C(=O)NCC2CCCO2)CCSC2(CCOCC2)C1 O=C(CCO)NCC1CC1CNC(c1ncc[nH]1)=O C1(C(C)C)CCC(C(=O)NCCC2(C#N)CCC2)N1C(=O)C=CCN1CCC1 c1(CCC)c(C(=O)NC2CC2NC(=O)C(C)c2ccco2)cnn1CCO C1(NC(C(CCCC)C(C)C)=O)CS(=O)(=O)CC1N=c1[nH]nc(-c2ccccc2)o1 N1(C(C(CC)n2cncn2)=O)CC2CCC2(CCNC(=O)C(=O)C(C)(C)C)C1 c1(C(N2C(CCNC(C3(C)CN(C)C3)=O)CCC2)=O)cncc(C#N)c1 C1(C)(C(C)C)CCC(NC(C=CCC(C)(C)NC(=O)CNC(=O)NC2CC2)=O)C1 N1(CC(N2CC(N(C(=O)CC3CCC(O)C3)C)C2)=O)CC2CCC1C2 N1(Cc2onc(C(C)C)n2)CCN(C(C)(C)CN(C(=O)CC2CCCC2)C)CC1 Cc1ccc(NC(C2CCN(C(=O)OC(C)(C)C)CC2O)=O)c2[nH]ncc12 c1(NCc2cc(C)[nH]c2)nc2c(c(=NCC(C)(C)OCCO)[nH]1)COCC2 C1(NC(c2n[nH]c(CC)c2Cl)=O)CCCCN(C(c2cc(N)ccc2F)=O)C1 S(=O)(=O)(c1ccc2[nH]c(=NCC3(C)CC3(C)C)sc2c1)N1CC(CCC)OCC1 c1(C(=O)NCCN(C(C2CC(OC)C2)=O)CC)c[nH]nc1C(F)(F)F c1(C(C)=O)cc(Br)ccc1NC(C1CC(O)CCN1Cc1cc(N(C)C)cs1)=O C(=O)(C1CCCc2nncn21)N1CCCC(NC(c2cc(C)c(C)[nH]2)=O)C1 C1(CNC(CC(CCC)C)=O)CCC2CN(C(=O)C(CCC)N(C)C)CC12 N1(C(CC(c2ccc(F)cc2)C)=O)CCC(CF)(NC(c2cc(Cl)n(C)n2)=O)C1 N1(C(CSCC=C)=O)CC2(C1)CN(C(c1sc3ccc(Cl)cc3c1C)=O)CCO2 C(C(=O)N(OC)C1CCOCC1)C1CCC(=C)CC1 N1(C(c2cnc(CC)[nH]2)=O)CC2CCCC(CNC(=O)CC3(CO)CC3)C2C1 c1(OC)ccc(O)c(C(C)(O)CNC(=O)NCCCC(O)C(C)(C)C)c1 C(=O)(C(O)CCCNC(C12CCC(C1)C2)=O)NCC(C)(C)N(C)C C(=O)(CCC(C)(C)NC(c1cnc(C)c(C)c1)=O)NCc1nc(C)c(C)[nH]1 N1(C(C2=NOC(C)C2)=O)CC2CCC1CN2C(=O)COCC1CCOCC1 C#CCC(CC(=O)N1CCC(O)(CC)C1)NC(c1sccc1C#N)=O C(=O)(C(C)C(C)(C)C)N1CC(OC)C(NC(=O)CCn2cnccc2=O)C1 N1(C(C(=O)Nc2ccc(C)cn2)C)CCS(=O)(=O)C(CCNC(C2CC2(Cl)Cl)=O)C1 c1(OC(C)C(F)(F)F)cc(NC(=O)Nc2cccc(CC#N)c2)ccc1F C1(C)(NC(c2cc(OCC)ncc2)=O)CCCN(C(c2cnc(C(C)C)[nH]2)=O)C1 c1(C(N2C(CNC(c3cnn4c3OCCC4)=O)CC2)=O)cc2c(nn1)OCCS2 c1(CC(=O)NCCN(C(=O)CC2CS(=O)(=O)C2)CCOC)cnc(Cl)cc1C Cc1cc(C#N)ccc1C(=O)NC1CC(C)N1C(=O)Cc1cncnc1 C1(C)(NC(C(CCC)OC)=O)CCCN(C(c2cccc(C3CC3(F)F)c2)=O)C1 CCC(CC)C(C)C(=O)N1CC(N=[N+]=[N-])CC1C(N1CCC(N2CC=CC2)C1)=O CC(C)(C#N)C(=O)NCc1ccccc1CNC(=O)CSc1nncs1 c1(C(C)NC(C2CCCCN2C(c2cnccn2)=O)=O)cccc(S(C)(=O)=O)c1 C1(C(N(C2CCC2)CC=C(C)C(F)F)=O)CC12CCN(C(C1CC1CF)=O)CC2 c1(C(N2CCC(CNC(C(n3ncc(C)c3)C)=O)C2)=O)nccc(Cl)c1C N1(C(CC(C=C)CC)=O)CCCCC12CC(NC(=O)COC1CCC1)C2 C1(CC)CC(C(=O)NC(C)C(F)(F)F)CCN1C(=O)C(CO)N(C)C C(CC(=O)N1CC(CO)C2(CC2)C1)(C(C)(C)C)NC(C(CC)C(C)C)=O Cc1ccc(C=CC(=O)NCC2(NC(c3ccc(C)nc3)=O)CC=CC2)nc1 N1(C(CN(CC)NC(N2CCC(C(N(C)C3CC3)=O)C2)=O)=O)CCCC(CC)C1 C1(O)(CC=C)CN(C(C2CC(=O)C2CC)=O)C1 c1(SCC)nccnc1C(N1CCC1CC1CC=CCC1)=O.C(=O)(CCCF)N C1(C(N(C2CCN(C(=O)CC3CCCOC3)C2)CCO)=O)COC2CC1C2 Brc1csc2[nH]c(CN(C3CCCCC3)CC3CC3)cc12 CCCC(C(=O)N(CCCNC(C1CC2(C1)CC1(CC1)C2)=O)CC)C(C)C C(=O)(CCC(C)NC(=O)C=Cc1ccnn1C)N(CCCCC)C C1(NC(C=Cc2n(C)cnc2)=O)CCCC12CN(C(C1NC(=O)OC1C)=O)C2 c1(OC)cc(C(=O)NCCC(C)NC(=O)C=C(C)c2cnn(C)c2)cc(Cl)c1 N1(c2ncnc(C)c2F)CCCC2(CCN(C(c3cccc(C#N)c3Cl)=O)C2)C1 c1(N(C)C(C2CC2CCNC(=O)COCC2CCOC2)=O)cc(CO)on1 C1(C(=O)NC2CN(C(C3(C4CCCCC4)CC3)=O)C3CC23)CN2CCCN1CC2 C1(C(=O)NC(C)(C)CCNC(c2ccccc2CC#N)=O)CCc2ccnn2C1 C1(C(C)C)CN(C(c2ccc(O)nn2)=O)CCN1C(=O)Cc1nc[nH]n1 O=S(=O)(c1ccccc1C(F)(F)F)N1Cc2ccc(SCCO)cc2C1 CS(=O)(=O)CC(=O)NC1CCOC(C(=O)NCc2ncc(Cl)cn2)C1 c1(CC#N)ccccc1C(=O)NCC1CC1CC(=O)NC1CCC(CO)CC1 Cc1nscc1C(=O)NC(CC1CC1)C(=O)NCc1nc(CO)n[nH]1 Cc1cc(O)c(F)cc1NC(C1(CCNC(=O)C(C)CO)CCOCC1)=O c1(C(=O)NCCCCNC(=O)CC(O)c2cncnc2)cc(Cl)ccc1O c1(NCc2c(OC)nsc2)cc(Br)ccc1S(=O)(=O)N(C)C(C)C1CC1 C(C(C)C(C)C(=O)NC1(CNC(=O)CSC)CC(F)(F)C1)OC C12(C(=O)NCCN(C(=O)COCc3nccn3C)C(C)C)CSCC1C2(F)F c1(CN(CC(F)(F)CN2CCOCC2)C)ncccc1Br C1(C(=O)NC(C2CCN(C(C3(C#N)CCOCC3)=O)CC2)C)CCC(=O)N(C)C1 N1(C(c2c(CC)nccc2)=O)CC2(C(N3CCCC(COC)C3)=O)CCC1CC2 c1(NC(C2N(C(C(C)C)=O)CCCC2)C)nccc(S(C)(=O)=O)n1 N1(C(C(=O)NC(C)CC2CC2)=O)CC2CCCC12 Cc1nc(Cl)sc1C(=O)Nc1ccc(CC(=O)Nc2cnn(C3CC3)c2)cc1 c1(C(N(CC(C)C)CCC#N)=O)ccnc(SCC(=O)NCc2cccnc2)c1 N1(C(c2c(C)cc(C(=O)OC)o2)=O)CC(CNC(C2CCCC2)=O)CC(C)C1 N1(C(C(C)C(F)F)=O)CC(C(=O)NC(C)CN2CCCC2)CCC1(C)C Cc1ccc(F)c(C(N2CC(N(C(=O)COCC3(F)CC3)C)C3(CC3)C2)=O)c1 N1(C(C2CCC(C(N)=O)CC2)=O)CCC(C2CC2)C1CN(C(=O)C1=C(Cl)CC1)CC c1(S)ncc(NC(=O)Nc2c(Br)n[nH]c2Br)cn1.N1(C(CSCC)=O)C(=O)CNC1=O N1(C(c2ncn(C)c2)=O)C2CCC1CC(F)(CNC(C1CCCCNC1=O)=O)C2 C(=O)(C(C)CC(C)(C)C)N1C(C)(C(=O)NCC(CC(=O)OCC)C)C=CC1 C12(C(N(CCCC=C)CC)=O)COCC1CN(C(c1ccc(CCC)cc1)=O)C2 C1(C(N2CCOC(C(C)C)C2)=O)C(CC)CCCN1C(=O)Cc1cccnc1O CC1CCC(C(N2CCCCCCC2)=O)CN1C(C1CN(C(=O)N(C)C)C1)=O N1(C(c2c(C)ccc(C)c2)=O)CCCC12CN(Cc1cc(F)cc(I)c1)C2 C=CCC(C(=O)NCCN1CCN(C(C2CCCCC2C(F)(F)F)=O)CC1)OC C1(CNC(CC2(N(C)C)CC2)=O)C2CN(C(n3ccc(C(C)(C)C)c3)=O)CC12 CC(C)(C#N)CC(=O)NC1CC(C(F)C(N2CCCC(F)(F)C2)=O)C1 N1(C(C(C)n2ccnn2)=O)CCC2(CC1)CC2CNC(c1coc(CO)c1)=O CCCC(CC)C(=O)N1CCC(NC(=O)COc2cnn(C)c2)C1C C1(CC(=O)NCC2C(NC(c3nc(C)nc(O)c3)=O)C2)COc2ccccc2O1 Cc1cc(NC(=O)C(=O)N(C)CC2CC2)c(C)cc1C(N1CCCCC1C)=O C12(CNC(c3nsnc3O)=O)CC(CCO1)N(C(C1CC3C=CC1CC3)=O)C2 C1(O)(CC(=O)NC2CCC(CNC(c3cncc(Cl)c3)=O)CC2)CCOCC1 C12(C(N3CC(C)(NC(c4n(C(CC)C)ncc4)=O)C3)=O)CCC(CC1=O)C2 C1(C(=O)NOC(C)CC)CC(C(=O)NCC2CCCC2)=NO1.N1(CC)CCOCC1 C1(NC(c2n(C)cnc2)=O)CCCCN(C(=O)NCC2CC2c2ccccc2)C1 c1(C(=O)NC2C=CCC(C(=O)NC(CCCC=C)C)C2)c(C#N)ncn1C C(=O)(C(C(C)(C)C)N1CCCC1=O)N1CCC(n2cc(CCSC)nn2)C1 c1(C2(NCC3(C)N(C)CC(OC)C3)CCC2)c(F)cc(Br)cc1F C1(CS(=O)(=O)NC(c2cccc(C)c2)CN(C)C)CC12CCCc1ccccc12 C1(O)(CNC(CSCC(N)=O)=O)CCCN(C(c2cncnc2C2CC2)=O)C1 C1(C(=O)NCC2(NC(c3[nH]cc(C)c3)=O)CCCC2)OC2CCC1CC2 c1(CCNC(C(=O)NC(C2CCOC2)C)=O)cnc(C(F)(F)F)s1 c1(OC)ncc(C(=O)N(C2CC3CC2N(C(C2(C)CS(=O)(=O)C2)=O)C3)C)c(C)n1 c1(NC(C2(C(=O)OC)CCNC2)C)ncnc2cc(C(C)(C)C)sc12 c1(NC(CCC2(NC(C3CC(OC)C3)=O)CCCC2)=O)ccccc1N=[N+]=[N-] Cn1nc(C(=O)NCC2CC3(CC3)CN2C(=O)CC2(C)CC2(F)Cl)c2c1CCC2 C(=O)(C(C)(C)CNC(C1CCC(NC(C2CCC(O)CC2)=O)C1)=O)NC C1(C(=O)NCC(C2CCC2)OC)CCCC(NC(c2nnsc2N)=O)C1 c1(COC)ccc(C(=O)NCC2(F)CN(C(c3ncoc3C3CC3)=O)C2)s1 C1(NC(C2(CC)CCNC2=O)=O)CCC2CC1CN2C(=O)Cc1ccn(C)n1 C1(C(=O)NCCCOCCN(C(=O)CCC2OCCO2)C)CCCC(C2CC2)O1 c1(C(N2CCC(n3cc(CCC#N)nn3)CC2)=O)cnn2cccc(F)c12 C12(NC(c3c(C)n[nH]c3)=O)CCCN(C(c3c(Cl)csc3Cl)=O)CC1C2 c1(SC)cc(C(N2CCCC2CCC(=O)NCC(C)(C)C2CCCO2)=O)co1 N1(C(c2c(C)nc(CCC)s2)=O)CCC(C)C(NC(=O)CC2(O)CCOC2)C1C C(=O)(C1=CS(=O)(=O)CCC1)NC(C)CCN(C(=O)C(F)CC1CCCCC1)C C1(NC(CS(CC)=O)=O)CN(c2ncnc(C)c2Br)Cc2nccn2C1 N=c1[nH]c(CCC(=O)NCC2C=CC(NC(=O)CCOC3CC3)C2)cs1 C(C(C)(C)C(=O)N1CC(C(=O)NC2C3CCCC23)C(C)C1)OC(C)C CC(CCCCNC(=O)CC1CC1(Cl)Cl)NC(C1CC(F)(CO)C1)=O c1(C(=O)NC2C(NC(CCc3nnc(CC)o3)=O)CCCC2)n[nH]cc1[N+](=O)[O-] c1(C(=O)NC2CC(C)(CNC(c3nsnc3O)=O)C2)n[nH]c2c1COC2 CCCC(C)(CCC)C(=O)NC1CC(CNC(c2ccnc(N(C)C)c2)=O)C1 CC1(C)CCC(C(N2CC(NC(c3cc(CC4CC4)on3)=O)C(CO)C2)=O)C1 CCCC(C(=O)Nc1cccc(CC(=O)NC2(O)CN(C(N)=O)C2)c1)N(CC)CC c1(SCCN2CCC(C(=O)NCCc3ccncc3)CC2)nc2ccccc2s1 C1(C(=O)NC)CCN(NC(C2C3CN(C(c4nccnc4Cl)C)CC23)=O)CC1 c1(CCC(=O)NC2CCC(CCN(C(C(C)(C)C)=O)C3CC3)C2)ccnc(Cl)c1 C1(OC)CC(NC(=O)CCc2ccccc2)CN(C(C2CC23CCC3)=O)C1 Cc1cccn2nc(C(=O)N(C3CCN(C(c4cncnc4)=O)CC3C)C)cc12 N1(C(C(C)S)=O)CCC2CCC(C1)N2C(=O)NC(=O)C(=O)O N1(C(=O)Nc2c(OCC#C)cccc2)CCc2[nH]c3ccc(F)cc3c2C1 c1(C(=O)Nc2cncc(C)n2)cnc2ccc(-c3ccc(F)c(C#N)c3)cn12 c1(C(C)NC(CNC(C)=O)(C)C)ccc(F)cn1 N12CCC(C1(C)C)C2=O.Cc1c[nH]nc1C1(CNC(=O)C(C)n2ccnn2)CC1 C1(OC)CN2CCCC2(C(=O)NCCc2nccc(Oc3ccc(F)cc3)n2)C1 N1(C(C2(NC(c3cc(C)oc3C)=O)CC2(C)C)=O)CCC(C)(C2CC2)C1 N1(C(CCSCCCC)=O)C(CNC(=O)CCc2ncco2)CC2CC12 CC(CCC(C)(C)C)C(=O)N(c1nc2ccccc2s1)Cc1ncnn1C CC(C)C(O)CC(=O)N1CC(F)(F)CC1CNC(C1CCN1C(C)(C)C)=O c1(N2C(C)CN(C(=O)CC(=O)NCC(F)(F)F)CC2)nc2ccc(F)cc2o1 CCCC(C(O)C(=O)NC(C)(CC=C)CC)NC(=O)C(=O)CC(C)C C1(CNC(C(CC#C)C2CC2)=O)C(C)CCCN1C(=O)C(O)Cc1ccccc1 C1(C)(NC(COCC(CC)C)=O)CCN(CCCl)C1 c1(C(N2C(CNC(CCOCC)=O)C(C)(C)CCC2)=O)cnc2n1CCCC2C C1(CNC(CCC2(C)CN(C(C3C4(CC4)C34CC4)=O)C2)=O)CCCC2(CC2)C1 c1(OC)cc(OC(C)C)cc(C(=O)NC2CCC(c3ccccc3)CC2F)c1 C1(C)(OC)CC(NC(=O)C(CNC(c2cc(C)nc(O)c2)=O)OC)C1(C)C C(=O)(C1=CCN(C(C2C3CN(C)CC23)=O)C1)NC(CC(=O)OCC)(C)C C1(CC(N2C(CC)CC(O)C2)=O)CCN(C(=O)CC2CCCC(=O)C2)C1(C)C C(=O)(CCC(C)(C)[N+](=O)[O-])N(CCCNC(c1cncc(C=C)c1)=O)C C=C(CCCNC(=O)C(C)(N)C1CCCC1)C(C)(C)C c1(NC(C2(OC)CCSC2)=O)cc(NC(c2ccc[n+]([O-])c2)=O)ccc1C C1(CC(=O)N(C2CC(NC(C3CCN(CC(F)(F)F)C3)=O)C2)C)C(C)(C)C1(C)C CC1CC(C)CCN(C(C2CC2CNC(C2CC3(CCO2)CC3)=O)=O)C1 c1(C(=O)NC(CC=C)CNC(c2c(C)csc2Cl)=O)ccc(C(C)(C)C)nc1C c1(CC)c[nH]cc1C(=O)NCC1OCCC1C(=O)NCC(c1ccsc1)O C1(CNC(COCCCC#C)=O)N(C(=O)CC(C)OC)CCCC1(C)C CC(CNC(C1CCOCC1)=O)C(=O)NCCN(C)C(C1CCC1)C CCCCC(F)C(=O)NC(Cc1ccon1)C(=O)N1CCC1(C)CC(=O)NC C1(O)(CNC(C(CC)SC)=O)CCCN(C(c2cc(OC)ccn2)=O)CC1 c1(C(CNC(CC(C)=O)c2ccccc2)(F)F)ccccc1F n1(CCCCCOC(C)=O)ccc(=NC(=O)CCc2ccsc2)[nH]1.CCC1C(=O)N1 Cc1cccc(CCNC2CCOC(c3ccncc3)C2)c1 C1(CNC(C=C(COC)C)=O)CC(C)(C)CN1C(=O)Cc1cncc(C)c1 C=CCCC(F)(F)C(=O)N1CC2(CCCC2NC(=O)C(c2ccc(F)cc2)F)C1 N1(C(C2CC(C)SCC2)=O)CC2CC(C1)C2NC(c1c[nH]nc1C1CCC1)=O S(=O)(=O)(c1ccccc1Cl)NC(C(=O)NC(CCCC)CC)N c1(C(=O)NC2(CNC(c3c(SC)snn3)=O)CC2)nn(C)cc1[N+](=O)[O-] C(=O)(C1CCCc2c[nH]nc21)N(C1CCN(C(=O)CSCCOC)CC1)CCC CC1=C(C(=O)N2CC3CC3C2CNC(C2C3CCCOC23)=O)CCC1 C=CC1(CC(=O)N(CCCC(=O)NC)C)CN(C(C2CC23CCC3)=O)C1 CC1CCC(NC(C2CCC(C(N)=O)C2)=O)CN1C(C12CC(CO1)C2)=O c1(C(=O)NCC2CN(C(C=COCC)=O)C(C)C2)nc(SC)n2ccccc12 c1(OC)ccccc1CC(=O)NC1(CNC(=O)C(C)c2ccsc2)CCC1 O=C1CC(C(=O)NCCC2CC2)N(C(C2CC=CC2)=O)C1 C1(c2onc(C(C)(C)C)n2)CCCN(C(c2cc(N)ccn2)=O)C1 N1(C(C(C)OCC=C)=O)C2CC1CN(Cc1ccc(CC)cc1)C2 C1(C(=O)NC2CCN(C)CC2)CC2CCC(C1)N2C(=O)Nc1ccc(N)c(F)n1 c1(C(=O)NCC(CNC(C2CCC(C)(CC)O2)=O)C)cc2nccnc2cc1F C#CCCCCCC(=O)NC1CCC(C)(CNC(=O)CCc2cc(OC)no2)C1 CC1Cc2cc(Br)ccc2CN1C(=O)NCCNS(=O)(=O)c1ccc(C(F)F)cc1 N1(c2ncc(C)c(O)n2)CCC2(NC(c3ccc(F)cc3Cl)=O)CCCC12 C=C=CCCC(=O)NC1(CCCNC(=O)CCCCSC)CC1 c1(CN2CC3C(NC(c4cc(C)ns4)=O)C3C2)cc(Cl)c(C)cc1O CC(C)(C)[Si](C)(C)OCCSCc1ccc(Cl)o1 C(=O)(C1=C(C#N)CCC1)NCCn1cc(C(N2C3CN(C)C(C3)C2)=O)nc1 C1(CCC)CN(C(=O)C(C)SC(C)C)CCN1C(=O)CCCC1CCC1 Cc1cc(F)ccc1C(N1CC(C)(C)CC1CNC(=O)CCc1ccnn1C)=O C(C)(c1cccs1)=CC(N1CC(OC)(CC(C)(C)C)C1)=O.C1(=O)C(CSCC)N1 C1(CCC(=O)NC2C(CNC(C3CCSC3)=O)CCC2)CCc2ccccc2C1 N1(C(CCCC#CC)=O)CCC2(C1)CN(C(C13CC(C1)C(C)O3)=O)CC(C)O2 Cc1n[nH]c(C)c1CC(N1CCCC(C(C)C(=O)N(C)CCO)C1)=O Cc1cc(=NC(CSC(C)(C)C)C(C)C)[nH]c(N2CCC(N(C)C)C2)n1 Cc1cnnc(O)c1C(=O)NCCC1CC(F)(F)CN1C(c1ccnnc1O)=O CCC(CC(=O)N1CCN(C(c2cc(OC)ncc2Cl)=O)C(C)C1)C(F)F N1(C(C2N(C)CCC2)=O)CCN(CC2CC2c2ccccc2OC(C)(C)C)CC1 c1(C(N2CCC3(C(C(=O)OC)C3)CC2)=O)n[nH]c2c(C)cccc12 CC(C)CCCC(C)C(=O)N1CCC(O)(CN(C(=O)CC(=O)N(C)C)C)C1 Cc1nc(O)nc(C)c1CC(N1CCCN(C(C2OC3CCC2CC3)=O)CC1)=O c1(OC)ccc2onc(CC(=O)NC3C4CC3N(C(=O)CC3CCCOC3)C4)c2c1 Brc1ccc(-n2nnnc2C(c2cn(C3CC3)cn2)NCc2cccs2)cc1 c1(C(N2CCC(CCOC)(NC(=O)C=CCO)C2)=O)cnc2c(C)c(C)ccn12 CC(C)C1=NOC(C)(C(N2CC(N(C(=O)CC3CCCCN3C)C)C2)=O)C1 Cc1cc(C(N2CC(C)CCC2C(=O)NCCC(C)F)=O)ccc1C#N N1(C(c2c(CC)nc(C)[nH]2)=O)CCCC(C)(NC(c2nn(C)cc2Cl)=O)C1 C=CCC(C(=O)NCCC1CCCN1C(=O)C(=O)Nc1ncc[nH]1)OC C=CCCCCCC(=O)NC1CN(C(=O)Cc2cncnc2O)CC1C c1(C(=O)NCC23CC(CNC(C(CC)O)=O)(OC2)C3)cccc(F)c1F N1(C(CC)C)CCN(C(C2(N)CC2)=O)CC1.C1(C)(C(=O)NC)CCC(=O)N1 C1(CNC(C(C2(O)CCC2)NC(c2cn(CCOC)nc2)=O)=O)CN(C)CCO1 c1(C(N2CCC(O)(C(CNC(C3(C)CC3)=O)(C)C)C2)=O)cc2c(Br)cccc2[nH]1 CC(C)(CC(=O)NCC1CCCC(NC(c2cc(=O)cc[nH]2)=O)C1)CC(F)F c1(-n2cc(C3OCCN(C(C4=NOC(C)C4C)=O)C3)nn2)cc(C#N)ccc1I C1(NC(CN2CCC(C(N)=O)CC2)=O)CCCCN(C(c2c(Cl)nsc2Cl)=O)C1 CC1CCN(C(=O)CCS(C)(=O)=O)CCN1C(=O)CSC(=N)N C1(N(C(CSCCOC)=O)C)CCCN(C(=O)Cc2ccnn2C2CCCC2)C1 C1(C(=O)NCCC(C)N(C(c2c(C)nc[nH]2)=O)C)CC=CCC1C CC(C)C(N=c1[nH]c(NCN2CCOC2=O)nc2ccccc12)C(C)N(C)C c1(C(=O)OC)cc(C(=O)NC(CNC(c2cscc2OC)=O)C(C)C)no1 c1(CC)ccc(NC(=O)C(C)=CCNC(=O)Cc2ccc(C)c(C)c2)cc1O C1(C)(CONC(=O)NCC(CC)(CC)c2nc[nH]n2)CCCNC1=O C1(C(=O)NCCCC2N(C(c3c(CC)nns3)=O)CCC2)CCC(O)CC1 Cc1cc(C2CC2)ncc1C(=O)NC1CCN(C(c2ccn(CCF)n2)=O)CC1F c1(C2C(=O)NCC3(CCC3)N2CC)ccc(OC(F)F)cc1.n1(CC)cncn1 C12(NC(C(C)(F)F)=O)CCC(CNC(c3ccc(=N)[nH]c3)=O)(CC1)OC2 N1(C(C2CC(C)=C(C)CC2)=O)CCOC2(CCN(C(C3NC(=O)C4CC34)=O)C2)C1 c1(NC(c2c(-c3cc(OC)c(F)cc3F)c[nH]n2)=O)nc(O)ccc1[N+](=O)[O-] N1(C(C2CC3CCC2O3)C(=O)NCC=C)CCCC(C2CCCCC2)C1 c1(C(=O)NC(C)CNC(=O)C(O)C2CCC2)cccc(-c2ccco2)c1 c1(C(=O)OC)cnccc1C(N1CCCC1(C)CC(=O)Nc1ccccc1C)=O c1(CCC(=O)NCCCNC(C2CC2c2cccc(Br)c2)=O)ccc(O)nc1 Cc1ncnc(C)c1C(=O)NCC1(NC(=O)CCC2CCCOC2)CCCC1 CC(C)(C(F)F)CC(=O)NCC(O)CCNC(=O)C(Cl)=CCl C1(NC(C(C)=CC)=O)CC2(C1)CC(CNC(=O)C(c1cccn1C)=O)C2 C1(C(N(CCCCN(C(C=Cc2c(C)ccs2)=O)C)C)=O)CCn2nccc2C1 C(=O)(C(C)CC(C)C)NCC(C)(CNC(=O)C(C)Cc1c(C)n[nH]c1C)OC c1(NC(C(C)O)C(=O)OC(C)(C)C)ccnc2c1CCO2 C1(NC(c2ccc(N(CC=C)C)cc2)=O)CC2CC1N(C(=O)C(CC)OC)C2 C1(CNC(C2C(NC(CC#N)=O)C2(F)F)=O)(OC(C)(C)C)CCCC1.C(=O)(N)OC N1(C(CC2(COC)CC2)=O)CC2COCCC2(NC(c2csc([N+](=O)[O-])c2)=O)C1 C1(OC)CC(CNC(=O)CCCOc2ccccc2F)N(C(c2ccc[nH]2)=O)C1 NS(=O)(=O)c1n[nH]cc1C(=O)NCCCNC(=O)C(F)(F)C(O)c1ccccc1 N1(C(C2CC(C#N)C2)=O)CCC(N2CCN(C(C3CCC4CC4C3)=O)CC2)CC1 C1(C(=O)Nc2cccc(C(C)C)c2)CNC(=O)CN1C(=O)CCc1csnn1 Cc1c(NCC(C)CO)nc[nH]c1=NCCC1CC=CCC1 c1(OCC)ccnc(CNCC2CCN(Cc3ccccc3)CC2)n1 N1(C(CC(C(F)(F)F)NC(c2c(CC)nn[nH]2)=O)=O)CCC12CCC(C)CC2 N1(C(C(COC)C(C)C)=O)CCc2c(F)cccc21.C1(C)CN(C(C)C)CCC1C N1(C(c2c(CC)nns2)=O)CCN(C(c2ccc(OC(C)C)nc2)=O)C(C)C1 Cc1[nH]nc(C(=O)NC2CCCC2CNC(c2sccc2Br)=O)c1C c1(C(N2C(CC(=O)NC(C(C3CC3)OC)C)CCCC2)=O)cccc2ccnn12 c1(CN2C(C(N(CCC=C)CCOC)=O)CC(F)C2)cc(Cl)ncc1NC N1(C(C(C)(C)C#N)=O)CCC(C2CN(C(=O)CC3OCCOC3(C)C)C2)CC1 Cc1nc(C(C)C)nc(O)c1C(N1CCN(C(C2C3CCCC23)=O)CC1)=O c1(C(c2cc(OCC)c(C)cc2)NC(C2CC(N)C2)=O)cc(Cl)cc(Cl)c1O C1(NC(c2c(C)coc2)=O)CCCCC1N1CCCC1.C12CC(C1)C(=O)N2 C=CCCCCCCC(=O)NC(CC)(CC)CCNC(=O)CC(C)(O)CC c1(C(N(CCCN(C(C2C(CCOC)C2)=O)C)C)=O)ccn(-c2cccnc2)n1 C1(NC(C(CCNC(C2C(C)CC2)=O)(C)C)=O)CCC(C2CC2)CC1 c1(OC)cc(F)c(CC(N2CC3CC(NC(=O)CC4CC4)C2C3)=O)cc1F CC1OC(C)C(C(N2CCC(O)(CNC(=O)C3=CCCS3)C2)=O)C1C c1(C(C)C(=O)NC2(C)CCN(C(=O)Cc3ccoc3)C2)ccc(C#N)cc1 C(=O)(CCC(=O)c1ccc(Br)cc1)NC1CC(NC(C(COC)C)=O)C1 C(CC(C(=O)NCCCSC)NC(C12CC1CN(C(=O)CC(F)(F)F)C2)=O)SC C(C1CCCC1)=CC(=O)NC1CC(CNC(CN(c2ccccc2)C(C)=O)=O)C1 C1(NC(c2cccc(CN(C)C)c2)=O)CCN(C(=O)COC2CCCC2)C12CC2 C1(=O)CC(C(F)F)CC(CC)O1.C(C(N)=O)(C1CC1)NC(=O)OC Cc1ncncc1C(=O)NC(C)C=CC(=O)NCc1ncoc1C N1(c2nnc(CC)c(CC)n2)CC2CC(NC(=O)CC3CC4CCC3CC4)C2C1 C1(F)CC(CNC(=O)C(C2CCCC2)NC(C2CC2CC)=O)C1.C(=O)(N)OC Cc1ccnc2c(C(N3CC(C)CCC3CNC(=O)C(C)(C)C3CC3)=O)cnn12 Cc1cc(F)cc(C(=O)NC2CCC2NC(c2c[nH]nc2[N+](=O)[O-])=O)c1N Cc1cc(CNc2cc(NCCSc3cnn(C)c3)ncn2)c(C)n1NC(N)=O CC(CN=C(NCC1CCOCC12CCC2)NCC(F)F)OC1CCCCC1 c1(C(=O)NCC2N(C(C3C(OC)CCC3)=O)CC2)ccc2ncn(C)c(=O)c2c1 c1(C(=O)NCC(CC)NC(c2scc(C)c2Cl)=O)cc([N+](=O)[O-])nn1C c1(NC(C2C(CC)CN(C(=O)CC(C)OC)C2)=O)cc(CO)cc(F)c1 c1(CC(=O)NC2CCCC2CC2CCCO2)cc(OC(F)F)ccc1O C1(C)(NC(C=CCC(C)(C)NC(C=C(COC)C)=O)=O)CCC(C)=C(C)C1 C(C(CCC)C(=O)NCC(C)(C)F)NC(COC1(C#C)COC1)=O C1(NCCc2cn(C(C)C(=O)O)nn2)CCCC1CNC(=O)OC(C)(C)C c1(C(N2CC(NC(CC3(COC)CC3)=O)C3C2C3)=O)cc(Cl)cc2c1OCC2 C1(CC(=O)NCC(CN(C(=O)COCCF)CC)(C)C)CCCCC1F C(=O)(C1CCCc2nn(C)cc21)NC(C)CNC(=O)C(c1cnn(C)c1)O N1(C(Cc2ccc(C(=O)NC)cc2)=O)CCC(C)C(NC(=O)CCCF)C1 CCCCC(=O)C(=O)NCC(C(=O)N1CC(NC(C)=O)C1)N(C)C CC1(OC(C)(C)C)CCN(C(N2CCOC(c3nc(C)no3)C2)=O)C1.C1CO1 CCCC(C(=O)N1CCC(C)(CNC(c2ccc(C(F)F)nc2)=O)C1)NC(N)=O C=C(C)CCC(=O)NCC1(C)CCN(C(=O)C(N2CCNC2=O)C)C1 C(CN=c1c(C(F)(F)F)c[nH]cc1Br)NCC(C)(O)C1CCOC1 N1(C(c2[nH]cc(C)c2)=O)CCN(C(=O)C(F)OC(F)(F)F)C2CCCC2(C)C1 c1(N(C)Cc2cc(C)no2)[nH]c(=NC2CCC(Cl)(Cl)C2)nc2c1ncn2C c1(CN2C(CNC(=O)NCCO)CCC2)c(C(F)(F)F)cccc1O N1(CC)CCCC(C2CCNCC2C)C1.c1(C2CN2)cnn(C)c1 N1(C(C(CC)NC(N)=O)=O)CCC2(CC(C(=O)NC34CC(C3)C4)C2)C1 c1(CNC2CC(NC(=O)C=CC3CCOC3)C2)ccc(C(C)(F)F)cn1 C(=O)(CCCC(F)(F)F)NCC(C)(C)C.CC1CC(=O)N2CC(C2)C(=O)N1 c1(C(=O)NCCC2CC(NC(c3cc(OC)n[nH]3)=O)C2)nn(C)cc1Cl CC1=NN(C)C(=O)C1CC(N1CC=CC1CNC(C1(CC2CC2)CC1)=O)=O C=CC(C(=O)N1CSCC1C(=O)N(CC(C)C)CC(C)C)OC C(CCCCCNC(C1CCCC(=O)O1)=O)N(C(CC1N(C(C)C)CCC1)=O)C C1(CNC(c2c(C)ncn2C)=O)CN(C(=O)CCC2CCCO2)CCC1C(F)(F)F CC1CN(C(c2ccccc2C(F)(F)F)=O)CCN1C(=O)CC1CCC(C)C1 C1(NC(C(CN(C)C)NC(C=C(C)C(F)F)=O)=O)CCC(C(=O)OC(C)(C)C)CC1 N1(Cc2cccc(C)n2)CC=C(CCNC(c2cc3occc3s2)=O)CC1 N1(C(C(C)SCCCC)=O)CCC(CNC(c2ccsc2COC)=O)C12CC2 c1(CCC)ncc(OC)cc1OCC1CC2CCC1N2 C1(NC(C(C)(C)SCCC)=O)CCCCC1CNC(c1ccc(C)nc1)=O Cc1ccc(Cl)cc1C(=O)NCC(C(C)(C)C)NC(c1cc(O)ncn1)=O Cc1cccc2cc(C(N3CCOC(CN(C)C(c4nncs4)=O)C3)=O)nn12 Cc1cnc(C)c(C(=O)NC(C)CC2CN(C(=O)C=Cc3cn(C)cn3)C2)c1 C1(NC(c2c(CC)n[nH]c2)=O)CC2CCC(C1C)N2C(=O)CC(C)(O)C1CC1 C1(NC(c2c(OC)cc(N)cc2)=O)CCN(C(C2CCSCC2)=O)CCC1CO C#CC1(NC(=O)C(CC)N(C(=O)C(C)CC(C)(C)C)C)CC2CCCC12 C12(CNC(C3OCCN(CC)C3)=O)CCC(CN(C(=O)C(C3CC3)OC)C1)C2 C123COCC1CN(C2)C3.N1(C(C(CCC)OCC)=O)CCCN(C(=O)OC)CC1 C1(C(=O)NC2CCC(C(N3C(C4(N(C)C)CC4)CCC3)=O)C2)CCC(C)(O)CC1 CC1(C)CC(=O)c2[nH]c(C(=O)NCC34CC3CN(C(=O)C3CC3)C4)cc2C1 c1(OC(C(=O)N(CCNC(c2nccs2)=O)CC)COC)ccc(Cl)cc1C C1(CCNC(c2c(COC)occ2)=O)NC(=O)NC1=O.C12(CCOC1)C(=O)N2 N1(C(c2ccn(C)c2)=O)CCN(C(=O)CCS(N)(=O)=O)C(c2ccccc2)C1 C1(NC(CCCCC(=O)NCC)=O)CCS(=O)(=O)C12CN(C(=O)C1=CCSC1)C2 c1(CC(=O)NCCCN(C)C(c2coc3c2COC3)=O)ccc([N+](=O)[O-])cc1 C=CCCCCN(C(=O)CCC1(C)CN(C(=O)COCC2CCCC2)C1)C c1(C(N2CC=CC(NC(C(CO)NC(C(C)C)=O)=O)C2)=O)cc2occc2s1 c1(C(=O)Nc2cn(C(CC)C)nc2)cccc(C)c1.c1(=O)c(=O)n1CCCO c1(OC)nc(C)c(C(c2nnnn2CC(F)F)NCC2CCCSC2)c(C)c1Cl Nc1sc2c(c1C(N1CC3(CCC(CNC(=O)C4=CCCC4)O3)C1)=O)CCC2 N1(C(C(F)=C(C)C)=O)CCC2(CC1)CC2NC(c1cnn(C(C)C)c1Cl)=O C#CCC(CC(F)F)C(=O)NC1CC(C(F)F)(NC(C2CC2NC(C)(C)C)=O)C1 Cc1cc(F)c(NC(=O)C(F)C2CC(NC(c3nccnc3C)=O)C2)cc1C Cc1ccc2c(c1)CC(C(=O)NCC1CCC1NC(c1cc(Cl)cnc1O)=O)S2 C(=O)(CC(C)(C)NC(=O)CCc1cncs1)N(CC(C)O)C1CC1 N1(C(C2C(OCC)C2)=O)CC(OCC)C(Nc2nc(C)n(-c3ccccc3)n2)C1 C(=O)(C(CC)C(C)(C)CC)N1CCN(CCCCCNC(C(C=C)(C)O)=O)CC1 C1(C(=O)NCC2CCCC(C)C2)CCN(C(c2ncc(F)cc2F)=O)C1(C)C C12(CCN(C(=O)CSC)CC1)C(=O)N(C)CCCC(=O)NC2.C1(OC)CC1.CCO C(N=c1[nH]c(=NC2CC(F)C2)[nH]c2ccsc12)C1C(CC)C1 N(C1=NCC2CCCN12)C(C(=O)N(C(C)(C)C)C)CCN=[N+]=[N-] n1(CC)nc(C(=O)NC2COCC2CNC(C2(C(N)=O)CC2)=O)c(C)n1 N1(C(C2CC(C)(O)C2)=O)CC2CCC1CN2C(=O)C1=NOC(C2CCCC2)C1 C(C)(CCCC(=O)N1CCC(CN=[N+]=[N-])C1)NC(C(CC=C)C)=O C(=O)(C1=CCCCCC1)NCCC1(C)CCN(C(C2CC(C(=O)OC)C2)=O)C1 c1(C(C(=O)NCC2(F)CN(C(=O)C(F)C3CC3)C2)O)ccccc1Br C1(CC)CN(C(=O)CCCNC(=O)OC)CCN1C(=O)CC(C)c1ccccc1 Cc1ccc2c(c1)CN(C(C1(NC(=O)CNC(=O)C(C)(C)C)CC1(C)C)=O)C2 C1(C(=O)NCCC(C)N(C)C(c2c[nH]c(=S)cn2)=O)CCOC(C)(C)C1 C=CC1(O)CCN(C(=O)C)C1.C1(C)CN(C(=O)C=C(C)C)C1 C1(NC(C(C)n2cnnn2)=O)CN(C(c2ccc3c(c2)CCC3)=O)CC2(CC2)C1 C(N=c1ccnc(N2CCOC(CCOC)C2)[nH]1)C1CCCN(CC)C1 N1(C(CC(C=C)C)=O)CCOCC(C)(CNC(c2c(Cl)c(C)nn2C)=O)C1 c1(CCNC(C(c2ccco2)NC(CC(C)n2cccn2)=O)=O)ccncc1F N1(CCC(=O)NC(C2CCN(C(=O)Cc3n[nH]c(=N)s3)C2)C)CCOCC1 c1(C(=O)NC(C2CCN(C(=O)CC3(C(F)(F)F)CCC3)C2)C)cccn1C c1(OC)cc(C(=O)NC2CC3CN(C(=O)C(C)O)CC23)c2c(c1)CCO2 O=C(C1CCOc2ccccc21)NCC1(CNC(C23CCCN(CC2)C3)=O)CC1 C1(C(c2cccc(C)c2)=O)CCC2(CC1)NC(=O)N(C)C2=O.c12cn(nn1)C2 C(=O)(C1CCc2ccccc21)N(C1CCN(C(=O)C(C)(C2CC2)OC)CC1)CC c1(CNC(=O)CCC(CNC(=O)CSC2CCCC2(C)C)OC)ccccc1Cl Nc1c(C(=O)NCCCN(C(=O)Cc2cncnc2)CCO)cccc1F c1(OC)ccc(Cl)c(C(N2CCC(O)(C(N3CCCC(F)(F)C3)=O)C2)=O)c1Cl c1(OCC(=O)NCCCC(C)NC(CSCCC)=O)ccc(Cl)c(C)c1 CC1NC(=O)CCC1N=c1[nH]c(=NCCCCN2CCOC2=O)[nH]c2c1CSC2 C1(NC(C2(Cl)CC2(F)F)=O)CCCN(C(=O)Cc2cccnc2O)C1 Cc1ccc(F)cc1C1(C(N2CC(CN(C(=O)CCF)C)C3(CC3)C2)=O)CC1 N1(C(c2c(C)coc2)=O)CCC(C)C(CC(=O)NC(Cc2ccco2)CO)C1 CC1CCN(C(C23CC(CC4CC4)(C2)C3)=O)C1C(=O)Nc1ccc(Cl)cc1 N#Cc1cc(S(=O)(=O)N2CCC(C3CN(Cc4cnc(Cl)s4)C3)CC2)ccc1F C1(C(=O)NCc2c(C)occ2)CC(=O)CN1C(C1CC(=O)C1(C)C)=O CC1(C(F)(F)F)c2cc(Br)ccc2CCN1C(=O)C1=NOC2CCCC12 c1(C(=O)NCC2CC(C)N(C(c3ccncc3)=O)C2)ccc(N=S(C)(C)=O)s1 c1(C(=O)OC)nc(N(C)CCOCCNC(=O)Cc2ccc(C)s2)c(F)c(Cl)n1 C1(C(=O)NCC(C)(C)OCC)CC12CCN(C(=O)C(C1CCCCC1)=O)C2 C(=O)(CCCCCCc1ccccc1)N(CCN(C(=O)CCCCSC)C)CC CC(C(=O)NCCCC1CN(C(c2cc(C(F)(F)F)c[nH]2)=O)CCO1)S(C)(=O)=O C(c1ccc(F)cc1)=CC(=O)NCC(C(C)(C)C)NC(c1ccc(N)cc1F)=O C12(CC(=O)NCc3cn(C(C)C)nn3)CCC1CN(C(c1ccnc(O)c1)=O)C2 N1(CC2CCCO2)CCC12CCCSC2.O=C1C(F)=C2CN1C2 N1(C(CC(C)CN(C)C)=O)CC2(C)CC1(C(=O)NC1C=CCCCC1)C2 N1(C(C#CC(C)C)=O)C2CCC1CC(NC(C1CCCCC1n1cccn1)=O)C2 N1(C(CC(=O)NCCNC(C2CCN(C)C2C2CC2)=O)=O)CC(O)C(C2CC2)C1 Cc1cn2c(n1)C(C(=O)NC1CCCC(NC(=O)CCc3cnoc3)C1)CCC2 C(C(C)C)(C(O)C(=O)N1CCC(NC(C2C=CCCC2)=O)C1C)OC c1(COC)cc(F)ccc1S(=O)(=O)Nc1ccc(C(=O)NCC2CCCO2)cc1 CCC(C)C(O)C(=O)N1CC2(NC(=O)C(N3CCC(C)CC3)=O)CC1C2 c1(CC(=O)NC(C(C)C)C(C)NC(=O)Cc2cncnc2)nc2c([nH]1)CCCC2 c1(OC)ccnc(C(=O)NC2(C)CC(NC(C3CC3(Cl)Cl)=O)C2)c1OC c1(CCCNC(c2nnco2)CO)ccco1 N1(C(COCCOCC)=O)CCC2(NC(c3ccncc3Cl)=O)CC2C1 CC1(NC(=O)CCc2cc[nH]n2)CCN(C(=O)CCC2CC2(Cl)Cl)C1 Cc1ccc(O)c(CN(C(=O)C2CC2)CC2CC(C)OC2C)c1 OC12CC1C2.c1(CN)cnc(-c2ccccc2)o1 C=CCCC(C(=O)N1CCCC(C)C1)NC(c1cc(C)cc(F)c1)=O C=CC1(C(N2CC(NC(c3ccoc3C3CC3)=O)C2)=O)CCCCC1 C1(C(=O)NCCOCCN(C(CCCCC(N)=O)=O)C)Cc2n[nH]cc2C(=O)N1 C1(NC(C2(COC)CN(C(c3cnccc3C(=O)O)=O)C2)=O)CCC(C)OC1 N1(C(C=CC=CC)=O)CCc2sc(CNC(C3(F)CC3(Cl)Cl)=O)nc2C1 c1(C(=O)NC2CCCCCC2NC(C2CCCSC2)=O)ccc2nonc2c1 CC1(C)C(Oc2ccccc2)CC1C(=O)NCCCCO.c1(C)cn(CCO)nn1 N1(CC(N2CCCC2CNC(C2(C3CCCO3)CCC2)=O)=O)CCCCCC1 C(=O)(CCCCCC#N)N1CC(C(N2CCC(SC)C2)=O)C(F)C1 C1(N(C(C2C(C(C)C)CCO2)=O)C)CN(C(c2coc(Cl)c2)=O)CCC1C C(N=c1cc(C)nc(C)[nH]1)C1N(C(CCc2nc(C)c(C)o2)=O)CCCC1 C1(O)(C(=O)NCC2CC(NC(c3ccc(C)nn3)=O)C2)CCCC(C)CC1 C1(CNC(c2cc(=O)cc[nH]2)=O)CN(C(=O)CCc2nc(O)n[nH]2)C2CC12 C1(CNC(c2ccn(CCNC(c3c(CC)[nH]cc3)=O)c2)=O)CC2CCC2C1 N1(C(C(C)N(C)C)=O)CC2CN(C(c3cccc4c3OCC4)=O)CC2(C)C1 c1(C(=O)NCC(C(C)C)NC(C(C2CCCC2)OC)=O)sc(C)cc1C N1(C(C(C)C2CCC2)=O)CCC2(CC1)CN(C(=O)Cn1nccn1)C1COCC21 C1(F)(C(=O)NC(C)CCCCNC(C2CCC2(C)C)=O)CCCCCC1 N1(C(C2CSC2)=O)CCC(CCCCCC(=O)NCC2(c3ncco3)CC2)CC1 c1(CN2C(CNC(=O)Nc3ccco3)CCC2)cc(F)cc(Br)c1 c1(C(N2CC(C)C(NC(=O)CCCC#N)C(C)C2)=O)ccc2nc(O)oc2c1 c1(C(N2CC3C(NC(CCCC(=C)C)=O)C3C2)=O)cc2c(=O)[nH]ccn2n1 Cc1csc(C(=O)N(CCC(C)NC(C2(C)CSC2)=O)C)c1C N1(C(c2cccc(CC)c2)=O)CCC2CN(C(C3(CC#N)CCCCC3)=O)C2C1 N1(C(C2(CC)CC2)=O)C2CCC1CC(C(=O)NCCCC(CO)=C(C)C)C2 Cc1c(C(=O)NC2(CO)CCCN(C(=O)C=CC(=O)N(C)C)C2)cccc1F C1(CNC(C2C(CC(C)C)C2)=O)(CN(C)C)CCN(C(C2(CO)CC=CC2)=O)CC1 c1(C(=O)NCCn2nnc(C)n2)ccc(CNC(c2sc(=N)[nH]c2C)=O)nc1 C1(NCC(=O)C2CCCc3sccc32)C(F)(F)C12CCOCC2 C1(C2CCN(C(c3cc4c[nH]cnc-4n3)=O)C2)(NC(c2cnco2)=O)CC1 c1(C(N2CCN(C(C3C4CCCCC34)=O)CC2CCO)=O)nccn2ccnc12 N1(C(c2n[nH]c(O)n2)=O)CCC2CN(C(C3(C(F)F)CCCO3)=O)CCC12 c1(C(=O)OC)cc(=NCC23CCCN2CCC3)[nH]c(Cl)n1 N1(CC(c2cccnc2)N(C)C)CC(c2cnn[nH]2)Oc2ccccc21 C12(C(N(CCN(C(c3cc(CCC)nn3C)=O)C)C)=O)CCOC1CCOC2 C(=O)(CC(C)NC(=O)CC=CCNC(=O)CC1CCC(=O)C1)OC C(=O)(C#CC1(C)CC1)NCC1N(C(CCC)=O)CC1 O=S(=O)(NCc1cc(I)ccn1)N1CCCC2(CCCNC2=O)C1 c1(C(=O)NC(C2CN(C(=O)C3=NOCC3)CCO2)C)cnc(S(C)(=O)=O)[nH]1 c1(CN(C)CC2CC3CC3C2)cc(C2CNC2)[nH]n1 N1(C(C(CC)CC)=O)CC2CCC2(CNC(=O)C=CS(C)=O)C1 CCCCC(O)CCC(=O)N1CCCOC(CNC(C2(C)CCN(C)C2=O)=O)C1 C1(CN)CCC(C(=O)NCC2CCN(CC3CCCC(F)C3)CC2)CC1 C(=O)(C(C)(C)CCCO)NC1CCC(NC(c2c(=O)ccn(C)c2)=O)CC1 N1(C(C2C(C)(C)OCC2)=O)CCC2(CCC2)C(NC(c2cnc(C(F)F)s2)=O)C1 CC1CCC(NC(c2cc(=O)n(C)cc2Br)=O)CN1C(c1cnc[nH]c1=N)=O Cc1oc(CNC(C2CCCC(=O)N2)=O)nc1C(=O)NC1(C(N)=O)CCSC1 CCCC(C)C(C)(c1nnnn1SCC)N.C(=O)(CC(C)(C)C)N1CC1.c1(C=O)nnnn1-c1ccccc1 C1(NC(c2nc(C(=O)OC)sc2)=O)CCCN(C(=O)C(C)C#N)CC1F C1(C(C)C(=O)N2CC(C(F)(F)F)C2)CCN(C(c2cncnn2)=O)CC1 N1(C(c2c(SC)scc2)=O)CCC2(CC1)C(NC(C13CCCC(C)(C1)OC3)=O)C2 N1(C(C(C)(CO)OC)=O)CCCC(C)(NC(C2CN3CCCC2C3)=O)C1 N1(C(CN2CC(C)C2)=O)CC(O)(CNC(=O)CC2(C)OCCO2)C1 c1(C(C(=O)N(C)CC2N(C(CC)=O)CC(F)C2)(C)C)c(C)[nH]c2ccccc12 CCC(C(=O)N(CCC(=O)NCC(C)(C)NC1CC1)CC)OC Cc1ccccc1CC(=O)NC1CN(C(c2sccc2CO)=O)CC1C(F)F c1(OC)ccc(CC(C)C(N2CCNC(CNC(=O)C(C)(C)O)C2)=O)cc1OC C1(CN(C(c2cc(C)c(C)[nH]2)=O)C)CN(C(C2(n3cccn3)CC2)=O)CC12CC2 c1(C(N2CC3CN(C(CCC(=O)NCC)=O)CC32)=O)c(OC)ccc(OC)c1OC c1(NC(C2CCc3n(cc(CC)n3)C2)=O)cccc(C#N)c1[N+](=O)[O-] c1(NCC2OCC(C)C2)[nH]c(=NCC2(C(F)(F)F)CC2)nc2c1ncn2C c1(N)c(F)cc(Br)cc1[N+](=O)[O-].c1(C(=O)OC)sccc1NC(C1CC(=O)N1)=O c1(NC(C(=O)NCCC(C)NC(C2C(C)(COC)C2)=O)=O)cccc([N+](=O)[O-])c1 c1(C(=O)NC2CCN(C(C3(C)CC=CCC3)=O)C2C2CC2)c(F)cccc1F N1(C(C2C(=C)CC2)=O)CC2=C(C1)CN(C(=O)CCn1nc(C)c(Br)c1C)C2 C1(CNC(Cc2c(C)nsc2)=O)(NC(=O)C(O)CC2CCCCC2)CCOCC1 c1(C(=O)NC2CC(CNC(C3(OC)CCSC3)=O)C2)cnc2c(c1)COCC2 c1(CC)cnc(Cl)[nH]c1=NC1CCN(C(c2nnn(C)c2C(F)F)=O)CC1C C1(NC(CCCCC#C)=O)CC2(CCC(CNC(c3cc(C)c(C)s3)=O)CC2)C1 N1(C(C2CC(C(C)C)C2)=O)CCCC(N(C(=O)C(C)C2CCCC2)C)C1 c1(C(C2CC2)NC(C)CCNC(=O)CC(C)C2CC2)c(Br)cnn1C1CCC1 N1(C(C(C)NC(N)=O)=O)CCCC2(C1)CC2(F)F Cc1ccc(C(=O)NC2CCN(C(c3cc(C(N)=O)cn3C)=O)CC2)cn1 c1(C(=O)OCC)cnc(NCc2nnc(CO)s2)s1 c1(C(=O)Nc2c(NC(=O)NC)c(C)ccc2)cc(C(=O)OC)c(Cl)cc1Cl N1(C(C(=O)NC(C)C)=O)CCCC(C2CN(C(c3cn(C)nc3Br)=O)C2)C1 CN1CCC2C(CCN2C(C2(C)CN(C(C3CCC4(CC4)C3)=O)C2)=O)C1 C12(NC(CC=CC)=O)CCOCC1CN(C(c1cccc(C#N)c1)=O)C2 CCCCC(CNC(c1cnccc1N(C)C)=O)NC(=O)CC(=O)NC1CC1 C1(C)(CC)CC(NC(c2ccc(C(C)(C)C)s2)=O)CN1C(=O)CC=C(C)C C(=O)(CCCC(=O)N1CCCC(N(C(=O)CC2CCCCC2O)C)CC1)N(C)C C1(CN(C)C(C2CCC(=O)N2)=O)CCCCN1C(c1ccc(=O)oc1)=O C(CC1=CCCCC1)N(C(CO)CO)C(C1CCCN1C1CC1)=O C1(CC(N2CCCC2CF)=O)(OC)CN(C(c2[nH]ccc2C2CC2)=O)C1 c1(C(N(C(CNC(C(F)=CC)=O)C2CC2)C)=O)nn(CCC)cc1Cl N1(C(Cc2cc(C)sc2)=O)CCC2(CC1)CC(NC(=O)CCC1CCCO1)CO2 c1(NCC(COCC)O)cc(C)c(S(=O)(=O)N2CCCC(C)(C)C2)cn1 c1(-c2ccc(C(C)NCC(C)(C)CC(F)(F)F)cc2)ccc2c(c1)C(=O)N(C)C2 c1(C(=O)NCC(C)NC(c2cc(C(F)(F)F)c[nH]2)=O)cccc2cccc(O)c12 C1(NC(c2cnc(OCC)s2)=O)(CF)CCN(C(=O)CC(C)n2cccc2)C1 C1(OC)CC2(C1)CC(C(=O)NCC(Cc1ccccc1)NC(=O)CC(C)C)C2 C1(NC(CCN(CC)CC)=O)CCC2CC1CN2C(=O)CCC(C)(C)OC CC1CN(C(=O)Cn2nnc(=N)[nH]2)CC1CNC(c1cn(C2CCCC2)nn1)=O C1(C(N2CCC(SC)CC2)=O)CN(C(=O)C=CC(F)F)C2(CCC2)C1 Cc1cc(CNC(C2CCN(C(=O)CCc3nc(C)no3)C2(C)C)=O)cc(F)c1 c1(C(=O)NCC2CCC(C)N(C(=O)COc3ccsn3)C2)cccc2[nH]ncc12 N1(OC(C(C)CCN(C)C)=O)CCOCC1(C)c1cn(-c2cccc(Cl)c2)nn1.CC C1(C(N(C)Cc2cncs2)=O)C2CCCC2CN1C(C1CCC(=O)N1C)=O O(N(CC)C(=O)C1CN(C(c2coc(N(C)C)n2)=O)C(C)C1)CC C1(CC(=O)N(CC(C)O)CCNC(=O)C(C)(C)C2CCC2)CCCC(=O)N1 C1(CCNC(CC(=O)NC)=O)CCCN(CC(=O)NCC2CCCO2)CC1 N(C)(C(=NCCF)NCC1C2CCC(F)(F)C12)CCOCCOC Cc1cccc2c1C(=O)NC(C)(C)N2C(c1cnc(C(F)F)o1)=O CCCC(C)(O)C(=O)NC1(CC=CC(N2CCC(n3cnnn3)C2)=O)CCC1 O=C1CC2(CCC2)C(C(N2CCN(C3CCN(C(=O)CSC(F)F)C3)CC2)=O)CN1 c1(C(=O)NC2CC(OCCC(=O)NC3CC3)C2)cc2ncccn2n1 C(=O)(C1=CC2C=CC(C1)C2)NCC(CC=C)NC(=O)CCc1cnn(C)c1C Cc1ccnc(C)c1C(=O)NCCN(C(c1cnn(C)c1)=O)Cc1ccccc1 C1(F)(CNC(CCn2ncc(C)c2)=O)CCN(C(=O)C(F)C(C)C)CC1 c1(C(N2C(C)CCN(C(C3CC(OC)C3)=O)CC2)=O)cc(O)nc2cnccc12 c1(C(=O)NC2CS(=O)(=O)CC2NC(c2ncccn2)=O)cnc2n1CCOC2 Cc1c(C(N2CCN(C(C3CNC(=O)C3)=O)CC2)=O)sc2[nH]cnc(=O)c12 C1(CC(=O)OCC)CN(C(=O)C(C)(N)C2CCOC2)CCO1 N1(C(C2(c3cn(C)nc3)CC2)=O)CCN(C(=O)CC2CCCC23CC3)CC(O)C1 c1(CNC(=O)NCC2CCOC2)ccc(CO)c(Cl)c1 N1(C(C2(CC#C)CCOC2)=O)CC(NC(c2cccc[n+]2[O-])=O)CC2(CCC2)C1 C(=O)(CCC(C)CNC)NCC1CCN(C(C(C)OCC=C)=O)CC1 C12CCCCN1C(=O)C1(CC1)NC2=O.C=CC(O)C(=O)OCc1ccccc1 n1(CCC(=O)OCC)nnnc1C(c1cc(OCC)cs1)NCC(C)F c1(CC)cc(C(N2CCC(N(C)C(c3ncccc3F)=O)C(C)C2)=O)cc(Cl)c1 N1(C(CSc2ccc(C)cc2C)=O)CC2CCCC1CN(C(c1ccsc1)=O)C2 C1(CNC(C(c2ccc(F)cc2F)C)=O)CC2CN(C(C3CCCS3)=O)CC12 C1(C(=O)NCC(CNC(C(C)SCCCC)=O)(C)O)CCC2(CCOCC2)O1 c1(C(=O)NCC2CCC(NC(c3cccc(CC#N)c3)=O)C2)cc2n(n1)CCC2 N1(C(Cc2c(C)n[nH]c2)=O)CC2CC1C2NC(C1(C(F)(F)F)CCCC1)=O c1(SCCN(C)C)cccc(CC(=O)NCc2ccccc2Cl)c1 C1(CNC(c2c(OC)ccc(Cl)c2)CC(=O)O)CNCC1C1CCOC1 N1(C(C(c2ccccc2F)(C)F)=O)CCC(CO)(NC(c2cnc(Cl)[nH]2)=O)C1 c1(C(=O)NC2(CC=C)CN(C(c3nsnc3O)=O)C2)coc2c1COC2 CC(C)(C)CC(O)C(=O)N1CC=CC1C(=O)NCCCCCCCO C1(OC)CC2C1CCN2C(c1ccn(CC2CCOCC2)n1)C(=O)NC1COC1 C1(C(N2C(C(=O)Nc3cn(CCCC#C)nc3)CC2)=O)CCCC2(C1)CC2(F)F c1(C(N2CC(N(C(CCC#C)=O)C)C2)=O)c[nH]c2ccc(C#N)cc12 c1(C(=O)NCCN(CC(C)O)C(=O)C=CC(=O)N(C)C)ccn2c1CCC2 c1(C(N2CCC(C(=O)Nc3c(C#N)cc(Br)cc3)C2)=O)ccc(O)c([N+](=O)[O-])c1 N#CC1(C(=O)NCCCOCCCNC(=O)C2=CCOC2)CC2CCC1C2 n1(CCC#C)c(N2CCC(C(C)(C)C)CC2)nnc1-c1ccc(C)o1 O=C(C(F)(F)CCn1cc(CCOC(=N)O)nn1)Nc1cccc(-c2nnco2)c1 C1(CCC)CN(C(C2CCC(=O)NC2)=O)CCN1C(=O)C=Cc1ccc(F)s1 C1(NC(CC2(CCNC(=O)Cn3nccn3)CC2)=O)(CSC)CC2CCCC12 CC(CC(C)NC(=O)C(F)(F)c1cscn1)NC(C1CCCCS1)=O c1(C(N2C(CNC(c3cc(OC)no3)=O)C(C)CC2)=O)cnc2[nH]c(C)nc2c1 c1(C(=O)OC)cc2c(s1)CCC2NC(=O)CCc1nc(-c2ccsc2)no1 c1(C(=O)NCCN(C(C(CC=CCC)C)=O)CCOC)ccc(CO)c(Cl)c1 n1(CC=C)nnnc1C(c1ncoc1COC)NC(C1(OC)CCC1)C c1(OC)cc(CO)cc(CN2CCC(O)C2C(N2C(C)CCC2C)=O)c1O C(=O)(C(C)CCCC(C)C)N1CC(CC(=O)NC(CC)C(=O)NC)OCC1 CC(C)(C)C(CNC(=O)CN(C1CCSC1)C)NC(=O)CN1C(=O)CCC1=O C1(NC(C2(c3ccn(C)n3)CC2)=O)CC(O)CN(C(=O)NC23CC(CCO2)C3)C1 N1(C(c2n(C(C)C)ncc2)=O)CC2CCCC1C2NC(C1CCCCO1)=O C(=O)(C1SCCc2sccc21)NC(CNC(c1cc(C)n(C)c1)=O)(C)C(C)C N1(C(CC2CN(C(c3n(CC)ccc3)=O)C(C)(C)C2)=O)CC2CCC(C1)C2O C1(C(C)(C)NC(CNC(CC)=O)=O)CCN(C(=O)C(F)=C2CCCC2)C1 C(CC(O)C(=O)NCC1CCN(C(C2CCCC2c2nc(S)n[nH]2)=O)CC1)SC N1(C(C2CCC(CNC(=O)COCC3CCCC3)CC2)=O)CC2CCOC2C1 Cc1ccc2c(c1)C(C(=O)N(C)CC1(NC(c3ccc(C#N)s3)=O)CC1)CC2 C12(C(N3CC(CNC(c4c(CC)oc(C)c4)=O)OCC3)=O)CCCN(CCC1)C2 N1(C(c2c(CC)cno2)=O)CC(NC(=O)CCCOc2cccc(C)c2)CC1C n1(CCC(=O)N(C)Cc2cn(Cc3ccoc3C(=O)O)nn2)ncn(C)c1=O C(C(C)(C)CC(=O)N(C1CCCN(C(=O)C(C)CC(N)=O)C1)C)OC N1(C(c2cccc(OC(C3CNC3)C)c2)=O)CCC2(CC(NC(C(C)C)=O)C2)C1 C1(C(=O)OCC)CCC(CCC(=O)NCCn2cc(CC(C)(C)CO)nn2)CC1 Cn1nccc1C=CC(=O)NC(C1CCOC1)CNC(=O)C(C)(C)n1cc(Cl)cn1 CCC(C)(C)CCCC(=O)N1CC(C(=O)NC(CO)CC(C)(C)C)C(C)C1 C1(C2CCC2)(C(=O)NC(C2CN(C(C3(CC(C)C)CCCC3)=O)C2)C)CC1 N1(C(Cc2c(C)nsc2)=O)CCC2(NC(=O)Cn3ccc(O)nc3=O)CCCC12 CC(C)CC(O)C(C)C(=O)NC1CCCCCC1NC(c1n[nH]c2c1CCC2)=O C1(C(N2CCC(N(C(=O)CCN3CCCC3=O)C)C2)=O)CC2CCC(C1)S2 C1(C(=O)NCCNC(=O)CC2(n3cccn3)CC2)CCS(=O)CC1 c1(CC)ncc(C(=O)NC2CCCN(C(c3ccnc(Cl)c3N)=O)C2)c(C)n1 C1(CC)CN(C(=O)COC(F)(F)F)CCN1C(C1CCN(C)C(=O)C1)=O N=c1[nH]c(CC(=O)NCC2(CNC(C3CC3CF)=O)CC2(F)F)cs1 C1(NC(CCCC(C)O)=O)CCN(C(=O)C(=Cc2c[nH]cn2)F)CCC1(F)F c1(C(=O)NC2CC2CNC(=O)CCc2cnc(O)[nH]2)nc(C(=O)OCC)cs1 c1(C(=O)NC2(CN(C(CN3C(=O)CN(C)C3=O)=O)C)CC2)nccc2cc[nH]c12 C1(CC)(NC(c2cc(F)cs2)=O)CCN(C(C2CCCNC2=O)=O)CC1 c1(C2(C(N3C(C(c4ccc(Br)o4)=O)CCC3)=O)CC2)ccnc2ccccc12 C1(O)(CCNC(C2CCCC2O)=O)CN(C(c2cc(C3CC3)[nH]n2)=O)C1 Cc1c(C(N2CC(CNC(=O)Cc3ccsc3Cl)CC2C)=O)cnn1CCO C1(CN(C(CNC(=O)NC)=O)C)(CNC(=O)COCC(F)(F)F)CCNCC1 C1(CNC(C(CC=CC)C)=O)CN(C(c2cnc(C(F)(F)F)nc2O)=O)CC1(C)C CCCCC(CNC(=O)CCc1cn[nH]c1)NC(=O)C(C)SCC c1(C(N2CC(C)CC(NC(c3c(CC)cno3)=O)C2)=O)cnc(N=S(C)(C)=O)s1 c1(CC)noc(C(=O)NC(C2CCN(C(=O)C(=O)NC3CC3)CC2)C)c1C Cc1ccc(OCCC(=O)NCCC(C)N(C(=O)CN(C)CCO)C)cc1 N1(Cc2cc(C)on2)CCCC1C1CCCCN1C(c1cc(C2CC2)no1)=O N1(C(CS(CC)=O)=O)CCCC(C)C1CNC(c1n[nH]c(C2CC2)n1)=O C1(NC(C=CC=CC)=O)C2CC1N(C(C1CC1c1ccccc1Cl)=O)C2 Cc1cc(C(=O)NC2CCC3CC2CN3C(=O)CCNS(C)(=O)=O)cc(C)c1C N1(C(c2cnc(C)s2)=O)CC(NC(=O)Cn2cccnc2=O)C(C)C1 C(CNC(=O)C(c1ccccc1)OC(C)C)(CCNC(C1C=CCC1)=O)OC N1(C(CCCCCSC)=O)CCC2CN(NC(=O)CC3CC(C)(C)C(=O)N3)CC12 N1(C(c2c(C)n(C)cc2)=O)CCC(N(C(=O)CSCCC(F)(F)F)C)C(C)C1 C1(NC(c2n(C(C)C)ncc2)=O)CCCN(C(C2C=CCC=C2C)=O)C1 Cc1nc(C(N2CCCC(N(C(=O)CCCc3ccc(Cl)cc3)C)C2)=O)nn1C c1(-c2onc(-c3cccc(SC)c3)n2)cnn2c(C)c(C)ccc12 c1(C(C)C)ccccc1CC(N1CC(C)(CNC(=O)CCCC2CCCC2)C1)=O C12(CNC(CN(CC)CC)=O)CCC(CNC(=O)C(C)n3ccnn3)(CC1)CO2 N1(C(C#C)C)CCN(C(=O)C(C)=CCNC(=O)CC(CC)SC)CC1 C1(C(=O)NCC(C)N(C(=O)COCC2CCCO2)C)CNC(=O)CC12CCC2 N1(CCOC)CCC2(CC1)CN(C(c1cn(C)nc1OC)=O)CCO2 C1(CN(C(C(COC)OC)=O)C)CN(C(c2cc(C)c(C)o2)=O)CCO1 c1(C(N2C(CNC(c3c(C)nc(C)o3)=O)CC(O)C2)=O)coc(S(C)(=O)=O)c1 Cc1cccc(F)c1CC(=O)N(CCC(C)NC(=O)CC1(N(C)C)COC1)C C1(C(=O)NCC(CNC(c2nc(C(C)C)oc2)=O)O)CC2(CC2)CN1C CC1(C)CCC(=CC(N2CC(CNC(C3CCCN3N=O)=O)C3(CC3)C2)=O)CC1 C(=O)(CC(F)(F)C(F)(F)F)NC12C(CN(C(c3c(N)c(O)ccc3Cl)=O)C1)CC2 CC(C)(C)C(C#N)C(=O)N1CCN(C(C2(C)COCCO2)=O)CC12CC2 Cc1cnc(N2CCC(C)CC2)c(S(=O)(=O)NC2CCCCN(C)C2)c1 Cc1ccc(Cl)c(O)c1C(N1C(C)C2CC1C2NC(C1CCN(C)S1(=O)=O)=O)=O c1(NC(C2C3CN(c4cc(C)nc(C)n4)C2C3)=O)ccc2nccn2c1C c1(C(N2C(CNC(C(C#C)(C)C)=O)CCC(C)C2)=O)onc2c1CCCC2 N1(C(CC2C(C)=NOC2=O)=O)CCC(CNC(=O)CCC(=O)OC(C)(C)C)C(C)C1 N#Cc1cc(C(=O)NCC2CCC(CNC(C3CCCCO3)=O)CC2)c[nH]1 C1(CC(=O)NC(C2CCN(C(C3CC(O)C3O)=O)C2)C)CC2CCC(C1)N2C c1(CC)c(Nc2cncc(SCc3ccn(C)n3)c2)cccc1Cl C(=O)(C#CC1CCCCC1)NC12CC(CNC(C3(C#N)CC3)=O)(C1)C2 c1(CC(N2CCN(C(C(C)SC)=O)C(CF)C2)=O)cccc2ccccc12 C=CC1(NC(C2CC2CNC(=O)COC2CC=CC2)=O)CCC1 C1(C(=O)OC)CN(C(C(=O)NC(C)(C)C)C2CC2(Br)Br)CCC12CCC2 CC(C)C(C(=O)Nc1ccsc1)C(C)NC(c1ccc2ncnn2c1)=O N1(C(CCN(CCC)C)=O)C2CCC(C(=O)NCc3n[nH]c(C)n3)C1CC2 c1(N2CC(NC(c3c(OC)cncc3)=O)C(C)CC2)ncn(C)c(=O)c1Br c1(CC)cccc(N(C(=O)C(=O)NC2CCN(C(=O)OC(C)(C)C)CC2)C)c1 c1(COC)ccccc1CN(C)C(C1CCCS1(=O)=O)=O C1(C(N2CC(CN(C(c3c(C)nsc3N)=O)C)C2)=O)CCc2c[nH]nc2C1 N1(C(c2cc(C(=O)OC)no2)=O)CCC(O)(C(=O)NCC2CCC(F)(F)CC2)CC1 C1(C(N2C(CNC(C3(O)COC3)=O)CC(COC)C2)=O)CN(C)CCN(C)C1 N1(C(c2c(Cl)ncn2C)C(=O)NC(c2ccccc2)C)CCN(C)C2(CCC2)C1 C(=O)(C1=CCCN(C)C1)N1CCC(C(=O)NCc2ccc(C#C)cc2)(CC=C)C1 C1(CC(=O)NCC2(COC)CCCO2)CC(C)N(C(c2cc[nH]c2)=O)C1 CC1(C)CC1(NC(c1cccnn1)=O)CO.c1(C(C(=O)O)S)ccccc1 C1(NC(CCN(C(CCC)C)C)=O)CC2CCC(C1)N2C(c1cnc(NC)cn1)=O Cn1c(C(N2CCCC(C(C)(C)C(=O)NCC3CCCCS3)C2)=O)ccc1C#N N1(C(c2c(CC)n[nH]c2)=O)CC(O)CC1(C)C(=O)NCCC1CC(F)(F)C1 Cc1ccnc2sc(C(=O)NC3(CO)CCN(C(C4(CO)COC4)=O)C3)c(C)c12 C1(C(=O)NC(CCC)C(=O)NCC2(C)CCC(=O)N2)CN(C)CC(C)O1 C=Cc1cc(C(=O)NCC2CCN2C(c2cc(C(F)(F)F)cc(O)c2)=O)cc(F)c1 c1(C(c2ccc(Cl)cc2)(CCC)NC(CCOCC#C)=O)ccccc1F C1(NC(C2C(OCCSC)C2)=O)CC2CCC1CC2NC(=O)CN1CCOCC1 c1(C(=O)NCC(CO)NC(C2(CCCC)CCC2)=O)cc2ccsc2n1C Cc1coc(C(N2CC(O)CC2CNC(=O)CCCn2ccnn2)=O)c1C CCC(C)C(C(=O)NCC(C)(C)CNC(=O)C(CC)C(C)C)N(C)C C(CO)(C(=O)Nc1c[nH]nc1O)NC(CSCCCCC)=O N1(C(C2C(C=C)C2)=O)CC(F)(F)CC1CCNC(c1cc(F)cc(Cl)c1)=O c1(CC(=O)NCC(C)(CNC(=O)CN(S(C)(=O)=O)C)OC)ccc2occc2c1 N1(NC(=O)CC(C)CCC2(NC(CCCOC(C)=O)=O)CCC2)CC2CCC1C2 CC1C(C(=O)NCC(C2CCC2)NC(=O)C=Cc2cncs2)CCN1C S(=O)(=O)(c1cccc(Cl)c1Cl)N1CC(NC(CCc2scc(C)n2)=O)C(C#N)C1 c1(OCC)ccc(N)c(C(N2CCCC2C2(NC(c3ccns3)=O)CC2)=O)c1 c1(C(N2CC(NC(c3c(OC)cccc3Br)=O)C(C)C2)=O)nc2ncccn2n1 C1(NC(c2c(CC)[nH]c(=N)s2)=O)CCC12CN(C(C1CCC(N(C)C)CC1)=O)C2 C(=O)(C1=CS(=O)(=O)CCC1)N1C(CCNC(c2cnc(SC)n2C)=O)CCCC1 S(=O)(=O)(c1ccc(N2CCC3(CC(F)C3)C2)nc1)N1CC(C)(C)C(CO)C1 C1(C2n3cc(nn3)C(=O)N(CCO)C23CCC3)CC1C1CCCC1.CO [N-]=[N+]=NC1CCC(OC(=O)CC(Cl)Oc2ccccc2)CC1 CC1CCC(NC(=O)CCN2CCCC2=O)CN1C(=O)CNC(N)=O C1(O)(C(=O)NC(CC)C(=O)O)CCN(Cc2ccc(C3CC3)cc2)CC1 c1(CN(C2CCCC(C)C2)CCC)c(C)nn(C)c1OC C1(NC(c2nc(C)[nH]n2)=O)CC(=O)N(C2CN(C(=O)Cc3ccc(Cl)cc3)C2)C1 N1(C(CCC=CCC=C)=O)CCC(NC(=O)COc2ccsn2)CC1C C(=O)(C1=CCC2CCC1N2C(c1ccc(N)c(F)n1)=O)N(C)Cc1nc(=O)o[nH]1 C=CC(C)N=c1[nH]c(=NCc2ccc(N(C)C)cc2)[nH]c2cc(OC)ccc12 c1(C(=O)NCC(C2CCC2)NC(C(C)O)=O)ccc(S(C)(=O)=O)cc1Br Cc1cnn(CC(=O)NC(CNC(C2CC(N3CCOCC3)C2)=O)CO)c1 C(=O)(C1NCCc2nn[nH]c21)NCC1CCCN(c2c(N(C)C)cccn2)C1 C1(N(C(C(C2CN(C(C3CCCS3)=O)C2)OC)=O)C)CCOC(C)(C)C1 C(C(CC1CC1)C(=O)NCCc1cn(C)nn1)NC(C1(C(N)=O)CC1)=O c1(C(C(=O)NCC2(OC)CCN(C(CCC#C)=O)C2)C)cc(C)cc(F)c1 c1(-c2cn(CC(=O)N(CC(F)F)C3CC3)nn2)ccc(C(=O)O)c(F)c1 O=C(C(F)Cc1ccccc1)NC1(CNC(C2CC2(Cl)Cl)=O)CC1 C1(N(C(C2(CC=C)CC=CC2)=O)CCC(c2coc(C)c2)=O)CC2(CCC(O)C2)C1 C=CCC(C(=O)NCCCc1ccnn1C)NC(=O)C(C)c1cc[nH]n1 C(c1ccccc1)=C(OC)C(=O)NC1CN(C(c2cscn2)=O)C1 c1(C(C2CCN(C(c3ccccc3)=O)C3(CC3)C2)=O)ccc2cc[nH]c2c1 C(=O)(C(C(C)(C)O)NC(C1CCCS1)=O)NCCC(CCC)O C1(CNC(CC=C=C)=O)CCCN(C(=O)CCc2ccc(C(F)F)cc2)C1 c1(SC)nccc(C(N2CCC(C)(CCNC(=O)CC(C)(C)SC)C2)=O)n1 N1(C(CCCC#N)=O)CCCCCC1C(=O)NCCn1cnnc1 C1(C(=O)NCC2=CCN(C(c3cnn4c3OCC4)=O)CC2)CCCCC(=O)C1 CC1(C#CC(=O)NC(C(=O)Nc2ccc(N=[N+]=[N-])cc2)C2(O)CCC2)CCCO1 C1(CNC(C(n2cc(COc3cnn(C)c3)nn2)C)=O)CCCCCN1C(N)=O c1(-c2onc(-c3nc(-n4cncn4)ccc3)n2)ccc2n[nH]cc2n1 c1(NC(CN(C(C(F)F)C2CCCO2)CC)=O)cc(C)c(C(=O)O)cc1C Cc1ccc(CNC(C2CCN(C(C3COCC3(C)C)=O)C2C)=O)cc1 Cc1cc(F)c(C(=O)NC2CC3CC2CN3S(=O)(=O)C(F)(F)F)c(F)c1 N#Cc1ccsc1C(N1CC=CC(C(N2CC(OCCO)C2)=O)C1)=O C1(NC(=O)OC(C)(C)C)(CNc2nccc(Cl)c2F)CCC2CCCC12 C1(N(C(=O)CCNC(N)=O)C)CCCN(C(=O)C=CC2C(C(=O)O)C2(C)C)CC1 c1(C(N2CCN(C(C3(C=C)CC3)=O)CC2CO)=O)cc2oc(Br)cc2s1 CN1CCOC2(CCN(Cc3cn(Cc4cc(C(=O)O)on4)nn3)C2)C1 C(CCCC(c1ccc(C(C)C)cc1)N(C(C)C(N)C1CCC1)C1CC1)OC c1(C(=O)NCC2N(C(c3noc(CC)c3C)=O)CCCC2)cc(S(N)(=O)=O)cs1 c1(NC)ccc(C(=O)NCC(O)CNC(=O)C(C)(C)CF)cc1F C12C3COC4(CN(C4)C1=O)C23.C=C1CC(NC(C2CC2OC(=O)OCC)=O)C1 C1(CC(=O)N(C)CC2CCCN2C(=O)CCn2cncn2)COC2(CCC2)CO1 C=CCC(CC)C(=O)NCc1ccc(C(N2CCC(N3CCC3)C2)=O)nc1 C1(C(=O)NC2C(CC(=O)NC(c3cncnc3)C)CCCC2)CC(C)(C)CCO1 c1(C(N2CCN(C(c3cn(CC)nc3)=O)CC2CO)=O)ccc2c(c1)CCCC2 c1(OCC)ccc2c(c1)NC(=O)CC(C)N2C(c1nsnc1O)=O c1(CC(=O)NCC(=O)NC2(CCCCNC(=O)CO)CC2)cccnc1 C1(NC(CSCCC)=O)CCCOC12CCN(C(=O)C(C)(F)C1=CCCC1)CC2 c1(CCC(=O)N(C(C)CCNC(=O)CCC[N+](=O)[O-])C)c[nH]c2ccccc12 c1(C(=O)NCC2CCC(NC(C=CC)=O)CC2)ccc(S(C)(=O)=O)cc1Cl CC1CCCC1N(C(=O)CNC(c1cn(C2CC2)cn1)=O)Cc1ncccn1 c1(NC(CC2CCN(C(c3n(C)c(C(F)(F)F)cc3)=O)C2)=O)cc(Br)cnc1O CCC(CC)C(=O)N1CCOCC1CN(C(=O)C(COC(C)C)NC(C)=O)C c1(OC)nc(C)ncc1C(=O)N(C1CCC(NC(c2cn(C(C)C)cn2)=O)C1)C c1(OC(C)C(=O)NC2CCC2NC(=O)Cc2c(OC)cccc2)cccc(Cl)c1 n1(C(C)(C)C)cnc2cc(OCc3cccc(SC(F)(F)F)c3)[nH]c2c1=O c1(-c2cn(CC(=O)N(C(C(C)NC)=O)C3CC3)nn2)ccc(-c2cncnc2)cc1 N1(C(c2cnc(C)[nH]2)=O)CCC(C2CC2)C1CNC(=O)CSc1ccccn1 N1(C(c2cnc(C(C)=O)s2)=O)CC2(COC(CNC(=O)C(C)CN(C)C)C2)C1 c1(-n2cc(-c3ccccc3)nn2)ccc(C2=CCSCC2)nc1 c1(C(N(C(C)CNC(C2(n3ccnn3)CC2)=O)C)=O)cc2c(F)c(F)ccc2[nH]1 C(CC(CC)C(=O)N1CCC(F)(NC(=O)CCNc2cccc(OC)c2)C1)=CC c1(C(N(C(CC)CNC(c2c[nH]nc2C(F)F)=O)C)=O)cccc(C#N)c1C CC1CN(C(c2cc(CCN3CCCC3)on2)=O)CC1NC(=O)CC1(C)CC1 N1(CC(N2C(C3(NC(=O)C=CCF)CC3)CCC2)=O)C(=O)CNC1=O c1(C(=O)NC(C(=O)OCC)CC2CC2)cc(C)on1.C1(CC(=O)N)CC(F)C1 C1(NC(=O)Cc2nccs2)CCC2(CC1)CN(c1cncc(Cl)n1)C2 c1(OC(C)=O)cccc(C(N2CCCC(C3CC(N)CCO3)C2)=O)n1 c1(C(=O)NCCCN(C(C(c2ccc(Br)s2)C)=O)C)cnc(C2CC2)o1 N1(C(c2cnc(C(C)C)nc2)=O)CC2(CNC(C34COCC3C4)=O)CC1CCO2 N1(CC(N2C(CN(C(Cc3ccn(CC)n3)=O)CC)CCC2)=O)CCN(C)CC1 C1(CCNC(c2c(C)coc2)=O)CC(F)(F)CN1C(c1ncc(C(F)F)s1)=O c1(OC)cncnc1C(=O)N(C(C)CCNC(=O)CCc1nnc(C(C)C)o1)C C1(CC(=O)N(C(CCCC)C)C)CN(C(C2(CC)CC2)=O)CCO1 c1(C(=O)NC(C2CCN(C(=O)C(O)Cc3cnc[nH]3)C2)C)cccc2c1CC(=O)N2 C(=O)(C(C)(C)C(N)=O)NC(CC(C)N(C(c1ccc(NC(CC)=O)cc1)=O)CC)C C(=O)(CCS(C)(=O)=O)NC(C(=O)N(C1CCNC1=O)CC)Cn1cccn1 c1(C(=O)NC2CCCN(C(C(CC)Cc3ccccc3)=O)C2)cc(N)cc(F)c1 c1(C(=O)NC2(C)CCN(C(C3(CC=C)CC3)=O)C2)ccc(Br)nc1O c1(C(CO)NC2(NC(=O)C=Cc3cc[nH]n3)CC2)ccc2ccccc2c1 c1(C(=O)NCC23C(CN(C(c4cc(C)c(F)cc4)=O)C2)C3)cc2c(s1)CCSC2 CC1(C)OCC2CC12C(=O)NCC1CCN1C(c1nocc1Cl)=O c1(C(=O)NCC(C)NC(C2(C)CC2)=O)cc(-c2ccccc2)n(C)n1 CCCC1C(=O)N1C.C(=O)(CSCC(N)=O)NCC=CCl c1(C(=O)NC2CC(C(CC)CC)OCC2)cc(S(C)(=O)=O)ccc1F CC1CCCC(CC(N2CCN(C3CCCC3NC(C34CC(F)(C3)C4)=O)CC2)=O)O1 CC1(C(=O)NCC#CC(=O)NCc2cn(C3CC3)nn2)CC1(F)F c1(N(C2N(C(C(CCC)C)=O)CCCC2)C)cc(C(F)(F)F)nc2ncnn12 c1(C(N2CCN(C(C#CC3(CC)CC3)=O)C(C)CC2)=O)ccc2oc(=O)oc2c1 N1(C(c2c(C)nccc2)=O)CCCN(C(=O)C(F)CC2CCCCC2)CC1C C(=O)(C(=O)N=c1ccn(CCNc2ccnn2-c2cccc(Cl)c2Cl)c(O)n1)NC CC1C(NC(C2(C)CC2Br)=O)CC2CCC1N2C(c1cc2c(F)cccc2[nH]1)=O c1(C(N2C3C(NC(c4c(COC)cc[nH]4)=O)C(C3)C2)=O)cccc2cnccc12 Cc1ocnc1CC(=O)N(C(C)CCNC(=O)CC1CC1C1CC1)C C=CCC(CC)C(=O)N(CCC(=O)OC)C.C1(C2CC2)C(=O)N1 C1(NC(c2n(C)ncc2)=O)COCCC1C1CC1.C1C(=O)N1CCOC(C)(C)C CCC(C(=O)NCC1CC(NC(C2CCCN2C)=O)C1)C(C)(C)CC N1(C(C2CC(COC)C2)=O)CCCC2(CCC2NC(=O)C(F)C(F)(F)F)C1 Cc1[nH]nc(Br)c1C(=O)NC1C2CC1N(C(=O)COCC1CCCOC1)C2 C12(CC)CC(C(=O)NCCN(C(=O)C(=O)NCC(F)F)CC)(CO1)C2 CC(=O)CCCCC(=O)N1CC2C(NC(C3CCCCN3CC(F)F)=O)C2C1 C(=O)(CCC(=O)NCC1CCCCC1NC(=O)C(C)(CC)OC(C)=O)OCC C1(C)(C(N(CC(CNC(CC2N(CC)CCOC2)=O)(C)C)C)=O)CCCS1(=O)=O c1(C(N2CCC(OC)C2)C(=O)NC2CCCCC2)ccc(C)c(C)c1F CCC(COC)C(=O)N1CC(C(=O)Nc2cscc2C)(CC)C1 C(=O)(CCC(C)(C)F)NCC1(O)CCN(C(C=C2CCC(C)C2)=O)C1 N1(c2cccc(-c3cscn3)c2)C(=O)NC(C2CCC2)C1=O.C=CC c1(NC)ccc(C(=O)NC(CC2CCC2)C(=O)NCc2nnnn2C)cc1 Cc1oc(-c2ccco2)nc1C(=O)NCC1(F)CC(NC(C2COCCO2)=O)C1 c1(-n2cc(CNC(CC(C)C)=O)nn2)cnn(C)c1C(N1CCOCC1CO)=O c1(C(=O)NCCN(C(C=Cc2ncc(C)[nH]2)=O)C2(CO)CC2)ccc(O)c(F)c1F C1(C)(CCC(=O)NCCCCC=C)CCCN1C(C1CCCCCC1)=O N1(C(c2cc(C(CC)CC)no2)=O)CC2(CCN(C(C3(F)CCOC3)=O)C2)C1 c1(CNC(=O)NC(c2occ(C(=O)OCC)n2)C)cc2cc(C)ccc2s1 N1(C(c2c(CCC)n[nH]c2)=O)CCCCC1CNC(=O)Cc1nocc1C(C)C C1(CC)C(C(=O)NC2CC(F)C2)CCCN1C(=O)Cc1nc(=N)[nH][nH]1 C1(C(=O)NCCC2(CNC(C(C)OC3CC3)=O)CCCC2)CCCC12CC2 c1(NC(C(CC)(O)c2ccccc2)=O)cnc2c(cnn2CC(=O)OC(C)C)c1 c1(C(=O)NCC(C)(CO)NC(c2cccs2)=O)cccc(-n2ccnc2O)c1 O=C(C(O)CC(F)(F)F)NCC12CCC(CC1)N2C(=O)CC1CCCO1 C1(C(=O)NCC2CCC(NC(c3cc(=NC)[nH]cc3)=O)C2)CC2C=CCC(C1)C2 COn1cnc(C)c1C(=O)NC1CCC(CCNC(c2cn(C)cn2)=O)C1 c1(CC(=O)NCCCNC(=O)CCNC(=O)Nc2ccco2)cc(F)ccc1F c1(C(N2CCN(C(C)C(F)(F)F)CC2)=O)cc([N+](=O)[O-])cc([N+](=O)[O-])c1Br CC(Cc1ccncc1)C(=O)NCC1CC1NC(=O)COC1CCOCC1 Cn1nc(CNC(C2CCS2(=O)=O)=O)cc1C(=O)NCCn1ccc(=O)cc1 c1(CC(=O)N(C)CC2N(C(c3c(C)csc3)=O)CCC2)ccccc1I C1(CNC(C2C(C)CC=CC2)=O)CN(C(=O)CCCC#N)C2CCN1C2 c1(OC)ccc(Cl)c(C(=O)NC2CC(CNC(c3ccno3)=O)C2(C)C)c1 N1(C(c2c(C)c[nH]c2)=O)CC(NC(=O)CC(O)C2CCCC2)Cc2ccccc21 C1(NC(c2nc(CC)oc2)=O)CCCC2CN(C(C34COCC3C4)=O)CCC12 N1(C(c2[nH]c(=NC)sc2)=O)CCC(CNC(=O)C(C)CS(C)(=O)=O)C(F)(F)C1 CC(C(=O)NC1CN(C(C2CC(F)(CO)C2)=O)CC(C)(C)C1)C(C)S(C)(=O)=O Cc1cccc(C)c1C(N1CCC(CCC(=O)NC2CC(O)C2)C1)=O N1(C(Cc2ncc(CC)[nH]2)=O)CCCN(C(c2cccc(O)n2)=O)CC1 c1(OC)ccc(C(N2CCN(C3CN(C(C4(COC)CC4)=O)C3)CC2)=O)c(N)c1 c1(NC(C2CC2F)=O)cccc(F)c1-c1ccc(OC2CNC2)nc1 C1(C(=O)NC(C(C)C)CNC(=O)C=CCO)CC(NC(=O)C(C)(C)C)CN1C c1(C(=O)NCCCOCCNC(CC(C)C2CC2)=O)ccc(OCF)cn1 N1(C(COCCCC#C)=O)CCCC(NC(=O)C(=O)NCC(F)F)CC1 c1(C(=O)NCC(C)(C)NC(CCc2c(OCC)cccc2)=O)c(C)cccc1C CCC(CC)(CC)C(=O)NCC1C(C)CCN1C(c1cccc(OCCF)c1)=O c1(OC)cccc(C)c1C(N1CCC(CF)(NC(=O)OCc2ccccc2)C1)=O N1(C(C(C)OC)=O)CC(C)(C)OCC1CNC(=O)CCSc1cccc(Cl)c1 c1(OC)ncc(CN2CCC(CC(=O)Nc3ncccc3CO)C2)cc1Br Cc1cnn2cc(C(=O)NCCCN(CCC(C)(C)C)C)cnc12 C1(C(N2CC(OC)C(C(=O)NCCCCCF)C2)=O)CC2(CC2)CN1C C(C)(C)(CCCF)NC(C(CN(C)C)NC(=O)CC1(CN(C)C)CCC1)=O c1(C(C(=O)NCC(CN(C(c2c(CC)scc2)=O)C)O)OC)ccccc1OC c12cc(n(C)n1)S2.CCC(CNC(=O)C(=O)NC1CC1)N(C)C c1(C(=O)Nc2cc(CCC)no2)ccc(C)cc1C.c12nc(cs1)C(=O)N2 C1(CNC(C=CCCC)=O)CCN(C(=O)C(F)(F)c2cnn(C)c2)CC1 CC1CC2CN(C(=O)CCOC3COC3)CC2N1C(c1cnc(C(F)(F)F)s1)=O N1(C(c2c(OC)ccs2)=O)CC2CCC(CNC(=O)CC3CCCC3O)C2C1 Cc1nc(-c2ccco2)sc1C(C)N(C(=O)CCc1nc[nH]n1)C C1(NC(c2c(C)coc2)=O)CC2(C1)CC(NC(c1ccn(C)n1)=O)C2 O=C(CS(=O)(=O)C1CC1)NC1CCC(CCCNC(=O)COC2CCCCC2)C1 c1(C(=O)NC2CCC(NC(c3c(C)nncc3)=O)C2)ccc2c(c1)C(=O)CCO2 C=CCCCCCC(=O)N1CCC(F)(CNC(C2(C(C)(C)C)CCCC2)=O)CC1 C=CCCCCC(=O)N1CCC(O)CC1C(=O)NCCCC1CCCCO1 C1(C(=O)NC2C(CNC(c3cccc(N)c3O)=O)C2)Cc2cc(F)cc(F)c2O1 Cc1nn(-c2ccc(F)cc2)c(C)c1CC(=O)OCC#CCN(C)C C#CC1CCCCN1C(=O)CC(c1ccc(OC)cc1OC)C(=O)O C(=O)(C1CCc2cccnc21)N1CC(C)N(C(C23CC2CNC3=O)=O)CCC1 CC(=O)C(C)CC(C)C(=O)NC1(C(=O)N(C2CCOC(C)(C)C2)C)CC1C C=CC1(C(=O)OC(C)(C)C)CN(CC2CN(C(=O)O)C2)C1.C1(C(=O)NC)CC1C c1(C(N2C(CCNC(C(C)=C(CC)C)=O)COCC2)=O)cnc2n1C(C)CCC2 N1CCN(CC)C2CCCCC12.C1(c2cn(CCCCCC)nn2)CCCCCC1 C1(C(=O)OCc2cccc(F)c2)CCC(=O)N1C(=O)CN1CCCCCC1 C(C)(C1OCCc2ccccc21)NC(c1ccc(OC)c(Br)c1OC)=O C1(C(=O)NC(C)CC(=O)O)C2CN(CC(=O)NC(c3cnn(C)c3)C(=O)O)CC12 c1(CC)ccoc1C(=O)N(CC(C)(C)N(C(C1CC(OC(F)(F)F)C1)=O)C1CC1)C c1(C(=O)NCCOC2CN(C(C3CC(C)SC3)=O)C2)ccc(C(F)F)cc1 c1(Cn2ncc(C)c2)cccc(F)c1C(=O)NNC(C1CC2CCC(C1)N2)=O C(=O)(CCCN=[N+]=[N-])NCCCN(C(c1cccc(CC)n1)=O)CCO n1(CC)ncnc1CNC(=O)C(CC(N)=O)NC(=O)CCCn1ccnn1 c1(-c2c(F)ncc(C)c2)ccc2nnc(C(N3CCOC(=O)C3)=O)n2c1 C(=O)(C1=CCC(C)(C)CC1)NCC1C(NC(COc2c(C)cc(Cl)cc2)=O)CC1 N1(C(c2cc(C)oc2C)=O)CCCCC(C(=O)NCC2(n3nccn3)CC2)C1 C1(OC)CCCCC1C(=O)N(C)CCN(C(=O)C(F)(F)c1cccnc1)C C(C(=O)NCC=CCC)=CCOC.C(=O)(C)NC(=O)CN(CC1CCC1)CC c1(C(=O)NC(CNC(C2C(C=C(C)C)C2(C)C)=O)(C)C)ccc(S(C)(=O)=O)s1 C1(C(N2CCCC(NC(=O)NCC(C)C)C2)C(=O)NCC=C)CCN(C(C)=O)CC1 O=S(=O)(c1ccc(SCOCC2CCC2)cc1Br)NCC1CCCC1 Cc1ccc2ccc(N3CC(CO)(NC(c4ncoc4C)=O)C3)nc2c1 N1(C(C2C(CC)CCCC2)=O)CC(CNC(=O)C(C)(C)C(C)C)C2(CCC2)C1 Cc1ccc(C(=O)NC(C)C(C(C)C)NC(=O)CC(C)(C)c2cccs2)nc1C c1(C(=O)NCC2(NC(CC(CC)OC)=O)CCCC2)cccn2cncc12 C1(C(=O)NC2(CCC)CC2)C=CCN1C(=O)C=CCN1CCOCC1 C(=O)(C1=C(C)CCC1)NCCn1ncc(C(=O)NC2CC(CC)C2)c1 C1(CC(=O)NCC2N(C(c3cc(C)c(Cl)s3)=O)CC(O)C2)CCCC(C)(C)C1 c1(C(=O)NCC(C(C)(C)C)NC(C(NOC)=O)=O)cc(C)cc(F)c1 c1(C(N(C(CNC(CCCOCC=C)=O)C2CC2)C)=O)cc(F)c(N)c(F)c1 c1(C(N(C2CCCN(C(=O)CN3CCCCCC3)C2)C)=O)ncccc1Cl N1(C(=O)NCCSCCC=C)CCC(=O)NCC1C C(=O)(C(C)SC(F)(F)F)N(CCN(CC(C)O)C(=O)CSS(C)(=O)=O)C(C)C C12(CNC(CC=CC)=O)CCC(CNC(=O)CCCC3OCCO3)(CC1)CO2 C1(CC)CC(C(=O)NC(c2ccsc2)C)CCN1C(=O)CC1CC(C)(C)CO1 C#CC1CCCC(NC(C2CCCC2CNC(c2cnnc(C)c2C)=O)=O)C1 C(=O)(C(O)C(C)CC)NCC(CC)NC(C1(c2cccnc2)CCC1)=O Cc1ncc(C(=O)NC2CC2CNC(=O)C=CC(F)(F)F)n1C c1(C(N(CCCNC(C(C(CC)O)C)=O)C2CC2)=O)ncccc1N=[N+]=[N-] C(=O)(C1=C(Cl)CCOC1)N1CC(C(C)C)N(C(c2cc(Cl)ncc2O)=O)CC1 C1(CS(=O)(=O)N(c2ccccn2)C(C)(C)CO)(CC)CC12CCC2 C(CC(C)(C)F)NC(CC1N(C(CN(C)C2CC2)=O)CC1)=O Cc1cc(C)c(NC(=O)CC2CCN(C(C34COCC3C4)=O)CC2)cc1C N1(C(C2N(C)CCN(C)C2)=O)CCC2CC2(C(N2CCCC2)=O)CC1 N1(Cc2ncn(C)c2)CCC2(CC1)CN(C(C1CC1F)=O)C2 N1(C(CCc2cc(C)no2)=O)CCN(C(C2CN(C)CCO2)=O)C(C)C1 N1(C(CSCCC)=O)CCC2CCC12CNC(c1c(I)ncn1C)=O c1(C2(C(=O)NC3(C(F)F)CCCNC3)CC(O)C2)ccc(Cl)cc1 N1(C(C(C)SCCN)=O)Cc2ccccc2C1.c12cc(I)ccc1N2 CC(c1ccccc1Cl)=CC(=O)NC(C1CCCC1)CNC(=O)C#CC(C)C c1(C(=O)NCC2(C)CCCN2C(C2CCC(C(N)=O)C2)=O)ccn2cncc2c1 CCCCC(CNC(C1CC(CCC)C1)=O)NC(=O)CSCc1cscn1 C=CCC(CC)C(=O)NC1(CO)CCN(C(=O)C(C)(C)c2cscc2Cl)CC1 N1(C(c2c(CC)[nH]nc2Cl)=O)CC2CCC(NC(=O)CNC(N)=O)(C2)C1 C1(C(=O)NCC2ON=C(CC)C2)CN(C(C2CCOC2)=O)C2(CCC2)C1 c1(OC(C(C)C)=O)cccc(F)c1.C12C(C1(F)F)Cc1cn(nn1)NC2 N1(C(C)=O)CCC(O)(C(C)CNC(=O)CN(c2ccc(Br)nc2O)C)CC1 C(CC(C(=O)NC)NC(c1c(CC)cns1)=O)NC(C)CC(=O)N(C)C C1(C(=O)NCC(CC(C)C)NC(=O)CCF)CCC(C)(C)CO1 c1(C(=O)NC(C(C)C)C(C)NC(=O)CCc2nncs2)cc2sccc2n1C CC1CC(C(=O)NCC2CCC(N(C(=O)CNS(=O)(=O)C3CC3)C)CC2)C1(C)C Cc1noc(C)c1CC(C)N(C(=O)CN(C(=O)Cn1nnnc1C)CC(C)C)C c1(C(N(CC)CC2CCCO2)=O)cnc2c(c1)c(C)nn2CC1C(C)(C)C1(C)C c1(C(=O)OCC(=O)NC(=O)Nc2ccccc2)ccnc(I)c1F Cc1nc(C)c(-c2nnc(N3CC=C(Br)CC3)n2CC2CCCC(C)C2)s1.SC N1(C(CC2C(=O)NCCCC2)=O)CCCC12CCN(CC(=O)NC1CC=CC1)C2 c1(C(=O)NCC2CN(C(C(CC)C)=O)CC2O)c(C)nn2cc[nH]c(=O)c12 N1(C(c2ccc(N)cc2O)=O)CCC(C2CC2)(NC(=O)CSCc2cccs2)C1 N1(C(CCC#N)=O)Cc2[nH]nc(C(=O)Nc3c(C#N)cccc3Cl)c2C1 C#CCCCC(C)C(=O)NCCC1(NC(=O)CCN2CCCCCC2)CC1 c1(SC)cc(C(=O)NCCN(C2CC(=O)NC2=O)C)c(C)o1 C1(OCC)CCCN(C(=O)C(C(C)O)NC(C2(OC)CCSC2)=O)C1 N1(C(CC2(OC)CCC2)=O)CC2CCCC2(NC(=O)CCc2cccc(F)c2)C1 Nc1cnc(C(N2CCCCC2CCC(N2CCC(F)C2)=O)=O)cn1 C1(NC(C2CC(C3CC3)C2)=O)CCCCN(C(=O)Cc2cccnc2O)CC1 c1(OC)ccc(NCCC(=O)NCC2CCCN(C(=O)CN(C)C)C2)cc1 C1(C(=O)NC(C(=O)NC(CC(=O)OCC)C2CC2)C)C2CCCCC12 N1(C(C(C)(CO)OC)=O)CCOC(C)(CNC(=O)CSC)C1 C1(C(C)C)SC(C)CC(N2CCC(O)C(C(N3CCC(CC4CC4)CC3)=O)C2)C1C C1(C(=O)NCC2CSCCO2)CCCCCN1C(c1n[nH]c2c1CCC2)=O C1(C(N2C(CNC(c3ccnc(C)c3N)=O)CC2)=O)Cc2ccc(F)cc2O1 Cc1c(Cl)ccc(C(N2CCC(C(F)F)(CNC(c3[nH]nnc3C)=O)C2)=O)c1O C1(C(=O)NC2(CN(C(CC3CCCN(C)C3)=O)C)CC2)CN=C2N=CNN2C1 N1(C(C2CC=C(C)CC2)=O)CCC(CNC(c2ccc(O)c(N)n2)=O)CC1C Cc1nn(C)c2c(NCC3CCCC3(C)C)nc(NC(=O)NCCCN(C)C)nc12 C1(C(=O)NCC(C)(Cn2cccn2)NC(C=CC(C)C)=O)CN(C)CC(C)O1 c1(C(=O)NCC2N(C(CC(C=C)(C)C)=O)CC(F)(F)C2)cnc2c(c1)CCCC2 N1(C(c2c(C)n[nH]c2)=O)CCOC(CN(C(=O)C(F)CC2CCCCC2)C)C1 c1(C(N2CCC(NC(C3(OC)CC3)=O)CC2C2CC2)=O)ccc2c(n1)CCC2=O c12cc(N3CCC(O)C(F)C3)nc(n1)CN2.c1(CCC)cc(C)no1 CN(C1CCc2ccc(Cl)cc21)C(=O)NCc1ccc2c(c1O)CCC2 C1(CC(=O)NCC(=O)NC)CCN(C(=O)C(CO)OC)C1(C)C c1(OC2(C(=O)NCCCC(C)NC(=O)Cn3cnnc3O)CC2)ccc(Cl)cc1 N1(C(c2cn(CCNC(CSCC#C)=O)nc2)=O)Cc2ccc(O)cc2C1 c1(SC)ncc(NC(c2nnnn2Cc2nnn(C)n2)(C)SC2CC2)s1 c1(OC)ccc(C(N2CC(CNC(=O)C(C)NS(C)(=O)=O)C2)=O)nn1 c1(C(=O)NC2(N(C(CN3C(C)CC3)=O)C)CC2)cnc(O)cc1C(F)(F)F C1(NC(c2nn(C)c(O)c2)=O)CC2CN(C(c3cnn4cc[nH]c34)=O)CC12 c1(C(=O)NC2CCN(C(Cn3ncc(C)c3)=O)C2)ccc(C)c(C#N)c1 c1(C(N(C2CN(C(C3CCC(C)(C)C3)=O)C2)C)=O)nc2ccccc2[nH]1 N1(C(C(CC)F)=O)CCC2(CCC2)C(CNC(c2cccc3cccnc23)=O)C1 c1(C(N(CC2N(C(CC(=C=C)C)=O)CCCC2)CC)=O)nnn2c1C(=O)NCC2 c1(C(C)=O)cccc(C(=O)NC2CC(NC(=O)Cc3n[nH]c(=N)s3)C2)n1 c1(OC)ccc(C=CC(=O)NC2(CF)CCN(C(C3(C#N)CC3)=O)C2)cc1F c1(OC)cccc2c(N3CC(N(C(=O)Cn4cc(CSC)nn4)C)C3)ncnc12 N1(C(C2CCC2)=O)CC2CC1CN2C(c1ncccc1F)=O CC1CCN(C(=O)CCCc2nc3ccccc3o2)CCN1C(=O)Cc1cnco1 CC1CCCCC1(CNC(=O)Cn1ncnn1)NC(=O)CSCC#N C(=O)(CC1=CCN(C(C2CC(F)(F)C2)=O)CC1)NC(C#C)C(C)C CC(CCS(C)(=O)=O)n1cc(C2CSCC2Br)nn1 CCC(C(=O)NCC(O)CCNC(c1ccccc1)=O)SC(C)C c1(C(N(CCC(C)NC(=O)Cn2nnc(=O)[nH]2)C)=O)coc(-c2ccccn2)n1 C1(C(=O)NC(C2CN(C(C3CN(C4CCOCC4)C3)=O)C2)C)COC(=O)C1 C1(NC(c2cc(CO)[nH]n2)=O)CN(C(=O)Cn2ncc(Br)n2)C2CC12 c1(CC)ccccc1-n1nnnc1-c1ccco1.C12(CC(O)C1)CNC2.SC S(=O)(=O)(c1cccc(Cl)c1)NC(C1CC1CNC(=O)N(CCO)C1CC1)=O C1(CNC(CCC#N)=O)CCCCC1NC(c1nn[nH]c1Cl)=O C=C1CCN(C(=O)C=CC(C)C)C(C(N2CCNC(=O)C2)=O)C1 c1(C(N(CCCCN(C(C2C(C)(C(=O)OCC)C2)=O)C)C)=O)cnc(C2CCC2)s1 O=C(C1=NOC2(CCOC2)C1)NC1CCN(C(c2ccc(F)c(C(F)F)c2)=O)C1 c1(CCC(=O)NC(C(CC)CC)C)cc(C)ccc1OCC C1(NC(CC=C)=O)CC(OC)CN(C(=O)Cc2csc(Cl)c2)C1 C(CN=c1[nH]c2cccc(Br)c2o1)CCNC(c1c(OC)nccn1)=O C(=O)(CCCC(C)C)N1CC(CNC(Cc2nc(C(C)OCC)sc2)=O)(OC)C1 c1(C(N2CCC(NC(c3cnc(C4CCC4)o3)=O)(CO)C2)=O)c(O)cccc1Cl C1(NC(c2cc(CC)no2)c2nnnn2C2COC2)(COC)COCC(=O)N1 Cc1nc2cc(C(=O)NCCC3CCCNCC3)c(F)cc2[nH]1 c1(CN2CC(NC(c3ccccc3)=O)C2)cc(F)c(O)cc1F CCCCC(O)C(=O)NCC1(NC(=O)CCC2OCCO2)CC(OC)C1 N1(C(C(=O)NCC)=O)CCCC(NC(c2oc(CC(C)C)nc2C)=O)C(F)C1 Cc1c(C(N2CCC(CN(C)C(C3CCC(N(C)C)CC3)=O)C2)=O)cncc1N c1(-c2cn(CC(=O)N(C3CCCC3)CCCOC)nn2)cc(Cl)ccc1F CC1CCC(CC(=O)NCCCCCCNC(=O)CCCN2CCCCC2)OC1 CC1CCN(C(=NCCC2(C)NC(=O)NC2=O)NC2CCCC2)C1 c12ccc(cc1)CS(=O)(=O)NC(=O)NC2.N1(C(C)=O)CCC(C(C)NCCC)C1 C1(N(C(C(C=C=C)C)=O)C)CCCN(C(=O)OC(C)(C)C)CC1 N1(C(C(C=C)(F)F)=O)CCN(C(c2ccc(C)n2CC)=O)C(c2ccncc2)C1 C1(CC(=O)NCc2cc(C(=O)NC3CC(C(C)O)C3)on2)COCC(C)O1 C(C(=O)NCCC(C)(C)NC(=O)Cc1ccc(F)cc1Cl)(C(C)(C)C)N(C)C C1(CNC(c2ccc(F)cc2C(F)F)=O)CC2CCCC2N1C(=O)CCC1CC1 O(NC(=O)C(CNC(=O)C(C)SC(C)C)CCC(C)(C)C)C(CC)C c1(C(N(C2CCN(C(=O)C(=O)NC3CC3)CC2)CCCC)=O)cccc(C)c1C c1(C(=O)NCCN(C(=O)CC2CCCOC2)C2CC2)cnc2ccccc2n1 c1(C(=O)NC2CC3CN(C(CC=C)=O)CC32)cc2cc(C(=O)OCC)cnc2[nH]1 O=S(=O)(c1cccc(=NC2CCCc3sccc32)[nH]1)N1CCOCC1C1CC1 C(=O)(C1=NOC2(CCC2)C1)NC(C(=O)NCc1c(CC)nco1)Cc1ccco1 N(C(=NCCCF)NCC1CCN(CC)C1)Cc1c(OCC)nccc1 C1(C(=O)NCC2CCCN2C(=O)CC2CCC(=O)NC2=O)CCC12CCOCC2 C(=O)(CC(F)(F)C(F)(F)F)N1CCC(Cn2cc(CCOC(C)=O)nn2)C1 N1(C(c2nc(C)oc2)=O)CC2CCCC2(NC(c2cccc3[nH]ccc23)=O)C1 c1(OC)csc2c1OCCC(=O)N1CC(C(C)C1)CNC2=O.C1(CO)CCCC1 c1(OC)cccc(CC(CC(C)C)OC)c1.C1(C2c3nnnn32)COC(C)(C)C1 c1(C(N2CC3CN(C(C(C(C)(C)C)O)=O)CC32)=O)cccc2ncsc12 N1(C(C)C)CC(CNC(c2ccc(CNC(C3CCO3)=O)s2)=O)CC1=O c1(N(C(C)(C)C)C)nc(=NCC2CCC(F)C2)[nH]c2c1CCC2 c1(C(=O)NC(C(C)C)(C)C)cc2c(s1)CCOC21CCN(c2ncccn2)CC1 C(CCOCc1ccccc1)(CC(C)C)NC(C1CCC(C(C)C)N1)=O C(=O)(CCCCc1cnn[nH]1)N(C1CN(C(=O)C=C(Cl)Cl)C1)C c1(C(=O)NCC(C)NC(=O)Cc2cnc[nH]2)cccc2nc(O)n(C)c12 c1(CC)[nH]nc(C(=O)NC2CC(CNC(=O)CSCc3ncc[nH]3)C2)c1Cl C(C(F)(F)C(=O)N1CCC(F)(CNC(=O)CSCCCc2ccccc2)C1)OC C(C(C)(C(C)C)NC(=O)C(F)=CCOC(C)(C)C)NC(C=COCC)=O.C1CC1 C(c1cnn(C)c1)=CC(=O)NC1C(CNC(c2c(CC)noc2)=O)COC1 C(=O)(C(CNC(c1ccc(O)nc1)=O)C(C)(C)C)NC(c1ccccc1O)C c1(C(N2CCC(NC(c3c(C)ccnc3)=O)CC2C)=O)cc2c(nn1)OCCS2 c1(CC)noc(C)c1CNC(C1CCN(C(C2C3CC4C(C3)C24)=O)C1)=O C1(NC(c2ccc(CC)nc2)=O)CC2CCC1C(NC(C1(OC)CCCC1)=O)C2 C(=O)(CCCC(C)NC(=O)C=CC(C)(C)C)NCC(CC=C)OC N1(CCC(C(=O)OCC)(C)C)C2CCC1CC(O)C2 N1(C(CC(C)(C)C(F)(F)F)=O)CC(C2CCCN(C(=O)CN3CCCC3=O)C2)C1 c1(C(=O)NCCC(CNC(C(N2CCNC2=O)C)=O)O)cccc(C(N)=O)c1F C=C(C)CCCC(=O)N1CCN(C2CCN(C(=O)C(C)C3(O)CCC3)C2)CC1 N1(C(CC2OCCN(C(CCOCC#C)=O)C2)=O)CCC2(CC1)CC(=O)N2 C(=O)(C(CNC(=O)C(CC1CCCC1)CC)CCC)NC(C#CC)(C)C O=C(CCCCCc1ccc(F)cc1)NC1CC(CNC(c2ccccn2)=O)C1 c1(CCC)ccc(Cl)cc1-c1nc(-c2cccc(N)n2)nn1CC1CCCOC1 C1(C(=O)NC(CC)CN(C(=O)CSC2CC2)C)CCC1(F)F C1(NC(CCCC(=O)OC)=O)CC2CN(C(c3cccnn3)=O)CCN2C1=O CCCCCC(C)(C)CNC(=O)C(C)N1CCC1CN(CC)CC.C(C)(C)(CC)O C1(NC(C(NOC)=O)=O)CC2CCC1C(NC(C1CC3COCC3C1)=O)C2 C=CCCC(CC(C)C)C(=O)N1CC(F)CC1CNC(c1cc(C)nn1C)=O N1(C(CC(=C)C)=O)CCC(NC(c2ncoc2C(C)(C)C)=O)CC1C Cc1ccc(C(N2CCCC(C)(NC(=O)C(C)C#N)C2)=O)cc1Br C1(CNC(CC2C(C)(C)C2)=O)CN(C(c2occ3c2CCC3)=O)CCC1(C)C c1(C(=O)NC2CCC(NC(CC(CC)CC)=O)CC2)c(O)nnc2c1CCC2 C1(C(=O)N(C2CCC(O)CC2)C)(COC)C=CCN1C(c1csc(C)n1)=O c1(SC)nn(C)cc1C(=O)NC(C1CCN(C(=O)C(C)N2CCCC2)CC1)C N1(C(c2ccc(C(C)=O)cc2)=O)CCc2ccc(NC(=O)C(C)N(C)C)cc21 C1(OC(CCc2cc(C)no2)=O)CCC(F)(F)C1 Cc1cc[n+]([O-])cc1C(N1CC(NC(c2nocc2Cl)=O)C(CC2CC2)C1)=O C1(C(=O)NC(C)CC(C)NC(=O)Cn2cc(N)cn2)(CC)CCNC1=O C(=O)(C(C)(C)C(=O)N1CC(NC(=O)C=CCN2CCC2)C(CO)C1)OCC N1(C(c2c(C)nc(COCC)s2)=O)CCN(C(c2cc(Cl)ncc2O)=O)C(C)C1 c1(NC(C2CCN2C(c2cc(Cl)sc2Cl)=O)=O)c(Cl)ccc2cccnc12 C1(C(=O)NCC2CCC(CNC(c3cc(C)oc3C)=O)CC2)CC2CC2CC1C Cc1ccc(C)c(CSCC(=O)NCCCCN(C)C(c2ccc(CO)o2)=O)c1 c1(C(C)=O)cn(C)nc1C(=O)NC(C)CC(C)NC(C1CCC(C)O1)=O O(NC(=O)CC(C)C(C)(C)NC(c1ccc(C)s1)=O)CC C(C)(C)(C(C)CC(=O)NC1CN(C)CC1(F)F)NC(CCSCC)=O c1(CC(=O)NC2(CCC(=O)NC(C)(C)C)CCC2)csc2c(OC3CC3)cccc12 Cn1cnc(C(=O)NC)cc1=O.C1(CC(=O)NCC2(CCC)CC2)CC(O)C12CCC2 C=CCC(C(=O)N)N(CC(F)C1CCC1)CCC1(N)CCCC1.C(#CC)OC N1(C(C(n2ncc(C)c2)C)=O)CC2CCOC2(CNC(C2(N(C)C)CC2)=O)C1 c1(C(N(c2ccccc2)CCCN(C(C(C)OC)=O)C)=O)cc2cccnc2[nH]1 Cc1noc2nc(=NC3CN(CC(C)(C)C)C4(CCC4)C3)[nH]c(N)c12 C(=O)(C1CCc2ccccc21)NCC(C)(C)NC(=O)C(F)=CCCF n1(CCC)cc(C(=O)NC2(C)CC(N(C)C)C2)c(C)n1.C12(CCC1)CC(=O)N2C C(CCCCCCN1CCC(C(C)O)C1)N(c1n(-c2cccc(C)c2)nnn1)C c1(CNC(=O)Nc2cn(C)cc2C#N)cccc2nc(O)[nH]c12 C1(CN(C(CC2(COC)CCCC2)=O)C)CCN(C(=O)C(C)NC=O)CC1 CC(C)C(C)(C)C(=O)NCC1CCCN1C1CCCC1.C12(C(=O)N)C3C4C5C3C1C5C24 c1(C(N(CC(O)CN(C)C(C2(C(F)(F)F)CCCC2)=O)C)=O)cc(C#N)ccn1 C(=O)(C(C)(C)C(F)F)NCCC1CC(NC(Cc2c(C)nc(S)s2)=O)C1 c1(C(=O)NCCCNC(C2(CCNC(c3ccco3)=O)CC2)=O)c[nH]nc1CO C1(N(C(=O)CC(N)=O)CC)CCC(NC(=O)CC2COCC2(C)C)CC1 C(C(O)C(C)(C)C)NC.C1(=O)C(C)N1C.C(COC)OC C1(C(=O)NCc2c(C(=O)NCC(C(C)O)O)[nH]cc2)CCCC(F)C1 c1(C(=O)NC2CCCN(C(c3n(CC)ccc3)=O)C2C)cccc2c[nH]nc12 N1(CCNC(C2C(C)CCO2)=O)CCC(NC(c2cnsn2)=O)CC1 CN1N=CC(CC(N2CCC(c3cccc(-c4ccc(O)nn4)c3)C2)=O)C1=O C1(C(=O)NCc2nnc(C(C)C)s2)CC(C#N)(c2ccccc2)C1 C#CCCCCC(=O)N1CC(=O)NCC1C(N1CCC(C(C)(C)C)C1)=O C1(C)(C(N(CCN(C)C)CC)=O)CCN(C(C2(COC)CC2)=O)CC1 C1(NC(c2cncs2)=O)CN(C(C2CCCCS2(=O)=O)=O)C2CCCCC12 c1(C(=O)NC(C2CN(C(C3(C=C)CCCCC3)=O)C2)C)c(Cl)oc2ccccc12 N1(C(C2(C#C)CN(C(=O)C(C)=C3CCCC3)C2)=O)CC(C)C(C)C1C C12(CNC(C(C(C)C)OCC)=O)CN(C(c3cc4n(n3)CCO4)=O)CC1CCO2 Cc1ccc(C=CC(=O)NCC(C(C)C)NC(c2cc[nH]c(=N)c2)=O)cn1 c1(N(CCC2(CC)CCC2)C)nnc(-c2ccccc2C)n1CC1CSCCS1 C(=O)(CC(F)(F)F)NC(C1(CNC(C2C(C)CC2)=O)CCC1)=O.C1(=O)CCN1 N1(C(C(C)(C)c2cccs2)=O)CC2CC(O)C1C2NC(C1CCCS1)=O C(=O)(CN(C)C(C)=O)NCCOCC(=O)N(CCC)CCOC N1(C(CC(=O)OC(C)(C)C)=O)CCN(C(c2cnnc(O)c2)=O)C(CC(F)F)C1 Cc1ccc(C(=O)NC2CN(C(C3(c4ccsc4)CC3)=O)C2)c(O)n1 c1(C(=O)NCCOCCN(C(c2c(C)ccnc2C)=O)C)sccc1S(N)(=O)=O N1(C(C(C)SCC)=O)CCN(C(=O)C(O)C2CCCC2)C(CCO)C1 CCCC(O)(CCC)CC(=O)N1CC(O)CC1Cn1cc(Cn2ccnc2)nn1 Cc1ccc2scc(C(N3CC4CCCC(C3)N4C(c3cnsc3)=O)=O)c2c1 C1(F)(CNC(C2(CC)CC2(F)F)=O)CCCN(C(c2ncccc2O)=O)C1 c1(C(N2CC(CN(C(C(C)C(F)(F)F)=O)C)OCC2)=O)cncc2ccsc12 C(=O)(C1CCSc2ccccc21)Nc1c(C#N)ccc(CCO)c1 c1(C(N(C(C)CNC(=O)CC2CC3(CC3)C2)CC)=O)ccc(Cl)cc1F Cc1cc(CC(N2CCCC2CCC(N2CCCC(C)CC2)=O)=O)ccc1O C(C)(C)(CC(=O)N1CC(O)(CN(C(=O)Cc2ccccc2C(F)(F)F)C)C1)OC c1(OC)cccc(C(=O)NC2CCCCN(S(=O)(=O)C(Cl)(Cl)Cl)C2)c1F CCCC(C)(O)C(=O)N(C1CCC(CNC(c2ccc(C)n2C)=O)CC1)C C(CC(O)CNC(=O)CC1CCCOC1)NC(=O)CSCc1cccnc1 c1(CNC(CCCC2(NC(CC(=O)N(C)C)=O)CCC2)=O)cnc(O)nc1O c1(OCc2cn(C3CCC(C(=O)NCCSC)C3)nn2)ccc(F)cc1 c1(C(=O)NC2(CNC(=O)COc3ccccc3F)COC2)cc(Br)ccc1O N1(C(=O)N(c2cccs2)CC2(C)CCCO2)CCC(Oc2ccccc2)CC1 C(N=c1[nH]c2cc(F)c(F)cc2s1)C1CCCCN(C(c2nc(CC)oc2)=O)C1 c1(C(N2C3CN(C(c4cc(I)ccc4F)=O)CC32)=O)cnc2ccccc2n1 c1(CC)n[nH]c(=NCN2C(=O)CCC(C(=O)NC3CCOCC3)C2)s1 Cc1cc(Cl)ncc1NC(C1(CNC(=O)CC2OCCC2(C)C)CC1)=O C1(NCC(N)CC(F)(F)F)CCc2c(cnn2Cc2ccccc2)C1 N1(C(C(CC)C)=O)CCCC(NC(=O)C(Cc2ccccc2)CC2CC2)CC1 CCC(C)C(C)C(=O)N(C1CN(C(=O)CNS(=O)(=O)N(C)C)CCC1C)C c1(CC)ccc(C)c(C(N2CCC(C)(CCNC(C3CC(OC)C3)=O)C2)=O)c1 N1(C(C(C2(C)CC2)NC(C(C)N(C(C)=O)C)=O)=O)CC(=O)N(C)CC1C n1(C(COC)C)cc(C(=O)NCC(n2cc(-c3csc(C)c3)nn2)C)cn1 c1(C(N(CCCN(C)C(c2cc(C(F)F)n(C)n2)=O)C)=O)ccc2ccoc2c1 N1(C(=O)COc2ccsc2)CC(C2CN(C(C3CCN3C3CCCC3)=O)C2)C1 c1(CC(=O)NC2CCC(F)(F)C2)cnc2n1CCOC2.n12cc(nn1)CSCC2 c1(CN2CCC(F)(C(N3C(C(CC)OC)CCC3)=O)C2)cnc2[nH]ccc2c1 N1(C(C2C(C)C2C)=O)CC(NC(c2ccnc(N(C)C)c2)=O)C2(CCOCC2)C1 C1(NC(CN(C(C)C)C)=O)C2CC3C(C2)C13C(=O)NC(C)C(C)(C)N(C)C CC1CCCC(C(=O)NCc2nocc2C(N(C)CP(C)(C)=O)=O)CC1 N1(C(CN(CCC)C)=O)C(CNC(=O)CCc2ccc(OC)cc2)CC2CC12 c1(C(=O)NCCC2CCCN(C(CC(COC)C)=O)C2)cn2cccnc2n1 n1(C(N(CCOCCNC(CCc2cnc(C)o2)=O)C)=O)cnc2ccccc12 c1(C(=O)NCC2(NC(C3N(C)CCCC3)=O)CC2)ccc(O)c(C(N)=O)c1 N1(C(C(C(C=C)C)C)=O)CC2(CCN(C(=O)CCCc3cccc(Cl)c3)CC2)C1 C1(NC(C(C)=C(CC)C)=O)CCC(O)CN(C(=O)C(F)CC2CC2)C1 N1(C(C2C(=C)CC2)=O)CCN(C(c2cccc3cncn23)=O)C2(CC2)C1 N1(C(CC(C)CF)=O)CC(NC(c2cncc(C(F)(F)F)n2)=O)CC(F)C1 c1(N(CC(C)NC(c2cncc(Cl)n2)=O)C)ncnc2ccc([N+](=O)[O-])cc12 N1(C(COc2ccc(CC)cc2)=O)CCC(N=c2[nH]c(C#N)c(Cl)s2)C2(CCC2)C1 N1(C(Cc2ccc(OCC)nc2)=O)CC2CCC1CN2C(=O)C=C1CCC1 c1(C(=O)NCCNc2ccc(C(=O)O)cn2)csc2c(NC3CC3)ncnc12 C1(CC(=O)NCC2(F)CC(CNC(c3ccn(CC4CC4)n3)=O)C2)CCC2CC12 c1(C(=O)Nc2cccc(C(=O)NC)c2)cc2c(C3=CCSCC3)cncc2s1 c1(-c2onc(C)n2)ccc(C(=O)NC(C)C(C)NC(C2(O)CC2)=O)cc1 C1(NC(CCn2cc(COC)nn2)=O)CN(C(=O)CC2CC2)CCC12CCOC2 C(=O)(CS(=O)CCC(F)(F)F)NC(CNC(C=CC)=O)(C)CC CC(O)(CC(=O)N1CCCC(F)(CNC(c2ncc(Cl)s2)=O)C1)C(F)(F)F C1(CNC(CCNS(C)(=O)=O)=O)CC2(CCC2)CN1C(C1CCOC(=O)CC1)=O C(CCCCNC(=O)CCc1cn[nH]c1)N(C(CC1C(C)C1)=O)C c1(CC)c(C(=O)NCCNC(C2CN(C(C34CC(C)C3C4)=O)C2)=O)cnn1C c1(-c2nc(C3(C)CCC4CC4C3)on2)ccc2c(c1)OCCO2 C(C)(C(=O)NC1CCN(C(c2cccc(Br)c2)=O)C1C(C)C)(C(C)C)OC N1(C(C2C(CC)CCCC2)=O)CCC(CO)(NC(c2csc(C(F)F)c2)=O)CC1 C12(NC(c3c(C)nc(CC(C)C)s3)=O)CCN(C(C3(S(C)(=O)=O)CC3)=O)CC1C2 C1(NC(c2cn(CCC=C)nn2)=O)CCN(C(C2(CC)CCCC2)=O)CC1 N1(C(c2cncc(C)n2)=O)CC2CCC2(CC(N2CCC2C(=O)N(C)C)=O)C1 Cc1c(C(N2CC3CCN(C(=O)CN4CC(=O)NC4=O)C3C2)=O)sc2nccn12 Cc1oc(CO)cc1C(=O)NCC(C)(F)CNC(C1(C)CCCC1C)=O N1(C(Cc2ncc(CC)[nH]2)=O)CCC2C(CCN2C(=O)C(C)NS(C)(=O)=O)C1 C(CCCCC(=O)N1CC(N(C(=O)CCc2cncs2)CC)C(C)C1)OCC c1(C(C)C)ccc(C(=O)NCC(C)CN(C(C2CCOC2)=O)C(C)C)o1 C1(NC(C(C)C(C)O)=O)CCN(C(=O)Cc2cccs2)CCC1CO C1(C(N(C)CCOCCNC(c2cc(=N)[nH]c(=N)[nH]2)=O)=O)Cc2cscc2C1 c1(CC(=O)NC(C)C(C)NC(C2(F)CCOCC2)=O)ccc(C(N)=O)nc1 N1(C(C2(CC#C)CCCO2)=O)CC2CC(NC(C3CCC(C)C(C)C3)=O)CC2C1 C1(CNC(C(C(=O)OCC)F)=O)CC(NC(c2ccon2)=O)C12CCC2 c1(-c2c(C(=O)NCCOCCC)[nH]cn2)nc(C2CC2)cc(C(=O)O)c1C CC(CN=c1ccc([N+](=O)[O-])c[nH]1)N(C(=O)Cn1ncn(C)c1=O)C Cc1cc(C(=O)NCC(C)CNC(c2ncccn2)=O)c2c(c1)CCCN2 C=C(C)C(O)CC(=O)NC(CNC(=O)C(C)(C)N1CCOCC1)C1CC1 c1(C(=O)NC(c2ccccc2)CNC(C(C)(C)C2CC2)=O)cnc2c[nH]nc2c1 N1(C(C)=O)CCCC(C(=O)N(C(C)C)CC2CN(C(C)Cc3ccc(C)s3)C2)C1 N1(C(c2c(OC)nsc2)=O)CC2CC2(NC(C23CC(C(F)(F)F)(CO2)C3)=O)C1 C#Cc1ccc(C(=O)N(CC(C)NC(c2cnn(CC(F)F)c2C)=O)CC)nc1 C1(NC(C2CCC(F)CC2)=O)CCN(C(c2cscc2C(F)(F)F)=O)C1C1CC1 c1(CN2CC(C(N3C4CCC3CC4)=O)OCC2)cnc(Cl)nc1Cl C1(C(N2CCN(C(C3(C)CCNC3=O)=O)CC2CO)=O)CNC(=O)CC12CCC2 Cc1cccc(NC(=O)CCNC(=O)Cn2ccc(C)c2)c1 C1(NC(CC2C(NC(CCC=CC)=O)CCC2)=O)CNC(=O)C12CC2 C12CCC(CC1)NC2=O.C(=O)(C(C1(C)CC1)NC(=O)CCN(C1CCC1)C)OC C(=O)(CCCCC(=O)N1CC2C(NC(=O)CCc3nnc(O)nc3O)C2C1)OC N1(C(C(c2ccccc2Cl)C)=O)CC(NC(=O)CCCC2CCC2)C(O)C1 C1(CC(=O)NCC(CNC(C(c2cccnc2)OC)=O)C)CCCC(F)(F)C1 CCCCC(C(=O)N1CCC(N(C(=O)Cn2nnnc2C2CC2)CC)C1)N(C)C CCC(C)CC(=O)NCC1CCCN1C(=O)C(C)=C1CCCC1 N12CCC(CC1)C2.C1(C(C)C)CCCN1C(=O)Cn1cc(C(C)O)nn1 CCC(C(C)(F)F)NC(=O)COCCNC(=O)CCC1CC1(F)F c12cccc3c1CCCN3C(=O)C=CC(=O)N2.c1(N(CC(C)C)C)ccccc1 C#CC1(C)CCCN(C(=O)C(CC2CN(C(C3(CO)CCOC3)=O)C2)OC)C1 c1(NC(C(COC)(C)C)=O)ccc(OC)c(-c2cccc(OC)c2)c1 Cc1ccc(N2CCC(C(N3CCCC(Oc4ccncc4)C3)=O)C2=O)cc1 N1(C(COCCC)=O)CC2CCCC(NC(=O)C(N3CCC(O)CC3)C)(C2)C1 c1(C(=O)OC)ccc(CN2CCCC(C)C2)c(O)n1.c12ccc(cc1)o2 C(c1cn(C)cn1)=CC(=O)NC1C(NC(c2ccc(C(C)=O)o2)=O)CC1 C(=O)(C(C)(O)C(F)(F)F)NCCCCC1CN(c2nnc(CC(C)C)s2)C1 Cc1nc(NCCC2CCC(NC(c3ccc(O)nc3)=O)C2)c2cnn(C)c2n1 Cc1nccc(C(N2CC(C3CC3)(C(N3CCCC3CCO)=O)C2)=O)c1N c1(CC)oc(C(N2CCCC(CNC(C3CCCC(C(C)C)C3)=O)C2)=O)cc1C c1(C(C)C)nccc(C(=O)NC(CNC(=O)C(c2ccc(O)cc2)N(C)C)CO)n1 C12CC3CCC1N(C3)C2=O.N1(C(C)C)CCCC(N(C)C)C1=O N1(c2nnc(C)o2)CCN(C(c2cc(C3CCN3OC(C)(C)C)on2)=O)C1=O c1(C(N2CCC(C(=O)NCN(C(=O)CN(C3CCC3)C)C)C2)=O)sccc1C#N C#CCCCCC(=O)NCC(C1CC1)NC(c1cccc(-c2ccccc2)c1)=O c1(C(C(=O)N(C(C)CO)CC)C)cccc(Br)c1 N(C(=NCCC1COC(=O)N1)NCc1ccnn1C)Cn1cc(CC)nn1 C1(NC2(N(C)C)CCCC2)CCC(C(=O)N(C(C2(C)CCCO2)=O)C2CC2)CC1 Cc1ncc(C(N2CCC(O)(CN(C)C(C3CCC(=O)N3C)=O)C2)=O)cc1N N1(C(CC2CCC(C)C2)=O)CCOCC(CN2C3(C(=O)NC4CC4)CC(C2)C3)C1 C1(OC)(CNC(=O)C(C2CCCCC2)NC(=O)C(CO)N(C)C)CCCCC1 C1(C(=O)NCCCC(C)NC(=O)CCC(F)(F)F)CCCC(C)(C)C1 c1(C(=O)NCCN(CCC)C(c2cc(-c3cccs3)on2)=O)c[nH]c(=N)cc1C C1(NC(C(C)NC(C)=O)=O)COC2(C1)CN(C(C1CC1c1ccccc1)=O)C2 C(=O)(C(CCC)S(N)(=O)=O)N1CCC(CC=C)(NC(C2CC(C)CCO2)=O)CC1 N1(C(C2CC(OC)C2)=O)CCCC(C(C)NC(C23CCC(CC2)C3)=O)C1 N1(C(CCc2scc(C)n2)=O)CCC(NC(=O)C(F)=CC2CC2)CC1C C1(O)(C(=O)NC2CCCC(NC(c3ccsc3Cl)=O)CC2)CC2(CCOCC2)C1 N1(C(C(C(C)NC(CC2C(CC)C2)=O)C(C)C)=O)CC2CCN(C)C2C1 C1(CC(=O)NC(C)(C)C(=O)NCCOC(F)F)CCC(C#N)C1 Cc1ccc(OCC(=O)NC(CNC(c2ccc(O)c(N)n2)=O)CO)c(C)c1 C1(C(=O)NCCCC(C)NC(=O)CC2CC(F)(F)C2)CCn2nnnc2C1 C1(NCC(CC(=O)O)c2ccccc2)CN(CCO)CC2(CCC2)C1 N1(C(C2(NC(c3cc(C)on3)=O)CCCC2C)=O)CC2CC(C)C2C1 C1(O)(CC(N2C(CCCNC(c3c(C)ccs3)=O)CCC2)=O)CCCCC1 C(=O)(CCCN(C)N=O)N(C1CCC(CNC(c2c(O)ccc(C)c2)=O)CC1)C C1(c2n(C)cnc2)CN(C(=O)C2=CCC2)CC1NC(c1cc(Br)c[nH]1)=O C(=O)(C(F)(F)C(F)F)N(C)CC1CCN(C(C2CC23CCCC3)=O)C1 Cc1cccc(S(=O)(=O)NC2CN(C(=O)CN3CCCC(C)C3)C2)c1 C(=O)(C(F)CC)N1CC(OCCC(N2CC(CC)C2)=O)C1 c1(C(=O)NCC2(NC(CC3(C)OCCO3)=O)CCC2)cccc(C#N)c1F CC(C)(O)CC(=O)NCC(CO)NC(c1cccc(OC2CCCC2)c1)=O c1(C(N(CCNC(CC(C)C(C)(C)C)=O)CC2CC2)=O)cc2c(cn1)COCC2 N1(c2cc(NCC3(CCOCC)CC3)nc(C)n2)CCC2(CCCCC2)C1 Cc1coc(C(C)C)c1C(=O)NC1CC(CNC(c2ncc(Br)cn2)=O)C1 N1(C(C2(C#C)CC2)=O)CCCC(C2(NC(=O)C(C)NC(=O)NC)CC2)C1 C(=O)(CC(C(F)F)c1ccccc1)NC(CC(C)NC(c1cnc[nH]1)=O)C c1(CNC(C(C)(C)COC)c2n(C(CC)C)nnn2)ccc2ccccc2c1C C(C(C)C)(C(O)C(=O)N(CCNC(C1(c2ccccc2)CC(C)C1)=O)C1CC1)OC c1(CCNC(C2CN(CCN3CCCC3)CCC2O)=O)ccc2c(c1)OCO2 c1(C(N2CC(CNC(c3cc(OC)n(C)n3)=O)C(O)C2)=O)nc2sccn2c1C C(=O)(C(C)(O)C(C)(C)C)NCC(C)NC(c1nccn2nccc12)=O C1(NC(Cc2nc(C)sc2)=O)CC2(C1)CC(NC(c1onc(C)c1C)=O)C2 CN1CC(NC(=O)CC2CCCN(C(=O)Cn3ccc(C4CC4)n3)C2)CC12CCC2 C1(C(N(CCC(=O)NCCCc2cc(C)no2)CC#C)=O)CC=C(C)CC1 N1(C(Cc2cc(CC)no2)=O)CCN(C(=O)CC2CC2C(F)(F)F)C(C)CC1C CC(C)C(CC(=O)NC(=O)C#CC(C)(C)C)O.C1C(C)C(=O)N1.C1CCC1 CC(CCC(=O)N(CCC(=O)NCCCO)CCN1CCCC1=O)N(C)C C1(F)(CNC(C=CCOC)=O)CC(NC(=O)C=Cc2cocn2)C1 N1(C(C2CCCC(C(=O)OC)C2)=O)C(C)CC2CN(C(c3c(Cl)cnn3C)=O)CC12 C(CC(C)C(=O)N1CCC(CC(=O)NC(CCOC)C(C)C)C1)=CC c1(-n2cc(CC(C(F)(F)F)N3CCOCC3)nn2)ccc2cccc(Cl)c2n1 CC(N=c1[nH]c(=NCC2CC(C(F)(F)F)C2)[nH]c2c1CSC2)C1CCOCC1 c1(NC(C2(OCC)CC(C(F)F)C2)=O)cnc(Cl)c(C)c1 c1(C(N2CCCC(NC(c3cc[nH]n3)=O)(CO)C2)=O)cc(Br)ccc1[N+](=O)[O-] N1(C(CCC(C)(C)F)=O)CCC2(CC1)CCN(C(=O)CC13COC(C1)C3)CC2 c1(C(=O)NC2C(NC(CCCCC=C)=O)CC2)ccc(C#N)c(OC(F)(F)F)c1 Nc1cc(F)c(F)cc1C(=O)NCC1CCCC1NC(=O)Cn1ccccc1=O C(=O)(C1CCc2ccccc21)N1C2(COC)CC(NC(c3c[nH]nc3F)=O)(C1)C2 C1(CC(=O)NC2COCCN(C(c3csc4ncsc34)=O)C2)CC2(CCC2)CO1 C=CCC(C)(CC)C(=O)N1CCOCC1CC(N1CC2(C1)CC2(F)F)=O c1(CC)nc(N2CCCC(NC(c3c(C(F)(F)F)cnn3C)=O)CC2)[nH]c(=N)n1 c1(C(N(C2CCN(C(=O)COCCF)C2)C)=O)nnc2n1CCC2 Cc1ccc(C(=O)NC(C)C(C)NC(c2cnn(C)c2C(F)F)=O)c(N)c1Cl N1(C(c2cc(C)c(C)s2)C(=O)NC2CC(C(=O)OC)C2)CCC2(CCC(O)C2)C1 N1(C(c2ccc(CCC)nc2O)=O)CCc2nc(NC(=O)CN(C)CC)sc2C1 c1(CC)ccc(=N)[nH]c1-c1cccc(CN2COCCC2CCO)c1 Cc1ccoc1C(=O)NCCC1CN(C(=O)C=CCN2CCCC2)C1 O=C(C#CC1CCOC1)NCC1(C(=O)NCC(F)C2CCC2)CC2(CC2)C1 N1(C(c2ccc(C(C)C)s2)=O)CCN(C(C2CSCCS2)=O)C(C(C)(C)C)C1 C1(CCNC(c2cc(CC(=O)OC(C)(C)C)sc2)=O)CC(O)C12CCC2 N1(C(=O)Cc2ccc(Cl)cc2)CCCC2C1CCN2C(=O)Cc1ccncc1 N1(C(c2c(CC)occ2)=O)CC(C2CCCN(C(c3[nH]c(=N)sc3C)=O)C2)C1 c1(NC(N2C(C(CC)O)CCC2)=O)nn(Cc2ccccn2)cc1Cl CC(C(=O)N1CCN(C)C(CNC(=O)CC(=O)NC2CC2)C1)C(C)(F)F c1(CC)c(C(=O)NCCNc2cnc(OC)cn2)cccc1C c1(C(=O)NCC2C(C)CN(C(=O)C(C)OCC3CC3)C2)c[nH]c2cccc(Cl)c12 c1(C(c2nnnn2CCCC2CC2)NC(C(=O)NCC(C)C)C)ccnc(F)c1 c1(C(N2C(C)CC(NC(c3csc(O)n3)=O)C2)=O)cccc2nonc12 C1(C(=O)NCC2CC(OCC)C2)C=CCN1C(=O)Cn1nnc(C)n1 c1(C(N2C(CNC(C3CCO3)=O)CCC2)=O)ccc(Cl)c(C(F)(F)F)c1 C1(C2CCNCC2)(C(=O)NCC(C(C)C)=O)CCOCC1 C#CCCCCCC(=O)NC(C)(C)CC=CC(N1CCC(C(C)OC)C1)=O c1(C(=O)NCC2N(C(Cc3n(C)ncc3)=O)CCOC2)noc2c(F)cccc12 c1(CC(=O)N(C2CCC23CCNCC3)C2CNC(=O)C2)cccc2ccccc12 C(CC(O)C(=O)NC1CN(C(C)C)CC1C)NC(Cc1c(C)con1)=O N1(C(c2c(CC)nns2)=O)CC(C)N(C(=O)CCN2C(C)CCCC2C)CC1C c1(C(=O)NC(C(C)(F)F)CS(C)(=O)=O)cc(=O)c2ccc(F)cc2o1 C1(C(=O)NCC=CCNC(c2c(C)nn(C(C)C)c2)=O)CN2CCN1C(C)C2 c1(CCN(CC(C)NC(C2CC(OCC)C2)=O)C)cccc(Cl)c1 C(c1ccnn1C)=CC(=O)N(C)CC1(CNC(=O)C=CCN2CCCC2)CC1 CCC(C)(CC(=O)O)NC(C1CCCN(CC(F)F)C1)=O c1(C(C)C)cc(C(=O)NCCN(C(C2CC2)C2CC2)CC2CC(=O)CO2)n(C)n1 C=CC(C)(O)CC(=O)NCCn1cc(CNC(C2CCC3CCC23)=O)nn1 c1(CC(N2C3(CN(C(c4ccc(=O)oc4)=O)C3)CC2)=O)nc2ncccn2n1 C1(C)(C(=O)NC(CCCNC(C2C(C)=CCS2)=O)(C)C)CCCCNC1=O N1(C(c2c[nH]nc2C2CC2)=O)CCC2C(C1)CN2C(=O)C1=CCCCCC1 CC(C)(CC(=O)N1CC(NC(c2sc(F)cc2Cl)=O)C(O)C1)CC(F)F c1(C(N2CC3CC2CN3C(c2cn3ccccc3n2)=O)=O)c(F)cc(Cl)cc1Cl c1(CC)cnccc1C(N1CC2C(C(N3CCCC(C(C)C)C3)=O)C2C1)=O CC(CNC(=O)CC(=O)N(C)C)CC(=O)Nc1ccc(F)nc1 N1(C(C(C)(C)NC(=O)NCC)=O)CCCC(CNC(c2cccc(CO)n2)=O)C1 c1(C(=O)NC2C(NC(c3c(O)ccc(C)n3)=O)CC2)cccc2c1COCC2 c1(C(C)=O)ccc(N(C)CCN(C)C(C23CCC(CC2)CC3)=O)c([N+](=O)[O-])c1 c1(NC(C=CC(CC)C)=O)nn(C)cc1N N1(C(C(C)=C(C)C)=O)CC(C2(NC(=O)CCOCc3ccccc3Cl)CC2)C1 C(CC1=CCOCC1)NC(CN(C(CCCN(C)C)=O)CC1CC1)=O C1(C(=O)NC2CN(C(CCCCC(N)=O)=O)CC2N(C)C)Cc2c[nH]cc2S1(=O)=O N1(C(C2C(CC)C2)=O)CCCC(C2CCN(C(c3ncn(C(C)C)n3)=O)CC2)C1 C1(NC(CN(CCC)C)=O)CC2(CCN(C(=O)C(C)CC(F)(F)F)CC2)C1 C1(C(=O)NC2(CSC)CCC2)C=CCN(C(=O)C(C(C)O)N(C)C)C1 Cc1ncc(C(=O)NCc2ccc(C(=O)NC(c3ncc[nH]3)C)s2)s1 C1(NC(c2n[nH]c(C)c2Cl)=O)CN(C(C23CC(F)(C2)C3)=O)CC1S(C)(=O)=O c1(CC)cnccc1C(N1CCC(CO)(NC(=O)C=Cc2ccco2)C1)=O N1(C(C(Cn2ccc(C)n2)C)=O)CC2OCCN(C(c3coc(C)n3)=O)C2C1 C(=O)(C(CC)C(=O)OCC)NCC(CCCC)NC(c1ccc(C(C)C)cc1)=O c1(COC(C(=O)NC2CCC(CNC(CSC)=O)C2)C)cccc(C)c1 N1(C(C(CC)OC2CCCC2)=O)CCC(C2(NC(=O)C3=CCCOC3)CC2)CC1 C(C(=O)N1CCCC1(C)C(N1CCC(O)(CO)C1)=O)(C(C)(C)C)OC Cc1cc(N2CCCN(CC(O)COC)CC2)nc(=NCCOC)[nH]1.C(C)C c1(C(N2C(C(C)NC(CC(C(C)C)O)=O)CCC2)=O)cncc2c(O)nccc12 C(=O)(C(F)CC(C)C)N1CCC(CN(C(c2cnc(C)[nH]2)=O)C)CC1 C1(C(=O)NC(N2CCCC(C(c3nccc(O)n3)C)C2)=O)CCC(F)(F)CC1 C(=O)(C#CC1CCCO1)NC1(C)CCN(C(c2nc(OC)c(C)s2)=O)C1 N1(C(C(C)(C)C)=O)CCCC(CCNC(=O)C(F)CC2CCC2)C1 C1(C(=O)NCC2CC(CNC(CCCOC)=O)C2)CC(=O)N(C)C1 Cc1ccc(C(=O)NCC2(c3ccccc3)CCCO2)c(Br)c1 C1(CN(C(CN(CCC#C)C)=O)C)COCCN1C(=O)C=Cc1ncc(C)[nH]1 C(=O)(C1=NOC(C)(C)C1)NC1C2(CCN(C(C(C)NC(=O)NC3CC3)=O)C2)C1 C1(NC(=O)CCCSc2ccccc2)(CO)CCN(C(=O)CC2CCC=CCC2)C1 C1(C)(NC(CN2CCC(C)CC2)=O)CCN(C(C2CC2C(F)(F)F)=O)CC1 C(=O)(C(CC)CCCCC)NC1C2(CC(NC(C3(CCCC)CC3)=O)C2)C1 C(=O)(C(C)(F)C(C)(C)F)N(CC(C)NC(c1n[nH]c(C2CC2)c1Br)=O)CC C1(C(=O)NC2C(NC(CCC(C)(C)F)=O)COC2)CSC(c2ccccc2)=N1 Cc1cn2cc(C(=O)NCCCCn3cc(CC(C)(C)CO)nn3)nc2s1 C#Cc1cnn(C)c1C(N1CCC2C(NC(=O)CC3CC4CC4C3)C12)=O CC1CCCC(C)N1C(N1CC2CC1CN2C(c1ccc(OC(F)F)cc1)=O)=O c1(CN2CC(NC(Cc3ccc(OC)cc3)=O)C(C)C2)cc(Cl)c(O)cc1F N=c1[nH]nc(C2CCCN2CC(=O)N(C(C2CCOCC2)c2cccs2)C2CC2)s1 C1(N(C)C(C2CCC3C(C2)C3(F)F)=O)CCSC12CN(C(C1CCCCCC1)=O)C2 Cc1cc(=NCc2ncc3ccccn23)[nH]c(N2CCN(C3CSC3)CC2)n1 Cc1ncnc(C)c1CC(=O)N(C1CCN(C(C2CC(C)(F)C2)=O)C1)C c1(C(=O)NC2(CCNC(c3ccc[n+]([O-])c3)=O)CC2)nc(C(F)(F)F)oc1Br C(C)(C)(C(O)CO)NC(C(CC)N(C(=O)C(C)CC1CC1)C)=O C(=O)(C(O)Cc1cnc[nH]1)NCC(CN(C(=O)C(F)OC(F)(F)F)C)O c1(C(=O)OCC)cc(C(=O)NCC(F)CNC(c2nnn(C)n2)=O)c(C)o1 CC1CN(C(c2ccc(CF)cc2)=O)C(C)CN1C(=O)C(O)CC1CCCC1 CCCC(C)CC(=O)N1CCCC(N(C)C(c2cccc(C)c2O)=O)C1 Cc1cc(Cl)cnc1S(=O)(=O)N1CCSC(c2ccccc2)C1 O=C(CC1OB(O)c2ccccc21)Nc1ccc(Cl)c(I)c1F C(=O)(C(F)(F)C(O)C(C)C)NC1CCCN(C(c2c(CC)n(C)nc2)=O)CC1 c1(C(=O)NCCNC(C(C)C(C)c2ccc(F)cc2)=O)cccc2nc(O)oc12 c1(C(N(C2CCN(C(c3cnc(CC)[nH]3)=O)C2)C2CC2)=O)cccc2oncc12 Cn1cc2ccc(C(N3CC(F)(C(=O)Nc4c(O)cccc4O)C3)=O)cc2n1 Cc1ccc(C)c(CC(N2C(C(=O)NC3CCC(C#N)CC3)CC3CC23)=O)c1 C1(C(N(C)CC2CCCN(C(c3c(OC)noc3C)=O)C2)=O)CCCCN1N=O N1(C(C2CC3(C(OC)C3)C2)=O)CC2(C1)CN(C(C1(CC(C)C)CCC1)=O)C2 c1(C(C)CNC(=O)NC2(c3cc(Cl)cc(Cl)c3)CCCCC2)nc2ccccc2o1 CC1(C)C(CNC(=O)COc2ccon2)CCN1C(=O)CCC(N)=O N1(C(CCn2c(CC)ncc2)=O)CC2CCC(C1)N(C(c1ncc(C)cn1)=O)C2 C(=O)(C1CCCc2nc[nH]c21)N(CCCNC(c1c(C)ccc(O)c1)=O)C(C)C N1(C(CS(=O)(=O)NC)=O)CC(C)N(C(=O)CCc2cscn2)CC1C c1(C(=O)NC2(C3CN(C(CCOCC#C)=O)C3)CC2)cncc2nnn(C)c12 C(C1CCC(=O)O1)=CCN1CCC(C2(C)N=N2)C1 CC1COC2(C1)CN(C(C1(CCNC(=O)CC3CSCCO3)CCCC1)=O)C2 c1(C(=O)NC(C(C)C)CCN(C(=O)C(C)CN(C)C)C)cccc2nn(C)nc12 C(=O)(C(C)CCCC(C)=O)N1CCC(CC#C)(C(=O)N(C2CCCN(C)C2)C)C1 CCC(C(=O)N1CCOCC1CNC(c1c[nH]nc1OCC(F)F)=O)C(C)C Cc1nc2cncc(C(N3CCC(CNC(=O)C4=CCSC4)C34CC4)=O)c2[nH]1 N1(C(CC(C)(F)F)=O)Cc2ccnn2CC(NC(=O)COCc2ccccn2)C1 C(CN=c1[nH]nc(C2CC2)o1)NC(C1N(C(N)=O)CCCC1)=O C(=O)(C(C)(C)C(F)F)N(CC(C)(C)NC(=O)CC1CC(C)(C)CCO1)C1CC1 c1(N2CC(CNC(C)=O)OCC2)nc2cc[nH]c2c(=NCCc2ccccn2)[nH]1 c1(C(=O)NCC2(CO)C(C=C)C2)cc(CNC(c2ccc(C)s2)=O)nn1C c1(C(N(CC(C)O)CCNC(C=CCCC(C)C)=O)=O)cc2sccc2[nH]1 CCCCC(CC(=O)NCCOc1cccnc1)OC(=O)C(O)C1CC1 CC(CNC(=O)CCC1CC1(Cl)Cl)(C1CCC1)NC(=O)CNC(c1ccsc1)=O C1(NC(Cc2ccc(C)s2)=O)CCCCC1NC(c1c(C2CC2)cnn1C)=O c1(C(=O)NC(C)CNC(c2cn(CC(N)=O)nn2)=O)cc2cn[nH]c2cn1 C#CCC(C)(CC)C(=O)NCCC(C)(C)NC(c1nc(C)n(-c2nc[nH]n2)n1)=O Cc1cccc(CN(C(=O)C(CCN(C)C)NC(=O)C(C(C)O)N(C)C)C)n1 N1(C(c2cc(C(C)(C)C)n[nH]2)=O)CCN(C(c2ccnc(O)c2)=O)C2(CCC2)C1 c1(C(=O)NC2CCC(N(C(CN(CC)CC)=O)C)C2)ccncc1C(F)F c1(C(=O)NCC(CNC(=O)CCc2ccncn2)F)c(O)cc(F)cc1F C1(N(C(C#CC(C)C)=O)C)CCN(C(=O)CCc2cccs2)CC1C c1(OC)ccc(CCC(=O)NCC2CCCC2NC(=O)Cc2cnns2)cc1O C=CC1COCC1NC(=O)C(=O)OC(=O)CC1CC2(CC2)C1 c12ccc(cc1)CCc1cn-2nn1.CC1C(=O)NCCO1.C(C)(C)(C)OC(N)=O N1(C(C(C)(C)O)=O)CCC2(CC(NC(c3ccnc(C(F)F)c3)=O)CO2)C1 c1(C(=O)OC(C)Cc2c(F)cccc2Cl)cc2n(n1)CCCCC2=O N1(C(C(CCC)NC(c2cc(OC)no2)=O)=O)CCCC(C)(COC)CC1 CS(=O)(=O)c1coc(CNC(C2CCN(CC(O)C(F)(F)F)CC2)=O)c1 Cn1ncnc1CCCNC(=O)CCC1CCN(C(C2CCC3CC23)=O)C1 Cc1cc2c(Br)ccc(C(=O)NC3(CF)CCN(C(=O)C(C)O)C3)c2o1 N1(C(C2N(C(c3cnc(Cl)s3)=O)CCN(C)C2)=O)CCOCC12CC2 N1(C(C2C(CCC)CCC2)=O)CCC2(CC1)CC(NC(=O)CC(C)C(F)F)CO2 CC1(CNC(=O)CCc2ccsc2)CCN(C(C2(CO)CCOCC2)=O)C1 C(=O)(C1CCCc2nn[nH]c21)NCC(CO)NC(C=Cc1c(C)cccc1)=O N1(C(COc2cccc(C)c2)=O)CC2(CC(NC(=O)CCC[N+](=O)[O-])CO2)C1 C1(NC(C=C(CCC)C)=O)CN(C(c2cnoc2-c2ccccc2)=O)CCC1O CC1CCC(NC(=O)CCCn2cncn2)CN1C(=O)C=CC(C)(C)C c1(OC)ccc2c(C(=O)NCC34CC(NC(=O)CC(C)CF)(C3)C4)cnn2c1 Cn1cc(CC(=O)NC2CCC2CNC(=O)CCc2ccc(F)nc2)c(Cl)n1 C(C1=CCCOC1)N(C(CCN(C(CNC(C1C(C)C1)=O)=O)C1CC1)=O)C C1(C=O)(CNC(=O)CCOC2CN(N3CCOCC3)C2)CC2(CC2)C1 CC1(CNC(C2(NC(C3CC3C(N)=O)=O)CCSC2)=O)C=CCCC1 Cc1c(CC(N2CCC(NC(=O)COCCOc3ccccc3)C2)=O)ncn1C C1(C(=O)NCCCC2(NC(CCc3cn(C)nn3)=O)CC2)CCC2(CC1)CC2 N1(C(C(CO)NC(c2nc(C)n(C)c2)=O)=O)CC2CC(N(C)C)C(C2)C1 Fc1ccc2c(c1)C1C(NC3(c4nnnn4C4CCCC4)CCSC3)C21 c1(C(N2C(CNC(c3n(CCC)ccc3)=O)CC2)=O)ccccc1N1CCCC1 c1(C(=O)NC(CC=C)CNC(C)=O)ccc(OC)c(S(C)(=O)=O)c1 CC1CC(NC(C2(CO)CCCC2)=O)CCN1C(=O)CC1CCS(=O)(=O)C1 c1(C(=O)NC2(C)CN(C(C(COC)COC)=O)C2)cc2cc(Cl)ccc2nc1C c1(CN2C(C(=O)NC(c3ccncc3)C)CNCC2)c(O)cccc1[N+](=O)[O-] c1(-c2c(C)nccc2)ccc(C(=O)N(C(C)(C)C)CC#N)c(Cl)c1Cl c1(CC(N2CCCC(CNC(C3CC3F)=O)C2)=O)coc2cc(Cl)ccc12 C(=O)(CCC(C)(F)F)NC(CNC(CC1N(C(C)=O)CCCC1)=O)(C)CO c1(NC2(C(=O)NC3CC(COC)C3)CCCOC2)ccc(F)cc1[N+](=O)[O-] C1(C(N2CCC(CCC)C2)=O)CC2CN(C(=O)C(C)(C)OC)CC2C1 N1(C(C(C=C)(C)CCOC)=O)CCC2(CCC2NC(c2ccc(O)nn2)=O)CC1 C(=O)(CCCC(F)(F)CO)N1CCCCC(NC(CN2CCP(C)(=O)CC2)=O)C1 c1(CC(C(=O)NC2C(CNC(C=C(COC)C)=O)C2)OC)ccc(C)cc1 CC1=C(C)CC(C)(C(=O)NCCCN(c2nccc(C(C)(C)C)n2)C)CC1 c1(CCC)ncc(C(=O)NC2CC2NC(C2CC(O)C2)=O)s1 N1(C(c2c(SCC)ncs2)=O)CC2CCCC2(NC(=O)C2=CCN(C(=O)OC)C2)C1 c1(C(=O)NCC2(C)CCN(C(C=C3CCC(C)C3)=O)C2)cc2c(s1)CN(C)CC2 CCC(C)(C)C(=O)N1CCCC1CN(C(=O)C(=O)N(C)C)C N1(C(C=CC(=O)OCCCC)=O)CC(NC(=O)C(C)CC#N)CC(O)C1 C(C)(C(C)CC)N(C(c1nncn1CC(C)C)C(=O)NC)C.CS C1(C(C)CNC(=O)CCC2CNC(=O)N2)CCN(C(c2cn(C)cn2)=O)CC1 N1(C(CCCNC(=O)C2=COCCC2)=O)CCCN(C=O)CC1 c1(CC(N2CCC(N(C(C(CC)O)=O)C)C2)=O)coc2ccc3ccccc3c12 S(=O)(=O)(c1ccc(NC(C)C2CC2)nc1)N1C(CCNC(C)=O)CCCC1 CCC(C)(CO)C(=O)NC1CCC(CC(N2CCOCC2CCO)=O)CC1 N1(C(C(C(C)NC(=O)CN2CCNC(=O)C2)C)=O)CC2(CCCCC2)C1 CC1CCCC1C(=O)NCc1c[nH]nc1C1CCN(C(=O)CN(C)C(N)=O)C1 C1(C(=O)NCCn2cc(Br)nn2)C2CC3C1C3C2F C(=O)(CCCCC(=O)OC)N1CCC(NC(C2(CC)COC2)=O)C1 C1(NC(=O)CC2CCCC2(F)F)CN(C(=O)C2=COCCO2)C2(CCCC2)C1 N1(C(C(C2CCOC2)OC)C(=O)NC2CC2)CC2CN(C(C)=O)CC2(C)C1 C1(=O)NNC(=O)CNC(=O)C2CC1C2.C12(CSC)CC(OC(C)=O)(C1)C2 C(CC1=CCCCC1)N(C(c1cc(SC)oc1)=O)C.C12CCCCC1C(=O)NC2 N1(C(C#CC(C)C)=O)CCCC12CCN(C(c1ccn3nncc3c1)=O)C2 C1(NC(C=CC)=O)CC(F)(CNC(C23CCCC2C3)=O)C1 Cn1c(Cl)c(C(N2CCC3CCC(NCC(O)CO)C2C3)=O)c2ccccc12 C1(C(N(C2CCN(C(c3cncc(SC)c3)=O)CC2)C)=O)CC(C)(C)CN1C Cc1cc(C(=O)N(C)CC2CCN(C(c3nocc3C)=O)CC2C)cc(C)n1 C1(OC)CN(C(=O)Cc2cscn2)C(C)(CNC(=O)Cn2cncn2)C1 N1(C(=O)CONC(c2ccc(O)nc2)=O)CC2C3CCC(C3)C2C1 C1(N(CCC)C(c2ccccc2)=O)CCN(CC#N)CC1.C(C(C)(O)C(C)C)S CCCC(C)(C)CC(=O)N1CCC2(CC2)CC1C(=O)NC1(C2CCC2)CC1 Clc1ccc(OCCNCCc2csc(-c3ccccc3)n2)cn1 N1(C(C(CCC)O)=O)CC2CC(C1)CN(C(C1(C3CCCO3)CCC1)=O)C2 c1(C(=O)NC2(CC=C)CCN(C(C3CCCCS3)=O)C2)ccc(N=[N+]=[N-])cc1 CC1(C#N)CCCN(C(=NCc2nc3c(s2)CCC3)NCC2CCCCO2)C1 C1(C(=O)NC(CCCNC(C=C(CCC)C)=O)C)CCC(C(=O)N(C)C)CC1 C1(CC(N2CCC(F)(CNC(CC3(C=C)CC3)=O)C2)=O)CN2CCC1CC2 C(C(C(C)C(C)C)NC(=O)CN1CCC(F)(F)C1)NC(c1c(C)cccn1)=O N1(C(C(CC)OC)=O)CC2CC(C(=O)NC3(COC)CCCC3)C(C2)C1 N1(C(C2CCSCC2)C(=O)NC)CCN(C2CCN(C)CC2)CC1 N1(C(C2CN(CC)C(=O)C2)=O)CC2CCCN(C(C3CCNC3=O)=O)C2C1 c1(C(=O)NCCC(CNC(C2(CC)CC2)=O)(C)C)ccc(F)c(F)c1N C1(NC(CCCOc2cccc(C)c2)=O)CN(c2ccnc(Cl)n2)CC(C)(C)C1 C1(C(N2C(CCCC)C=CC2)=O)CCN(c2nc[nH]n2)CC1 C(=O)(C(C)(CC)C(=O)NC1CN(C(=O)C(C)(C)OC)CC1C(F)(F)F)OCC CC1C(C(=O)N2CC(NC(c3ccc(F)cc3F)=O)CC2(C)C)=NOC1C C1(CNC(CP(C)(C)=O)=O)CCC2(CO1)CC(NC(C1CC(O)C1)=O)C2 c1(C(N(CCCOC)CCNC(=O)CSC2CCCO2)=O)ccccc1C C(C(O)C(=O)NC(C1CCCCC1)C)NC(C(F)=C(C)C)=O C1(C)(C(=O)NC2(CNC(C3C(C)CCCC3)=O)CCC2)CCC2(CC1)OCCO2 N1(C(c2cc(C)c(Cl)cc2)=O)CC2CN(C(=O)C=C3CCN(C)CC3)CC2(C)C1 N(C(=NCCc1ccccn1)NCc1ccc(C(C)C)cc1F)C(COC)C1CC1 N1(C(c2cc(Cl)nc(Cl)c2F)C(=O)NC(C(=O)OC)C)CCCN2CCCC2C1 N1(CCC=CC)CCC(=O)N(Cc2cccc(Cl)c2O)C1=O C(c1ccc(S(=O)(=O)N2CCOCC2)cc1)=CC(=O)NCc1cccc(C)c1O n1(CC)cc(C(=O)NC2CC(NC(=O)Cc3cc(C)nn3C)C2)c(C2CC2)n1 C12(C(=O)NCc3cc(C)[nH]n3)CCCC1CCN2C(c1cc2ncccc2[nH]1)=O C(=O)(C(C)CC(C)CC)N1CCC(c2c(CNC(CSCC=C)=O)cccc2)C1 CCC(CC)(CO)C(=O)NC1CCN(C(c2cccc(C3(C)CC3)c2)=O)CC1F N1(C(c2c(C)ccnn2)=O)CCC(C(N2CC3CC=CC2C3)=O)C(C)(C)C1 c1(C(=O)NCC2N(C(c3c[nH]c(=NC)s3)=O)CCCC2)ccccc1S(C)(=O)=O c1(CCOCCCNC(c2cccc(Cl)c2)(C)CO)cccc(F)c1 N(C1CN(C(=O)CCS(C)=O)CCc2ccccc21)C(c1cnc(C)nc1)=O N1(C(C=CC(=O)OCC)=O)CCCC1CCCNC(C)=O.C1CCC(=O)N1 N1(C(c2c(CC)nco2)=O)CC2CC(C1)N2C(C1COCC(C)O1)=O Cc1cc(=O)ccn1CC(=O)NC1CC2CC(NC(=O)CC(C)F)C1C2 c1(C(=O)NC(c2cccc(OCC)c2)COC)c(Br)nc2n1CCOC2 N1(C(CC2(NC(C)=O)CC2)=O)CCCC(CNC(=O)Cn2ccc(C)n2)C1 c1(C(N2CC(OCC(=O)NCCOC3CCC3)C2)=O)sc(F)cc1Cl C(=O)(CCN=[N+]=[N-])NC(C(=O)N(C(C#C)C)C)CC1CC1 Cc1ccc2nc(C(=O)NC3CCCC34CCN(C(=O)CC3CCC3)C4)cn2c1 CC(CCC(C)(C)C)C(=O)N(C)CC1(NC(=O)C2=CSCS2)CC1 Cc1cnn2c(NC(=O)COc3ccc(O)c([N+](=O)[O-])c3)cc(Cl)nc12 c1(C(=O)NC2CN(C(c3c(C)cc(C)nc3)=O)C3C2C3)ccc2c(c1)COC2=O CCC1=C(C(=O)N2CCC(C(=O)NOCC3CC3)C2(C)C)CCCO1 N1(C(CC2CCC(NC(c3c(CC)n[nH]c3)=O)C2)=O)CC2CCCC1C2 n1(CC)cncc1CNC(C1(CCNC(=O)C=Cc2ccc[nH]2)CC1)=O C1(NC(c2cnc(NC(C)=O)o2)=O)CN(C(=O)CC2CSCCS2)CC1F N1(C(C2C3CN(C(C(C(C)(F)F)F)=O)C2C3)=O)CC2(CCC(=O)NC2)C1 c1(C(=O)OC)ccc(N)c(SC2(c3noc(CN(C)C)n3)CC=CCC2)c1 N1(C(CCC2CCCN(C)C2)=O)CC2(CCCC2NC(=O)CCSC(F)(F)F)C1 N1(C(C=CSC)=O)CC(C)CN(C(c2ccc([N+](=O)[O-])c(N(C)C)c2)=O)CC1C C(=O)(C(CC(F)(F)F)N(CC(O)CN(C(=O)COCC(C)C)C)C)NC N1(CCNC(=O)Cc2cnc[nH]2)CCN(C(C2CC2C(F)(F)F)=O)CC1 CC(CCNC(=O)C(CNC(=O)CC1CC(=O)C1)C(C)(C)C)CC(C)(C)C C1(C(N2CC(CCCCNC(Cc3cn(C)nc3)=O)C2)=O)CCOC(=O)CC1 C1(NC(C(C(C)C)F)=O)CCN(C(c2cnns2)=O)C12CCC2 c1(OC)cc(C(=O)NCC2C3CN(C(C4(C)CC5C=CC4C5)=O)CC23)ccc1F C(=O)(C1CCCn2ncnc21)NC1CCCCN(C(c2c[nH]c(=NCC)s2)=O)C1 CCC1=NOC(CCNC(C2(CC)CCN(C(C3CC(C)(C)CO3)=O)C2)=O)C1 C1(CC(N2CC(CNC(CC)=O)N(C)CC2)=O)Cc2cc(C(F)(F)F)ccc2O1 C1(CC#C)(C(=O)N(CCCNC(=O)CC2CC2(Cl)Cl)C2CC2)CCOC1 c1(C(=O)NCCCN(c2nncs2)CC)ccccc1C c1(C(=O)NC(CC2CCC2)C(=O)NCCCO)ccc(SC(F)F)cc1 C12(CNC(C3N(C(C)=O)C(=O)CC3)=O)CCC(C1)N(C(C1CC1(C)C)=O)C2 C(Cc1cnc[nH]1)(C(=O)NCCC(C)O)NC(C=C(COC)C)=O CC1CC(NC(c2ncoc2-c2ccon2)=O)CN1C(=O)C=Cc1ccnn1C c1(NC(CC#C)=O)ccc2ccnc(NC(c3cc4cnccc4[nH]3)=O)c2c1 c1(C(N2CC(Cn3cc(C4CC=CCC4)nn3)C2)=O)ccc(O)cc1 N1(C(C(CC)OC2CCCC2)=O)CC(CNC(C2CC(n3cnnc3)C2)=O)C(O)C1 N1(C(C(C)OCC(C)C)=O)CCC(CCC(=O)N(C)CCCC=C)C1.C(C)N CC(C)C(C)(CNC(C1OCCC1C)=O)NC(c1cn(CC(F)(F)F)nn1)=O c1(C(N2C(CNC(CC(=O)NCC)=O)CC3(CC3)C2)=O)cc(C)c2c(c1)CCC2 c1(C(=O)NCC2(NC(C3C=CCCN3OC)=O)CC2)ccc(C)nc1C c1(C(N2CC(NC(CCCCSC)=O)C(F)C2)=O)cc(C)nc(O)n1 c1(CCC(=O)NCCOCCNC(CC(=O)N(C)C)=O)ccc(C(N)=O)nc1 C1(OC)CC2CC(c3nnnn3C3CC4(CC4)C3)(NC34CC(CO)(C3)C4)C2C1 N1(C(c2n(C)ccn2)=O)CCc2nc(CNC(C3CC3C3CC3)=O)sc2C1 C(=O)(C1=CCCN(C(=O)CC2(CSC)CC2)C1)N(C(C=C)C1CC1)C c1(C=O)cc(C)ccc1C.c1(SC)cccc(-c2noc(CNCC(N)=O)n2)c1 c1(C(N2CC(CN(C)C(c3cccc(OCCF)c3)=O)C2)=O)cnnc(O)c1 N1(C(C2CC(NCc3c(C)cccc3)C2)=O)CCCC2CCCCC12 N1(C(C2C(CC)OCC2)=O)CCC2(CC1)CC(NC(c1cncnc1)=O)CCO2 c1(CC(=O)N(CCOC)CCNC(c2ccc(Br)o2)=O)c[nH]c(=N)nc1O C(=O)(C(COC)CC(C)C)N1CC(CCOC)(C(=O)NCC(=O)OC)C1 CC1CN(C(c2ccco2)=O)CCC1CNC(=O)CCc1ccc(C(F)F)cc1 c1(CO)ccccc1-c1ccc(CN2CCN(CC3CC3=C)CC2)cc1 C1(N(C(CN2CCN(C(c3c(CC)noc3C)=O)CC2)=O)C)CC2CCC1CC2 CC1CCC(=CC(=O)NCCCC(C)NC(c2ccn(C3CCC3)n2)=O)CC1 C1(C(=O)NCCNC(COCC(=O)OC)=O)CC(C)=NO1 c1(C(N2CC(CC)N(Cc3ccc(O)c(O)c3)CC2)=O)cc(Cl)ccc1[N+](=O)[O-] N1(C(C(C)(C)F)=O)CCC(F)(F)C(CNC(C2(CC3CCCC3)CCCC2)=O)C1 C1(C)(CC)C=C(C(=O)NC2(C(=O)NCC(O)CC3CCC3)CCCCC2)C1 C1(C(=O)NCC(CNC(C2(NC(C)=O)CCCC2)=O)CO)CC=C(C)CC1 c1(C(=O)NCCNC(C2(C(=O)NCc3ccc(C)[nH]3)CCC2)=O)c(C)cnn1C N#CC1CC(C(N2CC(c3ocnc3CNC(c3ccc(C(N)=O)o3)=O)C2)=O)C1 N1(C(CNC(=O)NC)=O)CCN(C(=O)C=Cc2nc(C)co2)CC1C1CCC1 c1(CC(=O)NCCNC(CCc2scc(C)n2)=O)ccsc1S(C)(=O)=O c1(C(=O)NCc2cc(F)cc(Cl)c2)ccc(Cl)c2c(=O)cc[nH]c12 c1(NCCC(=O)NCCN(C(=O)C(C)Cn2ccnc2)CC)ccc(C)c(C)c1 C1(S(N)(=O)=O)(C(c2n(CCSC)nnn2)Nc2ccc(F)c(CO)c2)CCCC1 N1(C(c2c(CC)cc[nH]2)=O)CCC(O)(CN(C)C(c2ccnnc2O)=O)C1 N1(C(=O)OCCC(C)C)CCCC1CNC(=O)C(C)(C)c1cscn1 N1(C(C2CCC(=C)CC2)=O)CCC2(NC(c3ccc(CC)cc3)=O)CCCC12 C1(CCCNC(c2coc(O)n2)=O)CCCN1C(=O)CCCc1cccnc1 CC(C)C(O)C(F)(F)C(=O)NCCN(C(c1cnc(O)c(F)c1)=O)CC1CC1 c1(N(C)Cc2nccn2C(F)F)ccnnc1OC(F)F C1(N(C)C(=O)C2CC2)CCC(F)(CNC(C2(c3ccccc3I)CC2)=O)C1 c1(C(=O)Nc2c(CC)ccc(F)c2)cc([N+](=O)[O-])ccc1OC C=CC(C)(C)CC(=O)NCC(CCCC)NC(=O)C(F)(F)c1nccn1C N1(C(c2n(C(CC)C)ncc2)=O)CC(NC(C2CC(OCC)C2)=O)CC1C C(=O)(CS(=O)(=O)C(C)(C)C)N1CCC(C2(CO)CN(C(C(C(C)C)C)=O)C2)CC1 C12(C(=O)NC(CCOC)CNC(=O)CCc3ccn(C)c3)CC(C)(C1)OC2(C)C c1(NCc2cnc(CCC)s2)nccc(=NC(C)CS(C)=O)[nH]1 C1(CC=C)(C(=O)NCC2C(C(=O)NOCCN3CCOCC3)CC2)CC=CC1 C(C1=CCN(CCS(C)(=O)=O)CC1)N.C12(CCC1)C(=O)NC2.CCO c1(CCCC(=O)NC2CCN(CCCNC(CCC)=O)C2)ccc(C)cc1 c1(C(N2CC(N(C(=O)CC3CCC4CC34)C)C2)=O)cc2c(s1)CCC2 c1(NCCNC(N2CCCC(F)C2)=O)ncnc2[nH]cc(C3=CCS(=O)(=O)CC3)c12 NC(=O)CC(O)C(=O)N1CCCC(F)(C(N2CCC(CO)C(O)C2)=O)C1 C1(c2ccccc2)(OC(C(C=C)OC)=O)CS(=O)(=O)C1 N1(C(C(CCC)CC)=O)CCC(C2CC(NC(=O)Cc3sc(C)cc3C)C2)CC1 C12(C(=O)NC3CCC(NC(C(CCC)c4ccccc4)=O)C3)CCN(CC1)CC2 CC(CN(C)C)C(=O)NCC(C)(Cn1cccn1)NC(c1ccc(C(F)(F)F)[nH]1)=O c1(CC)ccc(CCNC(C)(CCI)c2nnnn2C2CCOC2)cc1 N(C1CCCn2ccnc21)C(C(CN=[N+]=[N-])NC(=O)CSC1CC1)=O C1(CNC(CNC(CCC)=O)=O)CCCN(C(=O)C(C)(CC2CCC2)OC)CC1 N1(C(COCC)=O)CC(NC(=O)CN2CCOCC2)CC1C.CSC C1(CC)C(C(=O)NC2CCC2(C)C)CCN1C(=O)CN(C)C(=O)OC c1(C(N2CCC(NC(c3ccc(CC)cn3)=O)C(F)C2)=O)ccn2c1CCCC2 n1(CCC)ccc(C(=O)NC2(CC(=O)NC(c3cnn(C)c3)(C)C)CCC2)n1 CCC(CC(=O)NCC(C)(C)CN(C)C(C1(F)CCCCC1)=O)SC C(=O)(C1=CCOCC1)NCC(CNC(c1cc(C2CC2)no1)=O)OC C(C)(C)(C(=O)NC(C)CN(C)C(c1cn(CCO)nn1)=O)OC.C12CC(C1)C2 Cc1ccc(Br)cc1C(=O)NCCCCCCN(C(=O)C(C)C1CCCO1)C N1(C(CC2CC(=C)C2)=O)CCC(C)=C(Br)C1 N1(C(C(CC2CN(C(C3OCCN(C)C3)=O)C2)F)=O)CCCC2CNC(=O)C12 c1(C(=O)NCCN(C)C(c2coc(C#N)c2)=O)cc(OC(F)F)cc(F)c1 C(=O)(C1=CCCSC1)NC1C(CCC)CN(C(c2c(SC)cnn2C)=O)C1 c1(C(N2CC(C(=O)Nc3cc4n(n3)CCC4)C2)=O)ccc(C(F)F)c(Cl)c1 c1(C(=O)NCC(CNC(c2cnn(C3CCC3)c2)=O)OC)cc(F)c(N)cc1F C(=O)(N=c1cc2n([nH]1)CCCC2)C1CC(C)(C)N(C(=O)CC=C(Cl)Cl)CC1 C1(CNC(C(C(CC)C)=O)=O)CCC2CN(C(=O)C(=Cc3cnn(C)c3)C)CC12 C1(O)(CNC(CSCC=C)=O)COCCN(C(c2csc(-c3ncc[nH]3)n2)=O)C1 N1(C(C2(CC#C)CCCO2)=O)C2CCC1CN(C(c1cccc(CCO)c1)=O)C2 C1(CNC(CN(CCOC)C)=O)CC(F)CN1C(=O)COCc1ccnc(O)c1 c1(CC(CO)NC(C2C(C)(C)CC=CC2)=O)ccc2ccccc2c1 C1(N(CCC(=O)NCC(C)(C)C)C(C2(COC)CC2)=O)CCCCC1.C1CC1 CN1C(=O)CCC1C(=O)NCCN(C1CCCCC1)C(=O)C=CC=C(Cl)Cl c1(CNc2cccc(-c3c(OC)cccn3)n2)cc(F)ccc1O N1(C(C(=O)NC(C(=O)OC)C)=O)CC(Cc2cccc(Br)c2)CC(C)C1 c1(C2CC(C(C)NC(=O)CCc3cnn(C)n3)C2)ccnc(C2CC2)n1 n1(CCC)nc(C(=O)N(C2CCNCC2)CC)ccc1=O C1(NC(CC2(COC)CC2)=O)CN(C(=O)C(C)(C)CC2CC2)CC1C(F)(F)F C1(C)(NC(C(C)OCCOC)=O)CCN(C(c2cccc(C3CC3)c2)=O)CC1 Cc1cnc(NC(c2ccccc2)C)nc1.C12CCCC1C(=O)NC2 Cc1cc(NC(c2nncs2)=O)ccc1NC(=O)C(C)n1cncn1 c1(C(=O)NCC(CNC(C(C)OCC)=O)OC)ccccc1NC C1(NC(C(CC)C)=O)CC12CCN(C(=O)C=Cc1cccc(CO)c1)CC2 N1(ONC(C2C(C)(C(N)=O)C2)=O)CCCC(Cn2ccc(C=O)n2)C1.CCO CCC(C)(C)CC(=O)NCCCC(C)NC(=O)C(C)C1CC1 CCCCCCCOCC.C12CN(CC1CCNC(=O)OC)C2=O c1(N(C)C)ncc2c(n1)CCC(NC(=O)C(=O)NCc1c(F)cc(F)cc1F)C2 C1(CC(=O)NC2CCC(CCNC(C3CCC(=C)CC3)=O)C2)CC2C=CC1CC2 c1(CC)oc(C(=O)N(C)CCC2CCN(C(=O)C=CC=C(C)C)CC2)cc1C N1(C(c2ccn(CCC)n2)=O)CC(NC(c2ccc([N+](=O)[O-])s2)=O)CC(F)(F)C1 C1(N(C(C2N(S(CC)(=O)=O)CCC2)=O)C)CC2CC1N(C(=O)CSC(C)C)C2 c1(CC)ccc(NC(C23CC(CO2)N(C(C2CC2(C)C)=O)C3)=O)c(C)c1 c1(OC(F)F)cc(C)ccc1C(N1CCCC(N(C)C(C2(OOC)CC2)=O)CC1)=O.C.C.O CC1CN(C(=O)C(C)(C)C2CCOCC2)CCC1Nc1ncnc(=N)[nH]1 C12(NC(C(CNC(Cc3cc(CC)no3)=O)O)=O)CCN(CC1)CC2 C=C(C)C1CCC(C)(O)C(NC(=O)NCC(O)CC(=O)OC(C)(C)C)C1 c1(C(N2CCC(N(C)C(c3cnc(O)c(Cl)c3)=O)C2)=O)ccc(C#N)cc1F CCCC(CC)C(=O)N1CCOCC1CNC(c1cnn[nH]1)=O C1(NCC2(N(C)C(C)C)CC2)CCCC1CN(C)C(c1c(OC)ccs1)=O N1(C(C(CC)=CC)=O)CCC(C)N(C(=O)Cc2ccno2)CC1 c1(C(N(C2CCN(C(c3cnn(C)c3)=O)C2)CCC)=O)n[nH]c(C2CC2)c1Br Cc1n[nH]c(=NC2CCN(C(c3cnc4oc(O)nc4c3)=O)CCC2(F)F)o1 c1(C(=O)NC2CCC(C(=O)NCC3(C(=O)OC)CCC3)C2)ccc(C)nc1Cl Cc1ccc(C(N2CCN(C)C(CNC(C3(CC(C)C)COC3)=O)C2)=O)c(O)n1 CCC(C)C(C)CNC(c1csc(CNC(c2cnn(C)c2C)=O)c1)=O c1(CNC(c2cccc(SCC(F)(F)F)c2)C)ccc(F)cc1Br C1(CNC(COCCC#C)=O)CN(C(c2cc(C(F)F)[nH]n2)=O)C2(CCC2)C1 C(=O)(CC(C)C(C)(C)C)N(CCC(=O)NCCC=CC)CCO c1(COC)cc(NC(=O)CCC(=O)N2CCCC(N3CCNCC3)C2)cc(C)n1 Cc1coc(C(=O)NCc2cccc(CNC(c3ccc(C#N)o3)=O)c2)c1C C(C1c2ccsc2CCN1C(c1cccc(F)c1)=O)NC(C12CC(C)(C1)C2)=O Cc1c[nH]nc1CNC(=O)COC1CCN(C(C2C(C)C2(F)F)=O)C1 C(c1ccc2ccccc2n1)=CC(=O)NC12C(CN(C(c3c(OC)ccs3)=O)C1)C2 c1(CN(C(=O)NC2N(C(C(=O)NC)=O)CCC2)C)ccc(Br)cc1N(C)C N1(C(C=CCN(CC)CC)=O)CC(=O)NCC1CNC(=O)Cc1ccon1 C(=O)(C1=NNC(=O)C1)NC1(C)CC(NC(c2cc(N(CCC)CCC)ccn2)=O)C1 N(C1c2ccccc2CC1NC(C12CCC(CC1)O2)=O)C(C1CC(=O)NC1)=O c1(NC(C(C)OC(COC(C2CCCC2)C)=O)=O)ccccc1C1CC1 Cc1cc(=O)n(C)cc1C(N1CC(C(N)=O)(CNC(C2(C)CCCC2C)=O)C1)=O Cc1ccc2[nH]c(C(N3CCC(C)C3CNC(=O)CC3C=CCC3)=O)cc2c1C c1(C(=O)NC2CC(NC(CC(C)C3CCCO3)=O)C2)csc2c1CCCC2 Nc1cc(C(=O)NC2(CF)CCC2)cnc1N.C12(C(=O)N)CC(CN1C1CC1)C2 N1(C(C2CC(=C)C2)=O)CCCC2(CC(NC(=O)C(C)(C)SC)CO2)C1 C1(NC(Cc2ccc(CC)cc2)=O)CC2CC(C1)N(C(C1(C)CCNC1=O)=O)C2 C1(C#N)(C(N2CCCN(C(C(=O)NC(C)C)=O)C(CO)C2)=O)CC2CCC1CC2 c1(C(=O)NCCC2CC(NC(CNC(CC)=O)=O)C2)[nH]nc2ncccc12 c1(-c2cc(C#N)c(NC(=O)Cn3ccnn3)cc2)nc2c(s1)CC(C(=O)O)CC2 CC(C)(F)CC(=O)NC1CCN(C(=O)C#CC2CC2)C1c1ccccc1 Cc1cccnc1S(=O)(=O)N1CCC(O)(Cn2ccnn2)C1 Cc1nc(C)n(CCC(=O)NC(C)CCN(C)C(C2CCCCO2)=O)n1 c1(C(C(=O)NCCN(CCC)C(c2csc(C#N)c2)=O)F)ccc(F)cc1 c1(C(N(C)CCC2CCN(C(C3CC3C#N)=O)CC2)=O)ccnc2ccccc12 CCC(C)(CNC(=O)C(n1cc(Cl)cn1)C)NC(c1ccn(C)c1)=O c1(C(=O)NCCCN(C(C2CC3CCC3C2)=O)CC)cc(C)cc([N+](=O)[O-])c1 N#Cc1ccc(C(N2CC3(CC(CC(=O)Nc4cc(Cl)ccn4)C3)C2)=O)cc1F C1(C(N(CCN(C(=O)C(F)(F)CO)C(C)C)C)=O)CC2CCCN2C(=O)N1 N1(C(C(=O)NCCN2CCCC2)=O)CCCC(CC2COC(=O)O2)C1 Cc1ncnc(C)c1CC(N1CCC(NC(C2CCOC(C(C)C)C2)=O)CC1)=O N1(C(C)=O)CCOC(Cn2cc(CNC(=O)C(C)(C)Cc3ccccc3)nn2)C1 C1(CC(N2CC(COC)(CNC(=O)C(O)CN(C)C)C2)=O)CCC(F)(F)C1 N1(C(c2cc(C)sn2)=O)CCC2(CCC2NC(C2CNC(=O)CC2(C)C)=O)CC1 N1(C(C(C)CN(C)C)=O)CCN(C(=O)C=CC2(C)CCOCC2)CC1C1CCCC1 CC1CC(NC(=O)CCC(C)(F)F)CN(C(c2cccc(C(F)F)c2F)=O)C1 N#Cc1ccccc1CCC(N1CCC(NC(=O)C=CC=CCO)C1C(F)(F)F)=O C12(CCCCC1)c1noc2n1.C(CC(F)(F)F)C1C(c2cocc2)C1 Cn1ccc(C(=O)NC2CCC2NC(C2CC(n3ccnc3)C2)=O)c1C1CCC1 C1(NC(CSC)=O)CCCC(C(=O)NC(COc2cncc(C)c2)=O)C1 c1(CC(=O)N(CCNC(=O)CC2CC=CC2)CC)ccc(O)cc1Cl c1(C(=O)NC(c2ccccc2)CC)nc(-c2ccncc2)no1 C(CCN=C1NCC(c2ccoc2)N1)c1c(F)cccc1 Cc1nc(Cl)ccc1C(=O)NC1(C)CCN(C(c2[nH]nnc2C2CC2)=O)C1 N1(C(c2cnn(C)c2N)=O)CC2CC1CC2CNC(=O)CCCCCF C1(C(=O)NC(C#C)C(C)(C)C)CCC2(CC2)N1C(=O)CS(=O)CC Cc1cc(C(N2CCC(CCNC(c3csc(Cl)n3)=O)CC2C)=O)c(N)c(F)c1 C(=O)(C(N=[N+]=[N-])C(C)C)NC(CC#C)C(=O)N1CCC(C)(O)C1 C1(CC(=O)NC(C(=O)N(CC(O)CF)C)c2ccoc2)CCOC1(C)C c1(CC(=O)NC(CN(C(C2(C(F)F)CC2)=O)CC)C)cc(C)on1 c1(C(=O)NCC2N(C(C(C)(C)c3cc[nH]n3)=O)CC2)nccnc1N c1(OC)cc(F)c([N+](=O)[O-])cc1CC1(C)CCS(=O)(=O)C1 c1(OC(C(N2CCC(C)(CNc3cc(C)ncn3)C2)=O)C)cccc(C)c1C N1(C(=O)NC(c2ccccc2F)CC)CCN(N2CCCC2)CC1C N1(C(C(CC2CC2)OC)=O)CC(C)(C(=O)NCC2CC3C=CC2C3)CC1(C)C C12(NC(CCOCCCOC)=O)CCN(C(c3cccc(Cl)c3N)=O)CCC1C2 N1(N(C)CC)CC(C)(C)CC1NC(C1CCOC1C=O)=O.c1(SC)cnn(C)c1 C(=O)(CCCCC(=O)NC(C)(C)C(=O)NCC1CCC1C)OC CCC(O)C(F)(F)C(=O)NCC(CC(=O)NC1(CCOC)CC1)C1CCC1 Cc1cc(N2CCC(CS(N)(=O)=O)C2)nc(N(CCCSC(F)F)C)n1 c1(N(C)CC2CN(c3cc(OC)nc(C)n3)C2)cc2cccnc2[nH]1 C1(NCC(N2CCCC(C(N(c3ccccc3)CC)=O)C2)=O)CCC(C)(C)CO1 N1(C(CC(C)(C)O)=O)CCC2(CCCCC2NC(c2cc(O)cc(O)n2)=O)C1 C=Cc1ccc(CNC(C2CCCN(C(=O)C=CSc3nc[nH]n3)CC2)=O)cc1 CCC(C)(C)C(C)CC(=O)NC1CCC(NC(C2CCCC3(CCC3)O2)=O)CC1 N1(C(C(c2cnn(C)c2)NC(c2ccnc(OC)n2)=O)=O)CCCC2(CCCO2)C1 CC(C(=O)N1CC(CNC(c2ccc(C3SCCCS3)cc2)=O)C1)C(F)F C(=O)(C(C)(C)CCOC)NC1C2(CC(NC(C(C=C)(F)F)=O)C2)C1 c1(NC2(c3n(C4C(OC)CCC4)nnn3)CCCSCC2)ccc(F)c(S(N)(=O)=O)c1 Cc1csc(=O)n1CC(=O)NC1CCC(C(=O)O)CC1 c1(OC)cc(CO)cc(C(=O)NCC(O)CCS(C)(=O)=O)c1OC(C)=O N1(C(c2ccc(C)cc2)=O)CC2(CCC(Nc3cc(C(C)C)nc(C)n3)CC2)C1 O=C(C1CCCn2cnnc21)NCC1C=CCN1C(c1cc([N+](=O)[O-])n[nH]1)=O C1(CC(=O)NCc2n(CC)ncn2)CCC(NC(=O)C=Cc2ccnn2C)CC1 C(=O)(CCS(=O)(=O)CC(C)C)NCCCN(C(C1CC=C(C)CC1)=O)C CCC(CC(=O)N1CC(F)CC1CC(N1CCC2(CSC2)C1)=O)CC(C)C CC1(NC(=O)CC2OCCCO2)CCC(NC(c2ccccn2)=O)C1 C1(c2cn(CCCC3(N(CCOC)C)CCC3)nn2)C(C)CCN1C(=O)OC C(CNC(=O)CCc1cc(C)no1)(CC(=O)N(C)C(C1(C)CC1)C)OC C1(C)(C(N(C(C=C)C2CC2)C)=O)CCCN(C(c2cc(C(N)=O)co2)=O)C1 c1(C(=O)NCC2C3CN(C(CSC)=O)C(C3)C2)cc(Cl)cc2cccnc12 CCN=C(NCCC(C)(C)O)N1CCC(F)(C#N)C1 S(=O)(=O)(c1c(Cl)cccc1Cl)NC(CCC(=O)O)CCc1ccccc1 N1(C(COCCCC#C)=O)CCCN(C(=O)C(C)Oc2ccc(F)c(F)c2)CC1C C1(CC)C(NC(=O)C2=COCCC2)CCCN1C(=O)CC1CC2CCC1C2 C1(CNCC(C(C)C)c2ccncc2)CC2OC1C1CC21 N1(C(CCC=CC)=O)CCC(O)(C(C)NC(=O)Cc2ccc(C)nc2)C1 C1(C)(CNC(CS(CC)=O)=O)CC(F)(F)CN1C(C1CC2(CC(=O)N2)C1)=O c1(-c2c(C)n[nH]c2)ccc(C(=O)NCC2CC2)cc1F.c1(N)ncncc1Cl N1(C(c2cc(CCC)[nH]n2)=O)CCC(NC(=O)CC(C)(C)C2CC2)C12CCC2 N1(Cc2cn(C3CC(NC(CC4CNC(=O)O4)=O)C3)nn2)CCn2cncc2C1 Cc1ccc(Cl)c(OCC(=O)NCCN(C(C2C3CC4C(C3)C24)=O)C(C)C)c1 c1(N2CC(NC(C(=O)OCC)=O)C(F)(F)C2)ccn2ncc(I)c2n1 C=CCC(C(=O)NC(CO)C(=O)NCc1ncc(CC)s1)C(C)C N1(C(CC(CCCC)NC(=O)CS(=O)(=O)CC)=O)CCC2=C(CCCC2)C1 C=Cn1nncc1C(N1CC(O)(C(F)C(=O)NCC2CCC(=O)C2)C1)=O Cn1ccc(CCC(=O)NCCOC2CCN(C(C3OCCO3)=O)C2)n1 N1(C(C(C)OCCOCC)=O)CCCN(C(c2ccccc2C(F)(F)F)=O)CC1 C(=O)(CN=c1[nH]c2c(c(=NC3CCCCC3)[nH]1)CCCC2)NCCC(=O)NCC N#CC1(CCNC(=O)CCc2ccccc2Br)CCNCC1 N1(C(CC(C)N2CCCC2=O)=O)CCC(NC(=O)CSCc2ncc[nH]2)CC1 Cc1cc(C(=O)NCCOC2CCN(C(=O)CC3(Cl)CC3(F)F)C2)cc(C)n1 C1(C(c2cn(-c3c(C(N(C)C)=O)n(C)nc3)nn2)=O)CNC(=O)C12CC2 Cc1nnccc1C(N1CC(C(=O)NCCNC(C2CC(C)(C)CO2)=O)C1)=O c1(C(CC(=O)NCCCN(C)C2CC2)NC(CCC)=O)ccc(Br)cc1 c1(C(N2CC(CCc3cn(CC(CC)CC)nn3)C2)=O)cc(C)ccc1F CC(C)C(C)CC(=O)NC1CCC(C(=O)NCC2CCCC2N(C)C)C1 N1(C(CC2CC(CC)C2)=O)CCCOC(CCNC(=O)CCc2cncs2)C1 c1(C(=O)NC2C(NC(=O)CCc3ccoc3)CC2)ccc(Br)o1 C1(C(C)NC(c2sccc2Cl)=O)CCCCN1C(c1ccc(C(F)F)nc1)=O C1(CNC(c2cc(CC)nn2C)=O)C(C)CCCN1C(c1csc(COC)n1)=O Cc1nc(CO)ncc1C(N1CCCN(C(c2cc(C(C)(C)C)no2)=O)CC1)=O c1(CC(=O)NC2CC(NC(c3c(CC)c[nH]n3)=O)C2)coc2c(F)c(F)ccc12 c1(C(=O)NC(CCNC(CC2CC(OCC)C2)=O)C)ccc(C)nc1N C(=O)(C1=CCCC1(C)C)NC(CC)=O.c12cccc(c1)CC(=O)N(C1CC1)CC2 C(=O)(C(C)CC(F)(F)F)NC(C1N(C(c2cc(C)n(C(C)(C)C)n2)=O)CCC1)C N1(C(C(C)(C)OC(C)C)=O)CCCCC(CNC(=O)NCc2ccc(Cl)cc2)C1 C1(CC(=O)NC2(CC)CC2)N(C(=O)OC(C)(C)C)CC1(C)C C(=O)(C1=C(C#N)CCC1)NC(c1sc(C)c(Br)c1)=O.C12CCN1CCCNC2=O CC(=O)CCCCCCC(=O)N1CCC2(CCOCC2C(=O)NCC(F)F)CC1 C1(NC(c2c(C)nn[nH]2)=O)CCCCC1CNC(=O)CCC(=O)NC1CCCC1 N1(C(C(CC)O)=O)CC(F)CC1C(=O)Nc1cnncc1C(N)=O C1(C(N2CC(OCC)C2)=O)CN(C(=O)CN2CCC(C)CC2)CC1C N1(C(C2CN(C(C(CC)NC(N)=O)=O)CC2C)=O)CC2CC1CN2C C1(NC(C(C)C(C)(F)F)=O)CCN(C(=O)CC(O)c2ccccc2)C12CCC2 C1(C(=O)NC2CC(CNC(C34CCCC3CC4)=O)C2)CCCN2CCCC12 N1(C(CN2C(C)CC2)=O)CCCCC(CNC(c2nn(C)nc2C(F)(F)F)=O)C1 C1(NCC2CC(C(N(c3ccccc3)C)=O)C2)(NC(C2CC(C)=NO2)=O)CCOC1 c1(C(N(OC)C2CCC2)=O)cc2ccncc2c(O)n1 C1(C(N)=O)(COC(=O)CCCc2nc(C3CCCC3)no2)CC1(F)F c1(C(=O)NCC2C(NC(COCCCC)=O)C2)ccc(CN(C)C)cc1 C1(C(=O)NCCCCN(C)C)CCOCC1NC(c1nccnc1N)=O C1(NC(CNS(N)(=O)=O)=O)C2CC(NC(c3c[nH]nc3Cl)=O)CC12 N1(C(CSCC)=O)CC=C(CC(=O)N2CCOC(CN(C)C)C2)CC1.C(=O)OC CC(CF)CC(=O)NCc1ccc(CC(C)NC(C2CC(C)(C)C2)=O)cc1 C1(C(=O)NC2(CO)CCN(C(c3cccc(CSC)c3)=O)C2)CCC2(CCC2)C1 C(CNC(c1cccc(OC(F)F)n1)=O)(C(C)(C)C)NC(C(CN(C)C)O)=O n1(CCC(=O)N(CC(C2CCC(CO)CC2)=O)C)cnc2ccccc12.CO c1(NC(C)=O)cc(C(N2CC3(CCC3NC(C3CCS(=O)(=O)N3)=O)C2)=O)cc(C)c1 CC1CCC(CNC(C2(CNC(N)=O)CCCC2)=O)CN1C(=O)CC1OCCO1 C(=O)(C#CC1CCC2(CC1)OCCO2)NC1C(CNC(C(C(CC)C)OC)=O)C1 Cc1c(C(=O)NCC2CCCC2NC(c2cn(C)nc2Br)=O)nnn1C C1(C(=O)NCC(C)(CO)NC(c2c(C)cc(CC)o2)=O)CC2(C1)CS(=O)(=O)C2 N(C1CCc2cc(CNC(C3CC(O)C3)=O)ccc21)C(c1ccc(CC)cn1)=O Nc1ccc(F)c(F)c1C(N1CCC2(CC(NC(C3CCCN3C=O)=O)C2)C1)=O C(CCCCC(=O)NCCN(C(c1ccc(CO)o1)=O)C1CC1)OC CCC(CC(C)C)C(=O)N1CCC(C(=O)NCC(n2ccnn2)C)(CC)C1 C1(CCC)COCCN1C(=O)CCN(C(=O)COC(F)(F)F)C1CC1 CCCCCC(O)C(=O)N1CCC(NC(c2nn(-c3ccccc3)nc2Br)=O)C1 C1(NC(C=Cc2ccc(CC)o2)=O)CC2CN(C(=O)C=CS(C)=O)CC2C1 n1(C(C)C)nc(C2CC2)cc1C(N1CC(NC(C2(C)CC=CCC2)=O)C(O)C1)=O c1(C(N2C(CNC(CC(C)OC)=O)CCC2)=O)cc([N+](=O)[O-])ccc1C(F)(F)F Cc1nc(C(=O)N(C2C3CN(C(C4CCN(C)C4C)=O)CC23)C)n(C)n1 c1(C(=O)NC(C2CCCOC2)C(=O)NCCCC2CC(C)C2)cc(O)cc(F)c1 N1(C(=O)Cc2cccs2)CCN(C(=O)C(F)(F)C2CC2)CC1c1cccc(F)c1 c1(N2CCCC(NC(C(=O)N(CCN(C)C)CCO)=O)C2)ccc(C)cc1C c1(C(=O)NC(C2CCCCN2C(c2nnn(C)n2)=O)C)cc2ccccn2c1 Cn1cnc2c(NCc3cccc(Br)n3)nc(=NCCCn3ccnc3)[nH]c12 c1(C(=O)NCC(CN(C)C(C2CCCN2CCCO)=O)(C)C)ccc(CO)cc1 c1(C(=O)NCC(=O)NC(C2CCCC2)C#C)cc(C)c(N)cc1F C(=O)(C1CCCn2nccc21)NCC1(OC)CN(C(=O)CC(C)(O)C2CC2)C1 CC(C(=O)NCC(C1CC1)NC(C12CC(C)(CCO1)C2)=O)C(F)(F)F C12CC(O)CN1C(=O)CCC1CCC(C1)NC2=O.C1(CC)(OC)CCC1 c1(OC)cnc(Cl)cc1C(=O)N(CCCNC(C1CC12CC2)=O)C(C)C C1(C(=O)NC(C(=O)NCC(C)CN2CCCC2)CC2CC2)CC(O)CN1C c1(CCC(=O)NC(CCOC)CNC(c2ocnc2C2CC2)=O)ccccc1Cl N1(C(c2c(C)nc(C)c(C)n2)=O)CCCC2(CCN(C(=O)CC(F)(F)Cl)C2)C1 C1(NC(Cc2n(C)ccc2)=O)CC(O)CN(C(c2cnc(O)cc2O)=O)C1 c1(C(=O)NC(COC)CC(=O)NC2C=CC(CO)C2)cc2cccnc2[nH]1 c1(C(N(CCC)CCNC(=O)C(C(C)C)n2cncn2)=O)cc(N)cc(O)c1C c1(C(=O)NCC2CCCN2C(C2CC2C2CC2)=O)cccc(-c2nc[nH]n2)c1 c1(OC)c(C(=O)NCC2CN(C(C34CC3COC4(C)C)=O)C2)occc1=O C1(C(=O)NC(CNC(C(CSC)O)=O)(C)CO)CN2CCN1CC2C C1(CNC(c2ccn(C(C)C)n2)=O)CN(C)CCN1C(=O)CCn1cc(Cl)cn1 N1(C(c2c3ncc(C)cn3nc2)=O)CCN(C)C2(CCC2)C(C)C1 N1(C(c2c(C)nc(Br)o2)=O)CCN(C(c2cc[nH]c2)=O)CC1c1ccccc1 c1(C(=O)NCC23C(C(=O)NCC4(C)CCCOC4)C2CCC3)cc(O)cc(=O)o1 c1(SCC(=O)NCC(CNC(c2cnn(C(C)C)c2N)=O)OC)ccccc1F C1(CCOC)(NC(C2(C)CCNC2=O)=O)CCN(C(=O)CNS(N)(=O)=O)CC1 N1(C(c2cnccn2)C(=O)NCCCOC)CCC2(C1)CN(C)C(=O)CO2 c1(C(N2CCC(NC(C(CCC)C)=O)C(F)C2)=O)ccc(C#N)c(F)c1 N1(C(CCCOC)=O)CCCCC(NC(=O)C=CC2CCCO2)C1 c1(SC)ccc(C)c(C(=O)NC2CCCCN(C(=O)CC3CCC4CC34)C2)c1 N1(C(C2CCC(CC)O2)=O)CC(NC(c2ncccc2OC)=O)CC2(CC2)C1 c1(C(N(CC(CNC(C2CC(SC)C2)=O)O)C)=O)cccc2[nH]ccc12 c1(C(N2C(CNC(C3C(COC)C3)=O)COCC2)=O)cnc2n1CCCCC2 C=CCC(C)(C)CC(=O)N1CCC(CC(N2CCC2C(C)O)=O)CC1 N1(C(C(n2cc(-c3ccsc3C#N)nn2)C)=O)CCOC(c2ccccc2Cl)C1 c1(CC)ccc(C(=O)NCC(C2CCN(C(C3(O)CCOC3)=O)CC2)F)cn1 c1(SC)cc(C(=O)NC2CN(C(=O)CC3CCOC3=O)CC2F)cc(Cl)c1 c1(N(C)Cc2c(C)cnn2C)nccc(=NCC2C(F)(F)C23CCC3)[nH]1 C#CCC(CC#C)C(=O)NCC1(O)CN(C(=O)CSCCC#N)C1 C12(C(N3CCC(N(CCF)C)C3)=O)CCCN1C2=O.c1(OC)cc(CO)ncn1 Cn1nccc1C=CC(=O)NCC1CC(CC(N2CCCCC2C2CCC2)=O)C1 N1(C(C(c2cccnc2)NC(CCC(=O)N(C)C)=O)=O)CC2CCCC(C1)N2C C1(C2CC2)(C(=O)NCC2(F)CC(NC(CNC(C)=O)=O)C2)CCOCC1 CC(C)C(CNC(=O)CCCN(C)C)NC(C1(C)CCCS1)=O C1(CNC(c2nc(C(N)=O)sc2)=O)C2CC1N(C(C13CCCCC1C3)=O)C2 c1(C(=O)NCC2CCN2C(C2CC23CC3(F)F)=O)cccc2c3c([nH]c12)CCC3 N1(C(C(CO)N(C)C)=O)CCN(C(c2cc(C3CCCCC3)no2)=O)C(CO)C1 c1(CNC(C2CCCCCC2)CC)cnc2ccccn12 c1(C(=O)NC2CCC(NC(c3c(C)nc(O)s3)=O)CC2)cnc(O)c(F)c1 C1(NC(C=C(C)C(C)C)=O)CC(O)CN(C(=O)Cc2cnn(C3CC3(F)F)c2)C1 c1(OC)cccc(C=CC(N2CC(N(C)C(c3ccn(C)c3)=O)C(C)(C)C2)=O)c1 C1(NC(C(CNC(c2n(CC)nc(C)c2)=O)C(C)C)=O)CCC(=O)NC1(C)C C(=O)(C1CCCn2cc(C(C)(C)C)nc21)NCCCN(S(C)(=O)=O)C C(=O)(CCCC(=O)NCCCCCNC(c1nc(C2CC2)cs1)=O)OCC C1(CNc2ccc(COC)cc2)(NC(=O)COCC(=O)OC)CC2CCC1C2 C1(=CC(N2CC(C(=O)OC)(NC)C2)=O)CCOc2ccc(OC)cc21 N1(C(COCCCC)=O)CCCC(NC(=O)CCC2CCCC(=O)N2)CCC1 CC(C)C1=NOC(C(N2CC(F)(F)CC2CCNC(=O)C=Cc2ccsc2)=O)C1 O=C(O)CC(CNC(c1cnn(Cc2ccccn2)c1)=O)CN1CCOC1=O c1(C(=O)NC2(C)CCN(C(c3cnccn3)C)C2)cccc2occc12 C1(NC(c2ccc[nH]2)=O)CN(C(c2cnn(CC3CCCC3)c2)=O)CCC1O CC1(C)CC(F)(F)CCC1C(N1CCN(C(c2cccc(Cl)c2)=O)C2CCC12)=O c1(OC)cc(C)c(CC(N2CC3(CCCN3C(c3ccoc3C)=O)C2)=O)c(C)c1 c1(C(=O)NC(CC=C)CNC(=O)C(C)N(C)C)ccc(C(F)F)cc1F c1(CC)cc(C(=O)NCC2COCCN(C(=O)CS(C)(=O)=O)C2)cc(Cl)c1 N(C1CCc2c(C)cccc21)C(=O)Nc1n(C)nc(C)c1Cl C1(OC)CCCC(CC(=O)N(CCCCCNC(c2c[nH]c(=N)s2)=O)C)C1 CC(O)C(C(N)=O)NC(c1ccc(CNC(C2(C)CCCC2)=O)cn1)=O N1(C(CCSCC)=O)CCC2CN(C(=O)C3=NOC(CC4(O)COC4)C3)C2C1 CC1CC(c2cn(-c3ncc(Br)s3)nn2)CCN1C(c1cc(Cl)sc1Cl)=O CC1CN(C(=O)COC2CC=CC2)CCC1CNC(=O)COc1ccccc1 C1(C(C)NC(C2CC2(Cl)Cl)=O)CCN(C(c2ncnn2C(C)(C)C)=O)CC1 c1(C(N(CCCNC(C2N(C)CC(C)(C)C2)=O)C)=O)nc2cncnc2nc1O C1(OC)CN(C(=O)CCC2CCCOC2)CC1NC(=O)CCc1cc(C)cs1 N1(CC(C)NC(C2C(C)C2(F)F)=O)CCN(C(C2CC3C=CC2C3)=O)CC1 C(=O)(CC1COc2cc(OC)ccc21)NCCC(C)(C)NC(C1C(COC)C1)=O Cc1ccc(C)c(OCCC(N2CC3(NC(=O)CC4CC(CF)C4)CC2C3)=O)c1 C1(C)(C(N2CC(OCCNC(CC(CC)C3CC3)=O)C2)=O)CC2C=CC1C2 N1(C(C2CC(=O)CC(=O)C2)=O)C2COCC1CC(NC(=O)C=Cc1cc[nH]n1)C2 C12(C(=O)NCc3ccn(C)c3)CCC(CC1)C2 c1(N)cccc2c1NCC2.c1(COCCC(=O)NC(=O)NC2CC2)ccccc1Br c1(C(N2CCC(NC(=O)CCC3CCC3)C23CC3)=O)nc(Br)n2ccccc12 C1(NC(C(CC)C(C)C)=O)CN(C(=O)C(C)(C)C2CCCC2)CC(F)(F)C1 C1(C(=O)NC2C3C4CCC(C4)C23)CCc2nnc(C3CC3)n2C1 N1(C(C(C)OCCC=C)=O)CC2CC1C2CNC(c1ccc(C(C)(C)C)nc1)=O N1(C(CCC2(C)N=N2)=O)CCC(NC(=O)Cc2ccn(CC(F)(F)F)n2)C1 Cn1cc(C(N2CC=CC2CNC(=O)CCN2CCOCC2)=O)cn1 C1(c2nnnn2CCCSC)(NCc2c(C)ncs2)CCCC(C2CCOCC2)C1 c1(NCCCN)cccc(Cl)c1.C1C(O)CN(CC(C)(C)C)N1C N1(C(CNC(C(CC)C)=O)=O)CCCCC(NC(c2cnn(CCO)c2C)=O)C1 CN1C(=O)C(NC(C2CC23CC(NC(=O)CSC(F)(F)F)C3)=O)CC1(C)C C(c1cc(F)c(O)c(F)c1)=CC(=O)NCC(F)CNC(c1cnnc(O)c1)=O c1(NC(C)=O)ccc(C(=O)NC2CC(C(=O)NC3(COC)CCC3)C2(C)C)nc1 N1(C(CCc2ccc(C)o2)=O)CCC(NC(C2CCN2S(C)(=O)=O)=O)C(O)C1 N1(C(CCC=C)C(=O)NCCC#N)Cc2ccc([N+](=O)[O-])cc2C1 N1(C(C2CC(CCC)OCC2)=O)CCC(C)N(C(C2CCC(F)(F)CC2)=O)CC1 C12(C(N(CC(COCC)O)C)=O)CC(CO)(CN1C(C1CNC(=O)N1)=O)C2 c1(C(N2CCCC(CCCCNC(C=CSC)=O)C2)=O)ccc2nn[nH]c2n1 c1(C(N2CCC(CC(C)C)C2)=O)cn2c(n1)CCN(C1CCC(C)(C)C1)CC2 N(C(=NCCc1cccc(C)n1)NC1CCCCC1)CC(CC#C)C1CC1 N1(c2ncc(C)cn2)CC2CCC(NC(C3CCCN3N=O)=O)CC2C1 c1(CC(=O)NCCOCCNC(=O)Cc2ccns2)ccc([N+](=O)[O-])cc1Cl C1(=O)CC(C(F)F)N1.c1(C(C2CC2)NC(C2(COC)CC2)=O)ccccc1 C(=O)(C(C)(O)Cc1ccccc1)NCC(CNC(C1(OCC)CCCC1)=O)C c1(OC)ccc(C(C(=O)NC2(C)CC2)N(C(C)(C)CC(F)(F)F)C)cc1SC C1(COC)(CNC(=O)CC(c2c(C)noc2C)C)CCCN1C(=O)C(C)C1CC1 C1(NC(c2ccc(C#C)cn2)=O)CC2CCCC(C1)N2C(=O)Cc1ccoc1C Cc1ccncc1C=CC(=O)NC1CCC(CNC(c2cc([N+](=O)[O-])n[nH]2)=O)C1 C#Cc1ccc(C(=O)NC2(CF)CCN(C(=O)CNS(C)(=O)=O)C2)c(F)c1 CC1CN(C(=O)C(C)N(C)C)CC1CC(=O)NC(CO)C1(C)CC1 C1(C(=O)N(C2CCN(CCOC)C2)C2CC2)CN(C(=O)CN2CCCC2)CC12CC2 Cc1occ(C(F)(F)F)c1C(=O)NC1CCCC(C(=O)N(C)CCN(C)C)C1 c1(C(N(CC(C)NC(C=CCC)=O)C)=O)ncnc(C)c1C N1(C(c2c(C)n[nH]c2)C(=O)NCC2CCOCC2)CCOC(CF)C1 c1(C(=O)NC(COC(C)=O)(C)C)nn(C)c(=O)cc1C.C12(CC1)C(=O)NC2=O N1(C(C(COC)(C)OC)=O)CCCCC(NC(C2CC(N3CCCC3)C2)=O)C1 C1(CNC(CC(=O)NCC#C)=O)CC2(CCN(C(c3sccc3Cl)=O)C2)CO1 Cc1c(NCc2conc2C(F)(F)F)ncc2ccccc12 N1(C(C2N(CCC)CCC2)=O)CCCCC1CC(O)C(F)(F)F c1(C(=O)NC2(C)CN(C(C3(CO)CC(C)(C)C3)=O)C2)cc2ccsc2s1 S(=O)(=O)(CCC(=O)NCC1CCN1C(c1cnc(C(F)(F)F)c(F)c1)=O)NC c1(CNC2C(C(=O)NCc3cc(OC)ncc3)CCC2)ccc(Br)cc1O c1(C(=O)NC2(CF)CCN(C(c3c(C)n[nH]c3C)=O)C2)ncc2[nH]ncc2n1 c1(C(=O)NC2(CO)CCN(C(c3c(CC)oc(C)c3)=O)C2)ccc(Cl)c(OC)c1 C1(NC(Cc2cccc(OC)n2)=O)CCC12CCN(C(C1CCC(F)CC1)=O)CC2 Cc1sccc1CC(=O)NCC(F)CNC(=O)C(F)(F)C1CCOCC1 C1(CC)CN(C(=O)CC2CCN(C)C2=O)CCN1C(=O)Cc1ccc(OC)nc1 C1(CNC(c2ccc(C)nc2O)=O)CC12CCN(C(C1(CO)CCCO1)=O)CC2 c1(OC(C)(C)C)cc(C(=O)NCC23CCC(C2)N(C(=O)C(N)=O)C3)ccc1C O=C1NC(C(=O)NCC2(CO)CCC2)C2CCC12.n12cc(nn1)C1(CCC1)C2 C12(CNC(C(C)Nc3cccnc3)=O)CC(CN1C(=O)CSc1cccnc1)C2 C(C(C)(C)C(=O)NC1CC2(C1)CC2NC(=O)CCNS(=O)(=O)C(F)(F)F)OC c1(CC(=O)NCC(CN(C)C(C2CC(=C(F)F)C2)=O)(C)C)cnc2n1CCCC2C C1(NC(c2nc(CCC)oc2)=O)CN(C(C2(N3CCCC3)CC2)=O)C(C)(C)C1 N1(C(CC2CC(OC)C2)=O)CCC2(CCCCC2NC(c2cscc2C(N)=O)=O)C1 N1(C(C2(CC)COC2)=O)CCCCC1CC(=O)NCC(F)CO c1(OC)cc(O)ncc1C(=O)NCCN(C(=O)CCc1nc(=N)[nH][nH]1)C1CC1 C1(C#N)(C(=O)NC2(C)CCN(C(C3CCCS3)=O)C2)CC2CCC1CC2 C(CC(C(=O)NC(C)(C)CN(C(=O)CCc1ccco1)C)OC)OC C12(NC(c3cnc(C(C)C)[nH]3)=O)CCN(C(C3(C4CC4)CC3)=O)CCC1C2 C1(Cc2c(NC(=O)NC(c3ccc(F)cc3)C)ccs2)CCCCCC1CO CC1CN(C(c2cnc(C3CCCO3)s2)=O)CCN1C(c1cc[nH]n1)=O c1(C(=O)NCC2(Cn3cc(CN)nn3)CC2)ccc(F)c(OC(F)(F)F)c1 C1(COCC=C)CCN(C(N)=O)CC1.c12ccn(n1)C(C(=O)OC)N2C c1(NC(N2CCN(c3snc(COC)n3)CC2)=O)cnc2n1CCS2 C=CCCC(C)(C)CNC(C(C)(C)C=C=C=C)c1nnnn1-c1ccccc1C N1(C(c2nc(NC(c3cc(I)ccc3F)=O)sc2)=O)Cc2ccccc2C1 N1(C(C2C3(CCN(C(C(C)(C)F)=O)CC3)C2)=O)CCc2ccncc2C1 c1(C(=O)NCC(C2CCCC2)NC(C(n2cnc(C#N)n2)C)=O)cnn(C)c1Cl CC(C)CC(C)(CNC(=O)CCOCCN(C)C)NC(C1CC1c1cccs1)=O Cc1nc(CSCC2CC3CC2C3)no1 C(=O)(CC1=NN(C)C(=O)C1)NCCC1(O)CCCN(C(C(C)SC(C)C)=O)C1 CC1CN(C(c2ccnc3ccnn23)=O)CCCN1C(C1CC=CCC1)=O N1(C(C2CCN(C(CC)=O)C2)=O)CC(NC(c2cccc[n+]2[O-])=O)C(O)C1 C1(NC(Cc2n(C)ccc2)=O)CS(=O)(=O)CC1NC(C1OCCO1)=O C(=O)(C(CC(C)C)C(C)C)NCC#CCNC(c1c(C)nc(N)cn1)=O N1(C(CC2CCN(C(C3C4(OC(C)(C)C)CC(C3)C4)=O)C2)=O)CCC(C)(O)C1 C(C)(CC(=O)N1CC(F)(CNC(C2(C)CC2(F)F)=O)C1)(C(F)F)N(C)C Brc1cnn2ccc(N3CCC(C4CCC4)CC3)nc12 N1(C(C(CCC)c2ccccc2)=O)CCCC(NC(=O)C(F)(F)COC)C1C C1(NC(C(C)NC(C)=O)=O)CCC2(CC1)CC(NC(=O)C(n1ccc(C)n1)C)C2 c1(C(=O)NCCc2c(OC)c(C)ccc2)ccc2nc(F)ccc2c1O c1(C(N2CCC(COC)(NC(=O)C=CC3CCCO3)C2)=O)ccc2nncn2c1 c1(CN2CCC(C#N)(NC(C3CCC(CCC)CC3)=O)C2)cc(C)c(Br)cc1F N1(N2CCc3ccc(Cl)cc32)CC2CCN(C)CCC2C1.C1(C=O)(CO)CCCO1 CCC(CC(=O)NC(C)C(C)(C)CO)N(C(=O)C=CC1(C)COC1)C Cc1ccc2[nH]c(C(N3CCC=C(CNC(C4CCO4)=O)C3)=O)cc2c1 CCCC(O)CC(=O)NC1CN(C(c2ccc(C3CC3)nc2)=O)CC1CCC c1(C(=O)NC(C2(O)CN(C(C(C)OC)=O)C2)C)cc2c(Br)c(F)ccc2[nH]1 C(=O)(CC(C(F)(F)F)P(C)(C)=O)NCC(CCNC(C(C)(C)CC(F)F)=O)O Cn1ncc2cc(C(=O)NCC(C)(O)CNC(c3ccc(C#N)s3)=O)sc12 c1(OC)cc(OC)cc(C(O)C(=O)NCC2COCC2NC(C)=O)c1 C(N=c1[nH]c(=NC(C)c2ccc(Br)s2)[nH]c2c1SCC2)CCC=CCCC C(c1cccc(F)c1)=CCC(=O)NC1CC(NC(C2CC2OC(C)(C)C)=O)C1 c1(C(N(CCN(C(CC=C=C)=O)C)C)=O)ccc(N2CCC(C)=N2)cc1 C1(NC(c2c(C)scn2)=O)CN(C(=O)C=CC(C)(C)C)CCC1c1ccccc1 N1(C(CC2C(C(=O)NC)C2)=O)CCCN(C=O)CC1.C1(C(=O)OC)(O)CC1 N1(C(c2ccc(OC)cc2)=O)CC=C(C(=O)NCCC(=O)N2CCCC2)CC1 C1(NC(=O)CN2CCS(=O)CC2)CN(C(=O)Cc2cc(F)cc(F)c2)CCC1F N1(C(C(Cn2cncn2)NC(c2c(CCC)n[nH]c2)=O)=O)CCOC(C(N)=O)C1 C(=O)(C(F)(F)C(C)O)NCCCC1N(C(c2ccc(OC)nc2)=O)CCCC1 C(=O)(CC(C)C(F)F)NC(c1cccc(C)c1O)C(=O)NC1C(CC=C)CCCC1 C(CCC(=O)N(CCN(C)C(c1occc1C(C)C)=O)C(C)C)OCCC C(CCCC(CO)NC(c1nn(C)cc1C(C)=O)=O)NC(c1ncn(CC)n1)=O N1(C(C2=NOC(C)C2)=O)CCN(C(=O)Cn2ncccc2=O)CC(O)C1 c1(C(N2CC(NC(CC(C)(C)Cc3ccccc3)=O)C2)=O)nccc2[nH]ccc12 C(C(CNC(=O)C(Cc1ccco1)NC(=O)CSc1ccccn1)C(C)C)OC c1(OC)ccc(C(=O)C(=O)NCC2CCC(C)CN2C(c2cccs2)=O)cc1Cl c1(CNC(c2coc(CNC(c3cc[nH]c3C3CCC3)=O)n2)=O)ccncc1F c1(C(=O)NC2C(CC)COC2)cncnc1C C1(n2cc(COC)nn2)CCN(C(c2c[nH]nc2-c2cc(Br)cs2)=O)CC1O N1(C(CCOC)=O)CCC(O)(CN(C)C(c2nccc(-n3ccnc3)n2)=O)C1 c1(OC)c(O)cc(C(=O)Nc2nc(CC(=O)NC(C)CF)cs2)cc1O C12(C(N3CCC(O)(CNC(C(CCN(C)C)O)=O)C3)=O)CCC(O)(CC1)CC2 C(=O)(C(C)C(O)C(C)C)N1CCC(=C)CC1C(=O)NC1CCSC1 C(=O)(C1CCCc2sccc21)NCCCCC1CN(C(c2c(C)nn(C)c2)=O)C1 N1(C(CCc2ncc(CC)[nH]2)=O)CCC(O)(C(C)CNC(=O)Cc2cc[nH]n2)C1 C(=O)(C#CC(C)(C)C)NCC(C)(C)NC(=O)CCCn1c(C)ncc1 C1(C(=O)NCCn2ncc(C)c2)CN(C(=O)CC23CCCC2C3)C(C)(C)C1 c1(OC)cc(OC)c(Cl)c(C(=O)NCC2CN(C(c3cc(OC)n(C)n3)=O)C2)c1 CC1(C#N)CCN(C(=O)C(C)(C)C2CCCN2C(C2CCC3(CC3)C2)=O)CC1 CC1C2CCC(C2)C1C(N1CC2(C)CC1(C(=O)NCc1cc(C3CC3)n[nH]1)C2)=O c1(C(=O)NC(C)(C)C2CC2)cc(S(=O)(=O)NN2C(C(CC)O)CCC2)cn1C C=CC(C)C(=O)N(CC(CC)NC(c1cncn1C1CC1)=O)C C(=O)(C(CO)C(F)(F)F)NC1CC(C(=O)NC(C2CCCO2)CC)C1 CCCCC(C)CCC(=O)NC(C)CN(C)C(c1ncc(OC)nc1OC)=O Nc1c(C(=O)NC(C2CCOC2)CNC(C2CC2C(F)(F)F)=O)cc(F)cc1F C(CC(C)C)(C(=O)NC(Cn1cncn1)C(=O)N1CCC(CCO)C1)NC(C)=O CC1CCCC(C)CN1C(=O)CC(C)(C)CNC(C1(CO)CCCC1)=O C(c1cc(OC)cc(OC)c1)=CC(=O)NC(C(C)NC(C(CC)CC)=O)C C1(C)(C(=O)NC(C(=O)OCCC)C)CC(O)CN1C(=O)CCc1cc(C)on1 c1(CC(=O)NCCCN(C(c2ccncc2)=O)CC2CC2)csc2nccn12 C1(C)(OCC(=O)NC(C)CNC(c2nnnn2C2(C)CC2)=O)CCCC1 C1(C(=O)NC(CC=C)CNC(c2cccn2Cc2cccs2)=O)CSCC(=O)N1 C1(NC(c2c(OC)nsc2)=O)(CO)CCCN(C(c2n[nH]cc2C)=O)C1 N1(C(C2=CC(C)(C)C2)=O)CCC(NC(C2CCC(C3CC3)CC2)=O)CC(C)(C)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])N(CCCOCCNC(C=CC=CC)=O)C.C(C)=O N1(C(C(CC)(C)COC)=O)C2CCC1CC(NC(c1cc3ccccc3o1)=O)C2 c1(N2CCCC(NCc3ccc(NC(C)=O)cc3)C2)nn2cc(C)nc2s1 N1(C(c2c(C)ocn2)=O)CC(N(C)C(C2CC2(F)F)=O)C(C)(C)C1 C1(C(=O)NCCN(CCOC)C(c2cc(Cl)ncc2O)=O)CC2COCC(C1)C2 N1(C(c2c(C)cc[nH]2)=O)CC2(CCN(C(C3CC3c3ccccn3)=O)CC2)C1 N1(C(c2ccsc2)=O)CC2CCC1C(CNC(C13CCC(CO1)C3)=O)C2 N1(C(CC(COC)C)=O)CCN(C)C(C(N2CC(CO)C2(C)C)=O)C1 C1(NC(c2cn(CC=C)nn2)=O)CC1C1CCCN(c2ncnc3c2CCO3)C1 Cc1cc(Cl)ccc1Oc1ccc(C(=O)NCC(C2CCC2)NC(=O)CO)nc1 C1(N(C(CC)C2CCO2)C)CC(C(=O)OC)C1 C1(C(=O)NCC(C)C)COCCN1Cc1cnc(Br)s1 C1(C(=O)NC(CC)CNC(c2nnsc2C)=O)CCCCC1O N1(C(C=C(C)c2cnn(C)c2)=O)CCC2(CCC2)C(CNC(=O)C(F)=C(C)C)C1 c1(C(N2CC(C)(N(C)C(c3cc(Br)c[nH]3)=O)C2)=O)ccccc1OC(F)(F)F C1(C(N(C(C2C(=C)C2C(=O)OC)=O)C)=O)CCCN(c2nnc(C#N)s2)C1 C1(C(=O)NC(C)(C)CCNC(C2CC2(C)C)=O)CCS(=O)(=O)C12CCC2 N1CC=CC1(C)C(=O)N.c1(CNC(C=CCN(CC)CC)=O)cn(CCF)nn1 c1(C(C(=O)N(CC(=C)C)C2CCC2)(C)C)c[nH]c2ccc(Br)cc12 c1(C(=O)NCc2c(C(=O)NC3C(CCOC)CCC3)scc2)ccc(N)c(F)n1 N1(C(c2cc(CC)[nH]n2)=O)CCCC(C2(NC(=O)C3=CCCCC3C)CC2)C1 C1(C)(NC(c2ccn(C)c2)=O)CCC(NC(=O)Cc2c(Cl)cccc2Cl)CC1 c1(C(=O)NCCC2N(C(C3C(OC)CC3)=O)CCCC2)cc(Br)cc(O)c1 C1(F)(C(=O)NCCCN(C)C(c2cc(OC(F)F)ns2)=O)C2CCCCC12 O(C1CCc2cc(Br)cnc21)C(C(c1cccc(F)c1)C)=O C(=O)(C(C(C)O)N(C)C)NC(C(CO)NC(c1cc(C(C)(F)F)n[nH]1)=O)C N1(C(C=CC(c2ccccc2)=O)=O)CC(NC(C2CCOC2=O)=O)C2(CC2)C1 C1(CNC(COCCN(C)C)=O)CN(C(=O)Cc2ccnnc2O)CC(C)(C)O1 C1(C(=O)NCC(c2ccncc2)O)(CC)CCCN(C(=O)C=Cc2cc[nH]n2)C1 c1(C(=O)NCC2CC(NC(C(CC=C)OC)=O)C2)ccc(N)cc1Br C1(CC)CCC(C(N2CCCC2(C(=O)Nc2ccccc2)C(C)C)=O)CC1 N1(C(CN2C(=O)COCC2)=O)CCN(C(c2cccc3cc[nH]c23)=O)C2CCC12 c1(CC)[nH]nc(C(=O)NCC2C=CCN2C(C2CC(C)(C(C)(C)C)C2)=O)c1Cl N1(C(C2C(C(C)C)C2)=O)CCC(C(F)(F)F)C(CNC(=O)C2=CC(C)(C)C2)C1 c1(SCCCC(=O)NCCC(CNC(C2(C)CC(=C)C2)=O)O)ccc(Br)cc1 C1(C(=O)NCC2CCN(C(CC)=O)C2)CC(O)CN1C(=O)Cc1c(Cl)cnn1C O=C(O)CCN=c1ccc(NCC=C(Cl)Cl)n[nH]1 Cn1nncc1-c1cnc(C(F)(F)F)s1 C1(CC)C(NC(c2ccccc2Br)=O)CCN1C(=O)C(C)NC(C)=O Cc1cnc(C(=O)NCC2(NC(=O)C(O)CN3CCCC3)CCCC2)c(C)c1 N1(CC(=O)N(CC(n2ccnn2)C)C(C)(C)C)CCCC1 N(C(=NCCc1cccs1)NCC(C)(C)C1CC1)C(C)CC1CCOC1 c1(C(=O)N(c2ccco2)CC)cnc2nc(N3CC4CC(N)C4C3)oc2c1 C1(CCOC)CCN(C(=O)Cn2ccc(C)c2)CC1.C12(CC1)C(=O)N(C)C2 c1(C(C)C)nocc1C(=O)NCC(C1(O)CN(C(=O)CN2CC3CC3C2)C1)(C)C c1(C(=O)OC)cccc(C(c2nnnn2C(C)(C)C)NC(c2ncc(C)o2)CC)c1 C=C1COCCN(C(c2cnc(C(F)F)s2)C(=O)NC2(C)CC2)C1 CC(C)(CS(C)(=O)=O)C(=O)NCC=CCNC(C1CC1CSc1ccccc1)=O c1(CCC(=O)NCCC(C)NC(=O)C(C)(C)CO)ccc(Cl)cc1Br C#Cc1ccc(C)c(NC(=O)CC2CCCC(NC(=O)CC(C)(C)C)C2)c1 c1(C(N2CCN(C(C(C(C)C)SCC)=O)C(C)C2)=O)ccc2c(C)noc2n1 C(=O)(C#CC1(C)COC1)NC(C1CCCN1C(C1CN(C)CCO1)=O)C CC1(C)CN(C(=O)CN2CCCS2(=O)=O)CC1CNC(=O)CCC1CCCO1 C1(O)(CCNC(C(COC)OC)=O)CCCN(C(c2cc(C3CCC3)no2)=O)C1 N1(C(CCCNC(C)=O)=O)CCC(O)(C2CCN(C(=O)C3=C(Cl)CCC3)CC2)C1 N1(C(CCC(CC)=O)=O)CCC(C2CC2)C1C(=O)NCCc1nnc(O)o1 C1(CCC)CC2CCC1(Cn1c(C3(SCC)CCCC(CC(=O)OC)C3)nnn1)C2 CC1CC(C(=O)N(C2CCCCC2)CCNC(=O)CNC(=O)C2CC2)CCS1 c1(CC)noc(CC)c1CC(N1CC(N(C)C(c2nc(CC)no2)=O)C(O)C1)=O N1(CCNC(C(=O)NC(c2c(OCC)cccc2)CF)=O)C(C)CCCC1C N1(C(CCC=C)=O)CCOCC(CNC(c2nn(C)nc2Br)=O)C1 C(CCO)(C(F)F)N(C(C(C1(O)CCC1)NC(CCC)=O)=O)C C1(C(=O)OC)Cc2c[nH]nc2CN1c1cc(Br)nc(C)n1 Cc1cc(C(N2CC(NC(C3(CCF)CCC3)=O)CCC2C)=O)c(O)nc1C c1(OC)ccc2c(N3CCNCC3C(=O)Nc3cc(O)ncn3)ncnc2c1 Cc1c(C=CC(N2CC(NC(=O)C(=O)NCC3CC3)CC2(C)CO)=O)cnn1C N1(C(c2ccn(CCC)n2)=O)CCC(C2CCN(C(=O)C(C)(C)CC#N)CC2)C1 c1(OC)ccc(CNC(=O)C(C2CCC(=O)CC2)F)c(OC)c1Br N1(C(CCOC(C)C)=O)CCN(C(c2ccccc2C(F)(F)F)=O)CC(O)C1 N(C(=NCC(C)C)N1CCC2(CCCC2)C1)C(C#C)C(C1CCC1)OC c1(CC)ccc(NC(C2CC(NC(=O)Cc3cccc(F)c3)C(O)C2)=O)cc1 c1(CC(=O)NC(C2(O)CN(C(C3CC4(C3)CC(O)C4)=O)C2)C)cccc(Cl)c1Cl c1(CC(=O)NC2CC(NC(CC3C(OC)CC3)=O)C2)cccc(OC(F)F)c1 N=c1nnn(CC(=O)NC(c2ccccc2)CNC(c2nn[nH]c2Cl)=O)[nH]1 c1(OC)nn(C)cc1C(N1CCCC1C(=O)NCC1(CCO)CCC1)=O O=C(C#CC1CCCC1)NC1COCCN(C(=O)CN2CCSCC2)C1 CCCC(C)CC(=O)N1CC2(CNC(C3CN(C)C3)=O)CCC1C2 C(=O)(CCC(O)C(C)(C)C)NCC1C(NC(c2nc(C)nn2C)=O)CCC1 c1(CC)cccc(OC)c1.C1(CC(=O)NC)CCCC12CC2.C1C(=O)O1 c1(C(N2CC(CC)N(C(=O)C3=CCSC3)CC2)=O)cnc2n1CCOC2 CCC(C)C(C)(O)CNC(=O)CCC(C)(C)NC(c1cnc(C)nc1)=O CP(C)(=O)CC(=O)NCc1ccc(CNC(C2CC(O)CN2C)=O)cc1 c1(OCC)cccnc1C(=O)N(C(CNC(=O)C=Cc1csnc1C)C1CC1)C O=C1NCCSc2cc(NC(C3CCC(F)(F)C3)c3nnnn3CCC3CC3)ccc21 C#Cc1ccc(CC(N2CCC(NC(=O)CCC3CC3(C)C)C(O)C2)=O)cc1 c1(NC(C2CCN(C(c3nnn4ccccc34)=O)C2)C)c(Br)cccc1[N+](=O)[O-] C(C(=O)N1CC(O)CCO1)c1ccccc1.N(C)(C(=NCCC(C)=O)N)C(CC)C C#Cc1cccc(C(N2CCC(NC(=O)C(C(C)(C)C)OC)C(CO)C2)=O)c1Cl c1(C(=O)NCC2CN(C(=O)CC3CCCOC3)C2)c(CC2CC2)cccc1Cl C(=O)(CC(CC1CC1)NC(=O)CCCOC(C)(C)C)NC(C(C)C)CCN(C)C O=C(C1=C(Cl)CCC1)NCC1(NC(C23CCCCC2C3)=O)CCCC1 c1(NC(C(C2C3CCCC23)N(C2CCC2(C)C)C)=O)ccc(F)cc1 N1(C(c2cccc(NC(C)=O)c2)=O)CC(C(=O)Nc2ccnc(C#N)c2)CC(C)C1 C=CC(CC)C(=O)N1CCCC1CNC(C1(c2ncc[nH]2)CC1)=O c1(C(=O)NC2C(NC(c3cc(OCF)ccc3Br)=O)C2)cccc([N+](=O)[O-])c1O c1(OC)noc(C)c1C(=O)NC(C)CCCCNC(c1cc(C)c(C)[nH]1)=O C(CC(C)C(=O)N1CCC(C)C1C(=O)NCCN1CCC(OC)C1)=CC c1(N(C)C)cc(C(N2CCC(NC(C3CCN(C(N)=O)CC3)=O)C2)=O)cc(Cl)n1 C1(OC)COCCC1CC(=O)OCC(=O)NCCCCN1CCCC(C)C1 C(C(C)(C)CC(C)C)NC(c1cc(CC)on1)=O.C(C(F)C(=O)NC)C1CNC1 C1(C(=O)NC(CCN(C(c2cc(C(CC)C)no2)=O)C)C)CN2CCN1CC2C C1(NC(C(OC)OC)=O)CC(C)CN(C(c2cncc3c2CC3)=O)C1 CC1=NS(=O)(=O)NC=C1C(=O)N1CC2(C1)CN(C(=O)C(CC(C)C)N(C)C)CCO2 C(=O)(NNC(=O)C(=O)NCC1CCCO1)N1CCC(O)CC(C)C1 C1(NC(c2c(C)ccnn2)=O)CN(C(c2ncn(C)c2C)=O)C2(CCCC2)C1 c1(CCC)sc(C(=O)NC(C)(CNC(=O)C(C)c2ccsc2)CO)cc1CC C12(CNC(c3ccc(C)s3)=O)CC(NC(c3cc(C(C)(C)C)nn3C)=O)(CO1)C2 C1(C2CC2)(CNC(COCC(=C)C)=O)CCN(C(c2cnsc2)=O)C1 C(=O)(CCCC(=O)NC12CC(CNC(=O)CC3CCCCC3(C)C)(C1)C2)NCC O=C(C#CC1CCCCO1)NCC1CN(C(=O)CN2CCC(CO)CC2)CCO1 C1(CNC(C2(CC#C)CCCC2)=O)CN(C(c2cncnc2C2CC2)=O)CCO1 C(CC(=O)NOC(CC(C)C)C(=O)O)(OC)OC c1(C(=O)OC)ccc(F)c(CN2CCC(F)(C(=O)NC3(CO)CCNCC3)C2)c1 O=C(N=c1nc(O)s[nH]1)c1ccccc1OCCF CN(C)NC(=O)CCC(=O)N(C1CCN(C(c2cc3cccnn3n2)=O)C1)C C12(NC(c3c(Cl)ccc(OC)c3F)=O)CCCC1N(c1nnco1)CCC2 c1(C(=O)NCC(CNC(c2ccc(OCC)nc2)=O)C)nccn2ccnc12 N1(C(c2c(CC)nc[nH]2)=O)CCC2CN(C(c3ncc(C)cc3OC)=O)CCC12 N1(C(Cc2c(C)onc2Br)=O)CCN(C(C2CC2F)=O)C(C2CC2)C1 C(=O)(C(C)(C)CN1CCOCC1)N(CCNC(C1CC(O)C1)=O)CC C#Cc1ccc(C(N2CC3(CC3)CC2C(=O)Nc2cnccc2CC)=O)c(C)c1 C1(NC(=O)Cn2ccnc2)CC=CCC1C(=O)N(CC(O)C(F)(F)F)C1CC1 C(=O)(C(O)C(C)(C)CC)NC1C(C=C)CN(C(=O)CN2CCOCC2=O)C1 Cc1nn(C)cc1C1CCCN1C(=O)Nc1ccc(Cl)[nH]1 N1(C(CCOCC#C)=O)CCSCC1CCNC(c1cc(C)n(C)n1)=O C1(CC(=O)NCCN(C(=O)C2=CCOC2)Cc2ccccc2)CCCC(O)C1 N1(C(c2ncn(CC)c2)=O)CCCN(C(=O)Cc2ccc(C)cc2F)CC1 c1(C(=O)NCC(CNC(C(C2CCOCC2)OC)=O)(C)O)cc(Cl)n[nH]c1=N Cc1cc(C(=O)N(C)Cc2ccc(CNC(C3(C#N)CCOC3)=O)cc2)ccn1 CC(C)(C)C(O)C(=O)NC(C)(CNC(=O)CCc1cc(Cl)cc(Cl)c1)CO C1(CNCCCN(S(C)(=O)=O)C)(CO)COCC2CCCCN12 c1(OC)cccc2c(C(=O)NC3CN(C(C4(COC)CC4)=O)C3)coc12 C1(NC(c2cc(CNC(c3n[nH]c(C)c3Cl)=O)no2)=O)CCCCC1C#N C#CCC(C)(C(=O)N(c1ccc(Cl)cc1)C)NC(c1cccc(C#N)c1)=O C12(NC(CC(CC=C)NC(=O)Cc3cc(C)cs3)=O)CC3CC(CC1C3)C2 c1(OCC)ccc(CN2CCCC2CCC(=O)NCc2ccsc2)cc1F C(=O)(C(F)(F)C(F)(F)C(F)F)N1CC2C(CNC(CS(CC)(=O)=O)=O)(C2)C1 C1(C(=O)NCC2(C#C)CCC2)CC2C=CC1CCC2 C(CN=c1[nH]cnc(=N)[nH]1)N(C)C(=O)OC(C)(C)C.C(=O)(CCC1CCOC1)O C(=O)(C1=CCC(C)(C)CC1)NCC1(C(=O)Nc2c(Br)cn(C)n2)CCCCC1 C1(CC)C(NC(C2(SC)CC2)=O)CCN1C(c1csc(-c2cccs2)n1)=O C(C1CCOCC1)=CC(=O)NCC(C(C)C)NC(=O)Cc1ccn(C)n1 c1(C(=O)N(C(CNC(C=CC(=O)OCC)=O)CCOC)C2CC2)cccc(F)c1Cl C1(CC(=O)NCCC(C)NC(=O)CNS(=O)(=O)C2CC2)CCCCN1C C(C(C)CCCC(C)C)NC(c1nnnn1C(C)(C)C)C1CC(=C)C1 C(=O)(C1=CCC2(COC2)OC1)N1CCCN(C(c2onc3c2CCCC3)=O)CC1 c1(C(=O)NCC2CC23CN(Cc2cncc(C(F)(F)F)c2)C3)ncc(Cl)cc1Cl C1(C(=O)NCC(=O)NCc2cccs2)CC(O)CN1C(=O)CCCCC1CC1 c1(OCC)cc(F)c(-c2n[nH]c3c2CN(Cc2cnn(CC4CC4)c2)C3)cc1F c1(C(=O)NCC2CCN2C(=O)CCOC2CC2)c(C(F)(F)F)nc2n1CCCC2 N1(C(C=CC(=O)N(CCNC(C2CC(C(C)C)C2)=O)CC2CC2)=O)CCOCC1 c1(OC)cccc(O)c1C(N1CCCC(CO)(NC(=O)CC2CC(F)(F)C2)C1)=O c1(NC(CC2(C=C)CN(C(C3(COC)CC(=C)C3)=O)C2)=O)cn(CC)nc1C#N C12(C(=O)OC)COCCC1(F)CN(C(=O)NCc1ccnc(S(N)(=O)=O)c1)C2 C1(C(N2CC(c3c(C)nn[nH]3)C2)=O)CC1C1CN(C(C2CC(O)C2)=O)C1 CC(CS(C)(=O)=O)C(=O)NC1CC1NC(c1cc(OC(F)(F)F)ccc1O)=O C1(OC)CC(CNC(c2ccsc2)=O)N(C(C2CC(C)OC2C)=O)C1 c1(C(=O)NC2(CO)CCN(C(=O)CCc3cncs3)C2)cc2ccccc2[nH]1 c1(C(=O)NC(CC)CNC(=O)C=CC(C)OC)cccc(C(C)(F)F)n1 C1(C2CCN(C(C3(CF)COC3)=O)C2)(NC(C(CC(C)C)OC)=O)CC1 n1(CC(=C)C)nnnc1C(c1ccoc1)NCCc1ccc(C)o1 C1(C(=O)NCC2OCC(CC)C2)CCCN(CC#C[Si](C)(C)C)C1 C1(NC(CC(CC)O)=O)CCN(C(C2(N3CCCC3=O)CC2)=O)CC1C C1(OC)CN(C(C2(C)CC=CC2)=O)C(C)(CNC(C2CCN2C)=O)C1 C(N=c1[nH]c2ccccc2o1)C1OCCCN(C(c2ccc(Cl)cn2)=O)C1 C(=O)(C1=NNC(=O)CC1)N(CC(C)NC(=O)C=CC1CCOCC1)CC C1(NC(Cc2cn(CC)nc2)=O)CC(F)CN(C(=O)CN2CCOCC2=O)C1 C1(C(=O)NCCCN(C(=O)Cc2cccc(OC)n2)CC)COC2CCCCC12 N1(C(=O)CCC2CCCO2)CCCCC2(CCN(Cc3ccc(Br)o3)C2)C1 c1(C(=O)Nc2ccc(CN3CCOCC3)o2)cc(C2=CCC(O)CC2)ccn1 c1(C(=O)OC)nn(C)cc1S(=O)(=O)NC1CCC(C(=O)O)CC1 c1(NC(C2(C3N(C(c4c(N)cccn4)=O)CCC3)CC2)=O)ncc(Cl)cc1O C1(OC)CC(CNC(=O)COCc2ncc(C)o2)N(C(=O)CC(C)F)C1 N1(CC(=O)N2CC2=O)Cc2ccccc2CC1C(C)C.C(C)(C)N(C)C c1(C(=O)NCC(C)N(C(C2CCC2)=O)CC)ccc(C(C)(C)C)nc1 C(=O)(CC(F)(F)F)NCC(=O)NCCCC(C)NC(=O)C=C1CCN(C)C1 O=C(N=c1ccnc(C(F)(F)F)[nH]1)C1CC(C(=O)Nc2ccc(F)nc2F)C1 c1(C(=O)NCC2N(C(c3c(C)ncc(N)c3)=O)CC2)cccc2[nH]cc(Cl)c12 N1(C(c2n(C(C)C)ncc2)=O)CCC(CNC(=O)CC2CC(=O)C2)CC1C N1(CC(C)NC(=O)CSc2ccccc2)CC23CCCCC2(C1)CN(C)C3=O c1(C(N2CC(NC(c3onc(C(C)(C)C)n3)=O)C2)=O)ccc2c(c1)C(=O)OC2 c1(C(=O)NC2C3CCN(C(C(C)=C4CCC4)=O)C32)cc(Cl)c([N+](=O)[O-])[nH]1 C(c1ccc(Cl)cc1F)=CC(N1CCN(C(C(CSC)(C)C)=O)CC1)=O CC(C)C(C(=O)NC1CC1CNC(c1cnccn1)=O)N1CCCC1=O N1(C(C(C)C2CCCO2)=O)CCN(C(C2CC(O)C2)=O)C(C)C1 C#Cc1ccc(C(=O)NC2CC2NC(=O)C(C)CN2CCOCC2)cc1Cl C1(CNC(c2c(COC)ccs2)=O)CCN(C(=O)Cc2cccc(Cl)c2)CC1C c1(NC(C2CCN(Cc3ccc(OC)cc3Br)C2)=O)ccc2c(c1)c(Br)nn2C C(=O)(C(O)CC(C)(C)C)NC(C1CCCC1)CNC(C(C)(C)OC(C)C)=O c12ccc([N+](=O)[O-])c(c1)NC(=O)C2.C1(CNC(CSCC)=O)(COC)CC1(F)F N1(C(c2cnc(Cl)cn2)=O)CC2CCN(C(=O)COCC(F)(F)F)C2C1 c1(C(=O)OCC)c(NC(CNC(=O)C(O)C2CCC2)C(C)C)cc(C)nc1O CC1CCCC1(C)CN(CCCCN(C(=O)CCNC(=O)CO)C)C C(N=c1[nH]cc(Cl)c(C)c1C#N)C1CN(C(C(C(CC)C)C)=O)CC1C(F)(F)F CN(Cc1ccc(Cl)s1)N1CC2(CC(C(N3CCCCC3)=O)CO2)C1 c1(C(=O)NC2C(NC(C3(CN(C)C)CC3)=O)CCC2)ccc(Cl)c(O)c1N c1(C(=O)NC(CNC(C(C)OCC(F)(F)F)=O)C(C)(C)C)c(N(C)C)cccc1F C(CN=c1ncc(C(=O)NC2CC(C)N(Cc3ccccc3)C2)c[nH]1)OC C1(C(N(CC(=O)N(C(CO)CO)CC)CC2CC2)=O)CCC(=O)O1 C(=O)(CS(=O)(=O)CC(F)(F)F)NCC(c1ccc(OC)cc1)NC(C=CC)=O CC#CCC(C(=O)N(CC)CC1CCOC1)NC(=O)C(C)C(C)(C)C C12(NC(c3c(C(C)C)nn(C)c3)=O)CC(CNC(=O)Cn3ccnn3)(C1)OC2C N1(C(c2c(SC)ccs2)=O)CCCC(NC(=O)Cc2c(C)noc2C)C(F)C1 c1(C(N2CC(O)(C(C)NC(c3cn(C)nn3)=O)C2)=O)ccc(F)cc1 c1(-n2cc(C)nc2)cccc(C(=O)NC(CCn2nnc(-c3ccsc3)n2)=O)c1 C(C)(CNC(c1cc(C(F)(F)F)cn1C)=O)(CC(C)C)NC(c1[nH]cc(C)c1)=O N1(C(c2c(CCC)n(C)nn2)=O)CCN(C(c2cccnc2O)=O)C(C2CC2)C1 n1(C2CCN(CCNC(CC(C)(C3CC3)OC)=O)C2)nnc2c1CCCC2.C(N)(=O)N C12(C(=O)NC(CCOC)C(=O)NC(c3nn[nH]n3)CC)CCCC1OCC2 Cc1[nH]c(-c2ccccc2)c(C)c1C(=O)NNC(=O)CCOCC1CCCO1 N1(C(C(C(C)C)N(C)C)=O)CCCC2(CCN(CCCS(C)(=O)=O)C2)C1 C1(OC)CC(CNC(=O)C(C(C)C)c2cccs2)N(C(c2ccnn2C(C)C)=O)C1 N(C(=NCCCCl)NCc1cscc1C(F)(F)F)C(C1CCCO1)C C=CCC(C)C(=O)N(CC)CC1CCN(C(=O)Cc2cccc(F)c2)CC1 n1(CC)nc(C)c(C(N2CC(CO)(NC(=O)C3=NOC(C(C)(C)C)C3)C2)=O)c1Cl N1(C(c2ccc(COC)s2)=O)CC(NC(=O)C=C(C)c2ccsc2)CCC(O)C1 Cc1ncccc1C=CC(=O)NCC(C)(C)CNC(=O)C(c1cccc(O)c1)C c1(C(N2C3CC(OC)(C3)C2)=O)nn(C)c2c1C(O)CCC2 N1(C(c2cnc(C)s2)=O)CC2CC(NC(C3(c4ccnn4C)CC3)=O)CC2C1 c1(NC(N2CCC3(CN(C(C(=O)NCC)=O)C3)C2)=O)cc(C)ccc1S(N)(=O)=O c1(CN2C(C(=O)Nc3c(C)noc3C)CC(O)C2)cc(Cl)cnc1Br C=CC(O)(C(=O)NCCN(C(=O)CCCO)CCC)C(F)(F)F.C(C)=O c1(C(=O)NC2CCN(C(C(C)NC(=O)NC)=O)CC2C)ccc2ocnc2c1 c1(C(C)C2CC2)ccccc1-c1nc(C2CC2)nn1C(C)C(F)(F)F c1(C(=O)NCC2C(CNC(C(C)(C)OCC)=O)C2(F)F)ccc(F)c(C)c1 C(=O)(C(CNC(C1(n2nccn2)CC1)=O)CC(C)C)N1CCN(CC#C)CC1 C(CCC(=O)N(C(C)C)C)O.C(C(=O)N(C1(CC(C)C)CC1)C)=CC CCC(COC)(CC)NC(C1(OC)CCSC1)c1nnnn1C1CCCC1 CC(CC(C)(C)C)C(=O)NCC(CC1CC1)NC(=O)CC(C)(C)Cc1ccccc1 C(=O)(CC(O)C(C)CC)N1CCCCC(C(N(CCCC)CCCC)=O)C1 C1(CNC(COCC(C)C)=O)(CNC(=O)Cc2ccco2)CC1(F)F C=CCCCC(C(=O)NCC1(C)NC(=O)NC1=O)NC(C1OC2CCC1C2)=O C(=O)(C(CNC(=O)CC(F)(F)F)CC(C)C)N(CCCC)CC CC1(C(N2C(C(N3CCCC3NC(N)=O)=O)CCC2C2CC2)=O)COCCO1 N1(C(C(C)OCCCC)=O)CCCC(C)(NC(c2ccn(C)c(=O)c2)=O)C1 Cc1nc(S)sc1CC(N1CCC(C(C)CNC(c2ccc(Cl)s2)=O)CC1)=O c1(NC(N2C(C=C)CCCC2)=O)cc(C)[nH]c(=NC)n1 c1(CC(=O)NC2C(C)CCN(C(C3CCCN3C)=O)C2)cc2ccccc2o1 C(=O)(C1CCCc2c[nH]nc21)N1C2C(C(Oc3snc(CCC)n3)CC)C(C2)C1 C(CN=c1[nH]c(=NCC2(C)CCCCC2(F)F)[nH]c2c1CS(=O)(=O)C2)C1C(C)C1 C1(C(C)NC(=O)COC2COC2)CCCN(C(c2scnc2Cl)=O)C1 C1(N(C(C(C(C)NC(c2c(C)[nH]cc2)=O)C)=O)C)CCN(C)CC1C C1(C#N)(C(=O)NCC2CC(NC(C(COC)O)=O)C2)CCCCC1 C1(NC(C2CC(C)(CC)C2)=O)CCC2CN(C(c3ccc(C)c(F)c3)=O)CC2C1 C1(NC(=O)Nc2n(C)nc(C3CCCO3)c2)CC(C2CCCC2)C1 Cc1cccc(C(=O)N(CCCCCNC(=O)CC2CCCC(C)C2)C(C)C)c1Cl Cc1sc(C(N2CCC(C(F)(F)F)CC2)C(=O)NC2COC2)c(C)c1Br c1(C(=O)NCC(CNC(c2nc(COC)oc2)=O)OC)cnc2cc(C)[nH]c2c1 C1(C(N2CCC(O)CC2)=O)(COC)C=CCN1C(=O)C(C)OCC(C)C N1(C(C(C(C)C)NC(c2cncc(N(C)C)n2)=O)=O)CCCC(C)(CO)C1 C1(C(=O)NCC2C(C(=O)NC3CN(CC)CC3C)CCN2C)CC(=O)CC(=O)N1 c1(C(=O)NCC2(CNC(=O)C3=CCOC3)CC2)cc(CSC)ccc1Cl C(CC(C(=O)NCCC1CCCN1C(C1CC1F)=O)OC)OC C1(NC(C(CSC)C)=O)CCN(C(c2ccc(-c3nc[nH]n3)cc2)=O)CC1O c1(C(=O)NC2CCC(F)(CNC(c3cnns3)=O)C2)cc(F)c(F)c(O)c1F C1(NC(=O)NCc2c(C)c(Cl)ccc2)CC2(CCC(CN)OC2)C1.N12CC(C1)C2 Cc1cccc(=O)n1CCCCN(C(=O)C(C)n1ccnc1)C(C)C C1(NC(CN(S(C)(=O)=O)C)=O)C2CCC1N(C(=O)Cc1cccnc1)C2 N1(C(C(CC2CC2)NC(CC2(CC)CCC2)=O)=O)C2COCC1C2 CN1CCc2ccc(C(=O)NC(C)(C)Cn3ccc4ccccc34)cc21 CCCC(C(=O)NC(C)C(C)NC(=O)C(c1ccccc1OC)(C)C)NC(C)=O C=CC(C)(CC)C(=O)NCCCN(C(c1cc(Cl)ns1)=O)C1CC1 C=Cc1cncc(C(=O)NCC2CCN(C(c3oc(C)cc3C)=O)CC2C)c1 c1(OC)cc(CN2CC(O)CC2C(=O)Nc2cnc(C)cn2)cc(C(F)(F)F)c1 c1(C(=O)NC(CCCCNC(CC(C=C)C)=O)C)c[nH]c2c(Br)cccc12 c1(CC(=O)NCC(C)CNC(=O)Cn2nnc(C(F)F)n2)n[nH]c2c1CCCC2 c1(C(=O)NCCCC(C)NC(C2(C(=O)NC)CCC2)=O)cc(F)cc(F)c1N c1(C(C(=O)NCC2CC(NC(=O)CCc3cc(Cl)cs3)C2)OC)cccc(Cl)c1 n1(CC)ncc2c(N(CC(C)NCC(C(C)C)OC)C)nc(NC)nc12 c1(-n2ccc(=NC(=O)C3CCCCN3S(C)(=O)=O)[nH]2)nnc(O)c2c1CCCC2 C(=O)(C1=CCCCO1)N1CCC(CNC(=O)CC2CCN(CC(F)(F)F)C2)C1 c1(C(N2CCC(C(C(=O)NC(c3ccn(C)n3)CC)(C)C)C2)=O)cnc(C)nc1 c1(C(N(C(=O)C(O)CCSCC)CC(C)O)=O)cc2ncccc2[nH]1 C(=O)(C1=NOC(C)(C)C1)N(C1CCCN(C(c2cccc(C)c2O)=O)C1)C c1(COC)ccc(C(=O)NCC2COCC2C(=O)NC2(OC)CCC2)o1 CCC(CC)(CO)C(=O)N1CC(CCNC(c2ccnc3c2CCO3)=O)C1 N1(C(=O)NC(C2CC3CCC2C3)C)CCC(Cc2cc(C(C)(C)C)n[nH]2)CC1 C1(NC(CN(C(C)=O)C)=O)CCCC(C(=O)NCCCOCCO)CC1 c1(C(=O)NC2CN(C(C(C)C3CCC3)=O)C(C)C2)cn2cnnc2cn1 C1(CNC(=O)CC2CCC2)CCCC(NC(=O)C=CC2CCC2)C1 C12(NC(CCc3ccc(C)s3)=O)CC1CN(C(c1cc(CO)oc1C)=O)C2 Cc1noc(C(=O)NC23CC(NC(C4C5CCC4(c4ccccc4)C5)=O)(C2)C3)c1C c1(N(CC(C)NC(=O)CC2CCCC(C)(C)O2)C)ccc([N+](=O)[O-])cc1Br C1(CN(C(CCNC(=O)OCC)=O)C)CCC(C(=O)NC(C)CC)O1.OCC c1(SCC(N2C(CNC(c3cc(CC)on3)=O)CCC2)=O)nc2ccccc2o1 C1(NC(CNC(CNC(C)=O)=O)=O)COCCC1C(N1CCN(C(=O)CO)CC1)=O C(C(C)(C)CNC(c1nocc1C(C)C)=O)N(C(=O)Cc1cscn1)CC C1(NC(c2nsnc2O)=O)CC2CN(C(c3ccnc(Cl)c3O)=O)CC12 C1(NC(c2c(OC)csc2)=O)CC(CNC(c2csc(Br)n2)=O)C1(C)C c1(C(=O)NCC2(C)CCC(NC(C(CC)CC)=O)C2)cccn2ccnc12 CCCCC(C)(F)C(=O)NCCCC1CCCCN1C(c1cccc(C)n1)=O N1(Cc2n(C)c3c(n2)c(Cl)ccc3)CCc2c(Cl)c(Br)cc(F)c2C1 N1(C(CCOC)=O)CCCC1CN(C(c1nonc1CC)=O)C1CC1 C(=O)(C1=NOC2COCC12)NCC1CCCC(C(=O)NC(C)(C)CCCF)C1 C1(NC(C=NOC)=O)CCCC(CNC(C2CC(c3ccccc3)C2)=O)C1 CCCCC(C(=O)NC(CNC(=O)CC(=O)N(C)C)CC)C(C)C C1(C)(NC(C2N(C(Cc3cc(C)sc3)=O)CC(O)C2)=O)C(C)(C)C1(C)C c1(C(C)(C)C)cccc(NC(=O)C(N2CCC(N3CC(O)C3)C2)C2CC2)c1 C1(NC(c2ccc(C)o2)=O)CCCC2CN(C(C34CC(C3)S(=O)(=O)C4)=O)CC12 Cn1cc(C=CC(=O)NC2(C(=O)NCCC(N)=O)CSC2)cn1 N1(C(CCc2onc(C)n2)=O)CC(NC(C2(N(C)C)CCC2)=O)C2CCCC12 C1(C(N2CC(C(C)CO)C2)=O)CC2CCC2C1 Cc1ncc2n1CCC(C(=O)NC1CC(F)CN(C(C3CN(C)CCO3)=O)C1)C2 CCCC(CC)CCC(=O)NC(c1nocc1C(=O)NCCC(C)N1CCCC1)C N(C(=NCCC1(O)CCCCC1)N1CCCC(CC(N)=O)C1)CCOC C=Cn1nccc1C(N1CCCC1CC(=O)NCC#CCSC)=O C(Cc1cn[nH]c1)(C(=O)Nn1nncc1CO)NC(C(C)(CO)OC)=O N1(C(C=C(CCC)C)=O)CCC2(C1)C(=O)N2.c1(CC2CC2)cccc(Cl)n1 c1(C(=O)Nc2cnn(CCC(C)C)c2C(C)C)cc2cc(Br)sc2s1 N1(C(CCCC(C)O)=O)CCC2CCN(C(c3c[nH]nc3C3CCCO3)=O)CC12 O=C(C1=COCC1)NC1CCCC(NC(=O)Cn2ccc(C3CC3)n2)C1 C1(C(N2CCOCC(NC(c3c(CC)csc3)=O)C2)=O)CS(=O)(=O)CC(=O)N1 CC1CN(C(=O)CCN2CCOCC2=O)CC1CNC(=O)CCc1nccs1 c1(C2C(C(=O)NC(CS(C)(=O)=O)c3ccccc3)C2)c[nH]c2c(Br)cccc12 c1(C(N2C(C(N3CC(C(CC)C)C3)=O)CC(F)CC2)=O)cc2ccccn2c1 c1(C(N(C)CC2CCCCN2C(c2ccc[nH]2)=O)=O)ccccc1S(C)(=O)=O c1(CC(=O)NCC(C2CCCCC2)NC(C=COCC)=O)ccc(C)nc1Cl C=CC1(CC(=O)NCCCN(C(C2C3CCCCC23)=O)C2CC2)CCCCC1 Nc1cc(F)c(C(N2CC(C3(NC(c4cccnn4)=O)CC3)C2)=O)cc1F C1(NC(C(C)(C)NC(Cc2c(C)n(C)cn2)=O)=O)CCCCCC1(C)C c1(OC)ccccc1OC1(C(=O)O)CCC1.c12ccc([nH]1)C(=O)NC1CN(C1)C2=O C12(CCC(C)(C)C1)C(=O)N2.c1(CO)ncccc1SC.c1(C(=O)OCC)cnc(N)s1 C1(n2cnnn2)(CC(=O)NC2C(NC(CC(=O)N(C)C)=O)C2)CCOCC1 C1(CNC(c2cccc(C(F)F)n2)=O)COCCN1C(c1nncs1)=O c1(C(=O)NCCOCCCNC(CCC(=O)OC)=O)cc(Cl)c(F)cc1Cl N1(C(c2cc(C)nn2C2CC2)=O)CCC(NC(C2(C)CCCCCC2)=O)CC1C c1(C(N(C2CCN(C(C3CN(C(C)=O)C3)=O)C2)CC#C)=O)cn(C)c(C(F)F)n1 Cc1ccc(COCC(N2CCN(C(=O)CCn3cncn3)CC2)=O)cc1F CC1CCCCC1n1nc(C2CC2)nc1-c1c[nH]c(Br)c1.C1(CO)CCC1 C(CC(C)C(=O)N(C)CC1CC1)OC.C12CCCN(C1)C(=O)C(=O)N2 N1(CC)CCOC(C(=O)NC2(C(=O)NC3C(C)CCC3C)CC(F)(F)C2)C1 C(C(=O)NCC(C1CC1)NC(=O)COC(=O)NCC1CCC1)OCC=C C(=O)(C(C(O)C(F)(F)F)C(C)(C)C)NCCN(C(C)C)C(c1cn(C(C)C)cn1)=O C1(C(=O)NCC2(F)CN(C(CSc3n(C)ccn3)=O)C2)CCCC2CCCN12 C1(N(C(CNS(CCCC)(=O)=O)=O)C)CCC2CN(C(=O)C(=O)C(C)CC)CC12 c1(CC=C)cccc(C(N2CCCC(CN(C)C(C3CC3F)=O)C2)=O)c1 c1(C(=O)NCCN(C(c2ccc(CCCCC)o2)=O)C)cc2c(s1)CCOC2 CCCC(C(=O)NC(CNC(=O)COc1cccc(Cl)c1CC)C1CC1)C(C)C c1(CC)c(C(=O)NC2CCCC(NC(=O)CCn3nc(C)nc3C)C2)nnn1C c1(C(=O)NCCOCCC(=O)NCCc2ccc(F)nc2)c[nH]c(=S)cn1 CCC(CCCC(=O)NC1CC2(CCCC2)C1)NC(C1(C)CC(F)C1)=O C1(C(N2CC(C3(NC(CCC(=C)Br)=O)CC3)C2)=O)CCc2nncn2C1 O=C(C1=COCC1)NC1CCC1C(=O)NCC1CCC(F)C1 c1(NC)ccc(C(N2CC=CC2(C)C(=O)NC(C)Cc2ccncc2)=O)nc1 c1(C(=O)NC(CC)CNC(C2CCC(N(C)C)CC2)=O)ccc2oc(C)nc2c1 N1(C(C(C)C2CCCO2)=O)CCC(C2(O)CN(C(=O)C3=CCCCC3)C2)CC1 c1(C(=O)NCC(CC(C)C)NC(=O)CS(C)(=O)=O)ccc2c(O)n[nH]c2c1 N1(C(C2CN(C(C3(OC(C)=O)CC3)=O)C(C)C2)=O)CCCCC(F)(F)C1 C1(NC(C=C(C)C2CC2)=O)CC=C(C(=O)N2CCCC(C(C)(C)C)CC2)C1 C1(NC(C2CCCC(NC(c3c(N)cc(F)cn3)=O)C2)=O)CC2CC1C(O)C2O N1(C(C2(SC)CC2)=O)CC2CC1CC2NC(=O)CCc1cccc(C2CC2)c1 Cc1ccn2cc(C(=O)NC(C3CC(NC(c4cnnn4C)=O)C3)C)nc2c1C N1(C(C=C2CCC(C)C2)=O)CC2(C)CN(C(C3CCC(=O)N3)=O)CC2(C)C1 CC(C)CC(CC(=O)NCC1OCCC1(C)C)NC(c1c[nH]c2cnccc12)=O C(=O)(C1CCc2cccc(F)c21)NC(C)CCNC(c1cnccn1)=O c1(C(=O)NCC2=CCN(C(C(C(C)C)C)=O)CC2)c(F)ccc2ccncc12 C(N=c1[nH]cc2ccnc-2[nH]1)C1C(C)CCN(C(c2cccc(OC)n2)=O)C1 c1(N2CCC(C)(c3ncc[nH]3)CC2)nc(N2CC3CC3C2)nc2ccccc12 c1(C(N2CC(NC(=O)CCn3ccc(O)nc3=O)C2)=O)c(F)cccc1[N+](=O)[O-] C1(NC(C2CC(CC)C2)=O)CCC2CC1CN2C(=O)Cn1nc(C)ccc1=O C(=O)(C1CCCc2cncn21)N(CCCN(C(C1N(C(C)=O)CCOC1)=O)C)C c1(C(=O)NC2(C3CN(C(C4(COC)CC4(F)F)=O)C3)CC2)nccn2nc(C)cc12 N1(C(C(C)OCC)=O)CCC(=CCNC(=O)COCCc2ccc(C)cc2)CC1 N1(c2cc(NCC(C)CC(C)O)nc(COC)n2)CCc2sc(Br)cc2C1 c1(CCOC)cc(=NC(=O)NC(c2ccccc2)c2ccc(C)s2)[nH]o1 O=C(C1=CCCN(S(=O)(=O)Cc2ccc(F)cc2F)C1)Nc1cc(Cl)cc(Cl)c1Br c1(C(N(C2CCCCC2NC(C2CCC(F)(F)CC2)=O)C)=O)cc2scnc2[nH]1 C1(C(=O)NCCS(C)(=O)=O)(CC)CCCN1C(C1CC(SC)C1)=O Cn1cnc2[nH]c(=NCC3(C)CCOCC3)nc(C(F)(F)F)c12 N1(CC)CCC2(CC1)CN(C(=O)C(C)(C)c1csc(C)n1)C2.C(=O)(CC)OO CC1(F)CCC(C(N2CCCC(C)(NC(c3ccnc(Cl)n3)=O)C2)=O)CC1 c1(CNCCCSC(c2nnnn2C2CCOCC2)C)ccnc(Cl)c1 C#CCC(C)(CC)C(=O)N(C)CC1CCCN1C(=O)C(C)=CCC C12(CCNC(=O)OC(C)(C)C)CCC1CN(C(=O)C(c1ccc(F)cc1)(C)F)C2 C1(CNC(C(C)CF)=O)N(C(=O)CC(c2cccs2)C2CC2)CCC1(C)C N1(C(C(C)=CC)=O)C(C(=O)NC2CONC2=O)CC2CCCCC12 c1(CC(N2CC(OC)(CNC(=O)CC3(C)CCOC3)C2)=O)cn2ccsc2n1 N1(C(C(C=C)OC)=O)CC2CC2(CNC(C2(C)COC2)=O)C1 c1(CC(=O)N(CCC(=O)NCC(C)OC)CC)ccn(C)c1 C1(NC(CCc2c(C)noc2C)=O)CCN(C(=O)COc2ccsc2Cl)CC1F C12CC=CCC1NC2=O.C(C(=O)NCCSCCCO)N(C)C(N)=O C(=O)(CC(CC)C(C)C)N1CCC(C(=O)Nc2cnc(CCC)nc2)C1 N1(C(CSc2c(C)n[nH]c2C)=O)CCC(C(=O)NC23CC(F)(C2)C3)C(C)(C)C1 CC(C)C(C#N)C(=O)NC(C1CCCN1C(=O)C(=O)C=Cc1ccccc1)C C(=O)(C1=CC2CCCCCCC12)NCCC1(NC(COCCCC)=O)CC1 c1(C(=O)NC(CCC)CNC(=O)C(COC(C)C)NC(C)=O)cncnc1C c1(COC)ncc(CNC(=O)C=CCNC(=O)C=CC(F)F)[nH]1 Cc1c(NCCN(C)C)nc[nH]c1=NCc1nc(-c2ccc(Cl)cc2)n[nH]1 C(=O)(CCCCCc1cccs1)NC1CN(C(c2cc(CC)c(C)s2)=O)C1 c1(CC)cc(F)ccc1C(=O)NCC(CNC(c1ccc(C(C)C)s1)=O)OC Cc1csc(=NCC(=O)N2CCCC(C)(NC(C3(C4CCC4)CC3)=O)C2)[nH]1 C1(Nc2cc(C(=O)OC)no2)CCN(C(=O)CN2CCN(C(C)C)CC2)CC1C c1(C(C2CC(O)C2)N(CC(O)CNC(=O)C=CC(C)(C)C)C)nnc(O)n1C C1(NC(=O)C2CC2)CCN(C(=O)Nc2nc(N3CCCCC3)no2)CC1 N1(C(COC(CC)C)=O)CCC(CO)(CNC(C23C=CC(CC2)C3)=O)CC1 CCC(F)C(=O)NCCC(Cc1ccccc1)NC(C1CC(=O)N(C(C)C)C1)=O CN1CCC(C(=O)NCC2CC2CNC(=O)Cc2csc(=N)[nH]2)CC1=O c1(CC(=O)NC2C3CN(C(C=CCOC)=O)C2C3)c[nH]c2cc(Cl)ccc12 N1(C(c2ccc(OC)nn2)=O)CC(N(C(=O)CC2CC=CC2)C)C2(CC2)C1 C1(C(=O)NCCCc2onc(C)n2)CC=CCN1C(=O)CC1CCCCN1C C(CCCCC=O)N(C(C(C)=CC=C)=O)C(CC#CC(F)(F)F)=O.NCC C(=O)(C1OCCn2ccnc21)NC(C)CN(C)C(c1cc2c[nH]nc2s1)=O Cc1[nH]c(=N)nc(O)c1CC(=O)NC1CC2CN(C(=O)CC(F)(F)F)CC12 N1(C(c2c(C)n[nH]c2)=O)CC(F)CC1C(=O)NCC1CC1[N+](=O)[O-] CC1CN(C)CCC1N(C)C(C1CCC(NC(c2ccnc(O)c2)=O)CC1)=O C(CN=c1ccc2c([nH]1)CCCC2)C1CCN(C(C(C)(C)O)=O)CC1 N1(C(C2(CC)CN(C(=O)CNc3cccnc3)C2)=O)CC2(CC2)CC1C c1(C(=O)NCC2N(C(C3C(C)=C3)=O)CCC2)ccc(C)c(S(=O)(=O)N(C)C)c1 N1(CC(=O)Nc2c(OC)cc(I)cc2)CCc2cccnc2C1 C12(NC(c3c(C)n(C4CC4)nc3)=O)CCCCC1CN(C(=O)CCP(C)(C)=O)C2 C1(C(=O)NCC(=O)NC(C)Cc2ncon2)CC2CC2C1 c1(CNC2CCC2NC(=O)NCC(COC)OC(C)(C)C)cccnc1 C1(NC(C(C)OCC#C)=O)CC2CC1CN(C(=O)C(C)OCC1CC1)C2 c1(C(=O)OC)n[nH]c(=NC2C(C)CN(C(=O)C(C)(C)S(C)(=O)=O)CC2C)s1 N1(C(C(CCC)C#N)=O)CCC2CCN(C(c3ccc([N+](=O)[O-])s3)=O)C2C1 CC(=O)CCCCC(=O)N1CCC(OCCNC(c2c(C)cccc2F)=O)C1 c1(C(=O)NCCOCCN(C(C2C(C)CC2)=O)C)ccc(CCC(N)=O)cc1 Cc1cccc2c1c(CN1CCN(C(=O)Nc3ccns3)C(C(F)(F)F)C1)cn2C N1(C(C(CCNC(Cn2nc(C)oc2=O)=O)O)=O)CCC2(CC1)CSC2 C#Cc1cccc(C(=O)NC(=O)COCCSC)c1.C(C(C)O)N(C(=O)CO)CC(F)F N1(C(C(C=C)OC)=O)CC(CCNC(c2cnns2)=O)OC(C)C1 C1(NC(CCCC)=O)CN(C(c2cc(C)n(CC3CCCC3)n2)=O)CCC1CO C#CC1CCCCN1C(=O)CC(=O)NCCNC(=O)C1=CCCOC1 C(=O)(C(C(C)(C)C)NC(C1C2COCC12)=O)NCc1ccc(OC)nc1 CCC(C)C(C(=O)N(C)Cc1ncco1)NC(C1C(C)(C)C1(C)C)=O CC1(C)COCC1C(=O)NC(c1ccccc1F)C(=O)NC(C)(CO)C1CC1 C1(NC(C(CCN(C)C)NC(=O)CC2CCC(=O)CC2)=O)CN(C)C(C)(C)C1 Cn1nc(Br)cc1C(N1CC(NC(c2ccncc2)=O)C(CC2CC2)C1)=O C(=O)(C1=NNC(=O)CC1)NCCCOCCCNC(c1cc(C#N)no1)=O C1(COC)CCCN1C(=O)CC(C)N(C(=O)Cc1cccs1)C N1(C(COCC=C)=O)CCC(C)(NC(=O)CC2CCCCCC2)C1 c1(CC)cc(C)nc(NC2CCC(NC(=O)CC3CCCCC3C)C2)n1 c1(CC(=O)NC2CC(NC(C3CCCO3)=O)C2)cc2nc[nH]c2cc1Br c1(OC)ccc(CC(N2CC3CCC2CN3CC(N)=O)=O)cc1[N+](=O)[O-] Cc1cn2cc(C(N3CCCC3CCCNC(C3CCCN(C)C3)=O)=O)nc2s1 C1(OC)(CNC(=O)C=CC2CCCC2)CCN(C(=O)CC2CCC2)C1 CCS(=O)(=O)CC(=O)N1C(C(=O)NC(CCO)C(C)C)CC2CC12 c1(C(N(C)CC2(NC(C3CCCC(CC)C3)=O)CC2)=O)cc(C)ccc1O C(=O)(CCC(=O)NCCC1(C(N2CC(OC)(OC)C2)=O)CCC1)NCC.C(=O)NC c1(CC(=O)NC)ccccc1NC(C1(NC(=O)CC2CCCC(=O)N2)CC1)=O CCCS(=O)(=O)CC(=O)N1CC(NC(=O)COc2ccc(Cl)c(Cl)c2)CC1(C)C c1(SCC)cnccc1C(=O)NCC(C)N(C(=O)CCC1CCCCN1C)C CC(C)CCC(O)C(=O)N(C)CC1CCCN1C(c1cccc(C(C)(C)C)c1)=O N1(C(C(c2ccc(C)s2)C)=O)CCC2C(C1)CN2C(c1cn(C(C)C)nc1C)=O C(=O)(C(CO)C(C)(C)C)N1CCNC(C)C1.C1(C(C)=O)(N2CCC2)CC1C(F)(F)F N1(C(C(c2n(C)ncc2)NC(c2cnsn2)=O)=O)CCCC2(CC2)C1 c1(C(=O)NC2CC(CNC(CCC(=C)C)=O)C2)cccc2sncc12 c1(-n2ncc(NC(C(CC)(C)F)=O)c2)ccc2c(c1)OCO2.N12CCCC1C2=O c1(N2CC(=O)NCCC2)nc(N2CCC(OCCF)C2)c2c(n1)CSC2 C1(C(=O)NC2CC(C(F)F)(NC(C3CCCOC3)=O)C2)CCC2CC1CO2 N1(C(C(C)(C2CCC2)NC(c2c(CC)cccn2)=O)=O)CC(C2CCCCC2)C1 C(=O)(C(C)C(C)(C)C)N1CC(c2c(CNC(c3c(C)cn(C)c3)=O)nco2)C1 C1(CN(C(=O)C=C(C)C(C)NC(=O)C(c2cnn(C)c2)C)CC)CCC(=O)N1 c1(Cn2c(=O)n(C(C(C=C)CC)=O)c(=O)n2-c2ccccc2)ccc2c(c1)COC2 O=C(C1=C(Cl)CCOC1)NC1CCNCC1 C(=O)(CCCCC(F)(F)F)NCC1OCC(C(=O)NC(c2cnc(OC)s2)=O)C1 N1(C(c2n(CCCC)ncc2)=O)CCC(C)C(NC(c2ncc(C(F)F)s2)=O)C1 C1(C(N2CCC(C)(OC)CC2)=O)CCc2ccnn2C1 C1(C(C2CCCC3(CC3)C2)=O)CC2CC(C1)NC2.CCCCCN(CCC(=O)NC)C CN=C1NCCCc2nc(no2)CNC(=O)N2C(CCC2)CN1.C(C)(C)(C)OCC C12(OCC(=O)NCCOC3CN(C(c4nc[nH]n4)=O)C3)CCCCC1C2 S(=O)(=O)(CCC(=O)N1CCCC(N(C)C(c2sc(CO)nc2C)=O)C1)NC C(=O)(C(C)(C)CC(=O)OC)N1CC(NC(CN(CCCCCC)C)=O)C2(C1)CC2 C1(C(=O)NC2(CSC)CCC2)CCC(C)N(CC(C)C)C1 S(=O)(=O)(c1cccc(CNC(=O)NC2C3CC3C3CC23)c1)NCCC N1(C(C(C(C)C)C(C)C)=O)CCC2(CCC(NC(=O)CC(C)n3cccn3)C2)C1 N1(C(C(C)Cc2ccc(C#N)cc2)=O)CCCN(C(=O)Cc2cnsc2)CC1C CC(C)CC(C)CC(=O)N1CCCC(C)C1CNC(=O)CC1(C)CCCCC1 C1(NC(c2cccn2C2CC2)=O)CC2CC1N(C(C1CCC1)=O)C2 N1(C(C(CC)N(CC)CC)=O)CCN(C(c2ccncc2F)=O)C(C2CC2)C1 Cc1cn2ccc(C(N3CC4CC(NC(=O)C(F)n5ccnc5)C3C4)=O)cc2n1 C1(COC)(NC(=O)Cc2cc[nH]n2)CCN(C(c2nccnc2C(N)=O)=O)C1 Cc1cc(C)n(CCCC(=O)NC2CCN(C(=O)Cn3ccnn3)C2)n1 N12CCN(CC1)C(=O)N2.c1(NC(C)Cc2nncn2C)cccc(Cl)c1 c1(NC2(c3n(CCSC)nnn3)CCC2)cc2n(n1)CC(O)CO2 CCCC(C)CCCC(=O)NC1CC(CCNC(c2c(C)nsc2N)=O)C1 c1nc2ccsc2c(=NC2CCCSCC2)[nH]1.Cc1cn2c(n1)CNCC2 Cc1ccc(C(=O)N(CCNC(=O)C(CC(C)C)n2ccnc2)C(C)C)c(O)n1 c1(OC)ccc(OC)c(CC(N2CC(NC(=O)CC3COC(=O)N3)C(C)C2)=O)c1 C12(CNC(C3(C)CCCC3)=O)CC(C1)C(NC(C1(C)CC=CCC1)=O)CO2 c1(C(=O)NC2CC(C(N3CC(C)OCC3C)=O)C2)cnc2ccoc2c1 CC1OCCOC1C(=O)NC(C(=O)NCCC(C1CC1)C1CC1)C1CCCO1 C1(CCCNCCCCCF)CCOC2(CCC2)C1 C(=O)(C(C)CC(C)(C)C)N1CCC(C)C1CNC(c1ccnc(C(F)(F)F)c1)=O N1(C(C(C)C2CCC2)C(=O)NC2(C)CC2)CCCC(c2nn(C)cc2I)C1 Cc1cccn2nc(C(=O)NCCC3CC3C)cc12 C12(CCCC1)CC(=O)N(C1CC1)CCNC2=O.n1(C2(SC)CC2)cncn1 CCC(C(=O)NCc1nocc1C(=O)NCC1CC1(F)F)NC(N)=O CC1CN(CCNc2ccn(-c3ccc(F)cc3)n2)CCN1Cc1ccccc1 C1(COC)(CNC(=O)C(C2CCCCC2)O)CCCN1C(c1ccnc(C)n1)=O C(C(C)C)(C(O)C(=O)N1CCCC1CCNC(C1(C)CCN(C)C1)=O)OC C1(CC=C)(C(=O)N(CCC2CC2)CC)CCN(C(=O)Cc2ncccc2C)C1 C1(CC(=O)NC2CN(C(COC(C)C)=O)CC(C)C2)COc2ccccc2O1 CCCCC(CC(=O)NCCCO)NC(=O)C(C)(O)C(C)(C)C c1(C(=O)NCC2N(C(CCNC(c3ccncc3)=O)=O)CCC2)ccc(F)cn1 c1(C(=O)NCC(CC=C)NC(C2CCS2(=O)=O)=O)cc(C(F)(F)F)cn1C N1(C(CC=C)=O)CCSCC1CCNC(=O)Cc1ccoc1 CN1CC2CN(C(c3c(Br)cc(Br)c(O)c3Br)=O)CCN2C1=O c1(Cn2cc(CCN(C(c3nc(Cl)ccc3Cl)C)C)nn2)nc2c(s1)CCCC2 C1(C(N2CCCCC(NC(=O)COC3CCOC3)C2)=O)CCCC12CCOCC2 C1(C(=O)NCC#CCNC(C2(C)C(CC)CCC2)=O)CCCCN1S(N)(=O)=O C1(C(N2CC(OCC)C(CNC(C3CCCC3CC)=O)C2)=O)CC(C(C)C)=NO1 CC1(CNC(c2csc(-c3ccsc3)n2)=O)CCCN1C(C1CC1F)=O CC(C)(O)CC(=O)N1CCC(C)(NC(c2cc(-c3ccccc3)ccn2)=O)C1 N1(CCC(c2ncc(F)cc2F)NC(C2CCOCC2)=O)CCN2C(=O)CCC2C1 c1(-c2n(C(C(C)C)C)nc(-c3ccc(Cl)cc3)n2)ccc(F)c(F)c1 C1(C(=O)NC(CC=C)CNC(c2cccc(F)c2Cl)=O)CCc2ncsc2C1 C1(C)(OC)CC2CC1CC2CNC1(c2nnnn2C2COC2)CC2C=CCC12 C1(OC)CCC2(C(=O)NCc3c[nH]nc3C(=O)NOCC(O)CO)CC12 N1(CC(=O)N(C2(N)CN(C(=O)CC(Cl)Cl)C2)CCCCl)CCC(O)CC1 N1(C(C(C)(C)c2ccccc2)=O)CC2CN(C(c3cccc(O)c3Cl)=O)CC12 Cc1ccnc(C)c1CNC(=O)C1=CCC(NC(C2CCNC(=O)C2)=O)C1 c1(NCC(=O)NCC2(CCNC(CC3CCC(C)C3)=O)CCC2)cc(Cl)ccn1 C1(C)(C(=O)NCc2ccc(C)nn2)CC(O)CN1C(=O)C=Cc1ccncn1 c1(OC)ccc2c(CC(N3CC(CC4CC4)C4(CCC4)C3)=O)coc2c1 C1(C(N2CCC(C)(NC(CC(=C)Br)=O)CC2)=O)CC2CCC1CC2(F)F C(=O)(C(C)(C)C(F)F)NC1(CO)CCN(C(C2CN(C)C2)=O)C1 C(C(C)(C)CNC(=O)Cc1csc(S)n1)N(C)C(C1CC1[N+](=O)[O-])=O C1(NC(CC(c2c(C)nn(C)c2C)CC)=O)CC1C1CCCN(C(=O)CCC#N)C1 N1(C(C(CC)O)=O)CCC(C)(NC(=O)C(C)(C)Oc2ccccc2)CC1 C1(CC=C)(C(=O)NCCCC(=O)OC)CN(C(=O)CC2COCCO2)C1 Cc1c(NC(C2C(CNC(=O)CCCC3CC3C)C2(F)F)=O)cccc1F O=C(C1Cc2c(Cl)cccc21)NC1(CNC(C2Cc3nccnc3C2)=O)CCC1 C12(NC(c3sc(C)c(O)n3)=O)CCC(CNC(=O)CC3CCCC3O)(CC1)OC2 C=C(Cl)C(C)(C)C(=O)N1CC(NC(=O)CC2(CO)CCN(C)CC2)C(O)C1 CC(CC1CCCO1)N=c1ccnc(N(c2cc(F)ccc2F)C2CC3(CC3)C2)[nH]1 C1(C(=O)NCCN(C(C(c2ccccc2Cl)C)=O)C)CCCCC(=O)C1 C1(NC(C(CN(C)C)O)=O)CC(F)CN(C(c2c[nH]c(Br)c2)=O)C1 N1(C(C2C(C)CC2)=O)CC2(CCC(CNC(c3cc(F)cc(F)c3)=O)O2)C1 C(=O)(C(C)(O)C(F)(F)F)NC1C(C(=O)NC(C(=O)OC)C)CCC1 C1(C(=O)NCCSC)CN(C(=O)C(N2CCOCC2)C)CCC1O C1(C(N(CC(C)NC(C2CSCCS2)=O)C)=O)OCC2CCCCC12 N1(Cc2cccc(OC)c2)CCC(NC(=O)C(C)Oc2nnc(CO)o2)C(C)C1 CCCCC(C)C(=O)NCC=C1CCN(C(c2cnc(O)n2CC)=O)CC1 C1(C(=O)NC2CCC(CNC(CC(=C)C)=O)CC2)CC2CCCCCCC12 N1(C(c2c(C)snc2)=O)CCCC1(C)C(=O)Nc1cccnc1 CC1(C)NC(=O)CC1C(=O)NCC1CN(C(=O)Cc2cc(C3CC3)on2)CCO1 N1(CC(=O)NCC2C(OC)(OC)CC2)CCCC(C)(NC(C)=O)C1 C1(C#N)(C(N(CCCC(=O)N2CC(n3ccnn3)C2)C(C)C)=O)CC12CCC2 C1(NC(=O)Nc2c(C)onc2Br)CCC(C)N(C(=O)OC(C)(C)C)C1 c1(COC)cc(C(=O)OCC2(C)CCCO2)cs1 C(=O)(C#CC1(C)CC1)NCC1C(CC(C)(O)C2CN(C(CC(CC)SC)=O)C2)C1 Cc1cc(F)ncc1C(=O)NC1CCN(C(=O)COc2cc(F)cc(F)c2)CC1 c1(SC)c(Cl)cncc1Cl.c1(NC(CN(C(C)COC)CCC)=O)ccccc1Cl N1(C(c2cc(C)c(C(F)F)cn2)=O)CCC(C2CC(NC(=O)COC3CC3)C2)C1 C(C1=CCN(C(c2occ3c2CCC3)=O)CC1)NC(C1(O)CCC(CC)C1)=O C1(C)(C(=O)NC(C2CCOCC2)C#C)CC(O)CN1C(=O)C(C)=CC1CC1 c1(C(N(C2CCCN(C(C(CC)OC)=O)C2)CC2CC2)=O)ccn2ccccc12 c1(C(N2CC(O)(C(C)NC(c3csc(CO)n3)=O)C2)=O)cc2ccccc2nn1 N1(C(c2ccc(C)cc2)=O)CCC(O)C(C(N2CCC(O)C(CO)C2)=O)C1 n1(C(C)C)ncc2c(NCC(C)C(C)C)[nH]c(=NC(C)c3ccccc3Cl)nc12 C1(C(=O)NC(c2n(C(C)C)ncc2)C)CCCN(C(C2CCC(=O)N2C)=O)C1 c1(C(N(CC(F)(F)F)CCC=C)=O)ccncc1C1=CCC(C(C)(C)C)CC1 C(=O)(CCC(=O)NCC1CCCN(C(c2n[nH]c(C)c2C(F)(F)F)=O)C1)OCC Cc1cccc(CC(N2CCC(NC(=O)CCC(F)F)C2C)=O)c1 n1(Cc2cn(CC(=O)NC3CNCC34CCC4)nn2)cnc2cccnc12 C1(C(=O)NC(C=CC(=O)N(CC(C2CC2)OC)C)(C)C)CCC(C)O1 c1(C(=O)NCC2N(C(C3(CC=C)CCC3)=O)CCCC2)nc(C)n(C)c1C c1(OC)ccc(C(N2CCN(C(C3CC3F)=O)CC2)=O)c(F)c1 C#CCC(C)(C(=O)NC(C)CC(C)CC)NC(=O)CCOC1C(OC)CCC1 N1(C(c2cn(C)nc2O)=O)CC(C)(C)CC1CNC(=O)CCNC(=O)C=CCl C1(C)(NC(c2ccc(C(=O)NCCCCC(=O)OC)nc2)=O)CCCCCC1 c1(C(c2n(CCOCC)nnn2)NC(C)CCOCC)ccc(Cl)nc1Cl c1(OC)ccc2c(c1)CC(C(=O)NC(CO)C(C)NC(=O)Cc1sccc1C)O2 Cc1oc(-c2cnn(C)c2)nc1CN1CCC1CO c1(CN2C(C(=O)Nc3c(C(CC)C)cccc3)CC2)c(OC)ccc(Br)c1F N1(C(c2cnc(S)nc2)=O)CCC(F)(C(N2CCC(OCCF)C2)=O)C1 C1(NC(C2(C)CCC2)=O)C=CCN(C(c2cnn(C(C)(C)C)c2N)=O)C1 c1(C(=O)NCC(CC)(C)NC(=O)Cn2cccn2)cc(C)c2c(c1)CCC2 N1(C(c2c(C(C)C)cco2)=O)CC2CCC2(NC(C2CC2(C)C(F)F)=O)C1 N1(C(C(=O)NC)=O)C2CCC1CN(C(c1cn(C(F)F)nc1C(F)F)=O)C2 c1(C(=O)NC(CC=C)CNC(c2ccnn(C)c2=O)=O)cccc2c1nnn2C C1(CCOC)(NC(C2CN(c3nncs3)C2)=O)CCN(C(=O)CC2(C)CC2)CC1 N1(C(C2=C(C)CC2)=O)CC(C(N2CCC(C3CC3)C2)=O)CC12CCC2 C1(CCC)CCCCC1C(=O)NC(C)(C)CNC(=O)CC(C)(C)c1cccs1 C1(C(=O)NCC2CCN(C(CNC=O)=O)C2)CC(O)CN1C(c1ccccn1)=O C12(C(=O)NC(C3CCCN3C(C3(N4CCCC4)CCC3)=O)C)CCC(CC1)OC2 c1(C(=O)NC2(C)CCCN(C(CC(C)F)=O)C2)cc2cc(Br)cn2cn1 C1(C(N(CC(=O)NCC)C)=O)(C(C)C)CCN(C(=O)CNc2c(C)csc2C)C1 N1(C(C(F)=CC)=O)CCOC(CCCNC(C2CC(=O)N(C)C2)=O)C1 N1(C(c2c(CC)nns2)=O)CCC2(CC1)CC2NC(C1(OC)CCCCCC1)=O C1(CNC(c2cc(SC)oc2)=O)CN(C(=O)C=C(C)C)C2(CCC2)C1 C1(CNC(C2C(C)C2)=O)CN(C(c2cc(C(=O)OC)nn2C)=O)CCC1(F)F CC1(C)COC(C(=O)NCC2CCN2C(=O)COC2CCCCCC2)CO1 n1(CCCSC)nnnc1C(c1ccn(C(C)C)n1)NC(C)CCC1CCCCC1 C1(NC(c2c(C)nn(C)c2)=O)CN(C(C2(COC(C)C)CC2)=O)CC1C1CC1 C(=O)(C(O)CCC(C)C)N1C(CN(C(c2noc(CC)c2C)=O)CC)CCCC1 c1(NC(=O)NCC2OCCN(C)C2c2ccccc2)cccc2c1CCCC2 c1(C(N2CCN(C(=O)C(C3CCCCC3)F)CC2C2CC2)=O)ccnc2[nH]ncc12 C1(C(=O)OCC#CCNCC)CN(C(c2cccc(C)c2)=O)CC1O N1(C(C2(CNC(c3cc(C)c(C)nn3)=O)CC(C)(C)C2)=O)CCCC(C)(O)CC1 c1(C2(CC3CCCO3)CCC2)ccc(F)cc1F.c12ccnc(n1)NCCN2C c1(OCC(=O)NCCC(C)NC(CC(C)C)=O)ccc(F)cc1O c1(NC(C(CCNC(COC)=O)(C)C)=O)c(F)cc(OC)cc1F.C12CN(C1)C2 C1(C(C)=O)CC(C(=O)NCC(C)CNC(=O)CC2(CSC)CC2)C1(C)C Cc1cn(C)cc1C(=O)N(C(C(=O)NCc1ncc[nH]1)C1CC1)C C(CC(C)C(=O)NCCOCCCN(C)C(c1cccc(O)c1)=O)OC Cc1cc(CNC(C2CCN2C(c2cnc(Cl)n2C)=O)=O)cc(C)c1 c1(CCC(=O)N(CC(C)O)CCNC(C(C=C)(C)O)=O)cccc(F)c1Cl N1(C(Cc2c(C)cccc2)=O)CCCC(C)(NC(c2ccc(Cl)nc2Cl)=O)C1 C1(C(N2CC(N(C(c3c(C)c(Br)sc3)=O)C)C2)=O)SC2C=CC1CC2 C1(CC(=O)N(C(C2(CCO)CC2)C)C2CC2)CCCC(=O)N1.C1(=O)CN1 c1(N2CC3C(C(N4CCC(O)C(O)CC4)=O)C3C2)ccc2ccc(Br)cc2n1 c1(C(=O)NCCN(C(C2CN(C3CCCCC3)C2)=O)CC)sccc1Cl C1(C2CC2)(NC(c2c(CNC(c3ccc(C)s3)=O)noc2)=O)CCCC1 c1(C(=O)NC2CCC(C(=O)NCC3C(=O)OCC3)C2)cccc2nccn12 c1(CC(=O)NCC2C=CCN2C(c2cc(C3CC3)on2)=O)ccc(F)cc1 C1(C(=O)NCCCN(C(=O)C=CC(C)(C)C)C)CCc2ncncc2C1 c1(NCC(C)(C2CC2)NC(c2cc(C3CC3)on2)=O)ccc([N+](=O)[O-])cc1C#N C1(C)(CNC(C2N(CC)CCOC2)=O)CN(C(=O)C(c2cnn(C)c2)=O)CC1C C1(CC(N2CC(CCNC(C(C)=C(CC)C)=O)C(C)C2)=O)CCCNC(=O)C1 c1(C(N(CCCCN(C)C(c2coc(CC3CC3)n2)=O)C)=O)ccn2ccsc12 N1(C(c2n(C)ncc2C2CC2)=O)CCN(C(c2ccnc(Cl)c2Cl)=O)CC(O)C1 C1(CN(C(=O)Cc2ccon2)C2CC2)CCCN(C(=O)CCc2nccs2)C1 N#Cc1csc(C(=O)NC2CCOCC2C(=O)NCc2cccnc2)c1 N1(C(CNS(CCOCC)(=O)=O)=O)CC(C)CN(C(c2nccn2C)=O)CC1C Cc1cc(C(N2CCC(CO)(NC(=O)C=CCN(C)C)CC2)=O)cc(C)c1N C(=O)(C1OCCc2ccccc21)N1C(C)CCC(NC(CC(CCC)O)=O)C1 C(=O)(C(O)CCCCC)NCC1(F)CC(CNC(C2C(=C)C2)=O)C1 S(=O)(=O)(c1cccc(=NCCCc2nc(C(F)F)n[nH]2)[nH]1)NC(C(C)(C)F)(C)C c1(SCCC(=O)NCC(C2CC2)NC(C2(CO)CC2(F)F)=O)ccccc1 S(=O)(=O)(c1[nH]c(=NCc2cncs2)ccc1Br)NCC(CC)(CN(C)C)CC C1(COC)CN(C(C2CN(C(C)=O)CCO2)=O)CCN1C(c1c(Cl)cnn1C)=O C(=O)(C(C)(C)C1CCN(C(=O)C(C)NC(=O)C(C)(C)C)C1)N(CCOCC=C)C c1(CN2CC3C(CNC(c4c(C)nc(CC5CC5)o4)=O)C3C2)nc(Cl)ccc1Cl C1(S(C)(=O)=O)(C(=O)NCC2(NC(CC3C(C)(C)CCCC3)=O)CCC2)CCCC1 c1(NC(CC)(C)C(F)(F)F)ccc(S(=O)(=O)NCCOCCN(C)C)cc1C#N C1(NC(C2CC(OC)C2)=O)CCC(C)(NC(=O)CCC2NC(=O)NC2=O)CC1 N1(C(C2CN(C(C3=CCCCC3C)=O)CC23CC3)=O)CCC2(C1)CC2(F)F C(=O)(C1Cc2ccccc21)NC1C(NC(C(CC(=O)N(C)C)(C)C)=O)CC1 C1(C(=O)NCCCN(CCCNC(C2CCCC2)=O)C)CCCC12CC2 CC1C(C(=O)NC2(CCO)CCOC2)CCN1C(=O)C(C)c1cccs1 N1(C(COCCCCCC)=O)CCC(C(O)CNC(C2(CO)CCOC2)=O)CC1 N1(C(C2CC2(F)Cl)=O)CC2(CO)CC1(C(=O)NCCc1ncccc1F)C2 C(CCCCC(=O)N1CCC=CC1C(=O)N(C1CC2CC2C1)C)OCC C1(OC)CCC(C(N2CCCC2C2(O)CN(C(C3CN(C(C)C)C3)=O)C2)=O)CC1 C(=O)(CC(C)(C)CC)N.C(CC(O)C(C)(C)C)c1nnc(C(CCCC)CC#N)o1 CC(C)(CC(=O)N1CC2(CCCC(CNC(c3ccoc3)=O)O2)C1)CC(F)(F)F N1(C(C(C)n2ccnn2)=O)CC2(CO)CC1(CNC(c1ccoc1)=O)C2 Cn1c(C(=O)NCC2CCCN(C(=O)CN3CC=CC3)C2)ccc1[N+](=O)[O-] C1(CNC(C2(SC)CC2)=O)CN(C(c2ccon2)=O)CC12CC2 C(=O)(C=CCCCC)NCC(CCCC)NC(=O)CNC(c1ccc(F)cc1)=O C(=O)(C(F)(CNC(C1CNC(=O)N1)=O)C(C)C)N1CCC(CCCC)CC1 CC(C)C(CNC(=O)NCC(C1CCCCC1)CO)C(C)C C1(C(N2CCC(N(C(=O)C#CC(C)(C)C)CC#C)C2)=O)OCC2CCCCC12 c1(NC(C)=O)cnc(C)c(C(N2CCC(NC(=O)CC3(C)CC3(F)Cl)CC2)=O)c1 N1(C(CC2C(OC)CC2)=O)CCN(CCN(C)C(C2CCCN2C(C)C)=O)CC1 N1(C(C(COC)OC)=O)CCC(COC)(NC(C2Cc3nccn3C2)=O)CC1 c1(OC)cc(Cl)ccc1-n1nc2nc1C2.C1(OCc2nnc(C)s2)CCCCO1 c1(CC(=O)NC(C)C=CC(=O)N(C)CCF)cccs1 CC1(C)CN(C(c2cc[nH]c2C2CC2)=O)CC1NC(c1cncn1C1CC1)=O c1(C(=O)NCC(C(C)(C)C)NC(CCC=C=C)=O)nn2cccnc2c1Cl c1(C(=O)NCC2CN(C(=O)CC3CCOC3)CCO2)cc2c(Cl)cccc2s1 C(C)(CO)(C(=O)NC(C)CNC(c1cccc(OC2CCC2)c1)=O)OC N1(C(C2C(C)CCO2)=O)CC2CN(Cc3occc3Br)CC2C1 C1(NC(c2n(CC)nc(C(F)(F)F)c2)=O)CC(O)CN(C(=O)CC2CC(C)C2)C1 N1(C(C(F)=CC)=O)CCC(C(C)(O)CNC(=O)CCC23CCC(CC2)C3)CC1 C1(C(N2C(C3(C(=O)NCc4c(C)csc4)CC3)CCC2)=O)CC2COCC2C1 CCCCC(Cc1cn(-c2cccc(OC)c2OC)nn1)CCC O=C(NNC(=O)NCc1cnc(Cl)cn1)c1ccccc1Br c1(C(=O)NCCN(CCCN(C)C)C(c2c(C)ccnn2)=O)cnc(Cl)c(N)c1 C1(CC(=O)NC(c2cnc[nH]2)C)COCCN1C(c1cncc(C(F)(F)F)c1)=O N1(C(C2CCN(C(CC3(CSC)CC3)=O)C2C)=O)CCOC(C#N)C1 N1(C(C2CC(C)(CC)C2)=O)CCC(CO)(NC(c2sc(C)nc2C(C)C)=O)CC1 C1(OC)CC2CC(NC(=O)C=CC3CCN(C(=O)CSC(F)(F)F)CC3)CC12 C1(C2CCC2)(C(N(CCCOCCNC(C(CC)N(C)C)=O)C)=O)CCC1 C(C(C)CC(=O)Nn1cnn(C)c1=S)NC(CCOCCSC)=O c1(OC)ccc(CCC(N2C(CNC(C3(OC)CC3)=O)CC3CC23)=O)cn1 c1(COC)nc(C)c(C(N2CCCC2C(C)NC(C2(O)CC2(C)C)=O)=O)s1 O=C1NC(=O)C2CN(C(c3cc(CNC(=O)C(O)C4CCC4)on3)=O)CC12 c1(OC)ccc(N(c2ccc(Cl)cc2Cl)C(C2CC(C(F)F)C2)=O)cc1F C(=O)(C(C)(C)C(=O)NC(C1(CNC(c2c[nH]c(C(F)(F)F)c2)=O)CC1)C)NC c1(OC)cc(Br)cc2[nH]c(C(=O)NC3CC3NC(=O)CCC(F)F)cc12 c1(C(=O)NCCCCC(C)NC(C2(CC)CCOC2)=O)ccc2c(n1)CCC2=O N1(C(C(CCC)F)=O)CCC2CCCC12C(=O)NCC1(C2CCC2)CC1 C1(NC(C(CC)(O)c2ccccc2)=O)CCN(c2ncccn2)C(C)C1 c1(C(N2CCCC(OC3CNC3)C2)=O)cc(O)ccc1I c1(N(C)C)ccc(Cl)cc1NCc1cc(-n2ccnc2)cc(F)c1 CC1CN2CCN1C(C(=O)NCC1CC(NC(=O)CC(C)(C)O)C1)C2 C1(F)(C(=O)NCC(CC)(C)NC(c2csc(Cl)c2)=O)CC=CCC1 O=C(C(O)C(F)(F)F)NCCCCC1CN(C(C2(N3CCOCC3=O)CC2)=O)C1 C(=O)(C1(O)CCCc2ccccc21)NCC(c1c(C)c(Cl)ccc1)O C1(C(N(C)CC2CCCN2C(=O)CC(C)(C)n2cnnn2)=O)CC2(CC(=O)N2)C1 c1(OC)cc(Cl)c(Cl)cc1C(N1CC=CC1C(N1CCC(O)C(F)C1)=O)=O c1(N2CCC(CC)C2)nc(N2CCn3nc(C(C)(C)C)cc3C2)nc2c1CSC2 C(c1ccc(Cl)cc1)=CC(=O)NCC1C=CC(NC(C(C)c2cc[nH]n2)=O)C1 C(=O)(C#CC1CCCOC1)NCC1N(C(c2c(F)ccc(N(C)C)c2)=O)CC1 c1(C(=O)NCC(CCC)C(=O)NCC(F)Br)ccc2n[nH]cc2c1 Cc1cccc(C(N2CCOC(C(=O)NCc3cnccc3Cl)C2)=O)c1C#N C(=O)(C(F)C(C)(C)O)NCC1CC(C(C(=O)N(CCC(N)=O)CC)F)C1 C1(N(C(c2ncc(OC)nc2)=O)C)CCCN(C(=O)C(C)OCCC(C)C)CC1 c1(N2CCCC(NC(C(C=CCCC)O)=O)C2C)ncnc2ccc(F)cc12 CCC1=C(C(=O)NC2CC2NC(c2cn3c(n2)SCC3)=O)CCCO1 c1(C(N(C(C)C(=O)NCCOC2CCOC2)C)=O)cscc1Cl Cc1ccc2c(N3CCN(C(=O)C(C)(O)CC(F)F)CC3)ncnc2c1 C1(NC(c2cc(C)c(C)[nH]2)=O)CC=C(C(=O)NCC(C)C2CCC2)C1 CS(=O)C=CC(=O)N(C1CC1)CC1CCN(C(C2(F)CCOC2)=O)CC1 N1(C(CC2(C)CC2(F)Cl)=O)CCC2CCC(NC(c3cc(Cl)nnc3O)=O)C1C2 N1(C(C(C)NS(CC)(=O)=O)=O)CCOC(C(C)NC(c2cnn(C)c2N)=O)C1 O=C(CCCn1ccnn1)NCC(C1CCOC1)NC(=O)Cc1ccon1 N1(C(c2c(COC)cco2)=O)CC2CCCCN2CC1CNC(=O)C=CCOC C(=O)(C(CNC(=O)C(O)CN(C)C)C(C)(C)C)N1CCCC(C#C)C1 N1(C(c2c(C)csc2Cl)=O)CC2OCCN(C(c3c[nH]c(=O)cn3)=O)C2C1 c1(CNC(C=CCN(C)C(C2CCSC2)=O)=O)ccc(Cl)cc1 N1(C(CCC2NCC(CCC#C)C2)=O)CCC(C=C)(C(=O)N)CC1.c1(C)ncncc1N CC(CC(=O)N1CCCC1C(C)(C)NC(=O)C=CC(F)(F)F)CC(F)(F)F c1(C(=O)OCCCC)ccc2c(Br)cccc2n1.c12nnc(o1)NC(=O)C2 C1(NC(C(C)CN(C)C)=O)CC(CNC(c2ccco2)=O)C1(C)C N1(C(Cc2c(C)scc2)=O)CCOC(CC(=O)NCC2CC(F)C2)C1 N1(C(c2c(CC)n[nH]c2)=O)CCC(NC(c2scc(C)c2Cl)=O)C(C)C1 N1(C(C(CC)CC)=O)CCCCC(NC(=O)CN2CCCCS2(=O)=O)CC1 Cc1ccc(C(=O)N(CC(C)NC(=O)C2=CCOC2)C)c(F)c1F C1(C(=O)NCCC(CC)CO)CN(C(=O)CN2CC3CC3C2)CC12CC2 c1(C(C)C)cc(C(=O)NCC2CCN(C(=O)C(C)NS(C)(=O)=O)C2)no1 C(C(=O)NCC1(C(=O)NOCC2(F)CCC2)CCCC1)(C(C)C)SC c1(C(=O)NCC(C)(C(C)C)NC(c2ccc(OC)cc2)=O)cnn2c1N(C)CC2 N1(C(COCCCC#C)=O)CC(CC(=O)NCCCOC(C)=O)CC1C C(C(C)(C)C(=O)NCCCCC(C)NC(c1cc(CN(C)C)on1)=O)SC C12(CNC(=O)CC3CCOC3=O)CC(CN1C(=O)CCC1CCCO1)C2 O=C(C1=CC2CCCC12)NCCc1ccccc1-c1ccc(Cl)cc1 C=C1COc2c(C(=O)NC3CC3CNC(c3ccncc3)=O)cnn2C1 C1(N(C(=O)CC2CC3(CC3)C2)CCO)CCN(C(=O)Cc2nc[nH]n2)CC1 c1(C(=O)NCCC2CC(NC(C3(OCC)CCOC3)=O)C2)cnc[nH]c1=N n1(C(C)(C)C)nnnc1C(C1CCC1)NC(C1CCCO1)c1cccs1 CC1CC=C(C(=O)N2CC3CN(C(c4cc(C#N)ccc4N)=O)CC3C2)CC1 Cc1nc(F)ccc1CN1CCCCC1C(=O)NCCC(C)C N1(C(CCN(C(C)=O)C2CC2)=O)CCCC1(C)C(=O)NCc1ccncc1C C(=O)(C1c2c[nH]nc2CN1C(=O)Cc1ccoc1C)NCc1c(C)cccc1 c1(C(N2CC(OC(C)C)C2)=O)ccnc(NC(=O)CNC=O)c1.C1CC1 c12ccc(cc1C(N)=O)c(=O)[nH]c(=O)c1c(cccc1)c(=O)[nH]2.C(CN(C)C)OC O=C1CC(=O)NC(C(=O)NC2(CC(N3CCOCC3CO)=O)CCCCC2)C1 c1(C(=O)NC23CC2CN(C(=O)Cn2nccn2)C3)ccc(S(=O)(=O)N2CCC2)o1 C1(O)(CNC(CS(N)(=O)=O)=O)CCN(C(=O)CCCc2cccs2)CC1 C1(C(N(C(CC)CC)CC)=O)CCN(C(=O)CSCC(=O)N(C)C)C1 N1(C(CC=CC)=O)CCC(N(C)C(C2CC(CC(C)(C)C)C2)=O)CC1 c1(C(=O)NCC2N(C(C3(C)N(C)CC(OC)C3)=O)CCCC2)c(O)ccc(Cl)c1F C(=O)(CCCCCCCCCO)NC(C)(C)CNC(c1cncc2ccsc12)=O C1(C(=O)NC(C(=O)NC)C2CC2)CCN(C(c2cc(C#N)c[nH]2)=O)C12CCC2 C#Cc1ccc(OCC(=O)NCC2(C)CN(C(c3cnn[nH]3)=O)CCO2)cc1 C1(C(N(CC(CN(C)C(c2ncoc2C(C)(C)C)=O)O)C)=O)OCCC1(C)C C(C1=CCN(C(=O)C2=CCCS2)CC1)NC(C(C)(C)c1ccccn1)=O C=CCC(C)(C)C(=O)N1CCC(CO)(CNC(C2CC2OCC)=O)C1 C1(NC(=O)CO)CCCC(CNC(c2csc(C(F)(F)F)c2)=O)C1 N1(C(c2c(C)con2)=O)CCN(C(=O)CC2CCOCC2)CC1CF C1(C(=O)Nc2cn(C)nc2)C2CCC(C2)C1NC(=O)Cc1csnn1 C1(NC(C(C)NC(N)=O)=O)CC(NC(=O)C=C(C)C(C)(C)C)C1(C)C C1(C(N2C(CN(C)C(c3ccc(Cl)o3)=O)CC(F)C2)=O)CC2(C1)CC(F)(F)C2 N1(C(Cc2ccc(OC)cc2)=O)CC2(C1)CN(C(C1(C)CC1Br)=O)CCO2 C1(OCC)(CNC(C2CC(CNC(C3CCCCO3)=O)C2)=O)CCCC1 C(C(F)(F)CCC(=O)N(C1CCCC(C)(C)C1)C)n1cc(C(C)OCC)nn1 CC1(C)C(CNC(=O)Cc2ccon2)CCN1C(c1ccc(Cl)cc1Cl)=O C(C1=CCCSC1)(c1n(CCC)nnn1)NC(C1CCCCC1)(C)C c1(OC(C)C(=O)N(CCCNC(C2SCCS2)=O)CCO)cccc(F)c1 c1(C(=O)NCC(N(C(CSCC)=O)C)C2CC2)ccc(-c2ccccn2)s1 C(=O)(CCCOc1ccccc1)NC1CC(NC(C(c2ccccc2)SC)=O)C1 CN=C(NCC=CC(F)(F)F)N1CN(C)C(=O)C1C CC1(NC(C2CCN(C(C3CCCCCCC3)=O)C2)=O)CCCC1(F)F c1(OC)ccn2cc(C(=O)NCC#CCNC(c3ccn(CC#N)n3)=O)nc2c1 C1(C(N2CC(C)(CC)C2)=O)CC(C)(C)CN1C(C1CC(=O)C1)=O C1(C(N2CC(NC(c3c(OC)ccs3)=O)C(CC3CC3)C2)=O)CC2(CCC2OC)C1 c1(CCC(=O)NCC#CCNC(Cc2nc(C)sc2C)=O)ccccc1[N+](=O)[O-] N1(C(c2ccn(C(C)(C)C)n2)=O)CC2(CCCC2NC(=O)Cc2cnsc2)C1 c1(CCCC(=O)N(C2CN(C(Cc3cnc(C)[nH]3)=O)C2)C)ccc(F)cc1Br C1(OC)(CNC(c2c(Cl)sc(C)c2C)=O)CCN(C(C2(C)CC2F)=O)CC1 N1(C(c2c(Br)csc2C(=O)OC)=O)CC2OCCN(C(=O)C(F)CC3CC3)C2C1 O(NC(=O)C(CNC(C1CC(=O)C12CCC2)=O)C(C)C)CC(C(C)C)O CC(C)C(C)CC(=O)NCC12CC(NC(C3SC4C=CC3C4)=O)(C1)C(C)O2 c1(C(=O)NC2CC(NC(C(Cn3ccc(C)n3)C)=O)C2)cc2cc[nH]c(=O)c2s1 S(=O)(=O)(c1ccccc1F)N(CC(N1CCN(C(=O)CCSC)CC1C1CC1)=O)C C1(C(=O)NCCC2CCN(C(CC3(C)CCC3)=O)C2)CCOCC12CCC2 c1(-c2cc(C(=O)N(CC3(O)CN(C(CCC=CC)=O)C3)CC)on2)nn(C)cc1O c1(SC)nccnc1NC(C1CCCC1C(n1cc(-c2ncccn2)nn1)C)=O C1(NC(c2cc(CCC)on2)=O)CCN(C(c2ccc(C3CC3)o2)=O)CC1(C)C N1(C(CC2CCC(NC(c3cn(C(C)C)nc3)=O)C2)=O)CCC2SC(=O)C=C2C1 c1(C(N(CCNC(C(=O)NCCOCCC#C)=O)CC)=O)n[nH]c(C)n1 N1(C(CCc2nnc(C)n2C)=O)CC2(CNC(C3(C)CC=CC3)=O)CCC1CC2 C=CCN=C(NCC(c1ccc(F)cc1)CO)NC1C(C)(C)C1(C)C C(=O)(C1=CC2CC=CCC12)NCN1CC(OCCNC(c2[nH]nc3ncccc23)=O)C1 N12CCC3(C=C(C(=O)N(CCOC)CC(O)CC1=O)C3)C2.C(CO)OC.CN C1(NC(CCOCCOC)=O)CC2CCC1(NC(c1cc(C)co1)=O)C2 C(=O)(C1CCCc2sccc21)N1CC(O)(CN(C)C(C2COCC(C)(C)O2)=O)C1 C1(C(=O)NC2CCC(NC(CN(C(=O)OC)C)=O)C2)OCCC1(C)C N1(C(C#C)C)CCN(C(=O)C(C2CC=CCC2)NC(=O)CN2CCCCCC2)CC1 N1(C(C2C(=C)C2C(=O)OC)=O)CC(F)CC1CNC(=O)C=CC1(C)COC1 C(CCCC(C)(C)C)NC(C(C(C)O)NC(=O)COCCF)=O C1(C(N2C3CN(C(N4CCC(C)CC4)=O)C(CC3)C2)=O)CCc2c(cnn2C)C1 n1(CC)ccc2cc(Cc3c(C(c4nnnn4C)N)nc(C)cc3)ccc12 C(CCCCCC)(OCC)NCCCn1nnnc1CC1CC1C1(C)OCCO1 CC1CN(C(c2cnco2)=O)CCC1N(C(=O)CCCC(=O)N(C)C)C CC1(NC(c2cnc(S)[nH]2)=O)CCN(C(c2cnc(CC(F)(F)F)s2)=O)C1 C(C)(C)(CN=c1[nH]c2c(c(=NCc3cc(F)cc(F)c3)[nH]1)CC(C)CC2)SC c1(C(=O)NCCC(C)NC(C2CCC(=O)N2)=O)csc(C2CCCC2)n1 CC(CC(=O)NC(C(=O)NCc1ncco1)c1cccs1)n1cccc1 CC(C)(C)CC(C(=O)N1CCC(CN=[N+]=[N-])C1)NC(=O)C1CC1 CC(N=c1[nH]c2c(c(=NC3CCN(C4CC4)C3)[nH]1)CSC2)c1c(F)cccc1F c1(C(=O)NC2CC(NC(c3ncc(OC)cc3F)=O)C2)cc2cc(F)ccc2[nH]1 C(CC(C)CCNC=O)NC(c1[nH]cnc1C)=O.Cc1cc2oc1=2 C1(CCCNC(c2c(C)nco2)=O)CN(C(c2cnccc2N(C)C)=O)CCO1 N1(C(c2cn(CC)nc2)C(=O)NCCSC)Cc2ccccc2OCC1(C)C c1(CC(=O)NC2C=CCN(C(c3cccc(OCC)c3)=O)C2)cnc(Cl)c(C)c1 N1(C(C(CC#C)C)=O)CCC(CCOC)(NC(=O)CC(C)c2cnn(C)c2)CC1 c1(OC)cccc(C(C(=O)NC2CC2NC(c2nc(C)sc2C)=O)OC)c1 c1(C(=O)NCC(C)NC(=O)CC(c2cccc(F)c2)O)ccccc1O C1(CN(C(=O)Cc2ccsn2)CC)CCCN(C(=O)Cc2cncnc2O)C1 O=C(C1Cc2ccc(Cl)cc21)N1CCC(C(F)(F)F)C1.C12CN(CCN1)C2=O c1(C(=O)NC(CNC(C23CCC2C3)=O)CO)ccnc(OC2CCC2)c1 N1(C(C(CCCC)O)=O)CCC12CCN(C(c1cc3cc(C)ccc3[nH]1)=O)CC2 CC(CC(C)NC(=O)CCC1CC1)NC(c1n[nH]c(-c2ccccn2)n1)=O C(C(=O)N1CCC(CN(C(=O)CSc2ccccn2)C)C1)(C(C)C)OC C1(NCC)CCN(c2nnnn2CCSC)CC1.C(C)(C#N)N N1(C(CCC2C(C)C2)=O)C2CCC1C(CO)C2.n12c(nnc1S)C(C#N)C2=O C(=O)(CC(C)COC)NCC1(C(=O)NCC(C)OCC#C)CC=CC1 CN1C(=O)CN(CC(=O)NCC2(CNc3ncnc4c3COC4)CC2)C1=O C(=O)(CCCn1cncn1)N(C(C)C(=O)NC(C)CSC)CC C1(C(=O)NC(C2CCN(C(c3csc(-c4cnc[nH]4)n3)=O)C2)C)CC(F)(F)C1 C1(C(=O)NCCN(C(C2(N(C)C)CCCC2)=O)C2CC2)CC12CCC(F)(F)CC2 C(=O)(C#CC1CCOC1)NC(C(=O)Nc1cnc(SC)nc1)CCN(C)C c1(C(N2C3CN(C(c4n[nH]c(C)c4C)=O)C(C3)C2)=O)c(C)ccc2ccccc12 C1(CN(C)C(c2cc(C#N)on2)=O)CCCN(C(=O)COC(C)(C)C)CC1 CC1(C)CC(C(=O)N2CCCCC(CNC(c3nc4cnccc4s3)=O)C2)=NO1 C(=O)(C1=NOC(C2=CC=CC=CC2)C1)NC(CC)CNC(c1cc(CF)on1)=O c1(CC)cc(C(=O)NCCC(O)CNC(=O)CN(C2CCSC2)C)ccc1O c1(C(=O)NCCC(C)(C)NC(C2(C=C)CC2)=O)cc(Cl)c(F)c([N+](=O)[O-])c1N C1(=O)C(O)CCN1.C12(CC)CC(NC(C3(C(=O)OC(C)(C)C)CCCC3)=O)(C1)C2.OCC N1(C(C(C2CC2)NC(C2CCC(CC)O2)=O)=O)CC(=O)NC2(CC2)C1 CCCS(=O)(=O)C(C)C(=O)NC(c1ccncc1Cl)=O.C12CCCN1C2(C)C c1(C(N2CCC(F)(NC(CNC(=O)OC)=O)C2)=O)cccc2c1nc(O)n2C Cc1ccc(-c2cc(NC(=O)C(C)OC(c3cnn(C)c3C)=O)n[nH]2)cc1 N1(C(C2(Cl)C(C(C)=O)C2)=O)CC(CC(=O)NC2CSC2)CC1(C)C C(=O)(C1=C(Cl)CCC1)NCC1C(NC(C(CC)Nc2ccccc2C(C)C)=O)C1 N1(C(C2(C)N(C)CCC2)=O)CC2(CC2)CC1CNC(=O)COCC1CCCC1 c1(CC)cc(N)c(C(=O)NCCCN(C(=O)CC(O)CN(C)C)CCO)c(F)c1 N1(C(=O)CC)CC(O)(C2CC2)C1.N1(CC)CCC(NC23CN(C2)C(=O)C3)C1 c1(OC)ccc2cc(C(=O)NCC3(S(N)(=O)=O)CCC3)[nH]c2n1 c1(C(N)=O)ccnc(C(=O)NC23CC2CN(C(C2CSCCS2)=O)C3)c1 c1(C(=O)NCC(C2CCC2)NC(C(COC)(C)OC)=O)cnc2c(C)cccn12 c1(C(=O)NC(CNC(C(CC)Oc2ccccc2F)=O)CC)ccc(N)c(Cl)c1 C=CCC(C(=O)NC(CNC(=O)CCN(C)CS(C)(=O)=O)CC(C)C)NC(C)=O C1(CCC)CN(C(c2ccncc2Br)=O)CCN1C(C12CC(O)C1C2)=O c1(C(=O)NC2CN(C(C(N3CCNC3=O)C)=O)CC2C(F)F)cc([N+](=O)[O-])c[nH]1 Cc1cc(C)n(CC(N2CC(CNC(C3CC3(C)Br)=O)C2)=O)n1 Cc1cc(C)c(C(N2CCC3CC23C(=O)NCCN(C)C)=O)cn1 CCCC(C(O)C(=O)NC1C2CCC(C2)C1CO)NC(C1(C#N)CC(=O)C1)=O C1(C(N(C(c2cccnc2)CC)C)=O)CC12CCN(C(C1CC=CC1)=O)CC2 C#CC1CC2CCC1N(C(=O)C(CNC(=O)C1=C(Cl)CCCC1)CC=C)C2 CCC(F)(C(=O)OCC)C(=O)NC1CCN(C(=O)COCCN(C)C)C1.C(C)(C)CC C(=O)(C(C)C(C)C(C)(C)C)N1CC2(CCN(C(CCc3cnc(C)s3)=O)C2)C1 CCC(CCC(=O)NCC(O)CC(F)(F)F)NC(c1cccnc1NC)=O N1(C(c2c(CCC)nco2)=O)CCN(C(=O)C(CO)OC)CC1 C1(C(=O)Nc2c(C)cc(Br)cc2)CCCC12CCN(C(c1ncc(C)s1)=O)C2 C(N=c1ccc(Br)c(S(=O)(=O)N2CCC(C(N)=O)C2C)[nH]1)c1c(CC)c[nH]n1 C(CCC(C(=O)NOCCC(F)F)NC(C1OCCOC1C)=O)OC CC1CCC(NC(c2ccc(C3CC3)cc2)=O)CN1C(=O)Cc1cccnc1 N1(C(c2cc(C)nnc2O)=O)CC2ON=C(CNC(=O)C3=CCCCC3)C2C1 c1(CC(CC)NC(=O)NC2C(C(=O)OCC)C2)ccc(O)nc1 C1(C(N2C3CC(NC(CSCC=C)=O)C3CC2)=O)COc2ccccc2C1 c1(C(N2CCC(CC=C)(NC(=O)COC3(C)CCCC3)C2)=O)cnccc1C#N C1(C2CCN(C)CC2)(C(=O)NCC2C(CNC(C(COC)(C)C)=O)C2(F)F)CC1 Cc1cccc2cc(C(=O)NC3CC(NC(C4CCCN4C(C)C)=O)C3)sc12 c1(CNC(c2cccc(C(=O)OC)c2)=O)ccc2nccn2c1.C12CCCN1C2 c1(C(=O)NC2(CNC(CC3(C)CC3)=O)CC2)cc(C(F)F)ccc1Cl C1(C(N(C)Cc2c(C)nsc2)=O)CCN(C(=O)CC2CCOC2(C)C)O1 c1(CC)ccc(C=CC(N2CC(O)(CNC(=O)Cn3ncc(Cl)c3C)C2)=O)cc1 CC(C)CC(CNC(c1cccs1)=O)NC(c1ccnn1CCN1CCCC1)=O C1(CNC(C=C(C)Cl)=O)CC(C)(C)CCC1NC(c1cncc(NC(C)C)c1)=O c1(C(C)C)ccc(C(=O)NCC2CCC(NC(C3(C)CSC3)=O)CC2)cc1 N12CCC(C(c3ccccc3)C1)OC1CCN(C1)C(=O)C2.CC(=O)OCCF Cc1snc(CC(=O)NCC2C3CN(C(C45COCC4C5)=O)CC23)c1C#N CCCCC(F)C(=O)NCCCN(C(=O)C(C)(C)C(F)F)C1CC1 C1(CC(=O)NC)CN(C(C2CC2c2ccn(C)n2)=O)CCN1C(c1ccn(C)n1)=O c1(C(=O)Nc2cccc(OCCNC(=O)NC3CC3)c2)cnc2ccccn12 C#Cc1cccc(C(=O)NCC2CCN(C(C3COCCN3CC)=O)CC2)c1C N1(C(C(CC2CCC2)OC)=O)CCN(CC(C)NC(C2(C)CC(C)(C)C2)=O)CC1 N#CC1CCC(C(=O)NCCCCCCNC(=O)C(F)CC2CCC2)CC1 c1(C(=O)OC)cc(C)cc2c1NC2=O.C1(C(=O)OC)CC1NC(C1CC1C)=O C1(CNC(CNC(c2nc(C)sc2)=O)=O)CC(O)CN1C(=O)CCC1CCCOC1 CC1(C)C(O)CC1N=c1[nH]c(N2CCC(C3CC3(F)F)C2)nc2c1SCC2 c1(NC(C)C)cncc(C(=O)NCC(O)CN(C(C2CC(C)(F)C2)=O)C(C)C)c1 N1(C(c2ccc(C(=O)NC)nc2)=O)CCOC(C)(CN)C1.C(C)(C)(C)O N1(CCCOCC)CCN(CCCCCNC(c2c[nH]nc2CC)=O)CC1 C(CNC(=O)CCc1ccc(Cl)cc1)(C(C)C(C)C)NC(c1c(C)cc(C)[nH]1)=O C1(CC(N2CCN(C)CC2)=O)CC2(C1)CN(C(=O)CC1CCC(=O)N1)C2 C1(C(=O)NCC(C)CN(C(=O)C(c2cccc(F)c2)O)C)CN(C)CCO1 C(=O)(CCC(C(=O)NC(C)(CNC(c1cnn(C2CC2)c1)=O)CO)N(C)C)OC N1(C(C(CC=CC)C)=O)CCC(C)C(N(C(=O)CN(C)C(C)=O)C)C1 C(=O)(C(C)CC1CN(C(=O)Nc2c[nH]nc2OC(C)(C)C)C1)NCC C(=O)(CC(CC(C)C)NC(c1cc2ccccn2c1)=O)N1C(CC=C)CCCC1 N1(C(C(C2CCN(C(c3cncc(C(F)(F)F)c3)=O)CC2)C)=O)CC(F)C(F)C1 C(CC(=O)Nn1ccnn1)N(C(C(C(=O)NC)CC)=O)C N1(C(c2cnc(C)s2)=O)CCCCC1CC(=O)NCC1CC2(CC2)CO1 c1(CN(C2CN(C(=O)OC(C)(C)C)C2)C)cc(Cl)cc(Cl)c1F c1(CC)ccc(C)cc1C(=O)NC(C1CN(C(=O)CCn2cnccc2=O)C1)C Cn1c(=O)ccn(CC(=O)NCC2CN(C(=O)CC3(O)CC3)CC2(C)C)c1=O CC1(C)CC(C(=O)NCCOCCNC(c2cn3cnnc3cn2)=O)CNC1=O c1(C(N2CC(NC(C(c3c(OC)cccc3)=O)=O)C(C)C2)=O)cc(Cl)ccc1N Cc1ccc(C(N2CC(NC(=O)CC3CCCSC3)CC23CCC3)=O)cc1C#N CC(CCCC(=O)NCCS(C)(=N)=O)NC(=O)C(C)NC=O C1(NC(C2C(C#C)C2)=O)CC2CN(C(=O)C=Cc3cnc[nH]3)CC2C1 CC1CC1C(=O)N1CCCC(O)(CO)C1.C1(C(=O)NC2CC2)CCOC1 C=CC1OCCC1C(N1CCC(C(=O)NCCCC(=O)NC2CC2)(CC)C1)=O C(C(C)(C)CC(=O)NC1CC(O)C1CC(N1CCC1(C)CCO)=O)OC C1(NC(c2coc(CO)c2)=O)COC2CN(C(C3CCC34CCOCC4)=O)CC12 c1(C(=O)NCCCCN(C(C2(C)N(C)CC(OC)C2)=O)C)ccc2cncn2c1 c1(CN2CCC(O)(C(=O)NC3CC3)C2)cc([N+](=O)[O-])ccc1Cl C(=O)(C1Cc2ccccc21)NC1CCN(C(c2c(OC)nccc2)=O)C(C2CC2)C1 Cc1cc(OCC(=O)NC2CCC(CCNC(=O)C(O)C3CCC3)C2)ccc1Cl c1(C(=O)NCC(N(C(=O)CCCn2ccnc2)C)C2CC2)cc(O)ccc1F CC(=O)CCCCC(=O)NC1CCCC(CC(N2CCOCC3(CC3)C2)=O)C1 Cn1nnnc1C(c1cnn(-c2ccccc2)c1)NC1CCSCC1 c1(C2N(C(C(C)(C)OC(C)=O)=O)CCC2)ccc(Cl)c(F)c1.C12CN(CCO1)C2 CC1CCCN(C(c2coc(C(N)=O)c2)=O)C1CNC(=O)COCC(C)(C)C C1(N(C(c2cnc(OC)s2)=O)C)CN(C(c2ccccc2Cl)=O)CC1O c1(C(=O)NCC2(F)CC(NC(c3nc(C)oc3)=O)C2)nnc(O)nc1O N1(C(c2c(C)c[nH]c2)=O)CC(NC(=O)CCn2cnc([N+](=O)[O-])c2)CC12CCC2 CCCC(CNC(c1ncnc(O)c1F)=O)C(=O)NCCc1cnn(CC)c1 N1(C(CS(=O)(=O)NC)=O)CCC(NC(=O)CC2CCC(C)(C)C2)C(F)(F)CC1 C12(C(=O)NCC(C(C)C)NC(c3cn(C(C)C)nn3)=O)CC3CC1(CO)CC3C2 C1(C(=O)NC(C2N(C(CCCOCC)=O)CCC2)(C)C)CS(=O)(=O)CC12CC2 c1(OC)cccc2c(N3CC4CC3CN4Cc3ncc[nH]3)ncnc12 c1(CNC(C2C(C(C)(C)C)C2)=O)ccc2c(c1)CN(C(c1c[nH]nc1F)=O)C2 C=CC(CC)CC(=O)NCC(CO)NC(=O)C(C)=CC1CC1 N1(C(C(CCOC)NC(c2cccnc2OC)=O)=O)CCCOCC1C c1(C(=O)NC2C(CC(N3CCC(C(=O)NC)C3C)=O)CCCC2)cc(=O)n(C)cn1 CC1Cc2cc(S(=O)(=O)NC3COc4ccc(Br)cc43)cc(Cl)c2O1 C1(C(=O)NC2C3(CC(NC(CCC#C)=O)C3)C2)CCC2(CC1)CNC(=O)C2 n1(CCC=C)c(N2CCOC(C)C2)nnc1CC(C)(F)F Cc1nc(CC(N2CCC(O)(C(C)CNC(=O)COC3CCCC3)C2)=O)c(C)s1 C=CC1OCCC1C(=O)NC1(CF)CCN(C(=O)CC2(CS(C)(=O)=O)CC2)C1 C1(CC)C(=O)NCCN1C(C1CCC1)=O.c1(S)ccc(OC)cc1 C1(C(=O)NC2(C)CC(NC(C3CCCOC3)=O)C2)C2CCCC(F)(F)C12 C(=O)(C(C)(C)CS(N)(=O)=O)N1C(C)CC(CNC(c2cc(C)cc(Cl)c2)=O)C1 c1(C(=O)NC2(CN(C(C3ON=C(C)C3C)=O)C)CC2)sc2ncccc2c1Cl CC(=O)CCCC(=O)N1CC(CC(=O)NCc2cccnn2)C2(CC2)C1 C(=O)(C1=CCCN(C(C2CN3CCC2CC3)=O)C1)N1CCC(C)(C)CC1 c1(C(=O)NCC(CN(C)C(c2cccc(CO)n2)=O)O)cccc2oc(O)nc12 C=C(C)CCC(C)(c1nnnn1CCCF)NCC(C)C(C)C c1(OC)cncnc1C(=O)N(C)CCOCCNC(c1ccc(O)nn1)=O N1(C(c2c(CC)noc2C)=O)CCCC(F)(CNCc2cnn(C3CC3)c2)C1 C1(CN(C(c2cc(CC)on2)=O)C)COCCN1C(=O)CCOC C(C(C)C(F)(F)F)N(C(C1(CNC(=O)CCCNC(N)=O)CC(=C)C1)=O)C c1(C(=O)NCC2(O)CN(C(C3C(Cl)(Cl)C34CC4)=O)C2)ccc2c[nH]nc2n1 c1(C(=O)NC2CCC(NC(CC34CC(C)(OC3)C4)=O)C2)ccc2oc(=N)[nH]c2c1 C(=O)(C1CCCc2nncn21)NC(CNC(C1(OC)CCOCC1)=O)CO c1(C(=O)NC2C3(CC(NC(C4(C)CNC(=O)C4)=O)C3)C2)nc2cccnc2s1 N1(C(C2CC(C)C2)=O)CCC2(CC1)CCN(C(=O)CCC(N)=O)C2 C=C(C)CN=C(NC1CCS(=O)(=O)C1)N1CCC(OC(=O)N(C(C)C)CC)CC1 C1(C(=O)NC2CCN(C(CCOC)=O)CC2)CCc2n[nH]cc2C1C C1(C(=O)NOCCC(F)(F)F)CCN1.c1(C2CN(C(=O)OCC)C2)ccncc1 c1(C(=O)NCCCOCCNC(C(C)O)=O)coc(S(=O)(=O)NC2CC2)c1 C1(CC)CN(C(=O)C(C(C)CC)N(C(=O)CCNC(=O)OC)C)CCN1C N1(C(CC(=C=C)C)=O)CC2(CO)CC1(C(=O)N(CC(O)CC)C)C2 c1(C(=O)NC2C(C)(COC)C2)cnn(CCNC(C2CC2C(F)(F)F)=O)c1 N1(C(C2(COC(C)C)CC2)=O)CCC2CN(C(=O)CN(c3ccsc3)C)CCC12 C1(c2n(CCCC)nnn2)(NCc2cnc(Br)cc2C)CCOCC1F c1(C(N2CCCC(N(C(C(CC=CC)C)=O)C)C2)=O)cc(CC)ccc1F C=C=CC(C)C(=O)N1CC(c2ocnc2CNC(=O)C(O)c2ccsc2)C1 N1(C(C2C(C(=O)OCc3ccccc3)C2)=O)CCCC1c1ccccc1 N1(C(C(C)OCOC)=O)CCCC1CN(C)C(C1(COC)CCCO1)=O CC(CNC(=O)N(C)C)CC(F)(F)F.C(=O)(CCCC(=O)OC)N1CCN(C=O)CC1 c1(C(=O)NCCCCN(C(=O)CC2CCOC2)C2CC2)cc(OCC(F)F)ccn1 c1(OC)cccc2c(N(c3ccc(C4CCCC4)cc3)C)nccc12 c1(C(=O)NC(CC)CCO)c(CNC(c2ccn(CCF)n2)=O)nnn1C N1(C(c2cc(OC)ncn2)=O)CCCC2CN(C(=O)CC3CC3)CCCC12 N1(C(C2(C#C)CC(=O)C2)=O)CC2(C=C(C(=O)NCC(O)C3CCC3)CO2)C1 c1(N(CC(=O)NCC)C)nc(=NCc2csc(Br)n2)[nH]c2ccccc12 C1(C(=O)NC(C(C)(C)NC(C(C)NC(=O)NC)=O)C)CC2(CCOCC2)C1 C1(O)(C(N2CCCC(CCCCNC(CCC=C(C)C)=O)C2)=O)CCCCCC1 CN1CCOc2c(CNC(C)(CCN(C)C)c3nnnn3CC(F)F)cccc21 C1(C(=O)NCC2CC(N(C)C)C2)CN(C(=O)CC2CCCOCC2)CC1C1CC1 C1(C(=O)NC2CC(n3cccn3)C2)CCNC2(CC2)C1 C1(CNC(C(C(C)C)OC)=O)CC(C)CCN1C(C1CC(=O)N(C)C1)=O C(=O)(C1CCCc2nc[nH]c21)NC1CCN(C(c2c(N)nc(Cl)cc2)=O)C1C1CC1 N1(C(CNC(C(CC)C)=O)=O)CC2CC(C1)C2NC(=O)CC1(C)CC1 N1(C(C2CCCSC2)C(=O)NC(C)C)CCCCC2(CCC2)C1 N1(C(C2C(OC(C)=O)C2)=O)CCCC(CNC(c2conc2C2CCCC2)=O)C1 c1(OCC(=O)NCC2C(NC(C(CC=CC)C)=O)CCCC2)c(C)cc(Cl)cc1C Cn1nc(C(N2CCN(C(=O)CCF)C3CCC23)=O)c2c1CCCC2O C#CC1(C(N2CCC(N(C(=O)Cc3ccc(C)nc3)CC3CC3)CC2)=O)CCCC1 C1(F)(C(N2CCC(OCC=C)C2)=O)CCN(C(c2n[nH]c(O)n2)=O)CC1 c1(NC(c2c(C)ncs2)=O)cccc(F)c1C(=O)Nc1ccc(Br)c(C)n1 c1(C(=O)NC(CNC(c2[nH]cc(C)c2)=O)C2CC2)ccccc1N1CCCC1=O Cc1coc(C(=O)N(C(c2ccccc2)CNC(=O)Cc2ccsc2)C)c1 C1(NC(c2cc(CCNC(=O)OC(C)(C)C)n[nH]2)=O)CC2CCCCN2C1 C1(NC(c2ccc(C(F)F)o2)=O)CN(C(c2cc(Cl)ccn2)=O)CC12CC2 c12n[nH]cc1C(=O)NC2.C(CC(=O)NCCOCCOC)SCCCC S(=O)(=O)(c1ccc(C#N)c(NC2COCC2F)c1)NCCc1n(C)c(Br)nn1 n1(CC)nc(C(=O)NCCC2CCCN2C(=O)CSCCC#N)c(Br)n1 c1(C(N2CCN(C(Cc3cc(OC)nn3C)=O)CC2)=O)sc2cccnc2c1Cl C1(CN(C)C(c2nsnc2O)=O)CCCC1NC(=O)Cn1cccn1 C1(CCNC(C2C(OC)C2)=O)CSCCN1C(=O)C(=O)Cc1ccc(Cl)cc1 C#Cc1ccc(C(=O)NCCC(C)N(C)C(c2ccn(CC(C)C)n2)=O)cn1 N1(C(C2C(C)CCCC2)=O)CCCC(C2CCN(C(C3CSCN3C)=O)CC2)C1 CC1(c2nn[nH]n2)CCCN(C(=O)CCC2CCOC2)C1 CCC(C)(C(=O)NCCOCCN(C)C(C1CCCS1)=O)OC N1(Cc2c(C(=O)NCC=C)cccc2)CC2CCC(C1)N2c1ccncn1 N1(C(C2C(CC)C2)=O)CCC(C)N(C(c2ccc(-n3ccnc3)c(F)c2)=O)CC1 C1(CC(=O)NC(c2cccc(O)c2)c2ccccc2)CN(C(CO)C2CC2)CC1O C#CC1(C(=O)NC2CC23CCCCCC3)CCN(C(C2CC(O)C(F)C2)=O)CC1 c1(C(N2CCN(C(CNC(C(CC=C)C)=O)C)CC2)=O)ccc2c(c1)COC2=O C(CN=[N+]=[N-])(C(=O)NCCC(C)(O)C1CC1)NC(C=C1CCC(C)CC1)=O C(c1ncccc1C)=CC(=O)N(C1CCN(C(C2CC2(F)Cl)=O)C1)CC C=CCC(CC=C)C(=O)NC(C)CCC(=O)N1CC(n2cccn2)(C(=O)OC)C1 c1(C(N2C(CNC(=O)C=CBr)CC(C)(C)C2)=O)[nH]nc2c1CCC2(C)C c1(C(=O)NC(CNC(c2ccc(OCC(C)C)cc2)=O)(C)C)cc(F)cc(Cl)c1 C(=O)(C(=O)CCC(C)C)N1C(C(=O)NC(CC=C)(C)CC=C)C(C)CC1 c1(CNC(CN2CC3C(NC4CN(CC=C)C(=O)C4)C3C2)=O)ccc(O)c(C)c1 c1(CSC2OCCC(NC(=O)OC(C)(C)C)C2)nc2cc(Cl)ccc2o1 c1(CC(CC)NCc2ncc(C3CCCN3)s2)ccc(C(F)(F)F)cc1 C1(NC(c2c(OC)nc(Cl)cc2)=O)CN(C(C23CCCC2C3)=O)CC(F)(F)C1 C(=O)(C(O)CNC(c1ccn(C(F)F)n1)=O)NC(c1nccs1)C Cc1ccc(Br)c(C(=O)NCC2CCCC2NC(=O)CC(C)C)c1 CC1CC(CNC(c2cnc(-c3ccccc3F)nc2)=O)CN1C(=O)CNC=O CS(=O)(=O)CC(=O)N1CCC(C2CCCCN2C(C2C3CCN2CC3)=O)CC1 C(N=c1[nH]c2ccc(O)cc2s1)C1CCCC(NC(CC2(C)CC2)=O)C1 C1(C(=O)NCCC=CC=C)CC(C)N1C(=O)CCn1cnc(=N)[nH]1 N1(C(C(C(C)C)C)=O)CCC2(CCC(NC(c3ccsc3Cl)=O)C2)C1 CCC(O)C(F)(F)C(=O)NC1CC2CCC1CN2C(=O)C(N1CCOCC1)C C1(C)(C(=O)NC(C)CN(C)C)CC(C(=O)OC)C1.N12CCCC1NC(=O)C2 C(=O)(C1(C)OCCc2ccccc21)N1CCCC(NC(C(C)C#N)=O)CC1 C(C(=O)NOCC1CCCO1)(C1CC1)NC(c1cc(OC)n[nH]1)=O c1(C(=O)NC(C)CCCNC(C2(C)C(C)(C)C2(C)C)=O)ncc(Cl)c(N)c1Cl c1(C(C)C(=O)NCC2CC(NC(=O)CCN(C)CCO)C2)ccc(F)c(F)c1 n1(CC(=O)N(CCC)CCNC(c2csnc2C)=O)nc(C)n(C)c1=O C1(C(N2C(CNC(c3c(CC)[nH]cc3)=O)CC(F)C2)=O)Cc2ccccc2C1 C(=O)(CCCC(=O)OC(C)(C)C)N(C)CC1CN(C(C2(OC(C)(C)C)CCC2)=O)C1 Cn1nc2c(c1C(N1CC3CC1C3NC(=O)CCC1CC1)=O)CSCC2 C1(NC(c2nn(C)c(Cl)c2)=O)(CO)CCCN(C(c2ccc(F)c(Cl)c2)=O)C1 C(=O)(CC(C(C)(C)C)NC(=O)COc1ccn(C)n1)N1CCC(O)(CC)C1 C1(C(=O)NCC2OCCN(C(C3C(C)OCCC3)=O)C2)CCc2nc(O)[nH]c2C1 n1(CC)cc(Cl)c(C(=O)NCC(C2CCCCC2)NC(C2CCC(C)(C)C2)=O)n1 Cc1ccc(CO)cc1NC(N1CC(C)(Nc2cccc(SCC(C)(C)C)c2)C1)=O C12(CNC(CCCn3c(C)ncc3)=O)CC1CN(C(C1C3CC4C(C3)C14)=O)C2 c1(C(=O)NCC2C(NC(CC(C)NC(N)=O)=O)C2)cnc2c(c1)CCCC2 S(=O)(=O)(c1ccccc1F)N1CCC(NC(=O)CNC=CC(=O)C(F)(F)F)CC1 C1(SC)CCN(C(=O)N(C(C)CCC=C)CC2(n3cnnn3)CC2)CC1 C1(NC(=O)OC(C)(C)C)CN(C(=O)CN2CCCC2c2cc[nH]n2)CCO1 Cc1c(C(=O)NCC2CCC2NC(=O)C(C)O)cnn1-c1ccccn1 Cc1cc(C(N2CC(CCNC(C3SCCC3C)=O)C2)=O)n(CC(F)F)n1 N1(C(=O)NC(CC=C)CNC(=O)C(C)CNC(=O)OC(C)(C)C)CC(=O)NC1=O C1(NC(Cn2c(C)cc(C)n2)=O)CC(NCC(=O)NCCC(F)(F)F)C12CCC2 CON(CCC(=O)NCCN1CCCCCC1)C(=O)C(C)OC(C)(C)C C(N=c1[nH]c(N2CCCOC(C3CCC3)C2)nc2c1COC2)c1c(C)n(C)nn1 c1(OC)ccc(Cl)c(CC(=O)NCc2ccc(NC(c3ncc[nH]3)=O)o2)c1F C1(CC)CC(C(=O)N(C)CCNC(C23CCCC(C2)OC3)=O)CC(=O)N1 O=C1CCC2CCN(c3ccc(C(c4ccccc4)=O)cc3)CC2N1 CCC(CC)CC(F)C(=O)NC1CC2(C1)CC2C(=O)NCCCC1CC(C)C1 C1(NC(=O)OC(C)(C)C)(CN)CCC1.C1(NC(C2CCCO2)=O)CC(C)C1 c1(C(=O)NCC(C)NC(C(COC)(C)OC)=O)ccc2c(c1)N(C)CCO2 c1(C(=O)OCC2(C)CCC(C(=O)OCC)C2)onc2c1CCCC2 c1(OC)nc(C)ccc1C(=O)NCCN1CC(NC(c2c[nH]c(=N)s2)=O)CC1=O c1(NC(=O)C(=O)NCCc2cc(O)nc(O)n2)c(C(N(C)C)=O)cccc1F Cc1cc(C(=O)NCc2ccc(CN(C(=O)C=CS(C)=O)C)cc2)c(C)nc1C c1(CC(=O)NC2(C)CN(C(COCC(=O)NC)=O)C2)cccc(C)c1 c1(C(N(CC(CC)NC(=O)C(F)Cc2ccccc2)C)=O)ccc(OC)c(C)c1 c1(C(=O)NCCOCCCN(C(=O)CCn2cnc(=N)[nH]2)C)ns[nH]c1=O Cc1nn(CC(N2CCCC(CC(N)=O)(NC(=O)CSC(F)F)C2)=O)c(C)c1CO c1(C2(C(=O)NCC(CO)NC(C3(C)CCC(=O)N3)=O)CC2)cccc(F)c1F C(=O)(CC(C)(C)SC)NCCCCNC(C=CC=CC)=O.C(N)=O CC(CCCNC(c1c[nH]nc1C(F)(F)F)=O)NC(c1cc(CF)on1)=O Cc1c(NC(C2CCN(C(C3CN(C)C3)=O)C2)=O)cccc1F N(C(=NCCN1CCOCC1)NC1CCS(=O)(=O)C1)Cc1cn(CCF)nc1 c1(Cn2c(N3C(C(C)C)CN(C)CC3)nnn2)ccc2c(c1)CCCNC2 Cc1[nH]nc(C(=O)NC2CN(C(=O)CC3CCC=CCC3)CCC2F)c1[N+](=O)[O-] CCCCCCC(C(=O)N1CC(NC(=O)CCCCC(=O)OC)CC(O)C1)OC C(=O)(C1CCCn2ccnc21)NC1(C)CCN(C(CC2CCN(C)CC2)=O)CC1 C12(CNC(CS(CC)=O)=O)CN(C(=O)CCc3ccnc(C)n3)CC(F)(C1)C2 C#Cc1cccc(C(N2CCCC(C)(CNC(c3ncn(CC)n3)=O)C2)=O)c1Cl C1(NC(C2C(C)CCC2)=O)CCc2onc(C(=O)NC(C3COC3)C)c2C1 Cc1nc(N2CC3C(NC(C4(C)CS(=O)(=O)C4)=O)C3C2)c2cnn(C)c2n1 Cc1cncc(C(=O)NCc2ccc(C(=O)NCC3CC(=O)N(C)C3)nc2)c1 C1(NC(C(CC=C)OC)=O)CN(C(c2cc(CC)nn2C)=O)C2(CCC2)C1 C1(C(=O)NCC(C(C)(C)O)F)C2CC(O)C(C2)N1C(c1cc(Cl)ns1)=O c1(C(=O)NCC2CN(C(Cc3c(C)nn(C)c3)=O)C2)cccc2c1CCC(=O)N2 Cc1cc(-n2cc(CCN(C(=O)CC3OCCOC3(C)C)C)nn2)cc(F)c1 N1(C(c2cc(CCC)[nH]n2)=O)CC(CNC(C2CC(CF)C2)=O)C(C)C1 CCC(CNC(=O)C(C)=C(C)C)NC(=O)CCNC(C1CC1C)=O N1(C(C2(C)CC(=C)C2)=O)CC2(CC(NC(=O)C=Cc3cnccn3)CO2)C1 N1(C(C(C(C)C)OCC)=O)CCC2(CC2NC(c2cc(C#N)c[nH]2)=O)C1 CC1(C(=O)NCCC2CCCN(C(=O)CCOC3CCCC3)C2)CCOCC1 Cc1cc(C(N2CCC(OC3CN(C(=O)C(C)(C)C(N)=O)C3)CC2)=O)n2nccc2n1 N1(C(c2ccc(C)s2)=O)CCC2(CCCN(C(=O)CCCCN(C)C)C2)CC1 N(C(=NCC(C)C1CCCC1)NCC(=Cc1cccnc1)C)CC=C c1(C(=O)NCCCOCCNC(c2cc3scnc3[nH]2)=O)cnc2[nH]cncc1-2 C1(NC(c2c(C)ocn2)=O)C=CCN(CC=C(Cl)Cl)C1 C(N=c1[nH]cnc2ccccc12)C1CN(C(c2c(C(C)=O)cccc2)=O)C(C)C1 C12CC3CCC1(C3)C(=O)N2.C(CCC(=O)N1CC(C)(OC)C1)OCCOC N1(C(c2c(CC)nc[nH]2)=O)CCCC12CCN(C(c1nnn3c1CCC3)=O)C2 CCCCC(=O)NCC1(C(=O)NC2COCC2CC)CC=CC1 c1(C(=O)NC2CCCC(NC(c3cc(CC4CC4)on3)=O)C2)cc(O)ccc1Br CC(O)CC(C)NCCCn1cccn1 C(C)(CN=c1nc2[nH][nH]cc-2c(O)n1)N(C(CCOCCOC)=O)CC CC1CCOCCN1C(=O)CCc1ccccc1 Cn1nc(C(N2CCC(C)(NC(=O)COCCF)C2)=O)c2nc[nH]c(=O)c12 N1(C(c2ccccc2Cl)C(=O)NCCSC)CCCCC1n1ccc(C)n1 c1(C(=O)NCC(C)N(C(C(C)OC)=O)C)cccc(C2(O)COC2)c1 c1(CC(N2C(CNC(CC(C)c3ccncc3)=O)C=CC2)=O)nc2ccccc2s1 C(=O)(C1CCCc2scnc21)NCC1N(C(c2cccc(C(C)=O)c2)=O)C2C(C1)C2 c1(SC)ncc(C(=O)NC(C)CC(C)NC(=O)Cc2c(C)cccc2Cl)c(O)n1 C1(NC(c2c(C)n(CC(C)C)nc2)=O)CCN(C(c2n[nH]cc2Br)=O)C1(C)C N1(C(C=Cc2c(C)n(C)nc2)=O)CCCN(C(c2ns[nH]c2=O)=O)CC1C N1(C(C)=O)CCCC(NC(C2C3CC2N(C(C2CC(O)CN2C)=O)C3)=O)C1 c1(C(=O)NCC(COC)C2CC2)ccc(C2CCCCC2)cc1C c1(C(=O)NC2C(NC(=O)Cn3ccnn3)CCCC2)cc(O)c2ccoc2c1 C1(C)(CC)CC(NC(C2(C(=O)OC)CC2)=O)CN1C(=O)Cc1cnc(C)o1 C(=O)(CCCCCNC(C)=O)N1CC2N(c3nccc(OC)n3)C2C1 n1(CC)nc(C)c(CC(N2CCC(CN(CCCCC3CCCC3)C)C2)=O)c1C C1(C(=O)NC(C)C(=O)NCC2CC3C=CC2CC3)CCc2nnnn2C1 CCC(CC(=O)N(CCNC(=O)C(=CC1CCCCC1)F)C1CC1)C(C)(C)C c1(C(=O)NCC=CCNC(c2cc(=O)cc(Cl)[nH]2)=O)ccn2ccnc2n1 N1(C(C2CCC(=C)CC2)=O)CCC(CCC)(NC(c2c(C)cccc2F)=O)CC1 C1(C(N(C(c2ccccc2)CC)C)=O)CCN(c2cnccn2)CC1 c1(NS(C)(=O)=O)ccc(C=CC(=O)NCCC(C)(C)NC(=O)CC2CCCO2)cc1 CCC(CC)(CN=c1[nH]c(=NCC(C)(C)CCO)[nH]c2cc(OC)ccc12)OC C1(C(C)(C)C)(NC(C(=O)NCCOC)=O)CCN(C(=O)CN2CC3C=CC2C3)C1 C(CCC(C)C(=O)N1CC(CCCCNC(=O)CCn2cncn2)C1)OC Cc1nc2ccc(C(=O)NCC3CCCCN3C(c3cnco3)=O)cc2nc1C CCCCCCCCC(=O)N1CC2CCC2(NC(=O)CCc2cncs2)C1 C1(OC)CN(C(=O)CC(C)O)CC1C(N1CC2C(C(N)=O)C2C1)=O Cc1nnsc1C(=O)N(C)CCN(C)C(C)C1CC1 C1(NC(C(F)(F)F)c2ccccc2)CC2CCC(C1)C2CN1CCCC1 C1(NC(c2ccc(C)o2)=O)CC2(C1)CC2C(=O)NC(CO)C(=O)N(C)C C(=O)(CC(C)(C(F)F)OC)N1CC(CC)(NC(C2CC(C#N)(NC(C)=O)C2)=O)C1 C1(CNC(c2c(SC)scc2)=O)CN(C(=O)C(C)C(F)F)C2(CCOCC2)C1 Cc1cc(C(C)C)ccc1CN(C)C(=NCC1CCCO1)NCc1ccccc1F N1(C(C2CC(CC)C2)=O)CCOCC1CN(C)C(c1sccc1C(=O)OC)=O C1(NC(c2c(C)cn(C(C)C)c2)=O)CC2CC1CN(C(=O)CCc1ccnn1C)C2 CC1(C)CN(C(c2ccc(C(F)(F)F)cn2)=O)CCC1NC(c1ccc(Cl)s1)=O Cc1cccc(-c2nnn(C(C)C)n2)c1.n12nc(cc1C)CC(=O)N2 c1(C(=O)NC2CCCN(C(=O)Cc3c[nH]nc3O)C2)ccc2cc[nH]c2c1F C(c1ccc(F)cc1F)=CCN1C(C(=O)NCCc2ncco2)CCCC1 O=C(C1CS(=O)(=O)c2ccccc21)C1(c2ccc(Cl)cn2)CCC1 N1(C(=O)CCCn2cc(C3C(CC4CC4)CCC3)nn2)CCC(S(=O)(=O)C(F)F)C1 Cc1c(Cl)c(C(=O)NC2COCC2CNC(=O)Cc2cc(Cl)n(C)n2)nn1C Oc1ccc2c(c1)CN(Cc1ccc(Br)c(CO)c1)CCO2 c1(OC)cccc2c1OCC(CNC(=O)NC1CCN(c3cc[nH]n3)C1=O)C2 CCC(CC)C(F)C(=O)NC1(CNC(c2cc(C)c(N)cn2)=O)CCCCC1C c1(C(N2CC(C)CC(NC(CNC(=O)NC)=O)C2)=O)cc(C)c(O)c(N)c1 c1(C(N2CCC(NCc3ccc4sccc4c3)C2)=O)ccc(F)c([N+](=O)[O-])c1 CN1CCOCC1CC(=O)NC1CC(CNC(=O)C(c2ccccc2)N(C)C)C1 CCC(CCC(=O)NCC1(O)CCCC1(C)C)NC(=O)CC1CCCN1C C1(N(C(CC(n2ccc(C)n2)C)=O)C)CN(C(c2sc(Cl)nc2C)=O)CCC1C Cc1nc(C2CCC2)oc1C(=O)NCC1CN(C(c2c(Br)nnn2C)=O)C1 Cc1ccc(C(N2CC(NC(c3cn(C)nc3C)=O)C(O)C2)=O)c(C)n1 c1(OC)ccc(C(N2CCC(NC(=O)CSC(F)(F)F)C2C(C)C)=O)c(F)n1 N1(C(CC)C)CCN(C(=O)CONC(C2CCC(=O)O2)=O)CC1 CC1CN(C(c2nocc2Cl)=O)CCN1C(C1COC2COCC12)=O N1(C(C2(CC(C)C)CC2)=O)CCC(CN(C(=O)CC2CSCCO2)C)CC1 c1(C(C(=O)NC(c2ccccc2)C)N(CCCC(=C)C)C)cn(C)nc1Br C1(NC(CCC(CCC)OC)=O)CCC2(CC1)CN(C(=O)CP(C)(C)=O)CCO2 c1(CN(C(C2N(C(C=CCN(C)CC)=O)CC2)=O)C)ccccc1C c1(C(c2n(CC(=C)C)nnn2)NCCC(O)C2CC2)ccc2cc(Br)ccc2c1 O=C(CC1=NNC(=O)C1)NC(CNC(C1CC1(F)F)=O)C1CCC1 S(=O)(=O)(c1ccccc1S(C)(=O)=O)N(c1ccc(OC)nc1)C(C1(F)CNC1)=O C1(CC)CN(C(=O)CCC2CCCN2C)CCN1C(=O)Cc1sccc1Cl C1(NC(C2(C)COC(=O)N2)=O)CN(C(C2CCCC23CC3)=O)C2(CCCCC2)C1 C1(NC(CCSCC)=O)CCN(C(C2CCN(c3ccccc3)C2=O)=O)CC1O C1(CNC(C(CC#C)O)=O)CC(C(=O)NCC2(O)CCC2)=NO1 C1(O)(CCNC(C(CC=CC)C)=O)CCN(C(C2CCCC2C(=O)OC)=O)CC1 c1(C(=O)NCCCC2(NC(=O)C3=CCCS3)CC2)cnn2cc[nH]c(=O)c12 N1(C(C2CS(=O)(=O)C2)=O)CC2(CCN2C(=O)COc2cccc(F)c2)C1 N#Cc1cccc2[nH]c(C(=O)NC3CC3CNC(c3ccsc3Cl)=O)cc12 CC(C)CC(CNC(=O)Cc1cc(C(F)(F)F)n[nH]1)NC(=O)CSc1nc[nH]n1 c1(SC)ncc(NC(C2C=CC(NC(C3CC(C)(C)C3)=O)C2)=O)cn1 Cn1cnc2cc(CN3C(=O)CN(CC4C(C)(C)C4(F)F)C3=O)cnc12 c1(CN2C(C)CCC(NC(c3c(C)cc(C)o3)=O)C2)ccc2c(c1)COC2 N1(C(c2cn(CCC=C)nn2)=O)CC2CN(C(c3ccsc3Cl)=O)CC2(C)C1 c1(OC)ccnc(C(=O)NC(C)C(C)NC(c2cc(C3(O)COC3)on2)=O)c1F C#Cc1ccnc(C(=O)NCC2(C)CCC(NC(c3ccc(C)c(F)c3)=O)C2)c1 c1(NC(COC(C2C(CC)CC2)=O)=O)cc(I)cc(Br)c1Cl CC1Cc2ccc(CNC(=O)N(C)Cc3ccc(NCC(N)=O)cc3)cc2N1 C1(CNC(c2cc[nH]n2)=O)CCN(C(c2ccc(F)cc2)=O)CC1 c1(CN2CCN(C(=O)NCc3cccc(Cl)c3F)CC2)sc2ccccc2c1Cl N(C1CCCc2occc21)C(C(CCSC)NC(C1CCN(C)CC1)=O)=O N1(C(Cn2ncc(C)c2)C)CCCC(CNC(=O)C(O)CC2CCCCC2)C1 c1(CNC2CCC(NC(c3c(C)ncs3)=O)C2)ccc(Br)cc1Cl C(CC(C)C(=O)NCC1CCC(C(=O)N(CC)Cc2ccc(F)cc2)C1)=CC N1(CC2COCC2(C)C)C(=O)CCOC1CCCC(CNC(CCC(C)N)=O)CC O=C(C1=CCCN(C(=O)Cc2cnsc2)C1)NC1CCCCNC1=O C1(CCC)CN(C(c2cnccc2Cl)=O)CCN1C(C1COCCC1(F)F)=O C12(NC(c3c(CC)oc(C)n3)=O)CCC(NC(=O)CC3CC(F)(F)C3)(CC1)C2 Cc1nc(C)c(-c2nc(C3CCCCC3O)nn2CCC(C)(C)C)c(O)n1 N1(C(CC2CN(C(C3(F)C(C)(C)C3(C)C)=O)CC23CC3)=O)CC2(CCNC2=O)C1 Cc1oc(C)c(C(=O)NCC2CC(C)CN(C(c3cc(F)c[nH]3)=O)C2)c1C c1(OC)nc(N2CCC2(C)C(=O)Nc2nccc(Cl)c2I)ncc1F c1(OC(CN(c2ccccc2OC)CCCC)=O)ccc(C(F)(F)F)c(F)c1 Cc1cc(C(=O)N=S(C)(C)=O)cc2c1NC(=O)CC2 C1(NC(c2ccsc2)=O)CC2CN(C(C3CCS(=O)(=O)N3)=O)CC2C1 c1(COC)ncc(NC(c2cc(CNC(c3ncn(C)c3C)=O)[nH]n2)=O)cn1 CC(C(=O)NCC1(CF)CCC1)N(C(=O)CCC1CCCO1)C1CC1 N1(C(CSCCNC(CCC(=C)OC)=O)=O)CC(C2=NOCC2)C1 C1(C(=O)NCC23CC(C(C)(C)C)(C2)C3)CN(C(=O)Cc2ccc(Cl)nc2)CCO1 c1(-c2c(C(=O)NC3C(C(=O)NCCCOC)C3)con2)ccc2c(c1)OCCO2 N1(C(COCCOCC#C)=O)CCC2CC12C(=O)NC(CSC)CO c1(CC(N2CC(OCCC(=O)NCC(=O)OC3CC3)C2)=O)cccc(F)c1 N1(C(CCC)=O)CCCC1(C(=O)NCC1CN(C)C1)CCC.C1(CO)CO1.C(C)C C1(CN(C(C=CCC)=O)CC2CC2)CCC(NC(=O)CCc2ncccc2C)CC1 c1(OC)cc(Cl)c(C(N2CCC(c3cccc(C(=O)O)c3)(C(=O)O)C2)=O)cc1Cl c1(Cc2n(CCCC)nnn2)ccc2cccc(C)c2n1.C1CCC(C)(C)N1 c1(C(=O)NCCCCNC(c2nc(CC)sc2)=O)cc2n(n1)CCCC2=O C1(C(N2CC(C3CCOC3)C2)=O)(Cc2ccccc2)CCCCC1 CCCC(CNC(=O)C(CC)OC)C(=O)N1Cc2ccccc2CO1 C1(N(C)C(C2CC(C)(C)CN2C)=O)CCC2CN(C(=O)Cc3cnoc3)CC12 C#CC1(NC(=O)CCC2(C)CCCN2C(C2CS(=O)(=O)C2)=O)CC2CCCC12 C1(O)(C(C)NC(=O)CCc2ccc[nH]2)CCN(C(c2c(N)cccc2Cl)=O)CC1 N1(C(c2n(CC)ccc2)=O)CCCC(C(C)(C)C(=O)N2CCC2C2CCOCC2)C1 c1(C(=O)NCC2CN(C(C(CC(CC)C)C)=O)C(C)C2)ccc(F)c2ccsc12 OC1CC2CN(CCCc3ccccc3F)C1C2 C1(CCOC)(NC(=O)COCCCC(C)C)CCN(C(=O)C(O)CN(C)C)C1 c1(C(N2CC(O)(C(C)NC(C3CC(C)(CC)C3)=O)C2)=O)cncc(C(=O)OC)c1 c1(C(N2CC(CC(C)NC(C(C)C)=O)C2)=O)ccc2c(c1)NC(=O)CCN2C c1(NC(c2c(OC)cccc2I)=O)cc(C#N)c(Br)cn1.N12CCC(O)C1C2=O C1(NC(=O)CCCn2cccc2)CCCC(c2ccccc2)C1 N(C(=NCCC1SCCS1)NCC1CCCO1)C(c1cccc(Br)c1)C CCCC(C(=O)NCCC1CCOCC1)NC(c1ccc(F)cn1)=O c1(OC)ccccc1NC(C)C(=O)NC(CNC(=O)C(C)OC)C(C)C N12CCC(CC1)C2=O.C(=O)(C=C)C1C(NCC=CC)C1.C(COC)OC(C)=O N1(C(c2cccc(C(C)=O)c2)=O)CCN(C(=O)Cn2nccc2C)CC12CC2 c1(C(N2CC(N(C(=O)CC3CCNC3=O)C)C2)=O)cn(C)nc1-c1cccnc1 C(C1CN(C(c2sccc2Cl)=O)Cc2ccccc21)NC(c1[nH]n(C)c(=O)n1)=O c1(C(N2C(CNC(C(ON=C(C)C)C)=O)CC(O)C2)=O)cc2cccn2c(O)n1 c1(NC(C2C3CN(C(=O)C=Cc4cnccn4)CC23)=O)ccc(F)c(F)c1F N1(C(C(c2ccco2)NC(COCC(C)C)=O)=O)CC(O)C(O)C1 C1(NC(c2c(C)ncn2O)=O)CC12CCN(C(=O)COCc1cccc(Cl)c1)C2 C(=O)(C(O)CC(C)(C)C)NCC1CN(C(C2CCC(CC)CC2)=O)CC1C C1(C(=O)NCC(C(C)C)NC(C2CCCCS2)=O)CCCC(C)CC1 c1(OC)nc(N(c2cnn(-c3ccccc3)c2)CC2CCNC2)ncc1F NS(=O)(=O)c1ccsc1C(N1CC(O)(CNC(=O)Cc2ccoc2)C1)=O C1(NC(C2(CNC(c3ccco3)=O)CC2)=O)CC2CCCCCC12 c1(C(N2CC(C(C)NC(=O)C=Cc3cccc(O)c3)C2)=O)cc2n(n1)CCCC2O CCC(C(N)=O)NC(C1CCN1C(c1cnn[nH]1)=O)=O C1(C(C(=O)NC)NC(c2cc(I)cs2)c2nnnn2CCCF)CC=CCC1C CC(C)C#CC(=O)N1CC2C(NC(c3nocc3C(C)(C)C)=O)C2C1 c1(C(C)C)ccc(C(=O)N(C)CCOCCNC(=O)CCc2ccoc2)nc1 c1(C(=O)NC(C)(CO)C(=O)NCCCC2CCCCO2)ccc(O)cc1F C12(C(N3C4C(NC(c5ccoc5)=O)CC(C4)C3)=O)C3CC(CC13)C2(F)F c1(C(=O)NC(C)CC2CN(C(c3cc(C#N)on3)=O)C2)ccc2ncccc2n1 c1(C(N(CC(CC)NC(=O)CCC2(C)CC2)C)=O)cc(Cl)c(F)cc1F C(=O)(C1=CCC2CCC1N2C(=O)CCOCC(C)C)NCC(CC=C)(C)CO C1(CC)(CC)CC(NC(=O)CCC2CC2(F)F)CN1C(c1ccon1)=O C12CCN(C1C)C2=O.C1(CC)C(CNC(c2cc(C(C)C)on2)=O)C1(C)C C(=O)(C1CCc2cc(F)ccc21)N1CCCC(CN(C(=O)CC(F)F)C)C1 c1(C(N2CCCN(C(C3C(COC)C3)=O)C(C)C2)=O)cc2nc(C)cc(C)n2n1 c1(C(=O)NC(CCOC)CNC(=O)C(F)Cc2ccccc2)cccc(F)c1 Cc1ccc(O)cc1C(=O)NCc1cc(C(=O)NC2(C3CC3)CCCC2)ccn1 CCCC(C)CCCC(=O)NCC12CCC1CN(C(c1cnc(C(F)F)s1)=O)C2 C(C)(C(=O)N1CCC(NC(c2cc(CCO)on2)=O)C1)(C(C)C)OC c1(C(=O)NCC(CNC(=O)C=CCF)F)ocnc1-c1ccccc1 CCCCCCC(C)C(=O)NC1(CNC(C2CCCN(CC(C)C)C2)=O)CC1 C123CC1CCN2C3=O.C(=O)(C(C1CC1)NC(C1(CCOC)CC1)=O)OCC C(C)(C(=O)NCCC(=O)NCCCNCC(O)COC(C)C)OC c1(C(=O)NCC2(CCNC(CCN(C)C(N)=O)=O)CC2)c[nH]nc1C(C)(C)C CON(CCCO)C(=O)C12CCC1CN(C(c1cc(C)c[nH]1)=O)C2 N1(C(c2cc(C)nnc2C)=O)CC2(C=C(C(=O)N3CCCCC3CF)CO2)C1 N1(C(CCCC#C)=O)CC(NC(c2sccc2F)=O)C2CCCCC12 n1(CC)ccnc1C(=O)NCC1C=CC(NC(=O)C=CC(F)F)C1 N1(Cc2n(C)c(C(F)(F)F)cn2)CCC=C(C(=O)NC(=O)CCc2ccc[nH]2)C1 C(=O)(C(C)CCCC(C)C)N1C(C(=O)NC(CC(C)C)C)CC2(CC2)C1 n1(CC(N2CCCCC(CC3CCC3)C2)=O)nc2ccccn2c1=O Cc1ccc(C#N)cc1NC(C1CCCC(NC(=O)CC2(C)CC2)CC1)=O N1(C(C2CC(OC)C2(C)C)=O)CC2(CNC(=O)C(C(C)(C)C)SC)CC(F)(C1)C2 CC1(C)CCCC(c2cccc(CNC(=O)NC34CC3CNC4=O)c2)C1 C1(CC)CCCN(C(=O)CC(C)C(F)F)C1C(N1CCCC(C(C)O)CC1)=O N1(C(c2c(N)ncc(C)c2)=O)CC(C)CN(C(c2occc2CN(C)C)=O)CC1C c1(O)ccc(C(C)C)cc1.c1(CC(=O)N(CC)CC)sccc1Cl.C1(=O)CO1 C1(NC(C(C(C)OC)NC(C2CCC(=C)CC2)=O)=O)C2CCC(F)(F)C12 C(N=c1[nH]c2c(c(=NC3CCC3C3CCCC3)[nH]1)CCC2)c1cc(O)nc(O)n1 c1(OC)ncc(F)c(=NC(=O)c2[nH]c(C)c(C(=O)NCCCCO)c2C)[nH]1 C1(C)(NC(Cc2n(C)ccn2)=O)CCCCC1C(N1CCOC(CF)C1)=O N1(CCNC(C(C2CC2)NC(C2ON=C(C)C2)=O)=O)CCNC(=O)C1 CCCCC(F)C(=O)NCC(C(C)C)NC(=O)CSCCOC c1(C(=O)NC(c2onc(CC)n2)CCC)oc(CC)nc1C.C12(CC1(C)C)C(=O)N2 C1(NC(=O)CC2(NC(C3CCCCO3)=O)CC2)CCCC(F)C1 C(CC(C)N(CC(C)NC(=O)COCC)C)SC.c1(C=O)cscn1 C(N=c1cc(C(C)=O)nc[nH]1)C1N(C(C2(C=C)CCOCC2)=O)CCC1 C1(O)(n2cc(CN(CCOC)C)nn2)CCN(C(c2nc(C)ccc2Br)=O)CC1 N1(C(C(C)NC(c2ccoc2)=O)=O)CC(NC(C2CC2Br)=O)C(C)C1 Cc1coc(C=CC(=O)NCC2(NC(c3ccncc3C3CC3)=O)CC2)n1 N1(C(C(C)SC(C)C)=O)CC2(C=C(C(=O)Nc3cncc(F)c3)CO2)C1 C1(NC(C(c2nccc(C)c2)(F)F)=O)C2CC1CN(C(C1CC=CCC1)=O)C2 CC1(C)CN(C(C2(C#N)CCCO2)=O)CC1C(=O)NCC(C1CC1)C1CC1.C12C=C1C2 N1(C(c2cc(C)n(C)n2)=O)CCC(C)(NC(=O)Cn2nnc(C3CC3)n2)CC1 C=CC1(CC(=O)NC2CCCC2C(N)=O)CN(C(=O)CCC(N)=O)C1 C(=O)(C(F)C(F)(F)C(F)(F)F)NC(CC(C)NC(C(CC)c1ccccc1)=O)C Cc1cc(C(=O)O)ccc1C(N1CCOC(C)(C(C)C)C1)=O c1(C(N2CC(F)(CNC(C=CC(=O)N(C)C)=O)C2)=O)ccc(C#N)nc1 CCC(C)(CCC(C)C)C(=O)NCC(C1CCCCC1)NC(=O)C(C1CC1)OC C1(NC(C(C)CC2CC2)=O)C(C)CN(C(=O)CSCc2ccccn2)CC1C c1(N2CCC(CC=C)(NC(c3cc(C(N)=O)[nH]n3)=O)C2)ncc2ccsc2n1 C(=O)(C(CC(C)C)ONC(c1oc(C)nc1C)=O)NC1C(CCOC)C1 c1(OC)ccc(CNC(C)C(C)OCc2ccc(Cl)cc2)cc1N C12CC(CCO1)NC(=O)CC1(CC1)N(N(C)C)C2=O.C1(COCC)(CC)CC1 c1(C(C)=O)cc(C(N2CCC(O)(C(C)NC(C3CCOC3C)=O)C2)=O)ccc1C c1(C(=O)NCCN(CCCCCC)C(=O)CC=CCC2CCC2)ccc(CF)cc1 C1(C(N(CCCNC(c2coc(C(F)F)c2)=O)CCO)=O)C2CCC(=O)C12 C(=O)(CC(C(F)F)n1ccnc1)N(CCNC(C1CCCSC1)=O)CC C1(c2c(C(=O)Nc3nnc(C4CCOC4)s3)cccc2)COCCC1(F)F N1(C(CCN(C)C)=O)CC2(CCC(NC(c3nc4ccccc4[nH]3)=O)C2)C1 c1(NC(C(CC)NC(C2CC2C(F)F)=O)=O)cc(C(=O)O)cc(Br)c1 CC1CN2CCN1C(C(=O)NC(CNC(=O)Cc1ccccc1CO)C1CC1)C2 C(=O)(C(F)CCC(C)(C)C)N1CC2C(C(N(C)Cc3nnnn3C)=O)C2C1 C1(CNC(=O)CCC2CCC2)CCN(C(c2cc3cccnn3c2)=O)CC1(F)F c1(CC)cc(C(=O)NC2(C)CC(NC(c3ccccc3)=O)C2)ccc1C(F)(F)F c1(C(=O)NC(CN(C)C)C(=O)NCc2ccnc(F)c2F)ccc2cccnn12 CCC(C(=O)N1CCC(O)C1C(N1CC2(C1)CN(C(C)=O)C2)=O)C(F)(F)F N1(C2(C)C(NC(C(C)NC(=O)CN)=O)C2)CCCCC1 C1(OC)CC(NC(C2(SC)CC2)=O)CN(C(=O)C=Cc2ccc(C)s2)C1 C1(CC(=O)NC(C)(C)COC(F)F)CCCN(C(=O)CCCNS(C)(=O)=O)CC1 CCCC(CCC)C(=O)N1C(C(=O)NC2(C(=O)OC)CC=CC2)CC1C C12(C(N(CC(C)NC(c3cc(Cl)cc(F)c3)=O)C)=O)CC(C)(C1)OC2(C)C C(=O)(C(C)(O)C=C)N1CCC(CC(=O)NCC(=O)NCC#C)C1 c1(CC(=O)NC(C)(C)CCNC(=O)COc2ccon2)c(F)ccc(Cl)c1F C1(NC(CCc2ncc(C)[nH]2)=O)CCN(C(=O)COc2ccccc2O)CC1C CC1CN(C(c2ccc(Cl)nc2N)=O)CCC1NC(c1c[nH]nc1C(F)F)=O c1(CC(=O)NC2CC(CNC(C(N3CCOCC3)C)=O)C2)cccnc1F S1(=O)(=O)C2=CNC(=NCCNC3CCN1C3)C=C2.CCC(C)COC C12(CC(F)(F)C1)CN2.c1(CC(C2CC(CNS(C)(=O)=O)C2)=O)ccccc1 C(=O)(C(O)CC(C)(C)C)NC(C(N1CCC(C)(c2ccccc2)CC1)C(=O)NC)C N1(C(c2c(I)cn(C)n2)=O)C2CC3CC1CC(C2)O3 C1(C)(C(N(CC(=O)NCC)C)=O)CCN(C(c2cc(OC)nn2C)=O)C1 Cc1c(C(=O)NCC(C(C)C)NC(c2cncc(F)c2)=O)cnn1CC(C)C C1(C)(CC)CCC(NC(C2(NC(c3coc(C(N)=O)c3)=O)CC2)=O)O1 C1(C(=O)NC2C(c3onc(C)n3)C2)CC1C1CN(C(=O)Cc2ccccn2)C1 C1(CNC(c2c(C#C)c[nH]n2)=O)C2CCCC1N(C(=O)CC1OCCC1(C)C)C2 c1(CC(CC)NC(COCCC(=O)NCC#C)=O)cccc(OC)c1F c1(N2CC3C(NC(C(C)C4CCOC4)=O)C3C2)ncnc2sc(C(F)(F)F)nc12 Cn1ncc([N+](=O)[O-])c1C(=O)NC1CCCN(S(=O)(=O)C2CC2)C1 CCCC(C)C(=O)N(CCC(=O)NCC(C)(O)CC)CCO C1(C)(C(N2CC(N(C(CCCC3C(C)C3)=O)C)C2)=O)CCS(=O)(=O)CC1 c1(CC(C)NC(c2cncc(C3CC3)c2)=O)ccc(CNC(C2(C#N)CC2)=O)cc1 CCCCC(C)CCC(=O)N1CCCC(C)(CNC(c2ncn(C(C)C)n2)=O)C1 C1(NC(C(C)C)=O)COC2(C1)CN(C(=O)CCC1(C)CCC(=O)N1)C2 O=C(C1=CCOCC1)NC1(CF)CCN(C(=O)C=Cc2cocn2)C1 N1(C(CCSC)=O)CC(OC)C(NC(c2ccc(CN3CCOCC3)cc2)=O)C1 C1(C(=O)NCC2(C)CC(NC(c3cn(C)nc3Br)=O)C2)CC2(C1)CC2(F)F N1(C(C(C(C)C)C#N)=O)CCOC2(CCC(NC(=O)CCN3CCCC3)CC2)C1 c1(CC)cscc1NC(=O)C(C1CCC1)NC(=O)C=Cc1cscn1 C1(CNC(c2cc3ccoc3s2)=O)CC2COCC2N1C(C1(C2CC2)CC1)=O N1(C(c2c(C)ncs2)=O)CC(NC(c2cnn(C3CCC3)c2)=O)CC1C C(=O)(CCC(F)(F)F)N(CC(=O)N(CC=C)CCN(C)C)C.OC N1(C(C2CCCC(C)C2)=O)CCC(CNC(=O)CNC=O)C1(C)C C1(C(=O)NCC#C)CC2CCC1N2C(C1CCC(C)(C)C1)=O c1(CC(=O)NC(COC)C(=O)NCC(F)F)cccnc1C N1(CCOC)CCN(C(Cc2ncoc2C)=O)CC1.C1(CCCN)C=CC=CC=C1 c1(CC)c[nH]cc1C(N1CC(CC(=O)NN(C)C)(CC2CC2CO)C1)=O C(C(O)CO)(C1CC1)NC(CN(CC)CC)=O.N12CCC1C2=O N1(C(CC(CC)OC)=O)CCCC(CC)C1C(N1CCCN(CCO)CC1)=O C(=O)(C1CCCc2c[nH]nc21)NC1CCC(NC(c2c(C)cc(=O)n(C)c2)=O)C1 C(=O)(CCc1cccs1)NCC1(CCNC(COCC=C)=O)CC1 C1(NC(=O)CCCNC(C2(F)CCCC2)=O)CCC(F)(C(=O)NCc2ccoc2)C1 Cc1ccccc1C=CC(=O)NCC12CC(CO1)N(C(=O)C(C)OCC1CC1)C2 C1(OC(C2CCC3(CC2)CC3)=O)CCC(=O)N(CC(F)(F)F)C1 CN1CCCC(C)(C)C1N(CCC1CC1)CC1CC1 c1(C(=O)NC2(CNC(C=CC3C(C)C3(Cl)Cl)=O)CC2)cccc([N+](=O)[O-])c1 c1(N2CCC(CCNC(C3(C)CCOCC3)=O)C2)ncnn2c(Br)ccc12 C1(C(=O)NCC2C(C)CCN2C(c2occc2Br)=O)CC(C2CC2)=NO1 c1(CCC(=O)N(C2CNC2)C2CC2)ccc2ccccc2c1.C12CCCC1C(=O)O2 c1(CNC(c2ccc(OCOC)cc2)=O)cc2cc(C)ccc2[nH]1 N1(C(C(Cc2ccco2)NC(COCCCN(C)C)=O)=O)CCC(C(=O)OC)C1 n1(C(C)C)cccc1C(=O)N(CCCNC(=O)C(F)(F)C1CCCC1)C1CC1 CCC(CNC(c1cc(C)c(CC)o1)=O)(CC)C(=O)NCC1CCCC1N(C)C C1(C(C)C)CN(C(=O)CNC(=O)C2CC2)CCN1C(=O)NC1CC2CC2C1 Cc1cc(Cl)ccc1OCC(=O)NC1CCCC1CNC(c1cnoc1C)=O c1(C(=O)NCCOCCN(C)C(C2CC(F)(F)CS2)=O)cccc(C2CC2)c1 C(=O)(C(C)CC(C)C(C)=O)N1CC(C(=O)N(C(CCO)C(F)F)C)(COCC)C1 C1(c2cn(CCNS(C)(=O)=O)nn2)CN(C(c2ccsc2C(=O)O)=O)CCO1 S(=O)(=O)(c1cc(C(C)C)ccc1C)N1C(c2nc(C)no2)CC(OC)C1 C(C(C)C(F)C(=O)NC(C)CN1CCCC1)NC(c1cncc(OC)c1)=O c1(NC(C2(OCCSC)CC2)=O)cc(Cl)nc(C2CC2)n1 Cc1cc(NC(C2CC(O)CN2C(=O)CCS(N)(=O)=O)=O)ccc1OC(F)F N1(C(c2cnc(CC)nc2)=O)CCN(C(=O)C(CO)N(C)C)CC1CCO C1(CNC(c2cccc(OC)n2)=O)CC2(C1)CN(C(C1(C)CC(C)C1)=O)C2 c1(NC(C(CN(C)C)NC(C(CCC)C#N)=O)=O)cncc2ccccc12 C(c1cccc(N)c1)=CC(=O)NCC(C)NC(=O)CC(=O)NCc1ccccc1 c1(CC(N2C(C(=O)OC)CCC(F)(F)C2)=O)cccc2occc12 N1(CC)CCOC(C(=O)NC(CCSC)C(C)C)C1c1ccccc1 O=C(C1=CCCCCC1)NC(C(=O)NCc1nncn1C1CC1)C1CCCO1 CC1CN(C(C2(C(F)(F)F)CC2)=O)CC1NC(c1ccc(C2(F)COC2)cc1)=O CC(C)CC(O)C(=O)NC1C=CC(C(=O)NC2CC(=O)N(C)C2)C1 CC(C)CC(C)(O)CN(C(CCc1nnc(-c2ccccc2F)o1)C(C)(C)C)C n1(CC)nc(C(=O)NC2CN(C(c3cnnn3CC)=O)C2)c(=O)c2ccccc12 C(=O)(CS(=O)(=O)CC)NC1(CC(=O)N(CCCC)CC)COC1 N1(C(c2c(COC)n(C)nc2)=O)CCCN(C(=O)CCCc2ccsc2)CC1 c1(NC2CCC(CCCC)C2)ccc(S(=O)(=O)NCCn2cc(Cl)cn2)c(Cl)c1 N1(C(C(C)(C)N2CCCCC2)=O)CC2OCC(NC(=O)CCF)C2C1 c1(-n2cc(N3CC(NC(C(CC)N4CCCCC4)=O)C3)nn2)ccccc1C CC(C)C(CCc1ccccc1)C(=O)NCCN(C)C(c1ccc(N)c(O)c1)=O N1(C(C2CN(C)C2)=O)CCN(C(=O)C(C)(C)F)CC1C1CCCC1 CC(CNC(=O)CSS(C)(=O)=O)(Cc1ccccc1)NC(=O)CC1CCCOC1 CC1(C)OC2(CCN(C(=O)NCC3CCCC3NS(C)(=O)=O)CC2)NC1=O N1(C(CN(CCOC)C)=O)CCCC(N(C(=O)Cc2cc(C(F)(F)F)n[nH]2)C)C1 C=CC1(CN(C(=O)Cc2nccs2)CCNC(=O)C(C)(C)n2cncn2)CCC1 c1(C(N(CCNC(C(C2CC2)OCC)=O)C2CC2)=O)cc(C(C)C)n(C)n1 CC1CN(C(c2csc(-c3cnn(C)c3)n2)C(=O)NCSC)CC(C)(F)O1 c1(CC(N2CCCC(C)(CNC(C=C(CC)CC)=O)C2)=O)csc2cc(C)sc12 C1(F)(NC(c2ccc(OC)cc2CO)=O)CS(=O)(=O)CC12CCC2 C12(CNC(C(CC)CC)=O)CCCC1N(C(=O)COCCCF)CCC2 c1(CCC=C)ccc(C(=O)NC2CCC(C)(CNC(=O)CCOC)C2)cc1 c1(OC)c[nH]c(C(=O)NCC2(NC(C3CNC(=O)N3)=O)CCCC2)cc1=O C1(NC)CCCC12CCCN(C(=O)CC(C)(C)C(=O)OC)C2 C1(CC)CC(C(=O)N(CCCn2cc(C3COC(C)(C)O3)nn2)C2CC2)CCC1=O O(C=C(C#N)C(=O)N1CCCC1CCNC(c1cc(CC)on1)=O)CC CCCCCCN(C)C(C1CCOC1CNC(=O)CNC(C1CC1C)=O)=O N1(C(C=CC(C)NC(c2c(C)ncs2)=O)=O)CCC(O)C1C N1(C(C=C(CC)C)=O)CC2CCC(C1)N2C(=O)C(C)Oc1cc(C)ccc1Cl C1(NC(CC(CC)C)=O)CN(C(=O)C(c2ccc(F)c(F)c2)(F)F)CC1(C)C C1(CN(C(C(C)=C(C)C)=O)C)CCCN1C(c1cc(Cl)no1)=O c1(-c2nnc(C)o2)cccc(COC(C2CC(=O)N(c3ccccc3F)C2)=O)c1 C12(NC(CC(=C)Br)=O)CCN(C(c3cnc(C4CC4)nc3)=O)CC1C2 C1(NC(C2(COC)CCCC2)=O)CCCN(C(=O)C=Cc2ncc(C)[nH]2)C1 CN1CCC(C(N2CC(CCNC(c3csc(-c4ccccc4)c3)=O)C2)=O)CC1 C12(C(=O)NCc3cc(C)no3)C(NC(C3CC3(C)Br)=O)C3CC1C2C3 Cc1ccc(O)c(CC(N2CCCC2(C)CNC(=O)COc2cc(C)on2)=O)c1 n1(CC(=O)NCC(C)NC(C(C)CN(C)C)=O)nc(-c2ccccc2)oc1=O N#Cc1cccc(Br)c1C(=O)NC1(CNC(c2cc(F)c(F)cc2Br)=O)CCCC1 C1(=O)CCCCCNCCO1.c1(OC(C(=O)OC)C)ccc(C(C)C)cc1 CC(C(C)(C)C)=CC(N1CC(F)(CNC(=O)CCCOCC2CCCO2)C1)=O Cc1c(-c2cccc(Cl)c2)o[nH]c1=NC(=O)N(CCCC1C(=O)NN=C1C)C1CC1 c1(-n2c(C(=O)NCC3(C(=O)NCC4CC4)CC3(F)F)cc(C)n2)c(F)cccc1F CCC(CC(C)C)C(=O)NCCC(C(C)C)NC(C1CNC(=O)CC1(C)C)=O n1(CC=C)cccc1C(=O)NC1CCCC1CNC(c1scnc1C1CC1)=O C(C)(C)(C(C)NC(c1ccn(CC(F)F)n1)=O)NC(C1(CCOC)CC1)=O c1(OC)nc(C)c(C(=O)NC2CCC(NC(=O)C(CC)N3CCCC3=O)C2)s1 CC1(c2cn(CCNC(c3ccccc3Sc3nccs3)=O)nn2)CCOCC1 N1(C(C(C)Cc2cccnc2)=O)CCCCC(NC(C2(n3cncn3)CC2)=O)C1 C1(NC(C2C(=C)C2)=O)C2CC3C(C2)C13C(N1CC(C)(C(F)(F)F)C1)=O Cn1cc(SCC(N2CC(F)(CNC(c3cc(O)no3)=O)C2)=O)cn1 c1(OC)ncc(F)cc1C(=O)NC1CCCC1CNC(c1cc(Cl)c[nH]1)=O C1(NC(=O)C=Cc2cscn2)COC2(CCN(C(c3ccccc3CO)=O)C2)C1 C=C(C)CCC(c1nnnn1CCCOCC)NCC1CCN(CC(N)=O)CC1 c1(C(=O)N(C(C2(CCNC(C3CC=CC3)=O)CC2)=O)C2CC2)cc(O)cc(=O)o1 c1(C(N2CCC(CCNC(=O)C=Cc3ccncn3)C2)=O)cncc2c[nH]nc12 C#CCCC(O)C(=O)N1CCN(C(C2SCCS2)=O)C(C)C1 CC1(C(N2CC3CCC3(CNC(C34CCC(F)(CC3)C4)=O)C2)=O)CCC12CCC2 c1(CC)cnn(CC(=O)NC(C)(CNC(=O)CC2CCCOC2)C2CCC2)c1 N1(C(c2c(CNC(c3c(CC)nn[nH]3)=O)cccc2)=O)CCCCC(C)C1 C1(CNC(c2cnc(C)s2)=O)CC12CCN(C(=O)CCn1cc(Cl)cn1)CC2 c1(C(=O)NC2CCN(C(C3CC(C)C3)=O)CC(O)C2)ccc(S(=O)(=O)N(C)C)cc1 c1(OCC(=O)NC2CCCCC2NC(=O)CCC2CCC2)cc(F)cc(Cl)c1 C12(CC)CN(C(c3nncn3C)=O)C(CNC(c3cc(Cl)cs3)=O)(C1)C2 c1(CN2C3CC(S(CC#N)(=O)=O)CC2CC3)ccc2sccc2c1 C(=O)(CCCCCC(C)O)NC1CC2CN(C(C=C(CCC)CCC)=O)C(C1)C2 C(=O)(CCCC(=O)N1CCC(NC(C2CC(F)(F)C2(C)C)=O)C1)OC Cc1nc(C(=O)NC2(C)CCN(C(=O)CCN3CCCCCC3)C2)ccc1C#N n1(CCCC)cc(C(N2CCC(CNC(=O)C=CCF)C2)=O)nn1 C(=O)(CC(C)(C)CC(C)=O)N.C(C(C)(C)CNC(=O)C(CO)N(C)C)N(C(C)C)CC N1(C(C(C#C)(C)C)=O)CCN(C)C(C(=O)Nc2ccccc2C)C1 CC1(C#CC(=O)N2CCC(NC(c3ccc4[nH]ccc4c3)=O)CC2)COC1 CC(C)(C)CC(O)C(=O)NCC1CCN1C(=O)Cc1csc(NS(C)(=O)=O)n1 C1(C(=O)NCCC(=C)CNC(C)=O)CCN(C(=O)C(CC)CC)CC1 c1(NC2C(OC)CN(c3ncccn3)C2)ccc(F)c(F)c1Cl N1(C(C(CNC(=O)OC)(C)C)=O)CCC2(CCCC2CNC(C2(C)CC2)=O)CC1 C(C(C(=O)NCC(N1CCCCC1)C)C(C)(C)C)NC(C(c1ccc(C)o1)C)=O N1(S(CCC)(=O)=O)CCCC(C(=O)N(CCCN(C)C(C23CC(C)C2C3)=O)C)C1 CC(C)C(C)(CNC(=O)C(O)Cc1cn(C)cn1)NC(=O)CCCn1cccc1 C1(CCNC(COCCOC)=O)CCC(NC(=O)CCCC2CCOCC2)C1 N1(C(c2nnn(C)n2)C(=O)NCCOC)Cc2nccn2CC(c2ccccc2)C1 c1(C(=O)NCCC(C)NC(c2cc(CC)nc(O)c2)=O)cnc2ccnn2c1C N1(C(c2c(CC)ccc(Cl)c2)=O)CCC2CN(C(=O)C(=O)NC3CC3)C2C1 c1(C(=O)NCC(C2CC2)NC(C2(OCC)CCCC2)=O)ccc(F)cc1SC CC1CN2CCN1CC2C(=O)NCC1CCN(C(=O)CCS(C)=O)C1(C)C N1(C(c2c(OC)ccc(C)c2)=O)CCN(C(C23CCC(CC2)OC3)=O)CC(O)C1 C(=O)(C(C)CC(C)C(C)=O)N1CCC(C(N(CCCC)CC)=O)(CO)C1 Cc1cc(C)n(CCCC(=O)N(CC(C)CNC(C2(O)CC2)=O)C)n1 c1(C(N2CC(CCCCNC(COCC(=O)NC)=O)C2)=O)cc(N)cc(F)c1 C1(NC(C(F)OC)=O)C2CC3CN(C(=O)CCc4cnc(C5CC5)o4)C1C3C2 C(c1ccc(SC(F)F)cc1)=CC(=O)NC1CN(C(c2cc(C)sc2)=O)C(C)C1 CC(C)C(C)CC(=O)N1CC(c2ocnc2C(=O)NCC2C3CCC(F)(F)C23)C1 C1(C(=O)NC(c2cnc[nH]2)C)Cc2c([nH]c3cccnc23)CN1C(=O)CCC(N)=O c1(C(=O)NCC(C2CC2)NC(c2cccc(C)c2F)=O)cnn2c1CCCC2C C#CCC(CC(F)F)C(=O)NCC(CC)N(C(=O)Cn1nnnc1C1CC1)C N1(C(C2N(CCCC)CCCC2)=O)CCCC(C)(NC(=O)C(C)(CSC)OC)C1 N1(C(c2cccnn2)=O)CCC2(CC1)CC(NCc1ncccc1F)C2 c1(C(N2CC(CNC(CC(CC)C)=O)C(F)(F)CC2)=O)cnc2n1CCCCC2 Cc1cccc(OCC(N2CCN(C)CC2CNC(=O)Cn2cnnn2)=O)c1C N1(C(c2cc(C)ns2)=O)CCN(C(=O)C(C(C)C)c2nc[nH]n2)CC1C(C)C N1(C(c2nc(C)nc(O)c2)=O)CC2C3CCC(C2C1)N(C(c1occc1C)=O)C3 C(=O)(C(C)CN(C)C)N(C1CCN(C(=O)CCOCCCCNC(C)=O)C1)CC#C c1(C(=O)NC2C(CNC(C=C(C)c3ccco3)=O)C2)cnc2n(c1=O)CCS2 c1(C(=O)NC2C(C)CN(C(CC(C=C)(C)C)=O)CC2C)ccc2c(c1)OCCO2 C1(NC(C(C2CCCC2)OCC)=O)CCCC2CN(C(C3COC(C)C3)=O)CC12 CC(C(=O)NC1CCN(C(=O)COC(F)(F)F)CC1F)C(F)(F)F C1(NC(C(CC)C(C)(F)F)=O)CN(C(C2CC(F)(F)C2)=O)CC2CCCC12 CCC(CC)(CO)C(=O)N1CCC(CNC(c2cc(OC)c(OC)cc2O)=O)CC1C c1(-c2c(C(=O)NCc3cc(C)on3)ncs2)ccccc1C C1(C(=O)NCC(c2cnc[nH]2)C)CSCN1C(=O)Cn1cccc1 CCC(C(=O)NCc1cc[nH]n1)N(C)C(C1CC(C)(F)C1)=O c1(COC)nc(C(=O)N(CCCCCNC(=O)CC2C=CCC2)C)co1 C1(C(C(=O)N(C(C(=O)OC)C)C2CC2)C)CCN(C(c2ccn(C)n2)=O)C1 N1(C(C2CCCCC(=O)C2)=O)C2CCCC1CC(n1cc(C(=O)O)nn1)C2 CCC(C)(C)CC(=O)NCC1CCN1C(c1[nH]c(C)cc1C)=O C1(O)(CCNC(c2cnc(OC)s2)=O)CCN(C(=O)CC2(O)CCCOC2)C1 C1(NC(CCc2cc(OC)no2)=O)CCCN(C(c2ccncc2)=O)C1C C1(NC(c2c(CC)ccs2)=O)CCC2CN(C(C3CCCOC3C)=O)CC2C1 N1(C(C=NOC)=O)CCCC2(NC(=O)COc3cc(F)cc(Cl)c3)CCCC12 Cc1[nH]nc2c(C(=O)NC3(CNC(=O)CC(C)F)CCCC3)cccc12 c1(C(=O)NCC2CN(C(C3C(C)(C)COC3)=O)C2)ccc(O)c(F)c1 Cc1ccc(C(=O)OCc2csc3cccnc23)c(=O)n1C N1(C(C(C)(C)OCCC)=O)CC2CC(C(N3CC(CO)C4(CC4)C3)=O)CC2C1 Cc1cnc(C(N2C3CC2CN(C(c2oc(C(C)C)nc2C)=O)C3)=O)cc1Cl Cc1cc(C(=O)NC2CC(C)N(C3CCN(C(=O)NC4CC4)CC3)C2)cc(Cl)n1 c1(C(=O)NC2CCCN(C(=O)Cc3sccc3Br)C2)cn2c(n1)CCCC2 C(=O)(CCCCC(C)C)OCC.C1CCCCC(=O)N2CC(O)(C2)c2cn1nn2 c1(OC)cccc(I)c1C(=O)Nc1ncc(CCNC(=O)CCC(C)C)s1 CCC(CC)(C(N)=O)NC(C1(F)CN(C(c2ccc(=N)[nH]n2)=O)C1)=O C1(OC)CC(NC(c2ccc(C)cc2)=O)CN(C(=O)C(C(C)C2CCC2)N(C)C)C1 c1(C(=O)NCC2N(C(CC(CCC)(C)O)=O)CCCC2)ccc(C=NOC)cc1 C1(C)(CC)CC(NC(=O)CC(C)(C)O)CN1C(=O)C(N)=O CCCC(C)CC(=O)NCC1(O)CCN(C(=O)C(c2ccccc2)C2CC2)C1 c1(C(C)CC(=O)NC(C)CCNc2ccccc2)ccc([N+](=O)[O-])cc1 C(=O)(C(C)(C)C(=O)NC1CCCCC1NC(C1CCCCS1)=O)OCC C1(CCC(=O)Nc2cn(CCCN3CCOCC3)nn2)CCc2ccccc2C1 c1(C(N2C(C)CC(CNC(=O)Cn3cncn3)C2)=O)cc(N)cc(F)c1 CCCCCC(F)C(=O)N1CCC(NC(c2c[nH]nc2CC)=O)C1 c1(C(=O)NC2CCCC(NC(CN3C(C)CCC3)=O)C2)cc2scc(Cl)c2[nH]1 c1(C(=O)NC2CN(C(C)=O)C2)ccc(NC2NC(=O)CC2C(F)(F)F)cc1F c1(CC(=O)NC2CC(F)(CNC(C(CC#C)C)=O)C2)cccc(C)c1C Cn1nc(O)cc1C(N1CCC(Cn2cc(Cn3cc(N)cn3)nn2)CC1)=O c1(C(N2CCC(NC(CCSCC(C)C)=O)C(F)C2)=O)ccc2nc[nH]c2c1 C1(C(=O)N(c2ccccn2)Cc2ccc(F)cc2)CC(F)(F)CC1O C12(C(N3CC(CN(C(CS(=O)(=O)NC)=O)C)C3)=O)CCCCC1NC(=O)C2 c1(C(N2CC3CC2CN3CCOc2cccc(Cl)c2)=O)cnn2c1CCCC2 c1(OCC(N2CC(NC(C(C)N3CCC3)=O)C2)=O)nn(C)cc1Br n1(CC)ccc(CC(=O)N(CCCCCNC(c2c[nH]nc2C)=O)CCO)n1 C1(C(=O)NC2CC(CCC(=O)NCc3ccc(C)o3)C2)(CC)CCNC1=O N1(C(c2c(OC)cnnc2)=O)CCC(C(=O)NCC2CCSC2)CC1C c1(NC(=O)NCC2CC2NC2COC(C3CCC3)C2)ccc(OC(F)F)c(Cl)c1 CN(C)S(=O)(=O)N(C)CC(=O)NCC1(NC(=O)C(c2cc(Cl)no2)OC(=N)O)CC1 c1(CC(=O)NCC(C(C)C)NC(c2ccnn2CCF)=O)cnccc1C(F)(F)F c1(C(=O)NC2CN(C(c3cc(C(C)C)nn3C)=O)C3C2C3)sccc1S(C)(=O)=O C1(CNC(=O)CCC2CCOC2)CC2CC2N1C(C1CC(=O)N(CC2CC2)C1)=O C=C(Cl)C(C)(C)C(=O)NC1CC2(C1)CC2NC(C1(C)CC2CCC1O2)=O c1(OC)ncccc1CC(=O)NC(C1CCCN1C(c1ccncc1Cl)=O)C N1(C(C(F)OC)=O)CC2CCCC(CNC(=O)CC3CCS(=O)(=O)C3)C2C1 C=CC(CCC)CC(=O)NCCOCCCN(C(=O)CC1CC=CC1)C c1(NC(CN(CC(CCCC)CC)C)=O)cc([N+](=O)[O-])ccc1Br C#CCCN=C(NCCC1(OC)CCC1)NCC1CC1.C(C(=C)Br)N(C)C C12(C(N3CC(CC)SCC3)=O)CC(C)(CN1C(=O)CCCC(C)C)C2 C1(C(=O)NC(CO)C2CC2)CC(O)CN1C(c1nc(Cl)sc1Cl)=O Cc1conc1C(=O)N(CC(C)O)CCNC(=O)Cn1ccc(CC(C)C)n1 N1(C(C2(c3ccc(OC)c(C)c3)CC2)=O)CCC(C2CC(F)(F)C2)C1 C(=O)(C(C)(O)CC(C)C)N(CC(=O)NCCC(C)N1CCCC1)CCC N1(CCC)CC(C(N2CC(NC(c3nocc3C3CC3)=O)C(F)C2)=O)CC1=O N1(C(C2C(c3c(C)ccs3)C2)=O)CCC(NC(=O)C(C)N(C)C)C(O)C1 N1(C(CC(CC)C2CC2)=O)CCN(C(c2cn(C)c(=O)cn2)=O)CC(CO)C1 C1(CNC(CCCOCC=C)=O)CC(C)(C)CN1C(=O)C(O)C(F)(F)F c1(CN2CCN(C(c3ccccc3[N+](=O)[O-])=O)CC2)cc(C2=CCS(=O)(=O)CC2)cs1 c1(C(=O)NC(CN(C(c2cc3nc(C)sc3[nH]2)=O)C)C)cc(C)cc2c[nH]nc12 N1(C(CSCCCC)=O)CCCC(N(C(=O)C(CO)N(C)C)C)C1 c1(N(C)Cc2cc(C)no2)ncc(N)c2ccccc12 CC1(C)CCN(C(=O)Cn2cnnc2)CC1C(=O)NCC1(C)CCC(=O)N1 c1(N(C(c2cccnc2OC)C(=O)NC)C)c(C)cccc1C C12(C)CCC(O1)C(=O)NCCCCCNC2=O.c1(CC)ccc(NCC(F)(F)F)o1 N1(C(C(C=CCCC)O)=O)CCC(CNC(c2ncccc2OC(F)F)=O)C(C)C1 c1(C(N2CC3(CN(C(C(c4ccc(O)cc4)C)=O)C3)C2)=O)cc(Br)cc(Cl)c1O C(C(=O)NC1CN(C(=O)CC(=O)Nc2nccs2)CC1O)(C(C)C)SCC c1(C(=O)NCCCNC(c2cc(C)cc(Br)c2)=O)c(C)oc(C)c1S(N)(=O)=O C1(F)(CNC(C2(C)CC2(F)F)=O)CCCN(C(=O)CCc2cnc[nH]2)CC1 C(=O)(CCCCC(N)=O)N1CC(C)C(NC(=O)Cc2cccs2)CC1 C1(C(=O)NCC2(F)CCN(C(COCC(C)(C)C)=O)C2)CCc2nccn2C1 c1(NC(C)=O)nc(C)c(S(=O)(=O)N2CCOCC(NC(C3CCCC3)=O)C2)s1 C1(NC(c2cc(C)ns2)=O)CN(C(c2cc(Cl)cnc2O)=O)CC2(CCC2)C1 C1(O)(CN(C(Cc2c(CC)con2)=O)C)CCN(C(c2ccc(CO)nc2)=O)C1 C(=O)(C1=CCC(NC(=O)C(C(C)C)OCC(C)C)C1)NC(C(=O)N(C)CC)C C(C(C)(C)C(=O)N1CCCC(OCCn2cc(CC3CCC3)nn2)C1)SC C(N=c1[nH]c(N2CCC(N3CC(O)C3)C2)nc2cc[nH]c12)C1(C)COC(=O)N1 c1(C(c2n(C(C(=O)OC)C)nnn2)NCCCNC(C)=O)c(Br)noc1C c1(OCC)sccc1C(N1CC(OCCNC(c2ccc(O)s2)=O)C1)=O c1(NCC(C)(C2CC2)OC)nccc(=NCc2cnc(C)c(Br)c2)[nH]1 c1(OC)ccc(CN2CC3C(C(=O)Nc4ncn5ccccc45)C3C2)cc1C#N c1(OC)ccc([N+](=O)[O-])c(NC2(C(N)=O)CN(C(=O)CCn3ccc(C)n3)C2)n1 c1(CNC2CC(CCC(=O)Nc3cn(C4CC4)nn3)C2)cnccc1Cl c1(C(=O)NC(CNC(C(CC)CC)=O)CO)c[nH]c2nc(Br)ccc12 C(CC(O)CC(=O)NCC1(F)CC(CNC(c2ccccc2OC(F)F)=O)C1)SC C=CCC(C)C(=O)NC(C1CCCN1C(c1cc(C2CCC2)nn1C)=O)C C1(C(N2CC(COC)(CNC(C3C(C)CC3C)=O)C2)=O)CCS(=O)(=O)CC1 CCC(C(=O)NC(C)CC1CN(C(C2(CC(C)C)CC2)=O)C1)OC1CCCCC1 c1(CN(C(=O)CCn2cc(CC3(Cl)CC3(C)C)nn2)C)ccc(C(F)F)cn1 c1(CC)ccc(Cl)c(C(N2CC3CC2CN3Cc2cccc(NC)c2)=O)c1 c1(CC)nc(C(N2CC(NC(=O)C(C)c3ccsc3)C(O)C2)=O)c(N)s1 C1(OC)(CNC(=O)CC2(CSC)CC2)CN(C(C2CCCN2C)=O)C1 C1(NC(C2CN(C(N)=O)C2)=O)CCOCC1NC(=O)Cc1cc[nH]c1 c1(C(N2CCC(N(C(=O)C(C)C(O)CC)CC)CC2)=O)cc(F)cc2nc[nH]c12 C1(C(=O)NC(CC2CC2)CC2CC2)C2Cc3c(Cl)cccc3C12 c1(CN(C(C2OCCN(C(C3(CC)CCCO3)=O)C2)=O)C)cccc(F)c1F c1(C(=O)NCC2C(NC(c3c(C(C)C)onc3)=O)CCC2)cccc(F)c1 C1(C(=O)NC2CN(C(CCOC(C)=O)=O)CC2(C)C)CNC(=O)C(C)(C)C1 N1(CC(CCC=C)C)CCC2CN(C(c3ccccc3)C)CC12 c1(C(N2CCN(C(CC(CCC)C)=O)CC2COC)=O)c(F)ccc(Cl)c1F C(=O)(C(CNC(C1(F)CC1)=O)CC1CCCC1)N(CCCC(O)CO)C c1(Nc2ncc(C(=O)OC)s2)cc(CO)ccc1NC(C1CC=C(C)CC1)=O C1(C(=O)NCC(N2CC(CC(COCP(C)(C)=O)(C)C)C2)=O)(OC)CCCSC1 c1(C(=O)NCCC2CN(C(=O)OC(C)(C)C)C2(C)C)cccc(Br)c1O CN1CCc2cc(C(N3C(C(=O)Nc4cc(I)ncn4)CC4CC34)=O)ccc2C1 N1(C(C2CCN(C(C)=O)CC2)=O)CC(F)(F)CC1C(N1CC(=O)NC(C)C1)=O N#Cc1ccccc1C(N1CCC1CO)CN1CCC(O)(c2cnn[nH]2)C1 C1(=O)C2=NOC(C2)OC(=O)N(C2CC3(CCC3)C2)C(C)CN1.C(C)(C)(C)OC N1(C(CCOCC#C)=O)CCC(C)(C)C1C(=O)NCC(C)(O)CO N1(C(C23CCCC2C3)=O)CC2(CCN(NC(c3[nH]cc(CC)c3)=O)CC2)C1 C1(C(N(CC(C)N(C(=O)C(c2ccccc2F)C)C)C)=O)Cc2nnsc2S1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCC1CCC2(CN(C(CCC3(C)CC3)=O)C2)O1 CC(C)(C)C(CNC(c1c[nH]c(Br)c1)=O)NC(C1(C)CC2CC2C1)=O C1(C(=O)NCCOCC(=O)NC)CN(C(c2coc(C(N)=O)c2)=O)CC(C)(C)C1 C1(CNC(C(C(C)C)O)=O)CCC2CN(C(=O)C(C3(O)CCCC3)F)CCC2C1 C(=O)(C(C(C)CC)NC(N)=O)NC1(C)CN(C(COC2(C#C)COC2)=O)C1 C(N=c1cc(C)nc(C2CCC2)[nH]1)C1CN(C(C(C(CC)C)C)=O)CC1(C)C C1(CC(N2CCC(Cn3cc(-c4cccnc4)nn3)C2)C)CCCC(C)(C)C1 Cc1cc(-c2nc(CC3CCCC3(F)F)n(CC(C)(C)CO)n2)c(C)o1 Cc1ccc(CNC(C2CCN(C(c3nn(C)c(C)c3Br)=O)CC2O)=O)c(F)c1 N1(C(C=CC(C)C)=O)C(C(=O)Nc2cnc(Br)cn2)CCC1C C12(CNC(CC(=O)N(C)C)=O)CC(NC(c3cc(F)c[nH]3)=O)(C1)C(C)(C)O2 C(=O)(CC(C)CCCCC)N(C1(C(=O)NCCC(=C)C)CCC1)C1CC1 N1(C(CCC#CC)=O)CC(C2CCCCN(C(c3cccnn3)=O)C2)C1 CC(C)(C)C(C#N)C(=O)NC1(CNC(=O)C=Cc2cccc(Cl)c2)CCCCC1 N1(C(c2nc(OCC)sn2)=O)CCCCC1C(C)NC(c1cc(Cl)c(Cl)[nH]1)=O C1(C2(O)CCN(C(C34CCCCC3CCC4)=O)CC2)(NC(C2CC2(Cl)Cl)=O)CC1 c1(OC)cccc(Cl)c1C(=O)NC1CCCC1C(=O)Nc1ccc(C)nc1 C1(NC(=O)CSc2ccccn2)CCCCN(C(C2(CO)CCCC2)=O)C1 c1(C(=O)OC)c(NC(C2CCC(NC(C3CCC(=O)N3)=O)C2)=O)ccnc1Cl c1(C(N2CCN(C(CNC(CCC)=O)=O)C(C(F)F)C2)=O)c(F)cc(N)cc1F c1(C(c2n(C)nnn2)NCc2cnn(C)c2Br)cc(F)cc(Cl)c1 C1(NC(C(C)=C2CC2)=O)CN(C(=O)CCC2CCC2)C2(CCCOC2)C1 C1(CNC(c2c(CC)cno2)=O)CCCCCN1C(=O)CC1COC(C)(C)C1 c1(NC(CCN(C2CC(O)(c3ccncc3)C2)C)=O)cccc(Cl)c1 C1(O)(C(N(CC(=O)NC)C)=O)CCN(C(c2nccc(C)n2)=O)CC1 C(=O)(C(S(C)(=O)=O)C1CC1)N(C(CNC(C(C)C1CCC1)=O)C1CC1)C CCC(CCC(=O)N1CCCC(F)C1)NC(C1CC2(CC2)CO1)=O C1(NC(c2n(C)ccn2)=O)CCC(C)(CNC(C23CC2CCC3(F)F)=O)CC1 N1(C(CN(C)CS(CC)(=O)=O)=O)CCN(CCN(C(=O)COC)C)CC1.C1CCC1 N1(C(C(C)C)=O)CC(CNC(c2ncoc2-c2cccs2)=O)C2(CCOCC2)C1 C1(NC(C2CC(N3CC(O)C3)C2)=O)CCCN(C(C2CCS(=O)CC2)=O)CC1 N1(C(C(C)OCCCC)=O)CCC(CO)(NC(c2cc(C(F)F)cs2)=O)C1 CC(C)(CCC(=O)N1CCC(CF)(NC(=O)C2=CCCOC2)C1)c1ccccc1 c1(C(N2CCC(OCCNC(CCCC(C)O)=O)CC2)=O)cnc2ccccn12 CC1(C)COCC1CC(=O)NC1(CCCCNC(C2CC=CC(O)C2)=O)CC1 c1(OC)cc(CCNC(=O)N(C2CCN(C)C2)C(C)C)ccc1F c1(SCC(=O)NCC(CNC(c2c(C(C)(C)C)c[nH]c2)=O)CO)ccccc1F C1(C(=O)NC(CCNC(C(C)C)=O)C)CC2CS(=O)(=O)CC2C1 C1(CNC(C(CC)(C)OC)=O)CC12CCN(C(C1CCCN(C(C)C)C1)=O)CC2 c1(OC)cnc(C(=O)NCC2CCCN(C(C3CC4CCC3C4)=O)C2)nc1 c1(C(=O)NC2C(CNC(CCCCCSC)=O)C2)noc2ccc(Cl)cc12 C(CCCCC(=O)N1CC(O)CC1C(C)C)NC(CN1CCC(C)CC1)=O c1(CC(=O)NC2CCN(C(c3cc(CO)[nH]n3)=O)CC2O)nc2c([nH]1)CCCC2 Cc1nsc(C(=O)NC(C)CN(C(=O)CC2CC(O)C2(C)C)C)c1N CC1(C)C2CC1CN(C(=O)CN(C1CCC1)C(C1CC(C)(O)C1)=O)C2 c1(CC)c(C(=O)NC2CC(C)(CNC(=O)CCC(=O)N(C)C(C)C)C2)cccc1F c1(C(=O)NCC(C(C)C)NC(=O)CCc2cccc(F)c2F)cc(O)cc(O)n1 CCCC(C(O)C(=O)NC(CC)C(N)=O)NC(=O)CN1CC(C)(OC)C1 Cc1c(Br)ccc(F)c1CN1CC(C)(CNC(C2CCCOC2)=O)C1 Cc1oc2nc(Cl)ccc2c1C(=O)N(CC(O)CNC(C1OCCO1)=O)C C(=O)(C1=CC2CCCCC12)N(C1CC(NC(c2ccc([N+](=O)[O-])c(O)c2)=O)C1)C c1(C(N2CCC(CNC(CC3(C)CC3F)=O)C2)=O)ccc(Cl)c2occc12 c1(C(CNC(=O)CCSCC(N)=O)N(C(=O)Cc2ccns2)C)cccc(O)c1 CON(CCC(=O)NC1CCn2ccnc2C1)C(=O)C1CCCCC1 O=C(N=c1cc(NC(=O)CSc2ncccn2)[nH][nH]1)c1cc(F)ccc1I Cn1c(C(=O)NC2CCC(CNC(c3ccsc3)=O)C2)cc2cc([N+](=O)[O-])ccc12 C1(CC(C)NC(c2cc(C)sc2)=O)CCN(C(=O)CC(C)O)CC1 N1(C(C2CCN(C)CC2c2ccnn2C)=O)CCNC(=O)c2sccc21 Cc1ccc(C(=O)C(=O)NCC(C)CNC(=O)C(C)n2ccnn2)cc1 C1(C(N2CCN(C(C(=O)OC)=O)CC2)=O)COCCN(Cc2cccn2C)C1 c1(CC(=O)NC2CCN(C(C3C(c4cn(C)nc4)OCC3)=O)C2)cnccc1Cl C1(C)(CC)C=C(C(=O)NC23CCC(CNC(=O)CCCC(=O)N(C)C)(C2)OC3)C1 CCCC(CC)CCC(=O)N1CSCC1C(=O)N(C(C)C1CC1)CC Cc1cc(F)c(C(N2CCC3C(C2)CN3C(=O)C(C)C)=O)cc1Br c1(CC)oc(C(=O)NC(C2CCN(C(C3CC3CC(C)C)=O)C2)(C)C)cc1C C1(NC(C2CC(C(F)(F)F)(OC)C2)=O)CCCC(NC(=O)Cn2nccc2C)C1 c1(N(CC)CC)ccc(C(=O)OC)cc1C(C)(C)O.n12cc(nn1)C1COCC1CC2 c1(C(=O)NCC=CCNC(CCCCSC)=O)nc2c(Br)cccn2n1 C1(NC(CCN(C)C)=O)CN(C(c2cc(C(F)F)no2)=O)CC2CCCC12 C(=O)(C1=CCSC1)N1CC(OCC)(CNC(C2CCC(OC)C2)=O)C1 C12(C(=O)OC)COCCC1(F)CN(C(=O)C=CC(C1CCCCC1)=O)C2 c1(OC)cncc(C=CC(=O)NC2C=CCN(C(c3ccoc3Br)=O)C2)c1 c1(OC)ccccc1NC(C1(O)CCN(C(=O)COCC(C)C)C1)=O C12=CC=C(C=C1)C2.c1(C(C(=O)NC)N(CCF)C2CC2)c[nH]nc1C c1(C(=O)NC(C(C)NC(c2csc(F)c2)=O)CO)ncc(C(F)(F)F)cc1Cl N1(C(C(CC)SC)=O)CCN(C)CC1C(=O)NCc1nnn(C)n1 c1(C(=O)NCC2(NC(C=CC(C)(C)SC)=O)CCOC2)cc(C#N)c(N)cc1O c1(C(=O)NC(C)C(=O)NCC2CCN2C(c2cccc(F)c2)=O)c[nH]cc(Cl)c1=O C1(CC(=O)NCC(CNC(C(CCOC)C)=O)(C)OC)CCC(C)(C)CO1 C(CC(C)P(C)(C)=O)N(CC)Cc1ccc(C(c2ccccc2)O)cc1 N1(C(C2(CC)CCN(C(c3cc(C(C)=O)c[nH]3)=O)C2)=O)CCC2(CC(OC)C2)C1 n1(C(CC)CC)nc(-c2cscn2)nc1-c1cc[n+]([O-])cc1 CC1(C(=O)NCC2CC(NC(=O)Cc3cncnc3)C2)CC2CCC1O2 CN1C(=O)CCCC1C(N1CCOCC1CNC(C12CC(C#N)(C1)C2)=O)=O C=CCC(C)C(=O)N1CC(CC)(NC(=O)CCCn2ccccc2=O)C1 c1(C(N2CC(C)CC(NC(Cc3c(C)ccs3)=O)C2)=O)cn(C)c(=O)c(C)n1 C(=O)(C1CCCc2n[nH]cc21)N(C1CCN(C(c2cnc(C)nc2)=O)CC1)C n1(CCC)nnnc1C(C1CCCCC1)NCC1(CCC)CCC1 C1(C(N2CCC(C(N(C3CCN(C)C3)CC#C)=O)C2)=O)CCN(C)C(=O)C1 c1(C(=O)NC(C(C)NC(c2c(CC)sc(=N)[nH]2)=O)C)cn2cccc(F)c2n1 c1(C(C)(C)Nc2c(C)cccc2)cccc(C#N)c1 c1(OCCC)ccc(S(=O)(=O)N2CCCCC(C)C2)cc1NC1CC1 C(CO)(CCCCNC(c1cccc(O)c1F)=O)NC(c1c(OC)cc(C)s1)=O Cc1ccc(C(=O)NCCCc2csc(C)n2)cc1-n1cccc1 N1(C(C2(C)CCCN(C)C2)=O)CC2CC(NC(C34CCC(CC3)OC4)=O)CC1C2 C(=O)(C1=CC2CCCC12)N1CC2C(NC(c3cccc(Br)c3F)=O)C2C1 C(N=c1[nH]c(N2CCc3sc(Br)cc3C2)nc2c1CSC2)C1N(CC)C(=O)CC1 C(=O)(CCCCCNC(N)=O)NCCC1CCN(C(Cc2nc(=N)[nH][nH]2)=O)CC1 c1(OC)ncccc1C(F)(F)C(=O)NCC(C)NC(=O)C(F)Cc1ccccc1 N1(C(c2c(OC)ccs2)=O)CC2(CCCCN2C(c2cc(C)c(C)nn2)=O)C1 C1(C(=O)NC2(CCOC)CCC2)C2CN(C(=O)CCCCC3CC3)CC12 C(=O)(C(C)C(=O)NC(C(=O)NC(c1cncc(F)c1)C)C1(O)CCC1)OC Cc1cnn(C(C)C(=O)NC2(C(=O)NC(C)Cc3ncn(C)n3)CC2(C)C)c1 c1(CC(=O)NC2CCCN(C(=O)CCc3ccc(F)cc3)CC2)ccc(O)cc1Cl C(C(CO)N=c1nc[nH]s1)NC(C1Cn2c(C)cnc2CC1)=O C(=O)(C(F)CC(C)(C)C)N1CC=C(C(=O)N(C2C(C)CCC2)C)C1 c1(-c2cc(C(=O)NCC=CCNC(CSC)=O)no2)ccc(C)cc1 c1(NC(C(C)CNC(c2cccnc2O)=O)=O)cn(C)nc1C#N c1(C(N2C(C)CCN(C(C3CC(C#C)(O)C3)=O)CC2)=O)nn2c(c1C)OCCC2 Cc1c2c(-c3cnc(Cl)c(C(=O)NCC(N4CCCC4)=O)c3)cccc2nn1C c1(NC(C(CC)(CC)CO)=O)cc(S(=O)(=O)NC2CCC2)ccc1OC CCS(=O)(=O)CC(=O)N1CCC(C2CCCN2C(c2cc(Br)n[nH]2)=O)C1 CN1CCCC1C=CC(=O)NCCCC1CN(C(c2ccnnc2)=O)CCO1 N1(C(C2CC2C(F)F)=O)CCN(C(c2snc3ccccc23)=O)C2(CCC2)C1 C1(C(CN)=O)CC12CCC2.N1(OCOC)CCCCC1 N1(C(CCCC(=O)NCCC)=O)CCC(F)(F)C(CNC(c2cc(F)cs2)=O)C1 c1(C(N(C(CC)C(=O)OCC)C)=O)cc(C(N)=O)cc([N+](=O)[O-])c1 Cc1occc1C(=O)NCC1CCN1C(=O)C(C)c1cccs1 C1(NC(CCCCSC)=O)CC2CCC1(NC(c1cccnc1OC(C)C)=O)C2 c1(C(=O)OCCOc2c(C)nc3ccnn3c2)ccc2c(c1)c(C)c(C)n2C N1(CCC(C(=O)OC)(C)O)CCCc2ncccc2C1 C1(C)(C(N2CC(NC(c3cc(C)ncn3)=O)C3(C2)CC3)=O)CCCCNC1=O C1(C(=O)NCC(CC=C)NC(c2ccc(CO)cc2)=O)CC(=O)C1(C)C C1(NC(c2ncn(CC)n2)=O)CCN(C(=O)CC2CC(SC)C2)C1C C1(CN(C(C=CC(=O)N(C)C)=O)C)CCCCN1C(=O)CC1(C)CCC1 c1(C(=O)NC(CC)CN(C(=O)C(O)CC2CCCCC2)C)c(C)cnn1CC C=CCC(CC(=O)N1CCOCC1CC)NC(=O)Cc1cccc(O)c1 CCC(C)(CO)C(=O)N1CCCC(CCNC(=O)Cc2cnc[nH]2)CC1 C1(CC)CCN(C(=O)Cc2cncn2C)C(C(=O)NC(C)CN=[N+]=[N-])C1 Cc1ccc(NC(C2COC(C(F)F)C2)=O)c(Cl)c1O C(CC(=O)NCC1=CCN(C(=O)C2=CS(=O)CCC2)CC1)(C(F)(F)F)OC C(=O)(C#CC1CC(F)(F)C1)N1CCCC(O)(CNC(C(C(=O)N(C)C)(C)C)=O)C1 c1(C(=O)NCCN(C(C)(C)C)C(c2cc[n+]([O-])cc2)=O)ncccc1F C(=O)(C(C)C(C)NC(c1sc(F)cc1C)=O)NC(C1CCCCC1)CC C(CN=C(NCc1ccc(C(F)(F)F)cc1)N1CC2C(C(=O)N(C)C)C2C1)SC CCC(CCOC)C(=O)NC(C)(CNC(=O)Cc1cc(C)nn1C)C(C)C C(CC)(CS(=O)(=O)c1ccccc1)Sc1n(CC)c(CC2CCCCN2)nn1 C1(C(=O)NCCC(C)NC(=O)C(C)(O)C2CC2)COC(=O)N1C c1(CN(C2CCN(C(c3ccc(C#C)cc3)=O)C2)C)cccc(F)c1C#N N1(C(CC2(C=C)CC2)=O)CCC(CO)CC1CNC(c1cnn(C(C)C)c1C)=O N12CC(C(C)C1)C2=O.N1(CCNC(C(C2CCC2)OCC)=O)CC2CC2C1 c1(Nc2c(F)cc(-c3cn(C)nn3)cc2F)ccc2c(c1)OC(F)(F)O2 c1(CC)cc(NC(C2COCCC2NC(c2cc([N+](=O)[O-])c[nH]2)=O)=O)cc(F)c1 n1(CC(=O)NC(C(=O)N(CC(CC=C)O)C)CN(C)C)cccnc1=O CC1(C)CC(NC(=O)COCC2CCCOC2)CN1C(c1cnn(C(F)F)c1)=O N1(C(c2c(CC)scn2)=O)CCN(C(=O)CCOc2cccc(C)c2)C(C)C1C c12cc(n(C)n1)C(=O)NC1(C)CC(C1)NC2=O.c1(CC)ccsc1OC c1(C(=O)NC2C(CNC(c3ccccc3)=O)CCCC2)[nH]nc2ncnc(O)c12 c1(CC(=O)NCCCCNC(C2N(CCC)C(=O)CC2)=O)cnn2c1CCCC2 C1(CC)CC12CCOC2.C(=O)(C(C)(C)N1CCCC1)N(C(=O)COC1CCOC1)C c1(CCC)cc(C(=O)NCC2COCCN2C(=O)Cc2ccccc2C)ccn1 c1(OC)cnc(C(=O)NCCC2CCCN(C(=O)C(C)C(C)C)C2)nc1 Cc1cc(C(=O)NCC2CCCCN(C(C3CCOC(C)(C)C3)=O)C2)c(C)cn1 c1(C(N2CC3C(NC(c4c(C)cnnc4)=O)C(C3)C2)=O)c(C)oc2ccccc12 C(=O)(NN=c1[nH][nH]c(=NC2COCC2c2ccccc2)s1)C1C(OCC)C1 CC(CCC(C)(C)C)C(=O)N1CCCC(Nc2ccc(C#N)nc2)CC1C CCCC(C(=O)OC)C(=O)N1CC(OC)CC1CNC(=O)COc1ccccn1 c1(OCC)ccc2cc(CN(C(C3CCSC(C)C3)=O)C3CC3)[nH]c2c1 c1(OC)c(C(N2CCCC(CNC(=O)CC3C=CS(=O)(=O)C3)C2)=O)cccc1N c1(C(=O)NCC(C)(CNC(C2CCCN2C2CC2)=O)OC)ncc(C)cn1 c1(C(N2C(CCNC(C3OCC(C)(C)C3)=O)COCC2)=O)cnc2ccccn12 C1(C(N2CCN(C(C3CCC3c3ccco3)=O)C2)=O)SC2C=CC1CC2 N1(C(c2n(CC)ccc2)=O)CCCC(CNC(=O)C(C)Nc2nc(C)cs2)CC1 c1(CC(=O)NC(CNC(C=C(COC)C)=O)C2CCC2)ccc(OC)cc1 C(C(C)CC(=O)NC(C1CCOCC1)C)NC(c1ccn(COC)n1)=O c12ccnc(c1)NC2=O.Cc1coc(C(N2CCC(C(=O)NC3CCC3)C2)=O)c1 C1(NC(c2cccc(N(C)C)c2)=O)CN(C(=O)CO)CCC1O Cc1nc(C2CC2)sc1C(C(=O)NC(C)CC#N)N(C(C)C)C1CC1 C(N=c1nc(O)c2ccccc2[nH]1)C12OCC(NC(C(C)N3CCC3)=O)(C1)C2 CS(=O)CCC(=O)N1CCC(CCNC(=O)CC23CCC(CC2)C3)CC1 C1(C(=O)NC(C)Cc2nn[nH]n2)(NC(=O)C=CC2CCCN2C)CCC(C)(C)C1 c1(NCC(=O)NCC(CO)NC(C2N(C)C(=O)CCC2)=O)ccc([N+](=O)[O-])cc1 FC1CCCCCC1N=c1[nH]c(-c2ccc3c(c2)COC3)nc2cc[nH]c12 N1(C(C2(C#C)CCCC2)=O)CCC(N(C)C(C2CN(S(C)(=O)=O)C2)=O)C(C)C1 C1(CCC(=O)NCC2C(NC(c3n(C)ncc3)=O)CCC2)CCCC(O)C1 C=CCC(C(=O)NC(C1CCN(C(c2c(C(C)=O)c[nH]c2C)=O)C1)C)NC(C)=O N1(C(c2c(C)nn(C3CC3)c2)=O)CCCC(NC(=O)CC2CCOCC2)C(F)C1 CC1COc2c(C(=O)NC3(CCF)CCN(C(c4ccccc4)=O)C3)cccc21 C1(C(C)NC(C2CCCN2S(C)(=O)=O)=O)CCN(C(=O)CCn2ccnn2)C1 Cc1ccc2c(c1)CC(C(=O)NC13CC(C1)N(C(C1CCCO1)=O)C3)S2 C1(CNC(CCCOCC)=O)CCCC(CNC(=O)COCc2ccccc2)C1 C1(C(N2CCC(NC(C3(COC)CC3)=O)C(F)C2)=O)C2CCC(C2)C1(C)C C1(=CCNC(Cn2ccc(C)n2)=O)CCN(C(C2(C#N)CC2C)=O)CC1 N1(CC(C)SC)CCC2CC(C(N3CC(C)NCC3C(C)C)=O)C2C1 CC(C)CC(C(=O)N(C1CCCC1(F)F)C)ONC(=O)CC1CC=CC1 CC1(C)CC(CC(=O)Nc2cccc(CNC(c3ccsc3)=O)c2)CCO1 C1(CNC(c2ccc(CN3CCCC3=O)cc2)=O)C2CC1N(C(=O)CCF)C2 c1ccc(Cl)cc1.CCCSC c1(C(N2C(C)CN(C(C(F)=CC)=O)C(C)C2)=O)cc(C#N)c2n1CCCC2 C12CN(C(C3CC3(F)F)=O)CC1C2.c1(C2(N(C)CC)CNC2)ccc(OC)cc1 CC1(F)CC2(CN(C(=O)CC3(NC(C4CCC5(CCC5)O4)=O)CCC3)C2)C1 C(CC)(CCCC(=O)N1CC(=O)NC(C)(C)C1)NC(C1CCC(=C)CC1)=O C1(CNC(C(P(C)(C)=O)O)=O)CC12CCN(C(c1cc(C(N)=O)cs1)=O)CC2 c1(OC)c(C(=O)NCC2CCN2C(c2cc(C(C)(C)C)n(C)n2)=O)cccc1Cl CC1=C(C(=O)NCc2cc(C(=O)NC(c3ccccn3)CO)on2)SCCO1 c1(OCC)nc(=NC(=O)C2=NOC3(CCC3)C2)[nH]cc1C c1(C(C)C)c(Cl)nc[nH]c1=NCC1(C(C)(F)F)CC1.C(=O)(C(N)=O)N c1(C(=O)NCC2CCC2NC(=O)C(O)CCc2ccccc2)cc(O)nc(O)c1 C1(C)(C(=O)NC(C2CCCC2)CNC(Cc2cc(C)sc2)=O)CCC(=O)C1 c1(C(N2CCCCC2c2ncc[nH]2)=O)sc2ccccc2c1Cl C#CCCCCCC(=O)NC(CC#C)C(=O)N(C)CCC1CCCN1C c1(C(=O)NCCN(C(=O)C(C)OCC(C)C)CC)cnc(C(C)C)nc1 c1(C)cccc(P(C)(C)=O)c1.C12CCC3(C1)CN(C3)N2.C(C=O)=C(C)C c1(C(=O)NCC2(CN(C(=O)CC3(C)CC3)C)CC2)cc[nH]c2nccc1-2 CC(CC(=O)c1ccc(F)cc1)C(=O)N(CC(c1ccccc1)O)C.c1ccccc1 CN1CCC(C#N)(C(=O)NC2CCCCC2CNC(=O)C2=C(Cl)CC2)CC1 c1(C(=O)NCC2CCN(C(c3cnn(C4CC4)c3)=O)C2)cccc(F)c1C(F)F N#CC12C3C4C1C1C2C3C41C(=O)NCCN(C(=O)CSCC(N)=O)C1CC1 N12CCC(F)(CC1)C2.c1(C(=O)NCc2ccn(CC)n2)cnc(OC)cc1C C=CCCC(C)(C)C(=O)N1CCCC(C(=O)Nc2cccc(C(C)C)c2)C1 N1(C(=O)CC2CCN(C(C3CCCC(O)C3)=O)C2)CCc2c(O)cccc2C1 C1(NC(c2ncc(OC)cn2)=O)CCCC2CN(c3cnc(C#N)cn3)CC12 CCC(CC(=O)N(CCC(N1CCCOCC1)=O)C1CC1)c1ccccc1 C(=O)(C1=C(Cl)CCOC1)N(C(C)CNC(C1(COCC)CCCCO1)=O)CC CC1=C(C(=O)NC2(CO)CN(C(=O)C(C)(O)C(C)C)C2)CCC(C)(C)C1 Cc1c(C(=O)NC2COCCN(C(C3CN(C)C(=O)C3)=O)C2)sc2nnc(S)n12 C(c1cnn(C)c1C)=CC(=O)N(CCOCCNC(C(n1ccc(C)n1)C)=O)C N12CC3(CC1CO3)C2=O.O=C1COCCN1CCCNC(=O)C(=O)NCC(F)F C(=O)(C1=C(Cl)CCCC1)NC1COCCN(C(c2c(C)ccc(OCC)c2)=O)C1 C(=O)(C(C)(C)CCF)NCC(C)CC(N1CC2CC2C2CC12)=O S(=O)(=O)(c1cccc(NCc2nc(C(F)F)nn2C)n1)N(CCF)CC C1(C)(CN(C(=O)C(F)(F)F)CCOC)Cc2ccccc2C1 N1(C(c2c(CC)n(C)nc2)=O)CCC2(CC2NC(=O)CCc2cncnc2O)C1 C(=O)(C(C)CCC(C)(C)C)N1CCC(CN(C(=O)CC2=CCCC2)CC)CC1 C1(NC(c2cc(C)oc2C)=O)COCCN(C(c2ccc(F)cc2Cl)=O)C1 c1(CCCCNC2(Cl)CC2(F)F)nc2ccccc2s1.O=C1CN1 n12cc(nn1)NC(=O)C2.C1(C(=O)NCC2(CN(C)C(N)=O)CC2)CC(C(F)(F)F)C1 N1(C(=O)C2=COCCO2)CC23CCCC2(C1)CN(C(c1ccnc(Cl)c1Cl)=O)C3 CC12CCCN(C1)C2=O.C1(C(N2CCCCC2)=O)CCCC1N1CCOCC1 CCCCC(O)C(=O)NC1(CO)CCN(C(=O)CC2COCC(C)(C)O2)CC1 CCCCC(C)CCC(=O)NCC1CCCN1C(=O)C(c1ccccc1)F C1(C(=O)NC2C(NC(C(C)c3cncs3)=O)COCC2)CC(=O)NC(=O)C1 C1(CNC(c2[nH]cc(C)c2)=O)COCCN(C(=O)C(C(C)O)N(C)C)C1 C(=O)(CCCC(C)(C)C)N1CC(C(C)C)C(C(N2CCC(OCC3CC3)C2)=O)C1 C1(C)(C(=O)NC(C)C(=O)NCCCCC2CC2)CC(=O)C1.C(CO)S c1(C(N2C(C(N3CCC(=C)CC3)=O)COCC2)=O)cc(F)ccc1OC C#Cc1cncc(C(=O)NCCc2ccoc2C(=O)N(CC)OCC)c1 S(=O)(=O)(c1cccc(F)c1C)N1CC2CCN(c3nc(OC)c(F)cn3)C2C1 c1(OC)cc(NC2CC3CC2CC3N)cc(OC)c1C N#Cc1ccccc1C(N1CCOC(C2CN(C(c3cnc(Br)o3)=O)C2)C1)=O C(=O)(CC1NC(=O)c2ccccc21)N1C(C)CCN(C(COC)=O)CC1 C1(C(N2CC(N(C(Cc3c(C)scc3)=O)C)C3(C2)CC3)=O)CCn2nccc2C1 c1(C(C(=O)NC(CC)(C)C)N(C)Cc2ccnn2CC2CCC2)ccnn1C C1(CC(=O)NCC(C(=O)NC)O)N(C(=O)CN2CSCC2=O)CCC1(C)C C1(C(N(C)C)=O)(NC(=O)C(F)=CCCF)CCC1 c1(C(F)(F)F)ccccc1N.n1(CC2CCCO2)cc(-c2ccnn2CC(F)F)nn1 N1(C(c2c(C)cc(C)nc2)=O)CCC2(CC1)CC2C(=O)N(CC(C)O)CCO c1(C(C(=O)NC(C)CC)N(CCOCC)C(C)C)cc(C)cc2c1CCC2 C12CN(CC1F)C2=O.Cn1cc(C(=O)C=CC(=O)NC2(CO)CC2)cn1 c1(CC(=O)NCC(C)N(C(C(C(CC)(C)C)O)=O)CC)c[nH]c2cccc(Cl)c12 Cn1ccc(C(=O)NC2(C(=O)NCC3(C)CC=CCC3)CC(CO)C2)cc1=O c1(CC2CC(NCC(c3n(CC)nnn3)C3CC3)C2)cccc(P(C)(C)=O)c1 N1(C(Cc2sc(C)c(C(C)C)n2)=O)CCC(C)(NC(=O)CC(Cl)Cl)CC1 CC(C)(O)CC(=O)NC1CCOC(CNC(c2cn(CC(F)(F)F)cn2)=O)C1 C#CCC(CCOC)NC(=O)NCC1CCCC1NC c1(C(=O)NCC2CC(F)(CNC(C3CC3F)=O)C2)ccc2ccoc2c1 C1(CC(C)NC(CSCC#C)=O)CN(C(=O)C(F)C2CCOC2)C1 CC(=O)CCCC(C)C(=O)NC1CC(CC(N2C3CCC2COC3)=O)C1 CC(CS(C)(=O)=O)N=c1[nH]c(N2CCOc3ncccc3C2)nc2c1CCCC2 C1(NC(C(C(C)O)NC(CN(CCOC)C)=O)=O)CC2CCCC2O1 N1(C(C(C)=CC)=O)CCC2C1CCCN2C(=O)COCCCC(C)C C1(NC(C23OCC(CC)(C2)C3)=O)CCC2CCN(C(=O)CNS(=O)(=O)NC)C12 N1(C(CCc2cnc(C)o2)=O)CC(NC(=O)C(C)Sc2nncn2C)CCC1C C1(C(N(C2CCN(C(C=CCOC)=O)CC2)C)=O)CC(COC)C12CCC2 N1(CC)CCN(C(C2CN(C(C3(OC)CCSC3)=O)CC(C)O2)=O)CC1C Cn1c(C(=O)NCC2CC(C(=O)NCc3cncc(Cl)c3)=NO2)ccc1C#N N1(C(C2CC(=C)C2)=O)CCC(C)C1CNC(c1ccc(C)o1)=O C1(NC(c2cc(F)cc(I)c2)=O)CN(C(c2cnco2)=O)CCC1F C1(COC(CN2CCC(OC)CC2)=O)CCC(=O)N2CCOCC12 c1(C(=O)NCC(N2CCOCC2CCO)=O)ccccc1Br CC1CCN(C(=O)C=Cc2nccs2)CCN1C(=O)C(N1CCCCCC1)C CC1(C)CCCCN(C(=O)NCC23CC(C2)C(c2ccccc2)O3)C1 c1(CC)ccsc1C(=O)NCc1ncoc1CCNC(c1ccc(C(C)C)s1)=O C1(CC#C)(C(=O)NC(c2cccc(C)n2)C)CCN(C(C2CC23CC3)=O)C1 C(N=c1cc(C)nc(N2CC3C(CO)C3C2)[nH]1)c1c(C)ccs1 Cc1cc(CCC(N2CCOCC2CCNC(=O)CCC(C)N(C)C)=O)nn1C c1(C(=O)NC(CCC)CNC(C2C=CCS2)=O)cccn(C)c1=O CCC(C)C(O)C(=O)NCCOC1CCN(C(C2CCC(C)(C)OC2)=O)C1 C=C1CC2(C1)CN(C(C1CCCC(NC(c3ncccc3F)=O)CC1)=O)C2 N1(CC(=O)N(C(c2ccccn2)=O)CC2CCCCC2)CCCc2ccccc21 c1(C(=O)NC2C3CN(C(C(C4CCC(C)CC4)CC)=O)C2C3)nc2ccccc2s1 N1(C(C(CSC)(C)C)=O)CCN(C(c2ccc(CCN(C)C)[nH]2)=O)C(COC)C1 CC(C)C(C)C(CNC(c1cc(C(F)(F)F)ccc1O)=O)NC(=O)CC(F)F C1(NC(C=CC=CC)=O)CS(=O)(=O)C12CCN(C(=O)C(C)CCC)CC2 c1(C(=O)NCCO)sc(C)c(C)c1Br.CCCCOCC(=O)NCCOCC.SCC C(=O)(CCC(C)(C)C#N)N1C(C(N2CCC(N(C(C)=O)C)C2)=O)CSC1 C(CCN=C(NCCS(=O)(=O)C(F)(F)F)NC1CCN(C(C)(C)C)C1)OCC N1(C(C2(OC)CC(CF)C2)=O)CCC(CCCNC(C23CC(O)C2C3)=O)CC1 CC1CC(CNC(=O)Nc2ccc(F)cc2)CN1N1CCCC(C(N)=O)C1 N1(c2c(C)c(NCCc3cnc[nH]3)ncn2)CCC(C2CCCOC2)CC1 c1(C(N(CCNC(C(C)(C)OC)=O)C)=O)cc(C)ncc1Br C1(NC(C(C)(CO)OC)=O)CC2CC1CC2C(=O)NCC1(n2cccn2)CC1 N1(C(c2nccc(Cl)c2F)=O)CCC2CCN(C(=O)C(F)(F)CO)CC2C1 CCC(CC)(CO)C(=O)NC(C)C(C)NC(c1cc(C2CC2)n(C)n1)=O N1(NC)CCCC1(c1ccccc1COC)C.c1(C)ccccc1 C1(C)(CN(C(=O)C=Cc2cocn2)C)CCCC1NC(=O)CN1CCSCC1 c1(C(=O)NCC2CC(NC(CCOCCCOC)=O)C2(C)C)ncc(F)cc1F c1(CC)nc(C)c(C(=O)N(C2C3CN(C(C4OCCC4(C)C)=O)CC23)C)o1 N1(C(c2c(CCC)n[nH]c2)=O)CCC2(CC1)CCN(C(=O)CCC1CC1)CC2C C1(CNC(c2ccc(CC)s2)=O)CCC(C)N(C(C2CCC(O)C2)=O)C1 c1(CNC(=O)NC2CCC(CCCCC)O2)nc(C)c(C)s1 C(CC(C(=O)NCc1cn(CC(N2CCC(O)(CO)C2)=O)nn1)N(C)C)OC C(c1ccccc1)=C(CC)C(=O)NC1CCCC1CNC(=O)Cn1cncc1C c1(OC(CC)C(=O)NC2(O)CN(N3CC(OC)C3)C2)ncc(F)c(OC)n1.C(=O)N Cc1ccccc1C(C)CC(=O)NCC(C)NC(=O)Cn1nnnc1C1CC1 c1(C(=O)NC(C2(O)CN(C(=O)C=Cc3cscn3)C2)C)ccc2nnn(C)c2c1 c1(C(N2C3CC(CN(C(C(C)OCCC#C)=O)C3)C2)=O)c[nH]c2nc(F)ccc12 N1(C(C=CC)=O)CCC(C(=O)NCC(C)(O)C(C)(C)C)(CC)CC1 c1(C(=O)NCC2(O)CCN(C(c3cncc(OC)c3)=O)C2)cc2c(s1)CCSC2 C(=O)(CCCC(F)(F)CO)N1CC(NC(=O)COc2cccc(F)c2)C(CO)C1 N1(C(CNS(C)(=O)=O)=O)CCC(C2(NC(C3CCS3(=O)=O)=O)CC2)CC1 C1(NC(CC2C(C)C2)=O)CN(C(=O)CN2CCC(N(C)C)CC2)CC1(C)C Cn1nc(C(=O)NC2CCC(CNC(C3CC(F)(F)C3)=O)CC2)cc1O Cn1ccc2cnc(N3CC4C(NCc5ccccc5S(N)(=O)=O)C4C3)nc12 C1(CNC(C=C(CC)CC)=O)CCCCC1NC(=O)COC1CC(F)(F)C1 c1(C(=O)NC(C2CCCC2)CNC(C(CCC)OC)=O)cnc2[nH]ccc2c1 C1(CC(=O)NC2(CCCC)CCCC2)OCCC1(C)C.C12(CCCC1)C(=O)NC2 Cn1ncc2c1CC(NCC(=O)Nc1ccc(F)c(F)c1F)CC2 C1(N(CC(C)C)C(=O)CC2CCC(=O)N2)CCN(C(C2CC2(F)F)=O)CC1 C(CCNC(=O)Cc1cccc(OC)c1)(C(C)C)NC(C1(COC)CC=CC1)=O c1(C(=O)NC2CC(CC(=O)NCc3c(CC)n[nH]c3)C2(C)C)cc2occc2[nH]1 C1(N(C(Cc2cc(CC)sc2)=O)CCO)CCCN(C(C2CC(C)=NO2)=O)C1 c1(C(N2CCC(C)N(C(=O)CC3C=CCC3)CC2)=O)cc2ccccc2c(O)n1 C1(CNC(=O)CCOC2CCCC2)CCN(C(C2CCCO2)=O)C1 C(C)(C)(CCC(=O)NC(C1CCN(C(C2CCCN(C)C2)=O)C1)C)OC c1(NC(c2c(C)n(C)nc2)=O)ccc2nc(C3=CCCC3)cn2c1 c1(CC)cc(C(=O)NCC(O)CN(C)C(c2cn(C)nc2C)=O)cc(N)c1 C12(C(=O)NC(CCC)c3ccco3)CC(CN(C(C3CCCC(=O)CC3)=O)C1)C2 C1(CCNC(C2(COCC)CCCO2)=O)CCCCN1C(c1[nH]c(O)nc1C)=O c1(C(N2CC3C(NC(CC(COC)C)=O)(CC3)C2)=O)cccc2c1CCC2 Cc1ccc(CC(C)C(=O)NCC2CCN2C(=O)Cc2ccco2)cc1 N1(C(CC2OCCN(C(C3(C#N)CCOCC3)=O)C2)=O)CCn2nccc2C1 C1(NC(C(C)=CCC)=O)CCC(C(=O)N(CC(=O)NC(C)(C)C)C)C1 c1(CNC(NC2C(C)C2)=NCCc2ccns2)cc2ccc(N(C)C)cc2o1 N1(C(CCc2scc(C)n2)=O)CCC(F)(CNC(c2cc(Cl)cn2C)=O)C1 C=C(C)CCCC(=O)c1noc(-c2ncnc(C)c2C2CC23CCOC3)n1 N1(C(C(COC)NC(C)=O)=O)CCCOC(CNC(=O)CCC(C)CN(C)C)C1 C(=O)(CCC(C)(C)NC(N)=O)NCC(CO)NC(COCC(=C)C)=O C1(NC(c2c(CC)c[nH]n2)=O)CC1C1CCN(C(c2nn[nH]c2Cl)=O)CC1 c1(C(=O)NC2CCN(C(C)=O)C2)coc2c1CN(C(c1ocnc1C1CC1)=O)C2 Cc1ccc(F)c(CNC(=O)C=CC(C)NC(c2occ3c2CCC3)=O)c1 C1(CC)CN(C(=O)C(C)(C)CCSC)CCC1NC(c1c(C2CC2)noc1C)=O N1(C(c2cc(C)no2)=O)CC(NC(=O)CNC(=O)NC2CC2)CC(O)C1 N1(C(c2cc(SC)oc2)=O)CCC(C)C1C(=O)NCC#CC1CC1 CC12CCOC(CNC(=O)CC3(NC(c4ncnc(O)c4F)=O)CC3)(C1)C2 c1(C(N2C(CCNC(c3c(C#N)scc3)=O)CCCC2)=O)cc2n(n1)CC(F)C2 N1(C(c2c(C)csc2)=O)CC(C(=O)NC2(C(N)=O)CC(O)C2)C(C2CC2)C1 CCC(C)(CC)C(=O)N1CC(CNC(c2cncs2)=O)OC(C(F)(F)F)C1 C1(C(CNC(C(C)OCC)=O)(C)C)CCN(C(=O)C(C)CC2CC2)CC1 N1(C(C=CCC)=O)CC(O)CC1(C)C(=O)NOCC1CC1 C(=O)(C1CC(C)(C(=O)O)c2ccccc21)OC.c12cc(ccc1[N+](=O)[O-])NC2=O CC(C)C(CNC(c1ccnn1CC(F)F)=O)NC(=O)CN(C)CCO C1(C(=O)NCCNC(COC)=O)(NC(c2ccccc2CF)=O)CCN(C)C1 C1(C(=O)NCC2C(NC(C3CCC(C)(CC)O3)=O)CCCC2)CN2CCN1CC2 N1(C(C(CC)C#N)=O)CC(C)CN(C(c2ccc(C3CCC3)cc2)=O)C(C)C1 c1(CC(=O)NC23C(CN(C(c4cccc(OC)c4)=O)C2)C3)cc(Br)ccc1C C12(CNC(C(c3c(OC)cccc3)(C)C)=O)CCCN(CC1)C2 CCCC(C)(O)C(=O)NC1CCN(C(c2cn(C)nc2I)=O)C1 Cc1c(C(=O)NCC(O)CN(C(=O)C(C)(F)C(F)(F)F)C)sc2[nH]cnc(=O)c12 C(=O)(C1=NOC(C2(O)COC2)C1)NCCCCCN(C(=O)COCC(F)F)C C1(C(N2CCC(C)(NC(c3cc(Cl)c(Cl)s3)=O)C2)=O)CC(S(C)(=O)=O)C1 N1(C(C(C(CC)CC)C)=O)CCC2(CC1)OC1(CO)CC2(NC(=O)C(C)CF)C1 C(=O)(C#CC1CCOCC1)N1CCC(C(N2CC(C)=C(C)C2)=O)C(C)C1 C1(NC(COCCOC)=O)CCN(C(=O)CC2CCOC(C)(C)C2)CC1F N1(CC(=O)NCCC(CNC(=O)C(=CC2CCCC2)C)OC)CCC(C)(C)C1 N1(C(C2(OCC)CC2)=O)CCC(NC(=O)NC2COCC2F)C1 c1(CN(c2cccc(Cl)c2)C(COc2c(C(C)O)cccc2)=O)cccc(Cl)c1F C(CC(C)(C)C(=O)NCC1(C)CCC(NC(C2(C(F)(F)F)CCCC2)=O)C1)OC c1(C(=O)NC2C(C(N(CCOC)C)=O)CCOC2)ccc(O)nc1C c1(C(=O)NCC(CC)N(C(=O)Cc2ccc(O)cn2)C)ccc(C)c(Cl)c1 C1(CCOC)(NC(=O)CC(F)(F)F)CCN(C(C2(C)CC(C)=NO2)=O)C1 C1(NC(C2CCN(C)C2)=O)CN(C(=O)CCC(C)(C)N(C)C)CC12CCC2 n1(CCC(=O)NCC=CCNC(=O)CC2(O)CCCCC2)nc(O)c2c1CCCC2 C(C(C)C(F)C(=O)N1CC(CN=[N+]=[N-])C1)NC(C1(CC#C)CCC1)=O C(=O)(C(C)(C)C(C)NC(=O)C(C)SC(F)(F)F)NCc1c(C)nc(C)[nH]1 c1(C(=O)NCC2C3CN(C(c4on(C)c(=O)c4)=O)CC32)ccc(Cl)nc1N C1(c2c(C)ncs2)CCCN(c2nnnn2CCCC(=O)Nc2nc(O)n[nH]2)C1 N1(C(C(C)C(C)(F)F)=O)CCC(NC(c2cncnc2)=O)C(F)(F)CC1 c1(CN2CCC(NC(c3cccc(Cl)c3F)=O)CC2)cc(F)cc(Br)c1F C1(C(=O)NC(C2CCN(C(C3(O)COC3)=O)C2)C)CCc2nnc(O)cc2C1 C=CCCC(F)(F)C(=O)NC(C)C(C)C(=O)NC1CC2CC2C1 Cc1cccc2cc(C(=O)NCCNC(c3c(Br)noc3C3CC3)=O)nn12 C#CCC(C)(C)C(=O)N1CCC(NC(=O)CCCCCc2cccs2)C(F)C1 c1(C(N2CCC(CCC(=O)N(CCC(C)C)C)C2)=O)ccc(CO)nc1 N1(C(C2C(CC)C2)=O)CCC2(NC(C3CCCC(C)CC3)=O)CCCCCC12 C(c1ccc(C(N)=O)o1)=CC(N1CC(O)(CN(C)C(C2COC(=O)O2)=O)C1)=O c1(C(=O)NCC(C)NC(C(C2CCOC2)OC)=O)c(N)cccc1[N+](=O)[O-] c1(N(C)C)nc2c(c(=NCc3n[nH]cc3CCCc3nncs3)[nH]1)CCCC2 C(C(=O)N1CCN(C(c2c[nH]ccc2=N)=O)CC1C)(C(C)(C)C)n1ncc(C)c1 C(CC(C(=O)NCC1CC(C)=NO1)NC(c1nncs1)=O)=CC C(CCCCCC(=O)N(CC(O)CNC(C1(CCCF)CC1)=O)C)SC C(=O)(C(C)(F)C(F)(F)F)N1CC(CCCC)N(C(c2ccc(COC)o2)=O)CC1 CCC(O)C(=O)NCC1(C)CC(N(C(c2ccccc2)C(=O)NC)CC)C1 C1(CC(=O)NCCCN(C(C2N(C(C)N(C)C)CC2)=O)C(C)C)CC(C)(C)CO1 C1(C(N2C(C=C)CCC2)=O)CCN(C(=O)c2cc(SC)nn2C)O1 C(C(C(=O)N(CCOC(C)=O)CC)C(C)C)NC(c1cnc(OC)s1)=O c1(C(N(C)CC2CN(C(c3cnc(O)o3)=O)CCO2)=O)[nH]cc2c1CCS2(=O)=O c1(COC)nccc(=NC2CS(=O)(=O)CC2NC(c2ccc(O)nc2)=O)[nH]1 CCC1C(=O)NCC2(CCCC2)C(=O)NCC2(C(C)C(=O)N1)CC2.CC C#CC1(F)CN(C(C2(C3CCCCN3C(C3CC3=C)=O)CC2)=O)C1 CC1CCCN(C(=O)CCn2ccnn2)C1CNC(=O)CCC(=O)N(C)C C(C(COC)C(=O)N1CC(N2CCN(C(c3snc(Cl)c3Cl)=O)CC2)C1)OC Cc1nc(F)ccc1CNC(C1(CCC(=O)N(C)C)CCCC1)=O c1(NCC(=O)NC)cnnc(O)c1Cl.c12ccc(cc1)NC(=O)C(C)OC(=O)C2 C(=O)(C(O)CCC(C)C)NC(C(=O)NC1C(C(=O)OC)COC1)C(C)(C)C C1(C(F)(F)F)(COC(C(CC)F)=O)CCOCC1 C1(CNC(C=CSC)=O)CN(C(=O)CC2(C)CC2(Cl)Cl)CCO1 C1(C2CCCC2)(NC(CC2CC(C)N(C(c3ncn(C)n3)=O)C2)=O)CCC1 C1(NC(c2cc(Cl)c[nH]2)=O)CC2(C1)CC(NC(C1CC(n3ccnn3)C1)=O)C2 c1(C(=O)NC2(CCOC)CCN(C(C3(C)CCCO3)=O)C2)sc(C)c(C)c1C c1(OC)cccc(CC(=O)NC(C)CC(C)NC(C2CCC(C)C2)=O)c1 C(=O)(C1=Cc2ccccc2OC1)NCC1(CNC(c2c[nH]c(=NC)s2)=O)CCCC1 c1(C(=O)NC2CCCNC2=O)cccc2ccnn12.c12ccc(cc1)C(=O)NC2C C1(NC(c2nc(C)nn2C)=O)CN(C(c2cccnc2F)=O)CC12CCOCC2 N1(C(C(CCCC)O)=O)CCC2C1CCCN2C(=O)Cn1ncc2cccnc12 CC(C)(C#N)CCC(=O)NC1(C2CC2)CCN(C(=O)Cn2cnnn2)C1 c1(C(=O)NC(CC)CNC(c2ccc(CCN(C)C)cc2)=O)ccc(C#N)cc1 Cc1ccc2[nH]nc(C(N3CC4(F)CCC3(C(=O)OCC(C)(C)C)C4)=O)c2c1 N1(C(CC)=O)CCOCC1CN(C(=O)C(C)(C)C1(O)CCOC1)C1CC1 CC1CN(C(=O)CC(c2cc(Br)ccc2F)=O)CC(C)C1NC(c1cc[nH]n1)=O CCS(=O)CC(=O)NC1(CNCc2ccc(C(F)(F)F)cn2)COC1 C(=O)(CC(C)C(F)F)N(C1CC(C(=O)NC(C)CN2CCOCC2)C1)C1CC1 c1(C(=O)NCC2CCN2C(c2sccc2SC(F)F)=O)ccn2ccnc2c1 c1(C(N(C)CC2(NC(C34CCC3CC4)=O)CC2)=O)nccc2[nH]ccc12 C1(CC(=O)NCCC2CCCN2C(C2(CF)CC2)=O)CN2CCN1CC2 S(=O)(=O)(c1cc(C)cnc1N1CC(CO)C2(CC2)C1)NC(CCC)C C1(COCC)(CNC(=O)C=Cc2ccc(NC)cc2)CCN(c2nnco2)CC1 CC1(C)CCCC(CN2CC(NC3CC3)C2)O1 c1(C(N2CCC(C(=O)NCc3c(CC)cc(F)cc3)CC2)=O)cc(F)c(Br)cc1Cl c1(C(=O)OCc2cc[nH]c2)ccnc(N2CCCCCC2)c1 CC(CN(C)C)CCC(=O)N(C)CC1CN(C(=O)Cc2c[nH]ccc2=O)CCO1 c1(CC(N2C(N(C(CCOCC#C)=O)C)CCCC2)=O)cccc(C#C)c1 C(=O)(C1=CC2CC(C1)CC2O)N(CC(c1ccc(Cl)c(Cl)c1)=O)C1CC1 C(N=c1[nH]cnc2[nH]ccc12)C1N(C(CNC(C)CCCOC)=O)CCC1 c1(C(=O)OC)nc(NCC(=O)Nc2cccc(SC)n2)ncc1Br C1(NC(CCCCSC)=O)CC12CCN(C(=O)CC(C)(C)F)C2 c1(C(=O)OC)cccc2c1N(C(c1ccc(Cl)cc1)c1nn[nH]n1)CCC2 c1(C2(O)CC(C(N(CCC)CCNC(=O)C(=O)N(C)C)=O)C2)cccc(Cl)c1 c1(C(CNC(c2ncoc2Cl)=O)O)cc2ccccc2o1 N1(C(C2(C(=O)OC)CCOC2)=O)CC2(CCN2C)C1.C12(CC=CC1)C(=O)NC2 S(=O)(=O)(c1ccc(NCCC(O)C2CCC2)nc1)NC(C=C)(C)CC c1(C(N2CC(CNC(CCSCCCC)=O)(OC)C2)=O)cc2n(n1)CC(F)C2 CCC(C)(C)C(=O)C(=O)N1CCCCCC1C(=O)N(C)CC1CCCC2CC12 N1(C(c2cccc(-c3cc[nH]n3)c2)=O)CCC2CC1CN(C(C1(Cl)CC1)=O)C2 C(C)(CCCNC(=O)C(O)Cc1[nH]cnc1C)NC(CCOCCCOCC)=O N1(C(CCn2c(C)ncc2)=O)CC2CC1CN2C(C12CCC1CC2)=O Cc1ccn(C(C)C(N2CCC(C(=O)NC(c3scnc3C)C)C2)=O)n1 C1(CCC)CN(C(=O)CCc2cnoc2)CCN1C(=O)Cc1ccccc1Br C1(CNC(C(C)CC(F)F)=O)CN(C(=O)CCC(C)(C)F)C2(CCC2)C1 N#Cc1ccc(Cl)c(C(=O)NC(Cc2cn(-c3ccccn3)nn2)C(=O)O)c1 Cc1ccc(C(=O)NC(C)CN(C)C(C2CC(C3OCCO3)C2)=O)c(N)c1 N1(C(C(C=C)(C)O)=O)CCC2(CC1)CC2CNC(c1conc1C1CCC1)=O O(NC(=O)CCc1ccc(Cl)s1)CC(=O)NCC(=O)NCC1CC12CC2(F)F C1(NC(C=Cc2scc(C)n2)=O)C2CC1CN(C(=O)Cn1cc(C3CC3)nn1)C2 C1(CNC(c2c(C(C)C)n(C)nc2)=O)CC2(CCC2)CN1C(C1COCCO1)=O c1(CC)cccc(CC)c1CC(=O)NC1(NC(=O)CC2(C)CCC2)CCOCC1 C(C(=O)N1CCC(F)(C(N)=O)C1)(C(C)O)NC(c1cc(OCC)n[nH]1)=O C=C(C)CCC(=O)NC1(CO)CN(C(C2CC3CC2CO3)=O)C1 C1(CCNC=O)CCC(NC(=O)Cc2ncsc2NC)C1.C(F)(CC=O)=CC C1(F)(CNC(c2ccc(C)o2)=O)COCCN(C(c2ccc(CO)c(F)c2)=O)C1 C1(NC(CNS(CCC)(=O)=O)=O)CC2CC(NC(=O)CC3CC3(Cl)Cl)CC12 C1(C(=O)NCC2N(C(c3c(N)cncc3)=O)C3C(C2)C3)CCC2(CCOCC2)C1 C1(C(N2C(C3(O)CN(C(=O)CC4CC(CF)C4)C3)CCC2)=O)CC12CCOCC2 c1(NC(C(C2CN(C(C)=O)C2)N(C2CCC2C)C)=O)c[nH]nc1C c1(CC(=O)NC2C(NC(C(CC#C)C)=O)C2)cc(F)cc(Br)c1 C1(C(=O)N(C)CC2(O)CN(C(c3cc(Cl)ncc3N)=O)C2)(OC)CCCC(C)C1 CCC(C)C(C)C(=O)NC(C)CCCNC(c1cnnc(Cl)c1)=O CC(=O)CCCC(=O)NC1CCN(C(c2ccc(Cl)cc2OC(F)(F)F)=O)CC1C C12(CCCC1)C(=O)OCC1(F)CN(C1)C2=O.C(=O)(CCC)N.C(=O)(C1CC1)N C1(CC)CC(C(=O)NC2CC(N(C(=O)CC=CC(C)(C)C)C)C2)C1 CC(CCCC(=O)NCc1cn(C2CC2)nn1)NC(=O)CN(C1CCOC1)C c1(NC(CC#C)=O)ncc(-c2ccc(-c3ccn(C)n3)s2)cc1C C1(NC(C(CC)C(F)(F)F)=O)CCC12CCN(C(C1CN(S(C)(=O)=O)C1)=O)CC2 C1(CCNC(CCC=C)=O)CCCN(C(=O)C(OC(C)=O)OC)C1 C1(F)(C(=O)NCC2C(CC(=O)NC(CCSC)CO)C2)CC=CCC1 C(=O)(CCCCCN=[N+]=[N-])NCCC(C(=O)NC(C#C)C(C)OC)O N1(C(c2n(C=C)nnc2)=O)CCC(NC(C2CC23CC(O)C3)=O)C(F)(F)CC1 N1(C(c2c(C)cns2)=O)CC(O)CC1(C)C(=O)NCCC(F)(F)CO c1(C(C(=O)NCC)N(CCC#N)C2CC2)ccc(=O)n(CC(F)(F)F)n1 c1(C(F)C(F)(F)F)ccc(CNC2CCCCC2N2CCCC2)cc1 O=S(=O)(c1ccc(NCc2cc(Br)cs2)nc1)NC1CCC=CCC1 c1(C(=O)NC(c2cn(CC)nn2)C)ccc(-c2cnco2)cc1 c1(C(N(CC(CC)NC(=O)CC(C)c2ccco2)C)=O)ccc2snnc2c1 C1(CN(CC(F)F)C)COCCN1C(c1cc(NC(=O)OC(C)(C)C)ccn1)=O C(=O)(CCS(N)(=O)=O)N(C1CCN(C2CCN(C(C3CCOCC3)=O)C2)CC1)C C1(NC(=O)C=Cc2ncco2)CC2(CCN(C(c3cc(CO)ccn3)=O)C2)C1 C(C)(C)(CCC(=O)N1CCC=CC1C(=O)OC)OC.c12nc(co1)C(=O)NC2 c1(OCC)ccc(C)nc1C(N1CC2CC1CC2NC(=O)CC(C(C)C)OC)=O c1(C(N2CCN(C3CCC3)CC2)C(=O)NC(C(=O)OC)C)ccc(Cl)c(C)c1Cl C1(C(=O)NC2CC3(C(NC(c4c(CC)n(CC)nc4)=O)C3)C2)CN2CCN1CC2 N#CC1CC2(CNC(=O)Cn3cc(C4CCCOC4)nn3)CC1C2 C1(C(N(CCOCCN(C(=O)C(F)CC2CCC2)C)C)=O)CC2COCC2C1 C(=O)(C1CSc2ccccc21)NCCC1=CCN(C(C2CN(C(C)=O)C2)=O)CC1 C1(N(C(=O)C=CC(F)(F)F)CC#C)CCN(C(=O)C(C)C2CCCO2)CC1 N1(C(c2c(C)oc(Cl)n2)=O)CC2CN(C(C3CC(F)(CO)C3)=O)CC2C(F)(F)C1 N1(C(C(CCC)CC(C)C)=O)CCC2(CCCN2C(=O)Cc2ccc(C)o2)C1 N1(C(C(n2cc(C)nc2)(C)C)=O)CCSCC1CCNC(c1ncccc1N)=O C(=O)(C1Cc2ccccc21)N1CC(NC(CC2C(C)(C)C2)=O)C1 C(c1nc2ccccc2o1)=CC(=O)N(CCNC(c1c(C)cnnc1O)=O)CC C1(CC(CC)NC(=O)NC2CC2F)(C(F)(F)F)Cc2ccccc2C1 C(=O)(C1CCc2nccn21)N1CC(NC(c2c(CCC)nco2)=O)CC12CCC2 C1(NC(c2c(OCC)cncc2)=O)CC2CN(C(c3ccc[n+]([O-])c3)=O)CC2C1 C1(NC(c2ccc(C)n2C)=O)CC2CC(C1)N(C(=O)CC1CC3CC3C1)C2 C1(NC(c2cn(C)c(=O)n2C)=O)CC12CCN(C(=O)C#CC1CCOC1)CC2 c1(C(=O)NC2COCCN(C(C(C)(F)F)=O)C2)occ2c1CCCC2 N1(C(C(=O)NC(C)C)=O)CC(NC(=O)Cn2ccoc2=N)CC(C)(C)C1 c1(-c2ncc(C(=O)NC(C)Cc3ccsc3)s2)ccccc1F N1(C(c2[nH]cc(CC)c2)=O)CCN(CCCNc2ccccc2Cl)CC1 CCC(CC(=O)NC1CC(CNC(=O)C(COC)C(F)(F)F)C(O)C1)C(F)F C1(C(N2C(C)CN(C(=O)C(F)=CCCF)CC2)=O)(C(F)F)Cc2ccccc2C1 n1(CC)ccnc1CN(C)CC1CN(C(=O)C(C)Oc2ccccn2)C1 CC(C)C(C)CN=c1[nH]ccc2cc(Oc3ccc(Cl)cc3)ccc12 c1(C(=O)NCCCCN(C(CCOCC(C)C)=O)C)cc2c(s1)CCS(=O)(=O)C2 N1(C(C2(C)CC=CCO2)=O)CC2CCCC2(CNC(=O)Cn2cncn2)C1 CCC(CC(=O)NCCCCCNC(=O)CC1CC=CCN1C)OC N1(C(C2N(C(C=CCCC)=O)CCC2O)=O)CCS(=O)C(C)C1 C12CCN(CCO1)C(=O)COC1CC(C1)NC2=O.C1(CC)CC=CCC1 CN1CCOC(C(=O)NCC2(F)CCCN(C(c3cc(N)c(F)cn3)=O)C2)C1=O c1(CSCC)cccc(C(=O)N(CCNC(=O)C(C)CO)C2CC2)c1 CC(CC(=O)NCSC1CCCN1CC(=O)Nc1cnns1)n1cccc1 Cc1nc(CC(=O)NC2CC(NC(c3ocnc3-c3ccccc3)=O)C2)c(C)s1 C=C(C)CC(C(=O)NCc1cn[nH]c1)NC(=O)C(C(C)C)SC n1(CO)cccc(C)c1=O.C(CC(C(=O)NC1CCC(CN)CC1)NC=O)SC C(C(C)(C(=O)NCCOC1CN(C(C2CCN(C)C2=O)=O)C1)OC)OC Cc1nc2c(o1)CCN(C(C1CCCCCN1C(C1CC(C(C)C)C1)=O)=O)C2 N1(C(C2C(C)(C)C2)=O)CCC(O)(CCNC(=O)C2=CCCCC2)CC1 C12(C(=O)Nc3c(C)c(F)ccc3)CC(C)(C1)OC21CCNCC1 C(=O)(C1=CCC(C)(C)CC1)NC(C(CO)NC(c1c(COC)cc[nH]1)=O)C c1(OC)ccc(N)c(C(=O)NCCC(C)NC(=O)CCOC2CCCOC2)c1 CCC(N=c1[nH]c(N2CCN(Cc3cnccn3)CC2)nc2cc[nH]c12)C1CC1 c1(C(=O)NC2C(NC(=O)CCOCC(F)F)CCC2)cn2c(n1)CCCC2 Cc1ccc(C(N2CCCCC2CNC(c2cnnn2C)=O)=O)c2cccnc12 C1(C(=O)NCC2(C(N)=O)CC2)CCCC(NC(c2cn(CN)nn2)=O)C1 c1(C(C)NC(=O)CCC2(NC(=O)C(N3CCOC3=O)C)CCC2)cccc(CO)c1 C1(C)(CCC)C(=O)NCCN1CC(=O)N(c1ccc(F)cc1)C(C1CCCC1C)=O c1(C(N2CC(NC(CC=C)=O)C(C)CC2)=O)ccc2nc(O)n(C)c2c1 C1(C)(CCNCCC(CCC)C2(c3nnnn3C)CC2)C2CC3CC(C2)CC1C3 CCCCC(CC)n1nc(-c2cscn2)nc1CN(C)C(=O)NCCO c1(CC(N2CC(F)(CNC(c3nc(OC)oc3)=O)C2)=O)cccc(C)c1Cl C1(NC(c2c(CCC)n(C)nc2)=O)CCCCN(C(=O)Cc2ccnnc2O)C1 C1(CNC(=O)CCNC(c2ccoc2)=O)CC2CCC1N2C(c1ccc(F)o1)=O c1(C(C)NC(C2N(C(C)C)C(C)(C)OC2)=O)cc(Br)cc2c1OCC2 C(=O)(C1=CCC(C)CC1)NCC(C)CNC(c1ccc(-n2nnnc2O)cc1)=O C1(CNC(c2ccc(C)o2)=O)(CO)CCN(C(=O)C=Cc2ccncc2)C1 c1(C(N2CC(CCn3cc(CC)nn3)C2)=O)c(N)c(C(F)(F)F)nn1C(C)(C)C N1(C(COCCCCC)=O)CC2CC2(CNC(c2cc(C(C)(C)C)c[nH]2)=O)C1 C1(C(C(=O)NCCN(CCCc2ncc(Br)cn2)C)(C)C)CCCN(C(=O)N(C)C)C1 Nc1ccc([N+](=O)[O-])cc1C(N1CCOCC1CNC(C1COCCO1)=O)=O c1(C2C(=O)N2N(CCCC(F)(F)F)C(C)(C)CC)noc2c1CCC2.C1(C2CC2)CC1.CC CC1CCC(C)N1C(=O)CNC1CC(C[Si](C)(C)C)C1 O=C(C1c2ccccc2CN1Cc1ccco1)Nc1ccc2ncnn2c1 c1(C(=O)NCCCCNC(c2ccn(C)c(=O)c2)=O)c(F)cc(F)c(F)c1F N1(C(c2nc(F)ccc2Cl)=O)CCCC2C1CCCN2C(=O)CCc1ccsc1 N1(c2cc(OCC)ncn2)CCC(c2ccccc2)C(C)C1.c1(N)cnc(Cl)cc1C c1(SCC(C)(c2nn[nH]n2)NC2CC2)cccc(C(F)(F)F)c1 C1(NC(=O)Cc2cc[nH]n2)CC2(C1)CC(NC(c1sccc1Br)=O)C2 C1(CN(C(C=C(C)C)=O)C)CCCCN1C(=O)CC(C)c1ccncc1 N1(C(c2nccc(C)c2)=O)Cc2ccc(C(=O)Nc3cc(Cl)cnc3C)cc2C1 C1(=O)CCCO1.C(=O)(CCCn1cc(C)cn1)N(C(C)=O)C(C)C CC1CC=C(C(=O)N(C(C)(C)CC(N2CC(=O)NCC2C(N)=O)=O)C)CC1 N1(C(C(CC)(C)C)=O)CCOC2(CCN(C(c3cccn3C3CCCC3)=O)C2)C1 C1(C)(C(=O)NC(C)CN(C)C(C2(F)CCOC2)=O)CC(c2ccccc2)=NO1 CC(CCCC(=O)NCC1CCCCCCC1)NC(c1cnn(C)c1)=O c1(C(=O)NC(CNC(C2(c3cc[nH]n3)CC2)=O)CO)cc2ncccc2[nH]1 c1(C(=O)NCC2(O)CC(Nc3cnc(F)cn3)C2)cc(Cl)ncc1F Cn1cc(Cl)c(C(=O)NC2CC3C(NC(C4CCCC4(C)C)=O)C3C2)n1 c1(C(=O)NC2CC(NC(C3=CCCC3C)=O)C(O)C2)cc2ccccn2n1 c1(C(=O)NC2CCCCN(C(c3n(CC)nc(C)c3)=O)C2)ccc(F)cc1C#N N12CC(CC(F)C1)OC(OCC)C2=O.C1(=C(C(=O)NC)F)CCCCC1 c1(N)cncc(Cl)n1.C(CCC(=O)N1CCC(CNCC)C1)OCCC N1(C(c2ncc(C)cc2C)=O)CC(NC(C2CC3CCC3C2)=O)C2CCCC2C1 C(=O)(CC(C)C(F)(F)F)NCCCC(C)NC(c1snc(Cl)c1Cl)=O C1(NC(c2c(Cl)cc(C)nc2)=O)CC2CCC(C1)C2NC(c1ncccc1F)=O c1(O)cn2cc(Cl)cc(Cl)c2n1.C1(OCC)CC(CN)CCN1C(=O)OC(C)(C)C C1(N(C(C(=O)NC)C2CCSC2)C2CCCC2)CCN(C)CC1 N1(C(CSCC(=O)OC)=O)CCn2c(CNC(=O)C(F)n3cccn3)nnc2C1 C(CCC(CCC)NC(=O)CCC(=O)N1CCOCC1)NC(C(C#C)(C)C)=O N1(CC(=O)NC2CCC(NC(C(C)(C)C)=O)C2)CCCS1(=O)=O N1(C(=O)CCC2CC2(F)F)CCC2CCN(c3cc(F)ncn3)CC2C1 c1(-c2cn(CC(N3CCOC4CC34)=O)nn2)cccc2[nH]ccc12 C1(C(=O)NCCSCC=C)CN(C)CCN1C(=O)CC(C)(O)C=C C12(CNC(C(CCOC)C)=O)CC(NC(=O)CC(C)C(C)C)(C1)C(C)O2 N1(C(C(C(=O)OC)OC)=O)CC2(CCCC2)C1C(=O)N(C)Cc1ccns1 c1(OC)cccc2[nH]cc(CC(N3CC(NC(C4(F)CC4)=O)CC3C)=O)c12 C(c1cccc(O)c1)=CC(N1CCC(NC(c2c(CC)nc(C)o2)=O)C1)=O c1(C(=O)NC(C(=O)NCC2(CF)CCC2)CC(F)F)cncc2[nH]ccc12 C1(N(C(C2(C)C=CCC2)=O)Cc2ccc(Br)cc2)CCCC2OCCC12 C1(C(N)=O)CN(C(=O)C(=O)NCCC2(C)CCCO2)c2ccccc2O1 O=C1CC(C(=O)NCc2ccc(C(=O)N(C3CC3)CC3CCOC3)nc2)=NN1 c1(OC)cccc(C(=O)NC2CC(C(N3CC4CC3CO4)=O)C2)c1F c1(C(=O)N(CC(=O)OCc2ccco2)C2CC2)cccc(-n2cncn2)n1 c1(C(N(C2CCN(C(C3CCSC(C)C3)=O)C2)CCC)=O)coc(C#N)c1 c1(NC(C(C2CC(NC(C3CCC(C)(O)CC3)=O)C2)F)=O)cccc2[nH]ccc12 N1(C(c2n(CC#C)ccn2)=O)CCCC(C2CCCN(C(=O)C(F)OC)C2)C1 Cc1ccc(-c2cnc(NCC3CC4CCC3O4)c(O)c2)c(C)n1 C(=O)(C(O)CC[S+](C)C)N(CCC)CCNC(c1cc(OC(F)F)ccc1O)=O c1(CCC(=O)NCC2C(NC(CC3(OC)CC3)=O)C2)nc(C)c(C)[nH]1 c1(C(=O)NC2(C)CC(NC(C3(CCC)CCNC3=O)=O)C2)ccc(C#N)cc1C C(=O)(C(C)(C)C(F)(F)F)NC1C2(CC(NC(C3C(CN(C)C)C3)=O)C2)C1 C1(NC(CSCCC)=O)CN(C(c2cc(OC)cc(Cl)c2F)=O)CC12CCC2 c1(C(=O)NC(CCOC)CNC(c2cccnc2)=O)c(C)cc(Cl)cc1[N+](=O)[O-] C1(C(=O)NCc2c(C(=O)NCC3(O)CCC(C)C3)occ2)C2C3CCC(C3)C12 C(=O)(C1=CC2CCC(C1)C2)NCC(C(=O)NC(C(C)C)CN(C)C)CC1CCCC1 C(C)(CC)(CC)CCN1CCCC1.c1(C(C(=O)NC)N(C)CC)ncoc1C C1(NC(CCC=C)=O)CN(C(c2ccc(S(N)(=O)=O)nc2)=O)C2(CCOC2)C1 C1(NC(Cc2cccc(OC)n2)=O)CC12CCC(NC(=O)CCC(C)SC)CC2 N=c1cc(C(=O)NC2CCC(NC(=O)Cn3cccn3)CC2)c(Br)c[nH]1 C1(NC(CN(CCOC)C)=O)CC12CCN(C(c1csc(C(C)C)n1)=O)CC2 c1(C(=O)NCC(=O)N(CCNC(C(CC)N2CCCC2=O)=O)C)ccccc1C N(C1CCCc2c1cnn2CCO)C(c1nc(C(C)(C)C)[nH]n1)=O c1(OC)cc(C(=O)NC(CNC(=O)C(C)SC)CC(F)(F)F)ccc1Cl C1(N(C(=O)CN2CCSCC2)C)CN(C(c2cccc(F)c2N)=O)CCC1O c1(CCC)ncoc1C(=O)NC(C)(C)CCNC(=O)C(F)OC(F)(F)F C1(CC)CCCC(NC(=O)C(CCNC(=O)Cc2ccnc(OC)c2)OC)C1 C1(NC(C2CCC(O)CC2)=O)CN(C(c2cnc(C(F)F)nc2)=O)CC2(CCC2)C1 C(=O)(C(C)CN(C)N1CCOC2(CCCN(c3cccc(C)c3)C2)C1)OC C1(O)(CNC(c2ccsc2)=O)CCCN(C(C2CCCOC2c2cc[nH]n2)=O)C1 C1(CNC(C(CC)F)=O)CC2(CCOCC2)CN1C(c1ccnc(C(N)=O)c1)=O N1(C(C(CCC)C)=O)CCN(C(c2ccc(Cl)cc2NC(C)C)=O)CC1C Cc1cccc(O)c1C(=O)NC1CC1CNC(c1cc(C)n(C2CC2)n1)=O N12CC(C(O)C1)CC1(CC1)C2=O.c1(CC(=O)N)ccsc1.C1(OCC)CC=CC1 c1(C(=O)NCC(CC)NC(C2CCCN2C(C)C)=O)cc(OC)cc(OC)c1 c1(C(=O)OC)cc(C(=O)NCCNC(=O)COCC2CCOC2)c[nH]1 C1(CNC(C(COC)O)=O)CC12CCN(C(c1cc(Cl)c(Cl)n1C)=O)CC2 N1(C(C2CN(C(C(CCC)C#N)=O)C(C)(C)C2)=O)CCC2OCCC2C1 c1(C(=O)NCC2C(CNC(c3nc(C)nc(O)c3)=O)C2)nc2nccc(C)n2n1 CC1(C)CCC(CC(=O)NCC(C(C)(C)C)NC(=O)C2=COCC2)C1 c1(OC)cc(OC)c(C(=O)N(CC(=O)O)C2CC2)cc1OC C12(CNc3ccc(C=C)cc3)CCCC1N(c1cc(C(=O)NC)nc(C)n1)CC2 C1(O)(CNC(=O)CCc2nc[nH]n2)CCN(C(=O)Cc2c(Cl)cccc2Cl)CC1 C(=O)(C(COC)CC(C)C)NCC(=C)CCNC(c1occc1COC)=O C1(N(C(C(CCC)OC)=O)C)CCC2CN(C(c3cc([N+](=O)[O-])c(C)s3)=O)CC12 N1(C(C2(CCN(C)C)CC2)=O)CC2CCC1C1CN(c3nnco3)CC21 CCC1=NOC(C(=O)NCc2cccc(NC(c3snnc3C3CCC3)=O)c2)C1 C=CC1(C(=O)NCC2CC(NC(=O)CSCC(N3CCCCC3)=O)C2)CCCCC1 c1(C(=O)NCCC(C)N(C)C(c2ccns2)=O)csc(-c2ncc[nH]2)n1 N1(C(C2(OC)CCN(C(C3CC4CCC3O4)=O)CC2)=O)CCCC2CC1C2(C)C C(C1=NOC2CN(C(c3c[nH]nc3C(=O)NC)=O)CC12)NC(CCC(=C)Cl)=O c1(NCCC(C)(OC)OC)nc2c(s1)CCCCCC2 N1(Cc2cccc(NC(C)=O)n2)CC(C(N2CC3CNC(=O)C3C2)=O)CC(F)C1 Brc1c[nH]nc1CSc1nnnn1-c1ccccc1.C12CCCN1C(=O)COCC2 C12CCCN1C(=O)CCS2.C(=O)(C(C)c1ccsn1)N(CCNC(N)=O)CC C1(C(=O)NCCC2C(C)CN(C(=O)CCCCC3CC3)C2)CCOCC12CCC2 C1(C(N(CCOC)CCNC(=O)C=CC(=O)N(C)C)=O)COC(C)C1 C1(C(=O)NC2CC(C(N)=O)C2)CC2C=CC1C2.c12cccc(c1)NC(=O)C2 O=C(C(O)C(F)F)NC1(O)CN(C(=O)C(F)(F)Cc2ccc(F)cc2)C1.CC(C)=CC C(C(CC(C)C)NC(=O)Cc1cnc(C(F)(F)F)s1)NC(C(C)(C)OC(C)C)=O C(CCC(C)(C)C(=O)N(C)Cc1nccn1C)NC(CC(CC)CC)=O C1(C(=O)NC(CCC)C(=O)NC)CCCCCN1C(=O)CN1CCSCC1 C1(CC(C)C)CCN(C(=O)C(C2(O)CCCCC2)NC(=O)CSC(C)C)CC1 N1(C(C2CCC(CCC)CC2)=O)CCCCC2(C1)CN(C(c1ccoc1Br)=O)C2 c1(C(C(=O)NCCC)N(C)CC2(O)CCCC2)cc(C)cc(Br)c1 Cc1ncn(C)c(=O)c1C(=O)NC1(C2CCCN2C(C2CC3CCC2O3)=O)CC1 c1(C(=O)NC2CN(C(C(C3CCC3)OC)=O)CC2O)ccc(F)c2ccccc12 c1(CC)cc(C(N2CC3C(CNC(=O)C(C)(CC)CO)C3C2)=O)ccc1O C1(C(=O)NOC)CCC(C)(C)N(CC(CC)C)C1 c1(C(=O)NC(C2CCCN(C(C3CC(C#N)C3)=O)C2)C)cnc2c(c1)CCC2 N1(C(C(=O)N(c2nc(C)c(C(F)(F)F)o2)CCC(N)=O)=O)CCc2ccccc2C1 N#Cc1ccc(N)c(C(N2CCCN(C(=O)CCS(N)(=O)=O)CC2)=O)c1 C=CC1(C(N2CCC(CC(C)C)CC2)=O)CCN(C(c2cc(Cl)cs2)=O)C1 C(=O)(C1CCc2snnc21)N(CCCNC(C(C)O)=O)C1CC1 C(=O)(CCCCC(=O)N1CCCC1CNC(C1(C)CCCC1)=O)OC C12CCN(CC1)C(=O)N2.n1(CC)nnnc1C(c1cc(C)on1)N(CC)CC N1(C(c2ncn(C(C)C)c2)=O)CCCC12CCN(C(c1cccn(O)c1=O)=O)C2 CC(CNC(c1cc(C(F)F)[nH]n1)=O)C(F)C(=O)NC1(C)CCCC1O C1(CC(=O)N(CC(C)NC(C23CSCC2C3)=O)C)(CO)CCCO1 c1(C(=O)NC2(CF)CCN(c3cc(CC)ncn3)C2)ccc(S(C)(=O)=O)cc1 C1(NC(c2ccn(CCOC)n2)=O)CC2CC1N(C(c1cnn(CCF)c1)=O)C2 N1(C(=O)OC(C)(C)C)CCC1CCCC(=O)NCCCC1CCCO1 C=CCC(C)(C)C(=O)NC1CC(CCNC(c2ccnnc2)=O)C1 c1(C(N(CCCNC(C2NC(=O)C(F)C2)=O)C2CC2)=O)nnc2ccccc2n1 CC(C)(O)C#CC(=O)N1CCC(C(=O)NCc2cn[nH]c2)C1(C)C c1(C(N2CC(C(C)NC(c3cc(O)ccc3O)=O)C2)=O)[nH]nc([N+](=O)[O-])c1Cl c1(C(=O)NC2N(CC)CCCC2)cc(N)c(Cl)c(O)c1.C1(=O)C(=O)NCC2C(C2)N1 C1(F)(C(=O)NCC(=O)N(CCOC)CC)COC1.C1CCNC(=O)CO1 N1(C(CCOCCNC(=O)CCOC2CC(F)(F)C2)=O)CC(O)(C2CCC2)C1 c1(COC(C(C)C(C)c2ccccc2Cl)=O)cn2ccccc2n1 c1(C(C)C)ncc(C(=O)N(CC(C)NC(=O)C(C)C2(O)CCC2)C)s1 n1(CC(=O)NCCC2CC(NC(C3CN(C(C)C)C3)=O)C2)ncc(O)nc1=O N1(C(C(C)=C2CC2)=O)CC(NC(C2CC2(Cl)Cl)=O)CC(C)(C)C1 Nc1sc2c(c1C(=O)NC13CCC1CN(C(c1cnc(O)s1)=O)C3)CCC2 C1(C(=O)NC(C#C)C)CCC2(CN(C(=O)CCc3ccn(C)c3)C2)O1 CCC(C)C(C)N=c1[nH]c(N(CC(CC)Oc2ccccc2Cl)C)nc(=NC)[nH]1 C1(C2CCN(C(=O)C(C)(C)C(C)(C)O)CC2)(NC(C(C=CCCC)O)=O)CC1 N1(C(C(C)OCC)=O)CCN(C(C2CC(F)(F)C2)=O)C(CC)C1 C(=O)(C(C)(C)S(C)(=O)=O)N1CC(C(C)NC(c2cc(C(=O)O)sn2)=O)C1 c1(C(N2C3C(CNC(CC4(OC)CCC4)=O)C(C3)C2)=O)cnc2[nH]cnc2c1 CC1COC(CN)CN1C(c1cccnc1N1CCCC1)=O c1(C(=O)NCC2COCCN(C(c3cc(C)ns3)=O)C2)ccnn2ccnc12 CC(C)C(C(=O)N1CCC(N(C(=O)C2=CCSC2)C)CC1)n1cnnn1 S(=O)(=O)(c1cccnc1NC1(CCF)CC1)NC(CNC(=O)OC)C N1(C(c2nc(CC)oc2)=O)CCC(CC(=O)NOCC2CCOC2)CC1 C=CC(CC)CC(=O)NCC(C)N(C(c1ccc2c(c1)CC2)=O)CC c1(OC)cc(C(=O)NC(c2ccc(F)cc2F)CNC(=O)C(C)(C)C)ccc1C CC1(C)COCC(C(N2CC(CNC(c3nn[nH]c3Cl)=O)C(F)(F)C2)=O)O1 c1(C(C)(C)C)nc2cc(CNC(=O)CCSCCC(=O)O)ccc2o1 C1(C2CC2)(NC(=O)CCc2ccsc2)CCN(C(C2CCNC2=O)=O)C1 c1(OC)cccc(OCCC#N)c1N(C)C(=O)NCc1cc(C)on1.OC C1(COC(C2CC(C(F)F)(NC(COCC)=O)C2)=O)CCCC(OC)C1 Cc1cn(C)cc1C(=O)NC(C)CN1CCN(C(C2(CN(C)C)CC2)=O)CC1 C(C(=O)NC1CCC(CNC(=O)C=CC(=O)N(C)C)C1)(C(C)C)n1ncc(C)c1 N1(C(c2cc(CCC)ncc2)=O)CCCCCC1CNC(=O)COC1(C)CCC1 O=C(CN1CCN(C(=O)CC(F)(F)F)CC1)C1CCCCc2ccccc21 Cc1ccc([N+](=O)[O-])cc1N(C(=O)CN(C(c1ccc(CO)o1)=O)C1CC1)C CS(=O)(=O)c1ccc(NC(=O)Nc2cc(C#N)c(Br)cn2)nc1 CC1(C)OCc2cc(C#N)c(=NCC3CCCN(C(=O)C=CCF)C3)[nH]c21 C(C(F)(F)CCC(=O)NC1CCC1)n1cc(C(C)NC23CC2CN(C)C3)nn1 c1(CNC(CC(C)NC(N)=O)=O)cccc(NC(=O)C(c2ccccc2Cl)O)c1 N1(S(CCOC)(=O)=O)CCC12CCC(OC)CC2 C(c1ccncc1)=C(C(=O)NC(CNC(CCOCCOCC)=O)C)C Cc1ccc(CCC(=O)N(C(C)CC(=O)NCCC(O)C2CCC2)C)o1 C(CC(O)C(=O)NCC1CN(c2nnc(C(F)F)o2)CCO1)SC C1(C(N2C(C)COCC2)=O)CC2CCC(C1)N2C(=O)CC(C)C CC1N(C(c2cc(CNC(C3(C#N)CC(=O)C3)=O)[nH]n2)=O)CCC1(C)C CC1CN2CCN1C(C(N1CCCCC1CNC(=O)Cc1ccccc1F)=O)C2 c1(C(N2C3CN(C(=O)Cc4cccc(Cl)c4)CC32)=O)cccc(I)c1Cl C(=O)(C1=NOC2COCC12)C1(CN2CC(N)C2)CC1 N1(C(C(c2ccccc2Cl)C)=O)CC2(CCCCN2C(C2COCCOC2)=O)C1 C(C)(CCC(=O)NCC(C)CNC(c1cc(C)nn1Cc1ccccc1)=O)OC C1(N(C(CCCN(C)C)=O)C)CN(C(C2C(Cl)(Cl)C23CC3)=O)CC12CC2 NS(=O)(=O)c1ccc(CC(=O)NC2CCN(C(=O)Cn3cnc(=N)[nH]3)CC2F)cc1 C1(NC(C2SCCCS2)=O)CCC12CN(C(=O)C(c1ccccc1F)O)C2 CC(C)C(O)CC(=O)NC1(C(=O)NCC2(C)CC3CCC2C3)CCSC1 c1(C(N(CCNC(C=C(CCC)C=CC)=O)CCOC)=O)ccc2c(n1)CCC2 N1(C(C(C)(C)O)=O)CC2CCN(C(C3CCC4CCCCC4C3)=O)CC12 Cc1nnc(O)c(C(=O)NC2CC(CNC(=O)COC3CCC3)C2)c1C C(=O)(C(O)CC[S+](C)C)N1C(CN(C(CCCN(C(C)=O)C)=O)C2CC2)CCC1 C1(NC(COC(CC)C)=O)CCN(C(c2ccc(NC(C)=O)cn2)=O)CC1F CCC1C(=O)Nc2ccc(C(=O)NCC(C3CC3)NC(c3cn(C)nn3)=O)cc21 C(C)(N=c1nc(N2CCC3CC3C2)c2c([nH]1)CCS2)c1c(C)noc1C CC1(C)CC(CC(=O)NCCC(F)(F)F)CN1C(=O)C=CC(F)F C1(NC(C2(SCC)CC2)=O)CC1C1CCN(C(C2CCCN2CC)=O)CC1 Ic1ccc(C(c2nnnn2C2COC2)NC2CC(C(F)F)C2)s1 C(N=c1ccc(C#N)c(C)[nH]1)C1C(C(F)(F)F)CCN(C(CN(CCC)C)=O)C1 C=C(Cl)CCCN=c1[nH]c(=NCC2(C3CC3)CCCC2)[nH]c2c1CSC2 N1(C(CN2CC(CC)C2)=O)CC2CC(NC(=O)C(C)OCCOC)C1C2 C1(O)(CN(C(=O)C(F)n2ccnc2)C)CN(C(=O)CCc2cncs2)C1 N1(C(CN(C(c2cc[nH]c3nccc2-3)=O)CC2CC2)=O)CCC2CCC(O)C1C2 c1(CC(=O)NCCNC(c2c(OC)cc(Br)cn2)=O)cc(Br)cc2c1OCC2 c1(C(N2CCN(Cc3c(OC)c(Br)ccc3)C3C2C3)=O)ccc(F)c(F)c1O C(c1ccccc1F)=CC(=O)N(C(CNC(=O)CC(F)(F)F)C1CC1)C N1(C(COC(C)(C)C)=O)CCC(O)(C(=O)Nc2cn(C3CCCC3)cn2)C1 C1(C(=O)O)C=CCCC1NC(c1cccc(N2CCCCC2)n1)=O c1(C(=O)NCC(C)CN(C(=O)CC2COCCO2)C)ccn2nccc2n1 c1(C(=O)NC2(CCNC(c3cn(CC)nn3)=O)CCCC2)ccc(C)cc1C c1(N2CCc3c(ccc(CC)c3)C2)nc(=NCCCF)[nH]c2c1CSC2.C1C(=O)N1 c1(C(=O)NCCC2(O)CN(C(C3(CC)CC3(F)F)=O)C2)cc2[nH]nc(C)c2cn1 C1(C#N)(C(N2CCC(NC(CCCN(CCC)CCC)=O)C2)=O)CC12CCCC2 C1(NC(Cn2c(C)ccn2)=O)CCCCC12CCN(C(=O)C(C)(C)N(C)C)C2 N1(C(C2CC(C)=C(C)CC2)=O)CCC(NC(C2CN(C)C2)=O)C(C)(C)C1 N1(C(c2c(SC)nn(C)c2)=O)CCCC2(C1)CN(C(C1(C)CCC(=O)NC1)=O)C2 c1(OCC)ccc(C)cc1C(N1CCCC(NC(=O)CC(=O)OC(C)(C)C)C1)=O N1(C(c2c(C)noc2C(C)C)=O)CCCC2CN(C(c3occc3F)=O)CCC12 c1(C(N2CC(CNC(C(COC)COC)=O)C(O)C2)=O)sc2cccnc2c1Cl c1(C(=O)NCC2CC(C(N3CCCCC3C3CCOC3)=O)C2)nnc(O)nc1O C1(C(=O)NC2CC(NC(C3CC(C(=O)OC)C3)=O)C2)Cc2nn[nH]c2C(C)C1 C1(C(N2C(c3cccc(OC(C)=O)c3)CCC2)=O)CC(C)(C)CC(C)(C)C1 Nc1cc(Cl)cc(Cl)c1C(N1CC2CCC1C2NC(c1ccoc1)=O)=O N1(C(C2CCCC2)=O)CC2CCC2(CC(=O)NC2CCC=CCCC2)C1 CC(C)(C(c1nnnn1CC(F)F)NCCC(N)=O)c1ccccc1 c1(OC)cnccc1C(=O)NCCCCCNC(C1CCC2(CC2)C1)=O c1(C(=O)NNC(=S)NC2CC(F)(F)C2)ccc2oc3ccccc3c2c1 C1(NC(c2nc(COC)oc2)=O)CC2CC1N(C(c1cccnc1O)=O)C2 C1(CC(N2CCC(c3cn(CCCC)nn3)C2)=O)CCN(C)CC1 N#Cc1ccc(C(N2CCCCC2C(O)C(F)F)=O)cc1[N+](=O)[O-] c1(C(=O)NC2CN(C(C(C)CF)=O)CC(C)(C)C2)c2c(nn1C)CCSC2 C1(NC(COCC)=O)CN(C(=O)CC2CSCCO2)CC1C(F)(F)F C1(CNC(c2scc(OC)c2)=O)CCN(C(c2cnc(C(F)F)s2)=O)CC1C c1(NC(C(C)Cn2cc(-c3nc(C4CC4)cs3)nn2)=O)cnn(C)c1S(N)(=O)=O CP(C)(=O)C1CCN(C(c2nc(-c3ccccc3)oc2Br)=O)C1 n1(CC)nnc2c(N3CCN(C)C(CNC(C4(CO)CCCC4)=O)C3)ncnc12 C=CC1(NC(=O)CC2CCCN(C(=O)CC3CCOC3C)C2)CCCC1 c1(SC2(c3n(CC=C)nnn3)CCC(=O)N(C3CC3)C2)c[nH]c(=O)c2ccnn12 C1(NC(C(c2cccnc2)OC)=O)CC2(CCCN(C(C3(C#N)CC3)=O)C2)C1 CC1(CCNC(=O)CC2CC(NC(c3c[nH]cc3CC3CC3)=O)C2)CCCO1 C1(NC(C(C)(OC)OC)=O)CC2CC(NC(C3(C)CCN(C4CC4)CC3)=O)CC12 N1(C(c2cc(CC)oc2C)=O)CCCN(C(=O)CN2CCCC2C)CCC1 c1(OC)ccc(C(=O)NC2CC(C)N(C(C3CCCC(N(C)C)C3)=O)C2)nc1Cl N1(C(c2cc(C(C)=O)sc2)=O)CCN(C(=O)Cn2nccc2N)CC(O)C1 c1(NC(C2CCCN(C(=O)N(C)C)CCC2)=O)n[nH]c2ccc(C(F)(F)F)cc12 C(=O)(CC(C(C)C)OC)NCCC(CC)(C)NC(c1ccc(C)cc1OC)=O C1(C)(CC(=O)OCC)CCN(C(=O)NC2CCN(c3ccncc3)C2)C1 CC1(C)CC(O)CN(C(=O)NCCC2(c3ccccc3)CCOCC2)C1 C(=O)(C(C)(O)CC(C)C)NCC(CC)NC(c1c(C)ccc(C)c1C(=O)NC)=O c1(C(N2CCCC(C(C)NC(c3csnn3)=O)C2)=O)cc(S(N)(=O)=O)cs1 N1(C(CCCC(=C)C)=O)CCC(NC(=O)COc2ccc(SC)cc2)CC(O)C1 O=C1OCC2CN(CCc3ccc(Cc4ccccc4)cc3)CCC12 CC1(C)CCCOC1C(=O)NCCCCNC(C1C2CCCCC12)=O C(=O)(CCC(=O)N(C)C)NC(C)C(CO)NC(C1CC(=O)N(O)C1)=O C1(NC(c2ccc(CO)o2)=O)CN(C(C2(C(F)(F)F)CC2)=O)Cc2nccn2C1 C(=O)(CCCS(C)(=O)=O)NCCCCC(C)NC(C1C2COCC12)=O c1(C(N2CC3CC3(C(N3CCOC(CO)C3)=O)C2)=O)cc(Br)c2ccccc2n1 CC1CCCCCCN1C(=O)C(CC1CCC1)NC(=O)C(C)c1ccsc1 C(=O)(C(C)(C)C(C)O)NCC1(COC)CCN(C(C2CCOC2CF)=O)C1 N(C(=NCC(F)(F)Cl)NC1CCC1)C(C(c1ccccc1)C)C c1(C(N2CCC(NC(COCCCC#C)=O)C(CC)C2)=O)ncnc2ccsc12 C1(NC(CCc2cccc(C)c2)=O)CN(C(c2ccc(Cl)c(O)c2)=O)CC1(F)F N(C1CN(C(=O)CCOc2cccc(Cl)c2Cl)Cc2ccccc21)C(=O)CO C(=O)(C#CC1CCCCC1)NCC(CNC(c1c(CC)con1)=O)CO C1(C(=O)NCC(c2ccccc2)NC(c2snnc2C)=O)(COC)CCCCC1 CCC(C)C(O)CC(=O)N1CCC(CO)(CNC(c2cc[nH]c2)=O)CC1 CC1CCC(NC(=O)C(C)(C)c2ccccn2)CN1C(c1cnco1)=O N1(C(C2C(C3CN(C(C4(F)CC5(CCC5)C4)=O)C3)C2)=O)CC23CCC2(COC3)C1 C1(F)(CN)CCC(OC(N(C(c2cn(C(C)C(=O)NC(C)(C)C)nn2)C)C)=O)C1 C1(C)(CNC(C=Cc2n(C)cnc2)=O)COCCN(C(C2CCNC(=O)C2)=O)C1 c1(N2CCCC(C(C)C)C2)nc(N2CC3CC3C2)c2c(n1)CCC(C)C2 N12CCC(C)(C1)C2=O.c1(C(=O)NC(CC)CSC)ccsc1C(F)F c1(C(=O)NC2(CO)CN(C(c3cnc(C(C)C)o3)=O)C2)ccc(C(C)(C)C)cc1 c1(C(=O)NC2CCN(C(C3CC4C=CC3C4)=O)CC2)ccn2ncnc2c1 C=CC(O)C(=O)NC(CN(C)C)C(=O)N1CCC(c2ccon2)C1 Cc1ncc2n1CCC(C(=O)NCC1CN(C)CCN1C(=O)CCOC(C)C)C2 O=C1CN(CC(N2CCC(Cc3cn(CCN4CC(F)(F)C4)nn3)C2)=O)CCN1 Cc1nc(CSCC(=O)N(C)CCNC(c2cn(-c3ccccc3)nn2)=O)cs1 CC1CC(NC(c2cnn(C3CCCC3)c2)=O)CN1C(=O)CC1COCCO1 N1(C(c2n(C(CC)C)ncc2)=O)CCC(C)(CNC(c2cnn(C)n2)=O)C1 c1(C(N2CC(CC)N(C(C3C(F)(F)C34CC4)=O)CC2)=O)cn2ccc(C)cc2n1 C1(O)(COC)CCN(C(=O)C(C2CCCO2)NC(=O)C=C(C)C)C1 Nc1cc(C(N2CC3CC3(CNC(C34COCC3C4)=O)C2)=O)cc(O)c1Cl c1(C(=O)NCCC(C)NC(C2CCCC2O)=O)cc(C(F)F)no1 Cc1ccc2c(c1)C=C(C(=O)NC1CC1CNC(=O)CCCC(N)=O)CO2 N1(C(C=CC(C)(C)C)=O)CCC(F)C(NC(c2ccc(C3CC3)o2)=O)C1 C1(C(=O)OCCC(C)(C2CCC2)NC(C(C)(F)F)=O)CN2CCCCC2CO1 N1(C(C(C=C)(C)C)=O)CCC(NC(C2(C)CC(OC)CN2C)=O)C(C)C1 n1(CC(=O)NCCC2CCCN(C(c3cc(CCO)on3)=O)C2)ncccc1=O C=CCC(CNC(=O)C=CC(C)(C)C)C(=O)NCC(C)(C)F C1(C(N(C(=O)C(C)=CC2CC2)C(C2(CC#C)CCC2)=O)C2CC2)C=CCOC1 C1(C(=O)NCC(C)NC(c2cccc(C(F)F)c2)=O)CCC2(C1)CC2(F)F N1(C(C(c2cncnc2)NC(CCC2CCC(=O)C2)=O)=O)CC=CC(O)C1 c1(C(=O)NC2CC(NC(=O)CSC(F)F)C2)cccc(-n2ccnn2)c1 n1(CC)cnc2[nH]c(=NCCSC(C)(C)C)[nH]c(=NC3CCC=CC=C3C)c12 c1(C(=O)NCCn2cc(CC(C)(C)CO)nn2)cc2sccc2s1 c1(C(=O)NCC(C)NC(c2c[nH]nc2C(F)(F)F)=O)cccc(C2CCC2)c1 N1(C(CC(C)c2ccncc2)=O)CCN(C(c2ccn(C(F)F)n2)=O)CCC1C C=CCC(C)(C)CC(=O)N1CC2(CCC2)CC1CNC(=O)CNC=O Cc1c(CC(N2CCN(Cc3ncco3)CC2C)=O)sc2ccccc12 C1(C(=O)NCCCN(C(c2c(C)coc2)=O)C2CC2)CCCN(S(C)(=O)=O)C1 N1(C(C2CCN(C)CC2)=O)CCC2(CCCN2c2cncc(Cl)n2)CC1 C1(C(=O)NC(CCC)(C)CC)CCC2(CC2)N1C(c1c[nH]cc1C)=O Cc1cc(F)cc(C(N2CC3CC(NC(c4c(I)cnn4C)=O)CC3C2)=O)c1O N1(C(C2N(CC)CC2)=O)CCC2CCC(NC(c3cccc4[nH]ncc34)=O)C1C2 c1(NCC=C=C)ccc(S(=O)(=O)NC(C)C(C)(C)OC)cc1Br C1(C(=O)NC(C)Cc2nnc(CO)s2)COCC(C)O1 N(S(=O)(=O)N1CCCC(C)C1)CC(C(C(C)C)O)(C)C C(=O)(C1=CCCOCC1)NC12C(C)OC(CNC(C3CN4CCC3CC4)=O)(C1)C2 c1(CC)cc(C(N2CCCC(NC(=O)C(F)=CCCF)C2)=O)cc(F)c1 CCC(C)(C)C(O)C(=O)NC1(CC(F)F)CC(C(N2CCN(CCF)CC2)=O)C1 N1(C(c2ccc(NC)cn2)=O)CCC2(NC(=O)CCC=C(C)C)CC2C1 C(=O)(C(F)C(=O)NC(C1(O)CCN(C(c2coc(Br)c2)=O)C1)C)OCC C1(NC(C2C(OC)C2)=O)CC(CO)N(C(=O)C=C2CN(C(C)=O)C2)C1.C(C=C)OC CCC(C(O)C(C)C)NC(=O)Nc1ccccc1Cl Cc1cn2cccc(C(=O)NC3(C)CCN(c4nc5ccc(N)cc5s4)C3)c2n1 c1(OC)c(Cl)ccc(C(=O)N(CCCNC(c2ccc([N+](=O)[O-])cc2)=O)C)c1F c1(-c2c(C)cc(C(=O)NCc3ccc(F)c(O)c3)nc2)cnc2ccccc2c1 CCC(CO)C(=O)N1CC(=C(F)CNC(C2CCCS2)=O)C1 C=C(C)C(C)(C)C(=O)NC(CNC(c1cnc(-c2ncccn2)s1)=O)CC(C)C c1(C(N2CCCC(NC(C(C(C)C)SCC)=O)CC2)=O)cc2c(ccn2C)[nH]1 N1(C(C2(COC)CC(=C)C2)=O)CCN(C(=O)C=Cc2cncs2)CC1 C(=O)(C#CC1CCOCC1)N1CC(O)(C(C)NC(C2(C)CCCC2(F)F)=O)C1 c1(C(=O)NC(C(C)NC(c2c(C)nc(CC)s2)=O)C(C)C)c(N)cccc1F c1(CC(=O)NCC(C)CN(C)C(C2CC2C(C)O)=O)ncc(Cl)s1 CCC(CC(=O)NCC(C)=CC(N1CCCC1)=O)NCCCC(=O)NCC(F)F Cc1nc(C(=O)N(C)CCC2CCCCN2C(C2CC=CCC2)=O)sc1C Cc1cccc(Br)c1C(C(=O)NC1CC2CC1CC2=O)NC(=O)CNC(N)=O C1(C(=O)NCC(c2csc(CNC(c3cnc(S)[nH]3)=O)n2)(C)C)CCOCC1(C)C CC1CCCN(C(=O)C(=O)N2CCN2C(=O)Cc2csc(=N)[nH]2)C1.C1(C)CC1 c1(OC)cc(C(=O)OC(C(N2CC(COC)C(C)CC2)=O)C)c(CO)cc1OC C1(C)(NC(C(C)OC)=O)CCCN(C(c2ncn(C(C)(C)C)n2)=O)C1 S(=O)(=O)(c1cc(NC(C2CCC(C(=O)O)CC2CCCC)=O)ccn1)N(C)C C(CC(=O)N1CCC(CO)(OC)C1)(CC(C)C)NC(c1c(COC)cc[nH]1)=O C1(C2CC2)(C(=O)NC(CCCC)CC)CN(C(=O)C(CO)OC)C1 n1(CC)ccc2c(C(=O)NC3CC3NC(=O)CSc3cnn(C)c3)cc(C)nc12 n1(CC)nc(C)c(=NC(=O)C2CN(Cc3cc(O)ccc3F)CC(F)(F)C2)[nH]1 N1(C(c2c(C)[nH]nc2Cl)=O)CC2(C1)CN(C(C1CCCC1CF)=O)CCO2 c1(N2CCC(C)(c3ccccc3)C2)nc(N2CCC(CCO)C2)c2sccc2n1 CCCCN=C(NCc1nccc(OC)n1)N1CCC(CC2CCCC2)C1 c1(C(=O)NC2CN(C(=O)C=CBr)CC23CC3)cccc2[nH]cc(Cl)c12 c1(C(=O)NCC2N(C(c3c(C)nc(C)o3)=O)CCCC2)cncc(C)c1Cl C=CCC(CC(=O)NC1(C)CCCC1O)NC(c1cnnn1C)=O C1(CNC(c2cnc(S)[nH]2)=O)CC12CCN(C(=O)CCc1ccc(F)cc1)CC2 C1(C(=O)NC2CC(OCC(=O)N(C(CC)CO)C)C2)COC(=O)N1 c1(C(N2CCC(OCCNC(C(C)OCCCC)=O)C2)=O)ncnc(O)c1F N1(C(COC)=O)CC2CCC1C1CN(C(=O)CC3(OC(C)(C)C)CCCC3)CC21 N1(CCNC(C2(COC)CN(C(=O)C(C)C(F)F)C2)=O)CCCCC1C c1(N2CC(CC(=O)NCC3(OC)CCC3)C2)ncnc2c1COC2 C(C(=O)NC(C)C)(C(C)CC(C)(C)C)N1C(COC)CCC1 S(=O)(=O)(c1ccc(=NCCNS(=O)(=O)CC)[nH]c1)N(CCCCCC=C)C c1(C(C(=O)NC2CCOC2)N(C(C)C)CC)cccc(C(F)(F)F)c1F c1(C(=O)NCC(CNC(C2C(C(C)C)C2)=O)(C)C)ccccc1CCC(F)(F)F C1(NC(C2C(C#C)C2)=O)CCN(C(=O)C=Cc2ccc(F)c(F)c2)CC12CCC2 C(=O)(CCCCC(F)F)N1CCC(CNC(CN(C2CCCCC2)C)=O)C1(C)C N1(C(CCC(=O)NCCC)=O)CCC(C(=O)NCCCc2cncnc2)C1(C)C c1(C(N2C(C)(C(=O)NCCC(CCC)O)CCC2)=O)cc(C)cc(O)n1 C(CC(=O)N1CCC2OCCC12)(C(N)=O)NC(C)=O CS(=O)(=O)c1nccc(N2CCN(C(c3c(Cl)ccnc3F)=O)CC2)n1 Cc1cn2cc(C(=O)NC34CCN(C(=O)Cn5cccn5)CC3C4)cc(C)c2n1 c1(C(=O)NCC2(F)CN(C(C(C3CC3)OCC)=O)C2)ccccc1C1(C)CC1 Cc1cnc2ccc(C(=O)N(C3CC(NC(=O)CCC(C)S(C)(=O)=O)C3)C)cn12 C1(NC(C(c2ccccc2)OC)=O)CCN(CCNc2ccc(=N)[nH]n2)CC1 N1(C(c2cc(=N)[nH]cc2)=O)CC2CCCC(NC(C34CCC(CC3)CC4)=O)C2C1 N1(C(C(C)SC)=O)CCC(F)(NC(=O)C(C)NC(=O)NC2CCCC2)C1 c1(SC)cccc(Br)c1CC(=O)NCC(C)(CC(C)C)NC(=O)C(C)O CC1(C)NC(=O)CC1C(N1CC(NC(=O)CC=CC(C)(C)C)C(CC2CC2)C1)=O C12(NC(C=CSC)=O)CCN(C(=O)C(CO)NC(=O)C(F)(F)F)CCC1C2 c1(C(CNC(=O)C(C)(N(C)C)N(C)C)NC(C2C(C)C2C)=O)cccc(Cl)c1 Cc1ccc([N+](=O)[O-])c(C(=O)NCC(CNC(c2cnsc2)=O)CO)c1C CCCCC(F)C(=O)N1CCCCCC1C(=O)NC(CC1CC1)CC1CC1 CC1(C)CC(C)(C(N2CCCCC(F)(F)C2)=O)CN1C(=O)C1=NOCC1 Cc1nccc(CCc2cc(N3CCC(c4ccncc4)C3)ncn2)n1 C12(C(N3CC(SC)C3)=O)CCC(C(=O)NCC3CCC(O)C3)(CC1)CC2 C(C)(CC(C)(C)CO)NC(CC1N(C(C(=Cc2cn[nH]c2)C)=O)CC(O)C1)=O N1(C(c2cc(C)nc(O)n2)=O)CCC2CCCN(C(=O)CCN3CCCC3)C2C1 C(=O)(CCCC(=O)N1CC2CC2(CNC(=O)CSCC2CCCCO2)C1)NC N1(c2nnc(CSC(C)C)n2CC2CCCCO2)CCC2(C1)CC(F)(F)C2 c1(C(=O)OC)cc(NC(CO)C(=O)N(C2(C)CC2(F)F)C)ccc1OC c1(C(N2CC(C(C)NC(c3c(CC)ncnc3)=O)OCC2)=O)cc(C)ccc1F CCS(=O)c1ccccc1C(=O)NCC1(OC)CN(C(C2(C)CC2)=O)C1 N1(C(C2(C(=O)NC3(CO)CCCC3)CC2)=O)C2CCC1C(CCN1CCCC1)C2 Cc1nc(Br)c(C(N2CCC(CO)(NC(=O)C(C)C3CCC3)C2)=O)s1 N1(C(c2c(OC)oc(C)n2)=O)CCC(O)(CCNC(c2cnc(C#N)s2)=O)CC1 CC1CN(C(=O)COc2cccnc2)CC(CCNCc2ccnc(O)c2F)O1 Cc1cnc(F)cc1C(=O)NC(C)CCCCN C(CCCCCC1CC1)CC(=O)NC.C(CC(=O)NCC(C)(C)O)=C(C)C c1(OCC(N2CCC(N(C(C)=O)CCO)C2)=O)ccccc1C.c1(C=O)nc(CS)cs1 c1(-c2cc(C(=O)NC(CCCC)COC)ncc2)ccc(OC2CC2)cc1C S(=O)(=O)(c1ccc(NCC2(CO)CC3CC3C2)c2cnccc12)N(C)CCF C=CC1(CC(N2CCCC(C3CCCN3C(=O)C=CCC)C2)=O)CCCCC1 C1(Nc2cc(OCC)n[nH]2)CCN(C(=O)CCN(CCC(C)(C)C)C)C12CCC2 C=CC1CN(C(C2CCC(NC(c3coc(CO)c3)=O)CC2)=O)CC1O c1(OC)cc(COCCNC(C2(O)CCN(C(c3cncs3)=O)C2)=O)ccn1 c1(C(C)C)ccc2cc(C(=O)NCC3CC3CNC(c3csc(C)n3)=O)[nH]c2c1 CCC(C)C(O)C(C)C(=O)NC1CCN(C(C2CC(=O)C2C(C)(C)C)=O)C12CC2 Cc1cccn(CC(N2CCC(NC(c3ccc(C(C)C)o3)=O)C(O)C2)=O)c1=O c1(C(c2nnnn2CCSC)NC2CC(=C)C2)ccc(Br)cc1OC(F)F CC#CC1CCN(C(C2(C)C=CCN2C(c2cc[nH]n2)=O)=O)C1 c1(N(CCC)C(c2cn(CCN3CCC(O)CC3)nn2)=O)cc(Cl)c(C)cn1 c1(C(=O)NCC(CC)(C)NC(c2n[nH]cc2COC)=O)cccc(C(N)=O)c1C CC(C)CCCCC(=O)N1CC(CC(=O)NC2C3CCCOC23)C(C)C1 c1(C(C)Sc2ccc(OOCc3ccccc3)cc2)cc(F)cc(F)c1 C(CNC(c1cccnc1C)=O)(C(C)C(C)C)NC(CCn1ncc(C)c1)=O N1(C(CC2CCCCC(=O)N2)=O)C2CCC1CC(NC(=O)C(Cl)=CCl)C2 c1(C(=O)NC(C(C)SC2CC(c3ccccc3)C2)=O)sccc1C#N CC1C(NC(c2cnccc2Cl)=O)CC2CCC1N2C(c1ncc(Cl)s1)=O C(=O)(CC(CNC(=O)CC(C)n1ccnc1)C1CCC1)N1CC(C)(CC)C1 C1(C(N2CC(C)C(C(N3CCOCC(O)C3)=O)C2)=O)CC2CC(=O)C1O2 N1(C(CCc2n(C)ccn2)=O)CC(NC(=O)CP(C)(C)=O)C(O)C1 c1(CNC(C2CCC(NC(c3c(C)cc(Br)o3)=O)C2)=O)cc(Cl)ccc1Cl C1(N(C(C(CNC(c2n(CC)nc(C)c2)=O)N(C)C)=O)C2CC2)CC2(C1)CC(C)C2 c1(C(=O)NCCN(C(=O)CC2CC(C(F)F)C2)CC)ccc2c(c1)NCCC2 C=CCN=c1[nH]cc(C(=O)NC2CN(C(=O)CSCC(N)=O)CC2C)s1 C1(C(N(CCCCNC(C(C)OCC2CC2)=O)C)=O)CCC(=O)N1C c1(OC)nc(NCC2(CCNC(C3(O)CC4CCC3C4)=O)CC2)ncc1C CCC(CNC(=O)CO)(CC)C(=O)NC1CCN(C(C)C)C1.c1(CO)nc[nH]n1 C1(C(N(CCCCNC(CSCCC)=O)C)=O)CCCN(C(C2CC2F)=O)C1 C1(C(N2CCCC(C(CNC(CC(=O)OC)=O)(C)O)C2)=O)CCCN2CCCC12 C(=O)(CCCC(C)(F)F)NC1C(SC)CN(C(c2ccsc2C#N)=O)C1 C1(NC(C(CC)(O)c2ccccc2)=O)CCN(C(=O)C2=C(C)CC2)CC1(C)C C1(C)(C(N(CC(CN(C)C(c2csc3cncn23)=O)O)C)=O)CCCNS1(=O)=O C1(CNC(COCCCCCC)=O)CN(C(c2cncc(COC)c2)=O)C2CC12 c1(C(N2CC(CNC(c3scc(C)c3)=O)N(C)CC2)=O)cccc2ncc(C)n12 N1(C(C2C(CC)C2)=O)CCC(C2(O)CN(C(c3cc4c(s3)CCCC4)=O)C2)CC1 C=CCC(F)(F)C(=O)NCC(C(=O)NC(CC1CC1)CC1CC1)N(C)C c1(C(=O)NC2(OC)CCN(C(=O)CC(C)NC(N)=O)C2)ccc(Cl)c(Br)c1 C=CC1(NC(=O)C(Cn2cncn2)NC(=O)Cc2cnsc2)CCC1 C1(NC(CCC(C)Nc2nnc(C3CCNCC3)s2)=O)CS(=O)(=O)CC1C C1(N(C(=O)C(=O)NCC2CC2)CC)CCCN(C(=O)Cn2ncn(C)c2=O)C1 C12(C(=O)NCC3N(C(C(N4CCSCC4)C)=O)CC3)CCCC1(C(N)=O)C2 N1(C(CCCN(C)C)=O)CCC(c2ccccc2)(CNC(=O)CCS(C)=O)CC1 c1(OCC)ccc(CN2CCSC(C(N3CCCCC3C#N)=O)C2)cc1Cl Cn1c(C(=O)NC(CNC(=O)CC2CCCCC2)CO)cc(Cl)c1Cl N1(C(c2c(C)nn(CCO)c2)=O)CC2CCCC1C2CNC(=O)CCc1ccc[nH]1 C1(CC)CN(C(=O)C=CI)CCC1NC(c1nocc1Cl)=O C1(NC(c2n[nH]cc2NCc2cncs2)=O)CCCC1C(F)(F)F n1(CCC)nc(C)c(C(=O)NCCC(=C)CNC(c2nn(CC)cc2Cl)=O)c1C c1(C(N2C(CCC(=O)NCCCc3ccncc3)CCC2)=O)ccc(F)nc1F c1(NC(=O)NC(c2cn(C)nc2)C2CCCCC2)sccc1C#N c1(C(N(C)CC2CCCN(C(CCC(=O)NCC)=O)C2)=O)c(F)cc(N)cc1F c1(NCCCN(C(C)C)C2CC2)nccc(=NCC(C)Cc2ccccn2)[nH]1 C1(CC)CCCN(C(c2cc(C)c(C)cn2)=O)C1C(N1CCCC(C(=O)OC)C1)=O C(CCN=C(NCC(F)F)NC1CC(=O)N(C2CC2)C1)N(S(C)(=O)=O)C C(=O)(C1=CCCC1(C)C)N(C)CC1CCCN(C(c2c(Cl)cnc(SC)n2)=O)C1 N1(C(C(c2cnn(C)c2)C)=O)CC2CC(O)C1C2NC(c1snc(O)c1Cl)=O CCCC(C)CC(=O)N1CCCC(N(C(=O)CCOCC)CC2CC2)C1 N1(C(c2cnc(C)nc2)=O)CC2(C1)CN(C(C1CC1(C)Br)=O)C2 O=C(C1=COCCC1)NC1CC(F)CN(C(c2cc(O)ncc2Br)=O)C1 N1(C(C(=Cc2cccs2)C)=O)CC(NC(=O)C(C(C)C)NC(C)C)C2(CC2)C1 c1(C(CC)CC)nc(C)c(NC(C2CCCC(C)C2)=O)o1 N(C(=NCCF)N1CCN2C(=O)NCC2C1)CC(CCCC)CCC Cc1c(Cl)cnn1CC(=O)NC1CC1CNC(=O)CCCc1cncs1 N1(C(C(CC(=C)C)OC)=O)CC2CC(C(=O)NC(CO)C(F)(F)F)C(C2)C1 C1(CNC(C2CCC(C(CC)=O)CC2)=O)COCCN(C(C2(CC)C=CCC2)=O)C1 c1(C2C(=O)N2)cn(C)nn1.C(CN=[N+]=[N-])N(C(=O)CN(C)C(C)=O)CC C1(OC)CC(NC(c2c[nH]nc2C2CCCO2)=O)CN(C(c2occc2C)=O)C1 C(=O)(C1=CC2CCCCCC12)NCCN(C(CSCCCC)=O)C1CC1 C(=O)(C(CN)C(C)C)N(C1CCCC1)CCOC c1(C(N(CC(=O)NCC=C(C)C)CC2CC2)=O)cc2ccccc2[nH]1 N1(C(CCCC)=O)CCN(C2CCCN(C(=O)CCN(S(C)(=O)=O)C)C2)CC1 N1(C(C(C)N(C)C)=O)CCc2ccccc2C(NC(=O)COc2cccc(C)c2)C1 c1(C(=O)NC(C)(CNC(=O)Cn2cc(N)cn2)C2CC2)cncc(F)c1 c1(C(=O)NCC2CN(C(Cn3nc(C)oc3=O)=O)C2)cc(N)c(C)c([N+](=O)[O-])c1 C=CCCCCC(=O)N1CCCC1(C(N1CCC(CC)C1)=O)CC N12CCC3(CC3C1=O)C2.C1(OC)CCC2(C(=O)NCCN3CCC4CC34)CC12 CCS(=O)(=O)c1cccc(C(F)(F)C(N2CCNCC2c2cccc(O)c2)=O)c1 C(=O)(C(O)CC(N)=O)NC1C(CC(=O)NC2C(OC)C(O)C2)CCC1 N1(c2ncc(C(=O)OC)nc2)CCCC2(NC(C3(C)CS(=O)(=O)C3)=O)CC2C1 c1(C(=O)NCC2CCN(C(C3CCC3C(F)F)=O)CC2)ccc([N+](=O)[O-])cc1F N1(C(CC(C=C)C)=O)CCN(C(=O)CN2CCCCCC2)CC(C)(C)C1 C1CN(C)N2CC(N(C)CC2C)N1.c1(-c2nc(C)[nH]n2)ccc(N(C)C)cc1 c1(C(=O)NC2C(NC(C(CC(C)(C)C)OC)=O)CC2)cccc2nn(C)cc12 c1(C2C(C(=O)NCCN(C(=O)CCc3cccn3C)C(C)C)C2)cc(F)ccc1Cl c1(C(=O)NCCNC(CC2OCC(C)(C)C2)=O)cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 CC(C(=O)NC1CCN(CC(F)F)CC1)C1=CCCC1.c12cccc(c1)NC2=O c1(C(=O)NCC2N(C(C3CCC(=O)NC3)=O)CCC2)c(F)cc(F)cc1Cl C=CCN=C(NCCSc1sccc1C)N1CCn2c(C(F)(F)F)nnc2C1 CN1C(=O)CCc2cc(C(N3CCCC(NC(=O)CCC4(C)CC4)C3)=O)ccc21 c1(CC(C)NCC2(OCC)CS(=O)(=O)C2)ccc(Cl)cc1Cl N1(C(C2N(C)C(=O)CC2)=O)CCC(C2CC2)(CNC(C23CCCN2CCC3)=O)C1 C1(NC(Cn2ncc(CC)c2)=O)CCN(C(=O)Cc2ccccc2)CC1CO O=C(C(O)C1=CCCCC1)NCC1CN(C(C2(C3CC3)CCC2)=O)C1 CCCCCCCCCC(=O)N1CCN(C(=O)CN(C)CCC)CCC1C CC1CC2CCCC2N1C(c1ccn(CCNC(c2cc(F)ccc2O)=O)c1)=O c1(C(N2CCC(CO)C2)C(=O)NCCC#N)ccc(C2CCC2)nc1 c1(C(=O)NCCCCN(C)C(C2CCC(=O)N2C)=O)cnn2cccc(Cl)c12 c12cscc1NN(CC1CC1)CCOC2=O.C1(C)CC1.C1(C)CC1 N1(C(CCSC)=O)CC2CN(C(C3(Cl)CC3(F)F)=O)CC2C1 c1(C(C(=O)NCCCN(C)C(C2CCCC2CF)=O)(C)C)ccc(Cl)cn1 c1(C(=O)OC(C)(C)C)cn(C2CCC(NC(N(CCC(=O)O)C)=O)C2)nn1 C(=O)(CC(C(F)(F)F)NC(=O)CCN1CCOC1=O)NCCC(C(C)C)N(C)C Cc1nc2c(F)cccc2cc1C(=O)NC1(C2CCN(C(C3CC3F)=O)C2)CC1 N1(C(C2(CC#C)CCCC2)=O)CCCCC(CNC(=O)CC2CC=CCC2)C1 Cc1ccn2ncc(C(N3CC4=C(C3)CN(C(=O)C(C)C3CCOC3)C4)=O)c2n1 c1(CC)cc(C(=O)N(CC(C)C(=O)NCC2CCC(O)CC2)C)nn1C C(=O)(C1=NOC(C)(C)C1)NCCOC1CCN(C(C2CC(C)N(C)C2)=O)C1 c1(C(N(CCC(C)(F)F)C)=O)ccc(C2CC2)cc1 CC(C)(C)C(CC(=O)NCC1OC(=O)NC1(C)C)NC(=O)CNc1ncccn1 N1(C(c2c(=O)ccn(C)c2)=O)CC(CNC(C2CC3CC2C3)=O)CC12CCC2 CCC(C)C1CC(=O)N1c1ccnc(C2CC2)c1.C(C(C)(C)n1cccn1)C(=O)NC c1(COC)cc(C(N2CCCCC2CCNC(c2ccnnc2O)=O)=O)n(C)c1 c1(CNC(CC(CC)NC(c2ccc(F)s2)=O)=O)cc(F)ccc1F C(N=c1[nH]cnc(Cl)c1[N+](=O)[O-])C1CCN(C(c2cc3c([nH]2)CCOC3)=O)C1 c1(C(N2CC(CNC(c3cncnc3C(C)C)=O)OCC2)=O)cc(O)ccc1O CN1N=C(C(=O)N2CCC(F)(CNC(c3cccc4c3OCC4)=O)C2)CCC1=O C=CC(CC)CC(=O)NCC1CN(C(c2cnc3n2CCS3)=O)CC12CC2 O=C(N=c1cc[nH]cc1O)C1CCN(C(C2CC(=O)N(Cc3ccco3)C2)=O)C1 C1(NC(CC(CC)C2CCC2)=O)C2CC1CN(C(=O)CC1(C)CCS(=O)(=O)N1)C2 c1(C(=O)NCC2CC(O)(CNC(C(CC)=CC)=O)C2)cccc(NC(=O)CC)c1 c1(SC)ncc(C(=O)N(CC(C)N(C(=O)C(CN(C)C)c2ccccc2)C)C)s1 Cc1c(C(N2CC(CNC(c3ccc(C(N)=O)cn3)=O)C(C)C2)=O)nnn1C c1(CCC(N2CCC(F)(CNC(C3(N(C)C)CC3)=O)C2)=O)ccc(Cl)c(F)c1 CC(C(C)C(=O)N(C)Cc1nccs1)NC(=O)CCC1CCCOC1 CCCCCC=CCC(N1CC(C(O)C(=O)Nc2ccnn2CC)C1)=O C12(NC(Cc3nc(CC)sc3)=O)CCN(C(c3ccc(F)cc3Cl)=O)CCC1C2 Cc1cc(O)ccc1N(C(=O)COC(=O)CC=CC(C)(C)C)C CC1CCc2sc(C(N3CCCCC3CNC(=O)Cc3cnnn3C)=O)cc2C1 N1(C(c2cc(OC)n[nH]2)=O)CCOC(C(C)NC(=O)C=Cc2cccs2)C1.C1CO1 C1(CC(=O)NCCOCCCNC(c2coc(Cl)n2)=O)CCCCC1O N1(C(C(C)N(C(C(C(=O)NC)(C)C)=O)C)=O)CCCN(C)CC1C N1(C(=O)Cc2cc(Br)ccc2F)CC2CN(C(C3(C4CC4)CC3)=O)CC2C1 C(F)(F)(C(F)(F)F)c1cc(CC(=O)NCC(C2CC2)NC(=O)Cc2cccs2)no1 c1(CC(=O)NC(C)CC(C)NC(=O)C#CC2CCC2)cc2ccccc2oc1=O N1(C(C2CC(SC)C2)=O)CCCC(C)C1CNC(c1cc(C)ccc1N)=O c1(NC(CC=C)=O)cnn(C(=O)NCCC2CC(OC)C2)n1 N1(C(CN2CC(C)C2)=O)CC(NC(=O)C=Cc2ccc(C(N)=O)cc2)C(C)(C)C1 c1(C(N2CCC(C(=O)Nc3c(OC)c(F)ccc3)C2)=O)cc(C)cc2[nH]ccc12 C1(NC(c2cccc(C)c2Cl)=O)COC2(C1)CN(C(C1CC3C=CC1C3)=O)C2 c1(OC)cc(C(N2CCCC(O)CC23CCC3)=O)c2sc(C=O)nc2c1 C12(NC(C(C)C3CCCC3)=O)CCCN(C(=O)C(c3ccccn3)O)CC1C2 c1(CC)ccc(C(=O)NCC2CC(NC(c3cnccc3C(C)(C)C)=O)C2)cc1 c1(-c2nc(C(N(C)CC3(O)CN(C(=O)OC(C)(C)C)C3)=O)on2)ccc(Br)cn1 C=CCCCC(C)(C)C(=O)N1CC(CCNC(c2cc(CO)on2)=O)(OC)C1 C1(CC(=O)N(CCOC(C)CCC)C(C)C(C)C)CCC(NC(=O)COC)CC1 c1(C(=O)NCC2CCCN(C(CC(C)SC)=O)C2)[nH]c2cc(F)ccc2c1C N1(C(CNC(C(CC)C(=O)OC)=O)=O)CCn2nccc2C1 CC1CC(CC(=O)O)CN1C(C1(C)CN(C(c2cccn2C)=O)C1)=O C1(N(C(=O)NC2(C(C)C)CCC2)C2CC2)CNC(=O)CC12CCC2 C1(CNC(CCNC(C)=O)=O)CC2CC2N1C(c1ccsc1C)=O CN1CCC(C(=O)NCC2CCCN(C(=O)C(C)(F)F)C2)S1(=O)=O C1(C)(NC(C(N2CCC(O)CC2)C)=O)CCN(C(=O)CCc2cncn2C)CC1 N1(C(C(C=C)O)=O)CC2CC1C2C(=O)NC(CC1CC1)CC1CC1 C(C)(CC(=O)N1CCCC1CCNC(=O)COC1CC(F)(F)C1)OC c1(NC(=O)NC2CC3CCC(C2)N3Cc2nc(Br)cs2)cccc2c1CCCO2 N1(C(c2cc(OC)ncn2)C(=O)NCCCSC)CCC(C2CC2(F)F)C1 c1(OCC)ccc(CCC(=O)NC2CC(CNC(C3(C)CC(F)(F)C3)=O)C2)cc1 C1(CNC(c2n(CC)cc(Cl)c2)=O)CN(C(c2cc(C(N)=O)c[nH]2)=O)CCCO1 C(=O)(C1=C(C)OCC1)NCC1(NC(=O)CCOC)CC(C(F)(F)F)(OC)C1 c1(CC)nc(C)c(C(=O)NCCCCN(CCCNC(=O)CN2CC3CC3C2)C)o1 N1(C(c2cc(CC)[nH]n2)=O)CC(C2CCN(C(C3C4COCC34)=O)CC2)C1 N1(C)CCc2ncnc(OC(C(CC)(CC(=O)OC)c3ccccc3)=O)c2C1 c1(C(=O)NCC(C)(C)NC(=O)CC2(O)CCCCCC2)ccc(P(C)(C)=O)s1 C(CNC(=O)CC1(C)CCS(=O)(=O)N1)(C(C)C(C)C)NC(C1C(OC)CCC1)=O c1(C(N2C(CN(C(C=Cc3occ(C)n3)=O)C)COCC2)=O)cccc(Cl)c1F C1(NC(c2ccc(F)o2)=O)CCN(C(c2cnc(S)n2C2CC2)=O)CC1F c1(C(CN(C)C)NC(=O)OC(C)(C)C)ccc(F)cc1.c12ccc(s1)CCC(=O)N2 Cc1cc(CO)oc1C(=O)NC1(CNC(=O)C(C2CCCCC2)O)CCC1 c1(C(=O)NCC2(C)CCC(NC(CSC(C)C)=O)C2)cc(F)cc2ccncc12 C(=O)(CC(O)C(C)C)N1CC(OC)C(NC(=O)COc2ccc(C(C)C)cc2)C1 N1(C(=O)NC2CCCC(CO)CC2)CCC2(CC1)OCC(O)C2O c1(C(=O)NC(CCCCNC(C2CC(SC)C2)=O)C)cncc2ncn(C)c12 CC(C)CCC(F)C(=O)N1CCC2C(NC(c3ccc[n+]([O-])c3)=O)C2C1 N1(C(CCC=CC(C)C)=O)CC2CCN(C(C3CN(C)CCO3)=O)CC2C1 C1(CNC(C(=O)OC)(C)c2ccccc2)Cc2ccccc2N(C)C1=O N1(C(c2c(C)nccc2Cl)=O)CCCN(C(=O)Cc2csc(Cl)n2)C(CO)C1 Cc1ccc(S(=O)(=O)NCCC(=O)NCc2cccc(-n3cncn3)c2)c(F)c1 CC1(CNC(c2cccnc2)=O)COCCN(C(C2(C#N)CCCOC2)=O)C1 c1(NC(C2(O)CCN(C(C(C)c3cccs3)=O)C2)=O)ccc(Cl)c(Cl)n1.C(=O)N C1(CNC(=O)CC2CCC(=O)O2)CC2CCC1N(C(C1(C(F)(F)F)CC1)=O)C2 CN1CCCC1CCNC(c1c[nH]nc1CCNC(c1csc(F)c1)=O)=O N1(C(C(C(=O)OCC)C)=O)CCCC(O)(C(=O)NCCC2(CO)CCC2)C1 O=C(C1=CCCCC1)NCCC1COCCN1C(=O)C(O)Cc1ccc(F)cc1 C(=O)(C(CC(C)N(CC(=C)C)C)N1CCCC(C)(CCC)C1)OC C(=O)(C(F)(CNC(=O)C1=CCCCCC1)C(C)C)N(C)Cc1onc(CC)n1 c1(C(=O)NCC(CCOC)NC(C2CN(C)C2)=O)cc2c(s1)CCCC2 c1(CC(=C)C(=O)N2CCC2(C)C(=O)NCC2(C3CCC3)CC2)ccc(F)cc1 C1(C(=O)NCC=CCNC(c2ccc(-n3cncn3)cc2)=O)CCCC2(CCC2)O1 C1(F)(CNC(c2cnc(SC)[nH]2)=O)CCC(NC(C2CCCCS2)=O)C1 C(=O)(C1(C)CC(C(C)C)c2ccccc21)NC(CNC(CCC(C)C)=O)CC C(C)(N=c1nc2sccc2c(N2CCC(CC(N)=O)CC2)[nH]1)c1c(C)noc1C N1(C(C(C)SC)=O)CCCC(N(C)C(c2cc(-c3ccco3)[nH]n2)=O)CC1 CC1CSCCN1C(=O)CC(CC1CC1)NC(=O)CCOCCN(C)C N1(C(c2cnc(OCC)s2)=O)CCCC(O)(CNC(c2cccc(N)c2F)=O)C1 c1(-n2c(C(C)(CCOC)NC(C3(CC)CC3)C)nnn2)ccc(OC(C)C)c(F)c1 C(=O)(CCC(N)=O)NCC(CN(C)C(C1(c2cccc(Cl)c2)CC1(F)F)=O)O CC1(C#CC(=O)NCCC2(C)CCN(C(c3cccc(F)c3O)=O)C2)CCCO1 C(=O)(C=CS(C)(=O)=O)N1CC(CN(C(=O)Cc2cncnc2)C)OCC1 C1(NC(c2c(C)nn(C3CCC3)c2)c2nnnn2C)CCn2cncc2C1 c1(C(C)Nc2ns[nH]c2=O)ccccc1[N+](=O)[O-].N12CC(CC1C)C2=O C=C(C)C1OCCC1CNC(=O)CC(C)CNC(=O)C(F)=CC1CC1 c1(C(N2CCc3cccc(Cl)c32)C(=O)NC2CCC2)csc2ccc(Cl)cc12 c1(COC(C2CCCC(CN)O2)=O)nc2ccccn2c(=O)c1Br C1(OC)CCN(C(c2cc(CNC(=O)C(O)C(C)(C)C)[nH]n2)=O)CC1C Cc1cc(N)cc(C(=O)NC23CC(C)(C2)OC32CCC2)c1F c1(C(N(CC=C)CC=C)=O)[nH]c(C)c(C(N2CC(C)SC(C)C2)=O)c1C N1(c2nnc(C3N(C)CCC3)n2Cc2cccs2)CCC12CCN(C)C2 C(C1=CCN(C(=O)C=CCCC=C(C)C)CC1)NC(CCC(C)SC)=O N1(C(CC)=O)CCCC1CCNC(C12CC(C)C1C2)=O C(=O)(C1=COCCC1)NCCC1CC(C(=O)NCCC2CCCCO2)C1 C(c1cccc([N+](=O)[O-])c1)=CC(=O)NC1CC1C(=O)NCc1cccc(O)c1 c1(C(N2CC(CCCNC(COCC)=O)OCC2)=O)cnc2[nH]c(C)nc2c1 C(CC(CNC(=O)COC(C)C)NC(=O)CCc1cccn1C)OC C1(NC(c2ccc(C(N)=O)cn2)=O)CCCCN(C(c2ccnn2C2CC2)=O)C1 N1(C(c2c(C)scc2)=O)CCC(NC(c2ccc(C(F)(F)F)[nH]2)=O)C(C)C1 C(=O)(C(CC(C)(C)C)NC(=O)C=CC1CCCCC1)N(C1C(C)COCC1)C C1(NC(c2ncn(C(C)C)c2)=O)CC2CC(NC(c3ccc(O)c(Cl)n3)=O)CC12 CN=S(C)(=O)c1ccc(C(=O)NCC(C)N(C)C(c2ocnc2C)=O)cc1 C1(CCC(=O)NC2C(N(C)C)COC2)CCCCN(C(=O)C(C)(C)CC2CC2)C1 c1(OC)ccc(F)nc1NC(C1CC1C(=O)Nc1cccc(C#N)c1)=O C12(CC)CCCN(C1)C(=O)C1(CC1)Cn1ccc(c1C)C(=O)N2.N1(CC)CCCC1 N1(C(C2CCC(OC)CC2)=O)CC2COCC(C1)N2C(c1ccncc1)=O C1(C)(NC(C(CC)COC)=O)CCCN(C(=O)CCc2ccccc2C(N)=O)C1 Cc1nc(Sc2c(NC3CCCN(n4c(C)ccc4C)C3=O)cnn2C)c(C)o1 C1(NC(C(C)SC)=O)CCSC12CN(C(=O)C(C)Cc1ccc(F)cc1)C2 C=CCCC(C(=O)OC)NC(=O)C(CC)NC(c1nscc1C)=O c1(CNC(C(=O)NCC2(O)C(C)(C)CCC2)=O)cc(Cl)cc(Cl)c1F FC1(F)CCN(c2ccnc(NCC3CCCN(C4CCCCC4)C3)n2)CC1 N1(CCn2c(C)cc(C)n2)Cc2ccc(O)cc2CC1C(N1CCCC(F)C1)=O c1(OC)c(Cl)cc(NC(=O)Nc2cn(C)nc2C(F)(F)F)cc1Cl c1(C(C)=O)cc(NC(=O)OC(C)(C)Cc2cccc(O)c2)ccc1F c1(NC(=O)NCC2C3CCCC23)ccc(-n2ccnc2)cc1 N1(C(CCC(C)C)=O)CC2(CCCC2)C1C(N1CCN(C(C)C)C(=O)C1)=O C(C(O)C(=O)NC(c1cn(C2CCCC2)nn1)(C)C)SC C1(CNC(c2c(C)ccnn2)=O)CN(C(c2coc(C(F)(F)F)c2)=O)CCC1C C1(NCc2ccnc(C)n2)CCCC(F)(F)C1O C1(C(N(C2CCN(C(C)=O)C2)CCC)=O)CCCN(C(C)CC2CCC2)C1 c1(C(=O)NCC2N(C(C=CCOCCOC)=O)CCOC2)coc2c(C)cccc12 c1(C=O)c(Cl)nc(SC)nc1Cl.N1(CC)CCOCC1CC(=O)NCC(=O)OCC C1(C(N2C(C(=O)NCC(N(C)C)C3CC3)CCC2)=O)CCCC(=O)C1 N1(C(C(N)=O)=O)CCN(C(=O)CC2C=CC=CC=C2)C(c2cccnc2)C1 Cc1csc(CNC(C2CC2CNC(C2CCC2)=O)=O)c1 N1(C(C=CCSC)=O)CC2CCN(C(c3ccc(Br)c(OC)c3)=O)CC2C1 CCC(O)C(F)(F)C(=O)N1CC(NC(=O)Nc2cccc(C(=O)O)c2)C(O)C1 N1(C(c2cc(Cl)ncc2Br)C(=O)NCCCOC)CCN(C)C2CC12 N1(c2ncc(C)c(C)n2)CCC12CCN(C(c1nc(Cl)ccc1F)=O)CC2 N1(C(CC=CC=C)=O)CC(C)(C)CC1C(N1CC(C(=O)OC)(OC)C1)=O N1(C(C=CCC)=O)CCC2CC12C(=O)NCC1CCCC(OC)C1 CCC(CNC(C1CC1(F)Cl)=O)(CC)NC(c1cncn1C)=O C1(NC(Cc2cc(OC)no2)=O)CC12CCN(C(C1CC1F)=O)CC2 c1(C(=O)NCCCc2cn(C(C(=O)NC(C)C)C)nn2)cnc2ccnn2c1C Cn1cc(SC=CC(=O)N2CC(O)(CNC(C3CN(C4CCOC4)C3)=O)C2)cn1 CC(C)(CC(=O)NC1CCC1NC(c1c[nH]nc1C(C)(F)F)=O)CC(F)F C=C(C)CC(C)C(=O)N1CCCC(CNC(=O)CCCOc2ccccc2F)C1 c1(C(N2CC(NC(CCCSC)=O)C(CO)CC2)=O)c(O)ccc2ccccc12 C1(C(C)(C)C)CC(CNC(=O)CP(C)(C)=O)CN(C(c2cncn2C)=O)C1 c1(N2CCC2)cc(C2CC2)nc(Cl)n1.C1(CC(=O)NC)CCC(=O)N1C.CO N1(C(c2cccc(OC)c2)=O)CCCC(F)(NCC(=O)NCCC(F)(F)F)C1 c1(C(=O)NC2CCN(C(C3(F)C(C)OCC3)=O)CC2)c(C(F)(F)F)cc[nH]c1=N C(C(C)=CC(=O)NCC(N(C)CC(C1CC1C(C)C)=O)C1CC1)OC N1(C(c2c(CCC)n(C)nc2)=O)CC2CCN(C(c3cc(C)nn3CC)=O)C2C1 CCN=C(NCC12CC(C1)C(C(F)(F)F)O2)NCC(C)CC(C)C N1(C(C(C)NS(C)(=O)=O)=O)CCC(O)(C(C)NC(=O)C2=CCSC2)C1 c1(C)ccc(C#N)cc1.CCC(COC)(c1nnnn1C(C)(C)C)NC(C)(C)C C1(CNC(c2c(C)scc2)=O)CC2CCC1N(C(=O)CNC(=O)NC1CC1)C2 c1(C(N2CCC(O)(CC)C2)C(=O)NC2COC2)cccc2sccc12 c1(C(=O)NC2C(NC(CCOCC)=O)CS(=O)(=O)C2)cc2n(n1)CCNS2(=O)=O C1(CC(=O)NCC#CCNC(C(c2ccnn2C)C)=O)CCCCC1C C(=O)C(C)(COC)CC.CCCC(CNC(=O)C(C)CC)OC C(c1ccncc1)=CC(=O)NC(CC(=O)NCC1(C)CN(C)C1)C1CC1 c1(C(=O)NCC2N(C(COC(C)C)=O)CC2)ccc2c(c1)Cc1ccccc1-2 C(=O)(CS(=O)(=O)C1CCCC1)NCCCNC(C1CCN(OC)CC1)=O Cc1cn(CC(=O)NC2CCN(C(c3cnc(S)nc3)=O)C2C)c2ccccc12 c1(C(=O)NCC(CN(C)C(C2CCCC2O)=O)O)cncnc1-c1ccccc1 C1(NC(c2c(CN(C)C)ccs2)=O)CCN(C(=O)C(=Cc2c[nH]cn2)F)C1(C)C C(=O)(C1=CCC(C)CC1)N1C(C(C)NC(C=CCN(CC)CC)=O)CCC1 c1(C(N(CC(C)(C)C)C2(NC(=O)CCCn3cccc3)CC2)=O)c[nH]nc1C(C)C c1(OC)cc(C(=O)NCCn2cc(CNC(C3SCCC3C)=O)nn2)ccc1F Cc1c(N(CC(=O)NC2(C#N)CCOC2)C2CCC2)cccc1Cl N1(C(=O)OC(C)(C)C)CCC(NC(=O)CC2CC2(C)C)C(C)(C)C1 CCCC(Cl)C(=O)N1CCC(O)(CNC(c2ccc(C(F)(F)F)cc2)=O)C1 C1(S(C)(=O)=O)(C(=O)NC2CC(C)(NC(C(CC=C)C)=O)C2)CCC1 Nc1nc(C(=O)NC2(CO)CN(C(=O)CC3CCC4(CCC4)O3)C2)ccc1O N1(C(C2CCC(C)(C)C2)=O)CC2(CC(C(=O)NCC=C(Cl)Cl)CO2)C1 c1(C(=O)NCCOCCN(C(c2nc(CC)oc2)=O)C)cc(O)ncc1Br Cc1ccnc(C(=O)NC2CCC2CNC(c2c(C)c[nH]c2CC(N)=O)=O)n1 c1(C(N2CC(C)C(NC(C3(c4cccnc4)CCC3)=O)C2)=O)cnc2n1CCC2 C1(CC(=O)NCC(CC)(CC)NC(C(CC)F)=O)CCCCC1(F)F Cc1cc(F)c(NC(=O)C(=O)NCC(C)CSc2ccccc2)c(I)c1 CCC1=NOC(CC(N2CC=CCC2C(N2CCC2C(=O)OCC)=O)=O)C1 C1(C#N)(NC(C2N(C(C3(OC)CCC(C)C3)=O)CC2)=O)CCOCC1 Cc1c(NC(C2CC2c2cccnc2)=O)n[nH]c1C1CC1 C1(C(=O)Nc2c(C)c(F)ccc2)COC2(CCN(C(=O)C(C)n3cccn3)CC2)C1 C(=O)(CC1=NN(C)C(=O)C1)NC1C(C=C)CN(C(C2(c3cccnc3)CC2)=O)C1 CC#CCCC(=O)N(C)CC1CCCN(C(=O)Cn2ncc(Br)n2)C1 C#CCCCCCCC(=O)N1CC(OCC(=O)NCCCC(C)CO)C1 C1(NC(C2(N(C)C)CCCC2)=O)CCN(C(=O)CC2CCSCC2)C(C2CC2)C1 C1(CC(=O)NC2(C)CN(C(CC=CC=C)=O)C2)(CO)CC2CCC1C2 Cc1ccc(F)nc1CNC(N1CC2(CC2)CC1C)=O N1(C(c2c(C)scn2)=O)CCC(CNC(c2c[nH]c3ccncc23)=O)C(F)(F)C1 C(=O)(CS(=O)(=O)CC(C)C)N1CCC(OCCNC(c2n[nH]c(C)c2C)=O)C1 Cc1csc2c(N3CCC(C(=O)NCC(=O)NC4CCCC45CC5)C3)ncnc12 C1(C(=O)NCC=CC)CCN2CCC1c1ncc(cn1)C2.c1(C)ccccc1.NC Cc1cc(C)c(C(N2CCC(NC(c3nncn3C)=O)C(F)C2)=O)c(=O)o1 C(=O)(C(O)C(F)(F)F)N1CCCC(CN(C(=O)C(=O)NCC(F)F)C)C1 N1(C(=O)CSc2cccnc2Cl)CC(NC(=O)C(O)Cc2cnc[nH]2)C2(CC2)C1 c1(OC)ccccc1C(N1CCC(CO)(NC(C2CC2(Cl)Cl)=O)C1)=O N1(C(C=CC)=O)CCC2(CC1)CCN(C(=O)C(c1ccn(C)n1)C)C2 N1(C(CNC(CCCC)=O)=O)CCN(C(c2csc(CC)n2)=O)CC1C1CCC1 Cc1nc(N)cnc1C(=O)NCC1CCCCN1C(c1cc(C(C)C)n(C)n1)=O c1(SC)cc(C(N2CC3(CCN(C(C4(N(C)C)CC4)=O)C3)C2)=O)c(Cl)cc1Cl CCC(CC(=O)NCCN1CCN(C(C2CCCCN(C)C2=O)=O)CC1)C(C)C N1(C(C2CN(C(C(CCC)OCC)=O)CC23CC3)=O)CCN2CCCCC1C2 CC1(C)CC(CNC(c2ccsn2)=O)CN1C(c1coc(O)n1)=O Cc1ccc(C(N2CCCC2C2CCN(C(c3csc(Cl)c3)=O)C2)=O)nc1 C1(CC(N2CCC(N(CCO)C(C3(C4CCC4)CC3)=O)C2)=O)CCC2(CC1)CC2 c1(C(=O)NCC2CC(C)N(C(c3n[nH]c4c3CCC4)=O)C2)ncsc1S(N)(=O)=O n1(CCCCC)nc(-c2cccc(OC(C)C)n2)nc1C1CCCS1 c1(CC(C(=O)NC(C(C)C)C2CCC2)NC(c2c(C)scn2)=O)cnn(C)c1O C1(C(CNC(=O)Nc2ccc(C3CCOCC3)cc2)O)CCC(F)(F)CC1 CN1N=CC(CC(=O)N(CC(C)(C)C(=O)NC2CC(C)(O)C2)C2CC2)C1=O C(=O)(CCCCCNC(=O)Nc1cc(C)ccc1C)NCC1(C)N(C(C)=O)CC1 C1(NC(CCC=CC)=O)CS(=O)(=O)CC1NC(=O)CCC(c1cccc(Cl)c1)=O c1(C2CC(=O)N2)cccc(COC(N2CCCC2C(=O)NC2CC2)=O)c1 c1(N(CC(=O)NCCNC(CS(CC)(=O)=O)=O)C)ncnc2[nH]cnc12 Cc1cc(Cl)ccc1C(=O)NC1CN(C(c2cc(Cl)on2)=O)CCC1C c1(C(=O)NC2CCN(C(C3C(CN(C)C)C3)=O)C2)cccc2c1OCC2 C(CNC(C1CCCC(O)C1)=O)(C(C)(C)C)NC(c1[nH]cc(C(C)=O)c1)=O C(=O)(CN=c1[nH]c(=NCc2cnc3ccccn23)[nH]c2c1CCC2)N(C)C C(=O)(C1CCCc2nncn21)N(C)CC1CN(C(=O)CCn2cnnn2)CCO1 c1(-c2cn(CCN(C(=O)CC3=CCCC3)CC)nn2)ccc(F)cc1Cl.C1CC1 CON1CCC(C(N2CCC(O)(CN(C(=O)C=CC3CCCC3)C)C2)=O)CC1 Cc1cc(C=CC(=O)NC(C)CN(C)C(C2CCC3(CC2)CC3)=O)c[nH]c1=N c1(OC)cc(=O)n(C)cc1C(=O)NCC1CN(C(=O)CC(C)C(F)F)CC1(F)F N1(C(c2c(NC(C)=O)c[nH]c2C)=O)CC2CN(C(=O)CC(C)(C)O)CC2(C)C1 C(C)(C)(CC(=O)NCc1nc(CNC(=O)CC2CNC(=O)O2)cs1)OC c1(OC)cc(C(=O)NCCC2CCN(C(c3ccc(C(N)=O)s3)=O)C2)sn1 C1(NC(CC2C(OC)CC2)=O)CC2CCC(C1)N2C(=O)CSc1cccc(C)c1 CC(O)CCCCCC(=O)N1CC2CCC2(NC(c2ccc3cncn3c2)=O)C1 c1(OC)ccc(F)c(C(N2CC3CC2C3NC(=O)C(N2CCC(C)C2)=O)=O)c1 C1(C(=O)NC2CC(CCNC(c3n[nH]c(=N)s3)=O)C2)CCCOC1C(F)(F)F C12(CNC(=O)Cn3cc(Cl)cn3)CCCC1N(C(c1cc[nH]c1)=O)CCC2 Cc1cccnc1C(N1CCOC(CCC#N)C1)=O c1(OC)cc(C)c(C(N2CC(NC(c3ccc4n[nH]cc4n3)=O)C2)=O)cc1Br C=C(C)CC(C(=O)NCC(C)(C)OCCO)NC(=O)C(F)CCC c1(OC)cc(Cl)ccc1CCNC(=O)C(=O)NC(C)CC1CCCOC1 C1(Nc2c(CCOC)cccc2)CCC2CN(C)CC12 Cc1ccc(C(=O)NCCOC2CCN(C(C3CC(=O)CO3)=O)C2)n1C c1(C(=O)NCCN(C(CC=C)=O)CCCN(C)C)cc(Cl)cc([N+](=O)[O-])c1O c1(N2CCC(=CC(C)(C)NC(=O)CC3CC(F)(F)C3)CC2)nc(C#N)ncc1Cl C1(NC(C(CC)C2CCOCC2)=O)CC2CC(C1)N(C(=O)CCS(C)=O)C2 Cc1cc(C#N)cnc1C(N1CCC(C2CCCN2C(c2ccoc2)=O)CC1)=O N1(C(c2cnc(OC)nc2)=O)CCCC(C)C1CNC(=O)CC(C)(C)O CC(CS(C)=O)C(=O)NCCC1(NC(=O)CCOCc2ccccc2)CC1 Cc1nc(CC(C)C)sc1C(=O)NC1CCN(c2ncc(C(F)F)cn2)C1C c1(C(=O)NCC2CCC(F)(CNC(C3(C)CCC(=O)C3)=O)C2)cnn2c1CCC2 c1(COCCCNC(C(=O)NCC#CCOC)=O)ccccc1 c1(CC(C)C)cccc(C(c2nnnn2C)NCCOCF)c1F c1(C(N2C(CNC(c3c(C(=O)OCC)cco3)=O)CC2)=O)ccc2c[nH]nc2c1 N1(C(CC2N(CC)CCC2)=O)CCCC(NC(=O)CCS(=O)(=O)N(C)C)CCC1 CN1C(=O)CCC1CC(N1CC2CC1(C(=O)Nc1cnn(C)c1Cl)C2)=O C(CC(C)CCCC(C)C)OC(c1c(SCC)cc(Cl)cc1)=O C(C(CC(C)C)C(=O)NCC12CC(C)(CCO1)C2)NC(C(C)=C1CCCC1)=O C1(CC(=O)N(CCC(C)NC(=O)Cc2cccc(Cl)c2)C)CCCCCO1 C12(NC(CC=C)=O)CCCC1(F)CN(C(c1cc(OC)cc(OC)c1N)=O)C2 Cc1occc1CC(=O)NC1CCN(C(=O)C(C2CCOCC2)F)C1 c1(OCC(=O)NCC2C(P(C)(C)=O)CCC2)ccc2cnccc2c1 c1(C(=O)NC(CC)CNC(c2cscc2Cl)=O)cc(Cl)sc1Cl Cc1c(F)cc(C(N2CCC(NC(=O)C(O)C(F)F)C(F)C2)=O)c(F)c1N C1(C(=O)NCCc2c(C)nc[nH]2)CSCCN1C(=O)C(C)n1cnnn1 N1(C(C(C)OCC2CC2)=O)CCC(O)(CCNC(C2(N=[N+]=[N-])CC2)=O)C1 C1(C(=O)NC(C2CCCN2Cc2n(CCCC)ccn2)(C)C)CC(F)C(=O)N1 c1(C(=O)NC2CN(C(CCN(CC)CC)=O)C(C)CC2)c[nH]c(=N)c2[nH]ccc12 N1(C(c2ccc(CN(C)C)cc2)=O)CCC2(NC(=O)CCCCC#N)CC2C1 c1(C(=O)NCc2ccc(N(CCCC)C)cc2)cc(C)c(CC)nc1O C(=O)(C1CCCn2ccnc21)N1C(CN(C)C(c2coc(CO)c2)=O)CCCC1 c1(C(=O)NCCCCC(C)NC(C2CC(C)(C)CO2)=O)ncnc2c1CCC2 N1(C(COC)=O)CCOC(CCCNC(=O)C(C)(C(C)C)C2CCCCC2)C1 c1(C(=O)NCC2CN(C(c3cc(=O)cc[nH]3)=O)CC2O)cccc([N+](=O)[O-])c1Cl C1(C(=O)NCCCCN(C)C(c2c[nH]c(C#N)c2)=O)C2CC2C2CC12 Cc1ccc(F)c(C(N2CCC(O)C(NC(C3CC3C(F)(F)F)=O)C2)=O)c1 c1(C(=O)NC2CN(C(C3(OC)CC3)=O)CC(C)C2)cc(OC)ccc1[N+](=O)[O-] C(CCC(C)C)(C(=O)N1CCNC(=O)CC1C)NC(c1cc(C)no1)=O C(CCC(O)C(=O)NCC(C)CN=[N+]=[N-])NC(c1c(CC)nn[nH]1)=O C(CC1=CCCCC1)N(C)C(C1CC(F)CN1CC(=O)NC1CCNC(=O)CC1)=O C(=O)(CCS(C)(=O)=O)N1CCC(C(=O)NC(c2ccn(C)n2)CC)C1C Cc1cnc2n1CCC(C(=O)NCC1(O)CN(C(C34CCCN(CC3)C4)=O)C1)C2 c1(C(=O)NCC(C)(CC)NC(CSCC)=O)cccc(Cl)c1Br C1(C)(CNC(c2c(CC)ocn2)=O)CCN(C(=O)CC(C)n2cc(Br)cn2)C1 N1(C(CC2N(C(C(C)OCCCC)=O)CCC2)=O)CCN(CC2CC2)CC1 C1(NC(CCN(C(CC)CC)C)=O)CN(C(c2cc(=O)cc[nH]2)=O)CC1C N1(C(C2(OCC)CCCOC2)=O)CCC(C(N(CC(COC)(C)C)C)=O)CC1 C1(C(=O)NCCN(C(=O)C(C)Cc2ccco2)CC)CC(O)(c2ccccc2)C1 c1(C(=O)NC(CNC(CC=C(C)C)=O)CC(F)(F)F)n[nH]c2c1CC(C)CC2 C#CC1CCN1C(C1C=CCN1C(=O)COCCSC(C)C)=O c1(NC)cnc(C(=O)N(CC(=O)N(C2CCC2)CCO)CC(C)C)cn1 N1(C(C2C(CCC)C2)=O)CC(NC(c2ccc(-c3cc[nH]n3)cc2)=O)CCC1C Cc1noc(C)c1CC(C)NS(=O)(=O)CCCC1CCC1 c1(CCCC)noc(CCC(=O)N(C2CCN(C(=O)CCN(C(N)=O)CC)C2)C)n1 N1(C(C(C(CC)CC)C)=O)CC(C)CN(C(=O)CSc2ccc(C)c(C)c2)CC1C C1(C)(C(NOCC(=O)N(C)CC2CCN(CC)C2)=O)CNC(=O)N1 c1(C(=O)NCC2CCN(c3snc(CCC)n3)C2)ccc2c(c1)N(C)CC2 C1(CCCCNC(C=C(CC)C)=O)CCN(C(c2cnn(C3CC3)c2C)=O)CC1 C1(C(N2C(C(C)NC(c3nn(C)cc3C(C)=O)=O)CCC2)=O)CC12CC(F)(F)C2 c1(C(N2CCC(C(N(CC(=O)N(C)C)CC)=O)C2)=O)cnc(O)c(C)c1 c1(C(=O)NC2CCN(C(c3c(CC)c[nH]c3)=O)CC2CC)cc(C)c(F)cc1Cl c1(C(=O)NC(C(C)NC(Cn2ccc(C)n2)=O)C)ccc2cccc(O)c2c1 N1(C(C2(C)CC2)=O)CC2CC1C2NC(c1cccc(CN2CCCCC2=O)c1)=O C(=O)(C(C)(C)CNC(=O)Cc1ccns1)NC(c1ccsc1)C C(=O)(C(C)(C)C)N(C1CC(CCNC(CSCCCC)=O)C1)CC c1(C(N2C(C)(CC)CC(NC(=O)CCC3CCC3)C2)=O)cc(=O)c(OC)cn1C C1(NC(C(CC)C)=O)C(C)(C)CN(C(c2cc(Cl)c(F)c(Cl)c2)=O)CC1(C)C c1(C(=O)NCC2CC(NC(c3cc[nH]c3)=O)C2)cnn(Cc2ccccc2)c1 N1(C(N)=O)CCCC(NC(C2CCC2CNC(=O)CCCC2CCCO2)=O)C1 C1(NC(CCOCCC)=O)CC2CC1CN(C(=O)CCc1c(C)noc1Cl)C2 c1(OC(C)C)cccc(CNC(C)C(=O)NC2CCC(C)C2)c1 C1(C(=O)NC(CCOC)C(C)C)CC12CCN(C(=O)C1=CC3C=CC1C3)CC2 c1(C(N2CCN(CC3CN(C(CC(C)F)=O)C3)CC2)=O)cc(C2CC2)nc(O)c1 N1(C(C(CC)Oc2ccccc2)=O)CCCCC1CNC(C)=O C12(NC(=O)C=Cc3cc[nH]n3)CC1CN(C(=O)CCOc1ccccc1O)C2 CCCC(C)CCCC(=O)N1CCC(O)(CCNC(=O)C2=CCOCC2)C1 C(CC1=CCN(C(=O)CC23CC(C2)C3)CC1)NC(c1c(C)n(C(C)C)cc1)=O N1(C(=O)CCC2CC2(F)F)C(=O)CN(CC23CCC(CC2)CO3)C1=O CC1=C(C(=O)NC(C)CCNC(C2CC3(CCC3)CO2)=O)C=C2CCCN=C2N1 C1(C(=O)Nc2cn(CC(C)C)nc2)CC2(CCN(C(=O)C(F)C(C)(F)F)C2)C1 C1(N(c2cccc(C(C)(C)C)c2)C(c2cc(OC)nn2C)=O)CCNCC12CC2 N1(C(C2CC(SC)C2)=O)CC(CC(=O)NCCC(C)(O)C2CC2)C2(CC2)C1 C=C(Cl)CC1C(=O)N1.c1(C(=O)NC2(CF)CCC2)cc2n(n1)CCO2 CC1CCN(C(c2cc[nH]c2)=O)CCN1C(=O)CCN1C(=O)NC(C)(C)C1=O C(=O)(C(=O)N(C)CCN(C(=O)CN(C(=O)Cn1cncn1)C)C)N(C)C C1(CNC(CNS(CC)(=O)=O)=O)CCN(C(c2cc3c(s2)CCC3)=O)C12CCC2 c1(C(=O)OC)cc(Br)c(NC(C23CC2CN(C(c2nccn2C)=O)C3)=O)c(I)c1 C(=O)(CC(=O)N(C)C)NC(C)CCNC(=O)CC1(CO)CC1.C(C)(C)(C)SCCS N1(C(C=C(C)C)=O)CCC2(CC1)CC(C)N(C(c1ncoc1C)=O)C2 N1(C(C2N(CC(C)C)CCC2)=O)CCC(N(C)C(c2cc(O)nn2C)=O)C(C)C1 Cc1nc2nccc(N3CC(CO)(NC(c4cc(C)oc4C)=O)C3)n2n1 C(CC(C(C)(C)C)NC(=O)COC1CCC(C)CC1)N(C(c1cnc(C)s1)=O)C C1(NC(C2(OC)CCOCC2)=O)CC2CN(C(=O)Cc3ccon3)CC12 S(=O)(=O)(c1ccc(OC)c(C(=O)O)c1)N(C(COCCC)=O)C(C)C N1(C(CC(=O)NCC)=O)CCC2(CCCN2C(C2CCC(C(=O)OCC)C2)=O)C1 Cc1ccc2cc(C(=O)N(C3CCC(NC(=O)CNC(=O)C4CC4)C3)C)ccc2c1 N1(N2C(C3C(NC(=O)C(C)(C)CN)C3(F)F)CCC2)CC=CC(OC(C)C)C1.CC=O C(=O)(C(=O)N=S(C)(C)=O)N1C(CN(C(C(c2ccc(O)cc2)C)=O)C)COCC1 c1(N2CCC(SCC)C2)ccncc1S(=O)(=O)NC(c1ccc(F)c(C)c1)C C1(CC(=O)NCC(CC)NC(c2c(C)nn(C)c2F)=O)CCCC(C)(C)C1 c1(C(=O)NCC(CC(=O)N(C(C)CS(C)=O)C)(C)C)cncc2[nH]ccc12 Cc1ccc(Br)nc1C(N1CCN(C2CSC2)CC1)C(=O)NCC1CCOC1 c1(CC(=O)N(C2CCN(C(c3cn(CC)nn3)=O)CC2)CCC)cccc(Cl)c1 C1(NC(=O)C(C2CCOCC2)O)CC2CCC1CC2NC(=O)C(O)C1CCC1 C(=O)(C(CC(C)(C)C)NC(C1(O)CCCCC1)=O)NC(CC)Cn1cncn1 C1(C(=O)NC2C(n3ncc(C)c3)C2)C2CCC(C2)C1NC(=O)C=CCF.C(C)(C)(C)O N(C1CC2CCCc3cccc1c32)C(CO)Cc1ccc([N+](=O)[O-])c(F)c1 CCCCC(C)(CO)NC(C1CC2C=CC1O2)=O.c12ccc(cn1)CNC2=O C1(C)(C(=O)NCC2CC(NC(C3(COC)CCC3)=O)C2)C=CCCC1 c1(C(N2CC(N(C)C(C34CC3CCC4(F)F)=O)C2)=O)nccc2[nH]ccc12 C1(CC(N2CC(CCC)(C(=O)N(C)CCOC(C)=O)C2)=O)CCCCN1C C1(C2CC2)(NC(CN(C)C(C2C=CCS2)=O)=O)CCOC1 N1(C(c2cn(CCC)nc2C)C(=O)NCc2nnn(C)n2)CCC2(CCSC2)C1 C1(C(=O)NC(C)CC2CN(C(C3CCOC3(C)C)=O)C2)CCC(=O)NC1 c1(C(N2CCC(CNC(CC(C)(C)OC)=O)C2(C)C)=O)ccc(S(C)(=O)=O)o1 c1(OC)ccnc(CN2CC(c3cccc(C)c3)(O)C2)n1 N1(C(C=C(CCC)C)=O)CCCCC1CN(C(=O)CCc1ccon1)C CC(=O)CCN=C(NCC1CC1)NC1CCC(c2nc(C)no2)CC1 C1(CNC(C(CC)COC)=O)CN(C)CCN1C(=O)C(c1ccc(C)o1)C N1(C(C=CC(C)C)=O)CCC2(CNC(=O)C(F)(F)c3nccs3)CCCC12 c1(C(=O)Nc2ccc(F)nc2Sc2ccncc2)nc2ccccc2[nH]1 C(=O)(C(=O)C(C)CC)N1CCC(CC=C)(C(=O)NC(c2ccnc(F)c2)C)C1 C1(CNC(C2CC(=C(F)F)C2)=O)CCCCN1C(C1CCC(F)(F)C1)=O n1(CC(=O)NCC(=CC(=O)N(C(C2CCC2)C)CC)C)nnc(C)n1 C1(NC(C=C(C)Cl)=O)CC2CN(C(=O)C=Cc3ccncn3)CC12 Cc1cncc(C=CC(=O)NC2CN(C(=O)CC(C)c3ccncc3)CC2C)c1 C1(CC(=O)NCc2c(C)scc2)CC(NC(=O)CCNC2CCOCC2)C(O)C1 c1(OC)cccc2cc(C(=O)N(C3CCCCNC3=O)C)c(=O)oc12 Cc1cc(=O)n(C)cc1NC(C1CCN1C(C1CN2CCC1C2)=O)=O CS(=O)(=O)CCCC(=O)N1CC2CC1C2NC(=O)CCC1CC1 c1(C(=O)NC2CN(C(=O)NC3CC3)C2)c(Cl)oc2ccccc12 c1(C(=O)NC(CC#C)C(=O)NCCCN2CCOCC2)ccnc(C)c1N N1(C(C(C=C)O)=O)CC(C2CCCN(C(=O)C=Cc3nnn(C)n3)C2)C1 C1(NC(c2cn(C)c(=O)cc2)=O)CCN(C(C2CC2C2CCCC2)=O)C12CCC2 C12(NC(C(C)NC(C3CCN(CC)C3)=O)=O)CC(CO)(C1)OC2(C)C Nc1cccc(C(=O)NC2CC(CCNC(=O)C(F)(F)c3ccccc3)C2)n1 N1(C(CC=CC)=O)CC2CC2(C(=O)NC(C)Cc2nc[nH]n2)C1 CCC(C)(C)C(C)CC(=O)N1CC2(C1)CN(C(c1cc(C3(Cl)CC3)n(C)n1)=O)C2 C#CC1CCCC(NC(=O)CCC2CCN(C(c3ncnc(O)c3F)=O)CC2)C1 C1(N(C)CC23CC(C#N)(C2)C3)CN(C(=O)CCCc2ccccc2)CC1(F)F CC(C)(Cc1cnn[nH]1)C(=O)NC1(CNC(=O)CNC(c2cccnc2)=O)CCC1 c1(NC(C)=O)cncc(C(N2CCC(NC(c3ccc(F)nc3)=O)C2CO)=O)c1 c1(C(N(CCNC(c2ncc(C#N)cc2F)=O)C2CC2)=O)cnc2ccccc2n1 N1(C(CCC(C)OCC)=O)CCC(CNC(c2cc(C)c(Br)o2)=O)C(C)C1 c1(C(=O)NCC2C(NC(CCc3ccn(C)c3)=O)C2)c(C2CC2)cccc1F c1(C(=O)OC)cncc(C(=O)NC2CC(NC(c3cn(CCOC)nn3)=O)C2)c1 Cn1nnc(C=CC(=O)NCC2CCCN2C(c2ccc(F)cn2)=O)n1 c1(C(C(=O)NCCN2CCN(C(C(C)NC(C)=O)=O)CC2)C)ccc(F)cc1F c1(C(=O)NCC(CNC(Cc2c(C)nc[nH]2)=O)C)ccc(CO)cn1 Cc1c(F)ccc(-c2cn(C(C)CNC(=O)C(C)(C)Cc3cnn[nH]3)nn2)c1F CC(CC(=O)NCC1COCC1NC(c1ccc(NC(C)C)nc1)=O)P(C)(C)=O C(=O)(C(F)(F)CNC(C1(NC(C2C=CCCC2)=O)CCCCC1)=O)OC c1(C(N2CC3CCN(C(=O)C=CC4CCCCC4)C3C2)=O)ccn2c(O)nnc2c1 N1(CC=C)CCC2(CCCN(C(C3CNC(=O)CC3(C)C)=O)C2)C1 C1(NC(C(C)Cn2cccn2)=O)CCCC(NC(=O)COCc2ccccc2)C1 CC(C)CCN=C(NCc1ccc(C(C)(F)F)cc1)NCC1CN(C(C)C)CCO1 N1(CCCC(N2CCC(C(C)NC(c3ccc[nH]3)=O)C2)=O)C(=O)CCC1=O C(=O)(C1=CCC(C)CC1)NCC1OCCCN(C(C2(COC)CC2)=O)C1 CC1CCC(CNC(=O)CCCNC(N)=O)N(C(=O)CCc2ccccn2)C1 C1(CNC(Cc2c(C)ocn2)=O)(NC(C2(CCF)CCCCC2)=O)CCOCC1 N1(C(C(C)NC(C)=O)=O)CCC(CNC(=O)CN2CC(=O)N(C)C2=O)C(C)C1 CC1CCC2(CC1)CCN2C(c1occc1CNC(c1cnc(O)c(F)c1)=O)=O c1(CN2C(C(=O)Nc3ncc(F)cc3Br)CC(O)CC2)ccc(Br)cc1[N+](=O)[O-] c1(OC)ccc(C(=O)NC2COCC2NC(C2(F)CCCCCC2)=O)cc1C N1(C(C2CCN(C(C3(C)C(C)C3)=O)CC2O)=O)CCC2(CC1)COC(=O)N2 Cc1cc(C#N)cc(C(=O)NC2CC3CC(C2)N(C(c2ccc(=O)oc2)=O)C3)n1 CC1C(NC(=O)CCc2ccncc2)CC2CCC1N2C(c1ccnc(Cl)c1)=O c1(C(N2CC=CC(NC(CC(CC)OC)=O)C2)=O)ccc2ncc(OC)nc2c1 c1(NC(C)=O)ccccc1CC(=O)NC1CN(C(C2CCOC(=O)N2)=O)CC1O N1(C(C#CC(C)(C)C)=O)CC2(C1)CN(C(=O)Cc1cccc(F)c1F)CCO2 CC1(O)CCCN(C(=O)C2=CCN(C(c3ncccc3O)=O)C2)CC1 c1(C(=O)NCC(C)(C)NC(c2ccc(COC)o2)=O)cnc2n1CCCC2 c1(NC(=O)NC2C(NC(C(c3cccnc3)C)=O)C2)cc2scc(Cl)c2[nH]1 N1(C(C2(Oc3ccccc3)CC2)=O)CCC(O)C(c2ccccc2)C1 N1(CC(=O)NC(CC)CNC(=O)CC2CCCC2C)Cc2ccccc2C1 C1(CNC(c2ccc(O)cc2)=O)CCCCCN1C(c1ccsn1)=O n1(CCNC(C2CN(C)C(=O)N2)=O)cc(S(C)(=O)=O)cn1 Cc1ccccc1C(C)CC(=O)NC1CCN1CC(O)COCc1cccnc1 c1(NC(C(C)OC(C2(CC)CCCCO2)=O)=O)cccc(Cl)c1C c1(CCC)nc(C(=O)N(CCN(C)C(C2CCCN2C(=O)NC)=O)C(C)C)co1 CCCCC(O)C(=O)N1CCCC(N(C)C(c2ccc(O)cc2F)=O)CC1 C1(CN(C(=O)Cc2ccccc2)CCNC(C(C)SC)=O)CCCC1(F)F c1(SC(C)(O)C(=O)NCCNC(c2csc(-c3ncc[nH]3)n2)=O)ccnc(O)c1 N1(C(C2C(OCC)C2C)=O)CCC(CO)C(NC(c2ncccc2Cl)=O)C1 c1(C(N2CCC(NCc3nn(CC)nc3C)C2)=O)nc[nH]c2nccc1-2 Cc1cc(C)c2nc(N3CCC(NC(c4ccnn4CCF)=O)C(F)C3)sc2c1 CC(C)CC(C)(C)C(=O)N1CCC(C)C(NC(c2ccccn2)=O)C1 Cc1cccc(NC(C23CC(CN2C(=O)Cc2cccnc2)C3)=O)c1C c1(NCC2C(OC)CC(OC)CC2)ccc2c(c1)CCCC2=O Cc1cc(C(N2CCOC(CC(=O)NC3CC3c3ccn(C)n3)C2)=O)ccn1 C1(C(=O)N(C2CC(NC(C3CCOCC3)=O)C2)C)(CC)CCOC1 N1(C(C(CCCC)NC(=O)CC2CCC(C)(C)O2)=O)CCCC2NC(=O)CC12 C(c1ccccc1[N+](=O)[O-])=CCN1CCC(F)(CNC(=O)CC2CCCCC2)C1 N1(C(c2ncc(N)nc2)=O)CCOCC(CNC(C2CC2C(N)=O)=O)C1 c1(C(C(=O)NC(CN(C(C2CC3(CC3)C2)=O)CC)C)C)ccc(C)s1 C(C(CC(C)C)NC(=O)CCN1CCCCC1)NC(CCc1cc(C)on1)=O c1(C(CC(=O)N(C2(C(=O)OC)CCC2)C)N)ccc(F)c(F)c1 CC(C)C(CNC(C1(Br)CC1)=O)NC(=O)COc1cn[nH]c1 O(NC(=O)C(CCSC)NC(c1cc(C)c(C)o1)=O)CCCC#C C1(CC)CCC(C(N2CCC(CNC(=O)CCCC3CCCCC3)C2)=O)O1 c1(OC)cccc(CNC(C2C(N)C3CCCCC23)=O)c1Br Cc1cnc(C(=O)NCC2C3CC2N(C(c2ccc(C4CC4)cn2)=O)C3)c(F)c1 Cc1cccc(CC(=O)NCC(CC(C)C)NC(c2ccc(F)cc2)=O)c1 N1(c2cc(OCC)nc(C)n2)CCC(C2CCCN(C(=O)C(C)C3CC3)C2)CC1 c1(C(=O)NC2CN(Cc3cccc(Cl)c3)CC2F)ccc2cccc(Cl)c2n1 CC(C)C(CNC(C1(CO)CCCO1)=O)N=c1nc(Cl)[nH]c(C)c1F CC1CN(C)C(C)CN1C(C1CN(CCF)CCC1(F)F)=O C1(NC(CCc2c(C)nn(-c3ccccc3)c2Cl)=O)COC2(CCCC2)C(C)C1 c1(OCC(=O)NC(C)(CNC(=O)CC2COCCO2)C2CC2)ccc(C#N)cc1Cl n1(CC=C)nnnc1C(C1CCCC1O)NCC1(CC)CC1 C12(NC(COC)=O)CC3CCC(C1C2)N3C(c1nn(CC(F)F)cc1[N+](=O)[O-])=O c1(C(C(N2CC(N(C(CC3(OC)CCC3)=O)C)C2)=O)O)ccc(Br)cc1F C(=O)(C(C)C(O)C(C)C)NC(CCNC(CC1(C=C)CCC1)=O)(C)C N1(C(=O)OC(C)(C)C)CC2CCCC2(NC(C2COCC2(C)C)=O)C1 c1(C(C(=O)NC(CNC(CC2CC(=C)C2)=O)(C)Cn2cccn2)C)ccc(C)cc1 C1(NCC(CN2CCN(C)CC2)O)CCC2(CCOCC2)CN1 N1(C(Cc2ccc(C)s2)=O)CC(C)(CNC(=O)Cc2cc(C)n(C)n2)CC1(C)C N1(C(C(C)(C)CO)=O)CC(N=c2ncc3ccccc3[nH]2)C(C)(C)C1 Cc1c(C(N2CC(C)(NC(=O)C3CCc4c[nH]nc43)C2)=O)[nH]c2c(C)cccc12 C(CC(=O)NCCCCC1CN(C(=O)COC2COC2)C1)NC(C1C(C)C1)=O CC(C)CCCCCC(=O)NCCC(N1CCCC1CN=[N+]=[N-])=O c1(C(N(C2CCN(C(=O)C(C3CCC(O)CC3)(C)C)C2)C)=O)cc(O)cc(F)c1F Cc1ccncc1CC(=O)NCC(CO)NC(c1cn(CC(F)F)cn1)=O C1(C(N(CCCCN(C)C)C)=O)(NC(C2COCOC2)=O)CCSC1 N1(C(C(CC(C)(C)C)O)=O)CCC2CN(C(=O)C(Cl)=CCl)CC2C1 C1(CNC(C2(CC#C)CC=CCC2)=O)CC2CCC1N(C(=O)C=C(C)C)C2 CC1CCC(C(F)(F)F)N(N(CCN2CCOC2=O)CCN(C)C)C1 c1(C(N(CC(=O)NCCCOC)CC)=O)cc2c(=O)n(C)c(=O)n(C)c2s1 N1(c2n(CCC#C)c(-c3cccn3C)nn2)Cc2ncnc(O)c2C1 CON(CCC(=O)N1CCN(C)C(=O)C1)C(=O)COCCCN1CCC1 Cc1ccc2[nH]c(C)c(CC(=O)NCC3(F)CN(C(=O)C(O)C(F)F)C3)c2c1 N1(C(C(CC=CCC)C)=O)CCCC2C(NC(c3cc(C)sc3N)=O)C(C)(C)C12 C=CCC(C(=O)OC)NC(=O)C(COCC)NC(c1ccncc1O)=O C(=O)(C(O)CC(C)(C)C)N1CC(CC(C)NC(=O)CCNC(=O)C(C)(C)C)C1 N1(C(C(C)C2(O)CCC2)=O)CCC=C(C(=O)Nn2nnc3ccccc23)C1 c1(C(N2C(CNC(c3n(C)nc(CC)c3Cl)=O)CCC2)=O)coc2c1CCCC2 C12(C(N(CC(CC)NC(c3cc(C(N)=O)no3)=O)C)=O)CCC(C)(C1)OC2 n1(CC2(CC)CC2)cc(C2CCCN2C(=O)CC(C)C2CCCO2)nn1 c1(C(=O)NCC(C)NC(C2C(OCC)C2)=O)c[nH]c2cc(C)ccc12 N1(CC(=O)NC2CCC(C)N(C(=O)CCc3ncc[nH]3)C2)CCc2sccc2C1 CCCCS(=O)(=O)NCC(=O)NC(C)CN(C(=O)CCC1CCC(O)CC1)C N1(C(c2coc(Cl)c2)=O)CCN(C(=O)Cc2sc(O)nc2O)C(CCO)C1 c1(N(C(C(C)OC2CCN(Cc3cccc(C)n3)C2)=O)C)cccc(Cl)c1Cl.OCC C1(=CC(=O)NC2CNC2)N=C(c2ccncc2)OC1=O.c12cc3n(n1)CCCN2C3=O C(=O)(C(C)(O)CC(F)(F)F)N(CCCNC(C(C1CC1)OC)=O)C(C)C c1(C(N2C(CC(N3CCCC(C)(O)CC3)=O)CCC2)=O)cnc2c(Cl)cccn12 Nc1cc(C(=O)NCC=CCNC(C2CCSC2)=O)ccc1-n1cnnc1 Cc1cncc([N+](=O)[O-])c1N1CC2CC1CN2C(=O)Cc1ccc([N+](=O)[O-])cc1 N1(C(CC(C)C)=O)CC2CC1C2NC(=O)C(C)Oc1ccccc1F C(=O)(CC(C(F)(F)F)NC(c1ccc(F)c(O)c1)=O)NC(c1ncnn1C)C n1(CC(=O)NC2(C3CCN3C(c3cnc4n3CCS4)=O)CC2)cc(F)ccc1=O CC(F)(F)CCC(=O)N1CCN(C(c2cnn(CCF)c2)=O)C(C(F)F)C1 c1(C(N(CC(CC)NC(=O)C(C)OC(C)(C)C)C)=O)nnc(C)cc1O C(CO)(C(=O)NC(c1ccn(C)c1)C)NC(C(C)=C1CCC1)=O n1(CC(=O)NCC(CC)(CC)NC(=O)CSCC(C)C)ccc(=O)cc1C c12cc(ccn1)CNC2=O.c1(C(C(=O)N(CC(=O)OC)C)=O)ccc(O)cc1 c1(C(C(=O)NCC(C)N(C(c2nnc(CC)s2)=O)C)C2CC2)ccccc1OC N1(C(COCC(=O)OC(C)(C)C)=O)CCCC(CCNC(c2cc(F)cs2)=O)C1 N1(C(CCNC(C)=O)=O)CCc2cccc(NC(c3ccc(Br)c(Cl)c3)=O)c2C1 C1(C(=O)NCCN(C2CC2)Cc2cc(CC)c(C)s2)CC(C2CC2)=NO1 c1(C(=O)NC2CCCCN(C(c3cncc(C)c3C)=O)C2)cc2ccncc2[nH]1 C(c1cccc(Br)c1)=CC(=O)NC(CNC(C=COCC)=O)CO CC1(C)COC1C(=O)NC(CNC(c1occc1Br)=O)C1CC1 Cc1cc(C(N2CCC(OC(C)C)C2)C(=O)NC2CCC2)c(C)cc1O N1(C(C(=O)NC(CCSCC)C)=O)Cc2cccnc2OCC1.C1C(C(C)(C)C)N1 c1(C(=O)NC23CC(NC(CSC)=O)(C2)C3)ccc(Br)cc1O c1(C(=O)NC2C(CNC(CC=C(C)C)=O)CCC2)c(Br)cnn1C(C)C C(=O)(C#CC1CCCC1)NC1C=CC(CNC(c2cccc(C(C)C)c2N)=O)C1 C1(CNC(C2(C(C)(F)F)CC2)=O)CN(C(=O)COCCN(C)C)CCO1 c1(CC(=O)NC2(CNC(CNC=O)=O)CCC2)cnc(C2CC2)[nH]1 c1(C(=O)NC)cn(CCC2CCN2C(=O)C(=O)Nc2ncc[nH]2)c2ccccc12 C1(C(=O)NC(C2CCOC2)CNC(c2c(CC)n[nH]c2)=O)CCCCN1CC C1(OC)CN(C(c2cnc(C(C)C)o2)=O)CC1NC(C1(c2cc[nH]n2)CC1)=O N1(C(=O)CCc2cncnc2)CCC(C2CCCN(C(C3CC(O)C3)=O)C2)C1 Cc1ccc(CC(=O)NCC2CCCN(C(C34COCC3C4(F)F)=O)C2)cc1C C1(NC(C2CCN(C(N)=O)C2)=O)CCN(C(=O)C=Cc2ncc[nH]2)C12CC2 c1(C(N2CC(NC(CC(=C)C)=O)C(C)C2)=O)cn2c(n1)CC(C)CC2 C1(C2CC2)(CNC(C(C=C)(C)CC)=O)CCN(C(=O)COCC(C)C)C1 CC1CN(C(=O)CC(C)(C)C)CCN1C(=O)C(c1ccc(Cl)s1)C C1(NC(=O)NCC(c2ccc(O)cc2)O)CCCN(c2ccncc2)C1 C(C(CC)CC)(c1onc(CCC(=O)OCCCC)n1)N.c1ccccc1 N1(C(C(C(CC)CC)C)=O)CCC2CN(C(=O)CC(C)C(F)F)CCC2C1 CCC(C#N)(CC)C(=O)N1CCCC(CN(C(=O)CCc2ncccc2C)C)C1 c1(-n2c(-c3cnon3)nc(C(C)O)n2)ccc(S(=O)(=O)c2ccc(Br)cc2)cc1 Cc1ccc(NC(C2CC(F)CN2C(=O)CCc2ccccc2F)=O)c(C)c1C C1(C(N(CCC#C)CCOC)=O)N(C(=O)Cc2nc(=N)[nH][nH]2)CC12CCCC2 c1(OC)cccc(C(=O)NCC2CN(C(c3cn(C4CCC4O)nn3)=O)C2)c1N S(=O)(=O)(c1ccc(NCCCN2CCN(C)CC2)cc1Cl)N1CC(C)=C(C)C1 N1(C(CC(CC)(F)F)=O)CC2(CCC2)CC1C(=O)NC1CN(C)CC1C C(CCO)(C(F)(F)F)C(N1CCN(C2CCC2)CC1)=O.N12CCC(C1)CCC2=O c1(OC)ccc(Cl)cc1C=CC(=O)NCC(C)N(C)C(C1CCOC1)=O C(c1c(Cl)cccc1Cl)=CC(=O)O.C(CCCC(=O)O)=C(CC(=O)OC(C)(C)C)Br N1(C(COCc2c(C)cccc2)=O)CC(C)N(C(=O)CCc2ccc[nH]2)CC1C c1(C(=O)NC2CC(NC(c3ccc(C(O)C(F)(F)F)cc3)=O)C2)cc(=O)cc(Cl)[nH]1 C(CCc1cnccc1C)(C(=O)NC1CC(F)(F)C1)NC(CCCOC(C)=O)=O C1(NC(c2cnc(-c3ccsc3)s2)=O)CCC2CCN(C(=O)C3=CCCC3)C12 c1(C(=O)NCC23CC2CN(C(=O)C2=CCCS2)C3)cc2ccccn2n1 CC(C)(C)CC(O)C(=O)N1CC(F)(F)CC1C(=O)NC1CCNC1=O N1(C(c2cccc(OC)c2)=O)CCC2(NC(=O)CCC3CC3(C)C)CCCC12 Cc1nc(-n2cc(C(C)N(C(=O)CCc3cnoc3)C)nn2)sc1C C(=O)(C(C)(C)C(N)=O)NC(CCOC)CNC(=O)CC1CC1c1ccccc1 CC1(C)CC(CC(=O)NC2Cc3nccn3C2)N(C(=O)CC2CC3(CC3)CO2)C1 CC1(C(=O)NCC2CCN2C(=O)Cc2csc(Cl)n2)CCc2ccccc2O1 C1(C(=O)NCC(C(C)C)NC(=O)CN2CCCNC2=O)Cc2ccncc2N1 c1(C(=O)NC(CNC(C(CC#C)(C)C)=O)C2CCC2)ncnc2c1OCCO2 c1(CN(C(C2CC(=C3CC3)C2)=O)CC2CCN(C)C2)c[nH]c2cccnc12 C1(NC(C(C)(C)CCCNC(=O)CCc2cncs2)=O)CCc2nncn2C1 C(CNC(c1ccc(=N)[nH]c1)=O)(CC(=O)N(C)C(C1CCCC1)C)OC N1(C(c2cc(OC)c(O)nc2)=O)CC2CN(C(C34CCCC3OCC4)=O)CC2C1 C12(CNC(C(C)OCCC(C)C)=O)CCC(CC1)N2C(c1cc2c(s1)CCC2)=O C(CCC1(C)CC1)(C(=O)N1CCC(O)C1)NC(C(CC)C1CCC(=O)N1)=O C(=O)(CS(=O)(=O)CCO)NC(C1CCCCC1)CNC(c1n(CC)nnc1C)=O N1(C(c2nc(COC)oc2)=O)CCCC(NC(C2CCCC2Br)=O)C1 N1(C(C2=NOC(CNC(C3C=C(C)CS3)=O)C2)=O)CC2(C1)NC(=O)NC2=O c1(C(=O)NC(CCCC)CNC(=O)CCN2CCCS2(=O)=O)cc(O)ccc1C C1(CC=C)(NC(c2[nH]nnc2C2CC2)=O)CCN(C(c2nnc(C)s2)=O)C1 c1(C(N(C2CCCN(C(CCSC)=O)C2)C)=O)ccc(O)c(OC)c1 C1(C(=O)NC2C(CNC(c3ccncc3)=O)COC2)CCC2(CCOCC2)O1 c1(CC(N2CCC(C(C(=O)NCC(C)OCCO)C)C2)=O)cccc(F)c1 c1(CC(N2CCC(OCCNC(c3cn(CC)nc3C)=O)C2)=O)cc(F)ccc1F n1(CCN(CC)CC)nc(-c2cc[nH]n2)nc1C(C)Sc1nccn1C N1(C(COCCN(C)C)=O)CC(CO)C2(CCN(C(=O)Cc3cccs3)CC2)C1 C1(C#N)(C(=O)NC2CC3(CN(C(C(C)NS(C)(=O)=O)=O)C3)C2)CC2CCC1CC2 N1(C(C2(C#N)CC2)=O)CC(C(=O)NCCC2CCCC23CC3)C2(CCC2)C1 Cc1cc(=NCC(C)CNC(c2snc3ccccc23)=O)c(C#N)c[nH]1 N1(C(c2cc(COC)on2)=O)CC(C2CCN(C(=O)C(C)=C3CCCC3)CC2)C1 C1(CC(=O)NCC(C(=O)NCC(=C)F)C)CCC(=O)C1C c1(C(COCCO)N(C(C)=O)C(=O)NC(C)(C)C)cc(C)cc(Br)c1 Cc1[nH]nc(C(=O)NC2(C(N3CCCC34CC4)=O)CC2(C)C)c1Cl C1(CC#C)CCN(C(=O)C=C(C)C2CCN2C(=O)C(C)OCCOC)CC1 CCS(=O)(=O)CC(=O)N1CC=CC1C(=O)NCC1CCN(C(=O)C(C)C)CC1 C=Cn1nccc1C(C1CCN(C(=O)CC2CNCC23CC3)CC1)=O n1(CN)cc2c(n1)C(=O)C2.C1(OCC)CCN(C(C2CC2OC(C)=O)=O)C1 c1(CC)cnc(O)c(C(=O)NCCN(C(c2nc(=O)n(C)[nH]2)=O)C(C)C)c1 c1(CC(=O)NCC(C(C)(C)C)NC(C(C(C)O)N(C)C)=O)csc2nccn12 CC(C)CCN(CC(=O)NC1(CCC(=O)NC2CC2c2ccoc2)CCC1)CC C(=O)(C1=NN(C)C(=O)CC1)N(CC(=O)NC1CCCC(C=C)C1)CC1CC1 N1(C(Cc2nnc(C)s2)=O)C2CCC1CC(CC(C)NC(c1sncc1C)=O)C2 Cc1ncc(C(=O)NCC2C(C)CCN2C(c2cc(Cl)cs2)=O)c(C(C)C)n1 N1(C(CC(=O)NCC2CC2)=O)CC(NC(c2occc2Cl)=O)CC12CCC2 c1(N(C(=O)C(n2nccc2C)C)CC)ccc([N+](=O)[O-])cc1F N12CCC(C)C1SCC2=O.c1(SCC(=O)NCC(=O)NC)ccc(C)cc1 c1(C(=O)NC(C(C)C)CCN(C(=O)C(C)CN(C)C)C)ccnc2ccsc12 C(=O)(C(F)(F)C(O)C1CC1)NCC(C)(C)CNC(C1CCCC(C(C)(C)C)C1)=O N1(C(c2c(C)ncc(N)c2)=O)C2CCC1CC(N(C)C(C1CCCC(C)C1)=O)C2 c1(C(N2C(CNC(c3c(COC)cco3)=O)CCCC2)=O)cc2n(n1)CCCO2 Cn1ncc2cc(C(=O)NCC3C4CN(C(C5CC(C)(C)CO5)=O)CC34)cnc12 Cc1c(C(=O)NC2CCC2CNC(=O)CCCN(C)C)ccc(F)c1F c1(CCC(=O)N(CC(CNC(Cc2c(C)cco2)=O)C)C)ccccc1C#N C12(NC(CCOCC#C)=O)CCC(CNC(=O)C(C)CC(=O)OCC)(CC1)CC2 Cc1cc(C(N2CCC(C)(CNC(=O)CCC3CCOC3)C2)=O)nn1C1CC1 C1(C(C)C(=O)N(CCC(N)=O)C2CC2)CCN(C(=O)CCOC2CCC2)CC1 CC1CC(N=c2[nH]c(N3CCC(C(F)F)CC3)nc3c2CCCC3)CCO1 c1(COC)ncc(C(=O)NC2CCC2CNC(c2cc(C3CCC3)on2)=O)s1 c1(OC)ccc(CN2CCCC(NC(=O)CCC3CCC3)C2)c(Br)c1OC CCCCC(O)C(=O)N1CCCC(O)(CCNC(=O)C(F)=CC2CC2)C1 Cc1nc(O)nc(O)c1C(=O)NCC1CC(NC(=O)CCCn2cncn2)C1 N1(C(Cc2c(C)ocn2)=O)CCCC12CCN(C(C1C(C)(C)C1(F)F)=O)C2 C1(C2CC2)(CNC(CNC(CC)=O)=O)CCN(C(c2cc(CO)[nH]n2)=O)C1 N1(C(CC(CC)(F)F)=O)CCC2OCCN(C(c3cnc4[nH]nnc4c3)=O)C2C1 C1(CNC(=O)COc2ccsc2)C2CCCOC12.C(C1C(=O)N1)OC N1(C(c2ccc(-n3cc(C(c4cnc(Br)s4)=O)nn3)cc2)=O)CC2CCCC2(CO)C1 C(=O)(C(F)C(C)CNC(c1cnc(O)cc1C)=O)NCc1cn(CC)nc1 C(=O)(C(CC)CCOC)N(CC(=O)NCC(CC)OC)C1CC1 CN1C(=O)OCC1NC(=O)NCCCCCCn1cc(-c2cncc(F)c2)nn1 C1(CNC(c2c(OC)cnnc2)=O)(CO)CCCN(C(C2CC2(C)C(F)F)=O)C1 c1(N(CCN(C)C)CC)ncn(C)c(=O)c1Br.C1(=O)CCC(=O)N2CCCC2N1 N1(C(c2n(C(C)C)ccn2)=O)CC(C(=O)NC2CCC3(CCC3)C2)CC(C)(C)C1 C1(OC)CCC(C)(C(=O)NC2CCCN(C(C3CCCN3C)=O)C2C)CC1 c1(CC(C(=O)NC(CNC(C(CSC)OC)=O)(C)CO)C)ccc(F)c(F)c1 c1(OC)cccc(CC(C)NS(=O)(=O)CC(C)C2CC2)c1F N=c1[nH]ccc(C(N2CC(O)(CNC(C3CCCS3(=O)=O)=O)C2)=O)c1Cl C1(C(=O)O)CC2CCCCC2N(C(CCCc2ccccc2)C=O)C1.C1(C)CC1 c1(CNC(C)=O)ccc(C(=O)NCC#CCNC(=O)CN(C)C(=O)C2CC2)o1 CCC(C)CCCC(=O)N(CCC(N1CC2(C1)CN(C)CCO2)=O)C1CC1 CCCS(=O)(=O)CC(=O)NC12CCC(CN(C(c3ccncc3Cl)=O)C1)C2 C12(C(=O)NCC3(CNC(c4cc(=O)cc[nH]4)=O)CC3(F)F)CCCCC1OCC2 C(=O)(C#CC1CCCOC1)N1CCCCC(NC(c2ccc([N+](=O)[O-])s2)=O)C1 c1(-c2n(CC=C)c(N3CCCC(c4nncs4)C3)nn2)ncc(C)cc1F c1(C(N(CC(O)CN(C)C(c2cc(C(F)F)no2)=O)C)=O)n[nH]c2c1CCOC2 N1(C(C2C(C)C2C)=O)CCN(C(=O)CCC(=O)c2ccccc2)CC(C)(C)C1 c1(C(N2CC=CC(NC(C(CCC)(C)C)=O)C2)=O)cc(F)cc(Br)c1O C1(CC)CCCCC1C(=O)NC1(CO)CN(C(c2cc(C3(O)COC3)on2)=O)C1 C1(COC)(CNC(=O)CCCOC)CCCN1C(=O)CCOc1ccccc1 c1(NCC2(OCC)CCCSC2)cc(N2CCC(COC)C2)nc(C(F)(F)F)n1 c1(C(N(CCNC(=O)CCc2ccon2)CC)=O)c[nH]c2ccc(F)cc2c1=O C1(CNC(CCOC2CCN(C)CC2)=O)CCCCCN1C(=O)CC(O)C1CC1 N1(C(=O)CN2CCCCC2=O)CCCC2(C1)CN(C(c1cc[nH]c1)=O)CCO2 C(CCCCCNC(=O)Cc1ccc(O)cn1)NC(C(C)CC1CCCCC1)=O O=C1NCC2(CCN(C(CC3CC3)C(=O)NC3COC3)CC2)N1 c1(NC)ccc(C(N2CCC(C(=O)NCC34CCC(CC3)C4)C2C2CC2)=O)cc1 c1(OC)cc(OC)c(CN2CC(F)CC2CN)c(Cl)c1 c1(CC)ccc(F)c(C(=O)NC2(CF)CCN(C(C3(OC)CCC(C)C3)=O)C2)c1 CCCCS(=O)(=O)NC(C)C(=O)NCCOC.C(=O)(CCO)N(CCOCCC)C c1(OC)cc(OC)c(C(N2CCC(N)C2)=O)cn1.N1(CCNCC)CCN(C)CC1 C12CCCCN1C2.C1(CNC(C2CCCCC2)=O)CCSCC1 C(=O)(C1=NOC(C)C1)NC1CCN(C(c2nnc(C)s2)=O)C1 N1(C(C2C(C(=O)OC)C2)=O)CC2C(NC(=O)Cc3cnc[nH]3)CS(=O)(=O)C2C1 C=CC(C)(C)CC(=O)N1C(C(=O)NC2CC3(CCCC3)C2)CCC1CC c1(C(=O)NCC2CN(C(C3CN(C(C)C)C(=O)C3)=O)C(C)C2)cc(Cl)ccc1F c1(CC(=O)NCC(CNC(C(C)NC(=O)OCC)=O)O)cccc(F)c1F CC(C)CS(=O)(=O)CC(=O)NC1CN(C(=O)CCCC(N)=O)CC1C1CC1 CC(C)(C)C(CNC(=O)NCc1cccc(C(C)(F)F)c1)C(F)F N=c1ccc(C(N2CCCC2CCCNC(C2CC3C=CC2CC3)=O)=O)c(Cl)[nH]1 C(N=c1nc(N2CCC(OCCF)C2)c2c([nH]1)CCCCC2)C1(P(C)(C)=O)CC1 CCCC(C)(O)C(=O)N1CCC(C(=O)NCCc2cccc(O)n2)C1 c1(C(=O)NCCCNC(C2CC(c3ccc(F)cc3)C2)=O)nnn2c1CSCC2 C(=O)(CCCC(=O)OC)N(CCCOCCN(C(C1CC(=C)C1)=O)C)C C1(NC(C2C(=C)C2)=O)CCC2CC1CN2C(=O)CCc1ccc(N(C)C)cc1 c1(C(=O)NC2CC(N(C(C(CC)O)=O)C)C2)cc(OC)cc2c1CCC2 C1(C#N)(C(=O)NCC(c2ccccc2)CNC(CC(=C)C)=O)CCSCC1 c1(C(N(C(=O)NCCc2c(C)noc2Cl)C)C)nc2c(s1)CCCC2 c1(C(=O)NC2CCCC2CNC(C2(c3ccno3)CCC2)=O)cc[n+]([O-])cc1 c1(OC)ccc(F)c(CC(N2CC=CC(NC(c3cnc(C(C)C)[nH]3)=O)C2)=O)c1 N1(C(C2CCSCC2)C(=O)NCSc2ccc(OC)cc2)CCCC(C)(O)CC1 N1(C(Cc2onc(C)n2)=O)CCCC(N(C(=O)CC2CC2(C)C)C)CC1 C1(F)(CNC(=O)Cn2ncnn2)CCC(NC(c2cc[nH]c2CC(N)=O)=O)C1 N1(C(C2CC(F)C(=O)N2)=O)CCN(C(=O)C=CC2CCCC2)C(CO)C1 N1(C(C(CC=CC)NC(=O)CN(C)C(=O)C2CC2)=O)CCOC(C)(CC)C1 c1(C(=O)NCc2ccc(CNC(C(C)(C)SC)=O)cc2)cncc(Cl)c1C c1(OC)ccc(C(=O)NC2CN(C(=O)C(N)=O)CC2C)nc1OC C1(NC(C2CC23CC3)=O)CCC2CCN(C(C3Cc4cscc4C3)=O)C1C2 N1(C(CCC2(C)CC2)=O)CCC2(CC1)CC2CNC(C1CC2(C1)CC1(CC1)C2)=O C1(NC(CCNC(C(C)(C)C)=O)=O)CCC2CN(c3cncc(Cl)n3)CC2C1 C(C(C)(C(=O)NCC1CC(NC(=O)CCc2ccnn2C)CC1O)OC)OC N1(C(c2c(C)noc2C(F)(F)F)=O)CC(CNC(c2cscn2)=O)CC(C)(C)C1 Cc1nc2ccnn2c(C)c1C(=O)NCCCCCNC(=O)C(C)NS(C)(=O)=O C(=O)(C(F)(F)C(C)(C)O)N1CCC(C)C(NC(=O)C(O)Cc2cnn(C)c2)C1 c1(OC)c(C(N(C(C(C)NC(=O)NC2CCCO2)C)C)=O)nnn1C C#CC1CCN(C(C2CC(NCCn3cc(-c4ccccc4)cn3)C2)=O)CC1 c1(C(=O)NCc2nc(CNC(CN3CCC(C)CC3)=O)sc2)cnn2ccncc12 Cc1oc(-c2cnn(C)c2)nc1C(=O)NCC1CN(C(C2CCOC2(C)C)=O)C1 C1(NC(C(C=C)(C)C)=O)CC(C(=O)NCCNS(N)(=O)=O)=CC1O N1(CCC(C)C)CCCC1C(=O)NC1CCC1CNC(c1ncnn1C1CC1)=O O(N(C)C(=O)CN=c1nc2c(cnn2C)c(NCC(c2ccsc2)C)[nH]1)CC N1(C(CCNC(C2CCc3nccn3C2)C)C)CCC(C)C(C)(C)C1 N1(C(c2ccc(C)cc2)C(=O)NCCOCC)CC(C)C(F)(F)C1 CC1CCC(CN(C)CCSc2nnc(N3CCCC3)o2)O1 N1(C(C(N2CCOCC2)C)=O)CC2CCC2(CNC(C2(F)CC3(CCC3)C2)=O)C1 c1(NC(C2(C)CCN(C(Cn3ncn(C)c3=O)=O)C2)=O)ccc(O)c(F)c1 N1(C(C(C2CC2)SC)=O)CC(CNC(=O)CCc2nc(C)no2)CC(C)C1 C=C1CC2(C1)CC(C(=O)NCCCOCCNC(=O)C(C1CCOCC1)C)C2 C1(C2CCN(C(=O)C(c3ccc(Cl)cc3)O)C2)(NC(C2CCC2(F)F)=O)CC1 C1(C(=O)NC(CC)CNC(=O)Cc2cnco2)CC=C(C)CC1 C1(NC(c2c(C)nns2)=O)CC(CNC(c2ccc(=O)oc2)=O)C1(C)C CCCCC(O)C(=O)NC1CCCC1CNC(=O)COc1ccc(Cl)c(C(C)=O)c1 c1(C(N2CCC(C)(CNC(C3(CF)COC3)=O)C2)=O)cccc(Br)c1F C(=O)(C1CCCn2cnnc21)NCC(C)CNC(=O)Cc1cccnc1Cl c1(CC(=O)N(C2CCN(C(=O)CC3CCCC3C)CC2)CC)cnc(Cl)cc1C C1(CC=C)CCCCN1C(=O)C(COCC)NC(=O)Cc1ccc[nH]1 Cc1c(CNC(C2CC(C)(F)C2)=O)sc2cncn12 N1(CCSC)C(=O)NC(c2ccc(C)nc2F)C2=C1CN(c1ccccc1)C2=O C1(C(F)(F)F)(C(=O)NCC2N(C(C(C)=C(C)C)=O)CC=C2)CC=CCO1 O=[N+]([O-])c1cnn(-c2ccccc2)c1NCc1ccc(C(F)(F)F)cc1F c1(C(N2CCC(N(CCO)C(C3(F)CCCCC3)=O)C2)=O)cc(Cl)cc(Cl)c1 c1(C(=O)OC)ncc(NCC23CCC2CCN3Cc2ccccc2)cc1Cl C1(C)(CC(=O)NCC2(NC(C(CC=CCC)C)=O)CC2)CCS(=O)(=O)N1 C1(NC(C2N(CC)C(=O)CC2)=O)CCN(C(c2ncc(N(C)C)cn2)=O)C1(C)C C1(NC(=O)CC2(O)CCN(Cc3nn[nH]n3)CC2)CCC2CCC1OC2 c1(Oc2ccccc2C2(C(=O)Nc3c(C)cn(C)n3)CC2)ccc(O)c(C(C)C)c1 C=C1CC2(C1)CC(C(=O)OCCc1ccc(CNC(=O)OC(C)(C)C)[nH]1)C2 C(CCCC(C)(C)C(=O)NNC(=O)c1ccc(C)s1)NC(C(CC)C)=O C(C#Cc1cn(C(C)(C)C)nn1)NC(C(CC(C)C)N1CCC(C(C)C)(CO)C1)=O N1(C(C(C)c2cncs2)=O)CCC=C(CNC(c2ccoc2)=O)C1 N1(C(CC(CC)(C)C)=O)CC2CC1CCN2C(c1cnc(C(F)F)s1)=O N1(C(CSCC#C)=O)C2CCC1CC(NC(C1CC(F)(F)CS1)=O)C2 C1(CC)C(C(N2CC=CC(O)C2)=O)CCN1C(c1cc(C(C)=O)c[nH]1)=O C(CS(=O)(=O)CC(=O)NCc1cnn(C)c1)OC.c12ccc(C)c(c1)NC2=O N1(C(c2n(C=C)ncc2)=O)CC(C)(C)OC2(C1)CN(C(=O)C(CC)=CCCC)C2 Cc1nc2cc(C(=O)N(CCCN(C(=O)CC3CC3CF)C)C)c(F)cc2[nH]1 Cc1cc(=NC(=O)C(=O)NC2CC3(CCN(C(C4CCOC4=O)=O)C3)C2)[nH]o1 Cc1noc(C)c1CSCC(=O)NC(C)C(C(C)C)NC(C1CC(O)C1)=O C(=O)(C1=CC2(CCOCC2)C1)N1C(CC)CN(C(=O)C(C2CCCC2)OC)CC1 C1(C(=O)NCCCCNC(CCC(C)(C)OC)=O)CC2CCCCN2C1 c1(OC)cnc(-c2ccc(-c3nccn3C)s2)nc1.c1nnc(C(F)(F)F)o1 N1(C(c2c[nH]c(=N)o2)=O)CCCC(C2(NC(=O)Cc3ccsc3)CC2)C1 C1(COC)(NC(=O)CC2CCCOCC2)CCN(C(=O)Cc2ccsc2Cl)CC1 Cc1nn(C)c(N)c1C(=O)NCC1CCN1C(=O)C(C)CO c1(C(=O)NCC(CO)NC(c2c(C(C)C)onc2)=O)ccc2c(c1)OCC(=O)N2 N1(C(C2(C)CCCN(C(C3CCCCC3O)=O)C2)=O)CCC2(C1)CC2(F)F C#Cc1cc(C(=O)NCC2CN(C(=O)Cn3cccn3)CC2(C)C)ccc1C C1(C)(C(N(C)CC2C3CN(C(=O)CS(=O)(=O)C4CC4)CC23)=O)CCCNS1(=O)=O CCC(CC(F)(F)C)C(=O)NC1CN(C(c2ccncc2C(F)(F)F)=O)CC1C C1(CNC(C2(CC)CN(C(C3CC3[N+](=O)[O-])=O)C2)=O)CC2(CC(=O)C2)C1 C#CCC(CC(F)F)C(=O)N1CCC2(CC1)CC2C(N(C)C[Si](C)(C)C)=O Cc1ccc(CN(CCO)Cc2cccc(-n3ccc(C)n3)c2)cc1 C1(CC=C)(NC(=O)COC2CCCOC2)CCCN(C(c2nocc2Cl)=O)C1 Cc1sc(C(=O)NC2CN(C(=O)CCN3CCC(F)C3)CC2C)nc1O c1(C(=O)NCC(C)CNC(=O)CC(C)C2CCCO2)ccc(Cn2cccn2)o1 CC1C(Cl)CCN1C(=O)CCC1CN(C(=O)C(C2CC3CC3C2)C2CC2)C1 C1(F)(CNC(C(SC)SC)=O)COCCN(C(=O)CCC2CCCC(=O)N2)C1 N1(C(COC(C)=O)=O)CC=CC1(C)C(N1CCC(CC(N)=O)CC1)=O C1(C(=O)NC23CC(NC(CC4C(C)OCC4)=O)(C2)C3)CN2CCC1CC2 Cc1cc(OC(C2CCC(=O)N2C(C2(I)CC2)=O)=O)cc(C)c1C C1(CCC=C)(C(=O)NC(C2(O)CN(C(C3(C)CCCO3)=O)C2)C)CCCC1 C1(C(N2CC(NC(c3n[nH]cc3C3CC3)=O)C2)=O)Cc2ccc(F)cc2O1 CC(CCc1ccccc1)C(C(=O)Nc1ccccc1Cl)N1CCC(CO)CC1 C1(C)(CNC(c2nc(-c3cc(SC)c(C)o3)on2)=O)CCC(C)=C(C)C1 N1(C(c2c(CC)cncc2)=O)CC2(CC(NC(C3CCC(C)(C)O3)=O)CO2)C1 CC1(NC(c2c[nH]c(C#N)c2)=O)CCCN(C(c2cnc[nH]2)=O)C1 c1(C(=O)NC2C3CN(C(c4cnc(C5CC5)o4)=O)CC23)cc2ncccc2o1 C(=O)(C1=NOC2COCC12)N1CC2(CCN(C(C34CC(C)(C3)C4)=O)C2)C1 C1(NC(CC2CC(CC)C2)=O)CCCC2CN(C(=O)Cc3nn(C)cc3Cl)CC12 c1(CCOC(C(C)(C)C(C)C)=O)ccc([N+](=O)[O-])cc1Br CCC(C)C(C(=O)Nc1ccc(C)c(CO)c1)N(C)CCc1ccccn1 c1(C(N(CC(C)O)CCNC(c2c(C)nc(C3CC3)o2)=O)=O)ccc(=O)n(C)c1 C1(NC(Cc2cc(C)nn2C)=O)CC(F)CN(C(c2cn(CC(N)=O)nn2)=O)C1 C1(C(C)NC(c2ccoc2)=O)CCN(C(c2csc(-c3cccnc3)n2)=O)CC1 C=CC(C)CC(=O)OC(C(C)OCCC)=O C1(N(C(CSCC(=O)OC)=O)C)CN(C(C23CC(C)(C2)C3)=O)CC1(C)C c1(C(C(=O)Nc2c(CC)noc2)NC(=O)C(F)OC(F)(F)F)c(C)cccc1Br C1(NC(C=C2CCC(C)C2)=O)C2CC1N(C(c1ccccc1-c1nc[nH]n1)=O)C2 CCC(C)C(O)CC(=O)NC1CC(C(=O)NCC2(C)CCN(C)C2)=CC1O C=CCC(C(=O)NC1CCN(C(=O)Cc2cncs2)C1C(C)(C)C)C(C)C c1(CC(=O)NC2CC(NC(CN(C)C3CC3)=O)C2)cc(C(F)(F)F)ccc1Cl c1(C(N2CCC3CN(C(C4CC45CCCCC5)=O)C3C2)=O)nccn2nccc12 c1([SH](CC)CC)nnc(CCc2cnn(-c3ccc(F)cc3)n2)n1N c1(OC)ccc(-c2nc(C3CCCN(C(C)C)C3)n(CC(C)C)n2)nc1 c1(NC(=O)NC(C)CN2CCC(c3ccccc3)C2)ccc(F)cc1 c1(-c2cn(CCCC(=O)NCC3(c4ccc(F)nc4)CC3)nn2)ccc(F)cn1 C1(CNC(CC2N(C(C=CCC)=O)CCC2)=O)CC12CCCCC2 c1(N(CCNC(c2sc(C(=O)OC)nc2C)=O)CC)nn(C)cc1CO CC1CCCCC1C(=O)NCCCCCN1CCN(C(=O)C=CC2CC2)CC1 Cc1nc(Cl)[nH]c(=NC2CCC3CN(C(c4ncc(F)cn4)=O)CC23)c1[N+](=O)[O-] c1(C(C(=O)N(CC)Cc2nnc(C(C)C)o2)F)ccc(C)cc1 N1(C(c2cc(OC)ns2)=O)CCN(C(C2CC2C2CCC2)=O)C(CF)C1 C(C(=O)NCCC(C)N(C)C(C1CC=CC1)=O)(C(C)C)c1cc(C)no1 N(S(=O)(=O)N1CCC(C)CC1)CC.N12CC(C)CCOC1=CC=CC=C2 C(=O)(C(F)C(F)(F)F)NC1(CNC(c2cnc(=N)[nH]c2)=O)CCOCC1 c1(N(C(C(CC)C)C)CCOC)ccc(F)cc1.C1(=O)NCCO1 C(C(=O)NOCCCCF)(c1ccoc1)NC(=O)CCCC1CCCC1 c1(CCCC(N2CCN(C(CC=C)=O)C3C2C3)=O)ccc([N+](=O)[O-])cc1 c1(-c2cn(CC(CCNC(CCNC(C)=O)=O)F)nn2)ccc(OC)cc1OC N1(C(c2cc(C)cc(Cl)n2)=O)CC(F)C(N=c2ncnc3[nH][nH]c(I)c2-3)C1 c1(CC)ccc(C(=O)NC2CCCCC2C(=O)NCC2(N(C)C)CCC2)nc1 N1(C(c2cc(C)sc2)=O)CCC(C(N(CCC#N)CCN2CCCC2)=O)CC1 C1(C(N2C(C3(NC(C(C)CC4CCC4)=O)CC3)CCCC2)=O)CC(S(C)(=O)=O)C1 C(C(=O)OCC1CCCN(C)C1)(C(C)(C)C)NC(CSC)=O C=CCCC(C)(C)C(=O)N1CC(CNC(c2csc(CCC)n2)=O)C2(CC2)C1 C1(C(N2CC3(CCC(NC(c4ccnnc4)=O)C3)C2)=O)CCN2CCCC2C1 c1(OCC(=O)OCC)cnccc1OCC(=O)NCCNC(C1CCCSC1)=O C(=O)(CCS(N)(=O)=O)N(C)CC1CCCN(C(C2(NC(N)=O)CCCCC2)=O)C1 c1(C(N2CC(C)C(CNC(C3CCCN3C)=O)C2)=O)ncnc(O)c1Br C(=O)(CCCCCN(C)C)NC(CNC(c1c(-c2ccc(C)o2)onc1)=O)(C)C c1(C(=O)NC(C(N2CCN(C(=O)NC)CC2)=O)CCC2CC2)ccc(O)c(F)c1 N1(C(C2CCC(=O)N2)=O)CCOC2(CCN(C(=O)Cn3ncnn3)C2)C1 c1(CNC2(C(=O)Nc3cc(C)no3)CC2)cc(F)c(-n2ccnc2)c(F)c1 c1(CNC(c2cc(-c3ccccc3)cs2)=O)cccc2c1CNC2 N1(C(C(=O)NCCSc2nc(C)[nH]n2)=O)CCC(C2CCNCC2)C1 c1(C(N2CCC(NC(c3nc(C)c(C)s3)=O)CC2C)=O)cccn2cnnc12 C1(C(N(CC(C(C)C)OC)C)=O)(CO)CCN(C(=O)C(C)Cn2ccnc2)C1 C(=O)(C1CCCCc2ccccc21)N1CCC(N(C(=O)C2=CCCCC2C)CC)C1 C1(C2CCN(c3ncncc3I)CC2)(NC(=O)CCNc2cccc(Cl)c2)CC1 C12(CCC=C)CN(CCO1)C1CCC(C1)OC(=O)C2.c1(OC)ccccc1 N1(C(C(C(C)C)CO)=O)CCC2(CC1)CCN(C(=O)CCc1ccc(F)nc1)C2 N1(C(CC(CCC)NC(=O)C=Cc2cscn2)=O)CCN2CCC1CC2 Cc1sncc1C(N1CCC(NC(c2cc(C3(C)CC3)n[nH]2)=O)C1)=O C1(NC(c2cccc3c2CCCN3)=O)CC1C1CCN(c2cncc(Cl)n2)CC1 N1(C(c2cc(CC)nn2C)=O)CCCC(O)(CCNC(C2(C)CCOC2C)=O)C1 c1(NC(N2CCC2c2cccs2)=O)ccc(F)cc1.c12ccccc1CN2 c1(C(N2CC(CNC(C=CC)=O)C3C2C3)=O)cc2ncccc2[nH]1 C1(NC(C(F)=CC)=O)CCCN(C(c2ccc(C)c(N)c2)=O)C1C c1(C(=O)NCC(C2CC2)NC(c2cnn(CC)n2)=O)c(C)cnnc1O N1(CC(=O)NC2C(NC(C(C)OCCOCC)=O)CCC2)CCCCCC1=O C1(CC(=O)NCC(CNC(C2C(C)(C)OC2(C)C)=O)OC)COCC2(CCC2)O1 C1(CCNC(C(CCOC)(C)NC(=O)OC)=O)COC2(CCOCC2)C1 C1(C(N2CSCC2C(=O)NCC(C)C(C)(C)C)=O)(CC)CCCCO1 CC(CCCCNC(=O)CC1CCCN1C)NC(=O)CCSc1n[nH]c(=N)s1 C1(CCNC(C2(CCNC(c3nnc(CCCC)s3)=O)CC2)=O)CCCCC1C C(C(=O)O)(C1CCc2ccccc21)NC1C(SC)COC1 Cc1ccc(C#N)cc1NC(C1C2CCC(C2)C1NC(=O)Cc1ccc(F)cn1)=O c1(C(=O)NCc2cncc(C(=O)NC(C)(C)C)c2)cc(F)cnc1O C12(CNC(Cc3c(C)nc(C)s3)=O)CCC(CC1)N(C(=O)C(C)c1ncco1)C2 c1(CCNC(C(C)OCCNC(C2(C(CC)=O)CC2)=O)=O)cc(C)ns1 Cc1cccc2c1CC(C(=O)NCC1CCCCNC1)O2 Cc1[nH]nc2c1CCC(NC(=O)N(c1ccc3c(c1)OCCO3)c1cncs1)C2 C1(O)(CNC(C2(COC)CCCO2)=O)CCCN(C(C2CCN(C)C2=O)=O)CC1 c1(C(N(CCNC(=O)C(C)(COC)OC)CC)=O)cccc2nc(C)cnc12 N1(C(c2cc(CC)[nH]n2)=O)CCC(O)(CCNC(c2ocnc2C2CCC2)=O)C1 C1(CNC(=O)CCn2cc(Cl)cn2)CC2(CC2)CN1C(c1cnn2c1OCC2)=O N1(C(c2c(C)n[nH]c2)=O)CCC(CNC(=O)CC(C)(C)CN(C)C)C(F)(F)CC1 C1(C(=O)NCCCOCCCNC(c2n(C)ncc2)=O)CC(C2CC2)=NO1 N1(C(CC2CC(OCC)C2)=O)CCC(NC(c2sccc2SCC(C)C)=O)CC1 c1(C(=O)OC2C(C)(C)CCC2)cc(F)cc([N+](=O)[O-])c1 N1(C(COCC(=C)C)=O)CCN(C(=O)C(C)SCOC)C(CC(F)F)C1 C(=O)(CC(F)(F)C(F)(F)F)NC(CC=C)CNC(c1cccc(C)c1N)=O C(C(CC1CC1)C(=O)NCc1cccc(C2CC2)c1)NC(C(C)C)=O CC1CN(C(=O)C(F)(F)c2csc(Cl)n2)CC1NC(=O)C(F)CC1CCCCC1 N1(C(C(C)OCC#C)=O)CC(F)(F)CC1CNC(=O)Cc1ccccc1O Cc1cc(C(F)(F)C(=O)NC2CCN(C(=O)CCC=CC(C)C)C2)cnc1Cl N1(CCC(N2CC(O)(CNC(C(C)c3ccsc3)=O)C2)=O)C(=O)NC(C)(C)C1=O c1(NC(=O)NC)cnccc1SCCOC N1(C(C(F)=CC)=O)CCC(C(C)(O)CNC(c2ccnc(C(F)F)c2)=O)CC1 CCCC(C(O)C(=O)N1CCC1(C)COC)NC(c1cc(C)c(N)cn1)=O c1(C(=O)OC)sc(=NCC2(CNC(C3(O)CCC(C)CC3)=O)CCC2)[nH]c1Cl C(C(=O)NNC(=O)C1CCCC(C)CC1)=CCCC(=O)OCC c1(C(=O)NCCNC(C23OC(C)C(CC2)C3)=O)cc2nnn(C)c2s1 C12(C(=O)NC(C)(C)CCF)CCC(NC(=O)CC(Cl)Cl)(CC1)C2 N1(C(CC(C)C2CC2)=O)CC2(CCC(NC(C3CCC(C)(C)O3)=O)CC2)C1 O=C(CN=c1cc[nH]cc1)N1CC2CN(S(=O)(=O)CC(F)(F)F)CC(C1)O2 c1(C(=O)NC2(CO)CN(C(C(O)NC(=O)OCC)=O)C2)cccc2nn[nH]c12 c1(C(=O)OCC)cc(C(CCC(=O)NC2CCC2)N(C(C)C(C)C)C)[nH]n1 c1(C(=O)NC2CCC(NC(Cc3onc(C)n3)=O)C2)cccn(CC(C)C)c1=O Cc1nc(C(=O)NCC2CN(C(=O)C(O)C3CC3)CC2C)cc(O)n1 C#CC1(N(C(C(COC)C(=O)OOCOC)C)C)CCCCCC1 CC1CCN(C(c2cn(C)[nH]c2=N)=O)CC1C Cc1ccnc(C(N2CCOC(CC(=O)NCC(C)C(C)O)C2)=O)c1F C1(NC(c2c(C)cc(C)o2)=O)CCC2(CC1)CCN(C(c1cc[nH]n1)=O)C2 c1(C(=O)NCCOC2CN(C(C3CC=CCC3)=O)C2)cc2ccc(Cl)cc2o1 C12(C3CCC13)C(=O)N2.C(CC)(CC)=CC(=O)NCC1(CC)CC1.CSC c1(C(C(=O)NC2C=CCN(C(C3(SC)CCC3)=O)C2)(C)C)cc(Cl)ccc1F n1(CC)nc(C(=O)NC2CC(CCNC(=O)C=C3CCCC3)C2)cc1C(F)(F)F N1(C(C2CC3(CC(NC(CC4CC(C)C4)=O)C3)C2)=O)CCCC(N=[N+]=[N-])C1 CCCCCC(O)C(=O)NCC(C)CNC(=O)CCCCO N1(C(C23C(CN(C(C(C(C)C)C)=O)C2)C3)=O)CCS(=N)(=O)CC1 C1(O)(C(C)NC(CNC(CC(C)C)=O)=O)CCN(C(C2CC2(Cl)Cl)=O)C1 N1(CC2CCCC(C)(N)C2)CCCc2cc(NC(=O)C(F)(F)F)ccc21 N1(C(Cc2c(C)n[nH]c2)=O)CCC=CC1C(=O)N(C)CCn1ccnc1C c1(OCC)cc(F)ccc1CN1CC2CN(C(=O)CC(C)c3ccco3)CC12 CCCC(C)CC(=O)NC1CC1CNC(c1cccc(NCC#N)c1)=O c1(C(=O)NCCC(=O)NC2CCC(N(C)C(C3CC=CC3)=O)C2)ccccc1F CCCCC(CC)CCC(=O)NC(C1CCCC1)CNC(=O)CCn1ccnn1 C(C)(C)(CC(F)C(=O)N1CCN(C)C(C)(C)C1)NC(CCCSC)=O c1(C(=O)NCC(CNC(c2cc(CC)ncc2)=O)F)cc2ccc(Cl)cc2s1 c1(C(CNC(N(c2ccccc2)CC=C)=O)C)snnc1C C1(C(N(C2CCN(C(c3coc(CS(C)(=O)=O)n3)=O)C2)CC)=O)CCCCC1 CC1(C)CC(C(N2CCC(NC(=O)CC3=CCOCC3)C(O)C2)=O)CC(C)(C)O1 c1(OC)ccc(C(N2CCN(C(=O)C(C)O)CCC2C)=O)c(Br)c1F C1(NC(CC(C)c2ccco2)=O)CN(C(=O)CC2CCCC2)CC12CC2 CCC(C)(O)C(=O)NCC1(NC(=O)C(n2ccc(C)n2)C)CC1 CC1C(C(=O)NCCC(C)(C)F)CCCN1C(=O)C1=CCCOC1 Cc1c(NCCOc2ccccc2F)ncnc1N1CCN(C)C(SCCO)C1 C(N=c1[nH]c(=NCC2(CCO)CCCC2)c2[nH]ccc2[nH]1)C1C(C)(C)C1 N1(C(CCCc2c(C)ccs2)=O)CCC(C2CC(NC(=O)CCC(C)C)C2)C1 c1(NC(C2CCN(Cc3cc4sccc4s3)CC2)=O)cc2ccccc2o1 C12CCC3(CC1)CC3C(=O)N2.N1(C(COCCOC)=O)CCC(C)(OC)C1 O=C(C1=NOC(CO)C1)N1CC(C2(N(C3CCCCCC3)C(C3CC3F)=O)CC2)C1 C1(NC(C(C)C)=O)(Cc2ccccc2)CCCN(C(C2CCC(F)(F)CO2)=O)C1 C1(C(=O)NCC2C(C)(C)CCN2C(=O)Cn2ccnn2)CCC2(CC1)CC2(F)F c1(C(=O)NCC2N(Cc3ccc(C)o3)CC2)nnc2n1CCCC2 CCCC(CCCNC(=O)C(C1CC1)OC)N=c1[nH]nc(CO)s1 C1(CC(=O)NCc2cc(C(C)C)no2)CC(NC(=O)C(F)C2CCCC2)C1(C)C C1(CNC(=O)NCC2(C3CC3)CCCO2)CC2CCCC(C1)N2C1CC1 N1(C(=O)NCC2CC(CO)CO2)CCC2(CCCNC2=O)CC1 N12CC(C(SC)C1)NC1(CC1)C2=O.c1(OC)ncoc1CNC(=O)OC(C)(C)C S(=O)(=O)(c1cc(-c2ccccc2)[nH]c1C)NCC(C(=O)OC)C CCC(CC)(CCNC(c1cc(C2CC2)cs1)=O)NC(c1oc(C)cc1C)=O Cc1ccc(F)cc1C(=O)NC1CC2CCC1N2C(C1CC1c1ccco1)=O c1(NC(=O)CNS(C)(=O)=O)cc(Br)cc(I)c1 C1(NC(=O)C=CC2CCOCC2)CC1C1CCCN(C(C2NC(=O)CC2Cl)=O)C1 c1(C(N(CCCNC(C(SC)SC)=O)CCO)=O)ccc(Cl)c(C)c1 C(c1nc(C)c(C)[nH]1)=CC(=O)NCC(CC)(C)NC(c1cnc(S)n1C)=O C(=O)(C1=CC(O)C(NC(=O)CCCC2CCCC2)C1)NCC1NC(=O)OC1 C1(CC=C)(NC(=O)C(C)N(C(c2ccn(COC)n2)=O)C2CC2)CCCC1 C1(CC)CCCN(C(c2c[nH]c(-n3cnnn3)c2I)=O)CC1 C1(C(N(CCNC(c2cccc(CF)c2)=O)CC)=O)CCC2C(C1)C2(F)F C1(NC(C(C)(C)C2CCOCC2)=O)CC(O)CN(C(c2coc(C3CC3)n2)=O)C1 c1(SCC(=O)NC(CC)CN(C)C(C2CC(C)(F)C2)=O)ccc(Cl)cc1 c1(C(N2CC(O)(CNC(c3cnc(CC)[nH]3)=O)C2)=O)ccc2nn[nH]c2n1 C(=O)(CCCCCNC(=O)CC1CC2CC1CC2O)NC(c1ncc(C)cn1)C C1(C(=O)NC(C2(OC)CCC2)C)C2CCN(C(c3cc(O)cc(F)c3)=O)CC12 C1(OCCNC(C(CC)c2cccnc2)=O)CCN(C(C2(C)C=CCC2)=O)CC1 c1(CN2CCN(C(C(C)n3cncn3)=O)CC2C#N)cccc2ccncc12 C1(OCC)CN(C(=O)CSC2CC2)CC1NC(=O)CC1CCC(O)C1 C(=O)(C1CCCc2nc[nH]c21)N(C)CC1OCCN(C(CS(=O)(=O)NC)=O)C1 C1(CC(=O)NC2CC(OCC(=O)NCCCOCCC)C2)CSCCO1 C1(N(C(CC2(C=C)CC2)=O)C)CCC(NC(C2COC2)=O)C1 c1(C(N(CCC)CCNC(=O)C(CC)C(C)C)=O)cc(NC(=O)NC)ccc1Cl O=S(=O)(c1ccc(C(=O)O)cc1Br)Nc1cccc(OCCF)c1 c1(C(N2CC3C4CC(CC4)C3C2)C)c[nH]c2cc(Cl)cc(Cl)c12 c1(C(N2CCC(C(=O)NCCC(C)(C)O)CC2)=O)cc(I)c(F)cc1F CCCC(C#N)C(=O)NCC12CC1CN(C(c1ccc(O)nc1C)=O)C2 N1(C(CCCCOC)=O)C2CCC1(CNC(=O)C(C)Oc1ccccc1F)CC2 c1(C(=O)NCC(CN(C)C(c2cnsc2)=O)O)ccc(OC(F)(F)F)cc1F N1(C(c2c(C)coc2)=O)CCCN(C(c2cccc(C(=O)N(C)C)c2)=O)CC1C N1(C(CCc2ccc(C)nc2)=O)CC2(CC(NC(c3ccsc3C#N)=O)C2)C1 C1(O)(CN(C)C(c2coc(Cl)c2)=O)CN(C(=O)CC2(C)CC2F)C1 Cc1ccc(O)c(CN2CCC(F)(C(N3CCOC(C(N)=O)C3)=O)C2)c1 CC1=C(C(=O)NCc2nc(C(=O)NCC3(CCO)CC3)c(C)o2)COCC1 C1(C(=O)NC(c2c(C)cccn2)C)CC2(CCC2)CN1C(=O)CCS(N)(=O)=O c1(C(C)NC(C(C=C)O)=O)ccc(CNC(c2csc(CC)c2)=O)cc1 C1(NC(C2CC(=C)C2)=O)CC(F)CN(C(=O)CC2CCCC(OC)C2)C1 c1(N2CCC(CC=C)(NC(c3nc(=O)n(C)[nH]3)=O)C2)nc(Cl)ncc1Br Cc1nc(C(=O)NC2CCC(CCNC(c3ccccc3N(C)C)=O)C2)c(C)o1 C(=O)(C1CCCc2ccnn21)N1C(CCC)CN(C(C2CC3(CCCC3)C2)=O)CC1 c1(NC(N2CC(C(C)C)C(C)CC2)=O)ccc(S(C)(=O)=O)nc1 C1(C(N2CCC(C(C(=O)N(CCCO)CC#C)(C)C)C2)=O)CCC(O)CN1C C1(NC(c2cn[nH]c2)=O)CCCC1CNC(=O)C(O)c1ccco1 C1(C(=O)NC(C)CC(C)NC(C23COC(CCO2)C3)=O)C2(CCC2)C12CCC2 C1(NC(CC(C)OC)=O)CN(C(c2ncncc2Cl)=O)C2(CCOCC2)C1 C12(NC(C3CCN(C(c4c(COC)cc[nH]4)=O)CC3C)=O)CC3CC(CC1C3)C2 C1(C(C)NC(C2CCCC2)=O)CCCN1C(=O)Cc1cnn(C)c1 c1(CONC(=O)NCC(CN(C)C)O)ncn2ccccc12 CC(C)(C(=O)NC1CCC1NC(C1COC(=O)N1)=O)c1ccsc1 C(CCS(C)(=O)=O)(C(=O)NC(C)(C)CN(C)C(C1CC1C(C)(F)F)=O)OC N1(C(c2c(C)nc(C(N3CCCC(C(C)C)CC3)=O)o2)=O)CCCC(N)C1C.CC C1(OC)CN(C(C2CCCCN2C)=O)CC1NC(C1(NC(C)C)CCC1)=O c1(C(=O)NC2CCN(C(c3cccc(N)n3)=O)C2)ccc(F)c(O)c1F N1(C(CCCCOC2CN(C(=O)COCCF)C2)=O)CC2(CO)CC2(CO)C1 CC1(C)CC(O)CCN(C(C2C=CCN2C(C2CCCC(O)C2)=O)=O)C1 c1(C(N2CC(N(C)C(c3cc4sccc4n3C)=O)C2)=O)ccc([N+](=O)[O-])cc1F C(=O)(C(F)(CNC(c1nonc1C)=O)C(C)C)NCC(CCC)(C)O C1(C(=O)OCC23COC(C(F)(F)F)(C2)C3)CCC2C3CCC(C3)C12 C(CC)(C(=O)NCC(F)CNC(=O)Cn1cnc(Br)n1)OCCOC C1(NC(C23OCC(C)(C2)C3)=O)CCCCN(C(c2ccnc(O)c2)=O)C1 c1(-c2c(OCC)cc(C(C)=O)cc2)ccc(Br)c(C)c1C C1(C(C)NC(c2csc(-c3cnc[nH]3)n2)=O)CCCN(C(=O)COC2(C)CCC2)C1 C(=O)(CS(N)(=O)=O)N(C(C)CNC(=O)C(c1cscc1Br)N(C)C)C c1(CC)nc[nH]c1C(N1CC(F)(CNC(=O)C(C)Cc2ccccn2)C1)=O C1(NC(C2CCC3(CC3)C2)=O)CC2CCC1N(C(c1cccc3[nH]ncc13)=O)C2 c1(C(=O)NC2CCCC(NC(Cn3nc(C)oc3=O)=O)C2)cc([N+](=O)[O-])oc1C CCC(C)C(O)C(C)C(=O)N1CC(C)(NC(=O)CC2CC(F)(F)C2)C1 CC(C)C(C(=O)NCc1ccc(C#N)cn1)C(C)NC(c1cccc(=O)o1)=O Cc1ccc(NCc2cn(C)nc2OCc2ccccc2)c(F)c1F n1(CCCC)nc(C)c(C(=O)NCCCN(C(C2COC(C)C2)=O)C(C)C)c1Cl Cc1cccc(NC(=O)Nc2cnccc2Cn2cccn2)c1C Cc1cc(C(=O)N)cnn1.N1(C(c2c(C)cco2)=O)CC(CO)C(O)C1 c1(CCNC(=O)NC(C#C)Cc2cccc(Cl)c2)nnc(S)n1C1CC1 Cc1ccc(C(N2CCCC(CN(C(=O)C=CC=C(Cl)Cl)C)C2)=O)cc1N N1(C(C(=O)NCC23CC(F)(CO2)C3)=O)CCC(C2CC2)C1 c1(C(N2C(C)CC(NC(C(NOC)=O)=O)C2)=O)cc([N+](=O)[O-])c[nH]1 Cc1cc(C)n(CC(=O)NC2CN(C(=O)CC(C)C)C3CC23)c(=O)n1 CCCCCCCC(=O)N(CC(CC)NC(c1c(F)ccc(F)c1Cl)=O)C C(=O)(C#CC1CCCCO1)NCc1ccc(CN(C(CCCC)=O)C)cc1 C1(NCCc2cn(CC(=O)NC(c3nnc(C)s3)C)nn2)OCCOC1(C)C C1(N(C(c2cc(C(=O)OC)no2)=O)CC)CCCN(C(=O)CC(C)(C)OC)CC1 N1(S(CC2(C(=O)OC)CCOCC2)(=O)=O)CCC12CCOC(C)(C)C2 C1(C(N2CCC(N(C(=O)Cn3cc(Br)cn3)C)C2)=O)COCC1(C)C CCCC(O)CC(=O)NCCCC(C)NC(c1ccc(C#N)o1)=O c1(OCc2ccc(C(=O)OC)cn2)ccc(Br)nc1OC C1(C(N(C2CCN(C(=O)CCC#N)C2)CC)=O)CC2(CCCCO2)C1 Cc1cnc(N)c(C(=O)NCC2CCN(C(c3cnc(C4CC4)s3)=O)CC2C)c1 C(=O)(C1CCCc2nncn21)Nc1cccc(CNC(c2cc(=O)cc[nH]2)=O)c1 C(=O)(CC(C(F)F)NC(=O)C(F)C(C)(F)F)NCCC(=O)N(CC)CC N1(C(C(CC)C#N)=O)CCC2(CC1)CC(CNC(C1(OCC)CCCC1)=O)C2 S(=O)(=O)(c1c[nH]ccc1=NCC1(CCOC)CC1)NCCCCCC=C CC1CC(NC(C2(C)CCOCC2)=O)CN(C(c2ccc(CO)nc2)=O)C1 N1(C(C2(CC)CCCC2O)=O)CCCN(C(=O)C(=O)Nc2ccc(C)cc2)CC1 c1(C(NC(CCCCN(C(C(COC)OC)=O)C)=O)C2CC2)cc(F)ccc1O C(=O)(CC(O)C(C)C)NCC(CNC(c1ccn(-c2c(C)cccc2)n1)=O)F c1(N2C(C(=O)N=c3[nH]nc(Cl)cc3Br)CC(OC)C2)ncnc2cccc(F)c12 c1(C(N(CCCNC(=O)C(O)CN2CCCC2)CC)=O)cc(Cl)c(Cl)s1 c1(C(N2CCN(C(c3cc(C=C)cc(F)c3)=O)CC2)=O)cc2ccc(O)nc2s1 c1(NC2CC(C)N(Cc3ccccc3)CC2)cccc2cccc(Br)c12 c1(C(C(=O)N(CCN(C(C(C2CC2)OCC)=O)C)C)C)ccc([N+](=O)[O-])cc1F C(=O)(CC(C)P(C)(C)=O)N1C2CC(CNC(c3scc(C)c3)=O)C1CC2 N1(C(C(CC)C(C)O)=O)CCCC2(C1)CN(C(=O)C=Cc1cc[nH]n1)CCO2 C1(NC(C(C)OCC#C)=O)CN(C(c2cccc(CN(C)C)c2)=O)CCC1F N1(C(C2CC2OC)=O)CCC(C(C)(C)CNC(C2CNC(=O)C2)=O)CC1.C(C)(C)(C)O S(=O)(=O)(c1ccc(Br)c([N+](=O)[O-])c1)NC(c1ncn(C)n1)C(=O)O C1(CC)CCCN(C(=O)CN(C)C2CC2)C1C(=O)NCc1cnccn1 C=CCC(CC)C(=O)NC12CCC(C1)N(C(=O)OC(C)(C)C)C2 O=C(C1=CC2CC=CCC12)NCC1(NC(c2csc(O)n2)=O)CC1 c1(CNc2scc(C(=O)OCC)n2)nc(OC)ccc1OC CCC(CC(=O)N1CCC(CN(C)C(c2ccnc(C(F)F)c2)=O)C1)SC C1(NC(C=CCCC(C)C)=O)C=CCCC1C(=O)N(C)CC1CCCO1 Cc1[nH]c(C(=O)NC(C)CNC(=O)CC(C)n2ccnc2)c(C)c1C CCC(C)CC(=O)NC1CCC1CNC(C1CC(CC(C)(C)C)C1)=O C1(CNC(C2(SC)CC2)=O)CC(C(F)(F)F)CN1C(=O)CC1(O)CCOC1 C12(NC(c3c(C)con3)=O)COCCC1CN(C(=O)CCNc1ncccn1)C2 N1(C(C=C(C)C(F)F)=O)CC(NC(c2coc(C(C)(C)C)n2)=O)CC12CCOC2 C1(C(N2C3(C)CC3CC2)=O)CC2C=CC1N(C(c1cnn[nH]1)=O)C2 C(c1cncc(F)c1)=CC(=O)NCC(CNC(CCn1c(C)ccc1C)=O)(C)C C1(c2n(CC3(OC)CCC3)c(N(C)C(C)C)nn2)CNC(=O)CC12CCC2 C(=O)(C(C)CCN(C)C)Nc1cn(C2CN(C(Cn3ncc(C)c3)=O)C2)nn1 C1(C(C)(C)NC(C(C)NC(C)=O)=O)CCN(C(c2csc(C3CC3)n2)=O)CC1 C1(O)(CNC(CN(C(CCC=CC=C)=O)C)=O)CCCCCC1 N1(C(CCC=C(C)C)=O)CC2CC1CN(C(=O)CCC(C)O)C2 c1(OCC)ccc(C(C)SCc2ncc(Cl)n2C)cc1.C(CC=O)C C(=O)(C1=NNC(=O)CC1)NC1C=CCN(C(c2cc(C(=O)OC)c(C)cc2)=O)C1 c1(-c2ccc3ncc(C(=O)NCCC(C)O)n3c2)ccc2c(c1)C(=O)NC2=O C(C(C)(C)CC(=O)NC(c1ccco1)CO)OC.C12(CC1)CC(=O)NC2 N1(C(c2cn(CC)nn2)=O)CCCC(N(C(=O)CCC2(C)CCC(=O)N2)C)CC1 c1(SC)ccc(Cl)c(C(N2CC=CC(NC(C3CC3C(C)C)=O)C2)=O)c1 CCC(CC)C(C)C(=O)NCC1(C(=O)NC2CC(n3cncn3)C2)CCC1 C=CCC(C(=O)N1CCCCC1CCCNC(C1(C)CC1)=O)c1ccccc1 c1(OC)ccc(F)c(C(=O)NC(C)CNC(c2cc(C)ncn2)=O)c1OC Cc1ccc2cccc(CN(C)C(=O)NCCNC(=O)C3CC3)c2n1 C(CCCC=C)(C(=O)N(C(C)C(C)CC)C1CC1)NC(C1(C=C)CCC1)=O CC(N=c1[nH]c(=NCc2nocc2Br)[nH]c2ccc(Cl)cc12)c1ncnn1C N1(C(c2occ(C)c2)=O)CC2(CCC2NC(c2cc(C3CC3)on2)=O)C1 C(=O)(C1CCc2cccc(OC)c21)NC(CCNC(C=C(CC)C)=O)C c1(C(N2CC(CNC(C(c3ccc(F)cc3)C)=O)OCC2)=O)ccc(N)c(O)c1 c1(C(N2C(CNC(CCSC)=O)C(C)CC2)=O)ccc(Br)c2cn[nH]c12 C#CC1(C(=O)NCCC2CC(CO)C2)CN(C(=O)Cc2cn(C)cn2)C1 c1(-c2cn(CC(OCC)OC)nn2)ncc(F)cc1C.N12CCC(CC1)C2=O C1(NC(c2c(COC)nn(C)c2)=O)C2CC3CN(C(=O)C(C4CC4)SC)C1C3C2 c1(C(=O)NC(C(C)NC(c2ccc(Cl)o2)=O)C)nnn2c1CCCCC2 N1(C(C2(OC)CCCC2)=O)CCCC(O)(CCNC(=O)C(O)CSC)C1 c1(C(=O)NCCC(=C)CNC(=O)Cc2cccc(OCC)c2)cncn(C)c1=O CCCC(C)(C)C(=O)NC1CC1CNC(c1ccnc(OC(F)(F)F)c1)=O c1(OC)nc(=NC2CC(F)(CNC(=O)CCc3cn[nH]c3)C2)[nH]c2[nH]cnc12 c1(CN2CC(NC(c3cc(Cl)nc(Cl)c3)=O)C(F)C2)cccc2cc[nH]c12 C1(NC(c2c(COC)cco2)=O)CC(C)CN(C(c2csc(C)c2C)=O)C1 c12ccc(Cl)c(c1)C(=O)NC2.Cc1ccc(-c2cnc(C(=O)NC3CC3)s2)cc1 Cc1nc2cc(C(=O)NCC(O)CNC(=O)CC3CCSCC3)cc(O)c2o1 c1(NC(C(C(C)C)NC(c2cocn2)=O)=O)ccc2c(c1)CCO2 C12(C(N3CC(NC(c4cc(C(N)=O)cc(C)c4)=O)C3)=O)CCOC1CCOC2 N1(C(c2c(C)noc2)=O)CCCC1C1CCCCN1C(=O)CCCCC(C)(C)C C12(CNC(c3c(C)n(C)nn3)=O)CCC1CCN2C(=O)Cn1c(C)c(C)sc1=O C1(NC(Cc2c(C)ccc(C)c2)=O)CCC(O)CN(C(C2CC(C)(C)CO2)=O)C1 c1(NC(CC2CN(C(c3c(C)ocn3)=O)C2)=O)cc(F)ccc1C(F)(F)F Cc1nsc2ncc(C(=O)NCC(=C3CN(C(=O)C=C4CCCCC4)C3)F)cc12 N1(C(CCCOCC)=O)CCN(C(=O)Cc2n[nH]c(C)n2)CC1c1ccncc1 c1(C(N2CC(CCNC(C3(C(C)(C)OC)CC3)=O)C2)=O)[nH]c(O)nc1C Cc1nccc(CCC(=O)N2CC(CCCCNC(=O)Cc3cn(C)nc3C)C2)n1 c1(CC(N2C(C(C)NC(C3CC(OC)C3)=O)CCC2)=O)cccc(F)c1O Cc1nccn1C(C)C(=O)NC1CCC1NC(c1cnc(-c2ccccc2)s1)=O c1(NC(=O)NCCCN(C(C)=O)C)ccc(N=[N+]=[N-])cc1 CC(F)(C(=O)NCC1(F)CC(CNC(c2cnc(Cl)c(Cl)c2)=O)C1)C(F)(F)F N1(C(=O)C=Cc2cnco2)CCC2(CCCN(C(c3[nH]cc4c3CCC4)=O)C2)C1 N1(C(C(F)OC)=O)CCCC2CN(C(C3(C)CCC(C)C3(C)C)=O)CCC12 N1(C(c2nn(CC)c(C)c2)=O)CC2CCC2(CNC(c2nccnc2C)=O)C1 C(=O)(C(C)C(F)(F)F)NCCC(=O)NC(C1CCN(c2c(OC)cnnc2)C1)C C1(C)(C(N2C(C)CC(NC(C3(n4cccn4)CCCC3)=O)C2)=O)C(C)(C)C1(C)C Cc1nc2cc(C(=O)NCCC(C)N(C(=O)CC3CCCO3)C)ccc2n1C CC1(C)CCC(C(N2C3CCC2C(CNC(C2CCCSC2)=O)C3)=O)CO1 N1(C(C(C=CC)O)=O)CC(NC(c2cnn(CCC(C)C)c2C)=O)CC(F)C1 c1(CC(=O)NC2(CNc3nnc(CCO)s3)COC2)csc(CC(F)(F)F)n1 Nc1ccc(Cl)cc1C(=O)NCCC1CCN(C(C2CC=CCO2)=O)CC1 N1(C(=O)C(O)Cc2ccc(Cl)cc2)CC2CCCC2(NC(C23CC(F)(C2)C3)=O)C1 C(=O)(C1CCc2c[nH]nc21)NC(C(C)C)CCNC(c1cc2c(ncn2C)s1)=O CCCCC(CC(=O)N(CCCF)CC)NC(c1cncc2[nH]ccc12)=O C1(O)(CN(C(CCNS(CC)(=O)=O)=O)C)CN(C(C2(C#N)CCC2)=O)C1 C1(C(N2CCC(C)(NC(c3cnc(Cl)s3)=O)C2)=O)CC2CCCCCC12 c1(OCCOC)cccc(CC2(C(=O)OC(=O)CCCOC(C)(C)C)CCC2)c1 CC(C(=O)NCCN1CCC(NC(=O)CCS(C)=O)CC1)C(C)(C)O C(=O)(C1=Cc2ccccc2C1O)NCC(CN(C)C(c1n[nH]c2c1CCCC2)=O)O Cc1cc(C(=O)NCCCCNC(C2(N3CCOCC3=O)CC2)=O)c(C)n1C c1(CC)nc(C(N2CCCC2(C)CNC(C23C=CC(CC2)C3)=O)=O)c(N)s1 c1(C(N2CC(COC)(NC(C3CC3C)=O)C2)=O)sc2cccc(F)c2c1Cl CC(C)(C)C(CNC(c1ccnc(C(F)F)c1)=O)NC(C1(n2ccnn2)CC1)=O CC1(C)CC(NC(C2CCS(=O)(=O)C2)=O)CCN(C(=O)COC(C)(C)C)C1 N1(C(C(CC)F)=O)CC(NC(c2cnc(S)[nH]2)=O)CC12CCC2 c1(CNCCC(C)(C)CO)c(CC#N)cccc1C(F)F c1(C2N(C(C(=O)NCC(C3CCC(C)CC3)(C)O)=O)CC2)ccc(F)cc1Cl CC1(C(=O)NC2CC2CNC(=O)COc2ccc([N+](=O)[O-])cc2)CCS(=O)(=O)CC1 c1(C(=O)NCC(CC)(C)NC(c2ccc(C(C)C)o2)=O)ccc2c(c1F)CCC2 C(C#Cc1cn(CCC2CCS(=O)(=O)C2)nn1)NC(Cc1cc(C(C)C)no1)=O N1(C(C2CCC(C(N)=O)C2)=O)CCCC(C)C1CNC(c1[nH]c(=NC)sc1)=O C1(C(N2CCC(COCCOCC#C)C2)=O)CCCC(C#N)C1 N1(C(C=C(C)c2cccnc2)=O)CCC2(CC1)CC2NC(C1(Cc2cn[nH]c2)CC1)=O c1(C(=O)NCC(C)(CNC(c2cc[nH]c2C)=O)OC)cc(F)cc(Cl)c1 CC12COCC1CN(C(c1ccc(CNC(c3cc[nH]n3)=O)cc1)=O)C2 C1(C(=O)NCC2CCNC2=O)CCN(C(C2(F)CC=CCC2)=O)CCO1 Nc1ccc(OC(CCOCCCCOCOC2CCNC2)=O)cc1 C(C)(CCC(=O)NC1CCCN(C(=O)CSc2nnnn2C2CC2)C1)SC C12(CNC(c3c(C)nn(C)c3)=O)CCCC1CCN2C(c1nccn1C)=O c1(C2(C(N3CC(CC)(NC(c4csnn4)=O)C3)=O)CCC2)ccccc1F N1(CC=O)CC(=O)CCC1=O.C1(CN(CCOCCCO)CC)CSCC(=O)N1 Cn1cc(Cl)c(CC(N2CC(NC(=O)C(C)(C)CO)C(C(F)F)C2)=O)n1 CCCCC(C(=O)NC1(CNC(=O)C(F)=CC2CC2)CCC1)C(C)C Cn1ccc(S(=O)(=O)N2CC3CCC(O)C3(C)C2)c1.c12ccc(cc1)NC(=O)C2 Cc1ncc(C(N2CCC(C(=O)NCC3CCCC3CF)C2)=O)c(=N)[nH]1 C(=O)(CCCC(=O)OC)NCC(=O)NCCCC(CO)NC(CCCC=C)=O C1(NC(c2nc(CCC)oc2)=O)CN(C(=O)C(CC)SC)CC12CC2 c1(C(C(=O)NC)CC(=O)NC)ccc(OCCOCCOCC(C)C)c(OC)c1 S(=O)(=O)(c1cc(C(=O)O)ccc1C=O)N(C)C.C12(N)CC3CC(O)(C1)CC(O)(C3)C2 Cc1cc(Cl)c(C(=O)NC2CCC(N(C)C(c3sccc3Cl)=O)CC2)s1 CC1(NC(=O)CC2CCCCO2)CC(C(=O)NCC2C3COCC23)C1 CCC(C)(CNC(=O)C(C)N1CC(C)C1)C(=O)NCCC1CC=CC1 c1(C(C)NC(c2nnnn2C)C2CC(OCOC)C2)cccc(F)c1C N1(C(CCNC(=O)NC)=O)CCC(NC(=O)Cc2cccs2)C1C(C)(C)C N1(C(C2N(CC)CC2)=O)CC(NC(=O)CCc2c(C)noc2Cl)CC12CCC2 N1(C(c2ccc(CNC(CSCC=C)=O)cn2)=O)CCCC(C)(C)C1C c1(C(=O)NC2C(NC(C3(COC)COC3)=O)C2)cc([N+](=O)[O-])cc(C)n1 CCCC(O)C(=O)NC(c1ccc(-c2cnn(CC#N)c2)cc1)C.C1CC1 C1(NC2(c3c(OCC(C)C)cccc3)CC2)CCN(CC=CCl)CC1C C1(C)(CNC(c2c(C)coc2C(C)C)=O)CC(F)(F)CN1C(=O)CC1CCOC1 c1(SC)ccc(CNC(=O)C(=O)NCC(=O)Nc2cc(Cl)c(Cl)s2)cc1 Cn1cc(NCc2ccccc2)c(C(F)F)n1.C1(CO)CN1 CN1CC(=O)Nc2ccc(C(=O)NC3CC(NC(c4cc(N)ccn4)=O)C3)cc21 C1(CC(=O)NCCCC(=C)Cl)C2CCCC2N1C(=O)C=CCN1CCC1 c1(C(=O)NCC(CC)NC(=O)CC2(O)CCC2)cccc(OC(F)F)c1 N1(C(c2ccc(CC)s2)=O)CC(C)N(C(=O)C(C)CC(N)=O)CC1C Cc1occc1C(=O)NCC(=O)N(CC(=O)NC(C)C(O)CO)C(C)C N1(C(CCC(C)SC)=O)CC2CCCC2(NC(=O)Cc2c[nH]c(=N)nc2O)C1 Cc1ccc(-c2ccnn2-c2cc(C)nn2C)c(OCCC(C)C)c1 C1(C(=O)NC2(CC=C)CN(C(c3nnn(C)c3N)=O)C2)CC(C(C)C)=NO1 N1(C(c2cc(C)nnc2)=O)CCC(C2CC2)(NC(C2CCCOC2)=O)C1 c1(C(=O)NC2(COC)CN(C(C3C(OCC)C3)=O)C2)c[nH]c2cc(C)ccc12 C1(C(=O)NCc2scc(C)c2)CCN(C(=O)CCc2nc(=N)[nH][nH]2)C12CC2 N1(C(CCCOC(C)=O)=O)CC(CNC(=O)C(CO)C(F)(F)F)C2(CCC2)C1 C1(CNC(c2cc(OC)ns2)=O)CCC(C)CN1C(=O)CCSC1CCCC1 c1(C(N2CC3(N(C(C(C)CO)=O)CC3)C2)=O)ccc(S(=O)(=O)NC(C)(C)C)cc1 c1(CC(=O)NC2C3CC(NC(=O)C(O)CN4CCCC4)CC23)cccc(O)n1 c1(C(=O)NCC2N(C(C(F)OC)=O)CCC2)cncc2c1CCNC2=O c1(CNC(=NCC=C)NCC(C)C(F)(F)F)nnc2n1CCOC2 c1(C(N2CCC(CNC(C3CC=CC3)=O)C2)=O)cccc2c1OCCO2 CC1(C)CC(O)(CC(=O)NCCC2CCN(C(C3CC4CCC(C3)O4)=O)C2)CO1 c1(OC(C)(C)C)ncc(C(N2CC(NC(c3cnc(Cl)[nH]3)=O)C2)=O)cn1 N1(Cc2ncc(OC)nc2)CCC2(CC2C(=O)Nc2sc(C)nc2C(F)(F)F)C1 c1(CCC(=O)NCC2(F)CC(NC(C(CSC)C)=O)C2)cccnc1Cl Cc1ccc(CN=C(NCC2CCCC2N(C)C)NC(c2cccs2)C)c(C)c1 c1(C(N(CC(=O)NCC(=O)NC2(C(=O)OC)CC2)C)=O)cc(C)n(C)n1 C1(F)(C(=O)NC2(CO)CC2)CCCN(C(=O)C(F)=CC2CC2)C1 CC(C)(CC(=O)NC1(CNC(=O)CNc2cc(F)cc(F)c2)CC1)C(F)(F)F c1(OC)nc(NC2CN(C(=O)C(=O)NCCCC#N)CC2(O)CO)ncc1Cl CCC(C)CC(=O)C(=O)NC(C(=O)NC1(c2cc[nH]n2)CC1)C1CCC1 N1(C(c2c(C)n(C)cc2)=O)CCC2(CC2)CC1C(=O)NC1(C(N)=O)CC1 c1(NC)c(C(=O)OCC)cc([N+](=O)[O-])cc1Br.N12CCNCC1C2=O C(=O)(C(C)S(N)(=O)=O)N1C(CN(C(CS(CC)=O)=O)C2CC2)CCC1 N1(C(c2cc(CC)on2)=O)CCc2ccccc2C(NC(=O)C(C)C2CCC2)C1 N1(C(c2cn(CC)nc2)=O)CC2CC(C)N(C(=O)C3=CCCCCC3)C2C1 CC(O)C(=O)NNC(=O)C12CCC(OC)C1CN(C1CN3CCCCC3CO1)C2 C(=O)(CC1CCOc2ccccc21)N(CCNC(C1C(C)C1)=O)C(C)C N1(C(c2nc(C(C)=O)sc2)=O)CCC2CN(C(=O)CC3COCC(C)(C)O3)CC12 C1(C(=O)NC2CC(CNC(C3(C#N)C(C)C3)=O)C2)CC2(C1)CC1(CC1)C2 c1(CNC(=NCC)NCC2COC(=O)O2)cc(C)cc(Br)c1 N1(C(CC(CCC)CC)=O)CCCC2CN(C(C3CC4(CCOCC4)C3)=O)CC12 C12(NC(C(CC)C)=O)CCN(C(c3cc[nH]c4nccc3-4)=O)CCC1C2 c1(C(=O)NCC(CNC(c2cccc(COC)n2)=O)O)ccc2c(c1)OCCO2 C1(C(N(CCNC(C2(OCC)CCCCC2)=O)CC)=O)OCC2CCCCC12 N1(CC)CCCC(NC(c2cnc(C3CCNCC3)[nH]2)=O)C1 C(=O)(C1OCCc2ccc(C)cc21)N1C(CNC(C=C(CC)C)=O)CCC1 N1(C(C=C(CC)C)=O)CC(NC(c2cnoc2-c2ccccc2)=O)C(O)C1 C#CCC(CC(F)F)C(=O)NC1CCCCC1NC(=O)C(N1CCOCC1)C CC1OCCN(C(=O)CCC2CC2(F)F)C1C(N1CCCC(C)CC1)=O Cc1ccc2c(c1)C(NC1CCCCC1C(F)(F)F)CCC2 C1(C(N2CCC(O)C2)=O)COCCC12CN(Cc1ccc(Cl)nc1)C2 C1(C)(NC(CC(C)(C)OC)=O)CCN(C(=O)C(Cc2cccc(Cl)c2)NC=O)CC1 c1(OC)cc(C(N2CC(C(=O)NCC3CCCOC3)C(F)C2)=O)ncn1 C1(CNC(C(CC)(C)C)=O)CCCC2CN(C(c3cc4ncccc4o3)=O)CC12 c1(C(N2CC(CN(C(=O)CC3CC(F)C3)C)OCC2)=O)[nH]nc2c1COC2(C)C Cc1cc(C(=O)N(CCCNC(C2CCCC(C)C2)=O)C)cc(Cl)c1 S(=O)(=O)(c1ccc(NC(CO)C2(C)CC2)c(C#N)c1)NCC(C1CCCCC1)C c1(CCNC(=O)C(N2CCCC(NC(C3CC4CC3C4)=O)C2)=O)ccc(F)nc1 S(=O)(=O)(c1c[nH]c(=NCCCN)cc1C)NC(c1c(C)n(C)nc1)C.C(N)(=O)N N1(C(C(C)(C)Br)=O)CCOC2CN(C(c3cnn(-c4ccccn4)c3)=O)CC12 C1(F)(CNCCCNC(CNC(CN(C2CCCC2)C(C)=O)=O)=O)C2CCCCC12 C1(CNC(C2ON=C(C)C2)=O)CN(C(c2cc(Cl)n(C)n2)=O)CCC1(F)F C1(NC2CN(C(COC)=O)C2)CC2(C1)CC(NC(=O)C(C)n1cccn1)C2 C1(CCOC)(NC(c2cc(C)sc2C)=O)CCN(C(=O)Cc2csc(C)n2)C1 c1(NCC)cccc(F)c1C(N1CC2(C1)CN(C(=O)CC1CCN(C)C1)C2)=O C1(C(=O)NCc2c(C(=O)NC3CCC(OCC)CC3)ocn2)CC(C)CC(C)C1 C(=O)(CC(C)CC(C)C)NC1(C(C(=O)NCCCCC)C)CCC1 C(=O)(CC1COc2ccccc21)NCCNC(C(c1cccc(C)c1)C)=O N1(C(C2CCN(C)CC2)=O)CCOC(C)(CNC(C2(S(N)(=O)=O)CCC2)=O)C1 C1(C(=O)NC(CC)CN(C)C(C2CCCCN2C)=O)CCC([N+](=O)[O-])CC1 c1(C(N2CCC(N(C(=O)CCCC(C)(F)F)C)C2)=O)cnc([N+](=O)[O-])n1C c1(OC(C)C(=O)NC2CCC(n3cccc3)CC2)ccc(Cl)cc1Cl N1(c2nc(C)nc(Cl)c2)CC2CCN(C(C34CC5CC(C(=O)N3)C4C5)=O)CCC2C1 C#CC1(NC(=O)C(F)CC2CN(C(=O)C(C)(O)C3CCC3)C2)CCC(C)CC1 N1(C(CC=CCC)=O)CCC2(CC1)CC2C(N1CCC(C)C1C)=O NS(=O)(=O)C1CCN(C(=O)C(=O)NCCSc2ccccc2)C1 CSC1=C(C(=O)N2CCC3(NC(=O)C(N4CCC(C)CC4)=O)CC3C2)CCCC1 C1(NC(c2c(CC)nco2)=O)CN(C(c2c(F)cc(C)cc2F)=O)CCC1CO c1(C(N2CC(COC)(COCCOC)C2)=O)coc2cc(C)ccc12.C1(=O)CN1 C1(C(N(C)CC2(NC(c3csc(=N)[nH]3)=O)CC2)=O)CCC(C(F)F)CC1 c1(CNC(C2CCN(C(C)=O)C2)=O)nn(C)c2c1CCC2.c12csc(c1)NC2=O C1(C(N(CC(=O)Nc2cnn(C)c2)C)=O)CCN(Cc2ccc(Br)s2)C1 N1(C(C23CCCC(OC)(C2)C3)=O)CC2CCC2(CNC(C2CC(CC)(CC)C2)=O)C1 C(CN=C(NCC1CCOC1)NCC1CSCCO1)C1(O)CCCC1 c1(COC)n[nH]c(=NCC2(F)CCN(C(=O)CC3CS(=O)(=O)C3)CC2)s1 c1(COCC(C)N(C(c2[nH]nnc2C)C(=O)NCS)CCC)ccccc1OC c1(CNC(C2(C)CCN2C(C2CCC(=O)N2)=O)=O)ncn2ccccc12 Cc1cn2c(n1)CC(C(=O)N(C1CCCCC1N(C(=O)C(O)CN(C)C)C)C)C2 C(CCCC(=O)NC1(CN(C(=O)C(C)CCc2ccccc2F)C)CC1)OCC N1(C(C2(NC(c3c(C)snn3)=O)CCC(C)(C)C2)=O)CC2CCC1C(O)C2 C1(C(=O)OC)CCC2(CCN(C(C3CCCC3(C)C)C(=O)NC3CC3)CC2)O1 N1(C(c2cc(C(C)NC(c3ccnc(SC)n3)=O)on2)=O)CCC(SCC)CC1 C(C)(C(CO)NC(c1cc(-c2csc(=N)[nH]2)c[nH]1)=O)NC(C1(OC)CC1)=O CCC(C)CC(C(=O)NC1CC(O)C1OC)NC(c1nnc(S)n1C)=O Cc1c(C(=O)NCCC(C)NC(c2ccn(CCF)n2)=O)c(C(F)F)nn1C c1(OCC(=O)NC2(C)CC(NC(C(c3cccnc3)C)=O)C2)ccc(F)cn1 c1(CC)n[nH]c(CC)c1CC(=O)NC1CC1NC(=O)Cc1cc(C)[nH]n1 n1(CC(=O)NCC(CNC(c2ccc(O)cn2)=O)OC)nc(C)ccc1=O N1(C2CCC(NC(CC3(C#N)CC3)=O)C2)CCN(C(=O)C=Cc2ccoc2)CC1 C1(c2nnnn2C2COC2)(Nc2c(C(=O)OC)n(C)nc2C)CCCCCC1C c1(CN2CCN(S(C3(CC)CC3)(=O)=O)CC2C#N)c(Br)cc(Cl)c2ccccc12 C1(C(N2CCC(N3CC=CC3)C2)=O)(CC)CCN(C(c2cccc(OC)c2)=O)C1 C1(CC(N2C(CNC(C(C)=C(CC)C)=O)CCC2)=O)NC(=O)C(C)NC1=O N1(CC)CCCCC1C(=O)NC(CCCOC)CNC(=O)CCNC(=O)OCC C1(NC(C(C)OC)=O)COC2CN(C(c3c[nH]c(=N)nc3C)=O)CC12 N1(C(c2cnc(C)s2)=O)CC(C(=O)NC(C(O)CO)C2CC2)C(C2CC2)C1 N1(C(c2c(OC)nsc2)=O)CC2CCCC1C2CNC(c1cc(O)nc(Cl)c1)=O CCCCC(C(=O)OCC)N1CCC(C(=O)NC2CC(F)(F)C2)(OC)CC1 c1(C(=O)NCCOCCCNC(C2(COC)CCOC2)=O)ccc2n[nH]cc2n1 C(=O)(CS(=O)(=O)CC)N1CCC(CC(=O)NCC(COCC)(C)C)CC1 Cc1cc(C(N2CC3CC(C2)N3C(c2cn3ccsc3n2)=O)=O)cc(Cl)c1 c1(C(N2CC(C)(CNC(c3c(C)nc(C)s3)=O)OCC2)=O)cc(C#N)ccc1O c1(CCC(=O)NC2CCN(C(c3ccc(OC)nn3)=O)C2)ccc(Br)c(C)c1 c1(CCNC(=NC)NCC(n2cc(C(F)(F)F)cn2)C)ccc(F)cc1 n1(C(CC)C)ncc2cc(C(=O)NCCC(C)(C)CNC(=O)C(C)C#N)cnc12 C1(C(N2CCC(C)(NC(=O)Cc3ccc(Cl)s3)C2)=O)CC12CCOCC2 c1(OC)cc(C#N)c(CC(N2C3CCC2CN(C)CC3)=O)cc1OC CC(C)C(CN(CCCN1CCOC1=O)C)c1nn[nH]n1 C1(CNC(CC)=O)CCC(NC(=O)CC2CC(O)C2)CC1.C(C)(C)OCC c1(C(=O)NC2CC(CNC(C(C)Cc3cccnc3)=O)C2)nccnc1C(N)=O C(=O)(C(CO)C(C)(C)C)N1C(C)(C)C(c2ccc(F)c(-n3cccc3)c2)C1 C1(C)(CNC(CCCCN(C)C)=O)CC(F)(F)CN1C(=O)CC(O)CN(C)C C#CCC(C)C(=O)NCCCCNC(c1cn(C)nc1-c1cccs1)=O CCC(CC)(C(=O)N1CC(CNC(C2CCN(C)C2)=O)C(F)(CO)C1)OC CC1CN(C(c2cnc(S)[nH]2)=O)CC(CCNC(C2(CN(C)C)CC2)=O)O1 N1(C(C(C=C)O)=O)CC2CN(C(=O)CCc3cncs3)CC2(C)C1 N1(C(C2=NOC(C)C2)=O)CCc2c(NC(=O)C3=CC(O)CCC3)cccc2C1 N1(C(C(C)NC(C)=O)=O)CCC2(C1)CN(C(=O)CCOSc1ccc(OC)cc1)C2 C1(C)(N(C(c2sc(I)cc2C)=O)Cc2ccc(F)nc2C)CCCN(CCC)C1 C1(C)(COC)CC(F)(F)CN1C(=O)NC1CC1C Cc1ccc2nsnc2c1C(=O)NCCC(C)CCNC(=O)C(=O)NCC(F)F C1(C(N(C(CCN(C(=O)CSC(F)F)C)c2cccs2)C)=O)CC2CCCCC12 Cc1cnc(Cl)n1CCNC(c1ccccc1SC1CCCC1)=O C1(OC)CN(C(=O)C(c2ccccc2)OC)CCC1CNC(=O)C(C)CC(C)C N1(Cc2cccc(COC)c2)CCC(O)(Cc2ccc(C)c(F)c2)CC1 C1(CCNC(C=NOC)=O)CN(C(=O)CCc2csc(C)n2)CC(C)O1 C1(C)(C(N(C(CC)C(=O)NCC(=O)N(C)CC)C)=O)CC(C)=NO1 C1(C)(NC(C(F)=CCC)=O)CCCN(C(C23CCCC2(C(N)=O)C3)=O)C1 C1(CNC(=O)CC2CCCCO2)CCC(NC(=O)Cc2coc(C(F)F)n2)CC1 c1(C(N2CCN(C(C(CCC)C(=O)OC)=O)CC2)=O)ccc2nc(CO)[nH]c2c1 c1ccc(Cl)cc1.C(C(O)CCNC(C1CCCN1C(N)=O)=O)NC(C(C)=CC)=O c1(C(C(=O)NC)=O)ccc(Cl)s1.C(C(=O)NCC1CC1)(C1CCOC1)OCC N1(C(COCCC)=O)CCC(C)CC1C(=O)N(CCN(C)C)C C1(OC)CC(NC(=O)CSC(F)F)CN(C(C2CCCS2(=O)=O)=O)C1 C1(CNC(=O)C2=NOCC2)CCN(C(=O)CCN2C(=O)CNC2=O)CCC1(F)F c1(OCCCN)ccccc1NC(=O)NC1(c2ccc(Cl)cc2)CC(C(N)=O)C1 Cc1cc(C(=O)NCC2(F)CC(NC(c3ncccc3Cl)=O)C2)cc(F)c1 CN1CCC(C)(C(N2CC3CC(CNC(=O)CCc4ccsc4)C3C2)=O)CC1 C(=O)(CCS(=O)(=O)NC=O)NC1CC2C(NC)C2C1.C1(=O)C(C)N1 CCCCC(CC)C(=O)N1CCC(CO)C(NC(=O)CC(CCC)OC)C1 N1(C(c2ccc(S(C)=O)cc2)=O)CC(C2CCCN(C(=O)C3=CCC3)C2)C1 c1(NC(C(=O)NC(CNC(c2cc(C(C)=O)on2)=O)CO)=O)ccc(F)cc1 c1(C(N2C(C(N(CC(C3CCC3)OC)C)=O)CCCC2)=O)cnc2n1CCC2 c1(NC(=O)NCC2CSCCS2)cnccc1Br C(CCCCCCO)NC(C1N(C(Cc2cccc(C)c2)=O)CSC1)=O N1(C(CSCC(C)C)=O)C2CCC1C(CNC(=O)Cn1nc(O)ccc1=O)C2 C(=O)(C1COc2ccccc21)NCCC(C)(C)NC(c1cccc(C)c1F)=O C1(NC(C(CC(N)=O)NC(C2CCC(O)CN2C)=O)=O)CC2CC1CC21CC1 CC1CC(CNC(=O)CC2CC(=O)NC(=O)C2)CN(C(C2CSCCS2)=O)C1 c1(OC)cccc(F)c1CC(N1CC(NC(=O)C(C)OC(C)=O)CC(F)C1)=O c1(N2CCC(COC)C2)nc(=NCC2(S(C)(=O)=O)CC2)[nH]c2c1CCCCC2 C1(C(N2CCCC(N(C)C)C2)=O)(CC)CCN(C(C2CCC3(CC3)C2)=O)C1 c1(CCCC)ccc(S(=O)(=O)NCC(O)CC=CCOC)cc1 c1(OCC)cccc(C(=O)NCC2C3CN(C(=O)C(C)c4ccsn4)CC23)c1 C1(C(N2CCC(CNC(c3c(CCC)occ3)=O)C2)=O)Cc2cc(C)ccc2S1 N1(C(C2C(=C)C2)=O)CCC2CN(C(c3cc(F)ccc3C3CC3)=O)CC2C1 c1(C(=O)OC)cccc(-c2nnc(N3CCCC34CC4)n2CC(F)(F)F)c1 c1(C2C(C(=O)O)C2)ccc(-c2ccsc2)nc1.C12CCCN(C1)C2 C(CCSC)(C(=O)N1CCCC1CNC(N)=O)NC(c1c(CCC)nco1)=O C1(NC(c2ccc(CC)c(F)c2)=O)CC1C1CCN(C(=O)C(C)(O)C2CC2)CC1 CC1CCN(C(c2coc(-c3ccsc3)c2)=O)C1c1cn(CCO)nn1 C#CCC(C)(C)C(=O)N1CCN(CC(=O)NC(C2(O)CCCCC2)C)CC1 CC(C)C(O)C(C)C(=O)NC1(CNC(=O)CNC(N)=O)CC1 N1(C(CC(C(=O)OC)C)=O)CCC2(CC1)CC(NC(C1CCNC(=O)C1)=O)C2 CC1CCCn2c(C(N3CC(CNC(=O)CN4CCCC4=O)C(C)C3)=O)cnc21 c1(OC)cc(CNC(C2(C)CCCN2Cc2ccc(C#N)cn2)=O)ccc1O C12(CNC(CCSCC#C)=O)CC(CNC(C3CCC3OCC)=O)(C1)C2 C1(O)(C(=O)NCC(CN(C(C(CC)(C)O)=O)C)(C)C)CC2CCC1C2 c1(CS(C)(=O)=O)nc(C(=O)NC2(CNC(C3(CF)CCC3)=O)CC2)cs1 C(CC(=O)NC1CCCN1C)(CCNC(C1CC1c1nc[nH]n1)=O)OC N1(C(=O)COC2CCOC2)CCC2(CC1)CC2CNC(c1ccc(CC)o1)=O c1(C(N2CC(C(C(=O)N(CCCCCO)C)O)C2)=O)cccc(F)c1 Cc1ccc(C)c(C(=O)NCC2C(C)CCN2C(c2cnc(C#N)s2)=O)n1 C1(NC(CCCCSC)=O)CN(C(=O)C(=O)NCC2CC2)CCC1CO C1(C2CN(C(c3cc(C(C)(C)C)on3)=O)C2)(NC(C=Cc2ncc(C)[nH]2)=O)CC1 C1(OC)CC2CC(c3nnnn3C3(C)CC3)(NCC3(C)CNC(=O)O3)C2C1 C1(CNC(C(=CC2CCC2)C)=O)CC2CCC1N2C(=O)Cn1ncc(Br)c1C CCC(C)(C)C(O)C(=O)N1CCCC(N(C(c2cc3c(s2)CCC3)=O)CC)CC1 C=Cc1cnn(C)c1C(=O)N(CCCNC(=O)CCc1cnn(C)c1C)C1CC1 c1(C(C(=O)NCC2CC(NC(CN(C)C3CC3)=O)C2)(C)O)cccc(F)c1 C(=O)(C(C)C(O)CCCCC)NC1CC2CN(C(C(CC=C)(C)C)=O)C(C1)C2 C1(C(N2CC(NC(CCC=C(C)C)=O)C2)=O)CCS(=O)(=O)C1(C)C C1(O)(C(C)NC(=O)C(F)n2cccn2)CN(C(c2coc(C3CC3)n2)=O)C1 CC1CCN(C(c2ccc(O)nc2)=O)C(C(=O)NCCC(C)(C)C)C1 N1(C(c2nnc(C)nc2)C(=O)Nc2ccccc2)CCC(C2(C)CC2)C1 Cc1cnc2cccc(C(N3CCCC3Cc3ccc(F)cc3)=O)n12 CCCCCC(O)CC(=O)NC(C)(CNC(=O)CCCS(N)(=O)=O)CO C1(O)(C(=O)OC)CCCN(C(C23CC(C2)C(c2ccccc2)N3)=O)C1 C#Cc1cnc(C(N2CC3CCC3(CCNC(C3(CC)CCC3)=O)C2)=O)c(C)c1 N1(C(COc2cc(C)on2)=O)CCCCN(C(=O)C(=O)Nc2cnn(C)c2)CC1 C(=O)(C(CCC(C)(C)C)N1CCCC(c2cnn[nH]2)C1)NCCCOC N1(C(c2cc(C)c(Br)nc2)=O)CCN(C(=O)C(F)CC2CCC2)CCC1C CC(O)CCCCCC(=O)N1CC(C)(NC(c2ccc(NC(N)=O)cc2)=O)C1 C1(NC(C2=NNC(=O)C2)=O)COC2(CCN(C(c3cncc4nc[nH]c34)=O)C2)C1 N(C1c2ccccc2CC1NC(=O)C=C(C)Cl)C(C(CC=C)(F)F)=O C1(NC(C(C)(C)NC(=O)NCC)=O)CN(C(=O)CCF)Cc2nccn2C1 c1(OC)nn(C)cc1C(=O)NC(C)CC(C)NC(C1CC(=O)N(CC(C)C)C1)=O C1(CC(=O)NCCC(N)=O)CCCCN1C(c1ccccc1-n1cncn1)=O c1(CNC2C(OC)C(O)C2)nc2cc(F)cc(F)c2o1 c1(C(N2CCOCC2)C)nc(-c2ccsc2)n(CC2CCC2)n1 CC1(C)OCC(CS(=O)(=O)NC(C2CCC(C3CC3)O2)=O)C(O)CO1 N1(C(c2scc(CNC(c3c(C)nns3)=O)c2)=O)CCC(CO)C(C)C1 Cc1cccc(C(O)C(N2CCC(C)C(NC(C3C(C)C3C)=O)C2)=O)c1F C1(C(=O)NCC(CCCC)O)N(C(=O)C(=Cc2cn[nH]c2)C)CCC1(C)C c1(N(CCOCC(=O)N(C(CCC)C)C)C2CC2)cccc(C(=O)NC)c1 S1(=O)(=O)c2ccc(cc2)COC(=O)CCCN1CC.C(C(C)(C)C)CC.C(C)(C)(C)O C1(NC(C(CC)OCC)=O)CC2(C1)CC(NC(C1CCC3(CC1)CC3)=O)C2 N1(C(C=CCC)=O)CCCC(C2CCN(C(=O)Cc3ccc4nonc4c3)C2)C1 O=C(CC1OCCc2sccc21)NCC12CC(CO1)N(C(c1cnccn1)=O)C2 O=C1CC(=O)CC(C(=O)NC2CCCCC2CC(=O)NCCC2CCCCC2)C1 CCCCC(CNC(=O)CN(C)C(c1ccsc1C)=O)CCC C1(C(=O)OCCC(=O)NCC#C)CC(=O)N(C)C1c1cnn(C)c1C c1(C(N(C(CNC(C2C(C=C)C2)=O)C)C)=O)csc(C2CCCCC2)n1 C(CC(=O)N1CC(=O)NCC1C(F)(F)F)(C(F)F)NC(=O)C=CC(F)F Cc1cc(N)cnc1Nc1ccc(C)c(C(N2CCCCC2)=O)c1 c1(C(N(C(C)CNC(C2(C)CCCS2)=O)C)=O)nccc2ccncc12 C12(C(=O)NCC3C(C)(C)N(C(c4ccc(N)cc4)=O)CC3)CCC(F)(CC1)CC2 c1(C(=O)NCC2N(C(C(CC)SC)=O)CC(C)(C)C2)cc2c(=O)ccn(C)c2s1 C(=O)(C1CCCc2nn[nH]c21)NC1(CO)CCN(C(C2(CC=C)CCC2)=O)CC1 N1(CC(=O)N(CCCN(C)C)CCNC(=O)C(F)=C2CCCC2)CC(=O)NC1=O Cc1cc(CCC(=O)NCC(C)NC(=O)CCC2CCC(=O)N2)c(C)s1 C12(C(N(C3C(C)CC3)C(C)C3CC3)=O)C3C4C1C1C2C3C41C C(=O)(C(C)(C)c1ccno1)N(C1(C(=O)OC)COC1)C(=O)Cn1cc(Cl)cn1 N1(C(c2c(CCC)nns2)=O)CCN(C(=O)Cn2ccc(C)cc2=O)C(CO)C1 c1(OC)cccc(C(N2CCCC2(C)CNC(=O)CC2CSCCS2)=O)c1 C(=O)(C(C)C(O)C(C)CC)NC1(C(N2CCC(OCCC)CC2)=O)CC1(C)C.C(=O)OC C#Cc1c[nH]nc1C(=O)NCc1cncc(C(N2CCC(OC(C)C)C2)=O)c1 Cc1cc(-n2cccc(Oc3cnc(C(C)O)nc3)c2=O)cc(C)c1 C(=O)(C1=CCC2CCC1N2C(=O)C(n1ccnc1C)C)N(CC(=O)NC)C C1(N(C(C(C)OCC2CC2)=O)C)CCCCN(C(=O)C=Cc2ccccc2)C1 Cc1ccc(CNC2C=CC(C(=O)Nc3ccnc(C(F)F)c3)C2)cc1Cl N1(C(CC2C(C)CCCC2)=O)Cc2occ(C(N3C(CO)CC3C)=O)c2C1 C(c1cccc(Cl)c1Cl)=CCN1CCC(NC(c2cc(C3(O)COC3)on2)=O)C1 c1(CC(=O)NC(CC)CN(C)C(C2CC2C)=O)coc2cc(CC)ccc12 N1(C(CCCC2C(C)C2)=O)CCC2(CC2)CC1C(N1CC2CCOC2C1)=O CC(C)C(CO)C(=O)NCCC(C)(C)NC(=O)C(C)CCNC(=O)OC(C)(C)C C(=O)(CCCC(=O)NC(C)CCCNC(c1coc(C2CCC2)n1)=O)NCCC c1(C(N2CCC2C)=O)cccc(Cl)c1C(N1CCOC(CO)C1)=O.CO C1(CNC(c2cnc(OC)c(C)c2)=O)CN(C(c2ccc[nH]2)=O)C2CCCC2O1 CC1(C)CC(CNC(=O)C=CSc2ccccc2)CN1C(c1cnsc1)=O c1(OC)cc(OC)c(CN2CCOC(C(=O)N(CCC#N)C(C)C)C2)cc1Br N1(C(C2CC(OC)C2)=O)CC(NC(C2CCCN2N=O)=O)CC12CCCCC2 C1(C(=O)NCC(C2CCC2)N(C)C(c2cncnc2)=O)OCC2CCCC12 N1(C(CC(CC)C2CC2)=O)CCCC(N(C)C(C2(F)CCCCC2)=O)CC1 c1(OC)cc(C(=O)NC2CCN(C(=O)CCC3CC3(F)F)C2)cc([N+](=O)[O-])c1N N1(C(C2C(CNC(C(C)C)=O)CCO2)=O)CCS(=O)CC1C N1(C(Cc2n(C)ccc2)=O)CC2ON=C(CNC(=O)Cc3ccc(Cl)cc3)C2C1 c1(C(N2CCCC(CNC(CC(CC)OC)=O)C2)=O)c(N)sc(C)c1C c1(OCC)cc(C(N2C(CNC(=O)C=CC(C)C)CC3CC23)=O)ccc1[N+](=O)[O-] C(=O)(C1=CCCCO1)N(C)CC1CCN(C(Cc2cnc(C)[nH]2)=O)C1 N1(C(C2C(C3C(C)C3)C2)=O)CCC2(CC1)CN(C(C1CC(F)(F)C1)=O)CC2CO N1(C(C=CCOC)=O)CC(NC(c2cccc(-n3cncn3)n2)=O)C2(CCC2)C1 c1(C(C)NC(C(C)(N(C(C(COC)N(C)C)=O)C)C2CC2)=O)nccc(C)n1 Cc1ccc(C(=O)NCC2(C)CN(C(c3cn(C)nc3Cl)=O)C(C)(C)C2)c(N)n1 CC1=CC(NC(=O)C(CC2CCOCC2)NC(=O)C(C)C#N)CCC1 c1(NC)cc(C(=O)NCC2C(NC(c3ncc(NC)nc3)=O)C2)cnc1O C1(CNC(N2CC(C(=O)NC)C2)=O)(Cc2ccccc2)CCOCC1 S(=O)(=O)(c1ccc(Cl)cc1)N(C1CCS(=O)(=O)C1)CC(F)F N1(C(=O)CCc2ccon2)CCN(C2CC(NC(C3(O)COC3)=O)C2)CC1 c1(-n2ncc(C(=O)NCCC3(NC(CC=C=C)=O)CC3)n2)ccc(F)cc1 Cn1ccc(CC(=O)NCc2cc(C(=O)NCCC3CCCCO3)no2)n1 c1(C(N(CCn2cc(C(CC)O)nn2)C)=O)cccc([N+](=O)[O-])c1Cl C(=O)(C(O)(C(F)(F)F)c1cn[nH]c1)NCCC1(O)CN(C(C(C)=C(C)C)=O)C1 N1(C(c2cc(CCC)[nH]n2)=O)CCCC(C(=O)NCc2onc(C)c2C)CC1 C(C(C)C(C)C(=O)NC(C)(C)CC(=O)NCCC(C)O)OC N1(C(COCCCC)=O)CCC2CCN(C(=O)C=CCOC)C2C1 CCC(CNC(=O)C(C)C(C)n1cccn1)(CC)NC(c1ccc(CO)s1)=O c1(OC)cc(C(N2CC(OCC(=O)NC3CC3c3cccnc3)C2)=O)nn1C c1(C(=O)NCC(CC=C)NC(=O)C(CC)SC)ccc2cc(Cl)ccc2n1 N1(C(C2(C)CCCS2)=O)CCCC(O)(CNC(c2cncc(Cl)c2)=O)CC1 CC1(CNC(=O)Cc2cc(F)ccc2F)CN(C(=O)C(F)CC2CCC2)CCO1 N1(C(c2cc(OC)nn2C)=O)CC(NC(c2n[nH]c(C3CC3)n2)=O)C2CCCCC12 c1(C(=O)NC(CCNC(c2c(C)cccc2C)=O)C)ccc(C#N)nc1O O=S(=O)(c1cncc(Br)c1Cl)NCc1csc(-c2ccccn2)n1 C1(C(=O)NCC2(OC)CCC2)CN(C(C2CCC(N(C)C)C2)=O)CC(C)(C)C1 C=C(C)CCC(=O)NCCC(C)(C)NC(c1ccccc1-c1ccncc1)=O CN1CCN(c2cc(C(=O)NCC3(NC)CC(F)(F)C3)ccn2)CC1 CC#CCCCC(=O)N1CCC(NC(c2ccncc2SCC)=O)C(CO)C1 N1(C(C)C)CC(NC(N2CCC(O)(CN(C)C)C2)=O)CC1=O.c1cccc(F)c1 c1(C(N(CC(CNC(C2(COC)CCC2)=O)C)C)=O)ccc2cc[nH]c2n1 C1(CNC(=O)CCN2CCC2)CC2(CCN(C(C3CCCO3)=O)CC2)CO1 Cc1[nH]c(C)c(C(=O)NCC2(O)CC(C(=O)NCC3(O)CCC3)C2)c1C c1(CNCc2cccc(C(N3CCN(C)CC3)=O)c2)ccc(F)c(F)c1F C1(C(N2CCC(NC(Cc3nnc(C)o3)=O)(CO)C2)=O)CCn2c(C)cnc2C1 N1(C(c2ccc(OC)s2)=O)CCN(C(=O)COCc2nc(C)no2)C2CC12 C(=O)(C(C)(C)CC(=O)N1CCC2C(C1)CN2C(C1CC(=O)N(C(C)C)C1)=O)OC C(=O)(CCCS(C)(=O)=O)N(C)CCC1CCCCN1C(C1CCSC1)=O Cc1sc(C(=O)NCC(C)CNC(c2cnn(C)c2CC(C)C)=O)nc1O c1(OCC(=O)NC2C(NC(c3cc(C)no3)=O)C2)c(F)cccc1F N1(C(c2cc(C(C)=O)oc2)=O)CC(NC(=O)CC2(N(C)C)CC2)CC(F)(F)C1 C1(C(N(CC)Cc2ncccn2)=O)CCCN(C(C2(CCCF)CC2)=O)C1C CC(C)C(O)C(=O)NCCC1(CC(N2CCC(n3cccn3)C2)=O)CC1 N1(C(C2CN(CC)C(=O)CC2)=O)CCN(C(=O)C2=CCCC2)C2CS(=O)(=O)CC12 C(C(=O)N1CCCC1CCNC(=O)Cn1nc(C2CC2)cc1C)(C(C)C)SC C1(O)(C(C)CNC(=O)C(O)CC2CCCCC2)CCN(C(=O)Cc2cc[nH]c2)C1 N1(NCC)CC2(CCC(Nc3cc(F)c(F)c(F)c3)O2)C1.c12cncc(n1)CO2 CC1(C(=O)NCC(C2CCOC2)NC(=O)Cn2c(O)nnc2O)CC=CCC1 N1(C(c2nn(C)c(O)c2)=O)CCCC2C(NC(c3ncccc3Cl)=O)C(C)(C)C12 c1(CN(C(c2cc(C(F)(F)C(F)(F)F)on2)=O)CC)cccc(C#N)n1 N1(C(COC(CC)(C)C)=O)CCN(C(=O)CN(C)C(=O)OC(C)(C)C)C(CO)C1 N(C1CC(C)n2ccnc21)C(COCc1c(C)cccc1)=O c1(C(C)NC(CONC(c2c(C)onc2)=O)=O)cccnc1F CC1CC(C)N(C(c2cn[nH]c2)=O)CCN1C(=O)C=C1CCSCC1 C=CC(C)C(=O)NC1CCN(CCCNC(=O)C(c2ccn(C)c2)C)C1 N#Cc1ccc(-c2cccc(CN3CCCCCC3CN3CCCC3)c2)c(F)c1 C1(CNC(c2c(COC)noc2)=O)CC(F)CN1C(c1cc(C)n(C2CC2)n1)=O C1(C(F)F)(CNC(c2ccc(F)s2)=O)CCN(C(=O)C=CC2CCOCC2)C1 N1(C(CNC(CC)=O)=O)CC(C2CN(C(=O)C=Cc3cccc(CO)c3)C2)C1 C(=O)(C1=NOC2COCC12)NC1C(C(=O)NC2CC(C)(C)C2)COC1 C1(NC(CN2CCP(C)(=O)CC2)=O)CC2CCC1N(C(=O)COC1CCCC1)C2 C1(C(=O)NCC(C)NC(=O)CCC=Cc2ccccc2)CCn2c(O)nnc2C1 CC1(F)CN(C(=O)C(c2ccc(Cl)c(Cl)c2)O)CCN(C(C2CC(O)C2)=O)C1 c1(OC)ccc(C(O)C(=O)NC2CCCN(C(=O)C(c3ccccc3)C)C2)cn1 C1(NC(C(C)(C)C)=O)CCN(C(=NCC2CC2)NCC2(C3CC3)CCCO2)C1 N1(C(C=CC)=O)CCC2(CC1)CN(C(c1ccnn1C1CCC1)=O)CCO2 N1(C(CN2C(C)CCCC2)=O)CCN(C(=O)C(O)CC(F)F)C(CO)C1 Cc1ccc(C(=O)NC2CC3CC(NC(=O)CC(C)n4ccnc4)CC23)c(O)n1 C#CCC(C(=O)NCC(C)(O)CNC(c1sc(C(C)C)nc1C)=O)C1CC1 C(=O)(C1=CCN(C(=O)CCN(C)CC)C1)NCC(CC)NC(=O)C(C)(C)C C(=O)(C1=C(C)CCOC1)N1C(C(=O)NCC=C)C(C)CC1 Oc1cc(Cl)ccc1-n1cc(CC2CCCN2C(c2cc(C3CC3)no2)=O)nn1 O=C1NC(CNC(=O)C(=O)NCC2CC2C2CCCCC2)CO1 CCC(CC)CCC(=O)N1CCC(F)(C(=O)Nc2cnc(Cl)nc2)C1 Cc1ccc(C(=O)NC(C)CNC(c2ccc(-c3cnc[nH]3)cc2)=O)c(Cl)c1 c1(C(=O)NCCCCNC(C2CCC(F)C2)=O)ccc2nnn(O)c2c1 N1(C(c2c(OC)cccn2)=O)CCN(C(c2ccc3c(c2)CCO3)=O)C2CCC12 N1(C(C(C)(C)c2nccs2)=O)CCC(C2CCN(C(=O)CC3CCCOC3)CC2)C1 N=c1[nH]ccc(C(F)(F)F)c1C(N1CC2(CC2)CC1C(=O)NCC1CC(O)C1)=O C1(NC(=O)CSc2n[nH]c(O)n2)COC2(CCN(C(=O)CCSC(F)(F)F)C2)C1 CC12CN(C(c3nonc3N)=O)CC1CN(C(C1CCCCC13CCC3)=O)C2 C(=O)(CCCCCN=[N+]=[N-])N1CC(C)C(CNC(C2CN(C)C2)=O)CC1 C1(c2ccn(C)n2)CCCN(C(c2cccc(F)c2)C(=O)NC2CCCC2)C1 c1(C(=O)NCC2C3CN(Cc4cc(C(=O)OC)[nH]c4)CC32)cccc(O)c1Cl C1(NC(CCOCCN(C)C)=O)CC2(C1)CN(C(=O)C(F)C1CCOC1)C2 c1(C(=O)NCCOCCN(C(=O)CC2COC(=O)N2)C)ccc(Cl)c(O)c1 N1(C(C(=O)NC2C3COCC2CNC3)=O)C2CCC(O)C1CCC2O C1(NC(c2n(C=C)ncc2)=O)CCSC12CN(C(c1ccnn1C1CCC1)=O)C2 c1(C(=O)NC2CC(CNC(C(C)(C)NC(C)=O)=O)OCC2)cc(O)cc(F)c1 c1(CC)nnc2cc(N3CC(NC(c4csc(O)n4)=O)CC4(CCC4)C3)ncn12 N1(C(C2CCC(C(C)C)CC2)=O)CC2CCC(C1)N2C(=O)Cc1cncn1C c1(C(=O)NC(CCCCNC(CC)=O)CO)cc2c(ccc3ccccc23)[nH]1 CC1CC(CC(=O)Nc2cc(F)ccn2)C(C)O1 CCCC(C)(O)CC(=O)N1CC(C)(OCCC(=O)NOCCO)C1 C(=O)(C1(C)OC(=O)c2ccccc21)NC1C(C)CN(C(=O)C=C2CCCC2)CC1 C(CC(C(=O)NC(C)CO)NC(=O)CCc1csnn1)=CC C1(=CC(=O)NC(C2(O)CN(C(C(OC)OC)=O)C2)C)CCC(C(C)(C)C)CC1 CC1OC2(C(=O)NCC=CCNC(c3cnccc3Cl)=O)CCC1C2 C=CCC(CC)C(=O)NC(C)(C(=O)N1CC(N(C)C)C1)C1CC1 N(C1CN(C(=O)Cc2cnn(C)c2)Cc2ccccc21)C(C(CC)(F)F)=O n1(CC)c(C(=O)NCC(C)(C)CNC(c2cc(C#N)on2)=O)cc2ccccc12 c1(C(=O)NC2(CC=C)CN(C(=O)C(F)(F)c3ccccc3)C2)cc(C)ccc1F C1(NC(c2csc([N+](=O)[O-])c2)=O)CC2(C1)CN(C(c1cc(CO)on1)=O)C2 c1(NC(C(=O)Nc2c(-c3nc(C)[nH]n3)cccc2)=O)ccc(C#N)c(F)n1 N1(C(CC(CC)CC)=O)CCC2CN(C(=O)CN3CCNC(=O)C3)C2C1 c1(NC(N2CC3C(CC(F)F)C3C2)=O)ccc(Cl)cc1Cl Cc1ccnc(C(N2CCC(NC(c3cnc(-c4ccsc4)s3)=O)C2)=O)c1 c1(OC)cc(C)ccc1Nc1cc(C)nc(NC(c2cnon2)=O)n1 N1(C(CCSC)=O)CCC2CCN(C(=O)CCCOc3ccc(F)cc3)C2C1 c1(C(CNC(=O)CCc2nc[nH]n2)OC(=O)CNC(C2CC2F)=O)ccc(O)cc1 CC(O)C(C(=O)NCCN(C)C(C1OCCC1(C)C)=O)NC(=O)OC(C)(C)C C(=O)(C1=CCCN(C(C2CCC(=O)N2)=O)C1)NC(C)CS(N)(=O)=O C1(C(=O)NCC(=C)Br)CNC(=O)CN1C(=O)CC1COCC(C)O1 N1(C(C2CCC(C(=O)OC)CC2)=O)C2CCCC1CC(NC(c1ccoc1)=O)C2 N1(C(C(CC)CNC(C)=O)=O)CCCC(C)(NC(=O)C(=O)OC(C)(C)C)C1 N1(C(CCC(C)(C)[N+](=O)[O-])=O)CC2C3CCC(C2C1)N(CC1CCCC1(F)F)C3 N1(C(c2cc(C)n(C)c2)=O)CCN(C(=O)COCC2CCCC2)C2CC12 c1(C(=O)NCC2CCCCN2c2ccnc3ncnn23)cc2cc(Cl)ccc2o1 C(=O)(CC(C(F)F)C(C)(C)C)NC1CN(C(C2(c3c(C)c[nH]n3)CC2)=O)CC1O C1(C(=O)OC)N(C(c2cc(C(C)(F)F)ccc2F)=O)CC12CCC2 CC1CC(n2nc(C3CCCC3)nc2-c2cc(-c3ccco3)[nH]n2)CCO1 c1(C(=O)Nc2cncc(Cl)n2)cn2c(n1)CCN(C(c1cnoc1)=O)CC2 CC(C)(C)CCC(=O)NC1(CCCNC(=O)CC2CCC3(CCC3)O2)CC1 c1(OC)cc(Cl)ccc1CNC1CC(C(=O)Nc2c(F)cccc2F)C1 N1(C(c2cc(C(C)=O)on2)=O)CCC2(NC(c3cccc(C4CC4)c3)=O)CC2C1 c1(C(=O)NCC(C)(C2CC2)NC(C23CCC(C2)C3)=O)ccc(Cl)c(O)c1N c1(N2C(CN3CC(NC(=O)C4=CCC4)C(F)C3)CCCC2)c[nH]c2c(Cl)cccc12 CCCC(C)NCC(C)CN C(=O)(C(C)(C)C1=CCSCC1)NCCOCCCNC(C(CC(C)C)NC(C)=O)=O C1(NC(CCSCCC)=O)CCN(C(c2cc(C(N)=O)co2)=O)C1C1CC1 C1(CC(N2CCC(NC(c3cnn(CC(F)F)c3)=O)C2)=O)CCCOCC1 CC1CCN(C(C2(NC(=O)CC3CCC(=O)C3)CC2)=O)CC1C c1(NC)cncc(C(=O)NCC(C2CC2)NC(C2CCCN2C(C)=O)=O)c1 c1(C(N2CCC(N(C(=O)C(C)n3ccnc3)CC)C2)=O)cc(N)nc(Cl)c1 C(C(F)(F)C(=O)NCC1(NC(=O)C(Cc2cnc[nH]2)OC)CCCCC1)OC Cn1cnnc1C1CCCC1NC(C1CC(N(C(=O)Nc2cncnc2)C2CC2)C1)=O c1(C(N(C)CC2CCN(C(C(C)(C)SC)=O)C2)=O)ccc2cnoc2c1 CC1(C)CCC(C(N2CC(C)(CCC(=O)NCC(F)C(C)(C)O)C2)=O)C1 c1(C(=O)NCCCC(C)NC(=O)CCNc2ccccc2)c(F)ccc(F)c1F CC1=C(C(=O)N(C(C)CN(C)C(C2CC3(CC3)CO2)=O)C)CCS1(=O)=O c1(CC=C)cc(C(=O)NCC(C)C(F)C(=O)OC)cc(OC)c1OC c1(OC)ccc(CCC(=O)NC2(C3CCCCN3C(=O)C(F)C3CC3)CC2)cn1 C=CC1(C(=O)NCC2CCC(O)C2)CCN(C(c2ccsc2)=O)C1 C(=O)(C(=O)C(C)(C)C)NCC(C)(C)CNC(c1nc(Cl)sc1Cl)=O c1(C(=O)NC2CCC(CNC(C(=O)NCC)=O)CC2)c[nH]c(=O)c2ccncc12 N1(C(c2cc(OC)ns2)=O)CCN(C(c2ncc(C(F)F)cc2F)=O)C(CF)C1 C1(C(=O)NC(C)CNC(=O)CC(C)(C)C2CC2)CC12CCC(F)(F)CC2 C1(OC)(CNC(c2cnnn2C)=O)CCN(C(=O)CC2(O)CCC2)C1 C1(CN(CC(CC)C)C(C2(N(C)C)CC2)=O)CCCCCCC1O N1(C(c2ccc(CC(C)C)s2)=O)CC2CC1CCC2NC(c1cccnc1O)=O CC1CCC(NCCOc2cccc(Cl)c2)CS1(=O)=O c1(C(=O)NCCCN(C(=O)C(C)CSC(F)(F)F)CC)cc(C)c[nH]1 c1(N(C)CCN(C)C)cc(N2CCOC(C(C)(C)C)C2)nc(CN2CCOCC2)n1 C(=O)(CC1=NNC(=O)C1)NC(=O)CC1CCC(C(F)(F)F)O1.C1(C)(N)CC1 N1(C(C(C2(O)CCC2)NC(C(C(C)C)C#N)=O)=O)CCC2CN(C)CC2C1 c1(C(CNC(C2CCCOC2)=O)NC(=O)CCc2csnn2)ccc(F)cc1 c1(C(N2C(CNC(CC(=C)Br)=O)COCC2)=O)cncc2c(F)cccc12 C1(NC(c2c(C)n(C3CC3)nc2)=O)CN(C(C2CC(C)(O)C2)=O)CC(F)(F)C1 n1(C(CC)C)nnnc1C(C1CC(OC)(OC)C1)NCCCSC C(=O)(C1Cc2c(Cl)cccc21)NCCC1CC(NC(C(C)CS(C)(=O)=O)=O)C1 CC1(C)CN(C(=O)CCCc2cccnc2)C(CNC(=O)CC2C=CCC2)CO1 C1(n2cccn2)COCC1C(N(C1(C(N(C)C)=O)CC1)C)=O.N12CC(C1)C2=O C1(C(N(C(CCN(CCCC2CCCCC2)C)=O)C2CC2)=O)CN(S(N)(=O)=O)C1 C12(CNC(Cc3c(C)nc(S)s3)=O)CCC(C1)N(C(=O)CN1CCC(C)CC1)C2 c1(C(=O)NC)ccc(N(c2nccs2)C(=O)COC2CC2Cl)cc1 C(=O)(C(C)(C)CNC(C12CCC(C(=O)O)C1C2)=O)OC c1(SCC(=O)N(C2CCN(C(CC(CC)SC)=O)C2)CC)ccc([N+](=O)[O-])cc1 c1(CNCC2OCCN(C(=O)OC(C)(C)C)C2)cccc2cnsc12 C(=O)(CCC(C)NC(=O)C=C(C)C1CC1)NCC(CC1CC1)OC N1(C(C2CC3CCC3C2)=O)CCC2OCCN(C(=O)Cc3cn[nH]c3)C2C1 c1(C(C)C)cccc(NC(=O)C(C2CCCC2)NC(=O)C#CC2CC2)c1 N1(C(C(=O)NC(c2ccc(Br)cc2F)C)=O)CCCc2c(Br)cccc21 C1(NC(=O)C(N2CCC(C(F)F)C2)=O)CCC(CO)CC1 C(C1=CCN(C(c2ncnc(O)c2F)=O)CC1)NC(=O)Cc1cnc[nH]1 C1(C)(OC)CCN(C(=O)CC2CCN(CC(=O)N(C)Cc3ccnnc3)C2)CC1 C(=O)(C(C)CC(N)=O)N1CC(CNC(C2(C)CC(C)C2)=O)OCC1 C(=O)(C(CNC(c1cc(C)c(C)s1)=O)(CC)CC)NCC1CCC(OC)C1 C1(C(=O)OCC)C2COC(C(=O)N(CCCNC(C3(Cl)CC3)=O)C3CC3)CC12 CC1CC(=O)CCC1C(=O)NC1CC(CC(=O)NCc2cnccc2Cl)C1 C1(C(=O)NCC2(C(N)=O)CN(C(CNC(C3C(C)C3)=O)=O)C2)CCC=CCCC1 c1(OC)ccc(COC(C2(SC(C)C)CC2(F)F)=O)cc1N Nc1ccc(C(=O)NCC2CC3CCC2N3C(=O)C(F)=C2CCCC2)nc1N C1(C(N)=O)COCC1C(=O)NC1(C(N2CCC(c3nn[nH]n3)C2)=O)CCC1 Cc1cnc(C(N2CCCC(NC(=O)CC3C=CS(=O)(=O)C3)C2C)=O)c(F)c1 C1(n2cc(CC34CC(C)(C3)C4)nn2)CCCN(C(=O)Nc2cc(C#N)cs2)C1 Cc1cc(C(=O)NCC2CN(C(C3C(C)C3C)=O)C3COCC3O2)cc(=O)n1C Cc1c(C(=O)NCC2C(C)CCN2C(c2cnc(C)n2C)=O)cccc1C#N N1(C(c2cnc(CC)s2)=O)CC2(CCN(C(=O)C(C)(C)C)C2)C1 c1(C(=O)NCC2(NC(C3C(C)SCCC3)=O)CCCC2)cnn(C)c1C#N c1(C(=O)NC2CC(N(C(=O)C(c3ccccc3)F)C)C2)ncccc1Br C=CC1CN(C(=O)Cc2cccc(C(C)C)c2)CC1NC(=O)C(C)OC C1(C(=O)NCCOC(C)(C)CNC(c2nc(C3CC3)cs2)=O)OC2CCC1C2 c1(OCCCC)ccc(C=CC(=O)NCC(C)N(c2ccns2)C)cc1 c1(NC2C(C(F)F)CCC2)cc(NCc2cncc(Br)c2)ncn1 N1(C(CC(=C)C)=O)CCC2(CO)CN(C(=O)C(F)(F)c3cnccn3)CC2C1 N1(C(C(=O)NCCC)C2CC(C(=O)OCC)C2)CCN2CCOCC2C1 CC(C)C(C)(O)C(=O)N1CC(CNC(c2ccc(Cl)cn2)=O)C(F)(F)C1 CC(CCO)NC(C1(N(C(=O)CC2CCCO2)C2CC2)CCC1)=O C1(C(=O)NCC(c2cnccn2)(C)C)(COC)CCCN1C(=O)C(C)NC(C)=O NC(=O)CCCCC(=O)NC1CCCCN(C(=O)C=CC=C(Cl)Cl)C1 CC1(CNC(C2CC3(CC3)C2)=O)CN(C(c2ccnc(Cl)c2N)=O)CCO1 CC(C)CC(C)C(=O)NCC1CN(C(c2ncncc2F)=O)CC(C(F)(F)F)O1 CC#CCCC(=O)NCC1CCCC(NC(C2CCCN2CCCCC)=O)C1 N(C(=NCc1ccc(CO)cc1)NCC1(CO)CC1(C)C)C(C=C)C Cc1ccc(O)c(NC(=O)CC2CCCCN2C(c2ccc(=N)[nH]c2Cl)=O)c1 C1(CNC(CCC)=O)CC2CN(C(=O)Cc3ncc(C)s3)CC12 CCC(CO)(C(=O)NCC1(C(=O)NCc2cccnc2)CC=CC1)OC C1(NC(=O)CCc2ccccc2F)COC2(CCN(C(c3coc(Cl)c3)=O)C2)C1 c1(C(N2C(CNC(Cc3nc(CC)sc3)=O)C=CC2)=O)cc2c(cc1N)OCO2 Cc1cnccc1C=CC(=O)NC1(C2CN(C(c3csc(CO)n3)=O)C2)CC1 c1(NC(C(CNC(c2cscn2)=O)O)=O)cnc(Cl)nc1 C(C)(C(=O)NCC(C(=O)N(c1ccoc1)CC1CC1)N(C)C)(C1(C)CC1)OC N1(C(c2n(CCOC)ncc2)=O)CCC2(CCCN2C(C2CCN(C)C2)=O)C1 c1(CC(=O)NCCC(COCCC(=O)OCC)O)cccc(F)c1F C1(CCC)(C(N2CC(O)(C(C)NC(c3cncc(F)c3)=O)C2)=O)CCNC1=O c1(OC)ccc(F)c(C(=O)NCC2CCCC2NC(=O)CNS(C)(=O)=O)c1Cl C1(COC2CCN(C(CCNC(C)=O)=O)C2)CCN(C(=O)CC2CCOC2C)CC1 CC(Cc1ccco1)C(=O)N(CCCNC(C1(C(F)F)CCCO1)=O)C1CC1 C(=O)(N=S1(=O)CCC2(CCNCC2)C1)c1c(C)cc(S(N)(=O)=O)cc1 N1(C(c2ccc(C#N)cc2)=O)CCC2CN(c3ccn4ccnc4n3)CCC2C1 C1(C(=O)NCCC2(NC(c3csc(C(N)=O)c3)=O)CC2)CS(=O)(=O)C1 c12n[nH]cc1C(=O)NC2CCO.C12(CCC1)C(=O)N2.C(CCO)SC Cc1c(OC(c2cnnn2C2CCN(C)C2=O)=O)ccc(Br)c1Cl Cc1cnnc(O)c1C(=O)NCC1CC(F)CN1C(C1CC2(C1)CC(F)C2)=O CN1N=C(C(=O)NC2CN(C(=O)Cn3cnc4c3CCCC4)C3CC23)CCC1=O c1(C(N(C(C(=O)NCc2cc(CO)on2)C2CC2)C)=O)cc(O)ccc1F C1(CC)CCC(C(=O)NCc2nc(CNC(=O)C(C(C)C)NS(C)(=O)=O)cs2)CC1 c1(C(=O)NC2CCC(C(=O)NCC3(C(N)=O)CC3)C2)ccc(O)nc1 N1(CC)CC(C)N(C(=O)CCN(C(=O)Cn2cccnc2=O)C)CC1C c1(C(C)C)ncc(Cl)c(C(N2CC(C)CCC2CNC(=O)CCP(C)(C)=O)=O)n1 c1(OC)nc2ccc(C(N3CC(NC(c4cc(CO)ccc4Cl)=O)C3)=O)cc2[nH]1 c1(C(N(CC(CNC(c2scc(C(C)=O)c2)=O)C)C)=O)[nH]cnc1C#N c1(-n2c(CNC(c3ncsc3-c3ccccc3)=O)ccc2)cccc(Br)n1 c1(C(=O)NCC2(C)CNC(=O)C2)ccc2cccc(F)c2n1 N1(C(CCCCCOCC)=O)Cc2ccccc2C1CNC(=O)C(C)=CC1CC1 C(=O)(CC(C(F)(F)F)NC(=O)C1CC1)NC1(C)CCN(C(C=CC(C)(C)SC)=O)C1 Cc1cccnc1CC(=O)NCC(C1CCN(C(C2CCC(O)C2)=O)CC1)F c1(NC2C(NC(C3CC=C(C)CC3)=O)CCCC2)nc(C)cc(C)c1C#N N1(C(C2(CC)CCN(C(c3cccnn3)=O)C2)=O)CC2CCC(C1)O2 n1(CC)nnc(C)c1CNC(=O)C(C)=CCNC(C1(O)CCCC1)=O C(C(=O)NCCc1ccccc1F)(C(C)(C)C)NC(C(C)n1ccnc1)=O N1(C(c2cn(CCC=C)nn2)=O)CCC(F)C(NC(c2ccc(Cl)cc2F)=O)C1 N1(C(Cc2scc(C)c2)=O)CCN(C(c2nnc(O)nc2O)=O)CC1CC(F)F c1(C(=O)NC(C2CN(C(c3cc(Cl)c(Cl)[nH]3)=O)C2)C)cn(C)c(=O)n1C Cc1sc2ccccc2c1C(=O)NC12CC1COC2(C)C c1(C(C)=O)ccc(C(N2CCOCC(CNC(C3(F)CC=CCC3)=O)C2)=O)cc1F C1(CC(N2CC(NC(c3cccs3)=O)C2)=O)CCCS(=O)(=O)C1 N1(C(CNC(=O)C2CC2)=O)CCC(N(C(Cc2n(C)ccn2)=O)CC2CC2)CC1 N1(C(CCCN(CCC)CCC)=O)CC2(CCN(C(=O)CC(C)NC(N)=O)CC2)C1 CC(C)CCCCC(=O)NC1CC2(C1)CC2C(=O)NCC1CCCN1C c1(C(=O)NC2CC3N(C(C4(OC)CCC4)=O)C(CC3)C2)cnn2c1C(C)CCC2 C1(C(N2C(CC(=O)NCC3(COCC)CC3)CC2)=O)C2(CC2)C12CC2.C(C)(=O)O C1(C(=O)Nc2cncc(C)n2)C2CCC(C2)N1S(=O)(=O)C1CC1 C1(NC(=O)CC2CC3C=CC2CC3)CCN(C(c2cncc(F)c2)=O)C12CC2 C1(NC(C2C(C)CCO2)=O)CCCC(C(=O)NC2CC3CCC2C3)C1 C1(C(=O)NCCN(CC(C)O)C(c2ccccc2)=O)CCCCC(=O)C1 c1(C(=O)NCC(C2CCN(C(c3ccn(CC)n3)=O)CC2)F)cc(Cl)ccc1N CCCCCC(O)CC(=O)NCCn1cc(C(N2CCC(n3cccn3)C2)=O)cn1 c1(CNC(C2CCC3(CN(CC=C)C3)O2)=O)sc2ccccc2c1Cl CCCC(C)CC(=O)N1CCC(N(CCO)C(c2cc(F)ccc2O)=O)CC1 C1(CCOC)(NC(=O)Cc2csc(=N)[nH]2)CCN(C(=O)C(C)(C)OC)C1 c1(C(N(C)CC2(NC(C3N(CC)CC3)=O)CC2)=O)cc(Cl)c(Cl)[nH]c1=N N1(C(c2cc(CC)sn2)=O)CCC(NC(C2CCC(N(C)C)CC2)=O)C(CO)CC1 C1(NC(C(=O)NCC)=O)CN(C(=O)COCC(=O)OC(C)(C)C)C2(CCC2)C1 c1(C(=O)NC2CC(CCNC(C(CC(=C)C)C)=O)C2)c[nH]c2cc(OC)ccc12 Cc1cc(-c2cn(C3CC(CNC(=O)C=C(Cl)Cl)C3)nn2)ccc1N O=C1NCc2ccc(NC(C3CC3NC(C3CCC3)=O)=O)cc21 CC1CC(CCNC(c2ccc(CO)o2)=O)CCN1C(=O)C(=Cc1c[nH]cn1)F c1(C(=O)NCC2C(NC(C3(CC=C)CCC3)=O)CCC2)coc2c(C)cccc12 CCS(=O)(=O)CC(=O)NC(C(=O)NC1CC(c2ncc[nH]2)C1)C1CCCO1 Cc1cccc(C(=O)NC2(CNC(c3cccn3CC3CCCC3)=O)CC2)n1 c1(CC(=O)NC2(C)CN(C(C3(O)CCOC3)=O)C2)ccccc1Cl CC1CN(C(C2CCS(=O)CC2)=O)CC1CNC(C1CN(S(C)(=O)=O)C1)=O C=CC1(C(=O)NC(C)C(=O)NC(C)C)CCN(C(c2cc(O)cc(=O)o2)=O)CC1 C(=O)(C1=NOC(C)C1)NC1(CO)CN(C(C2C(c3c(C)nn(C)c3)C2)=O)C1 CCCC(CC(C)C)C(=O)NC(C)(C)CCCNC(=O)C=CCOCC(F)(F)F N1(C(C)=O)CC2CC2(CNC(C2(C)CC(F)C2)=O)C1.c12ccc(nc1)OC2 c1(CC)cnn(CNC(C2(C(C)NC(C3CC(OC)C3)=O)CC2)=O)c1 C1(C(=O)NC(CC)C(N)=O)CCC2(CCN(C(=O)CCc3cccnc3)CC2)C1 c1(C(C)C(=O)N(CC(C)(C)CNC(=O)Cc2ccoc2)C)ccc(O)cc1 O=C(C1=C(Cl)CCCC1)NCC12CCCCC1C2(F)F N1(C(CNC(N(C)Cc2ccncc2)=O)(C)C)CCc2ccccc21 c1(NC(c2snc(CSC)n2)c2nnnn2C2CC2)cncnc1O c1(CCCC)ccc(CC(C)CNC(=O)NCCC2CCCN(C)C2)cc1 CCCCCC(=O)NC1CC(NC(=O)C(c2ccccc2)SC)C(O)C1 CN1C(=O)C(O)C(C(=O)Nc2ccc(Cl)cc2CCN)C1c1cccnc1 C1(CC(C)C)(C(=O)NCC(C)CNC(c2sccc2Cl)=O)CCNC1=O Cc1cc(C(N2CCC(C)C(NC(=O)CC3(C(F)F)CC3)C2)=O)cc(N)c1 C(=O)(C(C)(O)CC(C)C)N1CC(C(=O)NCCNC(C2(OC)CCOCC2)=O)C1 c1(N2CCC(C3CC3)(CNC(CN(S(C)(=O)=O)C)=O)C2)ncc([N+](=O)[O-])cc1C#N S(=O)(=O)(c1cncc(Br)c1)N1CC(N(C)Cc2cc(Br)c(Cl)cc2C)C2(C1)CC2 c1(CC)[nH]nc(C(=O)NCC=CCNC(=O)C(C)Cc2ccco2)c1[N+](=O)[O-] O=C(CC1=CCCC1)NCC1CCC(NC(c2ccc(-c3ccco3)o2)=O)CC1 N1(C(C2=C(C)OCC2)=O)CC(CNC(=O)CCc2ncccn2)OC(C)(C)C1 c1(C(=O)OCC)cccc(NC(=O)NC2(C3CCCO3)CC2)c1C c1(C(C(=O)NCCNC(C(CC=CC)C)=O)C)ccccc1S(N)(=O)=O N12CCOC(C1)C2=O.C(CC(=O)N(CC(N1CCCC1)C)C(C)C)NC(C)=O C(=O)(C1=CCN(C)C1)NC1C2(CC(NC(CCOCCOC)=O)C2)C1 C1(C(=O)N(C)CC2CN(C(=O)C(C)(C)OC)CCO2)(OC)CCOCC1 CC(C)(CC(=O)N1CC(NC(c2cnc(N)c(N)c2)=O)C(C2CC2)C1)C(F)F CC(C)C(O)C(=O)NC1CCCCC1CC(=O)NOCC(O)CO c1(N2CCC(CCCl)CC2)nc2ccccc2nc1N1CCC(S(C)(=O)=O)C1 N1(c2n(Cc3ccc(-c4c(Cl)cccc4)o3)nnn2)CCC2CCNC2C1 C(CC#CC)(C(=O)NC(c1ncc[nH]1)C)NC(Cn1ncc(C#C)c1)=O c1(CC(=O)NC(COCC)C(=O)NC(c2nccn2C)C)cccc(C)c1 c1(C(N2CCOCC(C3CC3)C2)C(=O)NCC(=C)C)noc2ccc(Br)cc12 CC1(C)C(CNC(=O)CC2CCC(O)C2)CCN1C(=O)CCc1ccc(O)c(Cl)c1 C1(C(N(CCCCNC(c2ncoc2C(C)(C)C)=O)C)=O)CC12CC(C)(C)C2 C(=O)(C1=C(Cl)CCOC1)NC1CC(F)(CNC(c2c(C#C)c[nH]n2)=O)C1 N1(C(c2c(SCC)cccn2)=O)CC2=C(C1)CN(C(C1(C)CC=CCC1)=O)C2 N1(C(COCC=C)=O)CCC(C=C)(C(=O)N(C2CCCC(C)C2)CC)C1 c1(NC(C2(c3ccc(Br)s3)CC2)=O)ccc(-c2ccc(OCC3CC3)nc2)cc1F C(C)(CO)(C(=O)N(CCC1CC1)CC1CC1)NC(C(C)=C(CC)C)=O c1(CC)cc(C#N)c(N2CCC(C(F)(F)F)(C(=O)OC)C2)nc1C C1(C(=O)NC)CCN(C(C2CC2C(=O)NC)=O)C12CCC2.c1(CC)cc(CCO)on1 C(=O)(C(C(C)C)OC)N1CC(CC=C)(NC(=O)C(C)(C)F)C1 Cc1nc(O)ccc1C(=O)NC1CCC(NC(=O)C#CC(C)(C)O)C1 c1(OCCC)ccc(C(=O)OC)cc1CNC1CC2(CCCCC2)C1 C1(C(=O)NC2CN(C(C(C3CCC3)OC)=O)CC2C)CC(c2cnn(C)c2)=NO1 Cc1cc(NC(C2CN(Cc3ccc(Cl)nc3)CCC2O)=O)ncc1Cl N1(C(c2c(CC)noc2)=O)CC2CC(NC(c3cnn(C(C)C)c3C)=O)C2C1 C1(NC(=O)NCc2cc(C(=O)OCC)[nH]c2)CC(C)SC(C)C1 Cc1ncc(C(N2CCC(CNC(c3cc[nH]c(=N)n3)=O)C(C)C2)=O)c(C)n1 C(=O)(C(C(=O)NCC(C)CNC(=O)Cc1ccc(F)cn1)C(C)C)OCC C(C(CC(C)C)C(=O)NCC1=CCN(C(=O)CC2SC(=N)NC2=O)CC1)OC Nc1ccc(Cl)c(C(N2CC=CC2CNC(=O)CCn2cnc([N+](=O)[O-])c2)=O)c1 n1(C(COC)C)cc(NC(C2CC=CCO2)=O)c(C)n1.C1CCCNC(=O)CO1 CCC(C)CCCC(=O)N(CCCNC(C1CC2CCCC(C1)C2)=O)C1CC1 N1(C(c2ncn(C(C)C)c2)=O)CC(F)(F)CC1CNC(C1COCC(C)(C)O1)=O S(=O)(=O)(c1cnc(NN(CC(COC(C)C)O)C2CC2)c(Cl)c1)NCC(C)(C)C CCS(=O)(=O)c1cccnc1C(N1CCC(CNC(=O)CN2CC=CC2)CC1)=O C1(NC(c2cc(C)c(O)cc2)=O)COC2C(NC(C3COC(C)(C)C3)=O)COC12 N1(C(c2cnc[nH]2)=O)CCN(N2CC(O)CC2CO)CC1 Cc1cc(C(N2CC(c3cn(CCCF)nn3)C(C)C2)=O)c(C)o1 C1(CC2CC2C(NOCCCC)=O)CCN(C(=O)C(OC)OC)CC1 c1(OC)ncc(Cl)cc1CNC(c1ccc(Br)nc1)C N1(C(c2ncnn2CC(F)F)C(=O)NCCOCC)CCC(C)(CO)C1 C1(C(N(CC(C)N(C(CC(C)C)=O)C)C)=O)CCC(F)CC1 N1(C(C2N(CCC)CCC2)=O)CCC(CC(C)NC(=O)COC(F)(F)F)CC1 C(=O)(CC(C)(C)OC)N1C(CCC(=O)NC(C(=O)NCC)CO)CCC1 c1(CN2CCN(CCNC(C(CC)C3COC3)=O)CC2)cn2nc(C)sc2n1 C1(CC)(NC(=O)C=CS(C)=O)CCCN(C(=O)C(c2cncc(F)c2)(C)C)C1 C1(C=O)CCCCC1O.C(C(=O)N(CC(O)CF)C)(C1CC1)OC c1(C(N2C(CNC(c3c(F)cccc3Cl)=O)COCC2)=O)cc(Br)c(O)c(Br)c1 c1(C(N2C(C)(CNC(C(CC#C)O)=O)CCC2)=O)cccc(Cl)c1F Cc1cncc(C(=O)N(C2CCCN(C(C3CC(C4CC4)C3)=O)CC2)CC)c1C N1(C(C(COC)C)=O)C2CCC(C(=O)NC3(C4CC4)CCC3)C1CC2 CCCCCC(CC)C(=O)NCC(C(=O)NCCOC1(C)CCC1)C(C)C CC(C)(CC(=O)N1CC2CCC1CN2C(C1(S(C)(=O)=O)CC1)=O)CC(F)(F)F N1(C(c2nc(CCC)oc2)=O)CCC(NC(c2cc(C)c(C)o2)=O)C(F)C1 N1(C(CN(C(=O)CCc2nccs2)C)=O)CCN(C(=O)CC(F)(F)F)CC1 N1(C(CCCC(CC)C)=O)C2CCC1C1CC1(NC(=O)CCOC1CCC1)C2 C#Cc1cccc(C(=O)N(C2CCC(NC(=O)CC3=CCOCC3)C2)C)c1C CCC(CC(=O)N1CCC(C)(CO)C1)N(C)C(C1CCC(=O)O1)=O N1(C(CC=CCC)=O)CC(=O)NCC1C(N1CCC2(CCC2)C1)=O Cc1nn(C)c(NC(=O)NCC2CC2C(F)(F)F)c1-c1ccccc1 N1(NC(=O)C(CCC)c2ccccc2)CCCN(Cc2cncc(Cl)c2)CC1.CC CCC(C(=O)NC1CC(Cn2cc(CCC3CCOC3)nn2)C1)c1cccnc1 N1(C(c2c(C#N)ccs2)=O)CC2(CCCC2)C1C(=O)NCC(=O)NCCO c1(OCCCC(=O)NC2(C)CN(C(C3CCCCN3C)=O)C2)cc(Cl)ccc1Cl S(=O)(=O)(c1c[nH]c2ncccc12)NCCCn1cc(C)nn1.CS(=O)(=O)N C12(NC(C(c3ccc(OC)cc3)CC)=O)CC(C1)N(C(c1ccnnc1S)=O)C2 CCCC(C(O)C(=O)N1CCC(F)(C#N)C1)NC(=O)CC(C)CC N1(C(CC(C)OC)=O)CCCC(C(N2CCC(c3ncns3)CC2)=O)CC1 C12(CC(F)(F)C1)C(=O)N2.CCC(C(=O)NC(C)(C)C(=O)N1CCCC1)OC c1(C(=O)NC2CC(CNC(C(C)SC(C)C)=O)CC2O)ncsc1S(N)(=O)=O OC1CCC2(CCCN(Cc3ccc(F)cc3Br)C2)C1 Cc1c(Cl)ccnc1C(N1CCN(C(c2csnc2Cl)=O)C(C(C)C)C1)=O c1(NC(c2ncccn2)CC)cc(Br)ccc1S(=O)(=O)N1CCn2nc(C)cc2C1 N1(C(CC=C=C)=O)CC(NC(c2cc(O)cc(Cl)c2)=O)C2CC2C1 C(c1ccnn1C)=CC(=O)N(C)CC1CCN(C(COCC(=O)NC)=O)C1 c1(C(N2CC(NC(CCCCCSC)=O)C(C)C2)=O)cc(F)cc2cnccc12 C#Cc1ccc(C(=O)NC2(C(N3CC(CC)(CO)C3)=O)CCN(C)C2)nc1 C1(C(=O)NCC(C)(C2CC2)NC(c2coc(Br)n2)=O)CC12CCOC2 C(=O)(C1=C(C)CCC1)NCCCC(N1C(C(=O)NCC(C(CC)C)C)COCC1)=O CC(C)CCCCC(=O)N1CC2CCC(C1)N2C(=O)Cn1ncn(C)c1=O Cc1cnc(N2CC3(CCC(CNc4ccccc4)O3)C2)c([N+](=O)[O-])c1 N1(C(Cc2cn(CC)nc2)=O)CCC(C2CC2)C1CNC(=O)C1=C(C)OCC1 C1(NC(c2n(CCC)ccc2)=O)CCCCCN(C(C2CCCNS2(=O)=O)=O)C1 c1(N(c2ccccc2)C)cc(NC(=O)N(C(C2CCCCC2)C(=O)O)C)ccc1F C(=O)(C(CC)CC)N1CC(C(C)(C)O)(CNC(CCOCCC)=O)C1 Cc1cnc2n1CCC(C(=O)NCC1(CNC(=O)CCCC#N)CC13CCC3)C2 C1(NC(CCC(=O)NCC)=O)CC1C1CCCN(C(c2c[nH]nc2C)=O)C1 C12(NC(C=CC(C)=O)=O)CC(CNC(C3CC3c3ccsc3)=O)(C1)C2 N1(C(CC2N(C)CCC2)=O)CCC2(CC(NC(=O)CCCc3cccnc3)C2)C1 C1(CC)(COCC)CCN(Cc2ccccc2)C1 C12(C(N(C3CCN(c4ncc(C(F)(F)F)cc4Cl)C3)CCC)=O)CC=CC(C1)OC2 Cc1cnc(CC(=O)NCC2CCC(NC(C3(C(C)C)COC3)=O)C2)[nH]1 N1(C(C2(OC)CCSC2)=O)CC2CCC(C1)C2NC(c1ccnc2ccnn12)=O CC(C)C1=NOC(C(=O)NCC#CCNC(=O)C(C(C)(C)C)OC(C)(C)C)C1 N1(C(c2c(C(=O)OC)nccn2)=O)CCCC12CCCN(C(C1CC1C1CC1)=O)C2 C#CC1(C(N2CCC(OCCCCC)C2)=O)CCCC1 C1(C)CCC(C)(C)CC1.n1(CC)nnnc1C(c1ccncc1)NCCn1cccn1 c1(OCC)cccc(C(=O)NCC#CCNC(=O)C(C)(C)C(C)O)c1N Cc1cc(F)cc([N+](=O)[O-])c1NC(C1C2CN(Cc3nc(Cl)ccc3F)CC12)=O CN(CCCC(=O)NCCC1CC(NC(=O)C#CC2CCC2)C1)N=O c1(C(=O)NC)cccc(C(N2CCC(O)(CNC(=O)CCC3CCOC3)C2)=O)c1 C(N=c1nc(O)c(Br)c[nH]1)C1(C)CCCN(C(c2ccc(C)nc2O)=O)C1 c1(C(C(=O)NCC(C)Cn2cc(CO)nn2)=O)cccc(F)c1 CC(C)(CCN(C1CCCCC1)C1CC1)CC(=O)OCCN1CCCNC1=O c12cccc(n1)C(=O)N1CCC(C1)CNC2=O.c1(CC)cn[nH]c1 c1(C(=O)NC2CC(F)(CNC(c3c(CC)[nH]nc3Cl)=O)C2)ccc(N)c(F)n1 Cc1nn(CC(=O)NC(C)(CNC(C2(C)CNC(=O)C2)=O)C2CCC2)c(C)c1Cl Cc1cc(F)c(Br)cc1C(=O)N(C(C)CNC(=O)CC(O)C(C)C)C CC1CN(C(C2CCCC(O)C2)=O)CC1NC(c1cc(C(F)(F)F)co1)=O CC(=O)CCCC(=O)N1CCC(O)(CCNC(C2CN3CCN2CC3)=O)C1 N1(C(CCSC)=O)CC2(C(=O)NC(C)(C)CO)CC1CO2 c1(CC(CNC(=O)CC2CCCNCC2)OC)cccc(Cl)c1 Cc1n[nH]c(C)c1C(N1CCN(C(CC(F)(F)C2CC2)=O)CC1)=O N1(C(COC)=O)CCC2CCN(C(c3cc(NC4CC4)ncc3Cl)=O)CC12 C1(C(=O)NCCC2(C(=O)NCCOCC#C)CC2)CC2CC2C1 CS(=O)(=O)c1ccc(CC(=O)NC2CCN(C(c3cc(C4CC4)on3)=O)C2)cc1 C1(NC(C(C=C=C)C)=O)CCC(C)(CNC(=O)CN2CCCS2(=O)=O)CC1 C12(C(N(CC(C)NC(c3ccccc3CC#N)=O)C)=O)CC(C1)C(C)(C)O2 c1(OC)cc(C)ccc1C(=O)N(C1CCN(C(=O)CCCC(C)=O)CC1)C c1(C(=O)NC2CCCN(C(CC(CC)SC)=O)C2)cccn2c(CO)nnc12 c1(C(=O)NCC(=O)NC(C)CNC(c2coc(Cl)n2)=O)ccccc1CC#N C1(NC(C=CCOC)=O)CCN(C(=O)C(C)N2CCCC2)CC1O c1(CN2C3CN(C(c4n(C)nc(C)c4Br)=O)C(C3)C2)ccc(O)c(Cl)c1 C1(CC(=O)NC2CCCC(C(=O)Nc3cnc(C)s3)C2)Cc2ccccc2C1 c1(C(=O)NC(C(=O)OC)C)cc(C(=O)C2CC2)on1.C(c1ccco1)=CC(=O)N N1(C(c2nc(OC)oc2)=O)CCCC12CCN(C(=O)CSc1nncn1C1CC1)C2 N1(C(CNC(CC)=O)=O)CC(NC(C2CS(=O)(=O)CCO2)=O)CC2(CC2)C1 N1(C(C(CC)C(C)C)=O)CC2CC(NC(c3cc(=O)cc(Cl)[nH]3)=O)CC2C1 Cc1cnc(C(N2CCOCC2c2nnc(C)o2)C(=O)NC2CC(F)(F)C2)c(C)c1 c1(C(=O)OCC)ccc(CN(Cc2ccco2)CC2(C)CC2(C)C)[nH]1 C1(NC(C=CCC)=O)CCCC1(C)CNC(c1cc(CC)on1)=O C1(CNC(=O)Cn2cccn2)C(C2CC2)CCN1C(c1ncc(C(F)(F)F)s1)=O N1(C(C(CNC(CC2COCC(C)O2)=O)N(C)C)=O)CCC(C2CC2)C1 c1(C(N(CCC(=O)NCC(c2ccncc2)O)C)=O)ccc(C#N)n1C N1(C(C(C2(C)CC2)NC(C(C(C)C)C(C)C)=O)=O)CCC2(CCOCC2)C1 c1(C(N2CC(F)(C(=O)NC(C3CCOC3)C)C2)=O)cc(C#N)ccc1Br N1(C(Cc2c(C)n[nH]c2C)=O)CCCCC(NC(c2ccncc2Br)=O)C1 N1(C(C2CC(C)N(C)C2)=O)CCC2(C=C(C(=O)N3CC(NC(N)=O)C3)C2)C1 N1(C(C(C)n2cnnn2)=O)CC2CCN(C(c3ccnc4ncnn34)=O)CC2C1 CN1CC(C(N2CCC(C3CN(CC4CCC5(CC5)C4)CCO3)C2)=O)CCC1=O c1(C(N(CCCNC(CCOC2(C)CCC2)=O)C2CC2)=O)cc(F)cnc1O c1(C(=O)OCC)c(NC(C2CCCN2C(=O)C(C2CCCC2)OC)=O)ncn1C S(=O)(=O)(c1ccc(C)cc1)N(C(C(=O)NCCNC(C1C(C#C)C1)=O)C)C N1(C(C23CC(C)C2C3)=O)CC2(CC(NC(c3n[nH]c4c3CCC4)=O)CO2)C1 C(=O)(C#CC1CCCCO1)NCC(C1CC1)NC(c1cc(CSC)c(C)s1)=O C(=O)(C1CCc2oc(C)nc21)N(C(C)CNC(c1cc(C)no1)=O)CC CC(C)C(CO)CCNC(C1CCN1C(C1CC(OC2CC2)C1)=O)=O c1(CC)cc(C(=O)N(CCCC(=O)NCCCNC(N)=O)C)n[nH]1 C12(CNC(C3CCC(=O)NC3)=O)CN(C(c3cnn[nH]3)=O)CC1CCO2 C1(C)(C(=O)NCC(C)(C)NC(C(CC)n2ccnc2)=O)CCC(=O)N(C)C1 N1(C(C(COC(C)C)NC(C)=O)=O)CC=CC(NC(C2(C)CS(=O)(=O)C2)=O)C1 C(=O)(C(C)(C)CCCO)N(C)CC1(CNC(C2(CC3CC3)CC2)=O)CC1 N1(C(COC)C)CCCN(C(=O)C#CC(C)C)C(C)C1 c1(C(=O)NCc2cc(NC(=O)NCCOc3ccon3)no2)cc2nc[nH]c2cn1 c1(C(C)NC(C(C2CCN(C(c3c(COC)ncs3)=O)C2)C)=O)c(C)noc1C c1(C(N2CCC(NC(C3N(CC=C)CCC3)=O)C2)=O)cc(C)c2ccccc2n1 C1(C(=O)NCC(CN(C(=O)CCn2ncn(C)c2=O)C)O)CCC2(CCC2)CC1 C(=O)(C(C)CC(N)=O)N1CCC(N(C(=O)C(C)OC)CC)C1 C1(C(N(C(C(N2CC(CCO)C2)=O)C2CC2)C)=O)CS(=O)C1 CC1(C)COC(CC(=O)NCC(=O)NCC(=O)NCC(F)F)C1 N1(C(C(F)=CC)=O)CC(C)C(NC(=O)Cc2cc(OC)ccc2F)C(C)C1 C(=O)(C(C)(C)C(O)C(C)C)NC1(CC)CCN(C(=O)C(C)C(F)F)C1 c1(C(C)NC(C)CN=[N+]=[N-])cc(F)ccc1C(N1CCCC1)=O CC(C)CN=C(NCc1ncn(C)n1)NCC1C(F)(F)C12CCCC2 N#Cc1cccc(C(=O)NCC2(NC(c3cccnn3)=O)CC2)c1 Cc1coc2c(C(N3CCCC(CCNC(=O)C(C)CC(F)F)C3)=O)cccc12 C1(C(N(CCN(C(=O)CC2OCCC2C)C(C)C)C)=O)OCCC1C N1(C(C(C)(C)C)=O)CCN(C(C2CCC(=O)O2)=O)C(CC(F)F)C1 CCC(CC(=O)N1CCCC1(C)C(=O)N(C)Cc1ncc(C)o1)CC(C)C c12cccnc1CNC2=O.CC1=NOC(C(=O)NCCCN2CC=CC2)C1 c1(C(=O)NC(C2(O)CN(C(c3n[nH]c(=N)s3)=O)C2)C)cccn(C2CC2)c1=O N1(C(c2ccc(CC)cc2)=O)CCN(C(=O)C2=NNC(=O)C2)CC1CC(F)(F)F C(=O)(C(C)N1CCCC1)N(CC(=O)NCC(=O)N(C)CC)C C12(NC(=O)NC3CN(C4CCCCC4c4ccc(F)cc4)C3)C(=O)C3CC1C2C3 C1(O)(C(=O)NC(C)CNC(=O)Cn2cnnc2O)CC(F)(F)C1 C1(NC(C=CCCC)=O)CC2(C1)CC2NC(c1ccc(C(C)C)nc1)=O C12(CC(=O)NC(C=C)C3CCC3)CCC1CN(C(C1(CCC)CC1)=O)C2 N12CCC(O)(CC1)NCCC2=O.N1(C(C)(C)CF)CCN(c2ccccc2)CC1 c1(C(=O)NCC(C)(C)NC(c2ccncc2)=O)csc(-c2ncccn2)n1 CC1CN(C(C2CC3(C2)CC32CCC2)=O)CC(C)N(c2ncc3ncnc-3[nH]2)C1 C(=O)(C(CC1CC1)NC(c1ccn(CCF)n1)=O)N(CCOC)CC C(=O)(CCCSC(F)(F)F)NC(C1CC1(F)F)C=C N1(C(Cc2c(C)noc2)=O)CCN(C(C)CNC(=O)CNC=O)CC1 c1(C(=O)NCCNC(c2cc(C(CC)C)no2)=O)cc(S(N)(=O)=O)c(C)o1 C1(CC)CN(C(=O)CC2(C)CCC2)CCN1C(=O)Oc1cncc(OC(F)F)c1 c1(C(=O)OCC)ccc(C(=O)NC2CC(C)N(C(=O)C=NOC)C2)nc1C c1(CC)ccc(CC(=O)NCC2CCC(NC(=O)CC(F)(F)F)C2)cc1 c1(C(N(CC(C)NC(C(c2ccc(F)cc2F)CC)=O)C)=O)cc([N+](=O)[O-])n[nH]1 c1(N2CCN(C(C=CC)=O)C(CO)C2)ncnc2c1CCC2 CC(C)CC(C)CNC(=O)NC(C(F)(F)F)C1CCC1 c1(NC(c2c(C)nc(NC(c3ccc(C(F)(F)F)[nH]3)=O)s2)=O)cnc(O)nc1O Cc1ccc(C(=O)NCC2CC(NC(c3ccc(O)nc3Cl)=O)CC2O)c(F)c1 CN1CCC(C)(C(N2CCC(CCC(N3CC(C)(C(F)(F)F)C3)=O)C2)=O)C1 CC1CCC(CC(=O)NCC(O)CNC(=O)C(F)=CCCF)OC1 N1(C(C(C2CCOCC2)C)=O)CCCC(CNC(C2CC23CC3(F)F)=O)C1 C1(CCC)CN(C(=O)CC(F)(F)c2ncccc2Br)CCN1C(=O)OC(C)(C)C O=C(NN=Cc1ccc(Br)cc1)C1(C(F)F)CCOC1 N1(C(CC2(C)CN(C(c3cncc(Cl)n3)=O)C2)=O)CCC(CO)C(F)(F)C1 CC1(C#N)CCN(C(=O)C(CC2CCCC2)NC(C2C3CCC(F)C23)=O)C1 N1(C(=O)CSc2n[nH]c3ccccc23)C2CC3C4CC(C3C2O)C1C4O C=CC(CC)C(=O)NC1CCN(C(C2C3CC(=O)CC23)=O)C1C Cc1nn(CC(=O)N(C(C)CCNC(=O)CC(C)C)C)c(=O)c2ccccc12 C1(C(c2n(CCOC)nnn2)NC(n2cnnc2)C)CC2(C1)CC(F)(F)C2 n1(CC)cnc2nc(N3CC4C(C)C4C3)nc(NCC(c3ncc[nH]3)C)c12 C1(CNC(C(CC)C#N)=O)CCN(C(c2ccc(F)c(Br)c2)=O)C12CC2 C1(CN(C(C2CC(C3CC3)C2)=O)CC)CCN(C(=O)CCc2nccs2)CC1 c1(C(=O)NCC2(C)N(C(C3C(C)(C)C3CO)=O)CCC2)ccc2nc[nH]c2c1 c1(OCC)ccc(CNC(C2CC(=O)N(OCc3ccccc3)C2)=O)cc1OC c1(NC(=O)NC2CC(C)(C)OC2=O)cnc2c(c1)CCCO2 C1(CNC(C=CC(N)=O)=O)CC(O)CN1C(c1cc(-c2ccc(Cl)s2)on1)=O Cc1ncc(Br)cc1NC(C1CCN(C(C2CC2C)=O)CC1O)=O c1(C(=O)NCC2C(NC(C(C3CC3)OC)=O)CC2)ccc2nonc2c1 C(=O)(C(C1=C(C)CCCC1)N(CC)Cc1cc(Cl)ccc1Br)NCC C1(CNC(C2CCC(COC)C2)=O)CC2(C1)CN(C(=O)C(F)=C(C)C)C2 N1(c2ccc(C(=O)OCC)cn2)CC(NC(c2c(C)cccc2F)=O)CCC1C c1ccc(N(c2csc(-c3nn[nH]n3)n2)C(=O)COC(F)(F)F)cc1 N1(C(CCc2n(C)ncc2)=O)CC(NC(C2(CO)CCOC2)=O)CC2(CC2)C1 CC(C)(C(=O)N1CCC(C2CCCO2)C1)C1CCN(C(c2coc(CO)c2)=O)C1 N1(C(C2CCC(=O)N2)=O)CC(C(N2CC(CO)(CO)C2)=O)C(C2CC2)C1 C1(S(N)(=O)=O)(C(=O)NCC(CNC(C(Cc2ccc(OC)cc2)C)=O)O)CCC1 N1(C(C2CCN(C(c3cc(CC)[nH]n3)=O)C2)=O)CCC(C)(CCO)CC1 c1(OC)c(C(N2CC3CCC(C3)C2)C(=O)NCc2cccs2)ccc(Br)c1F N1(C(C(CC)N(C)CC)=O)CCn2ncc(C(=O)O)c2C1 c1(CC(=O)NCC2C(NC(C3(C)ON=C(C)C3)=O)COC2)cccc2nsnc12 c1(C(N2CC(OCCNC(=O)CCCCC3CC3)C2)=O)cc[nH]c2nccc1-2 C1(NCCCC)C=CCCC1.c1(-c2cocn2)ccccc1 N1(C(CCC(C)(C)OC)=O)CC(C)N(C(=O)CCc2ccccc2C#N)CC1C N1(C(c2cc(CC)nnc2C)=O)CC2CCN(C(C3CC34CC4)=O)CCC2C1 c1(C(N2CCC(CCC)(NC(C3CCCCO3)=O)C2)=O)cc(O)nc(C)n1 CCC(CC)C(C(=O)NCC(CC1CC1)C(=O)NCC1CC(F)C1)OC CCCCC(O)CC(=O)NC1CCCC1NC(c1ccc(C(F)(F)F)c(O)c1)=O C1(C(=O)NC2(NC(C3CCCN(C(=O)OC)C3)=O)CC2)CCCC(C)(C)O1.C1CS1 c1(C(=O)NCC2C(NC(c3c(C)nc(C4CCC4)o3)=O)C2)cn(C)c(=O)cn1 C(CC(=O)NCc1cnco1)(C(F)(F)F)NC(c1c(CC)nc(C)o1)=O CCCC(O)(CCC)CC(=O)NC(CCN(C)C(c1cnc(C)s1)=O)C(C)(C)C N1(C(C2CCC(CC(n3cccn3)=O)CC2)=O)CCCN(C(=O)C(F)F)CCC1 C=C=CCCC(=O)NCC(C)(C)CNC(c1nocc1CC)=O c1(-c2nc(NC(C3(Br)CC3)=O)sc2)cccc(-c2ncc[nH]2)c1 C(=O)(C1CCCc2scnc21)N1CCOCC(CNC(C=CSC)=O)C1 C(CC(=O)Nn1cncn1)NC(CCNC(C1(C)CCC1)=O)=O c1(C(=O)NCCN(C(C(c2ccc(C)o2)C)=O)C)scc(C)c1Cl Cc1ccc(C=CC(=O)NCC2CC2NC(=O)CCC(=O)c2ccncc2)s1 C1(C(N2CC(NC(c3c(CC)con3)=O)C(O)C2)=O)CCOCC12CCCCC2 N1(C(C(C)NC(=O)CC(C)(C)C)=O)CCC2C1CCCN2C(=O)C(=O)N(C)C C(=O)(C(C)CN(C(=O)C(Cn1cccn1)NC(=O)CCc1cnn[nH]1)C)NC C1(C(=O)NCC(CNC(c2c[nH]nc2C(F)(F)F)=O)O)CCCCC12CCC2 C#Cc1c[nH]nc1C(N1CC(C(C(N2CC(C#N)C2)=O)OC)C1)=O c1(CC2(C(=O)NC(CC(C)=O)C)CC2)ccc(OC(F)F)cc1F c1(C(=O)NC2C(CC)CN(C(=O)Cc3cnns3)CC2)cccc2cncn12 N1(CCC(=O)NC(CCOC)CNC(=O)C(O)P(C)(C)=O)C(=O)NC(C)(C)C1=O Cc1cc(Cl)cc(CN=c2[nH]c(CC(=O)N=c3cc[nH][nH]3)cs2)c1O C#CC1COCCN1C(C1CCCCN1C(=O)Cn1ccnc1)=O Cc1cccc(Br)c1C(N1CCCCC1)=O.C12CCC(C1)N(C1CC1)C(=O)OC2 C(=O)(CN=c1cc[nH]cc1)NC(C(c1cn(C)nn1)NC(CCCN(C)C)=O)=O N1(C(COCCC=C)=O)CCN(C)C(CNC(=O)C(C)(C)c2cnn(C)c2)C1 Cc1ccc(F)nc1CNC(N1CCCCC1c1ccc[nH]1)=O C(=O)(C(C)CCC(C)(C)C)N(CCCCNC(c1nnn(C)n1)=O)C Cc1nc2ccc(C(N3CC(NC(=O)CC4(N(C)C)CCCC4)CC3C)=O)cc2[nH]1 c1(C(=O)NC(C)(C)CNC(=O)C=Cc2cnc[nH]2)c[nH]c2ccncc12 C(=O)(C(Cc1cccc(C#N)c1)N(C)N1CCCC1(C)COC)OCC C1(CNC(C(c2ccccc2F)C)=O)CN(c2ccnc(Cl)n2)CC(C)(C)O1 Cc1ccc(C(=O)C(=O)NC(C)CC(C)NC(=O)CC2CC2C)cc1 c1(C(N(C(C)CNC(c2ccc(Cl)nc2O)=O)C)=O)ccc2oc(O)nc2n1 N1(C(C(C)CO)=O)CCC2(CC1)CC2NC(c1ccc(C(F)(F)F)cn1)=O c1(C(N(CC(C)NC(C2CC2C2CC2)=O)C)=O)cc2ccc(F)cc2o1 C1(O)(CNC(C(C)(Cl)Cl)=O)CCCN(C(=O)C(O)c2cnc[nH]2)C1 C1(CC(=O)NCCCOCCNC(c2c(CC)nc[nH]2)=O)CC2C=CC1CC2 C(c1ccc(Cl)cc1)=CC(N1CC(O)(C(C(=O)NCCCCCCOC)F)C1)=O c1(C(N2CC(c3nc(CCC(=O)OC)on3)C2)=O)cn(C)c(=O)nc1O N1(C(Cc2ccc(CC)cc2)=O)CCCC(CC)(NC(=O)CCC#N)C1 C(CC1=CCN(C(c2csc(-c3cccs3)n2)=O)CC1)NC(C(C)CC(N)=O)=O c1(OC)cc(C(=O)N(C2CN(C(=O)C(F)(F)COC)C2)C)cnc1O c1(C(C(=O)N(C2CC2)CC)CC)ccc(F)c(F)c1F c1(C(=O)NCC(C2CCC2)NC(c2c(CC)c[nH]n2)=O)cc(C)c(N)cn1 CC(C)C(C(=O)N1CC(O)C(O)C1)NC(c1cnc(C(C)C)o1)=O C1(C(N2CC3(CC(NC(C4CCC(=O)O4)=O)C3)C2)=O)CCc2nccn2C1 N1(C(=O)COCCC2OCCO2)CC2CCN(C(c3cccc(F)c3)=O)C2C1 C1(COC)(NC(c2cccc[n+]2[O-])=O)CCCN(C(C2COC3(CCC3)C2)=O)C1 Cc1ccc(OCC(=O)NC2CC3(CC3)CN2C(=O)C2=COCCC2)cc1C CCC(O)C(C)(C)C(=O)N1CCN(CC2(NC(=O)C(C)c3cccs3)CC2)CC1 c1(C(=O)NCCC(C)NC(c2ccncn2)=O)ccc2c(c1)C(C)CO2 N1(C(=O)C=Cc2cnccn2)CC2(C(N3CC(O)(C4CC4)C3)=O)CC1CCO2 C(c1ccccc1C#N)=CC(N1C2CC(CNC(C(OC)OC)=O)(OC2)C1)=O c1(OC)cc(OC)c(OC)cc1CCC(=O)N(CCSc1cccc(I)c1)C c1(NC2CCN(C(C(CC)c3ccccc3)=O)C2)cccc(C)c1 c1(C(N(CC(CNC(C(c2cccnc2)OC)=O)O)C)=O)nccnc1N c1(C(=O)NC(CN(C(=O)CCC2CCOCC2)CC)C)coc2c1COC2 c1(C(N2C(C(C)C)CN(C(=O)C3=CCCC3)CCC2)=O)ccc2cnc(C)n2c1 S(=O)(=O)(c1ccc(NCC(C)(C)C#N)c(C#N)c1)NCc1ccc(OC)c(F)c1 c1(CC(N2C(CNC(CC(C)C(F)F)=O)C=CC2)=O)ccc2c(c1)CCCO2 N1(C(CSCC(N)=O)=O)CC2CCCC2(NC(c2ccccc2F)=O)C1 C1(NC(C2CC(CNC(CC=CC=C)=O)C(O)C2)=O)CC2(CCC2OC)C1 C1(CNC(C)CCc2ccccc2)C2CCN(CC2)C1 C1(C(=O)NCC#CCNC(=O)Cc2ccc(Cl)s2)CC2CCCCN2C1 N1(C(CC(=C)C)=O)Cc2nccn2CC(NC(=O)CCc2nc(CCC)no2)C1 C1(C(=O)NCC2N(C(C(F)=CC)=O)CC(OC)C2)CCC(=O)N(C(C)C)C1 S(=O)(=O)(c1cnc(OC)cc1OC)C(c1c(OC)ccc(F)c1)c1ccccn1 C1(NC(C(C)SC(C)C)=O)C=CCN(C(C2(c3ccc(F)cn3)CC2)=O)C1 c1(NC(C(CN(C)C(=O)OCc2ccccc2)(C)C)=O)cnn(C)c1C#N c1(N(C)CC2CCCC2)nc(=NCCn2ncc(Br)n2)[nH]c2ccccc12 CCCC(C#N)C(=O)N1CC(=C(F)CNC(=O)Cc2csc(C(C)=O)c2)C1 C1(CNC(c2cc(OC)nc(C)c2)=O)CC2(CCC2)CN1C(=O)C(=O)NC1CC1 N1(C(C2(CC#C)CCOC2)=O)CCCCC1CN(C)C(c1cncnc1)=O CCC(C)CC(C)(c1nnnn1C1CCCCC1)NC(c1cccc(Cl)c1)(C)C C(=O)(C(=O)C(C)(C)C)N1CCC(N(C)C(c2cc[nH]n2)=O)C1 N1(C(CN(CC)CC)=O)CCCC(NC(C2CCC(OC(C)C)CC2)=O)CC1 N1(C(c2cnc(SC)s2)=O)CCN(C(=O)CC(F)(F)F)CC1C1CCC1 Cc1ccc2cc(C(N3CC(N(CCO)C(C4CS(=O)(=O)C4)=O)C3)=O)cn2c1 Cc1cnc(C(=O)NCC(CNC(c2cc(=O)cc[nH]2)=O)CO)c(F)c1 N1(C(C2C(C)(C)CN2C(=O)Cc2ccc(F)nc2)=O)CCCC2OCCC2C1 N1(C(C(C(CC)C)NC(=O)C(=O)C2CCCC2)=O)CCn2nc(C)cc2C1 C(=O)(C(C)(C)CC(C)(C)C)NC(CC(C)C)CNC(c1n[nH]cc1Br)=O c1(C(=O)NCCC(C(C)C)NC(c2c(C)nco2)=O)oc2ccc(Cl)cc2c1C c1(CC(=O)NCCC2CCCN2C(=O)C(C2CC2)C2CC2)cccc(Br)c1 Cc1c(C(=O)NCCCCCN(C)C(C2CC23CCCC3)=O)ncn1C c1(-c2nc(C(C)C)nn2C2CSC2)cn2cc[nH]c(=O)c2n1 Cc1cc2c(cc1C)OC(C(=O)NCC1CCN1C(C1(O)CCOCC1)=O)C2 CC1(C)C(NC(=O)Nc2ccoc2C(F)(F)F)C2CCCOC12 CC(C)CCC(C)NC(=O)C(C1(C)CC1)NC(=O)CCCc1cnn[nH]1 C1(C(N2C(CNC(c3ccnn(C)c3=O)=O)CCC2)=O)CCC([N+](=O)[O-])CC1 c1(C(=O)NCC(C)(CO)NC(C2N(CCC)CCC2)=O)c(C)cnnc1O N1(C(CCC(=C)C)=O)CCCC(C2CCN(c3ccnc(COC4CC4)n3)C2)C1 c1(OCC#N)ccccc1Nc1cccc(-n2cnnc2)c1 C12(C(N3CC(N(C)CC)C3)=O)CC(CO1)N(C(=O)Cn1cc(C)cn1)C2 c1(NCC(C)(C)NC(=O)C(C)CC(N)=O)ncnc2c1nnn2-c1ccc(F)cc1 S1(=O)(=O)c2ccc(cc2F)CN1.c1(SC)cccc(C(C)(F)F)n1 c1(OC)c(C(F)F)cccc1CC(=O)NCC1CCN1C(=O)C=CCO N1(C(C23CC(C(=O)OC)(C2)C3)=O)CCC(C)CC(C)C1.C12CC3(C1)CC(C3)N2 CC(C)C#CC(=O)NC1COCC1NC(c1cccnc1N(C)C)=O N1(C(C2(CCNC(C=CCC)=O)CC2)=O)CCS(=O)C(C)C1 C1(OC)(CNC(C2CCCN2C(c2cc(Cl)no2)=O)=O)CCC(C)C1 C(=O)(C1SCCc2sccc21)NC1C(C)CCN(C(c2cnc3sccn23)=O)C1 N1(C(C2CN(CC)C(=O)C2)=O)CCc2sc(CNC(=O)CCCC(C)C)nc2C1 C1(NC(c2c[nH]c(=NC)s2)=O)CS(=O)(=O)CC1NC(=O)Cn1cnc([N+](=O)[O-])c1 C(=O)(C(CC)c1ccccc1)NC1(CCCNC(CCSCCC)=O)CC1 c1(C(=O)NCC2(CO)CC23CCC3)nc2ccccc2o1.C(=O)(C(F)n1cccn1)N Cc1cc(O)ncc1NC(=O)C(CNC(c1cccc(O)n1)=O)CC1CC1 Cc1c(C(=O)NC(CNC(=O)COc2c(F)cccc2F)C(C)C)c(Cl)nn1C CC(C)(C)CC(O)C(=O)N1CCC(CNC(C2(n3cncn3)CC2)=O)C(CO)C1 c1(C(=O)NCC2(C)COCCN(C(=O)C=C(Cl)Cl)C2)cc(S(C)(=O)=O)co1 n1(CC)cc(Cl)c(C(=O)NCC(C)NC(C2CN(C)C2)=O)n1 C1(CC)C(C(N2CCOCC2CC2CC2)=O)CCCN1C(c1cnco1)=O C(=O)(CCC(F)(F)CN=[N+]=[N-])N1C(C)(C)CC(CNC(=O)CSC(F)(F)F)C1 C(=O)(C(C)S(=O)(=O)C(C)C)N1CC(C(C)NC(CCN(CCC)C)=O)C1 CC(C)(C)C(C(=O)NC1CC(CNC(C2CCCS2)=O)C1)NC(=O)OC(C)(C)C N1(C(C(c2ccc(C)cc2)F)=O)CCC(NC(=O)CO)C12CC2 C(=O)(CC(C1CC1)NC(C1(NC)CCC1)=O)C(C1CC1(F)Cl)=O.CN C12CCN(CC1F)OC2=O.C1(N(C(C(C)CO)=O)c2cnn(C)c2)CCN(C)CC1 c1(OC)ncc(Cl)cc1C(=O)NCCC1CCN(C(=O)C(C)(C)N(C)C)CC1 N1(C(c2cc(CC)sn2)=O)CCC2CCN(C(=O)C(CC(C)C)OC)C2C1 N1(C(c2c(C)nc(O)cc2)=O)CC(C)CN(C(=O)CC2C=CCCC2)CC1C C(=O)(CC(CC)NC(=O)CCN1CCOC1=O)N(CC(CCC)O)C c1(NC(CC2CC(NC(CCC(C)=O)=O)C2)=O)ccc(C)c(C(=O)OC)c1 N1(C(c2ccn(CCC)n2)=O)CC2CCOC2(CNC(=O)C2=NOC(C)C2C)C1 N1(C(c2c(-c3cn(C)nc3)ocn2)=O)CCCC1C1CCCN1C(=O)COCCF C1(F)(C(=O)NC2(NC(C3CC(NC(=O)OC(C)(C)C)C3)=O)CC2)CCCCCC1 CCCC(C(=O)OC)C(=O)NCC(CC)NC(=O)C(c1cccc(Cl)c1F)(C)C Cc1cnc(C(=O)NCCOCCn2cc(-c3cccs3)nn2)cn1 S(=O)(=O)(c1ccccc1NC(=O)C(C)NCC(C1CC1)OCC)NC(=O)C1CC1 N1(CC(=O)NCCC2CC(NC(C(F)OC)=O)C2)CC2CC2C1 C1(CNC(C2CC3C(C2)C3(F)F)=O)CN(C(=O)Cc2cccc(Cl)c2F)CCCO1 C(=O)(CCS(N)(=O)=O)NC1(CNC(c2nnc(C)o2)=O)CCCCC1 C=CCC(CC=C)C(=O)N1CCCN(CCNC(c2ccc(OC)nc2)=O)CC1 C(CC(C)C)(C(=O)N1CCOCC(NC(=O)CCc2cc[nH]n2)C1)OC C(=O)(C1=CCCN(C(=O)CC(CC)C(F)F)C1)N1CCC(OCC=C)CC1 C(=O)(CC(O)CC(C)(C)C)NCC1(Cn2cc(-c3cc(C)c(F)cc3)nn2)CC1 C1(CNC(CCN(C(C)C)C(c2cccc(=O)o2)=O)=O)CC(O)C12CCC2 C1(C(=O)NC2CC(NC(c3c(C)nn[nH]3)=O)C2)CC(=O)N(c2ccccc2)C1 Fc1ccc(C2CNCC(c3nccn3CCc3nc(C4CC4)no3)C2)cc1 c1(NC(C2CCN(C(=O)COCC3CCCO3)C23CC3)=O)cnc2ccnn2c1 CC1(C(=O)NCC(C2CCCC2)NC(=O)COc2cccnc2)CC=CCC1 N1(C(CC2(C)CC2)=O)CCC2CCCC12CNC(c1nc[nH]c2ncnc1-2)=O N1(C(c2c(C)oc(CO)c2)=O)CCN(C(c2cnn(C)n2)=O)C(CCO)C1 N12CCN(CC1)CCNC(C)C2=O.c1(NC(c2cccs2)=O)ccccc1I C(C(C)(C)C(F)(F)F)NC(C1N(C(C(C)Cn2ccnc2)=O)CCSC1)=O CCC(CC)C(C(=O)NC1CC(C)CN(C(C2(C)COC2)=O)C1)N1CCCCC1 C(CCC(C)(C)NC(C1CCCCN1CC(F)F)=O)NC(c1nc(C)oc1)=O C#CC1(NC(C2(C(C)NC(C3CCN(OC)CC3)=O)CC2)=O)CCCOC1 Cc1cc(C(=O)NCC23CC2CN(C(C2(N4CCCC4)CCC2)=O)C3)c(C)s1 C1(c2n(CC(=C)C)nnn2)(NCc2ccccc2Br)CCCSCC1 C1(C(=O)NC(CCC)(C)CC)CN(C(C2CC2C(F)F)=O)C2(CCC2)C1 c1(NCNC(N(CC(O)COc2cccc(Cl)c2)C)=O)cc(OC(F)F)ccn1 N1(C(C(CNC(C2CC3(CSC3)C2)=O)O)=O)CCC2(CCC2)CC1 C1(C(N2CCCC(OC)C2)=O)CC2(CCN(C(c3cncnc3)=O)CC2)C1 C1(NC(Cc2scc(C(C)(C)C)n2)=O)CCCCC1NC(=O)Cc1cnns1 c1(CN(C(=O)C(c2ccccc2)C2CCCC2)C2CCCC2)ccccc1I Cc1ccnc(C)c1C(N1CCCC(CNC(c2nccnc2C(N)=O)=O)C1)=O Cc1occ(C(F)(F)F)c1C(N1CCCC(CCO)C1)=O N1(C(CCC)=O)CCC(CC(=O)N(C2CN(C(=O)Cc3sccc3Cl)C2)C)CC1 C1(NC(C=NOC)=O)C2CC3CN(C(c4cc[nH]n4)=O)C1C3C2.c12cccc(c1)S2 C(=O)(C1CCc2cccnc21)N(CCCNC(c1n[nH]c(C)c1Br)=O)C1CC1 CCC(C)(CNC(=O)CCc1ncccn1)NC(=O)COC1CCC1 n1(CCOC)cnc(=NC(=O)N(C2CC2)Cc2cc(C)cc(C)c2)[nH]1 C(=O)(CCCC(C)(C)CC)N1CC(O)(CN(C(C(C=CC)O)=O)C2CC2)C1 c1(OC)c(-c2nc(NC(=O)C(C)NC(c3cccs3)=O)cs2)c(C)nn1C C(=O)(C1=CCCC(C)(C)C1)NC(C(C(C)C)NC(=O)C#CC1(C)COC1)C.C1CO1 c1(CC(=O)NCC2N(C(C3CN(C(=O)NC)C3)=O)CCCC2)ccc(C#N)cc1 N1(C(c2ccn(CCC)n2)=O)CC(C(=O)Nc2csnc2C)CC(C)C1 c1(C(=O)NC(C(C)NC(CC=CC)=O)CO)nn(C)cc1S(N)(=O)=O CC(C)(C)C(=O)NCC(=O)NCCNC(=O)CC1CSC1 O=C(C1=CS(=O)CCC1)NC1CCCC1CNC(c1ccnnc1Cl)=O C1(O)(CC(N2CCN(C(=O)CC3CCCOC3)C(CF)C2)=O)CCCCCC1 c1(C(=O)NC(C2CC(NC(c3cc(OCC)ncc3)=O)C2)C)nc(C)ccc1F c1(SC)ccc(Cl)c(C(=O)NC2(C(=O)O)CC2C)c1 CC1CCC(CNC(c2cc(C3CCC3)nn2C)=O)N(C(c2cnco2)=O)C1 CC1CCN(C(c2ncccc2C(F)(F)F)=O)CC1NC(=O)CCSCC(N)=O N1(C(C2C(C)C2)=O)CC(CNC(c2cnn(-c3ccccc3)c2)=O)C(C)C1 c1(CNC2CCCN(C(c3c(CN)cccc3)=O)C2)ccncc1[N+](=O)[O-] C1(NC(c2c(NC)ccc(F)c2)=O)CCCCN(C(C2CC23CC(O)C3)=O)CC1 C1(NC(C2(CF)CCC2)=O)CC(CO)N(C(=O)CCc2ccc[nH]2)C1 C=CCCCCCCC(=O)N1CCCC2(NC(=O)Cc3c(C)cccc3Cl)CC12 C1(CC=C)(C(=O)NCC2(CC)CCOC2)CCCN1C(=O)CN1CCCNC1=O CC(CC(F)F)C(=O)N1CC=CC1(C)C(=O)NCCN1CCOCC1 c1(OC)ccc(F)c(C(N2CCN(C(c3cc(Br)c(C)o3)=O)C(CF)C2)=O)c1 Cc1ncc(N)cc1C(N1CC=CC1CNC(c1c[nH]nc1C(F)F)=O)=O Cc1ccnc2nc(C(=O)NC3CC(C)N(c4nnc(C(C)(C)C)o4)C3)nn12 N1(C(C2(Cl)C(C(C)=O)C2)=O)CC(C(=O)N(CC(F)F)CCO)C2(CC2)C1 N1(C(C2CCN(C(C(CCC)N(C)C)=O)C2)=O)CCC2(COC(C)C2)C1 C(C(CO)(CO)NC(=O)COCP(C)(C)=O)N(C)C(c1cncc(CN(C)C)c1)=O CN1N=C(C(=O)N2CCOC(C(=O)NCCc3cccc(Cl)c3)C2)CCC1=O CCC(C)C(CC(=O)Nc1cc(C)ccc1C)NC(=O)C(O)(COC)COC c1(C(C)C)n[nH]c(=NCC2CC(CNC(C34CCC(CC3)C4)=O)CO2)o1 C(=O)(C1Cc2ccc(F)cc21)N1CCC(N=[N+]=[N-])(C(=O)NCC(C(C)(C)C)OC)C1 N1(C(c2c(C)ocn2)=O)CCC(NC(C2CC23CCOCC3)=O)C12CC2 c1(NC(COCC)=O)cccc(C(C2(C)CCNCC2)C)c1 C(CC(C)(C)C)(C(=O)NC(C1CCN(C(C2(C(F)F)CCC2)=O)C1)(C)C)OC c1(N(C)Cc2cnn(C)c2)nc(=NCC2CC3CCCC3C2)[nH]c2ccccc12 c12ccc(cc1)c(=O)[nH]2.C1(CC(=O)N(CCCNC)C(C)C)CCC(C(F)(F)F)O1 C1(NC(C2C(C)(C)OCC2)=O)C2CC3C(C2)C13C(=O)NOCC1(F)CCC1 C12(C(=O)NCC(C)NC(=O)C(C)(CO)C(=O)NC(C)(C)C)CCC(C)(C1)OC2 CCC(O)C(C)(C)C(=O)NC1CCC1CNC(=O)CCc1cnco1 N1(C(C=C(CC)C)=O)CC(C)(C(=O)NC2CN(C(=O)OC)C2)C1 c1(C(N2CCC(O)(C(CNC(C(C)C)=O)C)CC2)=O)ccc2c(c1)CCCCN2 c1(C(=O)NC2CCC(C(=O)NC3(CC(C)=O)CC3)C2)sc(C)cc1C c1(-n2cc(C(C(C)(C)C)NCCn3ccc(Br)n3)nn2)c(F)c(F)cc(F)c1F O=C(CCCCCNC(C1CC1(F)Cl)=O)NCC1=CCCOC1 C1(C#CC(=O)NC(C)CC(C)NC(=O)C(c2cccc(F)c2)(C)C)(CC)CC1 c1(C(=O)NCC2C3CN(C(C(C4CC4)OCC)=O)CC32)cc(Br)cc(F)c1C C(=O)(CCCCC(C)C)N(C1CN(C)NC1=O)CCC c1(C(=O)NCC2(C(C)NC(c3c(C)cno3)=O)CC2)ccc(OC(F)F)cc1 C1(N(C(CN(CC(C)(C)C)C)=O)C)CCCC(NC(c2nnn(C)n2)=O)C1 C1(NC(C(C)C2CC2)=O)CC12CCN(C(=O)Cn1nnnc1C(C)C)CC2 CCCCCCOC(C)C(=O)NC(CN(C)C(C1SCC=C1C)=O)CC C(CC(C)(C)C)N(CCC(=O)N)C.C(CC(=O)NCCC(=O)N(C)CC1(CC)CC1)OC C(=O)(C(CCC(C)(C)C)NC(c1cc(I)c(F)cc1F)=O)OC CCC(CC(=O)N1CCC1c1ccc(C)cc1)C(C)(C)C.N1CC(C)C1(C)C CS(C)(=O)=Nc1cccc(C(=O)NC2CC3(C2)C(F)(F)C32CCC2)c1 C1(NC(C(CC#C)C)=O)CC2CCC1N2C(=O)Cc1csc(-c2ccoc2)n1 c1(C(N2C(CNC(C(Cc3ccc(F)cc3)OC)=O)CCC2)=O)c[nH]c(C#N)c1 c1(C(N(C)CC2CCCC(NC(=O)Cc3cn[nH]c3)C2)=O)cc2cn[nH]c2cn1 C#CCCCCCCC(=O)N1CCC(N(C(c2conc2C2CC2)=O)CC)C1 Cc1cncc(CCC(=O)NC2CC(NC(c3ccc(CO)cn3)=O)CC2O)c1 c1(OC)ccc2nc(N3C4CCC3CC(O)(C(F)(F)F)C4)sc2n1 C1(C(=O)OCCCO)CCCC(F)C1.C1CCC(=O)N1CC(F)(F)F N=c1[nH][nH]c(C(=O)NCCCNC(=O)CC2CC(F)C2)c1Br Cc1cc(OC2CCN(CC3CCCCN3)C2)ccc1N(C)C C1(C(N2CC(C(C(=O)N(CC(CC)O)C)OC)C2)=O)CN(C)CCN1C c1(CC2CCN(CC(=O)NC(C)(C)C)CC2)cccc2cc(O)ncc12 c1(OC)ccc(F)cc1C(N1CCC2(CC2C(N2CCCC2)=O)C1)=O c1(C(=O)NCC2N(C(C(C)NC(C)=O)=O)CCC2)cc2nccc(Cl)c2s1 C1(NC(CCc2nc(C)sc2)=O)COC2(CCN(C(=O)CC(C)C3CC3)C2)C1 CCCC(C)C(C(=O)Nc1ccc(COC)cc1)N1CCCC1C(C)CC C1(C(=O)NC2C3CN(C(COC(C)C)=O)C2C3)CC2(CCC(F)(F)CC2)CO1 n12c(nnc1C1CC1C(=O)N(OC)C)N1CCOC(C1)C2.C1C(=O)N1.N.C(C)C.S c1(C(N2CCCN(C(C=CC)=O)CC2C)=O)cc(F)cc2nc(S)[nH]c12 c1(C(=O)NC(C)CC2CN(C(=O)CCCOCc3ccccc3)C2)occc1F c1(NC(C(Cc2cn(CC)nn2)(C)C)=O)ccc(C)c(Cl)c1Cl.C12CC1CNC2 N1(C(c2n(C)ncc2)=O)CC2CS(=O)(=O)CC2(NC(=O)CCC2(C)CC2)C1 C(=O)(C1CCCc2c[nH]nc21)C(=O)CC1NC(=O)NC1=O.C12(CF)CN(C1)C2=O.N c1(C(C)=O)cccc(C(=O)N(C)CC2(O)CN(C(=O)C(C(C)C)NC(N)=O)C2)c1 N1(C(C2C3CCCCC23)=O)CC(NC(COc2c(C)occc2=O)=O)C2(CCC2)C1 C(N=c1[nH]c(C(=O)NCC(=O)NC2CCCC2)cs1)c1cccc(N)n1 C#Cc1cncc(C(N2CCN(C(=O)CCn3cc(C)cn3)CC2C(C)C)=O)c1 CON=CC(=O)N1CCC(N(C(=O)CCN2CCOCC2)C)C1 C1(=O)C2=CCC(C2)N1.C(=O)(CCNC(C1(CCC=C)CC1)=O)NCC#C c1(C(=O)NCCN(CC(C)O)C(C2C(C=C)C2)=O)cc2n(n1)CCC2 C1(C(=O)NCCC(C)CCNC(=O)CC(C)C)(CC)CNC(=O)C1 n1(C(C)C(=O)NC2CN(C(C3(N(C)C)CC3)=O)CC2F)cnc2ccccc12 c1(C(N2C(CCC3N(C(CC=C)=O)CCCC3)CCC2)=O)cnc(C)cc1Cl c1(C(=O)NC2(CNC(CC(C)CSC3CC3)=O)CC2)ccc(F)c(F)c1 c1(CC(N2C(CNC(=O)CCOC3CC3)CCCCC2)=O)nc2c([nH]1)CCCC2 N1(C(CS(=O)(=O)N(C)C)=O)CC2CCCC2(C(=O)NOCCC2CC2)C1 C(=O)(C(C)(C#N)CC)NCC1(F)CC(NC(C2ON=C(CC)C2)=O)C1 c1(C(N(CC(C)NC(C2(CCF)CCC2)=O)C)=O)ccc(C(F)(F)F)nc1 C1(CCC)CN(C(=O)C(C)=CCNC(=O)C(C)COC)CCO1 N1(C(C2C(CC)C2)=O)CCC2(CCC2)C(NC(c2cc(C3CC3)n(C)c2C)=O)C1 N1(C(C2(CCOCC)CCC2)=O)CC(C2(NC(=O)C(C)CC3CCCO3)CC2)C1 C1(CC(=O)NCCNC(c2c[nH]cc2-c2ccc(Cl)s2)=O)CCCCC1O C1(C)(NC(c2cc(C(=O)OCC)on2)=O)CCOCC1CO N1(C(C(C)SCCCC)=O)CC2CCCC(CNC(c3sc(O)nc3C)=O)C2C1 N1(C(C(COC)C)=O)CC2(CCN(C(C3CCC4(CCC4)C(OC)C3)=O)CC2)C1 C1(NC(c2c(CC)onc2)=O)CCC12CCN(C(C1CC(F)C1)=O)CC2 C(=O)(C(C)(C)C(=O)NC1CCCN(C(=O)C=C2CCC(C)C2)C1)NC c1(C(=O)NCc2cc(C)nc(Cl)c2)ccc2c(c1)CN(Cc1c(Cl)ccnc1Cl)C2 CC(C)(C#N)C(=O)NCC1CCCC1NC(c1sccc1C(C)(C)C)=O c1(NC(c2nccs2)CC)cnc(-c2ccncc2)cn1 CC1CN(C(C2CC2[N+](=O)[O-])=O)CCN1C(=O)CC1CCCCC1 Cc1ccc(Cl)c(C(=O)NC2CCC(CCNC(=O)CN3CCSCC3)C2)c1N N1(C(c2ccc(C)cn2)=O)CCOCC(F)(CNC(C2CCCN2C)=O)C1 CCC(CC)C(F)C(=O)N(CC(O)CNC(C1CCC(CC)CC1)=O)C c1(C(C(=O)NC(C)CCCNC(C2(C3CC3)CCCO2)=O)(C)C)ccccc1F c1(CCNC(C2CC2NC(=O)CNC(C2C(C)(C(F)F)C2)=O)=O)cnc(O)[nH]1 N1(C(c2c(C)nc(C)o2)=O)CCC(NC(=O)C(C)(C)C2CCOC2)CC1C C12(C(=O)NCC(CC=C)NC(=O)C(F)(F)c3cnccn3)CCCC1CCC2 C1(N(C(=O)CCC2CCN(C)CC2)C)CN(C(=O)Cc2cccn2C)CCC1O Cc1ccc(S(=O)(=O)N2CCCCC2)cc1NC(=O)CCCCCc1cccs1 C=CCC(C(=O)NCCOC1CCN(C(=O)C=CC(N)=O)CC1)C(C)(C)C c1(C(=O)NCC(=O)NCC2CCN2C(=O)C2CC2)csc(C(F)F)n1 c1(OC)cc(Cl)c(C)cc1C(=O)NCC1CC1CNC(c1occ2c1CCC2)=O c1(CNC(C(F)=CC)=O)c(C)nn2c1CN(C(=O)C(F)(F)C(F)(F)C(F)F)CC2 c1(CNC(c2c(CCC)nns2)=O)cccc2nc(-c3cccc(CC)c3)cn12 Cc1cc(C(N2CCC(NC(=O)COC(F)(F)F)CC=C(Cl)C2)=O)cc(N)c1Cl c1(C(=O)OC)ccc2c(c1)C(C(=O)NCCN(C)C(c1cnc[nH]1)=O)CO2 C1(C(=O)NCc2ncc(CC)[nH]2)CC(C)(C)CCN1C(C1CCCC2(CC2)C1)=O c1(C(C(=O)NCC(CNC(c2nnn(C(C)(C)C)n2)=O)F)O)ccc(F)cc1F C1(NC(C(CCC)N(C)C)=O)CC2C1CCN2C(=O)CC(=O)N(C)C C#CCC(C)(C)C(=O)NC(C)CNC(C1C=CCCC1)=O N1(C(C2OCC(C)(C)C2)=O)CCC2(CCCCC2NC(=O)CCc2cnn[nH]2)C1 Cc1cc(N(C)C)ccc1CNC(=O)C(CO)c1ccccc1.N12CC(C1)C2=O C1(NC(C=C(C)C)=O)Cc2ccccc2C1NC(c1cnc2c(n1)CCCC2)=O C1(C2CC2)C(F)(F)CSc2cc(ncn2)S1.CC(=O)OC c1(CC(=O)NCCOCCCCCC)cc(F)c(F)c(F)c1 C(=O)(C1=CCCOC1)N(C1CCCN(C(c2coc(N(C)C)n2)=O)C1)CC N1(C(CN(CCC)C)=O)CCC2(CCOC2)C(CNC(c2ncsc2C)=O)C1 CC(C)C(C(=O)NC1CCN(C(=O)C=Cc2cccs2)CC1)c1ccc(Cl)cc1 C1(C(N(C2CN(C(C3CC(C(F)(F)F)C3)=O)C2)C)=O)CCCC1S(C)(=O)=O N1(C(C2CN(C(CC3CC(=C)C3)=O)CC2(C)C)=O)CCCC2(CCCC2)C1 CC1(C)CCN(C(=O)Cc2ccon2)C(C(=O)NC2CCN3CCC2C3)C1 c1(CC)ccc(Cl)c(C(N2CC3CCC3(CNC(=O)CC3CCCS3(=O)=O)C2)=O)c1 C1(CC)CN(C(=O)CCOCCOC)CCC1NC(C1CC(=O)C1)=O C1(CC(=O)NC2C(O)CC2O)CN(C(=O)C(F)(F)C2CC2)CC12CC2 N1(C(c2nc(C)cn2C)C(=O)NC)CCN(C(C)C)CC1C c1(C(N(CC(C)NC(=O)CS(=O)(=O)C(C)C)CC)=O)cc(S(C)(=O)=O)cnc1O C1C(C(=O)NCC)CCCN1C(=O)C(C)OC.C(N)(=O)N(CCOC)C1CC1 C12(NC(CC3CC(OC)C3)=O)COC(CNC(C3CCC(C)C3)=O)(C1)C2 c1(OC)ccc(NC(=O)C(=O)Nc2cccc(F)c2)c(C)n1 C1(CNC(C2C(C(C)C)C2)=O)CCN1C(=O)C(C)n1cncn1 c1(C(N2CCC3(C(C(=O)N=c4[nH][nH]cc4Br)C3)CC2)=O)cccc2ccncc12 C(=O)(C#CC(OCC)OC)N1CCC(N(C2CCCC2)C(CNCCC)=O)C1 C1(CCCOC)CCCCN1C(=O)C(N1CCN(C(=O)C=C(C)C(C)C)CC1)=O Cc1cc2c(cc(C(=O)NCC(C)(C)CNC(C3(O)COC3)=O)n2CC2CC2)s1 C1(CC=C)(NC(=O)C=CC(F)F)CCN(c2nc(C(C)CC)ns2)CC1 C(C)(CNC(c1cc(Cl)cs1)=O)(CO)NC(CSCCCC)=O C(C)(C)(CC(F)C(=O)N1CC(N2CCOCC2)C1)ONC(c1c(C)nc(C)o1)=O c1(SCCNC(=NCCCCC)NCCNC(=O)NC)nccc2ncccc12 c1(CCNC2CN(C(CC=C)=O)CC(O)C2)ccc([N+](=O)[O-])c(C)c1 c1(C(C=CC(N2CCN(C(Cn3cccc(N)c3=O)=O)CC2)=O)=O)cc(F)c(F)c(F)c1 C1(CC)CN(C(C2CC2c2ccccc2Cl)=O)CCN1C(=O)CCc1ncc[nH]1 c1(C(=O)NCC(C)N(C(c2c(C)cc[nH]2)=O)C)c(C)nc2ccccn12 C1(CNC(c2coc3c2CSC3)=O)CC2COCC2N1C(=O)Cn1cnnc1 c1(CC)c(C(N2CCCC2C2CCN2C(=O)CN(C)CCOC)=O)nnn1CC C(=O)(CC(C(F)(F)F)n1ccnc1)NC1C2CN(C(C(CC)(C)O)=O)C(C2)C1 C1(C(N(C2CCC(CNC(C3(C)CCCCS3)=O)CC2)C)=O)CCC2(CCC2)C1 C1(NC(C=C(C)C)=O)CCC2CN(C(=O)CSCC(c3ccccc3)=O)CC2C1 C1(CC)OCCC1CNC(C1(SC(C)C(=O)NC(=O)Nn2ccnc2)CC1)=O CC1CCN(C(C2CC2c2ccco2)=O)C(C(N2CCCC(C(F)F)C2)=O)C1 N1(C(C(CCSC)(C)C)=O)CC(C)C(NC(C2COCCOC2)=O)C(C)C1 N1(C(CCc2onc(C)n2)=O)CCCCC(C(=O)NCCCCC(C)(F)F)C1 Cc1nn(CC(=O)N(CC(C)(C)CNC(C2SCCC2C)=O)C)c(C)c1C Cc1noc(C)c1C=CC(N1CCCCC1CN(C(=O)CC1C=CCC1)C)=O Cn1cccc(C(=O)NCC(CC2CC2)C(=O)NCC2CCCC2(C)C)c1=O C12(CNC(=O)Cc3cncs3)CC1CN(C(=O)Cc1cncc(Br)c1)C2 n1(CC)nc(C(N2CC(NC(=O)C=Cc3ccoc3)C(F)C2)=O)c(Br)n1 c1(NC(=O)NCCN(CCCC)CCc2cccc(Br)c2)ccc(F)cc1 Cc1cc(C)c(CC(N2CCC(N(C(=O)C(F)=CCCF)C3CCC3)CC2)=O)s1 CC(C)(CC(F)F)C(=O)N1CCC(F)(CNC(C2CCCN2C2CC2)=O)CC1 c1(CN(C(CCC#C)=O)C)cccc(N)c1.N12CCC(C1)NC2=O CC1CC(NC(=O)C=CC2CCCC2)CCN1C(C1CC2CCC1C2)=O N1(C(C(CCCOC)C)=O)CCC2(C1)CN(C(=O)CCCCCC(C)C)CCO2 Cc1cncc(C)c1C(=O)NCC1CCN1C(c1ccc(C(C)(F)F)nc1C)=O N1(C(CCC(C)OC)=O)CC(NC(=O)CCCc2cccnc2)C2CCCCC12 CC(C)C(C(C)NC(c1cc(Cl)ns1)=O)NC(=O)C(=O)NCCC(N)=O N1(CCC)CCCCC1C(=O)NC(C)(CNC(c1nc(C(C)(C)C)no1)=O)C1CC1 Cc1nn(C)c(C)c1CNC(C)(C)C(=O)N1CCC(C(C)O)C1 C1(NC(C2C(CC)N(C(c3cnn(C)c3Cl)=O)CCC2)=O)CCCCC1N=[N+]=[N-] c1(C(N2CC(NC(C(C)NCCCC)=O)C(C)C2)=O)ncc(F)cc1C(F)F c1(CNC(C2CCC(=O)C2)=O)ccc(CNC(C2CCCC(=O)C2)=O)c(F)c1 C1(C(=O)NCC2(OC)CCN(C(c3c(CC)nn[nH]3)=O)C2)C2CCCCCCC12 CC(C)CC(O)C(=O)N1CCCC(CNC(=O)CC2OCCC2(C)C)CC1 C1(CCN(CCC(=O)NCCC)C)CCN(C(C2(CF)CC(=O)C2)=O)CC1 Cc1cn2c(CCC(=O)N(C)CCNC(c3ocnc3C)=O)csc2n1 c1(OC)c(CN2CCCC2(C)c2ccc(C)o2)ccc(C)c1F N1(C(c2n(CC)ccc2)=O)CCC(C(N2CC(CC(C)(C)C)C2)=O)(CO)C1 c1(NC(C(N2CCC(c3c(OC)nccc3)CC2)=O)=O)cccc2c1OCCO2 C(=O)(CC(O)CNC(C1CCCCC1O)=O)N(c1cccnc1)C S(=O)(=O)(c1ccc(NC2(CO)CCCCC2)cc1Br)NC(C)Cc1nncn1C C1(C(=O)NCC(C)(C)C)CC2CC1CC2NC(=O)COC1CC1 C(=O)(C1=CC2C=CC(C1)C2)NC(CC#C)C(=O)NCCOCCCO C1(NC(CN(C(=O)Cc2cn[nH]c2)CCOC)=O)CC(=O)NC1=O C1(CNC(C2C(C)SCCC2)=O)CC2CCC(C1)N2c1nnc(C(C)(C)C)s1 N1(C(Cc2[nH]c(=N)sc2)=O)CC2CC(NC(=O)CCc3ncc[nH]3)CC2C1 c1(N(C)C)ccc(CNC2CN(C(=O)CCOc3ccccn3)CCN2)nn1 c1(CC(=O)NC2(CN(C)C(C3(CS(C)(=O)=O)CC3)=O)CC2)cccs1 C1(C(=O)NC(CCC(=O)NC(CC)(C)C(N)=O)C)CC2COCC2C1 N1(C(CC=C(C)C)=O)CC=CC1CNC(C1CCC(CCc2ccccc2)O1)=O CC1(C)C(NC(=O)CCCc2ncco2)C1CC(=O)NC1CC1c1ccccc1 C1(NC(c2scc(OC)c2)=O)CC(NC(c2cccc(=O)n2C)=O)C12CCC2 c1(C(C)=O)cnc(NCCCNC(c2nc(C)n(C)n2)=O)nc1C(F)(F)F c1(COCC)cccc(CNc2nc(C)ns2)c1 c1(CC(=O)NC(CNC(C(C)SCCCC)=O)(C)CO)cccc(OCC)c1F c1(C(N2CCC(CNC(c3c(C)ccn3C)=O)C2)=O)nc(C2CC2)ncc1Cl N1(C(C2(OC)CCSC2)=O)CCCC(NC(c2cc(C(C)(F)F)n[nH]2)=O)C1 N1(C(C=CC)=O)CCC(O)(NC(=O)CN2CCCNC2=O)C1 CC1CN2CC1C2=O.c1(CCN)cnccn1.C(=O)(C(=O)N(C)C)NCCSC c1(C(=O)OC)cc(C(=O)NCC23CC(NC(C4CCOC4C)=O)(C2)C3)c(C)o1 Cc1cnncc1C(=O)NCC(=O)NCC1(C#N)CC1 c1(C(=O)NC2C=CCN(C(C(CCC)N(C)C)=O)C2)cc[nH]c2nccc1-2 CC1OCCC1CC(=O)NC(C1CCCC1)CNC(C1CCCC1)=O c1(C(=O)NCCC2N(C(c3n(C)nnc3)=O)CCC2)cc2ccc(F)cc2[nH]1 C1(NC(c2cccnc2)=O)CN(C(C2CC3(C2)CC(F)C3)=O)C2(CCOCC2)C1 C(=O)(CCCCCNC(=O)C1CC1)N(C)Cc1c(C)n[nH]c1C c1(C(=O)NCC(C2(O)CN(C(C3(C#N)CC(C)C3)=O)C2)(C)C)ccnn(C)c1=O C1(NC(C2CCCS2)=O)CN(C(C2CCCS(=O)(=O)C2)=O)C2(CCOC2)C1 c1(C(N2CC(CCNC(C34CCC(OC)C3C4)=O)C2)=O)n[nH]c2ccc(F)cc12 C1(CNC(=O)C=CCC2(NC(C3CC3F)=O)CCC2)CCCC2(CC2)C1 CCC(C)(O)CNC(c1cc(CNC(c2sccc2C)=O)no1)=O c1(C(=O)OC)cnc(NCC2(C(=O)NCCN(C)C)CCC2)nc1C C12(CNC(c3c(CC)scc3)=O)CCC(CC1NC(c1cc(=O)cc(Cl)[nH]1)=O)C2 C(=O)(C(C)CC(C)C(C)=O)N1CC(OC)(CNC(C2CCCC(C)(C)C2)=O)C1 C1(C(N2CC(OCC3(NC(c4cc(C)nn4C)=O)CC3)C2)=O)CCCC(=O)N1C C1(C(=O)NC(CC#C)CO)(NC(=O)C(C2CCCC2)O)CCOCC1.CN C1(CNC(c2ccoc2)C)CCN(C(=O)OC(C)(C)C)C2C1C2(F)F CC1(C#CC(=O)N2CCC(Nc3ncc([N+](=O)[O-])cn3)C(F)(F)CC2)CCCO1 S(=O)(=O)(c1c[nH]c(=NCc2cc(COC)on2)cc1C)N(CCC=C)CC O=c1ccc(S(=O)(=O)NC2CCCC2c2ccccc2)n[nH]1 C(=O)(CC(O)CC(C)(C)C)NC(CNC(Cc1c(SCC)cccc1)=O)(C)CC c1(C(=O)NC2C(C(C)(C)C)NCCC2)ccc2c(Cl)ccnc2c1 Cc1nc2cncc(C(N3CCCN(C(c4cc[n+]([O-])cc4)=O)CC3C)=O)c2[nH]1 c1(OC)cc(C(=O)Nc2c(Cl)ccnc2Br)cnc1-c1cncc(C)c1 CCCCCC(=O)N1CCN(C(=O)CCc2ncc(-c3ccc(F)cc3)o2)CC1 N1(C(c2c(OC)c(C)cs2)=O)CCC2(CCCN2C(=O)Cn2cc(Cl)cn2)C1 N1(C(CC2N(C)C(=O)CC2)=O)C2CCC1CC(NC(=O)CC1C(C)(C)C1(C)C)C2 C1(NC(C(CCSC)(C)C)=O)CCCCCN(C(=O)Cc2cscn2)C1 N1(C(C2CCN(C(C3CN(C(C)=O)C3)=O)C2C)=O)CCCCCCC1C c1(OC)ccc(S(N)(=O)=O)cc1NC(C1CNC(=O)C1(C)C)=O C(=O)(C(O)C(C)(C)C)NCCCN(C)C(c1c[nH]cc1-c1cccc(Br)c1)=O c1(C(=O)NC2CC(CNC(=O)CC(F)F)CC2O)cc(Cl)cc(Cl)c1 CC1CN(C(c2cc(O)nc(O)n2)=O)CC(C)N(C(=O)Cc2cc[nH]c(=N)c2)C1 C1(C(=O)NCC2(SC)CC2)CC(OC)CN1C(c1ccncc1N)=O c1(OC)cc(C(=O)NCCCN(C)C(c2cnc(S)nc2)=O)sc1Cl N1(C(C(CC(C)(C)C)OC)=O)CCCC12CCCN(C(=O)C=C(C)C(C)(C)C)C2 C1(CNC(CC)=O)CN(C(C23COCC(C2)C3)=O)C(C)(C)C1 c12cc(Cl)ccc1NC(=O)C(O)C1CN(C1)C(=O)C2.C1(C(=O)OC)(CO)CC1 C1(CNC(C23CCC(C2)OC3)=O)CC2(CCN(C(=O)COc3ccon3)C2)CO1 c1(NC(c2c(C)nc(NC(c3cccn3C)=O)s2)=O)cccc2c[nH]nc12 C1(NC(C(C)N=[N+]=[N-])=O)CC(NC(C2(CO)CCC2)=O)C12CCC2 C1(C(=O)NCCC(C)(C)NC(c2nsnc2O)=O)CCCCN1N=O c1(CC)nn(C)c(CC(=O)NCC2(NC(C3CC3CF)=O)CCCCC2C)c1Cl C(=O)(C(C1=CCCCC1)N1CCCC(Nc2ccccc2F)C1)CCC1(C)CC1 C12(NC(C(C)c3ccsc3)=O)CCCC1N(C(=O)CC1CCC(C(F)(F)F)O1)CC2 CC1CCC(C)(NC(C2CCOC2CNC(=O)CN(C2CCC2)C)=O)C1 c1(C(N(C2CC(NC(=O)CCSC3CCCC3)C2)C)=O)cc(F)c(Cl)cc1Cl N1(C(C2N(C)C(=O)NC2)=O)C2CCCC1CN(C(=O)Cc1ccnn1C)CC2 Cn1cc(Cl)c(C(=O)NC2(CCC(=O)NCCCC3CCC3)CCC2)n1 c1(OC(C(=O)N(C2CCCN(C(=O)C3CC3)C2)CC)C)ccc(Br)cc1 C1(NC(Cc2c(C)n(C)cn2)=O)CN(C(=O)CN2CCCCC2=O)CC1N=[N+]=[N-] Cc1cc(C(=O)NC2C3CC2N(C(c2ccnc(O)c2)=O)C3C)ncc1F c1(C(C)C)ncc(C(=O)N(CCC(C)NC(=O)CC(=O)NC2CC2)C)s1 Cn1nncc1CC(N1CCC1CNC(c1cn(CCN2CCC2)nn1)=O)=O C1(CNC(C2C(C)C2c2ccccc2)=O)CC2CC2N1C(C1CC1F)=O CC(C)(C)S(=O)(=O)CC(=O)N1CC(CNC(c2cc(C(N)=O)on2)=O)OC(C)(C)C1 c1(C(=O)NC(=O)NC(C)C)cncc2c(F)cc(Br)cc12.C12CCCN1CC2 Cc1sc(C)c(C(=O)NCC2CC(O)CN2C(C2CCCN2C)=O)c1C#N c1(C(N2CC(CNC(c3n(CC)ncc3)=O)N(C)CC2)=O)cccc2scnc12 C=Cc1cnn(C)c1C(=O)NCC1CN(C(=O)C(C)OCC)CC1SC S(=O)(=O)(c1ccc(NC2CCC(O)CC2)c(Br)c1)N(CC)Cc1ccnn1C c1(C(N(CCOCCNC(c2c(NC)cnnc2)=O)C)=O)cccc(SC)c1F C(=O)(C1=CC(O)C(Nc2cc(C)ccc2F)C2CC12)OCC C1(COC)(NC(c2csc(O)n2)=O)CCN(C(C2COC(=O)O2)=O)CC1 O=C1CC(C(N2CCC(OCC(N3CCC(CF)C3)=O)C2)=O)CC(=O)N1 c1(C(C(=O)NC(CC)C)N(C)Cc2ccc(F)cc2)cccc(OC(C)C)c1 c1(NCCC(C(C)C)O)nc(N2CCOC(CO)C2)nc2c1ncn2CCO c1(C(=O)NCC2N(C(C3C(C(C)O)C3)=O)CCC2)cc(N)c(F)c(F)c1F C1(NOCCCCCNC(=O)Nc2ccc(F)cc2)(CO)COCC2CCCN12.O.C Cc1nn(C)c(C(N2CCN(C(c3nnsc3C)=O)C(C3CC3)C2)=O)c1Cl C1(CC(N2C(C)(CNC(C(N3CCN(C)CC3)C)=O)CCC2)=O)CCC2(CCC2)O1 N1(C(C2(C(=O)OC)CC2)=O)CCC2CN(C(c3cnc(Cl)cc3C)=O)CC2C1 n1(CC(=O)NC(C(=O)N(C(C(C)SC)C)C)Cc2cn[nH]c2)cnc(C#N)n1 C1(CC(=O)NCC2N(C(C=CC(C)(C)OC)=O)CC2)CCCC(C2CC2)O1 c1(OC)cc(Cl)c(CC(=O)NCC23CCC(CN(C(=O)CC#N)C2)C3)cc1OC C1(NC(C2CC(=C)C2)=O)CCCC12CN(C(c1cscc1Cl)=O)C2 C1(NC(CN(C(=O)Cc2cnn(C)c2)CC#C)=O)COC2(CCC2)C1 C1(C)(COC)CC(NC(=O)CC2CC3(CC3)C2)CN1C(=O)Cn1cnnc1 C(CCN=c1[nH]nc(O)s1)NC(c1c(C)cno1)=O C(=O)(C(F)C(F)(F)C(F)(F)F)NC(C)CNC(=O)C=Cc1cnc(C(C)(C)C)s1 c12ccc(c(F)c1)c(=O)n2C.n1(CC)nnnc1C(C1CC1)Nc1nscc1Br C1(C(=O)NCC2OCCN(C(c3cc(C)ns3)=O)C2)OCC2CCCCC12 C1(C(=O)NC(CCC)C(=O)N(CC(C)O)C)CC(=O)NC1(C)C N(C(=NCCSC)NCC(c1cccc(Cl)c1)OC)CC1(COC)CC1 C1(C(=O)NC(CC=C)CNC(C2CN(S(=O)(=O)CC)C2)=O)CN(C)C(=O)CCO1 C(=O)(CC(C)P(C)(C)=O)NC1C(C)CN(C(C2(C(C)(C)O)CC2)=O)C1 c1(CC(=O)NCC(C2CC2)NC(C2(CC)CC2)=O)ccc(Br)cc1 C1(C(N2CCN(C(=O)CCC[N+](=O)[O-])C(CCO)C2)=O)CCN2CCOCC12 c1(C(N2CC=CC(NC(C(C)CC3CCCC3)=O)C2)=O)nc(Cl)cc(N)c1Cl C1(CNC(CN(C)C2CC2)=O)COCC1NC(=O)CCC1(C#N)CCC1 c1(CNC(C2CC(NS(CCOC)(=O)=O)C2)=O)cnc2ccoc2c1 c1(C(C(=O)NC23CC(C)(C2)C3)NC(C(CCSC)O)=O)cc(F)cc(Cl)c1 N1(C(c2c(C)n(CC(F)(F)F)nc2)=O)CCN(C2CC2)CC1c1nccn1C C(=O)(CP(=O)(C(C)C)C(C)C)NCCC(C(C)C)NC(C1C(COC)C1)=O C(CC(C)(C)C)(C(=O)NC(C)C(C)(C)OC)NC(c1cnn(C=C)c1N)=O c1(OC)ccc2cc1C2=O.C12CN(CCS1)C2.c1(CC2CC2)cccnc1 c1(CC)csc(CC2CN(C(c3cc(NC(C)=O)cs3)=O)C2)n1.C1C(=O)O1 CC(C)(CNC(=O)CC1CC2(C1)CN(C(=O)C1=COCC1)C2)C1=CCCC1 c1(CC(P(C)(C)=O)C#N)cn(C2CCCc3cncn32)nn1 c1(C(=O)NCC(C)NC(CCc2c(OCC)cccc2)=O)ccc(C)n(C)c1=O C(=O)(C(C)(C)C(C)C)N(CC(=O)N(CCCC=C)C)C C(=O)(C1=CC(C)CC1)N1CCC(N(C(c2ccc(C(C)=O)nn2)=O)CCO)C1 c1(C(=O)NC(CC)CNC(C2(CC)CCOC2)=O)ncnc2c1CCC2 Cc1ccc(F)c(CC(=O)NCCCNC(c2ccc(OCCO)cc2)=O)c1 CC1(C(=O)C(=O)NC)CC1(Cl)Cl.c1(C(=O)NC2C(N)C2)cnn(C2CC2)c1 C1(C(=O)NCCCCCN(C)CC)CN(C(C2CCCC(C)CC2)=O)CCC1(C)C N1(C(C2(CCCC)CCC2)=O)CCOCC(C(=O)N(C(C)COC)CC)C1 C1(C(=O)NCC2CC2(Cl)Cl)CCCCN(C(=O)C=CC2CCCC2)C1 c1(C(N(C2CCC(NC(CCN(c3ncccn3)C)=O)C2)C)=O)cncc(O)c1 C1(C(=O)NC2(CC=C)CCOC2)(COC)CCCN(C(=O)CC2CC(C)C2)C1 CC1CCC(C(=O)NC2C(=O)OCC2(C)C)CN1C(c1cccnc1O)=O N1(C(C(CC)CC)=O)CCN(C)CC1CNC(=O)C(c1ccc(Cl)cc1)CO C1(CCC)CC(C(N2CCC2c2cn(-c3ccc(C)cc3)nn2)=O)CCO1 c1(C(=O)NC2CCN(C(C3(OC)CCCC3)=O)C2)cc2cc(F)ccc2s1 C(CCS(=O)(=O)C(C)C)SC.N12CCCC(C1)C(=O)NCCOCC=CC2=O N1(C(c2cc(NC(C)=O)ncc2)=O)CCN(CCc2ccccc2F)CC1C c1(NC(C2CC3(C2)CN(Cc2ncccc2F)C3)=O)cc(F)c(F)cc1Br C1(C(=O)NCC(CC)NC(c2ccc(C(C)C)cn2)=O)CCS(=O)(=O)N1 c1(OC)ccc(SC)cc1CN(S(=O)(=O)Cc1cc(Cl)ccc1Br)C Cc1ncccc1C(=O)N(CCOCCO)C.C(=O)(C(F)(F)F)N1CCOCC1 N1(C(C2(CC)CCC2)=O)CCCC(C(C)C(=O)NCc2cncc(C)n2)C1 Cc1cc(C(=O)NC2CCN(C(C3COC(=O)N3C)=O)C2(C)C)cc(F)c1 N1(C(CC2(OC)CCC2)=O)CCC(CCNC(=O)Cn2cc(C)cn2)CC1 c1(C(N(C)CC2CCCN(C(C(C)C)=O)C2)=O)c2c(cc3c1CCC3)CCC2 C1(C(=O)NCCCN(C(c2ncsc2Br)=O)CC)CC2CCC1O2 N1(C(CC(C)(C)C)=O)CCC(NC(C2(CCF)CCC2)=O)C(CO)CC1 C=C(C)C1OCCC1C(N1CCCC(N(C(=O)Cc2csc(C)c2)CCO)C1)=O C(=O)(C1=CC(C)(CC)C1)NCCCC1N(C(CC)=O)CCCC1 c1(COC(c2n[nH]cc2C2CC2)=O)[nH]nnc1-c1cccs1 c1(CC#N)ccc(NC(=O)CN2CCCCCC2)cc1.N12CCOCC1C2=O C=CC(C)(O)CC(=O)NCC1CC(C)CCN1C(=O)Cc1sccc1C C1(CC(=O)N(C(C)CCNC(c2cnn[nH]2)=O)C)(CO)CCCCC1 c1(C(C(=O)N(CC(=O)NCC2N(CC)CC2)C)OC)cnn(C)c1 c1(NC(C2(C)CCC(=O)NC2)=O)ccc2nnn(-c3ccccc3)c2c1 Cc1ccccc1C1=NOC(C(N2CC=CC2CNC(C2CCC2)=O)=O)C1 N1(C(c2nc(N(C)C)oc2)=O)CCN(C(c2csnn2)=O)C(c2cn[nH]c2)C1 c1(C(N2CC(CC=C)(C(N3CC(O)C(F)C3)=O)C2)=O)cccc2cncn12 N1(C(CCOCC#C)=O)CCC(C(C(C)C)NC(c2ccc(=N)[nH]n2)=O)CC1 Cc1cc(C(=O)NCCC(C)N(C)C(c2ncn(C(C)(C)C)n2)=O)n(C)n1 Cc1cccc(-c2cn(Cc3coc(-c4ccccn4)n3)nn2)c1 C(=O)(C1=CCCCO1)N1C(CCC(=O)NCC(C)CC2CC2)CCCC1 N1(C(=O)CSc2ccccc2)CCC2(CCCN2c2cc(Cl)ncn2)CC1 c1(C(N2CCCC(CN(C(CN(C)CC)=O)C)C2)=O)cccc(C(C)(C)C)c1N N1(C(c2nnn(COCC)c2N)=O)CC(CNC(=O)C(O)CCSC)CC12CCC2 c1(C(=O)NC2CC(CNC(c3ccnc(N(C)C)n3)=O)C2)nccc(Cl)c1O c1(C(=O)NCC(C)(C2CC2)NC(COC)=O)c(C)nsc1NC(C1CC1)=O C(CNC(=O)C(c1cnn(C)c1)O)(CCCC)NC(COCCC=C)=O c1(CC(=O)NC2CC(C(N3CCC(c4ccccc4)C3)=O)C2)ccc(O)c(O)c1 C1(C(=O)NCCCCCN(C)C(c2cn(C3CC3)nn2)=O)CCCCC1(F)F C(CC)(CCC(=O)N(c1ccccc1)C)NC(COCC(=O)NC)=O C1(NC(C2CCC(=C)CC2)=O)CN(C(=O)C(C(C)C)NC=O)CC(C)(C)C1 N1(C(C(CC#C)O)=O)CCN(C(c2cnn(C)c2Cl)=O)CC1CCOC c1(COC(C)(C)C)ccc2occc2c1.n1(CC(=C)C)nnnc1C(=O)N1C(C)C1 c1(CCS(C(N2CCCC3COCC23)=O)=O)cccc2cccnc12 C1(C(=O)NC(CCC)c2ccco2)CN(C(=O)C(CN(C)C)C(C)C)CCN1C c1(C(N(CCNC(C2(OCC)CCOC2)=O)C2CC2)=O)nc(C)sc1C N1(C(CN(S(C)(=O)=O)C)=O)CCCC(C(C)(C)C(=O)NC2(CO)CCC2)C1 c1(CC(=O)NC2CN(C(C3C(CCC)C3)=O)CC2O)cc(Cl)ccc1OCC N1(C(C2C=CCC2)=O)CC23CCCCC2(C1)CN(C(C1(C(F)F)CCCO1)=O)C3 C(=O)(C(CC1CC1)NC(=O)C(F)OC(F)(F)F)N(CC(C)O)CCF CCC(C)(C(=O)NCCCN(CCO)C(C1CCC(C)C1)=O)C(N)=O c1(C(=O)OC)ccc(C)c(NC(C2CC(C)CN2C(C2CNC(=O)O2)=O)=O)c1 c1(CC(=O)N(CCNC(C2N(CC)CCC2)=O)C2CC2)ccc(OC)cc1Cl N1(C(C(COC)O)=O)CC(NC(=O)C=Cc2ncc(C)[nH]2)CC(F)C1 c1(SCC(=O)NC2(C)CN(C(C3COCCO3)=O)C2)cc(Cl)ccn1 CC1(C)CC(C)(CNC(=O)C2=CCCCO2)CN1C(c1ccc(C(F)(F)F)s1)=O N1(C(c2cccnn2)=O)CCCC2(C1)CN(C(c1cc(Cl)ccc1O)=O)C2 Cc1[nH]c2ncccc2c1C(=O)NCC(O)CNC(c1nnn2c1CSCC2)=O C1(COC)CC(CNC(c2cn(C3CC3)nc2C)=O)N(C(c2oncc2C)=O)C1 N#Cc1nnc2ccccc2c1NCC1CCCN1C(=O)C1=C(Cl)CCOC1 Cc1nc(C(N2CC=C(CNC(=O)CCS(C)=O)CC2)=O)ccc1Br Cc1ccnc(C(C)(C)C(=O)NCC2CCC(NC(c3cn(C)c(O)n3)=O)C2)c1 C=CCCC(C(=O)NCC1CC1C1(C)COC1)NC(c1nocc1C)=O c12coc(n1)C(=O)NC2=O.CC1COCC(=O)N1.C1CO1.C1(SC)CC1 c1(C(N2CCC(CN(C(CSCC)=O)C)C2)=O)ccc(Cl)c(OC)c1F N1(C(c2cc(C)cc(O)c2)=O)CC(C)(C)OCC1CNC(=O)CCC1CCOC1 c1(N(CC(C(=O)NC)C)C)nc2cc[nH]c2c(=NCc2cc(C(N)=O)co2)[nH]1 n1(CCC)nc(C)c(C(=O)NC2CCC(F)(CNC(C3CC(C)C3)=O)C2)c1C Cc1nc2ccc(C(N3CCN(C(=O)C(O)CF)C(c4ncc[nH]4)C3)=O)cc2s1 c1(COC)cc(C(=O)NCC2CC2CNC(=O)CC2CCCO2)ccc1OC c1(C(=O)NC(C)CCCCNC(C2CC3CCC3C2)=O)cnc2c(ccn2C)c1 N1(C(C2(CC)CCCC2)=O)CC2CC1(CNC(=O)C(C)NC(C1CCCC1)=O)C2 N1(C(CC(CNC(CNC(C(CC)C)=O)=O)OC)=O)CCCC(C2CCC2)C1 C1(C(=O)NC2CC(C)CN(C(c3csc(O)n3)=O)C2)CC2COCC(C1)C2 N1(C(Cc2cn(C(C)C)nc2)=O)CCCCC1CN(C(=O)C(C)n1ccnn1)C C1(C(=O)NCCN(CCOC)C)CC=CCN1C(c1ccc(C)[nH]1)=O C(C1CCCC1)=CC(=O)NC(C1CC=CCC1)C(=O)NCC1CC(=C)C1 C(=O)(CCC(=O)N1CCC(CNC(c2cn(C(C)(C)C)nn2)=O)C1)OC CC(C(=O)NCC(C)(Cn1cccn1)NC(c1n[nH]c(=N)s1)=O)S(C)(=O)=O C(=O)(C1CCCc2ccnn21)N1CC(NC(=O)CCOC2COC2)C2(C1)CCC2 C1(NC(c2c(C)snn2)=O)CN(C(c2ccc([N+](=O)[O-])o2)=O)C2(CCOC2)C1 Fc1ccc(Br)cc1CNc1nc(-c2cccc(I)c2)n[nH]1 C(CCCCCF)N(C1(C(=O)O)CCOC1)C C(=O)(C1CCc2cccc(=O)n21)N1CCC(C)(NC(C2CCCCC2)=O)CC1 C1(NC(CCOCCOC)=O)CC(F)(F)CC1NC(c1nc(C)ccc1F)=O c1(OC)ncc([N+](=O)[O-])cc1Br.C12CN(CCO1)C(=O)C2 c1(OC)ncc(C(N2CCCC2(C)CNC(=O)C(C)(C)OC)=O)cc1C(F)(F)F C1(CCn2cc(C(C)(C)OC)nn2)CCN(C(c2cccc(C)n2)=O)CC1(F)F C1(C(C)(C)O)(CNC(C23CCCC2C3)=O)CN(C(C2(Br)CC2(F)F)=O)C1 C12(NC(C3CC(C#C)(O)C3)=O)CCCC1N(C(=O)CC1COCCN1C)CC2 n1(CC(=O)NCC2C(NC(C3CCC(N(C)C)CC3)=O)C2)cccc(N)c1=O C(CC(C)C)(C(=O)NCC(C(C)C)NC(c1cc(Cl)ccc1O)=O)OC C1(C(N(CCN(C(C(C(C)C)O)=O)C)C)=O)C2Cc3ccc(Cl)cc3C12 CC1(C)CCCN(C(=O)CCCOCC2CCCOC2)C1CCn1cncn1 C(C(CC1CC1)C(=O)NCCCC1CCC1)NC(C1N(C(C)(C)C)CC1)=O n1(CC#C)cnnc1C(=O)NCC1(CC(=O)NC2CNC(=O)C2)CC1 N1(C(C(CC)CC)=O)CCC(C(=O)NC2CC(C)(CO)C2)C(O)C1 N1(C(c2ccc(SCC)cc2F)=O)CC2COCC(C1)C2NC(=O)CCOC N1(C(C(C(C)C)NC=O)=O)CCN(C)CC1C(=O)NCCN(CCCO)CCO C(CCCC(=O)NC1CCCC12CC2)N(C(CC1ON=C(C)C1)=O)C(C)C C(Cc1cc[nH]n1)(C=O)NC(CC=CC(C)(C)C)=O.C(C(F)(F)F)(C1CC1)N C(=O)(C1=NOC(C)C1)NCC1(C(=O)NCc2cnc(C)[nH]2)CC1 C1(C(N2CCC(N(C(=O)CNC=O)CC)C2)=O)CCC(F)(F)CC1(C)C C(=O)(C(CC)CCCC)N(CCCCC(=O)NC1=CC=C1C(=C)C)C C1(NC(c2cccc3c2OCC3C)=O)COC2(CCN(C(=O)C=CC(F)(F)F)C2)C1 C1(C(C)(C)NC(CN(C(CC=CC=C)=O)CC2CC2)=O)CCCCC1O N#Cc1ccc(CNC(=O)C(c2ccoc2)NC(=O)CCC2CCC2)s1 Cn1[nH]c(C(=O)NCC2C3CN(C(C4CNC(=O)C4)=O)CC23)nc1=O N1(C(c2cccc(N)c2N)=O)CCCC(C2CC2NC(c2cccnc2F)=O)C1 N(C1CCc2ccccc21)(C(CCC=C)(C)c1nnnn1C1CC1)C1CCC1.CCS C#CCCCCCC(=O)NC(C)CNC(C12CCC(C(F)F)(CC1)C2)=O C12(CNC(CCCCSC)=O)CCCCC1N(C(=O)CCCCCNC(C)=O)CC2 C1(NC(Cn2ncc(C)cc2=O)=O)CCCC12CN(C(c1n[nH]c(C)c1O)=O)C2 C1(C)(NC(C=CC(CC)C)=O)CCCN(C(c2csc(-c3ncccn3)n2)=O)C1 N1(C(CN(CC)CC)=O)CCC(CCN(C)C(c2cnc(C(C)C)[nH]2)=O)CC1 C12(C(=O)NC(CN(C(=O)CC3(COC)CC3)CC)C)CC1COC2(C)C c1(C(N2CC(O)(C(C)NC(CS(CC)=O)=O)C2)=O)ccc(OC)c(N)n1 N1(C(CCCC(C)C)=O)CCS(=O)(=O)C(CCNC(=O)C2=CCC(C)CC2)C1 C1(NC(C(CCC)OC)=O)CC2CCC1N2C(c1ccn(CCN(C)C)n1)=O c1(OCC(C)OC)ccccc1C(N1CCCC(NC(=O)Cc2ccon2)C1)=O C1(C(=O)NCC2C(NC(C3CC=CCS3)=O)CC2)CCCCC1n1cccn1 C(C(=O)NCCCS(C)=O)(C(C)(C)C)NC(CC(C)c1ccco1)=O N1(C(C(C)n2cncn2)=O)CCC(O)(CCNC(=O)Cn2ccc(Br)n2)C1 c1(C(N2CCN(c3nc(C)c(C(=O)O)s3)CC2)=O)c(F)cc(Br)c(N)c1F c1(CC(=O)NCCOC(C)(C)CNC(=O)C(O)C2CCCC2)cccnc1Cl N1(C(C2(C)CC(=C)C2)=O)CC(CC(=O)NCCC2NC(=O)NC2=O)CC1(C)C C(C(C)(C)C#CC(=O)NCC1CN2CCC1C2)NC(CS(CC)(=O)=O)=O N1(C(CCCC(=O)NC(C)C)=O)CCC2(CC1)COC(CC(=O)O)C2 c1(CC)nc(C)c(C(=O)N(C2CCCCC2NC(=O)CN2C(=O)CCC2=O)C)o1 Cc1c(C(=O)NC(C)(CNC(=O)C(C)Sc2ccccc2)CO)cccc1Cl c1(NC(=O)CNC(C(N2CCS(=O)CC2)C2CCSC2)=O)ccc(Cl)cc1 C(=O)(C(C)C(F)(F)F)NCCOC1CCN(C(c2c(C)cc(CC)o2)=O)C1 Fc1cccc2nc(C(c3cccc(Cl)c3)NC3CC3)cn12 C1(CNC(C2(CCOC)CCCC2)=O)C2CCC(C2)N1C(c1cc(CO)on1)=O C1(C#N)(C(N(CCCCNC(=O)CN(C2CCSC2)C)C)=O)CCCOC1 c1(CC)ccc(Cl)c(C(=O)NC(C)CCNC(=O)CNC(c2ccncc2)=O)c1 C1(CN(C(=O)Cc2cnco2)C)CCCN1C(=O)CC1CCNC1 C1(CCNC2(c3n(C(C)F)nnn3)CC(CC(=O)OC)C2)CCC(F)(F)C(=O)N1 C(=O)(C1=CCCC1(C)C)NC1CCCN(C(C(CC)NC(N)=O)=O)CC1 c1(C(=O)NCCC2(CNC(C(C)(C)CO)=O)CC2)cc2ccnn2cn1 N1(C(C(=O)OCC(C(N2CCC(C)C2)=O)C)C)CC(C(F)(F)F)CCC1=O Cc1cc(CNC(c2cnnn2C)=O)oc1C(=O)N(C)CC1CC1(F)F NC1CCc2cc(C(=O)NCCc3ccc(Cl)cc3)ccc2NC1=O CCC(CC(C)C)C(=O)NC1COCC1CNC(=O)CCc1nnc(C2CC2)o1 C1(C2CCN(C(C3CNC(=O)CC3(C)C)=O)C2)(NC(c2c(CC)nco2)=O)CC1 c1(CC)cccc(C)c1NC(=O)C(c1ccc(NC)c(F)c1)N1CC(C)OCC1C Cc1cc(C(N2CCCC2C=CC(N2CCC=C(F)C2)=O)=O)cc(C)c1 C1(C)(C(N2CC3(CC(NC(C=CCOCCOC)=O)C3)C2)=O)CCCCNC1=O C(=O)(CC(C)C(C)(C)C)NCCCCCNC(c1ccn(C(C)C)n1)=O CC1(C)CCC(NC(=O)CNC(=O)CC(F)(F)F)C(Nc2ncccn2)C1 c1(OC(CC)C)cc(NC2CC2NCc2cc(N)cnc2Cl)nc(C)n1 c1(C(N2CC(CNC(C(C)OC3COC3)=O)OCC2)=O)cc([N+](=O)[O-])cn1C C#CC1CN(C(C2COCCO2)=O)CCN1C(c1n[nH]c(CC)c1Br)=O C(=O)(C1=CC2CCC=CCCC12)NCCCN(C(=O)CCF)C1CC1 c1(C(=O)NCC(O)CC(=O)NCC2C(C(C)(F)F)C2)cc(F)ccc1O c1(C(=O)NCC2CCC(NC(c3ccc(Cl)nn3)=O)CC2)ccc2sncc2c1 Cc1ccc2c(c1)CN(C(=O)CC13CCC1CN(C(=O)C(C)N1CCCC1)C3)C2 c1(C(N(C)CC2(NC(c3ccnn3C(C)(C)C)=O)CCC2)=O)cc(O)nn1C c12cc(C)nc(n1)N(C)C2.C(CCCCNC(=O)Cn1cc(C)cn1)SC CC1C(CC2CC(NC(=O)Nc3n[nH]c(-c4ccccn4)n3)C2)CCN1C c1(NC(C)=O)ccc(C)c(C(=O)NC2CN(C(C3(CCN(C)C)CC3)=O)CC2C)c1 N1(C(CSCC)=O)CCCC2(NC(C3COCCC3(F)F)=O)CCCC12 C1(CC)CC(O)CN1C(C1COCC1NC(=O)C1CC1)=O c1(C(=O)NC2CCN(C(c3cnc(C)s3)=O)CC2O)cncc2c1CCCC2 Cc1cc(CNC2CCS(=O)(=O)C2)cc(C)c1C(N1CCCC(C)CC1)=O Cn1ncc(C(=O)NC2C3CC4CN(C(C5CC(O)C5)=O)C2C4C3)c1S(C)(=O)=O N1(C(C2(CCOC)CC2)=O)CC(CN(C(=O)C(=O)OC(C)(C)C)C)CC1(C)C C1(C)(CC)CC(NC(=O)C(C)(C)NC(=O)Cc2cnc(C)s2)C1 C1(NC(c2c(C)cc(CC)o2)=O)CC(C2CCN(C(c3cscn3)=O)C2)C1 C=CC1(C(N2CCCC(N(C(=O)Cc3ncc(Cl)s3)C)CC2)=O)CCOCC1 C12(CNC(CCNS(C)(=O)=O)=O)CCC(CNC(c3sccc3Cl)=O)(CC1)CO2 Cc1cc(=NC2CC(NC(C3(CS(C)(=O)=O)CCC3)=O)C2)[nH]c(SC2CC2)n1 c1(OC(C(CC=C)(F)F)=O)ccc2cc(OC(F)(F)F)[nH]c2c1 c1(OC)cc(Br)cc(CN2CCNCC2C(=O)Nc2nc(C)cs2)c1O N1(C(CCCCCSC)=O)CCCN(C(=O)CCNC(=O)CC(C)C)CCC1 c1(NC(C)=O)ccc(C(N2CCCC(NC(c3ccc(C)nc3)=O)C2)=O)c(Cl)c1 c1(C(=O)NCC(C)NC(CC(CCC)O)=O)ccc([N+](=O)[O-])cc1Br CC1(NCc2csc(Br)n2)CC1(c1nnnn1CCCF)OC N1(C(C(=O)NC(C)C)=O)CC(NC(=O)CSc2ccccc2Cl)C(C)(C)C1 N1(C(C(CC)F)=O)CCN(C(=O)Cc2ccc(F)cc2C)C(c2cn[nH]c2)C1 N1(S(CCCCC)(=O)=O)CCC2(CCC2)CC1C(=O)OC C1(O)(C(=O)NCCC(CCNC(C(CC=C)CC)=O)C)CN2CCC1CC2 Cc1ccc(NC(=O)CCC(=O)N2CC(C(=O)Nc3nccs3)C(C)C2)cc1C N1(C(Cn2ncc(CC)c2)=O)CCn2ncc(CNC(C3(C)CCSCC3)=O)c2C1 C12CCN(CC1)C2=O.Cc1cnc(C(C)(C)NC(=O)C(C)Cc2ccco2)[nH]1 Cc1nc(CCC(N2CCCCC2CCNC(=O)C=Cc2cncs2)=O)[nH]c1C c1(CC(N2CC(C)CC(CNC(C(F)=CCC)=O)C2)=O)coc2ccc(C)cc12 c1(CC(N2CCC(NC(C(CCC)C)=O)CC2)=O)ccc(CC)c(F)c1 C(=O)(C(F)(F)C(O)CC)N1CC(OC(CC)CC)C1.N12CCC(C1)OCC2=O C=CCC(C(=O)NCCCCCc1cnc[nH]1)NC(=O)CCC1CC1(C)C N=c1nc2c(C(=O)NC3CC(O)CN(C(=O)Cc4cncnc4)C3)cccn2[nH]1 c1(CN2CC3N(C(c4cc(CO)ccn4)=O)C3C2)cccc2occc12 C1(C(=O)OC2CC(C)OC2=O)COC2COCC2O1 C1(CCC(=O)NCC2CCC2NC(=O)Cc2cc(C(F)(F)F)co2)CCCOC1 c1(C(=O)OCC)[nH]c2nccnc2c1NC(C1CN(Cc2ccc(C)cn2)C1)=O CC(C)CC(C)C(=O)OC(c1ccc(Br)c(N(C)C)n1)=O CC1C(C(N2CCN(C(c3n[nH]cc3-c3ccncc3)=O)CC2)=O)CCN1C Cc1cn2ccc(C(=O)NCC(C(C)C)NC(=O)C(C)CN3CCCC3)cc2n1 n1(CC(=O)NC(C)CCCCNC(c2cnns2)=O)nnc2ccccc2c1=O c1(C(C)(C)C)ccc(-c2nc(C(N3CCC(Br)C3)=O)cs2)cc1 Cc1nc(CC(N2CCC2CNC(=O)CCN2CCOC2=O)=O)n[nH]1 C1(CC=C)(NC(=O)C(CC(C)C)NC)CCCN(C(=O)CCNS(=O)(=O)CC)C1 CN(NC(=O)NCCc1ccc(Br)c(Br)c1)c1ccccc1 c1(CC)cc(C(=O)NC2CC2CNC(C2(O)CC2)=O)oc1CC CC(C)CC(C)CC(C(=O)NCCc1ccn(C)n1)NC(=O)CC1CC(C(C)C)C1 C#CC1CN(C(c2cnn(C)n2)=O)CCN1C(=O)C(F)C(C)(F)F c1(SCC#C)cccc(C(=O)NC(CNC(=O)C(C)(O)C2CCC2)C(C)(C)C)c1 c1(C(=O)OC)coc(C(=O)NCCCCCN(C(=O)C(C2CC2)SC)C)c1 N1(C(C2CCC(C)(CC)O2)=O)CCC2(CCC2)C(CNC(c2cc(C)c[nH]2)=O)C1 N1(C(CSCc2[nH]c(=N)sc2)=O)CC=CC(NC(=O)CC2CCC(C(F)(F)F)O2)C1 c1(C(N2CCCC(CCN(c3cnn(CC)n3)C)C2)=O)coc2ccc(C)cc12 C1(CCOC)CN(C(=O)C(F)=CC2CC2)CCN1C(=O)CC1CCCCN1C c1(N2C(C(C)C)CN(C(C3CNC(=O)C3)=O)CC2)nccc(S(C)(=O)=O)n1 C(=O)(CCC1=CCCCC1)N(C)CC1(O)CCN(C(CS(=O)(=O)NC)=O)C1 CCC(C)CCCC(=O)NC1CCCC(NC(=O)CC2(CC(=O)OC)CCCC2)C1 c1(CC(=O)NC(CC=C)CNC(C2(n3ccnn3)CC2)=O)ncccc1C n1(CCC)nc(C)cc1C(=O)NCC(C)(C)NC(=O)C(c1cncc(F)c1)C CC1CN(C(=O)C2=CCCCC2)CC(C2CC2)O1.C12CCCCC1NC2=O c1(C(N2CC(CC)(NC(=O)CC3(C)CC3)C2)=O)ccc(Cl)cc1Cl CC#CCC(C(=O)N1CC(N(C)C)C(O)C1)NC(=O)Cc1c[nH]nc1C CCC(F)(F)CC(=O)NCC1CN(C(C2CC(C)OC2C)=O)CC1C CC1C(C)(C)CNC(=O)N1.c1(C(=O)NCc2ccco2)ccc(CO)nc1 C1(C(=O)NC2CC(C(C)NC(=O)Cn3cccc3)C2)CC2(C1)OCCO2 Cc1c(C(=O)NC2(C)CC(NC(C3CCC=CCCC3)=O)C2)cccc1O c1(NC(C2N(C(Cc3scc(C)c3)=O)CCC2(C)C)=O)ccc2ncccc2c1 c1(OCC(N2CC(CNC(C3(C=C)CC3)=O)C(C)C2)=O)cc(Br)ccc1F CC1=C(C)CC(C(=O)NCC(O)CC(=O)NCC2(CO)CCCO2)CC1 C1(OC)(CNC(c2cc(C3CCCCC3)on2)=O)CCN(C(=O)C(C)C)CC1 C1(OC)CC2C1CCN2C(c1c(F)cccc1F)C(=O)NCc1nnn(C)n1 c1(SC)ccc(C(=O)NCC(C2CCC2)NC(c2ccnn2CCF)=O)s1 CCC(C)C(O)C(=O)NCC(CNC(C1(c2cccs2)CC1)=O)OC C1(NC(C(C)n2cccn2)=O)CCCN(C(c2n[nH]c(C(C)C)c2Cl)=O)C1 N1(C(C(C)N(C)C(c2cccnn2)=O)=O)CC(O)(C(F)F)C1 C(CN=c1[nH]c(N2CCN(CCS(C)=O)CC2)nc2c1CSC2)(C(C)C)OC C1(CNC(CC2C(CNC(C3(C(CC)=O)CC3)=O)C2)=O)CC=CCC1 C[Si](C)(C)c1cccc(-c2cn(CC(N3CCC3c3ccc(F)cn3)=O)nn2)c1 C1(NC(c2ccsc2)=O)CN(C(C2CCOC2=O)=O)CCC12CCC2 c1(C(=O)NCC(F)CNC(C2CN(C3CCC3)C2)=O)ccc(C#CC2CC2)cc1 Cc1cc(C)n(C)c(=O)c1C(=O)NCC1CC(NC(C2CCC(C#N)C2)=O)C1 Cc1cc(C(N2CCN(CC3CN(C(=O)C(C#N)C4CC4)C3)CC2)=O)oc1Br C1(C(N2CCC(C(F)F)(CNC(C3(Cl)CC3)=O)C2)=O)CCC(F)(F)CC1 c1(C(=O)NC2CN(C(C3C(CC)C3)=O)CC2CC2CC2)cc(N)ccc1C CN1CCOC(C(=O)NCC(CO)NC(=O)CCc2cncnc2)C1 Cc1cc(C2CC2CNC2CC(NC(=O)Cc3cnccn3)C2)on1 N1(C(C2(C#C)CC2)=O)CCC2CN(C(c3ccc(F)c(C(F)(F)F)c3)=O)C2C1 c1(CNC(C(c2ccco2)NC(C(CC)SC)=O)=O)oc(C)nc1C C(=O)(CC1=CCOCC1)N1CCC(C(=O)NCCOCCC(C)C)C1C C(=O)(C(CNC(C)(C)C)OC(=O)CCc1nc(=N)[nH][nH]1)OC C1(NC(C=Cc2nccc(C)c2)=O)CN(C(=O)CC(F)(F)F)CC12CCOCC2 N1(c2nc(OC)nc(OC)n2)CCC2CC2(NC(c2cncc(F)c2C)=O)CC1 c1(NC(C(CCC)OC)=O)ccc(NC(c2ccn(C(C)(C)C)c2)=O)cc1C N1(C=O)CCN(C(c2cc(SC(F)(F)F)c[nH]2)=O)C2(CC2)C1.CC(F)(F)C1(CO)CC1 C=C1CCCN(C(C(=O)NC2CC(C(=O)OC)C2)C2CC(C)C2)CC1 n1(CC(=O)NC(CCCCNC(COCC#C)=O)C)nc(C(F)F)c2c1CCC2 C(=O)(CC(C(C)C)NC(c1cccc(C)c1C)=O)NCc1n(CC)nnn1 C(=O)(C1CCCc2nncn21)N1C(C)(C)C(NC(=O)CC2CC2)CC1 Cc1cccc(C(=O)NC(C)CC(C)NC(c2c(F)cnn2C(C)C)=O)c1 C(=O)(C(F)C(C)CNC(C1CC2(CC(=O)C2)C1)=O)NC(CCC)CO Cc1cncc(C)c1C(=O)NC1CCC1NC(=O)Cc1cccc(Cl)c1Cl CCS(=O)(=O)c1ccccc1-c1cnc(NC(c2ccc(OC)cc2C)=O)c(O)c1 CC1(C)CCC(CCNC(C2CC=CCC2NC(=O)CCn2cnc(=N)[nH]2)=O)O1 C1(C(N(C)CC2CCN(CC)C2)=O)C(C2CC2)CCN1C(=O)C1=CCCOC1 CCCC(CC)CCC(=O)N1CCC(CCOC)(NC(c2ccc(O)nc2)=O)C1 c12ccccc1CC=CC2.C(=O)(CC(C)(C)C)N1CC(OC)C1 N1(C(CC2CC(=C)C2)=O)CC(F)(F)CC1CNC(=O)C(c1ccc(F)cc1C)(F)F N1(CC)CC2CC1CC2NCc1c(NC(=O)C=C(C)CN)nccc1 Cc1cc(Cl)cc2[nH]c(C(=O)NC3CN(C(=O)C4=CCCSC4)CC3C)cc12 N1(C(c2c(C)nc(C(C)OC)s2)=O)C2CCC1CN(C(c1nc(O)c(C)s1)=O)C2 N1(C(C2(C)CCOCC2)=O)CC(C2CCCCN(C(C3(C)CC3(F)Cl)=O)C2)C1 C1(NC(c2ccc(OC)nn2)=O)CCN(C(=O)CC2NC(=O)CC2(C)C)CC1F c1(C(=O)NCC2(CNC(C3(Cl)C(C)(C)C3)=O)CC2)ncn2c1CCC2 c1(C(C(=O)NCC(C)C)N(C)Cc2csc(CO)n2)cc2c(s1)CCOC2 C1(NC(=O)Cn2cc(-c3cnccc3Br)nn2)CC2CC3C(C2)C13 C1(NC(c2c(CC)nco2)=O)CC2(CCC(CNC(C3(N(C)C)CC3)=O)OC2)C1 CC1(C)CN(C(C2CC3(CC3)CO2)=O)CC1CC(=O)NOCC1CCCO1 C1(OC)CCN(C(=O)CC2(NC(=O)CN3CCOC3=O)CCCCC2)CC1C C(=O)(CC(C(C)C)C(C)C)NC1CCN(C(c2c(CC)nns2)=O)CCC1CO C=CC(C)CC(=O)NCCC(C)N(C)C(c1cccc(C(=O)C2CC2)c1)=O C1(NCC(n2cc(-c3cc[nH]n3)nn2)C)CCN(c2ccn(C)n2)C1 Cn1cnc(N2CC(C(N)=O)(CNC(=O)C=CSCc3ccco3)C2)cc1=O C1(CNC(Cc2c(C)ocn2)=O)CCCC2CN(C(=O)CCCS(C)(=O)=O)CC12 C(=O)(N=c1ccn(C2CC2(F)F)[nH]1)NC1CCCN(CCC(=O)OC)C1 c1(-c2c(C(=O)Nc3cnc(CCC)o3)cccc2)nccn2c(C)nnc12 Cc1cc(F)c2cc(C(=O)NCCC3CCCN3C(=O)Cn3ncnn3)[nH]c2c1 C1(NC(C2CCN(C(=O)COCCN(C)C)C2)=O)CC(CCC)(OC)C1 C(CCCCCC(=O)Nc1ccc2c(c1)COC2)NC(C(C)(C1CC1)OC)=O CCCC(C(=O)N1CCC1CN(C)C)NC(=O)C=Cc1ccco1 N1(C(C(COC(C)C)NC(C(CCC)NC(C)=O)=O)=O)CC2CCC(CO)(C2)C1 c1(C(=O)NC(CNC(C2CC(C)(C)OC2)=O)C2CC2)cccc(=O)n1O N1(CC(N2CC(C(C)NC(C3(C=C)CCC3)=O)C2)=O)Cc2ccccc2C1=O C(=O)(CS(=O)C(F)(F)F)NCC(C)(F)CNC(=O)C1=NOCC1 N1(C(C(C)=C(C)C)=O)CC2(COC(CNC(=O)C(N3CCOCC3)OC)C2)C1 c1(NCC2CC(F)(NC(C3=C(C)CCCC3)=O)C2)ncnc(N(C)C)c1[N+](=O)[O-] c1(CN(c2nnc(C3CCOC3)n2CCC#N)C)nc2c(s1)CCC2 N1(C(CCCn2cc(CSC)nn2)=O)CC(C)C(O)C1 NS(=O)(=O)CCCCCC(=O)NC1(C2CN(C(=O)C=Cc3ccccn3)C2)CC1 c1(C(=O)NCC2CCN2C(c2ccc(CO)o2)=O)cccc2nonc12 FC1(F)CC1C1CCN(c2ncnc(C3CCCC3)c2Br)CC1 C(=O)(C(F)(CN)N=C(NCC(C)(C)C#N)NC1CCCC1)N(C)C C(=O)(C(C)(CC)C(F)F)N(C)CC1CCC(NC(CCCC(=O)OCC)=O)CC1 c1(C(=O)OC)ccc(C(=O)NCC2CN(C(=O)COCC(C)(C)C)CCO2)cn1 N1(C(c2ccc(C(=O)OC)s2)=O)CCC(NC(c2cnn(C)c2C)=O)C1C C(=O)(CCC(=O)NN(C)C)N1C(CCC)CN(C(C2CC(C)(C)CCO2)=O)CC1 N1(C(Cn2cc(C(C)(C)SC)nn2)=O)CCCC(Cn2cc(C(C)O)nn2)C1 CC(CC(C)(C)C)C(=O)NC1CC12CCN(C(c1ccc(Cl)cc1F)=O)C2 C(CCCC#N)(c1n(C(C)(C)C)nnn1)NCCC=CBr CCCCC(C)C(=O)N1CCOC(CCNC(c2sc(C)nc2C(C)(C)C)=O)C1 c1(NC(c2ccsc2)=O)ccc2ccc(=NCCOCC(F)F)[nH]c2c1 N1(C(c2n(C(C)C)ccc2)=O)CC(NC(c2c(Cl)csc2Cl)=O)CC(C)(C)C1 N1(C(C2(SC)CC2)=O)CC2(CCC(NC(=O)C(N)=O)CC2)C1 C#CCC(C)(C(=O)NCP(C)(=O)OCC)NC(=O)CCCCCCC C1(O)(CNC(C2C3CCC23)=O)CCCN(C(c2ccccn2)=O)C1 c1(OC)ncccc1C(C)NC(N1CCCC(C(C)(C)C(F)(F)F)C1)=O N1(C(=O)NC(CC)=O)CC2CC(C1)C2.C(CN(C(C)C)C)NC(=O)OC C=CCC(C(=O)NC1C=CCCC1C(=O)NCC=CCl)NC(C)=O CC1CCC(NC(C2(C)CCCC2)=O)CN1C(=O)Cc1ccc(Cl)c(F)c1 C(=O)(C(C(C)C)C(C)C)NCC(CNC(c1nc(C(=O)OC)sc1)=O)OC Cc1cnccc1C(N1CC2C(CNC(c3c(C(F)(F)F)nn(C)n3)=O)C2C1)=O C1(C(=O)NCCCN(C(=O)CC2CCC3(CC3)CO2)CC)CCC2CC1C2(C)C N1(C(C(C(C)C)SC)=O)CC2(CCCC(CNC(=O)C(C)Cc3ccco3)O2)C1 c1(C(=O)NCC(CNC(CC(CC)C2CC2)=O)O)cc(N(C)C)cc(F)c1 c1(OC)ccc(C(N2CCCC(O)(CNC(=O)Cc3conc3C)C2)=O)cc1O C1(CCOC)(NC(C2CCC(=O)N2C)=O)CCN(C(c2sc(CO)nc2C)=O)C1 C1(C(=O)NC(C(=O)NC)C2CC2)C(C(=O)OC)CN1C(=O)CCCOC(C)=O CCC(CC(=O)N(C)CCN(C)C(c1cnn(CC(F)(F)F)n1)=O)CC(C)C N1(C(C(CO)OC)=O)CC2CC(NC(c3cncn3-c3ccccc3)=O)CC2C1 c1(OCC(=O)N(C2CCC(SCCOC)O2)CC=O)cccc(C)c1C N1(C(C(C2CC2)OC)=O)CCN(C(c2occ3c2CCC3)=O)CC1C Cc1cc(F)ccc1C(N1CC(N(C)C(C2CC2C)=O)C(C)(C)C1)=O C(=O)(CCCCCCCC1CC1)NC(C(C)C)(C)CNC(=O)CN(C)C1CC1 N1(C(CS(CC)=O)=O)CCCC2(NC(=O)COc3cc(C)ccc3F)CC2C1 C(C(COC)C(=O)N1CC(O)(CCNC(C2SC3C=CC2C3)=O)C1)OC C1(NC(c2ccc(C#C)o2)=O)CC2(C1)CC(C(=O)N(C)Cc1ccccc1)C2 C(N=c1cc(C)[nH]c(=NCC2CCCC2O)[nH]1)c1c(OC)cc(OC)c(Cl)c1 c1(C(C)C)nnc(CCC(=O)NC2(C3CCCN3C(=O)C=C3CCC3)CC2)o1 N1(C(c2ccc(CC)c(N)c2)=O)C2CCC1CC(NC(C1CC3C=CC1C3)=O)C2 CC1NC(C(=O)OCC(c2ccccc2)(C)O)=NN(CC(F)(F)F)C1=O c1(C(=O)NCC2CN(C(c3c(CC)n(C)nc3)=O)CC2C)cc(C)c(F)c(C)c1 c1(C(=O)O)cccc(C)c1.c1(C2C(C(C(=O)N3CC(C)C3)NC)C2)ccccc1 N1(C(C2(F)CCCC=C2F)=O)CCCN(CCSc2cccnc2Br)CC1 N1(CCNC(c2c(CC)cno2)=O)CCCN(C(=O)CC2(C)CCCO2)CC1 C1(CNC(C2(NC(c3cn(CCC)nc3)=O)CC(CO)C2)=O)CCCC(O)CC1 c1(C(N2CCC(F)(CNC(=O)CC3CNC(=O)C3)C2)=O)cc(F)cc2nc[nH]c12 Cc1nc(C=CC(=O)NCC(C)(C)CNC(c2ncn(C(C)(C)C)n2)=O)[nH]c1C N1(CCN(C(C2CCCCC2)C(=O)NC(=O)NC2CCCC2)C)CCOCC1.C(C)(C)(C)O C1(C(=O)Nc2cnc(C)c(C(F)(F)F)c2)CCN(CP(C)(C)=O)CC1 N1(C(c2cccc(CN(CC)CC)c2)=O)CCC(C#N)(CSC)CC1 C1(NC(c2nc(Cl)sc2)c2nnnn2CC2CC2)CC2CC3C(C2)C13 Cc1ccc(Cl)cc1C(=O)N(C1CN(C(C2(c3ccc(Cl)cc3)CCC2)=O)C1)C CN1CCC(C)(C(=O)NC2CCCC(NC(=O)Cc3cccs3)C2)C1=O C1(NC(C2C(=C)C2C(=O)OC)=O)CCOCC1NC(C1(C)CC=CCC1)=O Cc1ccc2oc(C(N3CC4(CCCN(C(=O)CN5CC(C)C5)C4)C3)=O)cc2n1 C(=O)(C(F)(F)C(C)O)N(CCC(C(C)C)NC(=O)CN1CCS(=O)CC1)C C1(CNC(C2(COC)N(C(C(CC#C)C)=O)CC=C2)=O)CC2C=CC1CC2 c1(C(=O)NC2C(NC(C(C(=O)OC)C)=O)CC2)c(C)cc(C)nc1OCC1CC1 N1(C(c2ccn(CC)c2C)=O)CC2(CC(NC(C3CC(C)(C)C3)=O)CO2)C1 CCN=C(NCc1ccc(CN2CCCS2(=O)=O)cc1)N1CCC2C(C1)C2(F)F C1(=O)CC(C)C(C)(C)N1C(=O)C(O)Cc1ccccn1.CC(C)C=CC(=O)NCCF Cc1cccc(C)c1NC(=O)C(=O)NC(CNC(=O)CC(C)(C)O)CO Cc1cc2sc(C(=O)NCC(C)CN(C)C(c3c(C)cccc3Cl)=O)cc2s1 N1(C(c2cccc(C(N)=O)c2)=O)CCN(C(c2cncc(O)c2)=O)C2CCC12 N1(C(C(F)=CC)=O)CC(C)(C)CC1CNC(C1(c2cccc(Cl)c2F)CC1)=O C1(CNC(C(C)(C)OC)=O)CCN(C(c2c(C)nnn2C)=O)C12CCC2 C(=O)(C1=NOC(CC2(O)COC2)C1)NC1CCC(NC(C2(C=C)CCC2)=O)C1 Cc1ccc(Br)nc1NC(N1CCC(c2cnc(Cl)s2)C1)=O c1(C(N(C(C)CNC(=O)Cc2ccon2)C)=O)cc2scc(Br)c2[nH]1 N1(C(CCCCSC)=O)CC2CCC(C2)c2ccccc21 C1(C)(CNC(c2c(CC)csc2)=O)CN(C(c2cc(OC)nn2C)=O)C(C)(C)C1 C1(CC)COC(C)(C)CN1C(=O)C(C)(C)CCl C1(COC)(NC(c2cnncc2C)=O)CCN(C(=O)CN(C)C)C1 C(=O)(CCCCC(F)F)N1CC2(CC(NC(c3cn(CCN(C)C)nc3)=O)C2)C1 c1(C(=O)NC(C(=O)OC)Cc2ccccc2)nc(C(F)(F)F)c2sccc2n1 C(=O)(CC(C)CNC(=O)CN(C)C(=O)C1CC1)NC1(CC)CCC1 Cc1ncc2n1CCC(C(=O)NCC1CN(C(c3n[nH]cc3Cl)=O)CC1O)C2 C12(NC(Cc3c(C)ncs3)=O)CCOC(CNC(C3CCCS3)=O)(C1)C2 Cc1ncncc1C(N1CC(CNC(c2cc(Br)sn2)=O)CC1C)=O N1(C(c2c(C(C)(C)C)[nH]cn2)=O)CCCC(NC(=O)CCn2cc(Cl)cn2)C1 C(=O)(C(C(C)C)NC(C1CC(O)(CNC(c2ccn(C(F)F)n2)=O)C1)=O)OC N1(C(C2C(CC)CCC2)=O)CC2=C(C1)CN(C(=O)CC1CCN(OC)CC1)C2 CC(C)(C)CS(=O)(=O)CC(=O)NC(CNC(C1(S(N)(=O)=O)CCC1)=O)C(C)(C)C c1(-c2ccc(CCNC(C3CCCC34CC4)=O)s2)cc(F)c(F)c(F)c1 c1(OC)ccc2ccccc2c1C(C)NCC(C)Oc1cc(C(F)(F)F)on1 N1(CC(C)C)CCCC(NC(C2CC2C(C)NC(C2CC2(Cl)Cl)=O)=O)C1 C1(CCC(=O)NCCc2ccn(CC)n2)CCN(C(C2CC2Cl)=O)CC1 Cc1cc(CCC(=O)NC2(CNC(C3CCSCC3)=O)CC2)n[nH]1 CC1(C)C(CNC(c2nccnc2N)=O)CCN1C(c1ccn(C2CC2)n1)=O C1(NC(=O)NCC2N(C3(CC)CC3)CCC2)CCCCCC1 c1(C(=O)NC(C2CCN(C(CC(C)O)=O)CC2)C)ccn(C(C)(C)C)c(=O)c1 c1(C(N2C(CNC(C3CC4CC4C3)=O)CC(O)C2)=O)ccnc2cc(F)cnc12 c1(C(c2ccc(Cl)c(Cl)c2)NC(C(=O)Nc2n(C)cnc2)=O)cc(Cl)cc(Cl)c1 c1(C(N2CC(O)(CNC(CC3(CC)CCC3)=O)C2)=O)c(O)ccc(F)c1C c1(C(N2CCC(C(C)NC(CCC=C)=O)C2)=O)nc(-c2ccc(F)cc2)oc1C C1(F)(C(=O)NC2CC(CCNC(C=CCCC=C(C)C)=O)C2)CC2(CCC2)C1 C1(C(N(CCC)CCC)=O)CN(C(=O)CC2CC3(CC3)C2)CC1C1CC1 N(C(=NCCCCl)NCC(C)(C)C(N)=O)C1CCC(C(=O)OC)CC1 Cc1nc2c(C(=O)Nc3cc4n(n3)CCC4)cccc2o1 C(=O)(C(C)CCC(C)(C)C)N1CC2(N(C(C3(COC)CC3)=O)CCC2)C1 c1(C(N2C(CN(C)C(c3coc(Cl)c3)=O)CCC2)=O)nn(C)cc1Cl N1(C(CNS(C)(=O)=O)=O)CCC(NC(=O)CC2CC(=O)NC(=O)C2)CC1C1CC1 C1(CC(=O)NC(C2CCOCC2)C#C)CC(NC(=O)C=CCCC)C1(C)C N1(C(c2c(CC)scc2)=O)CC2CCC1C2NC(=O)C(C)N1CCC1 C(C(CC(C)C)C(=O)NCC1(C(=O)NC(CCO)C2CCC2)CC=CC1)OC c1(C(N2CC3C(NC(C4C5COCC45)=O)C3C2)=O)cccc(S(=O)(=O)C(F)F)c1 c1(C(=O)NCC2C(NC(C3(C(=O)OCC)CCOCC3)=O)C2)ccc(=O)n(C)n1 C1(O)(CNC(C=Cc2ccc(C(N(C)C)=O)cc2)=O)CCC(F)(F)CC1 C1(C2(C)CC2)CCN(C(=O)NCC(O)CN2CCOCC2)C1 N1(C(c2cnc(CCC)s2)=O)CCN(C(C2C=C2C)=O)C2(CCC2)C1 N1(C(C(c2cnn(C)c2)C)=O)CCCC(O)(CCNC(=O)COC(F)F)C1 c1(COc2c(C(N)=O)cccc2)cc2cc(Br)ccc2s1.C12CN(CCO1)C2=O N1(C(C(CC#C)O)=O)CC(CC(=O)N(C2CCN(C)C2)C)CC1(C)C c1(-c2cc(C(=O)NCC(C)NC(=O)C(O)C3CCCC3)no2)ccccc1Br N1(C(C(C(C)(C)C)N2CCCCC2=O)=O)CC2CCN(C(=O)CC3C=CCC3)C2C1 C1(CC)CN(C(=O)C(=Cc2c[nH]cn2)F)CCN1C(=O)C1=CCN(C)C1 c1(CC)cc(C(N2CCN(C(c3cnc[nH]c3=N)=O)CC2)=O)cc(F)c1 C#CCC(C)(CC)C(=O)N1CC(O)(C(C)NC(=O)Cc2cccc(C)c2)C1 N1(CC)CCN(CC(=O)NC2CC(C)N(C(c3ccoc3Cl)=O)C2)CC1 N1(C(c2c(CC)nco2)=O)CCC2CN(C(c3cscc3CC)=O)CCC2C1 C1(NC(C(CC)CN(C)C)=O)CCCN(C(=O)C(C)C(F)F)C1C CC(C)C(CCN(C(=O)C(C1CCCCC1)N(C)C)C)NC(=O)CC(C)(C)C C1(NC(CSc2c(C)cccc2)=O)CN(C(=O)CC2CCCC2(C)C)C(C)(C)C1 N1(C(C(CC)COC)=O)CCN(C(=O)C2=NOCC2)C(C(C)(C)C)C1 N1(CCC)CCC(CNC(=O)NCC(c2cnn(C)c2)O)C1 N(C1COc2ccccc21)C(C1(C)CCCN(C(c2ncc(F)cc2F)=O)C1)=O N1(C(COc2c(C)cccc2C)=O)CC(NC(=O)CC(C)N(C)C)C2(CCC2)C1 N1(C(CC)=O)CCc2cc(C(N3CCC3C(=O)NC)=O)ccc21.C1(=O)CC(C)N1 C(=O)(C1CCCc2ncccc21)NCC(C)CNC(C1C(F)(F)C12CCC2)=O Cc1[nH]nc2c1CCC(C(=O)NCC(CNC(=O)CSCCN(C)C)CO)C2 N1(C(C2(C)CCCO2)=O)CCC2(CCN(C(=O)CCCC3CCCC(=O)N3)C2)C1 C1(N(C(C2CC(Cl)(Cl)C2)=O)CC)CCN(C(=O)Cc2ccno2)CC1 CCC(F)(F)CC(=O)N1CCC(C(=O)NCc2ccc(C#N)cc2)C(O)C1 n1(CCC(N2CCC(C)(NC(C3CC3C(F)F)=O)C2)=O)cc([N+](=O)[O-])cn1 C1(CN(C)C(C2CCC(=O)O2)=O)CCCN1C(C1CCCN1C)=O c1(C(=O)NCC(CC(C)C)NC(C(OCC)OCC)=O)ccc(SCC)c(F)c1 c1(N(C)Cc2csc(-c3ccoc3)n2)nc(N(CC(F)F)C)c2c(n1)COC2 N1(C(C(c2ccc(C)s2)C)=O)CC2CC2(NC(c2cnn(CCO)c2)=O)C1 c1(C(N(CC(C)O)CCNC(=O)CC2CCCOC2)=O)nccc2ncccc12 C(=O)(CC(C(F)(F)F)OC)NCC1CC(NC(C(C=C)OC)=O)CC1O c1(C(=O)NC2CN(C(c3c(CC)c(C)sc3)=O)CC23CC3)ccc(N)c(Cl)c1O C1(CC(=O)NC(C2CCCCC2)C)CCCN1C(c1cc(C(F)(F)F)c[nH]1)=O N1(CCOCCOC)CCC2(CC1)CC2NC(N1CC(O)CCC1C)=O C12(C(=O)NCCN(C(C=CC(C)(C)SC)=O)CC3CC3)CCC(C#N)(CC1)CC2 CC(C)CCCC(C)C(=O)NCC1(CC(=O)N(C)CC2CC2C)CC1 c1(C(N(CCNC(=O)C(F)C(C)C)CC)=O)sc2cncn2c1C C1(N(C(=O)C(C)SC)CCC)CCN(C(=O)CNC(C)C)C1 C1(=C(C(=O)N(C2CCN(C(=O)CC34CCCC3C4)C2)CC)F)CCCCC1 C1(C(=O)NC(COCCCC)C)CC(CCOC)CCN1C(=O)C(CC)SC O=S(CCc1nc(-c2c(F)ccc(F)c2Cl)no1)CC(F)(F)F c1(C2CCCC2)nc(C2(Cc3cncs3)CNC2)cs1 CC1(C)CCCOC1CC(=O)NC1(C(=O)NC2CCC(C3CC3)C2)CCSC1 c1(OC(C2(CC)CCCO2)=O)cc(C#N)ccc1C(C)NC(=O)OC(C)(C)C c1(C(=O)NC2C3CN(S(CC(=O)OC(C)C)(=O)=O)CC32)cc2c(F)cccc2[nH]1 C1(C(N2CCC(CC(=O)N(C)CC3CCOC3)CC2)=O)CCC(C2CC2)C1 C12(CCNC(C3CCCN(C)C3)=O)CCC(C1)N(C(C1CCC(C)CC1)=O)C2 Cc1coc(C(=O)NCC2CCCN2C(=O)CCc2cccc(N(C)C)c2)c1C N1(C(C2C(CC)CCO2)=O)CCCC(C(=O)Nc2cccc(CO)c2)C1 C(=O)(C(O)C(C)OC)NC1CC(NC(C23CC(C(=O)OCC)(C2)C3)=O)C1 Cc1cnc(NC2CCC(NC(=O)CC3CCCC3(F)F)CC2)nc1C c1(C(N2CC(O)(C(C(=O)NC(CCC)CC)F)C2)=O)cncc2[nH]ccc12 C(=O)(CC1CC(=O)c2ccccc21)N(C)CC1CCCN(C(C=CCC)=O)C1 c1(N2C(CNC(C3CCC3)=O)CCC2)ncnc2cccc(F)c12 c1(C(=O)NC(C2CCCN(C(=O)CNC(=O)C(C)(C)C)C2)C)cccc(Cl)c1Cl n1(CC)ccnc1C(=O)NC1CCC(N(C)C(C2CS(=O)(=O)C2)=O)C1 N1(C(CC2CCCN(C(Cn3ccc(C)n3)=O)C2)=O)CCOC(C)(C)C1C N1(C(c2ccc(C)n2C)=O)CC(O)C(O)C1CNC(=O)CCC1CC1 C1(CNC(CN(C2CCSC2)C)=O)CCC(C)(C)CN1C(c1cnn(C)c1N)=O C(=O)(CCCCN(C)C)NCC(=C)C(=O)N1CC(OCC(C)C)C1 CCCCN=C(NC1CC1c1c(Cl)cccc1Cl)N1CCC2(CCCC2)C1 CC(F)(F)CCCCN1CCS(=O)(=O)CC1 N1(C(c2c(C)coc2)=O)CC(NC(C2CC23CC3)=O)C(n2ccnn2)C1 c1(CN(CCC(=O)N(CC(CC)NC(C2CCC(OC)C2)=O)C)C)ccccc1 Nc1nc(Br)ccc1C(=O)NCC1CCN(C(=O)CN2CCCCC2)CC1O Cn1ccnc1C(=O)NCc1n[nH]cc1C(=O)NCc1nncs1 N1(C(C2(C#C)CN(C(C3(C(=O)OCC)CCC3)=O)C2)=O)CC2CCC2(CO)C1 N1(C(C2(CC=C)CCC2)=O)CC(CNC(c2cc(CC)no2)=O)C(C)C1 c1(C(N(C)CCOc2cccc(F)c2)=O)cc(Cl)c(F)nn1 c1(N(C=O)CC2CC3CC2C3)cccc2c1OCCO2 N1(C(C=CC)=O)CC2(CCCCN(C(C3CCOC(C)(C)C3)=O)C2)C1 N1(C(=O)CC2CC3(C2)CN(Cc2cccc(F)c2F)C3)CCC2COCC2C1 N1(C(C2N(C(CNC(CCC)=O)=O)CC(C)C2)=O)CCC(O)C(O)C1 N1(C(C2N(C(C)=O)CCCC2)=O)CCCC2(NC(C3CCCC(C)O3)=O)CC2C1 c1(N2CCN(Cc3ccc(C)cc3O)C3C2C3)ncc2[nH]ccc2n1 CCC(CC)(C(=O)NC1CN(C(=O)CC(C)(C)C)CC1c1ccccc1F)OC C(=O)(C1CC(=O)Nc2ccccc21)NCC(C)NC(c1ccc(C(C)O)cc1)=O CN1CC(C(=O)NCCOCCNC(c2cnc(O)n2C)=O)C(C(F)(F)F)C1 S(=O)(=O)(c1cc2sc(C)cc2s1)N1C(C(=O)OC)CC(c2ccccc2)C1 c1(C(=O)NC2C(C)N(C(C3CCC3(F)F)=O)CC2)cc2c(s1)CCOC2 c1(-c2cc(C(N3CCC(C(=O)OC)C3)=O)no2)cncc(F)c1 C1(NC(C(CCC)NC(N)=O)=O)CCN(C(=O)CCN2CCCCC2=O)C1(C)C Cc1nc2cccc(C(=O)NC(C)CC(C)NC(C3(C)CCCO3)=O)n2n1 C1(NC(COCC(C)C)=O)CCC(C)N(C(=O)C(C)c2ccco2)C1 n1(CC)cc(CCNC(=O)C(c2cccs2)NC(C2CCC(=O)O2)=O)cn1 Cc1cc(CCNC(=O)CC=CCNC(=O)C(C)CN2CCCC2)nn1C c1(C(N2CC3CC(NC(C(COC)(C)O)=O)C3C2)=O)ccc(C)c2cccnc12 N1(C(C(CCC)(C)O)=O)CCCC2(NC(C3CCc4ccccc4C3)=O)CC2C1 c1(OC)ccnc(C(=O)NCC2CCN2C(C2CCC3CC3CC2)=O)c1OC Cc1cc(C=CC(=O)NCC2CCN(C(=O)C#CC(=O)N(C)C)CC2)c[nH]c1=N CCCC(C)(CC)C(=O)NC1COCCN(C(C2CCCC2O)=O)C1 c1(NS(CC)(=O)=O)cc(N2CCCC2CF)nc(C)n1 CC1(C)C2CCC1(CC(N1CC3C(c4cn(CC(N)=O)nn4)C3C1)=O)C(=O)C2 c1(C(=O)NC(CCN(C(C2(CCOC)CCC2)=O)C)C)csc(C(F)F)n1 N1(C(C2(C)C(C)OCC2)=O)CCc2nnc(-c3cccc(C(F)(F)F)c3)cc2C1 C12CNCCOC1C(=O)N2C(C)C1CC1.CCCCNC1CC1 N1(C(c2ccc(CC)cn2)=O)CC(C)CCC1CNC(=O)CC1CC1CC C(=O)(C(C)(C)C(=O)N(CCC(C(C)C)NC(=O)C=CC(C)C)C)NC Cc1ncc(C(N2CC3C(NC(=O)C(C)SC(F)(F)F)C3C2)=O)cn1 Cn1ncc2cc(C(N3CCC(CO)(NC(=O)CNS(=O)(=O)C4CC4)C3)=O)sc12 c1(C(=O)NC2CC(C(=O)NCCC3CC(C)C3)CC2O)cnn(C)c1C#N C1(C(=O)NC(C2(O)CCN(C(C=C(COC)C)=O)C2)C)CCCC12CCOCC2 C1(NC(C2(C)CC(=C)C2)=O)C2CC(NC(c3noc(C)c3C(C)=O)=O)CC12 C1(C(=O)NCC(C)(C)CNC(=O)CC2CCCOCC2)CC2CCC1CC2 c1(C(C(=O)NCC(C2CC2)NC(C=Cc2nc(C)sc2)=O)=O)ccc(F)c(F)c1 C(=O)(C(CC(C)C)C(C)C)NC1(C2CCN(C(c3nc(C)oc3C)=O)C2)CC1 N1(C(C(CC)O)=O)CC2CCC1C(CNC(c1cnc(N)cn1)=O)C2 C1(NC(C2C3CCCCC23)=O)CCCN(C(C2CC23CCCCC3)=O)CC1 N1(C(=O)NC(C2CCC(C(C)C)CC2)=O)CC2CCCC(N(C)C)(C1)C2(F)F c1(OC)cc(S(C)(=O)=O)ccc1NC(C1CSCCN1C(c1cscc1C)=O)=O N1(C(COC)=O)CCC(NC(c2cnn(C3CC3)c2)=O)C1C(C)C N1(C(=O)COCc2ccccc2Br)CCC2(CCCN2C(=O)C2=NOCC2)C1 C(C(CO)(CO)NC(c1ncoc1C1CC1)=O)N(C(c1cn(CC)nc1)=O)C Cc1nc(C(N2CCSCC2CCNC(C2OCCC2(C)C)=O)=O)nn1C c1(C(N2C(CNC(CCCOCCC)=O)CC2)=O)c[nH]c2cc(C)ccc12 N1(CCC)CCC(NC(C2CC(CF)C2)=O)C1.C1(=O)C=C(C)CN1 C1(CN(C(CNC(CCC)=O)=O)C)CN(C(C2CCC3CC23)=O)CCO1 CC1CC2CN(C(=O)NCCO)CC2N1CCOC1CC1(F)F c1(C(C)C)ccccc1OCC(N1CCC(O)(CCNC2CCCN2C)C1)=O N1(C(C(C)OCC2CC2)=O)CC(NC(=O)COc2cccc(F)c2F)CC(O)C1 N1(C(c2c(C)c(C#N)[nH]c2)=O)CC2(CCCC2)C1C(=O)NCc1cnns1 CC1CCCN1CC(=O)NC1(C2CCCN2C(=O)CNC(=O)NC2CC2)CC1 CN1CCC(C(=O)NCC(F)(F)Cl)(NC(=O)Cc2ccccc2F)C1 n12c(csc1=Nc1ccc(S(C)(=O)=O)cc1)c1ccn(c3cnc2s3)n1.CO N1(C(C(C)(C)C)=O)CCN(C(CNC(=O)C=Cc2cc[nH]n2)C(F)F)CC1 c1(C(=O)NC(CC)(C)CNC(=O)C(C)(C)C#N)cc2cc(OC)ccc2n1C N1(C(C)=O)CCCC1c1nc(NC(=O)NCCc2cc(C)[nH]n2)no1 N1(C(CC2CC(CC)C2)=O)CCCCC(CC(=O)NCC(N2CC=CC2)=O)C1 CC1(C#CC(=O)NC2C3CCC(C3)C2C(=O)NCc2ncccn2)COC1 C1(CNC(C(C)(C)SCC)=O)CCC2CN(C(=O)Cc3cc(C)cs3)CC12 CCC(C)(C(=O)NCC1CN(C(=O)Cc2ccn(C(F)F)n2)CCN1C)C(N)=O c1(C(=O)NC2CC(N(C)C(C3CCCCNC3=O)=O)C2)nccc2c1CNC2=O C1(NC(CSC)=O)CN(C(c2cccnc2-n2nccn2)=O)CC1N=[N+]=[N-] N1(C(c2cc(OC)ncc2)=O)CCN(C(=O)CNC(C)=O)C(C)C1C c1(C(N2C(C)CN(C(C3COCCO3)=O)CC2)=O)cccc2nn[nH]c12 C1(CNC(C(C)Sc2nnnn2C2CC2)=O)CC2CCC1N(C(=O)C(C)(C)F)C2 c1(C(N2CCC(CC=C)(NC(=O)C(C)O)C2)=O)nc(Br)c2c(F)cccn12 C1(NC(C2(CCNC(CN3C(C)CCC3C)=O)CC2)=O)CCCCC12CC2 C1(NC(C(C)SC)=O)CN(C(=O)Cc2cnc(C(F)(F)F)s2)CC1F.C1C(=O)N1 N1(C(C(n2c(C)ncc2)C)=O)CC(C2(NC(C3CC3C#N)=O)CC2)C1 O=C(CCCCc1ccc(Cl)s1)NC(c1ccccc1CC(F)(F)F)C(=O)O C1(F)(CNC(C2CCC(=O)N2)=O)CCCN(C(=O)Cc2ccncc2Cl)C1 N1(C(C2(N)C(C)(C)C2)=O)CCC(C)(O)C(O)C1 Cc1ccc(C2(C(=O)NCC(CO)NC(=O)COCC(C)(C)C)CC2)cc1 N1(C(c2c(CC)c[nH]n2)=O)CCN(C(=O)CCCC2CCCC(=O)N2)C(CC)C1 C12(C(N(CC(C)C)CC)=O)CC(n3cc(-c4nccs4)nn3)C1C2 Cc1cn2ccc(C(N3CC(NC(C4SC5C=CC4CC5)=O)CC3C)=O)cc2n1 c1(CC)onc(C(=O)NCCN(C2CCCC2)C(c2cc(CO)ccn2)=O)c1C c1(C(=O)NCc2c(C(=O)NC(C)CC3CCC3)nco2)cccnc1O c1(C(N2CC3(CN(C(c4c(=O)ccn(C)c4)=O)C3)C2)=O)ccc2c(n1)CCC2=O c1(C(N(C2CN(C(C=Cc3scc(C)n3)=O)CC2F)C)=O)cc(Cl)cc(C)c1C C1(CC(=O)OCC)CCC(C(N2CCC(N(C(=O)CCOC(C)C)C)C2)=O)CC1 c1(OC)c(C(N2CC3CN(C(C4CCCC(=O)C4)=O)CC3C2)=O)cc(F)cc1F c1(C(=O)NC(CNC(CCCOCC=C)=O)CCOC)ccc(C)c([N+](=O)[O-])c1 c1(SCC)cccc(CC(=O)NC23CC(C2)N(C(c2ccnn2CCF)=O)C3)c1 Cc1cccc(COCC(=O)NC(C)C(C)NC(c2nc(Cl)c(Cl)s2)=O)c1 C1(C(=O)NC(C=C)C2CCC2)CC1C1CN(C(=O)CN=[N+]=[N-])C1 C(=O)(C1=NOC2COCC12)N1CC(O)(CN(C(=O)C#CC2(C)CC2)C)C1 c1(C2(CCN(C)C)CC2)ccncc1.C(=O)(CCN(CCO)C=O)O Cn1nc2c(c1C(=O)NCc1ccc(Br)c(F)n1)CCCC2 CC1CN(C(c2cnccc2C(N)=O)=O)CCC1CNC(=O)CN1CCC1 c1(C(C(=O)NCC=CCN(C(C(C=C)c2ccccc2)=O)C)=O)ccc(Cl)cc1 Cc1nn(CC(=O)NC2CCC2NC(=O)CC(O)C(Cl)(Cl)Cl)cc1[N+](=O)[O-] Cc1ccc2c[nH]nc2c1NC(C1CCCN(Cc2cc(Br)c[nH]2)C1)=O C1(O)(CCNC(CC(CC)SC)=O)CCCN(C(c2ccc(N)cc2OC)=O)C1 C1(N(C)C(c2ccnn2CCF)=O)CCC(NC(=O)CN2C(=O)CNC2=O)CC1 C(=O)(C(CC(F)F)Nc1nccnc1N)NCC(C(C)C)C CCC(C#N)C(=O)N1CCCC1C1(NC(c2ncccc2F)=O)CC1 c1(C(N(CCC)CCNC(=O)CC(C)(C)C)=O)cncc2c1CCNC2=O S(=O)(=O)(c1cccnc1NCC1CCCN1C(C)C)NC(CCCCC)CO Cc1cc(C(=O)NCC2CCN2CC=C(Cl)Cl)sc1C C1(C(=O)NC(C=C)C2CC2)CC=CCN1C(=O)CCCC#N C(C(C(=O)N1CC(F)(COC)C1)NC(c1cc(OC)no1)=O)OC N1(C(COC(C)=O)=O)CC23CCCCC2(C1)CN(C(=O)C(C)(C)C1CCCCO1)C3 c1(C(=O)NC2CN(C(C34C(C(N)=O)(CCC3)C4)=O)C2)ncnc2ccccc12 CC(C)CC(C)C(=O)NC1CN(C(=O)Cn2cnnc2O)CCC1C(F)(F)F N1(C(C(CC(C)C)C)=O)CC(C)CN(C(c2coc(S(C)(=O)=O)c2)=O)C(C)C1 CCC(CCC(=O)NCCC[Si](C)(C)C)NC(C1C2CCC(F)C12)=O Cc1nn(C2CC2)cc1NC(C1CC(C)N(C(=O)CN(C)C(C2CCC2)=O)C1)=O c1(C(=O)NC2(CC(=O)NCc3ccc(Cl)o3)CC2)cnc(CO)cn1 CC(N=c1[nH]c(Cl)ncc1[N+](=O)[O-])C1CCCN1C(C1CCN2CCCC2C1)=O c1(OC)ccc(F)cc1CC(=O)N(CC(O)CNC(C1CCCN1C(C)=O)=O)C c1(C(=O)NC2C(C)(C)CN(CC3CCCS(=O)(=O)C3)C2)ccc2occc2c1 c1(C(=O)NC2CN(C(c3ncsc3C(F)(F)F)=O)C2)ncc2n1CCCC2 c1(-c2ccc(NC(C(C=C=C)C)=O)cc2)ccnc2ccccc12 c1(C(=O)NCC2C3CN(C(c4ccccc4)C#N)CC32)cc2cc(Cl)ccc2s1 c1(OC)cc2c(C(=O)NCCNC(C3CC3C(=O)NC)=O)c[nH]c2cc1Cl Cn1cc(C=CC(=O)NCC(C)(C)C(=O)NCCn2ccnn2)cn1 c1(C(N2C(CNC(C3(C)CC(=CC)C3)=O)CC2)=O)cc(F)cc([N+](=O)[O-])c1Br Cc1sc(C)c2sc(C(=O)NC(C)CC(C)NC(C3CCCN3C3CC3)=O)cc12 C(=O)(C#CC1CCCO1)N1CCC(C)(NC(=O)CNC(c2ccccc2)=O)CC1 C1(CC)CN(C(c2ncoc2-c2ccon2)=O)CCC1NC(C1COC(C)C1)=O c1(OC)ccccc1C(=O)NCCC1(O)CCN(C(=O)CC2(C)CCOC2)C1 CC1(C)Oc2cc(C(=O)Nc3cccc(C(F)(F)F)c3C#N)cnc2NC1=O C(CC(C(=O)NCC(C)SC)NC(c1nn(C)cc1Cl)=O)=CC c1(C(N2CCC(C(C)NC(=O)C(F)=CCCF)CC2)=O)ccc(C#N)cc1F N1(C(CC2(OCC)CC2)=O)CC(O)C(O)C1CNC(=O)CC1CC1 C(=O)(C(CC1CCCCC1)C(C)C)N1CC(CNC(Cc2c(C)n[nH]c2)=O)OCC1 C(N=c1[nH]c(=N)[nH]c(=NCc2nccn2C2CC2)[nH]1)c1c(C)c(F)ccc1N C(=O)(C(CC)C(C)C)N1CCC(NC(COc2cc(CC)ncc2)=O)C1C C(=O)(CCS(=O)(=O)CC(C)C)N1CC2(CN(C(C(CC)(C)CC)=O)C2)OCC1 Cc1c(C(N2CCN(CCN(C)C(C3CCO3)=O)CC2)=O)cnn1CCC(C)C c1(OC)ccc(CNC(C2(C)CCCN2Cc2ccc(F)cc2O)=O)c(C)c1C C(=O)(C1CCCc2nccn21)N(CCCCN(C)C(C1(n2nccn2)CC1)=O)C C1(NC(C2CC3(CC(OC)C3)C2)=O)CC2(C1)CC21CCC1.C12(CC1)C(=O)N2 Cc1nnc2c(C(N3CC=C(CNC(c4nscc4N)=O)CC3)=O)cccn12 c1(C(N2C(C(C)O)CCC2)=O)ccc(-c2cccs2)o1.n12cc(nn1)CCCS2 c1(CN2CC(C)(CC(=O)NCc3cc(C)no3)C2)cccc2cc[nH]c12 c1(OC)cc(C(N2CCC(CNC(c3cccc(C)c3)=O)C23CC3)=O)ccc1F c1(C(N2CCC(C)(NC(C(C)SCCCCCC)=O)C2)=O)ccc(C)cc1CC Cc1cc(C(=O)NC(C)CC(C)NC(c2nnn3c2CSCC3)=O)cc(=O)n1C c1(OC)cc(C(=O)NC2CC(C)CN(C(c3ccc(O)c(Br)c3)=O)C2)ccc1Br c1(C(=O)OC)ccc(C(=O)NC(C2CN(C(=O)CC3(C)CC3(Cl)Cl)C2)C)nc1 C1(CNC(c2cc(OCC)no2)=O)CN(C(=O)Cn2cnc(=N)[nH]2)C2(CCC2)C1 C(=O)(CCCC(=O)N1CCOCC(CNC(=O)CC2CCCN2C(C)=O)C1)NC C1(CNC(Cn2c(C)ccn2)=O)CC2(CC2)CN1C(c1ccc(C2CC2)cc1)=O c1(C(=O)NC2CN(C(C3OCCN(CC)C3)=O)C2)cccc2sccc12 c1(C(=O)OC)ccc(CC(N2CC(NC(C3CC3c3cncn3C)=O)C2)=O)cc1 c1(C(=O)NC2CCN(C(CCCOCC=C)=O)CC2)ccc2ccsc2c1 c1(C(N2CC(CNC(C3C(CC)CCC3)=O)C2)=O)cccc(Br)c1 Cn1nc(C(N2CC3CC2CC3NC(c2ccoc2Cl)=O)=O)ccc1=O c1(OCC(N2CCN(S(=O)(=O)Cc3ccccc3)CC2)=O)ncccc1F CCCCCC(C)(C)C(=O)NC1CCOC(C(=O)N(CC(C)C#N)CC)C1 c1(CN2CCCC(C)(C(=O)NCc3cccc(I)c3)C2)ccc2nonc2c1 c1(C(=O)OC)oc2ccccc2c1CNC(c1cc(Cl)ccc1F)(C)C(=O)O C1(CC)CCCN1C(=O)CC(C)N(C(=O)C(N1CCOC1=O)C)C c1(C2C3(CCN)CC3CC2)ccc2cc(CNC(=O)OC)ncc2c1.C(C)(C)(C)O c1(C(=O)NC2CC(NC(C3CCCN(CC)C3)=O)C(O)C2)cc2ccncc2s1 CC1(C)C(C(N2CCCC(C#N)C2)=O)CCN1C(=O)C(=O)NC1CC1 C(CCC(=O)NCC1(F)CN(C(c2csc(C(N)=O)n2)=O)C1)N(C(C)C)C c1(C(N2CC(C(N)=O)(CNC(=O)C(c3cncn3C)O)C2)=O)cccn(O)c1=O N1(C(C(C)OCOC)=O)CCC(C(C)(C)CNC(=O)Cn2cc(CO)nn2)CC1 c1(NC2CCCN(CC=C)C2)[nH]c(=NCc2ccsc2)nc2sccc12 C1(C(N(CC(C)(C)NC(=O)CCn2cnnn2)C)=O)CCC2(CC2)C1 N1(C(c2cnc(C)n2C)=O)CCN(C(C2COC(=O)N2C)=O)C(C)C1 Cc1ccc(C(=O)NCCNC(=O)C(c2ccc(=O)n(C)c2)(C)C)c(C(C)C)n1 CCCC(C)(O)C(=O)N1CCN(C)C(CNC(c2ncc(Cl)nc2Cl)=O)C1 N1(C(C2C(C=C)CC2)=O)CCC(NC(=O)CCCC)C12CCC2 N1(C(C2CC3(CC(=C)C3)C2)=O)CC(CO)C2(C1)CN(C(=O)CCNC(=O)CO)C2 C(C(F)(F)C(=O)NC(C1CCN(C(C2COC(=O)N2C)=O)CC1)C)OC c1(C(N2CCC(O)(C(C)NC(=O)Cc3cscn3)C2)=O)cccc2nc(O)ccc12 c1(C(=O)NCC2CCCN(C(C(CCC)CC)=O)C2)cc(C)c(N)cc1Cl c1(C(=O)NCCN(C(=O)CCC(CC)OC)CCC)cnc(F)cc1C c1(C(=O)NCCC(=O)NCC(CNC(C=CCOC)=O)O)cccc(C)c1 C=CC(C)(CCOC)C(=O)NCC1CN(C(=O)Cc2cccs2)C2(CCC2)C1 C(C)(CNC(c1cc(=O)n(C)o1)=O)(CC(C)C)NC(C(C1CC1)SC)=O N1(C(c2cc(C)ns2)=O)CC(CC(=O)NCC(C)(O)C(C)(C)C)CC1(C)C CCC(O)C(F)(F)C(=O)NCC1C(C(N2C(CC=C(C)C)CCC2)=O)C1 C(=O)(C1=C(C)CCCC1(C)C)NCC1N(C(COC(CC)C)=O)CCCC1C C(=O)(C1CCCc2ccccc21)NC(C1CN(C(C(F)OC)=O)C1)C c1(C(C)C)ccc(C(=O)NC(C2(O)CN(C(C3(C)CCNC3=O)=O)C2)C)nc1 N1(C(C(CC#C)C2CC2)=O)CCC2(CC(NC(=O)CC3(C(=O)OC)CCCC3)C2)C1 c1(C(=O)NCC2(c3ccccc3)CC(NC(C3(C=C)CC3)=O)C2)ccc(C)cc1 c1(C(N2C3C(NC(C(CC)OC)=O)C(C3)C2)=O)c(OC)ccc2ncccc12 C1(C(=O)NC2N(C(c3nc(C)sc3)=O)CSC2)C2CN(c3cnn(C)c3)CC12 CCCC(C)(C)CC(=O)N1CCC(C(F)C(=O)N(c2cccc(CC)c2)C)C1 C(=O)(C1=C(Cl)CCCC1)NC1(C(N(CCOC)C2CC2)=O)CCCC1C c1(C(=O)NC(CC)CNC(=O)C(c2ccccc2)N(C)C)ncn(C(C)C)n1 C1(C(=O)OC)CC(C(=O)NCC2CC(n3cncn3)C2)C1(C)C CCCCC(C)C(=O)N1CCC(OCCNC(=O)COc2cc(C)on2)C1 C(=O)(C1CCc2cccc(=O)n21)N(CCNC(CC1(C)OCCO1)=O)C1CC1 N1(C(CC(CC)OC)=O)CCC2(NC(c3ccc(C(F)F)cc3Cl)=O)CCCC12 CC1CCc2[nH]c(C(N3CCC(=CCNC(c4ccnn4C)=O)CC3)=O)cc2C1 CC1(C)CCCc2c1n[nH]c2C(=O)NCC12CC(CN1C(C1CCCCS1)=O)C2 C1(C(=O)NC(CNC(C2N(C)CCC2)=O)C2CC2)COc2cc(O)ccc2C1 Cc1ncc(-c2cc(C(=O)NCCC(O)CNC(C34CC(CO)(C3)C4)=O)n[nH]2)s1 C1(C(=O)NC(C)CCCNC(=O)C(=Cc2c[nH]cn2)F)CC1C1CCOCC1 c1(C(=O)NC2CCN(C(CC3C(=O)NCC3)=O)CC2)nnc2n1C=CCC2=O C1(N(C(CSC)=O)C)CCCN(C(=O)C(C(C)C)NC(=O)N(C)C)C1 n1(CC(=O)NCC(C)(CNC(c2cncc(C)c2)=O)OC)ccccc1=O c1(-c2c(C(c3ncn(CCC)c3)=O)scn2)ccc(-c2ccco2)cc1 C(C)(C)(CCC(=O)N1CCCC(F)CC1)NC(C(C)NC(=O)C1CC1)=O c1(C(N2C(C(=O)Nc3c(OCC)ncnc3)CC(F)C2)=O)cc(C)ccc1O C1(NC(c2c(C)cncc2)=O)CN(C(c2ccc(C(N)=O)cc2)=O)CCC1O c1(C(N(C)Cc2n(CC)ccn2)=O)cn2c(n1)CCC(C)C2 c1(C(=O)NC23C(CCN(C(C(CC)=O)=O)CC2)C3)cc2ccccc2n1C Cc1ccc(C#N)cc1C(=O)NC(C1CC(NC(C2CC3CCC(C2)C3)=O)C1)C CC(C)C(=O)C(=O)N(CC(=O)NC1CC1(C)C)CC(C)C S(=O)(=O)(c1ccc(NC(c2ccccc2[N+](=O)[O-])C)cc1Cl)NCCC=C=C C=C1CC2(C1)CC(C(=O)NC1CC(CNC(c3c(C)noc3N)=O)C1(C)C)C2 C#Cc1ccc(C(=O)NCCC(C)(C)CNC(c2c[nH]c(=N)o2)=O)c(F)c1 Cc1cccc2oc(NCC3CN(C(C)C)CCO3)nc12.C(=O)C(C)(C)C N1(C(C2CNC(=O)N2)=O)CCCCC(CNC(c2n[nH]cc2C2CC2)=O)C1 O=C1CC(C(=O)N2CC(C(=O)NC3COCC3CO)C(F)(F)C2)=NN1 C1(C(=O)NC2CN(C(Cc3scc(C)n3)=O)C2)CCCCC(=O)N1 c1(CC(=O)NC2C3(CC(NC(C4(CC)CC4)=O)C3)C2)cc2ccccc2nc1O C1(C(=O)NCC=Cc2cccnc2)(CC)CCCN1C(C1CC(OC)C1)=O CC1(C(N2CC(O)(CNC(c3ccn(C4CCCCC4)n3)=O)C2)=O)CCCC1 N1(C(C2CCC(CC)O2)=O)CCN(C)C(C(N2CC3(CC3C(N)=O)C2)=O)C1 c1(N(C(c2scnc2Cl)C(=O)Nc2ccc(F)cc2)CCC)cc(C)cc(F)c1 C1(NC(=O)COCCCF)CCCC1CN(C(C1CCC(=O)N1)=O)CCO C1(CC)OCCC1C(=O)NC1CN(C(=O)COCc2ccccn2)C1 C1(c2ccc(C(=O)OC)cc2)C(n2cc(SCCCN)nn2)CCC(=O)N1C CCCCCS(=O)(=O)CC(=O)NC12CCCC1N(C(=O)Cc1cnc(C)s1)CCC2 C1(C(N2CC(n3cc(C)cn3)C2)=O)(NC(C=C(C)C(C)C)=O)CC(F)C1 C(=O)(CS(=O)(=O)CCO)NCCC1(O)CCN(C(CCSC)=O)C1 c1(C(N2CC(CCNC(c3cnc(N(C)C)s3)=O)C2)=O)cccc2cncn12 c1(C(N2CCCC2Cc2ccccn2)=O)cnc(-c2ccsc2)s1 CN1CCC(C)(C(=O)NCC2(C)CCCN2C(c2ccc(C#N)nc2)=O)C1=O C1(NC(CCOc2ccc(OC)cc2C)=O)C2Cc3ccc(Cl)cc3C12 N1(C(C2(OC)CCC2)=O)CC(OC)CC(NC=O)C1.c1(C2CC2)ccccc1F Cc1c(CNC2CCn3c(cnc3C)C2)sc2ccc(Cl)cc12 c1(C(N2CCCN(C(C(CCCCC)F)=O)C(C)C2)=O)cnc2c(C)cccn12 c1(C(=O)NC2(CCNC(C3N(C)CCCC3)=O)CCC2)cc2occc2s1 C1(C(=O)NC(C2CCN(C(C3(COC)CC3)=O)C2)C)CN(C(C)=O)CCO1 C1(C(=O)NCC2N(C(C=Cc3c(C)n(C)nc3)=O)CC2)CNC(=O)CC1(C)C C(CCCCCN(C)C(c1ncsc1Br)=O)NC(C1CCC(C)S1)=O Cc1cc(C(N2CC(=C(F)CNC(=O)Cc3cn[nH]c3)C2)=O)c(O)nc1C C=CC(O)(C(=O)NCC(CNC(c1ccc(Cl)cc1)=O)CO)C(F)(F)F C1(CNC(c2cnc(C(C)(C)C)o2)=O)(CO)CCN(C(=O)CC2CC(F)C2)C1 C1(CC(=O)NC(c2ccccn2)CC)CCCC1NC(=O)CNc1cnsc1C c1(NC(C)CNC(=O)CCC2(NC(=O)OC(C)(C)C)CCCC2)cncc(N)c1 c1(C2(CN(CC(C)(C)CN)C)CCC2)ccccc1OCC(O)CN(C)C c1(CC(N2CCCC(N(C(=O)COCC(F)F)C(C)OC)C2)=O)ccc(Cl)c(Cl)c1 S(=O)(=O)(c1nc[nH]c1F)NC(CCC)(N)C(F)F N1(C(c2cc(COC)on2)=O)C(C(=O)NCCCS(C)(=O)=O)CCC12CC2 CC1CCCC1(C(N1CCC1CC1CC1)=O)NC(C1CC(=O)C1)=O c1(OCC=C)ccc(C(=O)N(C)CC2(CO)CC2(F)F)cc1OC c1(C(N2CC(C=C)(CC(=O)NCc3cc[nH]n3)C2)=O)nccc2[nH]ccc12 N(C(=NCC1CCC1)NC1CCN(C2CCC2)CC1)C(C)CC(F)F Cc1nc2cc(C(N3Cc4cnn(C)c4C3)=O)ccc2o1 Cc1cc(Cl)c(Cl)cc1CN1CC2C(C(N3CCCCC3CO)=O)C2C1 c1(C(C)NC(=O)NC(c2cc(Br)ccn2)CC)ccc(F)c(C)c1 C=CC(CCC)CC(=O)NC1CC2CC(NC(c3cnn(C4CC4)c3C)=O)CC12 C1(C(N(CCCNC(CCOCCCOC)=O)C2CCC2)=O)CC2C=CC1CC2 c1(NCCc2ncn(CC)c2)cc(Cl)c(Br)cc1O C=CC(C)(O)C(=O)NC1CC(OCC(N2CC(C(C)CC)C2)=O)C1 C1(C(N2C(CNC(c3cc(Cc4ccccc4)ccn3)=O)CC2)=O)CC12CC(O)C2 C12(C(=O)NC(C)C)CCC(C(=O)NCC(C)NC(c3n[nH]cc3Cl)=O)(CC1)C2 C1(O)(CC(=O)N(CCN(C(C(C)CC2CCC2)=O)C)C(C)C)COC(C)(C)C1 C(C(C(=O)NCc1cc(C)cc(O)c1)C(C)(C)C)NC(CSCC)=O CCCCCC(O)C(=O)N1CCCC(NC(c2ccc3c(c2)NCC3)=O)CC1 c1(C(N2CCC(CNC(c3cc4c(s3)CCSC4)=O)C2)=O)cc2cccnc2s1 Cc1ccc(CC(=O)NCC2C(CNC(=O)Cc3occc3C)C2(F)F)c(O)c1 C(CC(O)CNC(=O)CCOCCN(C)C(C1CN(C)C1)=O)OC C1(NC(C2CN(C(C(C3CC(C)(C)C3)OC)=O)C2)=O)CC(C)(CO)C1 S(=O)(=O)(c1c[nH]ccc1=NCC1C(C)(C)C1(F)F)NCc1c(C)n[nH]c1 c1(CN2CC3C(C(=O)NCCCCC#C)(C3)C2)ccc(Br)c(OC)c1F c1(CC(N2CCCC(CNC(c3c(C)cc(Br)o3)=O)C2)=O)cccc([N+](=O)[O-])c1 C1(C(N(C)Cc2ncn(C)n2)=O)CN(C(C23C(=O)C4CC2C3C4)=O)CC1(C)C c1(CC2CCN(CC(=O)NCC(CC)SCC)C2)cc(C)c(C)cc1C C(=O)(CC(C)C(F)F)NCC(CCCC)NC(=O)Cc1ccco1 c1(NC(C2(COC)CNCCO2)=O)ccc(OC(F)(F)F)cc1C C12(C(=O)NC3CN(C(C(C)CN4CCOCC4)=O)C3)CCCCC1NC(=O)C2 Cc1n[nH]c(C)c1CC(C)C(=O)NC(C)(C)CCNC(=O)C=CC1CCCO1 C(=O)(C(COC)C(F)(F)F)NCCC1CC(NC(C(CCC)O)=O)C1 N1(C(CC2(C)CCOCC2)=O)CCCCC(CCC(=O)NC2CCC3(CC3)C2)C1 Cc1cccc(C(N2CCCC(N(C)C(C34CC(CC(F)F)(C3)C4)=O)C2)=O)c1F N1(C(CSC(C)C)=O)CCN(C(C2CCCSC2C)=O)CC(C)C1 c1(C(=O)NCCN(C(=O)CC2(CSC)CCCCC2)C)ccc2c(n1)OCC(=O)N2 c1(CCC(=O)N(CCN(CCSC)CC)CC)c(F)cccc1Cl C(=O)(C(=O)C(C)CC)NCCCCC(=O)NC1(CC=C)CCOC1 c1(CNC(C=C(CC)C)=O)ccc(C(=O)NC(c2ncco2)CC)nc1 c1(C(=O)OC)ccc(=NCCOCCNC(=O)CC2CCN(C)C2=O)[nH]c1 N1(C(c2cnn(C(F)F)c2)=O)CCC2C(CCCN2C(c2ccnnc2S)=O)C1 C1(C)(C(=O)NC2CN(C(c3cncc(CC)c3)=O)CC2O)CCCNS1(=O)=O O=C(C1=NOC2(CCC2)C1)NC(CC1CC1)C(N1CCc2nccnc2C1)=O c1(C(=O)NCCC2(CNC(c3n(C)nc(Cl)c3)=O)CC2)cnn2ccncc12 C(CCNC(C1(C)CCC(=O)C1)=O)(C(=O)NCCNS(=O)(=O)C1CC1)OC C1(NC(C(C)NC(N)=O)=O)CCOC12CCN(C(c1cc(Cl)ncc1F)=O)CC2 C1(NC(CC(CC)O)=O)CCCCN(C(c2ccc(N(C(C)CC)C)cc2)=O)C1 c1(CCC(N2CC(C)N(C(=O)COCCO)CC2)=O)cc2c(cc1Br)OCCO2 N1(C(=O)C=Cc2cn[nH]c2)CCC2(CNC(C3(CO)CCC3)=O)CCCCC12 N1(C(C2C(C)=CCS2)=O)CCCC(C)(C(=O)NCC=C(Cl)Cl)C1 C(C(C)(O)CC(=O)N1CCC(C(=O)NC2CCCC2C#N)C1C(C)C)OC C1(NC(C2CC(C)NC(=O)C2)=O)CN(C(c2ccc[nH]2)=O)CCC12CCC2 CN1CCN(CC(N2CC3(CNC(=O)OC(C)(C)C)CC2(C(=O)O)C3)=O)CC1=O c1(C(N2CCC(C(C)NC(C3C(C(=O)OC)C3)=O)CC2)=O)ccc(C)cc1F C12(CNC(C3N(C)CCOC3)=O)CC(C1)C(NC(=O)CN1C(=O)CNC1=O)CO2 Cc1cc(CNC(C2CCN(C(c3ccc(Cl)cc3)=O)C2C(C)C)=O)cc(C)n1 c1(C(=O)NC(C)CCCNC(=O)CC2(C)CC(F)(F)C2)ccc(F)c(N)c1F C(=O)(C(F)C(C)C(F)(F)F)NCC1(C)CCN(C(C(C)SCC)=O)C1 CN1CCCC(CN(C)C(c2coc(CNC(c3sccc3Cl)=O)n2)=O)C1 N1(C(C2N(C(C(CC)C#N)=O)CC(OC)C2)=O)Cc2cccc(C#N)c2C1 n1(CC)cnc(C(N2CC(C(C)NC(=O)CCn3ccc(C)n3)C2)=O)n1 C(c1cc(Cl)ccc1Cl)=CC(N1CCCC2(NC(c3c(C)onc3)=O)C1C2)=O C=CCCCCC(=O)N1CCC(CNC(C2CC23CCCCC3)=O)C1 C=CCC(C)(C)C(=O)NC(C)CN1CCN(C(c2n[nH]c(C)c2OC)=O)CC1 c1(C(N2C(C(C)C)CN(C(C3OCCO3)=O)CC2)=O)cc(=O)c2ccccc2o1 c12nc(C)c(s1)C(C)NC(=O)N2.C1(CC)CCN(C)C1c1cccc(Cl)c1 Cc1c(C(N2CC(CC(C)NC(=O)C(C)CF)C2)=O)cnn1CC(F)F c1(C(N(C2CCC(NC(=O)C(C)(O)C3CC3)CC2)C)=O)cccc(CF)c1 CC#CC1CCN(C(=O)C(CC2CCC2)NC(=O)CN2CC=CC2)C1 C1(CC(=O)NC)CN(C(c2cc(C)ccc2C)=O)CCN1C(=O)CC1(C)CC1(F)F C1(NC(Cc2onc(C)n2)=O)CN(C(c2cnc3cccnn23)=O)CC12CCC2 N1(C(C(CCCC)O)=O)CC2CCC(C1)N2c1cc(C)nc(C(C)CC)n1 C1(CCCNC(CSCC=C)=O)CCCCN1C(c1ccc(Br)cc1)=O C1(NC(CC2CC(C(=O)OC)C2)=O)CCCCN(C(c2cc(C)c[nH]2)=O)C1 c1(C(N2CC=CC(C(=O)OCC)C2)=O)cn(C)c(=O)c2cncn12 C1(CNC(CCCC(=O)NC)=O)CC2(CCN(C(C3OC(C)CC3C)=O)C2)CO1 c1(CC(N2CCC(NC(C3CCCC3)=O)C2)=O)ccc2c(c1)CCCO2 C(C(C(C)(C)C)NC(C1(C)CCCOC1)=O)NC(CCC=CC)=O Cc1c(C(=O)NC(C)CCN(C)C(c2ncccc2F)=O)[nH]ccc1=O N1(C(C2N(CC)CCC2)=O)CCC2(CC1)CC2C(=O)NCC1(CO)CC1 N1(C(c2ccn(COC)n2)=O)CCN(C(=O)C(=O)NCC(F)(F)F)C2COCC12 Cc1[nH]nc2c(C(N3CCC(NC(c4ccns4)=O)C(O)C3)=O)cccc12 C(CCCC(=O)NC1(CNC(=O)CC2COC(C)(C)C2)CCOCC1)N(C)C N(C1CCCc2cccc(C)c21)C(=O)NC(COC)COC C1(NC(COC(CC)C)=O)CC(C)N(C(=O)Cc2csc(Cl)c2)C1 n1(CC)ccc2nc(N(C3(Nc4cnccc4C)COC3)C(C)=O)ncc12 n1(CC(=O)NC2(C)CN(C(CN3CCC(C)C3)=O)C2)ccc2nc(O)nc(O)c12 CC1(C)CN(C(=O)CCC2CC(OC)C2)CC(CCNC(=O)CCCC#N)O1 N1(C(C(C)N(C(=O)Cc2ccccc2)CC)=O)CCCN(CC(O)C(F)(F)F)CC1 C(C(=O)NCCCSC)(C1=NOCC1)N(C1CCOCC1)CC C(=O)(CCCCC(N)=O)NCC(C)CNC(C1CC2CC1CC2O)=O N1(C(C2CC(C)CC(C)C2)=O)CCCC(O)(CNC(=O)CC2(O)CCC2)CC1 C1(C(=O)NC2CC(CNC(C3(C#C)CCCC3)=O)C2)CC1C1CC(F)(F)C1 C1(NC(c2c(C)c(O)ccc2)=O)CCN(C(c2cc(F)c[nH]2)=O)CC12CCC2 c1(CNC2CC(C(=O)N=c3cc(Br)[nH][nH]3)C2)c[nH]c2ccc(Br)cc2c1=O c1(C(=O)NCC(CNC(C2ON=C(C)C2)=O)C)nccc(C)n1 c1(CN(C)CC2CCCN(CCn3cc(I)cn3)C2)nc2ccccc2[nH]1 C(C(O)C(F)(F)C(F)(F)F)NCC1OCC(C)(C)C1 c1(OC(C)(C)C)cc(NC(=O)NCC(c2ccccc2F)F)ccc1Cl C(=O)(CCCCCN=[N+]=[N-])N(CCC)CCNC(=O)CC1(c2ccccc2)CC1 N1(C(CCCCC#C)=O)CCCC12CCN(C(=O)C(CO)c1ccccc1)C2 N1(C(CCN(C)CC)=O)CCN(C(=O)CNC(=O)Cc2ccc(Cl)s2)CC1 c1(C(=O)NCC2(OC)CN(C(c3snc(Cl)c3Cl)=O)C2)ccc2ccnn2c1 c1(CC)ccc(C(=O)N(C)CCNC(=O)C(Cc2ccccc2)OC)c(C)n1 c1(OC)cc(Br)ccc1CN1CCC2(CC1)CC2.n12cc(nn1)NCCC2 c1(C(=O)NC2CN(C(C3C(C)=CCS3)=O)CC2O)cc(C)n(-c2ccon2)c1C c1(CCO)cccc(F)c1.C1(C)(NC(C(C)N(C)C)=O)CN(C(=O)CNC(=O)C)C1 C1(C)(NC(CCC2CC(NC(C(CC3CC3)OC)=O)C2)=O)CCC(C)C1 C1(NC(=O)C2=CCCC2)CN(C(c2ccnc3ccsc23)=O)C2(CCOCC2)C1 c1(NC(CCC)C2CCCC2)ncccc1S(=O)(=O)NCC(c1cccc(Cl)c1)O N1(C(c2ccc(Cl)cc2C(F)(F)F)=O)CCCN(C(=O)C2CC2)CCC1 c1(NC(=O)NC2CC(CCNC(C(C(C)C)(C)O)=O)C2)ccc2c(c1)CC(=O)N2 CC(C)(O)C(F)C(=O)N1CCC(C=CC(=O)NC(c2cccnc2)CO)CC1 Cc1cn2ccc(C(=O)NC(C)C(C)NC(c3cc(Cl)cnc3O)=O)cc2n1 c1(C(=O)OC)ccc(C(N2CCCC(CCNC(=O)CSC)C2)=O)c(F)c1 C(CCC(=O)NO)N(C(=O)CCC1CCCN(C(=O)CC2NC(=O)NC2=O)C1)C c1(C(C)CNC2CC(c3ccccc3)CO2)ccc(F)c(F)c1 c1(C(=O)OC)c(C)noc1CNC(c1c(CNC(=O)O)cccc1)C n1(-c2c(C(N3CCCC4(C=CCO4)C3)C)cccc2)ncc2ccc([N+](=O)[O-])cc12 n1(CC)ccc(=NC(=O)C2(C)CCCN(C(c3cnc(C4CC4)nc3)=O)C2)[nH]1 N12CCCCC1CCC1CCCN1C(=O)C(C)CC2=O.CCCCOC1CCC1 c1(C(N2CCC(NC(C(CCC#C)O)=O)C2)=O)cc(Br)cc(C)c1C c1(C(NOC(C=C)C)=O)ccc2c(n1)CN(C(C1CCC(OC)CC1)=O)CC2 c1(C(N(CCNC(Cn2c(C)nnn2)=O)C)=O)ccc(O)c(CO)c1 C(=O)(C(O)C(C)(C)C)NC(CC=C)CNC(c1cccc(CC=C(C)C)c1)=O c1(C(C(F)(F)F)C(=O)NC(C=C)C2CCC2)ccccc1F Cn1ccc(C(N2CC3CC(C(N4CCC(C#N)C4)=O)(C3)C2)=O)cc1=O C1(NC(CC(CCC)O)=O)CN(C(c2cc(C(N)=O)no2)=O)CCC1(C)C c1(C(N2CCC(C(C(=O)OC)C#N)C(OC)C2)C)c(C)cc(C)nc1OC N1(C(CSCC)=O)CCC(C2CC2)C1C(=O)N(c1ccc(C)cc1C)C C1(NC(=O)Cn2cnnc2)COCCC1NC(C1CC1F)=O c1(CC)cc(-c2nc(CN3CCCCCC3)nn2CC2CC2)c(C)o1 N1(C(c2cc(CC)no2)=O)CCN(C(=O)CN(C(=O)C(CC)CC)CC)CC1 N1(C(=O)Nc2ccc(C)s2)CCC(c2ccc(Br)cn2)CC1 CC1CN(C(=O)COc2ccc(Cl)cc2)CC1CNC(C1C=CC=CC=C1)=O N1(C(C(CC#C)CC#C)=O)CCC2CN(C(=O)CCN(C)CC)CC2C1 CN=C(NCC1(C)CCC(=O)N1)N1CCC(c2csc(C)c2)C1 C1(CNC(c2c(CC(C)C)onc2)=O)COCCN(C(c2ccc(F)s2)=O)C1 Cc1ccc(C(=O)NCCCCC(C)NC(c2nncs2)=O)c(N=[N+]=[N-])c1 CC(CC(=O)NCc1cnco1)N(C)C(c1csnc1Cl)=O CCCCCCC(F)C(=O)N1CCCC(CO)(NC(=O)C(=Cc2ccco2)C)C1 N1(c2cc(COC)ncn2)CCC(O)(C(=O)N(CC(C2CCCC2)C)C)CC1 c1(CN2CC3C(NC(c4cnc(C)nc4)=O)C3C2)ccc(Br)cc1O c1(C(CC(=O)N(C)C)NC(C(CC)OC)=O)cccc(Br)c1 CCC(F)(F)C(C)(C)C(=O)N1C2CCC1C(NC(c1cc(C)nc(C)c1O)=O)C2 CC(C(CO)NC(=O)CCc1ccsc1)NC(c1cc(-c2ccccn2)no1)=O N1(C(C(c2c(C)ccnc2)(C)C)=O)CC2CCCCC2(NC(C2CC(C)C2)=O)C1 c1(C(=O)NCC(CNC(C2C(C)CN(C)C2)=O)(C)C)coc2cc(O)ccc12 C(=O)(C1COc2ccc(F)cc21)N1CC(C(C(N2CCC(CO)C2)=O)NC(C)=O)C1 C1(N(CC(C)C)C(C2CC2(C)C)=O)CCN(C(c2ccc(O)nc2)=O)CC1 n1(CC)ncc(I)c1C(=O)NC(c1ccc(Br)cc1)CC(C)C c1(C(=O)NC2C(CNC(C=CCC)=O)COC2)ccncc1OCCOC C(C(CNC(C1CCC(=O)N(C2CC2)C1)=O)C(F)(F)F)NC(CC)=O N1(C(CSCCCC)=O)CC2CC(NC(c3ccns3)=O)C(C2)C1 c1(C(=O)NC(CCC)CNC(=O)C(C2CCCCC2)C)c(C)n[nH]c1C Cc1ncc(NC(=O)C(C)CCCNC(c2cnnc(C)c2C)=O)cc1C#N C1(C(=O)NC2C(C(=O)NC(C(N)=O)c3ccco3)CCOC2)CCCC12CCC2 C(C)(C(=O)NCC1CCCN1C(c1cn(-c2cccnc2)nn1)=O)(C1CC1)OC C(=O)(C#CC1CCCOC1)N(CC(C)(C)CNC(C1(C)CCCCO1)=O)CC C1(c2cn(C(C)CNC(=O)C(C(C)C)n3cnnn3)nn2)(COC)CCOCC1 C1(NC(C(C)OCC(F)(F)F)=O)C2CC1N(C(C1(C#N)CCCC1)=O)C2 CCC(C)(C)C(C)CC(=O)NC(c1ccc(F)cc1)CNC(=O)CCC(F)(F)F CCC(CC(=O)NC(CN(C)C)C(=O)NC1CCNC1=O)C1CCC1.C1CCC1 c1(C(=O)NC(C2CN(C(COCc3ccc(C)cc3)=O)C2)C)cc(N)c(Cl)cn1 C(=O)(C(C)(C)C(=O)CC(=O)O)NC1CC(n2cc(C(CC)(C)O)nn2)C1 CC(C)(C)CCCC(=O)NC1CCN(C(=O)CCn2ccc(O)nc2=O)C1 C(=O)(C(=O)N=S(C)(C)=O)N.CC1(C)CC(CCNCCOC)C(=O)N1 c1(C(=O)NCC2N(C(C(N)=O)=O)CC=C2)cccc(C(F)F)c1 Cc1cc(CCC(=O)N(CCCCNC(=O)C(=C2CCCCC2)F)C)cc(C)c1 C(=O)(CCCn1ccnc1)N1CC(N(C(=O)CSC2CC2)CC)C1 C1(C(=O)NC(C)C(=O)NCCN2CCCC2)CC2(C1)CC2F C1(N(c2ccc(C(=O)Oc3c(Br)cn(C)n3)cn2)C)CCC12CCNCC2 C1(NC(C2(O)CCC(C)CC2)=O)CC2CN(C(c3ccccc3)=O)CC2C1 C1(NC(c2ccc(CC)c(Cl)c2)=O)CCC2(CCCN(C(=O)CC(F)(F)F)C2)C1 C=CCC(C(=O)NC1(CF)CCN(C(=O)Cc2cnns2)C1)C(C)C C1(C(=O)NC2CCCC2SC)(CC)CCN(C(=O)COCC(C)(C)C)CC1 CC(CC(F)F)CS(=O)(=O)NCc1cn(C(C)(C)C)c(=O)nc1O CC(O)C(F)(F)C(=O)N(CCCNC(C1(F)CCC1)=O)C1CC1 N1(C(C(=O)Nc2cc(C)c(C)nc2)=O)CC2CC(C1)C(N)C2CO N1(C(C(C2CC2)OC)=O)CCC2CN(CC(=O)NC3CCCC(C)C3)CC2CC1 c1(C(=O)NC2CN(C(COCC)=O)CC2(C)C)cc2c(cc1N)CCCC2 C1(CC(=O)NCCCCSCC)CCCN(C(=O)CC(=O)OC(C)(C)C)CC1 C12(CNC(CC3(C)CCN(C(c4c(C)[nH]nc4CO)=O)C3)=O)COC(C1)C(O)C2 CC1(Cc2cccc(Cl)c2)CN(C(C2(CO)CCOC2)=O)CCS1 C(C)(C)(CC(C)N=c1[nH]c(N2CCC3CCCCC3C2)nc2c1CSC2)OC C(C(=O)NOCC(O)C(C)(C)C)(OC)NC(C)C.C12(CC1)C(=O)NC2 CCCCC(C)CCC(=O)NCC1(F)CCC(CNC(=O)C(F)(F)F)CC1 C1(CN(C)C(c2ccncc2)=O)CN(C(c2ccccn2)=O)CCO1 N1(C(C2C(C(=O)OC)CC2)=O)CCCC(O)(CCNC(c2ccnc(S)c2)=O)C1 c1(OC)ccnc(OC)c1C(=O)NCC1(C)CC(NC(c2nc(=N)cc[nH]2)=O)C1 Cc1nc(C#N)ccc1C(N1CCC(F)C(NC(c2cnc3n2CCS3)=O)C1)=O c1(CC)cccc(C(=O)NC2CCN(C(C3CN(CC)CCO3)=O)C2CC)c1F Cc1cc(CC(N2CC(N(C)C(c3cnncc3)=O)C2)=O)no1 N1(C(C=CC(C)C)=O)CC2=C(C1)CN(C(=O)CNc1nccs1)C2 c1(C(=O)NCCCC(C)NC(C2OCCN(C)C2=O)=O)ncn2c1CCCC2 c1(C(N2CCC(C)(CNC(=O)Cn3nnnc3C3CC3)C2)=O)cc(F)ccc1F N1(C(=O)CC2(O)CCC2)CC(CO)C2(CCN(C(C3CCCSC3)=O)CC2)C1 CCCS(=O)(=O)C(C)C(=O)NCC1CCCN1C(c1cc2cc(Cl)ccc2[nH]1)=O CS(=O)(=O)C1(C(=O)N(C(CO)CCCCl)C(c2ccccc2)=O)CC1 C(=O)(C(C)C(C)NC(c1csnc1Cl)=O)NCc1snc(CC)n1 C1(ONC(C2COCC2NC(C2(CF)CCOCC2)=O)=O)CCC(O)C1O C(=O)(C(F)CC(C)(C)C)N(CC(N1CCOC(CCF)C1)=O)CCC c1(C(=O)NO)ccc2c(c1)OCC2.c1cccc(I)c1 N1(C(c2c(C)nco2)=O)CCN(C(c2cc(F)cc(Cl)c2Cl)=O)C2CCC12 c1(NC(CC2CC(NC(c3nccc(C)c3)=O)C2)=O)cc(F)c(F)c(F)c1Br Cc1cc(=NC(=O)C(=O)NC2(CNC(C3(C)CC4CCC(C3)S4)=O)CCC2)[nH]o1 CN=c1nc(N2CC3CC2CN3C(=O)NC(C)(C)C)[nH]c(=NCC(F)F)[nH]1 CCCC(C(=O)N1CCC(C(N2CCC(CCOC)CC2)=O)CC1)C(C)C c1(CC)cccc(-c2cccc(OCc3cccc(C)c3)n2)c1 C12(CNC(c3nc(C)sc3C)=O)CN(C(C3CCOC3)=O)CC1(C(F)(F)F)C2 C1(C(N(C)CC2CC2(F)F)=O)CCN(C(c2c[nH]nc2C2CC2)=O)CCO1 C12(C(CNC(CCc3ccc(C)s3)=O)NC(c3n[nH]c(C)n3)=O)CCC(CC1)C2 N1(Cc2cccc(NC(=O)CCOC(F)(F)F)c2)CCS(=O)(=O)CC1 C(=O)(C#CC1(NC(=O)OC(C)(C)C)CCCC1)N1CC2(CC(C(=O)OCC)C2)C1 C1(NC(CCC(N)=O)=O)CN(C(c2nnc(C(F)(F)F)s2)=O)CC(F)(F)C1 C1(CNC(CCC)=O)CCCCN(C(c2noc(-c3ccc(O)cc3)n2)=O)C1 C(CC(=O)N(C)CC1CCN(C)CC1)(C(C)(C)C)NC(C(CC1CCC1)OC)=O C1(CC(=O)NCC(CNC(COC)=O)OC)CC(F)(F)C1 c1(C(=O)OCC)cccc(C(=O)NCc2nc(C(N3CCCS3(=O)=O)=O)co2)n1 c1(C(N2C(CCNC(=O)Cn3cnnn3)CCCC2)=O)nnc(O)nc1O N1(C(c2c(OC)nc(C)cc2)=O)CC2CCC1C1CN(Cc3ccccn3)CC21 C1(NC(=O)CCCC2CC2)CC2CCC1CN2C(C1CC2(C1)CC(F)(F)C2)=O N1(C(c2c(N)ccc(C)c2)=O)CC(N(C)C)C2(CCC2)C1 C1(COC2CCN(C(c3sc(Br)nc3Cl)C(=O)NCC)C2CC)CCS(=O)(=O)C1 c1(C(=O)NCC(CNC(=O)CC(C)SC)OC)cnc(O)c(C(C)=NO)c1 c1(C(=O)NCCN(C(=O)C(C)(C)C#N)C)cc(C(=O)N(C)C)ccc1Br c1(C(=O)NCCCNC(CC(CC)C)=O)nc(C)ccc1C c1(OC)ccc(C(C)(C)CNCCC2CCCCN2C2CC2)cc1 c1(Cc2cc(C(N3CCN(C(=O)COC)CC3)=O)no2)cc(C)ccc1C C1(CC)CN(C(=O)CCC2CC2CC2CC2)CCN1C(=O)C(=O)NOC O=C(O)C#CC(=O)NC1CCN(C(=O)Cc2cc[nH]n2)CC1 Cc1cc(CNC(c2ccccc2NC2CC2(F)F)=O)c(O)c(Br)c1 N1(C(C(C2CCC2)OC)=O)CC(C)(C(=O)NC2CC=C(C(C)C)CC2)CC1(C)C N1(C(=O)C=C2CCC(C)C2)CC(C(C)C)C(C)C1.n12cc(nn1)CNC(=O)C2 n1(CCC(N2CC(C)(NC(c3c(C)cc(C)o3)=O)C2)=O)nc(O)c2c1CCCC2 N1(C(CC)C)CC(NC(C2CCCN2C(c2occc2OC)=O)=O)CC1=O C#Cc1cccc(C(N2CC(NC(=O)Cc3ccsc3)C(CCC)C2)=O)c1F C=CC(C)(CC)C(=O)N1CC(NC(=O)C2=CC(C)(C)C2)C(C(F)F)C1 c1(C(=O)NC(C)(CNC(=O)Cc2cnc[nH]2)C2CC2)cc2cnc(Cl)cc2s1 c1(C23CCCC2C3)ncnn1C1CCCC1.C1(CCc2occc2)CCCC1 c1(C(=O)NC(CC)CN(C(=O)CCc2c(C)noc2Cl)C)nccc(Cl)c1C c1(CNC(CCN(C)C(c2cccnn2)=O)=O)nnc(O)nc1O N1(C(C(c2ccccc2F)OC)=O)CC=CC(NC(=O)C=C2CCN(C)CC2)C1 C(=O)(C1=C(Cl)CCC1)N(CC=CC(=O)NCC#C)C N1(C(C2(CC=C)CCOC2)=O)CC(O)CC1C(=O)NC1CC(C)(CC)C1 Cc1nc(CC(=O)NCC(C)NC(=O)Cc2cscn2)oc1C N1(C(CCC(C)=O)=O)CCCC(F)(C(=O)N(C(c2ccccn2)C(C)C)CCO)C1 C(=O)(C(=O)N=S(C)(C)=O)NC(C1(O)CCN(C(C23CC2COC3(C)C)=O)C1)C C1(NC(c2c(C)occ2)=O)CCC(NC(c2cn(C(C)C)nc2C(F)F)=O)CC1 CCCS(=O)(=O)C(C)C(=O)NC1(CCNC(c2cc(C)sc2N)=O)CCC1 N1(C(c2nc(OC)oc2)=O)CCC2(C1)CN(C(c1c(C)n[nH]c1C)=O)CC(C)O2 C(c1cocn1)=CC(=O)NC1CCCC1CNC(=O)CCc1nc(O)n[nH]1 c1(C(=O)NCC(C)(C)NC(C2C(C)C2(F)F)=O)ccccc1CN1CCSCC1 C1(N(C(C(c2cccs2)SC)=O)C)CCCN(C(=O)CC2(C(F)(F)F)CC2)C1 N1(C(C2CCN(C(CCNC(C)=O)=O)CC2O)=O)CC(C)N(C)C(C)C1 C(=O)(C1=CNC2=NCCC2=C1)NCC=CCCC.C1(=O)C(C)=CCN1 N1(CCC)CCC(C(=O)N(C2CN(C(=O)CN3CCCC3C)CC2O)C)CC1 c1(CC)cccc2c(C(N3CCCC(N(CC(C)C(C)C)COC)C3)=O)c[nH]c12 N1(C(C=CC)=O)CC2(CC(NC(=O)C)C2)C1.c1(C[SH](=O)=O)cc(Cl)ccc1O CCC(C#N)C(=O)NC1CCCC(CC(=O)NCCCn2nccn2)C1 c1(OC)ccc(F)c(C(=O)NC2CCCCC2NC(=O)CCc2cccnc2)n1 Cc1ccc(C=CC(N2CC(O)(CNC(=O)CN3CCC3)C2)=O)o1 C1(C)(COC)CCN(C(=O)CC2CCCN(C(=O)C(C)C3CCCC3)C2)C1 C1(C(=O)NCCCCCNC(C(C)(C)c2cccs2)=O)CCCC(C2CC2)O1 c1(C(=O)NC(CCOC)C(=O)NCCC(O)CSC)ccc2cncn2c1 C=CC1CN(C(=O)CN(C)CCC)CC1NC(=O)Cc1ccc(F)cc1Cl CC1CN(C(C2(S(C)(=O)=O)CCC2)=O)CC1(C)CNC(=O)C(=O)NC1CC1 C1(NC(C(CN(CC)CC)F)=O)CCN(C(=O)Cn2ncnn2)C(C)C1 C1(CN(C(c2cn(C(C)C)nn2)=O)C)COCCN1C(c1cccc(Br)c1)=O C(=O)(C1=CC2C=CC(C1)C2)N1C(C)CCN(C(C(C)CC2CCCCC2)=O)CC1 Nc1cc(C(=O)N(CCCNC(=O)CC2CC2C2CC2)CCO)ccc1Cl CC1CC1(C)S(=O)(=O)NC(c1cccc(C2(C#N)CC2)c1)=O N1(C(C2CC2c2cncs2)=O)CCOCC1CNC(C1(O)CCC1)=O C1(C(N2CCC(OC)C2)=O)CCN(C(=O)C(C)C)CC1C N1(C(C2(OC)CN(C(C3CC4CCC3CC4)=O)C2)=O)CCCC(C(N)=O)(CO)C1 C1(NC(=O)CC2CC=CC2)CCCCC12CCN(C(c1c[nH]nc1C1CC1)=O)C2 CC1CC=C(C(=O)NCCC2(CNC(C3CCSC(C)C3)=O)CC2)CC1 c1(CNCC(=O)NCc2ccc(CC)s2)cccnc1OC CC1CCC(NC(c2coc(C3CCCC3)n2)=O)CN1C(=O)CC1(C)CC1(Cl)Cl N1(C(c2c(C)ncc(C)c2)=O)CCOC2(CCN(CCC3CCCCO3)CC2)C1 Cc1cc(C(N2CCC(C)C(NC(C3(C)CCCC3)=O)C2)=O)c(N)c(Cl)n1 c1(OC)c(F)ccc(F)c1C(N1CCN(C(C2CC2C2CCCC2)=O)C(C)C1)=O c1(CC2C(NC(N(C3CCN(C)CC3)CC)=O)CC2)ccc(C)cc1 c1(OC)c(C)cc(C(N2CCC(NC(c3sccc3Cl)=O)C2)=O)cc1C c1(C(N2C(C)C(NC(C3CCCSC3)=O)CC2)=O)ccc2c(=O)ccoc2c1 N1(C(c2cc(CC)sn2)=O)CCCOC(CNC(c2nccnc2C(N)=O)=O)C1 C(=O)(CCCC(F)F)N1C(C(C)NC(C(n2ccc(C)n2)C)=O)CCC1 N1(C(C(CC)OC)=O)CCCC(C)(C)C1CNC(C1CC2C=CC1CC2)=O CC(C)C(CCNC(=O)CC(O)c1ccccc1)NC(=O)CCCC1CC1 c1(C(=O)NC(C(=O)NC(CCC)CCC)CC=CC)cnn2c1CCC2 c1(C(C)C)ccccc1C(=O)NC(=O)N(CC(O)CN(C(=O)C(F)C1CC1)C)C C=CCC(CC)C(=O)NCC1(F)CCCN(C(=O)CCc2nc(CSC)no2)C1 C1(C(=O)NCC(C)NC(=O)Cn2cc(P(C)(C)=O)cn2)C2CCC(C2)S1(=O)=O N1(C(COC2CCN(C(=O)Cn3cccc3)C2)=O)CC(F)(F)C1C1CC1 Cc1c(C(=O)NC2CCCN(C(C3SCCCS3)=O)C2C)cccc1C1CC1 C1(C(CNC(C(C)OCCOCC)=O)(C)C)CN(C(=O)C(O)C2CCCC2)CCO1 c1(C(C(N2CCC(N(C(CNC=O)=O)CCO)C2)=O)C)ccc(F)cc1.C1CC1 c1(CC(=O)Nc2ccc(CNC(COC)=O)c(C)c2)ccc2occc2c1 C1(NC(CC2CCN(C(c3n(C)nc(O)c3)=O)C2(C)C)=O)CC2CC1C(O)C2O N1(C(C(CCO)N(C)C)=O)CC(NC(=O)CCc2ccsc2)CC12CCCC2 c1(C(N2CC(CC)C(NC(=O)CN(C)C(C)C)C2)=O)cc(Cl)c(F)cc1N c1(C(=O)NC2CC(C)(NC(=O)CC(=O)NCC3CC3)C2)cnn2c1OCC(F)C2 C(CCCCCCO)NC(C(C1CCCO1)NC(c1cc(OC)ns1)=O)=O S(=O)(=O)(c1[nH]c(=NCCC(N)=O)ccc1Br)N(CC)Cc1cccc(F)c1 N1(C(c2c(Cl)cn(C)n2)=O)CCC2(CCCN(C(c3ncnn3C)=O)C2)C1 c1(C(N(C2CN(C(C=CC(C)(C)SC)=O)CC2O)C)=O)ccc(F)c(F)c1F C(=O)(CCN(OC)C(=O)Cc1cccc(C#N)c1)NC1C(OCC)COC1 N1(C(C)C)CCCC(C(=O)NC2(CF)CCN(C(c3cccc(=O)o3)=O)C2)C1 CC(C(C)NC(=O)N(C)Cc1ccc(Cl)cc1Br)S(C)(=O)=O c1(C(N2C(CNC(c3nc(O)[nH]c(=O)n3)=O)CCC2)=O)c(Cl)nsc1Cl C(=O)(C(C)(O)CC(C)C)NC1CCN(C(CCOCC(C)C)=O)CC1(C)C c1(-c2cc(OC)c(F)c(F)c2)cccc2cc(C(=O)Nc3cccc(OC)n3)[nH]c12 Nc1cc(F)c(Cl)cc1C(=O)NCCCNC(C1(n2cnnn2)CC1)=O C1(C(=O)OCCc2nccs2)CCC(C2CCCCC2)CN1 c1(C(=O)NCC2CC3(CN(C(CC(CC)C)=O)C3)C2)cc2cc(Cl)cnc2o1 c1(C(=O)NCC(Cc2ccccc2)NC(C(C(C)C)C)=O)cccc2scnc12 C1(NC(Cc2nc(C)sc2C)=O)CN(C(=O)C(C#N)=CC(C)C)CCC1O N1(c2nc(C)c(F)cn2)CCC2(CC1)CC(C(=O)N=c1cco[nH]1)CO2 Cc1cc(C(=O)NC(C2(CNC(C3(F)CCCOC3)=O)CC2)C)ccn1 C1(C(=O)OC)CN(Cc2cc(CNC(C)C3CC3)on2)CC(F)(F)C1 N1(C(c2c(CC)oc(C)c2)=O)CC(NC(=O)CC23CCC(CC2)C3)CC(O)C1 N1(C(C(n2ccc(C)n2)C)=O)CCCC(CN(C)C(c2c(Cl)cnn2C)=O)C1 c1(OC)cncc(C(=O)NCC=CCNC(=O)CCCc2csc(C)n2)c1 CCN=C(NCC(Cc1ccc(F)cc1)CO)NCC1(F)CCOC1 N1(C(Cc2scc(CC)n2)=O)CCCC2(CCCCC2NC(=O)C(C)CCC)C1 N1(C(c2c[nH]c(=O)c3ccnn23)=O)CCCCC1C1CCCN1Cc1nccs1 C1(C(=O)NCC(O)CNC(C2CCCC2O)=O)(CC)CCCC1 C=CC(CC)CC(=O)N(c1ncc(F)cn1)Cc1ccc(F)cc1 NS(=O)(=O)c1cc(-c2ccc(CCNS(=O)(=O)C(F)(F)F)cc2)c(F)cc1Cl CCC(C)(C)C(O)C(=O)N(CCCN(C)Cc1ccc(C)o1)C C1(C(=O)NCCN(C(=O)CC2CCC=CCC2)CCC)CCC(F)(F)C1 C(C(C(=O)NCC1(O)CCOC1)C(C)(C)C)NC(CN(CC(C)(C)C)C)=O C1(C#N)(C(=O)NCC(C)NC(C2C(CN=[N+]=[N-])C2(C)C)=O)CCOCC1 C(CC(CC)(CC)NC(C1CC2CC2C1)=O)NC(C(C=C)O)=O Cc1cn2c(n1)C(C(=O)N1CCC(C)C(CNC(=O)C(C(C)C)C(C)C)C1)CCC2 c1(-n2c(C)nnn2)ccc(C(N2CCN(C(c3ccnnc3C)=O)CC2)=O)cc1 C1(C)(C(=O)NCC2(C)CCCN(CC3CCC3)C2)CC2CCC(C1)S2 C(N=c1[nH]cnc2ccc(NC(C(C)SCC)=O)nc12)C12CCC(CO)(CC1)OC2 N1(C(c2cnc(OC)s2)=O)CC2CCC2(CCNC(C2(C(C)=O)CC2)=O)C1 c1(CNC(=O)NCC(c2cc(C)n(C)n2)(C)C)cccc(F)c1Br C1(C)(C(=O)OC(C)(C)C)N=N1.C1(=O)CN(CC)C(=O)O1 C(=O)(C(CC1CC1)NC(=O)C(C)N(C)C1CC1)NCC(CSC)OC C(CC(=O)N1CCCCC1C(F)F)(C(F)(F)F)NC(C1(C)COC(=O)N1)=O CCCCC(O)C(=O)NC(CNC(=O)CCc1ccc(F)c(F)c1)C(C)OC N(C=CC(=O)C(F)(F)F)C(CC1CCN(C(C(c2cccc(O)c2)C)=O)CC1)=O C=C1Cn2c(C(=O)NC(CN(C)C(C3CC4CCC3C4)=O)(CO)CO)nnc2S1 CC1CCCN(C(=O)C(=O)NC2CN(C(c3c[nH]nc3C3CC3)=O)CC2C(F)F)C1 c1(C(N2CC(C(C)NC(Cc3c(C)ccc(C)c3)=O)C2)=O)ccc(N)c(Cl)c1O C=C1CC2(C1)CC(C(=O)N(CCCOCCNC(c1cnc(O)cc1C)=O)C)C2 N1(C(c2c(NC)cccc2)=O)CC(C(=O)NC(CCO)C(C)(C)C)C2(CCC2)C1 CC1CCN(C(=O)COc2ccsc2)C1CNC(c1cccn1C1CCCC1)=O Cc1cn2cccc(C(=O)N(C)CCN(C(=O)CCNC(=O)CO)C)c2n1 N1(C(CCCCC)=O)CC2CN(C(C3CCCC3)=O)CC2(C)C1 N1(C(CC(CCC)(C)C)=O)CCC2(CNC(c3ncc(C)cn3)=O)CCCCC12 C1(C(N2CC(O)(CC(=O)NCC#C)C2)=O)CSCC(=O)N1 CC(C)(C#CC(=O)N=c1ccn(-c2ccc(Cl)cc2)[nH]1)CC(F)F CC1CC(NC(c2cnc3sccn23)=O)CCN1C(=O)CCc1cnn[nH]1 Cc1onc(Br)c1C(N1CCOC(C(C)NC(c2cncc(F)c2)=O)C1)=O C1(NC(CC2C(C)(C)C2)=O)CCN(C(=O)CCc2cccc(F)c2Cl)C1(C)C c1(NC(c2c(CNC(CCc3ccc(C)o3)=O)ocn2)=O)nccc(C#N)n1 c1(C(=O)NCCOCCC(=O)N(C(C)C(C)C)CCC)cc(F)c[nH]1 C1(C(N2CC(C)(NC(c3ccsc3)=O)C2)=O)COc2ccc(F)cc2C1 Cc1ccnc(C(N2CCC2(C)CC(=O)NCC(C)(O)CCO)=O)c1N N1(C(C(=O)NCCCC(=O)OC)c2nc[nH]n2)CCC2NC(=O)NCC2C1 c1(CN(C(=O)C(CNC(=O)CC2(O)CCCC2)N(C)C)C)ccccc1 Cc1ncncc1C(N1CCC(N(C(=O)C(N2CCSCC2)C)CC2CC2)C1)=O c1(C(=O)NC(C)CNC(=O)C(C)S(C)(=O)=O)nc2n(c1Cl)CCCC2 c1(C(C(=O)N(CC2(F)CN(C(CCSCC)=O)C2)CC)C2CC2)ccc(F)c(F)c1 c1(C(=O)NC2C(NC(C(CC=C)CC=C)=O)C2)cnc2c(c1)CCCC2 n12cc(c(C)n1)NC(=O)C1CCN1C2=O.C1(CC)CC2C=CC1O2 c1(C(=O)NC(CC)(CNC(c2cc(C)ns2)=O)CC)c(C)cccc1Cl N1(C(C(C2CCC(=O)N2)C)=O)CC(C(=O)NOC2CCOC2)C(C2CC2)C1 C1(NC(CC2CC(=C)C2)=O)CCC(O)CN(C(c2ccn3c2CCCC3)=O)C1 CC1(C(N2CCC(NC(=O)CCCc3ccncc3)C2)=O)CC1(Cl)Cl N1(C(c2c(CC)cno2)=O)CCN(C(=O)CC2CCCOCC2)CC1CCOC N1(C(C2(C=C)CC2)=O)C2CCC1CN(C(c1nn(CC)cc1Br)=O)C2 c1(C(=O)NC2CC(CNC(C34OC(C)(C)C(C3)C4)=O)C2)ccc(Cl)c(N)c1Cl c1(N(C)C)cccc(C(N2CCC(C)(N(CCO)C(C3CCS3(=O)=O)=O)C2)=O)n1 C1(CC(=O)N(CC(CC)NC(C2(C)CC(F)(F)C2)=O)C)CCC(=O)C1C Cc1nc2cc(C(=O)NCCN(C(C3CC(CC(=O)NC)C3)=O)C(C)C)[nH]c2s1 CN1CCN(C(C2CCC(NC(=O)Cn3cnc(C#N)n3)CC2)=O)CC1(C)C N1(C(C(C)CNC(=O)CCCN2CCCC2)=O)CCC(C)(C#N)C1 c1(C(CC)C)cc(C(N2CCC2CNC(c2ccnn2C(F)F)=O)=O)on1 c1(C(C)(C(=O)NC2CC2C(=O)NC2(c3ccccc3)CC2)OC)ccccc1Cl N1(C(c2cc(C)oc2)=O)CCC2(CC1)CC2NCC(=O)Nc1c(C)cncc1C c1(C(=O)NCC2CCCCN2Cc2cccc(Cl)c2F)nccc2[nH]ccc12 c1(C(N2CCC(CCNC(c3n(CCOCC)ncc3)=O)C2)=O)ccncc1C Cc1cccc(C)c1C(=O)NC1CC2(C1)CC2C(=O)NC1COC2(CCC2)C1 c1(C(N(C)CC2CCCCN2C(c2sccc2Cl)=O)=O)ccc2occc2n1 N1(C(CCCC(N)=O)=O)CCCCC2C1CCCN2C(=O)C1=CCOC1 C1(C(=O)OC)CCCCN1C(C1(CNC(=O)C=Cc2ccc(C)o2)CC1)=O C(=O)(C1=CCCN(CC2CCN(C(c3ccc(F)cc3Br)=O)CC2)C1)OC c1(C(=O)OCC)ccc(C(=O)NC2C(NC(=O)CC3C(=O)NN=C3C)C2)cc1 c1(C(N(C2CCN(C(C3CC=CCO3)=O)C2)C)=O)ncc(F)cn1 C1(CC(=O)NCC(C)NC(C2(C=C)CCC2)=O)CC(C)(C)C(=O)N1 Cc1ccn2ncc(C(=O)NC3CCC(C)N(C(=O)CC4=CCCCC4)C3)c2n1 C#CC1(NC(=O)CCC2(NC(c3ccc(C(C)=O)[nH]3)=O)CCC2)CCC(C)(C)C1 C(CCC(C)CC(=O)NCCC(C(C)C)NC(c1cn(C2CC2)cn1)=O)=C(C)C c1(C(N2CCN(C(CP(C)(C)=O)=O)C3(C2)CC3)=O)cnc2nc(Cl)ccc2c1 c1(OCC)cnc(C(=O)NCC(CN(C(=O)C(C)OC(C)(C)C)CC)(C)C)cn1 c1(CC)cn2nc(Cl)cc(N3CCOC(c4ccc(Cl)c(F)c4)C3)c2n1 C(C(C)C)(C(O)C(=O)N1CC(CC(N2CC(C3CC3)(OC)C2)=O)C(C)C1)OC CC1CCN(C(=O)C(C)Cc2ccco2)CCN1C(C1(CN(C)C)CCCC1)=O c1(OC)cc(Br)cc(F)c1OC1CCN(C(C2CCCN2c2ncco2)=O)CC1 c1(C(N2CC(O)(CC(N3CCC3c3cccs3)=O)C2)=O)cc(Cl)ccc1Br n1(CCSC)nnnc1C(c1n[nH]cc1C)NCC1CCCC1 N1(C(C(C(C)C)(C)C)=O)CCC2(CC1)CN(C(C1CC3CCCCC13)=O)CCO2 c1(SC)cc(C(=O)NC2(C)CN(C(=O)CCc3cncs3)C2)ccc1[N+](=O)[O-] c12noc(n1)CCC(=O)OC2CC.C1(CCNC(C)=O)CN(C(=O)C(C)N2CCC2)C1 CC1CCCN(C(=O)COCc2ccccc2)C1CNC(=O)C=CC(=O)NC.C(CO)=C c1(C(=O)NC2CN(C(C(C)=O)=O)CC(F)(F)C2)cc2n[nH]cc2cc1Cl CCCCC(C(=O)N(CCC(C)NC(=O)CC1CCCC(C)(C)O1)C)N(C)C C1(C)(C(c2nc(CC(C)(C)C)cs2)C)CCN(C(=O)OC(C23CC(C#N)(C2)C3)=O)C1 N1(C(C2(C)C(C)(C)C2)=O)CC(C2CCN(C(C3CCCC34CCC4)=O)CC2)C1 CC(CCNC(c1cnoc1C1CC1)=O)CCNC(c1cccnc1)=O C(CC(C)(C)NC(=O)CCN1CCCC1)=CC(=O)NC1(CC(C)C)CCC1 c1(C(N(C)CC2(O)CN(C(Cc3c(C)cccc3)=O)C2)=O)cccc(Cl)c1F c1(OC)ccc(Cl)c(C(=O)OCCN(C)C(c2cnc(Cl)s2)=O)n1 C1(C(C)(C)CNC(=O)Cc2cccnc2)CCCCN1C(c1ccnc(O)c1)=O c1(C(=O)NC2CCN(C(CCC3CCC(=O)NC3)=O)C2)cc2[nH]ccc2cc1Cl CC1(C(=O)NC2CN(C(c3cnc(-c4cccs4)o3)=O)C2)CCCCC1(F)F C1(OCCN(C(c2ccc(CC)cc2)C(=O)NCCOCC)C)CCC(F)(F)CC1 c1(C(=O)NCCOCCCNC(C(C)CNC(N)=O)=O)ncnc2c1CCCC2 C1(C(=O)NCC(=O)NC(C#C)(C)C2CCCC2)CCC=CCCC1 c1(OC)cccc(NC(C2CC2NC(c2cc(Br)cc(F)c2O)=O)=O)c1C#N c1(N(C)CC2CCCN(C(=O)CC3CC3C3CC3)C2)ccc2ncnn2c1 N1(C(C(CC)C#N)=O)CC2OCCN(C(c3cccs3)=O)C2C1 C(=O)(CP(C)(C)=O)N1C(Cc2cn(CC(C)O)nn2)CCC1 O=C(CCCCC1CCC1)N(c1ccccc1)C(CCO)c1nn[nH]n1 N1(C(C(C=C)O)=O)CC(OC)C(NC(=O)Cc2csc(-c3cccnc3)n2)C1 N1(C(c2cn(CC=C)nn2)=O)CC2CC1CN(C(=O)CCn1c(C)csc1=O)C2 C(CCCOC)(C(=O)NC(c1cscn1)CO)NC(C(C(=O)OC)OC)=O C1(NC(=O)NCC2CCCOCC2)CC12CCOCC2 Cc1cc(=NC(=O)C(=O)N2Cc3ccccc3CC2CN)[nH]o1 CCC(C)C(O)C(=O)NCC1=CCN(S(=O)(=O)CC2CCOC2)CC1 c1(CN2CC(NC(C3C(CC)CCCC3)=O)C2)ccc(Br)c(Cl)c1 N1(C(C(CCOC)N(C)C)=O)CC2(CC(C(=O)N(CCS(C)(=O)=O)C)CO2)C1 C1(C(=O)NCc2c(Br)ccc(OC)n2)CC12CCN(Cc1cc(C)cc(C)c1)CC2 c1(C(C)C(=O)NC2CCCC2NC(C2CC(O)C2)=O)ccccc1[N+](=O)[O-] C1(NC(CC(=C=C)C)=O)CCN(C(=O)C(C)NC(C)=O)CC(C)(C)C1 N1(C(CN(C)C)=O)CCC2(CCC(NC(=O)COC3CCN(C)CC3)C2)CC1 C1(C(=O)NC2C(CN(C(c3nc(OCC)oc3)=O)CC)CC2)CCN(C)S1(=O)=O C1(C(=O)Nc2c(C)cc(O)nc2)C2CCCC2CN1C(c1ccc(Cl)s1)=O CCCCS(=O)(=O)CC(=O)NC(CNC(=O)C(C)C(C)(C)C)CO C(=O)(C1=CCCC1(C)C)N(C1CCCC(N(C)C(c2ccc(Cl)cc2)=O)C1)C c1(-c2cn(CC(N3CC(CCOC)C3)=O)nn2)ccccc1OCCN(C)C C1(NC(C2CC(=O)N2)=O)CCN(Cc2cn(-c3nccs3)nn2)CC1 N1(C(CN(CCOCC)C)=O)C2CCC1CN(CC1(OCC)CCSCC1)CC2 Cc1ccc(F)c(N(C)C(c2c(C(F)(F)F)coc2C(C)C)=O)c1 C(=O)(C(C)CC(=O)NCC1CC1CC(=O)NCCC1(CO)CC1)OC N1(C(C(C=C)OC)=O)CC(C2CCCN(C(c3[nH]nnc3CC)=O)C2)C1 C1(C)(C(N2CCCC(C(C)NCc3ccccc3)C2)=O)CCNC(=O)C1 c1(C(N(CC(CC)NC(c2cnnn2C)=O)C)=O)nc(Cl)c(Cl)s1 C1(C(=O)NCC(C)CNC(c2cc(C(F)(F)F)n[nH]2)=O)C(F)(F)C12CC2 N1(C(CCCCC)=O)CC(CNC(=O)CSCc2cccs2)C2(CCC2)C1 C1(C(N(C2CCN(C(C3CCN(c4ccccc4)C3)=O)C2)C)=O)CC2(CCC2)C1 c1(C(N2CCC(CC=C)(NC(C3CCSC3)=O)C2)=O)c(C)nc(C2CC2)nc1O c12nc(ncc1F)NC(=O)N2.N1(C(=O)OC(C)(C)C)CCOCC1Cc1ccco1 N1(C(CC(CCC)C)=O)CCC2CN(C(c3sc(C)cc3C)=O)C2C1 CC(C)CCC(=O)C(=O)NC1(C)CC(C(=O)N(C)Cc2cnn[nH]2)C1 C1(CNC(c2c(C)ccnn2)=O)CCCCN(C(c2cccc(C(N)=O)n2)=O)C1 CC1CN(C(=O)C(Cn2ccnn2)NC(=O)Cc2csnn2)CCC1N(C)C c1(CN(C(=O)NC23CC(C2)C3)Cc2ccc(OC)nc2)ccc(C#N)cc1C C1(NC(CNC(CC(C)C)=O)=O)CCC(NC(=O)C(N2CCCC2)C2CC2)CC1 c1(C(N2C(C(C)(C)NC(C3OCC(C)C3)=O)CCC2)=O)cn(C)ccc1=O N1(C(C(C)CCO)=O)CCCC12CCN(C(=O)C(C)NC(N)=O)CC2 N1(C(C2(F)C(C)C2)=O)CCc2nc(CNC(=O)Cc3ccc(O)cn3)sc2C1 N1(C(=O)C(F)(F)C(O)C2CC2)C2CCCC1CC(Nc1cc(C3CC3)ncn1)C2 Cc1cc(C(=O)N(C2CCC(NC(c3nn[nH]c3Cl)=O)CC2)C)cc([N+](=O)[O-])c1 C#Cc1cncc(C(=O)NC(C)(C(=O)NCc2ccc(OC)o2)C2CCC2)c1 c1(N(C)CC2CCN(C(C3CCOCC3)=O)C2)nc2ccc(O)cc2s1 C1(CC)C(=O)O1.C(C(=O)NCCF)N(C(=O)C=CC(=O)N(C)C)CC#C c1(C(C(=O)NCC2CCCO2)N(CC(C)(C)C)CC)cc(C)c(Cl)s1 n1(CC)cc(C(N2CC3C(CNC(C4(C)CC(=O)N(C)C4)=O)C3C2)=O)c(C(C)C)n1 N=c1nc(N2CCN(C(=O)C3=CCCS3)CC2)[nH]c(=NC2CCCC(C(N)=O)C2)[nH]1 Cc1noc(C)c1-c1cncc(F)c1.c12ccc(cc1)c1ccc(cc1)[nH]c2=O CC(C(C)(C)C(=O)N(C)CCC1CCCO1)NC(=O)CNC(=O)NCCO C1(NC(C(C)SC)=O)CC2CCC(C1)N2C(c1c(C(F)(F)F)coc1C)=O c1(CNC(c2cc(C)n(C)c2)=O)n[nH]c2c1CN(C(C1CC1C(N)=O)=O)CC2 C1(NC(C(CCN(C(=O)CP(C)(C)=O)C)O)=O)CC(C)(C)C12CC2 Cc1cc(C(=O)NCC(O)CCNC(=O)Cn2cccn2)c(F)c(Br)c1 C#Cc1ccccc1NC(c1ccc(NC2CCC2O)nc1)=O C1(C(N(CCNC(C(=O)NCCNC(C)=O)=O)C)=O)Cc2cncn2C(=O)N1 C1(CC(=O)NCCN(C(c2cnc(S)[nH]2)=O)CC2CC2)CCC=N1 Cc1cc2ncnc(N3C4CCC3C(C)C(NC(C3CC5CCC3C5)=O)C4)c2[nH]1 C1(CN(C(C2(CC#C)CCC2)=O)C)CCCN1C(=O)COC1(C)CC1 C1(NC(C2(C)CC(F)(F)C2)=O)C2CC1CN(C(=O)C(=Cc1c[nH]cn1)F)C2 N1(C(CC(CC)NC(c2cc(F)cc(Cl)c2N)=O)=O)CC2CCCN2CC1C C=CCC(F)(F)C(=O)NC1CCN(Cc2nnc(C(C)(C)C)o2)C1 C(=O)(C1=NN(C)C(=O)CC1)N1CC2CCC(NC(C(CCOC)(C)C)=O)(C1)C2 CC1(C(=O)NCC2CC3C=CC2O3)CCN(C(=O)C(C2CCOCC2)=O)C1 c1(C(=O)NCCOCCCNC(C2(C(N)=O)CC2)=O)ccnc(CO)c1 Cc1nn(C)c(C)c1OCC(=O)NCC(O)CCNC(c1csc(S)n1)=O C1(C(N(CC(O)C2CC2)C)=O)COCCN1C(c1cnn[nH]1)=O C1(CC#C)CCCN(C(c2cc(Br)co2)C(=O)NCc2ccccc2Cl)CC1 c1(C(N(C(C)CNC(c2ccco2)=O)C)=O)cccc(Cl)c1O C(=O)(NNC(=O)COC(c1ccccc1)=O)c1c(C)cco1 C1(C(=O)NCC(CCCC)NC(=O)CN2CC3CCC2C3)CC2CCCCCC12 c1(C(=O)NC(CN(C(CCC2CC(OC)C2)=O)C)(C)C)cnn2c(N)ccnc12 N1(C(C(C)OCC(C)(C)C2CCCO2)=O)CCCCC1C1CCN(CCF)C1 Cc1ccc2ncc(C(N3CC(N(C)Cc4cnc(Cl)cc4Br)C3)=O)n2c1 C#Cc1cncc(C(=O)NC2(CNC(C3(C#N)CCCC3)=O)CCC2)c1 C1(CC(=O)NC2CC(NC(C(c3cccc(Cl)c3)CC)=O)C2)CCC(C)(C)C1 C(=O)(CCC(=O)N1CCC(C(=O)NCC2(C(=O)N(C)C)CC=CC2)C1)NCC c1(C(N2CCC(N(c3ncncc3F)C)C2)=O)ccc(Cl)cc1 c1(C(N(CCN(C(c2c[nH]c(Br)c2)=O)CC)CC)=O)cc(O)n(CC)n1 c1(C(N2CC(F)(F)C2)=O)cnn2c1CN(C(c1c(Br)ccc(F)c1F)=O)CC2 CCCCC(O)C(C)C(=O)N1CCC(C2CCCN2C(c2nccnc2C)=O)C1 c1(C(=O)NC(c2cn(C(CC=C)CC)nn2)CC(N)=O)nnccc1C C1(C(=O)NCCN(C(C2CC(CCC)C2)=O)CCOC)CC(C)(C)CO1 N1(C(CSCCCC)=O)CCCC(C(=O)N(C(C)CCO)C)CC1 N1(C(C(CC=CC)C)=O)CCCCCC(NC(=O)Cc2cccnc2Br)C1 C1(O)(CS(=O)(=O)NC2(CC)CC(C)C2)CCOCC1 C1(C(N2C(CCNC(C(C)(C)C3CCC3)=O)CSCC2)=O)CC2(COCCO2)C1 CC(CC(C)(C)C)C(=O)NC(CO)C(C)NC(C1CCC(N(C)C)CC1)=O CCCC(C)CCNC(=O)COC1CCN(C(=O)CC2CCOC2)C1 C1(C(F)(F)F)(C(N(CCCCNC(=O)C(C)(C)CN(C)C)C)=O)CC2(CCC2)C1 c1(C(C(=O)NC2COC2)N(C)Cc2c(CCC)cccc2)cc(Cl)cc(Cl)c1 C1(C(=O)NC2(CC(=O)NC(c3c(C)ncs3)C)CCC2)CC(=O)CC(=O)N1 c1(C(N(CCC(=O)N(CCCCC)C)CC2CC2)=O)csc(=N)[nH]1 c1(C(C(=O)NCC(C)C)OC)ccc2c(c1)CCN(CC1CCCC13CC3)C2C CC(C(C)C(=O)Nc1cccc(C2CC2)c1)NC(=O)C=Cc1cccnc1 CC(C)(C)CC(F)C(=O)NC1(CCCC(=O)NC2CCOC2=O)CCC1 N1(C(C2(COC)COC2)=O)CCOC(C(=O)N(C2CCCNC2=O)C)CC1 c1(N2CC=CC(NC(C3CCC(CC)O3)=O)C2)nn2cc(C)nc2s1 C1(NC(CCOCC(C)C)=O)CCN(C(C2CCS(=O)(=O)N2)=O)CC(C)(C)C1 C1(C(=O)NCC2N(C(c3c(C)c(F)ccc3)=O)CCC2C)C2CCC1(C)C2(C)C CC1(C)CC(NC(=O)Cc2ccccc2[N+](=O)[O-])CN(C(=O)C=CC(F)F)C1 S(=O)(=O)(c1ccsc1C(=O)NCCCCNC(=O)C(C)CC(C)C)NC C1(NC(c2cccc(NC(C(C)C)=O)c2)=O)CC2(C1)CN(C(C1CCC(=O)O1)=O)C2 C1(CNC(CCCC)=O)CC(OC)CN1C(c1ccnc(SCC)c1)=O c1(C(N2CC(NC(C(CCC)CC)=O)C(O)C2)=O)ccc2ncn(C3CC3)c2c1 c1(-c2onc(C)n2)cc(C(N2CCOCC2c2ccc(C)cc2)=O)ccc1F c1(-c2nc(NC(C(C3CCC3)OC)=O)sc2)ccc(C)cc1 Cc1cc(NC(C2CCCCNC2=O)=O)nc(Br)c1 C1(NC(c2ccc(CCC)[nH]2)=O)CN(C(=O)CCN(C)CC)Cc2nccn2C1 C1(CC(=O)NC(C)(C)CF)CCCN1C(=O)CC1CCC1 C(=O)(C1=CC2(CCOCC2)C1)NC(C)(CNC(C1(C2CC2)CCC1)=O)CO c1(N2CCCC(C)C2)cccc(S(=O)(=O)N2CCCC2C2CN(C)CC2O)n1 N1(CC)CC(C)N(C(c2[nH]ccc2CNC(=O)C=CCOC)=O)CC1C N1(C(CCC2CCN(C(C3(OC)CCOC3)=O)CC2)=O)CCC2C(C(N)=O)C2C1 c1(OC)cccc(F)c1CN1CCOC(CC(=O)Nc2cnc[nH]2)C1 C1(NC(C(CCN(C)C)N(C)C)=O)CC2CCC1CN2C(C1CC(F)(CF)C1)=O N1(C(CCCOC)=O)CC(OC)C(NC(=O)CSc2nncs2)C1 c1(C(N(CCNC(C(C)(C(C)C)NC(C)=O)=O)C)=O)oc(S(N)(=O)=O)cc1C c1(NC2CC(CNC(c3c(C)nc(CC(C)C)o3)=O)C2)cc(C)nc2ncnn12 C1(SCCNC(=O)C=CCO)C2CN(C(c3ccnc(OC(F)F)c3)=O)CC12 C(=O)(C(CCF)NC(=O)CCNC(c1ccco1)=O)NC(C(=O)NC(C)C)C N1(C(c2scc(COCC)c2)C(=O)NCC2CCOCC2)CCCOCC1 N1(Cc2cc(CC)sc2)CC2CC1CN2C(=O)C(C)O c1(NC(C(C)c2ccco2)=O)cccc(NC(=O)NCCSc2ccncc2)c1 CCCC(C)CN(C)C(c1cc(CNC(C2CC(C)(O)C2)=O)[nH]n1)=O c1(OCC(N2CC(O)(C(C)NC(C(C(C)C)C)=O)C2)=O)cc(F)ccc1F CCCCCCC(F)C(=O)NC(C)CNC(c1sc(CC)nc1C)=O n1(CC(=O)NC(C)CCNC(=O)CC2CC2(Cl)Cl)ncc(C#N)c1N c1(CNC(=O)NC2C(NC(C=CCC)=O)COC2)cnc2sccn12.C(C)(C)(C)O N#Cc1cccc(F)c1CC(N1CC(NC(C2CCCO2)=O)CC(F)C1)=O n1(CCC)nnnc1C(c1cnc(C2CC2)o1)NC1CC(CSc2cccs2)C1 S(=O)(=O)(c1ccc(NC2CCCCC2OC(F)(F)F)nc1)NCC(C)C(F)F c1(OC)ccc2c(c1)CO2.C123CC(C1)(C2)CN3.C(=O)(CCF)OC(C)(C)C Cc1ccc(NC2CCOC(c3ccccc3)C2)nc1 Cc1cc(C(=O)NCC(C)N(C(=O)C2=COCC2)C)sc1-c1ccc(Cl)cc1 C1(NC(C(C)O)=O)CCC2(CCN(C(c3cnsc3)=O)CC2)C1 C=C1Cn2c(C(=O)NC3CCCC(NC(C4CC(O)(C#N)C4)=O)C3)nnc2S1 C1(C(=O)NC2CCN(C(COCC=C)=O)C2C(C)(C)C)CC12CCC(C)(C)CC2 C1(C(N(CCC)C)=O)CCC(C(C)C)N1S(=O)(=O)N=S(C)(=O)CC CCC(CC(=O)N1CCC1C1CCOCC1)NC(c1cc(C#N)cs1)=O c1(C(=O)NCC2CC3CN(C(C4C(=C)C4)=O)CC32)coc(S(=O)(=O)NC2CC2)c1 C1(C(=O)NC(C)CCNC(c2nc(Cl)ccc2N)=O)CN2CCCN1CC2 N1(C(Cc2c(C)nc[nH]2)=O)CC2CC(NC(=O)CCn3cnnn3)CC1C2 N(C1c2ccccc2CC1C)C(c1ccc(OC)nc1Br)=O C(c1ccccc1F)=CC(=O)NCCCN(C)C(c1cn(C)nn1)=O C1(CSC)CCCN(C(c2cc(CO)on2)=O)CC1.CCC(C)N1CC(=O)N1 N1(C(Cc2c(C)ccs2)=O)CCN(C(=O)COC2CCOC2)C(C2CC2)C1 C1(N(C(c2cnc(Br)n2C)C(=O)NCC2CC2)C)CCCCC1C(N)=O c1(C(=O)NC(C2CCCN2C(=O)CC2CCC(O)C2)C)ccc(C#N)s1 Cc1cc(C(=O)NCC2(COC(C)(C)C)CN(C(=O)C3CC3)C2)c2occc2c1 C12(C(=O)NC3CCC(NC(C4CC(C5CCC5)C4)=O)C3)CC(CO)(C1)OC21COC1 C=C(C)CCCC(=O)NC1C2CN(C(C3CCOC3)=O)CC12 Nc1cncnc1C(=O)NCC1(CO)CCN(C(=O)CN2CCNC(=O)C2)C1 c1(C(N2CC(CO)C3(CC3)C2)C(=O)NC(C)(C)C)ccc2ncccc2n1 N1(C(c2ccnn2CC(F)F)C(=O)NCCOC)CCC12CCN(C)C2 CC(C(=O)NCCOCCNC(=O)CCNc1cccs1)N(C)C CN1CCCC1(C)C(N1CC2C(c3cn(-c4cncc(OCCF)c4)nn3)C2C1)=O c1(OC)ncc(C(=O)NCCN(C(=O)C(O)CCSC)C)c(C(F)F)n1 C1(C(N(CCC)CCNC(=O)C(F)C2CCC2)=O)CC(C(=O)OC(C)(C)C)=NO1 N1(C(C(C)O)=O)CCC2CN(C(c3cncc(C4(N(C)C)CCOCC4)c3)=O)C2C1 C1(CC)CCCN(C(=O)CN2CCOCC2)C1C(=O)N(C)Cc1ccccc1C C12CCCCC1C(=O)N2C.C(C(F)(F)F)SC Cc1nc([N+](=O)[O-])cn1CC(=O)NCC1CC1NC(=O)C(C)(C)n1cccn1 CC1CN(C(c2ncsc2C(F)(F)F)=O)CCC1NC(=O)CN(C)C c1(CN2CCCC(N(S(=O)(=O)CC3CC3)C)C2)cc([N+](=O)[O-])c(O)cc1O c1(CCC(=O)NC(C2CCOC2)CNC(C=C(CC)CC)=O)nc(CC2CC2)no1 C(=O)(C(CCOC)SC)NCC1(C(=O)N(c2ccccc2)C)CC(=C)C1 c1(CC)cc(C)ccc1NC(C1C(C)CCN1C(c1cnc(C)nc1)=O)=O N1(C(C(C)SC(F)(F)F)=O)CC(CNC(c2nccn2C(C)C)=O)C2(CCC2)C1 CC(N=c1[nH]nc(C(F)(F)F)s1)C1CCCN(C(C2CC2(F)F)=O)C1 C1(CNC(C(CCC)CC)=O)CCC2(CC1)CC(NC(=O)Cc1ccccc1)C2 c1(OCC=C)ccc([N+](=O)[O-])c(C(=O)NC(CNC(=O)OC)CC)c1 C1(NC(c2c(C)c[nH]n2)=O)C2CC(NC(C3CC(N(C)C)C3)=O)CC12 c1(C(=O)NC2CC(NC(C3C(C)C3)=O)C2)ccc(CO)cc1F.C1(=O)CCN1 C(=O)(C(CCC(C)C)NC(=O)CC1CCSC1)NCCOCC C1(NC(C2(CC#C)CC2)=O)CN(C(C2CCOC(C(=O)OC)C2)=O)CC(C)(C)C1 C1(CNC(c2nn[nH]c2Cl)=O)CN(C(=O)Cc2cnsc2)CCO1 C1(C(=O)NCCOC)CCN(C(c2cc(OC)cs2)=O)C1C(C)C c1(C(C(N2CC(CCNC(=O)CCS(C)=O)(OC)C2)=O)(F)F)cccc(F)c1F N1(C(C2C(=C)C2)=O)CC(CO)C2(C1)CN(C(c1cn3ccncc3n1)=O)C2 Cc1cc(F)c(N)cc1C(=O)NC(C(C)NC(c1ccc(Cl)c(F)c1)=O)C(C)C c1(N(C(CNC(C=CCC)=O)=O)CC(C)C)nnc(N(C)C)o1 C1(CNC(C)=O)CCCCN1C(=O)CC1CCCC(C2CC2)O1 C1(C)(NC(CCNC(=O)NC)=O)CCN(C(C2CCCCC2)=O)CC1 c1(C(N2CC(C)(C(N3CCC4CC34)=O)C2)=O)cccn2nnnc12 n1(CC=C)c(=O)[nH]c(C2CCC(C)O2)c1C(=O)OC.c12ccc(c(F)c1)NC(=O)N2 c1(CC)ccc(C(=O)N(CCCNC(=O)CNC=O)CC2CCC2)cn1 C(=O)(CC1=Cc2ccccc2C1)N1CC2(OCC(NC(C3=CC(C)(C)C3)=O)C2)C1 Cn1cc(C(=O)NCC2CCN(C(=O)Cc3cnnn3C)CC2)c(O)nc1=O C(=O)(C(C)(C)COCC)NCC1(CC(=O)N(CCCCC=C)C)CC1 C(=O)(C(C)(C)CS(C)(=O)=O)N1CC(N(C(C(CSC)OC)=O)C)C2(C1)CC2 S(=O)(=O)(c1ccc(NCc2ccc(F)cc2Cl)nc1)NCC1C(C)(C)OCCO1 S(=O)(=O)(c1ccc(F)c(F)c1)NC12CC(NC(c3cc(C(F)(F)F)c[nH]3)=O)(C1)C2 C12(NC(c3cccc(F)n3)=O)CCC(C1)N(C(C1CC1(Cl)Cl)=O)C2 CCC(C(=O)NCC1CCCCN1C(c1cc(F)ccc1F)=O)C(C)O c1(C(=O)NCC(C)SC)cc(=NC(=O)CNC(=O)C(C)(C)C)[nH]n1C N1(C(C(C(CC)O)(F)F)=O)Cc2ccccc2C(CNC(C2(O)CCOC2)=O)C1 c1(C(=O)NC2C(NC(CCSc3ccccc3)=O)C2)ccc(SC(F)(F)F)nc1 c1(C)ccc2cccc(F)c2n1.c1(NC(c2sccc2N)=O)c(F)cc(Cl)cc1F c1(C(N2CCC(CCNC(CC(C=C)C)=O)CC2)=O)ccc(C(F)F)c(OC)c1 c1(C(C(=O)CCCCN2CCCCC2)=O)cnc2n(c1=O)CCS2.C1(N)CNC1 N1(C(C(C2CCN(C(c3c(C)occ3)=O)C2)C)=O)CCC(C#N)CC1 CC(C)C1C(=O)N1.C12(NC(=O)C(C)C#N)CC(C(=O)OC(C)(C)C)(C1)C2 c1(NC(C(CC#C)NC(=O)CSCC(N)=O)=O)cc(C)ccc1F c1(CC(C(N2C(CNC(C(C)=C(CC)C)=O)CCC2)=O)C)cccc(Cl)c1 C1(C(=O)NCC2N(C(C3C(C)CC3)=O)CCC2)CC(C)(C)CO1 C1(NC(CN(C)C(N)=O)=O)CCCC2CN(C(=O)CCn3ccnn3)CC12 N1(C(C(C(CC)C)O)=O)CC2CCC1C(NC(c1[nH]ccc1C)=O)C2 CCC(C)CCCCC(=O)NC1CCC(CNC(c2cncc(CO)c2)=O)CC1 CCCC(C(=O)N1CCN(C(=O)C=Cc2ccco2)CC1)OC CC1=C(C(=O)N2CCC(NC(C3CCS(=O)CC3)=O)C(C(C)C)C2)CCC1 C=CCCC(C(=O)NCCC(C)CCO)NC(=O)CCC(CC)OC c1(NCC(CCCC)NC(=O)CC2(CSC(C)C)CC2)nc(C)nc2c(C)csc12 Cn1c(C(=O)NCC2CC2NC(=O)CCc2ccc[nH]2)nnc1S CC1(C)CN(C(C2CC2c2cncs2)=O)CCC1C(N1CC(C)(O)C1)=O N1(C(CCCNC(C)=O)=O)CCC(C)C(NC(=O)C(C)Cc2ccco2)C1 c1(C(N2CC(CC(C(=O)C(c3ccc(F)s3)=O)F)C2)=O)ccc(CO)s1.NC N1(C(c2c(C)cc(F)cc2)=O)CC2CCCC2(NC(=O)Cc2cncn2C)C1 CC1(C)CC1(C)CNC(c1csc(O)n1)c1nnnn1C(C)(C)C C1(CNC(CCCCC)=O)CN(C(C2CC2C(=O)NC)=O)C2(CCC2)C1 c1(CC)ncc(C(=O)N(CC(C)NC(c2nc(=O)cc(N)[nH]2)=O)C)c(C)n1 N1(C(CC2(C=C)CN(C(=O)CC(Cl)Cl)C2)=O)CCOCC(O)C1 c1(CC(N2CCC3(N(C(C(N)=O)=O)CCC3)C2)=O)c[nH]c2cc(F)c(F)cc12 C1(NC(CCCN(C(C)=O)C)=O)CC2CCC1(NC(c1cc(C)n(C)n1)=O)C2 N1(c2n(CC(=C)C)c(-c3cc(O)nn3C)nn2)CC(C)OC2(CCCOC2)C1 CS(C)(=O)=Nc1ccc(C(=O)NCCCN(C(c2sccc2C#N)=O)C2CC2)cc1 c1(C(=O)NC2(CNC(C3(C)CCC(C)C3)=O)CCCC2)ccc(P(C)(C)=O)cc1 c1(C(N(CC(C)NC(=O)C(O)C(C)c2ccccc2F)C)=O)ccc(F)cc1N N1(C(C(C)CCNC(N)=O)=O)CC2(c3ccccc3)CC2(c2ccccc2)C1 C(=O)(C(C)(C)CCCNC(=O)NC)NCCNC(C(CC#C)C)=O c1(C(=O)NC(C(C)NC(CC(C)(C)OC)=O)(C)C)cnc2sc(C)cn12 Cn1cc([N+](=O)[O-])cc1C(N1CC2CCC(C1)C2NC(c1cscn1)=O)=O c1(NC(=O)OC)ccc(C(=O)NC(C)(CNC(C2CC2C(F)(F)F)=O)CO)cc1 C(CC(C)CC)(C(=O)N(C)CCN(C)C1CC1)NC(CCC=C=C)=O c1(C(N2C(C(=O)NCC(=O)OC)CCC2)C(=O)OC)c(Cl)c(C)nn1C Cc1ccc(NC(C2CCOC2CNC(c2nonc2N)=O)=O)c(C)c1O CCCC(C)NC(=O)CSC.CCC(C)(c1nccs1)NC(=O)O N1(C(C(C)SCCCC)=O)CCCC(NCCNC(c2coc(C(F)F)c2)=O)C1 Cc1ccc2c(CC(=O)NC3CCCN(c4ccccc4)C3)cc(=O)oc2c1 C(=O)(CC(C)CC(F)(F)F)N1C(C)(COC)CC(NC(=O)CCC2CC2)C1 C1(C(=O)NCc2sccc2Cl)CCCN(C(=O)CCc2nncs2)CC1 c1(C(N(CC(C)NC(=O)C(C)S(C)(=O)=O)CC)=O)nn2cccnc2c1Cl C=C(Cl)C(C)(C)C(=O)NCC1(CO)CCN(C(=O)Cc2ccn(CC(C)C)n2)C1 c1(CN(C(=O)C(C)C(=O)O)C(CC)C)nc(O)c2c(C)c(C)sc2n1 N1(C(CCOCCNC(c2ccc(C(C)=O)[nH]2)=O)=O)CCOCCC1C1CC1 C1(C(=O)NC(CC)COC(C)C)CN(CC2(C(=O)NC(C)(C)C)CC2)CC12CCC2 C1(CCCCNC(C(C)c2ccsc2)=O)CCN(C(=O)C=Cc2cn[nH]c2)CC1 C(c1ccc2c(c1)OCO2)=CC(=O)NCC1CCN(C(C2(F)CCOC2)=O)C1 c1(OCC)nccc(C(=O)NCCCN(C(=O)CCc2cnn[nH]2)C(C)C)c1F c1(OC)cccc(C(N2CCN(C(=O)C(CO)C(C)C)CC2C(C)C)=O)c1F CCC(CN1CCC1)N=c1cccc(S(=O)(=O)NC(c2cccc(F)c2)CF)[nH]1 C(=O)(C1=C(C)CCCC1(C)C)NCc1cn(CC(C)NC(C(CCC)C)=O)nn1 N1(C(c2c(C)cncc2)=O)CCN(C(c2cnn(CC3CCCC3)c2)=O)C2CC12 O=S(=O)(c1cccs1)NCC1(O)CCCN(Cc2cc(Cl)ccc2Cl)C1 N1(C(C2CC2F)=O)CCN(C(=O)CC2(CO)CCCC2)C(c2ccc(Cl)cc2)C1 c1(C(N(CCNC(C(n2ccc(C(F)(F)F)n2)C)=O)C)=O)ccc(S(C)(=O)=O)o1 C1(C)(CNC(C)=O)CN(C(C2(c3cc[nH]n3)CC2)=O)CC1C.C1(C)(CO)C(=O)N1 Cc1cc(Br)cc(C)c1C(=O)NCC1CC(NC(=O)Nc2cccc(Cl)c2Cl)C1 Cc1nc(NC2CC23CC(NC(=O)C(N2CCSCC2)C)C3)ccc1[N+](=O)[O-] Cc1nnc2n1CCCC2C(=O)Nc1cnc2n1CCS2 N1(C(c2c(C)nc(SC(F)(F)F)s2)=O)CCN(C(C2CC3CC3C2)=O)CC(O)C1 N1(C(C2CN(C(C)=O)C2)=O)CCC(C)C1CNCc1ccc(N2CCCC2)nc1 CC1C(NC(c2ccc(-c3ccccn3)nc2)=O)CCN1c1nnc(C#N)s1 c1(SCC(=O)N(CC(=O)NCCC(C)NC(c2cscn2)=O)C)ccccn1 C(=O)(C1CCc2c[nH]nc21)N(CC(=O)NCCSC1CCOC1)C(C)C C(=O)(C(C)(C)CN(C(=O)Cc1ccnn1C)C)NCCC1CC(C)C1 c1(C(=O)NCC(C2CCCC2)NC(=O)CC2(O)CCOC2)cc(Cl)c(Cl)s1 c1(C(N2CC(C(=O)OC(C)(C)C)OCC2)=O)cccc2c1COC2 c1(C(N(CCC)CCNC(=O)CCCc2ncc(C)o2)=O)ccc(C)c(F)c1F c1(C(N2CC(C=C)C(NC(=O)CCc3cnc[nH]3)C2)=O)cncc2[nH]ccc12 Cc1cccc(C)c1C(=O)NCC12CCC(C1)N(C(=O)C=C1CCC(C)CC1)C2 CN1CC2(CCN(C(=O)CC3C4CN(C(=O)C(C)(C)CO)CC34)CC2)C1 C(=O)(CC(C)(C)CC(F)F)N1C2CC(CNC(C(C)OCCCC)=O)C1CC2 C1(NC(c2cnc3ncccn23)=O)CCC2CN(c3nnc(C(F)F)s3)CC2C1 Cc1cc(=NC(=O)C(=O)NC2CC23CC(NC(=O)Cc2ccc(F)cn2)C3)[nH]o1 CC1(O)CON(C(=O)C(CNC(=O)C=Cc2ccc(C(F)F)o2)CC2CC2)C1 c1(COC)cc(C(=O)NC2CCN(C(=O)C(Cc3ccccc3)OC)C2)c(C)o1 Nc1c(F)ccc(Cl)c1C(N1CCOCC(CNC(=O)C=CC(N)=O)C1)=O C1(C(=O)NCC(C(=O)NCCNS(CC)(=O)=O)O)CCC(=O)CC1 C12CCCCC1(C1CC1)CC1(NC(C(COCC)C)=O)CC(C)(C1)C(=O)N2 C1(C2(C)CC2)(C(N(CCCCNC(C(CC2CCC2)OC)=O)C)=O)CC1 c1(C(=O)NC(CNC(C(CC)(C)O)=O)CC(C)C)c(C)cc(=O)oc1C c1(C(=O)NCC(CNC(c2coc(-c3cnn(C)c3)n2)=O)OC)cnc(C)[nH]1 C12(C(N(CC(=C)C)C)=O)CCN(C(=O)CC=C(C)C)CCC1C2 C=CC(CC)CC(=O)NC1C2CC1CN(C(C13CC(OC)C1C3)=O)C2 CN=c1[nH]cc(C(=O)NCCOC2CCN(C(=O)C3=NOCC3)C2)s1 CCCCS(=O)(=O)CC(=O)NC1CC1CNC(c1cc(OC)n(C)n1)=O C1(C(=O)NC2CN(C(CCC(=O)NCCC)=O)CC2C(F)F)CCC(=O)N(C)C1 c1(C(=O)NCC2CCCO2)c(NCc2cc(Cl)cc(I)c2)cccc1F C=CCC(CC=C)C(=O)N1CCC(NC(=O)CCCF)C(CO)C1 C(Cn1cccn1)(C(=O)Nn1cnnc1C)NC(c1[nH]cc(C)c1)=O N1(C(CC(=O)NCC)=O)CCC(C)C(NC(c2sccc2CO)=O)C1C Cc1ccc2oc(C(=O)NC(C)(C)CCNC(=O)CN3CC4CC4C3)cc2n1 N1(CCCN(CCNC(=O)CNC(c2cccnc2)=O)C2CC2)CCCC1=O N1(Cc2cc(NC(c3ccc(F)cc3F)C)ncn2)CCOCC(N)C1 CC12COC(C(=O)NCC3(O)CN(C(=O)CCCn4cncn4)C3)(C1)C2 c1(OCC)cccc2c1OC(C)(C)CN(c1nsc(N(C)C)n1)C2 C(=O)(CCS(=O)(=O)NC)NCCC1CC(NC(C=NOC)=O)C1 c1(CO)cc(=NCC2CC3CCCC3O2)[nH]cn1 c1(NC(C2C(C(=O)NCC3(CO)CC3)C2)=O)cnccc1C(F)(F)F c1(CC)nccn1C(C)CC(=O)NCC1CC(NC(=O)CC2(O)CCCC2)C1 c1(C(N2CC(CC(C)NC(=O)CC(O)C(C)C)C2)=O)ccc2cnccc2n1 C1(C(N2C(NC(CC(C(=O)OC)C)=O)CC2)=O)CC(C)(C)OC1(C)C c1(C(=O)NC(CN(C(c2ccc3nccn3c2)=O)CC)C)cc(F)c(N)cc1F Cc1nn2cccnc2c1C(=O)NC(CO)C(C)NC(=O)CN1CCCOC1=O C1(CNC(c2c(N(C)C)cccc2)=O)CCCN(C(=O)C2=CCCS2)CC1 CC1(C)C(C(N2CCCSCC2)=O)CCN1C(c1ncc(F)cc1F)=O N1(C(C(CC)(C)C)=O)CCN(C(c2ccc(C)c(C)n2)=O)C2(CCC2)C1 Cc1cc(CC(=O)OCC(=O)C(C)(C)C)cc(C)c1 C1(N2CCCC(c3nn(CC)c(C4(C)CCNC(=O)C4)n3)C2)CCC(=O)NC1=O C1(C(N(CCNC(C(c2ccc(C)cc2)F)=O)C2CC2)=O)CCOC(=O)CC1 Cc1c(C(=O)NC2(CNC(c3c(C(F)(F)F)cnn3C)=O)CCOC2)ncn1C N1(C(c2nc(C)nn2C)=O)CCC2(NC(=O)C(C)OCC(C)C)CCCC12 C(=O)(C1=C(C)OCCC1)N1CC(COC)(NC(c2sccc2Cl)=O)C1 N1(C(CCc2n(C)ccc2)=O)CCC2CCC(C1)N2C(C1(C)CC1(F)F)=O c1(C(=O)NC(C(C)(C)C)CNC(c2cncs2)=O)cc2cc(N)ccc2o1 C12CC(C(C(=O)CC3CC4(CC4)C3)=O)N(C1)C(=O)C(CC)N2.CCN.OCC c1(N2CCC(C(N3CCCCC(O)C3)=O)C2)cc(F)ccc1Br N1(C(C2(C)CCC2)=O)CCC(N(C(=O)Cn2nnc(-c3ccc(Cl)s3)n2)CCO)C1 C1(CC#C)(C(=O)NC2CCC2CNC(=O)CN2CCCS2(=O)=O)CC=CCC1 N1(C(c2csc(C)c2C)=O)CCN(C(=O)C=CCOc2ccccc2)C(CF)C1 N1(C(C(C)=CC)=O)CCC2(CC1)OCCC2NC(=O)Cc1cc(F)ccc1OC C(=O)(C(C(C)(C)C)SC)N(C(C)C(=O)NCCCCCCC1CC1)CC C(C)(CCC(C)(C)O)(c1n(CC=C)nnn1)NC1(CC=C)CCOC1 C(=O)(CC(C)(C)NC(=O)C(C)C1(O)CCC1)NC(CCOCC)C C1(N(C)C)CN(S(=O)(=O)CCCCCl)CC1(C)C.c12cc(no1)C(=O)N1CC2C1 c1(C(N2C(CNC(CC(C)C)=O)CC2)=O)cccc(Br)c1OC(F)F Cc1cccc(-n2nnc(C(=O)NCC(C(C)(C)C)NC(=O)CCCF)c2C)c1 C(=O)(C(C#N)(CC)CC)N1CCC(F)(CNC(CCCOCC=C)=O)C1 Cc1onc(C2CC2)c1C(=O)NCCC1CN(C(C2CCCOCC2)=O)CC1C N1(C(c2nnc(C)s2)=O)CCCC(CO)(NC(c2cc(O)nc(O)c2)=O)C1 c1(C(C)(C)C(=O)NCC2CN(C(c3cn(C4CC4)nn3)=O)C2)cccnc1F S(=O)(=O)(c1c[nH]ccc1=NC1CCCOCC1)NCc1cc(OCC#C)ncc1 N1(C(C2N(C(c3cccc(C)c3N)=O)CCOC2C)=O)CCC(=C(F)F)CC1 Cc1ccc(CC(C)C(=O)NCCC(C)CC=CC(N2CCSCC2C)=O)cc1 N1(C(c2c(C)cnn2C)=O)CC2CCCCC2(NC(C2CN(C3COC3)C2)=O)C1 N1(CC(=O)NCCNC(c2c(C)oc(C)c2Br)=O)C(=O)NC(C)(C2CC2)C1=O C12CC3(C1)CC(CCC(N)C3)C(CC=CCC)CC(=O)N2C(C)(C)C.C(=O)O C1(C2(C(N)=O)CC2)CCCN1C(=O)C(F)C1CN(C(c2cn(CCO)nn2)=O)C1 c1(CC(N2CC(CNC(C(C(C)C)OC)=O)C2)=O)nn(C)c(=O)c2ccccc12 N1(C(c2nc(Cl)sc2Cl)=O)CCC2(CCCN(C(C3CC4CCC3O4)=O)C2)CC1 C1(C#N)(C(=O)NCC(CC=C)NC(=O)Cc2cc(CC)n(C)n2)CCCCCC1 c1(CN2CC(CC)N(C(=O)Cc3ccc(C)cc3)CC2)c(F)ccc(C)c1F C(=O)(C(O)C(F)(F)F)N(CCNC(C1(Cc2ccccc2)CCOC1)=O)CC c1(N2CC(O)(CNC(Cn3ccc(C)n3)=O)C2)cc2nnc(C)n2cn1.C(F)F N1(C(Cc2c(C)con2)=O)CC(N(C)C(C2C(F)(F)C23CCC3)=O)C2(CC2)C1 Cn1cc(C(=O)NC2(CCNC(C3CC4CCC4C3)=O)CC2)ncc1=O c1(SC)ccc(NC(n2ccnc2C2OCCC2SCC(F)F)=O)cc1 C1(N2CCCCC2)(CO)CCCCC1.n1(C(C)C)nnnc1C(C1(C)CC(C)C1)N Cc1c(C(N2CC(NC(C3(F)CCOCC3)=O)CC2C)=O)ccn1CCO C=CCCCCCCC(=O)NCC1CCCC1C(=O)NCCC(C)(O)C1CC1 CC(C)C(F)C(=O)N1CCC(C(C)CNC(=O)CN(C)C(c2ccsc2)=O)CC1 N1(C(=O)CSC2CC2)CCCC2(CCN(C(c3csnn3)=O)C2)C1 c1(NC(=O)NC(c2n(CC)ncc2)C)ccc2nc(C)[nH]c2c1 N1(C(c2[nH]c(=NCc3ccc(CC)nc3)sc2)=O)CCc2cc(C#N)ccc2C1 C1(NC(c2cc(C)sn2)=O)CC2(C1)CC2C(=O)N(C(C)CC(C)C)C C1(CNC(c2cc(SC)nn2C)=O)CCC(C)CN1C(C1CCC(C)(C)OC1)=O c12ccc(cc1)C(=O)NC1CC1NC2.N1(S(CCOC)(=O)=O)CCCC1C(N)=O N1(C(CC(=O)OCC)=O)CCOC(C(C)NC(c2cn(C(C)C)nc2C)=O)C1 CCC(CC(F)(F)F)C(=O)N(C1CN(C(=O)CCNC(=O)COC)CC1O)C c1(C(N2C(C)CC(NC(C3C(C)(CC)C3)=O)C2)=O)cc(S(N)(=O)=O)co1 C1(O)(C(=O)NCC(C2CCCCC2)OC)CCN(C(=O)CNC(=O)C(C)(C)C)CC1 N1(C(C2C(C)N(C(=O)CCc3cncnc3)CC2)=O)C2CCCC1CN(C)C2 c1(NC(c2ccc(CC(N3C(CSC)CCC3)=O)cn2)=O)cc(CO)ccc1C C(=O)(C(C)C(C)c1ccco1)NC(CN(C(COCc1onc(C)n1)=O)C)(C)C Cc1ccnc(C(=O)NC(C)(C)CNC(=O)CCC2CCC(O)CC2)c1 Cc1cccc(C)c1CNC(=O)C(=O)NC12CC(C(=O)O)(C1)C2 CS(=O)(=O)C(CNC(=O)C(O)Cn1cncn1)CNC(c1n[nH]c2c1CCC2)=O c1(C(=O)NC(C)CCNC(=O)C(=CC2CCCCC2)F)ccc(=O)n2c1CCC2 c1(CC(=O)NCCN(C(=O)C(C)CNC(C)=O)CC)c(C)n[nH]c1C Cn1cc([N+](=O)[O-])c(=NC2CCN(C(C3CCC(N=[N+]=[N-])CC3)=O)CC2)[nH]1 N1(C(c2cccc(C)c2O)=O)CCC(C2CC2)(CNC(C2(C)CC=CCO2)=O)C1 C(=O)(C(CC)CCOC)N(C(CCNC(C1C(CC)CCCC1)=O)C)C N12CCC(F)(C1)C2=O.c1(CSCC(=O)NCC2(C)CC2)ccncc1.C(=O)(C1CC1)N CC(C)C(C(=O)N1CC(NC(=O)CCc2nc(O)n[nH]2)C1)c1ccccc1 n1(CC=C)cc(C(=O)NC(Cn2ccnn2)C(=O)NCCC(C)OC)cn1 C1(C(N(C(CC)CC(=O)NC2CCCCC2C)C)=O)CC2(C1)CC(C)C2 N1(c2nc(C)nc(C#N)c2)CCC2(CCCCN(C(c3ncccn3)=O)C2)C1 c1(OC)ncc(Cl)c(C(N2CCN(C(C3(F)CCOC3)=O)CC2CC(F)F)=O)n1 N1(C(C(C2CCN(C(C(C)(C)SC)=O)C2)C)=O)CCC(O)(CCO)CC1 N1(C(c2nc(Cl)sc2Cl)=O)CC2(C1)CN(C(C1CCS(=O)(=O)N1)=O)C2 O=C(CC=C(Cl)Cl)NCCCNCCCNC(c1ccnc(C(F)(F)F)c1)=O c1(CC(N2CC(NC(C=C(COC)C)=O)C(F)CC2)=O)coc2cc(Cl)ccc12 C1(C(=O)NC2CC(NC(C3(CC=C)CCC3)=O)C2)CC=CC(O)C1 CC1CN(C(c2ccoc2C(F)(F)F)=O)CC1NC(C1(C)CC2(CC2)C1)=O C1(C(C(=O)NCC(CNC(c2cc(C)n(C)c2)=O)OC)C)CCCCCC1 c1(NC(=O)NCc2cccc(Br)c2F)nc2c(o1)CCSC2 C1(NC(CCN(CCCCC)C)=O)CCCN(C(C2CC3CCC3C2)=O)C1 N1(C(C2CCCN(CC(C)C)C2)=O)CCC(NC(c2cnc(S)nc2)=O)C12CC2 CC1CCC(NC(c2cccc(C)c2)=O)CN1c1nccc(C2(C)CC2)n1.C(N)=O c1(C(=O)N(CCCc2cn(CC3(CC)CCC3)nn2)CC)c(C)[nH]c(C(=O)O)c1C C1(C(=O)OCc2cc(C)sn2)CCC(=O)C(C)C1(C)C c1(C(N2CCC(C)C2CNC(=O)C=CC(F)(F)F)=O)cc2ccc(Br)cn2c1 C=CCC(CNC(C1CC(SC)C1)=O)C(=O)Nc1ncccc1CC C1(C(=O)NCC(C)NC(COCCCOCC)=O)CC(n2cnnc2)C1 c1(C(N(CCC(C)NC(=O)Cc2cccc(Cl)c2Cl)C)=O)cnc2[nH]cncc1-2 CN=S(C)(=O)c1ccc(C(=O)NCCN(C(=O)CC2COCC(C)(C)O2)C)cc1 N1(C(CCS(C)(=O)=O)=O)CC(F)(CNC(=O)C(F)C2CCCC2)C1 c1(C(N2CCC(CNC(CCCC#C)=O)CC2C)=O)cccc2c1NCC2 S(=O)(=O)(CC(=O)NC1CCC(NC(=O)C(C)(F)F)C1)N(CC)CC N1(C(C(C)CNC(C2CN3CCN2CC3)=O)=O)CCC2(COC(=O)N2)C1 CC(CN(C(=O)Cc1nccn1C)C)C(=O)NC1(C2CCCO2)CCC1 N1(C(C(C)OC(C)(C)C)=O)CC(C)(C)C(C(=O)NC(C)(C)CCl)C(C)(C)C1 Cc1nc(C(N2CC(CC(=O)NCC3NC(=O)NC3=O)CC2C)=O)c(C)o1 N1(C(CN(C)C)=O)CC(OC)CC1CC(N1CCN(C(C2CSC2)=O)CC1)=O Cc1c(C(N2CCC(C(=O)NCc3ccc[n+]([O-])c3)(C(C)C)C2)=O)cncc1F c1(OC)cc(C(=O)NCCC2CCN(C(=O)C#CC(C)(C)C)C(C)C2)ccc1F Cc1cc(N)cnc1C(=O)NCc1ccnc(C(=O)NC2CCCC2(C)C)c1 C12(NC(c3c(Cl)c(C)n(C)n3)=O)COCCC1CN(C(c1cccnn1)=O)C2 C1(OC)CC(CNC(=O)CCSCC(N)=O)N(C(=O)C(C)C2CCC2)C1 Cc1ccc(Cl)c(NCC(N2C(C)CCCC2C)=O)c1 c1(OC)ccc(CN2CCC(C)(CNC(=O)COCP(C)(C)=O)C2)c(C)c1 c1(CC(N2C(C(=O)OC)CC(C(C)(C)C)CC2)=O)cn2c(n1)CCCC2 N1(C(CCCC(=O)N(C)C)=O)CCC2(NC(=O)CC(C)(F)F)CCCC12 C(=O)(C(C)C(C)(C)c1ccccc1)NCC(C)N(C(c1c(C)nc[nH]1)=O)C C1(C(=O)NC2CCN(C(C(C)OCC3CC3)=O)CC2O)CC1C1CCCCC1 N1(C(c2n[nH]c(C)c2C)=O)CC(NC(C2C(F)(F)C23CC3)=O)CC(C)(C)C1 c1(C(=O)NCC(CN(C(C(C)NC(c2ccoc2)=O)=O)C)C)cc2occc2s1 c1(OCC(=O)NCCC(C)N(C(=O)CC2CC3(CC3)C2)C)ccc(F)c(Cl)c1 C(=O)(C(F)(F)CCc1ccccc1)NC12C(CN(C(C(C)OCC)=O)C1)C2 c1(C(=O)NCC(c2ccc(C(C)(C)C)cc2)O)cc(N=[PH](C)(C)=O)ccn1 N1(C(c2cc(C)ns2)=O)CCCC(NC(C2CCC(C)(C)OC2)=O)C1C C1(CC)CN(C(=O)COc2ccc(F)cc2)CCC1NC(C1CNC(=O)N1)=O c1(C(C(=O)NCCCNC(C(C(C)SC)O)=O)=O)ccc(F)c(F)c1F N1(C(=O)CCc2ccc(Br)cn2)CCCC2C1CCN2C(c1cc(F)ccc1O)=O N1(C(=O)Cc2cccnc2)CCn2ncc(-c3cnn4c3CCC4)c2C1 CC1(CC(=O)NCC(O)CCNC(=O)C(c2ccccc2Cl)O)CCCCCC1 CCCCC(C(=O)N(C1CN(C(=O)C(C)CC2CCCC2)CCC1C)C)C(C)C c1(C(=O)NCC2C(NC(Cn3c(C)nnn3)=O)CCC2)cnn2c1CCCC2 N1(C(C(CC)(F)F)=O)CC(NC(=O)CCc2ccc(OC)cc2F)CC(C)(C)C1 c1(C)cccc(CN2CCCC2)c1.C12(CCOC)CCCC1(C(N)=O)C2 N1(C(C2C=CC(NC(=O)CCCC3CCCC3)C2)=O)CC2CCC(O)C(O)C12 N1(NCCC(=O)OC)Cc2ccc(NC(=O)CC3CCCN(CC)C3)cc2C1=O Nc1cncc(C(=O)NCC2C3CN(C(C4CCCC(O)C4)=O)CC23)c1 C(C(C(C)(C)C)NC(c1c(Cl)n[nH]c1C)=O)NC(C(C)(C)NC(=O)NCC)=O CCN=c1[nH]c(C(=O)NCC2CC(F)(CNC(C3C4COCC34)=O)C2)cs1 c1(CCSC)c[nH]c2ncccc12.c12c[nH]c(C)c1NC(=O)C1(CC1)N(C)C2=O N1(C(C=CC(=O)OCCCC)=O)CCN(C(=O)Cc2ccsc2C)CC12CCC2 c1(CC(=O)NCC(CC)NC(=O)CC2CCCOC2)cnnn1C C1(NC(CCC#CC)=O)CCN(C(=O)C#CC(C)C)C12CC2 C1(NC(C2CCCSS2)=O)CN(c2nnc(C3CCCC3)s2)C2(CCOCC2)C1 C#CC1(O)CC(C(N2CCCCC2CNC(c2oc(SC)cc2C)=O)=O)C1 c1(OC(C(C)Cn2ccnc2)=O)cccc(F)c1C#N C(=O)(C(O)P(C)(C)=O)NC(C)CCCNC(=O)CCc1nncs1 CN1N=CC(CC(=O)NCC(CC2CC2)C(=O)N(C2CC(F)(F)C2)C)C1=O CC1(C)CCCCC1=CC(N1CCOC(CNC(C23CCC2C3)=O)C1)=O C1(COC)CN(C(c2conc2C2CC2)=O)C1(C)C.C(=O)(C(C(=O)OC)OC)NC C(=O)(CCCCC(N)=O)NCC(CC=C)NC(C1(S(C)(=O)=O)CC(O)C1)=O Cc1nocc1CC(=O)NCCN(C(=O)C(F)=CC1CC1)CC(C)O c1(C(=O)NC(CC=C)CNC(C2CC2CC)=O)cc([N+](=O)[O-])ncc1Br c1(C(N2CCC(CNC(CCC3C(C)(C)C3)=O)C2)=O)cc2c(nc1O)CCCC2 O=C(CCCCO)NCC(=O)NCC#CCNC(=O)CSc1cccs1 n1(CC)ncn(NC(=O)C2CCC=CCC2)c1=O.c12[nH]ccc1CNC2=O N1(C(C(CC)SC)=O)CC2(C(=O)NCC3(C)CCCO3)CCC1CC2 C1(C(=O)NCc2c(C)non2)(NC(=O)COCCCF)CCN(C)C1 Cc1nocc1C(=O)NCC1(O)CN(C(=O)C(C)N(CC(F)(F)F)C)C1 C1(C(N2C(C(C(=O)NC(C(=O)OC)C)(C)C)CCC2)=O)C2CCC(C2)C1C c1(NC(CCC)CCCNC(=O)CCOCCOCC)ncc2ncnc-2[nH]1 O=S(=O)(c1c[nH]ccc1=NC1CCCC(C(F)(F)F)C1)NCC1(CC2CC2)CC1 C(=O)(C(CC(F)F)C1CCCC1)N(C(C)C)CCN(C)C(C1CC2CC2C1)=O N1(C(C2(O)CCN(Cc3ccc(OC(F)F)nc3)C2)=O)CCc2sccc2C1 c1(OC)ncc(CN2CCOC(CNC(c3conc3C)=O)C2)cc1Br C(=O)(C1=CC2(CCOC2)C1)NC12CC(CNC(C3C(COC)OCC3)=O)(OC1)C2 N1(C(CSCCN(C)C)=O)CCC(CNC(c2cc(C3CC3)on2)=O)C12CCC2 Cc1ccc2nc(C)c(NC(=O)N(C3CONC3=O)Cc3cccc(Br)c3)n2c1 n1(CCNC(c2c(CNC(C(CSC)C)=O)cc[nH]2)=O)cnc2ccccc12 CCCC(CCC)C(=O)N1CCC(O)(CN(C(=O)Cn2ccnc2C(C)C)C)C1 Cn1cc(C(=O)NC(C)(CNC(c2cc(C(N)=O)cs2)=O)C2CCC2)ccc1=O c1(CC(=O)NC2(C3CN(C(=O)CC4CC5(CCC5)C4)C3)CC2)cc(Br)ccc1F c1(OC)cc(N)cc(C(N2CCCC(OC(F)(F)F)C2)=O)n1 C1(NC(c2cccc(OC)n2)=O)CCOC12CCN(C(=O)C(O)P(C)(C)=O)CC2 c1(SC)cnn(C)c1C(=O)NC1CC(N(C(=O)CCC(N)=O)C)C1 Cc1cc(O)ncc1NC(=O)C(C)N(C(c1cc[nH]c(=N)n1)=O)C1CC1 CC(C)CC(C(=O)NC1CC(CCNC(c2ccc(Cl)c(F)c2F)=O)C1)C(N)=O c1(C(N2CC(N(C(=O)COCCC)CC#C)C2)=O)cnc2c(C)cccc2c1 c1(CN=C(NCC(C)(C)C)NC2CC(C(N)=O)C2)cnc2n1CCC2 Cc1ccc(C(N2CCC(CNC(=O)CSc3cccs3)C2)=O)n1C CC(C)C(C(=O)N1CCC(C(N2CC3CCCCC3C2)=O)O1)C1CCC1 c1(N2C(CC(=O)NCc3c(C)n[nH]c3)CCC2)nccc(Br)n1 C1(C2CC2)(NC(C2C(C(C)NC(=O)C(N)=O)C2)=O)CC1 C(=O)(C#CC1CCCOC1)NCC1CC(NC(c2c(C)cc(C)nc2)=O)CC1O Cc1cn(C)c(C(C(=O)NC(C)C)N(C2CCCC2)CCN(C)C)n1 CCCCC(=O)N1CSCC1C(=O)N(C)CCc1cccs1 C1(C(=O)OC)CCC(C(=O)NC(C)CNC(=O)CCCOC2CCOCC2)C1 C1(=O)N=C2NN=C(S2)C12CC2.CC1(C)CCN(CCO)C1 C(=O)(CC1=CCOCC1)NC(CC=C)CNC(=O)C(O)(C1CC1)C1CC1 c1(C(N2CC(CNC(C=CC(CC)C)=O)C(F)(F)C2)=O)cc2c(ncn2C)s1 C(=O)(C1=C(C)OCCS1)NCC(CC=C)C(=O)NC1COC(C)(C)C1 c1(C(=O)NCCN(C(C2C(CN)C2(F)F)=O)CC)ccc(F)cc1 C=CC1COCCN1C(=O)CC(C)N(C(=O)C(C)COCC)C Cc1cccc(C(=O)NCC(C2CCN(C(c3cc(C)c(C)[nH]3)=O)CC2)F)c1C C1(CNC(c2cn(C)cc2C(F)(F)F)=O)CCN(C(c2cncs2)=O)C12CCC2 C(=O)(C(C)(O)CC(C)C)NCC1(C(=O)NC2(C3(OCC)CCC3)CC2)CCCO1 C(C(C)CC(=O)NCC(C1CCN(C(=O)COCc2ncnn2C)CC1)F)OC C1(C(N(C2CCCN(C(=O)CN3CC(C)(OC)C3)C2)CC)=O)CC(=O)OC1(C)C CC(F)(C(=O)N1CC(CCNC(=O)C=CC(F)F)C1)C1CC1 C1(C(=O)NC2(CC=C)CCOC2)C2CC2CN1C(=O)CC1C(C)(C)C1(C)C C1(F)(CNC(COC(C)C)=O)CCCN(C(C2(C(C)(C)O)CC2)=O)C1 c1(CC)nn(C)c(CC)c1NC(=O)Nc1ccncc1C C1(CCC(=O)NCC(C2CC2)OC)CN(C(C2CCC(C3CC3)C2)=O)C(C)(C)C1 c1(C(=O)NC(CC)CNC(C2(n3cncn3)CC2)=O)cscc1C(F)F C(=O)(CCCc1ncco1)NC1(CNC(CN(c2ccncc2)C)=O)CCC1 O=C(C1=CC2CCCCCCC12)N1CCC1.c1(N)cc(C(F)(F)F)ccc1O c1(CN2C(C(=O)NC(c3ccc(Cl)cc3)CO)CC(=C)C2)cnc(OC)c(Br)c1 c1(C(N(C)CC2CN(C(CCOCC)=O)C2)=O)sc(C2CCCOC2)nc1C CCCCC(C(=O)NCCNC(=O)CC1(c2ccccc2)COCCO1)C(=O)O C(=O)(C1CCc2c[nH]nc21)NC1CCN(C(c2n(COC)ncc2)=O)CC(O)C1 c1(C(=O)NCC2C(NC(c3cn(CC)nn3)=O)CC2)ccc2c(c1)C(C)C(C)O2 C(CP(C)(C)=O)(C(=O)OC)N(C(c1cncc(OC)c1)C(=O)NC1CCC1)C c1(C(N2CC3CC2C3CNC(=O)C(F)(F)CC2CC2)=O)ccc2n[nH]cc2n1 C=CCCCC(C1CC1)NC(C1CC1C(C)NC(c1ccc(F)cn1)=O)=O C1(C(=O)Nc2cccc(OCC)c2)CCN(C(C2CC23CC3)=O)CC1C c1(NC(c2ccc(-c3cccc(OC(F)F)c3)nc2)=O)cccc2c1CCO2 N1(C(C2(C)CC(C)C2)=O)CCC(O)(CNC(c2cnccc2OC(C)C)=O)CC1 c1(NS(C)(=O)=O)nccc(=NCc2coc(NC3CC(C(F)(F)F)C3)c2)[nH]1 c1(OC)ncc(C)cc1NC(C1(NC(C2(C)CC3C=CC2C3)=O)CCC1)=O N1(C(c2cccc(CC)c2O)=O)CC2(CC(NC(=O)C(C)=CC3CC3)CO2)C1 Cc1cc(C)c(C(N2CCCC2CCC2CCCC2c2nn[nH]n2)=O)cn1 n1(C(C(=O)NCC(C(C)C)NC(c2c(C)cno2)=O)C)nc([N+](=O)[O-])cc1C N1(C(C2C(CCC)CCC2)=O)CCC2CCC(NC(=O)CCCCN(C)C)C12 CC12C3C4C1C1C2C3C41C(=O)NC1CCN(CCNC(c2c[nH]nc2C(F)F)=O)C1 C1(C(=O)NC(CNC(CCC(C)C)=O)C(C)(C)C)CCCc2ccccc2C1 n1(CC)ncc2c1CCCC2NCc1cccc2cccnc12 C1(C(N2C(CNC(CN(CCOC)C)=O)CC(COC)C2)=O)Cc2nccn2C1 C(CC(F)F)(C(=O)OC)NC(CN(C(=O)COCC(F)F)C)=O.C1(N)CC1 Cc1ncn(C)c(=O)c1C(=O)NCC1CC(NC(=O)COC(C)C)CCO1 c1(C(=O)NC(COC)C)oc(Cn2cc(CN3CCSCC3)nn2)cc1C C1(C(N(CCC(=O)NCc2c(C)n[nH]c2)CCCO)=O)CC1C1(C)COC1 N1(C(C(C)c2ccsc2)=O)CC2CCCCC2(NC(=O)CCc2cccnc2)C1 C(CC1=CCCCC1)NC(N1CC(N(C)C(C2CC(N(C)C)C2(C)C)=O)C1)=O c1(C(N2C3CC2CN(C(C2CC(n4cnnn4)C2)=O)C3)=O)ccc(F)c(CO)c1 Cc1nc(C(=O)N(C2CCCCC2)CCNC(c2sccc2OC)=O)sc1C c1(C(C)CC(=O)NCCCN(C(C)C(=O)N(C)C)C(C)C)ccc(F)cc1 C1(N(C)C)CN(C(=O)C(O)CCNC(c2cccc(O)c2)=O)CC1F C#Cc1c[nH]nc1C(=O)NC1CC2(C1)CC2C(N1CC(F)C(F)C1)=O C1(NC(Cn2c(C(=O)OC)cnc2)=O)CCCCC1CNC(=O)C(O)C1CCC1 C1(CC)(NC(=O)CCn2cncn2)CCN(C(C2CCS(=O)(=O)N2)=O)CC1 C(C(C)(C)CC(=O)NCC1CC1CC(=O)N(C1CC1)C(c1ccccc1)C)OC N1(C(C2CCN(c3cccc(C)c3)C2=O)=O)CCCC2(C1)N=N2 c1(C(=O)OC)ccc(CN2CCCC2C(=O)NC)s1.c1(C2COC2)ccccc1 c1(C(N2CC(COC(c3c(OCC)ccs3)=O)C(C)C2)=O)c(C)[nH]c(C(C)=O)c1C N1(C(C(C)N=[N+]=[N-])=O)CC2(CO)CC1(C(=O)NC1CCC1(C)C)C2 S(=O)(=O)(c1ccc(F)c(Br)c1)NCC1CCN(C(C(C)S)=O)CC1(F)F c1(CN2CCC(C(=O)Nc3onc(C)c3Br)C2)cc(Cl)cc(Cl)c1Cl C(=O)(C1=C(C)OCC1)NC1C(NC(CCCOCC=C)=O)CC1 C12(N(C)C(=O)NC(C)(C)C)CC1CN(C(C1CC=CCC1C(F)(F)F)=O)C2 c1(C(=O)NC(CC=C)CNC(=O)C(c2cncn2C)O)cnc(C(F)(F)F)cn1 C=C(C)CC(C)C(=O)NC(C)CN(C(=O)C(C)(C)C1CCCCO1)C CS(=O)(=O)c1cscc1C(N1CCC(F)(F)C(CNC(C2C3(CC3)C23CC3)=O)C1)=O C(=O)(C(C)N)OCC(=O)C(N(CCC)C(c1ccco1)N)=O.C(C)(C)(CC)O N1(C(c2c(NC)cccn2)=O)CCCC(CC)C1C(=O)NCCC(C)C(C)C c1(C(C)C)ccc(NC(c2cc(Cl)ccc2F)c2nnnn2C2CCCC2)cc1F C1(C(=O)NCCN(C(=O)Cc2csc(C)n2)CC)CCCCC(C)(C)C1 C12(CNC(c3cc(F)ccc3F)=O)CCC(CC1)N(C(=O)C(F)=CCCF)C2 N1(Cc2cn(CC)nc2)CCC2(CCN(C(=O)Cn3ccc(C)cc3=O)CC2)C1 C(=O)(CCCC(C)(F)F)NC1C(N(CC(=O)NC2CC2)C)CCCCC1 c1(OC)c(C(N2CCOC(CNC(c3ccc(CO)s3)=O)C2)=O)cccc1F N1(C(CCOCC(C)(C)C)=O)CC(NC(=O)CCC2CCCOC2)CC(F)C1 N1(C(CC)=O)CCC(C)(CNC(=O)CCc2scnc2C)C1 c1(C(N2CCC(CC#C)CC2)C(=O)NCc2ccccc2)cc(C#N)ccc1Cl N(C(=NCCCCl)NC1CCC(=O)NC1=O)CC1CN(C(=O)OC(C)(C)C)C1 N1(C(C23CC(NC(c4cc(C)nc(O)n4)=O)C(OC2)C3)=O)CC2(CCC(=O)N2)C1 CCCC(CC)C(=O)NC(c1ccccc1F)CNC(c1cnc(S)[nH]1)=O C(=O)(C#CC1CCOC1)NC1(CNC(COC(C)(C)C(F)(F)F)=O)CCOC1 C1(C(=O)NCCN(OC)C)CN(C(=O)C=Cc2nccs2)CC12CCC2 N1(CC(=O)NCCC)CC2CCC(NC(c3ccc4c(c3)OCCO4)=O)CC2C1 c1(CC)sccc1C(N1CC(CNC(c2cc(C3CC3)on2)=O)C1)=O C1(C(N2CC(CC(C(=O)N(C3CCC(C)C3)C3CC3)F)C2)=O)CCOCC1(C)C C(=O)(C(CO)C(F)(F)F)N(CCCC(=O)Nc1c(COC)csc1)C c1(C(N2CCN(C(CC3(OC)CC3)=O)CC2C)=O)c2cc(Br)ccc2nn1C N1(C(C2CC(F)C2)=O)CCCC(C2CCCN2C(C2(O)CCOCC2)=O)C1 c1(CNC(N(C)Cc2cc(OCC)ncc2)=O)cc(F)c(F)c(F)c1 C1(NC(COC2CN(C(C(C)(F)F)=O)C2)=O)CC2OCCCC12 CC(C)CC(O)C(C)C(=O)NC1CCC(NC(c2ccc(O)c(F)c2F)=O)CC1 c1(OC)ccc(C(N2CC(C)(C)C2CO)=O)c(C(F)(F)F)c1 CC(C)(C)C(O)CNC(c1nc(CO)cs1)c1nnnn1C1COC1 C(CCCCNC(C1CC1C(F)F)=O)NC(C1(OC)CC1)=O C(=O)(C(CO)C(F)(F)F)N(C)CC1CCC(NC(C2CC3CCC(C2)C3)=O)C1 C1(CC)CCCCC1C(=O)N(CCCNC(=O)C(F)(F)c1ccncc1)C C1(C(=O)NC(C)CNC(=O)Cc2ccc(CO)cc2)CCN(C2CC2)S1(=O)=O C(=O)(C(C)CCCc1ccccc1)N1CCC(C)(CNC(C=CCCC)=O)C1 C(C(CCN=c1[nH]c(=NCC2(SC)CC2)[nH]c2c1CSC2)C(C)C)OC C(c1cc(Br)ccc1CC)=Cc1ccc(CC=C)s1 CCCCS(=O)(=O)CC(=O)NC1C2CC1N(C(=O)Cn1cc(C(C)O)nn1)C2 c1(-c2cc(C)c(OCOC)c(C)c2)ccc2nc(C(N3CCCC(O)C3)=O)oc2c1 c1(C(N2CCC(COC)(NC(=O)CNC=O)C2)=O)coc2ccc(Br)cc12 N1(C(c2cnc(CC)o2)=O)CCCC(CC)C1C(N1C(CO)CC1C)=O C(=O)(CCCN(C)C)NCCC(C)NC(c1cccnn1)=O N1(C(C(C)CN(C)C)=O)CC2CCCCC2(CNC(c2c[nH]c(C#N)c2)=O)C1 Cn1cc(C(C2CCN2C(=O)CC(F)F)NC(c2cccnc2)=O)cn1 N1CC(c2cn(Cc3scc(C)c3)nn2)C(C)C1.c1(C=O)onc(CN(C)C)c1C c1(N(C)C(C2CCN(C(C3C(=C)C3C(=O)OC)=O)CC2)=O)nc2cccnc2s1 C1(C(N(C)CC2N(C(C#CC(C)C)=O)CCOC2)=O)CCc2cncn2C1 c1(O)ccc(C)c(C2CC2(F)F)c1.N12CCC(CC1)NC2=O.CC(=O)NCCO C1(C#N)(C(=O)NC(CCN(C(c2cccc(OCCC)c2)=O)C)C)CC2(CC2)C1 C1(F)(C(N(C)CC2N(C(c3c(C)cns3)=O)CCC2)=O)CCS(=O)(=O)C1 C(=O)(C1=CC2CCCCCC12)NCCC1CN(C(c2c(C)ncc(Br)c2)=O)C1 N1(C(c2cc(Br)cs2)C(=O)NC(CC)C)CCC(CN(C)C)CC1C CC1CN(C(C2CC(C)(C)C2)=O)CC2(CCN(C(=O)C(F)(F)c3nccs3)C2)O1 CSC1=C(C(=O)NC(C)(C)CCNC(=O)C(CC2CCCC2)C(C)C)CCCC1 CC1(C)CC(NC(C2(C)CCCNC2=O)=O)CCN(C(=O)COC2CCCC2)C1 CC(=O)CCN=C(NCC(C1CC1)C1CC1)N1CCN(c2nccs2)CC1 CC(=O)CCCC(=O)NCCC1CC(NC(c2cn3c(n2)SCC3)=O)C1 C1(N(C(c2cc(CCC)oc2C)=O)C)CN(C(C2CC(F)C(=O)N2)=O)CC12CC2 N1(C(c2c(C#C)c[nH]n2)=O)CCN(C(=O)C2=C(Cl)CC2)CC1CC(F)F N1(C(c2cocn2)=O)CCN(C(=O)Cc2cncnc2O)C2CCCCC2C1 N1(C(C(C)C)=O)CC(NC(C23CC(CN2C2CC2)C3)=O)CC12CCCCC2 N1(C(C(C(C)(C)C)CNC(C2CC3CCC3C2)=O)=O)CC2(CCC2)C12CCC2 C(=O)(C(C)(CN(CC)CC1CCCCO1)CC)N1C(CN2CCNC2=O)CCC1 N1(C(c2cccc(C#C)c2)=O)CCCC2CN(C(C3CCN3CC)=O)CCC12 N1(C(C(c2cncnc2)C)=O)CCCC(NC(=O)CSCCC(F)(F)F)CC1 N1(C(CC(CC=C)(C)C)=O)CC2CC3CC2C1C3NC(c1scc(C)c1Br)=O c1(C(=O)NC2C(CNC(C(C)NC(CC)=O)=O)CC2)cnn2c1NCCC2 c1(N(CCC)CCNC(=O)CN2CC3CCC2C3)nc2c(cc1C#N)CCOC2 CC1OC2(C(N3CC4CC4(NC(c4ccc5c[nH]nc5n4)=O)C3)=O)CCC1CC2 N1(C(C2CC(NC(C(C(C)C)C)=O)C2)=O)CC(C)OC(C)(C)C1C Cc1ccc2nc(C(N3CCN(C(=O)Cc4occc4C)C(CO)C3)=O)cn2c1 C1(OC)CCC(C(=O)NCCCCCCNC(c2nocc2CN(C)C)=O)CC1 c1(C(=O)NCC(CC)NC(c2ncccc2Br)=O)cc(C)c(O)c(C)c1 C1(N(C(=O)NC2(c3ccccc3C)CCC2)CC)CCC2COC1O2 c1(CC)ncc(Cl)c(C(=O)NC2C=CCN(C(c3ncnc(C)c3C)=O)C2)n1 c1(C(=O)NCC2CCN2C(=O)CC2C=CCC2)cccc(N2CCC2=O)c1 CC1CCCCCCN1C(C1CC2CCC1N2C(C1(CCF)CCC1)=O)=O C1(C)(OC(COC2CCN(C(C(C3CCC3)OC)=O)C2)=O)CC=CCC1 C1(N(C(C2CCC(=C)CC2)=O)C)CCN(C(c2ccncc2Cl)=O)CC1C c1(C(N2CCC(CN(C(=O)CC3C=CCCC3)CC)CC2)=O)cnc(O)c(F)c1 Cc1cc(C#N)cc(C)c1C(=O)NC1CC(CCNC(=O)Cn2nccc2C)C1 N1(C(C2CN(C)C2)=O)CCCC2CN(C(c3sc4nccnc4c3N)=O)CCC12 C1(C#CC(=O)NCCOC2CN(C(c3cc(C(N)=O)[nH]n3)=O)C2)(CC)CC1 C1(CNC(=O)COCCOCCO)CN(C(c2c(OC)ccs2)=O)CC12CC2 c1(C(C(F)(F)F)NC(C(=O)NC(CCCC)CC)=O)cccc2sccc12 N1(C(c2c(C)nn(C)c2)=O)CC2(CCCCN2C(C2(C)CCNC2=O)=O)C1 c1(NC(N2CC(CC(=O)Nc3cccc(OC(C)(C)C)c3)C2)=O)cc(F)cc(F)c1 N1(C(C(CSC)OC)=O)CCC(CNC(c2cccnc2N(C)C)=O)C(F)(F)C1 C#CC1CN(C(C2(CCNC(=O)CC3CC(=C)C3)CC2)=O)CCO1 c1(Cn2c(C3(NCCCC(C)(C)SC)CCC(CC)C3)nnn2)cc(Cl)ccc1O c1(NC(CN(CCCNC(C(N2CCNC2=O)C)=O)C)=O)ccc(O)c(CO)c1 C1(CNC(C=CC=CCC)=O)CN(C(c2cc(F)c(F)c(F)c2)=O)CCC1(F)F CC1CC(NC(N2CCCC2)=O)CN1CC(N1CCCC1)=O CC1(C)OCCC1NC(C1CC(CCNC(=O)CCN2CCCC2)C1)=O C1(CN)CCCN(CC(=O)Nc2ccccc2Oc2cccc(O)c2)C1 O=C1NCC(C(=O)N(C2(C(=O)NC3CC3CC3CC3)CCC2)C2CC2)N1 C=C(C)CCCC(=O)N1CC(CC(N2CCC(OC)C2(C)C)=O)C2(CC2)C1 N1(c2snc(CCC)n2)CCC(NC(=O)CNC(c2cnccn2)=O)C(C)C1 C1(CNC(c2c(OC)nsc2)=O)COCCN1C(=O)CCN1C(=O)CCC1=O C(=O)(C(F)(CNC(=O)C(c1cnn(C)c1)=O)C(C)C)NCC(=C)C C(=O)(CCCCc1cnn[nH]1)OCCCN(C)Cc1ccc(Cl)cc1 Cc1cccc(SC(C)C(=O)NCCNc2nc(CNC(=O)CC(C)C)cs2)c1 CC1(C)CN(C(=O)C(N)=O)CC(CNC(C2(C(=O)Nc3cccc(F)c3)CC2)=O)O1 c1(CC(=O)NCCCNC(C2N(CCC)CCCC2)=O)cc(F)ccc1Cl CSC1=C(C(=O)N2CCC(O)(CCNC(C3CCC(O)C3)=O)CC2)CCCC1 C1(C(N2C(C(=O)NCCC3ON=C(C)C3)CCC2)=O)CCCCC1(C)C CC1CN(C(C23CCC(C2)C3(C)C)=O)CCN1C(c1cn2c(n1)CCC2)=O N(C(=NCC1CCC2(CC2)C1)NC1CCCC1)C(C#C)Cc1ccccc1 Cc1ccc(C=CC(N2CCN(C(=O)CC(C)(C)F)C(c3ncc[nH]3)C2)=O)cc1 NS(=O)(=O)c1ccc(C(=O)NCC2CC2NC(=O)C=Cc2cscn2)c(C)c1 C(=O)(C(C)(C)CC(=O)NC(C1CCN(C(c2ccc(C)nn2)=O)C1)(C)C)OCC C1(CNC(c2cc(C)[nH]n2)=O)CCCC2(CN(C(=O)CN3CC4CC4C3)C2)O1 c1(C(=O)O)ccc(CNc2scc(Cl)c2Cl)cc1F.C12CC(F)CN(C1)C2=O N1(C(C(=O)C(c2ccccc2CC(F)(F)F)=O)=O)CCCC(O)(c2nn[nH]n2)CC1.OC c1(CC(=O)C(C=Cc2scc(C)n2)=O)ccc(Cl)c(O)c1.C(CCN)OCCN CC1(C)CCCN(C(C2(O)CCOC2)=O)C1CNC(c1ccc2c[nH]nc2n1)=O c1(C2C(C(N(C3CCN(C(c4sccc4CO)=O)C3)CC)=O)CC2)nncn1C CC(C)C(CNC(C1CCCC1F)=O)C(=O)NCC#CC(F)(F)F CCC(C)(CNC(=O)CSCC(N)=O)C(=O)NCc1cc(OC)ns1 N1(C(CC2CCCN(C(c3cccc(C)n3)=O)CC2)=O)CCCCC(C)(C)C1 CC1CC2CN(C(c3ccc(F)c(Cl)c3)=O)CC2N1C(c1cccc(N)c1F)=O N1(C(=O)NCC(CC)NC(=O)OC(C)(C)C)CC(C)(C)OC2CCCC12 C(=O)(C(C)CS(C)(=O)=O)NCC12N(C(C3(COC)CCCCC3)=O)C(CC1)CC2 N1(CC(=O)Oc2noc(C(N(CCC)CCC)=O)c2Br)C(=O)NC(C)(C)C1=O C1(NC(C2CC3(C2)CC3(F)F)=O)CCCN(C(c2cccnc2C(F)F)=O)CC1 N1(C(C(CC=C)(C)O)=O)CC2(C=C(C(=O)NCC(C)CC(F)(F)F)CO2)C1 C1(C)(CC(=O)NCC2CCN(C(C)=O)C2)CCN(C(=O)Cc2cnc(C)s2)C1 O=C1NCCN(C(C2C(O)CCN2C(=O)Cn2[nH]cnc2=N)=O)C1CCO Cc1snc2sc(C(N3CC(C)(NC(=O)CC4COCCO4)C3)=O)cc12 C1(NC(CSCCC)=O)CN(C(c2cccc(C3CC3)c2C)=O)C2(CCCC2)C1 c1(CNC(C2C(C(C)C)OCC2)=O)cccc(C(=O)NCC2=NOC(C)C2)n1 N1(C(c2ccc(NC(C)=O)cn2)=O)CC(NC(=O)C(F)CC(C)C)C(S(C)(=O)=O)C1 c1(C(=O)NC2CC(C)N(C(c3ccc(-c4cccs4)[nH]3)=O)C2)cc2n(n1)CCO2 c1(C(N2C(CNC(C(CC)=CC)=O)CC2)=O)ccc(F)c(C(F)(F)F)c1 C1(NC(COC(C)C)=O)CCC2(CC1)CN(C(=O)Cc1cncn1C)C2 C=CC1CCCN(c2nnc(CCSCc3nc(Cl)ccc3Cl)n2CC)C1 c1(C(=O)NCCCNC(=O)COC2CC(F)(F)C2)ccc(-c2cncnc2)cc1F C1(C(=O)NC(C)C(N2CCN(C)CC2)=O)CC(=O)N(C)C1c1cccs1 C=CC(CCC)CC(=O)NCC12CC(NC(=O)CCNC(=O)C=CCl)(C1)C(C)O2 O=C(C1=NOCC1)NCC(C1CCOC1)NC(=O)CC1CC1 C(C(C)(C)CCO)NC(C(C1CN(C(C2OCCC2C)=O)C1)OC)=O CN1CC(NC(C2CN(C(C3CCCCC3)=O)CC2(F)F)=O)C2(CC2)C1=O C1(NC(C2(CC#C)CC2)=O)CN(C(=O)CCCn2cccn2)CC1OC c1(C(=O)NC(C)C(CO)NC(=O)Cn2cc([N+](=O)[O-])cn2)cc2ccccc2[nH]1 C1(n2cccn2)(C(=O)N(CC(C)(C)CCO)C)CCN(C(=O)C=C2CCCCC2)CC1 c1(C(N2CCC(N(C(C3C(C=C)CC3)=O)C)CC2)=O)ccc(C)c(F)c1 N1(C(C(CCSC)O)=O)CC(NC(=O)CCc2cnc[nH]2)CC(O)C1 C1(C(N2CC(OC)C(C(=O)NC34CCCC3C4)C2)=O)CC(C2CC2)=NO1 C=C(Cl)CC(C(=O)NCc1cc(C)ns1)NC(=O)C(c1cnn(C)c1)O c12cc(ccc1O)CNC(=O)NC2C.c1(Sc2cccc(Br)c2)ccc(F)c(Cl)c1 C1(C(N(C2CCC2)C)=O)CC(NC(C2CC(F)C2)=O)CCO1 N1(C(C2CN(C(C)=O)C2)=O)CCC2(CCN(C(c3cc(O)cnc3N)=O)C2)C1 C(=O)(C1COc2ccccc21)N1CC(CN(CC(c2ccccc2)(C)O)C)C1 c1(N(C(=O)NCC(C)Oc2ccccc2Br)C)cccc(Br)c1Cl CCC(C)CCCCC(=O)N1CCC(NC(c2cccc(F)n2)=O)C(C)(C)C1 c1(OC)ccc(C(N2CCCN(C(c3c(C)n[nH]c3C)=O)CC2)=O)nc1N Cn1nccc1C=CC(=O)NCCCC1CCCN1C(c1c[nH]nc1F)=O Cc1[nH]c2ccc(C(=O)NCC(c3ccccc3)NC(C3CC3C)=O)cc2c1C c1(C(N(CC(O)CNC(C2CC(F)CN2C)=O)C)=O)cnc2cc(O)ccc2c1 C12(NC(C(c3ccccc3)OCC)=O)CCC(NC(=O)CSCC(F)F)(CC1)C2 c1(OC)ccc2cc(C(=O)NC(C)CC(C)NC(=O)CC(O)CN(C)C)[nH]c2c1 N1(C(=O)NCCNC(=O)Cn2cccc2)CCC2(CC1)OCC(O)C2O c1(N(C)C)ccc(C(=O)NCC2(NC(=O)CN3CC4CC4C3)CCOC2)cc1 C=C(C)CC(C(=O)N1CCN(C(=O)Cc2conc2C(C)C)C(C(C)C)C1)OC C1(CNC(C(C)=CC)=O)(OC)CN(C(c2cnc(-c3ccncc3)s2)=O)C1 C1(N(C(COCCC)=O)C)CCCN(CCc2cc[nH]n2)CC1 Cc1c(C(=O)NC2CC(NC(=O)CC3(CO)CC3)C2)oc2cc(Cl)ccc12 c1(C(N2CCCC(NC(C(C(C)C)SC)=O)C2C)=O)ccc([N+](=O)[O-])c(Cl)c1 c1(C(=O)NC(C2CCN(C(c3c(C)cncc3)=O)CC2)C)ccnc2[nH]cnc12 N1(Cc2[nH]nc(C(C)N(C)C)n2)CC2CCCN(C(c3csc4nccn34)=O)C2C1 N1(C(C(CCC#C)NC(=O)COCCOC)=O)CCCC2(CCCO2)C1 N1(C(Cc2c(C)ocn2)=O)CCC(NC(=O)C(N2CCC(O)CC2)C)CC1C C1(NC(c2n(C(C(=O)OC)C)nnn2)(C)CCBr)COc2cc(C)ccc2C1 c1(C(=O)NC2CN(C(CN(C(C)=O)C)=O)CC(C)C2)cnn2ccn(C)c12 C1(COC)CCC(C(=O)NCCN(C)C(=O)C2CC2)C1 c1(N(C(CCC(C)=O)=O)c2ncccn2)cnc2c(c1)CNCC2 c1(SC)cccc(N2CC3CC(NC(C4(S(N)(=O)=O)CC4)=O)CC3C2)c1[N+](=O)[O-] C1(CNC(C(C)OCC#C)=O)CCCC2CN(C(=O)CCc3nc(C)no3)CC12 Cn1nc(C(=O)NCC(O)CNC(=O)C=Cc2cccs2)cc1C1(Cl)CC1 CC(C)(CC(=O)NCCN1CCCN(C(C2CCC23CCCO3)=O)CC1)C(F)F C=CCC(C)C(=O)N(CCCN(C)C(c1cccc(OC(C)C)n1)=O)C c1(C(=O)NC(COCC)CO)cc(C2CCCC2)nc2c1cnn2-c1ccccc1 C(=O)(CCCCCCCCCO)NC(C)CNC(C12CCC1CC2)=O CCCCC(F)C(=O)N1CCN(C(=O)CN(C)C(c2cc(SC)c(C)o2)=O)CC1 C(=O)(CC(C)C(=O)N(CC(N1CC(SC(C)C)C1)=O)CCOC)OC c1(C(C)CC(=O)NCC2(NC(=O)CN3CCOCC3)CCCC2)ccc(F)cc1 O=C(CCCC(F)(F)CO)NCC1CN(C(c2cc3c(s2)CCC3)=O)CC1O c1(NC(CCC(=O)NCC2(CN(C(=O)CC(F)(F)F)C)CC2)=O)cccc(F)c1 c1(C(N2CC(CCCCNC(C3CCNC3=O)=O)C2)=O)cnn2cccc2c1 N1(C(CCN(OCCCCC)CC)=O)CCN(C(C2CC2(C)C)=O)CC1CC.CC Cc1cc(=NC(=O)C23CC2CN(C(c2ccc4cnc(C)n4c2)=O)C3)[nH]n1C C(=O)(C(C)(C)F)N(CCN(C(C(C)OCCC=C)=O)C)C Cc1cc(=NC2CCN(C(c3cn(C)nc3C(F)F)=O)CC2C)[nH]c(C2CCC2)n1 C1(F)(NC(C2CCC(=O)N(C3CC3)C2)=O)CC(N=c2ccnc(C3CCC3)[nH]2)C1 Cc1cc(C(=O)Nc2cc(NCCc3ccccc3F)ncn2)cc(C)c1 N1(C(CC2(OCC)CCC2)=O)CC2CC(CNC(=O)CSC)CC1C2 C1(C2C(O)CCC2)CN(CC(F)(F)F)CC1c1ccccc1Br CC1CCc2c(C(=O)NC3CCN(C(C4CC4CF)=O)C3)csc2C1 C=CC(C)(CC)C(=O)NCCCC(C)NC(c1ccccc1SC(C)C(N)=O)=O C1(NC(=O)CCC2CCC2)CCOC12CCN(C(=O)C=Cc1cccnc1)CC2 C(=O)(CC(=O)NC1CCN(C(c2sccc2C2CC2)=O)C1)OCC C1(S(C)(=O)=O)(C(=O)NCC2CC(OC)CN2C(c2sccc2C)=O)CCCC1 C(=O)(NNC(=O)COC(C)(C)C)c1nc(-c2cncc(C(=O)OCC)c2)n(C)n1 CCCCC(C)(F)C(=O)NC1CCCCC1NC(=O)CN=S(C)(C)=O C1(C(N2CC(O)(C(C)NC(=O)COCc3cccnc3)C2)=O)CCC(N(C)C)CC1 c1(C(=O)NC(C)CCCNC(c2cc(C(C)(F)F)n[nH]2)=O)cccc(F)c1Cl C(=O)(CCS(N)(=O)=O)NCCC1(O)CCN(C(c2c(OC)c(C)sc2)=O)C1 C1(c2nc(C(C)C)on2)CCCCN1C(=O)NC(CCO)c1cccs1 CC(C)(C#N)C(=O)NCC(CC1CCCC1)C(=O)NCC(c1ccncc1)O c1(Nc2c(N(CCOC)CC)ccnc2)ccc(C#N)o1 C(=O)(C#CC1(C)CCCO1)NCCC(C(C)C)NC(c1ccc(CC)c(Cl)c1)=O c1(C(N2CCCC(NC(C(C)(CO)OC)=O)CC2)=O)cc(Br)cc(F)c1F C1(CNC(C2CCCN(CC)C2)=O)CCCN(C(=O)C(C)(C)OC)CC1 C1(NC(C(CC2CCC2)OC)=O)CN(C(C)=O)CC1C c1(OCC(C(=O)NCC(C)(C2CC2)NC(C(CC)N(C)C)=O)(C)C)cccc(C#N)c1 c1(C(N(C2C3CN(C(C(C)NC=O)=O)CC32)C)=O)cc2nc[nH]c2cn1 C1(CNC(c2c(CC)ncs2)=O)CCCN(C(=O)C(C)N=[N+]=[N-])C1 N1(C(C)=O)CCC(C#N)CC1.n1(CCC)cnnc1C(C(=O)N)NCC(C)C CC1(C)C(C)(C(N2C3CC2CN(C(c2cc([N+](=O)[O-])sn2)=O)C3)=O)C1(C)C c1(C(=O)NCC(CO)NC(C(C)(C)F)=O)ccc(N)c2ccncc12 C(=O)(C1Cc2ccc(F)cc21)N1CC(NC(c2c(CCC)nns2)=O)C1 c1(C(=O)NC(c2ccsc2)CNC(C2C(CCC)C2)=O)ccc2sncc2c1 Cn1cnc(C(N2CCC(CNC(c3c(C(F)F)cnn3C)=O)C2)=O)cc1=O C1(CNC(c2ncn(C(C)(C)C)n2)=O)CC(C2CC2)C1 Cc1nn2c(c1CNC(=O)C(O)CC(F)(F)F)CN(C(=O)C(C)S(N)(=O)=O)CC2 c1(C(c2n(CCOC)nnn2)NCCOC2CC2)nc(Br)nn1C.C12CC(C1)S2 C1(C(NOCC(=O)NC2CC(=C)C2)=O)CCOCC1(C)C C(C)(C)(CCC(=O)NC(C)Cc1cn[nH]c1)NC(c1ccc(CC)cc1)=O c1(NC(C(CCC)C)c2nnnn2C2CC(F)(F)C2)c(C)cccc1F c1(C(N(CCC(C)NC(Cc2c(C)nn(C)c2)=O)C)=O)ccc(O)cc1F c1(OC)cnc(C(=O)NC(C)C(C)NC(C2CCCN(C(C)C)C2)=O)c(F)c1 N1(C(C2(C#C)CC(=O)C2)=O)CCC2(CC2C(N2CCC(OC3CCC3)C2)=O)C1 C1(C(N(CC(=O)NC)CCC)=O)CCCC1CNC(C1OCCC1C)=O C1(NC(C(=O)NCCC(N)=O)=O)CN(C(=O)CC2CC3CCC2C3)CC12CC2 c1(NC(C2N(C(CCCCNC(C)=O)=O)CC=C2)=O)cccc(C)c1C N1(C(c2c(SC)nccn2)=O)CCN(C(c2ccc(Cl)cc2Cl)=O)CC(O)C1 Cn1[nH]c(=NC(=O)NC(=O)CCCCF)ccc1=O C12(NC(C(F)=C(C)C)=O)CCN(C(C3CCN(c4ccccn4)CC3)=O)CC1C2 N1(C(CC=CC=C)=O)CC(OC)C(NC(c2cn(Cc3noc(C)n3)nn2)=O)C1 Cc1cc2c(C3CC3)c(N=c3nc4sccc4c(C4CC4)[nH]3)cnc2n1C CC1Oc2cc(F)ccc2C1NC(=O)Cn1cnc(=N)[nH]1 C1(NC(C(CCCC)O)=O)CC2CN(C(=O)CC(O)c3cc(C)cs3)CC2C1 C1(C(=O)NC2CCN(C(c3ccc(CCCCC)o3)=O)C2)C2CCN1CC2 c1(C(N2C(C)(CNC(C(CC#C)C)=O)CCC2)=O)cc(OC)ccc1[N+](=O)[O-] C(C)(C)(CCC(=O)NC1C=CCCC1)NC(COCC#C)=O c1(C(=O)NC2CCCCN(C(CC(C=C)CC)=O)C2)ccsc1S(N)(=O)=O c1(CCC(N2CC(NC(=O)C=CCF)CC3(C2)CC3)=O)cnc2c(=O)[nH]ccn12 c1(C(=O)NCCCOCCNC(CN(CCC#C)C)=O)oc(C)nc1C(=O)OC N1(C(c2cccc(C(C)C)c2)=O)CCN(Cc2cc(F)c(I)c(F)c2)CC1C#N C1(NC(C(C)(C)OC(C)=O)=O)CCN(C(C2CNC(=O)N2)=O)CC1 C1(NC(c2cc(C)nc(C)c2)=O)C(C)CN(C(c2cnc[nH]2)=O)CC1C c1(C(N2CCC(NC(C(CC#C)O)=O)C2)=O)ccc2nc(C(F)(F)F)[nH]c2c1 C(=O)(CCCC(F)(F)Br)N1CC(C(C)NC(=O)CN2C(=O)CN(C)C2=O)C1 c1(C(=O)NCC(C(=O)NCCCN(C)C)CC2CCCC2)cn2ccnc2cn1 CC#CCCCC(=O)NCCN(CCCCCC)C(C1CCC=CCCC1)=O C1(CNC(c2c(OC)n(C)nc2)=O)CCN(C(C23CC2COC3(C)C)=O)C1(C)C C1(C(=O)NCC2CCCC2Oc2ccccc2)(OC)CCN(C(=O)CSC)C1 C1(C(=O)OC)CC(=O)N(CC(=O)NC2CC2NC(=O)C(C)C2CCCC2)C1 C(=O)(C(C)(CC)C(N)=O)N1CCN(C(c2nc(COC)sc2)=O)C(CC(=O)NC)C1 N1(C(c2ccnc(OC)n2)=O)CC(NC(=O)CCc2ccn(C)n2)CCC1C c1(NC(C)=O)ccccc1C(=O)NCC1CCCN1C(=O)CNC(c1ccoc1)=O C1(CNC(c2cc(OC)nn2C)=O)COCCN(C(c2c(Cl)c(C)nn2C)=O)C1 C12(CNC(=O)CCCCO)CC(CO1)N(C(C1CC1C1CC1C)=O)C2 C1(C)(NC(c2c(CC)cncc2)c2nnnn2C2(C)CC2)CC=C(C)CC1 Cc1cc(C(=O)NC2CC(OCC(=O)N(C3OCCC3(C)C)C)C2)cc(O)n1 N1(Cc2cccc(C(C(=O)Nc3cccc(OC)c3)OC)c2)CCS(=O)(=O)CC1 C1(OC)CC(CO)N(C(C2CCN(C(=O)Cn3ncnn3)CC2)=O)C1 C=CC(C(=O)N(CCC(C)NC(c1cn(CCC(C)C)nn1)=O)C)OC C(=O)(C(O)CC(N)=O)N1C(CC)C(NC(=O)CCc2ccc(C(N)=O)cc2)CC1 c1(C(=O)NCCN(C2CCCCC2)C(C(C)NN2CCOCC2)=O)cccnc1 C(=O)(C1=CCCCCC1)N1CCC(NC(=O)Cc2n[nH]cc2Br)C(F)C1 C(=O)(C(O)C(C)(C)C)CNC(C1(CNC(C2C(OC)CC2)=O)CCOCC1)=O C=CCC(C)(C)CC(=O)NC1CN(C(=O)C(Cl)=CCl)CC1(C)C c1(NC(N2CC(NC(=O)OCC)C2)=O)nc2c(s1)CC(C)(C)CC2 N(C1c2ccccc2CC1NC(=O)CCCC1CC1)C(C(C(C)O)N(C)C)=O Cc1cc(C(=O)NCC2C3CC2N(C(c2nn(C)cc2Cl)=O)C3)nc(C)c1 C1(C(=O)NC(CCC)C2CCCC2)CN(C(c2sc(C)nc2C)=O)CCO1 CP(C)(=O)c1cc(NC(=O)C(N2CCSCCC2c2ccccc2)=O)ccn1 Cc1nc(CC(C)C)oc1C(N1CCOC(CNC(=O)Cn2cc(Cl)cn2)C1)=O N(C1c2ccccc2CC1NC(C1CCCC12CC2)=O)C(C(CCC)OC)=O c1(NC(C2(O)CCN(C(c3cncc(F)c3)=O)C2)=O)cncc(C(F)(F)F)c1 c1(OC)cc(CNc2cc(NC3CCCC4(CC4)C3)ncn2)ccc1OC(F)F N1(C(CCC(=O)NC)=O)CCN(C(C2CC2C(C)C)=O)CC(C)(F)C1 Cc1oc(-c2ccccc2)cc1CC(=O)NC1CN(CC=CCNC(C)C)CCO1 c1(OC)cc(NC(=O)COC)cc(F)c1.c12cscc1CC(=O)NCC=CCO2 c1(C(N2CCSCC2CO)=O)ccc(Nc2ccc(F)cc2)nc1.N12CC(C1)C2 CC1CC(c2nnnn2C(C)(C)C)(NC2CC2c2ccccc2)CC(C)S1 C1(C)(C(=O)NCC(C)C)CC12CCN(CCC1CCCCCN1)CC2 c1(CCC(=O)NCCN(C2CCCCC2)C(C2C(C#N)C2)=O)ccccc1F Cc1cccc(CCCC(=O)NCC2CC2CNC(=O)CC(F)(F)F)c1 N1(C(COCC)=O)CCC2CN(C(c3cnc(O)n3CC)=O)CC2C1 Cc1ccc(C(N2CCCCC2C(C)NC(=O)Cc2cc(C)n(C)n2)=O)cc1C C(=O)(C1=CC2CCCC12)NCC1N(C(C2CN(C(C)=O)C2)=O)CC2(CC2)C1 N1(C(CCOC)=O)CCN(C(=O)CNC(=O)Nc2ccccc2)C(C(F)(F)F)C1 C1(C(NOCC(CSCO)O)=O)CCC(C)CC1.CC(C)(C)CCN C1(NC(C2(C)CC2)=O)CC2(CCCN(C(c3ccnc(NCC(F)(F)F)c3)=O)C2)C1 c1(CC)cc(C(N2CCOC(CNC(C3CC(OC(F)(F)F)C3)=O)C2)=O)nn1C c1(CC)cc(F)c(C(=O)NCC(C)CNC(C2CN(C(N)=O)C2)=O)cc1F CC1(C)CN(C(=O)C(O)C(F)F)CCC1NC(c1ncn(-c2ccccc2)n1)=O CCC(F)(F)C(C)(C)C(=O)NCC(C)CNC(c1cnn2cc(C)cnc12)=O N1(C(CCCC=C)=O)CC2CCC(CNC(c3ccn(CC)n3)=O)C2C1 c1(C(=O)NC(CCOC)CNC(C2C(Cl)(Cl)C23CC3)=O)c(F)ccc(C)c1Cl N1(C(C2C(F)(F)C23CCC3)=O)CCCN(C(=O)C=CCOCC(F)(F)F)C(C)C1 N1(C(CCOCC#C)=O)CCC2(CCCN2C(c2ccnn2CCCC)=O)C1 C=CCCN=C(NCc1coc(C)c1)NCC1CCC(C)O1 CN1C2CC(CNCc3conc3C(C)(C)C)CC(O)C1CC2 c1(C(N2CC(NC(C(CC)SC)=O)C(C)C2)=O)csc(=NC2CC2)[nH]1 N1(C(c2ccnnc2)=O)CC2CCC(C1)N2C(c1c(O)cccc1F)=O C1(C2CCN(c3cnc(F)cn3)CC2)(NC(CC2CCN(OC)CC2)=O)CC1 C1(NC(c2cc(C)c(C)nn2)=O)CCC2CC1CN2C(C1(C2CCC2)CC1)=O CCC(C)(CO)NC(C1(NC(=O)Cc2nocc2C)CCCC1)=O N#Cc1cncc(CC(=O)NCC2CN(C(=O)CC3CC=CC3)C2)c1 c1(OCC(=O)NCC(CNC(=O)CC2(O)CC2)CO)ccccc1O N1(c2c(F)cnc(C)n2)CCC2(CCCCC2NC(C2(c3cccs3)CC2)=O)C1 N1(C(CC(CC)C2CC2)=O)CC(NC(c2cnc3n2CCC3)=O)CC1(C)C c1(C(C)C)nccc(=NC(=O)c2ccnn2C2CCCCC2)[nH]1 C#Cc1c[nH]nc1NCCC(N1CC(CNC(=O)C2CC2)OCC1)=O CC(C(C)(C)C)=CC(=O)N(C(C)CCNC(C1CC(CC(F)F)C1)=O)C(C)C.C1CC1 C(CC(=O)N1CC(CC)(NC2CC(CC(=O)OC)C2)C1)(C1CC1)SC CC(C)C(C(=O)N1CCCC(N(C(=O)CCCn2ccnc2)C)C1)NC=O N1(C(c2ccc(COC)o2)=O)CC(NC(=O)CCC2CCCN2C)CCC1C Cc1cc(N(C(C2COCCO2)=O)C(C)C)cnc1F.c12cccc(n1)NC2=O C1(CCNC(c2cccc(OC)n2)=O)CC(F)(F)CN1C(C1C=CC=CC=C1)=O CC(C)CC(CNC(c1cccc(N(C)C)c1)=O)NC(C1CCCCC1O)=O N1(C(C2(C(C)C)CCN(C(c3c(C)cns3)=O)C2)=O)CC(O)(C2CCCC2)C1 C(CCCCC(=O)N1CCOC(CNC(=O)C=Cc2cc[nH]n2)C1)OCC C(c1ccc2c(c1)OCO2)=CC(=O)NCC(C)CN(C(=O)C1=CCCOCC1)C c1(OC)ccc(C(N2CCCC(N(C)C(C3CC3CF)=O)CC2)=O)cc1Cl C(=O)(C(C)(C)CC(F)F)NCC(CC(=O)NCc1c(CC)nn(C)c1)C1CCC1 C1(C(N(C(CN(C(c2ncn(C(C)C)n2)=O)C)C)C)=O)CCC2(CCC2)C1 C1(NC(CCOC)=O)CCCN1C(=O)CN(C)Cc1ccccc1 Cc1nc2c(o1)CCCC2CC(=O)N1CCN(c2ncnn3c(Br)ccc23)CC1 N1(COC(C=C)C2CC2)CCCC(N2CCN(C(C)(C)C)CC2)C1 c1(NC(C)=O)ccccc1-n1cc(CN(O)C(C2CCCC(=O)O2)=O)nn1 C(C(=O)N(C)CCN(C)C(C1CCCN1C(=O)C(C)C)=O)(C(C)C)NC(=O)OC C(=O)(C(C)CC(C)(C)C)N1CC2C(NC(CNC(C(CC)CC)=O)=O)(C2)C1 N1(C(c2c(CC)n(CC)nn2)=O)CC=C(CCNC(=O)CCCC(F)(F)F)CC1 C1(C(=O)NCC(C)(COC)CC)(CC)CCCN(C(c2cnc(C)nc2)=O)C1 C(=O)(C#CC1CCCO1)N(C1CCN(C(c2ccc(C(C)C)o2)=O)C1)CC1CC1 N1(c2ccc(C#N)cn2)CC(NC(C2(C3CCC3)CCC2)=O)C2CCCCC12 N1(CC=C)C(=O)c2ccc(C(=O)NC(C)Cc3nc[nH]n3)cc2C1=O C(=O)(N=c1cc2ccccn2[nH]1)C1CN(C(CC(C)OC)=O)CC(C)(C)C1 c1(C(N)=O)cc(C(=O)NC2CCN(C(C3CN(C4COC4)C3)=O)C2)n[nH]1 C(C(C)(C(N)=O)NC(=O)NC1(c2ccccc2Br)CCC1)OC c1(C(=O)NCC2N(C(C=CC=CCC)=O)CC(O)C2)cccc2nccn12 C(=O)(C(C)CC(F)F)N(CC(CC)NC(C1CS(=O)C1)=O)CC C(=O)(C1CCc2ccccc21)NC1(CNC(c2ccc3c(c2)CN(C)C3)=O)CCC1 c1(CC)oc(C)cc1-c1nc(CCC(C)C)nn1CCC1CC1 N1(C(c2scc(C)c2)=O)CCCC(NC(=O)CC2CCCOC2)C1C c1(N(C2CCN(C(c3cc(COC)oc3C)=O)CC2)C)ccc(C#N)nc1 C#CCC(C(=O)NC)NC(c1cnc(CNC(=O)CC2CCCC(=O)N2)nc1)=O c1(CCC)cc(C(=O)NCC2(OC)CN(C(=O)C(C(C)C)SC)C2)ccn1 c1(OC)ccc(C)c(NC(c2c(CNC(=O)C(C(C)C)OC)nnn2C)=O)c1 c1(OC)ccc(Cl)cc1C(=O)NCC1CCC1NC(=O)C1=CCCS1 C1(C(C)C)CN(C(c2ccncc2F)=O)CCC1NC(c1cnn(CCF)c1)=O N=c1nc(O)cc(CC(N2CCCC2CNC(=O)COc2ccon2)=O)[nH]1 N1(C(C=C(CC)C)=O)CC2CC2(CNC(=O)C(C)(C)O)C1 N1(C(CC(C)n2cccc2)=O)CC2(CCNC(C3CCCN3C)=O)CCC1CC2 C(=O)(CCCCC(=O)NCC1(CCNC(=O)CCCC(F)(F)F)CC1)NC N1(C(C2CC(CC)C2)=O)CCCCCC(NC(=O)Cn2nc(C)oc2=O)C1 C(=O)(C#CC1CCOCC1)N1C2CC(CC(NC(CC3C(C)CC3)=O)C2)C1 C(=O)(CC(C(F)F)NC(=O)CCCF)NCc1cc(CC)[nH]n1 C(=O)(CC(F)(F)C(C)C)NC1CCN(C(c2c(C)nc(=N)[nH]c2)=O)CC1CO c1(C(=O)NC2COC3CN(C(=O)C=CBr)CC23)ccc2nonc2c1 c1(OC)cccc(C(C)C)c1F.N12CCC(C(Nc3ccccc3)C1)NC(=O)C2 CCS(=O)(=O)CC(=O)N1CC(CNC(c2cc(C3CC3)ns2)=O)C2(CC2)C1 c1(OCC)cccc(CC(=O)NC(CNC(=O)C(C)Cc2ccccc2)CC)c1 Cc1cc(C(=O)NCc2ccc(C(=O)NC3CSC(C)C3)cc2)nnc1O Cc1noc(C2CCCN2C(C2CC(n3cc(CCC4CCOC4)nn3)C2)=O)n1 C1(C(N(CCCCNC(c2cccc(OC(C)C)n2)=O)C)=O)OCCC12CCC2 c1(C(N2CCC=CC2C(=O)NC2CC(O)CC2O)=O)cc(F)ccc1F Cc1c(Cl)ccnc1C(=O)NC1COCC1NC(C1CC12CCC2)=O c1(C(N2C3C(C(N4CC(C)OCC4C)=O)C(C3)C2)=O)c[nH]c2cccc(Cl)c12 Cc1cc(O)ncc1C(c1nnnn1Cc1ccccc1)NC1(C)CC1(C)C CC1(C)CC(CC(=O)NC2(CO)CCN(C(=O)Cc3cccs3)C2)CCO1 C1(CC=C)(C(=O)OCC)CCN(C(c2cn(C(C)C)nn2)C(=O)NC2(C)CC2)C1 N1(C(c2ccc(CC)o2)=O)CC(NC(c2cscc2C)=O)C2CC12 C(C)(CCC(=O)N1CCN(c2ccc(CNC(=O)CCF)cc2)CC1)OC C1(CNC(c2nc(OCC)sn2)=O)CN(C(=O)CCC(C)CN(C)C)CC12CC2 C(C(CCCC)NC(C1(OCC)CCSCC1)=O)NC(C1CC(=C)C1)=O C(CCN=C(NCCC1CCCS(=O)(=O)C1)NCC(=O)OC(C)(C)C)SC c1(C(=O)NC2C(CNC(c3cc(=N)[nH]c(Cl)n3)=O)C2)c(O)nnc2c1COCC2 c1(NC(N2CC(n3ccnc3)C2)=O)cnn(Cc2cnco2)c1 C(CN=C(NCC(=O)NC1CC(Cl)(Cl)C1)NC1CCS(=O)(=O)C1)SC CCC(C(=O)NCC(O)CNC(c1ocnc1C)=O)OC1CCCCC1 C12(C(=O)NCC(CCOC)NC(c3ccncn3)=O)C3CCC(CC13)C2(F)F Cc1cc(C#N)sc1C(N1CCN(C)CC1CNC(c1cnccc1Cl)=O)=O C#Cc1cnc(C(N2CCCCC2CN2CC(C)(CC(=O)OC)C2)=O)c(C)c1 Cn1cc2ccc(NC(C3CC(O)CCN3Cc3ncccc3N)=O)cc2n1 N1(C(c2n[nH]cc2Br)C(=O)NCCSC)CCC(S(=O)(=O)c2ccccc2)CC1 C(=O)(CC(C)(C)C(=O)NC1CCN(C(=O)CNC(=O)NC)CC1C)OCC C(=O)(CS(=O)CC)N1CC(C(C(=O)NCCc2ncnn2C)OCC)C1 c1(NCc2c(C)nc(CCC)o2)nccc(=NCC2CC(C)(C)C2)[nH]1 c1(OC)ccc(C(C)N)cc1.n12cc(cn1)CN1CCC(C1)NC2=O c1(C(=O)NCC(CC=C)NC(c2cc(C(F)F)cc(F)c2)=O)ccc(N)c(F)n1 C(CC(CC)C(=O)N1CCC(C(N2CC=CC2CN(C)C)=O)CC1OC)=CC c1(OCC)cc(C(=O)NC2(C)CCN(C(=O)COC3CCC3)C2)cc(Cl)c1O c12ccc(cc1)CN2CC.N1(CC(N(CC(=O)NC)CC)=O)CC=CC1 Cc1nnc(CC(=O)NCCC2CCC(NC(=O)Cc3nncn3C)C2)o1 c1(C(=O)NCCC2CCC(NC(C3(CCCC)CC3)=O)C2)csc(C#N)c1 C1(OC)CCCCN(CC(=O)NCC(C)(Cc2ccccc2)C(C)O)C1=O C1(NC(C2C3CCC(F)(F)C23)=O)CN(C(C2SCCS2)=O)CC12CC2 c1(OC)cccc2cc(C(N3CCCC3CCCNC(C3CC3(F)F)=O)=O)[nH]c12 C1(NC(=O)COCc2ccccc2)CN(C(=O)C(F)(F)CO)CC1O CC1(N2CCC(O)(CO)CC2)CC2C=CC1C2 C1(NC(c2nn(C)c(O)c2)=O)CC2CCC1CN2C(=O)C(O)CC1CC1 Cc1ccc(C)c(F)c1-c1ccc(C=O)cc1Sc1ccc(CCc2cc(F)c(OC)cc2F)nc1 C12(NC(C(CC)C)=O)COC(C1)C(NC(c1ccc(F)cc1OC(F)F)=O)C2 N1(C(C2C(NC(=O)C(C3CCCCC3)O)CC2)=O)CCC(CC2CC2)CC1 c1(C(N2CC(C(C)NC(=O)C(C)C(F)F)C2)=O)ccc(OCCF)cc1F c1(C(=O)NC(C2(O)CCN(C(c3cc4c(s3)CCC4)=O)C2)C)cnc2n1CCC2 N1(C(CCN(CC#C)C(C2CCC(=O)N2)=O)=O)CCC(C(C)C)CC1 C(=O)(C(C)S(N)(=O)=O)N1C2C(C(=O)NCC(c3ccncc3)C)C(C2)C1 c1(C(=O)NC(C2CN(C(C3(O)CCC3)=O)C2)C)cccnc1-c1nncn1C c1(OC)cc(=NC(=O)C=CCC(C)(C)NC(=O)C(O)C2CC2)[nH]n1C c1(C(C(=O)NCCC#N)N(CC)CC2CC2)cnc(C)s1.n1(CN)cc(Br)cn1 C(C(C)=CC(=O)N(C)CCN(C)C(C1CC1Cl)=O)NC(C)=O n1(CC(=O)NC2(CNC(C3(C)CC3C(F)(F)F)=O)CCC2)cnc(=N)[nH]1 C1(NC(C(CSC)O)=O)CC2(CCN(C(c3cccc(CO)c3)=O)CC2)C1 C1(NC(N(CC)Cc2ccco2)=O)COCCN1Cc1ccc(F)cc1 C1(NC(c2cc(C(C)C)no2)=O)CCCC12CN(C(C1CC(O)CN1C)=O)C2 C1(C(N2CC(NC(c3ccc(C4CCC4)nc3)=O)C2)=O)C2CCCCC12 c1(NC(c2ncc(S(=O)(=O)N3CCCCCC3)s2)C)cc(N)cnc1Cl c1(C(=O)NCC(CC)(CC)SC)ccc(C(=O)OC)c(OC2CC2)c1 c1(C(=O)NCC(CCCC)NC(=O)CC2(OCC)CC2)cc(N)ccc1CC Cc1csc(=NCC(=O)NC2(CO)CN(C(C3CC4(C3)CC4(F)F)=O)C2)[nH]1 C1(NC(c2ccc(OCC#N)cc2)=O)CCCCN(Cc2cccc(Br)n2)C1 CS(=O)(=O)C1(CN2CCC(C3CCCCN3Cc3c(F)cccc3F)C2)CCC1 C1(C(C)NC(CCSC)=O)CCCN(C(=O)Cc2nc(C3CC3)nn2C)C1 c1(C(N2CC3C(NC(c4nncc(OC)c4)=O)(C3)C2)=O)nnc(O)nc1O C1(N(C(c2nocc2C)C(=O)NCC(=C)C)C)CCCC(C(N)=O)C1 c1(C(N2CCC3C(NC(c4cc(CC)c(C)s4)=O)C32)=O)cc(N)cnc1Cl c1(C(N2C(C(N3CCC(OCCC)C3)=O)C=CC2)=O)ccc(C2CCCC2)nc1 c1(OC)ccc(CN(c2ccc(OC3=CC=CC=CC=C3)cc2)CCC#N)cc1 Cn1cc(C(=O)NCCn2ccc(C(N3CCC(CCO)C3)=O)c2)nn1 c1(CC(N2C(CNC(C3N(C=O)CCC3)=O)CC2)=O)cc2ccccc2oc1=O c1(C(C(=O)NCC2N(C(c3n(CC)ccc3)=O)CC2)O)ccccc1F c1(CC)ccc(F)c(C(=O)NCC2CCCC(NC(c3[nH]ccc3C)=O)C2)c1F Cc1cc(C(=O)NCc2ccc(C(=O)NC(CC3CCC3)CO)cc2)c(C)s1 c1(CNC(C(COC)OC)=O)cccc2c1CCN(C(=O)COCCC(C)C)C2 C1(CNC(CCCCC#C)=O)CN(C(=O)CCCCOCC)CC(C)(C)O1 N1(C(c2ccc(SC)o2)=O)CCCC2(NC(=O)CC3(O)CCCC3)CC2C1 N1(C(C)=O)CCC(CCNCc2ncc(C(C)(C)C)s2)c2ccccc21 c1(OC)cnc(F)c(C(=O)NC(C)(C)CNC(C23CC(CO)(C2)C3)=O)c1 CN1CCN(C(=O)Cn2ccccc2=O)C(C(=O)NCCCSC(F)F)C1 N1(C(c2cn(CCC=C)nn2)=O)CC(C2CN(C(C3COCCC3C)=O)C2)C1 C1(N(C(CCCOCCC)=O)C)CN(C(=O)Cn2cnc(C#N)n2)CCC1C CCCCC(C(=O)NC1CCC1C(=O)NCC(C)C1CCC1)NC(N)=O C1(C(=O)NCC(CC)NC(c2c(Cl)nn(C)c2Cl)=O)CCCNS1(=O)=O c1(OC)ccc2c(C(=O)NCC3CCN3C(=O)C3=CCSC3)ccnc2c1 Nc1ccc(Cl)cc1C(=O)NCC12CC(NC(c3c[nH]nc3C3CC3)=O)(C1)C2 C1(C(N(CCCC(=O)NC)C)=O)CCN(C(c2cccc(C)c2C)=O)CC1(C)C N1(C(C2(CC)CC2)=O)CC2CC2(C(=O)N(c2ccc(O)cc2)C)C1 c1(C(=O)NC(C(C)NC(c2ccc(CC)o2)=O)C)cc2c(Cl)c(OC)ccc2[nH]1 c1(C(=O)NCC2CCN(C(C3C4CCCCC34)=O)C2)cc2cccnc2o1 c1(SC)ccc2sc(CN(C)CCCCCN)nc2c1 C1(C(C(=O)NCCN(C(c2c(SCC)cccn2)=O)CC)O)CCCCCCC1 Cc1cc(C#N)cnc1C(=O)NC1(C(=O)NC(C)C(C)n2cccn2)CCC1 c1(C(=O)Nc2nc(C)cc(C)n2)ncn2cc(-c3cncn3C)sc12 C1(F)(C(N2CC(NCc3cn(C)nc3)OCC2)=O)CCCCC1(F)F CC1(CCC(=O)NCCCNC(=O)CN2CC3C=CC2C3)NC(=O)NC1=O Cc1c(C(=O)NC(C)CNC(=O)COCc2cccnc2)cccc1O c1(C(N2CCC(N(C(C(CC)F)=O)C)CC2)=O)nc(-c2ccccc2)ncc1Cl c1(C(=O)NCCC(C)NC(C2C(SC)CCC2)=O)ccc2nc(O)cc(O)c2c1 C1(OC)CC(CCNC(C2COCCN2CC)=O)N(C(C2(CC(C)C)CC2)=O)C1 N1(C(C2(C)C(C)(C)C2)=O)CCC(C)(CNC(c2cnn(C(F)F)c2)=O)C1 C1(F)(C(N2C(CCNC(c3cc(COC)sc3)=O)CCC2)=O)C(C)(C)C1(C)C c1(C(C)NCCCCCCCl)cc(Cl)ccc1Cl C1(C(=O)NCC(CC=C)(C)CO)CCC(C)(C)N(C(=O)C=Cc2cn(C)cn2)C1 N1(C(CC)=O)CCC(C(=O)N(CC(C)CNC(=O)CC2(C(F)(F)F)CC2)C)CC1 c1(C(N2CC(NC(C#CC(C)(C)C)=O)C(F)CC2)=O)ccc2cncn2c1 c1(C(N(CCCN(C(=O)CN(C)C)C)CC)=O)cn(CC(=O)N(C)C)nn1 C1(C(C)NC(COCCCC)=O)CCCN(C(=O)CNC(=O)NC)C1 C1(CCOC)(NC(c2c[nH]nc2F)=O)CCN(C(=O)Cn2ccnn2)C1 c1(C(=O)NC(CNC(C2(C)CC2Br)=O)C2CC2)cc(O)cc([N+](=O)[O-])c1 c1(OCC(=O)N(CC(C)N(C)C(C2CCCC2O)=O)C)ccsc1Cl C1(NC(c2c(CC)scc2)=O)CC2CCC1N2C(=O)C(C)OCC1CCCO1 C1(C(=O)NC(C=C)C2CC2)CC(N=[N+]=[N-])CN1C(c1c[nH]c(C)c1)=O N1(C(C2C(C)CCS2)=O)CCN(CCCNC(C2C=CCS2)=O)CC1 CC(CC(=O)N1CCCC1(C)CNC(c1ccc(O)nc1Cl)=O)C(F)F C1(C(N2CC3C(CNC(c4ccon4)=O)C3C2)=O)(CC)CCNC1=O C1(C)(C(=O)NC(CC)CNC(=O)C(C)CC2CCC2)CCC(F)(F)C1 n1(CC2N(CCCOc3c(F)ccc(F)c3)C(=O)CC2)nnc2ccccc12 Cc1ccc(C(C)NC(=O)N(c2ccsc2C(F)(F)F)CC2CC2)cc1 C(=O)(C1=CCC(C)CC1)Nn1cc(C(C)NCc2cccc(C(C)=O)c2)nn1 CCC(CC)(CCNC(=O)CC1CCCC(=O)N1)NC(=O)CC1OCCCC1(C)C C(C)(N=c1[nH]c(N2CCC(N(C)C)C2)nc2cc[nH]c12)c1scc(C)n1 C1(CC)OCCC1C(=O)NCC(C)(C)CN(C(=O)C(C)NS(C)(=O)=O)C Cc1oc(C(=O)NC2CC(CCNC(=O)CCC3CCCO3)C2)cc1CO n1(CC(N2CCC(CC(C)NC(CCCOC)=O)CC2)=O)cnc([N+](=O)[O-])n1 CN1CC(C(N2CC(CNC(c3ccc[n+]([O-])c3)=O)C2)=O)C(C(F)(F)F)C1 N12CC(C(O)C1)N(C)CC1(CC1)CC2=O.C(=O)(CCCc1ccncc1)OC CC#CCCCC(=O)N1CC(NC(=O)CSCCN(C)C)CCC1C c1(N2CCC(=CC(=O)Nc3cnn[nH]3)CC2)ccncc1[N+](=O)[O-] c1(C(=O)NC2CC(C)N(C(=O)CC3CCCOC3)CC2)cc2n(n1)CCCO2 CC(C)(C)C(O)C(=O)N1CC2(CC(N3CCC(F)(N(CCCO)C)CC3)C2)C1 CC1CCC(=CC(=O)NC(C)(CNC(C2(n3cncn3)CC2)=O)C(C)C)CC1 N1(C(C(=O)NC)=O)CCCC1C(=O)N(CC(C)(F)F)C Cc1cc(O)ncc1C(=O)NCCN(C(=O)CC1COC2CC1C2)CC1CC1 n1(CC(=O)NC2CN(C(C3(CN(C)C)CC3)=O)CC2F)cnc([N+](=O)[O-])n1 C1(C(N(CC(c2ccccc2)N)C)=O)COC2(CCOCC2)O1.CCN CC1(C)CCN(C(c2cnc(C3CC3)o2)=O)CC1CNC(c1ccc(CO)nc1)=O N1(C(C2CC3(CCC3)CO2)=O)CCCCC1C1CCCN1c1cc(Cl)c(O)nn1 Cc1cccc(C)c1C(O)C(N1CCC(C2CCCN2Cc2ccns2)CC1)=O C1(NC(c2ccccc2)=O)CN(C(=O)CC(F)(F)Br)C2(CCC2)C1 c1(C(c2ccccc2)NC2C(NC(=O)C=CCF)CC2)ccc2c(c1)OCCO2 N1(C(C=CC(=O)OC(C)(C)C)=O)CC2CC2(NC(=O)CC(O)c2ccccc2)C1 c1(NCc2c(C)sc3ncccc32)[nH]c(=NC2CCCCCC2F)nc2ncn(C)c12 C1(C(N(CCCNC(C2(Cl)CC23CCC3)=O)C)=O)CC2(CCOCC2)C1 N1(C(c2cc(C(C)C)on2)=O)CC(CNC(c2cnc(=N)[nH]c2)=O)C(C)C1 N1(C(=O)Nc2cc(C)c(F)c(N)c2)CC2(CC(S(C)(=O)=O)C2)C1 C1(NC(COCCOCC)=O)CCCC12CCN(C(c1nnn(C)c1N)=O)CC2 Cc1ccc(C(CC2CC2)NC(C2CC(NC(=O)CCc3ccnn3C)C2)=O)cc1 C(=O)(NNCC(F)F)NC1(C(=O)OC(C)(C)C)CCOC1 C1(NC(C2(CCOC)CC2)=O)CCC2CC1CN2C(=O)C=Cc1nc(C)cs1 C1(NC(C(C(C)C)C)=O)CC(F)CN(C(c2ccc(CC(N)=O)cc2)=O)C1 C(=O)(C1=NNC(C(F)(F)F)C1)NCC(C1N(C(C(CC#C)C)=O)CCCC1)(C)C c1(NC2CN(C(=O)CC3CCS(=O)(=O)C3)C2)ncnc2c1CCC2 S(=O)(=O)(c1ccc(C(CC(=O)O)NC(=O)CCNC23COC(C2)C3)cc1)N(C)C N1(C(CS(=O)(=O)NC)=O)CCC2CCN(c3ncc(C)c(C)n3)CC2C1 c1(-n2cc(CC(C(N)=O)NC(C(C=C)OC)=O)nn2)cn2nccc2nc1C c1(C(=O)NC(C(C)(C)C)CNC(C2COCCO2)=O)ncnc2sccc12 C=CC1(CC(=O)NCC(c2cccnc2)O)CN(C(=O)CC2CC3C=CC2C3)C1 N1(C(C=NOC)=O)CCCCC1C1CCN(C(=O)C(C)Cc2c(C)noc2C)C1 N1(C(C(C)N2CCC2)=O)CCOCC1C(=O)NCc1ccc(NC(CC2CC2)=O)s1 Cc1[nH][nH]c(=NC(=O)C23CC2CN(C(=O)Cc2cccc(O)c2)C3)c1C C1(c2nn[nH]n2)(C(N2CC(OC)(CF)C2)=O)CC2(CSC2)C1 c1(C(N2CC(SC)C(NC(C3CCCCC(=O)N3)=O)C2)=O)cc(C)cc(F)c1N N1(C(N(CCCN(C(=O)Cc2cccc(Br)n2)C)C)=O)CCC(C)(O)C1 c1(C(C(=O)NCC(CNC(c2cncc(C)n2)=O)C)O)ccc(O)c([N+](=O)[O-])c1 CC1(C(=O)NC2CCC(NC(=O)CCSC(F)(F)F)CC2)CCC12CCC2 C1(C(=O)NC(C)C(=O)N(CC(F)F)CCO)CC2CC(=O)C1C2 Cc1nc(C(=O)NC(CNC(=O)C(C)Oc2ccccn2)C2CCC2)cs1 C(C(=O)N1CCCC(C)(CNC(=O)C2=COCCC2)C1)(c1ccccc1)=C(C)C N1(C(C(CC)=CC)=O)CC(CNC(=O)C(C(C)C)N(C)C)CC12CCOCC2 N1(C(CCCNC(C2C(OC)CCC2)=O)=O)CCN2C(=O)CCC2C1 CC(F)(F)CC(=O)NCC1(C)CC(NC(=O)C=Cc2cscn2)C1 Cc1c(NC(=O)CC2(C)CN(C(=O)COC3(C)CCC3)C2)ccc(Br)c1Cl N1(C(CC(C=C)CC)=O)CC(NC(C2CCC(=O)N(C)C2)=O)CC12CCOCC2 c1(C(=O)NCC2(OC)CC2)cc(CNC(=O)C(C)n2ccnc2)[nH]n1 Cc1c(CC(N2CCC(CF)(NC(=O)Cc3cnc[nH]3)C2)=O)cccc1Br Cn1cnc2cccc(C(N3CC(NC(c4cccnc4S)=O)C4CC34)=O)c12 C12(C(=O)NC3CN(C(CCc4ccn(C)n4)=O)CC(O)C3)CCC(F)(CC1)CC2 N1(C(c2nc(CC)oc2)=O)CCCC2(CCN2C(c2cc(Cl)ccn2)=O)C1 C1(C(=O)O)CN(C(=O)CCBr)CC12CN(C(C1CCCO1)=O)C2 CC(C)C(F)(CNC(C1C2CCC3C(C2)CC13)=O)C(=O)NC1(C2CCCCC2)CC1 C(CC(F)F)(C(=O)N(C)CCc1ccncc1)NC(CCC(C)OCC)=O c1(C(=O)NCC(C)(C2CC2)NC(c2cc(COC)[nH]n2)=O)cnc(O)n(C)c1=O Cn1cc(CN=C(NCC(F)F)NC2CCC2)c(C(F)F)n1 C1(C(N2C(CNC(C(C(C)C)N(C)C)=O)CC(O)C2)=O)CC(=O)NC(=O)C1 N1(C(C(C)(C)F)=O)CCCC(F)(CNC(C2(Oc3cccc(Cl)c3)CC2)=O)C1 C12(C(=O)NC3(CC=C)CCCC3)CC(CO)(CN1C(c1cnco1)=O)C2 C#Cc1ccc(C(=O)Nc2c(C)cnn2CC)cc1C c1(OC)ccc(CC(=O)NCCN(C(=O)CC(C)(C)OC)C)c(OC)c1 c1(C(N2C(CNC(C3(C4CCCCC4)CC3)=O)C=CC2)=O)cncc2n[nH]cc12 c1(C(=O)NCCNC(c2ccncc2Cl)=O)oc2ccccc2c1Cc1nn[nH]n1 c1(CC(=O)NCC(CCOC)NC(C2CCC(=O)NC2)=O)cc(C(F)(F)F)n(C)n1 C=CCCC(C(=O)O)NC(=O)Nc1ccc(CO)c(COC)c1 C1(NC(C(CO)N(C)C)=O)CCCCN(C(c2ccc(F)cc2)=O)C1 c1(C(=O)NC(C(C)NC(=O)Cc2ccc(CO)c(F)c2)C)c(O)cc(F)cc1F Cc1ncnc(C)c1C(=O)NCCC(C)NC(C1(CC(C)C)CCCC1)=O C1(NC(C2(c3cccc(F)c3F)CC2)=O)CC2CC(NCc3c(C)ocn3)C2C1 c1(N2CC3N(C(C(c4ccccc4F)C)=O)C(C3)C2)ncc2cn[nH]c2n1 N1(c2ccnc(NCCC(=O)Nc3c(Br)ccc(F)c3)n2)CCc2sccc2C1 c1(Sc2n(C)ccn2)ccc(C2(NC(=O)NC(c3ccccc3)=O)COC2)cc1 CC1(C)CC(=O)NCC1NCCCN1CCOCC1.N12CC(CC1CO)C2=O c1(CN2CCC(C#N)(C(N3CCC(C)(O)C3)=O)C2)ccc2cc(O)ccc2c1 c1(C(C(=O)NC(CNC(c2c(C)noc2N)=O)C)C)cc2ccccc2o1 c1(C(=O)NC2CCCN(C(c3c(OC)cccc3)=O)C2)sc(C)c(C)c1C N1(C(C2C(CC)CCN2C(=O)C=CCN2CCC2)=O)CCc2nc[nH]c2C1 CC1CN(C(=O)C(c2cc(F)cc(F)c2)C)CCCN1C(=O)CCC(C)(C)C N1(C(C(N2CCC(C(=O)OCC)(C)C2)=O)=O)C2CCCC1CC(F)(F)C2.C(C)(C)(C)N C=CCC(CC(F)F)C(=O)NCC1CCC(C)(C)CN1C(=O)CC1CCCN1C C1(C(N2CC=CC(NC(Cc3nn(C)c(Cl)c3)=O)C2)=O)CCCC(F)(F)CC1 C(=O)(CCC(CC)CCC)N1CCC(N(C(=O)C=CC=C)CC#C)CC1 c1(C(=O)NCC(c2ccccc2)CNC(C=C=C(C)C)=O)cn2cccnc2n1 c1(N2CC(NC(c3c(C)nn(C)c3)=O)C(C#N)C2)ncnc2c(C)cccc12 C#CCCCCC(c1nnnn1C1CCCCC1)NC(=O)CCc1ccc(C)cc1 CCCCCCC(O)CCC(=O)N(CC(O)CN(C(=O)C=CC=C(Cl)Cl)C)C N1(C(c2nc(C)sc2C)=O)CCOCC(C(=O)NC(c2nc(=O)o[nH]2)C)C1 n1(CC(=O)NC2CC(CNC(CCCCNC(C)=O)=O)C2)c(C)cc(C)nc1=O N#CCCCCC(=O)NC(CCOCCO)C(=O)NCCC1CC(F)C1 C12CN(CC1CC(=O)OC(C)(C)C)C(=O)N2.c1(C(C)NC(C)=O)ccsc1 C1(C(N2CCC(OCC)C2)=O)CCCCCN1C(c1ccco1)=O C1(C(N(CC#C)C)=O)CCCN(C(c2cccc(CC#N)c2)=O)C1 N1(C(C=COCC)=O)CCCC2CCN(C(=O)CCc3ccc(Cl)s3)CC12 N1(C(C2CC(CC)C2)=O)CCC1(C)CC(=O)NCC1CCCO1 C1(CC(=O)N(CC(=O)NCCOCC#C)CCC)CCC2CC12 c1(SC)cc(C(=O)N(C(C)(C(=O)NCCCCC2CCCO2)C2CC2)C)co1 O=C(C(O)C(F)(F)F)NCC1CC2CCC1N2C(c1ccnc(CO)c1)=O N1(C(CSCC=C)=O)CCC(CNC(c2cnc(C(F)F)nc2)=O)CC1C c1(C(=O)Nc2ccccc2Br)cc2ccc(-c3cc4ccccc4o3)nc2[nH]1 C1(O)(CNC(C(C)CC2CC2)=O)CCN(C(C2CC3(CCC3O)C2)=O)CC1 c1(C(N2CC(CNC(c3cncnc3C3CC3)=O)C2)=O)cc(OC(F)F)ccc1F n1(C2CCCN(CC=C(C)c3ccsc3)C2)cc2ccccc2n1 C1(NC(CC(CCC)C)=O)CN(c2ncc(I)cn2)CC12CCOCC2 N1(CCC(N2CC(O)CC(NC(COC)=O)C2)=O)CCCc2ccccc21 c1(C(=O)NC(c2cc(Br)ccc2Br)C)c(F)cc(Br)cc1Br C12(CNC(CCC#C)=O)CCCCC1CN(C(=O)C(C)(C)C1CCC1)C2 Cc1nc2sccn2c1C(=O)NCCN(C(c1ccc2cnsc2c1)=O)C(C)C C(C(CC(F)(F)F)NC(=O)CC1CC(C)(C)C1)NC(C(CC)O)=O C1(NC(c2cncc(C)c2C)=O)CC2(CCN(C(c3cnc(S)[nH]3)=O)C2)C1 N1(C(CCCC=C)=O)CCCCC(CNC(=O)C(C)S(C)(=O)=O)C1 c1(COCC)ccccc1CC(N1CCCC1CNC(=O)C(C)CN(C)C)=O N1(C(COCC)=O)CCC2(CCCN(C(=O)Cc3c(C)noc3C)C2)C1 CC1=NOC(C)(CNC(C2C=CCN(C(=O)C(c3cccnc3)O)C2)=O)C1 CCC(O)C(C)C(=O)NCCC1(NC(=O)CNC(c2ccc(Cl)cc2)=O)CC1 C(=O)(C#CC(C)(C)CNC(=O)CNc1ncccn1)NC1CC(C)OC1=O C1(C(=O)NC(CC)CNC(c2coc(C)c2)=O)CC(=O)N(c2cccc(Cl)c2)C1 c1(C(=O)NCC2OCC(CNC(C=C(CCN(C)C)Cl)=O)C2)cccc(N)c1 C(=O)(C(Cc1ccoc1)NC(=O)CC1CCCC1)N(CC)CC1CCOC1 c1(C(N2C(CC)CN(C(=O)CCCC(C)C)CC2)=O)nc(Cl)ccc1F c1(OCCC(=O)NCC2CC2NC(=O)Cc2ccco2)cccnc1 C=Cc1ccc(C(N2CC(C(=O)NCCCCN(C)C3CC3)C3(CC3)C2)=O)cc1 C(=O)(CCC(C)(C)F)N1C(C2(O)CN(C(C(C)CCOc3ccccc3)=O)C2)C1 Cc1c(Br)noc1C(=O)NC1CCCC1NC(=O)C(N1CCOC1=O)C C12(C(N3C4C(NC(CCc5ccc(OC)cc5)=O)C(C4)C3)=O)CCC(CC1F)C2 c1(-c2ccc(OCCC)nc2)ccc2c(C(=O)NCc3cnc(O)[nH]3)n[nH]c2c1 CCC1=NOC(C(=O)NCC2CCN(C(=O)NC(c3ccco3)C)CC2)C1 C(C1=NOC2CN(C(c3cc(C(F)F)[nH]n3)=O)CC12)NC(C=CC(C)(C)C)=O C#CCCCCC(=O)NCC1CC(F)CN1C(c1cccc(N(C)C)c1)=O N1(C(CCCSC)=O)CCC(C(=O)NC(C)Cc2cnc[nH]2)=C(F)C1 c1(N2CCN(CC)CC2)ccc(S(=O)(=O)NCC2CC3(CCC3O)C2)cc1Cl c1(C(N2C(C)CCC(NC(C(CCC#C)O)=O)C2)=O)oc2c(Cl)cccc2c1C C1(NC(c2n(CC=C)ccn2)=O)CCN(C(c2ccsc2Cl)=O)C1C C1(O)(C(C(=O)N(CCC(=O)NC)C)F)CN(C(C2COCOC2)=O)C1 C1(CC)CN(C(C2OCC3CCCC23)=O)CCN1C(=O)C(O)C(C)C C(Cc1ccsc1)(C(=O)N(CCCCNC(=O)Cc1ccc(C)o1)C1CC1)NC=O C1(CNC(C(CCC)CC)=O)CCCC12CCN(C(C1(C#N)CCCC1)=O)CC2 CC1CN(C(=O)C(C)(C)C2(O)CCC2)CCC(c2ccccc2)O1 c1(CCC(=O)N(CC#C)CC=CNC(=O)CC)nc(-c2ccc(C)s2)no1 N1(C(CNC=O)=O)CC2OC(C1)CNC2=O.c1(CO)nc(OC)cc(OCCO)n1 CCC(O)C(F)(F)C(=O)NCC1(OC)CN(C(c2cc(Cl)ccc2F)=O)C1 N1(C(=O)NCC(C)(C)Oc2ccccc2Br)CCC2(CCC(O)C2)C1 N1(C(Cn2c(C(C)C)ncc2)=O)CC2C(CNC(=O)CN(S(C)(=O)=O)C)C2C1 c1(C(=O)NC2(CNC(c3cc(-c4cccs4)[nH]n3)=O)CC2)c[nH]nc1F Cc1cc(N)c(C)nc1C(N1CCC(O)(C(C)NC(c2ccn(C)n2)=O)C1)=O N1(C(Cc2cc(C)on2)=O)CCCC(CC(N2CCC2C(=O)N(C)C)=O)CC1 N1(C(COCCCC)=O)CCCC1(C)C(=O)NCC1OCCC1C c1(OC)ncnc(OC)c1C(=O)N(CCCCNC(=O)CN(C)C)C C1(NC(CCSC)=O)COCCN(C(c2ccc(OC(C)(C)C)cn2)=O)C1 CCCCCC(C)CC(=O)NC(C)CNC(c1cc(-c2cnn(C)c2)no1)=O CN=c1cc(C(=O)NCC2(CNC(C3CCCCC3O)=O)CC23CCC3)cc[nH]1 Cc1c[nH]c(C(N2CCCC2(C)C(=O)NCCN2CCOCC2)=O)c1C Cc1ncc2n1CCOC2C(=O)NCCCCN(C)C(C12CCN(CC1)CC2)=O Cc1ncc(C(N2CC=CC2CNC(c2cn(C(C)(C)C)nn2)=O)=O)cn1 c1(C(=O)NC(C2CCN2C(=O)C(C2CCOCC2)F)C)cnoc1-c1cnc[nH]1 N1(C(CCC#C)=O)CC2CCC1CN2C(C1CCCN1c1ccccc1)=O C(=O)(C1CN(CCN2CCN2CC)c2ccccc21)NCN(CC(=O)OC(C)(C)C)C N1(C(C(C2CC2)OCC)=O)CC=C(C(=O)Nc2ccc(C)c(O)c2)CC1 CC(C(=O)NC1COCCN(C(C23CC(C2)C3)=O)C1)S(N)(=O)=O CC(CC(=O)N1CC2CC(NC(C3(n4cccn4)CC3)=O)C2C1)CC(C)(C)C N1(C(=O)NCC(C)OCC=C)CCC(c2ccnn2C)C1 Cc1c[nH]c(C(=O)NCCOCCC(=O)NCC2(C)CCOCC2)c1C C(CN=C(NCC1CC2CCC1O2)NCC(C)NC(=O)OC)SC c1(OC)ccc(C(N2CCN(C(C)Cn3cc(C(C)(C)O)nn3)CC2)=O)cc1Br C(=O)(C(C)CN(C)C(C1CCCC1OC)=O)N(CC)Cc1ccoc1 CCCC(CC)C(=O)NC1(C)CC(NC(c2cscc2F)=O)C1 C(=O)(CCCC(F)(F)F)NC(C1(C(=O)Nc2ccc(-c3ccon3)cc2)CC1)C Cc1cc(Cl)ccc1SCC(=O)NCCC1CCC(C)N(Cc2ccccc2)C1 CCCCC(CNC(=O)CN(C)C(C)C)NC(c1sc(C)nc1C)=O N1(C(c2c(C)cno2)=O)C2CCC(C2)C1CNC(c1ncsc1C(F)(F)F)=O C(=O)(C(C#N)C(C)(C)C)NC(C1CCN(C(COCCC)=O)CC1)C c1(C(=O)NC2CCCN(C(CC3CCN(C)C3)=O)C2)ccc2nn[nH]c2n1 c1(C(C)C(=O)NCc2csc(CCP(C)(C)=O)n2)cccc(I)c1 N1(C(c2nc(CC)oc2)=O)CCCCC1C1(NC(=O)CCc2cc(Cl)no2)CC1 c1(C(=O)NCC(C)(C)NC(Cc2ccc(C)c(O)c2)=O)cn2cccc(Cl)c2n1 Cc1ccc(CCC(N2CCC(CN(C(=O)CCC(C)(C)F)C)C2)=O)cc1C C1(NC(c2ccc(F)c(C(F)(F)F)n2)=O)CCC2(CCNC2)C1 CC(C)CCCC(C)C(=O)NC1C=CCN(C(c2cncc3nc[nH]c23)=O)C1 c1(COC(C(c2ccccc2)OCCC)=O)cc(Cl)c(F)c([N+](=O)[O-])c1N C1(C(=O)NC(c2cn(C)nn2)C(=O)N(CC(C)C#N)CC)CCCC(C)(C)C1 C1(NC(c2c(CCC)nns2)=O)(CC)CCN(C(C2CC(C#N)C2)=O)CC1 C(CC(C)(C)C(=O)N1CCC(C)(CCNC(C2CC2C(F)(F)F)=O)C1)OC c1(CC(C)SC)nc(-c2cccc(Cl)c2)nn1CC1COCCO1 N1(C(c2c(C)nc(O)cc2)=O)CCN(C(=O)CCCC(=O)NC(C)C)C2CCC12 c1(CNCCNC(C)=O)cccc2nc(C(F)(F)F)sc12 N1(C(COC(CC)(C)C)=O)CC(C(N2CCOC(CF)C2)=O)C2(CC2)C1 c1(C(N2CCCC(N(C(CNC(CC)=O)=O)CC)CC2)=O)nccc2nn[nH]c12 C(CCC1CC1)(C(=O)N(C)CC1CCSC1)NC(c1cc(C)no1)=O C(=O)(C(C)(C)C(=O)N1CC=CC(NC(=O)Cn2cc(Cl)cn2)C1)N(C)C N1(C(=O)C=Cc2cncs2)CC(N=c2nc(O)c(Br)c[nH]2)C2(CCC2)C1 C1(C(=O)NCCn2cc(C(=O)C3CC3)nn2)CCCN1C(c1cn(C(C)C)nn1)=O C(=O)(C(CCC(C)(C)C)N(C)Cc1ccc(N(C)C)cc1)NCC c1(C(=O)NCC2N(C(CC)=O)CCCC2)cc(Cl)ccc1N.C12CCCC1N2 C(=O)(C1=CCN(C)C1)NCC1(CCC(=O)NCCNC(C)=O)CCCC1 CC(C(=O)N1C(C(=O)NCC(O)C(C)O)CCC12CC2)S(C)(=O)=O N1(C(C(CNC(c2cc(C)ns2)=O)O)=O)CC(F)(F)CCC1C c1(OC)cc(C(N2CC(CNC(=O)C(C)=C3CCCC3)CC2C)=O)cc(F)c1F CP(C)(=O)C1CCC(C(=O)NC(Cc2cc[nH]n2)C(=O)O)C1 c1(C(N2CCC(CNC(C3(CC#C)CC=CCC3)=O)CC2)=O)n[nH]cc1[N+](=O)[O-] C#CCCCC(C)C(=O)NCC1CC(C(=O)NC2CCCCCC2(C)C)=NO1 C1(c2nnnn2C)(NC2C(C#C)CCC2)CNCCC1C C1(CC)CCCCN1C(C1CC(NC(C2(CC)CC2)=O)C(O)C1)=O c1(C(=O)NC(c2ccccc2)=O)ccc(CCc2snc(C(C)C)n2)nc1 C1(C(N2CCCCC(NC(CN(C)S(N)(=O)=O)=O)C2)=O)CCn2nncc2C1 C12(C(N(CCCNC(c3ccc(CO)cn3)=O)CC)=O)CCC(CC1=O)C2(C)C c1(C(=O)OCC)ncccc1NC(=O)NCc1ccc(SC2CCOCC2)o1 C(=O)(C(CNC(=O)C(C)C(C)(C)C)CC(C)C)NC(CCC)C(=O)NC C(c1ccccn1)=CC(=O)NC1(C)CC(NC(=O)Cc2cc[nH]n2)C1 C=C(F)C1(CC(=O)NC2CC(C(=O)NCC(=O)NOC)C2(C)C)CCC1 c1(C(N2CCC(C(N(C)Cc3cn(CC)nc3)=O)(CF)C2)=O)cccc(F)c1C O=C(CCCn1cccc1)NCC(C1CCCC1)NC(=O)CN1CCCCC1 C1(NC(NC(C(F)F)F)=NCCN2CCCCCC2)C2CC3CC(C2)CC1C3 c1(C(=O)NC2(CC(N)=O)CCN(C(CCCOC)=O)C2)cn2c(n1)CCCC2C O=C(C#CC1CCCCO1)NCC1CCN1C(=O)COc1ccc2c(c1)OCO2 N1(C(CC)=O)CC(O)CC1C(=O)NC1(C)CC(OCc2ccccc2)C1 C1(C(=O)NCC2=CCCN(C(c3ccoc3)=O)C2)CCc2nccn2C1 C(=O)(C#CC1CCC1)N(C(C(C1CC=CCC1)NC(=O)OC(C)(C)C)=O)CC c1(C(=O)NCCCCN(C(C=CCC)=O)C)ccnn1CC=CC N1(C(CC2C(C)=NNC2=O)=O)CCC(NC(=O)COC(C)C)C12CCC2 C1(CC=C)(NC(C2CC2C2CC2)=O)CCN(C(c2cc(OC)ncn2)=O)CC1 N1(C(C(=O)NCc2cn(C(C)C3CC3)nc2C)=O)Cc2ccc(C#N)cc2C1 Cc1cc(Br)ccc1C(N1CCCC(N(C)C(c2cn(C)cn2)=O)C1)=O C1(NC(CC=CCC)=O)CS(=O)(=O)C2CN(C(=O)C#CC3CC(F)(F)C3)CC12 c1(C(=O)NC(CC)CN(C(=O)CC2C=CCC2)C)cnc(S)nc1 C(CCC(=O)NCC1CCC1C(=O)NOCc1cccnc1)=CC(C)C c1(C(N2CCCC(CC=C)(NC(c3cc[nH]c3)=O)C2)=O)ccc2cccnc2c1 Cc1cccc2nc(CN=c3[nH]c(N4CCN(C5(C)CC5)CC4)nc(=N)[nH]3)cn12 CCC(CC)(CCNC(C1CC1c1ccn(C)c1)=O)NC(=O)Cc1ccc(O)cn1 C1(CNC(CCCCCC)=O)CC2(CCC2)CN1C(=O)C(CC)N1CCCC1=O c1(C(=O)NCC2N(C(C=C(C)C(F)F)=O)CC2)cc2n(c1)CCSC2 c1(C(=O)NCCCC(C)(C)NC(C(C)OC)=O)cn(C)c(=O)c(C)n1 Cc1ccc(SS(=O)(=O)CC(=O)NC(C)CNC(C2OCCO2)=O)cc1 c1(CNC(C(C)N(C(=O)CC2CCCO2)CC)=O)csc(C)c1 c1(C(=O)NC2CCN(C(CCN(CCCCC)C)=O)C2)n[nH]c2c1CC(C)CC2 Cc1ccnc2nc(C(N3CCC(C)C(CNC(c4cn(C)cn4)=O)C3)=O)nn12 CC(C)(C)CC(O)C(=O)NC12CC1CN(C(c1occ3c1CCCC3)=O)C2 N1(C(C(CC=C)C)=O)CCC(COC)(NC(=O)CC2CN(C(C)=O)C2)CC1 N1(C(C=CCCC)=O)CC(CNC(=O)C(C)Cc2ccco2)(COC)C1 CC(=O)CCCC(=O)N1CCCC(NC(c2ccc(Cl)nc2N)=O)C1 C1(NC(C2CC(SC)C2)=O)CCSC12CN(c1nc(C(C)(C)C)ccc1C#N)C2 c1(C(=O)NCC(=C)CCNC(=O)CC2CN(C)C2)c[nH]c2ccc(Cl)cc2c1=O c1(C(C(F)F)NC(CCC2C(C)(C)NC2)=O)ccccc1F N1(C(C2CC(NC(C(C3CCCCC3)C)=O)C2)=O)CCCC(C)C1CO CCCC(C(=O)N1CCCC1CNC(C1OCCCO1)=O)S(N)(=O)=O N1(C(CSC)=O)CC(NC(=O)C(C)Cc2c(C)n[nH]c2C)C(S(C)(=O)=O)C1 C1(CNC(C=CC=CC)=O)CC(C)N(C(c2nnn(-c3cccc(Cl)c3)c2C)=O)C1 C1(NC(c2c(CC)nco2)=O)CC2CCC1C(NC(=O)CCOC)C2 C(=O)(C1=CCCC1C)NCC(=CC(=O)NC(C=C)COC)C C1(C(=O)NCC2CCC(C(F)F)O2)C=CCN1c1nnco1 Fc1ccsc1C(C1CCC1)NC1CC2CC2C1 Cc1ccc(CC(=O)NCC(O)CCNC(c2ccc3c(c2)CC3)=O)c(F)c1F C(CN=C1NCC2CN(C)CC12)Sc1ccc(OC)cc1OC CC1(C)CN(C(=O)Cc2cnccn2)CC1CNC(C1CCC(=O)N1)=O c1(C(=O)NC2C(CC)CN(C(=O)C3=C(Cl)CCCC3)C2)coc2c1C(=O)CCC2 c1(C(=O)NCC2CN(C(C(N3CCC(C)CC3)=O)=O)CC2C)n[nH]c2c1COC2 Cc1cc(C)n(CN(C)C)n1.c12cc(cs1)C(=O)NC2.C1(NC=O)CC1CC1CC1 CC1OCCOC1C(=O)N(CCCC)CCOCCO.C1(F)(C(=O)N)CC=CC1 N1(C(c2cc(CNC(C(C)(CO)OC)=O)no2)=O)CC2(CCCO2)C1 C#CCCCC(=O)N(CCCOCCN(C)C(c1ccc(N(C)C)nc1)=O)C C1(CNC(C2OCCN(C)C2=O)=O)CC12CCN(C(c1csc(CO)n1)=O)CC2 O=C(C#CC1CCCOC1)NCC1CN(C(=O)Cc2ccc(O)nc2)CCO1 Cc1ccccc1C(C)(C)C(=O)NCCCCC(C)NC(=O)C(C)(O)C1CCC1 C12(CNC(CCOCCOCC)=O)CCC1CN(C(C1(O)CCSCC1)=O)C2 C1(C)(CNC(C2(C)CCC2)=O)CCN(C(C2CCC3C2C3(F)F)=O)CC1 c1(OC)ccc(C(=O)NCCN(C(=O)C(N2CCOC2=O)C)CC(C)O)s1 Cc1cccc(N)c1C(=O)N(C)CC1CCCCN1C(C1CCS(=O)(=O)C1)=O CC1(COC(c2cnc(-c3ccsc3)s2)=O)CCCCC1 C12(C(N3CC(CNC(C)=O)C(O)C3)=O)CC1COC2(C)C.c12ccncc1N2 N1(C(C2(CC)CN(C(=O)CC3(C)CCOC3)C2)=O)CCOC(C)(C)C1C Cc1cc(C(=O)NCC(C2CCCC2)NC(c2ncccc2F)=O)c(Cl)cc1F C1(CNC(CC(CC)C)=O)CN(C(C2CCCN2C)=O)CCC1(C)C C1(C(N(CCCN(C)C(c2sccc2Br)=O)C)=O)C(C)(C)C1(F)F c1(C(C(=O)NCCCCN(C(C(CN(C)C)(C)C)=O)C)(F)F)cc(Cl)ccc1Cl c1(C(N2CCC(C(C)NC(C(C)NC(=O)OC)=O)CC2)=O)cn2c(n1)SCC2 C1(C(=O)NC(C2(C(=O)NC3CC34CCCC4)CC2)C)CCCCCN1C Cc1nn(C)c(NC(=O)C(O)CC(C)C)c1Cl.n12cc(cn1)C(=O)N1CC2C1 Cc1ccc(SC(C)C(=O)N2CCCC2)c(NC(=O)CCC(C)C)c1 c1(C(=O)NCC2CCC(NC(C(C)NC(C)=O)=O)C2)ccc2scnc2c1 c1(C(=O)NCC2N(C(c3c(C)n[nH]c3)=O)CC2)cc(Cl)ccc1N C1(NC(C2CSC2)C)CCN(c2cccc(Br)c2)CC1 c1(N2CCCC(OCC=C)C2)nc2c(c(=NCc3nc(O)n[nH]3)[nH]1)COC2 N1(C(C(CC=C)(F)F)=O)CCC(C(N2CCCOCC2)=O)CC1(C)C c1(C(=O)NCCC(C(=O)Nc2c(CC)ncnc2)OC)cccc(CO)c1C N1(C(c2cccc(C)c2)=O)CC(C(N2CC(OC(F)F)C2)=O)CC(C)C1 c1(CCC)ccc(SCCCC(=O)NCCN(CC(=O)NCSC)C)cc1 C1(NC(c2cccc(C)c2)=O)C2CCC(C2)C1C(=O)Nc1ncccc1Br Cc1ccc2c(CN=C(NCCN(C(C)C)C(C)C)NCC3CC3(C)C)c[nH]c2c1 C1(C)(C(=O)NCCCN(C(c2cc(CCOC)on2)=O)CC)CCCNS1(=O)=O N1(C(C=Cc2n(C)ncc2)=O)CC2CCN(C(=O)C(O)P(C)(C)=O)CC12 N1(C(c2cc(F)ccc2C(F)(F)F)=O)CC2CN(S(=O)(=O)CCBr)CC2C1 N1(C(C2C(OC)(OC)CC2)=O)CC2(C(N3CC(C(C)OC)C3)=O)CCC1CC2 c1(C(=O)NC(C)CCCNC(=O)Cc2cccc(O)c2)ncnc2c1OCCO2 C1(CCC)CCCC1C(=O)NCC1CC(NC(=O)COc2cn[nH]c2)C1 c1(N(C)C)ccc(Br)cc1C(N1CC2C(C(N3CC4(CCC4)C3)=O)C2C1)=O C1(CNC(C2CCCC(C)CC2)=O)C2CCCC1N(C(=O)Cc1ccoc1)C2 C#CC1N(C(=O)NCC2CCCN(c3ccc(CC)cc3)C2)CC1(C)C C1(CN(C)C)CN(C(c2cccc(C(=O)NC3CCCC(N)C3)c2)=O)CC12CC2 c1(C(=O)OC)ccc(OC)c(C(=O)Nc2ncn(C(C)C)n2)c1 C1(OC)CN(C(C)=O)CC1n1cccn1.C12CCN(CC1)CC(=O)N2 c1(CC(=O)NC2COCCC2NC(C2(n3cnnn3)CC2)=O)ccc(Cl)cc1F N1(C(CCC(C)(C)F)=O)CC2CCCC2(CNC(c2nc(O)nc(O)c2F)=O)C1 c1(CC(N2CCC(N(C(C3C(CC)C3)=O)C)CC2)=O)cnc(Cl)cc1C C(c1cc(Br)ccc1F)=CC(=O)NCc1nc(C(C)(C)C)[nH]n1 C1(C)(CNC(C=C(CCC)C)=O)CC(F)(F)CN1C(=O)C(C(C)C)NC=O C1(F)(C(N2CC(NC(C3CC(C#N)C3)=O)C2)=O)CCN(Cc2ccc(F)cc2)C1 c1(CC)nc(C)oc1C(=O)NC1CCOCC1C(=O)NCCC1(C)CC1 N1(C(c2c(OC)ccs2)=O)Cc2ccccc2CC1CNC(C1CC(OC)C1)=O c1(C(=O)NCC(CCNC(c2c(CC)non2)=O)O)cc([N+](=O)[O-])cc(C)c1Cl c1(OC)cccc(C)c1C(N1CCCC(F)(CNC(=O)OC(C)(C)C)C1)=O Cc1snnc1C(=O)NCC(C)C(=O)NCC(O)CF C1(C(=O)O)CC(C)(C)CCN1C(=O)CC1CC(C)(C)CN1S(CCCC)(=O)=O C1(NC(C=CCCC=C(C)C)=O)C2CC3C1C3C2C(N1CCC(CO)C(O)C1)=O C(C(C)(O)C(=O)N1CC=CC(NC(=O)CS(=O)(=O)Cc2cccs2)C1)OC CC(CC(=O)NCC1(O)CC(C(=O)NCCCCCN(C)C)C1)C(F)(F)F N1(C(C(C(C)C)SCC)=O)CCN(C(C2(C)CC2)=O)CC12CC2 N1(C(CCCC2(C)N=N2)=O)CCOCC(NC(C2(CO)CCOCC2)=O)C1 C1(NC(C2C(=C)CC2)=O)CCCCC12CCN(C(c1cnc(C(C)=O)s1)=O)C2 C#CCC(CC(F)F)C(=O)NC(C(N1CC(F)CC1C)=O)C1CC1 c1(N2C(C)(C)C(CNC(C3CC34CC4)=O)CC2)nc(Cl)nc2[nH]cnc12 c1(C(C(=O)NCC(C)NC(=O)CCn2cc(Cl)cn2)O)cc(F)c(F)cc1F Cc1c(C(=O)N(C)CC2(NC(C3COC4(CCC4)C3)=O)CC2)cccc1F C1(C(=O)NCCC(C)N(C(=O)C=CC(N)=O)C)Cc2nccnc2C1 CS(=O)c1cccc(C(=O)NC2C=CC(CNC(c3cc(O)ncc3Br)=O)C2)c1 c1(OC)c(F)cc(C(N2CC3C(NC(=O)C(C(=O)OC)OC)C3C2)=O)cc1Cl c1(C(=O)NCC2CCN(C(c3ccc(COC)s3)=O)C2)n[nH]c2nccc(Cl)c12 c1(C(=O)NCC2N(C(c3n(CC)nnc3)=O)CCCC2)cccc2ncccc12 N1(C(c2cccc(N)n2)=O)CC(C2CCCN(C(C3CCC4(CCC4)C3)=O)C2)C1 C(=O)(C(C)C(O)C(C)C)NCCCCC(C)(C)NC(c1oc(C)c(CO)c1)=O c1(C(=O)NC(CCOC)CNC(=O)COCC(F)F)cccc2c(C)ccnc12 C(=O)(CC(C)(C)C(F)(F)F)N1C(C)C(NC(=O)CCC2NC(=O)NC2=O)CC1 CCS(=O)(=O)c1ccccc1C(=O)NCC1CN(C(C2CCC(C(N)=O)O2)=O)C1 C1(C(N(CCNC(c2c(OC)cco2)=O)C2CC2)=O)CC(C)(C)CCO1 CC#CCCCC(=O)N1CCC(C(C)(C)C(=O)NCC(CC)C(C)(F)F)C1 N1(C(C2CCN(C(C3CC(=O)N(CCN(C)C)C3)=O)C2)=O)CCOCC1C1CC1 c1(C(=O)NC2C=CCC(NC(c3ccc(OCC)nc3)=O)C2)ccc(C)c(OC)c1 CCCC(C(=O)NC(c1cnn(C)c1)C(N1CCCC(O)C1)=O)OCC c1(CC)nc(C(=O)NC2CC2CNC(=O)C=CC2CCCCC2)c(C)o1 N1(C(C2C(C)CC=CC2)=O)CCC(C2CN(C(C3CC4(CCC4)CO3)=O)C2)CC1 c1(C(=O)NCC2CN(C(C(CC)C#N)=O)C(C)(C)C2)ccc2ccc(C)cc2n1 C1(NC(c2ccc(CSC)cc2)=O)CN(C(=O)C=C(C)C)CC1CC(C)(C)C c1(NC(C)=O)cccc(CC(=O)NCCCC(C)NC(=O)C(O)C(C)C)c1 C(=O)(C1COc2cc(C)c(C)cc21)NC1(NC(C(CCOC)OC)=O)CC1 c1(NC(N2CCC23CCOC3)=O)cc(O)c2ccccc2n1 C(=O)(CS(=O)(=O)Cc1cccs1)NC(CCNC(c1c(CC)cncc1)=O)C c1(C(=O)NCC2C3CN(C(c4c(CC)[nH]nc4Cl)=O)CC32)c[nH]nc1S(N)(=O)=O c1(C(c2ccccc2)NC2(C(C)(C)C)CCOC2)cc(S(N)(=O)=O)ccc1O c1(C(C(=O)O)C(C)C)ccc(F)cc1C.c1(C(=O)OCC)nnc(C(=O)OCC)s1 C12(C(=O)NC3CCCN(C(C4CCCO4)=O)C3)CCC(C1)C(=O)NC2 O=C(C1=NOC2(CCCN(S(=O)(=O)C3C4CCCC4C3)C2)C1)Nc1ccccc1 Cc1ccc(F)cc1-n1nc(CC(C)C)nc1C1CC12CCC2 CCN=C(NCC1CCC1)NCC1CC=CCO1 Cn1cncc1CNC(=O)CC1CCN(C(C2CC2(C)C)=O)C1 CC1CCCCC1(CNC(c1nc(C(C)(F)F)cs1)=O)NC(c1nonc1N)=O C(=O)(C1=C(C)OCCS1(=O)=O)NC1CCC(CCNC(c2cc(OC)no2)=O)C1 C(=O)(C(C)(C)C(=O)NCC1(F)CCN(C2CCNC2=O)CC1)OCC C1(CC(=O)NCCCCCNC(=O)COC2CC(F)(F)C2)CC2(CC2)CO1 C(=O)(C1=CC2(CCOC2)C1)N(C(CC(=O)N(C(C)C(=O)N(C)C)C)(C)C)C Cn1cc(S(C)(=N)=O)c(NC(N2CC3OCCC2C3)=O)n1 N(C1CCOc2c(F)cccc21)c1ncnc(NC2CCC(OC)CC2)c1C c1(OC)ccc(C(N2CCC(NC(c3cc(SC)cc(F)c3)=O)C2)=O)c(F)c1F CC(CC(=O)NC1CN(C(c2occ3c2CCC3)=O)CCC1F)CC(F)(F)F C(=O)(CC(C)(C)CC(=O)N1CCCC2(NC(=O)Cc3nonc3C)CC2C1)OC c1(C(N2C(C)(C)C(C(=O)NCC(O)CO)CC2)=O)cnn2ccccc12 Cc1cccnc1C(=O)NCC1CN(C(C2CCC(NC(=O)N(C)C)CC2)=O)C1 C1(CCC(=O)NCCN2CCCC(OC)C2)CCCN(C(=O)CCC2CCC2)C1 N1(C(c2c(C)noc2C)=O)CC(NC(=O)C(C)(C)c2cscc2Cl)CC(O)C1 Cc1ccc(C(=O)NC2(CO)CCN(C(C3(C)CCOC3)=O)C2)cc1C#N N1(C(C(C(C)C)=O)=O)CCC(C)(C(=O)NC2CCC(F)(F)CC2)CC1 C1(NC(CNC(=O)NC)=O)(CO)CCN(C(=O)Cc2cc(Cl)ccc2OC)CC1 C(CC(N)=O)(C(=O)Nc1ccc(C)c(C(N)=O)c1)NC(C1CC(CC)(CC)C1)=O N1(C(C(C)=C(C)C)=O)CC2(C1)CN(C(c1cc3c(cc1Cl)NCC3)=O)CCO2 Cc1ccccc1C(C)NC(=O)C(F)CCCn1cc(COC(=N)O)nn1 N1(C(c2c(C)coc2C(C)C)=O)C2CCC1CN(C(C1(C)CC1)=O)C2 CC1CN(C(C23CC(C2)C3)=O)CC2(CCN(C(c3occ4c3CCCC4)=O)C2)O1 Cc1nnc2n1CC(NC(=O)NCC1COCCOC1)CC2 C12(NC(CSc3ccc(C)cc3)=O)CCC(C1)N(C(c1ncc(F)cc1N)=O)C2 C1(NC(=O)NC(CCCC=C)C2CC2)CCC2(CCN(C(=O)OC(C)(C)C)C2)C1 N1(C(C(c2ccccc2)C)=O)CCC2CN(C(c3cnn4c3CCCN4)=O)CC12 c1(C(N(C)C)=O)cccc(CN2CCN(C(C3(S(N)(=O)=O)CC3)=O)CC2)c1 C(=O)(C1CCCc2scnc21)NCCC(CCNC(c1c(CC)con1)=O)C C1(CCC)CN(C(=O)CN(C)C(=O)OCC)CC1NC(c1cccc(Cl)c1)=O Cc1c(C(N2CC(C)(CNC(c3ccc(Cl)c(Br)c3)=O)C2)=O)cccc1O C1(NC(=O)CNC(=O)NC2CC2)CCSC12CN(C(=O)CC=C(Cl)Cl)C2 C1(C(=O)O)CC2(CNC(=O)CNc3ccccn3)CC1C2 c1(N(CCCCNC(CNC(CC)=O)=O)C)ccc(S(C)(=O)=O)cc1 C1(CC)CC(C(=O)NC2CC2O)CCN1C(c1ccsc1C#N)=O C1(C(SC)=O)CCCN(C(c2ncccc2Br)C(=O)NC)C1 C1(C(N2CC(C(C(=O)OC)O)C2)=O)CN(C(c2ccnc(C)c2N)=O)CCN1C Cc1nc[nH]c1CC(O)C(=O)N(CCNC(=O)C(O)CN1CCCC1)CC1CC1 C1(NC(C(CC)OC)=O)CCN(C)C12CCCN(C(C1(CC)COC1)=O)C2 CC1(C)CN(N2CCN(S(=O)(=O)Nc3cccnc3)C2)CC1CCO N1(C(CCSCCC)=O)CC(NC(c2ncsc2Br)=O)C(C2CC2)C1 C1(C(N(CCCCO)CCCC)=O)CSCN1C(=O)C(C)n1ccnn1 C(=O)(C(C)(CC)C(N)=O)N1C(C)(COC)CC(NC(=O)C(=O)N(C)C)C1 c1(CC)nc2ccccn2c1CS(=O)Cc1nc(CC(F)(F)F)nn1C C(c1ccc(F)c(C)c1)=CC(=O)NC1CC(C)(NC(C(CC)N2CCCC2=O)=O)C1 c1(NC(C2(SC)CN(C(c3sc(O)nc3C)=O)C2)=O)ccc2ccncc2c1 C12(CNC(C3C(NC(C4C(C)(C)CO4)=O)CC3)=O)CCCN(CC1)C2 Cc1c(C(N2CC(N(C(=O)CC3CC3)C)C(F)C2)=O)nnn1CC1CCCC1 c1(C(N(CC(CC)NC(=O)C(C(C)C)N(C)C)C)=O)c[nH]nc1S(N)(=O)=O c1(C(=O)NCCN(C(=O)C(O)c2ccco2)C)csc2cncn12 CC1(C(N2CC3CC3(CNC(=O)COC3CC=CC3)C2)=O)CCC(=O)N1 c1(SC)ncc(C(=O)NC(C)CN(C(=O)CCSc2nncn2C)C)s1 C12(C(=O)NCC3CN(C(C4C(C)CC4)=O)C(C)(C)C3)CC3CC1C2C3(F)F C1(CC=C)(NC(c2n[nH]cc2F)=O)CCN(C(c2cc(N(C)C)ccn2)=O)C1 C(=O)(C(CC1CC1)N(C(=O)CCc1ccccc1)C1CC1)N(C)CCN(C)C1CC1 CON(CC1CCCCC1)C(=O)C(F)=CC1=CCCCC1 N1(C(C2(C3CC3)CCCO2)=O)CC2CC(C(=O)NCCC#CCO)(C2)C1 c1(C(=O)NC(CC)CNC(=O)C(O)C2CC2)c(C)noc1C(F)(F)F C1(C(=O)NC2CCC(C(N(CCCC)C(C)C)=O)CC2)CCC2CCCCN12 C1(OC)CCC2(C(N3CSCC3C(=O)NCCC(C(C)C)OC)=O)CC12 C(=O)(C#CC1CCOC1)NC1C(NC(c2cc(C)c(C)s2)=O)CCOC1 c1(C(=O)O)cc(CN2CCC(F)(C(=O)Nc3c(Br)ccnc3Br)C2)ccc1O C1(NC(C2C(C)CC(=O)N2)=O)CN(C(C2CC(=O)CO2)=O)CC2(CC2)C1 c1(N2CC(CCC)C(CC(N)=O)C2)nc(=NCCC(N)CC)[nH]c2c1COC2 C1(C(N(CC(Cc2ccccc2)NC(COCC)=O)CC)=O)CC(=O)N(C2CC2)C1 N1(C(=O)COC2CN(C(C3CCCCO3)=O)C2)CCc2cccnc2C1 c1(CC(=O)NC2(CF)CCN(C(c3c(CC)ocn3)=O)C2)cc(Cl)cc(Cl)c1 N1(C(CCSC)=O)CC(NC(=O)CCc2cncn2C)C(C2CC2)C1 S(=O)(=O)(c1ccc(F)cc1)CC(=O)NCCC(N1C(c2scc(C)n2)CCC1)=O C1(CC(=O)N(C)CCNC(=O)C2=CCCS2)CC(O)C12CCC2 c1(CSC)n[nH]c(CCNC(=O)CC)n1.C(=O)(C(C)C1CCCO1)N C1(CNC(C2(OC)CCSC2)=O)CN(C(C2CN(C3CCC3)C2)=O)CC1(C)C Cn1nc(C(=O)N(C2(c3ccccc3F)CC(N)C2)C(C)(C)C)nc1Br c1(COCC)nc(C)cc(=NC2CC3CN(C(c4csnn4)=O)CC23)[nH]1 C1(NC(C2(COC)CCC2)=O)CCC(C)N(C(=O)C2=COCCO2)C1 n1(CCC)cc(C(=O)NCCCC(C)NC(=O)CC(=O)Nc2nccs2)c(C)n1 C(=O)(C1CCc2snnc21)N1C(CNC(C2(C(=O)NC)CC2)=O)CC(O)C1 N1(C(C2C(C)=CCC=C2)=O)CCc2cccc(C(=O)NC(C)(C)CO)c2C1 C(CCCCCNC(C1C2CCC1(c1ccco1)C2)=O)NC(c1cocn1)=O C(C(N=[N+]=[N-])C(=O)N1CCC(CC(=O)NC(C)C(C)C(C)C)CC1)OCC CC1(NC(=O)C(O)C2CCC2)CCC(NC(c2cccc(CF)c2)=O)CC1 C(c1cnc(C)nc1O)=CC(=O)NCCNC(c1ccc(C(CC)(C)C)cc1)=O C1(C(N2CC(O)(CC=C)C2)=O)CC(F)CCN1C(=O)C(C1(O)CCCC1)F C1(NC(CNC(CC)=O)=O)CCCN(C(c2ccc(-c3ccccc3)s2)=O)CC1 N1(C(C(CC2CCC2)NC(c2cc(CO)[nH]n2)=O)=O)CCN(C2CCCC2)CC1 C1(NC(C2C(CNC(C(C)C3CCC3)=O)C2)=O)CCCC1(F)F c1(NCCCN(CCC)C)ncc(S(=O)(=O)NC2CCN(CC)C2)cc1Cl N1(C(c2cc(CC)no2)=O)CCOC(CCCNC(=O)C(C)NC(=O)NC)C1 c1(C(=O)NCC2(NC(c3ccc(Br)s3)=O)CCC2)ccc(OC(F)F)cc1 N1(C(CCCC)=O)CC(C)N(C(=O)C=Cc2ccc(C)s2)CC1C C(=O)(C(C(C)(C)C)C1CCC1)NC(CNC(c1cc(C)on1)=O)(C)C c1(C(C)NC(=O)CCNc2cccc(Cl)c2)nnc(-c2cccs2)n1C1CC1 c1(C(=O)NC(CC)(CNC(C2CC3CCC3C2)=O)CC)n[nH]c2c1COC2 CC(C)(C)CCCCC(=O)N1CC(=O)NCC1C(N1CC(CCO)C1)=O c1(NC(=O)CCC2CCC2)cn(-c2ccccc2)nn1.C1(N2CC2=O)CCOC1 Cc1cccn2ncc(CNC(c3cc4ccsc4cn3)=O)c12 CC1(NC(C23CSCC2C3)=O)CCN(C(c2cc(Cl)c[nH]2)=O)C1 c1(C(=O)NCC(C)CN(C)C(c2cc(=O)cc[nH]2)=O)ccc(-n2cnnn2)cn1 N1(C(C(C)=C(CC)C)=O)CC2(CNC(C3CC3(C)COC)=O)CC1CO2 Cc1cc(F)c(CC(N2CCC(C(C)(C)NC(C3CCCC3)=O)CC2)=O)cc1F c1(NC(CNC(Cc2cc(CC)no2)=O)CO)cc(N(C)C)nc(Cl)n1 c1(C(=O)NCC2C(NC(C)=O)CC2)cnc(Cl)c(F)c1N N1(C(C(C)OCCC#C)=O)CCC2CN(C(C3CC(n4ccnn4)C3)=O)CC12 C1(N)CCCCC1n1cc(CCC2CC2)nn1.N1(C(C(C)C2CCC2)=O)CCOCC1 C1(C(=O)NCC(C)(C(=O)NC(C)CCSC)OC)Cc2nccn2C1 CC1CC(c2ccoc2)CN1C(=O)C(O)c1cnc[nH]1 Cc1csc(C(=O)N(C(C)CN(C)C(c2cnn(-c3ccccc3)n2)=O)C)c1C CCCCC(O)C(C)C(=O)N1CCN(C(=O)C(COCC)N=[N+]=[N-])CC1CO C1(CC)CN(C(=O)C(O)C(C)C)CCN1C(=O)CCCN(C)C(C)=O c1(OCCC(C)C)cccc(C)c1.C(C)(C(=O)NCC1CC1CNC(=O)C)OC CC1=NNC(=O)C1CC(=O)N(C)CC1CCCN1C(=O)C(c1cnn(C)c1)C c1(C(C)C)nc(N2CC(C(C)NC(=O)Cn3nnnc3C3CC3)C2)cc(Cl)n1 C(=O)(C(C)(C)CNC(=O)C(C1CCN(C(c2c[nH][nH]c2=N)=O)C1)C)NC c1(C(N2CCCN(C(c3ccc(CC)[nH]3)=O)CC2)=O)sc2nnc(S)n2c1C C(=O)(C1CSc2ccccc21)NC1CC(CNC(C(=Cc2cccs2)C)=O)C1 C1(CC(N2CCC(NC(c3cc(C)ns3)=O)C23CC3)=O)CCC2(CCC2)CO1 C12(CCNC(=O)C(C3CCCCC3)O)CCC(CC1)N(C(=O)CN1CCCC1)C2 c1(C(=O)NCC2OCCCN(C(C3C(C#N)C3)=O)C2)cccc2ccoc12 C1(C(N2CC(O)(CNC(c3c(C)sc(Cl)n3)=O)C2)=O)OCC2CCCC12 C1(C(N2C(CNC(C(CCCOC)C)=O)CCCCC2)=O)CN=C2N=CNN2C1 C(=O)(C(CC1CCCC1)NC(C1CC1OC)=O)NC1(C(=O)NCC#C)CC1 C(c1nccs1)=CC(=O)NCC(C1CCOC1)NC(c1cc(C(F)F)on1)=O C1(CNC(Cc2cc(C)sc2)=O)(CNC(=O)CCC(C)(C)C)CC2CCCC2C1 C(CC(CNC(=O)C(O)c1cnc[nH]1)NC(c1csc(C(F)(F)F)n1)=O)OC CCCCCCCCCCC(=O)N1CCCC(N(C(=O)CCCC2CC2)CC)C1 c1(C(=O)NCC2(O)CCN(C(c3cncc(O)c3)=O)C2)cc2c(Cl)cccc2[nH]1 C1(O)(CN(C(C(CC)OC)=O)CC)CCN(C(c2ccnnc2C)=O)C1 N1(C(c2ccc(C)cn2)=O)CCC(C)C(NC(=O)CC(C)(C)O)C1 C#CC1(O)CCCN(C(c2cccc(CNC(C3CCSC3)=O)n2)=O)C1 C#CC1CCCN1C(=O)C(C)N(C(=O)CCC(=O)C1CC1)C Cc1nc2ccncc2c(=O)n1CC(=O)NCC12CCC(CC1)N2C(=O)CC#N c1(N(C)CCNC2CCCO2)cc(N2CCC(C3OCCO3)C2)nc(C(F)(F)F)n1 C1(CC(=O)NCCOC(C)=O)CCCCC1NC(=O)Cc1ccc(C)s1 c1(C(N(C(CN(C(Cc2nc(C)sc2C)=O)C)C)C)=O)cc2nc(Cl)ccc2s1 N1(C(CCCC)=O)CC(NC(c2cc(F)ccc2Br)=O)C(C2CC2)C1 C1(C(N2CCC(OC)(CNC(C3CNC(=O)C3)=O)C2)=O)CC2CCC(C1)C2 C(c1c(C)coc1C)=CC(=O)NCC(CCOC)NC(=O)CC1(C)CCCCC1 C1(C(=O)NCCOCCN(C(C(=O)NC)=O)C)CN(C(=O)C2CC2)CC1(C)CC CCCCC(C(=O)NCCC1CN(C(C2(Br)CC2(F)F)=O)C1)N(C)C Cc1cnc(F)cc1C(=O)NC1CC(C)N(C(C2CCN(CC(F)F)CC2)=O)C1 c1(OC)cc(C(=O)NCC2CCCCC2NC(=O)Cc2ccno2)c(F)cn1 c1(OC)ccc(NC(=O)C(=O)NC(c2cnsc2)C)c(C#N)c1 N1(C(C2C(CC)CCO2)=O)CC(C(=O)NCCCS(N)(=O)=O)C(F)C1 C12(C(N(CC(C)NC(=O)Cc3ccccn3)C)=O)CCC(C1)C2(C)C c1(CC)nncn1NC(=O)C(CCC(C)C)NC(c1cc(C#N)oc1C)=O C(=O)(CCCC(=O)NCC1C2CN(C(C3COCCO3)=O)CC12)NC(C)C CC1=C(C)CC(C)(C(=O)NCC(C2CCCC2)NC(C2(Cl)CC2(F)F)=O)CC1 CC(C(=O)NCC(C1CC1)N(C)C(c1cnnc(O)c1)=O)C(F)F N1(C(CC(=O)NCC#C)=O)CCC(C(=O)NCCC23CCCN2CCC3)=C(F)C1 Cc1nn(C)cc1CNC(=O)CC1CCCN1C(c1cc(F)c[nH]1)=O C(CC[Si](C)(C)C)NC(N1CCC(CCC(=O)OCC)C1)=O C1(COC)(NC(=O)C(C)C(F)F)CCN(C(c2cc(C)cc(C(F)F)n2)=O)CC1 CC(C)(C)C(CNC(C1(C)CC1C(F)(F)F)=O)NC(c1c[nH]cc1Br)=O C1(C(=O)NCC=CCSCCO)(OCCOCCOC)CC1 C(CC(O)C(F)(F)F)CCONC(CCN(C(C(n1ccc(C)n1)C)=O)CCO)=O CC1CN(CC(C2CCCCC2)=O)CCC1CS(N)(=O)=O N1(C(Cc2c(C)nc[nH]2)=O)CC(C)CCC1CNC(=O)CC1(C#N)CCCCC1 C1(COCC)CCN(C(=O)CCCNC(C2COCCN2C2CCCC2)=O)CC1 c1(C(CCO)NC(C(C)(C2CCC2)NC(=O)Cn2ccnc2)=O)cccc(O)c1 N1(CC(=O)N(CC(C)NC(=O)CC2CC(F)C2)C)CC(=O)NC1=O N1(C(C2(CC(N(C)C(c3cnc(O)o3)=O)C3CC3)CC2)=O)CCN(C2CCC2)CC1 C12(C(N(CC(COC)O)C)=O)CC(CN(C(=O)CCS(N)(=O)=O)C1)C2 c1(CC(=O)NC2CCC(NC(C=CC(=O)OCC)=O)C2)ccc(OC)c(F)c1 c1(C(N2CCCC(C(C)NC(=O)C3=CCSC3)C2)=O)c(F)cc(F)cc1F c1(C(C(=O)NCC)N(C2CCN(CC3CCCCC3)C2)C)cc(C)c(Br)c(Cl)n1 N1(C(C(C=CC)O)=O)CC2(C1)CN(C(c1cn(C)cc(F)c1=O)=O)CC2CO c1(C(C)(C)OCCCC=C)ccccc1S(=O)(=O)N(C)C C1(CNC(C(COC)C)=O)CCCCN(C(=O)C(C)N(C)C)C1 N1(C(C(C)NC=O)=O)CC(NC(=O)C=Cc2cccs2)CC12CCCCC2 C(=O)(C1CCc2nnc(C)n21)C1(C2N(Cc3c(C)cc(O)cc3)CCC2)CC1 Cc1cc(C)c(C(N2CCCC(N(C(=O)Cn3cccn3)C)CC2)=O)c(S)n1 C1(C(N2C(CN(C(C3CCCN3C)=O)CC)CCC2)=O)CCN(C)C(=O)C1 Cc1ccc(C(N2CC3C(CNC(=O)CCCCC(N)=O)C3C2)=O)c(O)c1C Cc1cn2c(CC(=O)NC3CC(NC(c4ccc(F)c(F)c4F)=O)C3)csc2n1 CN(C)S(=O)(=O)N(C)CC(=O)NCC1CCN(C(=O)CN2CC=CC2)C1(C)C c1(CN)cccc(NC(C2(F)CCN(NCC(F)(F)F)C2)=O)c1 c12cccc(c1OC)OC2.C1(C(=O)NCCCOC)C2CN(S(C)(=O)=O)CC12 c1(CC(=O)NC2C(OC(C)(C)C)COCC2)nc2cc(Cl)ccc2s1 Cc1cc(C#N)cnc1NC1CCCN(C(C2(F)CCCOC2)=O)C1 c1(C(=O)NC2CCCN(C(c3cc(C(F)(F)F)no3)=O)C2)cc2c(s1)CCC2 c1(NC(CC2N(C(C(C)Cn3cccn3)=O)CCC2)=O)cnnc(Br)c1 c1(C(=O)NCC#CCNC(C(N2C(CC)CCC2)=O)=O)cccc(C(C)(F)F)n1 c1(C(=O)NC(C(C)C)CNC(c2cn(C)ccc2=O)=O)cc(N)c(N)cc1F c1(-c2cn(CC(C(C)C)NC(=O)COc3cccc(Cl)c3)nn2)ccc(F)cc1 C(=O)(C(C#N)C(C)C)NCC(CCCC)NC(=O)C=Cc1cccs1 c1(C(=O)OC)ccc(C=CC(N2CC(C)(NC(=O)C(C3CC3)SC)C2)=O)o1 CC#CCCCC(C)(c1nnnn1C(C)C)NC(C)Cc1ccc(OCC)cc1 c1(C(=O)Nc2c(OC)ccc(O)c2)cc(-c2ccc(F)c(F)c2)cc2c[nH]nc12 C1(n2cc(C)nn2)CC(=O)N(c2cnn(C)c2)C1.C(=O)(C(C)C(C)C)N(C(C)=O)C C1(CNC(c2ccnc(C)n2)=O)CC2(CC2)CN1C(=O)C(C1CCCCC1)F Cc1nn(CCO)cc1C(=O)NC1CC(C)N(C(=O)COc2ccc(F)nc2)C1 N1(C(CCCCOC)=O)CCC2(CC2NC(c2ccncc2F)=O)C1 CN1CCOCC1C(=O)NCCn1cc(C(=O)NCC2CC(F)C2)nn1 c1(C(=O)NC2CCN(C(C3(C)C(C)(C)C3)=O)C2)ccc(-n2cnnn2)cc1Cl C1(=O)C(C)(C)CN1.CCCCCCOCC(N1CC(C(O)C(=O)N(C)C)C1)=O C1(NC(c2cnccc2Cl)=O)CCC12CCN(C(=O)CC1CCCCO1)CC2 C1(CN(C(=O)CN2CCOCC2=O)C)CCCCN1C(c1nccnc1Cl)=O C(C)(C(=O)NC1CCC1C(=O)N(CC(F)F)C)OCC=C c1(C(N2CCC(NC(C3(CO)CCCO3)=O)C(F)C2)=O)cc(Cl)cc(Cl)c1Cl c1(OC)cc(CN2CC(O)CC2C(=O)NCCCc2ccncc2)ccc1Br CC1(CNC(C2CC(F)(F)C2)=O)CCCN1C(c1cn(CC2CCCO2)nn1)=O c1(C(=O)OC)ccc2c(n1)CCCN2C(N1CC2CC2(c2ccccc2)C1)=O CC1(C)CC(C(N2CCC(C(F)(F)F)C2)=O)CN(C(C2OCCC2(C)C)=O)C1 C1(C(=O)NCc2n(C)nnn2)CCCCC1(C)NC(=O)CCc1cccs1 C1(CC(N2CCN(C(CC)=O)CC2)=O)CC(C)(C)CN1C(=O)CN1CCC1C C=C(C)C(C)(C)C(=O)N1CCN(C)C(CNC(=O)C(c2cccc(Cl)c2)SC)C1 N1(C(C2(c3ccccc3F)CC2)=O)CCN(C(C2CC3C=CC2C3)=O)CC12CC2 Cc1[nH]nc(C(=O)NC(C(=O)N(CCCC(C)O)C)C2CCOC2)c1C C=C=CC(C)C(=O)N(CCC(=O)NCCSCC)CC C1(C(=O)OC)CC2CCC(C1)N2C(CC(=O)OC(c1cn[nH]c1)C)=O c1(OC)nccc(CNC(C2CC(NC(C3COC(=O)N3)=O)C(O)C2)=O)n1 c1(CC(C)C)ccc(C(=O)NCC2CC2NC(c2cncc(Br)c2)=O)cc1 c1(OCCC)ccc(C(=O)NC(C)Cn2cc(CCSC)nn2)cc1 C(CCCCCNC(c1ccoc1C(C)C)=O)N(C(c1c(CC)noc1)=O)C C1(NC(c2cc(F)c[nH]2)=O)CCCCC12CCN(C(=O)C1=CCCC1)CC2 c1(NC(CC)CNC(C2CCCC2(C)C)=O)ccc(C#N)cc1[N+](=O)[O-] C(CC(=O)N1CCOCC1C(C)O)(C(F)(F)F)NC(CC1CC(CC)C1)=O C=C(C)CC(C(=O)OC)NC(=O)C(C(C)CC)NC(C1CCOC1C1CC1)=O c1(C(=O)Nc2cccc(Br)c2F)n[nH]c2c1CN(CC)C2.c12n[nH]cc1NC2=O c1(CCC(=O)NC2C(CNC(COC(C)C)=O)C2)cnn(-c2ccccc2)c1 C1(C(=O)NC2CC2)CC2CCC(C1)N2C(c1cnnn1C1CC1)=O c1(C(N2CC(NC(CSC)=O)C(CO)CC2)=O)cc2c(C)n[nH]c2cn1 C1(CC(N2CC(CCNC(C3CCC(C)(C)O3)=O)C2)=O)CCc2sccc2C1=O c1(C(=O)NC(C2CCOC2)C#C)cc(CNC(=O)Cc2ncoc2C)no1 c1(OC)ccc2[nH]cc(CN3CC4CC3CN4C(c3cc(C)ccn3)=O)c2c1 O=C(CCC(=O)N1CCOCC1)NCCn1cc(CCO)nn1.C1(CN)CCCO1 c1(NC)ccc(Cl)cc1C(=O)NCC(O)CNC(c1ncc(Cl)n1C)=O c1(OC)cc(F)c(C(c2nnnn2C2CCOC2)OCc2cnoc2)cc1Br S(=O)(=O)(c1cnn(CSc2ccccc2)c1)Nc1nc(CC(=O)OCC)oc1 c1(CNC(=O)Nc2c(C)cnnc2)ccc(S(=O)(=O)NCc2ccccc2)cc1 Cc1cn2c(n1)C(C(=O)N1CC(CNC(c3ccc(C4CC4)s3)=O)C1)CCC2 C(CC(F)F)(C(=O)NC1CCCC1(C)C)N(C(c1nnn(CC)c1C)=O)C N1(C(C(CCC)OC)=O)CC2CCC(C(=O)NCCOCC(C)C)(C2)C1 c1(CC(=O)NC(C)CCCNC(c2nccnc2Cl)=O)ccc(F)c(Cl)c1 S(=O)(=O)(c1ccc(-n2cnnc2)cc1)N1C2CN(C(CC(C)(C)C)=O)CC21 C1(C(N(CC(=O)NCCC)C)=O)CCC(CC)CC1.c12coc(n1)C(C)NC2=O Cc1ccc(-n2nc(CCCO)nc2C(C)Sc2ccccc2F)c(C)c1 c1(C(=O)NC2CC(C)(NC(C=NOC)=O)C2)ccc(C2CC2(Cl)Cl)cc1 N1(C(C=C=C(C)C)=O)CCC(C)(CNC(=O)CCC2CC(C)(C)CO2)CC1 c1(C(=O)NC2C=CC(CNC(C(CC)(C)O)=O)C2)cc([N+](=O)[O-])c2nsnc2c1 c1(C(=O)NCC(CNC(Cc2n(C)nc(C3CC3)n2)=O)O)ccc2cccnc2n1 N1(C(c2c(C)nsc2C)=O)CCC2(CCN(C(=O)C(F)(F)CC(C)C)CC2)C1 N1(C(C2N(C(C3CCC(C)(C)OC3)=O)C(C3CC3)CC2)=O)C2CCC1CC1(C2)N=N1 c12cccc(c1)C2.CN1CCC(N(C(c2csc(Cl)c2)=O)C2CC2)C1 c1(C2(C(=O)NCC3CCN(C(C45CCCC4C5)=O)C3)CCC2)cc(Cl)ccc1F c1(NCC(c2ccccc2C)(C)C)ccc(NC(=O)OCCN(CC)CC)cc1 N1(C(c2cc(C(CC)C)no2)=O)CCC(F)(CNC(=O)C(F)(F)CC2CC2)CC1 C(N=c1nc(N2CCCCC(C)(F)C2)c2c([nH]1)CSC2)c1cc(OCC)ncc1 C12(C(=O)NCC(CC)NC(=O)C(F)CC3CCCC3)CCC(O)(CC1)CC2 C1(CC(=O)NCCN(C(C(CCC)O)=O)CCC)OC(C)(C)OC1=O c1(NCc2nccc(NC(=O)NS(=O)(=O)c3ccc(Cl)s3)c2)nccc2[nH]ccc12 Cn1ncc2cc(C(N3CC4CC(C3)CN(C(=O)CSC(C)(C)C)C4)=O)cnc12 C1(C2CC2)(NC(C2CC=CCC2)=O)CCN(C(c2ccc([N+](=O)[O-])cn2)=O)C1 Cn1[nH]c(=NC(=O)C23CC(c4nnc(-c5ccncc5)s4)(C2)C3)cc1Cl N1(C(CCN(CCC)C)=O)CCN(C(C23CCC(C2)OC3C)=O)C(C)C1 N1(C(CCSC)=O)CCOC(C(C)NC(=O)CCCc2sccc2C)C1 N1(C(CCOCCC)=O)CCOC(CNC(=O)C#CC2CC2)C1 c1(C(=O)NCc2cc(C(N(CCC(=O)OC)CC=C)=O)n[nH]2)ccc(C)cn1 N1(C(c2c(OC)nsc2)=O)CCC2(C1)CN(S(=O)(=O)c1cnoc1C)CCO2 c1(C(C2CC2)NCC(C)(C2CC2)NC(c2c(C)scc2)=O)nccc(Cl)c1F C(C(=O)N1CCC(O)(CC(C)C)C1)(C(C)CC)N(C(c1cn(CCC)nc1)=O)C c1(C(N2C(CNC(C(CCC=C)(C)C)=O)CC2)=O)ccc2c(c1)CCC=C2 c1(C(=O)NC2(CCO)CN(C(c3ccc[nH]3)=O)C2)cc2c(cc1Cl)NC(=O)CO2 CC(CC(=O)N(C1CN(CC2CCN(C3CC3)C2)C1)C)c1cnn(C)c1 C1(NC(C(C)(C)OC)=O)CCC(C(=O)N2CC2)CC1.C1CN1.C(CO)OC c1(CN(C)C(=O)NC2(c3ccncc3F)CC2)ccc(Cl)cc1F C(CC(C(=O)N1CCC(CN(C)C(C2CC2CF)=O)C1)N(C)C)N(C)C c1(OCCC(=O)N(C)CC2CCN(C(C3OCC3(C)C)=O)C2)cccc(Cl)c1Cl C1(CO)C2CC3CN(C(=O)CCCNC(CCC(=C)C)=O)C1C3C2.c1ccccc1 c1(C(=O)OC)cnc2ccoc2c1.C12CCC(C1)OC2=O CC(C(=O)NCC1CCC1NC(=O)C(C)(C)Oc1cccc(Cl)c1)C1=CCCC1 c1(N2CC(C(C)CNC(C(C)OCCC=C)=O)C2)cc2nn[nH]c2cc1[N+](=O)[O-] c1(C(=O)NCCN(C(C2CCC3CC23)=O)CC)nccc2c1[nH]c1ccccc21 C(=O)(C1Cc2ccccc21)C(C(CC=CC)N)=O.C1(CN)C(C)(C)C1(C)C C(CN=c1ccnc(CC(C)C)[nH]1)N1CCC(c2c(OC)cccc2)CC1 C1(C2C(CS(C)(=O)=O)C2)CCN(C(C=C)C(F)(F)F)CC1 c1(C(=O)NC2CC(CCNC(C(c3ccc(C)s3)C)=O)C2)cccc(Cl)c1F c1(N2CCC(NC(c3cccc(C4(F)COC4)c3)=O)C2)nc2cccc(Br)c2o1 C(N=c1[nH]c(=NC2CCC3CC3CC2)c2sccc2[nH]1)c1c(Br)cns1 C(CS(=O)(=O)C(F)(F)F)OCCN(CCCCCC)Cc1cccc2c1OCC2 C(=O)(CC(O)C(C)C)NCC(CCOC)NC(=O)OC.C1(=O)CN1C n1(CC)c(C)nn(CC(=O)N(C(C)CNC(=O)C(CCSC)N(C)C)C)c1=O C1(c2nnnn2C(C)(C)C)(NC2(OC)CC(C[Si](C)(C)C)C2)CCOCC1F C1(CN(C(=O)CCSCc2nnsc2Cl)C)CCC(C)(F)CC1 c1(OC)c(Cl)cc(C(N2CCOCC2CNC(C2CC(F)C2)=O)=O)cc1Cl N1(C(Cc2scc(C)n2)=O)CC(C)CC1C(=O)Nc1nc(C)cs1 CC(C)CC(O)CC(=O)N1CCN(C(C2CC23CCC3)=O)C(C(C)(C)C)C1 c1(N(C(C2(C(=O)NC)CC2)=O)CCN(c2ccccc2)C)ccc(Cl)cc1Cl Cc1nc2ccc(C(N3CCC(F)C(NC(=O)C4=CCCSC4)C3)=O)cc2o1 C(C)(CCC(=O)N(CCCCCNC(=O)CC(C)c1cccnc1)C)SC C(=O)(C(O)CCCCC)N1C2(C(=O)NCCC(CC=C)(C)C)CC(C1)C2 C1(C(=O)NCCC(C)N(C)C(C2CCCN2C)=O)CC12CCOCC2 c1(C(=O)NCC(CNC(C(C)Cc2ccco2)=O)C)ccc(-n2cccn2)cc1 c1(C(=O)NCC2CCN(C(CS(CCCC)(=O)=O)=O)C2)ccccc1C#CC1CC1 c1(C(=O)NCCCC(C)NC(COCCCCC)=O)cc2c(s1)CCOC2 C1(C(N2CC(F)(CNC(c3cc(C(F)(F)F)c[nH]3)=O)C2)=O)(OC)CCOC1 c1(C(N2CCC(NS(C)(=O)=O)C2)C(=O)NCCSC)ccc2cccnc2c1Br C1(CCC)CCCN1C(=O)C(Cc1ccoc1)NC(=O)C(=CC1CCCC1)C C1(C(=O)NCC2C(CC)C2)CCCC1NC(c1cnoc1C)=O C12(C(=O)NCC(CCCC)O)C(NC(c3nccn3CC)=O)C3CC1C2C3 c1(C(N(C2CCCC2)CCNC(COCc2ncc(C)o2)=O)=O)ccc([N+](=O)[O-])s1 N1(C(CC2CN(C(C=C(COC)C)=O)C2(C)C)=O)CC(CO)OC(C)C1 c1(NC(C(=O)NC)CC(C)(C)C)ccc2c(c1)COC2(C)C C(=O)(C(O)CC(F)F)N1CCC(c2cn(NC(c3c(CC)non3)=O)nn2)CC1 N1(C(c2nc(CC)oc2C)=O)CCC2(CC1)CC(NC(c1cc(C)ns1)=O)CO2 C#CC1(C(=O)N(C)CCN2CCCC2=O)CCN(C(=O)CC2CC(C)=NO2)C1 c1(OC)cc(CC#N)cc(CO)c1CN=c1ccc(C(F)(F)F)n[nH]1 C1(CNC(C=CSC)=O)CC2(CC2)CN1C(=O)C(c1cccc(C#N)c1)C(C)C c1(C(N(CCN(C(=O)C(=O)NCC(F)F)C)C)=O)ccc2ncn(C)c2n1 C1(CNC(C2(F)C(C)C2)=O)CCN(C(c2cnn(C)c2F)=O)C12CC2 Cc1nn2c(C(=O)NCC3COCC3NC(c3sccc3C)=O)c(C)nc2s1 C1(CSCC=C)CC2(CCNCC2)C(=O)O1.C1C(c2ccccc2)C(=O)N1 Cc1c(C(=O)NCC2CC2NC(c2ccc(C#N)s2)=O)cnn1C1CCCC1 c1(CC(=O)NC2CCN(C(C3C=CCCC3)=O)C23CC3)c[nH]c2cc(Cl)ccc12 C1(NC(C(CC)OCC)=O)CCC2CC1CN2C(c1nc(Cl)cs1)=O CCC(C)(CO)C(=O)N(C)CC1CC(F)CN1C(c1sc(N(C)C)nc1C)=O N1(C(C2(NC(N)=O)CC2)=O)CCC(CCNC(=O)C=Cc2cnc[nH]2)C(F)(F)C1 N#Cc1ccccc1OCC(=O)NC1CC(O)(CNC(C2(C#N)CC2)=O)C1 c1(C(=O)NCC2C3CN(C(C4(C(CC)=O)CC4)=O)CC32)nc(Cl)ccc1Cl c1(C(=O)NCC(C)N(C(=O)CN2CCOCC2)CC)cccnc1C c1(OC)cccc2[nH]cc(CN3CCN(C(=O)Cc4cc[nH]n4)C4CC34)c12 N1(C(CCC(C)c2ccccc2)=O)CC(=O)NCC1C(N1CC2CC1CN2C)=O C1(CCNC(C=CC(CC)C)=O)CCN(C(=O)C(C)C2CC2)C1 N1(C(C(C)NC(C)(C)C)=O)CCCC(N(C(=O)CSC)C)C1.c1(C=O)ccccn1 C(=O)(CCCCCC(C)(C)C)NC(C(C)NC(C1CCN(C(C)C)CC1)=O)CO N1(C(C2(OC)CS(=O)(=O)C2)=O)CCC2(C1)CN(C(=O)C=CC1CCCO1)CCO2 C1(C)(C(=O)NCC2CCC(C(=O)NC(CCOCC)C)CC2)CC2CCC(C1)S2 c1(CC(=O)NCC2(F)CC(CNC(CCOC)=O)C2)ccccc1C C1(NC(C2(CC=C)CCC2)=O)CCC(NC(C2CCOCC2C)=O)CC1 c1(OCC)cnncc1C(=O)N(CCOCC)CC.C(=O)COCCO C1(C)(C(=O)NC(CC)CNC(c2csc(-c3ccsc3)n2)=O)CCCOC1 c1(CC)ccc(C(=O)NCCCC(C)NC(=O)COc2cnn(C)c2)cn1 N1(C(c2cc(C)[nH]n2)=O)CC(F)CC1CN(C)C(C1CCN(S(C)(=O)=O)CC1)=O C(=O)(CC1COCc2ccccc21)NCCNC(c1c(N(C)C)cc(Cl)cc1)=O c1(C(=O)NC2CC(N(C(=O)CC(F)F)C)C2)ccc(F)c(F)c1N N1(C(C(c2ccco2)NC(=O)CC2CC=CCC2)=O)CCCC2(CC2)C1 CCC(CC(F)F)C(=O)N1CC(CCNC(c2cccn2C(C)C)=O)OC(C)C1 N1(C(c2c(C(C)C)ncs2)=O)CCOCC(NC(C2(n3cnnn3)CC2)=O)C1 c1(CC(=O)NCCC(N2CCC(CN(C(C)=O)C)C2)=O)ccc2cccnc2c1 Cc1cc(C(=O)NC2COCCN(Cc3ccc(Cl)nc3Cl)C2)ccc1O CCC(CC)C(C(=O)N1CCCC1C(C)(C)NC(=O)C=Cc1cnccn1)OC Cc1ccc(C)c(C(=O)NCC(CNC(=O)C(C)Cn2ccnc2)S(C)(=O)=O)n1 C1(C2CN(C(C3CC3(F)F)=O)C2)(NC(C(c2cn(C)nc2)O)=O)CC1 C(=O)(C1COc2ccc(F)cc21)N1CC2(C(CO)CN(C(C3C(C)(C)C3)=O)C2)C1 O=C(CC1=CCCC1)NCCC1CCCN(C(=O)C(c2cccc(Cl)c2)(F)F)C1 C(C(C(=O)N1CC(N2CCCC2=O)C1)N(C(=O)Cc1cnnn1C)C)OC c1(OC)ccc(C=CC(=O)NC2CCC(NC(c3nsnc3O)=O)C2)cc1 c1(C(=O)NCC2C(NC(=O)CC3CC3(Cl)Cl)C2)cc(C(F)F)cc(F)c1 c1(C(=O)NC2CCN(C(CC)=O)C2)ccc(C(=O)NC2CCCCC2O)c(F)c1 C=CC(C)CC(=O)N(C)CC1CCN(C(=O)C(C)OCCOC)CC1 CS(=O)CCC(=O)N1CCC(CCCCCNC(=O)CC2(C)CCC2)CC1 c1(C(=O)NC2CCN(C(C3CC(NS(C)(=O)=O)C3)=O)C2)ccc(Br)c(O)c1 c1(C(=O)NC2CN(C(C(C)(C)OC)=O)CC2C)ccnc(F)c1N c1(C(N(CCCNC(=O)C(C)(C(C)C)OC)CC)=O)cccc2nc(O)oc12 C(=O)(CCC(C)(C)C)N1CCC(CN(C(=O)Cc2cnns2)C)C1 c1(C(=O)NCC2C(CNC(c3c(SC)n(C)nc3)=O)C2)cc2ncccc2o1 C1(C(=O)NC(C)C)CCCC(NC(c2ccc(Cc3ccccn3)cn2)=O)CC1 C1(C(=O)NCC(C(C)C)(F)F)CC(F)(F)CN1C(c1ccncc1N)=O c1(C(N2CCCC(c3cc(C(=O)OCC)on3)C2)=O)cncc2c1CCCC2 c1(CCNC(=O)NCC(C)Oc2ccccc2)c(C#N)cnn1C c1(C(=O)NC(C)CCNC(=O)CC2CCC(=O)N2C)cnc2c(c1)CCOC2 N1(C(CSCCC#N)=O)CCC2(CC1)CCN(C(=O)CCc1cc[nH]n1)CC2 c1(CC)ccc(C(=O)NCCc2n[nH]cc2C(=O)NCC2COCC2O)o1 C(=O)(C(O)CC[S+](C)C)NCC1N(C(c2c(OCC)nccc2)=O)CC2(CC2)C1 c1(C(=O)NCCN(C(c2n(C)cnc2)=O)C2CC2)c[nH]c2cccc(Br)c12 Nc1cc(F)c(CC(N2CC3CCC(C2)N3C(C2CCCC(O)C2)=O)=O)cc1F N1(C(=O)NCCCC(C)(F)F)CC(CO)Oc2ccccc21 C1(NC(C(CCOC)NC(c2cccc3c[nH]nc23)=O)=O)CC2(CNC(=O)O2)C1 c1(OCC(N2CC3C(CNC(CC(C=C)(C)O)=O)C3C2)=O)ccc([N+](=O)[O-])cc1 C(CN(C)C(C1CCCOC1C)=O)(CO)(CO)NC(c1n(CC)ncc1)=O c1(C(=O)NCC2(CCCNC(CCOCC#C)=O)CCCC2)oc(C)cc1C C1(CCNC(c2ccn(C(C)C)n2)c2nnnn2C)CCCCC1(F)F N1(C(c2ccc(CC)o2)=O)CC(CC(=O)N(C(C)(C)CO)CC)C2(CC2)C1 C(=O)(C1CCCc2c[nH]nc21)NCC(CNC(C(C(CC)C)NC(C)=O)=O)O Cc1ccc(-n2nc(CCCN(C)C)nc2CCCCc2ccccc2)cc1 c1(NC(c2nnnn2C2CCC2)C)cncc(-c2ccccc2)c1 CS(=O)(=O)c1ccc(C(=O)NC2CC3CN(C(=O)CCC(F)(F)F)CC3C2)cc1 C1(OC)CC(NC(c2cnn(C(F)F)c2)=O)CN(C(c2cccc[n+]2[O-])=O)C1 C1(C(=O)NCC2CC(CNC(C(C)CC3CC3)=O)C2)CC1C1(C)COC1 c1(NC(c2c(-c3ccc(N(C)C)c(F)c3)nccc2)=O)ccc(C#N)c(O)c1 CC(CCC(=O)Nc1ccccc1Cl)NC(=O)CC=C(Cl)Cl n12cc(nn1)CN(C(=O)CC#N)CCNC(=O)C2.N1(C(C)C)CCC1 c1(C(=O)NCC(CC)NC(C2CCOCC2)=O)c(C2CC2)nn2ccccc12 C(=O)(C1=CCC(C)CC1)NCCOC1CN(C(c2c(C)nc(COC)s2)=O)C1 C(=O)(C(C(C)CC)NC(=O)C(C)CC1CCCC1)NC(CCC=C)CO c1(Cc2onc(C3C(C)CCC3)n2)cc(OC2CCOCC2)ccc1F CS(=O)(=O)c1cncc(C(N2CC3C(C(=O)Nc4ncc(F)cn4)C3C2)=O)c1 c1(CC(N2C(C(=O)Nc3cnc(Cl)cc3I)C(O)CC2)=O)ccccc1[N+](=O)[O-] c1(C(=O)NC2C(O)CCN(C(C(CCC)(C)C)=O)C2)cc2nccnc2cc1F C(=O)(C1=NOC(C)C1C)NCCOCCOC1CN(C(C(C)C2CCCC2)=O)C1 CC1c2ccccc2N(C(=O)CN2CCCC3(CCCNC3)C2)C1C C1(C(N(CCOCCCNC(C=CCCC)=O)C)=O)CC2CC2C1 N1(C(Cc2cccc(OC)n2)=O)CCN(Cc2cc(F)ccc2OC)CC1C#N C1(C(=O)NC2CN(C(COC)=O)C(C)(C)C2)CC(c2ccccc2)=NO1 CC1CC(O)CCN(C(=O)C(c2cn(C)nn2)NC(c2cccc(=O)n2C)=O)C1 C(C(C)(C)C(=O)N(CCN(C)C(C1CCCC1OC)=O)C(C)C)OCC C1(F)(CNC(C(C)CCN(C)C)=O)CCN(C(=O)C(O)Cc2cnc[nH]2)CC1 C(=O)(C(C)CC(C)C)NC1(C2N(C(c3ccc(C(C)=O)cn3)=O)CCC2)CC1 C1(NC(CC(N(C(CC(C)(C)OC)=O)C)C2CC2)=O)CCCCC12CCC2 C1(NC(C2(C(C)(F)F)CC2)=O)(CO)CN(C(c2coc(Br)n2)=O)C1 C(=O)(CCCCN(C)C)NC(C(=O)NCC1C(C)C1(F)F)Cc1ccco1 S(=O)(=O)(C1CCN(Cc2ccccc2C2CN(CC3CC3)CCO2)C1)NC(C)C CC1(C)CC(CNC(=O)CC2CC(F)(F)C2)N(C(c2csnc2Br)=O)C1 C(c1cncn1C)=CC(N1C(C2(NC(CC3(OC)CCC3)=O)CC2)CCC1)=O N1(C(COCCCC(C)C)=O)CC2(CCN2C(=O)CCC2CCCO2)C1 C1(CCOC)CCCCN(C(c2nonc2N)=O)C1 N1(C(C2C(CC)C2)=O)CC(C2(NC(=O)CC3(O)CCOCC3)CC2)C1 N1(C(CCC(=C)Cl)=O)CCCC2(NC(c3ccnn3C(CC)CC)=O)CC2C1 c1(CC(=O)N(CC(C)NC(=O)CCc2cncs2)C)ccc(C#N)c(F)c1 N1(CC#C)CCC(C(N2CCC(C)C2CNC(=O)C(F)=C2CCCC2)=O)CC1 N1(C(C(C)OCC=C)=O)CCC(NC(C2CCC(C3CC3)CC2)=O)C(C)(C)C1 C(CC(C(=O)NCC1(C)CCN(C)C1)NC(=O)C=CC(C)(C)SC)SC C1(CC)(NC(=O)CC2CC=CCC2)CCCN(C(=O)CSCCN2CCCC2)C1 C(=O)(C(C)C(=O)NCc1occc1C(=O)NC1CCN(C(N)=O)C1)OC N1(C(c2n(C=C)ncc2)=O)CCN(C(=O)C(c2cccnc2)O)CC1C(F)F Cc1cnc(NCC(O)CC2CCCCC2)c(S(=O)(=O)NC)c1.C1(C)CCOC1 C1(NC(C2CC(NC(C3(OCC)CCOC3)=O)C2)=O)CCCN(C)C1=O C1(CNC(C(C(C)C)SCC)=O)CN(C(=O)Cn2nc(C)nc2C)CC(C)(C)O1 c1(CC(=O)N(C2CCCN(C(=O)CC3(O)CCC3)C2)C)cc2ccccc2s1 Cc1ccnc2ccc(C(N3CCN(C(c4cccnc4S)=O)C4CC34)=O)cc12 C1(CC)CCC(C(=O)NC2CCOCC2C(=O)NC(C)CCCCSC)CC1 c1(OCCOC)ccc(C(=O)NC2CCN(c3c(Br)cncc3Br)C2)cc1OC c1(CN2C(C(=O)Nc3cc(C)c(O)cn3)CC(F)C2)cc(F)cc(C)c1O C(=O)(C=C1SCC(=O)N1C)N1CCOCC(NC(C(=C)CNS(=O)(=O)NC)=O)C1 C1(C)(CC)CC(NC(c2cnoc2C)=O)CN1C(=O)CCC(C)(C)N(C)C C1(CCNC(c2cc(C(=O)OC)on2)=O)CN(C(C23CCC2C3)=O)CCS1(=O)=O N1(C(CC)=O)CCC(NC(C2CCC3(CC2)CC3)=O)C(CO)C1 C1(CCNC(CCn2ncc(C)c2)=O)CSCCN1C(=O)CSc1n[nH]c(C)n1 c1(NC(N2C(Cn3ncc(C)c3)CC(F)C2)=O)cc(F)c(O)c(F)c1 C(=O)(C(C(C)C)S(=O)(=O)C1CCCCC1)N(CCc1ncc(CCOC)[nH]1)CC N1(C(C=CC=CC)=O)CCC(C(=O)NC(c2cncnc2)C)(COC)C1 N1(C(C(CCC)(C)CC)=O)CCCC2(CC(NC(C3CC4CCC3C4)=O)C2)C1 N1(C(C2(CC)CC2)=O)CCC(C2CN(C(C3CCN(CC(F)(F)F)C3)=O)C2)CC1 C(=O)(C(C)(C)C(C)O)N(CC(C)O)CCNC(c1c(C)cncn1)=O c1(C2C(CC(=O)O)C2)ccnc(C(N2CCC(C(F)(F)F)C2)=O)c1 CC1(C)CN(C(=O)CSCc2cncs2)CC1CNC(=O)C(O)c1ccsc1 CC1(CNC(=O)CSC(F)F)CCN(C(C2CN(S(C)(=O)=O)C2)=O)C1 c1(C(N2CC(C)C(NC(=O)CC3CCN(C)CC3)C2)=O)nnc(Cl)cc1N C=CCCCCCNC(=O)C(CO)NC(=O)C(N1CCNC1=O)C Cc1cc(C(N2CC(NC(=O)CN(C)C)C3(CC3)C2)=O)nnc1C Cc1c(NC(=O)Cc2cccc(F)n2)nc2c(F)c(Br)cnn12 Cc1cc2nc(C(N3CC(c4ccccc4)C4(CCC4)C3)=O)cc(=O)n2o1 C(=O)(C(O)CC(N)=O)NC(C(=O)N(C(C(=O)OCC)C)C)CCF N1(C(C2=C(C)OCC2)=O)CC(CNC(c2ccccc2Cl)=O)OC(C)(C)C1 Cc1cc(-c2cnccc2CN2CCC23CCCOC3)cc(O)c1 N1(C(CC(=O)NCC#C)=O)CCC(F)(F)C(CNC(=O)C=Cc2ccccc2)C1 C12(NC(C=CSC)=O)CCCCC1CN(C(c1ccc(C(F)(F)F)o1)=O)C2 N1(C(C2(COC)C=CCC2)=O)CC2(C1)CN(C(=O)C(C)Cc1ccc(C)cc1)C2 C(=O)(C(CCS(C)=O)N(C)C)N1CCC(C)(NC(C=C(COC)C)=O)C1 C(C(C)(O)CNC(C1C2CCCC12)=O)NC(C1(CS(C)(=O)=O)COC1)=O C(C(C)(C)C(=O)NCC1CCCC(CNC(C23CCC(C2)C3)=O)C1)N(C)C C1(CNC(=O)NC2C(C)C2C)CC(F)CN1C(c1cnn(CCF)c1)=O c1(CC(=O)NC(CCCC)CNC(=O)C#CC2CCC2)cc(F)c(F)cc1F N1(C(CCN(C(C)=O)C)=O)CCC(NC(=O)CC2(C)CC2)CC1C1CC1 C1(CNC(C2CN(C(C)C)C(=O)C2)=O)CC2(C1)CN(C(=O)C(O)C(F)(F)F)C2 C1(CC(=O)NCCC=CC=C)CN(C(=O)CCCCC)CC1C c1(CC)n[nH]cc1C(=O)NC1(C)CN(C(=O)CC2CC(SC)C2)C1 N1(NC(=O)C=CCOC)CC(OC)CC1OC.C(C=O)OCCOCCOC C(=O)(C(CC(C)C)C(N)=O)N1CC(C=CC)C(C(=O)NOCC(C)OC(F)F)C1 CCC(C)(CC)C(=O)C(Cn1cncn1)OC(=O)NC1CN(C(N)=O)C1 N1(c2nccc(=NCc3scc(C)c3)[nH]2)CCN2C(CCS2(=O)=O)C1 Cc1cc(C(N2CC(NC(c3cccc(Br)c3)=O)C(C)C2)=O)c2c(C)noc2n1 Cc1nc2cc(Cl)cc(C(N3CC(NC(C4(F)CCC4)=O)CC34CCC4)=O)c2[nH]1 CCC(CC)(CC(=O)OC)C(=O)N1CC(NC(C2CCS(=O)(=O)CC2)=O)C2CC2C1 c1(C(N2CCC(CCNC(C(CC)C#N)=O)C2)=O)[nH]nc2ncccc12 Cc1cccc2c1NCCC2C(=O)NC1(CNC(C2(C)CC(F)(F)C2)=O)CC1 CC1CCN(C(=O)CCCC2CCC2)CC1CNC(C1COCOC1)=O c1(C(=O)NC(C(=O)NC(CC)C)C2CC2)cnnn1C Cc1cncnc1C(=O)N(C)CC1(O)CCN(C(C2(n3cccn3)CC2)=O)C1 C#CC1CCN(C(=NCCc2ccccn2)NCC2CCCC2CCC)C1 c1(C(=O)Nc2cccc(CCC)n2)[nH]c(C)c(C(=O)NC2CSC2)c1C CC(CCC(C)(C)C)C(=O)N1CC2(C)CC1(C(=O)NOC1(C)CCCC1N(C)C)C2 C12(CO)CCCN(C1)NC(=O)N2.c1(C)ccccc1.CC1(Br)CC1C(=O)OC C(=O)(C1=CCCC1)N1CCC(CCNC(C2C(C)C2)=O)C1 c1(C(=O)NC2C(OC)CN(C(=O)C(C#N)C3CC3)C2)cc2c(C)ccc(F)c2o1 c1(CN(C)C(C2CCCOC2)=O)cnn2c1CN(C(C1(F)CCCCC1)=O)CC2 c1(OC)ncc(C(=O)N(C2CCCN(C(=O)C(=O)NC3CC3)C2)C)nc1C c1(COC)noc(CNC(C2(C)CN(C(=O)Cn3cncn3)C2)=O)n1 C(CN=c1[nH]c2ccccc2s1)NCCOCCNC(C1CC2CC2C1)=O Cc1c(NCC(C(F)F)n2cccn2)ncnc1N1CCC1CO C1(C(=O)NC2CC(C)(C)N(C(=O)CCC3CCC3)C2)CCc2nnc(O)cc2C1 N1(C(C(C)OCCCC)=O)CCCCC1C1CCCN(C(c2cnc(C)cn2)=O)C1 N1(CC(=O)OC)CCN(Cc2nc(-c3ccoc3)n(-c3ccccc3O)n2)CC1 CC1=CCC(C)(C(=O)NCC2CC(O)(CNC(=O)C=CCOC(C)(C)C)C2)CC1 Cc1nn(CC(=O)NC2CCN(CCc3cn(CCCF)nn3)CC2)c(C)c1C CC(CN(C)C)N=c1[nH]c(=NCC2CCS(=O)(=O)N2C)c2cccc(F)c2[nH]1 C(C1c2ccccc2CCN1c1ncnc(Cl)c1F)NC(C=CC)=O C1(C(=O)NC2CC(NC(C34C(C(=O)OC)(CC3)C4)=O)C2)CC2OC1C1CC21 CC(C)(C)C(CNC(=O)C1=NNC(=O)C1)C(=O)NCCC1CC2CCC1O2 C(CN=c1[nH]cnc2c(F)cc(Cl)cc12)N1CCN(C(=O)Cc2cnoc2)CC1 C1(NC(c2n(CC)cc(Br)c2)=O)CC2CC(NC(c3nn[nH]c3Cl)=O)C2C1 N1(C(c2ccc(F)s2)=O)CCC2CCN(c3nnc(-c4ccon4)s3)CC2C1 c1(C(=O)NC2(COC)CN(C(=O)CC3CCC(=O)N3)C2)cncc2ccsc12 C1(CN(C(C=C(CC)C)=O)C)CCC(NC(=O)CNC(C)=O)CC1 C(=O)(C1CCc2c[nH]nc21)NCCCC(C)(C)NC(c1cnc(O)c(F)c1)=O C1(CNC(C(CC2CCC2)NC(c2nc(C)sc2)=O)=O)CC(C)(C)CCO1 c1(C(N(C2CCN(C(c3cc(C)[nH]n3)=O)CC2)CC)=O)cccc(CS(C)=O)c1 N1(C(C=CC=CCC)=O)CCCCC(CNC(c2cnn(CC)c2C)=O)CC1 C12(CNC(CCOC(C)C)=O)COCCN1C(=O)CN(C(=O)C1=CSCCO1)C2 c1(C(C(=O)NC(CC)(C)CC)N(C)CCNC(C)=O)ccc(C(F)(F)F)c(F)c1 N1(CCC(=O)N(C2CCN(C(CC(CCC)O)=O)C2)C)CCCc2ccccc21 C1(N(C(C2(CNC(C3CCOC3C(C)C)=O)CC(=C)C2)=O)C)CC(C)CC(C)C1 c1(C(=O)NC2CCC(NC(C3(CCOC)CC3)=O)C2)cc(C)ccc1OC(F)F N1(C(c2ccc(Cl)cc2)C(=O)Nc2c(C)cccc2)Cc2cccnc2CC1C CCC(C#N)C(=O)N1CCCC1CCNC(=O)CC1(C)CCCC1 c1(-n2c(C3N(C)C(=O)OC3)nc(C3CC3(C)C)n2)cc(F)c2ccc(Cl)nc2c1 C1(NC(N2CCC(C(N(c3cccc(F)c3)C)=O)C2)=O)CC2(CCOCC2)CO1 c1(NC(C2C(NC(c3cccc(Br)c3Cl)=O)CCC2)=O)cc(Br)nc(Br)c1 C1(NC(=O)NCCOc2ccccc2Br)C2CC3C(C2)C13C(=O)O CN1CCC(O)(C2(C(N3CCC(CN(C(=O)C4=CCCCO4)C)C3)=O)CC2)CC1 Cc1nn(C)cc1NC(N1CCC(O)(CC(=O)Nc2cccnc2C2CC2)C1)=O c1(C(=O)NC2C(NC(CSCC=C)=O)CCCC2)cnc(C)nc1OC c1(CC(=O)NCC2N(C(C(CN(C)C)(C)C)=O)CCC2)cc(F)cc([N+](=O)[O-])c1 CC1CN(C(C2CC(=C3CCC3)C2)=O)CC(CCNC(=O)Cn2ncccc2=O)O1 Cc1cccc([N+](=O)[O-])c1NCCNC(c1conc1C=Cc1ccccc1Cl)=O C=C(Br)CC(C)(C)C(=O)NCC1CCCCN1C(=O)C(C)=C(C)CC c1(C(=O)NCCc2ccc(CNC(CC(=C)C)=O)cc2)ccc2c(n1)CCCC2 c1(CNC(=O)NC(C)C(c2ccnn2C)C)c(F)cncc1Br Cc1cnc(CNC(=O)C(N2CCC2C(=O)NCC2CCCC2)=O)c(C)c1 c1(C(=O)NCC(C)NC(Cc2cnc(C)[nH]2)=O)cc(CN2CCOCC2)n(C)n1 C1(NC(C23CCC(OC)C2C3)=O)CC12CCN(C(c1cnncc1C)=O)C2 Cc1ncc(C(N2CC=CC2C(=O)NOCC2CCCO2)=O)s1 C1(C(N(CCN(C(=O)CC2COCC(C)(C)O2)C)C)=O)CC(F)(F)C1(C)C C1(CC(=O)NC(CNC(C=CCC)=O)(C)CO)CSc2ccccc2NC1=O c1(C(N2CCC(F)(CNC(CCC(C)N(C)C)=O)C2)=O)ccn2ncccc12 c1(NC(=O)NCCN(C)CCO)cc2cccnn2c1 N#CCCCCCC(=O)NCC1CCN(C(C2CCCS2)=O)C1 C1(NC(C(C2CC2)OCC)=O)CCCCN(C(=O)C(C)S(C)(=O)=O)C1 N1(C(c2c(CCC)n(C)nc2)=O)CCC(C)C(CNC(=O)CC(C)C)C1 C1(CC(=O)Nc2c(OC)csc2)CCC2(CCN(C(=O)OC(C)(C)C)C2)O1 c1(NC(N(c2cccc(C(=O)NCC3CC3)c2)CC)=O)ncn2c1COCC2 C1(C(N(CC(C)(CO)CO)CC(C)C)=O)COCCN(C(=O)Cc2ccco2)C1 C(c1c(Cl)cccc1Cl)=C(C)CN(C(=O)C(O)CC(N)=O)CC1C2CC3C(C2)C13 c1(C(C)=O)[nH]c(C)c(C(N2C3CCC2(CNC(=O)COCC(F)F)CC3)=O)c1C S(=O)(=O)(c1ccc(C#N)c(N2CC=CCC2)c1)NC1(C=C)CCC1 C1(CNC(CC2C(C)CCCC2)=O)CC2(CC2)CN1C(=O)CCc1cnc[nH]1 C1(CC)CC(CC(=O)NC2(CNC(c3ccccc3O)=O)CC2)CCO1 C1(N(C(c2ccc(CN(C)C)o2)=O)C)CCCN(C(c2ncncc2Cl)=O)C1 c1(C(=O)NC(CO)CCCCNC(c2nc(Cl)cs2)=O)cc2ccc(O)cc2[nH]1 C1(CC(=O)NCCCCSC)CCCC1(F)F.C(CC(=O)NC(C)(C)C)NC(COC)=O C1(N(C(CC2C(CC)C2(F)F)=O)CC)CN(C(=O)C=Cc2cccs2)CC12CCC2 c1(-c2cn(CC(CNC(C(C)NC=O)=O)(F)F)nn2)cccc(Cl)c1 C1(CNC(=O)COCCCF)CC2(C1)CN(C(=O)CCCc1ccccc1Cl)C2 N1(C(C(=O)NCC(=C)C)CC2CCCCC2)CCCC(F)(F)CC1C c1(CC(N2CCN(C(C(CC)C#N)=O)CC2CF)=O)ccc2c(c1)OC(F)(F)O2 C1(C(=O)NCC=CCN(c2ccccn2)C(=O)C(O)CF)CCc2nnc(O)n2C1 C1(CN(C)CCc2ncc(Br)cn2)CCN(C(C2(C)CC(C)(C)C2)=O)CC1 c1(OCC(N2CCCN(C(C(CC#C)O)=O)C(C)C2)=O)ccc([N+](=O)[O-])c(C)c1 c1(C(N(C(C)CNC(c2coc(C3CC3)n2)=O)CC)=O)occc1C(C)C N1(C(c2c(OC(C)=O)c[nH]c2C)=O)CCN(C(=O)C(C)O)CC1CO N1(C(C=CCNC(C(C=CC)O)=O)=O)CCS(=O)CC1 C(=O)(C(F)C1CCCC1)NCCN(C(=O)C(C)c1cccs1)CC C1(C(C=O)OCC)CC(F)(F)C1.N1CCC1CNC(=O)CC1(CO)CC1 n1(CC#C)c(N(C)CCC2CCOC2)nnc1Cc1ccccc1C C1(NC(CCSCCC)=O)CS(=O)(=O)CC1NC(=O)CCCC(C)C CC(C)C(C(C)NC(=O)CS(N)(=O)=O)NC(=O)C=CC1CC1 N1(C(c2cnn(C)c2N)=O)CC(NC(c2c(F)cccc2Br)=O)C(C#N)C1 CCCCCCC(=O)NC1CCC(N(C(=O)C(CCC)OCC)C)CC1 C1(NC(C(C2(O)CCC2)OCC)=O)CC(F)(NC(=O)CC2CN(C(C)C)C2)C1 N1(C(c2ccc(-c3nnn(C)n3)cc2)=O)CC2CCC(F)(C2)C1 CC1=C(C(=O)NC2CN(C(=O)COc3cc(F)cc(F)c3)C3CC23)CCCC1 C1(O)(CC(=O)N(CC(C)CNC(=O)CC2CCC2(C)C)C)CCCCCC1 CCC(C#N)C(=O)N(CCCN(C(=O)CCc1ccc(Cl)s1)C)C N1(C(Cn2cc(C(C)O)nn2)=O)CC(CNC(c2cccc(CO)n2)=O)C(C)C1 N1(Cc2cc(OC)c(O)cc2)CCCC2(CCN(C(c3cnc(O)[nH]3)=O)C2)C1 N1(C(CCC#C)=O)CCC2(CCC(NC(=O)CC(C)N(C)C)CC2)C1 C(=O)(C(C)(C)C(C)NC(=O)CC1(O)CCC1)NCC1C(C)C1 N1(C(c2c(C)occ2)=O)CCCCC(CNC(=O)CCNc2cncnc2)C1 c1(CC)cc(F)ccc1-n1nc(-c2ccc(SC(F)F)cn2)nc1CC1=CCCC1 C1(OC)CN(C(c2nc(C)n(-c3nc[nH]n3)n2)=O)C(C)(CNC(=O)C(F)F)C1 c1(CN2CCCC(N(CC(=O)OC(C)(C)C)CC)C2C)cc2ccoc2cn1 C1(CCNC(=O)CC2CC23CC3)CN(C(=O)C(F)=CC2CC2)CCO1 CC(F)CC(=O)NC(C)(C)CCN(C)C(C1CC(C)(C(C)(C)C)C1)=O C1(NC(C(CC=C)CC)=O)C2COCC1CN(C(c1[nH]cnc1CC)=O)C2 C12(C(=O)NCC3CC(N(C(CCn4c(C)ncc4)=O)C)C3)CCC(=O)N1CCS2 c1(C(=O)NC2C(CC(=O)NCCCC(C)CO)CCC2)ncccc1O C#CCC(C(=O)NOCC1CC1)NC(c1cc(CCOC)[nH]n1)=O c1(C(N2CC3C(CNC(C(CC)SC)=O)(C3)C2)=O)cc(Cl)cc(C)c1O CC(CCN(C)C)C(=O)NCC12CC(CNC(C3C4COCC34)=O)(CO1)C2 N(C(=NCC=CC1CC1)NCc1ccco1)CC1(C)CCCO1 c1(OC)ccc(CC(=O)NC2CCN(C(c3cccnc3N)=O)CC2F)c(F)c1 C(=O)(C(CN(CC(N1CC=CC1)=O)C)CC1CC1)NC(=O)CC1CCOC1(C)C Cc1ncc(C(N2CC(O)CCC2C(=O)NCC2CC3(CCC3)C2)=O)cc1C#N CC(N=c1[nH]c(=NC(C)CS(C)(=O)=O)[nH]c2c1COC2)C1CCOCC1 Cc1[nH]nc2c1CC(C(=O)N(C)CCOCCN(C(=O)C(O)C(F)(F)F)C)CC2 Cn1ccc(C(=O)NCC2CCC(NC(=O)C=C3CCSCC3)CC2)cc1=O N1(C(CSCC#C)=O)CCN(CC(=O)NCC2CC(CCO)C2)CC1 c1(OC)cccc(-n2nnnc2C(c2c(Br)nnn2C)NC2(C)CCOC2=O)c1 N12CCC3CC(C3C1)C(=O)Nc1cc2nc(CC)n1.C=C=CCOC c1(CNC(C(C2CC2)OCC)=O)cncc(C(=O)NC2CC(=O)N(C)C2)c1 C(C)(C)(C(N)=O)NC(C1(C)CC(NC(C2C(C(=O)OC)C2)=O)C1)=O c1(C(N2CCN(CC3CCC3)CC2)C(=O)NCC(C)C)ccnc(Cl)c1Br [N-]=[N+]=NCCCC(=O)NC1CCCCCC1NC(=O)C(c1ccc(F)c(F)c1)O C1(NC(CC(CC)SC)=O)CCC2(CCN(C(c3ccnc(Cl)c3O)=O)CC2)C1 C(=O)(C1=NOC(C)C1C)NC(CCC(=O)NC(CCOC)C)(C)C c1(C(=O)NC2(CC=C)CNC2)cccc2sncc12 Cc1scc(C(=O)NC2C3CC2N(C(c2n[nH]cc2Br)=O)C3)c1C Cc1cc(C(N2CCC(N(CCO)C(c3occc3C)=O)C2)=O)ccc1C1CC1 C(=O)(C(C)CNC(C1CC(O)(CC=C)C1)=O)NCc1ccc(C(=O)OCC)s1 c1(C(C2CC2)NC(CC=CCC)=O)ccc([N+](=O)[O-])cc1 C(=O)(C(C)CC(F)F)NC1(CC(=O)NC(CCC)CO)CCCCC1 N12CC(F)(F)CC1C2=O.c1(NC(c2ccc(COC)cc2)=O)nnc(Cl)cc1Br c1(C(=O)NC2(C)CCN(C(C3C(COC)C3)=O)C2)cnc2cccnc2c1 C1(CNC(C(CC)NC(C)=O)=O)CC2(CC2)CN1C(c1cc(I)ccc1OC)=O N1(C(C(=O)NCC2CC2)=O)CCCC(NC(c2ccncc2Br)=O)C(F)C1 N1(C(c2c(C)onc2C2CC2)=O)C2CCC1CN(C(c1ccncc1F)=O)CC2 N1(C(C2(COC)CCCCO2)=O)CCCCC(NC(C2CC3(C2)CC3(F)F)=O)C1 C1(C(=O)NCCCN(C(=O)CC2CC2C(F)(F)F)C)(NC(C)=O)CCCCC1.C(N)(=O)N c1(C(=O)OC)cccc2c1OCCO2.N12CCCN1C(C)C2.C(CCCCC=O)OC N1(C(C2(C)CC2)=O)CCC2(CC1)CC(NC(c1ccn3ccnc3c1)=O)CCO2 S(=O)(=O)(c1cncc(Br)c1)NCC(=O)NCc1ccc(C(F)(F)F)cc1 C1(C(=O)OC)CCN(C(=O)NC2CCC3CCC2O3)C2(CCC2)C1 C1(CC(=O)N(CC(=O)NCc2cnccn2)CC)C(=O)NN=C1C C=CCC(F)(F)C(=O)N1CC(NC(=O)Cc2nn(C)cc2Br)CC(C)C1 N1(C(c2c(C)cc(Cl)cc2)=O)CC2CN(C(C3CC(C)(C)OC3(C)C)=O)CC2C1 Cc1nc2ccc(C(=O)NC(C3CCN(C(=O)OC(C)(C)C)CC3)C(C)C)cc2[nH]1 C1(C(=O)NCCC2CCN(C)C2=O)CC2(CCN1C(=O)C(O)C(F)(F)F)CC2 N1(C(c2cc(C)c(C(F)(F)F)cc2)=O)CCC(CNC(=O)CCN(C)C)C(F)(F)C1 c1(C(N(CC(C)NC(C2CC(n3cnnc3)C2)=O)C)=O)cc(C#N)on1 CCCCC(CNC(=O)CSCCOC)NC(C1CCC(=O)NC1)=O C1(CNC(CN2CC(C)(OC)C2)=O)CN(C(C2CCOC2)=O)CC1(F)F c1(C(=O)NCC(CC)NC(c2cnc[nH]2)=O)ccnc(C(C)(F)F)c1 c1(C(N(CC(C)NC(C2(C)CC(C)C2)=O)CC)=O)cnn2c1CCCC2 Clc1cc(-n2nc(C3CSC3)nc2-c2cn[nH]c2)cc(Cl)c1Cl O(NC(=O)C(O)C1CN(C(c2cc[nH]n2)=O)C1)CC=CC=CC CC1CCN(C(c2ncoc2C(F)(F)F)=O)C(C)C1NC(=O)C=Cc1nccs1 CCC(O)(C(=O)N(C(CNC(c1ccc(C)nc1)=O)C1CC1)C)c1ccccc1 C(=O)(C(C)(C)S(C)(=O)=O)NCC1(C)CC(NC(C(C)Cc2ccccc2F)=O)C1 CCCCCCC(=O)NCC1COCCN1C(=O)C=CSC c12ccc(nc1)C(=O)NC2.C1(CC(=O)NC2C(CCOC)C2)CCCC12CC2 C1(NC(C)=O)C2CCC(C2)C1CN1CCC(Oc2ccc(CNC(C)=O)nc2)C1 C1(NC(C2CCN(C(C3(C)CCC4CC4C3)=O)CC2O)=O)CC(CO)C12CCC2 C1(n2cc(-c3cnc(C)s3)nn2)CCCCN1C(c1ccccc1CN(C)C)=O C(=O)(C(C)(F)CC)NC(C(C)NC(CCSC)=O)(C)C C1(N(C(=O)CC2(CO)CC2)C)CCCCC1NC(=O)CNC(C1(C(N)=O)CC1)=O N1(C(C2(CCNC(c3c(CC)[nH]cc3)=O)CC2)=O)Cc2ccnn2CC1C C1(C(=O)OC)CCCN(C(=O)NC2(CNc3ccccc3)CCN(C)C2)CC1 c1(C(N2CC(C)(C)C(CNC(=O)C(F)CC3CCC3)C2)=O)c(N)cc(F)cc1F C(=O)(C1=NOC2(CCC2)C1)NC(C1CCN(C(c2cccc3nccn23)=O)C1)C N(C1CCc2sc(CNCCC3(C)NC(=O)NC3=O)cc21)C(=O)OC(C)(C)C C1(C(=O)NC(C(O)CO)C2CC2)CN(C(C2(O)CCCCC2)=O)CC12CCC2 C=CCCN=C(NCc1cccc(C(F)(F)F)n1)NCc1ccn(C)n1 S(=O)(=O)(c1ccc(C(=O)NCC2(F)CC(NC(=O)C3=COCCC3)C2)cn1)NC C1(N(C)C(c2cc(C(F)F)no2)=O)CN(C(c2cc(O)nn2C)=O)CC1(C)C S(=O)(=O)(c1ccc2c(c1)C(=O)C(=O)N2)C(C)=O.n12c(C)cc(c1C)C=CC(C)CC2 Cc1c(C(N2CC(NC(C3CCNC3=O)=O)C2)=O)sc2[nH]cnc(=S)c12 C1(NC(CCCCCCSC)=O)CC2CCCC(C1)N2C(c1ncncc1F)=O c1(C(N(CCCN(C)C(c2ccc(C3CCC3)cc2)=O)C)=O)cnc(=N)[nH]c1 CCCC(C)CCN=c1cc[nH]cc1S(=O)(=O)NC1CCc2ccccc2C1 n1(CCC(=O)NCC2(C(N)=O)CN(C(=O)Cc3cc[nH]c3)C2)cc[nH]c(=O)c1=O C1(CNC(C2CN(c3cccc(C)c3)C(=O)C2)=O)(CO)CCCC12CCC2 c1(OCC(=O)NC2C(NC(CCCCCOC)=O)CCC2)cccc([N+](=O)[O-])c1 n1(C(C)C(c2ccc(Br)cc2)=O)ccc(=NC(=O)NCCN(C)C(C)C)[nH]1 CC(C)C(C(=O)NC1CC(CC(N)=O)C1)S(=O)(=O)C1CCCCC1 O=C(CC1OCCc2ccsc21)NCC1(CCNC(c2csc(CO)n2)=O)CC1 C(c1ccnn1C)=CC(=O)N(C)CC1(NC(c2c(OC)scc2)=O)CC1 N1(C(c2c(CC=C)cccc2)=O)CC2CCCC(C1)N2C(C1CC(C)(C)CO1)=O CCCCCCC(C)C(=O)NC1(C)CCN(C(c2cnc(COC)s2)=O)C1 C1(C(N(C2CCCN(C(c3c(SC)snn3)=O)C2)C)=O)CCc2nnnn2CC1 C(CN=c1[nH]cnc2c1CSC2)N(C(C1C(CC)OCC1)=O)CC1CC1 S(=O)(=O)(CC(=O)NCC1(F)CC(CNC(=O)C(c2cccc(F)c2)C)C1)NC C1(CNC(C2(C)CC2)=O)CCC(NC(c2sccc2C2CC2)=O)CC1 C1(=CC(=O)N(CCCCNC(Cc2nc(C)sc2)=O)C)CCN(C)CC1 N1(C(CCNC(c2cn(CC=C)nn2)=O)=O)CCCC(CO)C1 c1(C(N2CC(C)(NC(C(CSC)C)=O)C2)=O)cc([N+](=O)[O-])cnc1O c1(C(N(CCC)CCNC(=O)CNC(=O)NC)=O)cc[nH]c(=NC)c1 c1(NC(C2N(C(C=NOC)=O)C3C(C2)C3)=O)cc2c(cc1Br)OCCO2 Cc1cnc(Cl)[nH]c1=NC1CC2CN(C(C3(C)CS(=O)(=O)C3)=O)CC12 CN(C1CCN(C(=O)NC(C)(C)C)CC1)N1CC(CC2CC2)C2(CCOCC2)C1 N1(C(C=CCNC(C2(CC)CCCC2O)=O)=O)CCC(C)(O)C(O)C1 Cc1cc(C)c(C(N2CCSCC2C(=O)N(C)CC2CCOC2C)=O)s1 C(C(CC(=O)NCCC1CC=CCC1)NC(c1cn(C)cc1C)=O)OC C1(C(=O)NCC(CC)(C)CO)C2CCN(C(C3(n4nccn4)CC3)=O)CC12 c1(C(=O)OC)sc([N+](=O)[O-])cc1NC(C1CC1NC(=O)Cc1cccc(C)c1)=O C=CCC(C(=O)N1CCC(C)(NC(c2cc(C(C)(F)F)n[nH]2)=O)C1)NC(C)=O Cc1nc2ncnn2cc1C(=O)NC1CN(C(c2csc(=N)[nH]2)=O)C2CC12 c1(N2CCC(COC)C2)nc(N2CCN(C)C(=O)C2)c2ccccc2n1 c1(C(=O)NCC23C(CN(C(C)=O)C2)C3)sccc1C1=CCS(=O)(=O)CC1 n1(CC)ncc(C(N2CC(NC(=O)COC3CCCCC3)C(CO)C2)=O)c1C N1(C(C(CC)(CC)CCOC)=O)CCc2ccc(F)cc2C(C)C1 Cc1cc(Br)c2c(c1)CN(C(C1C3CCOC3C13CCC3)=O)CC2 c1(C(=O)NC(C(C)C)CNC(C2(O)CCC2)=O)cc(C(F)(F)F)ccc1Cl C#CCCCCCC(=O)NCC(C)(CC)NC(=O)C(C)OCCOCC n1(CC(=O)OC)c(C)cc(C(N2CC(NC(c3ccc[n+]([O-])c3)=O)C3CC23)=O)c1C Cc1c(Br)ccc(S(=O)(=O)N2CCCN(C3CCNC3=O)CC2)c1F c1(C(N(C(CNC(C=CC)=O)C)CC)=O)cn2c(Br)c(C)nc2s1 Cc1ccc(I)c(C(N2CCN(CCNC(C3CCC(C)O3)=O)CC2)=O)c1 c1(COC(C2CC2Cc2ccc(Cl)cc2Cl)=O)cc2cc(F)ccc2o1 Cc1nc(CC(=O)N(CC(C)N(C(=O)CCCc2ncco2)C)C)c(C)s1 C1(CC(=O)NC(C)CSC(F)F)N(C(=O)C(=O)C(C)(C)C)CCC1(C)C Cc1cccc(CNC(=O)CC2CC(F)CN2C(=O)CC2(C)CCCCC2)c1F c1(C(=O)NCC(C)Cn2cc(C3(O)CCOC3)nn2)cnnc(Cl)c1 C1(CC(=O)NCc2n(C)ncc2)CCCCN1C(=O)CCn1cnnn1 C(=O)(C(CC)(CC)OC)N1C(C(C)NC(C=CCN(C)CC)=O)CCC1 C1(NC(C2(COC)CC(=O)C2)=O)CCN(C(=O)C(Cl)=CCl)CC1C c1(CCC(=O)NC2C(CNC(C(C)(C)OC)=O)COC2)ccc(OC(C)C)cc1 C1(C(N(CC(CNC(CCN(C)CCO)=O)(C)C)C)=O)CC12CCC(F)(F)CC2 C1(NC(c2c(C)ccn2C)=O)CC2(CCC(NC(C3CC4C=CC3O4)=O)CC2)C1 c1(C(C(=O)N(C(C2CCCCC2)CC2CCOCC2)CC)=O)cccc2c1CCC2 C1(NC(C(C=C)O)=O)CC(OC)CN(C(c2c(C(F)(F)F)n[nH]c2C)=O)C1 C1(C(=O)NCC2(F)CC(CNC(Cn3c(C)cnc3)=O)C2)CC2(C1)CC2(F)F C1(NC(CC(CC)O)=O)CN(C(=O)COC(C)CC)CCC1CO CCCC1C(=O)NOCC(=O)N1.c1(C(=O)OC)c(Cl)cnn1C c1(C(=O)NC2C(NC(c3nc(N(C)C)oc3)=O)CC2)cc(Cl)sc1Cl c1(C(=O)NCC2C(NC(C(N3C(=O)CCC3=O)CC)=O)C2)ccc(Br)cn1 c1(CCC(=O)NCCCCCNC(C(CC)F)=O)c(C)nc(C(C)(C)C)nc1O N1(C(C2CN(CC)C(=O)C2)=O)CCN(CC(=O)Nc2ccccc2)CC1(C)CC Cc1cc(C(N2CCC(CN(C)C(c3cc[nH]n3)=O)C2)=O)cc([N+](=O)[O-])c1Cl Cc1ccnc(N(C(C)C(C)O)C(CNC(CNCc2ccccc2)=O)C)c1 C(CNC(c1cc(Br)sc1C)=O)(C(C)(C)C)NC(CC1(OCC)CC1)=O c1(CN(OC)C(=O)NCCCc2cn(CC(=O)O)nn2)cc(OC)c(F)c(F)c1 C1(C(N(C)C)=O)CCC(NC(C2(CS(N)(=O)=O)CCC2)=O)CC1 c1(C(=O)NCC(CNC(C2(CC#C)CCCCO2)=O)CO)c[nH]cc(Cl)c1=O N1(C(c2c(CC)cno2)=O)CC(NC(=O)C(=O)NCCl)CC12CCOC2.c1ncc[nH]1 C(=O)(C(O)CCC(F)(F)F)NC.C1(C(=O)NN2C(C)CCC2)CC2(CCOCC2)CO1 C(CCCC(C)NC(=O)Cn1nnnc1C(C)C)NC(C1C(C(=O)OC)CC1)=O C(=O)(C(C(C)(C)C)C1CCC(F)(F)CC1)NCCN(C(=O)C(F)C(C)(C)O)CCC Cc1cn2c(C(N3CCC(C)N(C(c4cnn5c4CCC5)=O)CC3)=O)cnc2s1 N=c1nc2c(c[nH]1)CC(C(N1CCCN(C(c3ccsc3)=O)CC1CO)=O)CC2 N1(C(C)C)C(=O)CCC1C(=O)NCC(C)(C)NC(C1CC1c1ccc(Cl)nc1)=O c1(CC(=O)NCCN(CCCN(C)C)C(C2C(C=C)C2)=O)ccccc1O C(=O)(C#CC(C)(C)CNC(=O)C(CO)N(C)C)NCCCc1onc(C)n1 c1(C(=O)OCC(CCCC(=O)OCC)=O)cc2n(n1)CCCNC2=O c1(OC)ccc(O)c(C(=O)N(CCC(=O)Nc2ccc(C(N)=O)cn2)C(C)C)c1 C1(C#N)(C(N2CCC2CN(C(C(C)CSc2cccnc2)=O)CC)=O)CCOCC1 N1(C(C2C(C)CCO2)=O)CCN(C(=O)CC2CC3CC3C2)CC1 c1(OC)ncc(Cl)c(C(=O)NCC2CCN(C(=O)Cc3nc[nH]n3)CC2C)c1Cl C(=O)(C(C)S(N)(=O)=O)N(CC1N(C(C2(C=C)CCC2)=O)CCC1)CC N1(C(C(CC)NC(N)=O)=O)CC(NC(C2(O)CCC2)=O)C(C)C1 C1(C(N2CCC(C(C)NC(=O)OC(C)(C)C)CC2)=O)CCCC(C(=O)O)O1 CC1CCCC(CCN(C(C2CCCN(C(=O)Cc3cnoc3)C2)=O)C2CC2)C1 C1(C)(CC(=O)OC)CCCN1C(=O)NCc1ccccc1-c1cn[nH]c1 S(=O)(=O)(c1ccc(Cl)cc1C(=O)Nc1ccc(Cl)c(F)c1F)N(C)C c1(C(c2n(CCC3(C)CC3)nnn2)NCC2CCC(=O)N2)cc(F)c(Cl)cc1F N1(C(C(C(C)C)c2cccs2)=O)CC2(CCN2C2CC2)C1 CC1(C)C=CC(NC(c2cc(CNC(=O)CSC3CC3)cs2)=O)CC1 N1(C(C2(CC)CCOC2)=O)CC2CC(C1)N2C(C1CC1CC(C)C)=O C(=O)(C1CCCn2cnnc21)NCC1N(C(Cn2ncc(C#C)c2)=O)CC1 N1(C(C(C)N(C2CC2)CC)=O)CCC2(CC(C(N3CC(C)N(CC)C(C)C3)=O)C2)C1 CCC(CC(F)(F)F)C(=O)NCCC1CN(C(=O)CC2CC3CC3C2)CC(C)O1 C1(N(C(=O)CCC2CCCN(C)C2)C)CC2CCC(C1)N2CC1CCOC1 CC1OC(C)(C)OC1(C)C(=O)OCC(c1ccccc1N1CCOCC1)=O CCS(=O)(=O)CC(=O)N1CCCCC(CNC(C2CNC(=O)C2)=O)C1 C1(CCCC)CN(C(C2CC(CC(F)F)C2)=O)CCN1C(=O)CNC=O N#CC1(C(=O)Nc2cccc(OCC3CCOC3)c2)CCOCC1 c1(C(N(CCNC(=O)NC)C2CC2)=O)ccnn1C1COC1 C=CC(CCC)CC(=O)NCC(O)CC(=O)NOC1CCOC1 N1(C(C(C)NC(CC)=O)=O)CCC(CNC(c2ccc(Br)o2)=O)C1(C)C CCCC(C)(C)CC(=O)NC1CCCC(NC(=O)COCCSC)CC1 N1(C(C(C2CCCO2)NC(CC(=O)NCC)=O)=O)CCC(C)(CC(=O)OC)C1 N1(c2n(CC3CCCO3)c(CNS(C)(=O)=O)nn2)CCC2(CC1)CC2(F)F c1(CCNC(C2C(C)CCCC2)=O)cn2c(n1)CCCC2 N1(C(C2(CC=C)CCCNC2=O)=O)CCN(C(=O)C2=C(Cl)CCC2)CC(O)C1 C(=O)(CCC(C)(C)F)NCC1CN(C(C2CCCC(Cc3c(C)occ3)C2)=O)C1 C1(NC(C2CCC(C(=O)OCC)C2)=O)CC(F)(F)CC1Nc1ncc(F)c(C)n1 CC1CCCC(C(N2CCC(C3CCCN3C(C3CCCC3)=O)C2)=O)CC1 c1(CC)n[nH]cc1CNC(=O)CN(C(=O)Cc1cncnc1)C1CCCO1 c1(C(N2C3CC(NC(C(C)(C)CF)=O)C2CC3)=O)sccc1S(N)(=O)=O C=CC1(CC(=O)NC2CCN(C(C)=O)C2C)CN(C(=O)COC)C1 c1(S)ccc2c(O)c(C(=O)O)sc2c1.c1(C2C(C)C(C(=O)O)C2)c(F)cccc1F C#Cc1cc(C(=O)NCCOC2CN(C(=O)C(F)(F)CC)C2)cc(N)c1 c1(CNC(C23N(C(C(N4CC(C)C4)C)=O)CC(C2)C3)=O)ccc(S(N)(=O)=O)cc1 c1(CC(=O)NC2C(C(N(CCC(=O)NC)C)=O)CCC2)sc(C)cc1C C1(C(=O)OC(C(=O)NC(c2cnccn2)C)(F)F)COC(Cn2cccn2)C1 C1(C(N2CC3OCC(C)C23)=O)(NC(CCCOC)=O)CCC(C)(C)C1 C1(C(=O)OCC)CC2(C1)CN(CCCC1CC(C(C)(C)C)C1)C2 C#CC1CCN(C(C2CC(NC(c3ccc(CO)s3)=O)CCO2)=O)C1 C=CCCC(O)CN(C)C(C1CCN(C(=O)CCCC2CCCC2)CC1)=O c1(CC(C)C(=O)NCC2(NC(C3CC3F)=O)CCC2)ccc(F)cc1 c1(N(C)C)ccc(NS(=O)(=O)C2(CC(=O)C3CC3)CC2)c(C(F)F)c1 N1(C(C(CCC)NC(=O)Cn2ccc(C)n2)=O)CC2(CC(N(C)C)C2)C1 C1(NC(=O)C(=Cc2ccccc2)F)C=CCN(C(c2cnc(S)[nH]2)=O)C1 c1(C(=O)NCC2C(NC(C3(CC=C)CC3)=O)C2)ncc(OC)nc1OC N1(C(CSCC(=O)OC)=O)CCC(CO)C(NC(c2oc(Br)nc2C)=O)C1 CC(CC(=O)N1CCCC(N(C(=O)CC(=O)OCCF)C(C)(C)C)C1)C(C)(C)C Cc1ccc(Cl)c(N)c1C(=O)NCCC(C)CCNC(=O)C(C)N(C)C c1(CC(=O)NCC2CCN(C(CC3CCC(=O)NC3)=O)C2)ccc(O)c(F)c1 c1(C(=O)NCCN2CCC(Oc3ccc(Cl)cc3)CC2)ccc(C(F)F)cc1 C(=O)(C1=Cc2ccccc2C1)N1CC2C(C(N3CCC(CCC)C3)=O)C2C1 C(CC(Cc1ccccc1)C1CCC1)N(c1nnnn1CCc1ccco1)C c1(C(=O)NC2C(CNC(=O)COC3CCOCC3)C2)ccc(Br)c(F)c1 C(=O)(CCC(C(C)C)NC(=O)CSc1nc[nH]n1)NCC(CC)CO O=C1NC(=O)C(c2ccc(C(N3CC(O)(CNC(=O)C=C4CCC4)C3)=O)cc2)N1 N1(C(CCC2CC(NC(C(CCC)OC)=O)C2)=O)CCCC(N=[N+]=[N-])CC1 C1(=O)C(F)C(=O)N2CC(C2)O1.C(CC(=O)NCCCN(C)CCOC)OC C(=O)(C(CC)CCCCC)N1CCN(C(CC=C)=O)CC1C(F)F CN1CCCC(C(=O)NC2CCC(CC(N)=O)CC2)C1.n12cc(nn1)COCC2 N1(C(Cc2c(C)noc2Cl)=O)CCCC2(NC(c3cc(C)n(C(F)F)n3)=O)CC2C1 Cc1cc(C(=O)NCc2cc(C(=O)NCCCC(=O)NO)on2)ccc1C#N C12(C(N3CC(C=C)(CC(N4CC(C5CCCCC5)C4)=O)C3)=O)CC(C)(CCO1)C2 N1(C(C(C(C)C)OC)=O)CCC2CN(C(C3COCCOC3)=O)CCC12 c1(OC)ccnc(C(N2CC(NC(=O)CSc3ccccc3Cl)C(O)C2)=O)c1N CC1=C(C)CC(C)(NC(=O)CCOCCN(C)C(C2CSCC(=O)N2)=O)CC1 N1(C(C(N2C(=O)CCC2=O)C)=O)CCC2CCN(C(=O)CCc3ncccn3)CC12 C1(CC(N2CC(C3(O)CCCC3)C2)=O)CN(C(=O)CC2CCCOCC2)CC1(F)F C(CCCCC(=O)NC1CCCC1NC(=O)Cc1ccccc1)N(C)C C1(NC(COCCCC)=O)CCC(NC(=O)Cc2sc(O)nc2O)CC1 CC(C)(F)CCC(=O)N1CC(CNC(=O)Cn2nc(O)ccc2=O)C(O)C1 C(=O)(C1CCCn2cnnc21)N1CCC2CN(C(c3c(C)sc(O)n3)=O)CC21 C1(C(N2CCCC(NC(Cc3n(C)nnc3)=O)CC2)=O)CS(=O)(=O)CC12CCC2 N1(C(CCn2c(C)cc(C)n2)=O)CC2CC(NC(c3cn(C(C)C)cn3)=O)C1C2 c1(C(C(=O)NCC(C)NC(c2c(COC)onc2)=O)C)ccc(Cl)c(Cl)c1 C1(NC(CS(C(C)C)(=O)=O)=O)CCCCC12CCCN(c1cncc(Cl)n1)C2 Cc1c(C(=O)NCC2(NC(c3ccsn3)=O)CC2)cnc2c(Cl)cccc12 CC1(C)CN(CC2CC(F)(F)CO2)CCC1C(F)(F)F c1(C(N2CCN(C(C3C(C)C3C)=O)CC2)=O)nnc(O)cc1O Cc1[nH]nc(C(=O)NC(C2CCN(C(C3CCCCC3F)=O)CC2)C)c1C Nc1c(C(N2CCC(NC(C3CCc4nccn4C3)=O)C2)=O)nc(O)nc1O N1(C(CC2CC(OC)C2)=O)CC2CC(C1)N(C(=O)CN(C1CC1)C(C)C)C2 C(=O)(C(C)C(C)c1ccc(F)cc1)NCCC(=C)CNC(=O)CC1(C)CCCCC1 N1(C(COCC=C)=O)CCC(CC(C)NC(=O)C(CC)SC)CC1 C1(CCOCCNC(c2c(C)[nH]nc2Cl)=O)CN(c2ccncn2)CCS1(=O)=O c1(C(=O)NCC(CC)NC(C2CC(=O)N(C)C2)=O)c(Br)c2ccccc2n1C C1(CNC(C(=O)NCCOC)=O)(CO)CCN(C(C2CCNC2=O)=O)C1 C1(C(=O)NC2CN(C(C3C(C)(C)C3(F)F)=O)CC23CC3)=CNC2=CC=CC=C1C2 N1(C(CC2N(C(C)=O)CCC2)=O)CCC(C2(NC(c3sncc3C)=O)CC2)C1 N1(C(c2ccc(C(C)=O)[nH]2)=O)CC(CNC(=O)CCc2ccc(C)o2)CC(C)(C)C1 C1(CC(=O)N(C(C#C)C)C)(NC(=O)CCNC(=O)COC)CCC1 N1(C(c2scc(C(=O)O)c2)=O)CCCC(c2nc(C(F)(F)F)cs2)C1 CCS(=O)(=O)C=CC(=O)N1CC2CCC1C(CNC(C1SC3C=CC1CC3)=O)C2 c1(C(CF)NC(=O)NC(C2CCOCC2)C(=O)OC)ccc2c(c1)OCO2 C(=O)(C(O)CN(C)C)NCCCN(C(C)C)C(c1cc(-c2ccncc2)no1)=O C(CC(C(C)C)NC(=O)CN(C)C(=O)C1CC1)NC(c1c(OC)ccs1)=O C1(C(N2CC(NC(C3N(S(C)(=O)=O)CC3)=O)(CO)C2)=O)CCN(C)C1=O N1(C(CC2C(C)(C)C2)=O)CCOCC2(COCCN2C(c2snc(Cl)c2Cl)=O)C1 c1(CC)ccc(N)c(C(=O)NCC2CC3CN(C(C4COCCO4)=O)CC23)c1 C1(C(=O)NCC=CC(C)(C)C)CCC(O)CN1C(C12CSCC1C2)=O c1(C(=O)OC)scc(-c2ccc(C)cc2)c1NC(=O)Cc1ccns1 c1(C(N(C2CCCN(C(C3CNC(=O)C3)=O)C2)C)=O)cnc(C(F)(F)F)cn1 c1(NC(CC2(NC(=O)CN3CCSCC3)CCC2)=O)cnccc1CO c1(C(C)C(=O)NCCCN(C(c2c[nH]c(=N)o2)=O)C2CC2)ccc([N+](=O)[O-])cc1F Cc1nc(O)ccc1C(N1CCC(O)(C(C)CNC(=O)CNS(C)(=O)=O)C1)=O Nc1cc(C(N2CCCC(NC(C34CCCN(CC3)C4)=O)CC2)=O)ncc1Cl c1(C(N2CC(CN(C(C(C3CCOC3)OCC)=O)CC)C2)=O)ccc(O)c(C)c1C C(CCCC(=O)NCC1CN(C(=O)CSC(C)(C)C)C2CC12)SC N1(C(c2c(CC)scc2)=O)CCCC2C(NC(c3cncc(NC)c3)=O)C2C1 N=c1nc2c(c[nH]1)CN(C(=O)C(N1CC(=O)NCC13CC3)=O)CC2 C1(O)(CNC(CCc2cn(C)nn2)=O)CCCN(C(C2(C)CC(F)C2)=O)CC1 N1(C(C(C=C=C)C)=O)CCC2(C=C(C(=O)N3CC(=O)NCC3COC)C2)C1 N1(C(CCCC#C)=O)CC2CCC1C1CN(C(c3cccc(N)c3F)=O)CC21 c1(NC2CCCC(NC(=O)CN3CCCC3)C2)nc2ccc(F)cc2s1 C1(C)(C(=O)NCC2CC3(CN(C(C4C(=C)C4)=O)C3)C2)Oc2ccccc2NC1=O c1(OC(C(N)NC2CCC2c2ccccc2)=O)ccc(F)cc1 C12(NC(CNC(CCC)=O)=O)CCC(CNC(c3cnsn3)=O)(C1)OC2 c1(OC)c(F)ccc(F)c1C(N1C2CN(c3nccc(Br)n3)CC12)=O c1(CC(C(=O)N(CCC(C)NC(c2c(CC)cno2)=O)C)C)ccccc1C C(C(C(C)C(C)C)NC(=O)CC1CCCC1)NC(C(c1ccc(CC)s1)=O)=O Cc1[nH]nc2ncc(C(=O)NCCCN(C(=O)C(C)(C)F)C3CCCC3)cc12 c1(C(N2C(CN(C(C3C(C)OCCO3)=O)C)CC(F)C2)=O)ccc(N)c(N)n1 C(c1cc(OC)cc(F)c1)=CC(=O)NCC1(O)CCN(C(C=CCCC)=O)C1 c1(CC)cccc2ccc(C(N3CC(NC(=O)C(O)CC)C(C4CC4)C3)=O)nc12 C1(NC(C(CCNC(C=CCC)=O)N(C)C)=O)CCn2cnnc2C1 C1(c2n(CC)c(N3CCC(C)(OC)C3)nn2)NC(=O)NC2=C1C(=O)NCCC2 C1(C(=O)NC(c2ccccc2)CC=C)CN(C(=O)CCC)CCO1 C1(NC(C(C(C)C)F)=O)CCN(C(=O)Cc2csc(C3CC3)n2)C12CCC2 CC1CCC(NC(c2cc(O)nc(Cl)c2)=O)CN1C(c1cc(Br)ncc1Br)=O C1(COC)(CNC(C2CSCC(=O)N2)=O)CCN(C(=O)C(C)(O)COC)C1 C(=O)(CS(=O)(=O)CC(C)C)NC(CNC(C(C(=O)NC)(C)C)=O)(C)CO N1(C(C(CCC)N(C)C)=O)CC2CCC1CN2C(c1cnoc1C1CCC1)=O C1(C(=O)NCC(CNC(c2ccc(C(C)C)o2)=O)OC)CCCCS1 C#C[Si](C)(C)CCCNC(=O)NCC1CC1C1CCCC1 N1(C(C2CC(F)C2)=O)CCOC(C(=O)NCC2(n3cncn3)CC2)C1 C1(C(=O)NC(CC)CN(C)C(c2csc(C(C)(C)C)n2)=O)CN2CCN1CC2 C1(C(=O)NC2(C)CC(C(=O)NCCC=CC=C)C2)CN(C)CCN1C CC1CC(CC(=O)NCc2nc[nH]n2)CN1C(c1csc(C#N)c1)=O c1(CNC(=O)NCCCC(C)(F)F)ccc(F)cc1Br Cc1c(Br)ccc(C(=O)NCC(O)CNC(C2CCCOC2C)=O)c1F c1(NC(C2CCCCN2C(c2cncc(Cl)c2)=O)=O)cccc(F)c1F N1(C(c2cc(C)c(O)nn2)=O)CCN(C(c2cnco2)=O)CC(C)(C)C1 CC(CS(=O)C(F)(F)F)NC(=O)C(=O)NC1CCC(=O)CC1 N(C(=NCC(C)C1CC1)N1CCC(NC(=O)C(C)(C)C)C1)CCOC C1(NC(C2(C(=O)NC)CCC2)=O)CC2CC(C1)N(C(=O)C(c1c(C)n[nH]c1C)C)C2 N1(c2ccnc(C)n2)CC2CCC1C(NC(C1CCC(C)NC1=O)=O)C2 c1(C(N2CCC(CC(=O)Nc3cc(-c4ccco4)no3)C2)=O)cc(Cl)cnc1F c1(C(N2C(C)CCC(NC(C3CCSC3)=O)C2)=O)nnc2c(F)cccc2c1O C1(C(=O)OC)CCC(C(=O)NCC2CN(C(c3cccn3CC)=O)CCO2)CC1 C(CCCCNC(=O)C(n1ccc(C(F)(F)F)n1)C)NC(C(C)OCC(C)C)=O O(NC(=O)CC(C)CNC(=O)C=Cc1cnn(C)c1)C(C1CCCCC1)C c1(CNC(C(C=C)CC)=O)cc(F)ccc1F.C12C=CCCN1C2=O c1(C(=O)NC(CCN(C(C(C(C)C)N(C)C)=O)C)C)cccc2nncn12 c1(C(=O)NCC2CC(NC(C(C)c3ccsn3)=O)C2)ccccc1-n1cccn1 C(C(C)(O)C(C)(C)C)NC(CCN(C(CCc1c(C)noc1)=O)CCCO)=O c1(C(N2C(CNC(C3(CC(F)F)CC3)=O)CC(OC)C2)=O)cc2oc(C)cc2[nH]1 N1(c2ncc(C)c(O)n2)CCC(NC(=O)CC(C)(C)c2ccccc2)CC(C)(C)C1 N1(C(C2N(CC)CCCC2)=O)CC(N(C)C(c2nnccc2C)=O)C2(CC2)C1 CS(=O)(=O)c1ccc(C(=O)NCC(c2cc(F)ccc2F)=O)[nH]1 S(=O)(=O)(c1ccc(NCC(C)(C)C)c(F)c1)N(CC(C)OCC(C)O)C c1(C(N2C(CNC(COC)=O)CC(O)C2)=O)ccc(N2CCCC2)c([N+](=O)[O-])c1 c1(OC)ccc(C(=O)N(C)CCN(C(=O)C(O)P(C)(C)=O)C(C)C)c(Cl)n1 O=[N+]([O-])c1ccc(F)c(CS(N2CCC3C(F)CC23)(=O)=O)c1 C1(C(=O)NCc2occ(C)c2)CCC=CC1NC(c1ccon1)=O C1(C(=O)OCC2(OC)CC2)CCN(C(=O)CCc2c(C)noc2C)O1 C1(C(N(C2CCN(C(c3csnc3Br)=O)C2)CCC)=O)OCCC1C C1(C(=O)NC2CN(C(c3c(C)noc3C)=O)C(C)C2)Cc2ccccc2C(=O)O1 C(=O)(CN=c1cc[nH]cc1)NC1CCC(NC(C(CC)=CCCC)=O)C1 c1(C(=O)NCC(C2CC2)NC(CCn2c(C)csc2=O)=O)ccn2cnnc2c1 C=CCC(C(=O)N1CC(C(N)=O)(CNC(c2cc(C3(C)COC3)no2)=O)C1)OC c1(OC)ccc(C(N2CCCC2)CNC(=O)CC(C)F)cc1.C1(C)CCC=CCC1 CC(C)C(C)(O)C(=O)NCC1CN(C(c2n[nH]cc2C2CCC2)=O)CC1C C(=O)(C1=Cc2ccccc2C1O)N1CC(C)C(CNC(=O)CCCS(N)(=O)=O)C1 c1(C(=O)NC2C3(C)CN(C(CNC(C)=O)=O)C2C3)c(F)ccc(Br)c1F c1(C(=O)NCC2C(C)CCN2C(=O)CC(C)(O)C2CC2)ccc2c(n1)CCC2 C1(C(=O)NC(c2nnc(O)o2)C)CCC(O)CN1C(c1cc(Cl)c[nH]1)=O c1(C(=O)NCC(=O)OC(C)(C)C)ccc2c(Cl)ncnc2c1.C12CN(CCS1)C2 N1(CCCNC(=O)CC2CCNC(=O)C2)CCN(C(=O)C(F)(F)NC2CC2)CC1 C1(CCC(=O)NCC2CCCN(C(C3C(C#N)C3)=O)C2)CCc2ccccc2C1 c1(CC(=O)NCC2(F)CCN(C(c3nc(C(C)C)oc3)=O)C2)c(O)ncnc1O CCC(C)CCC(=O)NCCN(C(C1CCC12CCCO2)=O)Cc1ccccc1 c1(CC(=O)NCC(C)NC(CCOCCOC)=O)ccc2c(c1)OCCCO2 C(=O)(C(N)C(=O)N(c1cccc(C)c1)Cc1nc[nH]n1)OC N1(C(C(C(=O)OCC)F)=O)CCC2CCN(C(=O)C(C)O)CC12 C1(C(=O)NC(CC)CC(C)O)(COC)CCCN(C(C2C3CC(=O)CC23)=O)C1 C1(C)(C(=O)NC2CC(CNC(c3c(SC)cccn3)=O)C2)CCN(C)CC1 c1(OCC)cc(C(N2CCCC2c2nc(CNC(=O)C(C)(C)C)cs2)=O)on1 C1(C#N)(C(N2C(CNC(CCOCCC)=O)(COC)CCC2)=O)CC2CC2C1 N1(CCCNC(C2C(C(C)C)OCC2)=O)CCN(C(c2cccnc2)=O)CC1 CC(C)(C)CC1CC1C(N1CCC1CC(=O)NCC(O)C1CCC1)=O c1(C(N2C(CCOC)CN(C(=O)C(C)CSC)CC2)=O)cc2ccccc2nn1 N1(C(COC(C(N2CCC(C)C2)=O)=O)=O)CCC(OC2CCC2)CC1 c1(OCC)ccc(Cl)nc1C(=O)NCC(C)(O)CNC(C1Cc2nncn2C1)=O N1(C(C(COC)N(C)C)=O)CC(C2CCN(C(=O)CN3CCS(=O)(=O)CC3)C2)C1 C1(NC(c2ccc(C)nn2)=O)CC2(C1)CC(NC(=O)Cc1cnsc1)C2 N1(C2CN(C(C3OCC(C)C3)=O)C2)CCN(C(=O)C(C)(C)n2cnnn2)CC1 c1(C(=O)NC2CCC(NC(C3(CC)COC3)=O)CC2)c(C)nn(CCOC)c1Cl c1(CNC(=O)NCC)ccc2oc(S)nc2c1.C1(=O)C(C2CCCO2)O1 C(=O)(CC(C)C(C)C)NCC(c1ccccc1)NC(c1oc(CC)c(C)c1)=O C=C(Cl)CC(C(=O)N(CC(C)(CC)OC)C)NC(C1CCCN1C)=O Cn1nc(C(=O)NC2CCC2NC(C2(CC3CCC3)CC2)=O)ccc1=O Cc1ccc(NC(=O)CC2CCN(C(c3ccccc3)=O)C2)c(CNC(C)C)c1 CC1CN(C(=O)CC(=O)NCC2CC2)CCCN1C(=O)C1=CCC1 N1(CC)CCCC(C(N2CC3CC3(C(=O)NC3(C)CC(F)(F)C3)C2)=O)C1 C(=O)(C(CCC(=O)N(c1c(C)cccc1)C)N1CC(C)OC(C)C1)NC1CC1 C(c1ccncc1)=CC(=O)N(C1CCCC(NC(=O)CCc2cn[nH]c2)C1)CC Cc1ccc2oc(N3CC4CCC(NC(c5nn(C)cc5C)=O)CC4C3)nc2c1 C1(NC(CCC=CCC=C)=O)CN(C(=O)Cc2ccnc(C)c2)C2(CCCC2)C1 CC1(C(=O)NCC2CC3(CC3)CN2C(=O)C=Cc2cn[nH]c2)CCC(F)(F)C1 N1(C(CC2(NC(Cn3ncc(C)c3)=O)CCC2)=O)CC2CCC1C(CO)C2 C1(C(=O)OCC(=O)NC(=O)CCc2cnc(O)[nH]2)CC(=O)N(C2CCC2)C1 c1(CNC(=O)NCc2cnc(C)[nH]2)c([N+](=O)[O-])ccc(Cl)c1Cl Cc1cc(C(=O)N(CC(O)CN(C)C(c2cnc(C(C)O)s2)=O)C)ccc1N C(=O)(C1CSc2ccccc21)C(=O)C(Cl)=CCl.C12COC3(C1)CN(C3)C2=O C(CCC(O)C(=O)NC1(C(N)=O)CCCCC1)NC(C1C(CC)CC1)=O N1(C(C(C(CC)C)OC)=O)CCC(C2CC2)(CNC(=O)CCc2cnccn2)C1 c1(C(=O)NCC(=O)NCC2N(C(c3c(CC)ocn3)=O)CC2)cc(Cl)cnc1O c1(C(N2CC(C(=O)NCCCN3CCN(C)CC3)OCC2)=O)ccc(I)c(F)c1F c12ccc(cc1)CN2.C(=O)(C(C)n1cnnn1)NCC(=O)N(C)CC1C(C)C1 C1(C(N(C2CCN(C(=O)C3=C(C)CCCC3)C2)CC)=O)CC12CCC(=O)CC2 c1(C(=O)Nc2c(OCC)cc(C#N)cc2)cncc2cnccc12 N1(C(CCc2n(C)cnn2)=O)CCN(C(c2ncc[nH]c2=O)=O)CC1CO C1(CNC(CCN(C(CC)CC)C)=O)COC(C)(C)CN1C(C1CC2CC2C1)=O c1(C(C(=O)NCCC(C)NC(C2COCC2C(F)(F)F)=O)O)ccccc1Cl CCCC(C)(C)C(=O)N1CC(O)(CCNC(=O)C(C)Oc2cccnc2)C1 c1(CC(=O)NC(CNC(C(C)Cc2cccnc2)=O)CO)cc(O)nnc1O C1(CNC2CN(C(=O)OCC)C2)C2CN(c3cc(Cl)nc(CS(C)(=O)=O)n3)CC12 N1(C(CCOC)=O)CCCC(N(CCO)C(c2sccc2CSC)=O)C1 N1(C(CCCOC(c2ccccc2C(F)(F)F)C)=O)CCC(C)(O)C1 Cc1cccc2[nH]c(C(=O)N(C)CCNC(c3c[nH]c4nccc(Cl)c34)=O)cc12 CC(C)(C)C(CNC(C1CCCC1O)=O)C(=O)NCC=CC(F)(F)F n1(CCC)cc(C(C(=O)NCC2(OC)CCC2)N(CC)CC2CC2)nn1 C(c1ccc(SC)s1)=CC(=O)N(CC(C)NC(=O)CCn1cnnn1)CC C(=O)(CCC(N)=O)NC(C)CNC(CN(S(C)(=O)=O)C(C)C)=O Cc1cc([N+](=O)[O-])c(NC(C2C3CN(Cc4cccc(Cl)c4C)CC23)=O)cc1Br C1(C(N2C(C)(CNC(C(CCOC)OC)=O)CCC2)=O)CC2OC1C1CC21 N1(C(c2ccc(CNC(C3C(CC)OCC3)=O)nc2)=O)CCc2ccc(C)cc21 c1(C(=O)OC2C(c3ccccc3)(C)C2)ccc2c(c1)CCN(C(=O)C#CC(=O)O)C2 CCC(CCC(=O)NCC(C1CC1)N(C)C(c1cc(C)ccc1)=O)OC.C(=O)(C1CC1)N N1(C(c2ccc(C)o2)=O)CCCC(C(=O)NC2(C3CCCO3)CCC2)C1 c1(C(N2CC(CC)C(NC(=O)C(C)(C)F)CC2)=O)ccc([N+](=O)[O-])n1C C(=O)(C(CO)C(C)(C)C)N1CCC(COC)(NC(=O)CCOC2CCCC2)C1 C(c1ccc2ncccc2c1)=CC(=O)NC1CCCC1NC(=O)CC1CCOC1 c1(C(=O)NC(CC)CNC(=O)CCCc2ccsc2)cccc(S(C)(=O)=O)c1 C=C(C)CC(C(=O)NC1CCC(Cn2cc(C(C)CC3CC3)nn2)CC1)OC N1(C(C2N(C(C)=O)CSC2)=O)CCC(F)(C(=O)NCc2ccc(Br)s2)C1 c1(OCC(=O)NC2CCCN(C(CCC3C(C)C3)=O)C2)cc(F)ccc1F C1(C(=O)NC2CC(CC(=O)NC)C2)C=CCCC1CN1CCC(N2CCC2)C1 C(=O)(C(C)n1ccnn1)N(CC(C)N(C(=O)Cc1cscn1)C)C Cc1ccc(S(=O)(=O)C2(C(N3CC(N)CC(F)C3)=O)CCCC2)cc1 c1(CC(=O)NC2COCCN(C(c3cccc(O)n3)=O)C2)cc2cccnc2[nH]1 c1(CC)ccc(C=CC(=O)NC(C)CN(C)C(c2ccnn2CC)=O)o1 n1(CC)nc(C)cc1C(=O)NCC1CCC1NC(=O)Cn1ncnn1 c1(C(=O)NCC2N(C(C(C3CC3)SC)=O)CCC2(C)C)ccc2nn[nH]c2n1 CCC(CNC(c1cc(C)on1)=O)(CC)C(=O)NC(C)CCOC C#CCCN=C(NCc1ccc(C2CC2)cn1)NC(C)CCS(C)(=O)=O N1(Cc2ncn(CCN(C(C)=O)CC)c2)CC2CS(=O)(=O)CC2(C)C1 CC1CN(S(=O)(=O)CCNC(=O)NC(c2ccccc2)C(F)F)CC(C)O1 O=C(CS(=O)(=O)C1CCC1)NC1CCCCN(C(=O)C=CC2CCOCC2)C1 CC1CCN(c2nnc(CCCc3csc(-c4ccsc4)n3)n2CCC)CC1C c1(C(=O)NC2CCC(NCc3cocn3)C2)ccc(C(F)(F)F)cn1 C1(NCC#C)CCN(C(=O)C(C2CCCO2)C2CC2)C12CC2.C12C(C1C)NC2=O N1(C(C=C(C)c2cccnc2)=O)CC2CC(C)N(C(C3CC3C3CCC3)=O)C2C1 Cc1ccc2c(N(C)Cc3cn(C)cn3)nc(=NC3CCCC3F)[nH]c2c1 C1(NC(c2cnc(C(C)C)[nH]2)=O)CC2(NC(C3CC(C)(C)CO3)=O)COC1C2 S(=O)(=O)(c1ccccc1C#N)N1CC2CCN(C(C#CC)=O)C2CC1 c1(C(=O)NCCC2CCCN(C(CC(=C)C)=O)C2)cc(NC(C)=O)ccc1F N1(C(C(CC)(C)OC)=O)CC2CC(C1)C2NC(=O)C(CC(C)C)c1cccc(Cl)c1 C(=O)(CC(C)(C)OC)NC(CC)CNC(C1(n2cc(Cl)cn2)CC1)=O C1(C(=O)NC(CNC(C(CC#C)O)=O)CO)CCCC2(CC2)C1 c1(C(N2CCC(C#N)(NC(C3C(C(=O)OC)C3)=O)C2)=O)c(C)ccc(F)c1O c1(C(N2CCCCC(CNC(c3ccsn3)=O)C2)=O)cc2cccnc2o1 C1(NC(C2CC(CC)C2)=O)CCCCN(CC(N2CCCCC2)=O)C1 O=C(Cc1coc2ccc(F)cc12)NN=c1ccn2ncc(I)c2[nH]1 C12(NC(CCC(C)OC)=O)CCC(C1)N(C(=O)CNC(C1CCCC1)=O)C2 CC1CN(Cc2cc(F)ccc2I)CCN1C(C1CC(O)C1)=O N1(C(C23CC(NC(C4CC(N=[N+]=[N-])C4)=O)(C2)C3)=O)CCC(C2CCOC2)C1 c1(C(=O)NCC2C(NC(C(C)Cc3ccccc3Cl)=O)C2)ccn(C)c(=O)c1 C12(NC(CC(C)(C)OC)=O)CCC(F)(F)CC1CN(C(=O)C(C(C)(C)C)OC)C2 N1(C(Cc2ccc(C)s2)=O)CCC(C(N2CCNC(=O)C2)=O)C1C1CC1 N1(CC(N2CC(CC(C(=O)Nc3c(OCC)c[nH]n3)F)C2)=O)CCCCC1=O N1(C(C(N)=O)=O)CCC(CNC(c2nc3cnccc3s2)=O)C(F)(F)C1 c1(C(=O)Nc2c(O)ccc(C)c2)n[nH]c2c1CN(C(C1CC1c1ccoc1)=O)C2 N1(C(c2c(CC)onc2)=O)CCC(N(CC(C)C)C(c2cc(C)c[nH]2)=O)CC1 C1(NC(=O)Cn2cc(-c3ccc(Cl)cn3)nn2)CCCN(O)C1=O c1(CNC(C=CCNC(CC2(CSC)CC2)=O)=O)ccc(C(N)=O)o1 CC(C)(C)C(O)C(=O)N1CCN(C2CCN(C(C3CC4(C3)CC(F)C4)=O)C2)CC1 c1(C(=O)NCC(C)N(C)C(c2cncc(F)n2)=O)cc(C2CC2)cnc1Cl O=C(CCCCN1CCCC1)NCC(O)CNC(=O)C(F)CC1CCC1 C1(NC(=O)C=CC2CCCC2)CC(F)CN(C(C2CCS(=O)CC2)=O)C1 C12(CNC(C(CC)CC)=O)CCC(NC(C3CC34CCCOC4)=O)(CC1)CO2 N1(C(c2cscc2Br)=O)CCC(CNC(C2(F)CC=CC2)=O)CC1 N#Cc1ccc(CN2CC(NC(=O)CCc3ccoc3)C2)c([N+](=O)[O-])c1 CCS(=O)(=O)CC(=O)NCC1CC2CC1CN2C(=O)CCN1CCN(C)CC1 c1(C(=O)NCC(C2CC2)NC(CNC(CC)=O)=O)oc2ccccc2c1NC(C)=O N1(C(C=CCCC(C)C)=O)CCC(C)C(N(C(=O)Cc2cc[nH]n2)C)C1 C1(OC(c2c(C)con2)c2nnnn2CSc2ccccc2)CC(C)OC(C)C1 N1(C(CNC(c2ccc(C)s2)=O)=O)CCCCC(NC(c2ccc(Br)o2)=O)C1 N1(CC(C)CO)CCN(C(c2ccsc2)C)CC1.c12ccccc1OC2C c1(NC(CCC=C)(c2nnnn2CCC2(C)CC2)C2CC2)cnc2ncccn12 N1(C(c2ncc(CC)s2)C(=O)NCCCF)CCCCC1C1CCCO1 c1(OC)ccc(Cl)cc1CC(=O)N(C(C)CN(C(=O)Cc1cccs1)C)C CC1=C(C)CC(C(N2CC3(C2)CN(C(=O)Cn2cnnc2)C3)=O)CC1 Cc1ccccc1C1C(C(=O)NCC2CCCN2C(=O)CN(C2CCSC2)C)C1 C(=O)(CCCCOC)NCC(C1CCCC1)NC(c1ccn(CCCC)n1)=O CCC(O)C(=O)NCCN(C(C1(CO)CC1(F)F)=O)CC Cc1ncc(C(=O)NCC(C)(C)CNC(C2CC(CF)C2)=O)cn1 c1(C(C(=O)Oc2ccc(Cl)c(C(F)(F)F)c2)(F)F)ccc([N+](=O)[O-])cc1 C1(NC(=O)C=CC2CCCC2)CN(C(=O)CC2CS(=O)(=O)C2)C2(CCCOC2)C1 C1(NC(COC(C)=O)=O)CCCC1CNC(C1(N2CCOCC2)CC1)=O c1(CCC(=O)NCCCC2CCN(C(=O)CC=C(Cl)Cl)CC2)ccc(F)cc1Cl C1(CC=C)(NC(=O)CCCc2ncco2)CN(C(=O)CC2CCNC2=O)C1 c1(C(N2CC(CNC(C(N3CCOCC3=O)C)=O)C2)=O)ccc2[nH]ccc2c1F N1(C(=O)OC(C)(C)C)CCC(NC(=O)CC(C)C(F)F)C(Cc2ccccc2)C1 C1(C(=O)NC(CNC(c2n(C)cnc2)=O)(C)C2CCC2)CCCC(C)(C)O1 c1(C(=O)NC2CCC(NC(C3C(CC)CC3)=O)C2)ccccc1OC(F)F C(=O)(C1=NN(CC)C(=O)CC1)NC(CC)CNC(C1CC2CCCCN2C1)=O c1(OC)cc([N+](=O)[O-])c2nccc(C(=O)Nc3cc(CSC)c4sccc4c3)n12 c1(CCC)ccccc1C(=O)NC1CCN(C(c2cc(CC)oc2C)=O)C1C C(CCC(C)(C)C(=O)Nc1ccc(NC(c2n[nH]cc2Cl)=O)cc1C)OC N1(CC(=O)NC(C2CCCN(C(c3cnn(C4CC4)n3)=O)C2)C)C(=O)CNC1=O C(=O)(C1CCCc2ccnn21)NC1(CF)CCN(C(C(C)C2CC2)=O)C1 C1(CN(C(=O)Cc2cocn2)C)CCCN(C(c2cnc(=N)[nH]c2)=O)C1 CCCC(C)(CC)C(=O)N1CC(CC(C)NC(=O)C(C(C)CC)OC)C1 C=C(Cl)C(C)(C)C(=O)NCCOCCN(C)C(c1csc(C(F)F)c1)=O c1(NC(C(CC2CCC2)NC(C2CC3(CCC3)C2)=O)=O)ccc(CCO)cc1 c1(C(N2CC3CCC(CNC(c4c(C)cno4)=O)(C2)C3)=O)cnc([N+](=O)[O-])cc1C C1(C(N2C(CCC(=O)N3CC(CF)C3)CCC2)=O)CC2(C1)CC(O)C2 CC(C)CC(CNC(c1cc(=N)[nH][nH]1)=O)C(=O)N1CCCC1(C)CO C(c1cc(Cl)c2c(c1)OCCO2)=CCNCCCCc1ccc(Br)cc1 c12ccc(OC)c(c1)NC2.C1(CC(=O)OC)(C)CNC1.C1(O)CC1 c1(OC)cccc(C(C)NC(=O)CN2CCC(N(C3CC4CCC3C4)C)CC2)c1 N1(c2ccnc(CC)n2)CCC2(CNC(=O)CSSC)CCCCC12 N1(C(C(C)OCC=C)=O)CCN(C(=O)Nc2cccnc2)CC1 Cc1cc(C(=O)N(c2cccc(Cl)c2)CCCO)c([N+](=O)[O-])c(O)n1 N1(C(C2(C)C=CCCC2)=O)CC(F)(F)CC1(C)CNC(c1cc(C(N)=O)c[nH]1)=O C(=O)(CCC(C)(C)O)OCC.C(=O)(C(CC(F)F)c1ccccc1)N1CCC(C)C1 N1(C(CCC(CC)C)=O)CC(C(=O)NCCC2CCC(C)(C)C2)CCC1(C)C C1(CC(=O)NCC(CNC(C2(CC)CCCCC2)=O)O)COCC(C)(C)O1 CCCCC(CC)C(=O)N(CC(O)CNC(c1cc(-c2csc(=N)[nH]2)c[nH]1)=O)C C1(NC(c2ccc(SC)o2)=O)CCSC12CN(C(=O)CC1CCC(C)(C)C1)C2 C(=O)(C(F)(F)CC1CCCO1)NCC1(C(C)NC(Cc2nc(CC)sc2)=O)CC1 CC(c1ccccc1C)=CC(N1CC(NC(c2[nH]nnc2C)=O)CCC1C)=O N1(CC(C)NC(=O)C(O)Cc2ccccn2)CCN(C(C2(O)CCC2)=O)CC1 Cc1cncc(NC(C2CCCC(F)C2)c2nnnn2C2CC(F)(F)C2)c1 C1(NC(c2n(C(C)C)ncc2)=O)CCC(N(C(=O)CC2CCN(C)C2)C)CC1 c1(-c2c(C(C)NC(=O)C(=O)NCC3(CCF)CC3)noc2)ccccc1F N1(C(C2(OCC)CCOC2)=O)CC(CC(=O)Nc2cncc(C#N)c2)C2(CC2)C1 C=CCCC(C(=O)NCCc1cocn1)NC(=O)C=CC1CC1 C1(NC(CC(C=C)(C)O)=O)COC2(CCN(C(c3cc(OC)ncn3)=O)CC2)C1 CC1CN(C(=O)C(=O)NCC(F)F)CC(CCCCNC(C2CSC2)=O)O1 C1(NC(C(C)(C)Br)=O)CCC2(CC1)CN(C(c1n[nH]c3c1CCC3)=O)C2 c1(-c2cn(CC3CN(C(C4(n5cc(C#N)cn5)CC4)C)C3)nn2)cn(C)nc1C C(C(=O)NC1CCCC1CC(N1CCC2CCC12)=O)(C(C)C)OC c1(OC)nccc(C(=O)NC2CN(C(=O)C(C)OCC3CCCO3)C2)c1F c1(C(N(C2CCCN(C(CCSCC)=O)C2)C)=O)sc2cncn2c1C N1(C(C(CCCC)O)=O)CCC(C)(C)C(C(=O)NCCC(O)C(F)(F)F)C1 CCC(C)(O)CCNC(=O)CC1CC(CN)C1 C12(CC)CC(C1)ONC2=O.c1(C(=O)NC2CN(C3CCC3)C2)cnc(C)s1 c1(C(=O)NC2CCC(N(C(COCCC#C)=O)C)C2)ccc(P(C)(C)=O)cn1 n1(CC(=O)NCC2C(NC(C(CC)(C)OC)=O)C2)ccc2cc(F)ccc12 Cc1nc(C(C)(C)C)sc1C(N1CC=CC(NC(=O)Cn2cc(C#N)cn2)C1)=O c1(C(C2(CCC)CC2)=O)nccc2c1NCCC2.C(C(=O)NC)N(CCOC)C C1(NC(CC2OCC(C)(C)C2)=O)CC2CC(C1)N(c1nnco1)C2 N1(C(CCc2c(C)ccnc2)=O)CCC2(NC(c3cnn4c3CCC4)=O)CC2C1 Cc1nc2cc(Cl)cc(C(=O)NC3CN(C(c4ccoc4)=O)CC3C(F)F)c2[nH]1 c1(C(=O)NCCOCCCNC(c2c(C)nccc2)=O)cccc(O)c1Cl Cc1noc(C)c1CCNC(=O)CCCCN(C)C(C1(C(=O)N(C)C)CC1)=O C1(CCS(CC(N=c2cc(C)o[nH]2)=O)(=O)=O)CCC2(CCOCC2)CO1 c1(-c2c(C(=O)OC)csc2)c(NC(c2cncc(N(C)C)c2)=O)csc1C C(=O)(C1=NOCC1)NCCCNC(c1c(CC)nc[nH]1)=O Cc1ccc(C(=O)OCc2ccc(NCCNCOc3ccccc3)nc2)cc1 C1(C(C(=O)NC)NC(=O)CNCc2nc(C(=O)O)n[nH]2)CC=CCC1 C(C(=O)NNC(=O)C(C)n1cccc1)c1cn(CCCC(=O)OC)nn1 Cc1cc[nH]c(=N)c1C(=O)NC1CC(NC(=O)COc2cccnc2)C1 CCC(C)(O)C(=O)NCC12CC1CN(C(=O)Cc1ccn(CC(C)C)n1)C2 c1(C(N2CC(C#C)(C(=O)Nc3cccc(O)c3)C2)=O)cnc(F)c(C)c1 N1(C(C=CCCC)=O)CCCC2(CNC(c3cc(OC)n(C)n3)=O)CCCC12 Cc1c(Br)cnn1CC(=O)NC(C)(C)CCNC(c1ccc(N)cn1)=O c1(NC(C(c2scc(C)n2)N2CCC(OCC3CC3)C2)=O)ccc(Cl)cc1F c1(CC)[nH]nc(C(=O)NCC(C(C)C)NC(=O)C(C(C)C)SC)c1[N+](=O)[O-] n1(CC)nc(C(N2CCC(NC(c3ncccc3OC)=O)CC2)=O)cc1C1CC1 c1(C(=O)NC2CCC(NC(C3CN(C)C3)=O)CC2)cc(S(N)(=O)=O)co1 C(=O)(C(C)(C)C(C)(C)C)NC12CN(C(C3CCCN(CC(C)C)C3)=O)C(C1)C2 c1(C(N2CCC(CCNC(C(CC)F)=O)CC2)=O)nnc2ccccc2c1O Cc1coc(C=CC(N2CCC(Cc3ccc(CC4CCCN4C)cc3)C2)=O)n1 N1(C(C(CC)CN(C)C)=O)CCCC(N(C(=O)C=CC2CCOCC2)C)CC1 N1(C(C2(COC)CC2)=O)CCCCC(NC(=O)CC(C(F)F)c2ccccc2)C1 CCCS(=O)(=O)CC(=O)OCC(=O)Oc1ccc(Br)cc1F C1(N)CC2C=CC1C2.C1(CC(=O)NCC(CC)OC)CCC(C)C1 c1(NC(C2(OC)CCN(C(=O)CC34CCCC3C4)C2)=O)cc(C)ccc1C C1(C)(CNC(CCC=CCC=C)=O)CCC(NC(C2COCCO2)=O)CC1 C1(NC(C2CC(C(F)(F)F)(OC)C2)=O)CCN(C(C2CC(F)(F)C2)=O)CC1F N1(c2cc(NCC)ncn2)CC2CC1CCC2NC(=O)C(C)(C)CCOC C1(CC#C)(C(=O)OC)CCCN(CC(C)(C)O)C1 C1(C(=O)NC(CC)CN(C(=O)C=CCN2CCCC2)C)CCC2(CCC2)OC1 C(=O)(C(CC)OC)N1CC(N(C(CC)=O)C)C1.C12CN(C1)C2=O N1(C(C(C)C2CCC2)=O)CCC(NC(C2(S(C)(=O)=O)CC2)=O)C(CO)CC1 CC(C(C)(C)C(=O)N1CCC(c2ncc[nH]2)C1)NC(C1CCCC(C#N)C1)=O Cc1ncc(Br)cc1C(N1CC(C(=O)NCCN2CCN(C)CC2)C(C)C1)=O N1(C(C2CCSC2)=O)C2CCC1CC(NC(=O)C(c1ccc(F)c(F)c1)(F)F)C2 C(C(C(=O)N1CC(O)(C(N)=O)C1)C(C)C)NC(CC(CC)OC)=O c1(C(=O)NC(CC)CN(C(C2CCC(=O)N2)=O)CC)ccnc2[nH]cnc12 c1(C(=O)NC(CC)CN(C(=O)COC2CC2(F)F)CC)cc2c(s1)CCOC2 C1(O)(CNC(C2CCCC2)=O)CCCN(C(=O)CCCn2ccnc2)C1 N1(C(c2c(C)c(I)nn2C)C(=O)NCCSC)CCC(O)CC1(C)C C1(CCC)CN(C(=O)C=Cc2cccnc2)CCN1C(=O)CCn1ccnc1C CC1=C(C(=O)NCCN(C2CCCC2)C(c2coc(C(F)F)n2)=O)SCCO1 CC(C)(C)S(=O)(=O)CC(=O)NCC1CCC(NC(C2CC(F)C(=O)N2)=O)CC1 c1(C(=O)NC(c2ccccc2)CNC(C(C)(C)F)=O)ccn2ccsc12 N1(C(C2N(CC)CCC2)=O)CCC2CN(C(c3ccc(NC)cn3)=O)CC2C1 C1(NC(c2c(OC)n[nH]c2)=O)CCN(C(C2CC(=O)NC(C)C2)=O)CCC1CO CC1OCCC1(O)CNC(c1c[nH]nc1CNC(=O)CC1CC(N(C)C)C1)=O c1(N2CC3(C(=O)OCC)C(C2)CS(=O)(=O)C3)nc2ccc(Br)cc2s1 c1(C(=O)NCCC2(C(=O)NCC3CCC3)CC2)cnc(Cl)s1 N1(C(C(CC=CC)C)=O)CC2CC(NC(c3ncc(F)cn3)=O)C(C2)C1 c1(C(=O)NCC2(C)CCCN2C(=O)Cc2cc[nH]n2)cccc(F)c1O c1(CN(C(CN(C)C(c2cncn2C)=O)=O)C2CCC2)ncc(Cl)cn1 CCC(C)CC(C(=O)N1CC2C(C(=O)OC)C2C1)NC(=O)CCN1CCCCC1 c1(C(=O)NC(CN(C)C(c2cc(C3CC3)[nH]n2)=O)(C)C)ccc(N)c(F)n1 c1(OC)cc(OC)c(-c2ncsc2C(=O)NCC2CCC(=O)N2)c(OC)c1 c1(CC)ncc(C(=O)NC2CCN(C(c3csc(C)c3N)=O)C2C)c(C)n1 C1(C(=O)NCC(C)(C)NC(C2CC(C)OC(C)C2)=O)Cc2cc(F)ccc2O1 Cc1cccn2cc(C(N3CC4CCCC(C3)N4C(=O)C3=CCCC3C)=O)cc12 Cc1cc(C(=O)NCC2CCC(NC(C3Cc4nccn4C3)=O)C2)cc(N)c1O c1(C(N2CCC(SC(F)F)C2)C(=O)NC2CCOCC2)cnc2sccn12 C1(C)(CNC(c2n(CCC)nc(C)c2)=O)CCCN(C(C23CC(C)C2C3)=O)C1 c1(C(=O)NCCCCN(C(C2C(C=C)C2)=O)C)ncc(C(=O)NC)cc1Cl CCCC(C)(C)CN=c1[nH]c(=NC2CCCCC2N2CCCC2)[nH]c2c1SCC2 O=C1CC(CC(=O)N(C2CCCN(C(C3(F)CCCCC3)=O)C2)CCF)CCCN1 c12cn(C)nc1C1(CCC1)C(=O)ONC2=O.C1(SC)CCCC1OC(C)(C)C Nc1cc(C(=O)NCCCOCCNC(=O)CC2CCC2)cnc1Cl C1(=CC(=O)NCC2(NC(=O)C=CC3CC3)CCOC2)CCCCCC1(F)F N(C1CC2(CCCC2)Oc2ccc(F)cc21)S(=O)(=O)c1ccccc1F CC(C)(C)CC(O)C(=O)NC(Cc1cc[nH]n1)C(=O)NC1(C(N)=O)CCCOC1 c1(C(=O)OC(C)(C)C)cc(F)cc2c(S(=O)(=O)N3CC(O)C(F)C3)ccnc12 c1(CC(N2CC(C)CC(NC(C(C(CC)C)O)=O)C2)=O)ccc2ccoc2c1 c1(C(=O)NC(CCNC(C2(C(=O)NC)CCC2)=O)C)cc(C2CC2C)on1 N(C(=NCc1ccc(Cl)nc1)NCC1CCCCO1)C(c1cccs1)C C1(CNC(CNC(C(C)(C)C)=O)=O)CCCCC1NC(c1cnc(C2CC2)o1)=O n1(CC)cc(C(N2CC(NC(=O)CCc3cncnc3)CC2C)=O)c(C(C)C)n1 N1(C(C2CCN(C(CC(CC)O)=O)CC2O)=O)CCN(CC)C(C)(C)C1 C=C(C)CC(C(=O)N1CC(CC(C)NC(=O)C2=CCCSC2)C1)OC N1(CC)CCC2C(CCN2Cc2c(F)ccc(F)c2I)C1 C(CCC(=O)NCCC1CCN(C(=O)C(N2CCOCC2)C)C1)OC C1(N(C)C(c2n[nH]c(C3CC3)c2Cl)=O)CC2CC1N(C(=O)Cn1cnnc1O)C2 c1(CC(=O)NCCCN(C(=O)Cn2nnc(C3CC3)n2)CC)ccsc1Br c1(C(=O)NC2(C(=O)NC34CCC(CC)(OC3)C4)CC2)c(C2CC2)nc2sc(C)cn12 C(=O)(C(C)(C)C(C)(C)O)NCC1C(NC(c2cn(CC)nc2C)=O)CC1 CC(C)C(C(C)NC(c1ncncc1Cl)=O)NC(=O)C=CC(C)(C)C N1(C(C2CC(=O)OC2)=O)CCCC2(CNC(c3cnoc3)=O)CCCC12 CC1(C)CC(CONC(C2(C(=O)NC3(C)CCOC3=O)CCCO2)=O)CO1 Cc1cncc(C(=O)NC(CC2CCC2)C(=O)NCCCNC(=O)C(C)C)c1 N1(C(CCC=C(C)C)=O)CC(CC(=O)NC(c2nn[nH]n2)C2CC2)CC1(C)C CCC(CC)C(C)C(=O)N(C)CC1COCCN1C(c1ccc(S(C)(=O)=O)o1)=O C(=O)(CCCCCF)N(C)CC1CCN(C(c2cccc(Br)c2N)=O)C1 CC1(C)COC(CCC(=O)N(CCNC(=O)C(F)=CCCF)C2CC2)C1 c1(-c2cc(OC)c(O)cc2)n[nH]c2c1CN(C(=O)C(C(C)C)n1cnnc1)CC2 N(C(=NCc1ccc(C)o1)NCC(C1CC1)OC)CC(C)(C1CCCC1)OC C(=O)(CCCCCn1cc(C2CCN(C)C2)nn1)N(C(C(=O)OC)=O)CCC#N c1(CC(=O)NC2C(C(=O)Nc3c(C)cc(O)cc3)C2)ccc(C)c([N+](=O)[O-])c1 C(=O)(CCP(C)(C)=O)NCc1cccc(CNC(CCC=C)=O)c1 N1(C(=O)Cc2ccc(Br)cc2F)CC2CCC1CN2c1ncc(I)cn1 n1(CC)nc(C(=O)NC(C)CNC(=O)C(O)C(F)F)c(Cl)c1Br CC1(C)NC(=O)CC1C(N1CCC(F)(CNC(=O)Cc2cncnc2)CC1)=O C1(NC(CN(C(C)C)C(c2cnn(C)n2)=O)=O)CCn2nnnc2C1 N1(C(C2N(C(C3CCCO3)=O)CCC(CC)C2)=O)CCc2nc(C)[nH]c2C1 C12CC3CCC(C1)N3C(=O)C(C1CC(C)(C)C1)N2.c1(C(C)=O)cnc(N(C)C)nc1 C12(NC(CCCC#C)=O)CCOCC1CN(C(c1noc3ccc(Cl)cc13)=O)C2 CCC(C)CC(=O)N(CCCCN(C)C(c1ccc(-c2ccccc2)nn1)=O)C N1(C(Cc2c(C)noc2)=O)CCC(CO)(CNC(=O)C(C)C(C)C)C1 Cc1cc(C)n(CC(=O)NC2CC(CNC(c3ncc(C)cn3)=O)C2(C)C)n1 C1(CCNC(C2C(C(=O)OC)CC2)=O)CCN(C(C2CC(=C3CC3)C2)=O)C1 C1(NC(c2n(CC)nnc2C)=O)CN(C(=O)Cn2ccc(C(F)F)n2)CCC1CO C1(C(=O)NCC(C)CN(C)C(c2ccc3ccoc3c2)=O)CCc2cncn2C1 C1(CNC(c2cn(CC=C)nn2)=O)N(C(=O)Cc2cc(C)nn2C)CCC1(C)C N1(C(c2ccc(C)[nH]2)=O)CCC2CCC(C1)N2C(=O)C(=O)NCC(F)F n1(CCC(=O)NC(C2CCOC2)CNC(CCC(=C)C)=O)ccc2cccnc12 C=CC(CC)CC(=O)NC1CCOCC1NC(=O)C(C)=C(C)C c1(C(=O)NC(C(C(C)C)C)CNC(C23CC(CO2)C3)=O)ccnc2c1CCC2 N1(C(c2c(C)[nH]c(C(F)(F)F)c2)=O)CCC(C2CCN(C(C3CCO3)=O)C2)CC1 O=C(N1CC(O)CCO1)C1(Cc2cccc(F)c2)CCCO1 c1(CC(=O)NC(C)CNC(=O)CSC(C)(C)C)nncn1C(C)C C1(NC(C2(CCN(C)C)CC2)=O)CCC(NC(C2(P(C)(C)=O)CC2)=O)CC1 c1(NC(N(C)Cc2cn(CC3CC(CCC)C3)nn2)=O)cccc(C)c1 C1(NC(COC2CN(C(C3(COC)CCCO3)=O)C2)=O)CCN(C)C1=O CCCN(CCO)N1CC(NC(=O)OC(C)(C)C)CC1C(=O)NC1CC1 CON1CC(C(=O)NC(C)(CNC(c2cn(C)nn2)=O)C2CC2)CC1=O c1(C(=O)NCCCCN(C(C(C)CC2CC2)=O)C)ccc(S(C)=O)cc1 C(C)(N=c1[nH]c2c(c(=NCC3CC3)[nH]1)CCCCC2)c1nc(C(C)C)sc1 C1(C(=O)Nc2ccc(CC)s2)C(C2CC2)CCN1C(=O)CC1CCC(=O)C1 c1(CC(=O)NCCN2CCN(C(c3c(C)ccs3)=O)CC2)ccccc1S(C)=O Cn1ccc2[nH]c(C(=O)NC3CN(C(C4CC45CC5)=O)C4(CCC4)C3)cc12 c1(CNC(COCC=C)=O)cccnc1CNC(c1ccc(OC)cc1)=O C1(NC(=O)CC2CC3(CC3)C2)CCC2(CC1)CN(C(C1CCCC1O)=O)C2 c1(C(N2CCCC(CN(C)C(c3cc(C)nn3C)=O)C2)=O)cnc2ncccn12 c1(CCCC(=O)N(CCCNC(c2cccs2)=O)C(C)C)csc2ccccc12 C1(C(N2CCN(C(C(C)=C3CCC3)=O)CC(O)C2)=O)CCc2ccc(F)cc2O1 c1(C(N2CC(O)(C(C)NC(COCCCOC)=O)C2)=O)sc2cccnc2c1Cl CC1CCN(C(C2CC2F)=O)C(CNC(=O)Cc2c[nH]nc2O)C1 n1(CC(=O)N(CC(CC)NC(=O)CCCn2ccnn2)C)nc(C)n(C)c1=O c1(CNC(CC2(C)CC2F)=O)ncoc1C1CN(C(C2CCCO2)=O)C1 C(C(=O)N1CCC(F)(Cn2cc(CN(C)C)nn2)C1)(C(C)C)OC(C)=O Cc1cccc(C)c1S(=O)(=O)CC(=O)NC1(C(=O)O)CC(C)C1 C1(C(C)C)CN(C(=O)CCc2nccn2C)CCN1C(=O)COCP(C)(C)=O n1(CC)cc(C(=O)NCC(C)(CO)NC(=O)C(CO)NC(N)=O)nn1 Cc1cc(OCCn2cc(-c3nccs3)nn2)ccc1NCC12CCC(CC1)O2 C1(O)(C(=O)NCCN(C(=O)CSc2nccn2C)C)CCOC1 N1(C(C=C(CC)C)=O)CC2(CCCC2NC(c2cc(C#N)no2)=O)C1 CC1CC(C)(C(=O)NCC(=O)NCC(=O)NCC2CC23CCC3)C1 Cc1ncc2c(n1)CCC(C(=O)NCCNC(c1coc(S(C)(=O)=O)c1)=O)C2 N1(C(c2cncc(C)c2)=O)CC2(CCCC2)C1C(N1CCC2(CC(F)C2)C1)=O c1(NC(C2CN(C(C3CN(C(C)=O)C3)=O)CC(F)C2)=O)coc2ccccc12 c1(C(N(CC(CNC(c2nc(CC)oc2)=O)C)C)=O)cc(Cl)c(F)c(Cl)c1 N1(C(C(C)OCC2CCCCO2)=O)CC2CCCC(C1)N2C(C1C2CCCC12)=O c1(C(=O)NC2CCN(Cc3c(OC)ccc(C(C)C)c3)C2)cccc2ccnn12 N1(C(CSC(C)C)=O)CCC2(CCCN2C(c2nn(C(C)(C)C)cc2Cl)=O)C1 n12cnc3c(ncnc13)N1CCC(CC1)CC2CO.C12(CCF)CCCCC1C2 C12(C)CCN(C1)C(=O)CSc1cccc(c1)C(=O)N2.C1(CSCC)CCCCO1 C1(OC)CC(CNC(c2cc(CO)c(C)o2)=O)N(C(=O)CC2C=CCCC2)C1 N12CC3CCCC1C3(NC(=O)OC(C)(C)C)CC(C)(C)CCN(CCCO)C2=O C1(N(C(c2onc(CC)n2)C(=O)NC(c2cccnc2)C)CC)CCN(C)CC1 Cc1ccnnc1C(=O)NC1C2CN(C(c3cnn(C4CCC4)c3)=O)CC12 C(CCCC(=O)NCc1ncoc1C1CN(C(=O)CCCC2CCCO2)C1)OC c1(C(N2CCCC(NC(C(C)(C)CC3CCC3)=O)C2)=O)cn2cc(Cl)cnc2n1 CC1CN(C(=O)CCC2CCCCN2C(=O)C=CC(F)F)CC1O c1(C(N2CCC(COC)C2)=O)cc(N2CCCC2)nc(Cl)c1 c1(N2CC(C)(C)C2)nccc(N2CCOC(C3(C)CC3)C2)n1 c1(C(=O)NC2CCN(C(CN(CC)CC)=O)CC2C(C)C)ccc2ccoc2c1 C1(COC)CN(C(c2cc(C)ccc2I)=O)CCN1C(c1cc(C)on1)=O N1(CCCCn2cncn2)CCCC(n2nccn2)C1 c1(C(N2C(CNC(C(COCC)C)=O)C=CC2)=O)ccc(Cn2ccnc2)cn1 N1(C(=O)COc2ccccc2)CCN(C(c2ccc(F)c(C(F)F)c2)=O)C2CC12 N1(C(c2ccn(C)c2)=O)CCCC(CCNC(c2c[nH]c(=O)cn2)=O)CC1 CCCCC(C)(F)C(=O)NCCOCC(C)(C)NC(=O)CCN1CCN(C)CC1 N1(C(c2cnc(C)[nH]2)=O)C(CNC(C23CCC(C)C2CC3)=O)CC2CCCC12 C1(CNC(Cc2nnc(C)s2)=O)CN(C(c2sc(Cl)cc2Cl)=O)CCC1C Fc1cc(-c2nc(-c3cc[nH]n3)nn2C2CC3CCC2C3)c2nncn2c1 c1(C(=O)NCC2CCCCN(C(=O)C(F)CC3CCC3)C2)cccc([N+](=O)[O-])c1 Cc1cc(C(=O)NC(C)(C)C(=O)N2CC(c3nn[nH]n3)C2)cs1 c1(CC(=O)NC2CN(C(c3cc(C)n(C)c3C)=O)CC2O)cccc([N+](=O)[O-])c1 C(CNC(C1CSCCN1C(=O)CN(C1CC1)C(C)C)=O)(C(C)(C)C)OC C(=O)(CC(CC)C(C)C)NCC(CC)N(C)C(c1c(C)nn(C)c1C)=O C=CCCCC(C)N=c1[nH]c(NCc2cccc(SC(F)F)c2)nc2ccsc12 C(C(COC)CC(=O)NCCC1CCN(C(=O)Cc2ccsc2C)CC1)OC C1(=O)C(CC)(CC)CCNCC(C)(C)CNC(=O)CCC(CC)N1C.OC c1(C(=O)NC2CCC(NC(c3c(C)n(C)nc3C(F)F)=O)C2)cccc2c1COC2 CC1CC(=O)CCC1C(=O)NCC1(NC(=O)C=Cc2cccnc2)CCOCC1 C1(CC(=O)OC)CCCCCN1C(C(=O)NC)C1CC(CCCC2CC2)C1 C1(C2(O)CN(C(C3CC(F)(CO)C3)=O)C2)(CNC(=O)Cc2ccc(Cl)cn2)CC1 C(=O)(C(C)C(C)C)NC(CN(C(C(C)NS(CC)(=O)=O)=O)C)(C)C c1(C(=O)NCC(C)(CNC(c2ccc(Cl)s2)=O)OC)ccc(CO)nc1 N1(C(C)=O)CCC2(CC1)OC1(C)CC2(NC(=O)CCCc2ccc(C)c(C)c2)C1 C1(C(N2CC(N(C(c3cc(C(C)=O)oc3)=O)C)C3(C2)CC3)=O)CC2C(C1)C2(C)C N1(C(c2c[nH]c(=NC)s2)=O)CCC(O)(C(C)NC(=O)Cc2cc[nH]n2)CC1 c1(C(=O)NC2CCN(C(CCSCCCC)=O)CC2C)ccc([N+](=O)[O-])c(N)n1 c1(C(N(CCNC(c2sccc2Cl)=O)C2CC2)=O)ccc(C(=O)C(=O)NC)cc1 N1(C(CC2CCC(C)O2)=O)CCCC(C2CCCCN2C(c2coc(Cl)c2)=O)C1 N1(C(C=CC(C)C)=O)CCC2C(C(=O)NCC34CCCC3OCC4)C2C1 C1(C(N2CC(C)(NC(Cn3c(C)cnc3)=O)C2)=O)CCn2ccnc2C1 N1(C(C2=C(C)OCC2)=O)CCC(NC(=O)C=CC2(C)CCOCC2)C2(CCC2)C1 C12(CNC(=O)CN3CC(=O)NC3=O)CCC(CC1)CN2C(C1CC(O)C(F)C1)=O C1(NC(c2cc(C)on2)=O)C(C)CCN(C(=O)CC2CCC(=O)NC2=O)C1C c1(OC)ccc(C(N2CCC(C(C)NC(=O)COC(C)(C)C)C2)=O)c(F)c1 C1(NC(c2c(C)nc(CC)o2)=O)CN(C(c2[nH]ncc2C#N)=O)CC12CCC2 c1(C(=O)NCCOCCOC)n[nH]c2ccc(C(F)(F)F)cc12 c1(NC(c2n[nH]cc2NC(=O)CCc2ccc(F)nc2)=O)ccnc(Cl)c1 c1(C(N(CCCC(=O)NC(CO)C2(C)CC2)C)=O)cccc2c[nH]nc12 c1(NC(=O)CCOC(C)C)cn(C2CC(CNC(C(C)NC(C)=O)=O)C2)nn1 c1(C(=O)NCC2C(NC(COCCCOC)=O)C2)[nH]c(=N)ccc1C c1(C(=O)NCC2N(C(C(CC)CC)=O)CC(O)C2O)cnc2c(ccn2C)c1 O=C(C1=CS(=O)CCC1)NC1CC2CN(c3nc(C(F)(F)F)ns3)CC12 c1(C(=O)NC(CNC(C(C(C)C)OC)=O)CC(C)C)cc2c(F)cc(F)cc2[nH]1 Cc1oc(CO)cc1C(N1CCCCC1C(=O)NCC(C)CC1CC1)=O N1(C(C=Cc2nc(C)sc2)=O)C2CCCC1CC(NC(C1(N(C)C)CCC1)=O)C2 Cn1c(C(=O)NCC2(NC(=O)OC(C)(C)C)CCCCC2)cnc1O N1(C(CNC(C)=O)=O)CCC(CNC(c2c(C)noc2-c2ccccc2)=O)C12CC2 C1(O)(CNC(c2cn(CC=C)nn2)=O)CCCN(C(C2CCC3(CC2)CC3)=O)C1 C(=O)(CCC1=CCc2ccccc21)NC1CC(NC(C(CCC)C#N)=O)C1 N1(C(Cc2cnc(C)s2)=O)CCN(C(=O)CSCC(N)=O)CC1c1cccnc1 C(=O)(C(C)C(F)(F)F)NC1C=CC(CC(=O)NC2(c3nc(C)on3)CC2)C1 C1(CNC(C(C(=O)OC)OC)=O)CCN(C(=O)CN2CC(C)(C)C2)C12CC2 C(=O)(CCN(OC)C(=O)C(C)C1CCN(C(=O)CCNC(C)=O)C1)OC c1(C(C)C)cnc(O)c(C(=O)NCCCN(C(=O)C(C)(C)COCC(F)F)C)c1 N1(C(=O)Cc2cnsc2)CCN(CCNC(C23CCC(C2)C3)=O)CC1 N1(C(c2n(CC#C)ccc2)=O)CC(CNC(c2ccccc2C#C)=O)CCC1C N1(C(C(C)Oc2cccc(F)c2)=O)CC(n2cc(C3CCCOC3)nn2)C(C)C1 C1(C(N(C)Cc2cnc[nH]2)=O)COCCC12CN(C(C1CCCS1)=O)C2 N1(C(CCNC(=O)OCC)=O)CCCC(C)C1CNC(c1ccn(C2CC2)c1C)=O Cc1ccc(C(=O)NC(CNC(c2cc[n+]([O-])cc2)=O)C(C)C(C)C)c(=O)n1C Cc1ccc(Cl)c(NC(=O)NC2CC3C2CCN3C(c2ccnc(C)c2)=O)c1 C1(CCOC)CN(C(C2CNC(=O)O2)=O)CCN1C(=O)COCCSC C1(NC(C(c2c(F)cccc2F)C)=O)CC(F)CN(C(=O)Nc2cnn(C)c2)C1 Cc1cc(=NC(=O)CSCC(C)(C)O)[nH]o1.C1CN=C2N=c3scnc3=C(N2)N1 N1(C(=O)C=CC(F)(F)F)CCN(C2CCN(C(c3cncc(N)c3)=O)C2)CC1 Cc1nc(N2CCCC(NC(C3CN(CC(C)C)C3)=O)CC2)[nH]c(=N)n1 C(=O)(CCC(N)=O)N(C1CCN(C(=O)C(=Cc2ccncc2)C)CC1)CC c1(Cc2ccccc2)c[nH]c(=O)cn1.OC12CN(C1)CC1N(CCC1)C2 N1(C(CN(CCC)C)=O)CCN(C(C2CCC(=O)NC2)=O)CC1c1ncc[nH]1 c1(NC(CN2CC(=CCNC(C3(CC)CC3)=O)C2)=O)cc(=O)n(C)cn1 C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CCC(NC(CC(CCCC)O)=O)CC1 N1(C(C)C)CC(C(=O)N(CCC(C)NC(=O)Cc2cccn2C)C)CC1=O C1(C(=O)NCCCCCN(C)C(C2CCC(F)CC2)=O)CC2CC1CC2O C1(C(=O)NC(C=CC(=O)N(CC(=C)C)C2CC2)C)CC=C(C)CC1 c1(CC)cc(C(N2CC3CC3(CNC(=O)CN3CCN(C)CC3)C2)=O)ncn1 CC1OCCC1(F)C(=O)NCCC1CCN(c2cc(C3CC3)ncn2)CC1 CC1CC(NC(c2csc(-c3ncc[nH]3)n2)=O)CCN1C(C1(C)CC(F)C1)=O N1(C(c2nnn(COCC)c2N)=O)CCCN(C(C2CC2(C)Br)=O)CCC1 N1(C(CNC(=O)NC)=O)CCC(C(=O)NC(C)CN2CCCCC2)C1(C)C c1(C(=O)NCC2CCN(C(C=CCC)=O)CC2C)cc(Cl)cc(Cl)c1OC C1(C(=O)NCCCNC(c2nc(C)nn2C)=O)CC(c2cnn(C)c2)=NO1 CCC(CC(=O)NCC(O)CCNC(=O)CCN(c1ccncc1)C)C1CC1 Cc1cc(=NC(=O)COCCNC(=O)Cn2cc(C#N)cn2)[nH]n1C C(C(=O)NC1CCC(NC(=O)C=CBr)C1)(C(C)C)NC(C(C)C)=O C(C)(N=c1[nH]c(=NC2CC=CCC2)[nH]c2ncn(C)c12)c1c(C)cc(Br)cn1 N1(C(C2CC(F)(F)CS2)=O)CCN(C(=O)CC(F)(F)F)CC1C1CC1 c1(NC(=O)C(=O)NC2CC(O)C23CCOCC3)cc2n(n1)CCNS2(=O)=O N1(C(C(C)=C(C)C)=O)CC(C2CCCCN(C(C3CCCCCS3(=O)=O)=O)C2)C1 C(CCCC(=O)N1CC(C)(C)C1C1CCN(C(=O)C(C(C)C)NC=O)CC1)OC N1(C(C(C)O)=O)CCCC(C2CCCCN2Cc2cn(-c3cccnc3)nn2)C1 C1(C(N2CCCS(=O)(=O)CC2)=O)CCC2(CCN(C(=O)C(Cl)(Cl)Cl)CC2)O1 c1(C(=O)NCCCN(C(C2CCSC2)=O)C2CC2)[nH]nc2ncccc12 CCC(CC(=O)Nc1ccc(C2C(OCC(F)(F)F)C2)cn1)(CC)c1ccccc1 C1(NC(c2cc(C)no2)=O)CCCN(C(=O)C(C)n2cccn2)C1C S(=O)(=O)(c1cc(F)c(F)cc1F)N1C2CN(C(c3cc(C)cc(C)c3)=O)CC21 c1(CC(=O)N(CCNC(C(C)N(C)C)=O)C)ncc(Cl)n1C C=C(C)CC(C(=O)N1CC2CC2(NC(=O)C(N2CCCCC2=O)C)C1)OC C(=O)(C(O)CCCCC)NCCOCCN(C(CCCCCC)=O)C C1(NC(COCCNC(c2cc(CC)ncn2)=O)=O)CC12CCCCCC2 CCCCCCC(=O)N1CCC(CCOC)(NC(c2ccc(CC)o2)=O)C1 C1(C(=O)NCC(C2CCC2)NC(CC=C(C)C)=O)COC2(CCC2)CO1 Cc1cnn(CC(N2CC(c3ccccc3)(NC(=O)Cc3n[nH]c(C)n3)C2)=O)c1 O=C(CC1=CCOCC1)NCC1CCN(C(c2c[nH]cc2C2CC2)=O)C1 C1(CC(=O)NCC2CC(NC(C(c3c(C)noc3C)CC)=O)C2)CCC(C)(C)O1 c1(C(=O)NC(CNC(C(C)SC)=O)(C)Cn2cccn2)ccc(S(N)(=O)=O)cc1 C1(NC(C2CC3CC3C2)=O)CCCC12CN(C(c1csc(Cl)c1Cl)=O)C2 C1(NC(CCNC(C)=O)=O)CCCC(NC(c2cn(C(C)C)nc2Br)=O)CC1 C(=O)(C1CCCc2c[nH]nc21)NCC1CC(O)(CNC(C(CCCCC)F)=O)C1 C1(c2onc(C)n2)CCCN(C(=O)Nc2ccccc2CCF)C1 N1(C(=O)CNC(=O)CN(C(C2CC2Cl)=O)CC2CC2)CCN2C(=O)NCC2C1 CCC(CCCC(=O)NC(CO)CCC(C)C)NC(C1(COC)CCC1)=O C1(C(=O)O)CC(C(F)(F)F)CN1C(c1ccc(-c2ccc(Cl)cc2)cc1)=O c1(OC)cccc2c(C(N3CC(N(C(=O)C(C)SC(F)(F)F)C)C3)=O)c(C)[nH]c12 c1(C(=O)NCC2COC(CC3CCC3)C2)n[nH]cc1[N+](=O)[O-].C12(CC1)C(=O)NC2 CCC(C)(C)C(=O)C(=O)N1CC2CC1CN(C(=O)COC1CCOC1)C2 C(=O)(C1=CCCC1)N(c1ccccc1)C(CNC(Cc1nc(COC)sc1)=O)C1CC1 c1(NC(C(N2CCC(CNC(N(CC)CC)=O)CC2)=O)=O)cc2cccnc2[nH]1 C1(C(N2CC(CC=C)(NC(=O)CCOC3CC3)C2)=O)CCC(OC)CC1 C1(CNC(C=C(C)Cl)=O)CC(C)N(C(c2cnc(C)s2)=O)C1 N1(C(Cc2c(CC)noc2CC)=O)CC2CCC1CN2C(C1CCC2(CC2)C1)=O c1(C(N2CCC(NC(C34CC(CC(F)F)(C3)C4)=O)C2)=O)ccc(C2CC2)nc1 C1(C(=O)NC(CC=C)CNC(=O)C(C)Cc2ccc(C)cc2)CCCCCC1 N1(C(C=C(CC)C)=O)CCCC(C(C)NC(c2ncc(C)cn2)=O)C1 c1(OC)ccc(C(C(N2CCC(NC3CCOCC3)CC2)=O)NCC2CC2)cc1 N1(C(c2cc(C)nn2C)=O)CC(C(N2CC(N3CC(O)C3)C2)=O)CC1(C)C C1(C(=O)NC2(CNC(C3CCO3)=O)CCOCC2)CC12CCSCC2 C1(CNC(CC=CCOC)=O)CCCC(NC(=O)CC2(O)CCOC2)C1 CC1CCC(CC(=O)NCCCNC(c2cnns2)=O)O1 N1(C2CCN(C(C=C(CC)C)=O)C2)CCN(C(=O)CCCc2sccc2C)CC1 C1(O)(C(N2CCC(C(C)O)C2)=O)CCN(CC=Cc2ccco2)CC1 N1(C(C(C)n2cncn2)=O)CCC(CO)C(NC(=O)CCN2CCN(C)CC2)C1 c1(CC)ccc(C(=O)NCCn2cc(C(=O)N(C3CC(C)(C)C3)C)cn2)[nH]1 C=CC(C)CC(=O)N1CCOC(CCNC(=O)CSc2nncn2C2CC2)C1 c1(SC(c2ccccc2)=O)ccc2nnnn2n1.N12CC3CC(C3C1)NC(=O)C2 c1(C(=O)NC(CC)CN(C(=O)C=C2CCOCC2)CC)cn(C)c(C)n1 C=C(C)CC(C)C(=O)N1CCC(CC(N)=O)(NC(C2CCC3(CC3)C2)=O)CC1 c1(C(=O)NCC2(F)CN(C(c3c(NC)cc(Cl)cc3)=O)C2)ccsc1S(N)(=O)=O c1(C(=O)NCC(C)N(C(=O)CC2CSCCS2)CC)cnc(C)nc1CC C(N=c1cc(C2CC2)nc[nH]1)C1CN(C(C(c2ccccc2)OC)=O)C1 n1(CC)ncc(C(=O)NCC2C(C)CCN2C(c2ccc(C(C)=O)o2)=O)c1C c1(C(N2C(C)CC(NC(C3CCC(COC)O3)=O)C2)=O)cc(C)c(O)nn1 N1(C(CCOC)=O)CCC2(CCC2)C(CNC(C2CC2C2CCCCC2)=O)C1 c1(NC(C2(C)C(C(C)(C)C)CCC2)=O)ccccc1-n1ccnc1 CC1CN(C(c2cnc(O)n2C)=O)CCC1C(=O)NCC1CCC(C)(C)CO1 c1(OC)nn(C)cc1C(=O)NCC1CCCC1NC(c1ccsc1)=O c1(CNC(C(C2CC2)SC)=O)ccc(C(=O)NCC(C)C)nc1 c1(C(=O)NCC(=O)NC2CC2)cncc(C(F)(F)F)c1 N1(C(C2ON=C(CC)C2)=O)CCC(F)(F)C(CNC(c2cc(C#N)c[nH]2)=O)C1 C1(NC(C(C)=C(CC)C)=O)CCC(C)(CNC(=O)C(C)OCCN(C)C)CC1 n1(CC)ncc(Cl)c1C(=O)N(C)CC1CCN(C(c2cnc(C(N)=O)cn2)=O)C1 CCCC(C)CCCC(=O)NCC1CC(C)(C)CN1C(=O)C1=CCSC1 c1(CNC(=O)NC2CC(CCC(C)SC)C2)nc(C2CC2C)cs1 N=c1nc2c(c[nH]1)C1CCCC(C2)N1C(=O)Nc1ccc(CO)cc1 N1(C(C2(OCC)CCCOC2)=O)C2CCC1CC(NC(c1cc(Cl)cnn1)=O)C2 c1(C(N(CCCNC(C(CC)c2cccnc2)=O)C)=O)ccc2n[nH]cc2n1 N(C(=NCCN1CCC(C)(C)CC1)NCC1CCCO1)CC1(OC)CCCSC1 C1(NC(CCSCCCC)=O)CCCN(C(=O)C(F)(F)C(C)O)CC1F C(=O)(C1NCCc2ccccc21)Nc1c(NC(C)=O)ccc(N=[N+]=[N-])c1 C1(NC2CN(C(C(=O)NC(C)CCO)=O)C2)C2CCC1(c1ccn(C)n1)C2 Cc1cc2c(cc1C(N1CCCC(C(C)(O)CNC(C3(O)CC3)=O)C1)=O)OCO2 N1(C(c2n(CC)nnc2)C(=O)NCCC2CC2)C(C(N)=O)CC2CCCCC12 CC1CN(C(=O)C(F)=C2CCC2)CC1NC(c1csc(-c2ccoc2)n1)=O N1(C(C2C(COC)C2)=O)CC(CCNC(C2(c3nccn3C)CC2)=O)(OC)C1 C1(C(=O)NC2CC(CNC(=O)Cc3cccc(Cl)c3)CC2O)OC2CCC1CC2 N1(C(c2n(CCC)ccc2)=O)CC(CCNC(c2ccc(C)cc2)=O)C(C)C1 C(C)(N=c1[nH]c(N2CCCN(CC)CC2)nc2ccsc12)c1c(CC)cncc1 Cc1nccc(C(=O)N(C2CCN(C(c3cnc(C#N)s3)=O)CC2C)C)c1N N1(C(c2n(C=C)nnc2)=O)CCC2(CC1)CC2CNC(=O)CCc1cc(C)[nH]n1 c1(C(N(C(CC)CNC(c2cn(CCOC)nn2)=O)C)=O)cnc2ccccn12 C1(NC(CC(c2ccccc2Cl)C)=O)CCN(C(=O)C=CC(=O)NC2CC2)CC1C C1(C(=O)NCC(C)(C)C2(O)CCC2)CC12CCC(F)(F)CC2 N1(C(C(CCC)OC)=O)CCCN(C(=O)COc2cccnc2)CC1C(C)C C(N=c1[nH]c(C)cc(=NC2CCC3CC2CO3)[nH]1)C1CCN(CC)CC1 C(CCF)(C(=O)NC1(CF)CCN(C(C)=O)C1)NC(C(C)N(CC)CC)=O C1(CC)CCCC1(C)C(N1CCN(CCCNC(=O)C2CC2)CC1)=O N1(C(c2c(C)cc(C)o2)=O)CCC(C)C(CC(=O)NC2CCCC(O)C2O)C1 CP(C)(=O)CC(=O)N1CCCC1C1(NC(=O)COc2ccc(Cl)cn2)CC1 C1(CNC(C(C)(C)F)=O)(CNC(c2cncc(Cl)c2)=O)CC12CCC2 C(=O)(CCCC(=O)C1CC1)N1CCC(N(C(=O)CCC2CC2)CC2CC2)CC1 O=C(CC(c1cccs1)N)NCc1ccsc1.N1(C)CCCC1 C(C(C)(O)CC(=O)N1CCC(C(=O)NCCC(F)(F)CO)(C(C)C)C1)OC C#Cc1cccc(C(N2CCC(N(C(=O)C(C)C(O)CCCC)CC)C2)=O)c1F c1(OC)c(Br)cc(F)c(OC)c1CNCCc1nccs1 C1(NC(=O)CNC(=O)C2CC2)CN(C(=O)CSc2nc[nH]n2)C2CC12 Cc1ccccc1OCCSc1ccc(NC(N2CCC(CCF)C2)=O)cc1 C12(C(=O)NCCC(C#C)C)C(NC(C3CN(C(N)=O)C3)=O)C3CC1C2C3 C(CCCCCC(=O)NCC1CCCN(C(=O)CC2CC(=O)NC(=O)C2)C1)SC C(Cc1ccoc1)(C(=O)NCCC(O)C1CC1)NC(=O)C=CCF c1(C(N(C)CC)=O)cc(S(C)(=O)=O)ccc1OC.c12cccc(c1Cl)C(=O)N2 N1(C(c2c(CC)cno2)=O)CCCC(F)(CNC(C2CC(F)(CO)C2)=O)C1 c1(C(N2C(C(C)(C)NC(C(C)C(F)F)=O)CCC2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 c1(C(=O)NC2(CC=C)CCN(C(C3CCN(C)C(=O)C3)=O)C2)cnc(Cl)cc1N CC1=C(C(=O)N(C(CC(C)C)C(=O)NN2CC(NC(=O)C3CC3)C2)C)SCCO1 N1(CC(=O)NC2CN(C(=O)CCSC3CCCCC3)CCC2O)CCCCS1(=O)=O C1(C(=O)NC2CC(NC(CSc3cc(C)cc(F)c3)=O)C2)CCc2nn[nH]c2C1 c1(C(=O)NC2(CC(=O)N(CCOC)C)CCC2)ccc(C)c(O)c1 C=CC(CC)CC(=O)N1CCCC(NC(=O)C(=O)Nc2ccc(C)cc2)C1CC C1(CC(=O)NCCN(C(C23CCC2C3)=O)Cc2ccccc2)CCOCC1 CCCN=C(NCc1ccc(CC(=O)Nc2ncn(C)n2)cc1)NCC C1(OC)CN(C(c2sc(CSC)nc2C)=O)CC1NC(C1(F)CCOCC1)=O N#Cc1cc(S(=O)(=O)CN2CCCC(CCN)C2)ccc1F.N12CCCC1C2=O CC(C)(C)C(CC(=O)N1CC(O)C(F)C1)NC(C1C(CF)C1(F)F)=O Cc1ccc(C(=O)NC2CC3CCC2N3C(=O)CC(C)c2cnn(C)c2)nc1C Cc1cccc(C)c1OCC(N1CC(NC(=O)CCc2ncco2)C(F)C1)=O c1(C(=O)NC2CN(C(C=C)=O)CC2c2ccccc2F)ccnc2ccncc12 C12CC3CN(CC13)C(=O)C1(CCOCC1)C2.c1(C(=O)OCC)csc(CO)n1 c1(C(=O)NC2CC(CNC(c3c(CC)nn(C)c3)=O)C2)cnc(C2CC2)nc1O c1(C(N2CCN(C(C=CCOC)=O)C(C(C)C)C2)=O)ccn2c(C)ncc2c1 Cc1cc(C)c(NC(C2(NC(=O)CCCn3ccnc3)CCC2)=O)cn1 O=C(CC1=CCN(C(C2CC=CCC2)=O)CC1)N(CCCO)CCO c1(C(=O)NC2CC(CCNC(C(Cc3c(C)nc[nH]3)O)=O)C2)csc([N+](=O)[O-])c1 CCC(C#N)C(=O)N1CCC1C(=O)N(CCCOC)C C1(NC(N(c2ccc(F)cc2)C)=O)CCN(C(=O)CC2CC(=O)NC2=O)CC1O c1(C(N(C)CC2(O)CCN(C(C(C)OCC#C)=O)C2)=O)cccc2nncn12 C(C(O)CC(=O)NCc1nocc1C(=O)N(C1CC=CC1)C)N(C)C Cc1ccc(SCC(=O)NCC23CC2CN(C(=O)CC(C)(F)F)C3)cc1C N1(C(C(C(=C)C)(C)O)=O)CC(C)(C)OCC1CNC(c1ccc(C2CC2)[nH]1)=O c1(C(N2CCCC(C(=O)NCC(=O)NC)CC2)=O)ccc2cncnc2c1 c1(NC(N2CC3C(N(C(C)C)Cc4ccccc4)(C3)C2)=O)c(F)ccc(F)c1F N1(C(C2C(C=C)C2)=O)CCC(F)(C(N2CCN(C(=O)CC)CC2)=O)C1 c1(C(=O)OC)[nH]c(=NC2CC23CC(NC(=O)C(C2CCCO2)C2CC2)C3)sc1C c1(C(=O)NCC2CCCCN(C(=O)Cc3cnns3)C2)cccn2cncc12 C1(C2CCN(C(c3cnc(S)n3C)=O)C2)(NC(CC=CCC)=O)CC1 C(=O)(CC(C(F)(F)F)C1CCCO1)NC1(CO)CN(C(C(C(C)C)O)=O)C1 N1(c2nc(OC)c(Cl)cn2)CCC2(CC1)CC(C(N1CC(O)C1)=O)CO2 C(=O)(C1=CC2CCCCCC12)NC(C(c1ccc(OC)cc1)OC)C C1(OC)CC(c2nc(-c3cc(C(=O)N(C)C)c[nH]3)no2)N(C(c2cccs2)=O)C1 C1(NC(c2ccccc2O)=O)CCC(C(=O)NC2CCN(C3CC3)C2=O)CC1 Cc1csc2c(N(C(CNC(c3cnco3)=O)Cc3ccccc3)C)ncnc12 C1(NC(COCCCC(C)C)=O)CN(C(C2CC(S(C)(=O)=O)C2)=O)CCC1C C1(C(C(=O)NCC(CC)NC(=O)C(C)=C2CC2)NC(C)=O)CCCCC1 C1(C(N2C(CNC(C=CC=CCC)=O)CCC2)=O)CCC(CCC)CC1 CC(C)(C(=O)NCC1(F)CC(NC(c2ccnn2C(C)(C)C)=O)C1)n1cccn1 N1(C(c2c(C(C)C)n(-c3ccccn3)nc2)=O)CCC(N)c2ccccc21 Nc1ccc([N+](=O)[O-])c(C(N2CCCC(NC(=O)C#CC3CCCOC3)C2)=O)c1 C1(C(N2CCC(OCCNC(C(=O)NC3CC3)=O)C2)=O)CNC(=O)CC1OC c1(C(=O)NCCCCC(C)NC(C2C(CC(C)C)C2)=O)cc2c[nH]cnc-2n1 C1(NC(c2ccc(SC)o2)=O)CC2CC(C1)N(C(=O)CC1NC(=O)NC1=O)C2 c1(Cn2c(-c3ccncc3)nc(CC(CC)C)n2)cc(C)ccc1Br C(C(C)(C)C(C)(C)C)NC(C1CN(C(=O)OCC)C1)=O.C1CC(=O)N1 c1(C(C(=O)NCc2cccc(N3CC=CC3)c2)=O)cc2ccccc2s1 c1(C(N(CCCNC(C2C(CCOC)C2)=O)C2CC2)=O)occc(=O)c1OC c1(CCNC(C(=O)NC(C(C)C)CCO)=O)cccc(Br)c1C C=C(Cl)C(C)(C)C(=O)NCC1CCN(C(=O)COc2cccc(C)c2F)C(C)C1 C1(NC(C2C(C(C)(C)C)C2)=O)CCC(NC(c2cncc(C(F)(F)F)c2)=O)CC1 C(C(COC)C(=O)NCCN(C(=O)CC1CCCOCC1)C)OC c1(-c2[nH]cc(NC(CCCC=C)C3CC3)c2)ccc(C(=O)O)c(OC)c1 C1(CN(C(=O)Cn2cnnn2)C)CCCCN1C(=O)Cc1cnns1 N1(C(CC2CN(C(COC(CC)(C)C)=O)CC2F)=O)CC(C)=CC(C)C1.C(C)(=O)O c1(NC(=O)CCCOC2CNC(c3ccccc3)C2)cccc2ccccc12 CCC(CN(C)C)CC(=O)NC1CCC(C)(NC(=O)CS(=O)(=O)CC)CC1 C1(N(C(c2nc(OCC)oc2)=O)C)CCC(NC(=O)CCC(=O)N(C)C)CC1 CCC(CC)CC(F)C(=O)OC1CC(N2CCNC2=O)C1 c1(C(=O)NCC(CO)NC(c2ccc(OC(F)(F)F)nc2)=O)c[nH]cc(F)c1=O C1(C(=O)NCC(C)OCC)CC=CCC1NC(=O)COc1ccn(C)n1 C(C)(C(=O)NCCC1(C(N2CCC(C(N)=O)C2)=O)CC1)(C(C)C)OC c1(C(=O)NC(c2ccsc2)C)ccc2c(c1)CCN(Cc1cc(Cl)ccc1Cl)C2 C(=O)(C(C)CC)N(C(CC)CO)Cc1sccc1C CCCC(C(=O)N(C)CC1CCN(C(=O)C(C)NS(=O)(=O)CC)C1)OC C(=O)(C(O)(C(F)(F)F)c1ccccc1)N1CC(CNC(c2c(CC)c[nH]n2)=O)C1 c1(OCC)cc(Cl)ccc1C(N1C2CCC1(CNC(C1CCC1(C)C)=O)CC2)=O c1(OC)nscc1C(N1CCCC1CC(=O)NC1CC1C(F)(F)F)=O N1(C(CCCOC)=O)CC(CO)C2(CCN(C(c3csc(C(F)F)n3)=O)CC2)C1 N1(C(CCN(CCCCC)C)=O)CCC(F)(CNC(=O)C#CC(C)(C)O)CC1 C1(C(=O)NC2CC(CC(N)=O)C2)(NC(C(=Cc2cn[nH]c2)C)=O)CCCC1C c1(CNC(c2n(CC=C)nnn2)C2(C)COC2)cnn(CC(C)C)c1C1CCC1 C(=O)(C(C)(C)S(C)(=O)=O)NC1CCN(C(C2(CC#C)CC2)=O)CC1F Cc1csc(=O)n1CCC(N1CCCCC1C1CCCN(CC(O)CCO)C1)=O C(=O)(C1=NOC2COCC12)N(CCC(=O)NC1C(COC)CCC1)C N1(C(CC)=O)CCc2[nH]nc(C(=O)NCCSc3cc(Cl)cc(Cl)c3)c2C1 C1(C)(C(=O)NCC(CC=C)NC(c2cc(C(C)=O)cs2)=O)CCCNC1=O CCS(=O)(=O)CC(=O)N1CCC(C)(CNC(=O)C(c2ccccn2)C)C1 CCC(CC)C(F)C(=O)N1CCC2(CC2C(=O)NC(C)(C)CN(C)C)C1 N1(C(C(C)OCCCC)=O)CCC(CNC(c2cn(CC3CC3)nn2)=O)CC1 c1(C(=O)OC)n[nH]cc1C(=O)NC(CNC(=O)CC1CC2CC2C1)C(C)C N1(C(C(C)N(C(C)=O)C2CC2)=O)CC=C(C(=O)NCC(C)CC2CCCC2)CC1 c1(C(N2CCCC(NC(=O)Cc3ccns3)C(F)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 c1(NC(C2(F)CCC2)=O)ccc(C2CCN(Cc3ccnnc3)CC2)cc1 N1(C(C(CSC)O)=O)CC(NC(=O)C(C)NC(C)=O)C2(CC2)C1 CC1CC(CNC(C2CCN(C)CC2)=O)CN(C(=O)C(C)N2CCCC2)C1 c1(NC(N(C(c2c(C)cccc2)C)C)=O)ccc(Cl)cc1C(F)(F)F c1(NC2CC(C)C(C)(C)CC2)ccc(S(=O)(=O)N(C2CCCCC2)C)cn1 CC1(C(N2CCCC2CNC(=O)C(F)(F)c2csc(Cl)c2)=O)CCNC1=O CCCC(C)(C)CC(=O)NCC1CN(C)CCN1C(C1CCC2(CCC2)OC1)=O c1(CNC(C(COCC)C)=O)cccc(NC(c2ccc(C3CC3)cn2)=O)c1 N1(C(C2CCCN2C(=O)CCn2cccc2)=O)CCCC(OC(F)F)C1 c1(C(=O)NCC2CCCC(NC(=O)CSC(F)F)C2)ccc2nc[nH]c2c1 C1(NC(c2c(C(C)(C)C)c[nH]c2)=O)COCC1CNC(=O)CCc1ccccn1 C1(C(=O)NC(CC#C)C(=O)NC2(C)CC2)CC(C)(C)CN1C S(=O)(=O)(c1ccc(-c2cccc(C)n2)s1)N(CC=C)C c1(C(=O)NCC(=O)NC(N2CC(F)(CCNC3CC3F)C2)=O)cccnc1 c1(CC(=O)NO)ccc(S(=O)(=O)N2CCN(C(C3CCCCCN3)=O)CC2)cc1 C(=O)(C1CCc2cccc(O)c21)N1CC(CNC(C=CCOC)=O)C(F)(F)CC1 CCCC(C)C(c1nnnn1CC)NCCCc1noc(C(C)(C)C)n1 C(=O)(C#CC1CCCCC1)N1CC(CC)N(C(C2CCC(=C(F)F)CC2)=O)CC1 N1(C(c2cc3[nH]c(=N)oc3cc2)=O)CCC2(CCC(NC(=O)CC3CSC3)C2)C1 CCC1=C(C(=O)N2CCN(C(=O)C(F)C3CCC3)CC2CC(F)F)CCCO1 C(CN=c1[nH]nc(C(N)=O)s1)=CCNC(C1=C(C)CCC1)=O c1(CC)ccc(C(=O)NC(C)(CNC(=O)C(F)(F)CNC(C)=O)C(C)C)c(C)n1 CCC(C)(C)CCCC(=O)NCC1CCN(C(=O)Cc2cc(Cl)n(C)n2)CC1C CC(C)CC(O)C(=O)N1CC(c2n[nH]c(CNC(=O)C(C)CN(C)C)n2)C(C)C1 c1(C(=O)NCCCCN(C(=O)C=CC(F)(F)F)C)ccc(C(C)(C)C)cc1N Cc1cccc(Br)c1C(=O)NC(CNC(=O)C(C)(C)n1cnnn1)C(C)C C1(CNC(c2cn(CCC)nc2)=O)CC2(CC2)CN1C(=O)CCC(=O)c1cccs1 C1(NC(C2(CC=C)CC2)=O)CN(C(=O)CCC#CC)C(C)(COC)C1 Cc1c(C(N2CC(C3CN(C(c4ccns4)=O)C3)C2)=O)cnc2ncnn12 c1(C(C2CC2)OCC(=O)NC2(CNC(CC=C(C)C)=O)CCOC2)ccc(Cl)cc1 CCC(C)C(CS(C)(=O)=O)N1CCC(C(=O)OCCOC(C)(C)C)C(C)CC1 C12(NC(C(CNC(C=C(CCC)CCC)=O)C)=O)CC3CC(CC1C3)C2 N1(C(C(C(=O)OC)OC)=O)CCCCC(N(C(=O)C(C)c2cccs2)C)C1 C(CCN=C(NCc1ccc(F)c(F)c1)N1CCC(C)(C#N)CC1)SC c1(OC(CC(=O)Nc2nccc(CC)c2)C)ccc(Cl)cc1C C1(C(=O)NCCCOCCNC(C2(C3CC3)CC2)=O)CC2(CC2)C1 C1(C(=O)NC2(CO)CN(c3ncnc(Cl)c3F)C2)C2Cc3ccccc3C12 c1(C(=O)NCCC(C)(C)C(=O)NCCO)cncc2[nH]ccc12 C(C(C)(CO)CO)N(C(=O)CC1COCCN1C(=O)CSC(C)(C)C)C C(CCCCC(=O)N1CC(CO)CC1CO)NC(=O)C(F)C1CCCC1 CC(C)CC(C)(CNCC1CCCCC1)NC(=O)CCC1CCCCC1 Cc1cc(N)c(C(=O)NCCNC(C2CC2Br)=O)c(F)c1 C1(NC(C=C)=O)CC2CCCC(C1)N2C(=O)C(C)Cc1cnc[nH]1 C(=O)(C1=NN(CC(C)C)C(=O)CC1)NC(C1CCCN1C(=O)CCCN=[N+]=[N-])C C1(NC(C(C2CCCOC2)OC)=O)CC2CC(C1)N(C(C1CCCN1C=O)=O)C2 N1(C(C2(CC#C)CCN(C(=O)C=CC3CCC3)C2)=O)CCOCC(C)(O)C1 c1(C(=O)NCC2(CC(=O)NCC(CC)O)CC2)cncc(NC)c1 C1(C)(CNC(Cc2n(C)cnn2)=O)CCN(C(C2(C)CCCCO2)=O)CC1 Cc1cccc(C(C)NC(=O)C(O)CNC(C2(Cl)CC2)=O)n1 C1(c2n(CC(=C)C)nnn2)(NCc2cc(OC)ns2)CCOC(C(C)C)C1 CON1CC(C(N2CC(C)(C(=O)NC3(CCO)CCCC3)C2)=O)CC1=O N(C(=NCCC1CCCC1(F)F)NCc1cccs1)CC1C(CF)CCCC1 c1(CN(C(=O)C(C)(C)CO)C)ccc(CNC(c2cccnc2N(C)C)=O)cc1 N1(C(C(CC)COC)=O)CC(NC(C23CC4CC2C3C4)=O)C2CCCCC12 C(C)(C(C)CCC)NC(=O)NCCCC#CC.C1CC1 c1(C(N(C(C)CNC(c2cccnc2)=O)CC)=O)cnc(N(C)C)o1 c1(C2(C)CC2OC(=O)C=C2CCCCC2)cccc(F)c1 N1(C(C(CC2CN(C(C3OCCC(C)C3)=O)C2)F)=O)CCC2(CCC2)CC1 C1(C(=O)NCC(CN(C(Cc2nc(C)sc2C)=O)C)C)CCc2c(n[nH]c2C)C1 c1(SC)ccc(C(=O)NCC(C)NC(c2c(C(N)=O)ccs2)=O)o1 C1(CC(N2CCCC(CN(C(=O)COC(F)(F)F)C)C2)=O)(OCC)CCOCC1 C(=O)(C1(C)CCc2ccccc21)N1C(CNC(CN(C(C)=O)C)=O)C(C)(C)CCC1 N1(C(C2CC(CC)OCC2)=O)CCCC(O)(CNC(c2nc(C)oc2C)=O)CC1 N1(C(c2sc(C)c(C)c2)=O)CCC(CNC(=O)Cc2cnsc2)C(O)C1 c1(-c2ccc(OC)nc2F)c[nH]c2ccc(C(=O)NCc3cccc(Cl)n3)cc12 C1(C(N(CCC(C)NC(c2cnc(-c3cccs3)o2)=O)C)=O)CCCC1C c1(CN2CC3C(C(=O)Nc4ccc(F)cc4O)(C3)C2)ccncc1[N+](=O)[O-] Cn1cc2c(n1)CC(C(=O)NC1COCCN(C(c3coc(C4CC4)n3)=O)C1)CC2 CCC(CCC(=O)Nc1ccccc1OC)NC(c1cnc(C)n1C)=O c1(OC)ccc(-c2ncsc2C(=O)Nc2ccc(OC(F)(F)F)nc2)c(Br)c1 C(=O)(C(O)(C(F)(F)F)c1cn[nH]c1)NCCC(CNC(c1c(C)n(C)nn1)=O)O N1(C(C(C)C)=O)CC2(NC(=O)C(c3cccn3C)=O)CC1C2 C(=O)(C1CCCn2ncnc21)N1CC(C(C)NC(C2CC3(C2)CC(F)C3)=O)C1 C1(CNC(=O)Cc2cncnc2)CC2(CCN(C(c3cnccc3Cl)=O)C2)CO1 c1(C(=O)NCCCN(C(c2ncoc2C2CC2)=O)CC)cnn2c1OCC(O)C2 c1(C(=O)NC(C(C)(C)C)CNC(c2ccc(Br)o2)=O)n[nH]c2c1CS(=O)(=O)CC2 C1(CNC(C2C=C(C)CS2)=O)COCCN(C(=O)C=CC(=O)N(C)C)C1 N1(C(C)C)CC(C(=O)Nc2cccc[n+]2[O-])CCC1=O.C12C=CCN(C1)C2=O N(C1CCOc2c(Br)cccc21)C(=O)Nc1cc(NC(=O)NCC)c(C=O)cc1 N1(C(CC2CC(=O)N2)=O)CCc2cc(NC(C3CC(O)C3)=O)ccc21 O(P(=O)(COC(c1cnc(C2CC2)nc1N)=O)OCC)CC c1(CC)oc(C(=O)OCC2C3CC=CCC23)cc1C C1(CC=C)(NC(c2ccc(CF)cc2)=O)CCN(C(C2C=CCCC2)=O)C1 c1(C(N(CC(C)NC(=O)C(C)(C)O)C)=O)ccc2c(c1)S(=O)(=O)NC=N2 CC(C)(C)C(O)C(=O)NC1CC1CN1C2(CCCCC2)C1=O.C(N)(=O)NC1CC1 N1(C(CCC)=O)CCCC(N(C(=O)C=CC2CCOC2)Cc2cc(C)nn2C)C1 C(=O)(C#CC1(C)CC1)NC1CCC(CNC(Cc2c(OCC)nccc2)=O)CC1 c1(C(=O)NCC(CCCC)NC(=O)C(O)CCSC)cc(N)ccc1SC Cn1ccc(=O)c(C(N2CC(OCCC(=O)N(C3CC3)Cc3ccoc3)C2)=O)c1 c1(CCC(=O)NC2CCCCC2c2nc(S)n[nH]2)ccc(Cl)nc1 C1(CNC(C(CC)OC)=O)Cc2ccccc2CN1C(=O)COC1CCCOC1 c1(CC)cc(C(=O)NC2CCCC(NC(C3(CSC)CCC3)=O)C2)oc1C N1(C(c2c(C)cns2)=O)CCC(CNC(=O)C(C)C(C)C)C12CCC2 C=CC(C(=O)NC(C)CC(C)C)c1ccccc1.C12CN(C1)C(=O)CCOC2=O c1(CC)conc1C(=O)NC(CC1CCCC1)C(=O)NC(CC1CCCC1)CO C=CCCC(C)(C)CNC(=O)CC=CC1CCCN1C(=O)Cc1cc[nH]n1 N1(C(C2(C=C)CC2)=O)C2CCC1C1CC1(NC(c1cc(C)cc(C)n1)=O)C2 C1(CCC(=O)NCCc2c(C)nccc2)CCCCN(C(=O)C(O)CC2CC2)C1 C1(C)(C(=O)NC2CC(C)(NC(c3n(CC)ccc3)=O)C2)CCCCC1(F)F C1(C(N2C(C#C)CCC2)=O)CN(C(c2ccccc2CC=C)=O)CCC1(C)C N1(C(CSCC)=O)CC2CCOC2(CNC(c2cn(C)nc2-c2ccoc2)=O)C1 C(=O)(C(C)(C)Cc1cnn[nH]1)NCC1(OC)CN(C(c2ccc(CO)o2)=O)C1 C1(CNC(Cn2c(C)cc(C(F)F)n2)=O)CC12CCN(C(=O)CCC1CC1)CC2 Cc1ccoc1C(=O)N(CC(=O)NCC(C)(C)C1CCCO1)C C1(C(CC)(C)C)CCC(CCl)CC1.C(=O)(NO)N c1(OC)ccc(C(F)(F)C(=O)NC(C2CCCN2C(C2(O)CCCC2)=O)C)cn1 C(=O)(C(O)C(F)(F)F)N(CC(CNC(c1n[nH]c(C)c1Br)=O)C)C C(CSC1CC1)(C(C)C)NC(=O)NC(CC)C N1(C(=O)Cc2ccc(Cl)nc2)CCN(C(C23CCCC2CC3)=O)CC12CC2 c1(N(C(=O)C(=O)N2CCCC2)C)ccnn1CC1CCCNC1 CC(CC(=O)N(C(CNC(=O)Cc1ncc(Cl)s1)C1CC1)C)C(C)(C)C N1(C(CCC=C=C)=O)CCCCCC(NC(=O)Cc2nnc3n2CCOC3)C1 c1(C(=O)NCCC(CC2(OC)CCCC2)=O)ccnc(C(=O)OC(C)C)c1.C1CCC1 C(=O)(C#CC1CCOC1)N1CC(CCCCNC(C2CC3(CCCC3)C2)=O)C1 C(CCCCCNC(=O)C(CO)C1CN(C(=O)OC)C1)NC(c1c(C)nco1)=O C1(CC)CN(C(=O)C2CC2)CCC1NC(c1ccc(=O)n(-c2ccccc2)c1)=O c1(C(N2CCC(NC(c3c(OC)cccc3)=O)C2)=O)cc2cccnc2s1 N1(C(C(C)=O)=O)CCN(C2CCN(C(=O)CC(C)C3CCCO3)C2)CC1 c1(C(N2CC(NC(C=C)=O)C(C)C2)=O)nc(Cl)ccc1F CC1(C)CC(NC(=O)C(c2cnn(C(C)(C)C)c2)=O)CN1C(C12COCC(C1)C2)=O N1(C(c2cn(CCOC)nc2)=O)CCN(CC2C=CCC2)C(C)C1 N1(C(C(COC)N(C)C)=O)CCOCC(CNC(=O)CCc2cc(C)on2)C1 C1(NC(c2ccc(CC)s2)=O)CCN(C(c2ccc(N)cc2C)=O)C(C)C1 N1(C(CC=C)=O)CCC(CN(C(c2cc(C3CCC3)[nH]n2)=O)CC)C1 C1(CC)CCC(NC(=O)C(CCNC(=O)CCCN(C)C(C)=O)OC)CC1 C12(C(=O)NCCOCCCNC(c3c(C)[nH]cc3)=O)CC1COC2(C)C C(C)(C)(C(=O)N1CC(CCO)(NC(=O)C(C)CN(C)C)C1)OC N1(C(CSC(C)(C)C)=O)CCN(C(=O)Cn2cc(CO)nn2)C(CC(F)F)C1 c1(C(N2CC(C(C(=O)O)O)C2)=O)c(Cl)cnn1C.c1(COC)cn(C)nn1 CN(Cc1ccc(C#N)cc1)N1CCOC(Cn2cccn2)C1 c1(CCC=C)ccc(C(=O)NCC(C)(O)CN(C(=O)C(C)O)CC)cc1 N1(C(C2(CC)COC2)=O)CCC(CCNC(=O)Cc2csc(Br)n2)C1 C1(OC)CC(O)C12CCN(Cc1cc(Br)cc(N)c1O)CC2 N1(C(C(C)OCCOCC)=O)CCOCCC1CC.N12CCC(C1)CCC2=O C1(N(C(c2cc(CNC(C(CCC)C)=O)no2)=O)C)CNC(=O)C12CC2 C1(C(=O)OC)(CNC(C2CC(N(C(C(CC)OC)=O)C)C2)=O)CC2(CC2)C1 C(=O)(CC1=CCN(C(c2cnc(O)o2)=O)CC1)NC1(c2nc(C)[nH]n2)CC1 c1(OC)cc(CCNCC(Cc2ccccc2[N+](=O)[O-])CO)ccc1S(C)(=O)=O CC(C)(C(=O)NCC(C)(C)C#CC(=O)NC1CCC(CO)C1)C(F)(F)F c1(C(N2CC(C(C)(C)O)(CNC(CCc3nc(C)sc3)=O)C2)=O)nc(=O)n(C)[nH]1 C1(OC)CNCCC1C(=O)NCc1cnc(N2CCNCC2)s1 C(=O)(C1=CC2CCC(C1)C2)NC(C(=O)N(CCC#C)CCO)CC(=C)C c1(NC(C23CCC(OC)C2C3)=O)cccn2cncc12.N12CCCCC1C2=O CN1CCN(c2ncc(NC(C3CCCCC3)=O)cn2)C(C(F)(F)F)C1 c1(C(N(CCNC(CN2C(C)CCC2C)=O)C)=O)cc(Cl)c(F)cc1F C1(N(C(=O)NC(c2nc(Cl)sc2Cl)C)C)CCC(C(F)(F)F)CC1 c1(C(N2CCC(NC(C(C(C)C)C)=O)C2C)=O)n[nH]c2c1CS(=O)(=O)CC2 C(=O)(C1CCc2ccc(Cl)nc21)NC1(CO)CN(C(c2c(C(N)=O)nccn2)=O)C1 c1(SCC(N2CCC(CNC(c3cscn3)=O)CC2)=O)ccc2c(c1)CCC2 C(=O)(CCCCCC(C)C)NC(CNC(COc1c(C)ccc(Cl)c1)=O)C C1(C)(CNC(c2nc(CCC)oc2)=O)CCCN1C(=O)C(CO)NC(=O)C(C)C N1(C(CCCCC)=O)CCOC(C)(CNC(C23CSC(C2)C3)=O)C1 Cc1cc(C(=O)N(CC(C)NC(C2(Nc3ccccc3)CC2)=O)C)c(Cl)cc1N c1(C(=O)NC2(CO)CCN(C(C3N(CC)CC3)=O)C2)cc(=O)c(Br)c[nH]1 C=C(C)CC(C)C(=O)NCC1CCCCN1C(=O)CCn1nc(C)nc1C C1(N(C(C(C2CCCC2)NC(C)=O)=O)C)CC2CCC(C1)N2C(=O)CC1CC1 C(=O)(C(O)CCC(C)C)N1CC2(N(C(CCCOC)=O)CC2)C1 c1(OC)ccc(C=CC(=O)N(CC(C)(C)CNC(=O)C(C)CS(C)=O)C)nc1 c1(CN2C(C)(C(=O)NCCSC)CCC2)cc2cc(F)ccc2s1 C1(OCC)COC2(C1)CN(C(C1(C3C(NC(C=C(CCC)C)=O)CCO3)CC1)=O)C2 C(=O)(CC(C)C(F)(F)F)NCC1N(C(Cc2c(C)cccn2)=O)CCOC1 C(=O)(CCCCC(=O)NCc1ccsc1C(N1CCCC12CCC2)=O)OC.C(=O)OC C1(C)(CCNC(C(C=C)OC)=O)CCN(C(=O)Cc2ccsc2)C1 CC1OCCN(C(=O)CSCC(F)F)C1C(N1CCCN(CC2CC2)CC1)=O N1(c2cc(OCC)ncn2)CCCC12CCN(C(C1(c3ccccc3)CC1)=O)C2 C1(C(N(C2CCN(C(CC(=C)C)=O)CC2)CC(C)C)=O)CCn2c(O)nnc2C1 N1(C(c2c(C)cc(SC)s2)=O)CCC2CCN(C(c3cnc(O)s3)=O)C2C1 c1(C(N(C2CCCN(C(=O)CCS(=O)(=O)NC)C2)CC)=O)csc2nccn12 C=CC1(CC(=O)NCc2cc(Cl)cs2)CN(C(c2cccnc2OC)=O)C1 c1(C(N2CCN(CCCNC(C3CNC(=O)C3)=O)CC2)=O)cc2c[nH]nc2s1 C(C(F)(F)C(F)(F)F)n1c(C)nc(-c2cccs2)n1 c1(C(=O)OCC)nn(C)cc1C(C(=O)NC1CCCSC1C)N(CCCSC)C N1(C(c2c(C(C)C)occ2)=O)CCC(C(=O)NC(C)CN2CCOCC2)=C(F)C1 c1(C(CC)C)ccccc1N1CCCS1(=O)=O.C1(=O)C(C)O1 N1(C(c2cc(COC)on2)=O)CCN(C(c2csc3cncn23)=O)C(C(C)C)C1 c1(NC(C2(C)CCN(CCCCCC)C2)=O)ccc(OC)cc1C c1(C(=O)NC(C2CCN(C(C3CCS3(=O)=O)=O)C2)C)ccc2oc(=N)[nH]c2c1 C1(NC(C2C(C(C)(F)F)C2)=O)CC(CO)N(C(=O)C=Cc2ccc(Br)o2)C1 CC(C)CC(C(=O)NCCCC(N1CC(=O)NCC1C)=O)C(C)C c1(OC)c(C(N2CCC(CNC(=O)CC3CCCCC3)C2)=O)oc2ccccc12 N1(C(c2c(COC)noc2)=O)CC2CCCC2(NC(c2ccnc(C)c2)=O)C1 c1(C(=O)NC2(COC)CCN(C(CSCC=C)=O)C2)cc(Cl)c(F)c(Cl)c1 C(CC(C)(C)C)(C(=O)N1CCCC(C)(C(N2CCC(CO)C2)=O)C1)OC N1(C(C2CCC(NC(C)=O)CC2)=O)CCCCC(NC(=O)CC(C)(C)CC)C1 c1(C(N(C(C)CNC(C2CC3(CCC3)C2)=O)C)=O)cc2c(ncn2C)s1 C(C)(CCC(=O)N1CCN(CC(N2CCC(C)(c3ccccc3)C2)=O)CC1)OC c1(C(C)NC(C(=O)NC2CC(C)C(=O)CC2)=O)ccc2c(c1)CCN2C c1(C(=O)NCC(CNC(c2c(C)nc(C)n2O)=O)CO)cccc(C=C(F)F)c1 Cn1ncc2c(C(=O)NCC3(O)CC(NC(=O)Cc4cnoc4)C3)ncnc12 N1(C(CC(C=C)CC)=O)CC(C)(C)CCC1CNC(=O)C(Cc1ccccc1)=NO C1(OC)CCN(C(=O)C(C)N(C(=O)C(O)C2CC2)C)C1C(C)C Cn1cc(CN2CCN(c3ncc[nH]3)CC2)c(=O)c2cnn(C)c12 Cc1ccc(C(N2CCN(C(C3CC3F)=O)CC2c2cccnc2)=O)c(=O)n1C C1(CC=C)(NC(C2CC2C2CC2)=O)CC2CCC(C1)N2C(C1(C(C)C)COC1)=O CC(C)CS(=O)(=O)CC(=O)NC1CCCN(C(C2CCN2S(C)(=O)=O)=O)CC1 N1(C(=O)CC2CCCCC2O)CC2CC(C1)N(C(c1cnc3[nH]ncc3c1)=O)C2 C1(C(=O)NCC2(C(N)=O)CN(C(C(F)OC)=O)C2)CCN(CC(F)(F)F)C(=O)C1 c1(OCCCC)ccc(CC(=O)NCC(F)CNC(C2(C)CCNC2=O)=O)cc1 c1(C(=O)NCC2(CN(C(=O)COC3CCOC3)C)CC2)ccc2occc2c1 N1(C(=O)OC(C)(C)C)CCCC(O)(C(F)(F)C(=O)NCC(C2CC2)SC2CC2)C1 c1(C2CC(F)(F)C2)cccc2nncn12.N1(C2(C(=O)NC)CC2)CCCOC1=O C1(CC(=O)NC2CCC(NC(C3(CCOC)CC3)=O)C2)CCC2(CC1)OCCO2 c1(CC2N(C(CN3CCC(OC)C3)=O)CCC2)ccccc1[N+](=O)[O-] N1(CC(C)S(C)=O)C(=O)CN(C2CC2(c2ccccc2)C(F)(F)F)C1=O c1(C(=O)NC(CN(C(C(CC)c2cccnc2)=O)C)C)noc(C)c1C(=O)OC CC1=C(C(=O)NC2CCC(CC(=O)NCC3C=CCC3)CC2)CCCO1 C(=O)(C(F)CC(C)(C)C)N1CCC(C(=O)NC(CCC)C#N)C1 C=CCCCCC(=O)NC1COCC1C(=O)NC1CCC=CCCC1 c1(CCC(=O)NC(CC)(CNC(=O)C(O)CSC)CC)cnc2n1CCCC2 c12cc(nn1C)S2.N1(C(COC)=O)CC(=Cc2cccs2)CC1=O C12CC(CN(C(=O)OC(C)(C)C)C1)N2.C1(CCC)(CO)CCCN1C(C)=O C1(C(C)C)CC(CC(=O)NC2CCCC2NC(C2(Cl)CC2)=O)CCO1 C1(NC(CCC#C)=O)CC(CCC(=O)N(CCC)CCOCCN(C)C)C1(C)C C(=O)(C1CCc2cc(Cl)ccc21)NCC(CNC(C(CCCCC)O)=O)CO C(C1CCc2ncnn21)N1C(CNC(c2cn3c(n2)CCC3)=O)CCC1 C1(F)(C(N(CCN(C(C2CCCN2S(C)(=O)=O)=O)CC)CC)=O)CC=CCC1 c1(OC)ccc(CNC(=O)C(N2CCN(CC(=O)OC)CC2)C2CC2(C)C)cc1 c1(C(N2CCCC(C(=O)NCC3(CO)CC=CC3)(CC)C2)=O)cnn2cccc2c1 CC1=C(C(=O)N2CCC(NC(=O)CC(F)(F)Cl)C(CO)CC2)C(C)(C)CCC1 CC(CCCSCCC(=O)OC(C)(C)C)c1ccccc1 N1(C(c2n(C)c(S)nc2)=O)CC2(C1)CN(C(=O)CCCCO)C2 C1(NC(CN(C2CN(C(Cc3c(C)ccs3)=O)C2)C2CC2)=O)CCN(C)C1(C)C c1(C(N2C(C)CC(C(=O)NC(c3ccncc3)C)CC2)=O)ccc2cc[nH]c2c1 c1(OC)ccc(-c2noc(C3CC4(OC)CC3C4)n2)cc1Br C(C(C)C(C)C(=O)NC1CCC(CNC(C2(CF)COC2)=O)CC1)OC N1(C(CCN(CCCCC)CC)=O)CCC2(CCCC2NC(=O)C(O)CC)CC1 c1(C(C(=O)NCCC2CCN(C(C=CCC)=O)C2)C)ccc(O)c([N+](=O)[O-])c1 c1(CC)nc(C)cc(=NC2C3CN(C(=O)C(C)Cc4cccc(Br)c4)CC23)[nH]1 Cc1cnc(O)c(NC(c2n[nH]cc2CNC(C2CCC3(CC3)C2)=O)=O)c1 Cc1cc(F)cnc1C(N1CCC(C)C(CNC(C2CCS(=O)(=O)C2)=O)C1)=O C=CC(C)(C)C(=O)NCC1(O)CCN(C(C2CCC2(F)F)=O)C1 N1(C(C(CCCC)O)=O)C2CCC1C(F)C(NC(c1ccc(CC)cc1C)=O)C2 N1(C(CSCCN(C)C)=O)CCCC(C(=O)NCC(C)(C)NC(=O)C(C)(C)C)C1 C1(Cl)(C(=O)NCC(C)(C)CNC(C2CN(CC(F)(F)F)C2)=O)CC12CCOCC2 N1(C(c2c(C)oc(C(C)(C)C)c2)=O)C2CCC1CC(NC(c1n[nH]cc1Cl)=O)C2 C#CCC(C)C(=O)NCCc1ccc(NC(c2cscc2C)=O)cc1 Cc1ccc(-n2ncc(-c3nc(C4CCOC4)no3)c2C)cc1 N1(C(CC(C)OC)=O)CCN(C(=O)Cn2cnc(C#N)n2)CC1COC c1(C(N2CC(NC(CC(C)(F)F)=O)C3(C2)CC3)=O)cc(F)cc(N)c1F C1(NC(C(C=C=C)C)=O)CN(C(c2cnc[nH]2)=O)C2CCCC12 C(=O)(C(C)S(N)(=O)=O)N1CC(CCNC(=O)Cc2ccc(C)c(C)c2)(OC)C1 C1(NC(C(=Cc2cccnc2)C)=O)CC(O)CN(C(c2c[nH]nc2Br)=O)C1 c1(C(=O)NC2CC2CNC(c2cnc3[nH]ccnc2-3)=O)cc(F)cc2cc[nH]c12 c1(C(N2CC(O)CC(NC(C3CCSC3)=O)C2)=O)cccc([N+](=O)[O-])c1Br c1(OC)cc(C(=O)N(CC(C)NC(C2(C)CNC(=O)C2)=O)C)cc(Cl)c1 C(C(C)(CO)NC(=O)C(C)CC1CC1)NC(COCCCOC)=O C(=O)(C(O)C(F)(F)C(F)(F)F)NCC1OCCN(C(c2c(C#C)cnn2C)=O)C1 Cc1ccnc2c(C(=O)ON3CCN(C(=O)C(c4ccccc4)=O)C4CC34)cnn12 C12(C(N(CCN(C)C)CCc3cccnc3)=O)C(N(C)C)C3CC1C2C3 C12CCC3(CN(C3)C(=O)N3C(CCC3)CNC1=O)O2.C1(CC)(CC)CCCCC1 c1(C(N2CC3C(CC(=O)OC)(C3)C2)=O)cc(Cl)c(OC)cc1NC(C1CCC1)=O c1(N2CCC(O)C2)cc(=NCc2cccc(Br)c2)[nH]c(Cl)n1 c1(C(N2CCC(NC(c3c(CC)n(C)nn3)=O)CC2)=O)c(F)ccc(Br)c1C c1(NC(C2CC(C)(CC)N(C(=O)Cc3nc(C)cs3)C2)=O)cc(C#N)ccc1C C1(CC)CN(C(C2(COC)COC2)=O)CCN1C(=O)CCS(N)(=O)=O c1(C(=O)NC2CCCC2NC(C2CC(n3ccnn3)C2)=O)coc2c1COC2 C1(F)(CNC(C2(C#C)CC2)=O)CCCN(C(=O)CCC(=O)Nc2nccs2)C1 CC1(C2CN(C(=O)C(c3ccccc3)NC(=O)C=CC(F)(F)F)CCO2)N=N1 Cc1cn2c(n1)C(C)CC(C(N1CCN(C(c3c[nH]nc3F)=O)CC1C)=O)C2 C1(NC(C(F)=C(C)C)=O)CC2(C1)CC(CNC(=O)Cc1c(C)noc1Cl)C2 C1(C(=O)NCc2c(C)noc2)CCC(C2CC2)N1C(=O)CC1CSCCO1 N1(C(c2c(CC)oc(C)c2)=O)CCCC(C)C1CNC(c1ccc(Cl)nc1)=O Cc1noc(C(C(C)C)NC(=O)COC2CN(C(C3CC4(CC4)C3)=O)C2)n1 C(=O)(C1COc2ccc(F)cc21)N1CC(O)(CNC(C2(C)C=CCCC2)=O)C1 c1(CC(C)C)n[nH]c(=NCCCC(C)NC(C2CCc3ncncc3C2)=O)s1 c1(C(C)NC(=O)C(CC2CCCC2)NC(=O)C=CC(C)(C)C)ccc(F)nc1 N1(C(COCCOCC#C)=O)CC(C)(C(=O)N(C2CCOCC2)C2CC2)CC1(C)C CC(C)CC(F)C(=O)NC1CC(CNC(c2cn(Cc3cccs3)nn2)=O)C1 C12(NC(CC3C(C)CCCC3)=O)CCCC1N(C(c1ccc(O)c(N)c1)=O)CC2 CC(C)CC(C(=O)NC(C)(C)CC1CCOC1)ONC(C1(C)CC=CCC1)=O N1(C(CCN(C)CC)=O)CC(NC(c2ccc(N3CCCC3=O)cc2)=O)CC1C C(=O)(C(C(=O)N1CCC(C(=O)N(C)CC2CCCC2(C)C)(CF)C1)OC)OCC N1(C(c2cn(CC(=O)O)nn2)C)CCOC(C)(CC(F)(F)F)C1 c1(C(=O)NCCNC(c2n[nH]cc2Cl)=O)ccc(SCC2C=CCC2)cc1 C1(OC)CN(C(=O)Cc2cn[nH]c2)CC1NC(c1c(C2CC2)cnn1C)=O Cc1cccc(C(=O)NCCC(=O)NCCC(C)c2cn[nH]c2)c1 N1(C(c2ccn(C)n2)=O)CC=C(C(=O)NC2CC(O)C2(C)C)C1 C(=O)(CCS(N)(=O)=O)NCCN(C(=O)C=CSC)CC N1(C(C(C(C)C)SCC)=O)CC(CO)C2(C1)CN(C(c1nn(C)c(C)c1Cl)=O)C2 C#Cc1cncc(C(=O)NC2(COC)CN(C(c3n[nH]c(C)n3)=O)C2)c1 C1(CCNC(C(C)NC(COC)=O)=O)CCCCN1C(c1cc(C)c[nH]1)=O C(=O)(C(F)(F)C(C)(C)O)N1CC(C(=O)NC(C)C(C)(C)CO)CC(C)C1 Cc1cc(C(=O)NC2CC3CC(C2)N(C(C24CC(C)(C2)C4)=O)C3)ccc1C#N C1(Cn2cc(-c3c(C)ccc(C)c3)nn2)CC2COCC2N1C(C12CCC1C2)=O c1(C(C)C)nc(Cl)cc(=NC2CCC(N(C(=O)CC3CCCC(=O)N3)C)CC2)[nH]1 C1(COc2cccc(NC(C(CC#C)NC(=O)CCC)=O)c2)CC2(CCCO2)C1 N1(C(c2cccc(SC)c2)=O)CC2CCC(C1)N2Cc1ccnc(F)c1 Cc1cc(C#N)ccc1C(N1CC(C)(CNC(=O)CCCCN(C)C)C1)=O CC(C)(F)C(C)(F)C(=O)N1CC(NC(=O)CC23CC(C2)C3)CC(F)C1 c1(OC)ccccc1CCC(=O)NC1CN(C(=O)CCc2cn[nH]c2)CC1C N1(C(C2N(C(C)C)CCC2)=O)C(CC(=O)NCCCCC2CC2C)C2CCCC12 c1(CNC(C(N2C(C=C)COCC2)(C)C)=O)cc(OC)c(OC)cc1Br c1(C(=O)NCC(COC)NC(c2nnn(C)c2N)=O)cc2c(s1)CCCC2 N1(C(c2c(C)n(C)cc2)=O)CC2(CCC2)CC1C(N1CC2CCC=CC12)=O C[Si](C)(C)CCCC(=O)N1CCCC(CO)CC1 c1(C(=O)NC(C)CC(C)NC(c2scnc2Cl)=O)cncc(Cl)c1 c1(C(=O)NCC(CO)NC(CCC(CC)C)=O)sc2ncccc2c1N N1(C(C(=O)NC)Cc2ccc(OC)c(F)c2)CCC(P(C)(C)=O)C1.C1(=O)CCN1 C(N=c1[nH]c(Cl)ncc1F)c1cccc(CNC(C(C(C)C)F)=O)c1 C1(c2nc(CSC)[nH]n2)CCCN(C(C2(C)CC=CCC2)C(=O)NCCC2CC2)C1 c1(CCC(=O)NC2CN(C(=O)Cn3cc(CO)nn3)CC2F)ccc2c(c1)CCO2 C(=O)(CC(C)(C)CC(F)F)NC(C1(O)CCN(C(C2CC2CF)=O)CC1)C c1(C(=O)NCC#CCNC(C(C)c2ccco2)=O)sccc1Cl C1(C(C(=O)NCC(CC)(CC)NC(c2ccns2)=O)O)CCS(=O)(=O)CC1 C1(N(C(=O)COCC2CCCS2)CC2CCCC2)CCN(C(=O)CC)C1 C1(C(N2CCC(CNC(CC(C)(C)OC)=O)C23CC3)=O)CCCC(C)(F)CC1 Cc1ccc(CCCNC(=O)NCC2CCC2)s1 N1(C(C(C)C)=O)CCC2(CC1)CC(NC(C1CC1(C)C(C)C)=O)CCO2 C1(O)(C(=O)NCC(CC)NC(c2c[nH]c(C(F)(F)F)c2)=O)CCCC(C)CC1 c1(NC(CCn2cc(C(CC)N(C)C)nn2)=O)ccc(Br)c(O)n1 C(CC(C(=O)OC(C)(C)C)OC(C1(c2cccc(Cl)c2)CCC1)=O)SC C(=O)(C(F)CC(C)C)NCCN(C(c1ccc(C)nc1O)=O)CC N1(CCCCCC)C(=S)NC(c2cc(C)c(Br)s2)C2=C1CCN(C)C2=O C1(NC(N2CCN(C)C(c3cccs3)C2)=O)CCc2nc(N(C)C)sc2C1 CN1CCC(N(C)C(C2CC2(c2ccccc2Br)F)=O)C1=O c1(C(N2C3CN(C(C4C(C=C)C4)=O)CC2CC3)=O)cc2c(C(N)=O)nn(C)c2s1 Cc1cc(NC(c2cc(C)on2)c2nnnn2C)c(C)c(C)c1 c1(C(N(C(C)C(N2CCCC2C(O)CO)=O)CC)=O)ccnc2cc[nH]c12 NS(=O)(=O)c1cc(CNC(N2CCCCC2Cc2cc([N+](=O)[O-])c[nH]2)=O)co1 N1(C(CC(=C)C)=O)CCCC(CCNC(c2cnn(CC(C)C)c2CC)=O)CC1 c12cccc(c1)S(=O)(=O)NCCN2.c1(CN(C(C)=O)C)ccc(C)o1 c1(C(=O)NC2(C)CCN(C(=O)CC3(N4CCCC4)CC3)C2)cc(O)ccc1Cl C1(NC(COCC=C)=O)CCN(C(C2CCC(F)(F)CC2)=O)CC1CO Cc1ncc(C(N2CCC(F)(C(=O)NC3CC(O)CC3O)CC2)=O)c(C)n1 C(=O)(C1=NOC2COCC12)N1CCOCC(C)(CNC(c2cc(CC)[nH]n2)=O)C1 N1(C(C2CCC(CNC(C3(CO)CCOC3)=O)C2)=O)CC2(CCCC2)C1 C1(NC(CN(c2ncccn2)C)=O)CCCCN(C(=O)Cc2cccc(F)c2Cl)C1 CC1CCCCC1(CNC(=O)CC1CC2(CC2)CO1)NC(C12CC(F)(C1)C2)=O N1(C(C2(COCC)CCC2)=O)CCCC(CC(C)C)C1.C1(CC(=O)N)CC2CC2C1 C[Si](C)(C)C1(CNC(=O)CCOC2CC=CC2)CC1.C1(NC(=O)CO)CCCOC1 C1(CNC(C2N(C(C)=O)CCC2)=O)CCN(C(C2CC2C2CC2)=O)C12CCC2 c1(C(=O)NC23CC(CNC(c4nc(CCC)sc4)=O)(C2)C3)ccc2sncc2c1 c1(CC(=O)NCC2C(NC(C=COCC)=O)CCCC2)cc2ccccc2o1 c1(CCC(N2CC(OCCNC(CN(C3CC3)CC)=O)C2)=O)ncc(C)[nH]1 c1(COCC(CN2Cc3c(nn(C)c3N)C2)O)ncnc2c(F)cccc12 c1(C(N2C(CNC(C3CC3CF)=O)CCC2)=O)cccc(C2CCOC2)c1 c1(C(=O)NC2C(CC)CN(C(=O)C(F)=CC3CC3)CC2)cn(C)c2ccccc12 Cc1noc(C)c1C(C)CC(=O)NC(C)CNC(=O)CCNc1ccccn1 C1(C(=O)NCC2N(C(c3cc(C)sc3)=O)CCC2)CCCCCS1(=O)=O N1(C(c2c(C)cco2)=O)CCC2(NC(c3cccc(N(C)C)n3)=O)CCCC12 N1(C(c2cccc(C(=O)OC)n2)=O)CC(NC(=O)C(C)C2CC2)CC2(CC2)C1 N1(C(COC(c2c(C)c(C)cc(C)c2C)=O)=O)CCCC2(CC1)CNC(=O)O2 N1(C(c2c(C)cc(=N)[nH]c2)=O)CC(C)CN(C(=O)CC23COCC(C2)C3)C(C)C1 C1(C(=O)NC(C)(CNC(=O)CCC(F)F)C2CC2)CC2CCC1CC2 C(CCS(C)(=O)=O)NC(c1cc(CNC(Cc2cc(C)no2)=O)no1)=O Cc1oc(CO)cc1C(=O)O.C1C=CCNC(=O)N1.C1(N)CC1 C1(CNC(C(C)OCCC=C)=O)C(CC)CCN1C(c1ncn(C)n1)=O C(CCC)(C(=O)NC(CCC)C(=O)N(C(C)C1CC1)CC)=CCC.C(C)=O C=CC(CCC)CC(=O)N(CCCOCCN(C(=O)CC1CCCOC1)C)C C(CO)(C(F)(F)F)NC(C(CC1CCOCC1)NC(c1cc(=N)[nH][nH]1)=O)=O C1(N(C(c2c(CC)ocn2)=O)C)CCCN(C(=O)Cc2ccccc2O)CC1 C(=O)(CC(F)(F)C(F)F)NC(CC(C)NC(C=CCC)=O)C CCCC(C(=O)NCc1ccnc(C(=O)Nc2cccc(CC)c2)c1)C(C)C N(C1CCCn2c(C)nnc21)C(C(C(CC)CC)NCCCOc1ccccc1)=O c1(-c2c(C(=O)Nc3nccc(Br)c3Cl)nccc2)ccc2[nH]nc(O)c2c1 CC(CC(C)NC(=O)CCn1cnnn1)NC(=O)CC(=O)N(C)C Cc1[nH]c(=N)nc(O)c1CCC(N1CCC(NC(c2cc(Br)c[nH]2)=O)C12CC2)=O Cc1ncncc1C(N1CCN(CCN(C)C(C2(Cl)CC23CCC3)=O)CC1)=O c1(C(=O)NCCOCCCNC(C2(CC#C)CCCC2)=O)cc(C#N)n(C)n1 c1(C(=O)NCCC(C)N(C(CCSCCC)=O)C)ccc(N2CCCC2)cc1Cl c1(CC(=O)NCC(CNC(Cc2cn(CC)nn2)=O)(C)O)ccc(Cl)nc1F C(=O)(C(O)C1=CCCCC1)NCC1N(C(C(C=C)(F)F)=O)C2C(C1)C2 c1(COC)nc(C(=O)NCCc2ccccc2)n[nH]1.c12cnn(c1)C2 N1(C(C2(C#C)CCCC2)=O)CC2(C1)CN(C(=O)Cn1ncc(O)nc1=O)CCO2 N1(C(c2cn(CCC)nn2)=O)CC(CNC(c2cncn2C)=O)CCC1C N1(C(C2ON=C(CC)C2)=O)CCc2ccc(C(=O)N(CCC(C)(C)C)C)nc2C1 C(=O)(C1=CCCOCC1)N1C(C(C)NC(c2ccn(C(C)C)n2)=O)CCC1 C(C)(C(C)C(=O)N1CCN(C(C)C)CC1)NC(c1cnc(CC)s1)=O S(=O)(=O)(CCCN=c1[nH]c2c(c(=NCCS(=O)(=O)N(C)C)[nH]1)COC2)NC C1(C(=O)NCCNC(C(C)Oc2cccnc2)=O)CC(c2ccccn2)=NO1 c1(C(N(CC(C)NC(=O)CCn2cnnn2)C)=O)cc(F)cc2ccncc12 N1(C(c2ccc(OC)nc2C)=O)CCC2CN(C(=O)CC(C)O)CCC12 c1(C(N2C(C)CC(NC(c3c[nH]c(Br)c3)=O)CC2)=O)cnn2cccc(Cl)c12 c1(CN(C(CCN(C(c2nc(C)sc2)=O)C)=O)C)cccc(O)n1 C1(C(N(C)CC2CCN(C(=O)COc3ccon3)C2)=O)CN(C)C(=O)N1 N1(C(c2ccc(-c3ccc(Cl)s3)cn2)=O)C2CC3C4CC(C3C2O)C1C4O N1(CC2CC3(CC(OC)C3)C2)C2CCC1CC(CCOC(C)(C)C)C2 c1(N(CC(C2CC2)OC)C)cc(=NCCC(=O)OC)[nH]cn1 C(=O)(C1=CCCN(Cc2cc(F)c(C)c(F)c2)C1)Nc1c(Br)ccc(OC)n1 C1(C)(C(N(C(C=C)C)C)=O)C=CCN1C(c1cnc(C2CC2)o1)=O c1(OC)ccc(C)cc1NC(=O)C=CC(=O)N(C(C)Cc1nccn1C)C1CC1 CC1CCCN(C(=O)C(=O)NC2CC(NC(C3(C)CCCOC3)=O)C2)C1 CC(C#N)CN=c1nc2sccc2c(NCC2(C)CC2F)[nH]1 C(=O)(C#CC1(C)CCCO1)N1C(CC(=O)NC2C(N(C)C)CCC2)C2CCCC21 c1(CC(N2C(C3(O)CN(C(CCCCC)=O)C3)CCC2)=O)cccc(F)c1O C1(CNC(CCCc2c(C)ccs2)=O)(NC(C2CC2C2CC2)=O)CCOCC1 C1(CC)(CNC(C2(c3ccccc3)CC2(F)F)=O)CCC(=O)N1 c1(C(=O)OCC)ccc(CN(C)CCN(C)C(c2cc[nH]n2)=O)cc1C CC(C)CC(O)CC(=O)NCCC1C(C)CCCN1C(c1csc(C2CC2)n1)=O CCCC(O)CC(=O)N(C1CCN(C(=O)C(C)(C)COC)CC1)CCC c1(SC)cccc(C(=O)NC(CNC(=O)C2=CCC2C)CO)c1[N+](=O)[O-] C(C(C)(C)C(=O)NCC1C=CCN1C(c1ccccc1N)=O)OC N1(C(C)=O)CC(O)CC1C(=O)NCC=CCNC(c1nn(C)cc1Cl)=O c1(C(=O)NCC2(O)CN(C(=O)C=C(Cl)Cl)C2)coc2c1CS(=O)(=O)C2 c1(COCC(=O)N(CCCNC(c2cccc(OC(F)F)c2)=O)C)ccccc1C c1(C(=O)NCC2CC(OC)CN2C(c2ncccc2F)=O)ccc(C)cc1C C1(C2CC2)(n2cc(-c3cnc(O)nc3)nn2)CCN(C(C2CCN(C)CC2)=O)C1 N1(C(Cn2c(C)ncc2)=O)CCN2CCN(C(c3cc(C(F)F)no3)=O)CC2C1 N1(C(c2c(OC)scc2)=O)CCN(C(=O)CC(C)(C)c2cccs2)CCC1C C12(C(=O)NCC3C(NC(C(C)CC(F)F)=O)CC3)CC3CC(C1)CC(C)(C3)C2 C(=O)(C(C)C(C)(F)F)NC1(CNC(CN2CCC(C)CC2)=O)CC(F)(F)C1 c1(C(=O)NC2C(C)N(C(c3cnc(O)n3C)=O)CC2)cnc2nc(O)ccc2c1 c1(C(=O)NC2C(OC)CN(C(C3CC(SC)C3)=O)C2)cnc(O)c2cccnc12 CCCC(CC(C)C)C(=O)N(C1CCC(NC(=O)C(C)SC(C)C)CC1)C CN1CCC(CC(=O)NCC2(C(N3CC4C=CC4C3)=O)CC2)CC1 N1(C(CONC(C(CCC=C)CCC)=O)=O)CCC2(CCOC2)CC1 C12CC(N=C3NC(=NC(=N)N3)NC1)C2.C(CCCNc1cnn[nH]1)SC C1(O)(CCNC(COCCCCC)=O)CCN(C(=O)C(C)(F)CC)C1 C1(CC(=O)NC2CCC(F)C2)CC2(C1)CN(C(C1CC1c1ccccc1)=O)C2 C(CS(=O)(=O)CC(=O)NCC1(C(=O)NCCc2cccn2C)CC1)OC C(=O)(CCCCCCC(=O)O)NC1CC(N(C)CC)C12CCCC2 C(=O)(C(C)(C=C)CCOC)NCCC(C)NC(CC(C=C)(C)C)=O Cn1cc(CC(=O)OC2CCN(Cc3ccccc3)C2=O)c2cc(Br)ccc12 N12CC(C(O)C1)C2=O.c1(C(=O)NC2CCN(CCC)C2)nc(Cl)c(CC)[nH]1 C(=O)(CC(C(C)(C)C)NC(C1CC1Cl)=O)NCC(=O)N(C)C N1(C(C(C)Cc2cnc[nH]2)=O)CCC2C(CCN2C(=O)C(N)=O)C1 c1(C(=O)NCC(CC)NC(c2n[nH]cc2OC)=O)cc(CO)c(C)o1 C1(C(=O)NC(CNC(CN(C)CC)=O)(C)CC)CCc2nc(O)[nH]c2C1 CC1(C(F)F)CCCC1NC(=O)NCc1ccc(NS(C)(=O)=O)cc1 C1(NC(c2c(CNC(c3ccc(C#C)cc3)=O)c[nH]n2)=O)CCn2ncnc2C1 N1(C(c2[nH]cc(C(C)=O)c2)=O)CC2CCC(N(C)C(c3ncccc3C)=O)C2C1 c1(C(=O)OCCN(C(=O)COC(F)(F)C(F)(F)F)C)cccc(C)c1.C1(=O)CN1 C(=O)(CC1=C(C)NS(=O)(=O)N=C1C)N1CC(C)CC(NC(C(COCC)C)=O)C1 CCC(O)C(C)(C)C(=O)N1CCCCC1CN(C)C(c1ccc2sccc2c1)=O c1(CC)cccc(C(=O)NC2CC(NC(=O)C(F)CC3CC3)C2)n1 c1(N2CCC(C(C)NC3CC3)CC2)ccc(F)cc1.C12CCCCN1C2=O CCC(C)(F)C(=O)NC1CC(CNC(=O)COCc2cc(C)no2)C1 N1(C(C2(CCOCC)CCCC2)=O)CC(NC(=O)CCC(C)(C)F)CCC1C c1(C(C)CN2CCC2C2CCC2)n[nH]c(=NC(=O)NC2CCCCC2)s1 CN1CC2CCC(C1)C2N(S(=O)(=O)Cc1sc(Cl)cc1Cl)C C1(C(C(=O)NCC(=C)C)N(C(C)C)CC)CCCC1(C)C Cc1n[nH]c(=NCCC(C)(C)NC(=O)C(C2CCOCC2)F)s1 CC(C(C)(C)C(=O)NCCN1CCNC1=O)NC(=O)Cc1ccccn1 N1(C(CCN(C(CCC)C)C)=O)CCC(NC(=O)C(O)C2CCCC2)CC1 CC#CCCCC(=O)NCC(CNC(c1ccccc1CN(C)C)=O)OC CP1(=O)CCN(CC(N2CC3(C2)CN(C(c2ncccc2Cl)=O)C3)=O)CC1 c1(C(=O)NCC(CC)(C)NC(=O)CCC2CCCN2C)cnn2c1CCC2 c1(CC(=O)NCCN(C(C(CC2CC2)OC)=O)C2CCCC2)cc(C)sc1C CC1=C(C(=O)NC2CCC2NC(C2CC(C(C)C)=NO2)=O)CCCO1 C1(NC(C(CCSC)O)=O)CCCC2CN(c3cc(C#N)nc(C)n3)CC12 C(c1cccc(OC)c1)=CC(=O)NC1CC(F)(CNC(C(CC)C)=O)C1 N12Cc3ccc(cc3C1)NC(=O)C2.C1(C(=O)NC(CCC)C)CCC(=O)N1 c1(CNC(c2n(CC)ccn2)Cc2ccc(C)cc2O)c(F)c(F)cc(F)c1F C1(NC(CSCc2nnc(COC)s2)=O)CCC(F)(F)CC1 N1(C(c2c(Cl)cn(CCC)n2)=O)CCC2C(CCN2C(=O)C=CC(C)C)C1 c1(C(C)=O)ccc(NC(C2CC2NC(=O)Cc2sccc2C)=O)cc1[N+](=O)[O-] C1(NC(CC(CC=C)NC(=O)C=Cc2ccc(C)o2)=O)C2CCC(C2)C1(C)C c1(CNc2nccc(OC(F)F)c2)c(N=[N+]=[N-])cnn1C c1(CC(=O)N(CCNC(C=Cc2occ(C)n2)=O)C(C)C)ccc2ncsc2c1 Cn1nc(C2=CCCCC2)c2ccc(C(=O)Nc3cc(O)ccc3Cl)cc12 CC(C)(C#N)CCC(=O)NCCC1CC(NC(C2CCCCN2C(N)=O)=O)C1 Cn1cnc2cc(C(N3CCC(NC(c4n[nH]cc4Cl)=O)C(O)C3)=O)ccc12 Cc1cc(C)c([N+](=O)[O-])cc1C(=O)NC12CC(C1)N(C(=O)CC(F)(F)C(F)F)C2 c1(OCC(=O)NCC(CNC(C(C)(Cl)Cl)=O)O)ccccc1C#N c1(C(C(N2CC(NC(C3CC(C)=C(C)CC3)=O)C2)=O)C)ccc(S(N)(=O)=O)cc1 C1(NC(c2c(C)nncc2)=O)(CO)CCCN(C(C2(C#N)CCC2)=O)C1 C=Cn1nncc1C(=O)NC1CCCC(NC(c2cc(CC(C)C)c[nH]2)=O)C1 c1(CCCOC(CN(C(C(C)C)CO)C)=O)cc2ccccc2o1 c1(N(CC(CC)OC)C)nc(=NCC(C(C)C)OC(C)(C)C)[nH]c2cc[nH]c12 c1(NCC(=O)NC2C(NC(C(C)c3cccs3)=O)C2)ccccc1C(F)F c1(C(=O)NC2CN(C(C3(C)C(C(=O)OC)CC3)=O)C2)c(C)noc1-c1cccs1 C12(C(=O)NC3(CCNC(CSS(C)(=O)=O)=O)CCC3)COCC1C2 c1(C(=O)NC2CN(C(CCC(C)SC)=O)CC2O)cc2nccc(Cl)c2s1 c1(C(=O)NCC(c2ccc(Cl)cc2)=O)n[nH]c2c(F)cccc12 S(=O)(=O)(c1ccccc1C(=O)N)NC(C)C(C)C(=O)O.C1(N)CC1 c1(C(N2CC(NCc3ccn(C)n3)C(O)C2)=O)ccc2cc(Br)ccc2c1 CC(C)C(C)(O)C(=O)NC(CNC(c1cc(-c2cccs2)on1)=O)CO c1(CC(=O)NC(CNC(c2c(C)sc(Cl)n2)=O)C)coc2cc(C(C)C)ccc12 C1(C(N2CC(C)C(NC(=O)CCn3ccnc3)C2)=O)CC2CCC1CC2 N1(CC)CCOCC1CC(=O)NCCC(C)N(C(=O)Cc1cnns1)C CC1CC2(CC(NC(=O)C(C(C)O)NC(C3CCS3(=O)=O)=O)C2)C1 Cc1ncc(C(=O)N(CC(C)NC(=O)Cc2ncccc2C)C)c(O)n1 c1(CC[Si](C)(C)C)cnc2[nH]c(=N)sc2c1.C12CCCC1C(=O)N2CCC CC1CC2CN(C(=O)CC(O)C(Cl)(Cl)Cl)CC2N1C(=O)CC(C)(F)F c1(OC)ccc(N2CCN(C(c3nnnn3C3(C)CC3)C3CCCS3)CC2)cc1 N1(CC)CCC(NC(=O)CC2(C)CCN(C(c3cnc(C)[nH]c3=N)=O)C2)C(C)C1 C1(OC)CC(CO)N(C(=O)CC(CNC(=O)CC2CCSC2)C2CCC2)C1 C(CCC(=O)NCC(C)NC(C1CC1(C)C(C)C)=O)OCC(C)C CC1CN(C(=O)Cc2c[nH]nc2O)CCCN1C(C1OC2CCC1CC2)=O c1(NCCCC=C)ncccc1S(=O)(=O)NCc1cccc(F)c1C C1CC2CC1CC2=O.CC1(C(=O)N(CCCF)CCO)CN(C=O)C1 N=c1[nH]c(=NCCn2cc(Br)nn2)[nH]c(=NCCC2CCCCO2)[nH]1 C1(C(=O)NCC(CC)NC(=O)Cc2nc[nH]n2)CCCCC1C(C)(C)C c1(C(N2C(c3cccc(C)c3)CC2)=O)c(C)cccc1O c1(C(N2C(C(C)NC(C3(COC)CCCO3)=O)CCC2)=O)cc(Cl)c(N)cc1F C1(NC(=O)CCc2cnoc2)CC2CC(NC(=O)Cc3nnc(O)s3)CC12 N1(C(C(CCCC)O)=O)CCCN(C(=O)Cn2cc(C(F)(F)F)nn2)C(CO)C1 C1(NC(=O)Cn2cncn2)CC2CC1CN(C(c1nn[nH]c1Cl)=O)C2 N1(C(C2(C)CN(C(C(C3CCCC3)OC)=O)C2)=O)CC2CCC(C1)C(=O)N2 N#Cc1cnc(NC(=O)CC2CC(NC(c3ccc(F)nc3F)=O)C2)cn1 c1(SC2CC(NCC(=O)NC(C3(CC#C)CC3)=O)CC2O)nc2ccccc2o1 C(=O)(C(O)CC(C)C)NC(C(=O)NC(CC)C(N)=O)C(C)OC Cc1ncc(C(N2CC=CC2(C)C(=O)NCCN2CCC(C)(C)C2)=O)n1C Cc1csc(C=CC(=O)NCCC(C)N(C(=O)Cc2ccco2)C)n1 c1(C(=O)NCC(C2CCCCC2)NC(CC2N(C)CCC2)=O)ccn2nccc2n1 N1(C(c2cccc(CC)c2N)=O)CC(C)(C)OCC1CNC(=O)Cn1cnnn1 CCC(O)C(C)C(=O)N1CC(C)C(C)(CNC(=O)CSCc2c(C)noc2C)C1 c1(NCC(=O)NCC(C)N(C(=O)Cc2scnc2C)CC)cccc(O)c1 CC1=NOC(=O)C1CC(=O)NCC1C=CCN1C(=O)CNc1cccc(C)c1 c1(C(=O)OC(C)(C)C)nc(C(=O)OCC2CCCS2(=O)=O)cn(N)c1=O c1(C(=O)NCC(C(C)(C)C)NC(CC(CC)C)=O)cc(S(N)(=O)=O)c(C)cc1C C1(CC(=O)NCC(C)(CO)NC(=O)C=CCN2CCOCC2)(CC=C)CCCC1 c1(COC)nc(NC2CC2C(=O)Nc2ccc(C)nc2C)cc(C)n1 c1(C(=O)NC2C(CC)CN(C(c3ccoc3C)=O)CC2)ccc(C)c(F)c1N N1(C(CN(CCOC)C)=O)CC(CNC(C2CCCN2C(=O)CC)=O)C(O)C1 N1(C(c2ncc(C)cn2)=O)CC2(CNC(=O)COC(=O)CO)CC1CCO2 C(=O)(C(CO)C(C)C)N1C(CN(C(c2ccc(OC)cc2)=O)C)CCC1 N1(C(C2C(NC(C=C(COC)C)=O)C=CCC2)=O)CCC(C2CCCC2)C1 c1(C(N2C(CN3CCCC3)C=CC2)=O)ccc(CNC(=O)CC2CC2(Cl)Cl)cc1F C(=O)(CC1=CCN(C(C2(Cl)CC2(F)F)=O)CC1)NC(CC(=O)NC)C1CC1 C(CC(C(C)(C)C)NC(c1cccc(N)c1F)=O)N(C(=O)CN(C1CCC1)C)C C1(C(=O)NCC2C(Cn3cc(C(C4CCC4)C)nn3)C2(F)F)CCCOCC1 N12CCc3ccccc3C1CN1C(=CC=C([N+](=O)[O-])C=NC(CCCl)C1=O)C2=O c1(C(=O)NCCC2N(C(C3CC(=O)NC3)=O)CCC2)cc2c(cn1)COCC2 C1(C(=O)NCCCCC2CCCN(C(COCC)=O)C2)CC2(C1)CC1(CC1)C2 Cc1c(CC(=O)NC2CCCC(NC(=O)CCn3ccccc3=O)C2)ncn1C C1(NC(C(Cc2cn[nH]c2)NC(CCOC)=O)=O)CCCCC12CC2 C1(CN(C(C=C(CCN(C)C)Cl)=O)C)COCCN1C(=O)CC1C(=O)NN=C1C C1(N(C(C)(C)C)C(=O)CC2CCCN2C(=O)CN)CCCCCC1 C12(NC(c3c(C)ncnc3)=O)CC(CNC(=O)C(c3ccccc3)C)(C1)OC2C C1(C(=O)NC(CC#C)CC)C2CCC(C2)C1NC(c1cn(CCN(C)C)nn1)=O C1(COC)(NC(=O)C(F)n2cccn2)CCN(C(=O)CCC2CC(C)C2)C1 c1(C(N2CC(CNC(c3cnc[nH]3)=O)C3C2C3)=O)cc(Cl)c2c(c1)OCO2 C1(C2(C(N(CC(CNC(COCC(C)C)=O)O)C)=O)CC2)CCCCO1 CCC(CC(C)C)C(=O)NC1CC1NC(c1cnnn1-c1ccccc1)=O C(=O)(CC(C)C(=O)c1ccccc1)N1CC(CC(C)NC(C2(C)CCCC2)=O)C1 C1(CNC(c2[nH]cc(CC)c2)=O)CCC12CCN(C(=O)C(F)(F)COC)CC2 C(=O)(C1=C(C2CC2C)N(C2CC2)C(=O)NC1c1ccccc1SCCO)OCC CCC(C(=O)OC)C(=O)NCC1(NC(c2cc(CCO)on2)=O)CCC1 c1(C(N(C(C)CN(C(=O)Cc2ccc(CO)cc2)C)C)=O)cn(C)c(=O)nc1O C1(C(N2CCC(CC(=O)N(C3CCOC3C)C)CC2)=O)(COC)CCCCO1 N1(C(CCC(CC)NC(c2cc(C(F)F)[nH]n2)=O)=O)CCC(C)(C2CC2)C1 CCCC(C)(O)CC(=O)NCC1(O)CCN(C(=O)CC(C)SC)CC1 c1(-c2c(CNC(c3cccc(Cl)c3Br)=O)cncc2)ccc([N+](=O)[O-])cc1 C#Cc1cnc(C(=O)NCCC2(CNC(C3CC(C)N(C)C3)=O)CC2)c(C)c1 Cc1cnc(-c2nc(CCCO)nn2C2(C)CCCCC2)c(C)c1 CC1CN(C(=O)C(Cc2cc[nH]n2)NC(c2cc(Cl)ns2)=O)CCC1CO CCN=C(NCCF)NCC.C1(CNC2CC2)(NC)CCCC1 CC1(CNC(=O)C2=CCCO2)CCN(C(c2ccnc(C3CC3)n2)=O)C1 S(=O)(=O)(c1ccccc1S(=O)(=O)Nc1ccc2ncccc2n1)NC1C(C)CN(C)C1 N1(C(CNC(=O)NCC2CCOC2)=O)CCCC(C)(OC(CN(C)CC)=O)C1 CCC(CCCO)NC(=O)C(N1CCCC1(C)C)=O.C1CO1 N1(C(CCC(=O)NCCC)=O)C2CCC1CN(C(C1CC(=O)N(C3CC3)C1)=O)C2 Cc1nc2ncccc2cc1CCC(=O)NNC(=O)c1coc(-c2ccccc2)n1 c1(C(=O)NC)ccc(C(=O)NCC2(O)CC(NC(C3(C#N)CCCO3)=O)C2)cc1 C12(C(=O)NC(C(C)C)C(C)NC(=O)C(=O)NC3CC3)CCC(CC1)CC2 c1(C(=O)NCC2(C(=O)NCc3snc(C)n3)CC2)c(C)cncc1C N1(C(=O)C2=COCCC2)CCCC(C2CCN(C(C3(C4CCCO4)CC3)=O)C2)C1 CCCCC(C(=O)NCC(C)C(=O)NC(C)C)NC(c1ccc(C)cc1)=O c1(C(=O)OC)c[nH]c2cc(Nc3cccc4ccc(C)nc34)c(OC)cc12 CC(CCCc1ccccc1)C(=O)N1CCCC(NC(=O)CCCn2cccn2)C1 C(c1ccc(Cl)c(Cl)c1)=CC(=O)NCC1CN(C(=O)C(Cl)=CCl)CC1O c1(NC(CC2(O)CCN(C(c3nc(C)oc3)=O)CC2)=O)ccc([N+](=O)[O-])cc1 c1(C(=O)NC(CNC(C2CC(OC)C2)=O)C2CC2)cnn2cc[nH]c(=O)c12 N1(C(c2cc(CNC(C3C(=O)NCC3)=O)sc2)=O)CC2C=CC1CC2 C1(N(C(CC)=O)CC2CC2)CCN(C(=O)Cc2ccn(CC3CCCO3)n2)CC1 Cc1ccn2ncc(C(=O)NCC3CC(C)(C)CN3C(c3ccnn3C)=O)c2c1 CC(C)(O)C(F)CNC(=O)CC1(C)CCN1C(C1CC=CCC1)=O N1(C(c2cc[nH]c(=N)c2N)=O)CCC2CCCN(C(=O)CC34CCCC3C4)C2C1 C1(CNC(c2ncc(CC)cn2)=O)CN(C(=O)CNC=O)CCC12CCC2 c1(C(N2CC(NC(=O)Cc3c[nH]nc3O)C(CO)CC2)=O)cc(F)c(F)cc1F N1(C(C#CC(C)C)=O)CC(C)(C)CC1CNC(C1COCCO1)=O N1(C(C2(C)CC(=C)C2)=O)CC2(CCC2NC(=O)C(C2CCCCC2)O)C1 C=C(C)CC(C)C(=O)NCC1CCN(C(c2c(C(F)(F)F)nc(C)n2O)=O)C1 c1(N(C(c2cc(-c3ccc(O)cc3)on2)=O)CC)ccc(N2CCC2)nc1 C1(C(=O)NCC(C(C)C)NC(c2c[nH]c(=NCC)s2)=O)CCc2cncn2C1 CC1=CC(C)CN(C(=O)C(CC(C)C)NC(=O)Cn2cc(C)cn2)C1 c1(C(=O)NCC(CN(C)C(c2ccnc(F)c2O)=O)O)cc2n(n1)CCC2 c1(C(=O)NCCC23C(CN(C(c4cc(C)ns4)=O)C2)CC3)nc2cccnc2s1 C1(OC)CN(C(=O)CCC(N)=O)CCC1NC(=O)CC1(CO)CC1 N1(C(c2c(C#N)ccs2)=O)CC2(CCC2)CC1C(=O)NCCC(C1CC1)C1CC1 C1(C(=O)N(C)CCN(C(=O)CC2C=NN(C)C2=O)C)(COC)CC(F)(F)C1 N1(C(c2c(Cl)cccc2Cl)=O)CCC(C2CCCN(C(C3CC4CC4C3)=O)C2)C1 Cn1ncc(C(=O)NCCN(CCOCCO)C(c2cc(Br)co2)=O)n1 C12(C(=O)NC3(C)CN(C(C4COC5(CCC5)CO4)=O)C3)CCC(CO)(CC1)CC2 C1(C(=O)NCC2(F)CC(CNC(=O)CCF)C2)CN2CCN1CC2 N1(C(COC2CN(S(C)(=O)=O)C2)=O)CCC(N(CC(F)F)CC(N)=O)CC1 C1(NC(=O)CC2CC=CC2)CC2CN(C(=O)Cc3ccnc(F)c3F)CC12 C=CC(CC)CC(=O)N1CCC(C)C(CNC(C2(C3CC3)CC=CC2)=O)C1 Cc1nc(C(N2C(C(=O)N(C3CCC3(C)C)C)CC3CC23)=O)c(C)s1 c1(C(=O)NCCNC(c2cccc(-c3nc(C)[nH]n3)c2)=O)cccc(=O)n1C CCC(C(=O)N1CCC(NC(c2cnc(N)c(Cl)c2)=O)C(F)C1)C(C)C c1(C(CC)C)nc(N2CC3(CN(C(c4cc5sccc5[nH]4)=O)C3)C2)cc(C)n1 N1(C(CC2CCN(C(c3c(C)cnn3C)=O)C2)=O)CCCC(C)C1CCO CC(CS(C)=O)C(=O)N1CC2CC1(CNC(=O)CCSCc1ccccc1)C2 c1(C)cc([N+](=O)[O-])c(Cl)cc1Cl.CC1(C(F)(F)F)CN(NC(c2sccc2N)=O)C1 Cc1c(C)c(C)c(C(=O)NC2CCCC(NC(C3CC3C)=O)C2)c(C)c1C C1(NC(C=CSC)=O)CCCC(CNC(=O)C(Cc2ccccc2)NC(C)=O)C1 c1(SC)ncc(C(=O)NC2CCC(NC(C3(NC(C)=O)CCC3)=O)C2)[nH]1 C(CC(F)(F)F)NC.C1(C(N(C2CN(CCCOC)C2)C)=O)CC(F)(CF)C1 CC1CN(C(C2OCCCO2)=O)CCCN1C(C1CN(C)CCN(C)C1)=O c1(OCC)ccccc1C(=O)NCC1CC(CNC(C2CCCC2(F)F)=O)CO1 CC(CC(=O)N(CC(C)(C)Nc1nc(C(F)(F)F)ns1)C)C1CC1 N1(C(c2ccc(CC)[nH]2)=O)CCC2(CC1)CC(NC(c1cn(C3CC3)nc1C)=O)C2 C1(NC(C2CCCCC2)=O)CCCN(C(=O)C(O)C(F)(F)F)CCC1 C1(NC(=O)Cc2ccc(Cl)c(C(F)(F)F)c2)CCCNC12CCC2 C1(C2CCN(C(C=NOC)=O)C2)CCCN(C(=O)C=Cc2cncs2)C1 C12(C)CCCN(C1)C2=O.C1(C(=O)OC)CCN(C(C2CCOCC2)=O)C1C CC(C)C(C)C(=O)NCCN(C(=O)C(C)OCc1ccccc1)C(C)C c1(SCC(N2CCC(NC(c3c(C)nns3)=O)C23CC3)=O)nnc2ccccn12 N1(C(c2cnc(CC)nc2)=O)CCCC2(CNC(C3C=CCS3)=O)CCCC12 Cc1ccnc(C(=O)NC2CC3(C2)CC3C(=O)N(C)Cc2cocn2)c1F c1(C(=O)NCC2C(NC(C3N(N=O)CCC3)=O)C2)cnc(C2CC2)nc1O C1(NC(C2CCCN(C(c3c(C)cnnc3O)=O)C2)=O)CC2(CCCCC2)C1 CC1CCCCC1CC(=O)NCCCCN(C(=O)CS(=O)(=O)N1CCCC1)C Cc1nc(C(=O)NCC(C(C)C)NC(C2(O)CC2(C)C)=O)nn1C C(CC(=O)NC(C)C(=O)NCCF)N(C(=O)C(C)C1(O)CCC1)CC C1(SCC)CCC(C(N2CC(CN(C)C(C3CCC(=O)O3)=O)C2)=O)CC1 c1(OC)ccc2c(C(=O)NC3(C)CN(C(c4cc(=O)cc[nH]4)=O)C3)ccnc2c1 C(=O)(CC(C(F)(F)F)NC(=O)CC1CCSC1)N(CCOCC#C)C C1(C(N2CC(O)(CN(C(c3cc(CC)on3)=O)C)C2)=O)CC(OC)C(OC)C1 c1(OCCOC)cc(C(=O)NC2CC(CNC(=O)Cc3cn(C)cn3)C2)[nH]n1 N1(CCCCC=C)CC2CCN(C(c3ccc(CC(C)C)cc3)=O)CCC2C1 C(CC(C)(C)C(=O)NC1CCC(CCC(=O)NCC2(C)CCCOC2)C1)OC N1(CC=CCC)CCC(NC(=NCC2CCCO2)NC)CC1.C1(C)=CC=C1 C(=O)(CCC(CC)CC)NCCCC(CCC)NC(c1nc(C)ccc1Br)=O C1(CC(=O)NC2CCN(C(Cc3cccc(CC)c3)=O)C2C)OCCOC1(C)C CCC(O)C(C)(C)C(=O)NCC1(F)CC(NC(c2cccc(CO)c2)=O)C1 c1(C(N(CCNC(CCn2ncn(C)c2=O)=O)C2CC2)=O)cnc2nccn2c1 N1(C(C=Cc2cnc(C)s2)=O)CCC(N(C)C(C2CCCC(=O)N2C)=O)C(C)C1 N1(C(CCCC)=O)CCC(C(F)CNC(C2(C)CC=CCC2)=O)CC1 c1(C(=O)NCCN(C(=O)C(C)C(C)C)CC)cncc2n[nH]cc12 C(=O)(CN1C(=O)Cc2ccccc21)NCC(CC=C)NC(C1CC(CF)C1)=O CN1CC2(CC2)CC1C(=O)NC1(C)CC(C(N2CCC(O)(C(N)=O)C2)=O)C1 c1(OC)ccc(F)c(C(N2CCCC2(C)c2cn(C3CCOC3)nn2)=O)c1F c1(NC(C2CCN(Cc3ccc(CO)o3)CC2O)=O)cccc2c(I)n[nH]c12 N1(C(C2CC(C)N2C(=O)Cc2ccccc2Br)=O)CC(C)C(C)C1 CC1OCCC1C(=O)NOCC(=O)NC1(C)CN(C(=O)COCCN(C)C)C1 c1(C(=O)NC(CN(C(c2cc(C3CCC3)on2)=O)CC)C)cnc(C)[nH]1 C#CC1(NC(=O)C(c2ccnn2C)NC(c2cc(C)cc(F)c2)=O)CCC(C)CC1 c1(C(=O)NC2(CO)CCN(C(c3ccncc3O)=O)C2)cc2c(=O)[nH]ccn2c1 C1(NC(c2c(C)cnc(F)c2)=O)CN(C(c2ccc[nH]2)=O)C2CCCCC12 Cc1nccnc1C(=O)NCC(O)C(F)(F)F.C1CC(=O)N1C(C)(C)C Cc1c(C(N2CCN(CCCNC(C3CCCC34CC4)=O)CC2)=O)nnn1C C(CCCCC(=O)NC(C)(C)CCNC(c1cc(-c2cccs2)on1)=O)OCC CC(C)(CF)C(=O)NCCC1CCN(C(c2ncc(C(F)(F)F)s2)=O)C1 C1(C(=O)NCC2(NC(=O)Cc3ccncc3F)CCCCC2)CC2C(C1)C2(F)F c1(-c2scc(C(c3ncccc3C)Nc3n(CC)nnn3)n2)ccc(Cl)cc1F c1(CNC(CCC2OCC(C)(C)C2)=O)ccc2c(c1)CN(C(=O)Cc1ccsc1)C2 C1(N(CCCO)C(c2c(C)[nH]c(C(C)(C)C)c2)=O)CCC2(CCNC2=O)CC1 c1(C(N2CCC(NC(=O)CC3CCCCC3(F)F)C2)=O)cnc2scnc2c1 C(=O)(CCC(C)(C)c1ccccc1)N(C1CC(NC(CNC(=O)OCC)=O)C1)C C=C(C)C(CC(=O)NC1CN(C(c2cnc(C)s2)=O)CCC1C)OCC Cc1cc(=NC(=O)CSCC(N2CC3CCC2C3NC(=O)C2CC2)=O)[nH]o1 N1(C(C2(C)N(C(C(CC#C)C3CC3)=O)CCC2)=O)CCC2CCCC2C1 C1(NC(C(N2CCCCC2)C)=O)(CO)CCN(C(c2cccc(CO)n2)=O)C1 N1(C(C2CSCCN2C(=O)Cc2ccccc2Br)=O)CCC2(CC1)COC2 C1(NC(C2C(OC)CCC2)=O)(CNC(C2CC=C(C)CC2)=O)CC2CCC1CC2 n1(CCCC(=O)NC(CN(C(c2cnc(C(F)F)s2)=O)CC)C)c(O)nnc1O N1(C(C2SCCS2)=O)CCc2cc(O)c(Br)cc2C1 CCC(C)(C(N)=O)NC(C1CCC(CNC(c2ccc(N)cn2)=O)CC1)=O C(c1ccc(F)c(F)c1)=CC(=O)NCCCC(CCC)NC(c1cc(C)no1)=O C1(C(=O)NC2(C(C)(C)OC)CC2)CC12CC(NC(=O)COC1CCC1)C2 CC1CC(C(=O)N2CCC23CN(C(C2COCCN2C)=O)C3)=NO1 CCC(C(=O)N1CCC(C2CCCCN2C(c2cc(CO)[nH]n2)=O)CC1)C(C)C C1(=O)C(CCF)NC(=O)C(=O)CN1.C1(=O)C(C)N1C.CCCCO.OC C1(CC(=O)NC2C(OC)COC2)N(C(=O)CN(c2ccncc2)C)CCC1(C)C CON(C)C1CCN(C2CCN(c3cncc(C)n3)C2=O)CC1 C(=O)(C(C)CC(C)CC)N1CCC(CNC(CC=CCC)=O)C12CC2 c1(C(=O)NC(C(C)NC(CCCC=C)=O)CO)cc2occc2n1C N1(C(c2c(C)noc2)=O)CCN(C(=O)CCc2cccnc2Cl)CC1C(C)C C#Cc1ccc(C(N2CCN(C(=O)C(C)N3CCC3)C(C(C)C)C2)=O)cc1 c1(C(=O)NC2C(C)N(C(=O)Cc3n[nH]cc3Br)CCC2)ccn2ccnc2n1 C(=O)(NNc1c(F)cc(Cl)cc1F)NC(C(CC)CO)C c1(C(=O)NC(CC2CCN(C(c3c(SC)ccs3)=O)CC2)C)cccc(Cl)c1Cl c1(NC(N2CCCC(NC(c3ncc(C)cn3)=O)C2)=O)ccc(C)cc1F N1(C(C(C(C)C)NC(C)=O)=O)CCC2CCC(NC(C3CCN(C)C3)=O)C1C2 N1(C(=O)NCC(CCC)CC)CCC2(CC1)OC(=O)NC2=O C(=O)(C(O)C(C)(C)C)NC1CCN(C(CC(C)SC)=O)C1 C(=O)(CC(C)C(F)F)NC(c1cccc(OC)c1)CNC(c1occ(C)c1C)=O CC1C(=O)CC1C(=O)NCC1CC(NC(=O)CCC2CCCO2)C1 c1(OC)cc(CNC2CN(C(=O)OC(C)(C)C)C3(CCC3)C2)cc(OC)c1Br C(N=c1nc2c(ncn2C)c(N(C)Cc2ncc[nH]2)[nH]1)c1cc(C)nc(C)c1 N#Cc1cnn2ccc(NCc3csc(NC(=O)CCCC(F)(F)F)n3)nc12 Cc1cc(C(N2CC(CNC(c3csc(C(C)(C)C)n3)=O)C3CC23)=O)ccc1F N1(C(C(C)N(CCC)C(c2ccn(C)c2CC)=O)=O)CCCC2CC1C2(C)C N1(C(CCc2onc(C)n2)=O)CCC2CCC12CNC(c1cccnc1F)=O c1(C(C(=O)N(CCC(=O)NCCOCCC=C)C)C)ccnn1C C1(O)(C(=O)NCCC2(NC(c3ccn(C)n3)=O)CC2)CCCC(C)(C)C1 C1(CNC(C2(C(=O)NC)CC2)=O)CC2COCC2N1C(c1cc(C#N)n(C)n1)=O CC1(C)C(O)CCN1C(=O)CC1(NC(c2cc(CO)on2)=O)CCC1 N1(C(c2n(CCOC)ccc2)=O)CCCC(CNC(=O)C(C)=CC(C)(C)C)C1 c1(OC(C)C)cccc(C(=O)NCC(O)CNC(=O)C2=CCCOC2)c1F C(=O)(C1=Cc2cc(OC)ccc2OC1)NC1C(CNC(C(CC)CC)=O)CCC1 FCCN=C(NCC1CS(=O)(=O)C1)NCC1(c2ccc(Cl)c(F)c2)CCC1 CC(C)(C)CC(O)C(=O)N1CC(NC(c2ccc(Cl)o2)=O)C(c2ccnn2C)C1 N1(C(CC2CCC(C)CC2)=O)CC2CN(C(=O)CN(C3CCCC3)C)CC2C1 C1(C(N2CCC(CSC)C2)=O)(NC(=O)C=Cc2ccc[nH]2)CCOCC1 CC(C(=O)N(CCNC(C1CCCCCN1C)=O)CCOCCOC)S(N)(=O)=O c1(C(=O)NCCN(CCOC)C(C2(OC)CCCCC2)=O)ccc(Cl)nc1O c1(CC)nc(C)c(C(=O)NC(C2CN(C(c3[nH]ccc3C)=O)CCO2)C)s1 C(=O)(C1CCCn2nccc21)N1CC(C(=O)Nc2ccc(O)c(O)c2)C(O)CC1 C(CC(C(=O)NCC(C)(C1CC1)NC(=O)C=CC(F)(F)F)NC(C)=O)SC N1(C(c2nc(C3CC3)cs2)=O)CCN(C(C2C=CCC2)=O)C(CF)C1 C1(NC(CCCN(C(C)=O)C)=O)C2CC3C(C2)C13C(=O)NC1CCC2(CC1)N=N2 N1(C(C=CCCC)=O)CC(CNC(=O)CC2CC2)C(O)C1 CC1(C)C2CN(C(c3cc(C(F)F)no3)=O)C(C(=O)Nc3ncnn4cccc34)C12 c1(OC)cc(Br)c(CN2CC3CC2CN3C(=O)Nc2ccc(CO)cc2)cc1O N1(C(=O)NC2CCC(N)C2)CCCC(N2CCCC2)C1 C#Cc1c[nH]nc1C(N1CCC(F)(C(=O)NCCC2OCCC2(C)C)C1)=O c1(CC)n[nH]c(=NC2CC(CNC(=O)C(c3c(F)cccc3F)C)C2)s1 c1(CC(=O)NCC(CNC(C(CC=C)(C)C)=O)CO)cnc2n1CCOC2 C12(C)CCCC1NC2=O.C(=O)(C(C#N)NC(C)(C)C)N(C(CN(C)C)C)CC.C(=O)O N1(C(c2cc(C)ns2)=O)CC(C)CN(C(C2(N(C)C)CCCC2)=O)CC1C N1(C(C(=CC2CCCC2)C)=O)CCC(N(C(=O)C(C)Nc2ccccn2)C)CC1 C1(C(=O)NC2CCN(CC)C2=O)CCN(C(=O)C=Cc2cc[nH]c2)C(C)C1 C1(NC(=O)COc2ccc(F)nc2)CN(C(C2CCO2)=O)CC1n1ccnn1 N1(C(c2nccc(OC)c2)=O)CCN(C(=O)Cc2ccc(F)cc2)CC1C(C)C C1(C(N(CC(N2CCCC2)C)C)=O)C2CC3C(C2NC(c2ccc(C#N)n2C)=O)C13 N1(C(C2(C)N(C)CCC2)=O)CCC(C2CCN(C(=O)CNC(=O)CC(F)(F)F)C2)C1 N1(C(c2c(OCC=C)cccn2)=O)CCN(C(=O)COC2CCCC2)C(CO)C1 c1(C(N)=O)ccc(C(N2CC(CO)C2)=O)cc1.Cc1cc(NC(c2nncs2)=O)no1 O=S(=O)(c1ccn(C2CC2(F)F)n1)N1CCC2CC1CC(O)CC2.c1(N)ccccc1 c1(C(N(CC(C)CNC(c2cccn2C2CC2)=O)C)=O)ncn(-c2nccs2)n1 CC(C(=O)NCCCNC(c1cn(C)nc1-c1ccccc1)=O)P(C)(C)=O N1(C(C(C)Oc2ccc(F)cc2)=O)CCN(C(=O)CCCF)C(C)C1 N1(C(c2ccc(C(F)F)o2)=O)CCC2C(CCCN2C(=O)CCC2CC2)C1 C1(O)(CN(C(c2cc(C)nn2C)=O)C)CCN(C(C2CCCCC2F)=O)CC1 N1(C(C(C=C)(F)F)=O)CCC2C(CCCN2C(c2ccc(P(C)(C)=O)nc2)=O)C1 C1(C(N2C(C#C)CCC2)=O)CC2CC1CC2NC(c1cnc(C)o1)=O S(=O)(=O)(c1cnc(Cl)nc1)N1C(C(=O)NCc2cncc(O)c2)CC2CC21 c1(C(N2CC(F)(CNC(CC(C)(O)C(F)F)=O)C2)=O)c(N)nn2ccccc12 c1(C(=O)NCCN(C(=O)CC2OCCC2C)CCOC)nnn2c1CCCC2 C1(NC(C(C)C)=O)CCCCC1NC(=O)CN(C1CCSCC1)C N1(C(c2cscn2)=O)CC2(CCN(C(=O)C(c3ccc(F)cc3)(F)F)C2)C1 c1(OC)ccc(C(N2CC(N(C)C(c3ccc(COC)[nH]3)=O)C(F)C2)=O)c(F)c1 Cc1cccc(C(=O)N(C(C)(C(=O)NC2CC2)C2CC2)C)c1O.C12CN(C1)C2 N1(C(Cn2ccc(C)cc2=O)=O)CCN(C(c2cnco2)=O)CCC1C C1(C(N(C(C)C)CCNC(=O)C=C2CCC(C)C2)=O)CCc2ccccc2C1 CC1(C)COC(C(=O)NCC(=O)NC2C=CCCC2)C1 C1(CNC(C=C(C)C(C)C)=O)CCCN1Cc1nc(CC2CC2)on1 c1(C(=O)NCc2ccnc(F)c2)ccc(NS(=O)(=O)CCCCl)cn1 N1(C(CC2(NC(C(C)CC3CC3)=O)CC2)=O)CC2CCOC2C1 c1(CC(=O)NC2CN(C(c3n(CCC)ncc3)=O)C(C)C2)c(OC)cccc1C c1(CNC(=O)NC2(c3cc(CO)cc(C)c3)CCC2)c(Br)cc(F)c(Cl)c1F Cn1nc(C(=O)NCC(CNC(=O)Cc2cnoc2)S(C)(=O)=O)c(Cl)c1Cl C=CCCC(CC(C)C)C(=O)NC(c1cn(C)nc1I)c1nnnn1C(C)(C)C C#Cc1cccc(C(=O)NCC2CC2NC(=O)C=Cc2ccc(Cl)cc2)c1C N1(C(c2ccsc2)=O)CC2CC1CN2C(c1ccc(Br)cc1C(F)(F)F)=O C1(OC)CC(C(=O)NCC2(C)CC(O)C2)N(C(=O)COC2(C)CCCC2)C1 CC1(C)OCCOC1CC(=O)NCCC1CCCN1C(=O)CC1(C)CCOCC1 C(=O)(C1=CCCCC1)N1CCC(CC)C1CNC(=O)CC1CC(OC(C)(C)C)C1 C1(NC(c2cncn2C)C)CN(C(=O)CSCc2ccccc2)CC1O c1(C(N(CCOCCC(=O)NC(CC#C)C)C)=O)ccnc(O)c1 C1(C(=O)NCC2CC(NC(C(C)n3cnnn3)=O)C2)CCC(C)CC1 c1(C(=O)NCC2(O)CCN(C(C(C)(C3CC3)NC(C)=O)=O)C2)cccc(F)c1C N#CC1(C(=O)NCCn2cnc(C(=O)NCc3cc(=O)cc[nH]3)c2)CCOC1 c1(-c2cccc(C)c2)nc(=NC(=O)C(=O)NC2CCOC2c2ccccc2O)s[nH]1 C1(C(=O)NCC(C)N(C)C(c2c(Br)nnn2C)=O)CC2C=CC1C2 C1(c2n(CS(C)(=O)=O)nnn2)(Nc2ccccc2I)CC2(C)CCOC12.C1CCC1 N1(C(CC=C(C)C)=O)CCCC2(NC(=O)CN(C)S(N)(=O)=O)CCCC12 C12(C(=O)NC(C(C)NC(c3sncc3Br)=O)C)CCN(CC1)C2 C=CCC(CNC(C)=O)C(=O)NCCC1CCN(C(=O)CC(=O)OC)C1 N1(C(C2(CSC)CC2)=O)CCN(C(c2cn(C)nc2C(F)(F)F)=O)C(C#N)C1 C1(NC(C2C(CC)C2)=O)CCC2(CCCN2C(=O)Cc2ccc(F)cc2)CC1 N1(C(C(C)CF)=O)CCN(C(=O)C=Cc2cnccn2)CC2(CC2)C1 Cc1cc(C(F)(F)F)c(C#N)c(N2CCN(Cc3cc(Br)cc(C)c3N)CC2)n1 CC1(C#CC(=O)NCC2(O)CN(C(C3CC3c3ccccc3Cl)=O)C2)CC1 N1(C(CCN(CCCO)C(C2C(CC)CC2)=O)=O)CCC(F)(F)C(C)C1 N1(C(c2cc(C)sc2Cl)=O)CCCC(NC(=O)CCCCC2CC2)C1C C1(CNC(=O)C=C2CCCCC2)CCCC2(CN(C(C3CC3Cl)=O)C2)O1 c1(C(=O)NC23CC(CNC(C(C)SC(F)(F)F)=O)(C2)OC3C)cccc2ccnn12 C1(NC(CN(S(C)(=O)=O)C)=O)CCC(NC(c2cc(C3(C)COC3)no2)=O)C1 Cn1c(C(=O)NC(CO)C(=O)NCCCc2cc[nH]n2)cnc1Cl N1(CC(=O)NCC(OCCc2cccc(C3CCN3)c2)OC)C2CCC1CC(F)(F)C2 [N-]=[N+]=Nc1ccc(Cl)cc1C(N1CC(c2ccc(C(=O)O)cc2)(O)C1)=O Cc1nn2cc(C(N3CCCC(CNC(c4onc(C)c4Br)=O)CC3)=O)nc2s1 Cc1ccc(F)c(C(N2CCC(N(c3cc(F)ncn3)C)CC2)=O)c1Cl C1(C(=O)NCC(C2(SC)CC2)OC)CCN(C(=O)CCc2nc(O)n[nH]2)C1 N1(C(C2CN(C)C2)=O)CCCC2(CCN(C(c3cscc3F)=O)C2)C1 CCC(CC)CC(=O)NCC1CC2(C1)CN(C(=O)CCC1CCOC1)C2 CCCC(CCC)CC(=O)NC1CC2CN(C(=O)CN3CC4CC4C3)CC12 C1(OC)CN(C(C2CCCC2)=O)CC1NC(c1cnoc1C1CCC1)=O c1(NCCNC(c2c(C)scc2)=O)ncnc2scc(-c3ccccc3)c12 c1(NC(N2CCC(Cc3ccco3)C2)=O)cnc2ccccc2c1 N1(C(N2CC(c3cnc(C)[nH]3)C2)=O)CCN(C(=O)NCC(c2ccco2)=O)CC1 c1(C(=O)NC2C(NC(=O)CCCOC3CCOCC3)C2)cccc(Br)n1 C1(CCC(C)C)CCN(C(C2CCCN2C(=O)CCOC2CC2)=O)CC1 CCC(CCC(=O)N1CCC=C(CNC(=O)CC(c2ccnc(C)c2)OC)C1)OC CC1(NC(=O)CC2CNC(=O)O2)CCN(C(=O)Cc2cc(C(F)(F)F)n[nH]2)CC1 c1(C(N2CCC(F)(CNC(c3coc(Cl)c3)=O)C2)=O)coc2ccc(Cl)cc12 C1(C)(OC)CC(NC(=O)C(F)CC2CN(C(=O)CC3(O)CCOCC3)C2)C1(C)C C(C(=O)NCCN(C(=O)C(O)Cc1ccccc1)C1CC1)(C(C)C)SC c1(OC)ccc(F)c(CN(CCNC(C23CCCC2(C(N)=O)C3)=O)C(N)=O)c1.C(=O)OC c1(OC)ccc(C(N2CCOC(CN(C)C(C3(CO)CC3)=O)C2)=O)nc1N N1(c2ccnc(N3Cc4c(C)ncn4CC3)n2)CCC2(CCC(C)CC2)C1 C(=O)(CCC(F)(F)F)N1C(C(=O)NCc2n(CCC)ncn2)CC=CC1 N1(C(C(COC)C)=O)CCC(C2CCC2)(CNC(c2nnc(S)n2C)=O)CC1 N1(C(C(CCC)O)=O)CCN(C(C2(F)CCOCC2)=O)CC1CC1CC1 N1(C(c2[nH]cc(C(N)=O)c2)=O)CCOCCC1C(=O)NCCC1COCCO1 Cc1cc(S(=O)(=O)N2CCCC(C)(C(N3CCOC(C)C3)=O)C2)ccc1Br C1(C(N(CCCO)CC#C)=O)C2CCC(C2)C1NC(=O)C1=C(C)CCC1 C1(CC(=O)NCC(=O)NC2(CCS(=O)(=O)N(C)C)CCC2)CC(O)C1(C)C N1(C(COCC)=O)CCC(CN2CCN(C(=O)C(F)(F)C3(O)CCC3)CC2)CC1 N1(C(c2c(N)n(CCO)nc2)=O)CCN(C(=O)CCC2CC2)C2CCCCC2C1 C1(CN(C(=O)CC2CC3C=CC2C3)CC)CCCCN1C(=O)C(C)C1CC1 C1(OCC)CC2CN(C(=O)C(CC(C)C)NC(C3(C#N)CC=CC3)=O)CC12 C1(N(C(CN2CC(CC)C2)=O)CC2CC2)CCN(C(=O)C=C2CCC(C)C2)CC1 C(C(=O)N1CCC(C(F)CNC(=O)Cn2ncccc2=O)CC1)(C(C)C)OC c1(C(=O)NCC(C)NC(C2(COC)CCCCO2)=O)cc(C)ccc1O N1(C(c2c(NC)ccc(F)c2)=O)CCC2CC1CN(C(=O)CCC=C(C)C)C2 C1(NC(c2ccc(C(F)(F)F)nn2)=O)CCC2(CC1)CN(C(=O)COC1CC1)C2 c1(CC(=O)NCCCCCCNC(C2(C(CC)(F)F)CC2)=O)nnc2n1CCOC2 C1(NC(C2N(C(Cn3ncc(C)c3)=O)CC=CC2)=O)CN(C)CCC1O N1(C(C2CC2(F)Cl)=O)CCCOC(c2cn(-c3ccccc3Cl)nn2)C1 S(=O)(=O)(c1ccc(N2CCOC(CC(N)=O)C2)cc1Cl)N1C(C)CN(C)CCC1 C1(C(N2C3C(NC(=O)CC4CCS(=O)(=O)C4)C(C3)C2)=O)CC12CCOCC2 C=CC1CCCCN1C(=O)COC1CC(NC(c2ccccc2SCC)=O)C1 C=CC(C)C(C)C(=O)NC1CN(C(C2(CSc3nnnn3C)CCC2)=O)C1 c1(C(N2CC(CC)C(NC(c3nccn3C)=O)CC2)=O)ccc2c(c1)COCO2 C(=O)(CC(O)C(C)(C)C)N1CC(C(C)NC(=O)C(C)NS(=O)(=O)c2cccs2)C1 c1(C(=O)NCC(C)(C)CNC(=O)C(CC(F)F)C2CCC2)ccc(N)cc1F CC(F)(F)CCCC(=O)NCC1CC(NC(=O)C(F)(F)c2ccccn2)CC1O C1(CN(C(c2cc(CC(C)C)on2)=O)C)CN(C(=O)CN(C2CC2)C2CC2)CCO1 O=C(N=c1ccn(C2CC2)[nH]1)C12CC1CN(Cc1ccc3occc3c1)C2 c1(NC2CN(C(c3n(C)c4c(c3)occ4)=O)C2)cc(Cl)c2c(F)cccc2n1 C1(C(=O)NC23CC(NC(CN(C)C)=O)(C2)C3)C2Cc3ccc(Br)cc3C12 C123CCC(CC1)(CO2)NC3=O.Cc1c(-c2nnc(SC(C)(C)C)o2)ncn1C N1(CCCC)CC2CCC1C(NC(=O)C(C)Oc1ccc(OC)cc1)C2 C(c1cncn1C)=CC(=O)N(C)CCSC1CC1.N12CCCC1CC1(CC1)C2=O N1(C(c2nc(CCC)oc2)=O)CC(C2CN(C(C3SC4C=CC3C4)=O)C2)C1 CC(C(=O)N1CCC(O)(CNC(C2CCC3(CCC3)C2)=O)CC1)C1=CCCC1 Cc1nn(CC(C)C)c(C)c1S(=O)(=O)N(C)CC1CCC1O C1(CN(C(=O)C(O)Cc2cnn(C)c2)C)COCCN1C(=O)CC1(C(F)F)CC1 C1(C(=O)NC2C(NC(c3ccc(F)c(Cl)c3F)=O)C2)CCc2cc(F)ccc2O1 C1(C(=O)O)CCc2nc(NC3(C=C)CN(C(c4ccc5n[nH]cc5c4)=O)C3)[nH]c2C1 c1(C(=O)NCC(C)(C)NC(=O)C(C)CF)cccc(C(N(C(C)C)C)N(C)C)c1 CCC(C)(COC)CNC(C12CC(NC(c3cnnn3C(C)C)=O)(C1)C2)=O C1(C(=O)NC2(CCC)CC2)N(C(=O)CC2CS(=O)(=O)C2)CC12CCCC2 c1(CC(=O)N(CCC(C)NC(=O)Cn2ncnn2)C)csc2ccccc12 C1(NCCNC(N(C)C)=O)CN(C(c2ccoc2)=O)CC1(F)F Cn1ncc(C(N2CC(F)CC2CNC(=O)CCCOC(C)(C)C)=O)c1F N1(C(c2c(C)scc2)=O)CCC2CN(C(c3cnc4n3CCS4)=O)C2C1 c1(C(C)C)nc2c([nH]1)CC(C(N1C3CCC1CN(C(=O)COCCF)C3)=O)CC2 c1(C(N(C(C)C)CCNC(=O)CC(C)C(F)F)=O)scc2c1OCCO2 c1(C(=O)NC(C2CCCN(C(c3cn(C)nn3)=O)C2)C)cccc2ncnc(O)c12 CC1(C)CC(NC(C2CC3CC2C2CC32)=O)CN(C(c2ccnc(Cl)c2)=O)C1 c1(C(N2CCC(NC(CSCC(=O)OC)=O)C2)=O)ccc2ccccc2n1 O=C(C1=CCCS1)NC1CCN(C(=O)C(O)CC2CCOCC2)CC1 C(=O)(C1Cc2ccccc21)NCC(C)NC(c1cc(C(=O)OC)no1)=O c1(C(=O)NC23CC(CNC(C4C(C)C4)=O)(OC2)C3)cc(S(C)(=O)=O)ccc1O c1(C(=O)NC2(C3CCCC3)CC2)cn(C)c(=O)n1C.CC1C2CCCN1C2=O c1(C(CO)Nc2cccc(C(=O)NCCCC(C)C)c2)cccc(Cl)c1Cl C1(CC(=O)N(CCC(N)=O)CC)C2CCC(C2)N1C(c1ncccc1CO)=O c1(C(=O)NC(C2CCN(C(c3c(CC)csc3)=O)C2)C)cc2c(nc1O)CCC2 c1(OC)ccc(F)cc1O.C1(CNC(C2(CSC)CC2)=O)C=CCN1C(=O)C C1(CNC(c2snc(O)c2Cl)=O)CCCC(CNC(=O)C=CSc2nc[nH]n2)C1 CC1CC(C(=O)N2CCC(C)(C)C2CNC(C23CC4CC2C3C4)=O)=NO1 c1(C(N(C2CCN(C(c3ccon3)=O)C2)C)=O)cnn2cc[nH]c12 c1(C(=O)NCCC(C)NC(C2(C(F)(F)F)CC=CCO2)=O)cc(F)c(F)cc1N C1(C(=O)NC(COC(C)=O)CO)CC(C)CN1C(c1cc(C(C)C)[nH]n1)=O CC1CCN(C(c2c[nH]ccc2=N)=O)CCN1C(c1cc(Cl)ccn1)=O N1(C(CC(CC)C)=O)CC(C)(C)OCC1CNC(c1cc(C)c(Cl)c(C)c1)=O c1(NC(C2CC(NC(c3c(C)nn(C)c3)=O)C2)=O)cccc(Cl)c1C c1(C(=O)NC(c2ccco2)CO)ccc(-c2ccccc2F)cc1 C1(C(N2CCN(C(CC)=O)CC2)=O)(NC(C)(C)C)CC2(CC2)C1 Cc1cc(C2CC2)cnc1C(=O)NCC(C1CC1)N(C(=O)CCC#N)C C1(N2C(=O)CCOCC2)CCCN(C(=O)CN(CC)CC)CC1.C1(SCC)CCC1 CCC(C(=O)N(C)CC=CC(=O)NCC1(CC(C)C)CC1)C(C)C n1(C(CC(=O)NC2C(c3onc(C)n3)C2(C)C)C)cnc2ccccc12 c1(C(N2CC(NC(C3(C(C)(C)O)CC3)=O)C2)=O)cnn(CSC2CC2)c1 C(c1cncn1C)=CC(=O)N(C)CCOC1CN(C(=O)COc2cnn(C)c2)C1 C1(C(=O)NCCN(C2CCN(C(C3CCCC3)=O)C2)OCC)CC2CCC1C2 C1(CNC(Cn2c(C)cc(C)n2)=O)CCCCCN1C(=O)C(C)CF N1(C(C2(OC)CCCC2)=O)CC2C(NC(=O)C=C3CCCCC3)C2C1 c1(C(=O)NC(C2CN(C(C=CC=CC)=O)C2)C)nn(C)c(Cl)c1Cl C1(C(=O)NCC(C)(C)OCC(=O)NC2(COCC)CC2)C=CC=CC=C1 C#CCCCCCC(=O)N(C)CCOCCCN(C(=O)C(F)CC(C)C)C C1(C(N2CCC(N(CC#C)C(C3CC3C)=O)C2)=O)CCCC(CF)C1 C=CCC(CNC(c1ccn(CCC)n1)=O)C(=O)NCC(O)CF N1(C(C(C)(C)C#N)=O)Cc2ccc(CNC(=O)C=CSc3ccccc3)cc2C1 CCCCC(C(=O)N1CCCC(CO)CC1)NC(c1cc(=N)[nH][nH]1)=O CN=c1[nH]c(=NCCC2CCCCO2)[nH]c(=NCCC2OCCC2C)[nH]1 c1(C(=O)NCc2cn(CC(COC)COCC(=O)O)nn2)cnn2cccnc12 c1(C(N2CCC(F)(CNC(c3cc4sccc4[nH]3)=O)C2)=O)cn2cnnc2cn1 c1(C(=O)NCC2C(CNC(=O)C=Cc3cn[nH]c3)C2)ncc2n1CCCC2 C(=O)(CCCCCC#N)NC(C(C)NC(c1cc(C)nc(C)n1)=O)CO Cc1nc(CO)sc1C(=O)NCCCCCC1CCN(C(=O)CC#N)CC1 C1(C(=O)NCCn2c(C)cc(C)n2)CC12CCN(Cc1cncc(Br)c1)C2 N1(C(C2(C#C)CC2)=O)CCCC(C(N2CCN(C(=O)C(C)(C)N(C)C)CC2)=O)C1 N1(C(C(C=C)OC)=O)CCCC(C2CN(C(c3cnc4scnc4c3)=O)C2)C1 S(=O)(=O)(c1ccc(-c2ccc(C(F)(F)F)cc2)o1)NCc1c(C)ccs1 C12(C(=O)NC(CC)C(C)NC(=O)COc3cccc(Cl)c3)CCN(CC1)CC2 c1(N2CC3C(CNC(C4CC(CC)(CC)C4)=O)C3C2)ncnc2cc(Br)ccc12 N1CCC2(CO)CN(C(c3cnccc3Cl)=O)CC2C1.CCC(CC)CC=O C=C(Cl)CCC(=O)N(CCN1CCCC1)CC.C12(CC(CO)C1)C(=O)N2 c1(OC)ccc(C)c(C(=O)NC(C)(CNC(=O)C(C2CC2)C2CC2)C2CCC2)c1 c1(C(N2C(CC)C(C(N3CC(C(C)OC)C3)=O)CC2)=O)cccc2occc12 CCCCC(CC)CC(=O)NC1CCCN(C(=O)CSCc2ccccn2)CC1 C1(CNC(=O)C(F)n2ccnc2)CN(C(=O)C(F)(F)Cc2ccccc2)CCO1 c1(C(=O)NC2C(CNC(c3nc(CCCC)sc3)=O)C2)cc(CC)oc1C C12(C(=O)OCC)C(NC(=O)CC3CCOC3)C3CC1C2C3.C12(CC1)C(=O)N2 C(N=c1nc(N2CCCC(C)C2)c2sccc2[nH]1)c1cccc(OC)n1 c1(C(N(CCN(C)C)C)=O)ccccc1CN1CC2CC2C1 CCCC(C)(O)C(=O)NCCCOCCOCCNC(=O)CSc1cnn(C)c1 C(C(F)(F)CCC(=O)NC1CCCN1)n1cc(C(C)N(C(N)=O)C)nn1 C1(NC(c2nccs2)=O)CCCC2CN(C(c3cnn(C4CCCC4)c3)=O)CC12 Cc1c(Br)cc(C(=O)NC2CCN(C(C3OCCOC3(C)C)=O)C2)c(=O)n1C CCCCCCN1CCC(CC(=O)OCC)C1.N12CCCC1C(=O)NCC2 C(=O)(CCOC1CCCC1)N(CCN(C(C)C)C(C1(C)COC1)=O)C N1(C(C(C)=O)=O)CCCC(CCNC(C2CCCSC2)=O)C1 C(=O)(CS(=O)C(F)(F)F)NCCC1CCN(C(C2C(CC)N(C)CC2)=O)CC1 c1(CCC)ccc(CC(=O)N(C2CC(CF)C2)C)cc1.C12CCN(C1)C2=O N1(C(c2n(CC)ncc2Cl)=O)CCCC(O)(CNC(=O)C(O)CSC)C1 N1(C(C=C(C)C(F)F)=O)CCC12CN(C(C1CNC(=O)N1)=O)C2.C1(C23C(C2)C3)CCCCC1 N1(C(C2(CC)CN(C(=O)CN(C)C(C)C)C2)=O)CC2(CCOC(=O)N2)C1 C(CCC(=O)NCC(C)(C)OCC(=O)NC1(O)CCSC1)OCCC C1(C(N(CCCCNC(Cc2cc(C)no2)=O)C)=O)CCCC(C(C)C)C1 N1(C(CNC(=O)OC)=O)CCC(C(=O)NC(C2OCCC2(C)C)C)(CO)C1 c1(C(N2CCC23CN(C(c2cscn2)=O)C3)=O)cnc(Cl)cc1Cl c1(C(N2CC(NC(c3cc(C)n(C)n3)=O)C(F)C2)=O)ccc2c(n1)NC(=O)CC2 Cc1ccc2ncc(C(N3CCC4CN(C(c5cnn(C)n5)=O)CCC34)=O)n2c1 N1(C(=O)C(F)OC(F)(F)F)CC2(C(=O)NCC3CCCSC3)CC1CO2 c1(C(=O)NC2CCC(NC(=O)CSc3ccccc3Cl)C2)cccc2nncn12 CCC(CC)CCC(=O)NC1CCC1NC(C1(Br)CC1)=O Cc1ccc(C(=O)NCC2CCCCC2NC(C2OCCCO2)=O)c(Br)c1 c1(C(=O)NCC(O)CCNC(C2CCC=CCCC2)=O)ccc2cnccc2c1 C(=O)(CCC(=O)N(C)CCN(C)C(c1c[nH]nc1Cc1ccccc1)=O)N(C)C c1(CC(=O)NC(C)CN(C(=O)C=CBr)C)cc(C(F)(F)F)n(C)n1 N1(C(c2ccc(OCC#C)cc2)=O)CCC(N(C)C(c2ccsc2)=O)C(C)C1 N1(C(CC2(C(=O)OCC)CCC2)=O)CCCC(N(C(=O)C=CI)C)C1 C(=O)(CC(C(F)F)n1cccn1)NCC(C)(C)CC1CN(C(=O)C#CC(C)(C)O)C1 C1(C(N2CC(OC)(CNC(=O)C(C)CC(F)F)C2)=O)CC2CCC(C1)C2O c1(C(N2CCCC(C)(CNC(c3c(SC)n(C)nc3)=O)C2)=O)cc2n(n1)CCO2 C1(NC(c2c(OC)c(Cl)ccc2)=O)CCC2(C1)CN(Cc1ccc(I)c(Cl)c1)C2 C=CCCCCCCCCC(=O)NC(CNC(C1CCCN1N=O)=O)CCCC c1(NS(C)(=O)=O)cc(C(=O)Cc2cccc(NC(C(CC)C)=O)c2)ncc1Br N1(C(C(C)CC2CCCO2)=O)CCN(C(c2cnc(C(C)(C)C)[nH]2)=O)CC1 c1(NC(C2(C)CCN2C(c2cc(Cl)c(F)cc2F)=O)=O)cnc2ccc(Br)cc2n1 N1(C(c2cnc(Cl)c(Br)c2)=O)CCN(Cc2ccc(OC(F)(F)F)cc2)C2CC12 c1(C(C)=O)cc(C(=O)N(CC(C)(C)NC(=O)CC2CC2(Cl)Cl)C)co1 N1(C(C2CCC(C(C)C)CC2)=O)C2CCC1CN(C(C13CC(CO)(C1)C3)=O)CC2 C1(C(=O)NCC2CC(F)(CNC(CCC=CCC=C)=O)C2)COCCN1C C(=O)(C(CCC)OC)NC(C1CC(NC(COCCCC#C)=O)C1)C CC(CC(C)(C)C#N)NC(c1c(C(F)(F)F)cccc1F)C C1(CC)CCCC1(C)C(=O)NCC(=O)NCC1COCCO1 N1(C(=O)OCC)CCC(C(N2CCC(CNC(C3(F)CC=CCC3)=O)C2)=O)CC1 c1(C(=O)NC(CNC(c2ncncc2F)=O)CO)c(F)cccc1Br c1(C(=O)NC(CNC(Cc2cc(COC)on2)=O)C2CC2)cccc2nn[nH]c12 c1(-c2onc(C(N3CC(CN(C(C4CC(SC)C4)=O)C)C3)=O)n2)cccc(F)c1 C1(O)(CNC(C2CSCN2CCF)=O)CN(C(=O)C(F)=CCCF)C1 N1(CC)CCOC(C(=O)N(CC(CO)(CO)NC(C2CC(=O)CCO2)=O)C)C1 C1(NC(c2c(C)oc(CNC(=O)C(C)CC3CCCC3)n2)=O)CCCCC1(C)C C1(CN(C(c2cnc(C3CC3)o2)=O)CC)CCCC12CC2 N1(C(C2(NC(CCCN(C(C)C)C)=O)CCOCC2)=O)CCOC2CCOCC12 FCCN=C(NCc1ccc2c(c1)CCC2)NC1CCCC2(CC2)C1 c1(OC)cccc(C(C)C(C)SC)c1.c1(S)ccccc1OC Cc1cc(C(=O)NC2(CCCNC(C34CCC(C3)OC4)=O)CC2)nc(C)c1 c1(CNC(c2ccc(-c3ccc(CC)cc3)o2)=O)ccc2ncccc2c1 c1(NC(C(CC(C)C)ONC(C2COCC(C)O2)=O)=O)cccc2ccncc12 C12(C(N3CCC(COC)(CNC(c4ccnnc4)=O)C3)=O)CCC(C)(CC1)OC2 C1(N(C(CC(C=C)C)=O)C)CCC2CN(C(=O)C(O)CC(N)=O)CC12 c12ccc(nc1)NC1C(CC1)CNC2=O.c1(C(=O)OC)cnc(CC(C)C=O)[nH]1 CCCC(C(=O)N(C1CCC(Cc2nc(C(=O)OC)no2)CC1)C)n1cccc1 c1(C(=O)NCCCCN(C(CC(=C)C)=O)C)c(S(C)(=O)=O)cnn1C C1(CNC(C2CC2Cc2ccccc2)=O)CN(C(=O)CC2(C)CC2)CCO1 CCC(F)(F)CC(=O)NC1CCN(CC(=O)Nc2ccns2)CC1O c1(CCC)cc(C(=O)NCC2(CNC(=O)CCC(C)N(C)C)CC2)cc(O)n1 N1(C(CN(C(CSCC=C)=O)C2CC2)=O)CC(F)(F)C(F)(F)C1 c1(CN2CCCC(C(N3CCS(=O)(=O)CC3)=O)CC2)cc2c(s1)CCCCC2 C(C(C)CC(=O)NC1CN(C(=O)Cc2cncn2C2CC2)C1)OC C(=O)(C(F)C(C)(F)F)N1CCCC(C(C(=O)NCCc2cn(CC)nn2)(C)C)C1 N1(C(C2OCCN(C)C2)=O)CCC(C)(C)C1CC(=O)NOCC1(F)CCC1 N1(CC(=O)NC(C2CCCN2C(=O)CSc2ccc(Cl)nc2)C)CC(=O)NC1=O N1(C(C2(CC)CCOCC2)=O)CCC2(CC(NC(c3sc(C)c(C)c3C)=O)C2)C1 CCCCC(C)CCC(=O)N1CC2CC1CN(C(c1cnn(C(F)(F)F)c1)=O)C2 C1(NC(C(C)N(C)C)=O)C(C)CCN(C(c2cc3ncccc3[nH]2)=O)C1C c1(OC)cc(OC)cc(C(N2CC(NC(c3nocc3Br)=O)C(C)C2)=O)c1 c1(NC(C2CN(Cc3sc(Cl)nc3Cl)CC2O)=O)cc(Cl)cnc1O N1(C(c2c(C)nsc2)=O)CCC(CO)(NC(=O)C(c2ccc(Br)s2)=O)CC1 N1(C(C2(F)CCN(C(CN(CCOC)C)=O)C2)=O)CC2CCCC(C1)N2C c1(N2CC=CC(OCC)C2)nc(C)nc2n[nH]cc12.N12CCC1C2=O C#Cc1ccc(C(=O)NCC(C(C)(C)C)NC(C2(CC)CC2)=O)o1 C1(NC(=O)NC(C(=O)O)C2CCCC2)CC(=O)N(c2cccc(C(F)(F)F)c2)C1 C(=O)(CCCCCCCC(=O)N(CCCNC(=O)CC1(C)CCCCC1)C)OC C(=O)(C#CC1(C)CCCO1)NC1(C)CN(C(=O)C=CCOc2ccncc2)C1 C(=O)(C(=O)C=Cc1cccs1)NCC1(CN(C)C(c2ccnn2C)=O)CC1 C1(C(N(CC=C)CC=C)=O)CCC(n2cc(C3CCN(C)C3)nn2)C1 c1(NC(C(=O)N(CCNC(C2C(C)C2C)=O)CC2CC2)=O)ccccc1 C1(COC)CN(C(c2cc(C)c(C)[nH]2)=O)CCN1C(C1CC(=O)N(OC)C1)=O CC1CC(C(N2CC(C)(NC(c3cn(C)c(=O)cn3)=O)C2)=O)CC(C)C1 C#Cc1cncc(C(=O)NC2CC3CC(NC(c4cnn(CCOC)c4)=O)C3C2)c1 c1(C(N2CCC(CC=C)(NC(c3nsnc3O)=O)C2)=O)cnn2c1CC(F)(F)C2 N#Cc1cc(NC(C2CC23CCN(Cc2cn[nH]c2)C3)=O)ccc1O c1(C(=O)NCC(CO)NC(CC(CCC)CCC)=O)c(C)ccc2ncccc12 C1(C(N(CCN(C(C)=O)C)C(C)C)=O)Cc2cc(C)ccc2O1.C1C(=O)N1 c1(C(N2CC(CC(=O)NCCC(C)CO)OCC2)=O)ccc(C#N)cn1 CCC(CC(=O)NCCc1ocnc1CNC(=O)C=Cc1c[nH]nc1C)C1CC1 O=C(CCc1ncnc2ccccc12)N1CCCc2nccn21 C1(CC(N2CC(OCC(=O)NCC)C2)=O)CN(C(c2conc2CC)=O)CC12CC2 c1(CNC2CC(CN)C2)ccc(S(=O)(=O)NC2(CO)CCSCC2)c(Cl)c1 C(=O)(CC(C)(C)C(=O)NCc1ccoc1C(N1CC2COC(=O)C2C1)=O)OCC c1(C(=O)NCCN(C(=O)Cn2ncn(C)c2=O)C)ccc(=O)n(C2CC2)c1 N=c1[nH]c2ncc(C(=O)NCC#CCNC(c3ccc4sccc4c3)=O)cc2s1 Cc1ccc(OCC(=O)OCC(=O)NCC(C2CCOC2)F)c(F)c1 N1(C(c2cn(CC=C)nn2)=O)CCC(NC(=O)C(C)(C)CC)C(O)C1 C1(N(C(C(CC)N(CC)CC)=O)CC)C2CC3CN(C(=O)C(C)=C(C)C)C1C3C2 CC1(C)CC2(CN(C(C3CN(C(C4CCC4(F)F)=O)C(C)(C)C3)=O)C2)C1 S(=O)(=O)(c1ccc(NC2C=CCCC2)cc1Br)N1CCCC(C)(CCC)C1 Cc1c(CC(=O)NCCNC(C2CC3CCC2CC3)=O)nc(Br)n1C Cc1nc2cccc(C(N3CCCCC(NC(=O)C(C)C(C)O)C3)=O)n2n1 c1(NC2C(CC)CC2)cc(Br)ccc1S(=O)(=O)N1CCN2CCOCC2C1 C1(NC(C=CC)=O)CCC12CCN(C(c1c(F)ccc(Br)c1F)=O)CC2 c1(C(=O)NCCNC(C23C(CN(C(=O)OC(C)(C)C)C2)C3)=O)cc(Cl)ccc1I N#CCC(C(F)(F)F)NC(=O)CC1CCCN(C(=O)NC=O)C1 c1(C(=O)NCCN(C(=O)Cc2cccnc2Br)CC)c[nH]c2cc(C)ccc12 N1(C(C(C)=C(C)C)=O)CCC2(CC1)C(NC(=O)CC(C)(C)O)CS2(=O)=O CC1CN(C(C2CN(C)CC(C)O2)=O)CC1(C)C(=O)NCc1cnns1 Cc1cnc(CNC2CCCCC2C(=O)Nc2ncc(Br)cc2C(F)F)cc1Br N1(C(C(CC)(F)F)=O)CCC(CNC(=O)Cc2ccc(C)o2)C(C)C1 N(C(=NCCCCc1ccccc1)NC(c1cnn(C)c1)C)C1CN(C(C)=O)C1 c1(C(=O)NC2C(F)CCN(C(C3C(C(C)(C)C)C3)=O)C2)cnnc2ccccc12 Nc1cccn(CC(=O)N(c2cccc(F)c2)C2CCC2)c1=O Cc1[nH]cc(C(=O)NC2CC(F)(F)CC2NC(=O)C(N)=O)c(=O)c1Cl c1ccc(Br)cc1.C1CCON(C)N1C.C(C)(C)(C)OC=O N1(C(C(C)(C)C#N)=O)CC(C2CCCCN(C(c3ccc4sncc4c3)=O)C2)C1 c1(-c2onc(COC)n2)cc(C)ccc1OCC(N1CCC(NC(C)=O)C1)=O c1(C(N(CCNC(=O)C(C)(O)C2CC2)CC)=O)snnc1C(C)C c1(C(N2C(C)(CCC(=O)NCCCC(=C)C)CCC2)=O)cc(C)ncc1C C1(c2ccc(C)o2)CN(C(CCC2(C#N)CC2)C(=O)Nc2ccccc2)CCO1 C#CCCN=C(NC(C1CC1CSCC)=O)N.C1(N(C)CC2CCCC2)CCCCC1 CCC(C)C(CNC(c1ccn(CCNC(C2CNC(=O)O2)=O)c1)=O)CO c1(OC)cc(CCC(N2CC(O)(C(C)(C)CNC(C3CCS3(=O)=O)=O)C2)=O)on1 c1(C(N(C2CC(NC(Cc3c(C)ncs3)=O)C2)C)=O)cnc(C(C)C)nc1 N1(C(COc2ccc(OCC(=O)NC)cc2)=O)CCN(C(=O)CSC)C(C)C1C c1(SC)cn(C)nc1C(=O)NC1CCC(CCNC(=O)CSc2nc[nH]n2)C1 C1(O)(C(=O)Nc2c(C(=O)OC)scc2)CCN(C(=O)CCOC(C)CC(C)C)C1 c1(CCC(=O)NC(C)CC2CN(C(=O)CCC3CC3(Cl)Cl)C2)cn(C)cn1 c1(C(N2C(CCNC(C(C)SC(C)C)=O)CSCC2)=O)cc2cn[nH]c2cn1 c1(OC)cccc(C(=O)NCC(C)(C)CC2CN(C(C34CCC(C3)C4)=O)C2)c1N C=CCC(C(=O)N1CC(=C(F)CNC(c2cnc(C(C)(C)C)[nH]2)=O)C1)OC C1(CCNC(C2CC2n2cc(C(=O)OC)nn2)=O)COCCN1CC(F)F Cc1cc(C(=O)NCc2n[nH]cc2C(=O)NC(C)CCC2CCCC2)ncc1N CC(C)CC(C)CC(=O)NC1C2CC1N(C(=O)CCc1ccc(Cl)s1)C2C c1(CN=C(NC(CC)C)NC2CCC(NC(N)=O)CC2)ccc(C)c(F)c1 C1(NC(COCC(=C)C)=O)COCC1CNC(=O)COCC1CCCOC1 N1(CC)CCOCC1C(=O)NCCn1cc(C(=O)NCC(O)C2CCC2)cn1 Cc1cccc(O)c1C(N1CC2(CCC2NC(c2cnn(C)c2)=O)C1)=O c1(C(=O)NCC(=O)COc2ccccc2Cl)cncc2n[nH]cc12 c1(C(=O)NC)ccc(C(=O)NCCCCCNC(=O)C(C2(O)CCCC2)F)cn1 n1(CC(=O)NC(CCNC(C(C(CC)O)(C)C)=O)C)ccc(=O)c([N+](=O)[O-])c1 c1(OC)ccc(NC(=O)Cc2ccccc2NC(C)=O)cc1S(N)(=O)=O N1(C(C2C(C)OCC2)=O)CC(F)CC1CN(C)C(C12CC(C1)C2)=O C1(NC(C2CC(CC)(CC)C2)=O)CCN(C(=O)C=Cc2nc(C)c(C)[nH]2)CC1C c1(C(N(CCCNC(=O)COC2CCOC2)C)=O)sccc1SC(F)F C=CC(C)(O)C(=O)N(C(C)CN(C(=O)CN(c1ccncc1)C)C)C C(=O)(CC(CNC=O)CC(C)C)NC(CCC)C(=O)NC1CCCN(CCC)C1 C1(F)(CNC(=O)CS(=O)(=O)Cc2cccs2)COCCN(C(=O)CC(F)(F)F)C1 N1(CCN(CC(CN(C(CN(CC(O)CC)C)=O)C)O)C)CCOCC1 N1(C(C(C)NC(=O)NC)=O)CC2CC1CN(C(C1CN3CCN1CC3)=O)C2 N1(C(=O)CC2(O)CCCCC2)CC(C2CCN(C(=O)CC3(C(F)F)CC3)CC2)C1 C1(CCNC(CC(C)c2ccncc2)=O)CN(C(=O)C(C)(C)F)CCS1(=O)=O N1(C(c2n(C(C)C)ncc2)=O)C(CNC(=O)CNC(N)=O)CC2COCC12 Cc1nn(C)cc1CC(=O)N(C)CC1CCCCN1C(c1ccc(F)s1)=O C1(C(N2CCOCC2CO)=O)CN(Cc2cccc(Cl)c2)CC12CC2 C1(CC)(NC(c2ncn(C)c2C)=O)CCCN(C(=O)CC2(O)CCCOC2)C1 CC(CC(=O)NCC1CCCCN1C(c1ccnc(C2CCC2)c1)=O)C(F)(F)F c1(OC)ccc(Cl)c(C(=O)NC2(C)CCN(C(=O)C(C(C)C)OC)CC2)c1F Cc1cnn2cc(C(N3CCCC4(NC(=O)CC5C=CCC5)CC4C3)=O)cnc12 C1(=O)N2CCC(O2)C1=O.N1(C(C2=CCN(C)C2)=O)CCOC(C)(C)C1CO C(CCS(C)(=O)=O)(C(=O)OCC(CCO)C(F)(F)F)NC(=O)OC(C)(C)C c1(OCC(=O)N(C(C)C)CCN(C(=O)CCC#N)C)ccc2c(c1)CCC(=O)N2 C(=O)(CCCC=O)N1CCC(C(C)CN(C(=O)C(C)CC2CC2)C)CC1.C(N)=O c1(CC(=O)NC2CCN(C(=O)CCCc3cnn[nH]3)C2)nccc2ccccc12 C1(OC)CC(CNC(=O)CCCC2CCCC2NC)N(C(=O)OC(C)(C)C)C1 N1(C(C2CC(CCC)C2)=O)CCC2(CC1)CCN(C(=O)C(=O)C(C)(C)C)CC2C C1(C(=O)NCc2ncc(C(N3CCCN(C(C)C)CC3)=O)cn2)(OC)CCC(C)C1 c1(C(C)C)cc(CN(C2CCN(CC3CC3)C2)C(C2(O)CCOC2)=O)on1 C1(NC(=O)NC2CCOC2)CCC2CC12.O=C1CN(C2CC2)C(=O)C2C1C2 N1(C(c2c(C)cn(C)c2)=O)CCC(C)C(NC(c2ccncc2Cl)=O)C1C c1(OC)nc(C(F)(F)F)c(C(=O)N(C2CCN(C(=O)OC(C)(C)C)C2)C)s1 C(CCCCC(=O)NCC1CCCN(C(=O)CC2CCNC(=O)C2)CC1)N(C)C N1(C(c2cnc(C)c(N)c2)=O)CCC(NC(c2cc(Cl)ncn2)=O)CC(C)(C)C1 Cc1cc2occ(CC(N3CC(O)(CN(C)C(C4CC4(F)Cl)=O)C3)=O)c2cc1C Cc1cc2ccccc2cc1C(=O)NC1CN(C(=O)C(C)c2ccon2)CC1C C(C)(CNC(=O)C(=Cc1ccccc1)C)(C(C)C)NC(CCCOC(C)=O)=O N1(C(CCC(=O)OCCC)=O)CCOCC(C)(CNC(=O)C(C)C2(O)CCC2)C1 N1(C(C(CNC(C(CC)C(=O)OC)=O)C)=O)CCc2cncnc2C1 Cc1cc(C(N)=O)sc1NC(=O)COC(C1C=CC1)=O N1(C(c2cc(C)ns2)=O)CC(NC(C2C(C)C2(F)F)=O)C(F)C1 c1(C(N2C3CC(NC(C(C)=C4CCC4)=O)C2CC3)=O)nnc2ccccc2n1 C1(N(CCCNC(C2CN(C(C)=O)C2)=O)C)CC2(C1)CC(F)C2.C(CN)O C1(CC(=O)NCCSCCC)CN(C(c2[nH]ccc2C2CC2)=O)CCC1C C(C)(CCC(=O)OC1CC1)NC(C(C1CCC1)OCC)=O.C1(C)(CC)C(=O)N1 C1(C(=O)OCC(=O)N(CC(F)F)C2CC2)CCCC1NC(=O)CC1CCCC1 C1(COC)(NC(=O)Cc2ncoc2C)CN(C(c2ccn(CCF)n2)=O)C1 C1(C(N2CCC(CCC(=O)NCC(c3cnn(C)c3)C)C2)=O)CCC(F)CC1 N1(C(c2c(OC)cncc2)=O)CCCN(CCNC(=O)C(F)C2CCC2)CC1 S(=O)(=O)(c1cc(F)c(C)cc1OC)NC(c1cccc(OCC)c1)C N1(C(C2CCN(CCC#C)CC2)=O)CCC(C)N(C(=O)Cc2cccnc2)CC1 O(NC(=O)C(C(C)O)NC(=O)CC1CC1COC)CC=C C(N=c1nc(NC2CCCC2O)c2c([nH]1)c(C)nn2C)C1CCN(CCC)C1 c1(C(=O)NC2CN(C(C(CC=C)C(C)C)=O)CC23CC3)cccc2c1CNC2=O C(=O)(CC(C(F)F)NC(C1CCCC1OC)=O)N(CCCF)CC C1(CC=C)(NC(C2CCCC2O)=O)CCCN(C(C2CCC3(C2)N=N3)=O)C1 C(=O)(CCCCCN(C)C)NCCC(CCNC(c1cncc(SCC)n1)=O)C c1(C(=O)NC(CCCCNC(CCC=C=C)=O)C)ccn(CC)c(=O)c1 C1(OCC(NNC(COC)=O)=O)CCc2ccccc2NC1=O c1(C(=O)NCC2CCCN(C(C(C(C=C)C)C)=O)CC2)cc(N(C)C)cc(C#N)c1 C1(CNC(c2c(CC)[nH]c(=N)s2)=O)CN(C(c2cncnc2)=O)C2CCCC2O1 c1(C(=O)NC2CCC(N(C(=O)COC3CC=CC3)C)C2)cnc2c(F)cccn12 c1(C(=O)NC2(C)CS(=O)(=O)C2)ccc(CNC(CC2CC(OCC)C2)=O)cc1 c1(CC(=O)CNC(c2cnc(-c3ccncc3F)cn2)=O)ccccc1F CCCC(C#N)C(=O)NC1CCCCCC1F.C12CC(C1)C(=O)NOC2 C(CC(=O)NC)NC(C)C.C(C(C)(C)C)=CCN(C(COCC#C)=O)C C12C3CC3CN1C(=O)C=CC(C)(C)NC2=O.C1(SC)CCCCCC1 c1(CC)oc2ccccc2c1CC(=O)NCC1CCN(C(=O)C=CSC)CC1C c1(CC(=O)NC2C(NC(C(C3CC3)SC)=O)COCC2)cc(C)cc(F)c1 N1(C(CC2CC(=C)C2)=O)CC(NC(=O)C(=O)NCC(F)F)CC1C c1(C(C)=O)cnc(N2CCC(O)C(C(=O)NN3CC(C)C(O)C3)C2)nc1C c1(C(N(CC(N2CCCC3(C2)N=N3)=O)CCOC)=O)n[nH]c2ccccc12 C12(CNC(CCSCCCC)=O)CC(NC(c3cc(CC)ccn3)=O)(C1)C(C)O2 C1(C(N2CCC(CNC(=O)C(c3cccn3C)=O)C2)=O)(NC(C)=O)CC(F)(F)C1 CC(C)C(C)(CN=c1[nH]cc2ccnc-2[nH]1)NC(c1cncc2sccc12)=O c1(C(=O)N(CC(CCOC)NC(CC(=C=C)C)=O)CC)c(C)[nH]c(C2CC2)nc1=O Cc1cnc(C)c(C(=O)NCCC2CN(C(=O)CCOCC(C)C)CCC2C)c1 C1(C(N2C(CNC(C(C)=C3CCCC3)=O)CC(O)C2)=O)CC12CCSCC2 Cc1n[nH]c(C)c1CC(=O)NC1(CNC(C2CC23CC3)=O)CCOC1 C1(CCCCNC(c2c(C)n[nH]c2)=O)CCCN(C(C2CCNC2=O)=O)C1 c1(C(=O)NC(CCOC)CNC(c2c(C)n[nH]c2C)=O)cnc2cc[nH]c2c1 Cc1ccc(F)cc1CC(N1CC(Nc2cccc(F)c2)C1)=O C(CC(=O)NCCC1CCC(C)(C)CO1)(C(N)=O)NC(C)=O c1(C(N2CCCC(CNC(C3C4CC(=O)CC43)=O)C2)=O)occ2c1CCCC2 CN1C(=O)NCC12CN(C(C1CN(C(C3(C)COCCO3)=O)CC13CCC3)=O)C2 C(=O)(CCCC(=O)NCC(O)CCNC(c1cc(Cl)ccc1OC)=O)NC C1(NC(=O)Cc2cc[nH]c2)CCOC12CCN(C(c1cncn1C)=O)CC2 C1(CNC(C(CC)OC)=O)Cc2ccccc2CN1C(c1cn(C(C)C)nn1)=O c1(C(N(C(CNC(C2CCOCC2)=O)C2CC2)C)=O)ccc(C2CCC2)o1 C1(CC)CN(C(=O)C=CCN(C)CC)CCC1CNC(C1CCCC1O)=O C1(NC(c2c(Cl)cn(C)n2)=O)CN(C(C2CC(F)(F)C2)=O)CCC1CO C(=O)(C(C(C)(C)C)NC(=O)C=CC1CCN(C(c2ccc(F)s2)=O)CC1)NC C#Cc1cnc(C(=O)NC(C)(CNC(=O)CCc2nncn2C)CC)c(C)c1 N1(C(C(CCSC)NC(c2cocc2C)=O)=O)CCCC2(C1)N=N2 Cc1noc(C)c1C(C)(C)C(=O)OCCn1ccnc1-c1nccs1 CC1(C)NC(=O)CC1C(=O)NC1COCC1NC(C1(C2CCCO2)CCC1)=O c1(NC(C2CN(C(C(F)=CCC)=O)CC2F)=O)ccc2ccncc2c1 c1(C(N(C2CN(C(=O)C(C)(C)OCC(F)(F)F)C2)CCOC)=O)nc(C)oc1C N1(C(CCCCNC(C)=O)=O)CCCC(NC(C2CCC(=O)NC2)=O)C1C N1(C(CNC(=O)OC(C)(C)C)=O)CCC2(CC1)CN(C(=O)CCF)C1COCC21 n1(CCCC)ccc(C(=O)NC2(CNC(=O)CC(C)SC)CC2)n1 c1(C(N2C3(CNC(C(C)C(C)N(C)C)=O)CC(C2)C3)=O)cc(S(N)(=O)=O)ccn1 c1(N2CCCC(CCC)CC2)nc2ccc(Cl)cc2c(=NCCCOCCO)[nH]1 C(=O)(C1=C(c2ccccc2)CCC1)NC1C(NC(C(CC)(C)OC)=O)CCOC1 C1(NC(CCC=C(C)C)=O)CC(C(=O)NCC(F)(F)C(C)C)C1(C)C N1(c2nc(SC)nc(C)c2)CC2CC(NC(c3ncc(Cl)s3)=O)CC2C1 C12(NC(CNS(NC)(=O)=O)=O)CCOCC1CN(C(c1sccc1C(F)F)=O)C2 N1(C(C(CCC)F)=O)CCC(C=CC(N2CCC(C(C)(C)O)C2)=O)CC1 O(NC(=O)CC(C(C)CC)NC(C12C=CC(CC1)C2)=O)CCCC Cc1nc2ncnn2cc1C(=O)NCCC(C)NC(c1ncc2ccccn12)=O c1(C(N(C2CC3CC2CN3)CCS(=O)(=O)N(C)C)=O)ccc(C)nc1Cl c1(NC(NOCCSCc2ccc(C)cc2)=O)ccc2ncnn2c1 N(C(=NCCCc1ccccn1)NCCC1CCOC1)C1CCCN(CC)C1 C(C)(C)(CCCC(=O)N1CCC(F)(F)CC1C)NC(c1nncc(OC)c1)=O CCCS(=O)(=O)CC(=O)NC1CCN(C(=O)Cc2occc2C(=O)OC)C12CCC2 c1(C(C)NC(CC(C)NC(C2N(CC)CCC2)=O)=O)ccc(F)cc1 n1(C(CC)C)nnnc1C1c2nc(cs2)CC2(CC2)CCN1.C1(C)CC1.C1(OC)CC1 C(=O)(C(O)CC(F)(F)F)NC1C(SC)CN(C(c2ccnnc2)=O)C1 C1(N(C(C(CC)F)=O)CC)CCN(C(c2cc(C3CC3C)on2)=O)CC1 C1(CC#C)(C(=O)NCC2CN(C(=O)C=Cc3sccc3C)CCO2)CCCCO1 c1(CCn2c(C(c3noc(=O)n3C)NCCC)nnn2)ccnc(CC2CCCO2)c1 C=CCC(C)(O)C(=O)NCC1CCC(NC(C2CCC3CC23)=O)C1 c1(C(C(=O)NCC2CC(NC(c3nc(OCC)oc3)=O)C2)(C)F)ccccc1F N1(C(Cc2nc(C)oc2)=O)CC(NC(C2CC3(CCO2)CC3)=O)C2(CC2)C1 C1(CCC)CCC(CN(c2cc(O)ncn2)CCN(C)C)CC1 C(=O)(C1CCCc2c1nnn2C)NC(CC(C)NC(c1c(SC)cccc1)=O)C N1(C(C2(NC(=O)NC)CCC2)=O)CCC(CNC(C2CCCCN2C)=O)CC1 c1(NC2N(C(CC)=O)CCC2)[nH]c(=NC2CC2CCOC)nc2c1ncn2CC C(=O)(C1=C(F)CN(C(=O)CC(C)(F)F)CC1)NCC(C#C)CC C1(CNC(Cc2n(C)ccc2)=O)CCN(C(C2(CCO)CC2)=O)CCC1(F)F c1(N2CC(CNC(N3CC(C)C=C(C)C3)=O)C2)ccc([N+](=O)[O-])cc1 O=C(C(=O)N=c1cc(C2CC2)n(C)[nH]1)Sc1ccccc1C1COC1 CCC(C)(C)C(O)C(=O)NCCC(O)CNC(=O)CC1CC2(CCC2)C1 N1(C(c2ncn(CC)n2)=O)CC(N(C)C(C2CCCC(OC)C2)=O)C2(CC2)C1 C(C(O)CC(C)(C)C)NC(C(CC)O)C c1(C(=O)NCC2(O)CC(NC(CC(CC)C3CC3)=O)C2)cnc2cnccc2c1 c1(C(=O)NC2CCCN(C(c3c(Cl)ncc(N)c3)=O)C2)ccc(O)c([N+](=O)[O-])c1 Cc1nn(C)c(C)c1C(=O)NCC1(CC(N2CCCC(C#N)C2)=O)CC1 O=C(CC(C(F)(F)F)NC(c1ncccc1Cl)=O)NCC1C=CCC1 N1(C(C(C=C)O)=O)CCC(NC(=O)NCc2cccc(OC(F)F)n2)C(F)C1 CC1C(NC(C2(CCSc3ccccc3)CC2)=O)CCN1C(C1CSCCS1)=O C(=O)(C1=CCc2ccccc21)NCC(C)(C(C)C)NC(CCOCCOC)=O CCCCC(CO)NC(=O)CCN(C(=O)CC1CCC(=O)C1)C1CC1 c1(C(N(C)CC2N(C(C(C)(C)OC(C)=O)=O)CCC2)=O)ccc2[nH]ccc2n1 N1(C(C(C)(C)OCC=C)=O)C2CCC1(C(=O)O)CC2.C(CC)O c1(C(N(C(CC)CO)C)=O)coc(CNC(=O)C(O)CNC(C)=O)c1 C1(C(N2CCC(CC)C2)=O)(CCC2CC2)CC2(CC2)C1.N1(CC=CC(=O)N)CCCC1 N1(C(CCSCC(C)C)=O)CCC(C)(NC(C2CCC2(F)F)=O)C1 c1(C2(C(=O)Nc3ccc(CC)cn3)CC2)ccccc1C#N N1(C(C(C)CC(F)F)=O)CCC2C(CCN2C(c2cc(Cl)n(C)n2)=O)C1 Cc1cc2c(CC(=O)NCC(F)CNC(=O)Cn3cc(C(F)F)cn3)csc2s1 C1(N(CCO)OCC(=O)O)CCN(Cc2cc(C)[nH]n2)C1(C)C C(=O)(C1=NNC(=O)CC1)N1CC=C(CNC(C2(CS(C)(=O)=O)COC2)=O)CC1 CC(=O)CCN=C(NCC1=CCN(C)CC1)NCc1cnn(C)n1 C1(C(N2CCCC(NC(CCCOCCC)=O)(CO)C2)=O)CCOCC12CCC2 C(CCCC(C)(C)NC(c1ccnnc1)=O)NC(C(C)CC1CCC1)=O c1(C(=O)Oc2ccc([N+](=O)[O-])c(C(F)(F)F)c2)cnc2nc(Cl)ccc2c1 C(=O)(C(C#N)C1CC1)NC1CC(NC(C2(C(N(C)C)=O)CC2)=O)C1 c12ncccc1S(=O)(=O)N1CC(C3(CC3)C1)N2.C(C(C)C)SC C1(NC(C2CN3CCN2C(C)C3)=O)CN(C(=O)COc2ccsn2)CC12CCC2 c1(C(=O)NCCOCCN(C)C(c2csc(O)n2)=O)nccc2nn[nH]c12 C1(NC(=O)CCc2ncc[nH]2)CC2CCCC(C1)N2C(c1ncncc1Cl)=O C(=O)(CC(F)(F)Br)NCC(CC=C)NC(=O)CC(C)OCCOCC c1(C2C(C(N(CCC(C)NC(c3nnn(C)c3N)=O)C)=O)C2)ccc(F)c(F)c1 C1(NC(CC=CCC)=O)CCC2(CC1)CCN(C(c1cc(OC)n[nH]1)=O)CC2 N1(C(C=NOC)=O)CC=C(CNC(=O)CCc2csc(C)n2)CC1 c1(C(N(CC(C)NC(c2ccc3nc[nH]c3c2)=O)C)=O)n[nH]c2c1CN(C)CC2 C1(C)(NC(c2c(CC)noc2)=O)CCN(C(=O)CSc2ccc(C)cc2)C1 c1(C(=O)NC(C(C(C)C)NC(C2CS(=O)(=O)C2)=O)C2CCC2)ncc(F)cc1F C1(C(=O)NCC2(NC(=O)C3=NOC(C(C)(C)C)C3)CCC2)CCC12CCOCC2 c1(C(=O)NC2CC(F)(CNC(CCOCCN(C)C)=O)C2)c(F)cccc1F N1(C(C(C)SC)=O)CC(F)CC1CNC(=O)C=C(Cl)Cl c1(NC(c2c(C)[nH]c(C)c2C)=O)ccc2c(c1)CCC2.C12CCC1CNC2=O c1(C(N(C)CC2(C)C(NC(c3c(C#C)c[nH]n3)=O)CCC2)=O)cc(C)nc(O)n1 c1(C(N2C(C)C(NC(=O)CN(C)C)CCC2)=O)ccn2cc(Br)cc2c1 C1(C(N(C)CCNC(c2cnsn2)=O)=O)CCC(c2nc[nH]n2)CC1 O=C(C1=NOCC1)NC1CN(C(c2cccc(C(F)(F)F)c2)=O)CC1O CC1CN(C)Cc2cccc(Br)c21.C12(C(=O)O)CCC(C(F)F)(CC1)CO2 C(C(C)CN=c1[nH]c(=NC2COC3(CCC3)C2)[nH]c2cc(C)ccc12)NC(=O)OC C12(C(N(CCC(=O)NC(=O)CCOCCC)CC#C)=O)CCCCC1C2 c1(C(N2C(C(C)NC(CC(C)C(F)(F)F)=O)CCC2)=O)cc(F)c(F)c(Cl)c1F C1(CNC(C(=O)NCC)=O)CCC(C(=O)N(C)CCC)CC1 C1(C(=O)NC(CC)C(=O)NO)CC(N=[N+]=[N-])CN1C(=O)CC1CC=CCN1C C#Cc1ccc(C(N2CCC=CC2C(=O)Nc2cnn(C(C)C)c2)=O)cc1 C1(C(=O)NCC2C(CNC(COc3cn(C)nc3)=O)C2)C(F)(F)C12CCC2 C=CC1(C(=O)NCc2c[nH]nc2C2CC2)CCN(C(c2cnc(N)cn2)=O)C1 C1(NCc2ccc(CC(C)C)cc2)CCS(=O)(=O)CC1 Cc1cc(C)c(C(=O)NC2CC2CNC(=O)C(C)Cc2ccco2)s1 N1(C(C(C)=C(CC)C)=O)CCC(C)(C)C1CNC(=O)Cc1nn(C)cc1Cl C12(C(=O)NCC(CC(C)C)NC(C(c3c(C)cccc3)C)=O)CCOC(C)(C1)C2 c1(C(=O)NCC(CC)NC(c2cc(C(C)=O)cs2)=O)oc(C(F)F)cc1C C(CC(C)C(=O)NCC1C(O)CN1C(c1csc(-c2cnc[nH]2)n1)=O)=CCC c1(C(N2C(CNC(=O)C(C)C)CC(OC)C2)=O)cccc2c1CCCCC2 c1(C(=O)NCC2CC3N(C(CC)=O)C(CC3)C2)ccc2c(c1)NC(=O)CNC2=O N1(C(CC(CC2CC2)NC(CCSCC)=O)=O)CCCC(C)CC1 N1(C(CCC=CC)=O)CC(NC(=O)Cc2cccc(C)c2Br)CC(C)C1 Cc1cc(C(N2CCC(C(C)NC(c3cscn3)=O)CC2)=O)cc(Br)c1C C1(C(N2CC(c3cccc(C)c3)C2)=O)CC(C)(C)CN1C(=O)OC(C)(C)C C1(NC(C2CC(C)(NC(Cc3cc(C)[nH]n3)=O)C2)=O)CC(CO)C12CCC2 CC(=O)CCCCC(=O)N1CC(C2CC2C(=O)NC(CO)CCC2CC2)C1 C#CC1CCC(C(N2CCC(NC(=O)C(c3ccc(Br)s3)C)C2)=O)CC1 c1(C(=O)NC2C(NC(COCP(C)(C)=O)=O)COCC2)cnc(O)c2ccccc12 Cc1cnn(C)c1S(=O)(=O)CCNC(=O)Cc1cc(C)n(-c2ccon2)c1C c1(CN(C(c2c(-c3c(C)cccc3F)cncc2)=O)CC)cc(Br)c(O)cc1O c1(C(N2CCC3(NC(C4(O)CCC4)=O)C(C2)C3)=O)cccc2scnc12 CC(C)C(CC(=O)N(C)CCNC(C1COC2(CCC2)C1)=O)C(C)C CCCC(CC)CCC(=O)N1CCCN(C(=O)Cc2ccc(O)nc2)C(CO)C1 C1(NC(C2CCN(C)C2)=O)COC2(C1)CN(CC1CCN(c3ccccc3)C1)C2 c1(CC(=O)NCC2CC(NC(C3C(C)OCC3)=O)C2)ccc(F)c(Br)c1 c1(N(C)CC2CCN(C(c3sccc3F)=O)CC2)nc(Cl)nc2s[nH]c12 C1(NC(C2(CCNC(CCCCC)=O)CC2)=O)CC2(C1)CC(CNC(C)=O)C2 Cn1c(O)ncc(C(N2CC(CNC(=O)CNC(c3cccs3)=O)C2)=O)c1=O C(=O)(C(CC)C(=O)N1CC(O)(CNC(=O)Cc2ccc(OC)c(F)c2)C1)OCC Cc1cc(C(=O)NC(CNC(c2cc(CCCO)on2)=O)C(C)(C)C)[nH]c1C n1(C(=O)N(CCO)C2CC2)ncn2nccc2c1=O CC1CCN(CC(N2CC(C(C)NC(=O)CNC(S(=O)(=O)C3CC3)=O)C2)=O)CC1 N1(C(C(n2cc(C(CC)O)nn2)C)=O)CCCC(NC(=O)CCCOC)C1 c1(OC)ccc2c(c1)CCN(N1CCN(c3cc(Cl)ccc3C)CC1)C2 c1(OC)cc(C(=O)N(CCNC(=O)C(=Cc2cccs2)C)C(C)C)cnc1OC C(C(C(=O)NCc1cn(C2CC2)cn1)NC(=O)CC1CC1)OC Cc1ccc(C(=O)N(CC(N)C(F)(F)F)Cc2ncc[nH]2)cc1 C(=O)(CS(=O)(=O)C(C)C)NC1CCN(C(Cc2ncc(C)s2)=O)C1(C)C C=CCC(C(=O)N1CC(C)C1C(=O)NC(C)C(C)C)OC C(=O)(C(C(C)(C)C)N(C)C)NCC(CNC(c1nn(C)c(F)c1)=O)(C)F CC1=C(C(=O)NCC2CC2CNC(c2ccc(O)c(C)c2)=O)CCCO1 C(=O)(C(CO)C(C)(C)C)NC(CCC)CCCNC(c1cc(C)c(Cl)s1)=O c1(NC(c2c(OC)ccs2)=O)nc(C)c(S(=O)(=O)N2CC3(CC3C(N)=O)C2)s1 c1(C(N(CCNC(=O)C(F)(F)C2CCCCC2)CC)=O)ccc2c(c1)C=CCC2 C(=O)(CCC#Cc1ccccc1)NC(C)CCN(C)C(c1ccccc1CO)=O CC(C)C(CCN(C)C(C1CC1(F)F)=O)NC(c1c(Cl)cnn1C1CCCC1)=O C1(C(=O)NC(C=C)(C)CC)CC=CCN1C(=O)CSC1CC1 N1(C(C(CC)n2cccn2)=O)CCCC(C)(NC(c2ccc(CO)s2)=O)C1 NS(=O)(=O)CCC(=O)NCCC1(C(=O)NCCC(F)(F)CO)CCC1 C1(=CC(=O)NCC(C)NC(=O)C2=NNC(C(F)(F)F)C2)CC2CCC(C1)N2C c1(C(C)=O)ccsc1C(=O)NC(CNC(=O)C(c1ccn(C)n1)C)C1CC1 c1(CC(=O)NCC2CCCN(C(C=CSC)=O)C2)cc2ccccc2c(=O)o1 C1(NC(C(COC)C)=O)CCSC12CN(C(=O)C=Cc1ccccc1OC(F)F)C2 c1(OC)nc(=NC(C)C2CCN(C(c3ccc(CO)o3)=O)CC2)[nH]c2[nH]cnc12 N1(C(CNC(CC(C)C)=O)=O)CC(F)CC1CN(C(=O)CC1CC2CC2C1)C CC1(NC(=O)C=CC(N2CCOCC2)=O)CCC(NC(C2CNC(=O)C2)=O)CC1 C1(C(N2CCC(NC(CCCCC#C)=O)C2C)=O)CCC2(CC1)CC(O)C2 c1(C(=O)Nc2ccncc2C2CC2)nc[nH]c2ncnc1-2.C1CCOCCN1C n1(CC(=O)NC(CCOCC)C)cc(CNC(=O)C(CCC2CCC2)OC)nn1 C1(NC(C2N(C(C(CC)(CC)OC)=O)CSC2)=O)CCCCC1N=[N+]=[N-] C1(NC(CCCC(CNC(COC2(C)CCC2)=O)CC)=O)CC2(C1)CC(C)(C)C2 C(=O)(CC(C)(C)C(=O)N1CCC(C)(CCNC(=O)C#CC2CC2)C1)OC C(N=c1[nH]c(C(C)C)ncc1C#N)C1CN(C(CN2C(CC)CCC2)=O)CC1C C(CCCC(=O)NC(C)(CO)C(F)F)N(C(CCSCCCC)=O)C1CC1 c1(CCNC(CCN(C(C(COCC)C)=O)C)=O)ccccc1F C12(C(=O)NCC3N(C(CCCC=C)=O)CC(C)(C)C3)CCCCN1CCC2 c1(C(N(C(C)C(=O)NCc2ccc(O)nn2)C)=O)ccnc2cc[nH]c12 N1(C(COCCC(C)C)=O)CCN(C(=O)C=CC2CCCO2)CC(C)(C)C1 C1(C(=O)NCC2(O)CC(NC(c3c(OC)n[nH]c3)=O)C2)CN=C2N=CNN2C1 N#Cc1ccc(CNC(c2scnc2-c2cc(C(=O)O)ccn2)=O)cn1 C(=O)(CS(=O)(=O)C1CC1)NCC(=O)Nc1c(OC)nccn1 c1(C(N(CCC(=O)N(C(C(=O)OCC)C)C)C2CC2)=O)cnc(N)cn1 c1(CC(=O)NCC(=O)NCC(CO)NC(=O)Cc2ccoc2)cc(F)cc(F)c1 c1(C(=O)NC(CNC(C2(COC)CC(=C)C2)=O)CC)cccc(C=C(F)F)c1 N1(C(C2CCC(C(=O)OC)C2)=O)CCN(C(C2CCCCCOC2)=O)C2(CCC2)C1 C1(C(=O)NC2(C(N3CC(CC=C)C3)=O)CC2)(CC2CC2)CCOC1 C(=O)(C#CC1CCCOC1)N1CCC(NC(c2cc(N)c(Cl)cn2)=O)CC1 N1(C(CCC(CC)OC)=O)CCCC12CCN(C(=O)C=Cc1cncc(C)c1)C2 C1(C(N)=O)CCC(N=c2[nH]c(=NCC3CC3C3CC3)[nH]c3c2CCCCC3)C1 N1(c2cc(C)nc(NCC(C)(F)F)n2)C(C)C2CCCCC2C1C N1(C(=O)CN2CCCS2(=O)=O)CC2C3CCC(C2C1)N(c1cc(F)ncn1)C3 C(C(=O)N1CC2C(CNC(=O)CN3CCOCC3)C2C1)(C(C)(C)C)SC C1(C)(C(N2CCC(NC(=O)NC)C2)=O)CN(C(=O)CC(O)C2CCCC2)C(C)(C)C1 c1(N2CCCC(C(=O)NC3(CO)CCC(C)C3)C2)ncc(Cl)c(O)n1 N1(C(C=CC)=O)CCn2c(CNC(C3(C)CNC(=O)C3)=O)nnc2C1 C(=O)(CCS(=O)(=O)C(F)(F)F)N1CCCC(C2CN(C(C(CC(C)C)C)=O)C2)C1 C1(C(=O)O)(NC(c2ccnc(OC(F)(F)C(F)F)c2)=O)CC(F)(F)C1 C1(C(CNC(c2cccn(CC(F)F)c2=O)=O)=O)Cc2ccccc2N1 N1(C(C2OCCN(CC)C2)=O)CC(NC(=O)COC(C)(C)C(F)(F)F)C(C2CC2)C1 C(C)(C)(CCCC(=O)N1CCC(CC(F)F)C1)NC(CC1N(C)CCC1)=O CN(CCCC(=O)NCC1(O)CCN(C(C2(C3CCC3)CC2(F)F)=O)C1)N=O N1(C(CNC(C(CC)C)=O)=O)CC2(CCN(C(=O)Cc3cccc(C)c3)CC2)C1 C1(CC=C)(C(=O)NCC(O)CC)CCCN1C(c1cnsc1)=O c1(C(N2CC(OC)C(NC(c3cnco3)=O)C2)=O)cc(N)ccc1C(F)(F)F C1(C(C(=O)NCC2(NC(CCC#N)=O)CCOC2)O)CCCCCCC1 C(=O)(C#CC1(C)CCCO1)N1CCC(C)CC1C(N1CCn2ncnc2C1)=O c1(C(N2CCCCCC(NC(C(CC)(C)C)=O)C2)=O)[nH]nc2c1CCCC2(C)C c1(C(C(=O)OCC)N(C(C)C(=O)NC(C)(C)CC)CCC)cccc(Cl)c1Br c1(C2C(=O)C(=O)C(C)(C)CN2C2CC2)cc(C)cc(Cl)c1.C1(CNOC)CCOC1 N1(C(CSC(C)(C)C)=O)CC2(C1)C(NC(C1CCS(=O)(=O)N1)=O)CCS2(=O)=O Cc1cc(F)ccc1CC(=O)NC1CC(C)N(C(C2CCC(C)C2)=O)C1 CC1(CNC(C23CSCC2C3)=O)CCCN(C(c2ccc(O)nc2)=O)C1 N1(c2n(C)ccn2)CCCN(C(=O)NC2CCC3(CCC3)C2)CC1 N1(C(c2ccc(NC)cc2)=O)CC2(CCC2NC(c2onc(C3CC3)c2C)=O)C1 Cc1ccc(C=CC(N2CCCCCC(NC(c3nc(Cl)cs3)=O)C2)=O)cc1Cl C(=O)(C1=C(C)OCCC1)N1C(CNC(CCCC#C)=O)C(C)CC1 c1(C(N2CCCCC(CN(C(C(CC(C)C)F)=O)C)C2)=O)ccc2occc2n1 CCCC(C)(O)CC(=O)NC1CN(C(c2cc(C(C)(C)C)n[nH]2)=O)CC1C C(=O)(CCCN(C)N=O)NC1(CCNC(c2c(OCC)cncc2)=O)CCC1 C1(C)(NC(C2(NC(c3c(CC)ocn3)=O)CC2)=O)CCCC1(C)C c1(C(N(C2CCCN(C(c3ccoc3C3CC3)=O)C2)C)=O)cnc(Cl)n1C N1(C(COCCC)=O)CCN(C2(CNC(=O)CCOCC)CC2)CC1 N1(CCC)CCC(C(=O)NC(C2CCOC2)C[N+](C(c2nc(Cl)cs2)=O)([O-])CC)CC1 C1(NC(c2cccc(NC(=O)NC)c2)=O)CN(C(c2cc[nH]n2)=O)CCC1(C)C C1(CC)CCC(C)CN1C(=O)CCCN(C(=O)Cc1cccn1C)C c1(C(=O)NC(CNC(Cc2cc(CC)nn2C)=O)C(C)C)cccc([N+](=O)[O-])c1 c1(C(=O)NCC2CN(C(c3c(CC)cccc3)=O)CC2C)nccc(Cl)c1Cl c1(C(=O)NC2CCN(C(=O)COCC3CCCO3)C2)c(Cl)cc(F)c(Cl)c1F C(=O)(CCC(C)(C)C(=O)N=S(C)(=O)CC1CCC(C(=O)OC)C1)OC C1(C)(C(=O)NCCCc2n(C)ccn2)CCCN(C(=O)C(F)n2ccnc2)C1 CCCCCCC(C)C(=O)N1CCCC1CN(C(=O)CCN(S(C)(=O)=O)C)CC N1(C(CN(CCC)C(c2cn[nH]c2)=O)=O)CCC(C)OC(C)C1 N1(C(C2CC(C)(CC)C2)=O)CC2(CCNC(=O)C(O)c3ccsc3)CCC1CC2 c1(NC2CC(NC(=O)C(N3CCCC4NCCC4C3)=O)C2)ccc2ccccc2c1 c1(C2C(OS(Cc3c(C#N)cccc3)(=O)=O)CO2)ccc2c(c1)OCCO2 Cc1cc(C)c(C(=O)N(C)CCN(C(=O)C(O)CC[S+](C)C)C(C)C)c(N)c1 C1(CC(=O)NCC(CC)(CC)OC)CC2(C1)CN(C(=O)Cc1ccn(C)c1)C2 n1(Cc2onc(C)n2)cc(C#CCNC(c2cc(Cl)cc(Br)c2F)=O)nn1 Cc1ccc(C(=O)NC2(C)CN(C(=O)Cc3ccc(C(=O)OC)cc3)C2)c(O)n1 c1(CC)ccc2occ(C(=O)NC3CCC(NC(=O)CCn4ccnn4)C3)c2c1 N1(C(CCCOC)=O)CC2CCC(C1CO)N2C(=O)C(C)Oc1ccccc1 c1(COC(CN(C)CC)OCC)cc(Cl)ccc1C c1(CNC(=O)CCC2CC2)nc(CNC(c2cc(Cl)cs2)=O)cs1 c1(NCCCc2cn(C)nc2)cc(F)cc(Cl)c1 c1(C(N2C3CN(Cc4cc(Br)cc(Br)c4F)CC23)=O)cc2n[nH]cc2cc1Cl C1(C(N2CCC(c3c(C)ncs3)CC2)=O)Cc2nccn2C1 C1(N(C)C(c2ccn(-c3ccccc3)n2)=O)CCC(NC(c2cc[nH]c2)=O)CC1 C1(C(N(C)CC2CCCN2C(c2cc[n+]([O-])cc2)=O)=O)C2CCCCC12 N1(C(C)C)CC(C)(C)OC2(CCOC2)C1.C12CCC(CC1)C(=O)N2.C1C(=O)N1 C(=O)(CC(C)(C)O)NCC1C(CNC(C=C(CCC)C)=O)C1 O=C1CN(C(=O)CN2CCOCC2)CCCN1.C12CCC(C1)N(CCO)C(=O)CC2 CC(C(C)(C)C(=O)NCC1CCCOC1)NC(C1COCCC1C)=O N1(C(COCCOC)=O)C2CCC(C(N3CC(C(N)=O)C(C)(C)C3)=O)C1CC2 C(c1ccc(OCC(N)=O)cc1)=CCOC(C)=O.CCCCC1CN1 C1(NC(c2n(COC)ncc2)=O)(CNC(c2scc(C)c2C)=O)CC2CCC1C2 C1(C(N2CC(OC3CCN(C(C#C)=O)CC3)C2)=O)C2CS(=O)(=O)CC12 N1(CC)CC2(CN(C(=O)C(C3CCC3)NC(=O)CC3CCCOC3)C2)C1 N1(C(CCCC(CC)C)=O)CCc2[nH]nc(CNC(=O)CCSCC(C)C)c2C1 CC(CC(F)F)C(=O)NCC(c1ccccc1F)NC(c1n[nH]cc1Br)=O c1(OC)c(C(=O)NC(CO)C(C)NC(=O)Cn2ncn(C)c2=O)cc(Cl)cc1Cl CN1CCC(C)(C(=O)OCC2(C(C)(C)C)CCN(C(=O)OC(C)(C)C)C2)C1=O c1(C(=O)NC(CSC)C(=O)O)ccnc(-c2cnn(CCCO)c2)c1 C1(CNC(c2c(Cl)cn(C)n2)=O)CC2(C1)CN(C(=O)COC1CC(F)(F)C1)C2 c1(C(=O)NC(C)C(=O)NCC23CC(CO2)C3)cnccn1 C(=O)(C1=NOC(C)C1)N1C(C(=O)NCC2(CCC=C)CC2)CC(O)C1 C1(OC)CN(C(=O)C(C)NS(C)(=O)=O)CCC1NC(c1ccc(C(F)(F)F)[nH]1)=O C1(NC(c2cnc(OC)s2)=O)CN(C(=O)C(C)(C)C2CCCO2)CC(C)(C)C1 c1(C(N2C(CCNC(CN(C(C)=O)C)=O)CCC2)=O)cccc2[nH]ncc12 C(C(COC)CC(=O)N1CC2CC(C(N3CC(Oc4ccccc4)C3)=O)C2C1)OC CCC1=NOC(CC(=O)NCC2CCCCN2C(c2cc(C(=O)OC)sn2)=O)C1 C(=O)(CC(O)c1ccccc1)N(CC(CN(C(=O)COCCCF)C)O)C c1(C(N(CC(C)NC(=O)C(C)CCCOC)CC)=O)ccc2nc(C)sc2c1 C1(NC(c2ccc(C)nn2)=O)CCCC12CN(C(=O)CCOCC(F)F)C2 N12CCC3CN(CC13)C(=O)Nc1cc(no1)C2.Cc1cccc(SC(F)(F)F)c1 c1(OC)cc(OC)c(C(=O)NCC2C=CCN2C(C2CC3(C2)CC(O)C3)=O)cn1 C1(NC(c2cc(C)c(C)nn2)=O)COC2(C1)CN(C(c1ccc(Br)o1)=O)C2 C1(C(=O)NC)CC(O)CN1S(=O)(=O)Cc1cc(CCN)no1 C1(NC(C(C)OCC)=O)CN(C(=O)CCC(C)(C)F)CCC12CCC2 Cn1ccc(CCC(=O)NC2CC(NC(=O)C=CC(F)(F)F)C2)c1 N1(C(C2C(OCC)C2)=O)CCCC2CN(C(=O)CSc3nccn3C)CC12 N1(C(C(C=C)O)=O)CCc2ccccc2C1CNC(c1sc([N+](=O)[O-])cc1Cl)=O C(=O)(C1=CCC(C)CC1)N1CC(NC(c2c(C)nc(C(C)(C)C)s2)=O)(CO)C1 N1(C(C2CC(C)(C)C2)=O)CC2CCCC(NC(C3(n4cncn4)CC3)=O)C2C1 C1(C(=O)NCc2c(C)cc(C)s2)N(C(C2CC2C(C)(F)F)=O)CCCC1(C)C N(C1c2ccccc2CC1NC(=O)CCC1CCOC1)C(CC(CC)(F)F)=O N1(C(CC2(CSC)CC2)=O)CCC2CCC(C1)N2C(=O)C(c1nc(C)cs1)C C1(CCCC)CCC(C(=O)NC(CN)CCc2ccc(F)cc2)CC1 CC(C(=O)N1CCCC(C2CCCN2C(c2cc(CCO)on2)=O)C1)C(F)F C1(C(=O)NC2C(NC(c3c(OC)c(F)ccc3)=O)C2)CCCCC(C)(C)C1 N1(C(c2c(C)con2)=O)CC2CS(=O)(=O)CC2(CNC(=O)C2=CCS(=O)(=O)C2)C1 c1(C(N(CCCNC(C=C(CC)CC)=O)C(C)C)=O)sccc1O N1(C(C2CCC(OC)CC2)=O)CCC2(CC1)CC2CNC(c1cnc[nH]1)=O C1(NC(C2(C(C)NC(C=CCOC)=O)CC2)=O)C=CCCCC1 C1(CCOC)CCCN(c2nnc(CSC)n2CCOc2ccccc2)C1 N1(C(C2C(C)OCC2)=O)CCCN(C(=O)CCN2CCN(C)CC2)CCC1 c1(C(=O)O)[nH]ccc1-c1cn(CC(=O)Nc2sccc2C2CC2)nn1 CCC(C(=O)NCCC(C)(C)C(=O)NCC1(O)CCCCC1)C(C)(C)CC c1(OC(C)C)ccc(C(=O)NCCCC(CO)NC(=O)C(O)c2ccsc2)cc1 C1(N(C(=O)Cc2scnc2C)CC)CCCN(C(c2csc(S)n2)=O)C1 N1(C(c2nc(C(=O)OCC)sc2)=O)CCC(C)(NC(=O)COCc2csc(=N)[nH]2)C1 N(C1=NCCSCN1)CC1CN2CCC1C2.Cn1cc(C(N)=O)c(-c2cccs2)n1 N1(C(C2N(Cc3ccc(C(C)(C)C)cc3)CC=C2)=O)CCC2(CCC2)C1 c1(NC(C)=O)cccc(CC(=O)NC2CCC2NC(c2cc(C)c(C)[nH]2)=O)c1 n1(CC)cnc2c(NCCCn3cncn3)[nH]c(=NC(C)c3ccsc3)nc12 N1(C(C2(OCC)CCCC2)=O)CCC(O)C(NC(=O)Nc2ccc(=O)oc2)C1 Cc1c(C(N2CCCC(NC(=O)CN(c3cnccn3)C)C2)=O)cccc1Cl c1(C(N(CC(CNC(C(=O)NC(C)C)=O)(C)C)C)=O)cccc(P(C)(C)=O)c1 C1(N(C(COS(CC)(=O)=O)=O)C)CN(C(=O)COC2CCCCCC2)CC12CC2 c1(C2C(C(=O)NC3CC(F)CN(C(c4cccnc4)=O)C3)C2)ccc(F)cc1F C1(NC(c2cc(C(C)C)no2)=O)CC=C(C(=O)NC(c2cc[nH]n2)C)C1 C(=O)(C(F)CCC(C)(C)C)NC12CCN(C(CCC(CC)=O)=O)C1CCC2 c1(C(=O)NC(CC)C(F)(F)F)cnn2cccc(-c3cc(OC)ccc3O)c12 C(=O)(CC(O)C(C)C)NCC(C1CCN(C(CNS(CCCC)(=O)=O)=O)CC1)(C)C Cc1cc(C(=O)NCc2ccc(C(N3CC=CC(O)C3)=O)s2)nc(C)c1 C(=O)(C(Cn1cncn1)NC(=O)Nc1cncnc1)OCC1(C)CC1 c1(OC)ccc(CC(=O)NCCC2(O)CN(C(=O)Cn3cc(Br)cn3)C2)cn1 C(=O)(C(C(=O)N(CCNC(c1n[nH]c(C)c1O)=O)CC)C(C)C)OCC C(=O)(CCCc1nncn1C)N(CC(C)N(C(C1(OCC)CCC1)=O)C)C Cn1nc(C(C)(C)C)cc1COC(c1cnn(C2CCOC2)c1C)=O N1(C(C(C)C)=O)CCC2CCN(C(c3cnn(C4CC4)c3)=O)CC2C1 c1(NC(C23CC(NC(c4c[nH]nc4[N+](=O)[O-])=O)(C2)C3)=O)c(CO)ccc(F)c1F C1(CC(=O)O)CCCC1NC(=O)NCc1ncco1 c1(C(N2CCC(CCCO)C2)C(=O)NCC(=C)C)ccc(CN(C)C)o1 c1(NC(c2ccc(C(=O)NC3C(C(N)=O)COCC3)[nH]2)=O)cc(F)ccc1Cl N1(C(c2c(SC)ccs2)=O)CCC(F)(CNC(=O)C(F)C2CC2)CC1 c1(Cn2ccnn2)cnn2c1NCC2 c1(CNC(c2csc(CNC(C3CCOCO3)=O)c2)=O)c[nH]ccc1=O CC1CCC(C(=O)NCC2C3CC4C(C3=O)C24)CN1C(=O)CCC1CCCCC1 c1(C(=O)NCCCCN(C(C(C)SC(C)C)=O)C)coc2c1COC2 C1(C(N2CC(O)(CNC(C3CN4CCN3CC4)=O)C2)=O)CCC(F)(F)CC1 Cc1cc(C(=O)NC2CCCC2NC(C2CN3CCC2CC3)=O)ccc1O CCC(C)(CC(=O)N1C2CCCC1CN(C(=O)C=Cc1cscn1)C2)C(=O)OC c1(C(N2CCC(C)(NC(C=CSC)=O)C2)=O)c(Br)cncc1[N+](=O)[O-] N1(Cc2cccc(C(=O)OC)c2F)CCC2(CC1)OCc1ccccc12 c1(N2CCC(CC)(CO)C2)nc(=NCCC2CCOC2)[nH]c2c1CCCCC2 CC(C)C(CCN(C)C(c1ncccn1)=O)NC(=O)C(C1CCCCC1)O N1(C(C=Cc2ccc(C)cc2)=O)CCCC12CCN(C(c1ccc(O)cn1)=O)C2 C1(NC(CCCCN(C)C)=O)CC12CCN(C(c1cc([N+](=O)[O-])n(C)n1)=O)CC2 C1(OCC)CC(O)CN1N(C)Cc1nnsc1SC c1(C(N2CCN(C(c3n[nH]cc3I)=O)CC2)=O)ccc2occc2c1 C1(C(N2CC(N3CCN(C(c4ccc(CO)s4)=O)CC3)C2)=O)C(F)(F)C12CCC2 CCC(CC(C)C)C(=O)N1CCCC(OCCCOC2CCC2)CC1 c1(C(=O)NC2C3CN(C(c4c(C)cc(OC)nc4)=O)C2C3)ccn2c1CCCC2 C=C1CC2(C1)CC(C(N1CC3CC(NC(=O)C4=CC(C)(C)C4)C1C3)=O)C2 C1(C(=O)NCc2occ(C(=O)NCc3nc(C)oc3)c2)CN(C)CCO1 c1(C(=O)NC(C)CC(C)NC(c2ccco2)=O)cc(Cl)ccc1OC(F)F Cc1cnc(N2CC(C(=O)NCCNC(c3ccc(C(F)(F)F)cc3)=O)C2)nc1Br c1(C(C)(C)C)nc2ncnc(NCC3CCN(C(=O)CC4NC(=O)NC4=O)C3)c2s1 c1(C(=O)NC(CNC(C(C)OCCC#C)=O)CO)c(C)nc(C)nc1C N1(C(C(C)Cc2ccncc2)=O)CCCOC(CNC(=O)CC2(C(F)F)CC2)C1 N1(C(C2C(NC(C(C)(C)OCC)=O)CC2)=O)CCCC(CC(N)=O)C1 N1(C(CCCCC(=O)OC)=O)CC(C2CCN(C(c3ccc(C)s3)=O)CC2)C1 C1(NC(C2C(COC)CCC2)=O)CN(C(=O)CN(C)C(=O)C2CC2)C(C)(C)C1 C1(NC(C(C)(C)C#N)=O)CC(NC(=O)Cn2nnnc2-c2ccsc2)C12CCC2 C12(C(=O)NC(CC=C)CNC(C3CCOC3(C)C)=O)CC(CO)(C1)OC21COC1 CC1CC=C(C(=O)NC2CC3CN(C(=O)CCC4CCOC4)CC23)CC1 S(=O)(=O)(c1cc(NC(C2(C(=O)OC)COC2)=O)ccc1F)NC(CCC)CO c1(N2CCC(N(C(C)=O)C)CC2)nc(NCCCCCF)c2ccsc2n1 N1(C(C(CN(C)C)NC(CCC(C)OCC)=O)=O)CCOC(C#N)C1 C(=O)(C(F)CC(C)(C)C)NCCn1ccc(C(=O)NC(C(C)O)C(=O)NO)c1 N1(C(c2cc(-c3cc[nH]n3)on2)=O)CCCN(C(=O)CCC2CC2Cl)CC1 S(=O)(=O)(c1cccc(N2CCC(N3CC(O)C3)C2)n1)N(C)CC1CCCS1 CC1(C)CN(C(c2ccc(C#N)s2)=O)CCC1NC(=O)Cc1ccc(F)c(Cl)c1 C(=O)(C(C(=O)OC(C)(C)C)C(C)C)NCCC1CC(NC(c2c(C)ocn2)=O)C1 N1(C(C(c2cccs2)SC)=O)CCC2(CCC2NC(=O)CC2CSC2)CC1 C(N=c1[nH]c2c(c(=NCC3COCCO3)[nH]1)CCC2)C1N(C=O)CCC1 C1(NC(CNC(CCCC)=O)=O)CN(C(c2cc(CC(C)C)c[nH]2)=O)CC1(C)C C(CCCCCCO)N(C(CC1(N(C(=O)CCc2ccoc2)C)CC1)=O)CN=O n1(C(CC)CC)nc(C(=O)NCC2(C)CCC(NC(=O)COC(C)C)C2)cc1C C(=O)(C1=CCCCC1)N1CC(NC(C2CCCCN2C2CC2)=O)C1 N1(C(C(c2ccccc2)OC)=O)CCC(CN(C)C(c2cc(Cl)nn2C)=O)CC1 c1(CCN(C2CCCC2)C(CNC(C=CC(CC)C)=O)=O)ncc(C)cn1 C(=O)(C(CC(F)F)NC(=O)CC1(CSC)CC1)NCC1(CO)C(C=C)C1 CC1CCC(O)(C(=O)NCC2CC(O)(CNC(C3CCCCO3)=O)C2)CC1 N1(C(c2nc(Cl)cs2)C(=O)NCCC)C2C=C(c3ccccc3)CC1CC2 C(C)(C)(CCCCC(=O)NCCC(C)NC(=O)C(C)NS(C)(=O)=O)OC N1(CC(C)C)C(=S)NC(c2scc(Br)c2C)C2=C1CCN(C(C)(C)C)C2=O C(=O)(C(C)CC(C)C)N(CCC(=O)NC(c1ccnn1C)CC)CC#C CCCC(C(=O)N1CCN(C(c2cc(N)ccc2F)=O)C(C)C1C)C(C)C c1(OCC(CC)OC(=O)CC2CC(C)C2)ccc2c(c1)OCO2 CC(C)(CC(=O)N1CCC(C)(CCNC(C23CCN(CC2)C3)=O)C1)CC(F)F C(CNC(c1sccc1C#N)=O)(CC(F)(F)F)NC(CN1CCC(C)CC1)=O c12onc(-c3ccccc3)c1C(=O)N2.C(C)(C)(C)OCCNCC=CCC c1(CNC2CCC(C#N)C2)c(F)ccc(Br)c1F c1(C(=O)NCCCN(CCO)Cc2ccnc(C)n2)nc(C)c(C)nc1C c1(C(=O)NCCC(CC)(C)NC(=O)CCC(C)C)cncc2ncccc12 Cc1cccc(C(F)(F)C(=O)NC2CC(CNC(=O)Cc3cncc(O)c3)C2)c1 Cc1nc2cc(C(=O)NC3CCC3NC(c3n[nH]c4c3CCC4)=O)ccc2s1 C(=O)(C1=CCCC1)NCC(C(C)C)NC(C(C12CC(SC)(C1)C2)OC)=O C1(CNC(COc2cc(C)on2)=O)CCN(C(=O)Cc2cncnc2O)C(C)C1 CC(C)(C)C(O)CNC(C1CC(=O)CN1C(=O)CN1CCOCC1=O)=O Cc1cc(C(=O)NC(C2CCCN2C(c2ncoc2C)=O)C)ccc1Br C1(C(=O)NCc2cnccn2)CCCN(C(=O)C(Cc2ccccc2)C2CC2)C1 c1(SCC)cccnc1CNCC(c1nc(=O)o[nH]1)C Cc1ccn(CCC(=O)NC(C(F)(F)F)c2cn(Cc3ccc(Cl)s3)nn2)n1 C1(NC(c2cnc(CC(C)C)s2)=O)CC2CC(C1)N(C(C1(C3CC3)CCC1)=O)C2 N1(C(c2c(C)c[nH]n2)=O)CC(NC(c2cc3occc3[nH]2)=O)CC(F)C1 Cn1cccc(C(=O)NC2(C)CN(C(c3c[nH]nc3-n3cnnn3)=O)C2)c1=O C(=O)(CC(C)CC(C)C)N(C1CN(C(c2ccc(C)c(C)n2)=O)CC12CC2)C C(C(=O)NCCc1ccncc1)(C(C)(C)O)NC(C(C)=C1CCCC1)=O c1(C(=O)NC2CC(OCCOC)CN(C(COC)=O)C2)cnc2ncc(Cl)cn12 C1(NC(=O)NCCC)CCC(C(N2CCCC(NC(CC(=O)NC)=O)C2)=O)CC1 N1(C(CNC(=O)C=Cc2nccs2)=O)CCCCC1CC(=O)Nc1ccccc1