SMILES CC1(C(N2CCC2n2cc(C3CCCOC3)nn2)=O)CCCC1(F)F N#CC1(C(N2CCCC(N3CCN(C(C4(O)CCCC4)=O)CC3)C2)=O)CCOC1 C1(C)(C(C)C)CN(C(c2sccc2CNC(C2(C(C)(C)O)CC2)=O)=O)CCO1 N1(C(C(CNC(c2[nH]cc(C)c2)=O)O)=O)CCC2(C1)CN(C)C2 C1(CNC(C(C)=C2CCCC2)=O)CCC2(CN(C(c3cc(C4CC4)cs3)=O)C2)O1 c1(C(=O)NC2C(OC)CN(C(=O)Cc3ccsc3C)C2)cn(C2CC2)c(C)cc1=O Cc1cc(NC(=O)C=CC(C)NC(c2c(C)cccc2O)=O)cc(Cl)c1 c1(OC)c(F)ccc(NC(N2CC(O)CC2CN)=O)c1F N1(C(C2N(CC#C)CCC2)=O)CCC(NC(c2c(C)cccc2Cl)=O)CC1C CCCC(C(=O)NCCC1CCC2CC12)NC(C1C=CCC1)=O C(=O)(C(C(C)C)NC(=O)CCCc1nn[nH]n1)NCCCC C1(NC(c2c(CC)nns2)=O)CCCN(C(=O)CCNC(=O)C=CCl)C1CC N1(C(c2cc(C#N)on2)=O)CC2(CCCC(CNC(C3CC(=O)N(O)C3)=O)O2)C1 C1(C(N2CCCC(CCN)C2)=O)CCCN(Cc2cccc(C3CCC3)c2)C1.CC N1(C(CC(C=C)(C)C)=O)C2COCC1CC(NC(c1ccc(O)nn1)=O)C2 C(=O)(C1=CCCO1)N1C(CC(=O)NC(c2ccccc2)C)CCC1 c1(C(=O)NC(CC)CNC(c2cnn3c2CCC3)=O)cc(F)c(C)cc1Cl C1(CC)(NCC(c2csc(=N)[nH]2)=O)CCCC1 CC(CCc1cn[nH]c1)N=c1[nH]c(=N)[nH]c(=NC(CCO)c2ccco2)[nH]1 c1(CNC(N2CCC(c3c(C)cccc3)(F)C2)=O)cc(Cl)cnc1C CON(C)CC(O)Cc1cn(C2CC(=O)N(C(=O)CCc3ccccc3)C2)nn1 C#CCC(C)C(=O)N1CCC(C)(NC(c2ncn(C(C)(C)C)n2)=O)C1 c1(C(=O)NCCN(C)C(C2CCCCC2C(C)(C)C)=O)ccncc1N N1(C(C(COC)C)=O)CCN(C(c2ccnnc2S)=O)CC1CF c1(C(=O)NCCCCC(C)NC(C2CCCCO2)=O)cc(O)ccc1Cl c1(C(N2CCC(O)(CCNC(c3cn(C)c(O)n3)=O)C2)=O)cc(Cl)c(F)c(Cl)c1 C1(C(=O)NCC(C)N(C)C)(NC(c2cn(CC3CC3)nn2)=O)CCCOC1 C1(CNC(CC(CC)C2CCC2)=O)CC2CCC1N(C(C1CC1C#N)=O)C2 c1(NC(C(N2CCC(CNC(c3cn(SCC)nn3)=O)C2)=O)=O)ccc(C)cc1 N1(C(c2ccc(C(C)C)s2)=O)CC(C2CC2C(N2CCS(=O)(=O)CC2)=O)C1 C(=O)(CCCCC(F)(F)F)N(C)CC1CN(C(=O)COCC2CCCO2)CCO1 C1(CNC(C(CC)(C)C)=O)CN(C(C2CN(CC(F)(F)F)C2)=O)CC1(F)F C1(C(=O)NC2(C(=O)NC(c3ncnn3C(C)C)C)CC(CO)C2)CC2CC(=O)C1O2 N1(C(CCNC(C)=O)=O)CC(NC(c2cc(-c3cccs3)nn2C)=O)C(C)C1 N1(C(CCNC2N(CC(=O)NS(CC)(=O)=O)CCC2)=O)CCC(C)(CO)C1 N1(C(C2C(Cl)(C(=O)OC)C2)=O)CCCC(C)(NC(C2CC3(CSC3)C2)=O)C1 c1(OC)cc(C(=O)NC2CCC(N(C)C(c3csnn3)=O)CC2)cc(Cl)n1 c1(C(N2CCCN(C(C(C)NC(C)=O)=O)CCC2)=O)coc2c1C(=O)NCCC2 c1(C(=O)NC2C3CN(C(c4c(C#N)ccs4)=O)CC2C3)cnc2[nH]ccc2n1 c1(CC)oc(C(N2CC(CNC(C3CCC(C(N)=O)O3)=O)C2)=O)cc1C N1(C(CCC(C)(F)F)=O)CC(C)(C)CCC1CNC(c1ccc(C2CC2)nn1)=O c1(C(=O)NC(CCOC)CNC(C2SCCS2)=O)ccc2c(c1)CNC(=O)N2 c1(N(C)CC)ccc(N=c2c([N+](=O)[O-])c[nH]c3ccc(F)cc23)c(F)c1 N1(C(CC(CC)O)=O)CCC(c2ccccc2)CC1C(=O)OC CCCCC(C)(F)C(=O)NCC(Cc1ccccc1)NC(C1CCOC(C)C1)=O c1(NC(C2CN(Cc3ccc(Cl)s3)CCO2)=O)cnc(Cl)c(F)c1 N1(C(CN(CC(C)C)C(C2CCC(C)C2)=O)=O)CCC(CC2CC2)CC1 N1(C(C2(C#C)CCCC2)=O)C2CCC1C(C)C(NC(C1CC1C=C)=O)C2 CC(C)CCC(=O)NCC(=O)NCC1CN(C(C2CCCC(C)C2)C2CC2)CCO1 CCC(CC)(CCN=c1cc(OC)nc(-c2ccccn2)[nH]1)CC C#Cc1cccc(C(=O)NCCCC(=O)N(C)C)c1.C(=O)(CO)N.C1(=O)CN1CCSC Cc1cc(C(=O)NC2CCCC2NC(=O)C(C)(C)n2cccn2)cn(C)c1=O C(CS(=O)(=O)CC(=O)N1CC(NC(=O)Cc2cnn(C(C)(C)C)c2)CC1C)OC CCCCC(C(=O)NCc1cc(C)ccc1O)NC(c1cncnc1C)=O N1(C(c2c(CC)noc2)=O)C2CCCC1CN(C(c1cccc(OC)c1Cl)=O)C2 C(C(=O)N1CCN(C2CN(C(c3ccc(O)nc3)=O)C2)CC1)(C(F)(F)F)OC C(CCC(O)C(=O)N(CC(C)O)CC(C)O)NC(CCC(C)C)=O N1(C(CC(=O)NCC#C)=O)CCC(C)C(N(C(=O)C(=O)NCC)C)C1 C(CCCCC(=O)N(C)CC1(O)CN(C(C2(COC(C)C)CC2)=O)C1)OC CC1CC(CNC(=O)Cn2cnnc2)CN1C(C1CC(F)(F)CS1)=O N1(C(CSCCSCC)=O)CC2=C(C1)CN(C(c1cncc(C(F)F)c1)=O)C2 N1(C(C)=O)CCCC1C(=O)NC1(CC2CC2)COC1.C1(C=O)CC(C)C1 Cc1cc(C2CCC2)ccc1C(=O)NCC1(O)CN(C(=O)C(C(C)C)N(C)C)C1 C1(NCC(F)(F)F)(SCCCC2CC2(Cl)Cl)CCCC1 C1(C)(COC)CC(NC(=O)CC2(C)CCOCC2)CN1C(c1ccn(C)c1)=O N1(C(COC2(C)CN(C(=O)CS(N)(=O)=O)C2)=O)CCN2CCOCC2C1 C1(C(=O)NCc2cc(C)sc2C)CC(F)CN(C(c2cc3sccc3s2)=O)C1 CCC(C)(C#N)C(=O)N1CCC(O)(CNC(c2nncnc2C(F)(F)F)=O)CC1 C1(NC(C(CC)CC)=O)CCCN(C(=O)Cn2ccccc2=O)C1CC C(=O)(CCS(C)=O)NC(CC)CNC(c1ccc(OC)s1)=O C1(F)(NC(c2c(C)c[nH]c2)=O)CCCN(C(=O)COCC2CCOC2)C1 Cc1cccc(C(O)C(C)NCc2ccc(F)cc2C(F)(F)F)c1F C1(F)(CNC(=O)CCc2cncs2)CCC(NC(c2cccnc2O)=O)C1 Cc1cc(F)c(-c2cn(CCC3CN(C(c4ccc(CO)s4)=O)C3)nn2)c(F)c1 N1(C(C(n2ccc(C)n2)C)=O)CC2CC(NC(C3CCOCC3)=O)C2C1 C(C(N=[N+]=[N-])C(=O)NCC(O)CNC(c1cnc(C2CC2)s1)=O)OCC C(CC(C(=O)N(CC(C)CO)C)NC(=O)Cc1cnsc1)=CC c1(C(C(=O)NC(C)C)N(C(C)C(C)C)CC)ccc(Br)c(F)c1 C1(CNC(C2(C3N(C(CC4(CC)CCOC4)=O)CCC3)CC2)=O)CCCCN1C.CO c1(CC2N(C(CS(N)(=O)=O)=O)CCC2)nc(O)c2sccc2n1.c12cn(nn1)C2 C#CC1CCN(C(C2C(NC(C3(N(C)C)CC3)=O)C2(C)C)=O)C1 N1(C(C=CC2N(C(Cc3c(C)scc3)=O)CCC2)=O)CCC2CN(C)CC2C1 CCCC(C(=O)NC1(C)CCN(C(c2sc(OC)nc2C)=O)CC1)S(N)(=O)=O Cc1cc(CC(=O)NCC2CN(C(C3C=CCC3)=O)CCO2)n(C)n1 C1(CNC(C(F)=C(C)C)=O)CN(C(=O)CC2(CS(C)(=O)=O)CC2)CC12CCOCC2 c1(OC)ccc(CNC2C=CC(C(N3CCCCC3C)=O)C2)c(O)c1 N1(C(C(CCSC)O)=O)CC2CCC1C2NC(C12CC3CC1C2C3)=O Nc1cc(Cl)c(Cl)cc1C(N1CC(NC(c2ccc(F)cn2)=O)C2CCCC12)=O N1(C(C2(OC)CCCOC2)=O)CCC(C2(NC(=O)Cc3csnn3)CCC2)CC1 N1(C(CCC(C)N(C)C)=O)CCC(C(F)(F)F)CC1CNC(=O)CC1(O)CCC1 c1(C(=O)NCCN(C(=O)CC(C)N(C)C)CC)cc(F)ccc1Cl CC(C)(CCCCNC(=O)C(CC(F)(F)F)C(N)=O)C(=O)NNC(=O)c1ccon1 c1(CC)nc(=NC2CC(NC(=O)C=Cc3sc4ccccc4c3C)C2)s[nH]1 C1(C)(CNC(c2c(CC)occ2)=O)CC(F)(F)CN1C(=O)COCC1CCCC1 C(S(=O)(=O)CC1CCCc2ccccc21)n1nnnc1OC.N12CC(C13CC3)C2.CC O=C(C#CC1CCCCC1)NCC1(NC(c2cnn(-c3ccncc3)c2)=O)CC1 c1(C(CC(=O)OC)C2(NC(=O)C3=CC(C)(CCC(=O)O)C3)CC2)ccc(C=O)cc1 Cc1cc(Cl)cc([N+](=O)[O-])c1C(=O)NC1CC(O)CN(C(=O)C=CC2CC2)C1 N1(C(COCC(=O)NC)=O)CC(C)N(C(c2cc(C)ns2)=O)CC1C Cc1c(Cl)cc(C(=O)Nc2ccc(NC(c3ccc(I)c(Br)c3)=O)cn2)cc1Cl N1(C(C(COC)NC(C)=O)=O)CCN(C(=O)C(C)N(CC(F)(F)F)C)CC1 C1(C)(CNC(c2cc(CC)[nH]n2)=O)CCCN(C(C2NC(=O)OC2C)=O)C1 C(CCC1CCC1)(C(=O)NOC(C)CC)NC(C(CC=CCC)C)=O C1(NC(C2C3CN(C(CCC(C)CN(C)C)=O)CC32)=O)CCn2ccnc2C1 c1(NC(=O)NCC(C(F)(F)F)OC)ccc(F)cc1F.C1C(=O)N1C1CC1 N1(C(C(C)(C)NC(N)=O)=O)CC2COCC(C1)N2C(c1cccc(C#N)c1I)=O N#Cc1ccc(C(=O)NC2CC23CCN(C(C2C=CCS2)=O)CC3)c(F)c1 c1(NC(N2CC(NC(=O)NC)C2)=O)ccc(CC(C)C)cc1 C(=O)(C1=NN(C)C(=O)CC1)CCOCCCC(=O)NCC1(C(=O)N)CCC1.CO c1(OC)ccc(C(N2CCCC(O)(CCNC(C3CC(OC)C3)=O)C2)=O)cc1C Cc1ccc(Br)c(C(=O)NC(C2CCCN(C(c3c(C)cnn3C)=O)C2)C)c1F Cc1cc(-c2ocnc2C(=O)NC(C)(CNC(C2CCC2F)=O)C2CCC2)on1 CN1CCc2cc(C(N3CC4CC4(CNC(C4(C(C)(F)F)CC4)=O)C3)=O)sc2C1 C1(C(=O)NCC(CC)n2cccn2)(OC)CCN(C(=O)CN2CC=CC2)C1 C1(CCNC(=NCC)NCC(=C2CCOCC2)F)C2CC3CC(C2)CC1C3 C12(CNC(C3CCCS(=O)(=O)C3)=O)CC(CO1)N(C(=O)Cn1ncnn1)C2 C1(C(=O)NCC(CC(F)(F)F)NC(C(F)=CCC)=O)CCCC2(CCC2)C1 C1(NC(C(C2CCCCC2)OC)=O)CCCN(C(c2ccc(C(=O)OC)[nH]2)=O)C1C C1(C(=O)NC2(CF)CCN(C(c3c(C#C)cn(C)n3)=O)C2)CCn2ccnc2C1 N1(C(c2ccnn2CC(F)(F)F)C(=O)CCCSC)CCCC2(C)CCCCC12.N C1(CC)(CNC(C2(CC)CN(C(=O)Cc3ccccc3Cl)C2)=O)CCC(=O)N1 C1(NC(C2(COC)CCC2)=O)CC2CC(NC(=O)CNS(C)(=O)=O)C1C2 C(=O)(C#CC1CCOCC1)N1CCCC(CN(C(c2cccc(C)c2C)=O)C)C1 c1(N(C)CC2CCCO2)ncccc1S(=O)(=O)NCc1cnc(Cl)c(Cl)c1 N1(C(C(c2ccncc2)C)=O)CC2CCC(N=c3cc(Cl)nc(C4CC4)[nH]3)C2C1 C1(C(=O)NCC(C)(C)N(C)C)CSCCN1C(=O)CSCC(F)F C(C(C)C)(C(O)C(=O)NCCCSC(c1ccc(C)cc1)C)OC N#Cc1cn(C2CCC(c3ncc[nH]3)C2)c(=O)n(C(=O)c2ccccc2Cl)c1=O CCC(CNC(=O)Cc1c[nH]nc1C)(CC)C(=O)N(CCS(N)(=O)=O)C Cc1ccncc1C=CC(N1CCOC(CCCNC(=O)CC2CN(C)C2)C1)=O c1(OC)cc(C(N2CCOCC2C2CC2)C(=O)NCC(C)C)cc(OC)c1Br CC1CN(C(=O)CC2CC2)CC1CNC(c1c[nH]nc1C1CCOCC1)=O C1(N(c2ncccn2)C(C2C(C(=O)OCC)CC2)=O)CCN(C(C)(C)C)CC1O N1(C(C2(C(=O)OCC)CC2)=O)CC(NC(C2(C)CCCCO2)=O)C(C#N)C1 C=CCC(C)(C)CC(=O)N1CC2CC(NC(C3CCC(=O)N(C(C)C)C3)=O)C2C1 C1(NC(Cc2scc(CC)n2)=O)CC2C1CCN2C(=O)CC(C)C(C)C c1(C(N2CCCC(NCC)C2)=O)c(C)cc[nH]c1=N N1(C(Cn2ccc(C)n2)=O)CCC2CC2(C(=O)NC23CCN(CC2)C3)CC1 C1(C(=O)NCC(C)NC(=O)CSCc2cscn2)CC2CCCCCCC12 N1(C(C(CCC)C)=O)CC2CC(C)N(C(C3CCNC4(CCC4)C3)=O)C2C1 C1(CC)CCN(C(=O)CCN(C)CCO)C1C(=O)NCc1ccc(OC)nn1 c1(N2CC3(CN(C(c4cnc(Cl)c(C5CC5)c4)=O)C3)C2)ccc(F)cc1[N+](=O)[O-] CC1C(NC(=O)CCC[N+](=O)[O-])CC2CCC1N2C(c1cnoc1C1CC1)=O C(=O)(C1=CCC(F)(F)CC1)NC12CC(CNC(C3(OC)CCSC3)=O)(OC1)C2 c1(C(N2CC3C(CNC(C)C)C3C2)=O)c(F)cc(Br)cc1F C1(NC(c2cc(Br)cnc2S)=O)CN(C(c2ncncc2F)=O)CC12CC2 C(Cn1cncn1)(C(=O)N=c1cc2n([nH]1)CCCC2)NC(C1CCC(=O)C1)=O C1(C(=O)OCCOc2ccc(F)cc2OC)(OC)CC(C)CC(C)C1 c1(C(N(C)CC2CN(C(C(C)N3CCC3)=O)C2)=O)nc(C2CC2)cs1 c1(CNC(c2ccc(C(=O)OC)o2)=O)ncc(C(N2CCC2C)=O)cn1 C1(c2n(CCCF)nc(-c3cccc(Cl)c3)n2)CCc2nncn2CC1 C1(C(=O)NCCn2cc(-c3csc(C4CC4)n3)nn2)CCC(F)(F)CC1 N1(C(Cc2nc(C)oc2)=O)CCN(C(=O)C(c2c(C)n[nH]c2C)C)C(CCO)C1 Cc1cc(C(=O)NC2CCCC(CN(C)C(c3occc3C(N)=O)=O)C2)nn1C C1(C(=O)NC(C#C)(C)C2CCCC2)COCCC1NC(=O)CC1C(=O)NN=C1C c1(CC(=O)N(CC(C)O)CCNC(C2(F)CC2C)=O)nccn1C C1(CC(=O)N(C(C)COC)CC=C)CN(C(=O)C(C)SC)CCC1C Cc1cc(N2CCC(C3(NC(=O)CC4CC=CCC4)CC3)CC2)nc(C)c1C#N C#Cc1cn(C)nc1C(N1C2CCC1C(NC(=O)Cn1cc(C(C)C)nn1)C2)=O c1(C(=O)NC2CCC(F)(CNC(c3ccns3)=O)C2)cc(Cl)c(F)cc1O CCCCC(C(=O)N1CC(OC)CC1C)C(=O)CC(=O)OC N1(C(C(CC)OC2CCCC2)=O)CC2CC2(CNC(c2cccnc2S)=O)C1 C1(COC)(CNC(C2CCCC2CN(C)C)=O)CCCN1C(=O)CSC C(=O)(C(C)CC(F)(F)F)NC1CC(C(=O)NC2(C(N(OC)C)=O)CC2)C12CCC2 c1(C(=O)NCCN(C(=O)C(O)Cc2cc(Cl)cc(Cl)c2)C)coc(S(C)(=O)=O)c1 C(=O)(CCCCC(F)(F)F)N1CC(C2CN(C(C(C)(C(C)C)NC(C)=O)=O)C2)C1 Cc1cnn(C)c1C(=O)NC1CCCC1NC(c1cnc(N2CCOCC2)s1)=O c1(C(N2CCC(C)(CC(=O)N3CC(OCC(F)F)C3)C2)=O)ccc([N+](=O)[O-])o1 c1(C(N(C2CCN(C(c3csc(C)c3)=O)CC2)CC#C)=O)cncc(F)c1 Cc1cc(C(N2CCC(C)C(N(C)C(c3cn(C)c(C)n3)=O)C2)=O)c(C)c(C)c1 N1(C(CC=C)=O)CCC2(CC(NC(c3cccnc3OCCO)=O)C2)C1 CCCC(C(F)(F)F)NC(C1(CCNC(=O)C(C)OCC(C)(C)C)CCCC1)=O C1(CNC(C(C)Cc2ccco2)=O)CCC(C(=O)N(C)CCF)CC1 c1(C(N2C(C(=O)NC3CCC(=O)NC3)C3CCCC32)=O)ccnc2cc[nH]c12 C1(C(N(C(c2ccc(OC)cc2)C(=O)O)C)=O)Cc2cc(C)ccc2S1 c1(C(N(C(CCNC(C2(CC)CCCC2)=O)C)C)=O)cnc2cc(C)ccn12 c1(C(=O)NCC2(C(N)=O)CN(C(CSCC(=O)OC)=O)C2)csc2c1CCC(C)C2 c1(C(=O)NCc2csc(-c3ccccn3)n2)ccn2ncnc2c1 CCC(CC)CCCN(C(=O)CC(C)CNC(C1(C)CC2C=CC1C2)=O)C O=C(CCC(F)(F)F)NCC(CO)NC(=O)CC1CCCS1(=O)=O C1(CCNC(CCC(C)(C)OC)=O)CCN(C(=O)CCC(C)(C)C#N)CCC1(F)F C(C1=NOC2CCCC12)NC(c1ncc(C)c(C)c1)=O CC(C(=O)NCC1CCC1C(=O)NC(c1nc[nH]n1)CO)=CC(C)(C)C Cc1cc(=O)c(C(=O)NCCCCN(C)C(c2cn3cccnc3n2)=O)cn1C N1(C(=O)COc2ccc(F)c(Cl)c2)CCC2(NC(C3CC4CC4C3)=O)CCCC12 C1(c2nc(C)[nH]n2)CCN(C(c2ccccc2)=O)CC1.C12CCN(C1)NC2=O CN1Cc2cc(C3CC3C(=O)NS(=O)(=O)c3ccc(CCN)cc3)ccc2C1=O C1(NC(CCCC=C)=O)CCN(C(C2(CCN(C)C)CC2)=O)CC(C)(C)C1 N1(C(c2snc(C)c2Br)=O)CC2CN(C(=O)C(O)C(C)C)CCC12 N1(C(C(C=C)O)=O)CCC(NC(=O)CCCN(C)C(C)C)C(CC)C1 CCC(C)CC(C)N(c1cncc(C2CC2)c1)C(c1ccccc1)C C1(NC(CSC(C)C)=O)CCCC(NC(C2COCCOC2)=O)C1 C1(=CC(=O)NC2CC(NC(C3C(C)(C)C3)=O)C2)CN2CCC1CC2 CC1(C)CC(NC(=O)CCc2ncco2)CCN(C(C2(C#N)CCOC2)=O)C1 c1(OC)ccnc(CCNC(C2CC3CCCC23)=O)c1OC CCC(CC(=O)NCCC1(O)CCN(C(=O)Cc2c(C)n[nH]c2C)C1)C(F)F C(=O)(C(C(C)C)n1cc(C)cn1)NCC(CNC(=O)Cc1cncs1)OC c1(C(N2CCC(NC(CC#C)=O)C2)=O)ccc(F)c(I)c1 C(=O)(C(C)(CO)OC)NCCN(C1CCCC1)C(c1cn(CCOC)nc1)=O CC(C)(C)CCC(F)C(=O)N1CCC2(CC1)CN(C(=O)Cn1ccsc1=N)C2 C1(NC(=O)C(O)COc2ccccc2)COC2(CCN(C(=O)CSC(F)F)CC2)C1 c1(CNCCNC(=O)C(c2ccc(Br)cc2)=O)ccc(F)c(F)c1F C(=O)(C1=C(Cl)CCOC1)N(CCOCC1C(NC(CCCOCC=C)=O)C1)CC N1(C(c2cnc(N)c3ncn(C)c32)=O)CCCC2C(CCCN2C(=O)C2CC2)C1 CC1=C(C(=O)N2CC(O)CC2CC(=O)NC2CCCCC2F)CCCO1 c1(OC)cc(C(N2CC(CN)C(C)(C)C2)=O)ncc1CO CC(C)(O)CCCC(=O)N1CC(CCNC(c2cncc(O)c2)=O)C1 c1(SCC=C)cccc(C(=O)NC(C)(CNC(c2cc(CC)n(C)n2)=O)CO)c1 N1(C(C(Cn2ccc(C)n2)C)=O)CCN(CCNC(=O)C(C)(C)CC2CCC2)CC1 C1(C(=O)NC2CC(C(C)NC(C(=Cc3ccco3)C)=O)C2)CCCOC1 N1(C(C)=O)CCCCC1CC(=O)NCC1CCN(C(C23CC(CC(F)F)(C2)C3)=O)C1 N1(CC(=O)N(CCOCCCN(C(c2c(CC)ncs2)=O)C)C)CCCCCC1 C12(NC(=O)CCCCc3cnc[nH]3)CCCC1N(C(=O)Cc1cnco1)CCC2 c1(CC)ccc(C=CC(=O)NCC2(OC)CN(C(C3CC3C(C)O)=O)C2)cc1 C(C)(CC(C)C(F)F)NC(C1N(C(c2c(C)cccn2)=O)CCSC1)=O N(C1CCc2cc(CNC(=O)C(=O)Nc3ncc[nH]3)ccc21)C(CCC(C)C)=O c1(NC(C(n2cc(C(CCC)=O)nn2)C)=O)coc(S(C)(=O)=O)c1 c1(OCCC(=O)NC(CCC2N(C(C=CC(C)C)=O)CCC2)=O)cccc(F)c1 N1(C(CC2(CNC(CCOCC(C)C)=O)CC2)=O)CCSCC(C)C1 Cc1cc(O)cc(=O)n1CC(N1CCC(C)C(NC(C2CC3(CSC3)C2)=O)C1)=O C1(COC)CN(C(c2cc(C)[nH]n2)C(=O)NCCC2(C)CC2)CC1C c1(C(c2nnnn2C(C)C)NC(CC(=O)NC)C)ccc(OC2CC2)nc1 CCCC(C(O)C(=O)NC1CCOCC1O)NC(=O)CCOC c1(CC(=O)NC2(CN(C(c3cnc(CC)nc3)=O)C)CC2)cccc(F)c1O c1(C(=O)NCCC2C=CCC2)ccoc1CNC(C1CC1(F)F)=O C1(CN(C)C(C2CC(=O)N(C)C2)=O)CN(C(=O)C=C(Cl)Cl)CCO1 C(C(O)CC(F)(F)F)NC(C1N(C(CCn2ccc(C)n2)=O)CC(F)C1)=O C=CCCCCC(=O)NCC(N1CCN(C(C2CC2C2CC2)=O)CC1)=O C#CC1(C(=O)NCC(O)CCC2CC2)CN(C(=O)C(O)CC=C)C1 c1(OC)cccc(NC(C2(CNC(c3cccc(Br)c3)=O)CCCO2)=O)c1 c1(C(=O)NS(c2ccc(C)c(Br)c2)(=O)=O)cc2cccc(Cl)c2nc1C N1(C(C(C2CCOCC2)OC)=O)CCC(N(C(=O)CC2CC(F)(F)C2)CCO)CC1 C12(C(=O)NCC(C)(CC)NC(C(CC=CC)C)=O)CC1CN(C(C)=O)C2 C(N=c1[nH]c2ccc(Br)cc2s1)C1CC(C)N(C(c2cccc(C3CC3)c2)=O)C1 CC1CCCCC1(CNC(=O)Cn1ccc(O)nc1=O)NC(=O)CC1(C)CCC1 c1(C(=O)NCC2(O)CCN(C(COCC#C)=O)C2)cc(OC)ccc1F FC1(F)CCCCC1n1nc(C2CCCO2)nc1-c1nnn(-c2ccccc2)n1 c1(C(C(=O)N(CC(CNC(c2cc(COCC)sc2)=O)C)C)C)ccccc1C C1(NC(COCCOCC)=O)CCN(C(c2cc(CC(C)C)on2)=O)C(C)C1 C12(CCNC(c3nc(C)n(C)n3)=O)CCC1CN(C(=O)CSC(C)(C)C)C2 N1(C(C23CCC(OC)C2C3)=O)CC(CNC(c2cncn2C)=O)CC(C)C1 Cc1c(C(=O)NCc2ccc(CCC(C)C)cc2)c2ccccc2n1C c1(SC(C)C(=O)NC2(CCNC(C3CC4CC4C3)=O)CCCC2)ccc(Cl)cc1 C1(NC(C(CC)C(C)C)=O)CC2CCCC(C1)N2C(c1nnsc1C)=O N1(C(C2C=C(C)CS2)=O)CCCC(C)(C)C1C(=O)NCC(O)C(F)F C1(NC(=O)OC(C)(C)C)CC2CCC1N(C(C1CCC3CCCCC3C1)=O)C2 C(CCCCC(=O)NCC1(C)CCC(NC(=O)COC2CC=CC2)CC1)N(C)C c1(C(N2C(CNC(c3csc(C)c3C)=O)C=CC2)=O)nc2c(s1)CN(C)CC2 Cc1nn(C)c(C(N2CCCC(CN(C(=O)CC(C)n3cccn3)C)C2)=O)c1Cl c1(C(=O)NCCc2ccc(OCCCC)cc2)ccc(F)c(Cl)c1 C(=O)(C(C(C)NC(=O)COCC1CC1)C(C)C)NCC(C)N(C)C Cc1nn(CC(N2CCCC(CNC(c3nc(C)n(C)n3)=O)C2)=O)c(C)c1C C#Cc1cccc(C(N2CC(NC(C3(n4cnnn4)CC3)=O)CC2C)=O)c1C N1(C(C(C=CC)O)=O)CC2(C1)CN(C(=O)Cn1cc(C(C)O)nn1)CCO2 C1(C(=O)NC(CC)C(N)=O)CN(C(C2CC(=O)CC(=O)N2)=O)CC12CC2 c1(OC)cc(C)ccc1S(=O)(=O)N1CCOC(C(N2CCCCC2C)=O)C1 C(=O)(C(C(C)C)N1CCN(C)CC1)N1CCC(CCNC(c2nnc(C)s2)=O)C1 c1(N2CCC(OC)C(F)C2)nc(N2CCCC(CO)CC2)nc2c1CC(C)CC2 c1(CC)cnc(O)c(C(N2C3CC2CN(C(C2OCCC2(C)C)=O)C3)=O)c1 C1(NC(C(CC)C)=O)CN(C(c2ccc(-c3cscn3)nc2)=O)CC(F)(F)C1 C1(C(=O)NCCC2CCN(C(C3(Cl)C(C(C)=O)C3)=O)CC2)CN2CCC1(C)CC2 CC(C)(CC(F)F)C(=O)N1CCC(O)C(NC(C2CCC=CCCC2)=O)C1 C1(C(=O)NCC(CNC(c2conc2-c2ccccc2)=O)O)CCC(CO)CC1 c1(NC(C2(C=C)CCC2)=O)ccc2cc(C)oc2c1 C1(NC(CCC)=O)CN(C(=O)C(=Cc2ccc(Cl)cc2)C)CC12CCC2 Cn1cc(C=CC(=O)NCc2cc[nH]c2C(=O)NCC(C)(C)CO)cn1 Cc1nc(S(C)(=O)=O)ccc1C(N1CC(CO)C2(C1)CN(c1ncccn1)C2)=O c1(-n2c(C3CN(CC(C)C)C(=O)CC3)nc(C3CCC3)n2)c(F)cc(F)cc1F c1(C(N(CCNC(=O)CCCc2cc(C)no2)CC)=O)n[nH]c2c1CCC2 N1(C(=O)COc2ccccc2)CC2(C1)CN(C(C1CCCCC1OC)=O)CCO2 C1(COC)CCCN(C(=O)NC(c2ccc(OC(F)F)cc2)C)CC1 C=C(Br)CCC(=O)NC1CCC(C)(CNC(=O)C=C(C)C2CC2)C1 C(=O)(C(C(CC)CC)OC)NCC1N(C(CC2CC(=C)C2)=O)CCCC1C C(=O)(C1=CC2CCCCCC12)NC1CC(NC(c2cc(C(C)C)cc(F)c2)=O)C1 CS(=O)(=O)c1cc([N+](=O)[O-])ccc1NC12CC3CC(CC1C3)C2 N1(C(c2cc(F)cc(N)c2F)=O)CCCC12CCCN(C(c1ccc(F)s1)=O)C2 C(=O)(C1CCCc2scnc21)N1CCC(N(C(c2ccc(CN(C)C)o2)=O)C)C1 c1(CNC(CC)CNS(C)(=O)=O)csc2ccc(Nc3ccccc3)cc12 CCCCC(CNC(c1ncc(CC)s1)=O)NC(=O)C(C)NS(=O)(=O)CC N1(C(c2c(C)nn(C(C)C)c2C)=O)CC(C)(C)C(NC(=O)CC(F)F)C(C)(C)C1 N1(C(=O)C2CC2)CCN(C(=O)CCC(F)(F)F)C2(CCC2)C1 c1(SCC)ccc(C(=O)NC2CCCC2NC(C2CCOC2C2CC2)=O)cn1 c1(C(N2CCN(C(C3(CC)CCNC3=O)=O)CC2)=O)ccc(=O)n(C)n1 c1(N2CCN(C(C3C(C)CCNCC3)=O)CC2)cc(S(N)(=O)=O)ccc1F C(=O)(CC1CCCc2ccccc21)NC(CNC(CC(C)CF)=O)C(C)(C)C N1(C(C2(C)C=CCN2C(C2CC=CC2)=O)=O)CCOCC2(CCC2)C1 C1(C(=O)NC2(C)CC(NC(C(CC)(F)C(=O)OC)=O)C2)Cc2ccc(F)cc2C1 C(=O)(CCCC(C)(C)CC)NC1CN(C(c2cc(CC)cc(C)c2)=O)CC(O)C1 c1(C(N2CC(C(=O)NC(CCC)C3CC3)N(C)CC2)=O)c[nH]c2ncccc12 c1(C(=O)NCC2CC(NC(CC3(C=C)CCC3)=O)C2)cc(Cl)c2c(c1)OCCO2 C1(C(=O)NC(c2cccnc2)c2nn[nH]n2)CCc2ccccc2C1 C#CCC(C(=O)N(C)Cc1cc(C)ccn1)NC(c1cc(CC)on1)=O C1(OC)CC(NC(=O)CCc2ccc(Br)nc2)CN(C(C23CC(F)C2C3)=O)C1 Cc1cc(Cl)c(C(=O)NC(C)CCCNC(c2cc(C(N)=O)on2)=O)cc1C C=Cc1ccc(C(=O)NCC2CCN2C(c2cc(Cl)n(C)n2)=O)cc1 C1(NC(c2cc(CC)no2)=O)CC2CCC(C1C)N2C(C1(C)CCCS1(=O)=O)=O c1(C(=O)NCC2(O)CCN(C(C3C(CC)C3)=O)CC2)ccnc2c1CCO2 CCCC(C(O)C(=O)N1CC(CO)C(C)(C)C1)NC(=O)C(F)=C(C)C N1(C(C(=O)NC(c2ncc(C)s2)CC)=O)CCCC2(CNC(=O)O2)C1 CC(C)CC(O)CC(=O)N(C1CCN(C(=O)CC(F)(F)Cl)CC1C)C Cc1cccc2cc(C(=O)NC(c3ccc(C(=O)O)c(C)c3)C)sc12 N1(C(C(C)CF)=O)CCCC(CC2N(Cc3cn(SC)nn3)CCC2)C1 C(CCC)(C(=O)N1CC=CC1(COC)CNC(C1CC(C(N)=O)C1)=O)=CCC N1(C(c2nc(C)n(-c3nc[nH]n3)n2)=O)CCC(CNC(=O)CC(C)(C)O)C(C)C1 CC(CC(C)NC(=O)C=CC(C)(C)C)NC(C1(NCC#N)CC1)=O C1(NCc2n(C)c(C3CCC3)nn2)CCN2CCCC2C1 NS(=O)(=O)c1csc(C(N2CC(NC(c3nncs3)=O)CC3(CC3)C2)=O)c1 C1(NC(c2ccc(C(C)C)o2)=O)CCCCC1NC(c1cc(Br)no1)=O C1(CCN=C(NCC(C(C)C)C)NC(C)C)COc2ccccc2O1 c1(C(N2CCN(C(=O)CSC(F)F)C3(CC3)C2)=O)ccc2nc(S)oc2c1 Cc1ccc(C(C)NC(C2(CF)CCN(C(=O)CC3CCOCC3)C2)=O)cn1 CC(CN=c1[nH]c(=NCc2ccc(Cl)c(Br)c2)[nH]c2cc[nH]c12)N(C)C c1(CN2CCCC(CC(=O)Nc3cncnc3Br)C2)ccc(Cl)c(F)c1 c1(N(C)C)cc(C(=O)NCC2CCC(NC(C3C4CCC3CC4)=O)CC2)ccn1 CCCCC(O)CC(=O)N1CC(O)CC1C(=O)NC1CCC2(CCCC2)CC1 n1(CC)nc(C2CC2)cc1C(N1CCC(C)C1CNC(=O)CC1CCCCO1)=O C1(CNC(C(C)SCCCC)=O)(NC(c2cc(C(C)(C)C)c[nH]2)=O)CCCCC1 C1(CC(N2CC(N(C(CC3ON=C(C)C3)=O)CCO)C2)=O)CC2CCC1CC2 c1(C=O)cc(C(F)F)ccc1F.N1(C(=O)NC(CN2C(C)CC2)C)CCOCC1 c1(NC(c2c(CNC(c3cccc(NC)c3)=O)c[nH]n2)=O)cc(F)ccc1O c1(OC)ccc2[nH]c(C(N3CC(CNC(=O)CSC)C(C)(C)C3)=O)cc2n1 CCC1=C(C(=O)NCC2CC(NC(c3oc(CC)nc3C)=O)C2)CCCO1 C1(N(C(Cc2cc(C)sc2)=O)C)CN(C(C2CCCN2S(C)(=O)=O)=O)CC1(C)C N1(C(C2N(C(c3c(C)cco3)=O)CC(F)C2)=O)CCn2ncc(C)c2C1 C1(CNC(COCC#C)=O)CC2CCC1N2C(=O)C(C)(C)Sc1cccc(Cl)c1 Cc1cc(C(N2CC(C3(NC(=O)CC(C)C4CCCC4)CC3)C2)=O)cnc1O C(=O)(C1=CC2CC=CCC12)N(CC(C)(C)CNC(=O)C(C)(C)CF)C c1(C(=O)NCC(C)(C2CCC2)NC(c2n[nH]c(C)c2F)=O)cc(Cl)cc(Cl)c1 C1(C)(C(=O)NCC(C)NC(c2cc(C3CC3)n(C)n2)=O)CCC12CCC2 CCCCCC(O)C(C)C(=O)N(C)CCN(C)C(c1ccc(SC)cc1Cl)=O c1(C(N2CCCCC2CO)=O)cnc2n[nH]c(-c3ccc4nsnc4c3)c2c1 C(=O)(CCCCN(C)C(C1CN(C)CCO1)=O)NCC(C(=O)OC)OC C1(CNC(c2cn(C3CC3)nn2)=O)CC2(CC2)CN1C(c1n[nH]c(C(F)(F)F)n1)=O N1(C(CCN(C(C2(OC)CCSC2)=O)CCO)=O)CCC2C(O)CC12 Cc1cc(-c2nc(-c3occc3Br)n(C3CCCC3)n2)c(C)o1 C1(C(=O)NC2(C)CC(NC(=O)CNC(=O)C3CC3)C2)CC1C1CC(F)(F)C1 C(=O)(C(Cc1ccccc1)CCS(C)(=O)=O)OCC(C)C(C)(C)C c1(C(N2CCCC(CCNC(CSC)=O)CC2)=O)ccc2c(c1)C(=O)CCCC2 c1(CCn2c(C(CCC=C)(C)NCCC3(C)CC3)nnn2)nc2cnccc2s1 N1(CC(C)NC(COCCC#C)=O)CCN(C(C2CC2=C)=O)CC1 c1(C(C)C)ccc(-n2cc(CN(CC(C)(F)F)CC3CC3)nn2)cc1 C(=O)(CCC(O)C(C)(C)C)N(CC(CC)NC(=O)CCC(=O)NN(C)C)CC C1(N)CC2C(C1)C2(F)F.c1(C2c3nnnn32)cc(Cl)c(Br)cn1.CC(=O)CCO N1(CC)C(=O)CCC1C(=O)NCCC(O)CNC(C1CC(N(C)C)C1)=O CCC(COc1ccc(Cl)cc1)S(=O)(=O)NC(c1cc(OC(C)=O)ns1)C c1(C(=O)NCC2(CNC(=O)COCC(F)F)CCCCC2)ccc(Cl)cc1F C1(C(=O)NCC(C)N(C)C(c2cc[nH]c(=N)c2)=O)CCCCS1(=O)=O N1(C(CCC2CCN(C(c3cnc(=N)[nH]c3)=O)CC2)=O)CCCC2CCCC12 N1(C(c2c(C)c[nH]c2)=O)CC(C(=O)NC2CCCC2CF)CC(C)(C)C1 N1(C(c2c(CC)cc(N)cc2)=O)CCC2CCCC(C1)N2C(C1CCC(=O)N1)=O C1(O)(CN(C(C2C(OC)CCCC2)=O)C)CCN(C(=O)C2=CCC2)CC1 C(=O)(C1CCc2c[nH]nc21)NCCN(C(C12CCC(OC(F)(F)F)C1C2)=O)CC CC1CCN(CC2CC2)CC1.c12cc(on1)CNC(=O)C(C)O2 CN=c1ccc(C(N2CC=CC2(C)C(=O)N(CC(O)CO)CCO)=O)c[nH]1 N1(C(c2cccc(NC)n2)=O)CC2(CCC2)CCC1CNC(=O)C(C)(CO)OC CC(CC(=O)NCC1CCN(C(c2cnn(CCN(C)C)c2)=O)C1)C1CC1 Cc1nn(C(C)C)c(C)c1CC(=O)NCC1CC1NC(c1nn(C)c(C)c1N)=O C1(CNC2CCCN(C(c3ccn(C)n3)=O)C2)COc2ccccc2O1 N1(CC(N2CCOCC2)C)C(=O)CN(CC2SCCS2)C1=O C1(CNC(CC2CCCC(C)O2)=O)CCCCCN1C(=O)CCN1CCCC1 CS(=O)(=O)c1cccc(-n2cc(C3CCCN3C(c3ccc(N)cn3)=O)nn2)c1 n1(CCOC)ncc(NC(=O)NC2C3CCC2CC3)c1C1CCOCC1 C(=O)(C(C(C)(C)C)OC)N(CCCCCC)CCNC(c1sc(C)nc1C)=O c1(OCCCCC)ccc(CNCCc2ccncc2Br)cc1 N1(C(C(C)n2ccnn2)=O)CC(CNC(=O)CCc2cncs2)CC1(C)C C1(C(=O)Nc2ccc(CC#N)nc2)CCN(C(C2CCCCO2)=O)CC1O C(C)(C)(C#CC(C)(C)O)NC(C)=O.CCC1C=CC(=O)N1 C1(CNC(CCCN(C)C)=O)CN(C(c2cc(C3CCC3)no2)=O)CCC1(F)F CC1CC(C(=O)NC23CCC(C(=O)O)(CC2)C3)CC(C)S1(=O)=O C(CC(C(C)C)NC(=O)CCNc1ccc(OC)cc1)NC(C(C=CC)O)=O C=C(Cl)CC(C(=O)N1CCC1CN=[N+]=[N-])NC(=O)C(n1nccc1C)C c1(C(=O)NC2CC(CNC(=O)C(F)CC3CCOC3)C2)ccnc2[nH]ncc12 N1(C(c2cnnc(Cl)c2)=O)CCC(CF)(NC(=O)C(Cl)=CCl)C1 c1(C(=O)NCC=CCSC)cn2c(n1)CN(C(c1ccc(Br)c(O)c1)=O)CC2 N1(C(=O)C=C2CCCC2)CCN(C(=O)CCc2ccc(O)nc2)C(CCO)C1 Cc1ccc2c(c1)CCC(C(=O)NC1CC1NC(=O)Cc1cc(C)[nH]n1)O2 N1(c2ccnc(NC(C3CCN(C(=O)C4CC4)C3)=O)n2)CCC2(CCSC2)C1 C12(C(N(C(C)CCNC(C3(C(F)(F)F)CC3)=O)C)=O)CCC(CC1)C2(C)C CCC(CC)CCC(=O)NC1CN(C(=O)CCCc2cccs2)C(CC)(CC)C1 C1(NC(c2n(CC)ccc2)=O)C2CC(O)C1N(C(=O)CC1CCC3(CC1)CC3)C2 Cc1ccc2c(c1CO)CCCN2Cc1nccn1-c1ccccc1 C1(CC(=O)N2CCC2)CCC(=O)NC1.C(C(C)(C)C)N(C)CCCS(C)(=O)=O N1(C(CC(C)C(F)(F)F)=O)CCC2CCN(C(=O)CCC(=O)c3cccs3)C2C1 C(C(CC(F)(F)F)NC(=O)CC1CC=CC1)NC(C1N(C(CCC)=O)CCC1)=O CN1CC=C(CC(=O)NCCCCC2CCCN(C(=O)C=CCO)C2)CC1 c1(C(N(C2CCN(C(=O)CCc3cc(Cl)no3)C2)CCC)=O)cnn(C)c1OC C(C(C)(C)CC(=O)NCC1(CCC(=O)NC2C(C(=O)OC(C)=O)C2)CCC1)SC C1(CC(=O)NCCC(C)N(C)C(C2CC2[N+](=O)[O-])=O)(OC)CCCC1 OC1CN(Cc2ccc(C3CCOC3)cc2)CCC12CCOC2 N1(C(c2cc(CNC(C3CCCSC3)=O)ncc2)=O)CC(F)(F)C(F)(F)C1 C1(CCNC(CNC(c2cc(C(F)F)[nH]n2)=O)=O)CCC2CC12 C(CC1=CCN(C(=O)CCC2CCOC2)CC1)NC(C12CCC(C)(C1)CO2)=O CC(C(C(=O)NCC(F)F)N(C)CC1(N(C)C)CC1)C1(C)CC1 C1(C(N2C(C(C)C)CC2)=O)CCN(C(=O)CC2CC=CCC2)O1 N1(C(C2C(C)(C)C2)=O)CCCC2CN(C(c3cnnn3C3CC3)=O)CCC12 CCC(CC)C(CN=c1nc(N2CCCCC(C)(C)C2)c2c([nH]1)CCC2)N(C)C CC1(C)CC(C(=O)NCC23CC(CO)(CO2)C3)CCN(C(=O)CCC#N)C1 c1(NC(=O)NCC2CCC(C(N3CCOCC3)=O)O2)ccnc2c(Br)cnn12 C1(C)(C(=O)NCCC2CCN(C(COCCCOC)=O)C2)CC(C)(C)OC1=O N1(C(CCc2cn(C)nn2)=O)CC(C2CC2)(NC(=O)C(C2(O)CCCC2)F)C1 N1(C(c2c(C)snc2)=O)CCC(C)(C)C(CNC(C2CC3(CC3)C2)=O)C1 c1(NCC(CC(C)C)C)ncc(-c2nn[nH]n2)cc1F C(=O)CCCC(CC)CC.CCC(C(=O)N1CC(N2CCCC2)C1)c1ccccc1 C(=O)(CC(C)(C)CC(=O)OC)NC1CCC(N(C(c2ccc(CSC)o2)=O)C)C1 c1(C(C(=O)NCC(C)NC(CC(=C=C)C)=O)O)cc(F)cc(F)c1 N1(C(=O)CC2CC23CC3)CCC2CN(C(c3cc(O)nc(Br)c3)=O)C2C1 c1(CC(=O)NCC(CNC(=O)C(C2CCCC2)C2CCCC2)O)ccnnc1O Nc1cc(C(N2CCC(NC(c3cc4occc4s3)=O)C(O)C2)=O)cc(O)c1Cl N1(C(Cn2ccc(C)c2)=O)CCCCC(N(C)C(c2cc(CCO)on2)=O)C1 C123C(C4CC1C2C4)NC(=O)C1(CCC1)NC3=O.C1(C(=O)OC)CC(OC)C1.C1CC1 n1(CC)nnc2c(N3CC4(CN(C(C5(CCF)CC5)=O)C4)C3)ncnc12 N1(C(C(C(C)O)NC(CC(C)C2CCCC2)=O)=O)CCC2(CC1)CC2 C(=O)(C#CC1CCOC1)N1CC(CN(C(C(C2CC2)OC)=O)C2CC2)C1 c1(C(=O)NCC(CO)NC(c2cnc(SC)s2)=O)ccc(C2CC2)nc1 Cc1cc(Cl)ccc1OC(F)F.C1(N2C(=O)CO2)CCCN(C(N)=O)C1 c1(C(N(C2CCN(C(=O)Cc3cnoc3)C2)CC)=O)cc2ccc(C)cc2[nH]1 c1(C(N(C(CCNC(c2cc(C)c(C)o2)=O)C)C)=O)csc2c1CCCC2 c1(C(N(CC(C)NC(C2(COC)CC=CC2)=O)C)=O)cn2ccnc2cn1 c12cccc(c1)C(=O)NC2.Cc1nc(C(=O)NCC2(F)CC(CN(C)C)C2)cs1 c1(C(C(=O)N(CC(C)NC(C2(c3ccccc3)CC2)=O)C)O)ccc(F)c(F)c1 C1(OC)CC(NC(C2(C)CC(F)(F)C2)=O)C12CCN(C(c1cccnn1)=O)CC2 C(=O)(C1=NOC(C(=O)OC)C1)NCC(CNC(=O)C(c1ccccc1)O)OC C1(CC)CN(C(c2cnn(CCO)c2)=O)CCC1CNC(C1CCC(C)S1)=O CC1CN(C(c2ccccc2F)=O)CCN1C(c1cccc(Cl)n1)=O c1(C(=O)NCCCSCC)cccc(NC(=O)C(C)(C2CC2)OC)c1 C1(c2nnnn2C2CC(C(=O)OC)C2)(NC(CCC)(C)C)CCN2CCC1C2 c1(C(C)NC(CN2CCOCC2)C(C)C)ccc(C(F)(F)F)cc1 c1(C(N2C3C(C(=O)NCC4(CC)CCC(=O)N4)C(C3)C2)=O)cnc(Cl)c(N)c1 Cn1nc(CNC(=O)CC2C3CCCC3N2C(=O)C(F)(F)C(F)F)n(C)c1=O N1(C(c2c(C)n(C)cc2)=O)CCC2(C1)CN(C(c1cc3ccsc3s1)=O)C2 C(CN=c1cc(SNCCOc2ccc(Br)cc2)nc[nH]1)NCCC1CCOC1 c1(C(=O)NCC(C2CCN(C(CC(CC)C)=O)CC2)F)ccc(Cl)c(N)c1 Cc1c(C(=O)NC(C)C(CO)NC(=O)C(c2cccnc2)C)cncc1Br N1(OCC)CCC(CCCNC(=O)C=CCN(C)C)CC1.C1(=O)NCCN1 C1(C)(C(=O)OC)CCC1(C)C(=O)NCC(C)NC(=O)CCc1cnc(C)s1 c1(C(N2CCCC(CNC(C(C)(C)OC)=O)C2)=O)cc2c(C)ccc(C)c2[nH]1 N1(C(C(=O)NC(CC)(C)C)C2CC2C)CCN(S(C)(=O)=O)C(C)C1 CC1COCCC1C(N1CC(CCNC(c2ccc(SC(F)(F)F)o2)=O)C1)=O C(=O)(CCCCC(C)C)NCCC(CC)(C)NC(c1cn2ccsc2n1)=O C1(CC)C(NC(=O)C#CC(=O)N(C)C)CCCN1C(=O)CCc1cnoc1 C1(CN)CC2(C1)CN(C(C1CC1C1CCC1)=O)C2.C12(CCCC1)C(=O)NC2 N1(C(CCc2ccn(C)c2)=O)CCC2CCN(C(=O)CC3CC3C(F)(F)F)CC12 c1(C(N(CC(=O)NCC2CCOCC2)CC)C)ccc(F)cc1 C1(NC(c2[nH]cc(C)c2)=O)COC2(CCCN(C(=O)C=C(Cl)Cl)C2)C1 N1(C(CNC(CC(C)(C)C)=O)=O)C2CCC1(CNC(c1cnc(C#N)s1)=O)CC2 N(C(=NCCc1ccc(OC)nc1)NCC1(CC(C)C)CC1)C(C=C)C c1(CC)ccc(C(=O)NCCCN(CCO)C(c2cc(C)c(C)s2)=O)c(C)n1 Cc1ccnc(O)c1C(=O)NCC1COC(CNC(C2CCC(C)(C)CO2)=O)C1 CC1CC(CC(=O)NCCc2noc(C(N)=O)n2)CN1C(=O)C=CBr C1(C(=O)NCCn2cc(C(=O)NCC(O)CF)nn2)CN2CCN1CC2 C#CC(C)(C)C(=O)NCc1cccc(C(=O)NCc2cccc(F)c2)n1 N1(C(c2c(C)sc(Br)n2)=O)CCCC(NC(=O)C=C2CCC2)C1C C1(C(N(C)CC2(C)CC2)=O)CC(NC(C2C(C)(C)C2(F)F)=O)C(O)C1 C=C=C(C)CC(=O)NCCCN(C(=O)CC1NC(=O)NC1=O)C(C)C CN(C)S(=O)(=O)N1CCC(C(=O)NC2CCCCN2S(C)(=O)=O)CC1 c1(C(N2CCC(NC(CC(COC)(C)O)=O)CC2C)=O)cc(Cl)cc(C)c1C CCC(CN(C)C)CC(=O)NCC1(CNC(=O)CSC2CCCO2)CCCC1 Cc1ccc(C=CC(=O)NC(C)CC(C)NC(c2scnc2Cl)=O)o1 C(C(O)C(=O)NCCOCCC(=O)NC(C1CCCO1)CC)=CC O=CN1CCCC1C(=O)NC(c1cccnc1)C(=O)NCC=CCO C1(NC(CSCc2nc(C)sc2)=O)CCN(C(C2CCOC2=O)=O)C12CCC2 C1(CNC(C2(CCC)CC2)=O)CN(C(=O)C(C)CN(C)C)CCC12CCC2 Cn1cccc1C(=O)C(=O)NC1CC1NC(=O)CCC1CCOCC1 C1(NC(C2CC(=C)CN2Cc2noc(CC)n2)=O)CCCCC1(F)F C(=O)(CCCC(=O)NC)N1CCC(CCNC(c2nc(COC)sc2)=O)CC1C N1(CC)CCOCC1CC(=O)NCCCC(C)NC(=O)CC1(OC)CCCC1 C1(C(N2C(c3cn(CC(C)C)nn3)CCCC2)=O)CCc2nnc(O)n2C1 N1(C(C(CC=C)OC)=O)CC2(CC(Cc3cn(C(CC)(CC)C(N)=O)nn3)CO2)C1 C1(C(=O)NCC2(O)CC(CNC(CCC=CC(C)C)=O)C2)CC2CCC1O2 Cn1cc(C(=O)NCC2CC3CCC2N(C(C2(C)CC2Br)=O)C3)c(=O)n(C)c1=O c1(C(=O)NCCC2(O)CN(C(c3cc4n(n3)CCO4)=O)C2)cncc2c[nH]nc12 c1(CNC(C(C)=C(C)C)=O)nc(C)c(C(N2CCC(F)CC2)=O)o1 C1(C(=O)Nc2cccc(C(C)F)c2)CN(C(=O)CCN2CCCC2)C(C)(C)C1 N1(C(C(CC=C)OC)=O)CCC(NC(C2(F)CCC2)=O)CC(C)(C)C1 N1(C(C(CSC)OC)=O)C2CCC1C1CC1(NC(=O)COCCOC)C2 c1(-n2ncc(NC(C3CC3CNC(C(CC)NC(C)=O)=O)=O)c2)ccccc1Cl C(=O)(C(O)CNC(=O)C(C1(O)CCCC1)F)NCC(C)(C)N(C)C N1(C(C(CC=C)OC)=O)CCCC(O)(CNC(c2ccc3ncsc3c2)=O)CC1 C1(C(=O)NCC(=C)C(F)(F)F)CN(Cc2cccc(F)c2)CCC1O CC1(C(=O)NC2CCN(C(c3cccc(Cl)c3)=O)CC2C(N)=O)CCCCCC1 C1(C(N(CC(CN(C(=O)C2=CCCCC2)C)O)C)=O)CC(S(C)(=O)=O)C1 C=CCCCC(C)(C)C(=O)NCC(C)C(=O)Nc1cnc(C)c(C)c1 O=C(C#CC1CCCO1)NCC1CC(F)(F)CN1C(=O)CN1C(=O)CNC1=O N12CC3CCC3(C1)CN(C(C1CCCCN1)=O)CCCCC2=O.C(C(C)C)SC c1(C(=O)NCC23CC2CN(C(c2cc[nH]n2)=O)C3)cc2c(Cl)cccc2s1 CC1CC(c2nnnn2C2CC2)(NCc2nc(=O)n(C)n2C)CN1CC(F)(F)F N1(C(C(C(C)C)NC(C)=O)=O)CC(C(=O)Nc2ccc(OC(F)F)cc2)C(C)(C)C1 CCC(C)(CC)C(=O)NC(C1CCCC1)CNC(=O)CCCN(C)C CC(C)(C)CC(O)C(=O)NCC1(F)CN(C(=O)COc2nc(O)nc(O)n2)C1 CC1CC(C(=O)NCCCC2CN(C(C3(C#N)CC3)=O)CCO2)=NO1 C1(N(C(C(C)(F)F)=O)C)CCC(NC(C2CCCCC2c2nc[nH]n2)=O)CC1 Cc1nccnc1C(N1CCCC1C1CCN(C(=O)CC2CCC(=O)O2)C1)=O C1(C(=O)NCCCN(C)C(=O)OC(C)(C)C)CN(C(c2cccnn2)=O)CCC1O c1(C2(NC(c3n(CCC)nnn3)c3nncn3C3CC3)CC2)ccccc1F c1(C(=O)NC(C(C)(C)NC(C(CC)n2ccnc2)=O)C)cc(Cl)cc2ccncc12 N1(C(C(COCC)C)=O)CCN(C(c2c[nH]nc2Br)=O)C2CCCC12 N1(C(c2ccc(NC)cc2Cl)=O)CC(CNC(=O)CN2CCOC2=O)CC(C)(C)C1 c1(C(=O)NC(C(c2ccccc2)NC(C(C)CO)=O)C)ccc2cc[nH]c2c1F C1(C)(C(N2CC(C(C(C)C)O)C2)=O)CCN(C(C2CC(C3CC3)C2)=O)CC1 c1(C(=O)NCCCN(C(C2CCC(=C)CC2)=O)C2CC2)cn(C)ccc1=O N1(C(C2NCSCC(=O)N2)=O)CCN(C(c2ncnc(O)c2F)=O)C(CF)C1 C1(CCNC(CCSCC(C)C)=O)COCCN1C(C1(C2CCCCO2)CC1)=O c1(C(=O)NCCCNC(c2ccc(OC)o2)=O)cn(C)nc1I c1(-n2cc(C(=O)NCC3N(C(C4CCC(=O)O4)=O)CC3)nn2)cccc(Cl)c1 c1(C(=O)NC2CC(NC(CCc3cnc(C)o3)=O)C2)scc(C)c1Cl C1(C(=O)NCC(CCOC)NC(CCCCC)=O)CS(=O)(=O)CCO1 c1(CC(=O)NCC2(C)CCN(C(CCC(CC)C)=O)CC2)cn2ccccc2n1 C1(NC(c2cnc3ccoc3c2)=O)CN(C(=O)Cc2ccsc2)C2(CCOC2)C1 c1(C(=O)NCC(CNC(C(C)C2CC2)=O)CO)cccc(-c2ccccc2)c1O N(C(=S)NNC(=O)C(O)C(F)(F)F)c1ccc(C(C)(C)C)cc1 C(=O)(C1CCCc2c1ncn2C)N.C1(N(C(C(C)SC)=O)CC2CC2)CCN(C)C1 C1(c2ccc(OC)cc2)(NC(c2ccccc2)CC2CC2)CC2(CCC2)C1 c1(C(=O)NCC(CC)(C)NC(=O)C=CC2CCC2)c(OC)ccc2cccnc12 c1(CCC)ccc(C(=O)N(C)CC2(NC(=O)C(C)(C)OC(C)C)CC2)s1 C1(C)(N(C(C(C2CCC(=O)N2)C)=O)C2CC2)CCCC1.C12CN(C1)C(=O)CO2 N1(C(C2N(C(c3cc(OC)n(C)n3)=O)CCC=C2)=O)CCN2CCC1CC2 Cc1cccc(CSCC(=O)NCC2CC(NC(=O)C3=COCC3)C2(C)C)c1 C1(C(=O)NCC2CN(C(CCc3nnc(C)n3C)=O)CC2O)COCC(C)(C)O1 N1(CC)CCOC(NC(=O)NC(C2(OC)CCCCC2)C)C1 C(=O)(C(C)(C)C(=O)NCCOc1c(-c2cn(C3CC3)nn2)cnn1C)OC CN1CCOCC1CC(N1CC(O)(CCNC(c2cc(C(F)F)no2)=O)C1)=O c1(C(=O)NC(CNC(c2c(CCC)nns2)=O)CC)c[nH]c2cc(OC)ccc12 c1(C(=O)NCC(CNC(C2ON=C(C)C2)=O)O)ccc(C(F)(F)F)cc1C#N C(=O)(C1CCc2c[nH]nc21)NC1CCN(C(Cc2cn(CC)nn2)=O)C1 c1(C(=O)NCC2C(C)CN(C(c3ccn(C)c3)=O)C2)coc2ccccc12 C1(NC(C2(C)CCCC2)=O)COC2(CNC(C3CCCC(F)(F)C3)=O)CC1C2 CC(C)C(O)C(C)C(=O)NCCCCCCC1CC1.C12CCCN1C2=O c1(C(N2CC(N(C(C(N3CCN(C)CC3)C)=O)C)C2)=O)ccnc(Cl)c1 N1(C(C2C(C(C)C)(COC)C2)=O)CCC(CNC(=O)Cc2cc(C(F)F)cs2)C1 C1(NC(=O)Cc2cnc[nH]2)CCN(C(c2ccc(O)nn2)=O)CCC1CO N1(C(C)=O)CC(CNC(c2ccc3nn[nH]c3c2)=O)OC2CCCC12 Cc1sc(C)c(C(=O)NCC2C(C)CCCN2C(c2cccc(O)n2)=O)c1Br CC1(NC(=O)Cn2ccc(=N)[nH]2)CCN(C(c2cccc(N(C)C)c2)=O)CC1 Cc1ccc(-c2noc(CN3CC(C)(NC(c4cccc(Cl)n4)=O)C3)n2)cc1F C(=O)(C(CNC(C1CCC(CC)CC1)=O)(CC)CC)N1C(C=C)CCC1 c1(C(=O)NCC2CCN(C(c3cn(CC(CC)O)nn3)=O)C2)c(Cl)c(C)nn1C CC1CN(C(c2cncc(N)c2)=O)CCCN1C(=O)CCC(C)(C)F c12cc(no1)CN1CC(C(O)C(=O)N2CC)C1.c1(SCCC(=O)OC)cccnc1 Cn1nc([N+](=O)[O-])cc1C(N1CCC(CCNC(=O)COC2CCC2)C1)=O c1(C(=O)NC2CCC(C(N(CC(=C)C)CC)=O)C2)cc(S(C)(=O)=O)oc1C c1(C(N(CC(C)NC(=O)CN(C2CCSC2)C)C)=O)ccc(C(C)C)c(F)c1 c1(C(=O)NCC(CC)NC(C2CC(C)CO2)=O)cc2c(Cl)nccc2o1 c1(CN(CC)CC2CCOC2)ccc(OC)c(Br)c1 CC1CN(C(=O)C2=CCN(C(c3nc(=N)cc[nH]3)=O)CC2)Cc2nncn21 c1(C(N2CC(NC(C(CC)(CC)OC)=O)C(OC)C2)=O)cc(N)c(F)cc1F c1(OC)cc(N(CCCNC(C)=O)Cc2cnn(-c3ccccc3O)c2)ncn1 N1(C(CC(C)SC)=O)CCCC2(CNC(c3cnc4c(c3)CCC4)=O)CCCC12 C1(C)(C(=O)NCC(CC)NC(=O)Cn2[nH]cnc2=N)CCNC(=O)C1 c1(OC)nc(N(C2CCCNC2)C(=O)Cc2ccc(C)c(C)c2)ncc1Br N1(C(CC(CC)SC)=O)CCN(C(=O)C(C)OC)CC(O)C1 C1(CNC(=O)C(F)=C2CCCC2)CC2CCC(C1)N2C(C1CCCC(F)(F)C1)=O C(=O)(C(C)C(O)C(C)C)N1CCC(C(c2ccccc2)C2C(C(CC)=O)CC2)C1 Cc1cccc(C(N2CCN(CC(N3CCOC(CCO)C3)=O)CC2)=O)c1I O=C(CC1=CCCCC1)NCC1CN(C(c2ccc(C(F)(F)F)cn2)=O)C2CC12 C1(C(N(C2CCN(C(c3c(CC)scc3)=O)C2)C)=O)CC(=O)N(C)C1 c1(SC)n[nH]c(=Nc2cnccc2C(=O)NCC(F)(F)F)s1 C1(C(=O)NCc2ccc(C)cc2)CCC2CCC1N2C(C1OCCC1(C)C)=O c1(C(C)C(=O)NCC2CC(NC(c3cnc[nH]c3=N)=O)CC2O)cc(F)cc(Cl)c1 c1(C(=O)NC2CCN(C(CC(=C=C)C)=O)CC(O)C2)cccc2c1OCC2(C)C c1(OC)cc(C(N2CC(C(C)NC(C3CC(O)CN3C)=O)C2)=O)cc(Cl)n1 c1(N(CC=C(C)C2CC2)C(N2CCCC(c3nc(=N)[nH][nH]3)C2)=O)cccc(F)c1 c12ccc(Br)c(c1F)C(=O)N2.N1(C(CCC)=O)CCCC1CC Cc1ccc(F)c(C(=O)NC2CC(NC(c3cncc(Cn4cccn4)c3)=O)C2)c1 n1(CCCN(C)CC2C(NC)CC2)cc(-c2cnn(C3CCOCC3)c2)nn1 c1(CC(=O)NC2C(NC(CCC(C)SC)=O)C2)c[nH]c2ccc(C)cc12 CC1CC(C(=O)NCc2ccnc(C(=O)NCCc3ncnn3C)c2)=NO1 c1(C(=O)NC2CC(C)N(C(c3ccoc3)=O)CC2)ccc2ccccc2c1 Cc1ccc(CC(=O)NC2(CNC(C3CC(C)(F)C3)=O)CCOC2)cc1[N+](=O)[O-] N1(C(c2ccc(OC)cc2)C(=O)NC)CCCC2CCN(CCCC(C)C)CC12 C1(NC(C2CN(CC(C)C)C2)=O)CCN(C(=O)C=Cc2ccncn2)CC(O)C1 c1(OC)ncc(C(N2CCCC2CNC(=O)C=Cc2nc[nH]n2)=O)cc1C C(=O)(CC(C)(C)C(F)F)NC1CCCN(C(C(Cc2ccccc2)N)=O)CC1 Cc1ccc(C(=O)NCCCCN(C(=O)CCn2ccnn2)C)c([N+](=O)[O-])c1 CC(=Cn1ccnn1)C(=O)N1CC(O)(CCNC(c2ccc(C)nc2O)=O)C1 c1(OCc2ncc(C(=O)NC(CC)CNC(=O)C(C)OC)cn2)ccc(F)nc1 c1(OC)cnc(Cl)c(C(=O)NC2CN(C(c3ccc(OC)c(Br)c3)=O)CC2C)c1 C1(NC(=O)Cn2cc(C(F)(F)F)nn2)COCCC1NC(C1CCCNC1=O)=O N1(CCNC(=O)C2=CCSC2)CCCN(C(=O)CC2NC(=O)NC2=O)CC1 C1(C)(CNC(CN(C(COC)=O)C)=O)CCN(C(C2CCOCC2(C)C)=O)CC1 Cn1nc([N+](=O)[O-])cc1C(N1CCCC(F)(CNC(=O)CN2CCCC2=O)C1)=O C1(C)(NC(CCCCNC(C(CC)CN(C)C)=O)=O)CCC(C)CC1 C1(NC(c2c(C)n(C3CC3)nc2)=O)CN(C(=O)CN2CCOC2=O)C(C)(C)C1 C1(C2CC2)(NC(C2OCCN(C)C2)=O)CCN(C(=O)CC(C)(C)O)C1 C(CCC(C)C(=O)NCC=CCNC(c1n[nH]c(C)c1O)=O)OC N1(C(C(C)NC(c2c(CC)noc2C)=O)=O)Cc2ccccc2C1C(=O)OC C=CCCC(F)(F)C(=O)N1CCC(C(C)NC(c2ccccc2Cl)=O)C1 N1(C(=O)Nc2ccc(CCO)cc2C(F)(F)F)CC2CCC(C1)C(=O)N2 c1(OC(CNC(C(C)OCC(=C)C)=O)C)ccccc1OC(F)(F)F C12(C(=O)NC3C(NC(=O)CCc4ccnc(Cl)c4)COC3)COCC1C2(F)F C=Cc1cncc(C(=O)NCC(C)(O)CNC(=O)C(=Cc2ccco2)C)c1 N1(C(C2(CC)CCCC2)=O)CC(NC(c2cnn3cccnc23)=O)C(N=[N+]=[N-])C1 C=C=CCC(C(=O)N1CCC(NC(c2ccccc2)=O)C1)NC(=O)OC(C)(C)C C(CNC(c1ccn(C2CCOCC2)n1)=O)(CC)(CC)NC(C1C(CC)C1)=O C(=O)(C1=CC2(CCOC2)C1)NC(CNC(C1=C(C)OCCS1)=O)CC(C)C C1(F)(CNC(Cc2cc(C)no2)=O)CCN(C(=O)Cc2ncccc2Br)CC1 Cc1cc(=NCC(C)(C)CC2CC2)nc(-c2ccncc2NC(C)C)[nH]1 n1(CCNC(C(C2CC=CCC2)NC(CC2(C=C)CC2)=O)=O)cc(C(=O)NC)nn1 CC1(C)CCN(C(c2cc(CCNC(=O)C=CCN3CCCC3)on2)=O)CC1 N1(C(=O)CC2CC2C(F)(F)F)CCC(Nc2ccc(Cl)cn2)CC1 c1(OC)ccc(C(N2CCOCC2CNC(C2CC2(C)Br)=O)=O)cc1O c1(C(=O)NC2C(CNC(Cc3c(C)nsc3)=O)CCC2)cnc(C(F)(F)F)cn1 CC1CN(C(c2cn(C)nc2O)=O)CC(C)CN1C(=O)CCc1ccnc(Cl)c1 Cc1nccc(CCC(N2CC(N(C)C)C(CNC(=O)Cc3cccn3C)C2)=O)n1 C1(C(C(=O)NCC=C)F)CCN(C(=O)C(c2ccccc2)O)C1 N1(C(c2cc(OC)ns2)=O)CCN(C)CC1C(=O)N(C1CCOC(C)C1)C Cc1cc(C(N2CC=CC2CNC(=O)Nc2cccnc2C)=O)c(O)nc1C C1(C(NOCCCOCC)=O)(CO)CN(C(=O)C(O)c2ccsc2)C1 N1(C(C(C)CN(C)C)=O)CC(C(=O)NCC2CCCNC2=O)CCC1(C)C c1(CN(C(CC)C(=O)OC)C)ccc(S(=O)(=O)N(C)C)cc1 C1(C(C(=O)Nc2ccc(OC)cc2)N(CC(C)OC)CC)CS(=O)(=O)CCO1 c1(C(=O)NC2CC(NC(C(=O)NCC)=O)C2)ccc(S(=O)(=O)CC)cc1 n1(CC)ncc(Cl)c1C(=O)NC1(CNC(c2ccn(CC(F)(F)F)n2)=O)CCC1 N1(C(c2ccco2)=O)C2CCC(C1)N(C(C1CCCCCC1)=O)C2 C1(C(=O)NC2C(NC(C3(CSC)CC3)=O)CC2)CCS(=O)CC1 C1(C(=O)NC(C=C)(C)CC)CN(C(=O)CC2COCC(C)O2)CC1N(C)C Cc1nn(C)c(-n2ccnc2)c1C(=O)N(CC(C)N(C(=O)Cc1ccco1)C)C C(=O)(C1=CC2CC(C1)CC2O)N1C2(CN(C(c3cccc(N)c3O)=O)C2)CC1 Cc1cn2nc(N3CCOCC(CNC(=O)C=C4CCN(C)C4)C3)sc2n1 N1(Cc2c(C)nn(CCO)c2)CCN(C2CC2)C(c2ccccc2Cl)C1 C(=O)(C1=CCCOCC1)NCC(CCNC(C1(C)ON=C(C)C1)=O)O C1(OCC)CCN(C(c2csc(CNC(=O)C=CC3CCOC3)c2)=O)CC1 C(=O)(C#CC1(C)CCCO1)NCC1C(C)(C)N(C(C2C3CCC(C3)C2C)=O)CC1 N#CC1CN(C(C2(C(=O)O)CC2)=O)CCN1C(=O)CCc1cncs1 C(C(=O)NCCCCN(C)C(c1cncc(C(F)(F)F)n1)=O)(C(C)C)OC(C)C CCN=C(NCC=Cc1ccc(Br)cc1)N1CCC(CC2CC2)C1 N1(CC(C)(O)C(N2CCc3sccc3C2)=O)CCOC2(CCS(=O)(=O)C2)C1 C1(C(=O)NC2CCCC(NC(C3(N4CCCC4)CC3)=O)C2)Cc2nncn2C1 C(CCNC(C1CCC(C)(C)O1)=O)(C(=O)NC1(CN(C)C)CC1)OC c1(C(=O)OCC)ccc(NC(=O)C(C)COC(C)(C)C)cc1Br N1(C(C2C(C#C)C2)=O)CCC(O)(CCNC(c2ccccc2C(=O)OC)=O)C1 C12(C(=O)NC(C3CCN(C(C(F)=CC)=O)C3)C)CC3CC(C1)CC(O)(C3)C2 CCCC(C)(O)CNC(C1(NC(=O)C(C)OCC2CC2)CCCC1)=O C1(NC(c2ccc(Cl)c(F)c2)=O)COCCN(C(c2cnc(S)n2C2CC2)=O)C1 c1(C(=O)NC(CNC(CCC(C)OCC)=O)CO)c(OC)cccc1O CC(C)CCCCCC(=O)NC1(C)CCN(C(C2CC2CF)=O)CC1 c1(CCNC(N(C(CC)CC)C)=O)c(OC)ccc2ccccc12 CC1(CNC(=O)C(N2CCN(c3cc(C(F)(F)F)on3)CC2)=O)CCC(F)(F)C1 c1(C(N2CC(NC(C(C)OCCOC)=O)C(F)CC2)=O)ccc(F)c2ccsc12 Cc1cccc(CC(N2CCC(CN(C)C(c3ccns3)=O)C2)=O)c1 C(=O)(CC(C)C(C)C(C)C)N1CCC(=CCNC(C2(OC)CCSC2)=O)CC1 CCC(C)C(C(=O)NCC1CN(C(c2c(Cl)noc2C)=O)C1)OC N12CC(C(C)C1)NC2=O.c1(C(C)C)nnc(C(N)=O)s1 N1(C(C)C)CCCC1C(=O)N(CC(C)N(C(=O)C(F)OC(F)(F)F)C)C C1(NC(COCc2onc(C)n2)=O)CN(C(C2CC3(C2)CC3F)=O)C2(CCC2)C1 c1(C(N(C2CCN(c3cc(C(C)C)ncn3)C2)CC)=O)cc(Cl)cn1C c1(C(N2CCC(CN(C(C(C)OCC)=O)C)C2)=O)cc(Br)cnc1O C(=O)(C(F)(F)C1CCCC1)NCCN(C1CC(OCOC)C1)CCC C(=O)(CCC(C)NC(c1cccc(F)c1)=O)NC(c1cnn(C)c1)CC N1(CCN(C(C2C3CN(CCCc4ccccc4)CC23)=O)CC)CCCCC1=O c1(C(N2CCC(N(C(C3C(CC)C3)=O)CC3CC3)C2)=O)cc(C)c(F)cc1F c1(SCC2CC2)cccc(F)c1.C1(NC(=O)CC2CCCOC2)CCN(C=O)C1 C(C(=O)N1CCC(C(=O)NCCCCS(N)(=O)=O)O1)c1ccc(C)s1 c1(C(=O)NC(C(C)C)(C)CNC(C2CC2C)=O)cc(F)c(Br)c(F)c1 Cc1cc(C(=O)NCCC(C)NC(c2ccoc2CC(N)=O)=O)c(N)c(F)c1 C1(CC)CCN(C(c2cncc(O)c2)=O)C1C(=O)NOCC1CCCO1 C1(NC(COCCCC)=O)CC2(NC(=O)CC(C)CCC)COC1C2 CCC(O)C(C)C(=O)N1CCC(CF)(NC(=O)Cn2cc(C(F)F)cn2)C1 CC1CCC(NC(=O)Cc2cnn(C)c2)CN1C(C12CCC(C1)OC2)=O C1(CC)(NC(C2COCCC2NC(=O)C(CO)OC)=O)CCCCC1 Cc1cc(C(=O)NCCCC(O)C(=O)N(C)Cc2ccn(C)n2)ncc1N c1(NC(CN2CCC(C#CC)C2)=O)cc(O)c(C)cc1C C=CC(C)(C)C(=O)NC1CC(C)N(C(c2cnn(CC(F)(F)F)c2C)=O)C1 C1(C(=O)NC2(CNC(C3CC=CC3)=O)CC=CC2)CC2C=CC1C2 Cc1cc(C(=O)NCC2(F)CCN(C(=O)C(C)CS(C)(=O)=O)CC2)c(Cl)cc1F Cn1c(C(=O)NC2CC(O)CN(C(=O)C3=C(Cl)CC3)C2)cc2c1CCOC2 C1(NC(C(C=C=C)C)=O)CCN(C(C2(Cl)CCCCC2)=O)CC1F C1(N(C)C(c2coc(Br)c2)=O)CCCCC1NC(=O)CCn1cc(Cl)cn1 c1(C(=O)NC(c2cn[nH]c2)C2CC2)ccnc(C(F)(F)F)c1 c1(C(=O)OCCN(CCCN2CCCC2)C)c(Cl)cccc1[N+](=O)[O-] c1(C(=O)NCC(CCNC(=O)COCC2(F)CC2)O)ccc2ccccc2c1F Cc1ccc(Cl)c(O)c1C(=O)NCC(O)CNC(=O)CCc1cn[nH]c1 c1(OCC)nc2ccc(C(=O)OCCNc3cc(C)nn3C(F)F)cc2[nH]1 O=c1n(C(F)F)ccn1CCc1noc(C2CC2)n1 N1(C(C2(COC)CCC2)=O)CCCCC(CNC(=O)CCCCCO)C1 c1(C(=O)NC2CC(CCNC(CCN(C)CC)=O)C2)cc2c(C)c(C)ccc2[nH]1 c1(C(=O)NCC2(O)CCN(C(CC3(C(=C)F)CCC3)=O)C2)cnc2ncccn12 C(=O)(CC1=Cc2ccccc2C1)N1CCCC(N(C)C(C2(C)CC2(Cl)Cl)=O)C1 C=CCC(F)(F)C(=O)N1CCC1CC(=O)Nc1nc(C)oc1OC c1(NC(C(Cc2cccc(C(=O)OC)c2)N(C)C)=O)nc(C)n2c1CCCC2 c1(C(N2CCN(C(C(C)=CC)=O)C(C3CC3)C2)=O)cnn2c1CC(C)CC2 N1(C(C2C(C)CCCC2)=O)CC2CC(C(=O)NCCC3(C)CC3)(C2)C1 c1(C(=O)NCC2CN(C(CCNC(COC)=O)=O)C(C)C2)c(F)cc(F)c(F)c1F N1(C(c2c(C)cccc2)=O)CC(C)N(C(c2ccc(Br)c(O)c2)=O)CC1C S(=O)(=O)(c1cccc(Cl)c1I)NC(c1noc(CCC(F)(F)F)n1)=O C1(c2nc(CCOC)nn2-c2ccccc2OC)CCC2CC(C)CN2C1 C(=O)(CC(=O)NCC(O)CNC(=O)Cc1nccs1)NCC c1(NC(CC2CC(=O)NC2)=O)nc2c(s1)CC(c1ccccc1)CC2 c1(C(N(C)CC2CCN(C(C3(CCOC)CC3)=O)C2)=O)ncc(Cl)cc1Cl C1(CCNC(C(C=C)O)=O)CCN(C(c2cnn(CCO)c2N)=O)C(C)C1 C1(CCNC(=O)Cc2ncc[nH]2)CCC(NC(=O)COCc2ccon2)C1 c1(CNC(=O)NC(CC=C)C)ncc(C(=O)OC)s1 c1(OC)ccc2nc(C(=O)N(C3CN(C(C4CC4F)=O)CC3(F)F)C)ccc2c1 C1(C(N(CCCNC(c2ccc(C)s2)=O)C2CC2)=O)CC12CC(F)(F)C2 N1(C(C2CN(C)CC(C)O2)=O)CCC2CCCC12C(N1CCCC(C)(C)C1)=O C(CC(=O)NC(C(=O)NC1(CCCF)CC1)C1CCCC1)SC C1(NC(C2N(C(c3cc(C)ns3)=O)CCC2)=O)CCc2ccccc2C1 C(C(C(=O)N(CCCC(C)C)C)C(C)C)NC(c1cc(C(C)=O)on1)=O.C1CC1 c1(C(=O)NC(CCC)C(=O)NCC2CC3CCC2O3)cnn(C)c1C#N N1(C(CC2C(C)=NNC2=O)=O)CCC2(CC1)CN(C(C1CC1F)=O)C2 c1(C(N2CCC(CNC(C3(F)CCCC3)=O)C23CC3)=O)cc(Cl)cc2c1OCC2 C(c1ccc2c(c1)OCO2)=CC(=O)NCCC1(NC(C2CC(CF)C2)=O)CCC1 N1(C(c2cc(C)nc(C)c2)=O)CC2(C)CN(C(=O)C(C)C(C)(F)F)CC2(C)C1 CC1c2c[nH]nc2CCC1C(=O)NC12CC(CNC(=O)CC3CC34CC4)(C1)C2 Cc1ccc(C(CNC(c2nnsc2C)=O)NC(C2C(C)(C)C2(F)F)=O)cc1 c1(CNC(c2c(OC)nsc2)c2nnnn2C2(C)CC2)ccc2occc2c1 Cc1cncc(C(=O)NCC(C)(CO)NC(c2sccc2-c2ncccc2O)=O)n1 C1(OC)CN(C(c2cccc(N)c2)=O)CC1NC(=O)CNC(=O)NC1CC1 N1(C(CCC2(CCC#C)N=N2)=O)CCN(C)C(C(=O)NCCCN2CCOCC2)C1 C1(NC(C(COC)C)=O)CC2(CCN(C(c3nnccc3C)=O)CC2)C1 CC(C)(C)CC(C)(C)C(=O)N1CCOCC(NC(C2CCC=CCCC2)=O)C1 N1(C(C(C)C(C)O)=O)CCC(NC(c2cccnc2OCC(F)F)=O)C(CO)C1 C(=O)(CC(C)(C)C(C)(F)F)NCC1CCN(C(C(C2CCOCC2)C)=O)C1 C12(NC(=O)Cc3ccsn3)CCN(C(C3(n4cnnn4)CC3)=O)CCC1C2 C1(C(N2CCCC(C(C)NC(=O)CCCC(C)=O)C2)=O)CCc2ccccc2C1 C(=O)(CC(C)CNC(C1COCC1C(N)=O)=O)NCC1(CO)CC(C)C1 C1(C(=O)NCC(C)(CO)NC(c2cccc(CC#N)c2)=O)CCCC(=O)N1 CC(C)(C)C(C(N)=O)NC(c1ncoc1CNC(C1CC1(C)C(F)F)=O)=O N(C(=NCCS(C)(=O)=O)NCCS(=O)(=O)Nc1ccccc1)CC(=Cc1cccs1)C Cc1cc(C(=O)N(C)CCNC(=O)C(c2ccc(F)cc2)(C)C)cc(=O)n1C C1(F)(C(=O)NC2CC(CO)C2)CCCN(C(c2cncc(Cl)c2)=O)C1 N1(C(c2c(C)cns2)=O)CCC2(CC1)CC2C(N1CC(O)CC1(C)CO)=O C(=O)(CC(C)(C)CC(=O)N1CCN(C(c2n[nH]cc2Cl)=O)CC(C)(F)C1)OCC C1(C(=O)OCC)CC(S(C)(=O)=NS(=O)(=O)c2cccc(OC(F)(F)F)c2)C1 Cc1cc(Cl)ccc1OCC(=O)NC1CCCC1CNC(C1CC2(CCC2)C1)=O c1(N(C(=O)N=S(C)(C)=O)CCCC)cc([N+](=O)[O-])c(C)cc1Br N1(C(COc2cc(C)on2)=O)CCCN(C(c2ccnc(C(N)=O)c2)=O)CCC1 C#Cc1cc(F)cnc1NC(C1CC1CNC(C1(c2cccc(Br)c2)CC1)=O)=O C(=O)(C1=C(Cl)CCCC1)NC(CC(=O)NCCC(C)N(C)C)CC1CCCC1 C12CCN(C1)C(=O)C=CCN2C(c1cc(C(C)C)no1)=O.N(C)CC C#CCC(C)(C)C(=O)NC1CCCC(CNC(=O)C(C)(O)CC)C1 C(=O)(C(C)(C)CSCC)NC(CC1(NC(c2nc(OCC)oc2)=O)CCC1)=O C1(C(=O)NC(C2C3CN(C(C4(C)CC(C)=NO4)=O)CC23)C)CCCCC(=O)N1 C1(NC(C2CCN(C(C3(n4nccn4)CC3)=O)C2)=O)C=CCCC1CO C(c1cncnc1O)=CC(=O)NCC1N(C(C(COC)O)=O)CCOC1 CC(C)C(C(=O)NC(CNC(c1cncc(C(F)F)c1)=O)C1CC1)NC(N)=O Cc1nsc(C)c1C(=O)NCC(O)CCNC(=O)C(F)n1ccnc1 N1(C(C(F)=CCC)=O)CCN(C(c2nc(C)ccc2Br)=O)C(CCO)C1 CC1C(NC(C2(O)CCSC2)=O)CC2CCC1N2C(=O)COC1CCOC1 C(=O)(C(O)CCNC(=O)C(CSC1CC1)NC(=O)C(CO)N(C)C)OC c1(C(N2C(CNC(c3cc(C)sc3C)=O)CC(C)(C)C2)=O)cc(F)c(O)c(Cl)c1 CC(C)CCC(CO)NC(=O)C(C)(C)C1CCN(C(=O)C(C)C(C)(C)C)C1 c1(OC)cc(CC(=O)NCC2(NC(=O)CCC3CC3(F)F)CC2)ccc1C c1(C(N2C3C(CNC(C)=O)CC(CC3)C2)=O)ccc2c(c1)C(=O)NCC(=O)N2 c1(C(=O)NC(C(C)C)C(=O)NCc2ccc(O)nc2)ccc(Cl)cc1Cl C12(NC(CC=C=C)=O)CC3CCC(C1C2)N3C(=O)C(C)Cc1ccc(F)cc1 C1(C(=O)NC2(CCNC(CSCC(N)=O)=O)CC2)CC(CC2CC2)C1 C1(C)(CNC(c2scc(OC)c2)=O)CCN(C(=O)Cn2nnc(=O)[nH]2)CC1 C1(C(N(C2CCCN(C(c3cccnc3)=O)CC2)C)=O)CC2(C1)CC2(F)F C#CC1(O)CCN(C(=O)COC2CCN(C(c3cccc(O)c3C)=O)C2)C1 N1(C(CCN(CC)CC)=O)CCC(C)(CC(=O)NC)C1.C1=CCNC1=O N1(C(CCC=C(C)C)=O)CCC2(CC1)CC2C(=O)N(C(C)C)CC1CCCO1 N1(CC)CCCC(C(C)NC(C(c2cnc(OC)cn2)N(C2CCCC2)C)=O)C1 C(=O)(C1CCCc2ccccc21)N(CC(C)NC(c1cc(C#N)ccc1N)=O)C Cc1ccnc(C(=O)NCC2(NC(c3c(Cl)cnn3C)=O)CC2)c1Br c1(C(N(C(C(=O)NC(CCOC)(C)COC)C)C)=O)ccc(=O)n(C)c1 C1(OC)(CNC(=O)C=CCCc2ccccc2)CCNCC1 Cc1ccc(C(=O)NCC2CCCN(C(=O)Cc3ccnn3C)C2)c2c1CCC2 C1(C(=O)NCCOCCNC(C(C)Cc2cnc[nH]2)=O)CCCN(C(N)=O)C1 N1(C(CC(CC)(F)F)=O)CC(NC(=O)Cc2cnccn2)CC12CCCCC2 CCC(C)(CNC(=O)C1CC1)C(=O)NCC(O)C(F)(F)F N1(C(C2CCN(C)CC2)=O)CC2(CC2)CC1C(=O)NC(c1ccc(Cl)cc1)CO C1(CC#C)(C(=O)NC2CCC2NC(C2CC3CCC2C3)=O)CC=CCC1 CC(C)(CC(F)F)C(=O)N1CC(CNC(C2CNC(=O)C2)=O)C(O)C1 CCCCC(O)C(=O)NCC1(COC)CCN(C(=O)CNC(N)=O)C1 N(C(O)=C1C=CN=NC1=O)c1ccc(OCC=C)c(Br)c1 C1(NC(c2nc(OCC)oc2)=O)CC2CCC1CC2NC(c1cnnc(C)c1)=O c1(C(N2C3CC4(NC(CCC=C)=O)C(C2CC3)C4)=O)ccnc2ccc(O)cc12 N1(C(C(C2CCCCC2)C)=O)CCC(NC(=O)CC(C)(C)c2ccccc2)C(C)C1 C(=O)(CCS(C)(=O)=O)N(CC(C)N(C(=O)COc1cccnc1)C)C CCCC(CC)CCC(=O)NC(CNC(c1cnc2[nH]ncc2c1)=O)CC(F)(F)F N1(C(CCOC2CN(C(c3cc(C)nnc3)=O)C2)=O)CC(CO)CC(C)(C)C1 N1(C(C2(SC)CCC2)=O)CCOCC(F)(CNC(c2cn3c(n2)COCC3)=O)C1 N1(C(=O)NCC2(OC)CC2)CC2CCC1C(C(=O)NC1COCCN1C=O)C2 N1(C(CCCNC(C=CC(C)(C)SC)=O)=O)CCn2c(C)cnc2C1 C1(CN(C)C(C2CC=CC2)=O)CCCN(C(=O)Cc2cn[nH]c2)C1 C1(NC(C2N(C(=O)NC)CCC2)=O)CC(COC)N(C(=O)C2=CCC2)C1 C12(C(=O)NC(c3ccc(Cl)cc3)C)CCC(C(N3CCCC(O)C3)=O)(CC1)CC2 c1(C(=O)NCC2(NC(C3CC(SC)C3)=O)CCCC2)nccc(Cl)c1F Cn1cc(C(O)CN)cn1.c1[nH]ccc1-c1ccccc1 N1(C(=O)OC(C)(C)C)CCC(O)C(C)(C)C1.C12CCC3CC13C(=O)N2 O=C1CCC2(CN1)CN(C(C13CC(CN(C(C4CCCOC4)=O)C1)C3)=O)C2 c1(NC(C2(C)N(C(C(CC)O)=O)CCC2)=O)ncc(Cl)cc1[N+](=O)[O-] N1(C(C2(CC#C)CCCC2)=O)CCC(CCOC)(NC(=O)CO)CC1 Cc1ccc(C(=O)NC2CC23CC(NC(C2CN4CCN2CC4)=O)C3)c(F)c1Cl C1(C(=O)NCC2(C)CCC(NC(=O)CCc3ncc[nH]3)C2)CN2CCN1CC2 C=C1Cn2c(C(=O)NCC3CC(NC(c4nc(O)c(C)s4)=O)C(O)C3)nnc2S1 C(=O)(C#CC(C)(C)CNC(c1cnc(C(C)C)o1)=O)NC(C(CCC)C)CO N1(C(Cc2cnc(C)s2)=O)CCC2CC1CN(C(C1CC(F)(F)CS1)=O)C2 C(c1ccc(N(C)C)cc1)=CC(=O)NC(C1CN(C(C2(C)CCC(C)C2)=O)C1)C C(C(C)N=c1cc(Cl)c(O)n[nH]1)NC(CC(C)OC)=O c1(C(C(=O)NCC(CNC(=O)C2CC2)OC)C)cccc(C)c1F Cc1ccnc2nc(C(N3CCC(NC(C4CCS(=O)(=O)N4)=O)C3(C)C)=O)nn12 c1(C(=O)NC(C2(O)CCN(C(c3cc(C)no3)=O)C2)C)ncn2ccccc12 C1(CNC(C(C)CN2CCCCC2)=O)CCCN(C(=O)C(O)CN(C)C)C1 c1(C(N2CCC(N3CCOCC3)CC2)=O)cnc(C(C)OC)nc1 c1(C2(N(C(C(=O)OCC(=O)NCC(C)C)=O)CCC)CCC2)ccccc1F C1(N(C(CC(CN(C)C)(C)C)=O)C)CCN(C(=O)C(C)(C)C#N)CC12CC2 N1(C(C(CC#C)NC(=O)CC(C)C2CC2)=O)CC2CC(OC)C(C2)C1 C1(n2cc(C(CC)(C)O)nn2)CCCN(C(=O)C=Cc2cc(C(=O)O)ns2)C1 c1(C(=O)NC2CN(C(C(C)N(C(C)=O)C)=O)CC23CC3)ccc2nc(O)oc2c1 Cc1cn2[nH]c(=NCC3CN(C(C4COC(=O)C4)=O)C3)sc2n1 N1(C(C(CO)OC)=O)CCN(C(=O)CCN(C2CCCCC2)C)CC1CC(F)F C1(O)(CNC(C2(C)CC2Br)=O)CN(C(=O)CSc2ccccc2)C1 C1(CNC(C(CC)OC)=O)(NC(C2CC3C=CC2CC3)=O)CCCCCC1 C#CC1CCN(C(=O)C(C)CNC(c2ccn(C)c2)=O)C1 c1(OCC)ccc(C)nc1C(=O)NCC1CN(C)CCN1C(=O)C(CC)SC c1(C(N2CC(O)(CNC(CC(CCC)CC)=O)C2)=O)cccc2c1OC(C)C(=O)N2 N1(c2nnc(COC)s2)CC2(CCC2)CC1CNC(C1CC2CCCC(C1)C2)=O C(=O)(C(C)(C)CC)NC(C=CC(=O)Nc1cn(CCOC)nc1)C N1(C(c2c(C)cccc2)=O)CCN(C(=O)Cc2ncncc2Cl)C(C2CCC2)C1 N1(C(c2ccsc2C(=O)NCC2CC2)=O)CC(OCC)CC(F)C1.C(=O)NC1CC1 c1(OC)ccc(C(N2CCC(C)C2CNC(=O)C(C)OCC(F)(F)F)=O)cc1Cl C12(NC(=O)Cn3cc(Br)cn3)CC1CN(C(c1cn(CCO)nn1)=O)C2 C1(CCC)CCCCC1N=c1nc2sccc2c(NCC(N2CCOCC2)C)[nH]1 N1(C(C(C)(C)OC)=O)CCC(N(C)C(c2ccc(CO)nc2)=O)C(C)C1 C(CC(C(C)(C)C)NC(c1cn(C2CC2)cn1)=O)N(C(C(C=C)CC)=O)C CC1CN(C(=O)CCC(C)(C)NC(c2cccc(=O)o2)=O)CCC1(F)F C1(C(=O)NCCOCC(F)F)(NC(C2CC(CC)C2)=O)CCN(C)C1 c1(N(C(C)=O)C(C)C)cc(C(N2CCCOCC2C)=O)ccc1Br c1(OCCNC(C(C(C)C)C#N)=O)ccccc1[N+](=O)[O-] c1(CNC(CCCC(CC)C)=O)ccc2c(c1)CCC2NC(=O)C=CC1CCC1 C#CCCC(=O)NC(C)(CNC(c1coc(CO)c1)=O)CC c1(C(=O)NCC(COC)NC(c2cccc[n+]2[O-])=O)cc(=O)c2ccncc2o1 c1(CN(C)C)ccc(C(=O)NCC2CC(O)(CNC(=O)CC3CCCO3)C2)o1 C1(CNC(C(F)=CCC)=O)CC(C)CCN1C(=O)C(CCSC)OC N1(C(C2CCC(C)O2)=O)CCC2(CC1)CN(C(C1CC(C#N)C1)=O)C1COCC21 N1(C(C2C(n3ccnn3)C2)=O)CCCCC1CCCOC.c1(C=O)nc(C)n(C)n1 C1(CN(C)C)COCC1CC1N(C(CO)=O)CCC1.C(=O)CCOCC(F)(F)F C1(NC(C(CC)C(C)C)=O)CCN(C(=O)C=CC2CCC2)CCC1CO c1(C(C)NCC(COCC)(C)C)ccc2ccccc2n1 c1(C(N2CCC(CN(C)C(c3sccc3Cl)=O)C2)=O)ncnc(O)c1F C=CCC(C)(C)C(=O)N1CC(C(=O)N(C)CC2CC(F)(F)C2)CCC1C Nc1cccc(C(N2CCC(OCCNC(C(=O)CCSC(=N)N)=O)C2)=O)c1O c12noc(c1Br)CNC2=O.C1(SCCC)CCC(=O)NC1 c1(SC)ccc(CCC(=O)NCCC2(O)CCN(C(C3(C)CC3(C)C)=O)C2)cc1 N1(C(c2oc(C)c(CO)c2)=O)CCC(C(=O)N(CC(N2CCCC2)C)C)C(C)C1 C(=O)(C(F)CCC(C)C)N1CCC(OC)(CNC(c2cccn2C2CC2)=O)C1 N1(C(C=CCOC)=O)CCC2(CC1)CC(NC(=O)C(C)CC(C)(F)F)CO2 N1(C(C(=O)NCCC2C(C)CCCC2)=O)CCC(C(C)C)C(F)(F)C1 C1(CNC(c2c(CC)nn(C)c2)=O)CN(C(C2(C)CCC(=O)N2)=O)CCC1C CCC(C(C)(C)OC)(c1nnnn1C1CC1)NCCS(=O)(=O)N(C)C C1(OC)CC(CNC(c2oncc2C)=O)N(C(C2CCCC(C(C)(C)C)C2)=O)C1 c1(CC(=O)NC2C3(CN(C(C=CCOC)=O)C3)CC2)ccc2oc(C)nc2c1 c1(C(N(CCC(C)NC(=O)C(C)c2cc[nH]n2)C)=O)ncc(C#N)cc1Cl C(=O)(C#CC1(C)CCCO1)NCC1N(Cc2ccc(OC)c(C)c2)CCC1 C1(C(=O)OC)CCCCOC(=O)CN1CC.c1(NC2CCOCC2)cccc(Cl)c1 C(=O)(C1Cc2ccccc21)NC1CCC(O)CC1.C1(CC(F)F)C(=O)N1C C1(NC(C(CNC(CC2N(C)CC=CC2)=O)CC2CC2)=O)CCC2(CCCC2)C1 C1(C(N(CC#C)CC2CCCO2)=O)CCC2CCC1N2C(=O)Cn1[nH]cnc1=N C(=O)(CC(O)(c1cccs1)n1cccn1)NCC(CNC(CC(=O)OCC)=O)O N1(C(C(CC(C)C)NC(C)=O)=O)CCCN(C(c2cccc(C)c2)=O)C(CO)C1 c1(CC)n[nH]cc1C(=O)NCC(CC)NC(c1cnc(-c2ccccc2)o1)=O N1(C(c2n(CC)ccc2)=O)CCOCC(C(=O)NC(C)(C)CC(=O)NC)C1 c1(CN(C(C2C3CCCCCC23)C(=O)NC(C)(C)C)C)cc(F)ccc1Br C1(C(=O)Nc2c(C(=O)OCC)cc[nH]2)CN(C(C2CCC=CCC2)=O)CC12CC2 c1(C(=O)NCC2C(CNC(C(CC(C)C)(C)O)=O)C2)cccc2nc(O)[nH]c12 C(N=c1[nH]c(C(F)(F)F)nc2c(F)cccc12)C1CC(C)(C)OC1 Cc1nc(O)sc1C(=O)NCC(C)CNC(=O)C(C)Cc1ccccc1Br C1(=O)C2=CCCN1C2.C=CC1(NC(=O)CN2CSCC2=O)CCC1 c1(CO)cc(CNC(C(=O)NC2CC2c2ccco2)C2CCC2)no1 c1(-c2ccc(C)o2)cc(NC(=O)NCc2c(C)noc2Cl)nn1C c1(OC)cc(C(F)(F)F)ncc1C(N1CC(c2nc(Sc3cccs3)n[nH]2)C1)=O CCCC(C(O)C(=O)NCC(CO)C(C)(C)C)NC(c1cnn(C)c1N)=O C1(CNC(=O)C(N2CCC(O)(Cc3ccsc3)CC2)=O)CC2(CCC2)CN1 c1(C(=O)NCC2CN(c3nccc(Oc4cn[nH]c4)n3)C2)ccc(F)cc1 c1(NC(C(CC2CCCC2)NC(CC(OCC)OCC)=O)=O)ncc(Cl)cn1 c1(C(CCC)NC(C2(N3CCOCC3)CC(O)C2)=O)cccc([N+](=O)[O-])c1 c1(C(C)=O)cccc(-c2cn(CC(=O)NCC(=O)NC3CCS(=O)(=O)C3)nn2)c1 c1(C(=O)NCCC(C)NC(=O)C(C)c2ccco2)cccc2c1CCC2=O c1(OC)cccc2c(C(=O)NC3CCCN(C(=O)C(Br)=C(C)C)C3)csc12 N1(C(c2ncc(CC)nc2)=O)CCCCC(NC(=O)CC2CCCC(F)(F)C2)C1 N1(C(CCC(=C)Cl)=O)CCN(C(c2cc(C3CC3)nn2CC)=O)CC1CO c1(C(=O)NCC(C(C)C)NC(c2cnc(C(C)OC)s2)=O)cccc2nncn12 c1(C(=O)NCC(CNC(CC(C=C)c2ccccc2)=O)O)scc2c1CCCC2 c1(C(=O)NC(C(C)NC(=O)Cn2ncnn2)C)conc1C1(C)COC1 N1(C(C#CC(C)C)=O)CCC(C(=O)N(C2CCOC2)CCF)C(C)C1 C1(NC(CSCC(C)C)=O)CN(C(=O)CCc2cn(C)cn2)C2(CCCOC2)C1 C1(C)(C(=O)NCCCCCCNC(C2C(C)(C)C2)=O)CCCNS1(=O)=O C1(NC(COCCN(C)C)=O)CCC2CC1CN2C(C1CCCCC1O)=O c1(C(=O)NCCc2c(C(N(CCC#C)C)=O)c[nH]n2)cc(C)nnc1O C1(OC)(CNC(=O)C(CO)c2ccccc2)CN(C(=O)C=CCOCC(F)(F)F)C1 Cn1nc2ccccc2c1C(N1CCCC(C2CC2NC(C2CCC2)=O)C1)=O C#Cc1cn(C)nc1C(=O)NCC1(O)CCN(C(=O)CC2CCCCC2C)CC1 C(=O)(CCC(C)N(C)C)N1CC2(C1)c1cn(nn1)CCO2.C=CC(Cl)C(F)(F)F C12(CNC(=O)NCc3cc(C)cc(Br)c3)CC3CC(CC(C3)C1)C2 c1(C(=O)NC2CC(CNC(C3(SCC)CCC3)=O)C2)cc[nH]c1C N1(C(C(C2CC2)CC)=O)CC(CNC(C2COCCN2C)=O)C(O)C1.C(=O)(OC)N C1(O)(CN(C)C(C2CC(O)C2)=O)CCN(C(c2conc2C2CCCC2)=O)C1 C=CCC(C(=O)OC)NC(=O)CC1C=CC(NC(c2cn(C)nc2COC)=O)C1 C1C(CC(C)C)C(=O)N1.c1(CCCC(=O)NCCC2ON=C(C)C2)ccc(N)cc1 c1(C(N2CCCCC(NC(C(CC=C)(F)F)=O)C2)=O)cccc2nonc12 c1(CC(=O)NC(C)(C)CNC(C2(CCF)CC2)=O)cc(Cl)ccc1Cl C1(OC)CC(C(=O)N(CCCCNC(=O)CCCC2CCC2)C)CC1OC c1(C(N2CCC(NC(C(COC)OC)=O)CC2)=O)ccc2ncncc2c1 c1(CC(=O)NCC2N(C(CSCC(N)=O)=O)CC3CC32)cccc2nsnc12 C1(C(N2CC3C(C(=O)NC4C(C)(C)C4(F)F)(C3)C2)=O)CC2(CCO1)CC2 c12cnnc(c1)C(=O)N2C1CCN(C(=O)Cc2ccon2)C1.C1(COC)CC1 CC1CCc2cc(C#N)c(N3CCC(NC(c4cn[nH]c4)=O)C(F)C3)nc2C1 C#CC1CCCN(C(=NCC2CN(C(=O)N(C)C)C2)NC(C)C=C)C1 c1(C(C)CC(C)(C)C)n[nH]c(=NC2Cc3cccnc3N2C)o1 CCC(C(=O)N1CC(C(C)O)C1)n1cccn1.C1=CCN(CC)C1=O C(=O)(C1=NOC(CC)C1)N(c1ccccc1C)CC(=O)NCCCCCNCC Cc1cc(N2CCCC(NC(c3cn(C(C)(C)C)nn3)=O)C2C)ncc1C#N C1(NCSC)CCOC(C)(C=O)C1.C#CCC(C=O)C1(OC)CC(C(=O)OC)C1 C1(NC(C(N2CCCCCC2)C)=O)(CNC(C2CCOC2=O)=O)CCCCC1 c1(C(=O)NCC2(F)CC(NC(CC(CC)C3CC3)=O)C2)cc([N+](=O)[O-])n[nH]1 N1(C(c2c(COC)nn[nH]2)=O)CCCC2(C1)CN(C(=O)CC13CCCC1C3)C2 C1(C(C)C(=O)N2CC(C(N)=O)C2)CCN(C(=O)C=C2CCC2)C1 C1(CNC(CC(=C=C)C)=O)C(C)CCCN1C(=O)Cc1ccc(N(C)C)c(F)c1 CCCC(O)CC(=O)NCCC1CCCN(c2ncn(C)c(=O)c2Br)CC1 CCCC(C)(C)CC(=O)NCCCCCC(=O)N1CCC(CO)C(O)C1 C1(NC(CC2CCN(C)C2)=O)CCCCCC1NC(C1SCCCS1)=O N1(C(C2CC(C#N)C2)C)CC2(C1)CN(Cc1nc(C34CC5CC3C4C5)cs1)C2 [N-]=[N+]=NCCCC(=O)NCC(O)CCNC(=O)C(Cc1ccccc1)C1CC1 C(N=c1[nH]c2c(c(=NCC3CC4(C3)CC4(F)F)[nH]1)CSC2)c1cc(O)cc(Cl)n1 C1(C(N(C2CCC(NC(c3cnc(Cl)cc3N)=O)C2)C)=O)C2CC3CC(C2)CC1C3 C(=O)(CCCC(C)(C)CC)N1C2CC(C(=O)NC(CC#C)C(=O)OCC)C1CC2 N1(C(C)C)C2CCC1CC(NC(C1(C(C)NC(=O)C3=C(Cl)CC3)CC1)=O)C2 N1(C(C=COCC)=O)CC(C)N(C(=O)Cc2nnc(O)s2)CC1C c1(OC)cc(Cl)c(Cl)cc1NC1(C)CC2CCC1C2 Cc1cc(C)[nH]c(=NCc2c(C3CC3)cnn2C)n1 C(=O)(C1=CCC(C)CC1)NCC(=O)Nc1cn(CCC)nc1 C#CC1CCCN(C(c2ccc(C)o2)C(=O)NCC)C1.C1(N)CCCCCC1 C1(C(=O)NCCOCCCNC(=O)CC2C=CCC2)COc2cc(Cl)ccc2C1 Cc1ccc(F)c(C(=O)NCCNC(=O)CC2CC23CC3)c1F CC(C)S(=O)(=O)C(C)C(=O)N(CC(O)CNC(=O)C=CCn1cncn1)C N1(C(C(=O)NC2CCOC2)C2(C)CC2)CCC(C)C(CC(=O)O)C1 C(COCCC)(C(C)(C)C)Nc1ccccc1.c1(O)ccccc1Cl.C12(CNC1)N(C)C2 c1(CC(C(=O)NC2CC(C)(NC(C=NOC)=O)C2)O)cccc(Cl)c1 c1(C(=O)NC2(CF)CCN(C(CC(C)F)=O)C2)ccc2nc(O)oc2c1 n1(CC(=O)NC(C2CCCN2C(c2cc[nH]n2)=O)C)nc2c(n1)CCCC2 c1(N2C3CS(=O)(=O)C(C3)C2)nc2c(c(=NCC(Cl)=CCl)[nH]1)SCC2 N1(C(CS(=O)(=O)NC)=O)CCOC2(CCN(C(C3CC(=O)N(C4CC4)C3)=O)C2)C1 C1(NC(C(C)C2CC2)=O)COC2(CCN(C(=O)C(c3ccc(F)cc3)C)CC2)C1 c1(SC)cccc(-n2nc(C3CCOCC3)nc2C(C)CS(C)(=O)=O)c1 C#Cc1ccc(C(=O)NC(CCCC2(NCCCS(C)=O)CCC2)=O)cn1 C(CCCC(=O)NC1CCN(C(c2cccc(C)n2)=O)C1C(C)C)OCCC=C C1(NC(C2CN(N(C)C)C2)=O)CC2CC1N(C(C1C(F)(F)C13CC3)=O)C2.C(=O)O C(=O)(C(CNC(=O)Cc1cccnc1)CC=C)NCC(COCC)O N#Cc1ccsc1C(=O)NCC1(F)CC(NC(C2CCCC(C3CC3)O2)=O)C1 C1(CCC)CCCN1C(C1(CC)CN(C(c2ccn(C(C)(C)C)n2)=O)C1)=O CC(C)(C)CCCC(C(=O)NC1CCC1)N1CCOC(C2CCC2)C1 C12(NC(CN3C(C)CCC3)=O)CCCC1CN(C(=O)C=Cc1ccsc1)C2 C1(C(=O)NCC2(CCNC(=O)C(F)CC3CCOC3)CC2)CCCC12CCC2 S(=O)(=O)(c1cc(C(=O)OC)c(Br)cc1F)C.N1(CCOC)CCC2CC12.OC N1(C(c2c(C)n(C3CCC3)nc2)=O)CC(C2(NC(=O)Cc3nccn3C)CC2)C1 C(=O)(CCCCN=[N+]=[N-])NCC1C(C)(C)C1C(=O)NCC1(O)CCCOC1 CC(C)CCCCCC(=O)NC1CCN(C(C2CC3(CCCC3)C2)=O)C12CC2 C12(C(=O)NC(n3c(C(=O)NCCSC(F)F)ccc3)CO)CCCC(=O)N1CCC2 CCCCC(C)(F)C(=O)N(C)CC1CCCN1C(c1cc(C)nnc1O)=O C1(CNC(CCN(C(C2(COCC)CC=CC2)=O)C)=O)OCCCC1(C)C c1(CC)nc(CC(C)C)oc1C(=O)ON1CCCC1C1(C)CC1 N1(C(C(CC)F)=O)CC2(CCN(C(=O)CCC3CC(F)(F)C3)C2)C1 CC1=C(C(=O)NC(CNC(=O)C(=O)NCCSC(C)C)CO)CCCC1 CC(C)C#CC(=O)N1CC(C(O)C(=O)NCC2CCC2)C1 C1(C(=O)NCCCc2nc[nH]n2)CC(F)(F)CN1C(=O)CN1CC=CC1 c1(OC(c2ccc(C(=O)OC)[nH]2)=O)ccc(OCC2CCCOC2)cc1C#N N1(C(CC(C)C)=O)CCOC2CN(C(=O)Cc3cnc4n3CCCC4C)CC12 C1(C(=O)OC)C=CCN(OC(=O)CC2(CC)CC2)C1.c12occc1CNC2=O N1(C(CCSCC)=O)CCCCC1C(=O)N(C1CCOCC1C)C C(=O)(CCC(=O)NC1COCC1NC(=O)CC1CCOC1)Nc1nnc(CC)s1 Cc1occ(C(F)(F)F)c1C(N1CCCC(N(C)CCc2cccc(N)c2)C1)=O C(CN=c1[nH]c(N2CCC(C3CCCO3)C2)nc2c1SCC2)N(CC)CC c1(OC)c(CC(=O)NC(c2ccccc2F)(C)C(N)=O)cccc1C#N C(=O)(CCCC(C)(C)NC(=O)C(F)=CC1CC1)NCCC1(C)CCOC1 C(=O)(NNC(=O)N)c1c(N)non1.C1CCCOC1c1cccc(F)c1 C1(NC(COC(C)C)=O)C2CC1N(C(=O)CCc1ccc(Cl)s1)C2C C(=O)(CCC1CCc2ccccc21)N(c1nc(C2CC2)nc(=NCC2CC2F)[nH]1)C c1(C(N(CCC)CCNC(=O)CS(N)(=O)=O)=O)cc2c(o1)CCCC2 C1(CC=C)(NC(=O)CN2CCOCC2=O)CCCN(C(=O)C(C)(C)CF)C1 c1(C(=O)NC2CC(CNC(c3cnc(Cl)s3)=O)CC2O)n[nH]c2c1CCC2 N1(C(C(C)CN(C(=O)C=CC(F)F)C)=O)CCCC(N(C)C)CC1 N1(C(c2ccc(COC)o2)=O)CCCC(C)(NC(C2(COC3CCC3)CC2)=O)C1 C(=O)(C1CCc2ccccc21)N1C(CNC(C2(COC)CCCC2)=O)CC(OC)C1 N1(C(Cc2cc(C)sc2)=O)CCC(F)(C(=O)NCCCC(O)CO)C1 N1(C(c2ns[nH]c2=O)=O)CCCC(C(N2CC=CC2CF)=O)C1 Cc1nc2cc(C(=O)NCC3CC(F)(F)CN3C(C3CC4CC4C3)=O)ccc2s1 c12nc(C)c(s1)C2=O.C1(CC)(NC(=O)C(C#N)CCCSc2ccccc2)CCCC1 c1(NCCOC)ccc(Cl)c(CNC(CN2CCCN(C)CC2)=O)c1 c1(OC)ccnc2c1CCCC2NC(N1C2CCC1CC1(CC1)C2)=O Cc1cc(O)ncc1C(=O)NC12COC(CNC(C34CCC3C4)=O)(C1)C2 C(=O)(CC(C(F)F)C(C)(C)C)N(CC(C)(C)NC(C(C(C)C)(C)C)=O)C c1(OCC(=O)NCC(C)N(c2cc(C(C)(C)C)c[nH]2)C(CC)=O)cc(Cl)cc(Cl)c1 C(=O)(C(F)(F)CCn1cccn1)N1CC(OCCNC(c2ccn(C)c2)=O)C1 C1(NC(C(OC)OC)=O)CCCC(CNC(c2cn(CCCF)nn2)=O)C1 c1(C(=O)NCC(C)NC(C2(CC)CCCC2)=O)ccc(-c2cscn2)cc1 N#Cc1cc(S(=O)(=O)NCc2ccc(C(N3CCCC3C3CC3)=O)s2)ccc1F Cc1cc(C(=O)NOCC(F)(F)F)cc(C)c1NCC1CCOCC1 c1(COC(CN(C2CCCN2N=O)S(C)(=O)=O)=O)noc2ncccc12 c1(C(OC(C=Cc2cccc(OC)c2)=O)C2CC2)c[nH]c(=N)nc1O C1(C(=O)NC2(C(N3CC(C(CC)C)C3)=O)CCCCC2)CC(=O)NC(=O)N1 C1(F)(CNC(CCSCC)=O)CC(NC(=O)C=Cc2cscn2)C1 Cc1noc(C)c1C(C)C(=O)N(C)CC1CCN(C(C2(N(C)C)CCC2)=O)C1 N1(C(c2cnn(C(C)C)n2)=O)CC(NC(c2cc(O)nc(O)n2)=O)CC2(CC2)C1 Cc1cccc(F)c1C(=O)NCC1(F)CC(CNC(c2cc(CO)on2)=O)C1 C1(O)(COC)CCN(C(=O)CC2C=CC(NC(=O)C=CC(F)(F)F)C2)C1 C=CCCCC(C1CC1)NC(C1(NC(c2[nH]nnc2C)=O)CC(C)(C)C1)=O C1(C)(C(=O)NCC(C)CN(C)C(C2(CC(C)C)CCNC2=O)=O)CNC(=O)C1 N1(S(=O)(=O)CC2CCCCC2)CCCCC1CC(O)C(F)(F)F FC(F)(CCCn1cc(C(=O)NC(C2CCCO2)C2CCC2)nn1)C(F)F N1(C(c2cnc(C(C)=O)s2)=O)CCC2CCC(C1)N2C(=O)CC(C)F O=C(C(Cc1ccccn1)CCCO)NCC1CCC1NC(c1cnc(Cl)[nH]1)=O C1(CNC(n2c(C)cnc2)=O)CCN(C(=O)C(C)NC=O)CC1O c1(NS(=O)(=O)Cc2ccccc2C(=O)O)ncnc2[nH]c(Br)nc12 c1(C(=O)NCCC2CCCN(C(CCC(C)O)=O)C2)cccc(C#N)c1 C(=O)(C(C)CC(C)(F)F)NCCC1CC(OC)C1.C12CCCN(C1)C2=O C1(C)(C(N2CCCC(NC(c3ccc(C(C)(C)C)s3)=O)C2)=O)CCCC1(F)F N1(C(C2(CC=C)CCC2)=O)C2CCC1CC(NC(=O)CCCF)C2 N1(C(c2c(C)nn(CC(F)F)c2)=O)CCC2(CCC2)C(NC(C2CCCC2)=O)C1 N1(C(c2c(Br)ccc(C#N)c2)=O)CCC2(CC1)CC(NC(C1(CCO)CC1)=O)C2 O=S(=O)(c1cc(I)cc(Br)c1Cl)NC1C(CO)CC1O C(=O)(C(O)CN1CCCC1)NCCC1(NC(=O)CSC2CCOC2)CC1 Cc1cn2c(n1)CCC(C(=O)NCC1(CN(C)C(C3CC4(CCC4)C3)=O)CC1)C2 C1(C(=O)OC)CCCCC1CNC(C1(O)CN(C(=O)Cc2ccc(F)nc2)C1)=O C1(CNC(Cc2c(C)cccc2)=O)CCCCCN1C(c1ccc(Cl)cc1Cl)=O c1(CC(=O)NC2(CC)CN(C(=O)C(c3ccccc3F)C)C2)c(C)cccc1F Cc1ccc2c(=NC3CCC3C#N)[nH]c(=NC(C)CCC(C)(C)C)[nH]c2c1 c1(CC(=O)NC2C3CN(Cc4noc5c4CCCC5)CC23)cc(F)c(F)c(F)c1 CC12CC(C1)C(C(N1CCCC(c3cccc(F)c3)C1)=O)CO2 N1(C(CC(C)(C)C2CC2)=O)CCC(NC(C2CCCCNC2=O)=O)C(F)(F)CC1 c1(OCC)ccc(C)nc1C(=O)N(CCCOCCNC(=O)C=C(CC)CC)C CC(C)(CNC(N1CCOCC(O)C1)=O)CS(N)(=O)=O C1(CCNC(c2ccc(Cl)cn2)C)CCC(C)(C)O1 Cc1cc(N2CCN(C)C(C(C)C)C2)nc(=NCC2CCCC2CO)[nH]1 c1(CN2C(CNC(c3c(C)cco3)=O)CCCC2)c(Br)ccc2c1OCO2 c1(CC)cccc(CNC(=O)COC2(C)CN(C(=O)CC3CSC3)C2)c1 N#Cc1ccc(=NCC2(F)CCN(C(C3CCOC(=O)N3)=O)CC2)[nH]c1 c1(C(N2C3C(NC)CC(C3)C2)=O)ccc2cccnc2c1 N1(C(C(c2cccc(Br)c2)C)=O)CCCC(C)(CNC(=O)C(C)(C)O)C1 Cc1cc(C)c(C(=O)NCc2c(C)nc(=N)[nH]c2C)c(C)c1 c1(C(C)(F)F)ccc(C(=O)NCC23CC2CN(C(C2CC2F)=O)C3)cc1 c12ccc(nc1)C(=O)N1C(CCC1C1CC1)C(=O)NCC=CC2.C1(COC)CC1.CC c1(C(N2CC(OCCC(=O)OC)C2)=O)cc([N+](=O)[O-])cc(C)n1 C1(NC(CNC(CC(C)C)=O)=O)CCN(C(c2ccc(CN(C)C)[nH]2)=O)C12CC2 C1(COC)CN(C(=O)Cn2ccc(C)n2)CCN1C(C1CCC(C)CC1)=O c1(CC(=O)NC(CC)(C)CCNC(c2ocnc2C)=O)ccc(O)c(C)c1 c1(C2(C)CC2)cc(C(=O)NCCC2CSCCN2C(=O)C(C)(F)F)n(C)n1 N1(C(C2(C=C)CC2)=O)CCC(NC(=O)Cc2cc(F)cc(Cl)c2)C(O)C1 N1(C(c2c(NC(CN3CCC(C)CC3)=O)cco2)=O)CC(C)OCC1C c1(OC)ncnc(NCn2cc(C3N(C(C4CC4C(=O)O)=O)CCOC3)nn2)c1F c1(-c2nc(OC)cc(CC)n2)cc(-c2nccn2CSc2nc[nH]n2)cc(F)c1 Cc1ncccc1CC(N1CCCC1C(C)(C)C(=O)NC(C1(CO)CC1)C)=O C(CC(=O)N1CCCOC(C)C1)(C(F)(F)F)NC(C1(CSC)CC(=O)C1)=O N#Cc1cccc(C(N2CCCC2CNC(c2cnn(C(F)(F)F)c2)=O)=O)c1 c1(C(=O)NCC(=O)NCCCCN2CCN(C3CC3)CC2)cccc2cncn12 c1(C(=O)NC2(n3cc(CN(C)C)nn3)CCOCC2)sc2cc(F)ccc2c1Cl c1(C(N2CC(N(C)Cc3ccc(C)cc3Cl)C2)=O)ccc(C#N)c(F)c1F Cc1cc(C(=O)NC2CCN(C(=O)Cn3[nH]cnc3=N)C2C2CC2)cc(C)n1 CC(C)CC(CNC(c1cccc(CCN(C)C)c1)=O)NC(=O)CCC#N c1(C(=O)NCCC2(OC)CN(C(=O)CCC3(C)CC3)C2)cnc(C)cc1C C(=O)(CCC(CC)CCC)N(C(CC(N1C(C#C)CC1)=O)C)C c1(C(=O)NCCCNC(CC(C)n2ccnc2)=O)cc(=O)cc[nH]1 Cn1cnc2c1CCCC2C(=O)N1CCCC(CNc2c([N+](=O)[O-])cnn2C)C1 C12(C(N3CC(CN(C(c4occ(C)c4)=O)C)OCC3)=O)CCCC(CO1)C2 c1(C(=O)NC2CC(CNC(CSCC(C)(C)C)=O)C2(C)C)cccc(O)c1F CCC(C#N)C(=O)NC(C(=O)N1CCOC(CC(=O)NC)C1)C(C)C c1(C(N2CC3(CN(C(C4CC(=O)OC4)=O)C3)C2)=O)cnc2ncnc(O)c2c1 c1(CC(=O)NC2CC(OC)CN(C(=O)CCF)C2)ccc2c(c1)OC(F)(F)O2 c1(CN(C)C(C2CC3CCC2N3C(=O)CCC(C)(C)C)=O)c(F)cccc1F N1(C(C(C(C)C)OC)=O)CCN(C(=O)COCc2ccc(C)cc2)CC(C)(C)C1 C1(C(=O)NCC(C(F)(F)F)n2cc(-c3c(C)scc3)nn2)CCC(=O)CC1C Nc1cccc2cc(C(=O)NCCN(C(c3cc(Br)no3)=O)CC3CC3)cnc12 Cn1c(C(N2CC3CN(C(=O)CCCc4cccs4)CC3C2)=O)cc2sccc12 N1(C(COCCCC)=O)CCC(C(F)C(=O)N(CCO)Cc2ccccc2)C1 C(=O)(C(=O)N=S(C)(C)=O)N1CC(C)C(NC(=O)Cc2cn3ccsc3n2)C1 c1(CC(=O)N(C)CC2CNCC2O)nn(C)c(=O)c2ccccc12 CCC(C(=O)NC(CNC(C1(F)CC1)=O)CC(F)(F)F)C(C)(C)CC Cc1oc2cc1CNC2=O.C1(C(N(CC(C)O)CCN)=O)CC1C1CC1 Cc1nc(O)[nH]c1C(=O)NCCC(C)NC(C1(F)CCCOC1)=O N1(C(C2(C)N(C(Cn3cc(C)c(O)nc3=O)=O)CC2)=O)CCC(O)CC(C)(C)C1 C12(C(N3C(C)CC(NC(=O)COC(F)F)CC3)=O)CCC(CC1)C2(C)C N1(C(C2C(NC(c3ccc(C)cn3)=O)CCC2)=O)Cc2ccc(C)cc2C1 c1(C(N2CCOCC(CNC(C(C)OCCC#C)=O)C2)=O)ccn2ncccc12 C(=O)(C1CCCc2cccnc21)NCC(C(C)C)NC(=O)CCSC(F)(F)F CCC(C)C(O)C(C)C(=O)N1CCCC(CC)C1C(=O)NCC1CCN1CC c1(C(N2C(CNC(c3cc([N+](=O)[O-])c[nH]3)=O)C=CC2)=O)cc2ccc(F)cc2[nH]1 C(=O)(C1OC(=O)c2ccccc21)NCC1CCN(C(CC2C(C)C2)=O)CC1 N1(C(c2ccc(C(C)(C)C)[nH]2)=O)CCN(C(=O)CCCN=[N+]=[N-])C2COCC12 c1(C(=O)NCC(CN(CC(C)C)CC)(C)C)cc(C)c(Cl)c(C)c1 c1(NC(C)=O)cnc(O)c(C(N2CCC(C)(NC(C3CC4CCC3C4)=O)C2)=O)c1 N1(CC(=O)NCC(C)CN(C)C(c2cc(O)nn2C)=O)CCOCC1=O N1(C(c2sccc2C(F)F)=O)CCCC2(CC(NC(=O)C=CC=C(Cl)Cl)CO2)C1 N1(C(CCC(C)OC)=O)CCCCC(N(C)C(c2c(C(F)(F)F)coc2C)=O)C1 CCCC(C)(C)CC(=O)N1CC(NC(c2cnc3c[nH]nc3c2)=O)C(C)C1 N1(C(C2N=C(C)SC2)=O)CC2(CCCC2NC(=O)CCOc2ccccc2C)C1 c1(NC(c2n(CC=C)nnn2)c2ccc(OC)s2)cccc2c1OCC2 N#Cc1ccccc1CCCNC(C1(O)CCCN(C(=O)COCCF)C1)=O CC(C)(COC(C1(C)CN(C(c2ccccc2)=O)CCO1)=O)C1=CCCC1 N1(C(c2cnc(CC(C)C)[nH]2)=O)CCC2CCN(C(=O)Cc3cncnc3)C2C1 CCC(CC(=O)NC1CC(C(=O)NC(CO)CC(F)(F)F)C1)C(F)F C(=O)(C(C)(O)C(F)(F)F)NC1(CNC(c2cn(CC=C)nn2)=O)CC1 N1(C(CCc2n(C)cnn2)=O)CCCC(C)(C)C1C(=O)Nc1ccc(O)c(=O)cc1 CCC(C)C(O)C(=O)N(CCCN(C(=O)CC1CC2CCC1CC2)C)C CCC(C)(O)C(=O)NCCC(C)(C)NC(c1ccc(C)o1)=O N1(C(C=C(CCC)CCC)=O)C2CCC1CN(C(C1CC13CCC3)=O)C2 n1(C(C)C)cncc1C(=O)NC1CC(N(C)C(C2CC2C(F)(F)F)=O)C1 C1(NC(C=Cc2ccc(CC)o2)=O)CCN(C(=O)CCCC2CCC2)CC(O)C1 CC1(CNC(c2n[nH]cc2NC(=O)C(F)C2CCC2)=O)CCCCCC1 C1(C(=O)NCCN(C(C(C)OCCOCC)=O)CC(C)O)C(CO)C1(F)F c1(CC)ccc2c(c1)N(C)CC1CN(C1)C2=O.c1cccc(OC)c1Br.OC C#CCCC(=O)N1CC(CNC(C2(CO)CCCO2)=O)(COC)C1 c1(C(=O)NCC2CCCC2NC(C23CC(CC(F)F)(C2)C3)=O)cc(O)cc(F)c1F C12(C(=O)OC)CCCC1(C(N1CC(C)(NC(=O)CC3CC3(Cl)Cl)C1)=O)C2 C1(NC(C(C2CC2)NC(C(C2CC2)OC)=O)=O)CCc2c[nH]nc2C1 c1(CC(=O)NCCN(C(c2cccc(OCCC)c2)=O)C)c(C)nc(O)nc1O C(CC(=O)N1CCC(NC(=O)CC(C)C(C)(C)C)CC1)(C(F)(F)F)OC C1(C(N)=O)COCC1C(=O)NC1CC(O)C1CC(=O)NC1CCCN1CCO c1(C(N(C(CCNC(c2c(C)cncc2)=O)C)C)=O)ncc(N)cc1Cl c1(C(=O)NC(CC=C)CNC(=O)C(C)P(C)(C)=O)cc2ccncc2s1 c1(C(=O)NCC(CNC(c2[nH]nnc2C)=O)OC)ncc2c(F)cccn12 c1(C(=O)NC2CN(C(C(CC)N(C)C)=O)CC(O)C2)[nH]nc2ncccc12 C(=O)(C1=Cc2ccccc2OC1)N1CC2C(NC(C(=O)NCC)=O)(CC2)C1 C#CCCC(O)C(=O)N(C1CN(C(c2ncncc2Cl)=O)CC1O)C C=CCC(CNC(C1CCCC(OC)C1)=O)C(=O)N1CCCCCC1 C1(CCOC)(NC(c2ncc(C(F)F)s2)=O)CCN(C(c2sc(C)cc2C)=O)C1 C1(C(=O)NCCNC(C(C)C)=O)CC(O)CN1C(=O)CC(C)C1CC1 c1(CN(C)CCNC(=O)NC2CSCCN2)cncc(C(F)(F)F)c1 c1(NC(C(CNC(c2cccc(CC)n2)=O)(C)C)=O)cnn2c1CCCC2 C(=O)(C(C)C(C)(F)F)NCC(C)CN(C)C(c1cc(I)c[nH]1)=O C1(c2n(CCC)nnn2)(NCc2ncc(CC(F)(F)F)[nH]2)CCCCC1CCO c1(CN(C(=O)CC2CSCCS2)C)ccc(CNC(=O)C2=CCSC2)cc1 c1(C(=O)OCC)c(NC(=O)C(C)CC)sc2c1CCC(C)(C)C2 C1(NC(C2CC(OCC)C2)=O)CN(C(C2C=CCS2)=O)CC1C(F)(F)F CC(C1=CCN(C)CC1)NC(=O)CC(C)Cc1nn[nH]n1 C(=O)(C1=CCCC(C)(C)C1)N(CCCNCC)Cc1ncccc1Cl c1(C(N2CC(CN(C)C(C3CC4CC3C4)=O)OCC2)=O)cnc2[nH]cncc1-2 Cc1ccc(C=CC(=O)N(C2CCN(C(=O)Cn3ccnc3)CC2)C)s1 N1(C(c2c(C)nc(OCC)s2)=O)CC(C2CN(C(=O)C(C)OCCOC)C2)C1 C1(NC(=O)C=CC2CCCO2)CCN(C(=O)CCOc2cccnc2)C12CCC2 N1(C(CN(C(C)=O)C)=O)CC(NC(c2cc[nH]c2C2CCCC2)=O)C(C2CC2)C1 N1(C(C2C(COC)C2)=O)CC2CCN(C(C3CNC(=O)CC3C(F)(F)F)=O)C2C1 C1(CNC(c2cncc(C(F)(F)F)c2)=O)CN(CCCC)C2CC12.c1(CC(=O)O)ccco1 c1(NC(c2ccco2)=O)ccc2c(c1)CN(C(C1(O)CCOCC1)=O)C2 N1(C(CCNC(=O)OC)=O)CCOC(CN(C(=O)C(O)C2CCCC2)C)C1 C(C)(C(=O)N=c1ccn(C2CN(C(=O)C=CC3CCC3)C2)[nH]1)N(C(C)=O)C1CC1 N1(C(C(OC)OC)=O)CCOC(CCCC2CCCN2C(C2CCOC2)=O)C1 N1(C(c2c(C)ccc(F)c2)=O)CCC2C(CCN2Cc2[nH]nc3ncccc23)C1 C1(CCOC)CCN(C(=O)C=C2CN(C(C3(OC)CCOC3)=O)C2)C1 C(=O)(CN1C(=O)Cc2ccccc21)NC1C(C)(C)CN(C(c2c[nH]c(Br)c2)=O)C1 N1(C(CN(CC#C)C(c2ccc(OC)s2)=O)=O)CC2CC(C)C2C1 C12(CNC(c3cn(C)nc3Cl)=O)COCCN1CCN(C(C1CNC(=O)C1)=O)C2 C1(NC(C(C=CC)O)=O)CCC12CN(C(c1cnc(Cl)[nH]1)=O)C2 C1(C(=O)NCC2N(C(c3nc(C)nn3C)=O)CCOC2)CC2CC(O)CC(C1)C2 C1(N(C(c2cccc(C(=O)NC)n2)=O)C)CCCCN(C(=O)C(C)C2CC2)C1 N1(C(c2ccc(CC)nc2OC)=O)CCN(C(=O)C(C)(O)C(C)(C)C)CCC1C Cc1ccc(OCC(=O)N(C2CN(C(C3(O)CCSC3)=O)C2)C)cc1 c1(NC(CCC=C(C)C)=O)ccc(NC(c2cc(Cl)cnc2O)=O)cc1C c1(N(C2CCN(S(C)(=O)=O)CC2)C(C)C)ccc2cc(Cl)ccc2n1 c1(C(=O)NCC(CC=C)NC(C2(CO)CCCO2)=O)cc(S(C)(=O)=O)co1 c1(CSC)ccc(CC2(C(=O)N)CNC2)cc1.c1(S)cccc(Cl)c1 C(=O)(CCCC(=O)NC1CCC(C)N(C(c2ccc(F)c(Cl)c2)=O)C1)NCCC C1(NC(C(CC)CO)=O)CCN(C(=O)Cn2nc(C)oc2=O)C12CCCC2 N1(C(C2C(OC(C)=O)C2)=O)CC2CC1CN2C(=O)C(C)=C1CC1 CC1CCN(C(C2CC3CCC2O3)=O)C1CNC(c1cc(C(C)(C)C)ccn1)=O C(=O)(CCCC(=O)N1CCCC1CN(C)C(c1c(C)nnn1CC)=O)NCCC N1(C(=O)CCc2cncnc2)CCCC2(CCN(S(=O)(=O)c3ccc(Br)s3)C2)C1 c1(C(N2C3C(NC(C4(COC)CC=CC4)=O)CC(C3)C2)=O)cc2n(c1)CCOC2 C12(COC)CC(NC(=O)CC3(C)CCN(C(=O)C4=CCSC4)C3)(CO1)C2 N1(C(C2CS(=O)(=O)C2)=O)CCC2(CCN(C(C3(C4(O)CCC4)CC3)=O)C2)C1 N1(C(CCCCSC)=O)CCN(C(c2ccnnc2C)=O)CC1CF c1(C(=O)NCCCNC(C2(CC#C)CCCCC2)=O)c(OC(F)F)cccc1Cl C1(CNC(C2C(=C)CC2)=O)CN(C(c2cnn(CC)n2)=O)C2(CCOCC2)C1 Cc1cc(C(=O)NC2CC(C)(CNC(c3cccc(OC(C)C)n3)=O)C2)cn1C c1(CC(N2CCC3C(NC(CCCC=C)=O)C32)=O)ccc2cccnc2c1 CC12CC(NC(=O)Cc3cncnc3)(C1)C1(CN(C(C3C=CCCC3)=O)C1)O2 S1(=O)(=O)c2ccc(c(Cl)c2)N1.C(CC(C)CCN(C)C)N.C=CCN(CCO)CC=C N1(CCNCc2cccc(C)c2)CCC2CN(c3cc(C#N)ncn3)CC12 c1(C(=O)NC2(C(N(C)Cc3nc(C)on3)=O)CCN(C)C2)ccc(F)c(O)c1 Cc1cc(N)n2ncc(C(N3CCCC3C(=O)NCCOCC3CC3)=O)c2n1 N1(C(C2C(C)=CCC=C2)=O)CC2(CCCC2NC(=O)Cc2ccc(C)cc2)C1 C1(C(=O)NC(C)CNC(=O)C(c2cccnc2)O)CC(C)(C)C1C(F)(F)F C(CC(F)(F)F)(C(F)(F)F)Nc1cnc(N(C(C(=O)N(C)C)=O)C)s1 N#Cc1cncc(NC(C2CCCCN(C(C3(C4CCCO4)CC3)=O)C2)=O)n1 N1(C(COCCSC)=O)CCC(C2CC2)(NC(c2cc(C(C)(C)C)n(C)n2)=O)C1 N1(C(CCc2onc(C)n2)=O)CC(CC(N2CCN(C(C)=O)CC2)=O)CC1(C)C C(=O)(CS(=O)(=O)c1ccccc1Cl)N1C(C)CCN(C(COCCC)=O)CC1 C1(OC)CN(C)C(C)(C(=O)N(C2COC2)C(C)C)C1.c12cccnc1NC2=O Oc1c(-c2cn(-c3ccc(OC(F)F)nc3)nn2)cccc1Cl C12(CNC(C3CN(C(c4ccccc4)=O)CCO3)=O)CCCC1OCC2 c1(NC(CC)CCOC)cc(N2CCOC(c3cnn[nH]3)C2)nc(C)n1 C1(NC(C2(SC)CC2)=O)CCCCC1NC(c1cc(C(C)C)nn1C)=O Cc1[nH]nc2c1CCN(C(c1ccc(-c3ccon3)cc1)=O)C2 CC1CCC(C(=O)NCCC2CC(NC(c3ccc(CSC(F)F)o3)=O)C2)O1 N1(C(CC(C)(C)n2cc(CCN(CCOC)C)nn2)=O)CCn2cc(C)nc2C1 c1(NC(C23CC(NCc4cc(Br)cnc4OC(F)F)(C2)C3)=O)cc(Cl)ccc1O N1(C(Cn2c(C)ncc2)=O)CC(NC(=O)CSc2ccccc2)C(F)(F)C1 n1(CC)nnc(C(=O)NCCN(C2CCCCC2)C(=O)CC2CCC(=O)N2)c1C N1(C(c2c(C)n(C)nc2)=O)CCc2cccc(O)c21 Cc1nc(-n2nc(C(C)O)nc2C2CC(=C3CCC3)C2)n(C)n1 Cc1nccc(N2CCC(OCCNC(=O)Cc3ccsn3)C2)n1 C1(NC(=O)C(=O)NC2COCCC2n2ccnc2)COc2ccccc2C1 CC(CNC=O)C(=O)N(C1CCN1C(=O)COC(C)(C)CO)C.c1(O)ccccc1 n1(C(N(C2CC2)CC2N(C(c3cncc(OC)n3)=O)CCC2)=O)ccc([N+](=O)[O-])n1 C#CC1(O)CC(C(N2CCOC(CCCN(C3CC3)C3CC3)C2)=O)C1 CCC(CC)C(C)C(=O)NCCC1CN(C(c2cc(C(F)F)[nH]n2)=O)CCCO1 C1(C(N2C(CNC(CCCCC)=O)CC(O)C2)=O)CCc2nnnn2C1 N1(C(C(CC=C)(C)N(C)C)=O)CCC2CCN(C(C3(C)CC=CC3)=O)CC2C1 C(C(N=c1cc(Cl)nc(C)[nH]1)C1CC1)NC(c1ccc(CSCCC)o1)=O c1(OC)ccc(O)cc1C(=O)N(CCCCN(C(=O)C(C)(C)N1CCCC1)C)C Cc1cc(C(=O)NCCCCNC(c2ccsc2Br)=O)ncc1CO N1(C(=O)CCSCc2ccccc2)CC2(CC(C(=O)NC3(C(F)(F)F)CCC3)C2)C1 N1(C(c2c(C)occ2)=O)C(CC(N2CCC(O)CC2C)=O)C2CCCC12 C12(C(=O)NC3C(NC(C4CC(=O)N4)=O)CC3)CC(C1)S(=O)(=O)C2 C(C(=O)NOCCO)=CCC1(CC(C)C)CC1.C1C(=O)N1CC#C N1(C(Cc2cn(C)nc2)=O)C2CCC1CN(C(C13CCCCC1C3Br)=O)C2 N1CCC2(NC(=O)C(=O)NC)CCCC12.n1(CC)cc(N(C)C(C)C)cn1 c1(C(=O)OC)cccc2c1CCOC2C(=O)NC1CCC2(CCCNC2)C1 c1(OC)cnc(NCC(C2CC2)NC(c2nc(C(C)C)oc2C)=O)nc1 Cc1ccc(N)c(C(=O)NC(C2CCCC2)CNC(=O)C(O)CC(C)C)c1 C1(C(=O)NCCCC(=O)NC)CC(OC)CN1C(C1(C(C)C)CC1)=O.C(C)(C)S c1(C(C)C)ccc(CC(=O)NCC2CCCN2C(c2ccnc(CO)c2)=O)cc1 C1(CNC(C(COC)C)=O)CC2(CCC2)CN1C(C1CC2(CCC2=O)C1)=O N1(c2ccc(-n3c(C)ncc3)nn2)CC2(CN(CC(=O)Nc3ccc(F)o3)C2)C1 c1(C(N2CC3N(C(C4C(=C)C4)=O)C(CC3)CC2)=O)ccc2c(c1)C(CC)C(=O)N2 C12(NC(=O)Cn3cc(CO)nn3)CN(C(=O)C=CC(F)(F)F)CC1CS(=O)(=O)C2 C1(C(C)C)CN(C(=O)C2=NOC(C)C2)CCN1C(=O)Cc1cc(C(F)(F)F)n[nH]1 C(=O)(CCCn1cc(C2C=CCN2C(c2csc(-c3cn[nH]c3)n2)=O)nn1)OC Cn1cnc2ccc(C(N3CC(NC(C4CCCSC4)=O)C(O)C3)=O)cc2c1=O c1(CNC(N(c2cscn2)C)=O)ccc(N2CCOCC2)c([N+](=O)[O-])c1 CCCCC(CNC(c1csc(=NC)[nH]1)=O)NC(=O)COCCOC CC1CCCC(C(N2CCCC2C(=O)NCC2(n3nccn3)CC2)=O)CC1 C1(C)(C(=O)NCC2N(C(CCc3nnc(N(C)C)o3)=O)CC2)CC(C)(C)C1 Cc1cc(C(=O)Nc2cccc(C(F)(F)F)c2)c(C)n1Cc1ccccn1 c1(CN2CCC(C#CC)C2)n[nH]c2cccc(C(=O)N(C)C)c12 c1(NC)ccc(C(=O)NC2(C)CN(C(c3[nH]ccc3C3CC3)=O)C2)cc1 N1(C(c2ccc3scnc3c2)=O)CCCCC2(CCN(c3nnns3)C2)C1 C(C)(C)(C(=O)NCCOCCN(C(=O)C=CC1CCCC1)C)OC Cc1c(NC(=O)C(c2ccnn2C)N)cccc1CO.c12c[nH]cc1CNC2=O C1(COC)CN(C(=O)C(c2ccccc2Cl)C)CCN1C(=O)Cc1cncnc1 N1(C(c2c(C)scn2)=O)CCC(NC(C23COC(CF)(C2)C3)=O)C(F)C1 C(=O)(C(O)CC(N)=O)N1CCC(CC(=O)NC2C(C)COCC2)CC1 C1(CCCCCC)CCCN(C(=O)C(=O)N(c2ccc(CC)s2)CCCC2CC2)C1 Cc1[nH]nc(CO)c1C(=O)NCC1C2CN(C(c3cnc(N(C)C)cn3)=O)CC12 c1(C(=O)NC(CCNC(C2(CC=C)CC=CC2)=O)C)cccc2c1oc(=O)n2C c1(C(N(C)CC2(NC(CS(=O)(=O)NC)=O)CC2)=O)nccn2nccc12 c1(CN2CCCC(NC(c3ccn(C4CCC4)n3)=O)C2)cc(Cl)ncc1F C#Cc1cccc(CC(=O)NCCOC(C)(C)CNC(C2SCCC2C)=O)c1 C1(CNC(C=CC(CC)=CC)=O)CN(C(c2ccncc2C)=O)CCC12CCOC2 C1(NC(c2cscc2C2CC2)=O)CCCN(C(c2cnncc2)=O)C1 c1(N(C)Cc2cnc[nH]2)nc2cc[nH]c2c(=NC2CCC(=O)N(C)C2)[nH]1 c1(C(C)(C)C)ccccc1NC=O.C1(NCc2ccc[nH]2)CCCN1C(=O)O C(=O)(C(C)(C)C(C)C)NCC1CCCC(NC(c2cc(C)sc2)=O)C1 N1(C(C(C)(C)NC(CCc2n(C)ncn2)=O)=O)CC2CC3CC2C1C3 O=C(CS(=O)(=O)CC(F)(F)F)NC1CN(C(=O)COC(F)(F)F)CC1O N1(C(CCC(=O)NCC)=O)CCN(C(=O)C(CO)OC)CC1c1ccccn1 c1(-n2c(N3CC(CNc4cc(C)ns4)C(C)C3)nnn2)ccc2n[nH]cc2c1C n1(CC)ncc2cc(C(=O)NCC3CC(CNC(C4(Cl)CC4)=O)CO3)cnc12 Cc1cc(O)ccc1CC(=O)NC1CC(CNC(=O)C(C)N(C)C2CC2)C1 C1(C)(COCCNC2CCCCN(C(=O)OC(C)(C)C)C2)CCS(=O)(=O)CC1 C1(N(C(=O)Cc2ccsc2)CCC)CCN(C(=O)CSC2CCOC2=O)CC1 c1(C(=O)NCC(C)CN(C)C(c2cc(O)nc(O)n2)=O)ccnc2ccncc12 c1(C(CN(C(C2CC(F)(CF)C2)=O)CC)O)cccc(C(F)(F)F)c1 C1(O)(CC(=O)NCC(C)Sc2nc[nH]n2)CCN(C(=O)CCC2(C)CC2)CC1 c1(OC)cnc(Cl)[nH]c1=NC1CC(CCNC(=O)CC2CCCC(C)C2)C1 Cc1cc(C(=O)NCC23CC(CO2)N(C(C2CC(O)C2)=O)C3)cnc1C(F)F c1(C(N(C2CCN(C(C3C(CCC)C3)=O)C2)CC2CC2)=O)cc(O)nc(Br)c1 C1(CNC(C(C)SCCCC)=O)CC2(CO1)CN(C(C1(C)CS(=O)(=O)C1)=O)C2 Cc1scnc1C(N1CC(NC(=O)CNC(=O)OCC2CCCC2)C1)=O N1(C(c2c(CC)n[nH]c2)=O)CCCCC1CCNC(C1CC2CCC1C2)=O C12(CCNC(C(C)(C)SC)=O)CCC1CN(C(=O)C(C)(C)c1cc[nH]n1)C2 CN1CCOCC12COCCN(C(C1CCCC3CN(CC4CC4)CCC13)=O)C2 C1(CNC(COCC)=O)(CNC(=O)CC(C)F)CC1(F)F c1(CC)ccc(O)c(C(N2CCC(C)(CCNC(c3cnc(C)[nH]3)=O)C2)=O)c1 N1(CCCc2cn(CCC)nn2)CCOC(c2nc(C)no2)C1.c1ccccc1 c1(C(C)N(C)CC2CC2C2CC2)ccc(C(N)=O)nc1 c1(C(N2CCC(CNC(C3(C)CC(=C)C3)=O)(OC)C2)=O)c(Cl)cncc1Cl N(C(=NCCC1(C)CCCC(=O)N1)NCCN1CCOCC1(C)C)C(COC)C N1(C(C)=O)CCC2(CCCC2N(C(=O)CCC(C)=O)Cc2ccccn2)CC1 C1(NC(C2CC=C(C)CC2)=O)CC2CCC(C1)N2C(C1(C)CC(C(F)(F)F)C1)=O c1(CCNC(c2cccs2)=O)n[nH]cc1NC(=O)Cc1csnn1 C1(F)(C(=O)NCC2(O)CN(C(c3c(C(C)C)ocn3)=O)C2)CCOCC1 Cc1c(CC(N2CCCC(CNC(c3cc(Br)cs3)=O)C2)=O)[nH]c2ccccc12 Cc1ncc2c(n1)CC1CCC2N(C(C2CC2C(F)F)=O)C1 N1(C(C2C(COC)CC2)=O)CCN(C(C2(NC(=O)N(C)C)CC2)=O)CC1 c1(C(N(C(C)C(C)C)CC)=O)cccc2ccn(C)c12.C12CN(C1)C(=O)N2 C1(C(=O)NCCC(C(=O)NC2CCCOC2(C)C)OC)C2CCC(C2)C1C C1(C(F)(F)F)(C(=O)NC2CC(C(N(C(CN(CC)CC)C)C)=O)C2)CC=CC1 N1(C(c2ccnc(C)n2)=O)CC(NC(=O)C(C)NC(=O)C2CC2)CC(O)C1 S(=O)(=O)(c1ccccc1C#N)Nc1cc(COCC)cc(NC2CC(SC)C2)c1 CC(C)(F)CCC(=O)NCC1(O)CCN(C(c2conc2C2CCCO2)=O)C1 c1(OC)ccnc(C(=O)N(C(C)CNC(c2cnc(C(C)O)s2)=O)C)c1OC C(c1ccncn1)=CC(N1C(CC(=O)NCC2(COC)CCOC2)CC1)=O CC1Cc2cc(C(N(C3CN(C(=O)CC45CCC(CC4)OC5)C3)C)=O)ccc2O1 c1(CN2CC(C(N3CC4C(NC(C)=O)C4C3)=O)C2)ccc(C)c(F)c1F C1(C2CCN(C(=O)C(CO)C(C)(C)C)CC2)(CNC(C2(C)CC2)=O)CCOCC1 Cc1cccc(C(=O)NC2COCC2NC(c2ccc(CO)o2)=O)n1 C(C)(C)(CCC(=O)N1CCCC(O)(C(=O)NC2CC2C2(C)COC2)C1)OC N(C(=NCc1nc(C(C)O)n[nH]1)N1CC(c2ccccc2)C(C)C1)C(C)C c1(C(C(=O)NC2CCCC(NC(c3nnn(C)n3)=O)C2)(F)F)cc(Cl)ccc1Cl c1(C(C)C)ncccc1C(=O)NC(C)CCCNC(C1CC12CC2)=O C(=O)(C1=CC2(CCOCC2)C1)N1CCN(C(CCc2cc(C)on2)=O)C(C)C1 c1(CC)ccc(N(C(c2n[nH]c(C)n2)C(=O)NCCCF)CC)cc1 c1(C(N(CC(=O)O)Cc2scc(C)n2)=O)cccc2cc(Cl)ccc12 N1(C(C(C)N(C(c2cc(OC)n[nH]2)=O)CC)=O)CC2CCC(CC2)C1 Cc1cc(F)ccc1CCC(=O)NC1CN(C(c2nc(Cl)ccc2N)=O)CC1F C1(C(=O)NOCC(C)(C)O)(NC(Cn2ncc(C)c2)=O)CCCOC1 C12CCN(C1C(C)C)C(=O)CN(CC(F)(F)F)C2=O.c1(CC)cc(Cl)n(C)n1 N1(C(C23CC(CCC)(C2)C3)=O)CCC(F)(C(=O)NC2C=CCC2)C1 c1(N2CCC(NCCC(C)(C)CCCO)C2)nc(NC(C2C(CCC)C2)=O)cc(C)n1 C(C(C)(O)C(=O)N1CCN(C2CCN(C(=O)CCC3CC3(F)F)CC2)CC1)OC CC1CCCC(C(N2CC(C(C)NC(c3cnnn3C)=O)C2)=O)CC1 C1(CCC)CCCC1C(=O)N(CCC(=O)NCCc1ncc(C)o1)CC c1(OCC(=O)OC)ccc(CNC(N)=O)cc1CC(C)C.C1(=O)CO1 C(N=c1[nH]c2c(c(=NCc3cnc4n3CCC4)[nH]1)CCCC2)c1nc(CC)sc1 Cc1cc(C)c(CC(=O)NC(C)C(C)NC(=O)CC2COCCOC2)c(C)c1 c1(C(=O)NCC#CCNC(C(C)C2CCOC2)=O)cc2n(c1)CCCC2 c1(C(=O)NC2CCN(C(CC3COC(C)(C)O3)=O)CC2F)ncc2n1CCCC2 C1(C(=O)NCC(=C)CCNC(C2CCCS2(=O)=O)=O)CCOCC12CCCC2 c1(N(C(C)C)C)ccc(C(=O)NCC2(NC(C34CSCC3C4)=O)CC2)cc1 C1(NC(CCNC(COC)=O)=O)CC(NC(=O)CN(C)C)C(O)C1 N1(C(c2[nH]nc(OC)c2Cl)=O)CCC2CCN(C(=O)C(c3cnn(C)c3)C)C2C1 C1(CNC(C2(COC)CCCC2)=O)CN(C(=O)C(N2CCOC2=O)C)CCCO1 c1(C(=O)NC(CNC(c2n(CC)nnc2)=O)CO)cnn(CC)c1C1CC1 O(NC(=O)CCS(C)(=O)=O)C(C(=O)Nc1n(CC)ccn1)C C1(F)(C(N)=O)CCCN(C(=O)Cc2cncnc2O)C1 C=CCCC(O)CN(C)C(C1(F)CCN(C(=O)CCNC(=O)COC)C1)=O C(=O)(C(C)CC(=O)c1cccc(F)c1)NC(C(C)C)(C)CNC(=O)CC1CSC1 C#CC1(O)CCCN(C(c2cnc(OC)cc2C)C(=O)NCCCC)C1 c1(C(=O)NC(CC)CN2CCCC2)conc1C(C)NC(=O)C(C)n1ccnc1 N1(C(CN(C(=O)C(F)COC)CCC)=O)CCCC(F)C1 C1(C(=O)NCC2(F)CC(CNC(C(C)OCCCC)=O)C2)CCC2(CC1)CC2(F)F C(=O)(C1=C(C)CCOC1)NC(C1N(C(CC=C)=O)CCC1)C CCC(C)C(CNC(=O)CCN(C(=O)CCc1cn(C)cn1)C1CC1)OC C1(C(N(C2CCN(C(c3cnc(C)s3)=O)C2)C)=O)CCC(=O)N1CCC(F)(F)F N1(C(C(C=C)O)=O)CCN(C(c2cccc(SC)c2)=O)CC1CCC Cc1[nH]c(C)c(C(N2C3CCC2(CNC(C2CC4C=CC2C4)=O)CC3)=O)c1C c1(C(=O)NC(CC)CO)cc2cc(-c3cccc4c3ccn4C)cnc2[nH]1 c1(CNC(C(N)C2(CCC3CC3)CC2)=O)cccnc1 C1(O)(CNC(C=CC)=O)CCN(C(=O)Cc2ccnc(Br)c2)C1 C1(NC(C2C3(CN(C(C(C)Oc4ccccc4)=O)C3)C2)=O)CC2CC1OC(=O)N2 c1(C(=O)NC2(CNC(C3C(OCC)C3)=O)CCCC2)cccn2nnnc12 CCC(CC)CC(F)C(=O)NC(C(=O)NCc1nocc1C(C)C)C(C)C c1(CC(=O)NC(CN(C(c2cn(CC=C)nc2)=O)C)C)ccc2c(c1)CCCO2 Cc1cccc(CCC(=O)N2CCC2c2ccc(Br)cc2Cl)c1Br C(=O)(CC(CC)CC)NCC(=C)CCNC(=O)CCc1cccc(OC)n1 CC1OC2(C)CC1(C(N1CCC1CNC(c1cnsc1)=O)=O)C2 C1(C(=O)NC2CC(NC(C(c3cnn(C)c3)C)=O)C2)C2COCC12 N1(C(CC=C=C)=O)CC(C2CCCN(C(c3cc(C(C)(F)F)on3)=O)C2)C1 c1(NC(=O)CCOCCC(c2ccc(C)cn2)C)cc(Cl)ccc1Cl CN1CCCC(C(N2CCN(C3CN(C(=O)CC4CCSC4)C3)CC2)=O)C1 C1(CC)C(NC(=O)COCCC(C)C)CCN1C(C1CCNC(=O)C1)=O c1(C(C(=O)NCC2(O)CC(CNC(=O)Cn3cncn3)C2)=O)ccc(Cl)cc1 C(C(F)F)(C(C)(C)C)NC(c1cc(CCNC(c2n(C(C)C)ccn2)=O)on1)=O C(C(C(=O)NCC(O)CC(F)(F)F)C(C)(C)C)NC(CN(CC(=O)OC)C)=O C1(C(N2CC(C#C)C2)=O)(COC)C=CCN1C(c1ccc(O)cn1)=O CCCCCCCCC(=O)N1CCC2CN(C(c3scc(OC)c3OC)=O)CC12 N1(CC)CC2CCC(C1)N2CCF.C12(CC=CCC1)C(=O)NC2 c1(OC)nc(C2C(n3cc(NC(=O)NC(C)(C)CN(C)C)nn3)CC2)ncc1F c1(C(=O)NCC(CNC(C=CCOC)=O)C)cc2occc2s1 C1(CNC(C(CC)OC)=O)CCCCN(C(=O)C(F)(F)C2(OCC)CCC2)CC1 C(=O)(C1=NN(C)C(=O)CC1)N1C(C(=O)NCc2cc(C)cc(C)n2)CCC(C)C1 c1(C(N2C3C(NC(c4ccoc4C4CC4)=O)CC(C3)C2)=O)cc2c(s1)CCOC2 C(CC(=O)NCC(C)(C)NC(=O)CCOCC(F)(F)F)C(C)=O.C(CN(C)C(N)=O)N C=C(C)CC(C(=O)N(C(C)(C(=O)NCCC(O)C1CC1)C1CC1)C)OC Cn1ccc(C(C)(C)C(=O)NC2CN(C(=O)CC3CC3c3ccccc3)C2)n1 c1(C(=O)NCCN(C(c2ccc(O)nc2C)=O)CC)ccc(C)cc1[N+](=O)[O-] N1(C(c2cncc(C)n2)=O)CC2(CCC2)CCC1CO N1(C(Cn2nc(C)n(C)c2=O)=O)CCCC2(NC(c3ncncc3Cl)=O)CC2C1 Cc1nc(-c2nn[nH]n2)ccc1NC(C1CCCN(c2nccs2)C1)=O Cc1cncc(C(=O)NC2CCN(C(c3cc[nH]c3C3CC3)=O)C2C(C)C)c1C C1(CC)C(C)CCCN1C(c1cc(=O)c(NC(c2ccn(CCC)n2)=O)c[nH]1)=O N1(C(c2c(C)oc(Cl)n2)=O)CC(NC(c2cn(C)nc2Cl)=O)CC12CCOC2 c1(C(N2C(C(C)(C)O)CCC2)=O)ccc(F)nc1 c1(O)ccc(F)cn1.CC1(c2cn(CCO)nn2)CN(N2CCC(C=O)C2)C1 c1(N(CC(=C)C)C)nc(=NCC23CCCCC2C3(F)F)[nH]c2c1CSC2 c1(C(=O)NCC2(C)CC(NC(c3ccoc3CC(N)=O)=O)C2)ccc(F)cc1F c1(NC(=O)NC2COCC(C)(C)C2)nc2ccc(Cl)cc2s1 C1(OC)(OC)CC(C(=O)OC2CCN(c3cc(C)nn3C)C2=O)C1(C)C C1(NC(C2CC(CCNC(C3(CO)CCCC3)=O)C2)=O)CCc2nn[nH]c2C1 Cc1cc2n(n1)CCN(C(C1CC(C)N1C(=O)CC(C)CC(C)(C)C)=O)C2 CCCC(C)(C)CC(=O)NC1CCCCN(Cc2cc3sccc3[nH]2)C1 C(=O)(C(O)C(C)C)NCC(C)N(C(C(C)OCCC=C)=O)C N1(C(C(CC)N2CCCC2=O)=O)CC(OC)CC1CNC(=O)CC(C)C1CC1 c1(C(=O)NCC2(NC(c3cc(COC)[nH]n3)=O)CCC2)ccc2[nH]c(=N)oc2c1 c1(OCC(=O)NC2CC(CCNC(C3OCCC3C(F)(F)F)=O)C2)ccccc1 C(c1ccc2[nH]ccc2c1)=CC(N1C2CN(C(C(C(C)(C)O)F)=O)C(C2)C1)=O C1(CCC)CCCC1C(=O)NC1(COC)CN(C(c2cnc(S)[nH]2)=O)C1 Cc1ccc(C(N2CCC(CCC(N3CCC(CC4CCC4)C3)=O)C2)=O)c(C)c1 C1(O)(CNC(C2C(C=C)C2)=O)CCCN(C(c2ncccc2C(F)F)=O)C1 CC(C)C#CC(=O)N(CCCCn1cc(C2CCCN2C)nn1)C1CC1 c1(OC)ccc(OC)c(C(=O)NC2CCC(NC(C3CN(C)C(=O)N3)=O)C2)n1 N1(C(c2c(OCC)n[nH]c2)=O)CCC(O)(CCNC(c2c[nH]nc2C)=O)C1 n1(CC(=O)NCC(C)N(C(=O)Cc2ccc(Cl)cc2Cl)C)cc(F)ccc1=O c1(C(N2CCC3(CC2)CC3(F)F)C(=O)NC(C)(C)C)cc2c(cc1Br)OCO2 C1(C(N2CCCC(CCCC)C2)=O)CCC2CCC1N2C(c1ccc(C)[nH]1)=O N1(C(C2OCCN(C)C2=O)=O)CC2OCCN(C(c3cscn3)=O)C2C1 C=CC(C)C(C)C(=O)NCC1(F)CN(C(=O)C(C)(C)C2CC2)C1 c1(CCC(=O)NC2CN(C(C3(C)CCCS3)=O)CC2O)ccc(F)cc1Br c1(C(=O)NCCn2cccc2)nc2ccc(-c3cc4ccccc4[nH]3)cc2s1 c1(C(=O)NC2(CC=C)CN(C(c3cnc(OC)c(C)c3)=O)C2)cc(C)c(C)nn1 Cn1cc(C=CC(=O)NCCC2(CNC(N)=O)CC2)nn1.C1(CO)C(=O)N1 c1(NC(C(CCF)NC(C(C(=O)OC)OC)=O)=O)cnc2ncnn2c1 c1(C(N2C(CNC(C(C)(C)N3CCCC3)=O)CC2)=O)ncc[nH]c1=O C(=O)(CC(F)(F)F)NCC(=O)N(CCCCC1C(CC)(CO)CC(=O)N1)C Cc1cc(C(C)C(N2CCC(O)(CCNC(C3(N(C)C)CC3)=O)C2)=O)cc(C)c1 c12ccccc1C(C)(C)c1cn-2nn1.c1(C(N(C(CC)(C)C)CC)=O)ccccc1 O=C(CC1OCc2ccccc21)NCCNC(c1c[nH]c2cc(Cl)c(Cl)cc12)=O N1(C(C2CCCN(C)C2)=O)CC(NC(=O)CCOC2COC2)CC12CCCCC2 c1(OC)nc(C(=O)NC(C2CCCCN2C(=O)C2=CC(C)(C)C2)C)cc(O)n1 N1(C(c2nc(C)sc2C)C(=O)NCCCF)CCCCCCC1 c1(C(N2CCC(F)(CNC(c3cnc(O)o3)=O)C2)=O)cc(F)cc([N+](=O)[O-])c1 N1(C(C2N(C)CC(C)(C)C2)=O)CCC2(C1)CN(C(C1(N(C)C)CCC1)=O)C2 N1(C(C(C=C)CC)=O)CCC(C)(C)C(CNC(=O)CCSC(F)(F)F)C1 C(=O)(CC(CCC)NC(C1(C#C)CC1)=O)NCc1ccncc1O C1(CNC(c2cc(C)nn2C2CC2)=O)CC2CCC(C1)N2C(C1CC=CCC1)=O C1(NC(CCCc2[nH]c(=N)sc2)=O)CC2CC(NC(=O)Cc3ccoc3)C1C2 n1(CC(=O)NCC2CCCC(NC(C(C)CCO)=O)C2)c(=O)oc2ccccc12 Cc1cnc(C(=O)NCC2(C)CCN(C(c3cscc3C3CC3)=O)C2)cc1C#N Cc1oc([N+](=O)[O-])cc1C(=O)NCC1CC(O)(CNC(C2CC23CC3)=O)C1 c1(C(=O)NC2(C(=O)NC(CCC=C)C)CC2C)n[nH]c(COC)c1C N1(C(CC2CC(=O)NC2)=O)CC(NC(C2CN(CC(F)(F)F)C2)=O)C2(CC2)C1 C(CCC(C(=O)NC1CC(CO)(CO)C1)NC(c1cc(C)c[nH]1)=O)OC C1(CNC(C(c2cccs2)NC(C=NOC)=O)=O)CCC(=O)NC1 CCC(C)CCCC(=O)NC1(CCC(=O)NCC(O)Cn2cccn2)CCC1 c1(CCC(=O)NCC2CN(C(C3C(Cl)(Cl)C34CC4)=O)C2)c(Cl)cccc1Cl c1(C(N2CC(O)(CCNC(C3CC(C)OC3)=O)C2)=O)cccc2c1CCS2(=O)=O Cc1onc(Br)c1C(=O)NC(C)CCN(C)C(c1ccccc1F)=O c1(CNC(C(C)C2CC2)=O)ccc(C(=O)NCC2CCCO2)nc1 C1(CC#C)(C(=O)NC(CN(C)C)CC)CCN(C(c2scnc2Cl)=O)C1 C1(C(Cn2c(N3CCC(C)CC3)nnn2)=O)CC2CNCC2(c2ccccc2)C1 C1(NC(c2c(C)cncn2)=O)COC2(C1)CN(C(c1ncc(F)cn1)=O)C2 Cc1nc(C(N2CC(CNC(c3csc(CO)n3)=O)C(O)C2)=O)c2ccccn12 CCC(CC(C)CO)NC(=O)CCCCN(C(=O)CCC1(C)CC1)C Cc1ccc2c(c1)N(C(c1coc(CNC(=O)COCC3CCOC3)n1)=O)CC2 N1(C(c2ccc(CCC)cc2)=O)CCCC2CN(C(=O)CCC(C)SC)CCC12 C(C(CC)(CC)NC(=O)C(O)C(C)c1ccccc1)NC(C=C(CC)CC)=O CS(=O)(=O)c1ccc(F)c(C(=O)NCc2cc3n(c2)CCNC3)c1 CC(C)(CC(=O)NC1CCC(CNC(=O)CCn2cnc([N+](=O)[O-])c2)C1)C(F)F N(C(=NCCCF)NCCOCCN(c1ccoc1)C)CC=C c1(C(C)=O)cccc(C(=O)N(C)CC2CCN(C(c3ccsn3)=O)CC2)c1 N1(C(C(C)(C)OCC)=O)CCN(C(=O)C(=Cc2cccnc2)F)CC(C)(F)C1 C(=O)(C(C)(C)C(=O)NCCN(CCCN(C)C)C(=O)Cc1ccccn1)NC C=CCC(C)(O)C(=O)N1CCC1CNC(c1cc(C)c(O)nn1)=O N1(C(Cn2ccc(C)cc2=O)=O)CCC2C(NC(c3ccc[nH]3)=O)C2CC1 S(=O)(=O)(c1cnc(NC2CC(O)C2(C)C)c(Cl)c1)N(C)Cc1c(OC)cccc1 C1(C(=O)OC2(CC(=O)NCCC(N3CCCC3)=O)CC2)SCCCS1 Cn1cnc2cc(C(N3CCCC(CC(=O)NCC4CCC(C)(C)O4)C3)=O)ccc12 c1(C(=O)NCCC#C)cc(F)ncc1NC(c1ccc(CCO)cc1)=O CCC(CC)C(=O)N1CCN(C2CCN(C(=O)CCC3CCCCO3)C2)CC1 C1(C(N)=O)CCC(NCC2CC3CCC2O3)CN1 N1(C(C2CC(OC)C2)=O)CC(c2cn(CC3CCCOCC3)nn2)C(O)C1 N1(C(C23CCC(OC)C2C3)=O)CCC2(C1)CN(C(c1cc(F)ccc1Cl)=O)C2 c1(C(C(=O)NC2CCOC2)N(C2CCCC2)Cc2scc(C)n2)cnccc1C C1(CC)(NC(=O)C(C)O)CCN(C(c2csc(I)c2)=O)CC1 C1(=O)CC(CNC(c2ccc(OC)s2)=O)NCC1=O.c1(OCC)ccccc1.CO C(=O)(C#CC1(C)COC1)N1CCN(C(C2(OCC)CCSCC2)=O)CC1CCO Cc1cc(O)ccc1C(=O)NCC1CCC1NC(=O)C(C)(C)C1CCCCO1 N1(C(C2CC(C(F)(F)F)(OC)C2)=O)CCC(C)(NC(c2ccc(C)cc2)=O)C1 CC1(C)CC(CC(=O)NC2CCC2)N(C(C2COCCO2)=O)C1 c1(CCNC(COCCNC(=O)CCC2N=N2)=O)cccc(O)n1 C1(CN(CC(CC)OC)C)(NC(=O)CSC)CCc2cc(Br)ccc2C1 c1(CC)ncc(Cl)c(C(=O)NCC(C)(C2CC2)NC(c2sc(=N)[nH]c2C)=O)n1 c1(OC)ccc(-c2nccn2CN2CCCC(C)(CCO)C2)cc1OC N1(C(CCSC)=O)CC2CCOC2(CNC(c2n[nH]c3c2CCC3)=O)C1 C(=O)(C=CS(C)=O)N(C1CCN(C(c2cncc(O)c2)=O)C1)C N1(C(c2n(CCC)ncc2)=O)CCC2(CCN(C(=O)C(C)NC(N)=O)C2)C1 C(=O)(CCCCCn1cc(CCCCc2ccn(C)n2)nn1)O.C(C)(C)(C)O C1(SC)CCc2nc(C)[nH]c2C1.c12cccc(c1)N(C(=O)CN1CCOC(C)C1)C2 c1(CN(C(c2cn(CC#C)nc2)C(=O)NCCC2CCC2)CC)ccccc1Cl C1(C(=O)NCC(CC=C)NC(C2(F)CCCCC2)=O)CCCSC1C c1(CC)ccnc(C(=O)NC2CCCC(C(=O)N(C)C(C)C3CC3)C2)c1 CC1(CNC(c2csnc2Cl)=O)CCCN1C(C12COCC1C2)=O c12ccc(cc1F)-c1nc(cs1)C(=O)N1CC(C1)N2.N1(CC)CCCS1(=O)=O O=[N+]([O-])c1c[nH]c2c(Br)cccc2c1=NC1CC(OCCO)C1 CC(C)CC(F)(F)C(=O)NCC1(C)CCCN1C(=O)CC(N1CCOCC1=O)C c1(NC(C)=O)ccc(C(N2CCC(CC(=O)N(C)Cc3ccsc3)C2)=O)nc1 c1(C(=O)NC(C)CCNC(=O)CSCc2ccncc2)[nH]cc2c1CCC2 C12CCCN1S(=O)(=O)C(C)COC2=O.CCCSCC1CC1 CC1=C(C(=O)NCCC(C(C)C)NC(=O)CC(c2c(C)noc2C)C)SCCO1 CC1Cc2ccccc2C1Nc1nccc(-c2ccns2)n1 C1(C(N(CC(C)N(C(=O)C=Cc2ccoc2)C)C)=O)CC(C)(C)OC1(C)C c1(C)nnc2n1CCN2C.C1(CCC)CCCCO1 c1(C(=O)NCCCNC(CC(C)C2CCCO2)=O)cc(Cl)c(F)cc1F c1(C(=O)NC2CCCN(C(COCCC(C)C)=O)C2)cc2occc2s1 c1(COC)nc(N2CCCCC(N(C(C)=O)CC)C2)cc(C)n1.C1(=O)C(C2CC2)O1 C=C(Cl)C(C)(C)C(=O)N1CCC2(CC2NC(c2cc(C(=O)OC)co2)=O)C1 C1(NC(c2cncc(-n3c(C)c(C(=O)O)cn3)c2)=O)CCS(=O)(=O)C(C)C1 C1(NC(CC2C(C)(C)C2(C)C)=O)CC2(CCN(C(=O)C(F)CC3CCC3)C2)C1 N#CC12CC(C(=O)NCC3(NC(=O)C(F)=C4CCCC4)CCOC3)(C1)C2 c1(CCC(=O)NC2C(NC(C(CN(C)C)O)=O)C2)ccc2ccccc2n1 C1(NC(C2(CC(N)=O)CCCC2)=O)CCOC12CCN(C(C1CCO1)=O)CC2 Cc1ccc(C(=O)NC2CC(n3cc(C4CCC(O)(C(=O)O)C4)nn3)C2)c(C)n1 c1(C(=O)NCC23CC(NC(C4CC(C)OC4)=O)(C2)C3)noc2c1COCC2 CC1C(NC(=O)C#CC(=O)NC2CC2)CCN1C(c1cn(CC(F)(F)CO)nn1)=O CC(C)CC(C(=O)NC)N(C(=O)CC1CCN(CC#N)C1)C Cc1ccc(C(=O)NC(CN=[N+]=[N-])C(=O)NCC2(O)CCC2)c(C)n1 N1(C(C2(CCO)CC2)=O)CC(O)(C(F)C(=O)NC2CC2c2cccnc2)C1 c1(C(=O)NC(C(N2C(C)(CCC)CC2)=O)CO)ccncc1F C1(CC(=O)N(CCNC(c2ccc(CC)s2)=O)C(C)C)CCCS1(=O)=O C(=O)(CC(C1CC1)NC(=O)CC1COCCO1)N(C1CCNC1=O)C N1(C(Cc2c(C)occ2)=O)CCC(O)(C(C)NC(c2ccco2)=O)CC1 CC1CC2CN(C(C34COCC(C3)C4)=O)CC2N1C(=O)Cn1cnnc1 CC1(C)CC(C(N2CCC3CC23)=O)CN1C(=O)Cn1cc(Cl)cn1 C1(CNC(C(CCC)C#N)=O)CC2CCCC2N1C(=O)Cc1nc(C)cs1 C=CCCC(F)(F)C(=O)N1CC(CNC(C2CCCCCC2)=O)C(F)(F)C1 N1(C(CC2(NC(CC(C)CN(C)C)=O)CCC2)=O)CCC12CC(O)C2 C1(CCC)(NC(C2(CC)CCCO2)=O)CCCN(C(C2(CO)CCCCO2)=O)C1 CN=c1ccc(C(N2CC3(CC3)CC2CNC(c2cn(CCO)nn2)=O)=O)c[nH]1 c1(NC(C(C)NC(c2c(C)cn(C)c2)=O)C(C)C)nc2ccc(Br)cc2o1 C(=O)(C(C)(C)CO)NCCN(C(C)C)C(c1cnn(C(F)(F)F)c1)=O C1(NC(C(C)OCCCCN(C)C)=O)(NC(=O)C2CC2)CC(F)C1 C1(C(=O)NCC(=C)CCNC(C2(C(=O)NC)CC2)=O)C2Cc3c(Cl)cccc3C12 CC1CN(C(c2n[nH]cc2-c2ccccc2)=O)CC1CCNC(c1cn[nH]c1)=O C1(C(N(CCCCNC(c2cc(CO)nn2C)=O)C)=O)CCn2c(O)nnc2C1 c1(CNCC(=O)OC)nc(N2CCC(C)(SC)C2)cc(C(F)F)n1.C(C(O)C)OC N1(C(c2ccc(CC)s2)=O)CC(CC(=O)NC(c2ccccc2)C)CC1(C)C N1(C(C(CO)NC(N)=O)=O)CC(NC(c2cc(Cl)cnn2)=O)CC12CCCC2 CC(CCC(C)(C)C)C(=O)N(CCC(C)NC(=O)COc1ccc(F)c(Cl)c1)C C1(N(C(=O)COCCc2cccs2)C)CC2CC1N(C(=O)Cc1ccnn1C)C2 N1(C(CC2(C)CC2)=O)CCN(C(=O)COc2ccc(F)cc2)CC(O)C1 C1(C(N2CC3CC3C2)=O)Cc2nccnc2CN1C(=O)CC1CCOC1 Cc1cc(C(=O)NCC2CC(NC(=O)C3=CCCC3C)C2)cc2nc[nH]c12 c1(C(=O)NCC2OCCN(C(Cc3cc(C)ncc3)=O)C2)cc(CO)ccc1C c1(C(N2C(C(C)(C)C)C(NC(C3CCCC(=O)O3)=O)CC2)=O)c[nH]cc(Cl)c1=O CC1(c2cccc(C(F)(F)F)c2)CCCN(C(=O)Nc2ccc(B(O)O)cc2)C1 C(CC(=O)NCCC1CCCC2CC12)(C(F)F)NC(=O)C1=NOCC1 C(C)(CC(=O)NCCCOCCNC(=O)CCc1nccs1)(C(F)F)N(C)C C12CCN(C1C(C)C)C(=O)CNC2=O.Cc1ncc(CCC(F)F)s1 CCC1=NOC(CC(N2CCN(CCNC(C3CCCN(C(N)=O)C3)=O)CC2)=O)C1 c1(OCC)ccsc1C(=O)N(CC(CC)NC(c1cnc(O)o1)=O)CC C1(F)(COC)CC(N=c2cc(C)nc(COC)[nH]2)C1.N12CCC(C)(C1)C2=O C1(C(=O)NC2(CC=C)CN(c3nc(CC4CCC4)ns3)C2)CCC2CCCCN12 C(C)(CCCC(=O)NC1CCCCC1C#N)NC(c1cc(C)nn1C)=O n1(CC)cnc(C(=O)NC(C)C(C)NC(C2(c3ccsc3)CC2)=O)c1 C(C(CC(F)(F)F)NC(c1ccnc(N2CCCC2)c1)=O)NC(C1C(OC)C1)=O N1(C(C2CCN(OC)CC2)=O)CCCC2(CCCCC2NC(=O)C(C)N(C)C)C1 C1(O)(C(C)NC(=O)CCNC(=O)CO)CCN(C(C23CC=CC(C2)OC3)=O)CC1 N12CC(O)CC1CC(=O)NCC1C2CCCCC1.[N-]=[N+]=NCC=O N1(C(c2ccc(OC)cc2C)=O)CC2CCC(C1)N(C(c1cn(C)c(O)n1)=O)C2 C(CC(C(=O)NC(c1ccccc1O)C)NC(=O)C(C)c1cc[nH]n1)=CC N1(C)CCN(C(=O)CNC(=O)C(F)(F)F)C(C)C1.C1(OCC)CCCC1C(=O)O CCCC(C(=O)Nc1ccccc1COC)NC(=O)C(C)(C)SCC N1(CC(=O)NCCCN(C(=O)CC2CC(F)C2)C)CCCC1 C=C(Cl)CC(C(=O)N1CCC1(C)CCC)NC(=O)CC1C=CCC1 C1(O)(C(C)NC(C(C)SCC)=O)CCN(C(c2cc(CN(C)C)n(C)n2)=O)CC1 C1(C)(C(=O)NC(C=CC(=O)N(CC(C)C)CC)C)CC(F)C1 c1(CNC(C(CC2CCC2)NC(CN(C)C(=O)C2CC2)=O)=O)cccc(F)c1O CC(CC(=O)NC1CCCN(C(c2cn(C)cn2)=O)C1C)P(C)(C)=O C1(NC(C2CCC2)=O)CN(C(C2CCC(F)(F)CC2)=O)C2(CCOC2)C1 C1(C(=O)NC2(C)C(NC(Cc3c(C)ncs3)=O)CCC2)CC2(C1)CC(O)C2 C1(C(N2CCCC(CCNC(C(CSC)(C)C)=O)C2)=O)CC(F)(F)CCC1(C)C c1(C(=O)NCC(N(C(c2c(C)n[nH]c2)=O)C)C2CC2)cnc(O)c2ncccc12 N1(C(CC(=O)OCC)=O)CC(=O)CC1C(=O)NCc1cc(CC)cs1 Cn1nc(CNC(=O)CC2CC2CNC(=O)C(F)n2ccnc2)n(C)c1=O c1(C(N(C2CCN(C(c3cncc(C)n3)=O)C2)CC)=O)cn2c(n1)CC(C)CC2 C1(NC(C(C)(C)c2ccccc2)=O)(CO)CCN(C(c2ccccc2Cl)=O)C1 Cc1ccc(C(=O)NCCN(C(=O)CCc2cncn2C)CCOCCO)c(F)c1 c1(COC(C2(Cc3ccccc3)CCOC2)=O)coc(Br)c1 C1(OC)COCCC1N1CCN(CCN2C(C(=O)NC3CCCC3)CCC2)CC1 C(=O)(C(F)C1=CCCCC1)N(C1CCC(NC(Cc2c(C)n(C)nc2)=O)CC1)C N1(C(C23CCC(C(N4CCCCC4)=O)(CC2)CC3)=O)CCc2ccc(F)cc2C1 C1(C)(C(=O)NCCCC(C)NC(c2ncn(C(C)(C)C)n2)=O)CCC(F)(F)CC1 C12(CC(=O)NC3C4CN(C(C(CC)OC)=O)CC43)CC3CC(C1)CC(O)(C3)C2 c1(C(=O)NC(C(C)NC(CN(C(C)C)C)=O)C)cnc(N2CCCC2)nc1 C(CN=c1[nH]cc(C#N)c(=N)[nH]1)N(C(C=C(CC)C)=O)C C(C)(C)(CC(C)NC(C1CCN(C(c2ccc(Cl)cn2)C)C1)=O)SC c1(C(c2nnnn2C2CCC2)CC(C)(C)OC)cnc2n1CCC2 N1(C(C(CC(=C)C)C)=O)CCC(F)(F)C(CNC(c2ccsc2COC)=O)C1 c1(Cc2cn(CC(=O)NC(C)C(=O)N3CCCC3)nn2)ccc(Cl)c(Cl)c1O N1(C(C2C(NC(c3c(C)ccnc3)=O)COCC2)=O)CC2CC(O)CC2C1 N1(C(CC2(C)OCCO2)=O)C(C(=O)NCCN2CCNC2=O)CCC1C1CC1 C(=O)(C1=NN(C)C(=O)CC1)NC(COC)C(=O)NC(C)C.C12(CC1)C(=O)OC2 C12(NC(C(CC)C3CCOCC3)=O)CC(CNC(c3csc(C)c3)=O)(C1)OC2C C(CC)(CC(=O)NC1CCCOC1)NC(Cc1c(CC)con1)=O O=C1Nc2ccc(NC(C3CCCCCS3(=O)=O)=O)cc2C1=O C12(NC(c3c(C)cnnc3)=O)CCN(C(C3(c4ccc(Cl)cc4F)CC3)=O)CC1C2 Cc1nc(N2CCN(C3CCCCC3)CC2)ccc1[N+](=O)[O-].C123CC(C1)(C2)C(=O)N3 Cc1ccc(C(=O)NC(C(=O)NC2CCCCC2(C)C)C2CC2)cc1O C1(C(=O)NCc2scc(CNC(Cn3ncn(C)c3=O)=O)n2)CCC(C)(C)OC1 C1(C(C)NC(c2c(CCC)nco2)=O)CCCCN1C(c1coc(CC)n1)=O c1(C(=O)NCC2N(C(C3(COC)CCCO3)=O)CCC2)nn(C)c(Cl)c1C(F)(F)F C1(NC(C(CC2CCC2)NC(c2c(CC)ncnc2)=O)=O)CCCCC12CC2 C1(C(=O)NC(C)CNC(C2Cc3cscc3C2)=O)CC2(CO1)CC(F)(F)C2 N1(C(C(C=C)(C)C)=O)CC(CC(N2CC(CO)C(O)C2)=O)OC(C)C1 C1(C(=O)NCC(C)N(C(=O)Cc2cccc(CC3CC3)c2)C)CCCCC1(F)F N1(C(C2(F)CCCN(C(c3ccc(CC)o3)=O)C2)=O)CCCC12CCOC2C N1(C(CCc2nc(C)sc2)=O)CCC(C)C(CNC(=O)C=CBr)C1 C(c1cccc(Cl)c1)=C(C)C(N1CCC(NCC23CCC(CC2)C3)C(C)C1)=O n1(N(CC)CC)c(N2CCC(CC3CCCCC3)C2)nnc1-c1ccc(C)o1 Cc1[nH]c2ccccc2c1C(N1CCC1CNC(=O)CCc1cn[nH]c1)=O C(=O)(C1=CC2CCCCCCC12)NC(C)CN(C)C(c1ncc(F)cn1)=O N1(C(C2(C)CN(C)C(=O)C2)=O)CC2CCN(C(C3(C4CCC4)CC3)=O)CC2C1 c1(NC(C2C3CN(C(COC(C)=O)=O)CC32)=O)ccc2nncn2c1 CC1C(NC(=O)Cn2nccn2)CCCN1c1ncc(I)cn1 c1(NCCN2C(C(=O)NCC3CCOC3)CCC2)n[nH]c2ccc(Cl)cc12 CCCCCCCCCCC(=O)N1CCCC(C)(C)C1CNC(=O)CC(=O)OC N1(C(CC2C=CC(NC(C3CC4(CCC4O)C3)=O)C2)=O)CCc2nn[nH]c2C1 C1(C(=O)NC(c2ccccc2)C)CN(C(=O)Cn2ccnc2)CCN1 Cc1nc(C(CNC(=O)C(C)NC(=O)OC(C)(C)C)NC(C)CCO)cs1 N1(C(c2ccc(OC)c(F)c2)=O)CCCN(C(C2NC(=O)CC2C)=O)CCC1 CCC(CC)CCCC(=O)N1CCOCC1CC(=O)NC(Cc1cnc[nH]1)CO C12CC3CCC1N3C2=O.C(C(C)NC(C(=O)CC1CCC1)=O)N(CC)CC c1(C(N2CCN(C(C(C)=CC)=O)C(C)C2)=O)sc2cc(C)cc(C)c2c1Cl C(=O)(C(C)(O)C(F)(F)F)N1CC(CNC(CSC(C)C)=O)OCC1 c1(NC(C2C(CNC(C(COC(C)C)(C)C)=O)OCC2)=O)ccc2occc2c1 N1(C(CSCCN(C)C)=O)CCN(C(=O)C=Cc2cnccn2)C(C(C)(C)C)C1 c1(OC2CCCC(CC(=O)NC3(CNC(=O)C=CCO)CC3)C2)ccc(F)cc1 C1(C(C)NC(=O)CCc2nc(O)n[nH]2)CN(C(c2ccc(Br)cn2)=O)CCO1 CC1(O)CCCN(C(=O)CONC(C2C3CC4C(C3=O)C24)=O)CC1 C(=O)(CC(F)(F)C(F)(F)F)NC1(C2N(C(C(CN(C)C)O)=O)CCCC2)CCC1 CC1CN(C(=O)CNC(C2(C(=O)Nc3ccc(F)cc3)CC2)=O)C(C)C1C C1(NC(Cc2nc(C(C)=O)sc2)=O)CCN(C(c2cc3sccc3s2)=O)C(C)C1 C1(COc2ccc(C(=O)OCC)cc2)CN(N2CCN(C3CC3)CC2C)C1CC C1(C(=O)NCC(CC)(CC)CO)CC12CCN(C(C1(Cl)CCCCC1)=O)CC2 N1(C(c2cccc3nc(CO)cn23)=O)CCCC2(CCNC2=O)C1 C1(C(=O)NC(C(C)(C)NC(CCOC)=O)C)CCN(C(C23CCC(C2)C3)=O)CC1 C(=O)(C(C)(C)C1=CCSCC1)N(CC(C)NC(c1cnc(OC)nc1)=O)CC C(=O)(C1=CCCCC1P(C)(C)=O)N1C(CNC(C2(CO)CCC2)=O)CC(OC)C1 c1(C(=O)NCCCCNC(C2CC2c2ccco2)=O)cc2cccnc2[nH]1 C1(CCCC)CN(C(=O)C(C)n2ccnc2)CCN1C(c1cocn1)=O C12(NC(CN(CCC)C)=O)CCCC1N(C(c1occc1CC)=O)CC2 C1(NC(Cc2c(C)con2)=O)CCSC12CN(C(=O)C(C)CS(C)(=O)=O)C2 Cc1ccc(C(=O)NC2CCC2NC(c2cscc2Cl)=O)c(C)c1 C1(NC(c2c(C)con2)=O)CC(C)N(C(c2cccc(NC(C)(C)C)c2)=O)C1 C1(C(=O)NC(C(=O)NC)CC2CC2)CC(C)CN(C(c2ccc(O)nc2)=O)C1 CC1NC(=O)OC12CN(C(C1(CNC(c3csnn3)=O)CCCO1)=O)C2 c1(C(N(C(CNC(=O)C(F)C2CCCC2)C2CC2)C)=O)cccc2ccnn12 Cc1cn2cc(C(N3CC4(CCC4)CC3CNC(c3n[nH]cc3Cl)=O)=O)sc2n1 C1(C(NOCC(=O)OC)=O)N(C(=O)Cc2cccc(C)c2)CC12CCCC2 Cc1nn(C)c2c(NCC3CCC4CC34)nc(NC(c3cnsc3)C)nc12 c1(C(=O)NC2CC(CNC(C3CC3(F)Cl)=O)C2)cc2ccccc2nc1O c1(C(N2CCN(Cc3ccccc3)CC2CF)=O)cc2nccn2c(O)n1 N1(C(CSc2n(C)cnn2)=O)CC(NC(=O)C2=CCCCO2)C(C)(C)C1 C12(C(N(C3CCC(NC(c4occ(C)c4)=O)C3)C)=O)CC3CC1C2C3 Cc1nc(CN2CCCC2c2ccccc2)sc1C1CC1 Cc1coc(C(C)(C)C)c1C(N1CCCC(CN(C)CCc2n[nH]c(=N)s2)C1)=O Cc1cc(C(=O)NC(C2CCN(C(C3CCS(=O)(=O)N3)=O)C2)C)c(O)nn1 c1(C(c2ccnn2C2CCC2)NCC(C)(C)OCC)nnnn1CC(F)F N1(C(CN2CCN(CC)CC2)=O)CC2COCCC2(NC(c2cc(Cl)no2)=O)C1 C(=O)(C(CCN(C)C)NC(C1CCC1)=O)NCCNC(CCC=C(C)C)=O C(CCCC(=O)N(C1CCN(C(=O)C=CS(C)=O)CC1)C)N(C(C)C)C Cc1nnc2n1CCC(CNC(N1CCC(OC(F)(F)F)CC1)=O)C2 Cc1cc(C(c2nnnn2C2(C)CC2)NCC2(CS(C)(=O)=O)CCC2)cc(C)n1 N1(C(C(C)NC(=O)NC)=O)CC2CCCC(CN(C(=O)C(C)S(N)(=O)=O)CC)C2C1 c1(N2CCC(C)(NC(=O)CCC3CCC(=O)NC3)C2)ncnc2ccc(Cl)cc12 c1(CC(=O)NC(COCC)C)ccc(C(C)(C)C)cc1.C1(=O)C(=O)NCCN1 CCC(O)C(C)C(=O)NC1CCC(C)N(Cc2ccccc2Br)C1 CC1CN2CCN1C(C(=O)NC1CCC(CCNC(=O)Cc3cnc[nH]3)C1)C2 CCCC(CNC(c1ccn(CCC)n1)=O)C(=O)NC1(c2nc[nH]n2)CC1 C12(NC(C3CN(C)C(=O)C3)=O)CCCC1N(c1ncnc(=N)[nH]1)CCC2 C#CCCCCCC(=O)N1CC2CCC1C(NC(c1cn(C)nc1SC)=O)C2 CCCCCCCCC(C)C(=O)N1CC2COCC(C1)N2C(c1oncc1C)=O C1(CCC(=O)NC2(CSC)CCC2)Cc2ccccc2NC1=O C1(C(C)NC(C2CCN(C3CC3)C2=O)=O)CCN(C(=O)C=CC2CC2)CC1 c1(C(C(=O)NCC(CC=C)NC(=O)CCc2cncs2)OC)cc(F)cc(F)c1 c1(C(=O)NCC2CN(C(c3c(C)scc3)=O)CC2O)cccc2ncsc12 c1(C(N(C(CCC)C)CCO)=O)nnc2n1CC(C(F)(F)F)CC2 Cc1cc(C(=O)N(C(C)CNC(=O)CCCCCF)C)cc(C)c1 c1(C(=O)NCCC(C)NC(c2cnc(C(C)OC)s2)=O)ccc2n[nH]cc2c1Cl C12(NC(C3CC(C)N(C(=O)C(C)(O)C(F)(F)F)C3)=O)CC(CO)(C1)OC21CCC1 C(=O)(CC(O)C(C)(C)C)NCCCCCCN(C)C(c1cccc(C(N)=O)n1)=O N1(C(c2cnc(CCC)s2)=O)CCC2C(NC(c3c(C)nn(C)c3F)=O)CC12 C1(CC(=O)NC(C)C=CC(=O)NC(CC2CCC2)CO)COCCOC1 C1(CNC(C2CN(C)C(=O)N2)=O)C2CCC(C2)N1C(c1ccc(C2CCOC2)s1)=O Cc1cccc(C(=O)NCC2CCC(C)CN2C(=O)CC23CCC(CC2)C3)c1O C(=O)(CC(C)(C)N(C)C(C1SCCCS1)=O)N1CCC(C(=O)NC)C1 N1(C(C(C)SCCCC)=O)Cc2n[nH]cc2C1C(=O)NCc1cn(C)nn1 C1(CNC(c2c(NC)cccn2)=O)CN(C(=O)CCC2OCCO2)CC(C)(C)C1 C=CCC(C(=O)OC)NC(C1(CC=C)CCN(C(c2cnn(CC)c2)=O)C1)=O C(=O)(C(CCC(C)C)NC(=O)C(F)C(CC)CC)NCCCCCCC=C c1(CC(N2CCC(CNC(C3(CCOC)CC3)=O)C2)=O)ccccc1S(C)=O c1(CNC(c2c(C(=O)OCC)n(C)nn2)=O)cc(C#N)ccc1O Cc1cc(Cl)cc(C)c1NCC(=O)OCC(C1CCc2nccn2C1)=O c1(NC2(C)CC(NC(C=Cc3cnc(C)s3)=O)C2)nc2cccc(Br)c2o1 c1(NC(CC)=O)cnccc1C(=O)OCCCC1CCOC1 C#CCCCC(C(=O)NC1COC1)N(C(C)(C)C)CCN(C)C CS(C)(=O)=Nc1ccc(C(=O)NCC2CCCO2)s1 C1(OCC)(CNCC(C)Cn2nc(C)cc2C)CCC(C)C1 c1(N2CCC3(CN(C)C3)C2)ccc(S(=O)(=O)N2CCC3(C2)OCCO3)cc1Cl N1(C(CCOCCOCCCOC)=O)CC(O)(NC(=O)CN2CCSCC2)C1 C(CC1=CCN(C(C2CC2c2ccco2)=O)CC1)NC(c1c(C)ccnn1)=O Cc1cnc(C(=O)NC2CN(C(=O)Cc3cccc(F)c3)CC2F)cc1Br C(=O)(CC(C1CC1)NC(=O)CC1(NC(=O)Cc2cncnc2)CCCC1)NC c1(C(=O)NC2CC3CN(C(c4[nH]cc(CC)c4)=O)CC32)snc2ccccc12 c1(C(N2CCC(Cn3cc(Br)cn3)C2)=O)ncc(C(=O)O)s1 c1(C(=O)NCC2CN(C(Cc3cccc(C(N)=O)c3)=O)C2)cc(Cl)c(F)cc1Cl CCC(CCCC(=O)N1CC2(CSC2)C1)NC(C1CC(CC)(CC)C1)=O C1(C(N2C(CN(C(C(CC)OC)=O)C)COCC2)=O)CCC=CCCC1 C1(C(=O)OCC)CCCC(NC(C2N(Cc3ccc(CC)s3)CCC2)=O)C1 c1(C(=O)NC(CC)(C)CNC(=O)C(C(C)C)n2ccnc2)cc2ccccc2o1 CC(C(=O)N(CCCOCCNC(=O)CCc1ncco1)C)c1cccs1 CCC(CC(=O)NC(CNC(C1CC2(C1)OCCO2)=O)C1CCC1)C(F)F C12(NC(=O)C=CC3CCCCC3)CC3CCC(C1C2)N3C(C1CC1C(F)(F)F)=O c1(CNC(C(N2C(=O)CCC2=O)CC)=O)cc2n(n1)CCN(C(=O)CCF)C2 C1(C(=O)NCCN(C(C(CC)=CCCC)=O)CC)Cc2nnc(C)n2C1 c1(C(=O)NCC2CC3(CN(C(c4[nH]c(=N)sc4)=O)C3)C2)cnc2c(c1)CCCO2 C1(CCOC)(NC(c2nc[nH]c2C)=O)CCN(C(=O)C(C(C)C)SC)C1 C(N=C(NCC(F)F)N1CCC(Nc2ccncc2)C1)C1C(CCC)C1 C#Cc1ccc(OC)c(C(=O)NC(C2CN(C(=O)C(CC)CC)C2)C)c1 c1(C(N2CC(NC(c3c(COC)n(C)nc3)=O)C(F)C2)=O)nc(C)c(C)[nH]c1=O C(=O)(C(CCC(N)=O)N(C)C)NCCC1OCCN(C(c2c(C)ccn2C)=O)C1 CCCC(O)(CCC)CC(=O)NC(C)C(C)NC(c1cccc(O)c1Cl)=O C1(C(N2CCC(COC)(NC(c3nc(=O)n(C)[nH]3)=O)C2)=O)CCN2CCOCC12 c1(CCCC(N2C(CCCC#C)CCC2)=O)cccc(C(=O)OC)c1 N1(C(CCC#CC)=O)CCC2CCN(C(=O)C=Cc3ccsc3C(F)(F)F)CC12 C1(C(N(C2CCN(C(c3cnc(C(C)C)o3)=O)C2)CC)=O)CCCCC1(C)C c1(COC)ccc(C(=O)NC(CO)C(C)NC(=O)C(C)CC2CCCCC2)o1 Cc1cc(NC(CNC(c2cnoc2-c2ccco2)=O)C(C)(C)C)ncn1 O=C(CCCCC(F)F)N1CCCCC1CNC(C1Cc2ccncc2N1)=O c1(C(C)(C)C)nccc(=NC(=O)C2CCC(CC(=O)Nc3n[nH]cc3I)CC2)[nH]1 Cc1ccc(SCC(N2CC(CNC(=O)Cn3ccnn3)C(C)C2)=O)cc1 c1(OC(CC)C(=O)N2CCC(C(N(C)CC3(OC)CC3)=O)C2)cccc(C)c1C C#Cc1ccc(OCC(=O)NC2CC(O)(CNC(=O)Cc3cnc(C)[nH]3)C2)cc1 C1(N(c2cccc(-c3ccsc3)c2)C(C(C)NS(CC)(=O)=O)=O)CCNCCC1C c1(C(=O)NC23CCN(C(COCCCC)=O)CC2C3)cnc2onc(CC)c2c1 N1(C(c2n(C(C)(C)C)ccn2)=O)CC(NC(=O)CSC2CCCCO2)C2CC12 c1(C(=O)NC2CCC(CCN=c3[nH]ncs3)C2)cc(Br)ccc1F C1(ONC(=O)C2CC2(C)C)CCOCC1.C1=CCN(C)C1=O.C1CCC1 C1(NC(c2n(C(C)C3CC3)ncc2)=O)CCC=CC1O CC(O)CCCC(=O)NC(CNC(=O)C(C)(C)CC1CCOC1)CO C(=O)(C1=C(C)N2CCN=C2C=C1)NCC(CC)(CC)NC(=O)COc1ccsn1 c1(CNC(c2n(CCCSC)nnn2)c2cnc(Cl)s2)cccc(C(C)(F)F)c1 C=CCC(CC(C)C)C(=O)N(CCNC(=O)CCC(C)CN(C)C)N(C)C1CC1 CC(C)CCC(=O)C(=O)N1CCN(C(=O)Cc2ccc(C(C)C)cc2)CC1C N1(C(CCCOCC=C)=O)CC2CC(NC(=O)Cc3cccs3)C(C2)C1 c1(C(N(C2CCN(C(C3(n4cnnn4)CC3)=O)C2)C)=O)cnn(C2CC2)c1N C1(C(N2CCC(C=CC(N3CCN(CC)CC3)=O)CC2)=O)CC2(C1)CC(CO)C2 C1(CC(=O)N(C)CCOCCN(C(=O)CSCC(N)=O)C)CCOCC1(C)C n1(CCOC)cc(CC(=O)NC(C2CCCN2C(=O)Cn2cnnc2)(C)C)cn1 C1(CNC(C(=O)NCC=CC)=O)CN2CC3CC2(CO1)C3 c1(CC(=O)NC2CN(C(c3cnc(O)nc3O)=O)CC2F)cc(F)ccc1F C(=O)(CCCCC#N)NC(CC)C(=O)NCc1cnn(C)c1O c1(C(N(CCNC(CCC(C)N(C)C)=O)CC2CC2)=O)c(F)cccc1Cl N1(C(C=Cc2ccc(CC)o2)=O)CCC(C(F)(F)F)C(NC(=O)CN(C)CC)C1 C(C(CO)(CO)NC(C1CCC1c1nc(S)n[nH]1)=O)N(C)C(C1CCCC1O)=O CC1(C)CCN(CC(=O)NCC(C2CC2)NC(=O)CNc2cccnc2)C1 c1(C(N2C(CC(=O)NCCCc3nccs3)CCC2)=O)cc2n(n1)CCO2 CCC(C)(O)C(=O)N1CCC(NC(=O)C(CCSC)OC(C)=O)C1 C1(C(=O)NCCC(C)(C)NC(C(C)=C(C)C)=O)Cc2n[nH]cc2C(=O)N1 CC(O)CC(C)(C)CNC(=O)CSc1nnc(-c2ccc(Cl)cc2)o1 N1(C(CC(C(C)C)c2ccon2)=O)CC2CCN(C(=O)C(C)(C)C)CC2C1 C1(C(N2CCC(C(=O)Nc3cnc(CCCC)nc3)C2)=O)CCC(=O)N(CC)C1 C1(C(N)=O)CCCCC1SC1(F)CC(NC(CN(CCC)C(=O)OC(C)(C)C)=O)C1 CC1CCCCC1(CNC(c1c[nH]c(Br)c1)=O)NC(c1nc(F)ccc1Cl)=O Cc1cn2cc(C(=O)NC(C)C(C)(C)NC(c3ccc(C(C)C)o3)=O)ccc2n1 CCCC(C)(O)C(=O)NC1CC(C)CN(C(C2(CO)CC2)=O)C1 C(=O)(CCC(=O)c1cc(C)sc1C)NC(CC=C)CNC(c1sccc1COC)=O C1(NC(CC(=C=C)C)=O)CN(C(=O)C(C)N(C2CC2)CC)CC12CCOCC2 C=CC1COCCN1C(=O)C(Cc1ccoc1)NC(c1oc(C)nc1C)=O C1(C(=O)NCC2(F)CCN(C(c3ccsc3Cl)=O)CC2)CC2C=CCC(C1)C2 c1(C(N2CCC(NC(C(N)=O)=O)C(CO)CC2)=O)ccc2c(c1)CCCS2(=O)=O CN1CCC(=CC(=O)NCC(F)CNC(=O)Cc2cnc(C(C)C)[nH]2)CC1 c1(C(=O)NC2CC(OC(C)C)C2)coc(CNC(=O)CC2CCOC2=O)n1 N1(C(=O)Nc2cccc(CC)n2)CCc2ccc(-c3cnc(C)nc3)cc2C1 C1(CNC(CN(C(C)C)C)=O)CN(C(=O)C(=Cc2cccc(F)c2)F)CCN1C N1(C(c2nc(Cl)cs2)=O)CCC2(CO)CN(C(=O)Cn3ccnn3)CC2C1 N1(C(C2CC(C)(C(=O)OC)C2)=O)CCCC(O)(NC(=O)COc2ccccn2)C1 N1(C(C2C(CCOC)C2)=O)CC(NC(c2cnc(O)c(F)c2)=O)CC1(C)C C12(CNC(COCC(C)C)=O)CCCC1N(C(c1ccc(C#N)cn1)=O)CCC2 N1(C(c2c(C)scn2)C(=O)NCCC2CC2)CCC2(CC1)COCC(=O)N2 Cc1ccc(O)c(C(=O)NCC2(CNC(C3CCS3(=O)=O)=O)CC2(F)F)n1 c1(OC)ccc(CC(=O)NCCN2CCN(C(=O)CCSC)CC2)cc1Cl C1(=CCNC(C2C(C)(C(F)F)C2)=O)CCN(C(=O)C(F)(F)CO)CC1 N1(C(C2C(C)C2)=O)CCN(C2CN(C(=O)Cc3ccc(Cl)cc3)C2)CC1 C1(C(=O)NCCCc2n(C)ncc2)CC1C1CN(C(=O)CN2CC=CC2)C1 C12(CN(CC=C)C(c3ccc(C(=O)OC)cc3)C)CCC(CC1)CO2 C1(C(=O)NC2CCC(NC(C3(CO)CCCCC3)=O)C2)CC12CCSCC2 C(=O)(C1=CNC2=NCCCN12)N1C(CCNC(C2CC(OC)C2)=O)CSCC1 C(=O)(C(O)CC(F)(F)F)N1CCC(OCCn2cccn2)C1.C12(CCC1)CC(=O)N2 C1(CNC(=O)CCCCO)CCN(C(c2ccc(F)nc2)=O)C12CC2 C1(CC)CN(C(=O)C(CCC2CC2)NC(c2cc(C)nnc2O)=O)CCCO1 C=C(C)C(C)(O)C(=O)NCC(C)(C(C)C)NC(c1cc2sccc2s1)=O Cc1nc2ccnn2c(C)c1C(=O)N(CC(C)(C)NC(c1nccs1)=O)C c1(-n2ncc(C(=O)NC(CC)CNC(=O)Cc3ccsn3)c2)ncc(Cl)cn1 CN1N=C(CC(=O)NCc2ccc(CNc3ccnc4ncnn34)cc2)CC1=O N1(C(C2(C(C)C)CCCN2C(c2nonc2N)=O)=O)CCC2(CCCO2)C1 c1(OC)ccc(Cl)cc1C(=O)NCC(C1CCCC1)NC(C1COCCOC1)=O C1(C(=O)NCCN(C(C)C)C)CCC(CNC(=O)CSC(F)(F)F)C1 C(=O)(C1=C2CCN=C2NC=C1)NC1CCC(NC(CN2CCC(=O)NC2=O)=O)C1 N1(C(c2cccc(C)c2)=O)CCN(C(=O)CC2CCC2(C)C)CC1CS(C)(=O)=O N1(C(C(C(C)C)C)=O)Cc2ccccc2C1CNC(=O)CC1CC=CC1 C(=O)(C(F)CC(CC)CC)NCCC(C)(CC)NC(CC(CC=C)(C)C)=O Cc1nc(-c2ncc[nH]2)sc1C(=O)NCC(O)CNC(=O)CCc1cncs1 C(C1(C)CCOCC1)=CC(=O)NCC(C)CCNC(=O)COC(C)(C)C C=CC1(C(=O)NCC2=NOC(C)C2)CCN(C(C2CC23CCCC3)=O)C1 C1(NC(CC2(COC)CC2)=O)CCC(C)N(C(c2cc[nH]c2)=O)C1 C1(NC(CC2CC(NC(COC)=O)C2)=O)CC12CCCC2 c1(CC)nn(C)c(CC)c1C(=O)NCC1CCCN1C(c1nc(=O)n(C)[nH]1)=O c1(C(=O)NC2CCC(N(C)C(c3cn(C)nn3)=O)C2)ncc([N+](=O)[O-])n1C N1(Cc2c(C)nc[nH]2)CCCN(C(c2ccc(Br)c(C#N)c2)=O)C(C)C1 c1(NCc2cn(CC)nc2)cc(=NC2CCN(C(C)C)CC2)[nH]c(COCC)n1 c1cnc2c(=NCCc3c[nH]c4ncc(Br)cc34)[nH]cnc2c1.N12CC3CC1CN23 S(=O)(=O)(c1c[nH]c(=NCCCC2CCCO2)cc1C)NC(C=C)Cn1cncn1 N1(C(C2C(=C)CC2)=O)CC2(CCC(NC(=O)CC3C=NN(C)C3=O)CC2)C1 C(C)(CCC(=O)N1CCN(CC2CN(C(=O)CCCNC(N)=O)C2)CC1)OCC C(=O)(C(C)(C)O)N1C(C(=O)NCCNC(COC)=O)CC1 c1(C(N(CCNC(C2(C(C)(C)C)CC2)=O)C2CC2)=O)cc(S(N)(=O)=O)c[nH]1 N1(C(c2ncccc2F)C(=O)NCCSC)CCC2(CCCC2)C1 c1(C(=O)NC2CCC2NC(=O)C(F)(F)c2ncccn2)ccc2c[nH]nc2n1 C(=O)(CS(=O)(=O)CC)N(CC(CCCC)O)Cc1cn(CC2COC(=O)C2)nn1 N1(C(C(C(C)O)C)=O)CCCC(C)(C)C1CNC(C1CC=CCO1)=O C1(CC(=O)NCC(CC)N(C(=O)CCC=CC(C)C)C)C=CCCC1 c1(C(=O)NCCCN(C(c2c(CC)nc(C)[nH]2)=O)CC)cccc2c1C(=O)NC2 c1(C(=O)NC2C3CN(C(COCc4onc(C)n4)=O)C2C3)cccc2c1ccn2C N1(CC(C)NC(C2(F)CCOC2)=O)CCN(C(=O)Cc2cnn(C)c2C(F)F)CC1 c1(NC)ccc(C(=O)NCC2CC(F)CN2C(=O)CCCc2nc(C)no2)cc1 N1(C(C(COCCO)NC(=O)COC2CCOC2)=O)CCCC(CCCO)C1 CC1(C)CCC(C(=O)NCC2(F)CCOCC2)CN1C(=O)CC1CSCCO1 c1(C(=O)NCC(C)N(C)Cc2cc(C)on2)cccc2ncnn12 CC1CN(C(=O)C(O)C(C)(C)C)CCC1NC(C12CCCN(CC1)C2)=O c1(CNC(C(C)OCC)=O)ncccc1C(N1CCC(C(C)CO)CC1)=O Cc1ccc(C)c(C(=O)NC2(CO)CCCN(C(C3(n4cncn4)CC3)=O)C2)c1 C1(C(=O)NCC(COC)(F)F)(CF)CCN(C(c2ccccc2C2CC2)=O)C1 C(CC(C)C(=O)NCC(C)(C(C)C)NC(c1cc(C)sc1C)=O)=CC N1(C(c2cnc(C)[nH]2)=O)CCCC(NC(C2CCC(N(C)C)CC2)=O)CC1 C(=O)(C1=CC2C=CC(C1)C2)NC1C(CNC(c2c(Cl)ccc(OC)n2)=O)CC1 c1(SC)nc(CC(=O)NCC2CC(C(=O)N(CC3CCOCC3)OC)C2)cs1 Cn1c(C(=O)N(CCNC(c2cn(Cc3cccs3)nn2)=O)C2CC2)cnc1O CN1CC2CN(C(C3CCN3C(=O)CC3OCCO3)=O)CC2(C)C1 C(C(C(=O)N1CCC(O)(C(N)=O)C1)C(C)(C)C)NC(c1cc(C)no1)=O Cc1cc(C(=O)NC(C)CCCNC(c2cnccc2Cl)=O)n(C(C)(C)C)n1 C1(NC(c2cccc(OCC)c2)=O)CC2CC1N(C(C1ON=C(C)C1C)=O)C2 C1(CC(=O)NCC2(NC(C(CN(C)C)O)=O)CCC2)CC(C)(C)OC1=O c1(C(=O)NCC(C)NC(Cn2c(C)cc(O)cc2=O)=O)c(C)nn2cccnc12 CCC(CNC(c1ccccc1C(F)F)c1nnnn1C1(C)CC1)CCCO C(=O)(CC(C)CC(C)(C)C)NC1CCN(C(c2scc(C)c2C)=O)CC1CO c1(CN2C(C3CCN(C(CCC(=C)C)=O)CC3)CCC2)ccc2c(c1C)CCC2 c1(CC)ccc(C(=O)NC23COC(CNC(C4CCOCC4)=O)(C2)C3)cc1Cl C12CCC(CC1)NC2=O.CCC1C(=O)C(=O)CC2(CC(=O)N1C)CC2.OC C(CN=c1cc(C)nc(NC2CCC(C(N)=O)C2)[nH]1)N(CC)Cc1cccc(C)n1 n1(C)cc([N+](=O)[O-])nc1C.C(C(CC)(CC)C(N)=O)Sc1n(CC)c(CCN)nn1 C1(NC(c2c(C)onc2CO)=O)CCN(C(=O)CCCCC2CC2)C(C)C1 C1(OC)CN(C(=O)C(C(C)C)NS(C)(=O)=O)CC1C(=O)NCC1CC(=O)N(C)C1 C12(NC(c3c(CC)ccc(C)c3)=O)CCCC1CN(C(=O)C=CSC)C2 C1(CN(c2cc(F)ccc2F)C(CNC=O)=O)CC2(CO1)CC(F)(F)C2 N1(C(C(C)C(F)F)=O)CC2CC(C1)CN(C(c1cc(F)c(F)c(F)c1)=O)C2 C1(N(C(C2(CNC(=O)C3CCCC3)CC(=C)C2)=O)CCN2CCCC2)CCS(=O)(=O)C1 c1(OC)cccc(-c2nc(Cc3ccc(C)s3)n(CCC3CCCC3(F)F)n2)n1 N1(S(C)(=O)=O)CCN(CC(N2CCC(CCC)C2)=O)CC1.C(c1cscn1)=CC(=O)N(C1CC1)N.N c1(OC)nc(C)ncc1C(=O)NC1CCCCN(C(c2cnc(C)[nH]2)=O)C1 CCCCC(CCCC)C(=O)NC1CC(CN=c2[nH]c3cccnc3s2)(F)C1 CCS(=O)CC(=O)N1CCCCC1CCCNC(=O)Cc1coc(C)n1 C=CCCCCCCC(=O)NC1CC1CNC(C1(c2ccccc2)CCCCO1)=O C(=O)(C(C)(C)C1=CCN(C(c2cccnn2)=O)C1)NCCCCCC(C)(C)C C(CN=C(NCC)NCC(C)NS(C)(=O)=O)C1(NC(S(CC)(=O)=O)=O)CC1.C(C)(C)(C)O C1(NC(c2c(NC(C)=O)cccn2)=O)CN(C(c2n[nH]c(C)n2)=O)CCC1C C=CC(C)(O)CC(=O)N1CCC(C(C)N(C(=O)C(C)N(C)C)CC)CC1 Cn1ncc2cc(C(=O)NCC34CCC(CC3)N(C(C3CCS3(=O)=O)=O)C4)sc12 C1(SC(C(=O)N2C(C(=O)OC)CC2)CC)CC2(CC(NC(=O)Cn3cncn3)C2)C1 CC(C)(CC1CC1)C(=O)NCC1C2CN(C(=O)Cc3ccc(Cl)cn3)CC12 C(CCNC(C1CCCN1C(C)C)=O)(C(C)C)NC(c1nc(CCC)sc1)=O c1(NCC(N2CC3C(CNC(CCOC)=O)C3C2)=O)ccc(C)nc1O c1(-c2cc(C)c(F)cc2)ccc2sc(C(=O)Nc3c(C#N)cnn3C)cc2c1 c1(CN(C(CCOCC)=O)C)cc(Cl)cc(Cl)c1F N1(C(CC(COC)C(C)C)=O)C(C)CC2CN(C(c3cc(C#N)c[nH]3)=O)CC12 C(=O)(CC1=NN(C)C(=O)C1)NC(C1CCCN(C(=O)C=CC2CCOCC2)C1)C C1(CNC(c2cnc3n2CCC3)=O)CN(C(=O)C(F)CC2CCC2)C2(CCC2)C1 CCC(CC)(CCNC(=O)CCCCSC(F)(F)F)NC(=O)C1=C(Cl)CC1 c1(OCC)cc(CN2CCC(C)(C(=O)NC3CCCOC3)C2)cc(Cl)c1 Cc1ccoc1C(=O)NC(CC1CC1)C(=O)NCC(O)Cn1cccn1 C(=O)(C(C)(C)C(=O)OC)NCC1(C(=O)NCC(CC2CC2)OC)CC(=C)C1 CC1CN2CCN1C(C(=O)NCC(C1CCC1)NC(c1csc(C3CC3)n1)=O)C2 C(=O)(C1CCCc2nncn21)NCC1(CNC(c2ccc(C#C)cn2)=O)CCC1 C1(C(N(CC(=O)Nc2ccc(O)cc2F)C(C)C)=O)Cc2ccccc2C1 c1(C(=O)NC2(CNC(c3c(NC)scn3)=O)CC2)c(Cl)c([N+](=O)[O-])nn1C N1(CC(=O)NCc2c(OC)cccc2Cl)C(=O)NC2(CCc3ccccc3C2)C1=O C1(CCCNC(C(CN(C)C)O)=O)CN(C(=O)CC2(C)CC2)CCO1 C(C)(C(C(=O)N(C1CCOC1)CCF)NC(=O)CC1CCOCC1)OC C1(C(N2C(CCNC(CC(C=C)C)=O)CCC2)=O)Cc2ccncc2N1 Cc1cn2cc(C(=O)NC(C)(C)CNC(=O)C(C)C(C)O)cc(C)c2n1 CC(C(=O)N1CCN(C(=O)CC2OCCC2(C)C)C(CF)C1)C(F)(F)F CN(C)NC(=O)CCC(=O)N1CC(CNC(C2(CO)CC2)=O)N2CCC1C2 c1(C(N(CC(N2CC(OC)C(F)C2)=O)CC(C)C)=O)cc(C#N)n(C)n1 CC1(NC(C2OCCC2CC2CCC2)=O)CCN(C(=O)CCN2CCOCC2)C1 c1(OC)cc(C(=O)NCC(C2CC2)NC(=O)CC(C)(C2CCC2)C2CCC2)ncn1 C(=O)(C(=O)N=S(C)(C)=O)N1C(C)C(NC(c2c(N(C)C)cccc2F)=O)CCC1 Cc1cccc2cc(C(=O)NCC(CO)NC(c3cc(C#N)ccc3Cl)=O)nn12 CC(F)(F)C(F)C(=O)NC1CCCC1CC(=O)NCCC(O)C1CCCC1 c1(C(N2CCC3(CN(C(C4(C)COC4)=O)C3)C2)=O)ccc2cnccc2n1 c1(CN2CCC(C(=O)NCCCC)C(O)C2)ccc(C#N)cc1S(C)(=O)=O C1(N(C(=O)C=CC2CCOCC2)C)CN(C(=O)C(F)OC(F)(F)F)CC12CC2 Cc1ccc(CCC(=O)NCCCNC(=O)C(Cl)=CCl)c(Br)c1 c1(NC(C2N(Cc3c(C)scn3)CCC2)=O)cccc(F)c1C c1(OCC(=O)NCCC2(OC)CN(C(C(C)(C3CC3)OC)=O)C2)ccccc1C C1(C(=O)NCC(CC=C)NC(c2cnnn2C)=O)CCN(S(N)(=O)=O)CC1 C(=O)(C#CC(C)(C)C)NC1(C)CCC(NC(C(C)OCc2ccc(O)cc2)=O)C1 c1(CCC(=O)NCC2(NC(c3ccc(C)cn3)=O)CC2)ccc(F)cc1Cl C=CCCN=C(NCCC(C=CC(F)(F)F)N(C)C)NC(C)CCF C(N=c1[nH]c(Cl)ncc1C(C)C)C1N(C(c2n(C=C)ncc2)=O)CCCC1C c1(CC)ccc(C(N2CC(NC(c3cn(C)nn3)=O)CCC2C)=O)c(C)n1 C(=O)(C(=O)N=S(C)(C)=O)NC1C(NC(C2(C)CN(C)C(=O)C2)=O)CC1 N1(C(C(C)OCC)=O)CC(C)N(C(=O)CC2(C)CCCCC2)CC1C N1(C(Cc2ccc(C)nc2)=O)CCCC2(NC(=O)C(F)C3CCC3)CC2C1 c1(CC(=O)NC2C(C(N(CCCO)CC)=O)CCC2)cccnc1O C1(C2CCCN(C(=O)C(C)(C)n3ccnn3)C2)(NC(C2CC(C)C2)=O)CC1 N1(C(CC(C(C)OC)NC(=O)C(C)(C)n2cncn2)=O)CC2(C=CCO2)C1 CC(C)(CSc1ccccc1)C(=O)NCCNC(=O)CN1C(=O)CCC1=O N1(C(C)=O)CCCC1C(=O)NCC=CCNC(c1ncoc1C1CCCC1)=O N#Cc1cc(N2CCCCCC2)ccc1N1CCN(c2nc[nH]n2)CC1 c1(CC(=O)NCCCCC(C)NC(C2CSC2)=O)cc(Br)ccc1F N1(C(C=CCCC)=O)CCC(NC(=O)CC2(F)CCCCC2)C12CC2 c1(CCC(=O)NCC2C(NC(C(F)=CC)=O)CCC2)cnc2ncccn12 C(C(C)C)(C(O)C(=O)N1CC=CC(C(=O)NCC2CC23CCC3)C1)OC C(N=c1[nH]c(C)cc(=NCC(C)(C)SCCO)[nH]1)c1ccn(CCC)n1 N1(C(C2(CC)CNC(=O)C2)=O)CCC(C(=O)NC2CCOC2=O)CC1(C)C c1(C(=O)OCC)cc(C(N2CC(N(C)C(C3(C(n4nccn4)=O)CC3)=O)C2)=O)c[nH]1 C1(C(=O)NCCCN(C(C(C(C)C)NC(C)=O)=O)CCO)CCCN(C)C1=O N1(CC)CCCC(NC(=O)CC(C2CC2)NC(c2ccoc2C)=O)C1 C1(NC2(c3n(CC(=C)C)nnn3)CCOC2)CCCC=C1Br N1(C(c2c(COC)cco2)=O)CCC2(CC2C(N2CCC3C(C(N)=O)C3C2)=O)C1 N1(C(C2CCS2(=O)=O)=O)CC=C(CCNC(C23CC4CC2C3C4)=O)CC1 c1(C(N2CCCN(C(C(C(=O)OC)C)=O)C(C)C2)=O)cc(OC)cc([N+](=O)[O-])c1 CC(C)(C)C(CC(=O)NC1CN(C(=O)CCF)CC1C(F)F)C(F)F C#CCC(C)(C(=O)NCCCOC1CC1)NC(=O)C1=CCCC1 C1(NC(C2CC2(F)F)=O)CC2CCC(C1)N2c1ncns1 N1(C(C2COCCO2)=O)Cc2occ(C(=O)NC3CCC(F)(F)C3)c2C1 N1(C(C=CC(C)(C)SC)=O)CCN(C(c2cnc(C)nc2C(C)C)=O)C(CO)C1 O=CCC(=O)Oc1ccccc1.N1(C2C(C(N(C3CC3)C)=O)C2)CC(NC=O)C1 c1(N(CCCNC(C(C=C)(C)C)=O)C)cc(OC)c(OC)cc1F c1(CNC(C2(SCCN(C)C)CC2)=O)ncsc1S(N)(=O)=O.c12cn(nn1)CC2 C1(CC(=O)NC(CC(=O)NC)C)C2CCCC2N1C(=O)CC1(OC)CCOC1 C#CC1(C(N2CC(OC)CC(F)C2)=O)CCN(C(c2oncc2CC)=O)C1 C1(C)(C(=O)OC)CCC1(C)C(=O)NCC(C)(C)CN(C(=O)C(F)C1CC1)C C(C(C)(C)CC(F)F)NC(C1(COC)C=CCN1C(c1cc([N+](=O)[O-])c[nH]1)=O)=O N1(C(c2ccn(CCOC)n2)=O)CCCC(CCNC(=O)CN2CCC(C)C2)C1 Cc1nncc(CNC(C2CCOC2CNC(C2CC(=O)CCO2)=O)=O)c1C c1(C(=O)NCC2CCN(C(=O)C=Cc3ncco3)C2)cc2c(s1)CCOC2 c1(C(N(CCNC(CSCC#C)=O)CC2CC2)=O)oc2ccccc2c1Cl c1(C(=O)NCC2(O)CCN(C(c3c(CC)con3)=O)C2)cc(=O)c(OC)cn1C c1(C(N2CC(CNC(CC=C)=O)C(F)(CO)C2)=O)c(Br)nc2n1CCOC2 c1(C(=O)NC2CCC(NC(C(C)OCCCC)=O)C2)cc(F)cc2c1CCC2 C1(NC(CCCCOC)=O)CCN(C(=O)CNC(=O)CCc2cnc[nH]2)CC1O Cc1ccn(CCC(=O)NC2(CCNC(=O)CCCN3CCCC3)CCC2)n1 c1(CC(=O)N(C2(CO)CC2)CCNC(=O)CSC(F)F)ncc(F)cc1F C1(CNC(C(C)(C(C)C)NC(C)=O)=O)COC(C)(C)CN1C(=O)Cc1ncoc1C N1(C(C(CCOC)OC)=O)CC2(CCC1CO)CC2.C1(C=O)CC(=O)N(C)C1 CCCC(C(=O)NCC(C)(CO)NC(c1nn(CC)cc1Cl)=O)C(C)C c1(CC(C(=O)NC2CCN(C(C3C(C=C)C3)=O)CC2)C)ccc(F)c(F)c1 c1(C(=O)NC(C)CNC(C2(Cl)CC23CCC3)=O)ccc(P(C)(C)=O)cc1 N1(C(C(=O)Nc2c(C)ncnc2)=O)CCCC(C)(C(=O)O)C1 C(=O)(C(CO)NC(N)=O)N(C1CCN(C(c2csc(-c3ccoc3)n2)=O)C1)CC C1(C(=O)NCCCCC#C)CN(S(=O)(=O)Cc2ccccc2Cl)CC1O c1(N(CC(=O)N(C2CCN(C(C3C(C)CC3C)=O)CC2)CC)C)ccc(Cl)nn1 c1(C(=O)NCC2CC(NC(C3(C)CCNC3=O)=O)C2)cccc2cc(O)ccc12 C1(C(=O)NC2CC(NC(c3cc(F)cs3)=O)C2)CCc2ccnn2C1 C(CCCCC(=O)N(CC(C)(C)CNC(c1ccccc1N(C)C)=O)C)SC C1(CC)CC(O)CN1C(C1C=CCN(C(c2ncncc2N)=O)C1)=O C1(NC(CCN(C(CC)CC)C)=O)(CNC(=O)C(C)SC)CC(F)C1 C(=O)(C1=CCCCO1)NC1CCC(C(=O)NCC(C)(C)C(F)F)C1 C1(C(=O)NC2C(OC)CN(C(=O)C=CS(C)=O)C2)(OC)CCCCCC1 c1(OCC(N2CC(N(C)C(c3c[nH]nc3C3CC3)=O)C2)=O)ccc([N+](=O)[O-])cc1 c1(CC)c(C(=O)NC2(C)CCN(C(=O)CC(O)C3CCCC3)CC2)cccc1C Cc1ccc(C(=O)N(C)CCNC(=O)CN(S(C)(=O)=O)C)c2ccccc12 C1(CC)CCCCC1C(=O)NCCN(C(=O)Cc1csc(C(C)C)n1)CC1CC1 c1(OC)cccc(C(C)CC(=O)N2CC(NC(=O)C(C)C)C2)c1 n1(CC)nc(C(=O)N(C2CC(NC(=O)CC3C(C)C3(F)F)C2)C)c2c1CCOC2 C1(C(=O)NCCCN(C(=O)COCCc2ccccc2)C2CC2)CC12CCC2 C1(C(=O)NCC(=CC(=O)Nc2c(OC)nn(C)c2)C)CC2CCCC2C1 CC1CC(NC(c2ccccc2F)=O)CCN1C(c1nscc1Br)=O C(=O)(CCN=c1[nH]c(=NC(C)CN2CCCC2OC)[nH]c2c1CCCC2)NC CC(C)C(CCNC(=O)C(=O)NC1CC1)NC(=O)C(C)(Cl)Cl c1(C(=O)NC2(C)CC(NC(=O)C=C3CCSCC3)C2)cnc2sccn2c1=O c1(-c2nc(CCC)nn2C2CCN(C)CC2)ccc(C#N)c(COC)c1 C1(C(=O)NCC(CNC(c2ccc(Cl)o2)=O)CO)CCC(=C2CC2)CC1 c1(C(N2C(C(=O)NC(CC(C)(C)C)CO)CNC(=O)C2)=O)cc2ccccn2c1 CC(C(=O)NCCCOCC1CCC1)NC(=O)NC1(C)CC1 C1(CC)CN2C(C)(C1)CNC(=O)c1nnc2n1C.C(C)(C)(C)OC(=O)OC(C)C C(N=c1[nH]c(N2CCC(c3ncccn3)C2)nc2c1CSC2)c1nc(C)nn1C c1(CC)cc(Br)ccc1C(=O)NC1CC(C(=O)Nc2sc(Br)cc2C#N)C1 CC(C)C(C)(O)C(=O)NCC(C)(C)OCCNC(c1ccc(OCF)cc1)=O c1(C(N2CC(CNC(C3(CC=C)CCC3)=O)(OC)C2)=O)c(C)cc(C)nc1O CC(C)CC(C)CC(=O)N1CCC(F)(CNC(c2cnc3[nH]cnc3c2)=O)CC1 Cc1c(C(=O)N(C2CCN(C(C3CCc4ccsc4C3)=O)C2)C)c(O)ccc1F c1(COC)ccc(C(=O)NCC(O)CCNC(=O)C(N2CCOC2=O)C)o1 O=C(CCN=c1ccc(OC(F)F)c[nH]1)N1CCC(C(c2ccco2)=O)CC1 c1(C(=O)NCCNC(c2cccc(C)c2F)=O)c(C2CC2)nc2sccn12 C(CC(=O)N1CC(NC(C2(C)CCCC2(F)F)=O)C1)(C1=CCCC1)OCC CC1(C)C2CCC1(C(N1CCCC(NC(=O)Cc3ccsc3)C1)=O)CC2 N1(C(c2ccc(Br)cn2)C(=O)NCc2ccc(F)cc2)CC2CCCC12 C1(CC(=O)NC(C(=O)N(C(CF)CF)C)Cc2ccco2)CCCC12CC2 Cc1ccc(C(N2CCOCC(CCNC(=O)COc3ccsn3)C2)=O)cc1C C1(C(C)(C)O)CN(C(C2CCN(C(=O)NC3(n4ccnc4)CC3)CC2)=O)CCO1 C1(OCC(=O)N(CC(CC)O)C2CC2)CCN(C(=O)C(COC)OC)CC1 C(=O)(CC(C)C(F)(F)C(F)(F)F)NC1CCCN(C(Cc2cnc(C)o2)=O)C1 N1(C(C(C)(C)F)=O)CCC2(CC1)CC(C(N1CCCC1c1ccncc1)=O)C2 CN1CCN(C(C2CC2(F)Cl)=O)C(C(N2CCC=C(F)C2)=O)C1 Cc1c(CC(N2CCC(NC(C3CC(=C4CCC4)C3)=O)C2)=O)cccc1Br c1(C(=O)NCC2C(NC(C(C)Cc3ccco3)=O)C2)cc2ccsc2c(O)n1 c1(-n2cc(CC)nn2)cc(F)ccc1C(=O)NCC1(c2ccc(Cl)cc2)CCC1 C1(NC(=O)CCC2CCC(OC(F)F)CC2)Cc2ccc(Cl)cc2N(O)C1=O N1(C(c2scc(C(N)=O)c2)=O)CCC(NC(c2ccsn2)=O)C1c1ccccc1 N1(C(=O)NC)CC(N(C)C)CC12CCCCC2.c1(OC)cc(Br)cnc1NC Cc1ccc(OCC(=O)NC2(CCCNC(c3c(NC)cncc3)=O)CC2)cc1 C1(C(=O)Nc2cc(SC)nn2C)CC(C)CN(C(=O)CC2CCCN2C(C)C)C1 C1(C(=O)NCc2cscn2)C2CCC(CC2(F)F)N1C(=O)CCN1CCCC1 C(=O)(C(C(=O)N(CCCNC(c1ccc(C)nn1)=O)Cc1ccccc1)OC)OC C1(C(=O)NCC2CCCC(NC(=O)CCCCN3CCCC3)C2)CC2C(C1)C2(F)F c1(CNCC2(C(=O)OC)CC2c2ccc(F)cc2)cn(C)c(=O)nc1O Cc1cccc(C(=O)NCC2CC(O)CN2C(c2ccc(Br)c(O)n2)=O)c1C C1(C(=O)OC(C)(C)C)N(C(=O)OCCC23CC2CCC3N)CC12CCC2C(C)(C)C C(C(C)C(=O)NCCC12CC(CO1)C2)NC(C(C)N(C(C)=O)C)=O c1(CN(C2(C)CC(O)C2)C(C)=O)cc(C)nn1CCO c1(OC)cc(Cl)c(Cl)cc1C(N1CC(NC(=O)C(F)=C2CCC2)C(O)C1)=O Cc1nc(C2CCC2)sc1CC(=O)NCC(CCO)c1ccncc1 C(=O)(CN1C(=O)Cc2ccccc21)NC(CN(C(c1cnccc1Cl)=O)CC)C CC(C)(C)C(=O)C(=O)N1CC2(CC2)CC1CNC(C1CC(CC(F)F)C1)=O c1(C(=O)NCC(O)CNC(C2COCC3(CCC3)O2)=O)cc2cc(Cl)ccc2s1 c1(C(=O)NC2CC(CNC(=O)C(O)Cn3cncn3)C2)[nH]c2ccccc2c1Cl C1(NC(C2CCC(F)CC2)=O)CC1C1CCCN(C(=O)CCc2cnn[nH]2)C1 C1(N=[N+]=[N-])(C(=O)NCCC2C(C)C2)CCN(C(=O)CCn2cccn2)C1 N1(Cc2c(NC(N(C)C)=O)cccc2)CCC2CCOCC2C1 C1(NC(C=CC(C)(C)NC(C2CNC(=O)N2)=O)=O)CCn2nccc2C1 Nc1cc(F)c(F)cc1C(N1CC(CNC(C2CC23CCOC3)=O)C1)=O C1(OC)CC(CC(=O)NCC2CC2NC=O)C1.C(C(F)F)N C1(O)(C(C(=O)NCC(CSC)OC)F)CN(C(=O)CCN(C)CCO)C1 c1(CC)[nH]nc(C(N2CC3C(C2)N3Cc2cc[nH]c2)=O)c1F c1(CCNC(C2CC3CC3N2C(c2c(Cl)csc2Cl)=O)=O)ncccc1F C1(C(=O)NCC2CC(OC)CN2C(=O)CCCc2cccs2)CC(C(C)C)=NO1 CC(C)C(C(=O)N(CC)C1CC1)NC(N)=O.c1(NC(=O)C(C)N(C)C)ccccc1 Cc1c(C(N2CCC(CS(N)(=O)=O)C2)C(=O)Nc2ccc(Br)cc2)ccnc1F c1(C(C)C)ccc(C(CCCNC2CCCC2N)N(C)C)cc1 CCCCC(CC)C(=O)NC(C1(CNC(=O)CCSc2ccccn2)CC1)C C1(C(N(C)CC2CCN(C(CSCC#C)=O)CC2)=O)CC2CCCC2C1 c1(CCC(N2CCC(CCC)(CO)C2)=O)ccc2c(c1)CCO2 CC(C)(C)CCC(=O)N(C1CCCN(C(=O)Cc2cc(F)ccc2Cl)C1)CCF C(=O)(CCCCN=[N+]=[N-])NC(CCCC)C(=O)NC1CCC(CO)C1 O=C(C1Cc2ccc(Cl)cc21)N1CCC2CCC(C1)N2C(c1cc(Cl)c(Cl)[nH]1)=O C1(CNC(C2N(C(C(CCC)OC)=O)CC=C2)=O)CCCC12CCC2 CCC(CNC(=O)CC1CC(O)C1(C)C)(CC)NC(=O)C(CC)Oc1ccccc1 N1(C(c2c(CC)non2)=O)C(CNC(c2cc(C(N)=O)on2)=O)CC2COCC12 N1(C(c2ncc(C)cc2C)=O)CCC2(CC1)CCN(C(C1CCSC(C)C1)=O)C2 Cc1cc(C)c(C2CCCN2C(=O)C(=O)N2CC(CC#N)C2)c(C)c1 C=CCCCC(C(=O)N1CCN(CCO)C(=O)C1)NC(=O)C(F)CCCC c1(C(NOC)=O)cccc(OC(=O)C=Cc2ccccc2)c1 c1(C(CC(=O)NC2CC(C(F)(F)F)C2)NC(CSC)=O)ccc(F)cc1 [N-]=[N+]=NCCCCC(=O)NCC(CO)NC(=O)CCCNC(N)=O C1(C(=O)NCCC=CC)CC2(CCN1C(=O)C(C)N1CC(C)C1)CC2 c1(C(N(C)CC2CCCN2C(=O)Cc2cnnn2C)=O)cc2c(=O)cc[nH]c2s1 C(=O)(C1c2ccccc2CN1C(=O)CSc1nc[nH]n1)Nc1cnn(C)c1Cl c1(CC(=O)NCC2(NC(C=C(C)Cl)=O)CC2)cc(C)cc(C)c1 N1(C(C(=O)NC)CCCOCc2ccccc2)CCCC2(C1)NC(=O)NC2=O N1(C(C)C)CCCC(C(=O)NCC2CCCCN2Cc2cnc[nH]2)C1 Cc1cccc(C(=O)NC2CCC(NC(=O)CCC=CC(C)C)CC2)c1C(F)(F)F C1(C(=O)NCCCOCCNC(c2cc(C(C)C)nn2C)=O)NC(=O)C2CCC12 Cc1[nH]c2ccc(NC(N3CCN(CCC(C)C)CC3)=O)cc2c1C C1(C(N2CCC(=CCNC(C3C(C=C)C3)=O)CC2)=O)CC2CCC(C1)C2F CC1(C)C(C(=O)NCC2CC(O)(CNC(C3CCC(C(N)=O)CC3)=O)C2)C1(C)C Cc1ccc(C(=O)N(C)C)cc1S(=O)(=O)CCO.C1(=O)C(Cc2ccccc2)N1 C1(C#N)(NC(c2ccc(N3CCC(C)C3)cc2)=O)CC2CCC1CC2 N1(C(C2(NC(C3CC(OC)C3)=O)CCC(C)(C)C2)=O)CCN(C(C)=O)CC(C)C1 C1(C#N)(C(=O)OC)CCN(C(=O)NC2CCCC2C(C)C)C1 C1(C(=O)NCCC2(NC(c3sccc3C)=O)CCCC2)(NC(C)=O)CCCCC1 C1(C)(COC)CC(NC(=O)Cn2cnnn2)CN1C(C1CCCN(C(C)C)C1)=O C(=O)(CCCC1CCOCC1)N(CC(C)(C)NC(C(C)c1ccco1)=O)C C(CCN=C(NCCS(C)(=O)=O)NC(c1ccc(SC)cc1)C)SC C(CN=c1cnc(C(=O)OC)c[nH]1)C1(COC)CCC1 N1(C(C(C(C)C)F)=O)CCN(C(=O)CNC(C2CCC2)=O)C(CCO)C1 N1(C(c2ncc(C)c(C)c2)=O)CC2(C1)CN(C(=O)CC(C)C1CC1)CC2CO C1(C(=O)NCCC(C)NC(C2(O)CC3(CCOCC3)C2)=O)CC(C)(C)C(C)(C)C1 C(=O)(C(C)CCOC)N(CCC(=O)NC(c1nccn1C)C)CC#C c1(C(=O)NCCNC(C2N(C)C(=O)NC2)=O)cnc2ccc(F)cn12 c1(C(N2C(CNC(C(C)SC(C)C)=O)CC(O)C2)=O)csc2c1CCCC2 N1(C(c2n[nH]c(C)c2Cl)=O)CCC2CN(C(C3(C(F)F)CCCO3)=O)CC2C1 Cc1cc(=NCC2CCN(C(c3cc4c(s3)CCC4)=O)CC2C)[nH]c(C)n1 C(=O)(C1CCCn2ncnc21)N1CCC(NC(=O)Cn2ncc3ccccc23)C1 c1(C(=O)OC)cc(Cl)n[nH]c1=NCCN1CCC(OC(F)(F)F)CC1 c1(C(=O)NC(C(=O)NCCN(CC(C)C)CC)c2ccco2)nccc(C)n1 c1(CN2CC(CNC(C(CC)(C)OC)=O)OCCC2)ncc(C)c(OC)c1C C#CCC(CC(=O)Nc1ccc(O)c(CO)c1)NC(=O)CC1CCC2CC12 CCCC(C#N)C(=O)N1CCCCC1CNC(c1c(C)nn(C(F)F)c1C)=O N1(C(C(=O)NCC2CCCO2)C2CCSC2)CCCCC1CCF N1(C(C(CC)C)=O)CC(C2CCN(C(=O)Cc3ccc(CC(C)C)cc3)CC2)C1 N1(C(Cc2c(C)cco2)=O)CC(NC(=O)C(C)n2ccnn2)C(N=[N+]=[N-])C1 C12(C(=O)NC3CN(C(C)=O)C3)CC(NC(=O)C(C)(C)c3ccccn3)(C1)C2 C1(NC(c2c(C)nc(C)s2)=O)CC2CCC(C1)N2C(C1CCCC(C#N)C1)=O C1(C(N2CCC(N3CCN(C(C4(O)CCOC4)=O)CC3)C2)=O)CCCNS1(=O)=O CC(CC(=O)NC12CCC(CC1)CC2)C(C)(C)NC(c1cc2cc[nH]c2cn1)=O N1(C(c2cccc(CNC(C3(CC)COC3)=O)n2)=O)CCC(C2(C)CC2)CC1 N1(C(c2cccc(C)c2Cl)=O)CC2=C(C1)CN(C(=O)C(N1CCCC(O)C1)C)C2 S(=O)(=O)(c1csc2ccccc12)N1CCN(C(=O)Cc2ccc(O)cn2)C2C1C2 C1(C(=O)OCC(=O)NCCCN(CCCN(C)C)C)CN2CCCC1CC2.C(CF)O c1(C(C)C(=O)NCC2(NC(=O)CC3COC(=O)N3)CCOCC2)cccc(Cl)c1 C(C)(C(=O)NC1CCCC(CC(=O)NCCN(C)C)C1)(C(C)C)NC(C)=O N1(C(=O)C(F)(F)F)CCN(Cc2ccccc2)CC1NCC12CCC(CC1)CC2 c1(C(=O)NCC(CNC(C2C(CC)C2)=O)F)cc(Cl)c(Cl)cc1C c1(C(=O)NCC2C3CN(C(CCC4CCC(=O)NC4)=O)C2C3)ccc([N+](=O)[O-])[nH]1 C1(C(F)(F)F)(C(=O)OC(C)(C)C)CC=CCO1.C12CCC(C1)C(=O)NC2 CCCC(CNC(=O)C(O)CCN(C)C)C(=O)NCC1(F)CN(C)C1 C1(NC(c2cccc(NC(C)=O)c2)=O)C2CCC1CN(C(=O)C(F)(F)C(F)F)C2 c1(CC)cc(=NC(=O)C(CC(C)C)N(CC(=O)NCC(F)F)C)[nH]n1C C1(C)(C(N(CCC(C(C)C)NC(=O)C(C)S(C)(=O)=O)C)=O)CCCS1(=O)=O c1(CCC(=O)NC(C2CCCCC2)CNC(CCOC)=O)nc2cc(Cl)ccc2s1 C(C(CC(=O)NCCC(=O)NO)C1CCC1)NC(C1C(CCOC)C1)=O C1(C(N(CC(C)C)CC)=O)CC2(C1)CC(O)C2.C1C(C)NC(=O)CS1 CC1(O)CCC(CC(N2CCCCC(NC(=O)C(C)S(N)(=O)=O)C2)=O)CC1 C1(O)(CCNC(c2ccc(CCC)[nH]2)=O)CCN(C(=O)CCc2ccsc2)CC1 c1(C(C(=O)N(CC(O)CNC(=O)CSCC2CCCO2)C)(F)F)ccc(F)cn1 C(CC(C)C)(C(=O)NS(CC1N(Cc2cn(C3CCCC3)nn2)CCC1)(=O)=O)OC n1(C(C(N2C(CCNC(c3c(C)csc3)=O)CCC2)=O)C)c(C)cc(O)cc1=O C1(CCC)CN(C(=O)CC2(CC)CCC2)CCN1C(=O)COc1ccccn1 N1(C(C(CC)(C)O)=O)CC(CNC(c2cc(C)ccn2)=O)OC2(CCC2)C1 CN1CCCC(O)(CC(=O)NCC(C)(C)CCNC(C2CC(O)C2)=O)C1 Cc1cnc(C(N2CC(NC(C3CCSC(C)C3)=O)C(O)C2)=O)cn1 CCC(C)(C)C(=O)C(=O)N1CC(C(O)C(=O)NCCOC2CC2)C1 C(=O)(CC(C)(C)CC)NCC=CCNC(Cc1cc(CC)nn1C)=O C1(CN(C(=O)CCC2CC2(Cl)Cl)C)C2CCCC1N(c1nnc(C3CC3)o1)C2 N1(C(CC(C)CF)=O)CCN(C(c2ccc(CN(C)C)cc2)=O)CC1C1CC1 Cc1ccc2[nH]c3c(c2c1)CCCC3Nc1ccc2ccc(C)nc2c1C N1(C(CCC=CC)=O)CCC2(CC1)CC2NC(=O)Cc1nc(Cl)c(C)c(=NC)[nH]1 C(CC(C)(C)CC(=O)N1CCC(CCC(=O)NC2COC3(CCC3)C2)CC1)OC C1(C(=O)NCCC2(CN=c3nc(CC)[nH]s3)CC2)CCC2(CCCC2)C1 c1(C(=O)N)cccc2oc(=N)[nH]c12.C1(COC(C)C)CCCCC1.C12(CC1)C(=O)NC2 c1(C(C)(C)C)cc(C(=O)NCCOC2CCN(C(C3(C#N)CCC3)=O)C2)on1 CCCCCCC(=O)N1CC(N2CCC(NC(=O)C(C)CC3CCCCC3)C2)C1 N1(C(c2cccc(C)c2)=O)CC2(CC(NC(c3oc(C4CC4)nc3C)=O)CO2)C1 C1(F)(CNC(COCc2c(C)ncs2)=O)CCCN(C(C2CCCCC(=O)N2)=O)C1 c1(C(N2CC(CC(=O)NCc3c(CC)nns3)C2)=O)cnnc(-c2ccccc2)c1 N1(C(C=Cc2cn(C)nn2)=O)CCC2(CCC2NC(C2OCC2(C)C)=O)CC1 CCC(=O)CCC(=O)N1CCC(F)(C(=O)NCC(C)C(C)O)CC1 c1(C(N2CC(CNC(C(C)OCC=C)=O)C(O)C2)=O)ccc(-n2cnnn2)cc1 C1(C(N2C(C(N3CC(c4ccc(C)o4)C3)=O)CC2C)=O)CCCCCN1C C1(CCNC(C2(N(C)C)CCCC2)=O)(CC(=O)NCCOCC)CCSCC1 CC(c1cccs1)=CC(=O)NC1CCN(C(=O)C(=Cc2cccnc2)F)C1 Cc1ccc(Br)c2c1C(NC(=O)N(C(C(C)(C)C)c1ncccn1)C(C)C)CC2 N1(C(c2cnc(SC)nc2)=O)CC(NC(c2ncc(Br)cc2C)=O)C(C#N)C1 c1(C(C)C(=O)NCC(c2ccccn2)C)cc(F)cc(F)c1 c1(CC)cc(CC(=O)NC(C2CN(C(C3(N(C)CC)CCC3)=O)C2)C)on1 C1(OC(N2CCCC(c3c(OC)ccc(F)c3)C2)=O)CCC12CCCCC2 C(=O)(CC1=CCCCC1)NCC1(CNC(C2CCC(OC)CC2)=O)CC1 C1(OC)CC(NC(=O)CC(C)(C)C2CC2)CN(C(C2C(C)(C)C2(C)C)=O)C1 c1(OCC(=O)NCC(N(C)C(C2CC3CC3C2)=O)C2CC2)ccc(F)cc1O N1(C(=O)C=CC(F)(F)F)CC2CC1C2NC(c1ccc(C2CCCCC2)o1)=O c1(-c2nc(CNC(=O)OC(C)C)nn2C2CCOC(C)C2)cc2oc(Cl)cc2[nH]1 C12(CNC(C(COC)(C)C)=O)CN(C(=O)Cc3nn(C)cc3C)CC1CCO2 C1(C#N)(C(N(CCC)CCNC(=O)Cc2cncc(C)c2)=O)CCN(C)CC1 CCC(C#N)C(=O)N1CC(F)CC1CNC(=O)CC1NC(=O)NC1=O c1(C(=O)NC(CNC(C2(COC)CCOCC2)=O)C)ccc2nc(C)[nH]c2c1 CCCCC(CCCC)C(=O)NCC1C(C)CCN1C(c1ccc(F)c(Cl)c1)=O CN1CC(NC(C2CCN(C(C3COCC3C(N)=O)=O)C2)=O)C2(CC2)C1=O C(=O)(CCCCNC(C1(C)CCCC1O)=O)N(C)CC1SCCS1 c1(-c2ccc(CCC)s2)nc(CS(C)(=O)=O)nn1CCCCO N1(C(C)C)CCC(C(=O)NC2CCC(NC(=O)CN3CCCC3)C2)CC1 CCCCCC(O)C(=O)N(C1CCCC1)CCCNC(=O)CCCC(C)=O N1(C(Cn2cc(C)c(O)nc2=O)=O)CCN(C(=O)CC2CC(=O)C2)C(C)CC1C c1(C2CC2C(=O)NCCCCCNC(C2CCC(C(C)=O)O2)=O)cccc(C)c1 C(CC(C(=O)N1CCC(SC)C1)NC(=O)CCc1cnccn1)OC C(=O)(C(CC(C)CC)NC(=O)Cc1cccc(F)c1)NC1C(C#C)CCC1 C1(C(=O)NC(CNC(c2cnc(CCCC)s2)=O)CO)CCc2nccn2C1 c1(CNC(C(CCOCC)NC(=O)CCc2ccccn2)=O)cc(C)cc(F)c1 CCC1CCCc2sc(NC(=O)C(=O)NCCSc3ccc(F)c(F)c3)nc21 C1(C(=O)NCCCNC(c2cnn[nH]2)=O)(CO)CC12CCC2 C1(C(C)NC(=O)NC2CCCC2C)CCN(CCCO)CC1 C(=O)(CCCC(C)(C)C)NCCC(CC)(CC)NC(=O)Cn1ccc(Br)n1 C(=O)(CC(CNC(c1cc(C)sn1)=O)C1CCC1)N(C(C)CO)CC c1(C(=O)NCC2(C(=O)NC3CCC(C#C)C3)CC3(CC3)C2)cc(C#N)oc1C N1(C(Cc2cc(C)on2)=O)CC2CCC1CN2C(=O)C(C)C1CCCO1 c1(C(N2C(CNC(C3CC(C)N(C)CC3)=O)CC2)=O)[nH]cc2c1CCS2(=O)=O c1(NC(C(=O)N(CCC#C)C)=O)ccc2c(O)ncc(F)c2c1 C1(OC)CC(C(=O)N(CC(N2CCCC2)C)C)N(C(=O)CCc2ccn(C)c2)C1 Cc1cc(C)c2c(c1)CN(C(=NCC1CC13CC3(F)F)NCc1cccs1)CC2 N1(C(CC=C=C)=O)CC2CC1CC2NC(c1ccc2c(c1)CC2)=O N1(C(CC=CC=C)=O)Cc2ccccc2CC1CNC(C1OCCC1C)=O N1(C(C=CS(C)=O)=O)CCC2CN(C(c3c[nH]c(C(=O)OC)c3)=O)C2C1.OC=C C#Cc1cc(C(=O)NC2CN(C(=O)CCCc3ccsc3)CCC2F)cc(N)c1 C=CCC(CC)C(=O)N1CCC(C(N2CC=CC2(C)CO)=O)C1 c1(C(N2C(C3(NC(c4ccc(OC)o4)=O)CC3)CCC2)=O)ncnc(O)c1F CCC(C)CC(CO)NC(=O)C(c1ccccc1)NC(=O)C=CC1CCCCC1 C1(C(=O)NCC(C(C)C)(C)NC(=O)C(O)P(C)(C)=O)CCS(=O)(=O)C1(C)C Cc1cc(C#N)cnc1C(=O)NC1(C(=O)NC(CF)C(F)(F)F)CCC1 c1(C(=O)NCC(C)NC(c2coc(C3CCC3)n2)=O)cccc2ncnc(O)c12 Cc1c(Cl)ccc(C(=O)N(C(C)CNC(=O)CCc2ncc(F)cn2)C)c1N CCN=c1[nH]cc(C(N2CC(NC(C3(C)CCCO3)=O)CC2C)=O)s1 C12(CNC(=O)C(O)C(F)F)CCC(NC(c3cc(Cl)cnc3O)=O)(CO1)C2 c1(C(=O)OC)ccccc1-c1ccc(OC2CCN(C(=O)NCC3CC3)C2)nc1 C(C(CNC(C1CC12CCCCC2)=O)S(C)(=O)=O)NC(C(C(C)C)F)=O CCC(CC)(CCNC(C1CC(C)C1)=O)NC(c1nc(-c2ccco2)sc1C)=O C1(CNC(C2CCC(C)O2)=O)C(C2CC2)CCN1C(C1CCCCC1O)=O C1(CCC)CN(C(=O)Cc2cnc[nH]2)CC1NC(=O)CC1(O)CCOC1 C12CC3(CO1)CN(C3)C(C1CC=CC1)C(=O)N2.O=CNCCC1CC1 CC(C)CCC(=O)C(=O)NCC(C)(C(C)C)NC(c1cnsn1)=O c1(CCNC(C(C)N2CCCC2)=O)cc(C(=O)NC2(CC3CCC3)CC2)no1 C(=O)(CCCC1(N(C(=O)Cc2cnc(C)s2)CC)CCC1)NC(c1nncn1C)CC C1(NC(CN(C(=O)OCC)C)=O)C2CC3C1C3C2C(N1CC(n2ccnc2)C1)=O c1(C(=O)NCC(CC=C)NC(C2(C)CC2)=O)ccc2c(c1)nc(C)c(=O)n2C N1(C(C(c2cccc(F)c2)C)=O)C2CCC1CC(N(C)C(c1cscn1)=O)C2 N1(C(c2c(OC)scc2)=O)CCN(C(C2(OC)CCC(C)(C)C2)=O)CC12CCC2 c1(OC)c(CNC2C3CN(C(c4cccc[n+]4[O-])=O)CC23)cccc1F c1(CC)[nH]nc(C(=O)Nc2nc(CC(=O)Nc3cnn(CC(C)C)c3)cs2)c1F c1(C(=O)NC(CCOC)C(=O)OC(C)(C)C)c(N(C(=O)OC)C)cccc1F C12(C(=O)NC(CNC(CCOCC#C)=O)(CC)CC)CC(CO)(C1)OC2C C(CCC(C)C)(c1n(CCOCC)nnn1)NC(CSC)Cc1ccccc1 C1(NC(C)=O)CC(N=c2[nH]c(=NCCCN(C)C)c3cccc(F)c3[nH]2)C1 c1(CC)c(C(=O)NCCCCN(C(=O)C(N2C(C)CCC2C)C)C)ccn1C N1(C(c2[nH]cc(C#N)c2)=O)CC2CC(C(N3C4COCC3C4)=O)CC2C1 C1(NC(CCc2c(C)nn(C)c2)=O)CN(C(c2cccn2C)=O)CCC1CO Cc1nc(Cl)cc(Cl)c1C(=O)NCCC1CCCN(C(=O)C(C)(C)CCl)C1 c1(NC(C2C(c3ccc(C)cc3)CCCC2)=O)ccc(Cl)c(C)c1 c1(C(N2C(CNC(C3CN(C(C4(CC)CC4)=O)C3)=O)CCC2)=O)ccc(C#N)[nH]1 c1(C(C)NC(c2ccc(Cl)s2)=O)cccc(-c2noc(C(F)F)n2)c1 C(=O)(CCCCCSC)N1CC(CN(C(C2N(C(=O)NC)CCC2)=O)C)OCC1 c1(C2C(C(C(=O)N(CCOCC#C)C)NC(=O)C=C3CCC3)C2)ccco1 C1(C(N(C(CC)C)CC)=O)CCCN(C(c2nccn2C)C)CC1 c1(C(=O)NCCCNC(C2CCC(C(=O)OC)C2)=O)c(C)oc(C)c1Br C12(NC(CC(CC)C3CC3)=O)CCC1CN(C(c1cnn(CC)c1Cl)=O)C2 C1(NC(CC=CCC)=O)(CC)CCN(C(C2CCN2CC)=O)CC1 N1(C(c2cccnc2OCC)=O)CCC2CCN(c3cc(Cl)nc(Cl)n3)CC2C1 N1(C(C(C)(C(c2ncn(CCCC(=O)OC)c2)=O)C2CC2)=O)CC2CC2(CO)C1 N1(C(c2cnc(C)s2)=O)CC(CC(=O)NC(c2cn(C)nn2)C)CC1(C)C c1(CC(N2CC3C(C(=O)NCCC(=O)N(C)C)(C3)C2)=O)ccc2ccccc2c1 c1(OC)ccc2oc(C(N3CC(NC(=O)C(CCSC)N(C)C)C3)=O)c(C)c2c1 N1(C(c2scc(C)c2)=O)CCC2CCCN(C(=O)CC3CC4(CCC4)C3)C2C1 C1(CN(C(C2C(C#C)C2)=O)CC)CCCN(C(c2oc(CO)nc2C)=O)C1 Cc1cnn(C)c1C(=O)NCC1CCN(C(C2COCCC2C)=O)C1 C12(C(N3CC(C)C(NC(=O)CN4CCCNC4=O)CC3)=O)CCC(F)(CC1)CC2 S(=O)(=O)(CCC(=O)N1CCC(CNC(c2ccnc(OC)n2)=O)C12CC2)NC C123COC(C1)(C2)CNC(=O)C3.c12ccncc1C2.C12(CC1)C(=O)N2.CSC C(=O)(C1=NNC(=O)C1)NCC1C(NC(Cc2cccc(COC)c2)=O)CCC1 C1(CC)(CC)CC(NC(c2cccc(O)n2)=O)CN1C(c1cnc[nH]1)=O CC(C)C(O)(C(=O)N1CCC1CNC(=O)CN1C(=O)NC(C)(C)C1=O)C(F)(F)F C1(NC(CCCN(C(c2c(CC)cc[nH]2)=O)C)=O)CC(C2CCC2)C1 C1(N(C(COCCCCC)=O)CC)CCN(C(=O)CCN2CCC2)CC1 C(C(C)C)(C(O)C(=O)NCC(C)CC(=O)NCC(CO)C1CC1)OC c1(N(C)C)cnc(C(=O)C(N2C(C)(C)C(=O)OCC2)=O)nc1.C(C)(C)(C)O.C1(CO)CC1 c1(CCC(N2CC3C(NC(C(C)OCCC=C)=O)(C3)C2)=O)ccc2cnn(C)c2c1 C(C1CCN(C(c2cscn2)=O)CC1)=CC(=O)NCC1(C)CC1(F)F O=C(CC(C(F)F)NC(C1(CC2CC2)CC1)=O)NC1CC(=O)NC(=O)C1 c1(C(=O)Nc2cccnc2OCCCF)ccc2ncsc2c1 C1(N(C(C)(C)C)C(C2(C#C)CC2)=O)CCN(C(=O)OC(C)C)C1.C(C)(CC)NC=O N1(C(c2cncn(C)c2=O)=O)CC2CN(C(c3ccnc(O)c3)=O)CCC12 Cc1cc(C(N2CC(NCc3c(O)cccc3F)C(O)C2)=O)ncc1Br C=CCC(C)(CC)C(=O)N1CC2(CC(CN=[N+]=[N-])C2)C1 Cn1ncc(CCC(=O)NCCC2CCN(C(C3(O)CCC3)=O)C2)n1 c1(C(=O)NCCCN(C(CC2C(C)=NNC2=O)=O)CCO)noc2c1CCCC2 c1(C(=O)NC(CC)CNC(c2ccn(C)c2)=O)ccccc1OCC1CC1 C12(N(C)C(c3ncoc3CNC(=O)CN3CCCC3=O)=O)CCCCC1OCC2 C(=O)(C1=Cc2ccccc2OC1)NCC1N(C(c2c(C)c(F)ccc2)=O)CC1 CCCCCCCC(=O)NCC1(C(=O)NC(CO)CC(F)(F)F)CCC1 C1(NC(C(CC)n2cncn2)=O)CC2(CCCN(C(=O)CC3CC4CC4C3)C2)C1 N1(C(C(CCC)F)=O)CC(F)(F)CC1(C)CNC(=O)CCC1CCCN1C c1(CSCC(C)C)ccc(C(=O)NC2CCCC2NC(c2cnsc2)=O)o1 CC(CCCCCO)NC(C1CCCCC1CNC(=O)CC1OCCO1)=O C1(CN(C(c2cnnn2C)C(=O)NCCCCCC)C)CCCC(COC)C1 C1(CC#C)(C(=O)NC2(C(=O)NCC(O)COCC3CCC3)CC2)CCCCO1 N1(C(C2(C#N)CCN(C(c3csnn3)=O)C2)=O)CCc2c(O)n[nH]c2C1 C1(OC)CCN(C(=O)CC2C=CCCC2)C(C)C1 c1(C(=O)NC2CC(C)(CNC(C(C)C3CCC3)=O)C2)ccnc(N2CCCC2)c1 CC1CCCN(C(=O)CN2CCC(O)CC2)C1CNC(c1cnn(CCO)c1)=O C(C(C)(C(=O)N(CCCC(=O)N(C)CC1(C#N)CC1)C)OC)OC C1(NC(CSCCC)=O)CN(C(=O)CNC(C)=O)C(c2ccccc2)(SCC)C1 C12(NC(c3sc(C)c(O)n3)=O)CCCCCC1N(C(c1n[nH]c(=N)[nH]1)=O)CC2 c1(CC)c(C(=O)N(c2ccc(N3CCCCC3)nc2)C)[nH]c(C)c1CCOC Cc1cc(C(=O)NC2CC(NC(=O)Cc3c(F)cccc3Cl)C2)cc(C)c1O c1(CN(C(C2CCN(Cc3cnn(C)c3)CC2)=O)CC)cccc(Br)c1 C(=O)(CS(=O)(=O)CC)N(C1CCCC1NC(c1nc(C(C)OCC)sc1)=O)CC c1(C(=O)NCC2C3CN(C(c4nc(COC)oc4)=O)CC32)ccc(N)c(Cl)c1O Cc1nc(O)nc(O)c1CC(N1CC2CC1C2NC(c1csc(C2CC2)n1)=O)=O CC(C)C(CC(=O)NC(CO)C(C)NC(=O)CS(N)(=O)=O)c1ccccc1 C1(C(=O)NCC(CC)(C)Cl)CN(C(c2cc(C#N)cs2)=O)CCN1C C1(OC)CC(C(C)(C)C)CN(C(=O)CC2CCC2)C1 C1(CNC(C(C)N(C)C)=O)CN(C(=O)CC2CC3C=CC2CC3)CCC1C C(=O)(C(C)(C)C(=O)NC1CCCC(CC(N2CC(F)(F)CC2CO)=O)C1)N(C)C C1(NC(CN(C)C(c2ccccc2)=O)=O)CC2CCC1N2C(C1COC(=O)C1)=O O=C1CCN(C(c2ccn(-c3ccccc3)n2)=O)C(C2CC2)C1 C1(NC(c2c(C)cc(F)s2)=O)CCC2(CCN(C(C3(N=[N+]=[N-])CC3)=O)CC2)C1 C1(NC(COC)=O)CC12CC(NC(C1(CO)CCCCO1)=O)C2 Cc1ccc(C=CC(=O)N(C2CC(C#N)C2)CC(=O)NCC(O)(CO)CO)cc1 C(CNC(=O)CCc1cn[nH]c1)(C(=O)NC(C)(C)C1CC1)OC C1(N(C)CCO)CN(C(=O)OC(C)(C)C)CC1CCOc1cccc(F)c1 N1(C(C(C=C)CC)=O)CCC(C)CC1C(=O)NC1CCCOC1 c1(OCCC(=O)NCC2CCCC(NC(CCNC(C)=O)=O)C2)cc(F)cc(F)c1 C1(CC)CN(C(=O)CC)CCN1N1CCC(c2cnn(C)c2)C1 C1(CC#C)(C(=O)NC(C)(CC)CCO)CCN(C(c2ncn(C)c2C)=O)C1 C1(CCC(=O)NC(c2cc(Br)no2)(C)C)CCCN1C(=O)COCCO C1(NC(CC(CC)C)=O)CCN(C(c2csc3ccccc23)=O)CC1(C)C C=CCC(F)(F)C(=O)NCC1(CNC(=O)C=CC(C)(C)NC(C)=O)CCC1 c1(C(=O)NC2CN(C(c3c(OCC)n[nH]c3)=O)CC(O)C2)cc(F)cc(F)c1O C(C1CCOCC1)=CC(=O)NCCC1CC(NC(=O)COc2cccnc2)C1 S(=O)(=O)(C=Cc1ccccc1)N1CCN(c2n(CC3CCC(C)O3)nnn2)CC1 C1(C(=O)NCCCCCNC(CNC(=O)NC)=O)COCCC1C c1(C(N2CCN(C)C(CNC(C3CCC(C)(C)C3)=O)C2)=O)ccc2cc[nH]c2c1 c1(CN2CC(NC(CC3CCCN(C)C3)=O)C(O)C2)cccc2nccnc12 c1(C(=O)NC2C(CNC(C(c3cscn3)N(C)C)=O)CCC2)ccc2c(c1)CC2 C1(C(N(CCC=C)CC)=O)CC(O)CCN1C(c1ccccc1C#N)=O c1(C(N2CC(CCCCNC(C3CC(OC)C3)=O)C2)=O)nn(C)c2ccc(F)cc12 CC(CCNC(C1CCCCN(C(=O)Cc2cnns2)C1)=O)C(C)(C)C N1(C(c2c(C(C)C)ocn2)=O)CC2CC(C1)CN(C(C1NC(=O)CC1C)=O)C2 N1(C(c2c(C(C)NC(=O)C=Cc3cn(C)nn3)noc2)=O)CCC(O)CC1C1CC1 N1(C(CC2(CC=C)CCCC2)=O)CCC(NC(=O)C(C)CCCC)CC1C c1(OC(c2nc(C)n(-c3ccc(I)c(F)c3)n2)=O)cccc(C#N)c1 c1(C(=O)NC2CC(CNC(c3ccoc3Cl)=O)C2)ccc2cnccc2c1 c1(OC)ccc2c(c1)CC(C(c1nnnn1C)Nc1ccc3nc(C)sc3c1)CC2 Cc1ccc(C(=O)NCC2CN(C(=O)C(c3cccn3C)=O)CCC2C)c(C)c1 c1(C2(C)CC2)cccc(C)c1NC(=O)C(CCC1(C#N)CCC1)N(CCO)CCO C1(C(=O)NC2C3CN(C(=O)CCOC4CCCOC4)CC23)CCc2nn[nH]c2C1 C=C=CCN=c1[nH]c2c(c(=NCC3(C)CCOCC3)[nH]1)CCCC2 C1(C(=O)NC(C=C)COC)(NC(c2[nH]ccc2CC)=O)CC(O)C1 C1(NC(C(C)SCC)=O)CC2(CCCN(C(C3CN(c4nncs4)C3)=O)C2)C1 C1(NC(c2onc(C)n2)=O)CCN(c2ncns2)CCC1CO C1(F)(CNC(CN(C(C)=O)C)=O)CCN(C(=O)Cc2cscc2Br)C1 C1(F)(C(=O)NCC2C(NC(Cc3ccc(C)nc3)=O)CC2)CCCN(C)C1 CCCC(C#N)C(=O)N1CCCC(C(N2CCCC(C)(C)C2)=O)C1 N(C1=NCCC(=O)NC2CC(F)(C2)C(=O)NCCN1)CS(C)(=O)=O.C=CCOC C1(C2CCCCC2)(C(N2CCCC(NC(=O)CC3CCOC3)CC2)=O)CC1 c1(C(N2CCCCC2CCC)C(=O)NCC=C)ccc(OC(F)F)c(C)c1 c1(C(CC2CC2)NCCN(C2CC2)CC)nnnn1C1COC1 c1(OCCC(=O)NC(C)CCCNC(=O)CC2CCCC2)ccccc1F C(=O)(C1=CCS(=O)(=O)C1)N1CC(N(C(c2ccc(C#C)o2)=O)C)C(C)(C)C1 c1(C(N2CCC(CC(C)NC(C#CC(C)C)=O)CC2)=O)ccc2ncccn12 CCC(C)C(C)C(=O)NCCCOCCN(C(=O)Cn1ccnn1)C C1(OC)CC(CNC(c2ccnnc2Cl)=O)N(C(c2ncnn2C)=O)C1 c1(C(=O)NCC2(NC(c3cc(CCCCC)[nH]n3)=O)CC2)ncnc2cc[nH]c12 C1(CC#C)CCN(CC(=O)SC2CC3CC3C2)C1 C(=O)(C(C)(C)CC(F)(F)F)NC1COC2C(NC(c3cc(C)ncc3)=O)COC12 C12(NC(C3CC(OCC)C3)=O)CCCC(NC(=O)CCn3ccnn3)(C1)C2 C1(C)(C(N(CCCN(C)C(c2csc(Cl)c2)=O)C)=O)CCNC(=O)C1 C1(CC(=O)NCC(CNC(C2(F)CC3(CCC3)C2)=O)CO)CC(=O)NC(=O)C1 N1(C(CCCOCC)=O)CCC(C(C)C(=O)NC2CCOC2C(C)C)CC1 c1(C(=O)NC(C(C)NC(=O)C=CS(C)=O)CO)ccc(C(C)(C)C)c([N+](=O)[O-])c1 N(C(=NCCCCOC1CCC1)NC1CC1)Cc1c(C)noc1C C=CCCCC(C)(C)C(=O)N(C)CC1CCN(C(=O)C(O)CC2CCOCC2)C1 c1(C(N2CCC(C)(CCNC(CNC(CC)=O)=O)C2)=O)cc(F)c2c(c1)CCC2 N1(C(c2cc(CNC(CC3CCC(=O)N3)=O)sc2)=O)CCC2(CCC2)C(O)C1 C(C(CC(C)C)C(=O)NC1(CO)CC(F)(F)C1)NC(C(CC(C)C)O)=O c1(C(=O)NCCC2CC(OC)CN2C(C2COCCO2)=O)cn(C)c(=O)n1C N1(C(=O)Oc2ccc(F)cc2)CC2CCC(F)(F)C2C1 c1(C(N(C2CCN(C(C(C)OC)=O)CC2)CC2CC2)=O)ccc2cncn2c1 c1(NC(c2ccc(Cl)cc2)c2ccn(C)n2)nccc(F)n1 C12(C(=O)NC3CN(C(C=CCCC=C(C)C)=O)CC3C)CC(C)(CCO1)C2 c1(C(=O)NC2C3OCC(NC(COCC#C)=O)(C3)C2)ccc2c(c1)C=CCC2 c1(C(=O)NC(CN(C(=O)CCOC)CC)C)nsnc1O CC(=Cn1ccnn1)C(=O)NC1CCC1CNC(=O)CCCc1ccc(C)s1 CC1CC(NC(c2cnc(O)c(Cl)c2)=O)CN(C(c2ccco2)=O)C1 C1(NC(CCn2ncc(C)c2)=O)CCN(C(=O)COc2cc(C)on2)CC(C)(C)C1 C(CC(=O)N1CCOCCC1C)(C(F)F)NC(CCSCCCC)=O C1(C(=O)NCC2CN(C(=O)CC(F)F)CC23CC3)(OC)CCS(=O)(=O)C1 CC(CNC(c1ccc(F)nc1)=O)C(F)C(=O)N1CC(C)(O)CO1 C1(C(C)NC(C(CC(=C)C)OC)=O)CCN(C(=O)CCOCC)CC1(F)F C1(CN(C(C2(C)C(C)C2)=O)C)CCCN(C(=O)C(C)(C)CC2CCC2)C1 N1(C(c2c(C)cc(C)s2)=O)CCC2CN(C(c3ncc(F)cc3F)=O)CCC2C1 c1(C(=O)NC2C(CNC(=O)CCC(F)(F)F)COC2)cccn2cnnc12 N1(C(C2CC(C)NC(=O)C2)=O)CCC2(CCC(NC(=O)C3=NOC(C)(C)C3)C2)C1 CC1(C(=O)NCCC2CCN(C(=O)Cc3cn[nH]c3)C2)CC=CCC1 N1(C(CCCNS(C)(=O)=O)=O)C2CCC1CC(NC(C1CC(=O)N(C)C(=O)N1)=O)C2 C1(C(=O)OC)CCC(C(=O)NC2CCCCC2NC(C2CC(OC)C2)=O)CC1 N(C1CCc2cccnc21)C(C1C(C)(C)CCN(C(=O)Cc2ccco2)C1)=O C1(C(N(C(C)CN(C)C(c2cn(C(C)(C)C)nn2)=O)C)=O)COCCN1C c1(C(N(C2CCCN(C(C3(C)CC4CCC3C4)=O)CC2)C)=O)ccc(F)cc1Cl C=CCC(CC(C)C)C(=O)N1CC2(CCC(NC(=O)C(O)C(F)F)CC2)C1 C(=O)(C#CC(C)(C)C)N(C)CCOCCC(N1CCCCC1CCN(C)C)=O C12(NCCN(C(C(=O)NCC(C)S(C)(=O)=O)=O)C)CC3CC(C1)CC(O)(C3)C2 c1(C(COCC(=O)NC2C(NC(C3(C#N)CC3)=O)C2)=O)ccccc1 CC1COc2ccc(CCN=C(NCC3C4COCC34)NCC3CCC3)cc21 CCC(O)C(F)(F)C(=O)N1CCCC(C(C)C(=O)N(C)CCC2CCC2)C1 c1(C(=O)NC(C)CCNC(C2(C(F)F)CCC2)=O)cc2c(Br)coc2cn1 CC1CCCC(C(=O)NC2CC(CNC(C3(CC(F)F)CCC3)=O)C2)CC1 N1(CCC(=O)N(C(C)C)CCNC(=O)CC2CC(=O)C2)CCCCC1C CCC(C)(O)C(=O)N1CCC(NC(=O)COc2ccc(O)cc2)C1 C=CCCC(C1CC1)NC(=O)COC1CC(CNC(=O)CC2CC(=C)C2)C1 c12ccc(cc1)C(=O)N1CC(C1)CNC2=O.C1(NC(C)=O)OCCC1C C1(CC=C)(NC(=O)CC(O)CC)CCN(C(c2nc(C)oc2C(F)(F)F)=O)C1 N1(C(C(C)c2ccco2)=O)CCC(O)(CCNC(c2occc2C2CC2)=O)C1 c1(C(N(CCC(C)N(C)C)CC)=O)ccc(-n2cnc(C(N)=O)n2)nc1.C c1(CC)cc(OC)ccc1C(=O)NCC1COCCN1C(=O)Cc1ccnn1C n1(C(C)C)ncc(C(=O)NCC(C(C)C)NC(C2(C)CC=CCC2)=O)c1Br c1(C(NC(=NC)NC(C)C)C2CC2)ncc(CNC(C)=O)s1 C#CCC(CC(=O)NCCc1scnc1C)NC(=O)C(C)(C)COC Cc1ccc(C(=O)NC(=O)C(C)NCc2ccnn2-c2cccnc2)cc1 N1(C(C(C)OCC)=O)CCN(C(=O)C(C(C)C)n2cncn2)CC(O)C1 C12(C(=O)OCCC3CC3)CC(CC1C(c1ccc(F)cc1)=O)C2 Cc1cc(CNC(C2(C)CCN(C(=O)CCC(C)(F)F)C2)=O)cnc1F c1(C(N2C(CC(=O)NC(CC)C(=O)OC)CCC2)=O)ccc(C(=O)C(F)(F)F)cc1 N1(C(c2c(C)cno2)=O)CC2CC(NC(c3cnn(C)c3C(F)(F)F)=O)CC1C2 C1(C)(C(=O)NCCN(C(C2(COC)CC2)=O)C)COCCO1 c1(CNC(=NC)NCc2ccc(N3CCN(C)CC3)cc2)ccccc1C(C)C c1(OC)cc(C(N2CCC(C(C)C(=O)NC3CCC(=O)NC3)CC2)=O)ncn1 C1(C(N2CC(CC(=O)OC)NCC2)=O)CN(C(C)=O)C2(CCOC2)C1 Cc1cc(C(=O)NC2CCC(C)N(C(=O)CCOC3CCCC3)C2)c(N)c(Cl)c1 N1(C(C(CCC)NC(c2cn(CC3CC3)nn2)=O)=O)CC2CC2(CC2CC2)C1 c1(C(=O)NC(C(C)NC(C=CC(C)C)=O)(C)C)ccc(C#N)n1C CCCCCC(C)CC(=O)N1CCC(CO)(NC(=O)CCc2cc[nH]n2)C1 N1(C(C(C)OCC(F)(F)F)=O)CCOC(CCNC(=O)C(=O)NN2CCCC2)C1 c1(N2CC(COC)OCC2)cc(Br)ccc1S(=O)(=O)N1CC2CCC1C2 c1(OC(C)C(=O)NCC23CC(CN2C(c2ccoc2)=O)C3)ccc(Cl)cc1 N1(C(C)=O)CCOC(C(N2CCCC2C2(NC(C3CC=CCO3)=O)CC2)=O)C1 N1(C(C2C(C)OCCO2)=O)CCC(C(=O)NCCCC2(C)CC2)CC1C N1(C(c2cc(Cl)n[nH]2)=O)CC2CCN(C(=O)CCC3CC3(F)F)C2C1 Cc1cc(NC(=O)CC(CNC(C2(Cl)CCCCC2)=O)C2CCC2)cc(C)c1F Cc1nc(C(N2CC(CC(=O)NC34CC(C3)C4)C(C)C2)=O)cn1C C=CCN=C(NCc1ccoc1C)NCc1ccsc1C(=O)OC(C)(C)C C1(NC(=O)CCc2ccsc2)(CO)CCCN(C(=O)C(O)C(F)(F)F)C1 c1(C(=O)NC(C)CNC(c2cc(-c3ccncc3)no2)=O)nnn(C)c1Br Cc1ccc(C(=O)N(C)CC2CN(c3ncnc(C(C)(C)C)n3)C2)cc1 c1(C(N2CCC3(CN(C(CCNS(C)(=O)=O)=O)C3)C2)=O)cccc2nc(O)[nH]c12 O=C(C1=C(Cl)CCOC1)NCCC(Cc1ccccc1)NC(=O)Cc1cnc[nH]1 c1(C(NNCc2cc(C(=O)OC)cc(Br)c2)=O)nn(C)c2c1CCCC2 c1(NC(=O)NC2CC(CS(C)(=O)=O)C2)nc(Cl)cs1 C1(CC(C)N(C(CO)=O)C)CN(CC)C1.C1(=O)COCCN1.OC Cc1occ(C(F)(F)F)c1CC(=O)NC1COCCC1NC(=O)C(C)C(F)F C(N=c1[nH]c(=NCc2cncnc2)c2[nH]ccc2[nH]1)C1(C)C=CCCC1 CC(C)(CCCC#N)C(=O)NCC1CCCN(C(=O)CC(F)(F)C(F)F)C1 C(C)(CCCCNC(c1ccc(C(C)(C)C)cn1)=O)NC(CCN(C)CC)=O C(CC(O)CC(=O)N1CCOC(CCNC(=O)Cn2nnc(C)n2)C1)SC Cc1cc(N(C)C(c2cc(CN(C)C)n(C)n2)=O)nc(=NCCCCN(C)C)[nH]1 C1(CNC(=O)COCC2CCC2)CC12CCN(C(C1CC(=O)N(O)C1)=O)CC2 c1(CC(=O)NC2CN(C(c3ccc(F)cn3)=O)CC23CC3)cc(Br)ncc1Br C(C)(C(CC(=O)NCC(C1CC1)C1CC1)NC(c1c[n+]([O-])c(C)cn1)=O)OC C1(CCSC(C)C)CN(C(C23CC(n4cc(CCN(C)C)nn4)C2C3)=O)CCO1 C12(CC)CCCN(C1)CC(=O)N2C.c1(NC)cccc(C#N)c1 N1(C(C(C)(C)C#N)=O)CC2CCC(NC(=O)CC3(O)CCOC3)CC2C1 N1(C(CC(CC)C)=O)CCC(C(N2CCC(NC(=O)NC)CC2)=O)C(C)(C)C1 c1(NC(C2(F)CCN(Cc3ccsc3Br)C2)=O)ccc(F)c(CO)c1 C=CCC(CC=C)C(=O)NCC1CCN(C(C2CCC2(C)C)=O)CC1C NC(=O)CCCCC(=O)N1CC(CNC(=O)CCC2CC2)OC(C(F)(F)F)C1 C1(CNC(=O)Cn2ncccc2=O)CCN(C(=O)CC2CCC(=O)O2)CC1(F)F C(C(=O)NCc1ncoc1C1CN(C(c2ccc(C)nc2)=O)C1)(C(C)(C)C)SC Cc1ncccc1CC(=O)NCCC(O)CNC(=O)Cc1ccns1 CC1CC2(C1)CC(N=C1N=C(C3=C(CSC)N3)N1CCC1CC(C)=NN=CSC(C)CC1)C2 N1(C(CC(=O)NCC#C)=O)C2CCC(C(=O)NCC3(O)CC3)C1CC2 N1(C(C(CC)=CCCC)=O)CCC(F)(CN(C(=O)CC2CCC(=O)NC2)CC)CC1 Cc1cc(-c2ccc(CN3CCC(C(=O)O)CC3C)cc2F)cc(C)c1 C#CC1(C(=O)NC2CCCC2NC(=O)CCc2ccc(Cl)nc2)CCOCC1 CS(=O)c1cccc(NC(c2ccccc2I)=O)c1 S(=O)(=O)(c1cccnc1NCCS(C)=O)NC(c1c(C)nc(Cl)cc1)C c1(C(=O)NCC23CC(CNC(C(C(C)C)C)=O)(OC2)C3)occ2c1CCC2 Nc1cc(C(=O)NCC(CO)NC(=O)C(F)=CC2CC2)ccc1Br c1(C(N2CCC(NC(C(C)Cc3cnc[nH]3)=O)CC2)=O)cc(C#N)ccn1 c1(OC)cc(F)c(CC(N2CCC3CCC23CNC(=O)C(C)(F)F)=O)cc1OC C1(CN2CC(C(C3CCN(C(=O)CC4=CCCC4)CC3)=O)C2)CC12CCSCC2 C1(NC(C(CCSC)(C)C)=O)CCN(C(=O)C(C)(C)c2ccc(Cl)s2)CC(O)C1 c1(OC)cc(NC(=O)OC(C)(C)CC2CCOC2)ccc1F C12(C(=O)NCCNC(c3cc4n(c3)CCOC4)=O)CCCCC1CC(F)(F)C2 CCC(CNC(c1cc(CO)on1)=O)(CC)NC(=O)C(=O)NCCNC(C)=O c12nc(cc(N3CCCC(CCF)C3)n1)N2.n12cc(nn1)C2.C1(CSC)CC1 c1(C(N2CC(C)(C)C(NC(c3cn[nH]c3)=O)CC2)=O)ccc2c(c1)C(=O)CC2 CCCC(C)(CC)C(=O)N1CCN(CC(C)NC(c2cc(C3CC3)ns2)=O)CC1 CC1(C)CC(NC(C2C=CC(=O)N=N2)=O)CN1C(=O)CCOc1ccccc1Cl c1(C(=O)NCC(CNC(C(c2c(C)cncc2)C)=O)C)ccnc(Cl)c1O c1(C(=O)NC2CC(C)(CNC(C(CC)CC)=O)C2)ccc(C=NOC)cc1 Cc1oc2ccccc2c1CC(N1CCN(C2CCCC2O)CC1)=O Cc1nnc(CCC(=O)NCC2(F)CC(CNC(C3CCCC3C)=O)C2)n1C c1(C(=O)NC(C)CN(C(=O)CN2CCCC2C(N)=O)C)cnn2cccc2c1 N1(C(c2ccc(C)c(CO)c2)=O)CC2(C1)CN(C(=O)CC1CC1(Cl)Cl)CC2CO CCCC(C)(C(=O)OC)NC(c1ccncc1-n1cc(CN2CCOCC2)nn1)=O Cc1nc(C(=O)N(C)CCOCCN(C)C(C2(C#N)CC(=O)C2)=O)c(C)s1 C=CC1(C(=O)NCC(C)OC)CCN(C(=O)CCOc2cccc(C)c2C)CC1 c1(NC(C(CC)C)=O)ccc(SCC(C)C)c(Cl)c1.N12CCN(CC1)CC2=O c1(C(=O)NCC(COC)NC(c2cocn2)=O)cccc(N(C)C)c1 O=C1CCc2c(C(=O)OC(C(F)(F)CBr)c3ccccc3)cccc2N1 CCCC(CC)CCC(=O)NCCC(CNC(c1ncn(C(C)C)n1)=O)OC(C)=O C#Cc1ccc(CCC(=O)NC2(CNC(c3ccc(Br)c(F)c3)=O)CC2)cc1 C1(NC(C=CCOC)=O)CCC(C)(CNC(=O)CCCc2csc(=N)[nH]2)C1 C(=O)(CC(O)C(C)CC)NC1CC(NC(c2cc(CCC)nc(O)c2)=O)C1 c1(CC)ccc(C(N2CC(NC(=O)COC3(C)CCCC3)CCC2C)=O)cc1F C1(C(=O)NCCc2cn(-c3nccc(C)n3)nn2)CCc2ccccc2CC1 CC(C)C(C(=O)N1CC(C(O)C(=O)N(CC(C)(C)C#N)C)C1)C1CCC1 C1(CN(C)C(=O)NCCC2CCN(C(=O)C3CC3)CC2)CCCC(O)C1 C=CCCC(CC(C)C)C(=O)N1C(CNC(c2coc(Br)c2)=O)CC2COCC12 C1(CN(C(=O)C=C2CCOCC2)C)CCN(C(=O)COC2CCCOC2)CC1 C1(CNC(=O)COCC(F)F)C(CNC(c2cncnc2)=O)C1(F)F C#CC1(O)CCCN(C(C23CC(C)(CN2C(c2c(O)cccc2F)=O)C3)=O)C1 C1(NC(c2cc(CC)n(C)n2)=O)CN(C(c2ccn(CC)n2)=O)C2CCCCC12 c1(C(=O)NCC2C=CCN2C(c2cocn2)=O)ccc(OC(F)(F)F)cc1Cl N1(C(c2c(C)c[nH]n2)=O)CCC2(NC(c3[nH]nc([N+](=O)[O-])c3Cl)=O)CCCC12 C(CCCC(c1nnnn1C1CCCCCC1)NC(C)(C)CCF)(OC)OC O=C(C1=CC2CCC(C1)C2)NCc1cc[nH]c1C(=O)NCC1CCC(O)CC1 C1(C)CCCN(C(=O)C(=O)N(c2ccco2)NCCOC)C1.N(C)C N(C(=NCCN(C)CCO)N1CC2C(NC(S(C)(=O)=O)=O)C2C1)C(C)C N1(C(C(C=C)(C)CC)=O)CC2CCN(C(=O)CSc3n[nH]c(O)n3)CC2C1 CN1CCN(C(c2[nH]ccc2CNC(=O)CN(CC(C)(C)C)C2CC2)=O)CC1 N1(C(C(C)C(C)(F)F)=O)CCC2(CCN(C(=O)CCC(=O)N(C)C)CC2)C1 C1(N(C(c2ccc(C)s2)=O)C)CN(C(c2sccc2NS(C)(=O)=O)=O)CCC1CO C1(C(=O)NC2CN(C(=O)C(F)CC3CCOC3)C2)OCC2CCCC1C2 c1(C(=O)NCC2(C)OCCN(C(CC3(C)CCCC3)=O)C2)onc2ccccc12 C(C(C)(F)CNC(c1ccc(Br)s1)=O)NC(C=CCN(C)CC)=O n1(CC(N2CCCCC(NC(C(C)(C)C3CC3)=O)C2)=O)cnc2c(N)ncnc12 C1(NC(C(C)(C)c2cnsc2)=O)C(C)(C)C(NC(C2CCCOCC2)=O)C1(C)C N1(C(C(C)CC2CC2)=O)CCC(N(C(=O)CCOCC2CCC2)C)CC1 C1(CC=C)(NC(=O)Cn2cncn2)CCN(C(c2cncnc2CC)=O)C1 CCC(C)(CNC(=O)C=CCOC)C(=O)N(C1CCCCC1C)C N1(C(CC2C(C)C2)=O)CCC(C)C(NC(=O)CCC2(C)N=N2)C1 N1(C(CCC(=O)NCCC)=O)CC2(CCN(C(=O)C(O)CC)CC2)CC1C C1(NC(CS(=O)(=O)NC)=O)CCCC12CN(C(=O)C=C(C)C(F)F)C2 N1(C(Cn2c(C(C)C)ncc2)=O)CCC2(NC(=O)CCN3CCC3)CCCC12 c1(N(CCCOCC2CC2)C)ccc(S(=O)(=O)NCC2(Cl)CC2(F)F)cc1Br N1(C(CC(=O)NCC)=O)CCC(CO)C1(C)C.c12ocnc1CCNC2=O C1(C)(CNC(C(C)NC(C)=O)=O)CCCN(C(=O)CCS(N)(=O)=O)C1 C1(COC)(CNC(=O)OCCC#N)CC1C(F)(F)F CCC(CC)C(F)C(=O)NC(CN(C)C)C(=O)NCCn1ccc(=O)cc1 C1(C(NNC(=O)c2n[nH]c(=N)s2)=O)Nc2ccccc2NC1=O Cc1ccccc1CC(=O)NCCC(C)NC(=O)C(=O)NCC1CC1 C1(CNC(C2C(C)(C(C)C)C2)=O)CCCCN1C(=O)CCC1CC1(F)F C1(N(C(C(C)(COCc2ccccc2)OC)=O)C)CCCCCCC1 N1(C(C(C)OCC=C)=O)CC(C(=O)NCC2OC(=O)CC2(C)C)CC(C)C1 N1(C(c2sccc2CO)=O)CCC(OCC(=O)N(C2CC2)C2CC2)C1 C1(CNC(c2c(CC)scc2)=O)CN(C(=O)C(=O)NC)CCO1 CCS(=O)CC(=O)N1CCC(C)C1CNC(=O)Cn1cc[n+](C)c1 c1(NC(C(=O)NCC2CCC(C3CC3)O2)=O)ccc(S(=O)(=O)CC2CC2)cc1 C=CCCC(O)CN(C(=O)C(C)(C)CNC(C1CCC(=O)O1)=O)C Cc1ccc(-c2ncccc2C(N2CCOC(CCO)C2)=O)cc1COC(F)F C=C=C(C)CC(=O)NCC1(O)CN(C(c2ccc(-c3ccccc3)nn2)=O)C1 N1(C(C(C)n2ccnc2)=O)CCCCC(CC(N2CC(O)C(O)C2)=O)C1 C=CC(CC)C(=O)NC1CCOC(CNC(=O)Cc2ccn(C(C)C)n2)C1 C(C(C)C(C)C(=O)N1CC2CC1(CNC(c1c(Cl)cnn1C)=O)C2)OC C(=O)(C1CCCc2cncn21)NC1(C2CCCN(C(C3CC(C)(O)C3)=O)C2)CC1 C(=O)(C(CCC(C)NC(C)CC(c1nnnn1C1COC1)OC)C(=O)OC)OC Cc1cc(F)ccc1NC(C1(C)CCN(C(C2CC2C(C)C)=O)CC1)=O N1(C(c2cnc(N(C)C)s2)=O)CC(O)CC1CNC(C1CC2C=CC1C2)=O Cc1cnn(C)c1CC(=O)NCCCN(C(=O)CCS(C)=O)C1CCCC1 c1(C(=O)NCCCO)ccc(SCC(=C)CCNC(=O)CCc2cncs2)cc1 C1(C(N2C(C(C)(C)NC(c3cc(F)c[nH]3)=O)CCC2)=O)CCCCS1(=O)=O C1(C(C)C)CN(C(=O)CONC(=O)C(C)OC(C)(C)C)CC(=O)N1 c1(C(=O)NC2C(OC)CN(C(C34CC(C3)C4)=O)C2)cnc2n1CCC(C)C2 c1(CN2C(CC(=O)NC(COCC)C3CC3)CCC2)ccc(F)c(C(F)(F)F)c1 C1(C(F)(F)F)(NC(=O)NCC(c2ccnc(Cl)c2)(F)F)CCc2ccccc21 c1(OC)ccc(C(N2CC(CNC(=O)CCc3ncc(C(F)(F)F)[nH]3)C2)=O)cc1 N1(C(Cc2nn(C)c(Cl)c2)=O)CCN(C(C2(C)COCCO2)=O)CC1C1CC1 N1(C(C=C(C)C(C)(C)C)=O)C(C(N2CCSCC2CN(C)C)=O)CCC1C1CC1 C1(CCCOC)CON(C(=O)c2cnc(N(C)C)s2)C1 c1(OCC)cccc(CC(=O)NC)c1.c12ccn(n1)C2.C1(C(=O)NC2CC2)CCC1.C c1(C(=O)NCC2(C(=O)NC3CCCC3C(=O)NC)CC(=C)C2)cc(C)c(C)[nH]1 c1(SC)cc(C(=O)NC2CC(NC(=O)Cc3ccn(C)n3)C2)cc(Cl)c1 CC(C)(F)CCC(=O)N1CCC(CO)(CNC(c2cccnc2)=O)C1 N1(C(C(=O)NC(C)Cc2ncon2)=O)CCC(OC)C(F)C1 C(c1cnn(C)c1)=C(C)C(=O)NCC=CCNC(C1CC12CCOC2)=O N1(C(C(c2cccs2)NC(COCCCOC)=O)=O)CCOC2CC12 N1(C(c2cc(Br)cc(C)c2F)=O)CCC2CCCC(C1)N2 N1(C(C2CN(C)C2)=O)C2CCC1CC(N(C)C(c1ccc(O)cc1)=O)C2 C(=O)(C(C)CC(=O)NC(CCOC)C(=O)NC(C)CC(=O)N1CCOCC1)OC C(CCCCC(=O)NC1CN(C(=O)CC=CC(C)(C)C)CC1C(F)F)SC C(=O)(C(CNC(C1C2CC(=O)CC12)=O)CC(C)C)NCCc1ncc(C)o1 C(=O)(CS(=O)(=O)c1ncc[nH]1)N1C(C)C(O)CCC1.c12cccc(c1)OC2 C1(C)(C(=O)NC2(CNC(c3nc(C)sc3)=O)CCCCC2)CCCCCC1 C(=O)(C1=CCCC1C)NC(CCCCNC(CCc1ccnc(C)n1)=O)C Cc1cnc(F)cc1CNC1CC(F)(CNc2cc(=O)n(C)cn2)C1 c1(CC(C(N2CC(F)(CC=C)C2)=O)F)ccc(C(=O)OCC)cc1 N1(C(CNC(C(CC)C)=O)=O)CC2CC1C2NC(C1(CC)CC1)=O n1(CC(=O)N(CCCN(C(=O)CN2C(=O)CCC2=O)C)C)cnc2ccccc12 Cc1cccc(C=CC(=O)NC(CC(=O)NCC(C)CN(C)C)C(F)F)c1 Cc1cc(C(N2CC(=C(F)CNC(=O)CN(S(C)(=O)=O)C)C2)=O)nn1C(C)C CN1CCN(C(C2C3CCCCC23)=O)C(CNC(c2cnn(C)c2Cl)=O)C1 c1(NC(C2CC3CC3N2Cc2cc(Br)c(Br)s2)=O)c[nH]c2cnccc12 c1(SCCC)nc2ccc(-c3cn(CCc4ccccc4)nc3C)cc2o1 c1(CC)ccc(CNC(=O)NCC2(O)CCCC2(C)C)c(OC)c1 c1(C(=O)NCCC(C)NC(c2ccc(=O)oc2)=O)occ2c1CCOC2 N1(C(C(C)c2cc[nH]n2)=O)CCC(C)(C)C(NC(=O)Cn2nc(O)ccc2=O)C1 C1(C(N2CCN(C(C#C)C)CC2)=O)CCN(C(c2occc2C)=O)C(C)C1 C#Cc1cnc(C(=O)NCCC2(C(=O)NC3CCCC(CC)C3)CCC2)c(C)c1 N1(C(c2cc(OC)c(F)c(F)c2)=O)CC2CN(S(=O)(=O)c3cnccn3)CC2C1 C1(N(C)C(C2CCCN(C(=O)C(=O)NCC(F)(F)F)C2)=O)CCOC(C)(C)C1 Cc1nccc(C(=O)NCC(c2ccccc2)NC(C2(C)CC2C)=O)n1 c1(C(=O)NCCC2(O)CN(C(C(C)OC)=O)C2)cc(C(N)=O)cn1C C(C(C)(C(=O)N(C)CC1CCOCC1)NC(=O)C(O)C1CCC1)SC C(=O)(C1=NOC(C)C1C)N1CC(C(=O)NC(CC#C)(C)C)C(CCC)C1 N1(CCNC(c2coc(C(F)F)c2)=O)CCCN(C(C2CC2C2CC2)=O)CC1 C(C1=CCN(C(=O)C(O)CCC)CC1)NC(C1CCN(S(C)(=O)=O)C1)=O N1(C(C(COCC)C)=O)CCC(C(=O)NCC2=CCCCC2)CC1(C)C N1(C(C2CCOCC2)C(=O)NCCCOC)Cc2cccc(F)c2C1 C1(C(=O)NC2(C(=O)NC(C)C)CC2)CC2(C1)CC(F)(F)C2.C1C2CC1N(C=O)C2 c1(NCCN(C(C(=O)NCC)C2CCSC2)C2CC2)cccc(Cl)c1 N1(CCC(=O)NC(C2CCCCC2)C(=O)NCc2ccncn2)CSCC1=O C1(C)(CNC(CCC(=C)Cl)=O)CN(C(C2CCCN2CCCC)=O)C(C)(C)C1 C1(NC(C2(C)CC3(CC3)C2)=O)CN(C(=O)CC2(C)CCC2)C2(CCOCC2)C1 N1(C(c2c(CC)nccn2)=O)CCN(C(c2cncn2C(C)C)=O)CC1C c1(C(N(CCN(C(C(F)=C(C)C)=O)C(C)C)C)=O)ccc(O)c(Cl)c1 C1(N(C(COC(CC)C)=O)C)CCCN(C(c2cnc(Br)s2)=O)C1 c1(CNC(=O)CN2CCCCC2)cnc2[nH]ncc2c1.C123CCC1CCN2C3=O N1(C(c2ncsc2C)C(=O)NCC(=C)C)CCC2(CC1)CC2C(=O)OCC CC1(C)CN(C(=O)Cc2ccc(N)cc2)CC1NC(c1c(F)cccc1Cl)=O N1(C(CC2CC(OC)C2(C)C)=O)CC2CCC1CN2C(=O)CC1CCCCCC1 C1(O)(C(CNC(c2c(SCC)cncc2)=O)C)CCN(C(=O)C(F)OC)CC1 N1(C(C(C)=C2CCC2)=O)CCC2(CCN(C(c3ncccc3N)=O)CC2)C1 C(CS(=O)(=O)C1CCCCC1)NC(c1n(CCSC)nnn1)c1cnc(SC)[nH]1 C1(N(CC(C)(C)O)C(=O)NC(C)C(F)(F)F)COC(C)(C)C1 N1(C(CC=CCC)=O)CCC2(CC1)CCN(C(c1ccnn1C(C)C)=O)CC2C N1(C(COCCC=C)=O)CCCCCC(NC(=O)C(C)Cc2ccccc2Cl)C1 C1(C)(CNCc2c(C(c3nnnn3C)C)con2)CCCN(CCO)C1 Cc1ccc(NC(C2CC2C2CN(C(C3CCCCC3)=O)C2)=O)cc1C#N C1(NC(c2cc(CF)on2)=O)CC2CCC1C1CN(C(=O)C=C(Cl)Cl)CC21 CCCC(CC1CCCC1)C(=O)N1CCC(CO)(NC(=O)Cc2ccoc2)CC1 CCC(C)CCC(=O)NC1(C)CCCCC1C(=O)NC(CN(C)C)CCO N1(C(C(C)SCCCC)=O)CCC2(CC1)CC2N(c1cc(C)nc(CO)n1)C S(=O)(=O)(c1ccc(N2CCCC(N(C)C3CC3)C2)c(F)c1)N(CCOC)C Cc1ccc(C(=O)N(CC(O)CN(C(=O)CCC2CCCCO2)C)C)cc1CO C1(CNC(CCC)=O)CC(O)CN1C(=O)NCCCC1CCCCO1 N1(C(CN(C(=O)OCC)C)=O)CC2CC1C2C(N1CC(N2CCC2)C1)=O C1(C(C(C)C)NC(c2nocc2Cl)=O)CCN(C(C2C(C#N)C2(C)C)=O)CC1 c1(C(=O)NC2CC(F)(CNC(C3C(C)(C(C)C)C3)=O)C2)ccc2oc(O)nc2n1 Cc1nnn(C)c1C(=O)NC(c1ccccc1)CNC(C1CCC(F)CC1)=O CC(C)C(C(C)NC(=O)Cc1cnsc1)NC(=O)CCc1cncc(F)c1 CC(C)(C(=O)C(=O)CC)C1CCOC1.c1(C(=O)NCCCN)n[nH]cc1Cl N1(C(C2CC(C)C2)=O)CC2(CC2)CC1CNC(c1ncc(C(F)(F)F)s1)=O Cn1nc(C(=O)NC2CC(NC(=O)CCc3ccoc3)C(O)C2)cc1C(F)(F)F N1(C(c2c(CNC(C3ON=C(CC)C3)=O)cc[nH]2)=O)CCC2(CC(CO)C2)C1 CN1CCOC(C(=O)NCC2CN(C(C3CC34CCSCC4)=O)C2)C1=O Cc1nn(CCCC(=O)NC(C)(CNC(=O)C(C)n2ccnc2)C(C)C)c(=O)o1 C1(C)(C(=O)NCc2cc(C(N3CC(C(C)OC)C3)=O)n(C)n2)CCC(=O)NC1 C(=O)(CC(C)CC(C)C)NCC(C1N(C(COC(C)=O)=O)CCC1)(C)C c1(C(=O)NCC(CO)NC(c2c(C)[nH]nc2C(C)C)=O)cnc2[nH]cnc2c1 C(c1ccc(F)cc1F)=CC(=O)NCC(CNC(c1cnc(C)nc1C)=O)(C)O N1(C(C2C(O)CCN(C(c3ncc(Br)nn3)=O)C2)=O)CCOc2ccccc2C1 CC(CN(C)C)CCC(=O)N1C2CCC1C(CNC(c1cc([N+](=O)[O-])n[nH]1)=O)C2 c1(N2CC(NC(c3cc(C(C)C)[nH]n3)=O)CC3(C2)CC3)nc2cc(Br)ccc2o1 Cc1c(Cl)cnc(N2CC(c3cc(O)no3)C2)c1C#N O=C(C1=C(Cl)CCCC1)NC1CCC(NC(c2cnn(CCF)c2)=O)CC1 CC1CN(C(c2cncc(C(F)(F)F)c2)=O)CC1Nc1ccncn1 C1(=O)CC(C2CC2)C(=O)NCCC12CC2.C12(CCC1)C(=O)NC2.C(=O)NC.CO CC1(C(=O)NCC2CCN(C(=O)CC3CCC(=O)C3)CC2O)CCCC1(F)F c1(C(N2CC3C(CNC(C(C4CCC4)OC)=O)C3C2)=O)cncc2ncn(C)c12 N1(C(C23CC(F)(C2)C3)=O)CC2(C=C(C(=O)N3CC4C=CC3C4)CO2)C1 C1(NC(C(CCOC)NC(C2CC(O)C2)=O)=O)CC2CCC1CC2 c1cc2n(n1)CCO2.C12CN(CCO1)C(=O)C1CCC(CC1)OCC2.CC N1(C(CC2CCN(c3ccnc(OC)n3)CC2)=O)CCCC(C)S(=O)(=O)CC1 c1(CC)cc(C(=O)NCC2(CNC(C3CC3COC)=O)CC2)cs1 Cc1cn2cc(CC(=O)N(CC(O)CNC(C3(CSC)CCCO3)=O)C)nc2s1 c1(C(=O)NC(C)CC2CN(C(C3CCC3(C)C)=O)C2)ccc(F)c2cnccc12 CC(O)CCCCCC(=O)NC1CC2CCC1N2C(c1ccn(CCO)c(=O)c1)=O C(=O)(C1CCOc2ccc(Cl)cc21)NCC1(C)OCCN(c2cc(C)ncn2)C1 C1(C)(CNC(CCSCCC)=O)CN(C(c2ccc(C(=O)OC)o2)=O)C(C)(C)C1 CC(=Cn1ccnn1)C(=O)NC1C2CCN(C(C3(C#N)CC4(CC4)C3)=O)CCC12 C1(CNC(c2cnccn2)=O)CCN(C(c2ccc3cc[nH]c3c2)=O)CC1(F)F n1(CCCSCC)nnnc1C(c1cc(Cl)no1)NC(c1cnn(CC)c1)(C)C c1(C(C)NC(=O)C(C2CCCC2)NC(C2CC2F)=O)cccc(O)c1 N1(C(C2=CC(C)(C)C2)=O)CCCC2(CCN(C(C34CCCC(C)(C3)OC4)=O)C2)C1 C1(C(N2C(C)(C(=O)OC)CCC2)=O)C2CC(O)C(C2)N1C(c1ccc(C)cc1F)=O C(=O)(C(CCF)NC(=O)CC1C=CCC1)N(C1C(C)C1)C C(=O)(CC1OCCc2sccc21)N(CCOCc1ccnc(Br)c1)C C1(C(C(=O)NCC(C)N(CC(C)O)C)C)CCn2cncc2C1 c1(CC(=O)NCC(C)(CSc2ccccc2)OC)c(C)cccc1F C1(C(N2C(CN(C(=O)CCc3cc[nH]n3)CC)CCC2)=O)CC(=O)N(C)C1 S(=O)(=O)(c1cccnc1Cl)N1CCCCC(NC(c2n(C(C)C)ncc2)=O)C1 N1(C(c2n(CC)ncc2)=O)CC(NC(=O)CNC(=O)CNC(C)=O)C2(CCC2)C1 C(=O)(CCCC(C)(C)C#N)N1CC(O)(C(C)NC(CSCCC(C)C)=O)C1 N1(C(C(C)SC(C)C)=O)CCCC(F)(CNC(c2n[nH]c3c2COCC3)=O)CC1 C1(NC(CNC(=O)OCC=C)=O)CC(NC(=O)CS(C)(=O)=O)C12CCOCC2 N1(C(CCCCN(CCC=C)C)=O)CCOCC(C)(NC(=O)CCCOC(C)C)C1 C12(NC(c3c(CC)c[nH]c3)=O)COC(C1)C(NC(=O)CC1CC3(CC3)CO1)C2 c1(C(=O)NC(C(C)(C)NC(CC(COC)(C)O)=O)C)ccc(C(C)C)cc1F N1(Cc2c(OCC)cccn2)CCc2cc(CCO)ccc21 N1(C(COCP(C)(C)=O)=O)CCN(C(c2nccnc2N)=O)C2CCC12 C1(CC=C)(C(=O)NC(c2n[nH]c(C)n2)C)CCCN1C(=O)C(C)OC1CC1 c1(C(=O)NC(C(C)C)CCNC(C2CC(=O)N(CC3CC3)C2)=O)ccc(O)c(O)c1 C1(OC)CCN(C(C2CC(N(C(=O)CCc3ccco3)CC3CC3)C2)=O)C1 CC(C)C(CC(=O)N=c1ccn(CCO)[nH]1)NC(C1CC(C)C1)=O CCCN=c1nc(NCC(C)(C)C2=CCCCC2)c2c([nH]1)c(C)nn2C C1(CCNC(CC=CCC)=O)CCCN(C(=O)CC2=CCCC2)CC1 CC1(C(N2CC(C)(OCC(=O)NC3CCNC(=O)CC3)C2)=O)CCC(=O)NC1 C12(C3CC3)CN(C1)C2=O.C1(CC(=O)OC)CCCCC1NC(=O)COCCN(C)C C1(c2cn(CCN(C(=O)CC(C)(F)F)CC)nn2)CCS(=O)(=O)C1 C(=O)(C(C(C)C)N(C)Cc1ccc(OC)cc1)NCCC.C(C)(CC)SC C1(=O)C(F)C(C)CN1.C(=O)(C(C)(C)NC(=O)C=CCCC(C)C)OCC c1(SC)ccc(C(=O)NC2COCC2NC(C2CN(c3nnnn3C)C2)=O)s1 N12C(CCC13CCC3)C2=O.c1(CC(OC)OC)cn(CCCC(=O)O)nn1 N1(C(C2(CC)CN(C(=O)CCn3ccnn3)C2)=O)CCC(COC)(COC)C1 N1(C(C(F)=CC)=O)CCC2C(C1)CN2C(c1cc(OC)ccc1C)=O C(=O)(C(C#N)C(C)(C)C)NCCN(CCC)C(c1cnc2[nH]cncc1-2)=O C(=O)(CC1=CCOCC1)NCCC(CNC(c1nn(CC)nc1C)=O)OC c1(NC)ccc(C)cc1C(N1CC(O)(CN(C(=O)C(C)(C)CO)C)C1)=O C1(C(C)C)C(C(=O)N(CCCCN(C)C)C)CCN1C(=O)CC1CCCC2CC12 C1(C(=O)OC)CCC2(CCN(S(=O)(=O)c3ccccc3)C2)C1 CCCS(=O)(=O)C(C)C(=O)N1CC2CN(C(C3(C)CC3)=O)CC2(C)C1 CCC(C(=O)N1CCC(CNC(C2CN(CC(F)(F)F)C2)=O)C1)OCC C1(C(N2CC(C)(NC(=O)Cc3ccon3)C2)=O)CCC2CC1CO2 N1(C(c2cccc(C#C)c2)=O)CCC2CCN(C(=O)C=C(C)C#N)CC2C1 n1(CC=C)cc(C(=O)NCC2CCCN2C(=O)C(C)SC)c2ccccc12 C(=O)(C(C)(C)C(O)C(C)C)NCC1OCC(C(=O)NCC(COC)(C)C)C1 C(c1cccc(Cl)c1)=CC(=O)NCC(CC)(CC)NC(=O)C(F)CC1CCOC1 C(=O)(CC1=CCCCC1)N(CC(C)NC(=O)Cc1cc(C)ccc1OC)CC Cc1ccc2cc(CN3CCC(O)CC3C(N3CCC(CO)C(O)C3)=O)sc2c1 N1(C(C=COCC)=O)CCC(O)(CN(C(=O)C(O)C(C)C)Cc2ccccc2)CC1 Cc1ccc(CS(N2CC(C)(F)C2)(=O)=O)c(F)c1 O=C(CCN=C(NCCC1CCOCC1)NC1CCOC1)N1CCCC1 c1(C(=O)NCC2(C(F)F)CCN(C(c3n(C)ccc3)=O)C2)cccc([N+](=O)[O-])c1 C(CC(=O)NCCCCN(C(=O)CCSC(F)(F)F)C)NC(=O)OC CC1CN(C(=O)CN(C)Cc2ccc(F)cc2)CCN1C(c1ccc(O)nn1)=O C(=O)(C1CNc2ccccc21)N(CCCN(C(CC(CC)C)=O)C)C c1(C(C(=O)NCCCN(C(CCNC(COC)=O)=O)CCO)O)cc(Cl)ccc1F C(=O)(CC1COCc2ccccc21)NCC(C)(C)NC(CC1CCN(C)C1)=O C=CCC(CO)CN=C(NC(C)CCC)NC1CCOCC1 CC1CC(CNC2CC2)CCN1C(C1CC(F)(F)C1)C(=O)Nc1ccccc1 CC(C)CC(O)C(=O)NCc1ncoc1C1CN(C(=O)CC(C)CF)C1 c1(C(=O)OC)cc(S(=O)(=O)NCC2CC3(C2)NC(=O)NC3=O)cc([N+](=O)[O-])c1C c1(C(=O)OCC)nc(C(=O)NC(C)(CNC(=O)CN(C)C=O)CC)cs1 C1(NC(c2ccoc2Br)=O)CCN(C(c2cnns2)=O)CC12CCC2 C(C(C)C(F)C(=O)NCc1ccns1)NC(c1c(C)nncc1)=O C1(C2(C(=O)NCC(CNC(=O)CCC3OCCO3)F)CC2)CCCCO1 C12(N(C)C(c3cscn3)=O)CC(CNC(C3CCCC(F)C3)=O)(C1)OC21CCC1 Cn1cc2cc(C(=O)NCc3cc([N+](=O)[O-])ccc3N3CCOCC3)ccc2n1 Cc1cncc(C(=O)NCC(F)CNC(=O)Cn2cc(CN(C)C)nn2)c1C c1(C(=O)NCCCCN(C)C(C2CC2(C)C)=O)nn(C)cc1Br Cc1ccn(CC(N2CCCC(C)C2CNC(C2(NC(N)=O)CC2)=O)=O)c(=O)c1 c1(OC)ncccc1S(=O)(=O)N1CCC(C(=O)Nc2c(C)cccc2Br)C(O)C1 c1(C(N2C(CNC(C3CCC(F)CC3)=O)C=CC2)=O)c(Br)nc2n1CCCC2 C1(NC(C(C(C)C)NC=O)=O)CN(C(c2ncnc(O)c2Cl)=O)CC1N=[N+]=[N-] c1(C(=O)NCC(C)CNC(=O)COC2CCOC2)cccc(Cl)c1OC(F)(F)F N1(C(CCn2ncc(C)c2)=O)CCC2(CCCCC2NC(C2CCC2)=O)C1 C(C(C)CC(=O)NCC(O)C1CC1)NC(C=CC(C)(C)SC)=O CC1CN(C(=O)C(=O)NC2CCN(S(C)(=O)=O)CC2)CCN1C(=O)C(C)C(F)F N1(C(C(CSC)(C)NC(=O)C(F)CC(C)(C)C)=O)CCC2CN(C)CCC12 c1(C(=O)NCCCC(C)(C)NC(C(C2CC2)OC)=O)ccc2nnn(O)c2c1 c1(CCC(=O)OC)nc(-c2cccs2)no1.N1(CCF)CC1 c1(CCOCCOC)cccc2c1OCC2CC(=O)N1CC(NC(=O)C=CCF)C1 C1(N(C(=O)COCC(F)F)CC)CCN(Cc2cn(CC3CCOC3)nn2)C1 c1(CN2CC3CN(C(c4c(C)cccc4Br)=O)CC32)ccc(Cl)c(Cl)c1O C1(C(N(C2(C)CC2)C)=O)CC(C)(C)CN1C(C1OCCC1(C)C)=O N1(C(=O)CCCc2cc(Cl)ccc2F)CC2C3CCC(C3)C12 C1(CNC(C23C(C(N)=O)(CCC2)C3)=O)CCCCN(C(C2CCC2(F)F)=O)C1 c1(C(N2CC(C(C)C)C2)=O)cncc(CNC(=O)Cc2cncnc2)c1 C1(NC(CC2(C=C)CC2)=O)CN(C(=O)CCc2cccc(OC)n2)CC1COC C12(NC(c3cc(CC4CC4)c[nH]3)=O)CCCC1CN(C(C1CC3CCC3C1)=O)C2 C(=O)(C(C)CCCOC)NCCN(C(CC1(C=C)CC1)=O)C1CC1 N1(C(C2C(CC)C2)=O)CCCC(C(N2CCCC(OC3(C#N)CCCC3)C2)=O)CC1 C1(C(N2CCC(C)(NC(C(CCCC)C)=O)CC2)=O)CCc2cn(C)nc2C1 C1(NC(CCCC=C)C)CON(C(=O)OC(C)(C)C)C1 C1(F)(C)CCC(CO)C1.C1(C)(C2(CCC=C)CC2)CS(=O)(=O)C1.C12CC1C(=O)NC2 c1(CC(=O)N(CC(C)N(C)C(c2cccc(CC#N)c2)=O)C)ccc(F)c(Cl)c1 CC(N=c1nc(N(C)CCN(C)C)c2c([nH]1)COC2)c1ccoc1 N1(C(CCOCCOCC)=O)CCC(C)(NC(c2ccn(CCF)n2)=O)CC1 C1(N(CC(=O)OCC)C)CC1(F)F Cc1cc(F)c(F)cc1NC(=O)CC1CCCN1C(c1cncc(O)c1)=O C1(C(N2CC(CNC(C3CCN(C)CC3)=O)C2)=O)CCCC12CCC2 c1(C(C)C)nc(=NC2CN(C(c3cc(F)ccc3Cl)=O)CC2C)s[nH]1 CN1CCN(C(=O)CCOC2COC2)CC1CNC(C1(C2CCOCC2)CC1)=O N1(C(CCOCC)=O)CCC2(CC2C(=O)NCc2nccs2)C1 C12(CNC(C3(CCS(N)(=O)=O)CC3)=O)CCC(NC(C3CC=CCO3)=O)(CO1)C2 C1(C)(NC(C2C(=C)C2)=O)CCN(C(c2oc(SC)cc2C)=O)CC1 N1(N(CCOCc2cccs2)C)C(=O)CN(CCCC2CC2(Cl)Cl)C1=O c1(C(N2CCC(CC(N3CC4COCC4C3)=O)C2)=O)c(F)cc(I)cc1F Cc1cnc2n1CCC(NCC1(CCO)CN(n3cccn3)C1)C2 CCCC(C(=O)N1CCCC1C(C)NC(=O)CC1CC2CC2C1)OC C1(C(=O)NC(C#C)CCC)CC=CCN1C(=O)C(C1CC1)SC CC1=NOC(CC(=O)NC2CCN(C(=O)Cc3csc(Cl)c3)C2)C1 C1(C(=O)NC(C2=NNC(=O)C2)=O)CCC2CN(c3cc(C(F)F)ncn3)CCC2C1 C(CC(=O)N1Cc2ccccc2CO1)OC1(C)CCCN(C(=O)CCC2CC2)C1 c1(SC)ccc(C=CC(=O)NC2CCN(C(C3CCCN3C=O)=O)C2)cc1 Cn1ncc(CNC(C2C3CC4C(C3)C24)=O)c1C(=O)NCc1cncs1 Cc1cc(C(=O)NCC(C)(C(C)C)NC(=O)Cc2ccc(Cl)cc2Cl)nnc1C C1(C(F)F)(CNC(C(C)OCC#C)=O)CCN(C(c2cn(C3CC3)cn2)=O)C1 c1(CNC(=O)C(=O)OC)ccc(NCC2C(CCC)CCC2)c(Cl)c1 c1(C(=O)NCC2CCC(NC(CC(=O)NCC)=O)C2)cc(C)c(O)c([N+](=O)[O-])c1 c1(C(N(C(C)CCNC(=O)CSc2nc[nH]n2)C)=O)c(O)cc(Cl)cc1F Cn1c(C(N2CCCC2CNC(=O)CC2CCC(F)(F)CC2)=O)cc2sccc12 c1(N2CCCC(C)(OC)C2)[nH]c(=NCc2ccc(C)cc2Br)nc2sccc12 CCC(C)C(C(=O)NC12CC1CN(C(=O)C(C)(C)OCC(F)(F)F)C2)N(C)C c1(C(=O)NC2CCN(C(C3CCCC4CC34)=O)CC2F)cc2ncccc2[nH]1 C1(NC(C(CC)OCC)=O)CCN(C(=O)CSCc2ccccc2)CC1C(C)C C#CC12CC(CN1C(=O)C(CC(=C)Cl)NC(=O)C(C)OC(C)=O)C2 C1(CCC)CCCC1N(C)CCOCCOC.C(=O)(CSCCCl)N C(=O)(C(C)CC(=O)OC)NCC1(F)CCC(NC(CCC#CC)=O)C1 C1(NC(CC(CC)C)=O)CN(C(C2(OCC)CC2)=O)CC1(C)C.c1cccc(C)c1 c1(C(=O)NCC(CO)NC(C2(C)CC3CCC(C2)S3)=O)c[nH]c2c(Cl)cccc12 c1(C(N2CCN(C(=O)Cn3cccn3)C3CC23)=O)ccc(C(C)(C)C)c(O)c1 CC1CCCC=C1C(=O)NCC(C1(O)CN(C(c2ncsc2C(C)C)=O)C1)(C)C N1(C(c2c(C)cccc2)=O)CC(C2CCCCN(C(C3CCCS3)=O)C2)C1 N1(C(C2C=CCN2Cc2cc(-c3ccccc3)no2)=O)CCn2c(Br)nnc2C1 C1(C)(C)CC(=O)N1.c1(C(C(N2CC(CCCCOC(C)=O)C2)=O)C)cccc(F)c1 C(=O)(C(CNC(=O)Cc1cncnc1)CC1CCCC1)NC(c1ccncn1)C S(=O)(=O)(c1cnccc1N1CCCC(C#N)C1)NCC(C1CCCC1)OC Cc1ccc(NC(C2CCCN(C(c3ccc(F)cc3C)=O)C2)=O)c(CO)c1 C1(N(C(c2ccc(C(N)=O)s2)=O)CCF)CCCN(C(=O)Cc2sccc2Cl)C1 c1(C(C)NC(=O)COC2CN(C(C3CC(O)C3)=O)C2)ccc(O)cc1 CC1(C)CN(CCC2CCCNCC2)CC2(CN(C(=O)OC(C)(C)C)C2)O1 C1(C)(C(N(C(C)CNC(C2CCCN2C(C)=O)=O)CC)=O)CNC(=O)C1 Cc1cc(C(N2CCC(N(C(=O)C(c3cccnc3)C)C)C2)=O)n(C(F)F)n1 c1(OC)ccnc(C(=O)NCCCNC(c2coc(SC)c2)=O)c1N c1(C(N2C(CC(N3CC(N(CCC)C)C3)=O)COCC2)=O)ncc(C)cc1C N1(C(C(C2CCCC2)OC)=O)CCN(C(=O)C(C)OC(C)=O)CC1 C(=O)(C1=CCCC1(C)C)N1CCC(NC(c2cnc(OC)nc2)=O)C12CC2 CC(C)(C#N)CCC(=O)NC12CC(NC(=O)CCc3ccc(F)cc3Cl)(C1)C2 c1(C(=O)NC(C)(C)CNC(=O)C=CBr)ccc(C(F)(F)F)nn1 N1(C(CC2C(CC)C2)=O)CCOC(C(=O)NCCC2=CCOCC2)CC1 CC1(C)CCN(C(=O)C(O)c2cnco2)CC1CNC(C1(CCO)CC1)=O CCC(C)(CNC(C1CCN(C(C2CCC(F)CC2)=O)C1)=O)C(N)=O C1(C)(CNC(c2c(CC)cc[nH]2)=O)CCCN(C(c2cc(C)sc2C)=O)C1 N1(CCN(C)C(=O)O)CCOCC1.C1(N(C)CC)CCN1C(=O)C1CC1 c1(N(C(CCCC)=O)CC(CO)NC(=O)C(C)(O)CC)ccc2cccc(Cl)c2n1 C1(C)(N(C)C)CCN(C(C2(NC(=O)CC3CCCC4CC34)CC(F)C2)=O)C1 c1(C(=O)NCCN2CCC(O)(C(=O)NCC)CC2)sccc1S(=O)(=O)N1CCCC1 c1(C(=O)NC2COCCC2NC(=O)C(O)CC2CCCCC2)ccc(CO)nc1 C(CC(C(=O)NCC=CCNC(=O)Cn1nnc(=N)[nH]1)OC)OC n1(CC)cc(Cl)c(NC(N2CCCC2C(N2CCCC2)=O)=O)n1.c12cccc(c1)N2 C1(C(=O)NCC(CN(C)C(c2csc(C3CC3)n2)=O)O)Cc2cc(Cl)ccc2O1 N1(C(c2ccc(CCC)cc2)=O)CCN(C(=O)Cc2ccn(C)n2)C(COC)C1 C#Cc1cccc(OCC(N2CC(NC(c3cscc3SC)=O)C3(CC3)C2)=O)c1 c1(OC)cc(C(=O)NC(CNC(c2nc(C)oc2C)=O)CO)ccc1[N+](=O)[O-] C1(NC(C2(C)CC(=C)C2)=O)CC(C(=O)N2CCSC(C)C2C)=CC1O C1(CN(C)C(C2CC2)=O)CCCN(C(C2CCCCS2)=O)C1 N1(C(CCn2c(C)nc(C)n2)=O)CC(CNC(=O)CC2OCCO2)CC(C)C1 C(=O)(CCCCCNC(=O)CCn1cncn1)NC(C#C)CC1CC1 c1(CC)nc(C(F)(F)F)ccc1C(=O)NCC1CCCN1C(=O)CC1CC1 c1(C(N2C(C)C(NC(C3CCC(O)C3)=O)CC2)=O)c2c(c[nH]c1=N)CCC2 c1(CNC(C2N(C(CC3CC(NC(C)=O)C3)=O)CCC2)=O)cnnc(O)c1 C1(CC)CN(C(c2nccc(C)c2N)=O)C(C)CO1.C123CC(C1)(C2)NC3=O c1(N2CC3C(C(=O)Nc4ccc(C#N)cc4)C(CC3)C2)ncc2ccc(F)cc2n1 N12CCC3CN(CC13)C1(CC1)C2=O.C1(COCC)CCCCO1.C1(=O)NCCN1 N1(C(C(c2ccccn2)C)=O)CCC2C(CCCN2C(=O)C(C)c2ccco2)C1 C(=O)(C1=CCC(F)(F)CC1)NC1C(C)CCN(C(CSc2c(C)cccc2)=O)C1 c1(CC(=O)N(CC(C)NC(C(C)OCCOCC)=O)C)sccc1C C12(C(=O)NCC(CC(C)C)NC(C3OCCOC3C)=O)CCCCCC1OCC2 C1(CC(N2CCC(CNC(C(C)N(C(C)=O)CC)=O)C2)=O)C=NN(C)C1=O c1(C(C)C)cc(C(N2CC(CCNC(=O)CC(C)(F)F)C(C)C2)=O)ccc1F N(C(=NCCCC1CCCC1)NC1C=CCCC1)C(C)COC(F)F c1(C(N2CCC(CCNC(C(C(C)(C)C)SC)=O)C2)=O)ccc2nc(C)cn2c1 N1(C(C2(CC)CCCCN2C(c2ccccc2)=O)=O)CC2(CCNC2=O)C1 Cc1nc(C)n(CC(N2CC3CC2C3NC(=O)CCC2CC2C(F)(F)F)=O)n1 C(=O)(CCCCCNC(=O)CCOc1cncc(Cl)n1)N(CC(C)NC(N)=O)C N12C3CCC1CN(CC3)C2=O.C1(C2(CC(=O)OC)CC2)CCc2nc[nH]c2C1 Cc1cc(N(C)CC2CCOCC2)nc(=NCC(C)c2ccc(Cl)cc2)[nH]1 c1(C(N2CCCC(C(C)C(=O)N(C(C)CN(C)C)C)C2)=O)cncc2[nH]ccc12 C1(C)(C(N2CCC(C(C)NC(c3c(C)c[nH]c3)=O)CC2)=O)CCCCNC1=O N1(C(C(=O)NC(C(=O)OC)C)CCC2CC2)CC2(CNC(=O)C2)C1 C1(NC(C(C)Sc2nncn2C)=O)CCN(C(c2ccn(C)c2)=O)CC1F C1(C(=O)OC)CC12CCN(N(C)C(C)C1CN(C3CCC3)C1)CC2 c1(N(C)C)n[nH]c2ccc(NC(C3CC(CCN(C)CCn4cncn4)C3)=O)cc12 c1(C(=O)NC(C(C)C)CNC(=O)CC2CCCCO2)cc(F)cc(Br)c1O C(CC(C)C(=O)NCC(O)CNC(c1onc(C)c1C)=O)=CCC C1(N(C(C2CCC(CC)CC2)=O)C)CCCCN(C(c2ccc([N+](=O)[O-])s2)=O)C1 CN(C1CCc2cc(F)ccc21)C(=O)CC1CC(=O)C1 N1(C(c2ccc(CC)s2)=O)CCC2CN(C(c3ccc(Br)o3)=O)CCC2C1 Cc1ccc2c(c1C)C(NC(C13CC(CN)(C1)OC31CCC1)=O)CC2 C=CC(C)(C)C(=O)NC1CC(NC(c2cnn(C(C)CC)c2C2CC2)=O)C1 C1(C(N(CC(c2ccccc2)O)C)=O)CC2(CCC(N)CC2)C1 Cn1cc(C(=O)NCCN2CCN(C(C3CCC(C)(C)C3)=O)CC2)cc1Br CCCS(=O)(=O)CC(=O)N1CCC(NC(C2CC3(CC3)CO2)=O)C(CO)CC1 N12CCCC(CC1)C2=O.C(=O)(C1=CCCCO1)NCC1N(C(C(C)(C)C)=O)CSC1 c1(CC(=O)NC2CC(CNC(c3c(C)ccc(O)c3)=O)C2)ccc2c(c1)COC2 C(C(=O)NC1CCC(CNC(c2nn[nH]c2Cl)=O)C1)(C(C)C)OC(C)C C12(Nc3nc(C)nc(Cl)c3)CCCC1CN(C(c1ccsc1C)=O)C2 c1(C(CC)C(=O)NC(C)(CNC(=O)CSC(F)(F)F)C2CC2)ccc(Cl)cc1 C1(C(=O)NC2(CC=C)CCN(C(=O)Cc3cnns3)C2)CCn2ccnc2C1 C12(NC(C(N3C(CC)CCC3)=O)=O)CCC1CN(C(=O)Cc1ccc(F)cn1)C2 C(=O)(C(C)C(O)CC(C)C)NC1(C(=O)Nc2ccc(C)cc2F)CC(O)C1 c1(OC)ncc(F)c(N2CCCC(N(C(=O)CCN3CCCC3=O)C)CC2)n1 C1(NC(C=CCCC(C)C)=O)(CO)CCCN(C(=O)C(C)C2CC2)C1 c1(-c2cc(C(=O)NC(C)CCNC(=O)C(C)(C)F)on2)c(F)cccc1Cl O=C(CCCCCO)N1CC2(CC2C(=O)NCC(F)CO)C1 C1(CCCOC)CN(C(=O)CC(=O)NC2CC2)CCN1C(=O)C=Cc1ccn(C)c1 C1(C(=O)NC2(CNC(c3cc(OC)c(O)nc3)=O)CCC2)CCCC2(CCC2)O1 Cc1cc(=O)n(-c2ccc(Cl)cc2)cc1CNC1COCC1C(N)=O c1(CC)ccc(C(CNC(C23CCC(C2)C3)=O)NC(c2ccncc2Cl)=O)cc1 c1(-c2cc(C(=O)NCCC3(O)CN(C(C=CCC)=O)C3)no2)ccc(F)cc1F CCC(C)(CNC(=O)C=Cc1cn(C)nn1)C(=O)NCC1CCC(O)CC1 c1(C(N(CCN(C(C2C(C)C2)=O)C)C(C)C)=O)cccc(-c2cccc(Cl)c2)c1 c1(C2CN(Cc3c(C)nn(C4CC4)c3)C2)cc(F)cc(Br)c1 c1(C(N2C(CNC(C3CC(F)(CO)C3)=O)CC(OC)C2)=O)cc2cccnc2o1 c1(C(N2CC3C(CNC(CCCSC)=O)(C3)C2)=O)cc2nc(C)[nH]c2cc1F c1(C(=O)NCC2(C)CCN(C(CCCC)=O)C2)ccccc1S(=O)C(F)(F)F C1(n2c(N3C(=O)OCC3)nc(-c3cccn4ccnc34)n2)CCC12CCNCC2 c1(OC)ccc(C)c(C(=O)NCC(C)(C)CNC(=O)Cn2cc(C)ccc2=O)n1 c1(CC2(C(C)NC(=O)OC(C)(C)C)CC2)c(I)cnn1C(C)(C)C C=CCCCC(C(=O)NCCC(F)(F)COC)NC(C1CCCCC1(C)C)=O CC1C(NC(=O)C(C)N2CC2)CCCN1C(c1ncoc1C(C)(C)C)=O N1(C(=O)CCOC2CC2)CCC2(C1)CN(C(c1cc[nH]c1)=O)C2 S(=O)(=O)(c1ccc(N2CC(COC)CC(C)C2)cc1Cl)NCCCC c1(C(C(=O)NC(C2(O)CN(C(C(C)OCCN(C)C)=O)C2)C)O)cccc(F)c1 C(=O)(CCCC(C)(C)NC(=O)C(C1CCCC1)SC)NC(CC#CC)C C(=O)(CC(C)C(=O)NCCOC1CCN(c2ccnc(C(C)(C)C)n2)C1)OC c1(C(N(CCCNC(COCC(=O)NC)=O)CCO)=O)cnn2c1CN(C)CC2 c1(C(=O)NC2CCCC(NC(CC3C(C)CCC3)=O)C2)ccc(O)c(F)c1 C1(N2CCC(OC)CC2)CCC(N=c2nc(NCC(C)C)c3nc[nH]c3[nH]2)CC1 c1(C(=O)NC2CCCC2CSC)ccc(N(C(=O)CCCCC2CC2)CC)c(C)c1 Cc1ccn(C(C)(C)C(=O)NC2CC(C)(NC(c3c[nH]cc3C)=O)C2)n1 c1(NC(C(COCC)C)c2nnnn2CC2CCCO2)cc(Cl)ccc1C C(=O)(C1=C(C)OCCS1)N(C1(C(=O)NC2C=CC(SC)C2)CCC1)C1CC1 C1(C(=O)NCCC(C)F)(Cc2ccccc2Cl)CCCN(C(=O)OC(C)(C)C)C1 C(N=c1[nH]cnc2[nH]ccc12)C1CCC(NC(=O)CC2CCCCC2O)C1 C1(NC(c2scc(OC)c2)=O)CCCC12CCN(C(c1cc[nH]c1C(C)C)=O)C2 C1(CCNCC)CCCN(C(=O)CCCC2CCC2)C1.C12(CC(C)C1)C(=O)O2 N1(C(=O)OC(C)(C)C)CCC(F)(F)C(NCCc2ccnc(OC)n2)C1 C(=O)(CCCS(C)(=O)=O)OC(N1CC(CC(CNC(C(C)C2CC2)=O)(C)C)C1)=O N1(C(c2cn(CCC)nn2)=O)CC2CC(C(=O)N(C)Cc3cncn3C)CC2C1 C(=O)(C1CCc2ccccc21)NC(COCC)C(=O)NC1CCCN1C=O C1(O)(CNC(c2cnc(CC(C)C)s2)=O)CCN(C(=O)C(F)=CC2CC2)C1 c1(C(N(CCC(C(C)C)NC(=O)C#CC(=O)N(C)C)C)=O)cccn2ncnc12 C1(CN(C)C(c2nc(Cl)sc2Cl)=O)CN(C(=O)CN2CCOC2=O)CCO1 N1(C(CCCCCN(C)C)=O)CC2OCCN(C(c3ccc(F)c(N)c3)=O)C2C1 C1(NC(COC)=O)CCCN(C(C2CCS2(=O)=O)=O)C1C CC(C)(CO)C(=O)Nc1cccc(NC(=O)Cc2ccn(C(F)F)n2)c1 C(=O)(C(C#N)(CC)CC)NC(CCC)CNC(=O)CNc1ccccn1 c1(N2CC3C(C)C3C2)[nH]c(=NCCC2CCCCO2)nc2scnc12 C1(CNC(c2n(C)ccc2)=O)CCCCCN1C(c1cc(=O)cc(Cl)[nH]1)=O c1(C(=O)NCCSCCn2cc(-c3c(C)ccs3)nn2)ccc(C(C)F)cc1 O=C(C1=CCCOC1)NC1CC(CNC(c2cnn(C3CC3)c2Cl)=O)C12CCC2 C1(C(=O)NCc2cnc(C)o2)CCN(C(=O)C2CCC3(CCC3)C2)O1 C1(CNC(C(=Cc2ccccn2)C)=O)C2CCC(C2)N1C(=O)CC(C)N(C)C C1(C#CC(=O)NCC(C)CN(C(=O)C=Cc2ccc(Cl)cc2)C)(CC)CC1 N1(CCC(=O)NC2CN(C(=O)C(O)C3CCC3)C2)CCCCC1=O CC#CCC(C(=O)NCC(C)C(C)O)NC(c1n[nH]c(C)c1Cl)=O N1(C(c2cnc(COC)s2)=O)CCCC2(NC(=O)Cc3nncn3C)CCCC12 c1(OCC)ccc(Br)cc1COC(C1CC1Nc1cnc[nH]1)=O CC(C)C(C)C(C)CC(=O)N1CCC(O)(CNC(c2ncoc2C2CC2)=O)CC1 C1(NC(C=Cc2nnc(C(C)C)o2)=O)CCN(C(=O)CSC2CC2)CC1O C#CC1CN(C(C2CCC(=O)N2)=O)CCN1C(=O)CCC1CC1(F)F c1(C(=O)NC2C(C=C)CN(C(C3CN(C)CCO3)=O)C2)nnc2ccccc2c1N C1(CNC(CC=C=C)=O)CN(C(=O)C(C)Cc2cnc[nH]2)CCCO1 c1(C(=O)NCC2N(C(CC(=O)OCC)=O)CCC2CC)cccc([N+](=O)[O-])c1Br C12CCCCC1N(CC)C2=O.C1(NC(=O)CCn2cccn2)CC(O)C1 C=CCCCC(C(=O)N1CC(O)(C(=O)NC)C1)NC(=O)CSC(C)C c1(OCCC#C)ccc(C(N2CCC(O)(CN(C(=O)CCCF)C)C2)=O)cc1 C1(CC)C(C(=O)NC(CC2CCC2)C(=O)NCC2(OC)CCC2)CCN1C Cc1ccc2n[nH]cc2c1C(=O)NCC(O)CNC(=O)C(F)(F)C(C)O c1(C(=O)NCC2C(NC(Cn3c(C)cc(C)n3)=O)C2)c[nH]c(=O)c2ccnn12 C1(C(=O)OC(C)(C)C)OCCC1NCC(F)(F)F.C12(CC1)C(=O)NCC2 C=CCCC(C)C(C)N(CC(N1CCC(C)C1(C)C)=O)C(C)C C(CN(C1CCOC1)N1CCCc2n[nH]cc2C1)c1c([N+](=O)[O-])cccc1 CC(=O)CCCC(=O)N1CCC(C(F)C(N2CCN(C)CC2CO)=O)C1 C1(OC)CN(C(C2CN(C(C)C)C2)=O)CC1NC(=O)Cn1ccc(C2CC2)n1 c1(C(N2CC(CNC(c3n(C)cc([N+](=O)[O-])c3)=O)C2)=O)ccn2c(O)nnc2c1 N1(C(C2=CCN2C(C(CC=C)CC)=O)=O)CCC2CCC(C1)N2C c1(OC)ccc(CC(=O)NC(C2CCCC2)CNC(=O)C2=CCCC2C)cc1F c1(CC(=O)NCC23N(C(C(C)OCCC=C)=O)CC(C2)C3)cccc(OC)c1N c1(NC(COC2(C)CN(C(CC(CC)O)=O)C2)=O)c[nH]c(=N)c(C)c1 C1(NC(=O)Cc2ccc3nc(O)[nH]c3c2)CCC2(CC1)CC2N=c1[nH]nco1 C1(CC#C)(C(N2CC(C)(NC(c3cn[nH]c3)=O)C2)=O)CCOCC1 Cc1ccc(C(F)(F)F)cc1C(N1CC(NC(c2cnc3n2CCC3)=O)C1)=O N1(C(c2n(CCOC)ccc2)=O)CCCCC1C1(NC(C2(C)CC(C)C2)=O)CC1 c1(C(=O)NC2CC(N(C(C3C(OCC)C3C)=O)C)C2)c(CC)nnn1C C1(OCC(=O)NC2(CC(F)CO)CC2)CCN(C(c2csc(O)n2)=O)C1 c1(C(N2C(CNC(CCC#CC)=O)C(C)CC2)=O)cc(OC)cc2ccoc12 c1(OC)cc(CC(=O)NC2CCCN(C(c3nccnc3N)=O)C2C)cc(F)c1 C1(NC(CN(C2CC2)CC)=O)CC2(CCN(C(=O)C(C(C)C)c3ccncc3)C2)C1 C1(C(C)NC(=O)CCSc2ccncc2)(Cn2cc(COC)nn2)CCCCC1 N1(C(C(P(C)(C)=O)O)=O)CCCC12CCN(C(c1cc(CC3CC3)on1)=O)CC2 c1(NCc2c(NC(C(C(=O)OC)C)=O)nccc2)ccc(OC(F)F)c(O)c1 C#CCCCCC(=O)N(CC(=O)NCC1=NOC(C)C1)CC C1(=O)CC(=O)N(CC)C(CC)CN1.c1(C(=O)NCC(O)CC)ccccc1OCC n1(CCC(=O)NCC(C)N(C)C(C2CCOC2)=O)cccnc1=O c1(C(N2CCC3(NC(C=CSC)=O)C(C2)C3)=O)sc2ccccc2c1Cl c1(C(C)C)ncc(C(=O)NC(CNC(c2cnnn2C)=O)Cc2ccccc2)s1 C12(C(N3CC(C)C(N(C)C)C3)=O)CC(CO1)N(C(=O)CC1(O)CCCC1)C2 C(=O)(C(CC)C(=O)N(CC(F)C(N1CCCC(OC)CC1)=O)C)OCC C1(C(=O)NCC(=C)CCNC(c2cccc(OC3CC3)c2)=O)CCC(C)(C)OC1 c1(C(=O)NCC23N(C(C(CN(C)C)(C)C)=O)CC(C2)C3)cc(C(N)=O)cc(Cl)c1 C1(CC(=O)N(CCC)C)CN(C(=O)CC23CCCC2C3)CC1C c1(N2CC(CN(C(CC(CCC)CC)=O)C)OCC2)ncc([N+](=O)[O-])cc1F N1(CCCNC(CC2CC(=C)C2)=O)CCN(C(=O)C=C(CC)CC)CC1 C#CCC(CC#C)C(=O)N1CC2(CC2)CC1CNC(C1(C2CC2)CC1)=O N1(C(Cc2cc(C)sc2)=O)CC(C)(C)OCC1CNC(=O)COC1CCCC1 c1(CC)ccc(CN=c2nc(-c3ccc(Cl)cc3Cl)o[nH]2)cc1C Cc1cc(F)cc(C(N2CCCC(CNC(=O)CNS(=O)(=O)N(C)C)C2)=O)c1C CC1(CC(N2CCOCC(NC(C3CCCCC(=O)N3)=O)C2)=O)CCCCCC1 C1(CNC(C2(CCC)CC2)=O)C2CN(C(=O)CSC(C)(C)C)CC12 C1(CC)CN(C(=O)C(O)CNC(=O)CC2(C#N)CC2)CCO1 C=CCC(C)C(=O)NCCN(CCOCCO)C(c1coc(C2CCC2)n1)=O CC1=C(CNC(c2ncsc2C)c2nnnn2CCSC2CC2)CCC1 N1(C(c2n(CC)ccn2)=O)CCC(C2(NC(=O)CCc3cncc(F)c3)CC2)C1 C(=O)(C(CCCCC1CC1)N(C)Cc1ccc(Cl)s1)NCCOC C(C(C)(C(=O)N1CCOC(C(N)=O)C1)NC(=O)Cc1nocc1C(C)C)SC Cc1nn(C)c(C)c1C(N1CCCC1CCCNC(c1csc(C(C)C)n1)=O)=O c1(C(=O)NCC(C)NC(C2(OC(C)C)CCC2)=O)cc2ncn(C)c2cn1 Cc1cnc2c(C(=O)N(C)CC3(NC(=O)CC4CCCCN4C)CC3)cnn2c1 N1(CC(=O)NCCOCc2c(OC)cccn2)Cc2c(F)cccc2C1=O CCCC(C#N)C(=O)NCCN(C(=O)CCc1ccnc(Br)c1)C(C)C c1(C(=O)NCC(C)(C2CC2)NC(C(C)c2cccs2)=O)nccc2ccncc12 C1(C(=O)NC(C)CCN(C(=O)CSc2ccccc2F)C)CCOC2(CCC2)C1 c1(C(=O)NCC(CNC(=O)CCCN2CCCCC2)O)c(N)c(F)cc(F)c1F c1(OCc2nc(-c3cc(F)cc(Cl)c3)on2)ccc2ncccc2c1 c1(CC)ccc(C=CC(=O)NCC2(CCSC)CC2)o1.C1(=O)CCCCN(C)N1 c1(C(c2nnnn2C)Nc2ccc3nc(C)[nH]c3c2)cc(C)cc2cnn(C)c12 c1(OC)ccc(Br)cc1C(C)NC(=O)N(C(c1ccccc1)CN(C)C(C)=O)C C1(NC2CC(F)(CCNC(COc3cn(C)nc3)=O)C2)CC2C=CCC(C1)C2 c1(CNC(=O)N(CCO)Cc2cncs2)ccc(-n2cc(Cl)cn2)cc1 C=CCC(F)(F)C(=O)NC1CC(C(=O)NCC(C)C(C)CC)C1 C1(CC(=O)NCC2CN(C3CC3)C2)CN(C(=O)NCCc2cccs2)CC12CC2 N1(C(C2C(CNC(C3N(CC)CCCC3)=O)CC2)=O)CCC2(CNC(=O)C2)C1 C(c1sccc1C)=CC(=O)NC(CNC(C(C=C)C)=O)C1CC1 N1(C(CCS)=O)CC2COCC2C1.Cc1nocc1C(=O)C(c1cccs1)O C(=O)(C(CO)C(F)(F)F)N1C(C(=O)NCCSCCO)CCOCC1 C(=O)(C(C(C)C)N(C1CCN(C(C)C(=O)NC)CC1)C)N(C(C)C)CC C#CCCC(O)C(=O)N1CCC(CC(N)=O)(NC(=O)C(F)C2CCCC2)CC1 Cc1cccc(CCNC(C2(CNC(=O)CCC3(C)N=N3)CC(F)(F)C2)=O)c1 C(C(C(=O)N1CCCCC1CN(C)C)C(C)C)NC(COCC=C)=O Cc1c(C(=O)NC(CNC(c2c[nH]nc2F)=O)C2CCC2)oc2ccccc12 C=CC(F)(F)C(=O)NC(C)(C)CC(=O)N(CC(N)=O)CC(N)=O c1(C(=O)NC2C(C)CCN(C(Cc3nc(CC)sc3)=O)C2)ccc(C)c(=O)n1C c1(C(=O)NCC2(CCNC(C3CCCC3)=O)CC2)nc(Br)c2n1CCCC2 C(=O)(C(C)(C)CC(=O)NCCCOCCNC(=O)CC(C)N(C)C)OC C=C=CCCC(=O)NCC(CCC)NC(C1CC(=O)N(OC)C1)=O C1(CNC(C2N(C(C3(OCC)CCC3)=O)CCCC2)=O)CCCC12CCC2 C1(CC)CCCN(C)C1.C12CCN(C1)C(=O)CC2.C12CN(C1)C2=O.C(C)(=O)O c1(N(C)CCOCCO)ccc(Br)cc1.c12cn(nn1)C2.C1CCCO1 C1(NC(C2CN(C3CC3)CCO2)C)CCC(C(=O)NCc2nc(C3CC3)no2)CC1 C(=O)(CC(O)CC(C)(C)C)N1CC(C(N2CC(O)(C(C(=O)NC)F)C2)=O)OCC1 CCCCCCC(C)C(=O)N1CC(CC(=O)Nc2cc(C)c(O)c(C)c2)C(C)C1 Cc1cc(F)c2ccccc2c1C(=O)NC1CCN(C(=O)CCNC(=O)CO)C1 c1(NCC2CCN(C)CC2)[nH]c(=NCC(C)(C)C2(SC)CCC2)nc2c1ncn2C C1(C(c2nnnn2CC(F)F)OCC)(NCCC(C(C)C)OC)CCS(=O)(=O)CC1 c1(CCC(=O)N(CCNC(c2conc2C(F)(F)F)=O)CC)nnc(C)n1C C1(C(=O)OC)C(O)CCN1C(=O)C(CCSC(C)=O)NCc1ccccc1 C(=O)(C(C)CC(F)(F)F)N1CCC(O)(CN(C(Cc2cn(CC)nc2)=O)C)C1 C=C1CC(C(=O)NC)N(C(C2CCN(Cc3ccc(C)s3)CC2)=O)C1 C1(C(=O)NC(C)C2CC2)CC12CCN(C(c1ccc(Cn3ccnc3)cc1)=O)C2 N1(C(CSCC)=O)CCC(C2(NC(c3cc(C4CC4)cs3)=O)CC2)C1 n1(CC(N2CC3CCC(C(=O)NC4(SC)CC4)CC3C2)=O)ncc2cc(C)cnc12 n1(CCOC)cc(NC(c2conc2CNC(C2CCC(O)C2)=O)=O)cn1 C1(CNC(C(C)SCC)=O)CCC2CN(C(=O)CC3CC(C)=NO3)CC12 C1(N(C(c2ccn(CCC)n2)=O)C)CN(C(c2cn(CCO)nn2)=O)CC1F C1(C(=O)NCC2C(C)(C)N(C(=O)C3=CCSC3)CC2)CNC(=O)CC1(C)C C1(C(=O)NCC2(C(N)=O)CC2)CCN(C(=O)C(F)C2(O)CCCCC2)O1 N1(C(c2nc(CC)[nH]n2)=O)CCCC(C(N2CCC(C(N)=O)CC2)=O)C1 c1(CC)occ(C)c1C(=O)NCc1noc(CNC(CC2(CCO)CC2)=O)n1 C1(c2onc(-c3cc(OC)c(Br)cc3)n2)Cc2cccc(OC(F)F)c2O1 N1(C(C2CC3(CN(C(c4cc[nH]n4)=O)C3)C2)=O)CC2CCCCCCC12 Cc1cc(C(N2CCC(NC(c3cc4c(s3)CCC4)=O)C2)=O)cnc1C(F)F CN1CCCC(C)(CNC(c2cc(CCN3CCCCC3CO)on2)=O)C1 c1(C2CC(c3ncccc3F)(C(=O)OC(C)(C)C)C2)ncnc2cccc(Cl)c12 C1(CNC(C(c2cccc(C#N)c2)(C)C)=O)CCCCC1(C)C C12(CNC(=O)NC(C)CN3CC4CCC3C4)CCC(O)(CC1)CC2 C1(CNC(c2ccccn2)=O)CCCN(C(=O)CCC(C)C)C1.C(=O)(CCN)NCC c1(NC(C2N(Cc3ccc(OC)cc3O)CCC2)=O)ccc(OC)c(OC)c1Cl N1(C(C=C(C)C(C)(C)C)=O)CCC(C(F)(F)F)C(CNC(C2(C)CCC(=O)O2)=O)C1 N1(C(C2CN(C)C2)=O)CCCCC(C2CN(C(C3CCCN(C(N)=O)C3)=O)C2)C1 CC1CCc2[nH]c(=NCC3(C)CCCC3)nc(N3CC(C)S(=O)(=O)C(C)C3)c2C1 C1(CNC(COCCCC)=O)CN(C(=O)CCOC)CCC1(F)F c1(C(C)NC(C2CC2C(=O)N(c2coc(Cl)n2)C(C)C)=O)csc2ccccc12 C1(NC(c2cccc(N(C)C)c2)=O)CCN(c2ccnc(C#N)n2)C1(C)C N1(C(Cc2c(C)con2)=O)CCN(C(=O)C(c2c(C)noc2C)C)C(CO)C1 c1(CNC(C(=O)NCCCC2N(C(CCC)=O)CCC2)=O)ccnc(F)c1 c1(OCCC)ccccc1N(C(c1scnc1Br)C(=O)NC)C C1(C(=O)NC2(CC=C)CC2)CC12CCN(C(=O)CCc1cnn(C)c1)C2 N1(C(=O)NCC2(COC)CCOC2)CCC(N2CCNS2(=O)=O)CC1 CCCCCC(CC)C(=O)N1CCCC(F)(CNC(c2cnn(C)c2C)=O)C1 C1(CNC(c2n(CCSC)nnn2)c2csc(Br)c2)CCC(F)(F)C1 c1(OCC(=O)N(CCC(C)NC(C(CC)n2ccnc2)=O)C)ccccc1CC c1(C(CN(C)C)NC(=O)NC2(CCCC)CC2)ccnc(OC)c1 N1(C(C2(CCOCC)CCC2)=O)CCCN(C(c2[nH]nnc2C(F)F)=O)CC1 c1(C(=O)NCCC(C(C)C)NC(c2c(C)n[nH]c2)=O)cc2cnccc2o1 c1(C(=O)NCC2CN(C(c3c(CCC)occ3)=O)C3C2C3)c(F)ccc(F)c1O c1(C(=O)NC2CC(C)N(C(=O)Cn3cc(N)cn3)CC2)coc2ccccc12 CC(C)(CC(=O)NCC(CC(F)(F)F)NC(=O)C1CCc2nccn21)C(F)(F)F N1(C(c2c(C)onc2)=O)CCC(C)C(NC(c2cc3sccc3s2)=O)C1C c1(CC(N2CC(C(C)NC(C(C3CCOC3)OC)=O)C2)=O)ccccc1C CN1CCN(C(c2ccoc2)=O)C(CNC(C2(Cc3ccccc3F)CC2)=O)C1 O(NC(=O)CC(C(F)(F)F)NC(=O)C(CC(CC)CC)CC)CCN1C(=C)C=N1 N1(C(Cc2nc(C)c(C)[nH]2)=O)CC(NC(c2cc3sccc3[nH]2)=O)CC2(CC2)C1 Cc1nn(C)c(F)c1C(=O)NCC1(C)CCC(NC(C23CC(CCO2)C3)=O)C1 C1(C(=O)NCC2C(CNC(=O)CCc3cc(Br)cs3)C2)CCCCCC1 c1(CC(=O)N(C(CCNC(COCCCOC)=O)C)C)ccnc(F)c1 N1(CC)CCOC(C(N2CCCCC2CNC(c2cccn2C(C)C)=O)=O)C1 c1(C(N2CC(CNC(C3CC(=C)C3)=O)(COC)C2)=O)coc(S(N)(=O)=O)c1 c1(C(C)NC(=O)OC(C)(C)C)cc(S(=O)(=O)NC(C2CCCC2C2CC2)=O)c[nH]1 C=CCCCC(C(=O)NC1CC(CC(=O)OC)C1)NC(c1ccc(F)cc1)=O C1(CNC(C2CCC(OC)C2)=O)CCC2CN(C(C3CCN3C(C)(C)C)=O)CC12 N1(C(c2c(COC)scc2)=O)CCC(C)(CNC(C2CC(C)=NO2)=O)C1 c1(NC(=O)NC(c2cn(C(CC=C)CC)nn2)(C)C)ccnnc1C C1(NC(C(C)=C2CCC2)=O)CN(C(=O)CC(c2cccc(F)c2)C)C(C)(C)C1 N1(C(CCC=C=C)=O)CCN(C(=O)CC2CCCC2C)C(CCC)C1 CC(CCO)C(=O)N(C)CCOCC(N1CCC(N)C1)=O.c1(N)ccccc1 c1(CN2CCC(C(=O)NCC(F)F)C(O)C2)ccc([N+](=O)[O-])cn1 C(=O)(CCC(F)(F)F)NCCOCCCNC(C1CC1C1CC1)=O N1(C(=O)C(F)C2CCC2)CC2CC1CN2C(=O)Cc1nc(C2CC2)cs1 N1(C(c2sc(C)c(O)n2)=O)CCN(C(=O)CN2CCSCC2)C(C)C1C N#Cc1cc([N+](=O)[O-])ccc1CNC(=O)CC(C(N)C(=O)O)c1ccccc1 C1(CNC(CSCC)=O)CCCCN(C(c2cc(OC)ccc2Cl)=O)C1 C1(C(=O)Nc2cccnc2F)CN(C(c2ccc(Cl)cc2I)=O)CCC1O c12ccc(cc1)[nH]2.C1(OCC)CC(C(=O)NCCNC(=O)Cc2cnoc2)C1 N1(CCCC)CC(C(=O)NCC2(NC(C3CNC(=O)N3)=O)CCC2)CC1=O CC1C(NC(=O)C2=CS(=O)CCC2)CC2CCC1N2C(=O)CCCS(C)(=O)=O CN1CCC2C(CCCN2C(c2cc(Br)cnc2Br)C(=O)NCc2ccco2)C1 CCC(CC)(CC)C(=O)NC1CC(NC(C2CC(O)CN2C(C)=O)=O)C(O)C1 N1(C(C(CC)CN(C)C)=O)CC2CCN(C(=O)C=C(C)Cl)CC2C1 c1(CCC(=O)NCC(CNC(c2cc([N+](=O)[O-])c[nH]2)=O)OC)ccc(Cl)c(Cl)c1 c1(OC)ccc2cc(C(N3CC4(CNC(=O)C(C)OC)CCC3C4)=O)nnc2c1 c1(OC)cnc(Cl)c(C(=O)NC2CCC(C)(NC(=O)CC(O)C3CC3)CC2)c1 c1(C(C(=O)NC2(CO)CN(C(C3N(C(C)=O)CSC3)=O)C2)C)c(C)nn(C)c1C c1(C(=O)NC2(CCNC(=O)CC=C(Cl)Cl)CCC2)nnn2c1CCC2 C1(NC(C(=O)OC)C2CC2)CCN(C(C)(C)C)C1=O N1(C(C(=O)N(CC)Cc2ccc(O)cc2)=O)CCCCC1C c1(NC(C2(CC)CC(O)C2)c2nnnn2C(C)C)ccc(C)c(C(F)F)c1 CC1=C(C(=O)NCC2(F)CCC(NC(C3(C(F)(F)F)CCCC3)=O)C2)CCCC1 CCCCCC(=O)NC12CC(C(N(C[Si](C)(C)C)CC3CC3)=O)(C1)C2 C1(NC(CCCOCCOCCOC)=O)CN(C(=O)CN2CCCC2)C2CC12 N1(C(C(C)OCCC=C)=O)CC(C(N2CCCC(C)(C#N)C2)=O)C2(CCC2)C1 C1(C(=O)NCCC(C)N(C(c2cnc(OC)c(C)c2)=O)C)CC2(C1)CC(C)(C)C2 C(=O)(C1=NN(C2CC2)C(=O)CC1)N(CCCN(C)C(c1cn(C)nn1)=O)C CCC(C)(C)CCNC(=O)C(Cc1cn[nH]c1)NC(=O)CC1CNC(=O)O1 C1(CC(N2CCN(C(c3c(Cl)ncc(N)c3)=O)CC2)=O)CCc2ccccc2C1 C(=O)(C(CNC(c1ncnc(C)c1C)=O)C(C)(C)C)NC1(CC(=O)OC)CC1 Cc1cnc(C(=O)N(C)CC2CCN(C(c3ccc(C(C)F)cc3)=O)C2)nc1 c1(C(=O)OC(C)C(C)(C)C)ncccc1CCNC(=O)OC(C)(C)C N1(C(C2C(C)CC(C)O2)=O)CCN(C(=O)CCN2CCCCC2=O)C2(CCC2)C1 C(C(C)CC(=O)N(C1CCN(C(c2cnc(CC3CC3)s2)=O)C1)CC1CC1)OC CC1CN(C(=O)COc2ccsn2)CCC1N(C)C.C12(C)CN(C1)C(=O)CC2 c1(C(c2n(C(C(=O)OC)C)nnn2)NCC2CCCCC2)sccc1S(N)(=O)=O N1(Cc2ccc(C#N)cc2F)Cc2cc(C(N3CCSCC3)=O)cnc2C1 Cc1ccc(CN2CCC(NS(=O)(=O)c3cn[nH]c3)CC2)cc1O C1(CNC(CC=C)=O)CN(C(=O)COC2CCC(C)CC2)CC1C C1(C(=O)NCCN(C(c2cc(C3CC3)ns2)=O)C(C)C)(OC)CC(C)C1 Cc1cccc2c(N3CCOc4ncccc4C3)nccc12 c1(C(N(CCCNC(C2CCSCC2)=O)CC)=O)ccn(C(C)C)c1C c1(OC)ccc(COC(c2ccccc2C(C)=O)=O)cc1F C1(C(N(C(CC)C(=O)N(C)CC2(O)CCC2)C)=O)CC2C(C1)C2(C)C N1(C(COCCCC#C)=O)CCC(C)(NC(C2(C)CC3(CC3)C2)=O)C1 c1(NC)ccc(Cl)c(C(=O)NC2CC(C)N(C(c3cn(C)c(C)n3)=O)C2)c1 N1(C(C(CC)N2CCCC2)=O)CC2CC1(c1cn(CCn3cccn3)nn1)C2 c1(NC(c2ccc(N3CCCC3)nn2)=O)cccc(CNC(N(C)CC)=O)c1C c1(CNC(C2C=CCN(C(=O)C3=CCCC3)C2)=O)ccc(NCC(F)(F)F)cc1 N1(C(C2CCN(C(=O)NCCCC)CC2)=O)CCC2(C1)NC(=O)N(C)C2=O CCC(CO)C(=O)NC(C)CC1CN(C(=O)C(F)(F)c2csc(C)c2)C1 C(=O)(C(F)C(C)C(F)(F)F)N(CC(C)NC(C(n1cc(C2CCC2)nn1)C)=O)C c1(C(C(C)=O)NC(N(CC=C)CCOC)=O)ccccc1 n1(CC)ccc(C(N2CC3CC(C2)C3NC(=O)CC(O)C(C)C)=O)cc1=O N1(c2nc(C)nc3c2c[nH]n3)CCC2(CCN(C(=O)CCCS(C)(=O)=O)C2)C1 n1(C)c(C2CC2)nnc1S.C(=O)(C(O)C1C(C(=O)NC)C1)N(CCCN(C(C)C)C)C N1(C(c2ncc(C)cn2)=O)CCC2(CCCN(C(c3ccc(F)cc3)=O)C2)CC1 n1(CC)ncc(C(=O)N(CCCNC(c2n[nH]c(C)c2F)=O)C)c1Br Cc1cc(C(N2CCC(C(F)F)(CNC(=O)Cn3ccnc3C)C2)=O)sc1C c1(C(N2CC(C)C(NC(C3OCCO3)=O)C2)=O)cccc2c1OCC2 c1(C(N2CCC(C(CNC(CCC(=C)Cl)=O)O)CC2)=O)nccc(N)c1Cl c1(C(N(CC(C)NC(c2cc(C)nn2C)=O)C)=O)ccc(Cl)c(F)c1F N1(C(Cc2nc(COC)sc2)=O)C2CCC(NC(=O)C3=CCN(C)C3)C1CC2 C1(C(=O)NCCC(C)NC(c2ccc(F)s2)=O)CC2(CC2)C1 c1(N2CCC(CC=C)(NC(C3CC(F)(CO)C3)=O)C2)ncnc(Cl)c1C(C)C C12(NC(C(C)c3cccs3)=O)CCCN(C(c3cc(Cl)ncc3Cl)=O)CC1C2 C1(CNC(C(CC=C)NC(C2(CO)CC2)=O)=O)CC(C(=O)OC)=NO1 n1(CC)cc(C(=O)NCC23CC2CN(C(c2cccc(=O)o2)=O)C3)c(C(C)C)n1 c1(CC(C)C(=O)NC2(C(=O)NC3CC(F)C3)CC2)cccc(C(F)(F)F)c1 N1(C(c2c(NS(C)(=O)=O)cc(Br)cc2)=O)CCC2(CCC(C(=O)O)NC2)CC1 C=C(C)C1OCCC1C(N1CC(C(=O)N(C)CCOC)C(F)(F)C1)=O CCCCC(C(=O)N1CC(O)CC1CNC(c1n[nH]cc1C1CCC1)=O)C(C)C C(C(C(C)C)NC(=O)C=CC(=O)OC(C)(C)C)NC(C1(OC)CCC1)=O C1(NC(C2C(=C)CC2)=O)CN(C(c2ccc(OC)nc2C(F)(F)F)=O)CC12CC2 C12(NC(c3cn(CCCC)nc3C)=O)CCC(CC1)N(C(c1cnc(S)n1C)=O)C2 C1(NC(=O)Cc2c[nH]c3ncccc23)CC2CC1CN(C(=O)Cc1ccns1)C2 c1(CN2CC3C(C(=O)NCc4ccc(C)nc4)(C3)C2)[nH]nc2ncccc12 CC1(C)C(C(=O)N=c2ccc(C#N)n[nH]2)CCS1(=O)=NC=O CCC(C#N)C(=O)N1C(CNC(=O)CSc2nncn2C)CC2CC12 C1(C(C)C)CN(C(=O)C(C)(C)c2ccno2)CCN1C(C1CC1C)=O CCCC(CCCNC(=O)C=CC(=O)N(C)C)NC(=O)C=Cc1cnc(C)s1 O=C(CC(O)CNC(c1ccc[n+]([O-])c1)=O)Nc1ccccc1C1CC1 C1(N(c2cccnc2)C(=O)NCC(=O)NC(C(=O)NC)CC)CCCN(C)C1 CC(=O)CCC(=O)NC(c1nc(C(=O)NCCCCCC2CC2)co1)C C1(C(=O)NC(CN(C(=O)CNC(C)=O)CC)C)CC2C=CC1C2 Cc1ccc(NC(C2CC(O)CN2C(c2ncc[nH]2)=O)=O)c(C(=O)N(C)C)c1 c1(OC)ncc(Cl)cc1C(=O)NC1CN(C(=O)C(C)OC)CC1F N1(C(C(C=C)O)=O)CC(NC(c2cccc(Br)c2Cl)=O)CC(F)(F)C1 N1(C(c2c[nH]c(=NC)s2)=O)CC(NC(=O)CCc2ccnn2C)CC(O)C1 Cn1nnc(C(N2CCC(C(C)(C)C(=O)NC(c3nc[nH]n3)CO)C2)=O)c1N CC1CC=C(C(=O)N2CC3C(CNC(=O)CCSc4ccc(F)cc4)C3C2)CC1 CC(C1Cc2ccccc21)NC(=NCCF)NCc1cccc(C(C)(C)C)n1 C1(CNC(C2CC(CC)C2)=O)CCC2(CN(C(=O)Cc3c(C)ncnc3C)C2)O1 N1(C(C2CCC(C)C2)=O)CCCC(C2CCN(C(C3(C4CC4)CCC3)=O)C2)C1 C1(CN(C(COC(CC)(C)C)=O)C)CCN(C(=O)C(c2cncnc2)C)C1 CC1CN(C(=O)CN(C2CC(C#N)C2)C(c2cccc3cc[nH]c23)=O)CC(C)(C)C1 C(=O)(C(C(=O)NCCC(O)CNC(=O)CN1CCOCC1)C1CC1)OCC CC1=C(C(=O)NC2CCOC2C(=O)N(C(C)C)Cc2cc(C)on2)CC1 c1(OCC(N2CC3C(CNC(C4CCC(=O)O4)=O)C3C2)=O)ccc(F)c(F)c1 C1(C(N(CC(O)CO)C)=O)(NC(C2(C3(C)OCCO3)CC2)=O)CCSC1 S(=O)(=O)(c1cnn(C)c1)N1CC(CC(=O)Nc2c(OC)cc(F)cc2)C1 Cc1cc(C(=O)NCC2CN(C(C3SCCC3C)=O)C2)c2cnccc2c1 C(=O)(C1=COCC1)N(CC(CC)NC(c1nc(Cl)cs1)=O)CC c1(-n2cc(C(=O)NCCC(=O)NC(C(=O)OC)C)nn2)ccc(Cl)cc1Cl N1(C(CC(=O)OCC)=O)CC2CC(C(=O)NC(c3cccc(C)n3)C)(C2)C1 N#Cc1c[nH]c(C(=O)NCC(CO)NC(=O)Cn2nnc(C(F)(F)F)n2)c1 Cc1nn(CC(N2CCC2c2cn(C3CCCOC3C(C)C)nn2)=O)c(C)c1C n1(CC(=O)NCCC(C)NC(=O)COCC2(F)CC2)ncc2ccccc2c1=O c1(N(c2cccc(Br)c2)C(N2CC3CC3C2)=O)ncn2cc(-c3cccs3)sc12 c1(NC(CC2CCCN(C(CNC(CCC)=O)=O)C2)=O)cc(Cl)c(O)cc1Cl C1(C(=O)NCCC(C)N(C(=O)C(c2ccc(O)cc2)=O)C)(COC)CCC(=O)N1 C(=O)(C=CS(C)=O)NCC(CNC(C1CCC(C(=O)OCC)C1)=O)C c1(C(=O)NCC2N(C(c3ccc(C)cc3)=O)CC(O)C2)cc(C)cc(C)c1C C(CCOC)(C(=O)NC1CC(CCC(N)=O)C1)NC(c1c(CC)cco1)=O N1(C(CC)C(=O)NCC(F)CNC(C2(F)CCCC2)=O)C(=O)CCC1=O n1(Cc2onc(-c3ncc(OC(C)C)nc3)n2)nnc2ccccc12 c1(N(CC(C(=O)Nc2cncnc2O)c2ccccc2)C)cc(C#N)cnc1C N1(C(CC(C)(F)F)=O)CCOCC(CNC(C23CCC2C3)=O)C1 CC(CN=C(NCc1cccs1)NCc1cccc(Cl)c1)CC(C)(F)F N1(C(C2CCN(C(C(CCC)C(C)C)=O)CC2O)=O)CCCC2C1CCN2C c1(C(N2CC(C)(N(C(=O)CNC(N)=O)C)C2)=O)ccc(-n2cccn2)nc1 N1(CC(=O)N(C)Cc2ccco2)CCC2(CC1)CC2CO CC1CN(C(c2sccc2C2CC2)=O)CC1NC(C1(S(N)(=O)=O)CC1)=O c1(C(=O)NC(CC)(C)CNC(C2(COC)CC2)=O)cnn2ccnc(C)c12 N1(C(C2C(SC)CCC2)=O)CC2CC(C1)C2NC(C1CC2CC2C1)=O c1(C(C(=O)NCCCSCC)N(C)CC2CCC(C)CC2)ccc(F)cc1F C(CCCCCC1CC1)N(C)C(C1CN(C(=O)C(c2cncn2C)O)C1)=O CCC(C#N)C(=O)N1CC(CO)(NC(C2CC(=O)N(c3ccccc3F)C2)=O)C1 c1(C(=O)NCC(CCCC)NC(C2C(=C)C2)=O)ccc(N)c(Cl)c1 N1(C(CCOCCC)=O)C2CCC1CC(N(C(=O)C(F)(F)CC)C)C2 C#Cc1cccc(C(=O)NC2CC(O)CN(C(=O)CCC3CCCC3)C2)c1F c1(C(=O)NC(CCN(C(C2(COC)CC=CC2)=O)C)C)cc(OC(F)F)n(C)n1 N1(C(CCCN(C(C)=O)C)=O)CCC2(CC1)CC2NC(=O)C(F)(F)CC1CC1 CCCC(C)CCNC(=O)CNC(=O)CNC(c1c[nH]c(=N)o1)=O C1(NC(c2nc(C(=O)OC)sc2)=O)CN(C(=O)CCCN(C)C)CC2CC12 n1(CC)ccnc1C(=O)NCc1ccc(C(=O)NCC2CCCSC2)s1 c1(NC(C(C)(N(C(CC=CCC)=O)C)C2CC2)=O)ccn2nccc2c1 CCCC(CNC(=O)CCC1OCCO1)C(=O)N(C)CC1CCC(C)CC1 Cc1cc(=NC(=O)C(=O)N2CC(O)(CN(C(=O)C(c3ccnn3C)C)C)C2)[nH]o1 c1(C(N2C(CNC(C3NC(=O)C4CCC34)=O)CC2)=O)ccc(Cl)cc1C(F)(F)F N1(C(c2c(Cl)c(C)n(C)n2)=O)CCC(NC(C2OCCCO2)=O)C(C)(C)C1 CCCC(C)(O)CC(=O)N1CCC(C)(C)C1CNC(c1ccn(C(C)C)c1C)=O N1(C(c2ccc(COC)o2)=O)CCC(N=c2cc(Cl)c(O)n[nH]2)C1 c1(CC)ccc(C(=O)NCC2CC(C(=O)N(C3CC3)Cc3cccnc3)C2)o1 O=C(C1CCc2cccnc21)N1CC2CCC(C1)C2CNC(C1(F)CCCC1)=O c1(C(N(CCCN(C(=O)C(c2cccn2C)=O)CC)CC)=O)nc(C)ccc1F C1(C(=O)NC2CCC(COC)C2)CC=CCN1C(C1CC1C(C)C)=O C(C)(C)(CCNC(=O)C=C(Cl)Cl)N(C(C1(C(CC)=O)CC1)=O)CC c1(OC(C)(C)C)ccc(F)cc1CC(=O)NCc1coc(-c2ccc(F)cc2)n1 C12(CC(=O)N(C)Cc3cnc(C)s3)CCC1CN(C(c1ncc(C)cc1F)=O)C2 c1(NC(CC)(CNC(C2CSCCS2)=O)CC)nc(C)nc(=N)[nH]1 c1(C(N(CCCN(C)C(c2cnn(C)c2)=O)C)=O)cccc(S(C)=O)c1 C(=O)(C(F)CCC(C)C)NC(CC)CN(C(=O)CCOCC(C)(C)C)C.C(CSC)O C1(C(=O)OCC)=C(O)N=NCC1NC(=O)Nc1cnn(-c2nccs2)c1 C(=O)(C(O)CCCCC)N(C(C(=O)NC(CC=C)(C)C(F)F)C(C)CC)C CC(CCNCc1ccccn1)N=c1[nH]n2cc(C(F)(F)F)nc2s1 Cn1nc(C2CCCN2C(c2cc3cc(Br)cn3cn2)=O)c2ccccc2c1=O c1(C(N2C(C)C(NC(=O)C(O)C3CCCC3)CC2)=O)cn(C)c(=O)cn1 c1(C(=O)NCC(CNC(C2CCC(C(=O)OC)C2)=O)O)nccn2cc(C)nc12 N1(C(C(CCC)N(C)C)=O)CC(C)(C)OCC1CNC(c1cc2[nH]ccc2s1)=O CCC(C(=O)NCC1CCCN1C(c1c(OC)ccc(C)c1OC)=O)C(F)(F)F O=C(CCCc1ncco1)NCCCNC(c1[nH]ccc1C1CCCO1)=O C(=O)(CCC(=O)C(C)(C)C)NC(COC)CC(=O)NC1CNC(=O)C12CC2 C(CCC(=O)NCCCNC(=O)CCCc1ccc(C)s1)NC(=O)NCC#C.SCC N1(c2snc(CCC)n2)CC2CC(NC(C3(n4cc(Br)cn4)CC3)=O)C1C2 C1(CNC(C(C=CC)O)=O)CN(C(C2CC2c2ccccc2)=O)CC12CCC2 C#CC1(C(=O)Nc2cnn(C)c2Cl)CN(C(=O)CC2CC(OC)C2)C1 c1(C(N(CCNC(CCc2ccnc(C)n2)=O)C2CC2)=O)cnn2cccnc12 N1(CCOC)C(=S)NC(c2ncc(Br)cc2OC)C(C(=O)OC)=C1C(C)OC C(=O)(C1=CCCCO1)NCc1ccc(C(N2C(C(CCC)C)CCC2)=O)s1 Cc1ccncc1CNC(=O)C=CC(C12CC(C1)C2)=O C#CCC(O)C(=O)NC1(CO)CN(C(c2cccc(-c3ccccc3)c2)=O)C1 c1(NC2CN(C(c3cnc(C)o3)=O)CC2C)ncc([N+](=O)[O-])cc1Br c1(OCC#C)cccc(NC(=O)CN2CCOC(CNC(=O)CC)C2)c1 c1(-c2cn(CCN(C(=O)Cc3cnsc3)C(C3CC3)C)nn2)cccc(C)c1F C1(NC(C2(COC)CC2(F)F)=O)CCN(C(C2CSCCS2)=O)CCC1CO C1(CN(C)C(c2cc(Br)ccn2)=O)CCN(C(C2CCC(C(N)=O)C2)=O)CC1 O=C1CC(CC(=O)NC2CCCC(NC(c3coc(C4CCC4)n3)=O)C2)=NN1 N1(C(c2nncc(OC)c2)=O)CCCC1C1CCCN1C(c1cccnn1)=O Cc1ccc2c(NC(=O)NCC3OCCCC3(C)C)[nH]nc2n1 c1(C(N2CC(OCCC(=O)N(C)CCn3cccn3)C2)=O)ccncc1N(C)C C1(NC(C(C)NS(CC)(=O)=O)=O)CN(C(=O)C#CC2CC2)CC1CC1CC1 N1(C(c2c(-c3cn(C)nc3)[nH]cn2)=O)CC2CC(C1)CN(C(C1CC1F)=O)C2 N1(C(CCCC2C(C)C2)=O)CCCN(C(C23CC(C(=O)OC(C)(C)C)(C2)C3)=O)C(C)C1 c1(C(C(=O)NC2COC2)N(C2COCCN(C)C2)C)nn(C)c2c1CCC2 c1(C(N(CCCNC(=O)C(C2CC2)SC)CC)=O)nccc(Cl)c1C C1(O)(CCNC(C2CCCCCCC2)=O)CCN(C(C2CC2C(F)F)=O)CC1 C(C(C)(CO)CN=c1[nH]c(=NC(C)CC2CC2)[nH]c2c1CSC2)OC C1(C)(C(=O)NC(C(C)NC(c2ccc(C)nn2)=O)CO)CC(C(C)(C)C)=NO1 c1(-c2cn(CCC3CN(C(Cc4nc(CC)sc4)=O)C3)nn2)cc(Cl)ccc1OC c1(CC)cc(Cl)c(C)c(S(=O)(=O)N2CCc3c(F)cccc3C2)c1 C=CC1(C(=O)NCC2(O)CCCC2(C)C)CCN(C(=O)C(C)CC2CCCC2)CC1 CC(CCC(=O)NCCC1(CNC(C2CCCN2C)=O)CC1)N(C)C C(C(CO)(CO)NC(=O)C=C1CCC1)N(C(c1ccn(CC(C)C)n1)=O)C n1(CC)nnc2c1C(C(=O)N1CCC3OCCC3C1)CN(C(c1cn[nH]c1)=O)C2 N1(C(CCCCC#C)=O)CC(NC(=O)C(C)OCCOC)CC2(CCC2)C1 c1(CC)nc(Cl)c(F)c(=NCC2(CO)CCN(C(=O)C3=CCCS3)CC2)[nH]1 C12(NC(c3c(SC)ccs3)=O)CCCC(NC(c3cnc(O)n3C)=O)(C1)C2 N1(C(C2(C)CCC(C)C2)=O)CC2CN(C(c3cc(C(C)(C)C)no3)=O)CC2C1 c1(C(N2CCC(O)C(O)CC2)=O)cnn2ccc(-c3ccc4[nH]ccc4c3)cc12 C1(Cl)(C(N(C)CCOCCN(C(=O)C(C)(O)c2ccccc2)C)=O)CC12CCC2 c1(OCC(=O)NCC(CNC(CC2(C=C)CC2)=O)F)ccccc1C(N)=O C1(C(=O)NC2C(Cn3cc(-c4n(C)ccc4)nn3)CCC2)CC(F)C(=O)N1 c1(N2CCCC(C(C)C)C2)nc(N(CCS(C)=O)C)nc2c1CCCC2 c1(C(=O)NCC(CNC(CCCC2C(C)C2)=O)(C)O)c(Cl)ccc2c[nH]nc12 N1(C(C2CC(NC(c3c(C#N)cccc3)=O)C2)=O)CCc2c(F)cccc21 N1(C(CC(C)OC)=O)CC(CNC(=O)CSc2cccc(C)c2)C(C)(C)C1 c1(C(=O)NCCC(C)NC(=O)Cc2ccccc2Cl)ccc(-c2cn[nH]c2)cc1 n1(CC)c(C)nn(CC(=O)NCCC2(NC(=O)CCC[N+](=O)[O-])CCC2)c1=O c1(CN2CC(NC(C)=O)C(F)C2)n[nH]c2cccnc12 C1(C(N2CCN(C(COC(C)C)=O)C(C)C2)=O)C2CCCC1CCC2 C(=O)(CC1NC(=O)c2ccccc21)N(C)CC1CCCN1C(=O)CNC=O c1(C(=O)NCCN2CCN(C(CC3C(C)C3)=O)CC2)c[nH]c2cc(F)c(F)cc12 c1(CC(=O)NCC2C(NC(C3(C)N(C)CCC3)=O)CCC2)cncc2ccccc12 Cc1csc2cc(C(N3CC(NC(=O)CCC4(C)CC4)C4CC4C3)=O)[nH]c12 C1(OC)CC(CNC(C2CC2F)=O)N(C(=O)Cn2cc(Br)cn2)C1 N=c1ccc(C(=O)NC2(CNC(=O)CN3CCCCC3=O)CCOC2)c[nH]1 N1(C(C(CO)NC(=O)OC(C)(C)C)=O)CCC(C(=O)NC2COC2)CC1 C(=O)(C1=CCCC1(C)C)N1CC(COC)N(C(c2cnc(N(C)C)nc2)=O)CC1 CC(C)C(C)C(CNC(C12CCC(CC1)O2)=O)NC(c1cc(=O)n(C)cn1)=O C=C=CCC(=O)NC1CCC1C(=O)N(C1CC1C1CC1)C CCCC(CCC)CC(=O)N1CCC(CO)C(NC(=O)CSCCC(C)C)C1 C(=O)(CS(=O)(=O)C1CC1)NC1CCC(C)(NC(=O)C(C2CCCCC2)F)CC1 c1(C(=O)NCCn2ncc(C)c2)ccc2c(n1)CN(C(c1ccc(Cl)o1)=O)CC2 C1(CC(N2CC(C)C(CNC(=O)CN3CSCCSC3)C2)=O)CCCC(C)(C)C1 C(=O)(C(C)C(O)CC(C)C)NCC#CCNC(c1c(C)c(Cl)cnc1)=O c1(NC(N2CC(C3CCCC(=O)C3)C2)=O)ccc2c3c(cccc13)CC2 c1(C(N2CC(C)C(NC(=O)C(c3cccn3C)=O)C2)=O)cc(Cl)ncc1F c1(C(CC)NC(=O)C(c2ccc(I)cc2)C)cc(C)ccc1C c1(C(=O)NC2C(C)CN(C)CC2)cc(O)nc2c1CN(C(C1CC(=O)CS1)=O)CC2 c1(C(=O)NCC2N(C(C(C)Cc3ccncc3)=O)CCC2)cc(C(C)C)cnc1O CCCCC(F)C(=O)NC1CC2CC(NC(c3cccc(C)c3Cl)=O)C1C2 N1(C(Cc2c(C)non2)=O)CCC(C)C(NC(c2cnc3sccn23)=O)C1C C1(OC)CN(C(c2cc(-c3cnn(C)c3)[nH]n2)=O)CC1NC(=O)C(C)(C)F CCCCCC(O)CC(=O)N1CC2CCCC2(NC(C2CNC(=O)N2)=O)C1 Cc1[nH]c(C(=O)N(CC#N)CC#N)c(C)c1C(=O)Nc1nc(Cl)cnc1I C1(C(N2CC(OC)C(OC)C2)=O)N(C(c2ccncc2)=O)CCC1(C)C CC#CCC(C(=O)N1CC2(CC(F)C2)C1)NC(=O)CCC1(C)CC1 c1(C(N2CCOC(c3ccccc3C)C2)C(=O)NC)ccc(C(F)(F)F)c(Cl)c1 c1(C(=O)OC(CC(CC)C)C)cccc2cccc(OC)c12 Cc1ccnc(C(=O)NC2CCC2CNC(c2cnc(C(F)(F)F)nc2)=O)n1 Cc1ccc(NC(C2(C)CCN(C(=O)Cn3cc(Br)cn3)C2)=O)c(Br)n1 C(CCC(C(=O)NC(c1ccccn1)C)NC(=O)C(C)C1CCCC1)OC CC(C)C(F)C(=O)N1CCC(C(C)CNC(C2CN(C3CCOCC3)C2)=O)CC1 C1(O)(C(C)NC(CC(CC)C)=O)CCN(C(c2cnc3sccn23)=O)CC1 c1(C(N2CCC(C)(C(=O)Nc3ncnc(Cl)c3Br)C2)=O)cc2cccn2cn1 c1(C(=O)NC(CNC(C(F)=CC)=O)(C)C2CCC2)ccnc2c(F)cccc12 Cc1nn(C)cc1C(N1CCC1CNC(=O)C(c1ccc(Br)cc1)C)=O CCC(CC(=O)N1CCOC(CF)C1)NC(C1CC1CC(C)C)=O C1(C(=O)NC(C=CC(=O)NCC2(CC=C)CCCC2)C)CCCN(C)C1 C12(NC(CC3(C)OCCO3)=O)CCCCCC1N(C(c1cncnc1)=O)CC2 C=CCN=C(NCC(C)(O)Sc1ccc(F)cc1)NCC(C)COC CCCC(CC)CCC(=O)N(CC(C)(C)CNC(=O)C(OC)OC)C C1(CNC(CCc2cn(C)nn2)=O)CCN(C(c2cccc(O)c2Cl)=O)C12CC2 N1(CCC(C(C)C)CO)CCC2(CCC(O)C2)CC1 S(=O)(=O)(c1cnc(N2CC(C3CC3)OC(C)C2)c(Cl)c1)NCc1ccc(CC)s1 N1(C(C2(C)CCNC(=O)C2)=O)CCCC2(C1)CN(C(C1COC(=O)N1)=O)C2 c1(N2C(C(=O)NC3CCCCN(CC)C3)CCCC2)c([N+](=O)[O-])c(C)nn1C N1(C(Cc2c(C)occ2)=O)CC(C(=O)N(CCN=[N+]=[N-])CCO)C(C)C1 C(CC(C(=O)NC12CC1CN(C)C2)NC(=O)CCN1CCOCC1)=CC c1(NCCN)cnc2ccccc2c1.c12cccc(c1)C(=O)N(C)CC(=O)N2 C(=O)(C(C)(C1CC1)OC)N.C(C=O)SCC.C1(=O)CN1C(C)C N1(C(C23CC(NC(C(C)NC(C4CCC4)=O)=O)(C2)C3)=O)CCCC(C)C1C C1(NC(c2ccc(C)nc2CCN2CCC(C)C2)=O)CCC12CCNCC2 C(=O)(CCCC(=O)N1CCC(N(C)C(C2CC(C)(C)CN2C)=O)C1)OC N1(C(C=CCOC)=O)CC(F)CC1CN(C(=O)Cn1nnc(C)n1)C C1(C(=O)NCC(C)(C)NC(C2(C(F)(F)F)CCCC2)=O)CC=CCC1 c1(C(N2CCC3(NC(CCn4ccc(=N)[nH]4)=O)C(C2)C3)=O)cnc2ccoc2c1 C1(C(N2C(CN(C)C(c3cccnc3C3CC3)=O)CCC2)=O)CCC2(CCC2)C1 N1(C(CC(CC)NC(C)=O)=O)CC(C(=O)NC(C)(C)CN2CCCC2)C(F)(F)C1 C1(C(N2C(C)(CNC(c3cccc(N)c3)=O)CCC2)=O)CCCCC1(C)C c1(CN2C(C(=O)Nc3ccc(C(=O)OCC)cc3)CC2)cccc2ccoc12 N1(C(CC(C)(C)OC)=O)CC2(C(=O)N(C(C)C(C)C)C)CCC1CC2 C(C(C)(O)CC(=O)NCCC(C)NC(=O)CN1CCC(C)(O)C1)OC N1(C(C=CCC=C)=O)CCC(N(C(=O)CCc2cccc(OC)n2)CCSC)CC1 c1(C(=O)OC)cnc(C(=O)NC2CC(CNC(C3(C)COC(=O)C3)=O)C2)cn1 C(=O)(C1=C2CCCN=C2NN1)N1CC(CC(C)NC(C2CC3(C2)CC3F)=O)C1 C1(NC(=O)Cc2ccsc2)CC2(C1)CC2NC(=O)C(O)Cc1ccccn1 n1(CC(N2CC(C)(NC(=O)C(c3ccccc3Cl)O)C2)=O)cc(S(C)(=O)=O)cn1 C1(C(=O)NCCN(C(CC=CC=C)=O)CC2CC2)OCCC1C(F)(F)F c1(OC)ccc2c(C(=O)NCC(C)CNC(=O)CCCCC(N)=O)n[nH]c2c1 C1(N(C(=O)CC(C)(C)C)C(C)C#N)CCN(C(C2(CO)CC(C)(C)C2)=O)CC1 C(=O)(C1Cc2ccccc21)NCCCOCCCNC(CCSCCC)=O C=C=CC(C)C(=O)N(C(C)(C)CC(=O)NC(C(=O)OC)C1CCC1)C c1(CNC(=O)NC(c2c(C)cccn2)CO)cnc(OCC(F)(F)F)c(C)c1 CC(C(=O)NC(C1(CN2CCCNCC2)CC1)=O)C(C)(C)c1ccccc1 c1(C(=O)NCC(CC(=O)N2CCC(C)(NC(C)=O)C2)OC)cnc(O)c(F)c1 C(=O)(CCCC(F)(F)F)N1C(C(C)C)(C(=O)N(C)Cc2cn(C)cn2)CCC1 C(=O)(CC1=CCCCC1)N1CC(C)(CNC(=O)Cc2nc[nH]n2)OCC1 c1(C(=O)NCC(CNC(C(CC)=CC)=O)O)cnc2c(c1)NC(=O)CN2C C1(NC(c2cc(C)c(Br)s2)=O)CN(C(c2cc(C#N)c[nH]2)=O)CC(C)(C)C1 N(C1CCC(NC(c2ns[nH]c2=O)=O)c2ccccc21)C(C12CCC(CC1)C2)=O C1(C(N(CCNC(=O)C(=Cc2cccnc2)F)C2CC2)=O)CCc2c[nH]nc2C1 C(c1ccc(Cl)cc1)=CC(N1CC(CSC)C(NC(=O)CCN2CCCC2)C1)=O C1(CCCOC)CN(C(c2cscc2F)=O)CCN1C(c1cc(COC)on1)=O N1(C(Cc2c(C)ccnc2)=O)CC(NC(=O)CCOCC(F)F)CC12CCOC2 N1(C(C(C)(C(C)C)OC)=O)CCN(C(=O)C=Cc2ccccc2)CC(O)C1 CS(=O)CCC(O)C(=O)NCC1(NC(c2cnc(=N)[nH]c2)=O)CCC1 N1(C(C(CCCCC)F)=O)CC2(CCN(C(=O)COCCC)CC2)CC1C n1(C(C)C)cc(N(C(=O)CC2CN(C(=O)C(n3cc(CC#N)nn3)C)C2)C)nn1 C(CO)(C(F)(F)F)NC(CC=CCNC(CCOC)=O)=O C1(C(=O)NC(CN(C(C2CCC2C(N)=O)=O)CC)C)=NC(C)=CC=CC=C1OC C12(CNC(c3ocnc3C(F)F)=O)CCC1CN(C(c1cc([N+](=O)[O-])c[nH]1)=O)C2 N1(C(c2c(C)cc(C#N)s2)C(=O)NCC2CCCO2)CCC2CCCCC12 n1(CC(C(=O)N(CCCCCC=C)CC(O)CCOC)(C)O)c(C)cccc1=O c1(C(=O)NCC(CC)(C)NC(=O)CC2CC(C)C2)cc(Br)c2nccn2c1 c1(C(=O)NC2CC(NC(c3c(C)cn(C)c3)=O)C2)nnc(O)cc1O C1(C(CC)(C)C)CCCC(C(F)(F)F)C1.c12n[nH]cc1CNC(=O)NCCN2 c1(C(N2CCN(C(C(CC(C)C)O)=O)CC2CF)=O)noc2c1CC(F)(F)CC2 CC1(C)CC(CCNC(N2CC(CC(F)F)C2)=O)N(C(=O)Oc2ccccn2)C1 c1(C(=O)NCCN(C(CC)=O)C2CCC2)ccc(Cl)nc1OCCN(C)C C1(C(=O)NCCN(C(=O)CCC2CCCO2)CCOC)Cc2nnc(C)n2C1 C(=O)(CCCC1c2nnnn2N1)NCC.C12(C)CC(C(=O)OC)(C1)C2 N1(C(=O)Cc2ccccc2)CCC2CN(CC(=O)NCc3cccs3)C2C1 C12(CCC)CCCN1C(=O)CONC2=O.C1(SC)CCCC1.C(=O)(C(C)C)NC c1(NC(c2nc(C(C)Oc3cnccc3N(C)C)sc2)=O)cc(F)cc(C#N)c1 N1(C(C(CC)n2cccn2)=O)CCN(C(=O)C(=C2CCCCC2)F)CC1CC1CC1 c1(CCC(=O)NC2CCC(N(C)C(C3CCCCO3)=O)CC2)nnc(O)nc1O C(=O)(C1=NOC(C)C1C)NCc1nc(C(N2CC3C(COC)(C3)C2)=O)c(C)o1 CC(C)CC(CNC(C1(c2cccs2)CC1)=O)C(=O)NC1(C)CCCC1C C(=O)(C1CCCc2nc[nH]c21)N(CCCCCNC(C1CCS(=O)(=O)C1)=O)C Cc1nc(-c2cccn2-c2ccccc2F)n(-c2cccc(C(=O)N(C)C)c2)n1 N1(C(C(n2ncc(C)c2)C)=O)CC2CC2C1C(=O)N(CC1CC1)CC1CC1 C(C)(C)(CCCC(=O)N1CC2(CNC(=O)C2)C1)NC(C1CC(SC)C1)=O c1(C(=O)OC)cc2c(Nc3cc(N4CCCC(N(C)C)C4)ncn3)nccc2o1 c1(C(N2C(C(C)(C)NC(C(C)OCCC#C)=O)CCC2)=O)cc(F)c(F)cc1O CC1=C(C)CC(C(=O)NCCC2CSCCN2C(C2CCC(=O)CC2)=O)CC1 C1(OC)CC(COCC2(C(=O)OCC)CCC2)N(C(=O)C2CC2)C1 C1(n2cc(C(CC)O)nn2)CCN(C(=O)C(c2cccc(C(=O)NC)c2)(F)F)CC1 C12(NC(C=C(CCC)C)=O)CC1CN(C(c1cccc(NS(N)(=O)=O)n1)=O)C2 CCCC(C)(O)CC(=O)NCC1CCN(C(=O)CCC2CCCO2)C(C)C1 c1(C(CNC(C(C)(C)OC)=O)NC(c2[nH]ncc2C#N)=O)ccc(Cl)cc1 N1(C(c2nc(C(C)C)sc2)C(=O)NC2COC2)CCCC2(CCC2)C1 c1(C(=O)NC2(C(N3CC(N4CCC4)C3)=O)CCCC2)cccc(F)c1F C(=O)(C(=O)C(C)(C)C)NC(CCN(C)C)C(=O)N(C)CC1(O)CCOC1 c1(OC)cc(N)cc(C(N2C3CCC2CN(C(=O)NC(C)C)C3)=O)c1OC c1(C(=O)OC)cccc(CNC(c2nnnn2NC2CSC2)C2CCOC2)c1 C1(NC(C(c2ccc(OC)cc2)=O)=O)CCN(C(c2c[nH]c(C#N)c2)=O)CC1C c1(OC)cc(C(=O)OC)c(C)c(Br)c1.C1(=O)C(=O)NCCCOCCCN1 c1(C(=O)NCC2(CNC(=O)CSc3cn[nH]c3)CCC2)cnccc1Cl C1(C(N2CC(N(C(CC(=O)NC)C)C)C2)=O)C2CC3C(C2=O)C13 c1ccccc1.CC(C(C)NC(C1(O)CC1)=O)NC(=O)C(C)OC1CCCC1 N1(C(C=COCC)=O)CCC2C(NC(c3ccc(-c4nnc(C)o4)cc3)=O)CC12 c1(C(N2CCC(C)C(C)C2)C(=O)NCCSC)cc2ccoc2cn1 Cc1nc(NC2CC(CNC(=O)Cn3ccsc3=N)C2)ccc1[N+](=O)[O-] C1(C)(CC)C=C(C(=O)N(C2CC(NC(c3cn(C4CCC4)nc3C)=O)C2)C)C1 CCCC(C(=O)NCCC1CC(C)(C)CO1)NC(=O)C#CC1CC1 CC1OC2(C)CC1(C(N1CCCC(O)(CNC(C3CCC(=O)N3)=O)C1)=O)C2 c1(N(C)Cc2cc(Br)cnc2O)c(C#N)cccc1C#N c1(C(N2CC3CCN(C(c4cnn[nH]4)=O)C3C2)=O)cn(CCO)c(=O)nc1O c1(OC)cc(CCC(=O)N(C)CC2(O)CN(C(=O)C(C)S(N)(=O)=O)C2)ccc1Cl C=C(Cl)CC(C(=O)NC(c1nc(C)no1)CO)NC(C1CC2(CC2)CO1)=O CC(C)C1=NOC(C(=O)NCC2CN(C(C3(C(C)C)CCC3)=O)CC2(C)C)C1 CCC(O)C(F)(F)C(=O)N1CC(O)(CN(C)C(c2ccc(=N)[nH]c2)=O)C1 c1(CNC(COC)(C)COC)nccc(=NC2CC(=C3CC3)CCC2)[nH]1 CC1CN(C(=O)CNc2nccs2)CCC1C(=O)O.C12(CC1)C(=O)N2 C(=O)(C(C)(C)CCCF)NC12C(CN(C(C(CCC)NC(C)=O)=O)C1)CC2 Cn1ccc(=O)c(C(=O)NC2CC(CC3CC3)C2)c1.C1CC(=O)NC12CC2 c1(NC(CN(c2cnccn2)C)=O)cccc(NC(C2(C)COC(=O)C2)=O)c1 C12(C(=O)Nc3nc(C)c(C(=O)NCC4CC5CC5C4)s3)CC=CC(C1)OC2 CC(C)(C)C(O)C(NC(=O)NC1C2COCC12)c1ccccc1 c1(CC)c(OC)cccc1C(=O)NC(C)(CNC(=O)C(C)n1cncn1)CC C(=O)(C(F)(F)C(O)C(C)C)NCCCN(C(c1cc(C)nc(CO)n1)=O)CCO N1(C(C(Cn2ccc(C)n2)C)=O)CCCC(O)(CN(C(=O)CNS(N)(=O)=O)C)C1 C12(CN(C(CC)C(F)(F)F)CCCO)CCCOC1CCN(C(=O)CSC(C)=O)C2 Cc1cc(C(=O)NCC2CC3CCC2N3C(C2(C)CCCCC2)=O)nc(O)n1 CCC(CC(=O)NCC1CCC(OC)CC1)N(C(=O)C(F)=CCCF)C CCCC(CC(=O)N1CCCC1(CC)CC)NC(C1(C)CCCCC1)=O c1(C(N2CC(F)(CNC(C=CCCCC)=O)C2)=O)cccc(CC2CC2)n1 C1(F)(CNC(c2cc(SC)oc2)=O)CCN(C(=O)C(F)C(C)C)C1 CCCCC(O)C(=O)NC1CCN(C(=O)C(C)Oc2ccccn2)CC1O c1(CN2CC(C(N3CC(C(N)=O)OCC3)=O)OCC2)ccc(Cl)c(O)c1 c1(SCC)cc(CC(N2CC(C)(NC(C3CC(=O)N(C4CC4)C3)=O)C2)=O)n(C)n1 CC(C)C1=NOC(C(=O)NC(CC(=O)N(CC(C)(C)C2CC2)C)C(F)F)C1 Cc1cc(N2CCC(NC3CCCSC3)CC2)ncc1S(=O)(=O)NC1CCC1 C1(CNC(C(C)(C)NC(=O)NCC)=O)CN(C)CCN1C(=O)CC(C)(F)F C=C=C(C)CC(=O)NC1CCCC1NC(c1c[nH]nc1OCC(F)(F)F)=O Cc1ccc(C(c2nnnn2-c2c(C)cccc2C)NC2CC(OC)C2)c(C)c1 CC1(COC)CC(C(=O)N(C2CCC2)CCO)CCN1C(C1CC1(Cl)Cl)=O N1(C(C=C(CCC)C)=O)CCCC(CC)(NC(C2CC3(CCC3OC)C2)=O)C1 C(=O)(C(=O)N=S(C)(C)=O)N1CCC(C(N2CCN(CC(C)C)CC2)=O)CC1C N1(C(C2N(C(c3c(CC)cccn3)=O)CCN(C)C2)=O)CCCN(C)CC1C C12(CNC(C3SCCS3)=O)CC1CN(C(C1CSCC(=O)N1)=O)C2 N1(C(CC)=O)CC2(CCN(C(=O)CC3CCCN(C(C)(C)C)C3)C2)C1 N1(C(C2N(C(=O)OC(C)C)CCCC2)=O)CCc2sccc2C1c1ccc(F)cc1 c1(C(=O)NCC2(CNC(C3(CC)CC=CC3)=O)CC2)cc2c(cc1Cl)OCCO2 C(CC(C(=O)NC(c1nnc(O)o1)C)NC(C1CC(=O)C1)=O)N(C)C CC1CC(C(=O)NC(c2ccccn2)C)CCN1C(=O)C1=C(Cl)CCC1 C1(O)(C(=O)OCC)CCN(C(=O)C(N)Cc2cccs2)C1 n1(CC)ccc(C(=O)NC23CC(C(=O)NCC4(C)NC(=O)NC4=O)(C2)C3)c1C CC1(C)CN(C(=O)CN(C(=O)C=CCF)CC2CC2)CCC1O c1(C(C)(C)C)ncoc1C(=O)NCC1(NC(C2CC(F)C2)=O)CCOC1 C1(O)(CC(=O)NCc2ccc(Cl)c(F)c2)CCCN(C(c2ccc(F)cc2)=O)C1 C(=O)(C(F)(CC)C(=O)OC)NCC1CCCN(C(C(c2ccc(CC)s2)=O)=O)C1 c1(C(=O)OC)scc(OC(C)=O)c1Cl.N12CCC(CC1)n1[nH]cc(c1=N)C2=O c1(C(=O)NCCOCCNC(C2(n3ccnn3)CC2)=O)cc2n(n1)CCO2 CS(=O)(=O)c1cccnc1C(N1CCC(CCNC(=O)CC(F)F)C1)=O c1(C(=O)NCC2(NC(C(C)SCCCC)=O)CCOC2)ccccc1NC N1(C(C(CC)N(C)C)=O)CCC2(CC1)CN(C(c1cccc3oc(C)nc13)=O)C2 c1(N2CCN(C(CC)C)CC2)ncc(S(=O)(=O)NC2(ON)CCSC2)cc1Cl Cc1nc(C2CCC2)oc1C(=O)NCC(C1CC1)N(C)C(C1COC1)=O C1(NC(CN(C(COC)=O)C)=O)CCCC(NC(=O)CCn2cncn2)CC1 C12CC(=NO1)C(=O)NC2.C(CCN(C)C)(C(=O)N(CCC(=O)OC)C)OC c1(CN2CC(Cn3cc(CSCC)nn3)OCC2)nc(C)c(C)nc1O c1(C(N2CCCC(C)(CNC(C(C)NC(=O)OC)=O)C2)=O)cc(F)c(N)cc1F c1(C(N(CCC(C)NC(CCNC(C)=O)=O)C)=O)csc2c(F)cccc12 N1(C(c2[nH]cc(C)c2C)=O)CCCCC(C(=O)NCCC2CCCO2)C1 C(=O)(C1CCCc2nn[nH]c21)NCCCNC(C1C2(CC(C)(C)C2)C1)=O C1(C(=O)C)CCC2(CC2)CO1.c1(C(=O)NCCOCCNC(=O)C2CC2)ccccc1 Cc1ccc(S(=O)(=O)N2CC(O)CC2CNC(c2c[nH]nc2C)=O)cc1 S(=O)(=O)(c1cnc(NC2C=CCC2)c(Cl)c1)NC(CCSCC)C [N-]=[N+]=NC1CCN(C(=O)C(C2(O)CCCCC2)NC(=O)C(F)=CC2CC2)C1 c12ccc(cc1)S(=O)(=O)NC(=O)N2.N1(C(=O)NC)CCC(C(C(C)C)NC)C1 C1(C(=O)NC2CN(C(C)C)C(=O)C2)CC12CCN(C(C1CS(=O)C1)=O)C2 C(=O)(CCCCCF)NC1C(NC(c2c(C)n(-c3cccc(Cl)c3)nn2)=O)CC1 c1(C(=O)NCC(C)NC(C(c2c(C)noc2C)C)=O)cncc2nnn(C)c12 C(=O)(CCCCCCCC)Nc1ccnc(C(=O)NCCOCCOCC)c1 c1(C(N(CCNC(=O)C(O)CN(C)C)CC)=O)ccc2ncccc2n1 C1(OC)CN(C)C(C)(C(N2CC(NC(=O)CC3CCCCO3)CC2(C)C)=O)C1 Cc1nnc2cnc(C(N3CC4CC3C4CNC(=O)CCS(C)=O)=O)cn12 n1(C2CCN(C(=O)NCCc3cc(C)cc(C)c3)CC2)c(O)nc2ccccc12 c1(C(=O)NC2CN(C(C3C(COC)C3)=O)C2)cc(-c2csc(CO)n2)c[nH]1 C(=O)(C#CC(C)(C)O)N1C(C)C(C(N2CCC(CN=[N+]=[N-])C2)=O)CC1 N1(C(c2cc(CCC)[nH]n2)=O)CCCCC(N(C)C(C23CC(CCO2)C3)=O)C1 C(=O)(C(C)N=c1cc[nH]cc1)NC(C)CCCCNC(c1ccnnc1)=O C1(C(=O)Nc2c(C(N)=O)occ2)CN(C(=O)C(O)C(F)(F)F)CCN1C Cc1c(C(N2CCC(O)(C(C)CNC(C3CC(F)(CO)C3)=O)C2)=O)cccc1N C1(C)(C(=O)NCCC(C)(C)NC(C(C)OCCCC)=O)CC=C(C)CC1 Cc1cccc(CNC(c2cccnc2CNC(=O)CNC(=O)C(C)(C)C)=O)n1 N1(C(CCC)=O)CC2(CNC(=O)C(C)C(C)COC)CC1CO2 Cc1nc(C)c(C(N2CCCC2(C)CNC(c2c(C)noc2C)=O)=O)s1 C1(C(=O)NC2(C)CCN(C(c3cccc(C(F)F)c3F)=O)C2)CC12CCSCC2 CN(C)NC(=O)CCC(=O)N1CCC2C(NC(=O)CCC3CCCCC3)C2C1 Fc1cc(F)c2cccc(-c3nc(COc4ccc(I)cc4)n[nH]3)c2c1 C1(NC(c2cccc3scnc23)=O)CC2CCC1N(C(C1SCCS1)=O)C2 CC1=C(C)CC(C(N2CCC(C(=O)NC(CO)C(C)(C)C)C2C(C)C)=O)CC1 C(=O)(C(C)C(=O)N1CCC(CC(=O)NCCC2CC(C)(C)CO2)CC1)OC c1(C(C)=O)cn(C)nc1C(=O)NCC(C1CC1)NC(c1cc(C(C)C)no1)=O C1(C(=O)N(CC(=CC(=O)NCC#C)C)C2CC2)OCCC1C(C)C c1(CC)c(C(=O)NCCC2(O)CN(C(=O)CC(C3CC3)C3CC3)C2)cnn1C CCC(C(=O)OC)C(=O)N(C)CCNC(c1cscc1C)=O C#Cc1cncc(NC(=O)CC2CC3(C2)CN(C(=O)Cc2cscn2)C3)c1 N(C(=NCC(C)N(C)C1CC1)N1CCC2(CC1)CCS(=O)(=O)CC2)C(CC)C CC(C)C(C(=O)N1CCCC1)N(C)CCNC(C1CSCCS1)=O C1(c2ccccc2)(CNC(C2C(C)CC2)=O)CC(NC(c2cnc[nH]2)=O)C1 N1(C(C2(C)C(C)CCC2)=O)CCc2nc(-c3ccc([N+](=O)[O-])cc3F)sc2C1 C(=O)(CCC(C)(C)[N+](=O)[O-])NCC(CNC(Cc1c(C)n(C)cn1)=O)C(F)(F)F CCC(CC(=O)N1CC(OC)CC1C(=O)N(CC(C)C)C)SC1CCCC1 Cc1cn2c(C(c3nnnn3C(C)C)Nc3cc(Cl)ncc3N=[N+]=[N-])c(C)nc2s1 c1(C(=O)NC2CCCN(C(C3C(C)C3C)=O)CC2)cc(O)ccc1[N+](=O)[O-] CCCCC(CNc1ncc(I)cn1)NC(c1sncc1C)=O N1(C(C(COCC)C)=O)CC(OC)C(NC(C2CN(CC(F)(F)F)C2)=O)C1 CCS(=O)(=O)CC(=O)N(C1CCN(C(=O)CN2CCCC2SC)C1)C c1(-c2cn(CC(C)NC3CCCC3)nn2)ccc(F)cc1.C1CCN1C1CC1 CCCCC(O)CCC(=O)N1CCC1CNC(=O)CC1(O)CCCCC1 c1(C(N2C(C(C)C)C(NC(C3CC(O)C3)=O)CC2)=O)ccc2sccc2c1 C1(NC(CC2(C(=O)NC)CCC2)=O)CCN(C(=O)Cc2ccsc2C)CC1C c1(C(=O)NCC(CNC(CS)=O)F)cc(OC)c(OC)c(Cl)c1.C#CCOCC=C N1(CC(N2CC(F)(CNC(COCCSC)=O)C2)=O)CCCCC(O)C1=O NS(=O)(=O)C1CC(NC(=O)CSc2cccc(F)c2)C1.c12nc(no1)C2 C#Cc1cccc(NC(=O)NCC(=O)NC2(C)CNC2=O)c1.C(CO)OC c1(C(N2CCC(NC(C3N(C(C)C)C(=O)CC3)=O)C2C)=O)ccc(=O)n(O)c1 Cc1cnn(CC(=O)NCC2(O)CC(NC(=O)CC(C)O)C2)c1 c1(OCC)cc(C)c(C(N2CCC(c3ccc(F)cc3C)C2)=O)cc1C c1(-n2cc(C3N(C(CCn4c(C)csc4=O)=O)CC3)nn2)ccc2cnn(C)c2c1 CC(C)(C)CC(F)C(=O)NCC1(C(N2CCN(CC3CC3)CC2)=O)CC2(CC2)C1 N1(C(=O)OC(C)(C)C)CCCC(C(=O)NC2CC(NC(C3CCOCC3)=O)C2)C1 c1(CNC(CC2C(C)C2)=O)c(Br)cccc1[N+](=O)[O-].C12CC(F)CN1C2 N1(Cc2ccc(C#N)s2)CCN(C(c2c[nH]c(=O)cn2)=O)C2CC12 N1(C(C(C2CC2)OC)=O)CCN(C(=O)C(N2CCCC2)C2CC2)CC1C c1(OCC)ccc(CCC(=O)N2CC(CCNC(c3sccc3SC)=O)C2)cc1 C1(CNC(=O)C=Cc2ccncc2)CCCCN1C(=O)CCCc1ccncc1 N1(C(CC=CC=C)=O)CC(C(N2CCCC(C#N)C2)=O)C2(CCC2)C1 C1(C)(CC)CCOC1Nc1cc(NC(=O)C(C)COCCOC)ncn1 Cc1cc(=NC(C)C2CCCC2)[nH]c(=NCCSCCC(F)(F)F)[nH]1 C1(NC(CC2(COC)CC2)=O)CCCC1CNC(=O)C(C)(C)C1CCC1 CC(C)C(O)C(C)(C)C(=O)NC1CCCC1NC(c1cc(O)cc(O)n1)=O N1(C(CC(CCC)C)=O)CCCC2(CC(NC(=O)CSc3nncs3)C2)C1 c1(C(=O)NC(CNC(C(C)CN(C)C)=O)C)ccc(F)c(C2(C)CC2)c1 CCCC(O)CC(=O)NCC12CC(NC(=O)CSCC(N)=O)(C1)C(C)O2 c1(CC(=O)NCCN(C(C2CC2F)=O)CC)csc(CC(C)C)n1 CC(C)C(C(=O)NCC(C(C)C)NC(=O)CCOCC(F)(F)C(F)F)C1CCC1 C1(NC(C(C)=C2CCCC2)=O)CCC(C)N(C(c2cnc(N(C)C)nc2)=O)C1 c1(OC)cccc2c1CCN(c1nnc(C3CC4CC3CC4OC)n1C)C2 CC1(C)C(C(=O)NCc2cccc(C#N)n2)CCN1C(C1CC(=O)NC(=O)C1)=O S(=O)(=O)(c1ccc(F)c(F)c1)N1CC(NC(c2cc3n(n2)CCC3)=O)C(F)C1 c1(C(C)NC(c2sncc2Br)C(=O)NCC)ccc(I)cc1 CC(CCC(C)(C)C)C(=O)N1CCCC(N(C)C(c2ccnn2C2CC2)=O)C1 N1(C(CCC2CC(NC(C3N(C)CCCC3)=O)C2)=O)CC2(CCNC(=O)O2)C1 C=CCCCC(C)(C)C(=O)NCC1CCCCCN1C(=O)CC(C)(O)CCC c1(C(=O)NC2CN(C(C(C)NC(COC)=O)=O)C2)cc(O)no1.C1CO1 C(=O)(C(O)CC(F)(F)F)NC1(CC=C)CN(C(c2ccc(O)c(Cl)n2)=O)C1 C1(CNC(=O)C(C)n2cccn2)(NC(CC2(C)CC2)=O)CCCCCC1 c1(C(=O)NC2(C)CC(NC(c3c(C(C)C)scn3)=O)C2)cccc2ccnn12 C1(CNC(C2(CC(C)C)CCC2)=O)CC(O)CN1C(c1cnc(Br)s1)=O c1(C(=O)NC(C)C(c2ccccn2)C)cc(NC(c2cnn(C)c2)=O)cc(Br)c1 N1(C(c2cc(C(C)=O)sc2)=O)Cc2ccccc2C(CNC(=O)C(C)C(F)F)C1 N1(C(COCCC=C)=O)CCC2C(CCN2C(c2ccc3c(c2)C(C)CO3)=O)C1 C(=O)(CC1=CCCCC1)NC(C)C(=O)NCCN(C)C.N12CCCN(C1)C(=O)C2 C1(CC)C(C(=O)NCCC2CC(=O)C2)CCN1C(=O)CC1CCC(C)(C)C1 c1(C(N2C(CC)CN(C(=O)C(C)C(C)(F)F)CC2)=O)cc2n(c1)CCCC2 C1(CNC(c2c(C#N)cncc2)=O)CCN(Cc2c(O)cccc2O)CC1(F)F c1(C(=O)NCC2(C)CC(NC(=O)CCSC(F)(F)F)C2)cnc2ccccn12 c1(C(N2CC(OC)(CNC(=O)C(C)CN(C)C)C2)=O)sc(C(F)(F)F)cc1C C(=O)(CCCCC1CC1)NCC1(OC)CCN(C(=O)COc2cccnc2)C1 C1(COC)CC(N=c2[nH]c(=NC3CN(CC(F)(F)F)C3)c3c([nH]2)CCCC3)C1 C(=O)(C1=CCCC1)NCC(C(C)C)NC(c1cnoc1-c1cccs1)=O C1(C(=O)NC(C(C)NC(c2nn(CC)c(O)c2)=O)C(C)C)CN(CP(C)(C)=O)C1 C1(C(=O)NC2CCCC(C#C)C2)CN(C(=O)C(C)CO)CC1C1CC1 Cc1cc(C(=O)NCC(C2CC2)NC(=O)C(F)(F)c2csc(C)c2)co1 N1(C(c2cc(OC)ncc2)=O)CCC2(CC2NC(C2(N(C)C)CC2)=O)C1 N1(C(C2CCC(CN(C)C)C2)=O)CC(F)(F)CC1CNC(c1[nH]cnc1C#N)=O C1(OC)CC(CCNC(=O)C(C)=C2CCC2)N(C(=O)C(F)F)C1 c1(CC)ccc(C(=O)NCc2csc(CNC(=O)Cc3c[nH]c(C(N)=O)c3)n2)[nH]1 C=CCCCC(C)(C)C(=O)NC1CCC1C(=O)NC1COCC(C)(C)C1 c1(CCC(N2CC3C(NCc4ncc(Cl)s4)C3C2)=O)cccc(Br)c1 c1(C(=O)NCC(CC)NC(=O)CC2C=CCCC2)cnnc(C)c1 c1(C(=O)NCC2CC(NC(C3(CCF)CCC3)=O)C(O)C2)c(F)cc(F)cc1Cl N1(C(c2cccc(CC)n2)=O)CC(NC(c2cccc(F)c2O)=O)C(C2CC2)C1 CC1C(NC(c2ccc(C(F)(F)F)[nH]2)=O)CCN1C(C1CC2CCCC12)=O c1(OCC#C)ccccc1NC(=O)CC1CCCCC1C C(C(=O)NC1CCC1C(=O)NC(C)(CO)C1CCCC1)(C(C)(C)C)OC CCC(CC(F)(F)F)NC(=O)N(c1ccc(CN2CCOCC2)c(C)c1)C(C)C CCC(CC(=O)N1CC(CNC(C2CC2(F)F)=O)(OC)C1)C1CC1 C(=O)(C1=CCCC1(C)C)NCC(CC)(CC)NC(C1CCN(C)C1=O)=O N1(C(C(COC)C)=O)CC2CC2(NC(c2ccc(-c3nccn3C)cc2)=O)C1 C1(CNC(C(COC)N(C)C)=O)CCCCN1C(=O)CC1CCCOCC1 C=CCC(C)(C)CCNC(=O)CN(C(C1CC(=O)C12CCC2)=O)CC C(CCN=c1[nH]c(-c2ccccc2)nc2c1CCCCC2)c1n[nH]c(=N)s1 C1(NC(=O)CNC(c2cn[nH]c2)=O)CCOCC1NC(C1CC(F)(CO)C1)=O C1(C(N2CC(F)(CNC(=O)C(O)(c3cccs3)C3CC3)C2)=O)CCCCS1(=O)=O c1(CCC)c(C(=O)NCC(c2ccccc2)Nc2nccc(C3CC3)n2)cnn1C Cc1cc(Cl)cnc1C(N1CC(CC(=O)OC(C)(C)C)C1)=O c1(C(=O)NC(CC)CN(C)C(C2CC3(CCC3)C2)=O)cccc2cncn12 C(=O)(CCCCC(N)=O)Oc1c(C(NOC(C)C)=O)nn(-c2ccccc2)c(=O)c1 C1(CNC(c2c(C)cncn2)=O)CCC2CN(C(=O)C=CCN(C)C)CC12 C1(S(C)(=O)=O)(C(=O)NCCOC2CCN(C(C3(CCOC)CCCC3)=O)C2)CC1 C1(CN(C(=O)CCCn2cc(C3CCOCC3)nn2)C)CC(O)CN1C C1(O)(CCNC(C)=O)CCN(C(c2ccccc2-n2cccc2)=O)C1 c1(C(N2CC(F)CC(NC(C(C=C)O)=O)C2)=O)ncnc2c1ccn2C C1(NC(CC(CC)CC)=O)CCC2(CC1)CC(NC(C1CCC(C3CC3)O1)=O)C2 CC1CC(O)CCN(C(C23C(NC(=O)CCCCCF)C4CC2C3C4)=O)C1 CC(CC(=O)N1CSCC1C(N1CCCC(C)C1CO)=O)CC(C)(C)C C1(OCC)CC2(CCCN(c3ccnc(Br)n3)C2)C1 c1(C(=O)NC(C)CN(C(=O)COCC(F)F)C)cc(Cl)nnc1O.C1(C)(O)CCCC1 CC(C)CCCOCC(=O)N(CC(C)(C)NC(C1CCS1(=O)=O)=O)C CCCC(CC1CCCC1)C(=O)N1CCCN(C(c2c(C)nnn2CC)=O)CC1 c1(C(=O)NC(CCOCC)C(=O)NCCC2CCOC2(C)C)ccc(F)cc1F N(C1COc2c(F)cccc21)C(=O)NCC1CCN(c2ccccc2)C1 c1(C(=O)NCC(CC)(C)NC(C2Cc3ccccc3S2)=O)ccc2[nH]ccc2c1 N1(C(C(C)N2CCC2)=O)CCN(C(c2ncccc2O)=O)CC1c1ccccc1 C1(C(=O)NCC2(NC(c3nc(C(C)OC)sc3)=O)CCC2)CC(C)(C)OC1(C)C C1(F)(C(N(C2CN(C(=O)Cc3ccc(Br)cc3)C2)C)=O)CCOCC1 c1(C(=O)NCCN(C(c2c(C)cnn2C)=O)C(C)C)cc2cccnc2cc1F N1(C(c2n(CC#C)ccc2)=O)CCC2CC1CN(C(=O)CNC(N)=O)C2 c1(C(N2CC(NC(CCCC)=O)C(OC)C2)=O)cc2c(O)ccc(F)c2[nH]1 C#CCC(O)C(=O)N1CCC(CN(C(=O)COCC(=O)OC)C)C1 c1(C(N2CCCC(CCC(N3CCOC4CC34)=O)C2)=O)c[nH]ccc1=O c1(CCC(=O)N(CCO)Cc2cc(C)no2)ccc(OCC(F)(F)F)cc1 C1(NC(C(C)(O)C2CCC2)=O)CCN(C(c2c[nH]nc2S(N)(=O)=O)=O)CC1F c1(N(CC(CC)(C)NC(C)=O)C)ccc(S(=O)(=O)N2CCC(CN(C)C)C2)cn1 C1(C)(CNC(C(CC2CC2)OC)=O)CC(F)(F)CN1C(=O)C(C)OC c1(C(=O)CBr)oc2ccccc2c1Cc1cnco1.C12(CCCC1)C(=O)N2 N1(C(CCNC(COC)=O)=O)CC2OCC(NC(c3cc(C4CC4)[nH]n3)=O)C2C1 Cc1cn2c(n1)CCC(NC(=O)Nc1c(C)nn(CC(F)(F)F)c1C(F)(F)F)C2 N1(C(CCc2ncc(C)[nH]2)=O)CCN(C(c2c(C)cncc2C)=O)CC1C(C)C CCCC(C)CCN=c1[nH]c2c(c(=NCCC3(C)CC3CO)[nH]1)COC2 C(=O)(CS(=O)(=O)C1CCCC1)N1CCC(C2CC2)(CNC(CCC(C)C)=O)C1 C1(NC(Cn2ncc(C)c2)=O)COCCC1NC(C1(Cl)CC12CCC2)=O C1(NC(CC2ON=C(C)C2)=O)CC2CC1N(C(c1n[nH]c(C)c1C)=O)C2 Cc1c(I)c(C(=O)N(c2nc(C(=O)NCCN(C)C3CC3)cs2)C)nn1C C1(CC=C)(CNC(=O)CCc2cc(C)[nH]n2)CCCC1.N12CCC(C1)SCC2=O.NCC C(CCC(C)C)(c1nnnn1C1COC1)NCC1C(CC(=O)OC)C1 C12(C(=O)NCC3C(C)CN(C(=O)C(C)OC4CCCCC4)C3)CC(C)(C1)OC2C c1(CNC(C(C)NC=O)=O)cc(C(=O)NC(c2ccccn2)C)cs1 Cc1cc(CC(=O)NC2(CNC(=O)CC3CC34CC4)CCCC2)ccc1O C(CCS(=O)(=O)c1ccc(Br)cc1)c1n(C)nc2c1CC(C)CC2 C(=O)(C1=CC2C=CC(C1)C2)NCC1(NC(CCc2cc(C)nc(C)c2)=O)CC1 c1(OCC)cccc(CC(N2CCC(C)(NC(c3csnc3Cl)=O)C2)=O)n1 N1(C(C(C)SC)=O)CCC2(CCCC2CNC(c2ccc[nH]2)=O)CC1 c1(CCn2c(N3C(C)C(C)(C)CC3)nnc2C2CC2)nc2cc(Cl)cc(Cl)c2[nH]1 C12(NC(c3ccc(O)nn3)=O)CCN(C(C3(CC(F)F)CC3)=O)CCC1C2 C(CC(=O)NC1C(O)CC1O)(C(F)(F)F)NC(c1c(OC)scc1)=O c1(C2(NC(N3CCCC(NC(CC(C)C)=O)C3)=O)CC(C)C2)c(F)cccc1F N1(C(C(c2ccccc2F)(C)C)=O)CC2(CCC2NC(C2C=CCC2)=O)C1 c1(C(=O)NCC2C(CNC(CCCSC(C)(C)C)=O)C2)ccc(Cl)c(S(C)(=O)=O)c1 C1(C#N)(C(=O)NC(CNC(c2c(C)scn2)=O)C(C)(C)C)CC2CC2C1 N1(C(c2c(C)onc2)=O)CCN(C(=O)CCCC(F)(F)F)CC12CCC2 C1(CNC(C(C)Nc2scc(C)n2)=O)CN(C(=O)CC2CC3(CCC3)C2)CC1C c1(C(N(CCC(C)NC(CCn2ccc(C)n2)=O)C)=O)cnccc1C(N)=O N1(C(CCc2ccc(C)o2)=O)CCOCC(CNC(=O)CN2CC(C)(C)C2)C1 CC1CCN1CC(=O)N(C)CCNC(=O)NC(C)C CCCCC(F)C(=O)NCC1CCC(NC(C2CCCNC2=O)=O)CC1 C(=O)(NN1CCCC(C(=O)O)C1)C1(N)CCCN(C(C(C)C)=O)C1 N1(C(CC(CC)O)=O)CCCCC2(CCN(C(=O)CC3CCC4(CCC4)O3)C2)C1 N1(C(CC(CC)C2CC2)=O)CCCC(C2CCN(c3nccc(C)n3)C2)C1 c1(C(=O)NC(CN(C(=O)C(C)Cc2ccncc2)CC)C)cc(C)cc(Br)c1 c1(C(=O)NC(CCNC(CCOCCOCC)=O)C)cnc(C)s1 c1(C(=O)NC2(C(CNC(c3cccs3)=O)C3CC3)CCC2)noc2ccccc12 C(=O)(C(C)CC(=O)NCCCCNC(C1CCCN1C1CCCC1)=O)OC N1(C(C(C)C#N)=O)CC2(CCC(CNC(=O)C=CC3CCCC3)O2)C1 N1(C(CC(CC)C)=O)CC2(CNC(c3cn(CCCF)nn3)=O)CC1CO2 N12CC3CCCN(C3C1)C(=O)c1cnc2s1.c1(C(C(=O)OC)C)cnn(C)c1 c1(C(N(CCCCNC(=O)Cc2ccn(C)n2)C)=O)ccccc1C1(C)CC1 Cc1ccc(C(N2CC(NC(=O)Cc3cc(Br)ccc3Br)C(C)C2)=O)cc1F C(CC(=O)NCC(C)N(C)C(c1cnn(CCOC)c1)=O)(C1=CCCC1)OCC C(=O)(C(C)(C)C1=CCSCC1)NCCC1CCC(NC(C2(CC(C)=O)CC2)=O)C1 N12CC(CC(C)C1)C2=O.N1(CC=O)CC(=O)N(C)C1=O.N1(CC)CCN(CC)CC1 Cc1ccc(I)cc1Cn1nc(-c2ccco2)nc1-c1ccc(F)cn1 C=CC1CN(C(=O)C(C)SCC)CC1NC(c1ccc(N)cc1O)=O CC(CNC(c1ccc(Cl)o1)=O)CC(=O)NC1CC12CC(O)C2 C1(CNC(C(CCC)(C)C)=O)C2CCCC1N(C(c1cc(=N)[nH]n1C)=O)C2 Cn1ccnc(C(=O)OCc2cccc(CS(N)(=O)=O)n2)c1=O C1(NC(c2nc(CCC)oc2)=O)CC2CCC1N2C(=O)CC(C)c1ccco1 N1(C(c2c(C)nccn2)=O)CCC2C1CCCN2C(c1nn(C)c(C)c1Br)=O c1(C(=O)NC2(CC=C)CCNC2)ccc2nc3n(c2c1)CCC3 C(=O)(CN=S(=O)(C)c1ccccc1)N1CC2(CCN(C(CCC#CC)=O)C2)C1 C1(O)(CNC(c2c(C)occ2)=O)CCCN(CC(O)COc2ccccc2)C1 CC1Cc2sc(C(=O)N(C)CCNC(c3cccc(O)c3Cl)=O)cc2C(C)C1 N1(C(c2cc(OC)nn2C)=O)CCN(C(C2CCC(=O)N2)=O)CC1c1ncc[nH]1 CC(C)(C(=O)NCc1cnns1)NC(=O)CC1COCCO1 C1(NC(CCC(=C)Br)=O)CCC2(CC1)CN(C(c1cc(C)sn1)=O)CCO2 c1(C(N(CC(O)CN(C)C(c2c[nH][nH]c2=N)=O)C)=O)ccc2c(O)n[nH]c2c1 c12ccc(C)c(c1)NCCN(C1CCN(CC)C1)C2.NC Cc1cc(C)c2c(N)c(-c3nc(-c4cccc(F)c4Br)no3)sc2c1 CCCC(C#N)C(=O)N1CC2(CC(NC(=O)C(CC)C(C)C)C2)C1 C(=O)(CN=S(C)(C)=O)NCCC1CC(OC)CN1C(c1ccc(C(N)=O)cc1)=O Cn1cc(CCC(=O)NCC(O)CNC(C2(CO)CCCC2)=O)nn1 C(=O)(C1=NOC2(CCOC2)C1)N(CCCNC(C1COCCN1CC1CCC1)=O)C CCC(O)C(C)C(=O)NCC1CC(NC(c2cn(C)cc(Br)c2=O)=O)C1 N(C(=NCCCn1cnc(C(N)=O)n1)NC1CCc2sc(Cl)cc21)CCO C(N=c1[nH]c(=NCC2CCCCS2)c2ccccc2[nH]1)C1C(C(C)C)OCCC1 C1(O)(CCNC(c2csnn2)=O)CCN(C(c2ccc(O)c(F)c2)=O)CC1 c1(C(=O)Nc2cccc(C#C)c2)cn2c(C)ccc(-c3cccc4c3CCC4)c2n1 c1(OCC)cc(C(N2CC3(CC3)CC2NC(=O)CCNC(C)=O)=O)ccc1OC c1(N(CC(CCC)C)C)nc(=NC(C)c2nnc(CSC)s2)[nH]c2c1CCC2 C=CC(CCC)CC(=O)NCC(C)CNC(=O)Cc1cnn(-c2ccccc2)n1 C1(C(=O)NCC(CNC(=O)CCCSC)OC)(OC)CCC12CCC2 N1(C(C=C(C)C2CC2)=O)CC2(CCC(NC(=O)Cn3cc(C(C)O)nn3)CC2)C1 c1(N(C)C)ccc(C(=O)NCCCOC2CCN(C(=O)C(F)C3CC3)CC2)cc1 c12cc3c(cccc3[nH]1)NC(=O)C1CCN(CC1O)C2.n1(CCC)cc(CN)nn1 Cc1csc(C=CC(=O)NCC2CC(CO)CO2)n1.C(=O)CCCc1cnn[nH]1 C1(CNC(C(F)OC)=O)CCN(C(c2ccc(C)nc2O)=O)C12CC2 N1(C(CC2CN(C)C2)=O)CC2(CO)CC1(C(N1CCC=C(F)C1)=O)C2 c1(C(N(CCNC(C2N(C=O)CCC2)=O)CC2CC2)=O)cc2sccc2[nH]1 C#Cc1cc(C(N2CCC(CN(C)C(C3(c4ccno4)CC3)=O)C2)=O)cc(Cl)c1 N(C1c2ccccc2OCC1F)C(c1ccc(C2CC2)cc1)=O C1(CC)CN(C(=O)CCOCC(N)=O)CC1C(=O)N(C1CCC1)C1CC1 N1(C(C(CCC)OCC)=O)CCC2(CCC2)C(NC(c2occc2Br)=O)C1 C12(C(=O)NCC3CC(CC)C3)CCN(C(=O)C=C=C(C)C)CCC1C2 c1(OC)ncc(NC(C2(C)CCCN2C(=O)CN2CCOC2=O)=O)cc1Br c1(OCC(=O)N(CCCCNC(=O)CC2CCC3CC23)C)cccc(F)c1F C1(C(=O)NCC(C(C)(C)C)NC(C2ON=C(CC)C2)=O)CC2CCC1CC2 c1(OCC(N)=O)ccc(CC(=O)NC2CC(NC(=O)C(F)(F)SC3CC3)C2)cc1 C(=O)(C(C)CC(N)=O)NCC(N1CCN(C(CC=CC)=O)CC1)=O c1(CC(=O)N(C)CC2CC2C)c[nH]c2ccc([N+](=O)[O-])cc12 c1(C(n2cc(CCCNC(=O)C(C)CF)nn2)CC)cccc(O)c1 N(C(=NCC1CC1)N1CCS(=O)(=O)C(C)(C)C1)Cc1ccc(C(F)(F)F)o1 N1(C(c2cnc(OC)nc2)=O)CCC(C)(C)C(NC(C2CCCN2C)=O)C1 c1(C(N2CC(OC)(CNC(c3cn(C(C)C)cn3)=O)C2)=O)cc(F)cc(C)c1N N1(C(C(C)N2CCCC2)=O)CCOCC(F)(CNC(=O)CCc2cn[nH]c2)C1 c1(OC)ccc2[nH]c(=NCCc3ocnc3C)nc(N3CCSC(C)(C)C3)c2c1 CCC(CC(=O)N1CCCC(C(N2CC[Si](C)(C)C2)=O)(CC)C1)C(F)F Cc1cnc(C(=O)NC2COCC2CNC(=O)C(N2CCCCCC2)C)c(F)c1 c1(C(N2CCC(C3N(C(C(F)OC)=O)CCC3)C2)=O)nc(Cl)sc1Cl c1(C(N2C3C(NC(CC=C=C)=O)C(CC3)C2)=O)c(C2CC2)nc2sccn12 Cc1ccc(CCCn2cc(CN(O)C(=O)N(C3CCCC3)C)nn2)o1 C(=O)(C(C)(C)C(C)(F)F)NC(C1CC(NC(c2c(C)occ2)=O)C1)C C1(C(=O)NCc2c(C)con2)CCN(C(c2cnn(C(F)F)c2)=O)C(C(C)C)C1 C1(C(=O)NC(C)CCNC(=O)CC2CC2(Cl)Cl)CCOC2(CCCCC2)C1 C1(OC)(OC)C(NC(=O)C(N2CCC(C)(CCO)C2)=O)CC1(F)F Cc1ncc2cc(C(N3CC4CCC(C3)N4C(C3(C#N)CCOC3)=O)=O)[nH]c2n1 CCCC(CC)C(=O)NCCC1CCN(C(=O)CN(C)CC)C1 CC(C)(COCC(F)F)C(=O)NC1CCOCC1NC(=O)CC1C=CCC1 C1(NC(Cn2c(CC)nnc2S)=O)CC12CCN(Cc1cc(C)nc(C)c1)CC2 CC1(C)CC(CNC(=O)C(CCF)NC(C2CC3(CC3)CO2)=O)CCO1 C(=O)(CCCCC(F)F)NC(C1CCOC1)CNC(=O)Cc1nnc(O)s1 c1(CNC(C2CC(O)CN2C(=O)C(O)Cn2cncn2)=O)ccc(F)c(Cl)c1F c1(C(=O)NCC(CC)NC(C2CC3CCC2O3)=O)ccc([N+](=O)[O-])cc1 c1(C(=O)NC(CNC(c2nc(C)sc2)=O)(C)CO)cccc2occc12 C(=O)(CN=c1cc[nH]cc1)NCC1C(NC(=O)COc2ccccc2Cl)CCC1 C(CCC(=O)N=c1ccn(CCc2ccccc2)[nH]1)C1C(C)CCC1 CC(C(F)C(=O)NC(C)CC1CN(C(c2sccc2C2CC2)=O)C1)C(F)(F)F c1(C(=O)NC2CC(NC(c3n(C)c(Cl)cn3)=O)C2)cccn2cncc12 C1(C(N2C(C)(CCC)CC2)=O)CC(C)CCN1C(c1cc(O)nn1C)=O C1(CNC(C(=O)N(CCC)Cc2ccc(Br)cc2F)=O)CC12CCOCC2 c1(C(=O)OC)cc(C)c(C(N2CC(CC(C)NC(c3cnn(CC)c3)=O)C2)=O)o1 c1(C(=O)NC2CC2CNC(C2CC2c2ccsc2)=O)cccc(=O)[nH]1 c1(OC)cccn2ncc(C(=O)NC3COCC3NC(c3nc(=O)n(C)[nH]3)=O)c12 CC(=O)CCCC(=O)NC(C(=O)N(C1CC1)Cc1ccoc1)C(C)C c1(C(N2CC(CC)N(C(=O)CCCSC)CC2)=O)ccc(C)c(C)c1F N1(C(c2c(C)nc(C3CC3)s2)=O)CCCCCC1CNC(c1ccc(CO)o1)=O c1(C(=O)O)cnn2cccc(F)c12.N12C3CCC1CN(C3)Cc1c([nH]cn1)C2=O CC(CS(=O)(=O)NC(C)(C)CC1CCOC1)CS(C)(=O)=O c1(CNC2CC(CC(=O)NCc3c(C)ncs3)C2)cc([N+](=O)[O-])c(Cl)cc1F N#Cc1c(Cl)nc[nH]c1=NCC(CNC(=O)C=Cc1ccccn1)C(F)(F)F N1(C(C(=Cc2cn[nH]c2)C)=O)CC(CNC(=O)CSC2CCOC2=O)CC1(C)C C1(NC(c2ccc([N+](=O)[O-])[nH]2)=O)CN(C(c2cccs2)=O)C2CCCC12 c1(C(N2CC(CNC(CCC#CC)=O)C(C)C2)=O)cc2n(n1)CC(F)C2 c1(C(=O)NCC2CCCC2)c(-c2ccc(F)cc2Cl)ccc2c1OCO2 C1(NC(c2n(C)ccn2)=O)CN(C(=O)C(C)(C)C(N)=O)CC12CCC2 C(=O)(C1=NOC(CNC(C2CNC(=O)N2)=O)C1)N1C(C)(CCC(=O)NC)CCC1 C=CC(C)CCNC(=O)CCCC1(NC(=O)CCc2cccs2)CCC1 CCC(CCCC(=O)NCC1CCOC(C)(C)C1)NC(c1ccc(C)cn1)=O C12(NC(c3c(C)nc(CC)s3)=O)CC(CNC(=O)C=C(C)C(C)(C)C)(C1)OC2C CC1(C)CCCC(C(N2CCC(C(F)F)C2)=O)C1 N1(C(c2sccc2F)=O)CCN(C2CCN(C(c3[nH]nnc3C3CC3)=O)C2)CC1 C1(C(=O)NCC(=C2CN(C(=O)CN(C)C(C)=O)C2)F)(OC)CCCCCC1 CC(C)(CCCNC(C1CC(C)(C)C1)=O)NC(C1CC1C(F)(F)F)=O c1(OC)ccc(Cl)c(CC(=O)NC2(CO)CN(C(C3CCN(C)S3(=O)=O)=O)C2)c1 C1(C(=O)NC2C(NC(c3ccc(-c4ccccn4)s3)=O)CC2)CCC=CCCC1 CC1C=C(C(=O)NCCN(C(=O)CC2CC3(COC3)C2)CC2CC2)CC1 C12(CNC(CC3(C)CCCO3)=O)CCC(CC1)N(C(c1ccnn1C(F)F)=O)C2 Cc1cc(Cl)cc(Cl)c1NC(=O)C(=O)NCc1scnc1C(C)C N1(C(C2C(C)(C(F)F)C2)=O)CC(CNC(=O)CC2(CO)CC2)C2(CCOCC2)C1 N1(C(Cc2cc(CC)no2)=O)CC(O)CC1C(=O)NCCCc1cncnc1 n1(CC(=O)NC2(C)CC(NC(c3nc(OC)c(C)s3)=O)C2)nc(C)ccc1=O C1(C)(C(=O)NCC(CC)(CC)NC(c2ccc(CN(C)C)[nH]2)=O)CC2CCC1C2 N1(C(CCCCCCC)=O)CC2COCC(C1)C2NC(c1cc2occc2[nH]1)=O C(=O)(N=c1ccn(CCF)[nH]1)N1CCC(CCC(=O)NC2CC23CCCCCC3)C1 CCCC(CCC)=CC(=O)NCC1CC(C(N2CC(F)(CC)C2)=O)C1 c1(OC)ccc(C(F)(F)F)nc1NC(N1CCCCC1C(c1ccccc1)(C)O)=O N1(CC)CCC(CO)CC1C.c12c(nnn1C)C(=O)N1CCC(CC1)C2 C=CC(C)CC(=O)NCC(O)CCNC(C1(CC)CC(C)(C)C1)=O N1(C(C)=O)CCC(NC(=O)NCCc2cscc2Br)CC1 C(=O)(C1=CCCN(c2cc(N3CC=CCC3)ncn2)C1)OCC CC1(NC(c2ccc(C(F)F)cn2)=O)CCN(C(=O)C=CC2CC2)C1 C(=O)(C(C#N)C(C)(C)C)N1C(C(=O)Nc2cccc(C)c2F)C(C)(C)CC1 c1(CC)cnc(Cl)[nH]c1=NC1CCCN(C(=O)Cn2nc(C)cc2C)CC1 C(=O)(C(CCC(C)C)NC(c1sccc1F)=O)NC(C(CC)C)CO C1(NC(c2c(CC)oc(C)n2)=O)CC12CCC(NC(=O)CCCNC(=O)OC)CC2 c1(CC)ncccc1C(=O)NC(CCF)C(=O)NCc1ncsn1 c1(Cn2c(-c3c(C)oc(Cl)n3)nc(CCCN(C)C)n2)ccc(O)c(Cl)c1 CC1CN(C(C2(C)CN(C(=O)CC3CCCN(C)C3)C2)=O)CCCO1 Cn1ncnc1CCCNC(=O)CNC(=O)CNC(=O)CC1(C2CC2)CC1 C(CC(=O)NNC(=O)c1cccc2ccccc12)(C(F)(F)F)NC(C)(C)C O=C(N=c1[nH][nH]c2c1COCC2)C1=CCCN(C(=O)CCc2nccs2)C1 c1(C(N(CC(=O)NC(C2CCOCC2)C)C2CC2)=O)ccncn1 c1(C(N2CCCC(C(=O)NC3CCS(=O)(=O)C3)CC2)=O)c(O)cc(O)cc1O c1(C(N2CCC(CC#C)(C(=O)NCC(C)OC)C2)=O)ccc(O)c(CC)c1 c1(C(N2CC(CNC(c3c(OCC)nccc3)=O)C(C)C2)=O)ccnc(O)c1F C1(C(N2CC(O)(C(C)NC(C(c3scc(C)n3)C)=O)C2)=O)CCC(=O)NC1 Cc1c(NC(c2cc(Br)ccc2CN)=O)cc(C(C)(C)C)n1C c1(C(N(CCOCCN(C(CCC(C)O)=O)C)C)=O)ccn2ncnc2c1 c1(C(N(CCC(C)NC(c2c(OC)nc(C)cc2)=O)C)=O)ccccc1S(C)=O C12(C(N3C(CN(C(=O)CN4CCC(C)C4)CC)CCC3)=O)CCC(F)(CC1)CC2 c1(OC)ccc2occ(C(N3CCOC4CN(C(=O)COC(C)C)CC34)=O)c2c1 C=Cc1ccc(C(=O)NC2CC3(C2)CC(Nc2ncncc2I)C3)cc1 CCCCC(CC(=O)N1CCCCC1CF)NC(C1C(C)C1(F)F)=O N1(C(C=CC(CC)C)=O)CC(CNC(=O)CCCC2CCC2)(OC)C1 c1(C(N2CC(C)CC(NC(C(C)NC(N)=O)=O)C2)=O)cncc(P(C)(C)=O)c1 CC1CN(c2nc(NCc3ncc(Cl)cn3)c3ccsc3n2)CCC1(F)F c1(C(=O)NC(CNC(C(COCC)C)=O)C(C)C)cc2c(nc1N)CCC2 N1(C(CC(C)O)=O)CCCC(NC(c2nnc(S)n2C)=O)C1C CCCC(C(=O)NC1CC(N)C1)NC(=O)CNS(=O)(=O)Cc1ccccc1 C(N=c1nc(N2CCC(OCC(N)=O)C2)c2c([nH]1)COC2)c1cc(CC)ncc1 Cc1cc(N)cnc1C(=O)NCCCCC(C)NC(C1(CO)CCCCO1)=O C(=O)(CCCC(C)(C)CC)NCC1C(OCC)CN(C(C2(C#N)CC(F)(F)C2)=O)C1 N1(C(C2C(=C)C2)=O)CC(NC(=O)CC2CCS(=O)(=O)C2)CC1C c1(C(C)C)cc(CC(=O)NCC(C)(F)CNC(C2(CF)CC(=O)C2)=O)on1 C(=O)(CC(CN(C)C)C(F)F)NC1C(NC(c2c(C)cccn2)=O)C1 C1(CC=C)(C(=O)NCCCCCN(C)C2CC2)CN(C(=O)COc2ccsc2)C1 Cc1nc(NC2CCCN(C(=O)Cc3cccnc3)C2)c2sccc2n1 c1(C(=O)NCC2N(C(CC(=O)OC)=O)CCOC2)c(Cl)c([N+](=O)[O-])nn1C C1(CC(N2CCC(NC(CC3CC(CC)C3)=O)(CF)C2)=O)CCCCC1(C)C C(CO)(C(C)NC(=O)C(CO)NC(N)=O)NC(C1(CCC)CCC1)=O c1(C(N2C(CNC(c3cc(CCC)oc3C)=O)CC2)=O)cc2nc[nH]c2cc1F N1(C(c2c(C)nc(C)o2)=O)CC(CNC(=O)C(O)CN(C)C)CC12CCC2 CCC(C)CC(=O)NCCCCSC.c12nn(cc1Br)c(=O)[nH]2 c1(CC(=O)NCc2cc(OC)c(O)cc2)cnc2ccccc2c1 CC1CCC(CNC(c2cccc(O)c2F)=O)CN1C(c1cncs1)=O c1(C(N2CCCC(N(C(C)Cc3ccc(F)cc3)C)C2)=O)coc2c1CSC2 C1(NC(c2ccnc(N3CCCC3)c2)=O)CCC2(CC1)CC2NC(C1CCO1)=O C(CC(N)=O)(C(=O)NC1CCCC(O)C1)NC(c1c(CC)n(C)cc1)=O N1(C(c2c(COC)ncs2)=O)CCCC2CN(C(=O)C(C)(O)C(C)C)CCC12 CC(C)C(F)(CN)C(=O)Nc1ccccc1-c1ccc(OC(F)(F)F)cc1 Cc1cc(F)cc(C(=O)NC2CC(NC(=O)Cc3ncn4c3CCCC4)C2)c1N C#Cc1cnn(C)c1C(N1CCC(CC(=O)NCc2ccc(F)cc2)CC1)=O c1(C(=O)NCC2CC(O)(CNC(C(CCCC)O)=O)C2)ccc2c(c1)nnn2C O=C1Cc2cnc(N3CC4CCC(C3)N4Cc3cc(C(F)(F)F)ccc3O)nc2N1 c1(C(=O)NC2CC(CNC(=O)C=CC3CCCC3)C2)cc(CO)ccc1Cl C1(CC#C)CCCN1C(=O)CC1(N(C)C(C2(C3CCCO3)CCC2)=O)CC1 c1(C(=O)NCC(CCOC)NC(=O)C(C(C)C)N(C)C)occ2c1CCCC2 N1(C(COCCCC)=O)C2CCC1CN(C(c1ccno1)=O)CC2 C1(C(=O)NCc2ccc(CC)o2)CC(F)C(=O)N1.N12CCC(C1)NC2=O c1(C(N2CCN(C(C3CC(O)C3)=O)CC2CCO)=O)cc2c([nH]1)CCCC2 c1(CC(=O)NC(CN(C(=O)CCc2cc(C)cs2)CC)C)cnccc1C CC(Cc1cnn(C)c1)C(=O)NC1COCC1NC(c1cn(C2CC2)nn1)=O CC1CN(C(=O)CN(C(=O)CC2(NC(N)=O)CC2)C)CCC1O C1(CNC(C(CC)C)=O)CN(C(=O)CCSc2cc(C)oc2C)CC1O C12CC3(CCN(CC3)C(=O)C1N(C)C)C2.Cc1snnc1N.C(C)(C)(C)C(=O)O CC1(C)CN(C(=O)C2=COCC2)CC1CNC(c1ccc(Cl)cn1)=O C12(C(N3CCCC(C)C3CO)=O)CCC(CC1)N(C(=O)Cc1ccc(O)cn1)C2 N1(C(C2OCCN(C(C)C)C2)=O)CC(CNC(=O)CCC(F)(F)F)OC(C)(C)C1 C12(CN3C(C(=O)OC)CC3)CC(CC)(CN1C(C)(C)C)C2.CCC1CC(=O)N1 C(CNC(=O)C1=CCCC1)(CC(=O)NC(c1ccc(C)cc1)C)OC CC1(C)CC(S(C)(=O)=O)CN1C(=O)NNC(=O)c1cc(Br)c[nH]1 C1(CN(C(c2c(C)n[nH]c2)=O)C)CN(C(=O)CN2CCCNC2=O)CCO1 Cc1ncnc(C)c1CC(=O)NC(C)C(C)NC(=O)COc1ccc(O)cc1 c1(CC(CO)N(C(C(CO)C2(C(=O)O)CC2)=O)CCO)cccc(OC(F)(F)F)c1 C#Cc1cnc(N2CCCC2CNC(C2CC2C2CC2C)=O)nc1 N1(C(c2cnco2)=O)CC2CN(C(c3c(O)cccc3Cl)=O)CC2C1 Cc1ncnc(C)c1CC(=O)NCC(CO)NC(=O)C(c1cccnc1)C C1(CC)CN(C(=O)C(O)CN(C)C)CC1C(=O)NCCc1cccnc1 c1(NC(CC2CCC(=O)NC2=O)=O)ccc2nc(O)[nH]c2c1.C12CCCCN1C2 N1(C(c2cc(C)n(C)c2)=O)CC2(C1)OCc1cc(-c3cccc(C#N)c3)ccc12 C1(C(=O)NC2C3(CC(NC(c4ccn(C(C)C)n4)=O)C3)C2)CCC2CCC1O2 C=CCC(CCCCC)C(=O)OCC(C12CCC(OC)(CC1)CC2)=O C1(NCc2ccn(C)n2)CC(C(=O)NCC(O)CN(C)C)C12CCC2 c1(C(C)(C)C)ccc(C#N)c(NC2CCC(C(=O)NC3CCCC(F)C3)C2)n1 Cc1ccccc1-n1cc(C(=O)NCCCN(C(=O)Cc2ncc[nH]2)C2CC2)nn1 C1(CC(N)=O)(OC)CCN(C(c2nsc(N3C4CCC3CC4)n2)=O)CC1 C(=O)(CCCC(N)=O)N1CCCC(CN(C(c2cn(CC)nn2)=O)C)C1 c1(C(N(CCCNC(=O)CC2CC(N(C)C)C2)C)=O)cnn2c1OCC2 C12(C(=O)NCCOC3CCN(C(c4c(C)nsc4)=O)C3)CC1Cc1c[nH]nc12 Cc1nc2cc(O)nn2c(C)c1CCC(=O)NC(CNC(C1(CF)CC1)=O)CO Cc1cc(C)c(C(=O)NC2COCC2NC(C2(F)CCCN(C)C2)=O)c(C)n1 C(=O)(CS(=O)(=O)C(C)(C)C)N1CCC(C(C)NC(=O)C(N2CCNC2=O)C)CC1 N1(C(Cc2cnc(C)s2)=O)CC2CC1CN2C(c1snc(C)c1N)=O N1(OC)C(=O)CCC1CC(=O)NC1N(C(=O)COCCN2CCCC2)CCCC1 N1(C(c2cc(OC)ncc2)=O)CC=C(C(=O)NC(C)CCSC)C1 C(C(C)(O)CC(=O)N1CC(CO)(NC(c2cc(C)nc(O)c2)=O)C1)OC C1(C(N2CC(C(C(=O)NCC=C(C(=O)OC)C)O)C2)=O)CCC(=O)CC1C C1(NC(C(C(CNC(C2(CC)CCC2)=O)C)F)=O)CC2C(O)C(O)CC12 C1(OC)CCCC(CN=c2[nH]nc(C(=O)Nc3ccc(OC4CC4)cc3)o2)C1 C1(NC(C(=O)NCC2(OCC(N)=O)CCCCC2)=O)CCOCC12CCC2 C1(CC)(CC)CC(NCCC(C)(C)NC(c2cc(COC)on2)c2nnnn2C)C1 C1(NC(c2cc(CNC(C3C(C)(C)COC3)=O)oc2)=O)CC(=O)NC(=O)C1 c1(C(=O)OCC)nc2n(c1Br)CC(C(C)C)CC2.C1(C)C(=O)N1C1CC1 c1(C(=O)NCC2N(C(C#CC)=O)CCOC2)ccc(Br)c2ncccc12 c1(C(=O)NCCCCCN(C(CCN(CCC)C)=O)C)sc2ncccc2c1N c1(CNCCC2(C(=O)NCc3cc(C)no3)CC2)cncc(C#N)c1 c1(CC)ncc(C(N2CCC(OCCNC(C3CCN(C)C3)=O)C2)=O)c(O)n1 Cc1cccc(Cl)c1-n1cc(Cc2ccccc2Cl)nn1.C1(C(C)(C)C)CCN1 N1(C(C(C(CC)O)C)=O)CCOC2(CCN(C(c3ccnc(SC)c3)=O)C2)C1 C1(NC(c2cncnc2)=O)CC(CNC(c2cc(C3CC3)ccn2)=O)C12CCC2 C=CC(C)(O)C(=O)NCC(=C)CCNC(c1csc(CO)n1)=O N1(C(CC=C)=O)C2CCC1CC(NC(=O)C(c1ccc(Cl)c(Br)c1)(F)F)C2 CCC(CNC(C1CCN(C(=O)NC)CC1)=O)N=c1cc(C(C)(C)C)nc(Cl)[nH]1 c1(C(N2CC(C(C)NC(=O)CC3C=CCCC3)C2)=O)n[nH]c2cc(OC)ccc12 c1(OC(C)C)ccc(C(=O)NCCNC(=O)CC2CCCC(=O)C2)cn1 C1(C(C)NC(CCNS(CC)(=O)=O)=O)CCN(C(=O)CC2(O)CCCOC2)CC1 c1(CN(C)Cc2cncc(OC)c2)cc([N+](=O)[O-])ccc1F C1(NC(c2c(CC)ocn2)=O)CC(F)CN(C(=O)CCCc2ccccc2)C1 C(=O)(C(C(C)C)NC(=O)C1CNC(C(=O)NC2CC(C)(C)C2)(C)C1)OC.OC C1(NC(C2CCCN(c3nccs3)C2)=O)CN(C(=O)C2=CCC2)CC12CC2 C(=O)(C(F)(F)C(F)(F)F)NCC1(F)CCN(C(c2ccc(OC)c(N)n2)=O)C1 N1(C(c2c(C)oc(CO)c2)=O)CCN(C(c2coc(C3CC3)c2)=O)CCC1C c1(C(=O)NCC(=C)CCNC(=O)C=CCOCC(F)(F)F)n[nH]c(CC)c1C C1(C)(COC(C2CN(C(C3CN(C(=O)NC)C3)=O)CC2(C)C)=O)CC(C(C)C)=NO1 c1(C(N(C(CN(C(C(C)C2CC2)=O)C)C)C)=O)ccccc1C(F)(F)F C(=O)(C1=CCCCC1C)NC(CC=C)CC(=O)NC(c1nc(C)no1)C CC1CCCCN1CCN(C(=O)CCCN(C)C(C)=O)C(C)(C)C N1(C(C(COC(C)=O)C)=O)CCC(CO)(NC(c2coc(-c3ccsc3)c2)=O)CC1 N1(C(CCC=C)=O)CCC(O)(CCNC(C2(CSC)CCCO2)=O)C1 C(=O)(CCC(C)CN(C)C)NC(CC)CNC(c1cnn(-c2ccccc2)c1F)=O N1(CC)CCCC(CNC(C2(n3ccnc3)CCC2)=O)C1=O CC1CN(C(c2cnn(CCNC(C3(O)CCC3)=O)c2)=O)CC(=O)N1C C#CCC(CC(=O)N1CCCC(CC2CC2)C1)NC(=O)C(=O)C(C)(C)C Cc1cccc(CC(=O)NCC2CCN2C(=O)Cc2ccc(C#N)nc2)c1C c1(C(C)=O)cc(C(N2CC=CC2C(=O)NCC2COCC2O)=O)no1 N1(C(C(CCCC)C)=O)CCC(C)(C)C(CNC(c2cnn3ccn(C)c23)=O)C1 c1(OCCOC(C(C(C)(C)C)c2ccc(C)cc2)=O)cccc2ccn(C)c12 C1(C(=O)OC)(CSCC#C)CCN(C(=O)CCCn2cccn2)CC1.C(C)C c1(-n2c3nc(n2)C3C)ccc2c(c1)OCO2.C(C)(C)OC N1(C(CCN(CCC)C)=O)CCC(CC(N2CCC(C)(C)C2C)=O)C1(C)C C1(CNC(CC(C)F)=O)COCCN(C(c2ccc(N)c(Cl)n2)=O)C1 N1(C(CCOCCN(C)C)=O)CC2(NC(=O)COCC3CCCC3)CCC1CC2 C1(NC(C(c2cccs2)NC(CC(CC)OC)=O)=O)CCN(C)C1(C)C c1(C(N2CC3(CCN(C(CCCCCSC)=O)C3)C2)=O)cnc2ncnn2c1N C12(NC(c3c(OC)n[nH]c3)=O)CCN(C(c3cn4c(n3)SCC4)=O)CC1C2 N1(C(CN(CC(N)=O)Cc2cn(-c3n(C)ccn3)nn2)=O)CCC(F)(CO)C1 c1(C(=O)NC(C2CCCC(C)C2)CC)cc2nc(C)ccc2o1 c1(C(=O)OCC)coc(CCCN(C(=O)Cn2cc(COCC)nn2)C)n1 CC1CCN(C(=O)CC2CCC3CC3C2)CC1CNC(C1CCOCC1(C)C)=O N1(C(CCCNC(C)=O)=O)CCC2CC2(NC(C2(CNC(N)=O)CC2)=O)CC1 C1(NC(C2CCC(CC)C2)=O)CCC(N(C(=O)C(c2cccnc2)=O)C)CC1 Cc1ccc2c(c1)CC(C(=O)NCC(C)N(C(=O)C1=NOC(C)C1)C)S2 c1(OC)nc(C)ccc1C(N1CCC(CN(C)C)C1)C(=O)NC1CC(F)(F)C1 CCCCC(C(=O)NC(c1cn(C)nn1)C(=O)NC1CN(C)CC1O)N(C)C C1(C(=O)NCC2N(C(CCn3c(C)csc3=O)=O)CCOC2)CC2OC1C1CC21 c1(OC)cccc(NC(C2CN(Cc3ccc(F)c(O)c3)C2)=O)c1Br c1(OC)cc(C(N2CC3CC(CNC(C4CC4CF)=O)C3C2)=O)cc(N)c1OC C(=O)(C1OCCc2ccccc21)N(C(C)CNC(C12CC(C)(C1)OC2(C)C)=O)C c1(SCC)cnc(O)cc1OC.c12ccccc1-c1cn(nn1)CCC21CC1 C#CCCCC(C)C(=O)NCC1CN(C(=O)CC2=CCCCC2)CC(C)(C)O1 c1(CC)cccc(NC(C2CCOCC2)=O)c1.N1(C=O)CCC(C)C1 Cc1c(F)ccc(C(=O)NC2CC2NC(=O)CC2CC3(CCC3)CO2)c1N N1(C(C=CCOC)=O)CCN(C(c2cc(-c3ccoc3)[nH]n2)=O)C2CCC12 c1(CN(C(=O)NCC(C)(C2CC2)SC)CC)c(Cl)ccc(F)c1N c1(C(N2CC3COCC3C2)C(=O)NC)cc(OC)cc(Br)c1 N1(C(=O)OC(C)(C)C)CC2CCN(Cc3ccc(Br)c(C#N)c3)CC2C1 CC(C)(CC(F)C(=O)NCC1CCCC12CC2)NC(=O)CC(C)(C)C(F)F C12COC(C)(C)CN1C2.CC(C)C(C(=O)N(C)C)n1cnnc1 C1(C(N2CC(Nc3nc(OC)c(F)c(C)n3)C(C)C2)=O)CCc2cnn(C)c2C1 C1(NC(C#CC2(C)COC2)=O)CCC2(CC1)CCN(c1nc(Cl)ncc1C1CC1)C2 C(=O)(C1CCc2cccc(=O)n21)N(C)CC1(O)CN(C(CCSC)=O)C1 c1(C(N(C2CCC(NC(c3cn(C(C)C)nn3)=O)CC2)C)=O)cc2n(n1)CCC2 c1(C(=O)NC2C(CNC(C3C(C#C)C3)=O)C2)cccc(F)c1 C(=O)(CCCC(C)(F)F)N(CC)CC1CCCN1C(c1cc(O)cc(O)n1)=O N(C(=NCC(F)(F)C1(O)CCCOC1)NCc1ccc(Cl)nc1)C(CC)C C1(NC(CSCC=C)=O)(CNC(C2CCCOCC2)=O)CCCCCC1 C1(C(N(C)CC2CCCCN2C(c2sccc2F)=O)=O)CCC(C)(C)OC1 C1(C(N2C(CC)CC2)=O)C2CC3C(C2NC(C2CCC(O)CC2)=O)C13 C1(C(=O)NCc2cc(C)nc(C)c2)CN(c2ncccc2[N+](=O)[O-])CCC1(F)F CC(C)C(C(=O)N1CC(NC(c2ncccc2Cl)=O)CC1C)n1cncn1 C1(C(=O)NCC2(C(=O)Nc3cncc(N(C)C)c3)CC(=C)C2)CCOC1(C)C N1(C(C(c2ccc(OC)cc2)=O)=O)CCN(C(=O)C=CC(C)C)CC1CF n1(CCC=C)nc(-c2ccccc2Cl)nc1C1CC(=O)N(CC(C)C)C1 N1(C(C=Cc2occ(C)n2)=O)CC(C2CN(C(c3ncc4[nH]ncc4n3)=O)C2)C1 c1(C(c2nnnn2C2CC2)NC2(COC)CCCOC2)c(C)sc2ccc(Cl)cc12 C(=O)(CCCN(C)C(c1nccn1C)=O)N(CC(F)F)CCOC C1(C(N(CCCOCCNC(C2C=CCCC2)=O)C)=O)CCCN(S(N)(=O)=O)C1 C(=O)(CC1COc2cc(O)ccc21)NC1(CNC(C2C(C)C2(F)F)=O)CCC1 c1(C(=O)NCCCCCNC(C(C)OCCC#C)=O)ccnc2cc[nH]c12 C1(C(=O)NCC(C)N(C)C(C2CCC(=O)O2)=O)C(F)(F)C12CC2 C(=O)(C(COC)CC)N(CCN(C(c1c(COC)cc[nH]1)=O)C(C)C)C C1(C(=O)NCC=C2CCN(C(c3ccncc3F)=O)CC2)CCc2cncn2C1 CC1CC(NC(=O)C=C(Cl)Cl)CN(C(C2CC(C3CC3)=NO2)=O)C1 c1(N(CCOCCN(C(C(CC=C)NC(C)=O)=O)C)C)cc(C#N)ccc1N C1(C(=O)NC2CC(N(C(=O)C=CS(C)=O)C)C2)CC2CCC1C2 Cc1cc(C(=O)NCC2(C)CCCN2C(=O)COc2ccc(Cl)cn2)cc(O)n1 C1(NC(C2C(C)=CCS2)=O)CCN(CCNC(=O)CC2CCCN2C)CC1 C(C(=O)OC(C)(C)C)(C(=O)NC1CCC(NC(=O)CC2CCC(C)(C)C2)C1)OC N1(C(c2cc(C)sc2)=O)CCC2(CCC2)C(CNC(c2cc(F)cc(F)c2)=O)C1 c1(C(=O)NCCCC2CCN(C(C3CCC(C)C3)=O)CC2)cc2cccnc2[nH]1 c1(OC(C)(C)C)ccc(C(=O)NCC(C)(C)CNC(=O)CC23COCC2C3)cc1 C1(C#N)(C(=O)NC2CC(F)(CNC(C3(OC)CCCCC3)=O)C2)CCOCC1 C(C(CC(C)C)C(=O)NCCCCNC(C1(C(C)(C)C)CCCCC1)=O)OC c1(C(N2CCC(CC3CCCO3)C2)C(=O)NC)ccc(Cl)c(F)c1F C=CCC(CC)C(=O)N(CC(C)CNC(=O)CSc1ccccc1C)C N1(C(c2ccc(COC)o2)=O)CC2CC(NC(c3coc(C)n3)=O)C2C1 N1(C(CSCC(=O)OC)=O)CCN(C(C2(C#N)CCC2)=O)CC1CC1CC1 N1(C(C2CNC(=O)N2)=O)CCC(CO)(NC(=O)CCC2NC(=O)NC2=O)CC1 CCCC(CCC)C(=O)NC1CCCC12CN(C(=O)C(CC)c1ccccc1)C2 N1(C2(C(=O)NC3(C)CC(NC(CCOC)=O)C3)CC2)CCCCC1=O CCC(CN(C)C)CC(=O)N1CC(CO)(NC(c2cccc(CO)c2C)=O)C1 c1(N(CCNC(CCn2ccc(C)n2)=O)C)ccc(OC(F)F)c(O)c1 CS(=O)(=O)c1ccc(C(=O)NC2CN(S(=O)(=O)Cc3ccccc3)C2)cc1Cl N1(C(CCC(=O)NC)=O)CCCCCC1C(=O)NC1CCC2CCC12 CCC(CCC(=O)N(C1CC2CCC1O2)C)NC(=O)C=Cc1nccs1 C1(C(N2CCC(c3ccc(F)cc3)(OC)CC2)=O)Cc2cccnc2C1 N1(C(CNC(c2c(OC)cccc2)=O)=O)CCN(c2nccc(C)n2)CC1C c1(C(=O)NC2C=CC(CNC(=O)C=CC(F)(F)F)C2)cc2n(n1)CCCC2 C(=O)(C(C)(C)CC(F)(F)F)N1CC(COC)(CNC(C2COC(C)C2)=O)C1 C#CCC(C)(C)C(=O)NCC1(CNC(c2c[nH]nc2CC)=O)CC12CCC2 c1(C(N2CC(NC(CC(C(C)C)O)=O)C3(C2)CC3)=O)cnc2[nH]nc(O)c2c1 C1(C(=O)NC2CC(C=C)C2)CN(C(=O)Cc2ccc(C)s2)CC1C=CC C(=O)(C(F)CC(C)(C)NC(=O)C#CC1CCOC1)NCCC1CC(C(=O)OC)C1 C1(NC(C2CN(CC)C(=O)C2)=O)CCN(Cc2cncs2)CC1O C1(C)(C(=O)NC2CC(C)(NC(C(C)N(C(C)=O)C)=O)C2)CCOC(C)C1 c1(C(=O)NC(C2CCCN2C(=O)CC2CC3CC3C2)C)cn(CCO)nn1 C1(C(=O)NC2C(CNC(c3c(C(C)C)noc3)=O)C2)CC(F)(F)CS1 C1C(CC(C)C)C(=O)N1.c1(COCCC(C)C)ccc(CC(F)(F)F)cc1 Cc1cccc(F)c1CN(C)C(C1CN(C(c2cc([N+](=O)[O-])cs2)=O)C1)=O C1(C(=O)NCC(C)N(C)C(C2CCC(C)(C)O2)=O)(CN2CCCC2)CCNC1=O Cc1nc(O)ccc1C(=O)NCC(CNC(=O)C(=O)N(C)C)C(F)(F)F N1(C(CC(c2ccc(Cl)cc2)C)=O)CCOC2CNCCC12 Cc1cnc(C(=O)NCCc2n[nH]cc2NC(=O)Cc2ccsc2)s1 c1(CC(N2CCC(O)(CCNC(C3(SC)CC3)=O)C2)=O)cc(F)c(C)cc1F CCCCC(O)CCC(=O)NCC1CN(C(c2ccc(N)cc2C)=O)CCN1C c1(C(=O)NCCN(C)C(c2occ3c2CCOC3)=O)ccc(Cl)c2cccnc12 c1(C2CN(C(C#C)=O)C2)nccc(=NC(=O)c2c(OC)ccc3ccccc23)[nH]1 C1(CC)CN(C(=O)C(C2CCOCC2)O)CCN1C(c1cc(Cl)ccc1Cl)=O C1(C(=O)NC(C(=O)NCC)C)CN(C(C2(F)CCC2)=O)CCO1 c1(OCC)cnc(C(=O)NCCO)c(Cl)c1.c1(C(=O)NC)ncn(CC(C)(C)C)n1 n1(CC)nc(C(N2CC=CCC2C(=O)NCCN=S(C)(C)=O)=O)cc1C C=C1CC2CCCC(C1)N2C(=O)CC(C1CC1)NC(c1ccnn1C1CC1)=O N1(CC2CCC(C)(C)C2)C(=O)CN(CCC2(C)CC2(F)Cl)C1=O C(=O)(C1CCCc2sc(=N)[nH]c21)NCC(=O)OCC1(C)CC1(F)F CC1CCN(C(=O)Cc2cncnc2)C1CNC(c1ccc(-c2ccccn2)o1)=O N1(C(C(C)NC(c2cccc(F)c2)=O)=O)CCC(NC(=O)C2=CCCS2)C12CCC2 c1(OCC=C)cccnc1C(N1CCCC1CNC(=O)CCNS(C)(=O)=O)=O C1(CCOC)CN(C(c2nnc(Cl)cc2N)=O)CCN1C(C1CN(C)CCO1)=O CC(C)(C)C(CNC(C12CC(C1)C2)=O)NC(c1ccn(C(F)F)n1)=O Cc1nc2cc(C(=O)NCC3(C)CC(NC(C4CC4C(C)(C)C)=O)C3)cnc2[nH]1 C1(NC(C(=O)NCCOCCCOCC)=O)CCCCN(C(C)C)C1 c1(C(C(N2CCC(N(C(=O)Cc3cscn3)CC)C2)=O)(F)F)ccc(C)cc1 C1(C(C(=O)NCC(CC)CO)(C)C)CCCN(C(=O)C(O)CCSC)C1 CCCCCCCC(F)C(=O)N1CCC(C)(CCNC(c2cc(F)n(C)n2)=O)C1 N1(C(CC(C2CC2)NC(C(CC)NC(C)=O)=O)=O)CCC2(CCSC2)C1 N1(C(c2ccc(C#C)cn2)=O)CCCCC(N=c2[nH]c(Cl)ncc2[N+](=O)[O-])C1 N1(C(c2n[nH]c(C)c2F)=O)CCC2(CCCN(C(=O)CN3CCCCCC3)C2)C1 N1(C(CN(C)S(N)(=O)=O)=O)CCC(CCNC(=O)C2=CCCCO2)C(F)(F)C1 N1(C(c2c(C)nc(O)cc2)=O)CCCC(C)(C)C1CNC(C1(C(N)=O)CCC1)=O c1(COC(CC2N(C(CSC)=O)CCC2)=O)cccc(O)c1F c1(CN2C3CC(CNC(COCC)=O)C2CC3)nc2ccc(OC)nc2s1 c1(C(=O)NC(CN(C(CC2N(CC)CCC2)=O)C)C)ccc(F)cc1SC C1(CNC(C2C(=C)C2)=O)CCCC12CCN(C(c1cnn(C)c1Cl)=O)CC2 Cc1ccc2c(c1)SC(C(=O)NC1CC(NC(c3coc(O)n3)=O)CC1O)C2 C(=O)(CC(C)CC(C)(C)C)NC1(C)CC(NC(c2c(NC(C)=O)c(C)ccc2)=O)C1 N1(C(C2(COC)CC2)=O)CC(COC)(NC(C2COCCO2)=O)C1 N1(C(C(C)=C2CCC2)=O)CCC2(C(=O)Nc3cc(Cl)cnc3C)CCCC12 N1(C(CN2CCC(OC)C2)=O)CCCC12CCN(C(=O)CCC(=O)OC(C)(C)C)C2 c1(C(n2cc(CN3CCCC3c3nccs3)nn2)C)cccc(Br)c1 S(=O)(=O)(c1ccc(N(CC(O)C2CC2)C)c(C#N)c1)NCc1c(C(C)C)nn(C)c1 c1(-c2ncc(C(=O)NCC=CCNC(c3ccns3)=O)s2)cccc(F)c1 N1(C(c2c(CC)n(CC)nn2)=O)CCC(C2(NC(=O)CC3(C)CC3(F)Cl)CC2)C1 Cc1ncn(C)c1C(=O)NC1CCC(CN(C)C(c2cc(Cl)cnn2)=O)CC1 N1(C(c2cn(CC)nn2)=O)CC(CNC(=O)COC2CCOCC2)CCC1C N1(C(c2c(C)n[nH]c2C)=O)CCC2(CC2NC(C2CC(C)C2)=O)C1 C1(CCNC(C2CCCC2)=O)CN(C(=O)C(F)=C2CCCC2)CCCO1 C1(C(=O)NC(CC=C)CNC(=O)CC23CC(C2)C3)CCc2nncn2C1 C(=O)(C(C)CC(C)C(C)=O)NC1C(CC)N(C(c2cscc2OC)=O)CCC1 c1(C(N(CCN(C)C(C2CSCCS2)=O)C)=O)cnc(N(C)C)s1 N1(C(C2ON=C(C)C2)=O)CC2(CC(C(=O)N(C)Cc3cccnn3)CO2)C1 C1(NC(C2(C)ON=C(C)C2)=O)CC(C(=O)NC(C(N)=O)C(C)C)=CC1O C1(CNCC(COCC)F)CC=CCC1C(F)(F)F C(=O)(C(CC)NC(=O)Cn1cc(CC)cn1)N(CC(=O)N(CC)CC)C c1(-c2cc(F)c(SC)c(F)c2)cc2c(s1)CCN(Cc1cccc3[nH]ncc13)C2 c1(Nc2cccc(Cl)c2)cccnc1N(C(=O)CNc1cccc(F)c1)C1CC1 N1(C(CCC)CC2(C(O)C(C)C)CC2)CCN(C(c2ccccc2SC)=O)CC1 C(=O)(CC(O)CNC(C1CC(C)=NO1)=O)NC(C(=O)NCC(C)C)C C1(CNC(c2cn(CCC)nc2)=O)CCC(C(N2CCC2C(C)O)=O)CC1 c1(C(=O)NC2CN(C(c3c(N)ccc(C(C)=O)c3)=O)C2)cc(S(N)(=O)=O)sc1C c1(OC)cc(OC)c(NC(C2CN(C(c3ccc(C)s3)=O)CCN2)=O)cn1 C(C(C)(C)C(C)(C)C)NC(C(C)(C1CCCC1)NC(CC(=O)N(C)C)=O)=O c1(C(=O)NCCC(C)NC(c2c(COC)cccn2)=O)oc2ccccc2c1C Cn1nnnc1SC1(C(=O)NCC#CCNC(=O)COC2CCC2)CC1 c1(C(CNC(C(CC=C)NC(=O)OC(C)(C)C)=O)OC)ccc(OC)nc1C CCCCC(CC)C(=O)NCCCOCCN(C)C(C1CSCCS1)=O C(CS(=O)(=O)CC(=O)N1CCN(C(c2cnn(C)c2)=O)CC1C1CCCC1)OC c1(C(=O)NC(C2(CNC(c3ccnn3C)=O)CC2)C)cc(Cl)cc(F)c1N c1(C(=O)NC2CC(C)N(C(c3cncn3C)=O)C2)cc2c(Cl)cccc2s1 N1(C(C(C)OC)=O)CCC2(CC1)CN(C(c1cc3c(ncn3C)[nH]1)=O)CC(C)O2 C#Cc1ccc(Cl)c(CNC2N(C(=O)OC(C)(C)C)CC2(C)C)c1 Cc1cc(F)ncc1C(=O)NC(C1CCN(C(=O)CCc2cccs2)C1)C c1(C(C)C)sc(Cl)nc1C(N1CCN(CCNC(=O)C(C2CCC2)OC)CC1)=O C(C(F)(F)C(F)(F)F)OCCC(=O)NCC(C1CCCC1)NC(C(CC)SC)=O Cc1cc(Cl)cc(N)c1C(=O)NC1CN(C(=O)CCN2CCCC2)C(C)(C)C1 C1(NC(=O)CC(O)C2CC2)CC2CN(C(=O)CCCCC3CC3)CC12 Cc1ccc(CC(C)NC(=O)NC(c2cc(C)ncn2)C)nc1 c1(C(N2CCC(C)C(NC(C3(F)CCCC3)=O)C2)=O)cc2ccccc2o1 C(CNC(C1CC1c1cccs1)=O)(CO)(CO)N(C)C(c1c[nH]c(C(N)=O)c1)=O C1(C(=O)NC(C(=O)NOCc2ccccc2)C2CCCC2)CCn2nncc2C1 C1(NC(C(C)CF)=O)CCCCC12CCN(C(c1ccc3c(c1)C(=O)NC3)=O)C2 C1(CN(C(C=CC)=O)C)CN(C(c2cccc(C3CC3)c2)=O)CCO1 Cc1cccc(Br)c1OCC(N1CCC(=CC(=O)Nc2cccnc2Cl)CC1)=O C1(CNC(c2ccc(F)s2)=O)CC2(CCN(C(c3cc[nH]c3C3CCC3)=O)C2)CO1 C1(NC(c2c(OC)c(C)cs2)=O)C2CC1CN(C(C1(C)CCCO1)=O)C2 C(=O)(C1CCCn2cncc21)N1CCCCC(N(C(=O)C2=C(Cl)CC2)C)C1 c1(NC(C)(C)C)c(O)ncc2c1CCC2.c1(N2CC(C)COC2=O)ccccc1 C1(NC(Cc2ccc(C)nc2Cl)=O)CN(C(=O)Cc2ccsc2)CCC1(C)C c1(C(=O)NC(CC)CNC(c2cnsn2)=O)ccn(C)c1C1CCC1 Cc1ccnnc1CC(c1nnnn1C1CCC1)NC(C1(c2ccon2)CC1)=O N1(CC=O)CCCC(OCCCC2(O)CC2)C1.C(CCF)O c1(C(=O)NCCN(CCC)CC)cc([N+](=O)[O-])c[nH]1.N12CCN(CC1)CC2 c1(C(N2CCC(NC(C(CCC)O)=O)C2)=O)ccc2cc(C(C)C)ccc2c1 CCCCC(O)C(=O)NCC(C)NC(=O)C(C)(C)COC(C)(C)C C1(NC(c2n(C(C)C)ncn2)=O)CC2CN(C(=O)C(C)(C)C#N)CC2C1 c1(OC)ccc(Cl)c(C(=O)NCCC2CCN(C(=O)C3=COCC3)C(C)C2)c1 c1(C(=O)NCC(CNC(CCCOC)=O)F)c[nH]c2cccnc12 c1(C(=O)NCC(=O)NCCN(C(c2ccncc2)=O)CC)cc(C)n(C)c1 c1(NCc2ccc(C)cc2F)ccc(S(=O)(=O)NCC2CCC(C(N)=O)O2)cc1Cl Cc1cc(C(=O)NC(C2CN(C(=O)CC3CC4(CC4)C3)C2)C)ccc1N n1(CC(=O)OC)cnc(C)c1C(=O)NC(CNC(C1(O)CC1)=O)CCOC CCCC(C(O)C(=O)NCc1cncc(F)c1)NC(=O)C(C)CCOC C(=O)(C(O)C(C)C)NCCOCCNC(c1n(CCC)ccc1)=O N1(C(CCNC(C)=O)=O)CCC(C(N2CCN(C(C)(C)C)CC2)=O)C(O)C1 CC(CO)(CO)C(=O)NC1CN(C(C2(C)CCC2)=O)CC1F O=C1OCc2c(CC(=O)N(C(C3CCCCC3)C(=O)O)C3CC3)cccc21 N1(Cc2ncc(C)o2)CCCC(C)C1C(C)NC(C1COC(C)(C)OC1)=O CN1CCOCC1C(=O)NC1(CC(=O)NC2(C(N)=O)CC2)CCC1 CC(C)CCCCCC(=O)N1CCCC(F)(C(=O)NC(C)CN2CCCC2=O)C1 c1(C(N2CCC(COC)(NC(=O)CCC3CCCO3)C2)=O)ccc(Cl)c(C)c1N CCC(O)C(F)(F)C(=O)NC1CCN(C(=O)CCC=Cc2ccccc2)C(C)C1 c1(OC)ccncc1CNC(=O)C(CC1(C#N)CCC1)NC(=O)CN1CCCC1 C1(F)(CNC(=O)C(C2CCCCC2)O)COCCN(C(C2(CO)CCCC2)=O)C1 c1(C(=O)NCC(C)CNC(c2cc(Cl)ccn2)=O)cc(O)nc2c1CCCC2 C(=O)(C(CCC1CC1)NC(c1ccc(C)nn1)=O)NCCCC C1(C(=O)NCC(C)O)COCCN(CC(O)CN2CCOCC2)C1 CC1(C)OC(=O)CC1C(N1CCOC(CC(=O)NOCCC2CC2)C1)=O c1(C(N2CC(OCCNC(C(C(C)C)C)=O)C2)=O)cc2cccnn2n1 C1(CNC(COC2CN(C(C=CC=CCC)=O)C2)=O)COC2(CCC2)C1 c1(C(=O)NCC2CCN(C(c3ccc(SC)cc3)=O)C2)cccc2c(C)[nH]nc12 N1(C(c2ccc(OC)s2)=O)CCOCC(c2cn(-c3cc(C)ccc3C)nn2)C1 Cc1cnc2c(C(=O)NCC(C)NC(C3Cc4cc(F)ccc4O3)=O)cnn2c1 C=CCC(CC(=O)N1CCCC1CCCC)NC(C1(OC)CC1)=O C(=O)(C(CC(C)C)CC(C)C)N(CCCCCNC(Cc1ncc(C)o1)=O)C Cc1c(C(N2CC(C)(NC(c3coc4c3COC4)=O)C2)=O)oc2ccc(Cl)cc12 c1(C(=O)NCC(CNC(CCCCOC)=O)O)ccc(=O)n(CCO)c1 C1(C(=O)NC(CNC(c2c(C(C)C)[nH]cc2)=O)C)CC2(C1)CC1(CC1)C2 C(=O)(C1=NOC(C)C1)NC(C(=O)NCC1ON=C(CC)C1)Cc1ccoc1 N1(CC(=O)N(CC(c2cscc2C(F)(F)F)=O)CC(=O)O)CCc2ccccc21 S(=O)(=O)(c1[nH]c(=NCC2(C)SCCCS2)ccc1Br)N1C2CC(OC)CC1CC2 C(=O)(C1CCc2ccc(Cl)nc21)NCCN(C(C1=C(C)OCC1)=O)C Cc1sc(O)nc1C(=O)NC1CCN(C(c2cncn2C)=O)C1c1ccccc1 Cn1cc2c(C(=O)NCC3C4CN(C(c5nscc5N)=O)CC34)cccc2n1 c1(C(N2CC(NCc3cc(OC)cc(O)c3)C(C)C2)=O)cc(Cl)cc(Cl)c1O C1(NC(c2c(CC)ocn2)=O)CC(C)CN(C(=O)C(C)N(C(C2CCCO2)=O)CC)C1 C(c1cccnc1)=CC(=O)NCC(C)(C)NC(C(n1ncc(C)c1)C)=O c1(C(=O)NCCCCCN(C)C(c2cc3ccsc3s2)=O)cccc2nonc12 C1(C(=O)NCCCOC(C)=O)CC2C=CC1N(C(c1cc(F)ccc1C)=O)C2 c1(OC)c(F)ccc(NNC(=O)OCc2nnc(C(F)(F)F)s2)c1F C1(CN(C(=O)C(C)(C)C2CCN(C(=O)Cn3cncn3)C2)C)CCCNC1=O CC1(C(=O)OC)CCCN(CC(C2CCC(C(N)=O)O2)=O)C1 C#Cc1cc(C(=O)NCC(CO)NC(c2ccc(O)nc2)=O)cc(F)c1 N1(C(C2C(COC)C2)=O)CCC(NC(c2cc(C3CCC3)cnc2F)=O)C(F)C1 CC(C)CCC(O)C(=O)NCC12CCC(NC(=O)CC3SC(=N)NC3=O)(CO1)C2 N1(C(c2c(CC)occ2)=O)CCC12CN(C(c1csc(S)n1)=O)C2 N1(C(=O)C(N2CCCc3[nH]ccc3C2)=O)CC(O)CC2CCCCC12 C1(NC(CC2C=CC(NC(C3CCC(C)O3)=O)C2)=O)CCOCC1(C)C O=C(N1CC2COCC2O1)c1ccc2c(Br)[nH]nc2n1 c1(C(=O)NCCC2OCCCN(C(CC(C)C)=O)C2)cnc2cnccc2c1 C1(NC(c2cccc(C(C)C)c2)=O)CCN(C(=O)C(F)CC2CCC2)C1(C)C Cc1cc2ccc(C(=O)NC3CC(C)(NC(c4ccc(F)cc4)=O)C3)cc2[nH]1 c1(NC(C2C(NC(=O)C3=CCC3)C2)=O)cc(-c2cccc(Cl)c2)ncn1 c1(C(=O)NCC(C2(O)CCN(C(CCC)=O)C2)C)cc2c(s1)CCC2 c1(OC)ccc(Cl)c(C(=O)N(C2CCN(C(=O)CN(C)S(N)(=O)=O)C2)C)n1 CCC(CC(C)C)C(=O)N1CCC(CN(c2nccc(C#N)n2)C)C1 c1(C(=O)NC2(C)CN(C(C3CCCC(N(C)C)C3)=O)C2)cnc2cccnn12 n1(CC(=O)NCC2CN(C(C3C4COCC34)=O)CCO2)cnc2sccc2c1=O C1(C(N(CCCOCCN(C)C(C2CC2C(C)(C)C)=O)C)=O)CC=CC1 C1(CC(=O)NC(c2ccccc2NC2CC2)=O)CCCN(S(=O)(=O)C2CC2)C1 CC1CN(C(=O)C(C2CC2)N(C)C)CCN1Cc1cn(C)ccc1=O c1(C(C(=O)NCCC)N(C(CC#C)C)C)cc(Cl)sc1Cl N1(C(CCNC(N)=O)=O)CCN(C(=O)CC(F)(F)Cl)CC1CC1CC1 C#Cc1cc(C(N2CCC2CNC(=O)CN2CCCS2(=O)=O)=O)ccc1C C1(C2CCN(C(C3CC4(CCCO4)C3)=O)C2)(NC(=O)CC2(CO)CC2)CC1 c1(N2CC(C)=C(C)C2)nc(N2CCCC(C(N)=O)C2)nc2cccnc12 CC1CCC(C(=O)NCC=CCl)CN1C(=O)Cc1cccnc1O C1(NC(C2CSCCS2)=O)CN(C(c2ncncc2Cl)=O)CCC1F C(=O)(C(CC(C)(C)C)NCCNC(=O)COC)N1CC(CC(C#C)C)C1 N1(C(c2cc(OCC)n(C)n2)=O)CC2CC1CCN2C(=O)CC1=CCCCC1 C1(C)(CC)C=C(C(=O)N(CCNC(c2ccc[n+]([O-])c2)=O)C2CC2)C1 C1(C(N2CCN(C(C(C)=CC)=O)C(CC(F)(F)F)C2)=O)CC2(C1)NC(=O)NC2=O Cc1cc(NC(=O)C(C)N(C(=O)CCC(C)(F)F)C)cc(C)c1F C1(C(C)NC(=O)C(C#N)C2CC2)CCCCN1C(c1ccc(C(F)(F)F)cc1)=O N1(C(c2cn(CC=C)nn2)=O)CCCCC(CNC(c2cc(Cl)ccc2C)=O)C1 C(C(COC)C(=O)N(CC(c1ccccc1)O)C)NC(C1(C(=O)OC)CC1)=O C1(NC(C2(CCC)CC2)=O)CCCC(NC(c2ccccc2SCCO)=O)C1 C(=O)(CC(F)(F)C(F)F)NCC12CCC(NC(CC(C)n3ccnc3)=O)(CC1)C2 C1(NC(C2(CC)CC2)=O)CCCCCN(C(c2cc(F)c(Br)cc2N)=O)C1 c1(N2CCN(C(c3n(OC)cnc3C)=O)CC2)cc(F)cc2c(Br)ccnc12 c1(C(N2CC(NC(CC3(C)CCC3)=O)C2)=O)cccn2nncc12 [SH](=O)(=O)c1ccc(F)cc1Cl.CN1CCN(C2CCNC2=O)CC1(C)C c1(NC(C)=O)cnc2ccc(NC(=O)C(N3CCC4(C3)CNC4(C)C)=O)cn12 S(=O)(=O)(c1cc(Cl)c(F)cc1F)N1CC(C)C(C(=O)O)C1C N1(C(Cc2c(C)ocn2)=O)CC2CCCC2(CNC(=O)CSc2cccs2)C1 CCCC(O)C(=O)N1CC(C(=O)NC2CCOC2C)(COC)C1 c1(C(N2C(CCCNC(c3c(C)cn(C)c3)=O)CCC2)=O)cc(O)ccc1N c1(CN(C)C(c2csc(-c3cnn(C)c3)n2)=O)ccc2c(c1)OCCO2 c1(CC)cc(C(=O)N(C2CN(C(C3CC34CCOC4)=O)C2)C)sc1C C(=O)(N=c1ccn(C2CC2)[nH]1)C1C(=O)N1.c1(C(=O)O)[nH]nnc1CO CN(C)NC(=O)CCC(=O)N1CCC2CN(C(=O)CC3CCC(O)C3)CC2C1 N1(C(c2c(OC)csc2)=O)CCN(C)C(CNC(=O)C=Cc2cc(OC)ns2)C1 C(N=c1[nH]cnc(C)c1OC)C1CCC(NC(c2ccc(OC)cc2)=O)C1 C(c1ccccc1Cl)=CC(=O)NC1CC2CC1N(C(=O)CNc1nccs1)C2 c1(C(N(CCC(F)(F)F)CC(=O)O)=O)ncn2c1CCC2 N1(C(C(=O)NC(C)C)=O)CC(C)(C)OCC1CNC(c1ccc(F)c(F)c1F)=O N1(C(c2cccc(-c3cn4ccccc4n3)c2)=O)CCN2CCOCC2C1 N12CCOC(C)C1C2=O.CCCC(C(=O)NCc1nocc1C)OCC c1(CC(=O)NC2CN(C(CCOCC)=O)C2)ccc(F)cc1F n1(CC)ncc(C(=O)Nc2ccsc2Cl)c1C1CC1.C12CC(C1)CNC2=O c1cc(C2CCOCC2)c2c(c1)CCN(N1CCOCC1C1CC1)C2 c1(C(C(C)CN(C)C(=O)NCCS(C)(=O)=O)C)ccc(OCCCC)cc1.C=CCO N1(C(=O)Cc2ccnn2C2CCOCC2)CCN(C(=O)C=CCF)C(CO)C1 C(=O)(C1=CC2CCC(C1)C2)N1C(CO)CC(OC)C1.C12CC(C1)NC(=O)CO2 N1(C(C(=O)NC(CC)=O)C)CC2CC(NC(c3ncccn3)=O)CC1C2 c1(C(N2CC(CC3(O)CC(NC(C4(CC)CCCC4)=O)C3)C2)=O)ccc[n+]([O-])c1 CC(CC(=O)N(CC(O)CN(C(=O)Cc1ccc(O)c(F)c1)C)C)C(F)(F)F C1(CNC(C2C(=C)CC2)=O)CCCCN1C(c1cccs1)=O C#CCCCCCNC(=O)CC1(C)CCN(C(=O)C(C)(C)N(C)C)C1 C12(C(N3CC(NC(CC4(C)CCCCC4)=O)(CF)C3)=O)CCC(C1)C2(C)C C1(CC(=O)NCC(C)CNC(=O)C(C)(C)n2ccnn2)COCC(C)O1 Cc1cccc(SCC(N2CC(C3CCCCN3C(=O)CC3CCOC3)C2)=O)c1 N1(C(c2c(OC)csc2)=O)CCN(C(c2cc(CO)n(C)n2)=O)C(C(C)C)C1 c1(CNC(C(C)N(C(C2CC23CCOCC3)=O)C2CC2)=O)cccc(F)c1O C(=O)(C1=CC2CC=CCC12)NC1(C)CCN(C(c2cc(OC)n[nH]2)=O)CC1 C#Cc1ccc(F)cc1C(=O)NCC1CN(C(C2(SC)CCC2)=O)CCCO1 C(=O)(CCC(F)(F)C(F)F)NC(CNC(CNC(c1ccc(C)cc1)=O)=O)(C)C C(=O)(CCC(=O)OC=O)N(C1CCN(CCCO)CC1)CC.C1(N)CCS(=O)(=O)C1 C1(C(=O)NCC2OCCN(C(c3cccc(SC)n3)=O)C2)CCCCNC1=O N1(C(CCN(C(C)C)C(c2ccc(CO)cn2)=O)=O)C2CCC1COC2 C1(NC(=O)CC2COCCN2C(=O)Cc2cccnc2)CC(O)C(O)C1O N1(C(c2ccc(OC)nn2)=O)CCC12CN(C(c1cc(Cl)c(C)cn1)=O)C2 C1(CNC(c2n(C(C)(C)C)nnn2)c2cscc2Cl)(CO)CCCCCC1 Cc1cc(Cl)ncc1CC(=O)N(C1CCN(C(C2CSCC(=O)N2)=O)C1)C C(=O)(C(C)C(C)(C)C)NC1(CCNC(C2C(C)COCC2)=O)CC1 c1(CC(=O)NCCOCCCNC(C(C)NCCCCCC)=O)ccccc1C c1(CC(=O)NCC2CC(O)(CNC(C(C)=C3CCC3)=O)C2)cc(C)cc(F)c1 N1(C(c2c(CCCC)ccs2)C(=O)NC)CCSCC1(C)C c1(OC)c(C(N2CC(CNC(=O)C(C)(C)C#N)C(C)C2)=O)oc2ccccc12 N1(C(C2(C=C)CCN(C(C3CCC(OC)CC3)=O)C2)=O)CCN(C)CC(O)C1 C1(CC(N2CCC(N(CC#C)C(C3(C)CC3(F)F)=O)CC2)=O)CCOCC1(C)C c1(C(C(=O)NCC(C)CC)N(CCCC)CC2CC2)ncnn1CCF N1(C(c2c(CC)ccs2)=O)CCC(C)(CCNC(=O)CC(C)C2CCCC2)CC1 C1(O)(CC#C)CCN(C(=O)CCCC(C)NC(c2cnc[nH]c2=N)=O)CC1 C(=O)(C(F)(F)C(O)C1CC1)NC1CC(N(C(c2ncn(CC)c2)=O)C)C1 C1(C(=O)NC(CCCCC)C2CC2)N(C(C23CCCC2C3(F)F)=O)CCC1(C)C CCCCC(CC(=O)NC1CN2CCC1(C)CC2)NC(=O)C(c1cnn(C)c1)O c1(C(=O)NC(C2CN(C(=O)C=CC(F)(F)F)C2)C)snnc1C1CCC1 CC(C(C)(C)C)=CC(=O)NCC(O)CN(C)C(c1cc(C2CC2)sn1)=O C(CC)(C(=O)NCCCCc1cnc[nH]1)N(C(C(C)NC(CC)=O)=O)C c1(C(=O)NCCC(CC)(C)NC(c2ccc(CO)s2)=O)cc(F)ccc1O CCC(O)C(F)(F)C(=O)N1CC=C(C(=O)NCc2ccc(CO)cc2)CC1 c1(C(N(CCNC(c2cc(C)c(O)nn2)=O)C)=O)cc2ccc(F)cc2s1 C1(C(=O)NCC2C(NC(c3cn(C(C)(C)C)nn3)=O)CCC2)CC2(C1)CC2(F)F C1(CNC(C(C=C)(F)F)=O)CC2CCCC2N1C(=O)Cc1cncnc1 C1(OC)CC(NC(=O)OC(C)(C)C)N(C(=O)NCC(c2nc(C)cs2)C)C1 N1(C(C2(C#C)CCCC2)=O)CCN(C(=O)CC2(CO)CC2)C(COC)C1 CC#CCC(C(=O)NC1CCCC(C)C1)NC(=O)C=CC(C)CC c1(C(=O)NC2CCC(NC(c3cnnn3C3CC3)=O)C2)noc2ccc(Cl)cc12 C1(C(=O)NCC2CCN(C(=O)C(c3ccc(F)cc3)F)C2)CCc2nn[nH]c2C1 C1(CCC)CN(c2cc(N3CCC(c4ccc(F)cc4)C3)ncn2)CCO1 n1(CC(=O)NC(CN(C(=O)C(C(C)(C)C)SC)CC)C)cnc2ccsc2c1=O c1(CC)[nH]c(=N)sc1C(N1CCC(N(C)C(c2c[nH]nc2C)=O)C1)=O c1(C(N(C2CCCC(NC(c3cc(O)cc(=O)o3)=O)C2)C)=O)cn(C)ccc1=O C1(N(C(=O)CC2C=CCC2)CC#C)CCN(C(C2CC(n3cnnc3)C2)=O)CC1 C1(NC(C(C)SC(C)C)=O)C2CCCN(C(c3ccns3)=O)C2C1(C)C C(=O)(C(CCC)OCC)NCCCCNC(C1(C=C)CCC1)=O C(C(C)(O)C(=O)NCCC1CCCN(C(=O)CC2CC(C)=NO2)C1)OC c1(NC(C2C3CN(Cc4c(C)c(Br)cnc4)C2C3)=O)cc(C#N)ccc1F c1(C(=O)NC2C(NC(C=CC(CC)C)=O)C2)cccc(OCc2cccs2)c1 N1(C(CNC(=O)OC)=O)CCC(N(C)C(c2ccnc(OC)n2)=O)C(C)C1 C(N=C(NCCN(C)C)N1CCC(C2CCOC2)C1)c1c(C)cc(Br)nc1 N1(C(CC2CC(C)C2)=O)CCN(C(=O)CN(C)C2CC2)C(=CC2CCCC2)C1 C(CC(C(=O)NC)NC(=O)CCOC(=O)NCC(C(C)CC)N(C)C)OC N1(C(C2CC3CC2C2CC32)=O)CCCC(C2CCN(c3ncc4ncnc-4[nH]3)C2)C1 C12(NC(c3c(CC)scc3)=O)CCCCC1N(C(=O)C(C)(F)F)CC2 n1(C(=O)NC(c2ccccc2)C(C)NC(=O)CC(C)(C)C)nnc2c1CCCC2 C(CC(O)C(=O)NCC(O)CCNC(=O)CN1CCCNC1=O)N(C)C CC(C)CN(Cc1cccs1)N(C)Cc1ccc(C(F)(F)F)c(F)c1 C1(CCOC)CN(C(c2cnco2)=O)CCN1C(=O)C(COCC(F)(F)F)OC CCCC(C(=O)N1CCOC(c2cn(-c3ncc(Cl)s3)nn2)C1)NC.C1(O)CC1 N1(C(C(CC(=O)OCC)C)=O)CCC2(CCC(NC(=O)CSCC(C)C)C2)CC1 Cc1cn2ccnc(C(N3CC(NC(=O)C(F)CC4CCCC4)C(F)C3)=O)c2n1 C1(C)(C(=O)NC2CC(CNC(C(CCC)OC)=O)C2)COC(C)(C)OC1 c1(C(=O)NCC2(O)CN(C(c3nocc3C3CC3)=O)C2)cccc2sccc12 N1(C(CSc2ccc(NC(CCCC#N)=O)cc2)=O)C2CCC1CN(C(N)=O)C2 N(C(=NCCCOC1CC(F)(F)C1)NCCN1CCCCC1)N1C(C)(C)CCC1 Cc1ccn(CC(C)(O)C(=O)N2CC=CC(NC(=O)COC3CCC3)C2)c(=O)c1 C1(NC(=O)OC)CC2CC1CC2NC(CO)C(N)=O Cc1ccc(Cl)cc1OCCCC(=O)NCC(C)CN(C)C(C12CCC1C2)=O C#Cc1ccc(C(=O)NC2(COC)CCCN(C(=O)CCC(=O)C3CC3)C2)nc1 c1(CC)cnccc1C#N.C12(C(=O)NCCCC3CCCC3O)CCCN1C2=O c1(C(=O)NC(C2CCCC2)CNC(C(C2CCC2)OCC)=O)cscc1C(N)=O C1(C(N2CC(CCNC(=O)C(C)CSC)(OC)C2)=O)COCC1(C)C N1(C(CC2(NC(C)=O)CC2)=O)CCC(NC(=O)C(C)(F)C(C)(C)F)C(CO)CC1 N1(C(CCCCCSC)=O)CC(=O)N2CCOCC2(CNC(C2CCCS2)=O)C1 C(C#Cc1cn(CC(F)(F)CN(C)C)nn1)NC(C(C)P(C)(C)=O)=O N1(C(C(F)OC)=O)CC(NC(c2ccccc2O)=O)C(C(F)F)C1 C(C)(C)(CCCC(=O)NC(CN(C)C)C(C)(C)C)NC(C1CCC(OC)CC1)=O c1(OCC(=O)NC2C(n3cc(C(C)(O)C(=O)O)nn3)COC2)ccccc1F C1(NC(CCCc2ccc(C)s2)=O)CCCN(C(c2c[nH]cc2C(F)(F)F)=O)C1 C1(CC)CCC(C(=O)OC)CN1C(c1cc(OC)ccc1OC(C)C(C)C)=O c1(NCC(N2CC(NC(c3c(F)cncc3Cl)=O)C2)=O)ccccc1[N+](=O)[O-] c1(CC(=O)Nc2ccc(NC(C3(COC)CC=CC3)=O)cc2)cc(C)ccc1C C1(C(=O)NCC(C)(C)NC(c2ccc(CO)o2)=O)(C(F)F)CCCO1 C1(CNC(C(n2c(C)ccn2)C)=O)CN(C(C2(CO)CCCCO2)=O)CCO1 c1(NC(c2cn(CC)nc2)=O)cc(NC2CN(S(C)(=O)=O)C2)cc(Br)c1 CC1(C)CC(CNC(c2cccnc2CO)=O)CN1C(=O)Cn1ncccc1=O c1(CN(C(=O)C(O)C2CCC2)CCCNC(C2CC2(Cl)Cl)=O)ccccc1 c1(C(=O)NCCC(C)NC(C2CC2C(F)(F)F)=O)cc(F)cc(S(N)(=O)=O)c1 C1(NC(=O)C=CCOCc2ccccc2)CCN(C(C2(C3CC3)CC2)=O)CC1 c1(CC)sc(C(N2CCC(C(C)NC(=O)CS(=O)CC)CC2)=O)cc1C N1(C(CC(CCCC)O)=O)CCC(C(=O)NCCC2CCC(=O)CC2)=C(F)C1 c1(C(=O)NCC2(NC(c3ncc(Cl)s3)=O)CCOC2)ccc(O)cc1 N1(C(CC(C)CC(C)(C)C)=O)CCC2(CCCC2NC(=O)CCC(Cl)Br)CC1 c1(-c2cn(CCCCNC(CC=C=C)=O)nn2)cc(Cl)cc2ccccc12 N1(C(c2n(C(CC)C)ncc2)=O)CC2CCC1C(CNC(=O)C=CC=C(Cl)Cl)C2 C1(C(=O)OCC)CN(C(=O)C(=O)NCCOCCC(N)=O)CC12CCC2 c1(NC(C2N(C(c3cc(OC)c(F)cc3)=O)CC(F)C2)=O)ccc(Cl)c(F)c1I C(=O)(C(CC(C)C)NC(c1cnn(C(C)C)c1)(CC)c1nnnn1C)OCC N1(C(c2occ(C)c2)=O)CCC(NC(=O)Cn2nc(C)oc2=O)C2(CCC2)C1 N1(C(C2CC3CC3C2)=O)CCCCCC1CNC(COCc1nnc(C)s1)=O c12ccc(=O)n(c1)C1(CC1)COC2=O.CCCC(F)C(=O)OC N(C(=NCC(C)C)NCC1CC(=O)N(c2ccccc2)C1=O)CC1C(C=C)C1 c1(C(=O)NC2CC(NC(c3scc(C)c3)=O)C2)ccc(-n2cncn2)nc1 Cc1cc(C)c(NC(=O)CC(c2cccs2)NCc2cc(F)cc(I)c2)cc1C N1(C(C(=O)NCC)=O)C2CN(c3ncc(C(=O)OC)cn3)CC12 C12(CNC(C3(CC#C)CC3)=O)CC(NC(C3CCCN3C3CCC3)=O)(CO1)C2 C(C(=O)OC)(C(C)(C)C)c1scc(C)n1.c1(NC(=O)NCCC)c(C)c[nH]c1CC(N)=O c1(OC)ccc(C(N2CCCC(NC(C3CC(=C(F)F)C3)=O)C2)=O)cc1Cl C1(NC(C(CCC)F)=O)CC(CNC(C2CC(OC3CC3)C2)=O)C12CCC2 n1(CC)nc(C2CC2)cc1N1CC(C(N)=O)C1.C(=O)C(C)(C)C N1(C(C=C(CC)C)=O)CCC(C2(NC(=O)CN3CCS(=O)CC3)CC2)C1 N1(C(C=C(CC)C)=O)CC2CCC(NC(=O)C(F)(F)C(C)O)CC2C1 c1(N)ccc2ncccc2c1.Cc1nc(CCC(=O)N)cs1.C12CC1CNC2=O c1(C(=O)NCCN(C(=O)CCc2cnn(-c3ccccc3)c2)CC)ccncc1 C(CC(O)C(F)(F)F)NC(CCN(C(C(COCC)C)=O)CCCO)=O C(=O)(C(O)(C(F)(F)F)C1CC1)N1CCCCC(NC(c2cc(C)c(F)cn2)=O)C1 C(=O)(C1=C(C)CCOC1)NC1C(NC(CCN(C)CC)=O)COCC1 N1(CC(=O)OC(C)(C)C)CCC(CC(N)=O)C(NC(c2cnn3c2OCC3)=O)C1 C1(CNC(c2cncc(O)c2)=O)COCCN(C(C2CCC(N(C)C)CC2)=O)C1 N1(C(CC2ON=C(C)C2)=O)CCCC1(C)CNC(=O)COCC(C)(C)C N1(C(c2c(C)n(C3CCC3)nc2)=O)CCCN(C(C2CC(C)(F)C2)=O)C(C)C1 c1(CC)ncnc(CC)c1.N1(C(=O)C=CC(F)(F)F)CCOC(CCCOC)C1 C=CCC(C)(C)CC(=O)N1CCC(CC)C1CNC(C1CC(C)(O)C1)=O N1(CC)CCC(N(C(=O)C(CCOCCO)NC(=O)Cc2csnc2C)C)CC1 C#CCC(CC#C)C(=O)N1CCC(CF)(NC(=O)Cn2nnnc2C(C)C)C1 C1(CC=C)(NC(=O)C(F)OC(F)(F)F)CCN(C(c2cc(C)c[nH]2)=O)C1 C(=O)(CC(C)(C)CC(F)(F)F)N1C(CO)CC(Cn2cc(C(=O)OC)nn2)C1 C(=O)(C1CCCc2n[nH]cc21)NC(CNC(c1n(C(C)C)nnc1)=O)(C)C1CC1 C(=O)(C(F)CCC(C)(C)C)NCC(CNC(c1ccc(C)cc1Br)=O)O N1(C(C2CC=C(C)CC2)=O)CC(C2CCCCN(C(c3sc(F)cc3C)=O)C2)C1 c1(C(=O)NCC#CCNC(C=CC)=O)ccc2cc(C(C)C)ccc2c1 c1(C(=O)NCC(C(C)C)NC(C2CCOC2)=O)cnn2c(C)cccc12 S(=O)(=O)(c1ccc(C)c(C(=O)O)c1)N1C(CC)C(C(=O)OC)CCC1 N1(C(C(C)NC(CC)=O)=O)C2CCC1CN(C(C1CN3CCN1CC3)=O)C2 n1(CCC(N2CC(COC)(NC(c3csnc3C)=O)C2)=O)nc(C2CC2)oc1=O C1(C(N2CCC(C(C)NC(c3c(C)scc3)=O)CC2)=O)CSc2ccccc2O1 C1(NC(COC(CC)(C)C)=O)CCCCC1N(C(=O)C(n1ccc(C)n1)C)CC C(C(=O)N1CCCO1)NC(C(C1CC(C#N)C1)NC(C1OC2CCC1C2)=O)=O C1(C(N2C(C3(OC)CC3)CCC2)=O)Cc2cccc(NC(C=C(CCC)C)=O)c2O1 O=S(=O)(c1ccc2nc(N3CCC(S(N)(=O)=O)C3)sc2c1)NC1CC1 c1(C(N(CC(O)CNC(=O)CCn2ccnn2)C)=O)ccc(C2CC2)s1 C12(C(=O)Nc3cc(CC)c(F)cc3)CCN(C(=O)C=CC3CC3)CCC1C2 C(=O)(CC(CCC)NC(C1(C)CCCOC1)=O)N1CC(C#CC)C1 C1(C(=O)NCC(CNC(CCCCOC)=O)C(F)(F)F)CCc2nc(C)cn2C1 CC1CN(C(=O)CCCS(N)(=O)=O)CC(C)N(C(=O)Cn2cnc(=N)[nH]2)C1 O=C(C(F)CC1CN(c2nc(C(F)(F)F)n[nH]2)C1)NCCCc1nn[nH]n1 C(=O)(CCCC(F)F)NC1CC(C(C)NC(=O)C(C)Cn2cccn2)C1 c1(C(N2CC3CC(NC(Cc4cc(C)ns4)=O)C3C2)=O)cnn2c(C)cccc12 c1(C(=O)NCC2CC(NC(C3(OC)CCCC3)=O)C2)cnc2occc2c1 C(=O)(CC(C)CC(F)(F)F)N(CC(C)NC(Cc1nnc(C)o1)=O)C c1(CNC(C)(CC(Cl)Cl)c2nnnn2C2CCCCC2)cccc2ccsc12 C1(C(N(CCN(C(c2n(CC(C)C)ncc2)=O)C(C)C)C)=O)CC2C=CC1CC2 C(C(=O)OC(C)(C)C)(C(=O)NC1CN(C(=O)Cc2cc(Cl)n(C)n2)CC1C)OC Cc1cnc(N)c(C(N2CC(CNC(=O)CCOCC(F)(F)F)CC2(C)C)=O)c1 c1(CNC(C(C(C)NC(CC(C)OCC)=O)C)=O)cccc(=O)n1C c1(NC(=O)NC2(c3cnc(NC(C)=O)s3)CC3(CCC3)C2)cccc(Cl)c1C C(C)(C)(CCCC(=O)N(C)CC1CC1)NC(C(COCC)C)=O Cc1cc(CC(=O)NC2CCN(C(C3(F)CCOC3)=O)CC2)ccc1CO c1(CC)ccc(CNC(C2(C)N(C(=O)NC(C(=O)OC)C3CC3)CC2)=O)cn1 N1(C(C(CC)CNC(=O)C=CCOC)=O)CCCOC(CC)C1 N1(C(=O)NC23C(C)OC(C)(C2)C3)CCOc2ccccc21 C1(C(=O)NC2(CCNC(CC(C)n3cccc3)=O)CCC2)COC2(CCC2)C1 C(=O)(C(C)(C)C1=CCN(C(=O)C=C2CCC2)C1)NCC1CCN(CCC)C1 c1(C2CN(C(C(N3C(C(N)=O)C(=O)NCC3)=O)=O)C2)cc([N+](=O)[O-])ccc1F O=C(NNc1c(F)ccc(F)c1Cl)c1cc(S(=O)(=O)N2CCOCC2)c[nH]1 C1(NC(CCCCOC)=O)CN(C(=O)CCc2cc(C)no2)C2CCCCC12 c1(C(N2CC(C)N(C(C3CCCC34CCC4)=O)CC2)=O)coc2c1C(O)CCC2 CC(C)C(CCCO)NC(=O)CC1(N(C)C(c2ccc[nH]2)=O)CC1 Cc1ccc2nc(C(=O)NC3CC(C)CN(C(=O)C(F)C4CCC4)C3)cn2c1 C1(CC#C)CCCCN1C(C1CCCN(C(=O)CC=CCC)C1)=O Fc1ccc(N=c2scc(-c3cnccn3)n2CC2CCC(F)C2)cc1 c1(C(N2CCN(C(C=C3CCC(C)C3)=O)CC(O)C2)=O)coc2c(F)cccc12 C(=O)(CN=c1cc(Cl)nc(C2CCCO2)[nH]1)NC1C(=C)COC1 C1(CCC)CCC(C(=O)NCC(C)CNC(=O)OC)CC1.C1CCC(=O)N1 N1(C(C2(C(F)(F)F)CC(=C)C2)=O)CC(NC(=O)C(CC)SC)C(C)C1 N1(C(c2cc(C(C)C)cc(C(F)(F)F)c2)=O)C2CCC1C(O)CCC2O C=CCC(C)(C(=O)NCC1CCC(NC(=O)Cn2cccc(O)c2=O)C1)N(C)C C1(CCC)CN(C(c2sc(O)nc2C)=O)CCN1C(c1cc(Cl)sc1C)=O C(CC(C(=O)NC1(C(=O)NC(C(N)=O)C2CCC2)CSC1)N(C)C)SC N1(C(C(COC)C)=O)CC2CC(NC(c3c(OC)cccc3OC)=O)C(C2)C1 CCC(CC)C(F)C(=O)N1CCC(C(C)(C)C(N2CC[Si](C)(C)C2)=O)C1 c1(C(=O)NC2CCCC(NC(CCn3ncc(C)c3)=O)C2)ccc2occc2n1 C(c1ccc(Oc2cccc(C)c2)o1)=CCN(CCOC)Cc1cccc(C)n1 C1(C(=O)NCCNC(c2ccccc2Cl)=O)CCC(CNc2ccccn2)CC1 c1(C(=O)NCC(CNC(C2CCN(C)C2=O)=O)O)cccc2c1CCCC2 c1(NC(C2(C)CC2Br)=O)ccccc1C(=O)OC.c1(S)ccccc1 c1(C(N(C(CC)C(=O)NCCC2(SC)CC2)C)=O)nccc(C(C)(F)F)n1 N1(C(c2ncc(CC)[nH]2)C(=O)NCC(F)F)C2CCCC1CC(N(C)C)C2 N1(C(COC(C)=O)=O)CCC2(CC1)CC2C(=O)Nc1cncc(Cl)c1 CCCCC(C(=O)N1CCN(C(=O)CSc2nnnn2C)CC1)N(C)C c1(-c2cn(CCCCCCNC(C3(CO)CCCC3)=O)nn2)ccc2nonc2c1 c1(CC(N2CCCC(N(C(C3(C=C)CC3)=O)C)C2)=O)ccc(C)c([N+](=O)[O-])c1 C(=O)(CCS(C)(=O)=O)NC1(c2ccccc2)CN(c2nccc(SC)n2)C1 c1(OCCCCC)cccc2c1OCCC2=O C(=O)(CC(O)CC(C)(C)C)N1CCCC(C)(NC(CCCC#CC)=O)C1 c1(CCN(C(C2CN(C)C(=O)C2)=O)CCO)n[nH]c2c1CCC2 c1(CC)ccc(C(=O)NC2(C)CC(NC(C3CCSC(C)C3)=O)C2)cc1 C(=O)(CCCS(N)(=O)=O)N1CCC(NC(Cc2n(C)nc(Cl)c2)=O)(CO)CC1 C1(OC)CC(CNC(c2csc(C(F)F)c2)=O)N(C(=O)CN2CCC(C)CC2)C1 c1(C(N(CCC(=O)N(C)CC2CC2C)CCC)=O)ccncc1O c1(SCC)ccccc1C(=O)NCC1COCC1NC(C1CCS1(=O)=O)=O Cc1[nH]nc2c(COC(=O)CC3CN(C(C)C)CC(C)O3)cccc12 c1(C(=O)N(C(C(CC)C)=O)CCC2CCCN2C)cnc([N+](=O)[O-])n1C C(=O)(CCCCC1CC1)N(C1CCN(C(C2CC23CC3(F)F)=O)C1)CCC CCC(O)(C(=O)NCC(CC)NC(c1ccn(CC)n1)=O)c1cccc(Cl)c1 Cn1cc(CNC(=O)C(C)(C)C2CCC2)c(O)nc1=O C(=O)(CCCC(=O)N1CC2(C(=O)Nc3c(C)cccc3Br)CC1CO2)OCC c1(N2CCC(CNC(=O)NCC(CO)OC)CC2)cc(O)nc(C)n1 n1(CC(=O)NCC2(NC(CCC3C(C)OCC3)=O)CCCC2)ncccc1=O N1(C(c2ncc(COC)s2)C(=O)NCCCC2CC2)CCCC(C(O)C(F)F)C1 C1(C(=O)NC2(CC=C)CCCC2)CN(C(c2cnn(C)c2C2CC2)=O)CC1OC c1(CNC(CN(C)CCO)=O)cc2c(cc1N)OCO2.C(C)(C)(C)O c1(CNC(c2c(Cl)cnn2C)=O)ccc(C2(C(=O)OC)CCCC2)cc1 c1(C(c2n(CC=C)nnn2)NCC2(CCCO)CC2)cc2ccccn2n1 N1(C(C2CCC(C(C)O)CC2)=O)CC2CC(NC(=O)C(C)NC(=O)C3CC3)C1C2 C#CC1(C(=O)NCC2(C)CCN(C(=O)CCc3cnccn3)CC2)CCOCC1 C(CNC(c1cn[nH]c1)=O)(CO)NC(=O)COCC1CCCO1 Cc1cc(Cl)cc(C)c1C(=O)NCC1C(C)CCCN1C(c1n[nH]c(C)c1Cl)=O N1(C(C(COCC)C)=O)CCN(C(c2csc(C(F)F)c2)=O)C(C)C1 C(=O)(C(C)C(O)CC(C)C)NCC(C(=O)NC(CCCC=C)C1CC1)OC CC1CN(C(=O)COc2ccccc2Cl)CCC1CNC(=O)CC(=O)N(C)C c1(NC(C23CC(NC(C=CC)=O)(C2)C3)=O)c(Cl)c(CC)nn1C c1(C(=O)NC2(CNC(CC3C(C)=NNC3=O)=O)CC2)cnc(=NCCF)[nH]c1 c1(OC)cc(CN2CCC(O)C(C(=O)NCCCS(C)(=O)=O)C2)ccc1I c1(C(N2C(CNC(c3c[nH]c4cnccc34)=O)CC2)=O)cc(F)c(F)c(Cl)c1F CC(C)(O)C(C(=O)NC1CCCC1C(C)(C)C)NC(=O)C(=O)NCC(F)F c1(CC(=O)NC2CC(NC(Cc3c(C(=O)OCC)ccs3)=O)C2)cn(C)nc1C C(CCCCC(=O)Nc1cc(F)cnc1O)N(C)CCO.C1CCCC(=O)N1 CCCCC(C(=O)NC1CC=CCC1C(=O)NCC(c1cnc[nH]1)C)N(C)C c1(NC(CC2(NC(c3ccc(Cl)s3)=O)CC2)=O)csc(Cl)n1 N#Cc1cccc(CN2CC3CC3(C(=O)NCCCN(C(COC)CO)C)C2)c1Cl c1(OCC(=O)NCC(CNC(C)=O)OC)ccccc1C(C)=O Cc1ccc(C(N2CC(NC(C3CC=CC3)=O)C(C3CC3)C2)=O)c2c1CCC2 C1(C#N)(OC)CC(C(N2CC(n3cc(C4CCCC(O)C4)nn3)C2)=O)C1 n1(CC)nc(C2CC2)cc1C(=O)NC1CC(NC(=O)C(C)OC2CC2)C1 C(=O)(C(C)CC(N)=O)NC(CNC(C1(C)ON=C(C)C1)=O)C1CC1 CC(CCNC(=O)CNC(=O)CN)n1ccnc1 c1(CNC2CC(NC(c3ccc(C)c(C#N)c3)=O)C2)ccc(S(N)(=O)=O)cc1 c1(C(N(CC(C(=O)NC(CC(C)C)(C)C)C)C)=O)cc2ccccc2[nH]1 N1(CCOC)CCC(CNC(c2cscc2SC(C)(C)C)=O)C1 C1(C(=O)NC2C=CCN(C(=O)CCC3CCCCC3)C2)CC12CCOCC2 c1(C(N(C(C)CN(C(=O)CN2CCCS2(=O)=O)C)C)=O)noc2c1CCCC2 N1(C(c2ccc(SCC)cc2)=O)CCC(C)(NC(c2ccc(Cl)o2)=O)CC1 c1(C(CC)NC(=O)C(N2CCCC2c2cnn(C)c2)=O)cnc2cc(C)nn2c1 C12(NC(=O)CCc3ccc(F)nc3)CCN(C(C3CCC3)=O)CCC1C2 C(C(CCC)C(=O)N(C(C)(C)C)C)NC(=O)Nc1cccn(CCCC)c1=O c12ccc(o1)C(=O)NC2.C1(Cl)(C(=O)OC)CC1C(=O)NC1CC1c1nc[nH]n1 N1(C(C(C)NC(C=C)=O)=O)CC2OCC(C(=O)NC)C2C1 Cc1cnc(C(N2CCN(C(c3nccc(Cl)c3F)=O)CC2C)=O)c(F)c1 C(=O)(CS(=O)(=O)C1CCCC1)C(C1CC2CN(c3ncnc4sccc34)CC12)=O CCCCN(C)N1CCCC(NC(N2CC(=O)NC(C)(C)C2)=O)C1 N1(C(c2n(C(CC)CC)nc(C)c2)=O)CCOC2CCN(C(C3CC3F)=O)CC12 C1(C(C)C)CN(C(c2ccccn2)=O)CCN1C(=O)C=Cc1csc(Br)c1 c1(N(C(C)CCNC(c2ccc(Cl)cn2)=O)C)cc(O)nc(O)n1 C1(C(=O)NCCOCC#C)CCCCCCN1C(c1conc1C(C)C)=O C1(C)(OC)CCCCCC1.C12(CCCC1)CCC(=O)C(=O)CO2.C(C(C#N)N)OCC C1(C(=O)N(CC(C)(C)NC(C2CC2C(N)=O)=O)C2CC2)CCCC12CCOCC2 N1(C(C(C)=C2CC2)=O)CCCC(C2CCN(C(C3(C4CCCO4)CCC3)=O)C2)C1 c1(C(N(CCN(C(C)C)C(C2CC(n3ccnn3)C2)=O)C)=O)cnccc1Cl c1(OC(=O)NCC2CC3CN(C(=O)OC(C)(C)C)CC32)ccc(CO)cc1F N1(C(C)=O)CCCC(c2nnnn2CCNc2cc(Cl)cc(Cl)c2)(N(C)C)C1 N1(C(CC(C)C)=O)CC(NC(c2nn(C)c(C(F)(F)F)c2Cl)=O)CCC1C Cc1ccc(OC(=O)CCc2cnccn2)cc1C.c12ccc(cc1)c(=O)[nH]2 C(C(=O)NCC1(C)NC(=O)NC1=O)(C(C)(C)O)NC(c1cc(OCC)n[nH]1)=O c1(C(N2CCC(F)(CNC(CCCCN(C)C)=O)C2)=O)nccc(Cl)c1Cl N1(C(c2ccc(OC)nn2)=O)CC(NC(c2nc(C)c(C)s2)=O)CC1(C)C c1(C(=O)NCCC(=O)NC(CNC(C(c2ccccn2)C)=O)(C)C)cncnc1 c1(C(N2CCC(C(C)C(=O)Nc3cncc(Cl)c3)CC2)=O)c(N)cccc1F n1(CCCC(=O)N(C2CCN(C(CC3CNC(=O)O3)=O)C2)CCO)ccccc1=O CC1(C)CN(CCC(Cl)(Cl)Cl)CC1NC(c1ccccc1)=O n1(COC(=O)CC2=CCCC2)cc(NC(=O)C(CC(F)F)OC)ccc1=O c1(C(=O)N(c2nnnn2C2CCOCC2)c2cnsc2)nnnn1CCCF C(=O)(C1=CCC(C)(C)CC1)NC1(CNC(c2c(C)n3c(s2)cnc3)=O)CCC1 c1(SC)cnn(C)c1C(=O)NCC12CC1CN(C(=O)CC1CN(C)C1)C2 S(=O)(=O)(c1ccc(NC2CCOC(C3CC3)C2)cc1Cl)NCC1(C)CSC1 C1(CC(=O)NCCC2CN(C(C)=O)CCO2)(CNC(C)=O)CCCCC1 N1(C(c2ccc(C(C)(C)C)o2)=O)CC(F)(F)CC1CNC(C1CCC=CO1)=O N1(Cc2cccc(CC)c2)CCC(O)C(C(=O)NC(CC#CC)C)C1 c1(NC(C23C(CN(C(c4ccnc(F)c4)=O)C2)C3)=O)cccn2ncnc12 c1(C(=O)NCCC2N(C(c3nc(C)oc3)=O)CCOC2)cccc2nnn(C)c12 C(=O)(C(O)CC(C)(C)C)N1CC(CCNC(c2c(C)snc2)=O)OCC1 C1(COC)(NC(=O)NC(C)C(=O)NC2(C)CSC2)CCCO1 N1(C(C(COC)O)=O)CCC2(NC(c3cncc(CO)c3)=O)CCCCC12 CC(C)(C)C(CC(=O)NC12CC(Nc3ncnc(Cl)c3[N+](=O)[O-])(C1)OC2C)C(F)F CC(CCCNC(c1cncs1)=O)NC(=O)C(c1ccccc1)NC(N)=O c1(CC(N2C(C)(CC(=O)NCCCNC(C)=O)CC2)=O)ncc(F)cc1F C(CCCCC(=O)NCC1CCC2(CCC2)O1)NC(C(CCC)C)=O N1(C(CC(C)NC(=O)CCC(N)=O)=O)CCC2(CCOC2)C1 C(=O)(C1=CC(C)(C)C1)N1CC(CNC(C2CCC(C(C)C)CC2)=O)C1 c1(OC)ccc2c(CC(=O)NC3(C(N4C(CO)CC5(CC5)C4)=O)CC3)coc2c1 c1(C2(ON)CCC2)cn(CC(=O)NC2CC(F)(CO)C2)nn1 CCCCCC(CC)(c1nnnn1CCC1(C)CC1)NC(COCC)CCO c1(CC)cc(Cl)ccc1C(=O)N(CCNC(=O)CC1CCC2CC12)CC c1(C(N(CC(C)NC(c2cncc(-c3ccoc3)c2)=O)C)=O)ccc(=O)oc1 N=c1nc2c(c[nH]1)CC(C(=O)NC1(CNC(c3cc4c([nH]3)CCCC4)=O)CC1)CC2 C12(C(N3CC(C(N)=O)(COC)C3)=O)CCC(CNC(C(CSC)O)=O)(CC1)CO2 O=[N+]([O-])c1cc(F)c(CNCCCOCC2CCOC2)c(F)c1 Cn1nc(CCNC(C2CCCN2c2ccc(Cl)cc2)=O)n(C)c1=O N=c1[nH]c(=NCCC2CC2C(F)(F)F)[nH]c(=NCCCc2c[nH]nc2C2CC2)[nH]1 C1(NC(C(c2ccnn2C)NC(c2cn(CCC)nc2)=O)=O)CC(C)(C)C1OC Cc1cc(=NC(=O)C2CCOC2NC(=O)N2OC3CCC2CC3)[nH]n1C c1(CC)cccc(NC(C2CCCN2C(c2ccc(C(C)O)cc2)=O)=O)c1 C1(N(C)CCNC(c2cc(Br)sn2)=O)CCCN(C(=O)N(C)C)C1 C=CC(C(F)(F)F)NC(=O)C(CCC1CCC1)NC(=O)CCCn1ccnc1 CC(=O)CCCC(=O)N1CCN(c2cc(O)nc(C)n2)C(c2ccccn2)C1 c1(C(N(CC(CC)NC(c2ccc(C(N)=O)o2)=O)C)=O)ccc2occc2c1 O=C(CCC(=O)c1cccnc1)NCCC1CCC(NC(c2csc(S)n2)=O)C1 N1(C(c2ccc(F)c(C)c2)C(=O)NC)CC2(CNC(=O)C2)C1 S(=O)(=O)(c1ccc(Br)cc1NC1C(n2cccn2)C1)N1CCCC(CCC=C)C1 C(=O)(C1=CCCN(C(c2cccc(C#N)c2F)=O)C1)Nc1cc(OC)cc(F)c1 c1(CC(N2CC(C)(C)C(CO)CC2)=O)cccc2ncccc12 Cc1nc2ncccn2c1C(=O)Nc1nccc(Cl)c1Cl C(=O)(C#CC1CCCCC1)N1CC(C)(CNC(C2CSCC(=O)N2)=O)OCC1 C1(CC)C(C(N2CC(c3ccn(C)n3)C2)=O)CCCN1C(=O)C=CC1CC1 C1(NC(c2c(OCC)cccc2)=O)CC2CC(NC(=O)C=C(C)C(C)(C)C)C2C1 c1(NC(CC2C(NC(C(C)OCCOC)=O)CC2O)=O)cc(C)c(F)cc1O C(=O)(C1CCOc2ccccc21)N1CC(CC)(NC(=O)CCc2cnoc2)C1 C(=O)(C1SCc2cccnc21)NCC1(CCNC(C(C(C)C)(C)C)=O)CC1 C1(CC(c2nnnn2C2COC2)NCCOC(C)(C)C)CCS(=O)(=O)CC1 O=C1CCN(C(=O)C2=CCC(NC(=O)C3=COCCC3)C2)CCCN1 CCC(COC)NC(=O)COCCN(C(=O)C(O)C1CCCC1)CC c1(C(=O)NCC23C(CN(C(C)=O)C2)CCCC3)cc2c(nc1O)CCCC2O N1(C(CCN(S(CC)(=O)=O)C)=O)CC(NC(=O)C(C)SC)C2(CC2)C1.N(C)CC N1(C(c2ccc(CNC(C(C)N(C(C)=O)C)=O)o2)=O)CC2CCCC2C1 C1(C)(CCNC(c2nn(C)nc2Br)c2n(CCCCCC)nnn2)CCCCC1 CC(C)(C)C(C)(C)C(=O)NCC(O)CCNC(c1ccc2occc2c1)=O c1(C(CNC(C(C)O)=O)NC(c2ccccc2NCC#N)=O)cc(F)cc(Cl)c1 N1(C(c2c(N)c(F)ncc2)=O)CC(NC(c2ccc(CO)o2)=O)CC12CCC2 N1(C(Cc2cn(C)nc2)=O)C2CCC(C2)C1CNC(c1cc(F)c[nH]1)=O N1(C(CC2CCCC(C)(C)C2)=O)CCC2(CC1)CC2CNC(=O)CSCC(N)=O c1(C(N2CC(NC(=O)OC(C)(C)C)C2)=O)ccc([N+](=O)[O-])cc1Cl.CC1C(=O)N1 CC1(C)CC(N=c2ccnc(C3CC3)[nH]2)CN(C(c2ccn(C3CCC3)n2)=O)C1 N1(C(C2CN(C(C=C(C)C)=O)C2)=O)CC(O)(C(C)NC(C2CC(C)CO2)=O)C1 C1(C(=O)NCC23CC(NC(CNC(CC(C)C)=O)=O)(C2)C3)COc2ccccc2O1 N1(C(C(C)NC(=O)NC)=O)CCCCC1CC(=O)NCC1CC(=C2CC2)C1 Cc1cc2cc[nH]c2cc1C(=O)NCC1CCN(Cc2cc(C#N)ccc2Br)CC1 C1(F)(CNC(CSC(C)C)=O)CCN(C(c2sccc2Cl)=O)CC1 CN1CC(C)(C)CC1C(=O)NC1(CC(N2CCN(CCO)CC2)=O)CCCCC1 C1(C(=O)NC2C=CCN(C(=O)C=CC3CCCC3)C2)Cc2ccccc2S1 N1(C(C(CC=C)CC)=O)CCC2(CCCN2C(c2cc(C)c(C)[nH]2)=O)C1 C=CCCC(C(=O)N1CCC(C)(CO)C1)NC(=O)C(C1CCCCC1)C c1(C(N2C3C(NC(c4cnco4)=O)C(CC3)C2)=O)ccnc2ccccc12 C1(O)(CNC(C(C)CC2CCC2)=O)CCN(C(C2CCC(O)CN2C)=O)CC1 CC1(C)c2cc(Br)ccc2NC1C(N1CCC2C(C(N)=O)C2C1)=O C(CCCC(=O)N1CCCCC1C)NC(C1(CC#C)CCCO1)=O N1(CCN(C)C(c2ccc(C3CC3)o2)=O)C(=O)CCC1=O.C12(CC1)C(=O)N2 C(CCC(O)C(=O)NCCOC1CC1(F)F)NC(c1nn(C)c(O)c1)=O Cc1cc(CN2CCC(NC(=O)CCc3ccoc3)C(O)C2)ccc1F C(=O)(CC(C)C(C)(C)NC(c1c[nH]c(=S)cn1)=O)NCC(c1nccs1)C C1(C(N(CCOCCC(=O)NCC(C(C)C)C)C)=O)CC(=O)OC1(C)C c1(C(N2C(CNC(C(C)OCC)=O)COCC2)=O)coc2cc(F)ccc12 CC1CN(C(=O)C(c2ccc(Cl)cc2)C)CC1Nc1cc(C(C)(C)C)ncn1 c1(CC)nc2n(n1)CCCC2N=c1[nH]c2c(c(=NCCN(C)C(C)C)[nH]1)SCC2 c1(C(N2CC(O)(CCNC(c3c(C)cn(C)c3)=O)C2)=O)c[nH]c2cccc(F)c12 C1(NC(C2CCC(CC)O2)=O)CCN(c2ccc(C(F)(F)F)cn2)CC1O c1(OC)ccc(C(=O)NC(CN(C(=O)CCNC(c2ccoc2)=O)C)CC)cc1 c1(C(=O)NCC2CC(C)N(C(C3CNC(=O)C3)=O)CC2)ccc(F)c(F)c1F C1(O)(C(C)NC(CC2(COC)CCCC2)=O)CCN(C(C2CCSCC2)=O)CC1 C1(C(N(CC(C2CC2)OC)C)=O)(C(C)C)CCCN1C(=O)CC1(C)CCC1 C1(NC(c2sccc2C2CC2)=O)CCN(C(C23CCC2C3)=O)CC1O C1(N(C(C(=Cc2cnc[nH]2)C)=O)C)CN(C(c2nc(=N)cc[nH]2)=O)CC1(C)C C1(CCNC(C(C)(C)C2CCOC2)=O)CCCCN1C(c1cc(C(N)=O)no1)=O c1(N2CCC(C)(NC(=O)CCn3cccn3)C2)ccc([N+](=O)[O-])cc1 c1(NC(=O)NC(CC)Cc2ncc(-c3ccc(Cl)cc3)s2)cccc2cccnc12 CCCC(C)CC(=O)NC(CCCOC)C(=O)N1CCCC1(CC)CN(C)C S(=O)(=O)(c1cnc(NC2CCOC2)c(Br)c1)NC(c1ccc(C2CC2)cc1F)C N1(C(Cc2c(C)nn(COCC)c2C)=O)CC2(COC(NC(=O)CSC(=N)N)C2)C1 c1(C(=O)NCC(C)CNC(c2nc(C(C)(C)C)no2)=O)ccc(C2(C)CC2)cc1 c1(C(=O)NC2C(C)(C)CN(C(=O)CC3CCOC3)C2)ccc2ncccn12 c1(C(N(CC(C)C)C)=O)ccc(CN(C(=O)CCC(=O)OC(C)(C)C)C(C)C)nc1 C1(NC(C(C)c2cncs2)=O)CCC2(CCN(C(=O)C(C)(C)C3CCOC3)C2)C1 C1(C(N2CCC(N(C)C(c3sccc3C3CC3)=O)C2)=O)CC2C=CC1C2 C1(CCC)(NC(=O)C(C)(C)C)CCCN(C(C2(Sc3ccc(F)cc3)CC2)=O)C1 c1(C(=O)NCC(O)CNC(C23CC(c4ccccc4)C2C3)=O)c(Cl)cncc1Cl C(CCCCC(=O)N1C2CCC1COC2)NC(C(C)CCn1cccn1)=O N1(C(CCCOCC)=O)CCC(C2CCCN(C(c3ccncn3)=O)C2)C1 C(=O)(CCCC(=O)c1cccc(Cl)c1)NC(C1CN(C(=O)CC2CC2)CCO1)C Cc1[nH]c(-c2ccccc2)c(C)c1C(=O)NC1CC1(F)F.C12CC1NC2=O C(C)(C(=O)N(CCOCCO)CCC(=O)CCN)OC.C(CNC(N)=O)=C C1(NC(c2n(CCC)ccc2)=O)CCCCC1C(N1CCC(CC(=O)OC)C1)=O c1(C(=O)NCCCC(CCC)NC(C2(CF)CC2)=O)c[nH]c2ccncc2c1=O N1(C(Cc2cc(C)no2)=O)CC2=C(C1)CN(C(C1COC3COCC3O1)=O)C2 C(=O)(C1=CCCN(Cc2cc(F)ccc2C)C1)Nc1cccc(CCC)c1 c1(C(=O)NC2CCN(C(=O)Cc3cccnc3)C3CC23)nccc2n[nH]cc12 c1(C(N2CCC(NC(Cc3c(C)n(C)cn3)=O)CC2)=O)cc2c(cc1O)OCO2 C(C)(CCC(=O)NC(C)(CNC(=O)CCCCN1CCCCC1)C1CC1)OCC Cc1[nH]c(C)c(C(=O)N(CCCNC(c2ccc(CCF)cc2)=O)C(C)C)c1C C(CC(C)N=c1[nH]c(=NCCc2c(F)cncc2F)c2cccc(F)c2[nH]1)SC C(=O)(CCCCC(F)F)NCCCNC(C(c1cn(C)nc1)(F)F)=O C1(CCNC(CC(C)(C)F)=O)CCN(C(=O)C=CC2CCOCC2)CC1(F)F C12(NC(COCCN(C)C)=O)CCC(NC(=O)C(c3cccnc3)O)(CC1)C2 c1(CC)ccc(C(N2CCC(C)(CNC(c3cnn(C)c(=O)c3)=O)C2)=O)c(F)c1 Cc1ccc(N)c(C(=O)NCC2CCCC(NC(=O)CN=S(C)(C)=O)C2)c1 N1(C(Cc2c(C(C)C)con2)=O)CCOCC1CNC(=O)COCC(F)(F)F c1(OC)cncc(C(N2CCC(N(C(=O)CCC3CC3)CCO)C(CO)C2)=O)c1C c1(OC)ccc(O)c(C(N2CCCCC(NC(=O)Cc3cnc(C)s3)C2)=O)c1 c1(C(N2CC3C(CNC(=O)CC4CC4(Cl)Cl)C3C2)=O)n[nH]c2c1CCC2 C#CC1(C(N2CCC(N(C(=O)C(C)C3CC3)CC3CC3)CC2)=O)CCCC1 N1(C(c2cccc3c[nH]nc23)=O)CCOC2(C1)CN(C(C13CCCC1CC3)=O)C2 c1(C(=O)NCC(C)CN(C)C(C23CC(C)(C2)C3)=O)cccc(F)c1C#N C(=O)(C(O)CCCNC(C1(CF)CC1)=O)NCCn1c(C)ncc1 N1(C(c2cc(OC)no2)=O)CCC(NC(c2csc(Cl)c2Cl)=O)C(OC)C1 CC(C(=O)NCC1CC1CNC(C1CC2(CCC2)CO1)=O)S(C)(=O)=O CCCCCCC(CC)(CC)C(=O)NC(CNC(C1CCC(C)(C)C1)=O)CC C(=O)(C(C)(C)S(=O)(=O)C1CC1)NCC(C)(C)NC(=O)CC1OCCO1 CCC(CC)CC(=O)N1CCCC(C2CCCCN2C(=O)C(C)=CC(C)(C)C)C1 C1(NC(Cn2ncc(C)c2)=O)C2CCC1CN(C(=O)Nc1ccccc1)C2 C(=O)(CC(C(F)(F)F)OC)NCC(CCOC)NC(=O)CCN(S(C)(=O)=O)C C#Cc1ccc(C(=O)N(CCN(C(=O)C=CSC)C)C(C)C)cc1F c1(NC(CCN(C(=O)CC2CCCOC2)CC)=O)ccccc1F C1(C(C)=O)OC2CCC1CC2.c12ccc(s1)C(=O)NCC(C(C)C)NC2=O C1(C2CCN(C(=O)CC3CC(F)C3)CC2)(NC(CSS(C)(=O)=O)=O)CCC1 C1(CC(=O)NC(C)(C)CCNC(C2CC(O)C2)=O)COCC1(C)C C1(NC(C=CCCC(C)C)=O)CCN(C(=O)CCNc2cccnc2)CC1C c1(C2CC2)ccsc1C(=O)NC1C(COC)COC1.n12cc(nn1)CNC(=O)C2 C=CCC(CC)C(=O)NC1(C2CN(C(=O)C(=Cc3cnn(C)c3)C)C2)CC1 CCCCC(C)C(=O)NCCOCCNC(C1(c2ccccc2)CC12CCC2)=O N1(C(C(c2ccc(Cl)cc2)(C)N(C)C)=O)C2CC2C2CC12 C1(CNC(CC=CCC)=O)CC2(CCN(C(=O)C(C)SC(F)(F)F)C2)CO1 CCC(C(=O)N1CCCC1CNS(=O)(=O)CC1CCOC(C)(C)C1)C(C)(C)CC C1(C)(CC)CC(NC(=O)CCn2ccnc2)CN1C(=O)Cc1cccnc1 N1(C(C2C(NC(C3C(C)=CCS3)=O)CC2)=O)CCn2c(C)cnc2C1 CCC(C(=O)OC)C(=O)N1CC2CC1(CNC(C1CN(C3COC3)C1)=O)C2 N1(C(C2CC3(CC(NC(c4cncc(C)n4)=O)C3)C2)=O)CCc2cnccc2C1 Cc1nc(C)c(CNC2COC2)c(C)n1.N12CCC3CN(C3C1)C(=O)CCNC2=O c1(C(=O)NCC(C(C)C)NC(C2CC=CCO2)=O)nn2ccccc2c1Br N1(C(c2nncc(CCC)c2)=O)CCC=C(CNC(=O)CCCC(F)F)C1 N1(C(C(CCC)(C)C)=O)CC=C(CCNC(C2(C3CC3)CCC2)=O)CC1 C=C(C)C1CN(C(=O)C(C)(C2CC2)N(C(=O)CCN=[N+]=[N-])C)CCO1 c1(C(N2CCC(NC(C=C(C)C(C)(C)C)=O)C2C)=O)nc(OC)ccc1F N1(C(c2c(C)nn(C)c2)=O)CC2CCOCC2(NC(=O)CCCc2ccsc2)C1 c1(CC)ncsc1C(=O)NCC(C(C)C)NC(=O)Cc1cncnc1 c1(C(C)OC)ncc(C(=O)NCCCN(CCSC)C(c2cnc(Cl)[nH]2)=O)s1 C1(C(=O)NCC(CC=C)NC(c2cncc(Cl)c2C)=O)C2CCCCCC12 CC1CCCN(C(C2CC(CNC(C3CC4CCC4C3)=O)C2)=O)C1 c1(C(N)=O)ccc(C(=O)NCCOC2CN(C(=O)Cc3cncn3C3CC3)C2)s1 N1(C(c2c(C)c(C#N)ccc2)=O)CC2(CCCN(C(C3(C(N)=O)CCC3)=O)CC2)C1 c1(C(C(=O)NC2(CC)CCC2)F)ccc(F)cc1.C12CCN(C1)C(=O)C2 c1(CC)ccc(C(=O)N(CC(C)CNC(=O)C(C)N(C)C)C)cc1[N+](=O)[O-] C1(NC(=O)CCOc2ccccc2F)CCCC2CN(C(=O)Cn3ccnn3)CC12 C1(CC)(NC(c2coc(C#N)c2)=O)CCN(C(c2ccccc2COC)=O)CC1 C1(C(N(CCNC(c2c(C)snc2)=O)CCOCCO)=O)CCCC1(F)F C1(NC(C(C)N(CC(F)(F)F)C)=O)C2CN(C(c3csc(C#N)c3)=O)CC12 N#Cc1cc([N+](=O)[O-])cnc1N1CC2CN(C(=O)CCn3cccn3)CC2C1 C#CCCCCCC(=O)NCCOCCC(=O)NC(CCC=C)C(C)C C1(NC(C(OC)OC)=O)C2CC(O)C1N(C(c1cccc3nn[nH]c13)=O)C2 Cc1cc(=NC2CC(C)NC(C)C2)[nH]c(=NCC)[nH]1.S(C)(=O)(=O)N C(=O)(C(C)C(=O)N1CCCCC1C1CCN(C(=O)CCc2cnn(C)n2)C1)OC N1(C(C2(CC=C)CCCC2)=O)CCCC(O)(CNC(c2sccc2COC)=O)C1 C(=O)(CCCC(F)(F)CO)NCCCCCNC(CC1C(C)(C)CCCO1)=O C1(NC(c2c(CNC(=O)CSc3cn[nH]c3)cco2)=O)CC2(CCC2)C1 CCC(CCC(=O)N1CC(N2CC(O)C2)C1)NC(c1ccnnc1C)=O c1(OCC)c(Cl)cc(C)nc1C(=O)NCC1(O)CN(CC2CC2CC(C)(C)C)C1 C(=O)(C1=NOC(C)C1)NCC(C1CCCCC1)NC(C1(COC)CC1)=O c1(NC(CC2N(C(C3CC(C)C3)=O)CCC2)=O)c([N+](=O)[O-])ccc(Cl)c1Cl CC(C)C(C)C(C)CC(=O)N1CCN(C)C(CF)C1 N1(C(c2c(COC)ncs2)=O)CCC(NC(c2cncc(N(C)C)n2)=O)C1(C)C CCCC(CC)(c1nnnn1CCC1(C)CC1)NC1(C)CC2CC2C1 S(=O)(=O)(c1ccc(Br)cc1Br)NCC1OCCN(C(C(CCCC)O)=O)C1 N1(C(c2c(CC)nn(C)c2)=O)CCCC(CNC(c2ccnc(F)c2Cl)=O)CC1 C1(C(=O)NCC=CCC(=O)NCC(CC)N(C)C)CCC(=O)C1 C1(CC(=O)NCC(C2CC2)NC(c2csc(C3CC3)n2)=O)CC(O)C12CCC2 N1(C(CNC(C)=O)=O)CC(C(F)(F)F)CC1C(N1CCC(N(C)C)C1)=O c1(C(N2CC(C#N)C(NC(=O)Cn3cccn3)C2)=O)cccc2[nH]ccc12 C(=O)(C(C)(O)CCc1ccccc1)N1CC(C(C)NC(c2c(C)nns2)=O)C1 c1(CN(C)C(=O)NC2(C)CCN2CCCn2ccnc2)cccc(O)c1 C(CCS(=O)(=O)c1ccc(CCCNS(=O)(=O)c2sc(Br)cc2C)cc1)OC c1(OC(F)(F)F)ncc(C(N2CCN(C(=O)CSC(F)(F)F)C(CO)C2)=O)cc1Cl.CO c1(CN(CC(=O)NCC(C)OCCCCCC)C2CC2)cnc(OC)cc1C N1(C(C(F)=CC)=O)CCC(NC(c2ccc(F)c(C(F)(F)F)c2)=O)C(F)C1 Cc1ccc(C(N2CCC(C)C2CNC(c2ccn(C3CC3)n2)=O)=O)cc1CO c1(C(=O)NC2CCN(C(=O)CNc3ccccc3)CC2F)ccccc1[N+](=O)[O-] N1(C(C2C3(CCN(C(c4ncccn4)=O)C3)C2)=O)CCSC2(CCC2)C1 c1(C(=O)NCC(C)N(C(C(CC)=CC)=O)C)cnc(CC(C)C)cn1 CC(C)C(C#N)C(=O)N1CCCC(N(C)C(c2ccc(N(C)C)cn2)=O)CC1 CN=c1[nH]cc(C(=O)NCC2CN(C(C3(O)CC3)=O)CCO2)s1 C(=O)(C(C)(F)C(C)(C)F)N1C2C(CNC(C(C)(C)N3CCOCC3)=O)C(C2)C1 CC1(C(=O)NCC2CC2CNC(=O)C(c2cccc(N)c2)O)CCNC1=O C(=O)(CS(=O)CCC(F)(F)F)NCCC(C)NC(c1cn2cc(F)ccc2n1)=O C(c1ccc(Cl)cc1F)=CC(=O)NCC(CNC(C1CC2CC2C1)=O)OC C1(NC(c2cc(C(F)(F)F)on2)=O)CC2CC1N(C(c1n[nH]cc1Cl)=O)C2 CCC(Cc1ccccc1)C(=O)N1CCC1CNC(C1(CCCSC)CC1)=O c1(N(C)C)ncc[nH]c1=NC(=O)CC(N)C(C)(C)C C#CCC(CC(F)F)NC(c1ncoc1CNC(C1CC1CCOC)=O)=O C1(NC(C2OCCC(C)(C)C2)=O)CCC2(CCN(C(C3(CO)CCOC3)=O)C2)C1 CC1(C2(N(CCC(=O)N3CC(C4CCCC4O)C3)CCCO)CC2)CC1 C(CCN(C)C(c1cc(Cl)cnn1)=O)(C(C)(C)C)NC(COCCOCC#C)=O C1(F)(COc2ccccc2)CCCN(C(=O)C(C)(C)C(C)(C)CNC(=O)OC)C1 C1(N(C(=O)C=CCN=[N+]=[N-])CC=C(C)C)CCC2(CC1)CC2 C1(NC(CS(CC)=O)=O)CC2(CCN(C(c3cc4c(cn3)CCCC4)=O)CC2)C1 N1(C(c2c(CC)c[nH]c2)=O)CC2CN(C(C3(C)CCNC(=O)C3)=O)CC2(C)C1 C1(NC(c2c(C)cco2)=O)CN(C(=O)CCSc2nnnn2C)CC2CC12 c1(CC)cc(C(=O)NCC2(CCNC(=O)CCC(=O)N(C)C)CC2)ccc1Br Cc1cc(CNc2ccc(N(C)C)cc2F)n2nc(C)cc2n1 c1(OC)cccc(CNC(C(CC2CC2)C(=O)N2CCC(OC(C)(C)C)C2)=O)c1 N1(C(C(C)OC2CCCC2)=O)CCN(C(c2cccc3[nH]ccc23)=O)CC(C)(C)C1 CC1(F)CCC(C(=O)Nc2ccc(C(=O)NC3CCC(OCF)CC3)cc2)CC1 Cc1cccc(OCC(C)NCc2ccc(Cl)cn2)c1 c1(CC(C)N(CCCc2ccccc2)C(=O)OC)ccccc1F.CC Cc1ccnnc1C(N1CCCC(CCNC(c2ccnc(C(N)=O)c2)=O)C1)=O N1(C(C2CCCN(CCC)C2)=O)CCCC(O)(CNC(c2cc(Cl)cnn2)=O)CC1 Cc1ccc(SCCNC(c2ccno2)=O)cc1 N1(C(C2N(C(c3cc(C(C)=O)[nH]n3)=O)CC(F)C2)=O)C2CCC1CN(C)C2 C(CC(C(C)(C)C)NC(c1sccc1C#N)=O)N(C(C1CC(C#C)(O)C1)=O)C Cc1cc(C(N2CCCCC2c2ocnc2C(=O)O)=O)cc(F)c1 N(C)(C1=NS(=O)(=O)c2ccccc21)C(C1C(NC(c2nc(C(C)N)oc2)=O)C1)=O CCCCCCC(CC)NC(=O)C(=O)NS(=O)(=O)CCOC c1(C(=O)NCC2(F)CCC(NC(c3ccns3)=O)C2)cc(O)cc(Cl)c1Cl c1(OCCC(=O)NC2(CF)CCN(C(C(CCC)O)=O)C2)ccc(Cl)c(F)c1 C(=O)(CC1OCc2cc(Cl)ccc21)NCc1nc(CNC(CCC(C)C)=O)sc1 n1(CC)ccc(C(=O)N(C(C)CNC(c2ccnnc2)=O)C)n1 C1(C)(CC)CC(NC(C2CCCC2)=O)CN1C(=O)CCCn1cc(C)cn1 N1(C(c2cccc(C)c2)=O)CC(CNC(=O)C=C2CCCC2)CC12CCC2 N1(C(C2(CC#C)CCCC2)=O)CCC(C)C(C)C1 C1(C(=O)NCC(C#C)CC2CCC2)CC(C)(C)CN1C(=O)COC1CC1 c1(C(=O)OC)ccc(CNC(=O)CCCC2CCCC(=O)N2)c(Cl)c1 C(=O)(CC(F)(F)C(F)(F)F)N(C(C)CN(C(=O)COC1CCOCC1)C)C Cc1noc(NC(C2CCCN(S(=O)(=O)Cc3ccc(Br)cc3)C2)=O)c1C C1(CCC(C)C)CCCN1C(=O)N(CCN(C)C)CC1CCN(C(C)(C)C)C1 CC(C)C(F)(F)CC(=O)N1CCCC1CNC(=O)CCC(=O)c1ccc(O)cc1 C(=O)(C1Cc2ccc(Cl)cc21)NC1CN(C(Cc2cc(C)[nH]n2)=O)C(C)(C)C1 C12(C(N(CCC(=O)OC)CC=C)=O)CC(CN1C(c1cnc(COC)s1)=O)C2 c1(C(=O)NCC2(C)CCN(C(C(C3CC3)OC)=O)CC2)cc2sc(C)cc2s1 C(C)(CCCCOCC(=O)NCCNC(=O)COCc1ccccc1C)OCC#C N1(C(C(CC=C)OC)=O)CC2CCN(C(c3cnn(C)c3C3CC3)=O)CCC2C1 CN1CCN(C(c2occ3c2CCC3)=O)C(C(=O)NC2CCC(F)CC2)C1 C=CCC(CC)C(=O)NCCC(C)(CC)NC(c1ccnc(OC)n1)=O C(CNC(=O)CCc1cnn[nH]1)(CNC(=O)CCOCCN(C)C)OC C1(C(=O)NCC2C(C(=O)OC)CC2)(CNC(=O)C(F)CC2CCOC2)CC2(CC2)C1 C1(C(N2CCC(C(C(=O)NC(COC)(C)C3CC3)C)C2)=O)CCCCC1(C)C c1(CCOC(C23C(CN(C(=O)OC(C)(C)C)C2)C3)=O)cccc(C#N)c1 C(=O)(C1=C(Cl)CCOC1)N1C(CNC(=O)CC(C(F)F)c2ccc(F)cc2)CC1 c1(CC)cc(C(=O)NCC2CCN2C(c2coc(N(C)C)n2)=O)c(C)o1 N1(C(CCOCC#C)=O)CC(NC(=O)CS(N)(=O)=O)CCC1C C(CNC(C1CC12CCOC2)=O)(CC)(CC)NC(CC1CC(=C)C1)=O C1(C(=O)NCC2(C=C)CCC2)(NC(=O)CCc2nc(CC)no2)CCCCC1 N1(C(=O)C=CCN2CCC2)CCCCC(C2CN(C(c3cnsn3)=O)C2)C1 C1(=O)CCCCN=C2NC(=NCC3CCN1CC3)NC1=C2CCC1.C(C)(C)(C)NC C1(NC(C(=O)NC(c2cn(-c3cccnc3)nn2)C)=O)CCC(C)CC1 c1(NC(C2CCCN(C(=O)C(F)(F)F)C2)=O)ccc2c(c1)OCO2 c1(C(=O)NCC23N(C(c4cc(C)[nH]n4)=O)CC(C2)C3)cc2ccc(F)cc2s1 O=C(CCc1cccnc1Cl)NNC(=O)C(=O)c1nn[nH]n1 c1(CCN(C(=O)Cn2cc(-c3csc(CC)n3)nn2)CC)nc(C)c(COC)o1 N1(C(C(CCSC)O)=O)CCC(N(C)C(c2cnncc2C)=O)C2(CC2)C1 CCCCCC(O)CC(=O)NC1CC(NC(c2ncccc2OC)=O)C1 O=C1CC(C(=O)NC(C(F)(F)F)C2CCCOC2)c2cccnc2N1 N1(C(C(C(C)C)N(C)C)=O)CC2(C1)CN(C(c1cocn1)=O)Cc1ccccc1O2 C(CC(C)C)(C(=O)NCc1cnn(C(C)C)c1)NC(C(CCSC)O)=O N1(C(c2[nH]nc(OC)c2Cl)=O)CCN(C(C2CC3CCC2O3)=O)CC(O)C1 c1(C(=O)NC2(CF)CN(C(CC)=O)C2)cnc2c(c1)NCC2 N1(C(C(CCC)CC2CCCC2)=O)CCC(C(c2ccc(C)nc2)=O)C(C)(C)C1 N1(c2cc(NCc3nnc(CC)o3)nc(C)n2)CCC(C2CNC(=O)C2)C1 Cc1ccc(Cl)cc1NC(=O)NC1(C)CN(C(c2c(C)nn(CC(C)C)c2Cl)=O)C1 C1(CNC(CCC(=O)NCCCn2c(C)cc(C)n2)=O)COCCN(C(N)=O)C1 Cc1cc(F)ccc1C(F)(F)C(=O)NCC1CC1NC(=O)CN(C)CCO c1(C(N(CC(CNC(c2cnc(C(C)C)s2)=O)C)C)=O)cnc2c(c1)CCOC2 CC(Cc1ccco1)C(=O)NCC1(CNC(=O)CCOC2CCOC2)CCC1 C=CCC(C(=O)N1CCC(C(=O)N(C)CCN(C)CCO)C1)C(C)C C(c1ccc2c(c1)OCO2)=CC(N1CCN(C(C2CCS(=O)(=O)N2)=O)C2CC12)=O C1(C(=O)NCCC2(CNC(CNC(=O)OC(C)(C)C)=O)CC2)CC(=O)CS1 c1(C(=O)NCC(=O)NCC2(OCCOCC#C)CC2)cc(C)c(C)c(F)c1 C1(C)(CNC(c2cnn(CC)c2C)=O)CN(C(=O)CCCC2CCCO2)CC1C N1(C(c2[nH]c(=NCC)sc2)=O)CC2CCC1CN2C(=O)C=Cc1ccc(Cl)cc1 C(CC(O)C(C)C)NC(C(CC1CCC1)NC(C(OC)OC)=O)=O c1(C(N2CC(CC)SCC2)=O)n[nH]c2c1CN(C(=O)Cc1c[nH]nc1C)C2 C1(N(C(C(CCC)O)=O)C)CN(C(=O)CN2CCCCCC2=O)CC12CC2 C(=O)(C1=C(C)CCOC1)N1CCC(C(=O)Nc2c[nH]ccc2=O)(CC)C1 N1(C(CCC)=O)CCC2(CCN(C(=O)Cc3sc(C(C)OCC)nc3C)C2)C1 C(CC(C(=O)NCCc1cnn[nH]1)NC(=O)C(CC)n1cncn1)=CC Cc1nc(C(N2CCC(O)(CCNC(C3CC(C)OC3C)=O)CC2)=O)ccc1C#N CC1(C)CC(C)(CNC(C2CCCN2C2CCCC2)=O)CN1C(c1nc[nH]n1)=O c1(C(=O)NC2C(CNC(C=C(CSC)C)=O)CC2)coc2ccccc12 C(=O)(CCCCCCNC(C1C(C#N)C1(C)C)=O)NC(C)C(C)(C)O c1(SC)cncc(C(=O)NC2(C)CCN(C(C3CCN(S(C)(=O)=O)CC3)=O)C2)c1 C1(CC#C)CN(C(C2(C=CC(F)(F)F)CN(CCC)C2)=O)CCO1 CCCCC(F)C(=O)N(CCC(N1CC(CO)(CO)C1)=O)CCO C1(CCNC(CN(CCC)C)=O)C(C)CCCN1C(=O)Cc1nc([N+](=O)[O-])n[nH]1 c1(CC(C)C)cc(C(=O)NCCCNC(C2CC(C)(C)C2)=O)no1 C1(CNC(C2CC(C)CN2C(=O)C(F)OC(F)(F)F)=O)CC(C(N)=O)=NO1 CCC(CC(F)(F)F)C(=O)NCCC(C)N(C(=O)CCSc1c(C)noc1C)C C1(NC(c2[nH]cc(C#N)c2)=O)C2CCC1N(C(C1CC(=C3CC3)C1)=O)C2 CC(CN=c1ccnc(Cl)[nH]1)N(C(=O)CC(O)c1ccccc1)C C#Cc1cncc(C(=O)NC2CN(C(=O)Cc3cccn3C)CCC2O)c1 N1(C(C(C=C)O)=O)C2CCC1CN(C(=O)Cc1cccc(OCCC)c1)C2 c1(CN2CCC(NC(c3ncc(CC)nc3)=O)C2)cc(Cl)ccc1Br c1(C(=O)NC(Cc2c(C)[nH]n(CCC(C)C)c2=O)=O)cc2cccc(Br)c2[nH]1 C(c1ccccn1)=C(C(=O)NC1CN(C(c2c(COC)ncs2)=O)C1)C C1(NC(CNC(C)=O)=O)CCN(C(=O)Cc2csnn2)CCC1CO C#Cc1cc(C(=O)NC2(C(=O)NCC3CC4C=CC3C4)CSC2)ccc1C Cc1cc2c(cc1Br)N(C(=O)C(=O)NCCCOC1CCCOC1)CC(C)O2 CCC(C(=O)N1CCCN(C(C2OCC3CCCC2C3)=O)CC1)C(C)(F)F Cc1cnc(C(=O)N(CC(C)(C)CNC(c2ccc(C(C)(C)C)cc2)=O)C)nc1 C1(CC)C(NC(=O)C(CO)NC(N)=O)CCN1C(C1(N(C)C)CC1)=O C(C(C(=O)N1CC(CNC(c2cc(OC)no2)=O)C(C)C1)C(C)(C)C)OCC=C C1(CC(=O)NC2CC(CNC(c3c(CC)n(C)nc3)=O)C2)CCC2(CC1)CC2 Cc1csc2cc(C(=O)N(CCC(C(C)C)NC(C3C(C)(C)C3(C)C)=O)C)[nH]c12 c1(C2C(c3ccccc3)N(C(C3CCCC3)=O)CCC2)ccc(C#N)c(C)n1 C(=O)(C(CCC1CC1)NC(=O)COC1CCOCC1)NCCC=CC(C)C CCCC(C(=O)N(C)OCC(F)(F)F)NC(C1CCOCC1(C)C)=O C12(NC(C(CSC)C)=O)CC(C)(C1)OC21CCN(C(=O)CCC[N+](=O)[O-])CC1 N1(C(C2C(CCC)CCC2)=O)CCCC(N(C)Cc2cccnc2C)C1 c1c(C)[nH]c(C(N(C(C)C)NCCC(=O)NC)=O)c1C.c1(N)ncccc1F C1(NC(C=Cc2n(C)ncc2)=O)CC(CNC(=O)Cn2nnc(=O)[nH]2)C12CCC2 N1(C(=O)C=Cc2ccc[nH]2)CCCC2(CCN(C(C3CC4C(C3)C4(F)F)=O)C2)C1 CCCC(C(=O)NC1CCCCC1CNC(=O)C=C1CCCCC1)NC(N)=O N1(C(CC[SH](CCC)C2CC2)=O)CCC2C(C(=O)N(CC(C)C)CC)C2C1 N1(C(CC(C)F)=O)CC(C2CCCN(C(=O)C(c3ccc(F)cn3)(F)F)C2)C1 C(=O)(C1=CS(=O)CCC1)NCC1N(C(C(Cc2ccccc2)OC)=O)CC1 c1(C(N2C3CC(CNC(C4C=CC=CC=C4)=O)C2CC3)=O)ncn2ccccc12 Cc1c(-n2nnnc2C(c2cncn2C)NCC(Cl)Cl)cccc1Cl N1(C(c2csnn2)=O)CC(C2CN(C(C3(CCN4CCOCC4)CC3)=O)C2)C1 C1(NC(COC2CC(NC(c3n(C)ccn3)=O)C2)=O)CC2C=CC1C2 c1(C(N(CCCNC(c2c(C)coc2C)=O)CC)=O)cc2c(O)cccc2n1C c1(NC(C)=O)ccc(NC(=O)CCCCN2CCCCC2=O)cc1Cl C(C(=O)NC(C)CC)(C1=CCSC1)N1C(CCCCC)CCC1 C1(C(=O)NCC2(O)CCOC2C)(CC)CCN(C(C2CC23CC3)=O)CC1 Cc1ncc(C)c(N2CCCCC2CNC(c2cc(C#N)c[nH]2)=O)n1 c1(C(=O)NCC(C)N(C(C(C)SC(C)C)=O)C)cncc(Cl)c1 N1(C(c2c(C)coc2)=O)CCC(C2(NC(C3CCCC3O)=O)CC2)C1 C(=O)(C1=CC2C=CC1C2)NC(CC)C(=O)NC1CC2CC(OC)C2C1 C1(C(=O)NN(C(C)C(C)OC)C(C2CCN2C(C)(C)C)=O)(CC)CCCO1 N#Cc1ccc(N2CC3C(NC(C4CCC(F)CC4)=O)C3C2)nc1 Cc1nc(O)c2c(n1)CCN(C(C1C=CCN1C(c1cc(Br)ccn1)=O)=O)C2 c1(N(C)C)cc(NC2C3CCC23)ncn1.C1(CC=O)CCN(CO)C1 N1(C(CCOCCOC)=O)CCC(NC(=O)C(O)CSC)C1C(C)C C1(CNC(c2ccc(CCC)[nH]2)=O)C(C)CCCN1C(=O)CC1CC1 C(=O)(C1=NNC(=O)C1)NCC1(OC)CCN(C(=O)CN(C2CCSC2)C)C1 CCC(CC(=O)NC1CC1NC(=O)C(c1ccc(OC)cc1)=O)c1ccc(C)cc1 c1(C(N2CCC(CN(C(c3cc(C)ncn3)=O)C)CC2)=O)ncnc2c1CCC2 C1(CNC(C2(C)CCCC2)=O)CN(C(c2c[nH]ccc2=O)=O)CCO1 Nc1c(C(=O)NC2CN(C(C3CC3c3nnc(O)s3)=O)C2)cc(F)cc1F c1(C(=O)NCCOCC)nc(CNC(c2cc(CC)[nH]n2)=O)oc1C C1(NC(C=CCC)=O)CN(C(C2CCc3n[nH]cc3C2)=O)CC2(CC2)C1 c1(CC(N2CCC(C(C)NC(CC)=O)C2)=O)cccc(F)c1Br CC1(C)CCC(CC(=O)NC2CC3CC2N(C(=O)CCc2cc[nH]n2)C3)OC1 CC1(CC(=O)NOC(=O)CCS(N)(=O)=O)Cc2c(Cl)cccc2C(=O)O1 N1(C(COCCCC(C)C)=O)CCCC1C1CCCCN1C(c1cccnc1)=O c1(C(=O)NC2CCC(NC(C3(C)CNC(=O)C3)=O)C2)cncc2c[nH]nc12 c1(C(=O)NCC2(O)CN(Cc3c(OC)cc(O)cc3)C2)ccc(F)c(F)c1Cl C1(NC(=O)Cc2ccc(C3CC3)cc2)CN(C(=O)CC(Cl)Cl)CCC1C(F)(F)F C(c1cccc(F)c1)=CC(=O)NCCC(C)CCNC(=O)COC(F)(F)F c1(C(=O)NC(c2cn(CCCCO)nn2)C)cc(C#N)ccc1F c1(CC(N2CCN(C3CCN(C(C(CC)=CC)=O)C3)CC2)=O)ccc(F)c(Cl)c1F C1(NC(C(C)CC2CC2)=O)CN(C(c2cc(Cl)cn2C)=O)CC1c1cnn(C)c1 C1(C(=O)O)CCC(C(F)(F)F)CN1CC(O)Cn1nc(C(F)F)oc1=O C#Cc1ccccc1CC(=O)NC1(C2CCCN2C(=O)C(C)C2CC2)CC1 C(=O)(C1CCSc2ccccc21)NCC1N(C(c2c(F)ccc(C)n2)=O)CC=C1 Cc1cc(O)cc(=O)n1CC(=O)N(CC(C)(C)CNC(C1CC(N(C)C)C1)=O)C N1(C(C(C)NC(=O)NC)=O)CCC(C2(O)CN(C(=O)CC3CCC(=O)N3)C2)CC1 C(=O)(CCCN(C)C)N1CC(CC(C)NC(C2CCC2(F)F)=O)C1 C(=O)(C(c1cccs1)NC(=O)C=CC(F)F)N(C)CCSC1CCOC1 C1(CC(N2CCC(C(C)NC(c3cn(C4CC4)nn3)=O)C2)=O)CCCC(C)(C)C1 c1(CNC(c2c(C)cns2)=O)ccc(CNC(C2CCC(C)S2)=O)c(F)c1 N1(C(CSC)=O)CC2CC(C1)CN(C(=O)Cc1cccc3ccccc13)C2 C(=O)(C(C)(C)C(=O)OC(C)=O)N(CC(CN(C(=O)OCCCF)C)O)C c1(C(=O)NC2CCN(C(C(CC)Oc3ccccc3F)=O)C2)cc(Cl)cnc1O c1(C(=O)NC2CC(N(C(c3nc(OCC)oc3)=O)C)C2)nn(C)cc1COC c1(C(=O)OC)ccc(S(=O)(=O)N2CCC3CN(Cc4cnn(C)c4)CCC23)n1C C(=O)(CCCCC(N)=O)NC(C(=O)NCC1CC(CC)C1)CO N1(C(C(C)N(CC(C)C)CCC(C)C#N)=O)CCCC(CC(=O)N2CCCC2)CC1 CC1(C)CCC(CN2CCCC(NC(c3cc(Cl)ns3)=O)C2)O1 C1(COC)C(O)C(O)CN1Cc1cn(CC2COCC2n2ccnc2)nn1 C1(C(=O)NC2CCC(NC(c3cc[nH]c3C3CCC3)=O)C2)(COC)CCOC1 Cc1cc2[nH]c(C(=O)NC3CC(CNC(c4ccc(S(C)(=O)=O)o4)=O)C3)cc2s1 C#Cc1cn(C)nc1C(=O)NC(CC(F)F)C(=O)NC1CCCC1OC C1(C(=O)NC(CC(=O)N(CC)CC)C2CC2)C2CCC(C2)C1N Cc1csc2cc(C(N3CCN(C)C(CNC(C4C(C)(C)C4(F)F)=O)C3)=O)[nH]c12 c1(CNC(=O)NCCC(CCC)C)cc2cnn(C)c2nc1Cl c1(OC)ccc(CC(N2CC(C)CCC2CNC(=O)C=C(C)C2CC2)=O)cc1OC Cc1c(C(N2CCN(C(C3CCCS3)=O)CC3(CC3)C2)=O)sc2ncnc(N)c12 CCC(CC(=O)NC1CCC(O)CN(C(=O)CSc2cc(C)on2)C1)C(C)(C)C C(=O)(C(C)(C)C(C)(F)F)NCC(C(=O)NC(c1nn[nH]n1)CC)N(C)C N1(C(C23CC(NC(c4c(C)n(C)cn4)=O)(C2)C3)=O)C(C)CCC1(C)C N1(C(C2(C(C)(C)C)CCCC2)=O)CCC(NC(c2cc(CO)ccn2)=O)C(O)C1 c1(-n2cc(SC(CCC(=O)Nc3nc(COCC)sc3)C)nn2)cc(C)ccc1C N1(C(C(C)OCC2CCCO2)=O)CC2(C1)CN(C(c1cccc(=S)n1O)=O)CCO2 N1(C(CN(C(C(OC)OC)=O)CC2CC2)=O)CC(C(N)=O)(SC)C1 C1(C(N2CCC(NC(C3CC4(C3)CC(O)C4)=O)C2)=O)CC12CC(F)(F)C2 c1(CNC(CC2C(C)CCC2)=O)ccc2c(c1)CN(C(=O)C(C)(C)F)C2 c1(C(=O)OCC)cc2sc(=NC3CCN(C(=O)C(C)S(C)(=O)=O)C3)[nH]c2n1C c1(NC(C(CC=C)c2ccccc2)=O)ncnc2cccc(OC)c12 C1(C(=O)NC2(C=C)CC2)C2CC3C(C2NC(C2CC(=O)CC(=O)C2)=O)C13 c1(C(=O)NCCCC2OCCN(C(C3(C)CC3)=O)C2)n[nH]c2c1CCCC2 C12(CNC(C(CC)CC)=O)CCC(CC1)N2C(c1cccc(F)c1)=O O=S(=O)(c1ccc(NCCCSC(F)(F)F)nc1)NCC1C=CCC1 C#CCC(C)(C)C(=O)NCC1CC1NC(=O)Cc1cc(Cl)n(C)n1 C1(C(N2CC=CC(NC(c3cc(C)c(C)nc3)=O)C2)=O)CCc2n[nH]cc2C1C C1(CNC(C(C)OCC=C)=O)CN(C(c2ccn(C)c2C(F)(F)F)=O)CCO1 C(=O)(C1=CC2C=CC(C1)C2)NC(CC(=O)NCc1[nH]cc(C(N)=O)c1)C(F)(F)F C=C(Br)CN=c1nc(N2CCc3nnnn3CC2)c2c([nH]1)CCC2 C(N=c1[nH]c2c(c(=NCC3(CO)CCCC3)[nH]1)COCC2)c1scc(C(N)=O)n1 C1(NC(c2ccc(C3CC3)o2)=O)CCN(C(=O)C=Cc2ccoc2)CC1F N1(C(CCCc2ccc(C)s2)=O)CC(NC(=O)CCNS(C)(=O)=O)CCC(O)C1 N1(C(C2CN(CC)C(=O)C2)=O)CCCC(C)(NC(C2CCOCC2)=O)C1 N1(C(C(CSC)O)=O)CC(C)(C)CC1CNC(=O)C(c1ccc(Cl)cc1)(F)F CC(C)(O)C#CC(=O)NC(CC1CCC1)C(=O)NC1CC2CC2C1 C(c1ccc(C)cn1)=CC(=O)NCCC1CCN(C(C2(OCC)CCC2)=O)C1 C(=O)(CCCCC(C)(C)C)N1CC(CCNC(CN2CCC(C)CC2)=O)(OC)C1 CC(C)CC(C(=O)N(CC(C)NC(C12CCC(C(F)F)(CC1)C2)=O)C)C(N)=O Cc1[nH]c(-c2ccccc2)cc1C(=O)Oc1cccc(-c2ccc(Br)s2)c1 N1(C(c2cn(C(CC)C3CC3)nn2)C(=O)NC)CCCC(Cc2ccccc2Cl)CC1 C12(CNC(C(CCC)C)=O)CCCCC1N(C(=O)CCC(C)(C)F)CC2 C1(CNC(C=C(C)C)=O)CN(C(C2CSCN2C(=O)C(C)(C)C)=O)CCO1 c1(C(=O)NCCC2CC(NC(C=COCC)=O)C2)cc(OC)cc(C)c1N C(=O)(CC(C)(C)C(=O)OCC1CC(C)(C)C1)NCCN(CCCOC)C c1(CCC)nc(C)c(C(N2CCC(N(C)C(c3cnn(CC(C)C)c3)=O)C2)=O)o1 N1(c2nnc(CC)s2)C2CCC1CC(NC(=O)CC1CC1(C)C)C2 CCCCCC(=O)NC(c1ccc(CNC(C2CCCN2C=O)=O)cc1)C c1(C(=O)OCC)c(F)cc(C(=O)NCCN(C)C(C2(F)CC(NC)C2)=O)cc1F N1(C(C(C(C)C)SC2CCC2)=O)CCC2(CCN(C(=O)C(F)(F)C(F)F)CC2)C1 N1(C(c2cc(CNC(C(C)NC(CC)=O)=O)no2)=O)CC2CC=CC1C2 C1(CC(=O)NCC(N2CCN(C(C3(C)CC(C)C3)=O)CC2)C)CCCC(C)(C)C1 CC1CCn2cc(C(=O)NCC3(CCNC(C4CCCCS4)=O)CC3)nc2C1 c1(NC(C(=O)NCCn2nc(O)c3c2CCOC3)=O)cccc2c1CNC2=O N1(C(c2cccc(NC(C)=O)c2)=O)CCCC(C2CC2NC(C2(O)CCC2)=O)C1 c1(CNC(C=CC=CC)=O)ccc(C(=O)Nc2cccc(OC)n2)nc1 c1(OC)ccc(CN2CCCC2C(=O)NCc2ccc(CO)cc2OC)c(F)c1 C(CC(=O)NNC(=O)C1CCCC(C)C1)NC(c1c(CC)cccc1)C c1(C(=O)NC(C(C(=O)NCC(COC)(O)CO)C)C)c(C)ncnc1C c1(C(N2CCCN(C(C(C)OCC(C)C)=O)C(C)C2)=O)ccc2nc(=N)[nH]n2c1 C1(C)(NC(N(CC(=O)NC)C)=O)CCN(C(c2cccs2)=O)C1 C(CCc1cccc(F)c1)(C(=O)NCC(F)F)N(CC(C)C)CCC C1(C(=O)N(c2ccccc2)CCO)CCCCN(C(C2C=CCS2)=O)C1 CC(C)(O)C#CC(=O)NCC=CCNC(C1CCCC(c2ccccc2)O1)=O N1(C(=O)NCc2cnc(C(=O)OC)o2)CCC(n2nnnc2C(F)(F)F)CC1 C1(NC(C(C2CCN(C(C3C(OC)CCC3)=O)C2)F)=O)(CO)CC(F)(F)C1 C1(NC(c2coc(C3CCC3)n2)=O)CCC12CCC2 C1(C(=O)NO)CCCN(Cc2cccc(-c3ccncc3)c2)C1=O C(=O)(C(CC(C)(C)C)OC)NC1CCC(CCC(=O)NC(C#C)C(C)(C)C)C1 C(=O)(C(C)(C)CS(C)(=O)=O)NC1CCC(NC(C(CCC)CC)=O)CC1 c1(C(=O)NC(CCNC(C(C2CC(F)(F)C2)SC)=O)(C)C)cc(C(C)C)ccc1F C1(C(=O)N(CC(CC)=O)C2CCCC2)CC2CC2N1CC.c12ccc-1s2 c1(-n2ccc(C)n2)ccc(C(=O)N(C(C)CCNC(c2cc(Cl)ns2)=O)C)cc1 N1(C(C2(C3(F)C(F)=C(F)C(OC)=C3F)CC2)=O)CCc2cccc(Br)c2C1 CC(C)C(C(=O)NCC(C)NC(c1cccc(NC(N)=O)c1)=O)NS(=O)(=O)C1CC1 CC1(C)CN(C(=O)CSc2cccnc2)CCC1NC(c1cc([N+](=O)[O-])n[nH]1)=O C1(C(=O)OC)CCC(C)N(C(=O)CCc2cccc(C(=O)O)n2)C1 N1(C(C(C)=C(CC)C)=O)CC(C(=O)NCC2=CCCC2)C(CC(C)(C)C)C1 CCC(C)C(O)C(C)C(=O)N(C1CCCCN(C(c2ccc(C)n2C)=O)C1)C N1(CCC)CCC(C(N)=O)CC1.C1(C(=O)OC)(COC)CNC1 C=CC1(CC(=O)NC2CCOCC2C(=O)NC2CCCC2C(C)C)CCOCC1 C1(N(C(COCC(=C)C)=O)C)CCCN(C(=O)CCc2scnc2C)C1 c1(C(N(C2CCN(C(=O)CC(O)C3CCCC3)CC2)C)=O)cn(C)nc1C(F)F N1(C(C(C)c2ccsc2)=O)CC2N(C(C3C=CCC3)=O)CCC2(C)C1 c1(-c2onc(C3C4(C)CCCN4C(=O)O3)n2)ccc2[nH]cc(CSC3CC3)c2c1 c1(C(=O)NC2C(CNC(c3cc(C)c(C)nc3)=O)C2)ccnc2ccc(F)cc12 O=C(C1NCCn2nccc21)NC1CC(N2CCCC2)C1 Cc1cc(N2CCC(CC(C)NC(c3cc4occc4s3)=O)CC2)c(C#N)cn1 C1(OC)CN(C(c2ncc[nH]c2=O)=O)CC1NC(c1c(Cl)nsc1Cl)=O CCS(=O)(=O)CC(=O)N(CC(C)(C)C(=O)Nc1cn(C)nc1C)C C(CN=C(NCC(C)(F)F)NC1CCCC1)(S(C)(=O)=O)C1CCCC1 C1(NC(C=CC(=O)OCCCC)=O)CC2CC(C1)N(C(c1nnn(C)n1)=O)C2 CC(C)(C(=O)N1CCC1C1CC1)C1CCN(C(=O)NC2CCOC2)C1 Cc1nc(C(N2CCC(C)N(C(c3ccnnc3O)=O)CC2)=O)c(C)n1C1CC1 Cc1cnc(C(=O)NC2CN(C(=O)C(=O)Nc3ncc[nH]3)CC2C)cc1Br C1(NC(C2(C(=O)OC)C(=C)CC2)=O)CCN(C(=O)CC2CCC23CCC3)CC1F N1(C(c2n(CC)ccn2)=O)CCCN(C(=O)CC(C)(O)C(F)F)CC1C c1(CC(=O)NC2(CNC(CCCOCCC)=O)CCCCC2)cc(Cl)cnc1C C(=O)(CCN=[N+]=[N-])NCC1(C(=O)NCc2n(CC)cnc2)CCCO1 N1(C(C(C)SCCCC)=O)CCC2(CCCC2CNC(=O)COCCCF)CC1 N1(C(C(CC)OC)=O)C2CCC1C(NC(c1cc(F)ccc1Cl)=O)C2 c1(C(=O)NC(CNC(C(CC)(C)COC)=O)(C)C(C)C)cc2ccncc2[nH]1 C1(NC(c2c(C)ccs2)=O)COCCC1NC(c1csc(C(F)F)c1)=O Cc1cc(F)c(C(N2CCN(S(=O)(=O)CBr)CC2)=O)cc1-c1cccn1C N1(C(C(COC)OC)=O)CCCC(CO)(NC(C2(CN(C)C)CC2)=O)C1 c1(CC)ccc(C(=O)NC2CC(C)(NC(c3nc(CC)ncc3Cl)=O)C2)cc1N C1(CC)CN(C(OC(F)F)=O)CC(CC(=O)O)O1.c12ccc(cc1)C(C)O2 Cc1cc(=NCCn2ccnc2)[nH]c(NC(c2cccnc2)C)n1 Cc1csc(=NCC(=O)N2CCCC(CNC(c3ccc(Cl)cc3F)=O)CC2)[nH]1 CC(C)C(C#N)C(=O)NC1CCC(C(=O)NCCC(C)(C)N(C)C)CC1 c1(C(N2CCC(CNC(C3CC(O)(CC#C)C3)=O)C2)=O)sc(C)cc1Cl n1(CC)nc(C)c(C(=O)NC2CC(O)(CNC(=O)C(=O)NC(C)C)C2)c1Cl c1(C(N(C(C)CCC2CC2)C)=O)cn(C)c2ccccc12.c1(C(=O)N)ccoc1C1CC1 CCCCC(C(=O)NCC1CCOC(C)C1)NC(=O)CNC(C1CC1C)=O c1(CC(=O)NCC(Cc2ccccc2)NC(C(C)CF)=O)ccc(S(N)(=O)=O)s1 N1(C(COC2(C)CN(C(CSC(C)C)=O)C2)=O)C(C)CCC1C n1(CC(N2CCC(CNC(c3c(C)oc(C#N)c3)=O)C2)=O)nc2c(n1)CCCC2 Cc1cc(C(=O)N(CCCNC(C2(C(F)F)CCCC2)=O)C2CC2)nn1C C=CCC(CC(=O)NC1CC1CC(C)C)NC(C1C(CF)C1(F)F)=O c1(CNC(Cn2cc(CC)nn2)C)cccc2cnn(C)c12 C1CN=C2C=C(N=CN2)N1.c1(CNS(C)(=O)=O)c(Cl)cccc1Cl c1(C(N2CC(CN(C(=O)CCC(C)(C)F)C)OCC2)=O)ccc(F)c(F)c1F N1(C(c2ccc(C)o2)=O)CCN(C(=O)CC2CC(C3CC3)=NO2)C(CF)C1 C1(CNC(C(C)CN(C)C)=O)CN(C(=O)Cc2nncn2C)C2COCC2O1 c1(CCNC(C2CCN(CC(C(C)(C)C)O)CC2)=O)cccc(F)c1F c1(C(=O)N(C(c2ccccc2)C(=O)NCC(F)(F)F)CCO)ccnn1CC(F)F CC(C(C(=O)NC1CCCCC1)N1CCC(CCC2CC2)C1)C1CC1 n1(CC(N2C(CNC(CNC=O)=O)C=CC2)=O)c(S)nc2ccccc2c1=O c1(OC)cc(C(N2CCC(C(C)CNC(=O)CCCCC#N)CC2)=O)ccc1Cl c1(C(=O)NC2CCCC(NC(C3CCOC3C(F)(F)F)=O)C2)csc2nnsc12 Cc1ccc(F)cc1C(N1C(CNC(=O)Cc2ccccc2F)CC2CC12)=O c1(CC(N2CCC(NC(C(C)(C)SC)=O)C(F)C2)=O)ccc2c(c1)COCC2 c1(C(C(=O)NC2(COC)CN(C(=O)CCC(C)(C)C)C2)C)cccc(C#N)c1 C(=O)(CC(C)(C)CC(C)=O)N1C(CCNC(C=C(C)C2CC2)=O)CSCC1 c1(C(N(CC(C)CNC(=O)Cc2cnnn2C)C)=O)cccc(C#CCO)c1 N1(C(CCc2c(C)ncs2)=O)CCCC(C(=O)NCc2ccc(N)cc2Cl)CC1 C(CCS(=O)(=O)c1cccc(C)c1)NC(COCCC)C C1(C(N(CCC(=O)NC)C)=O)CC2CCN(C(C3CCC=CO3)=O)CC12 Nc1ccc(Br)c(C(=O)NCc2cn(-c3ccc(Cl)cc3Cl)nn2)c1F N1(C(Cc2c(C)scc2)=O)CCC(C)C(NC(c2c[nH]nc2-c2ccoc2)=O)C1 C1(NC(C2(CC=C)COC2)=O)CCC(C)N(C(c2scnc2C(F)(F)F)=O)C1 N1(C(CC)=O)CSCC1C(=O)NC1CCN(C(C2(C(=O)N(C)C(C)C)CC2)=O)C1 c1(C(=O)OC)cnc(Cl)cc1NC(C1(C)CCN1c1cc(OC)ncn1)=O CC1(c2cn(CC3CC(NC(c4cc(Br)n[nH]4)=O)C3)nn2)CCCC1 C(C(C(=O)NCC1COCCN1C(=O)CCn1nc(C)cc1C)C(F)(F)F)OC C1(C(=O)NC(CC)CCOC)(CC)CCN(C(=O)Cc2cc(C)on2)C1 C1(NC(CCCNC(C)=O)=O)CCN(C(C2CN(C(N)=O)C2)=O)C(C)C1 c1(OC)ccc2c(c1)C(Nc1ccc(Cl)c(C(F)F)c1)CC2 C1(CC(=O)NC(c2c(C)nn(C)c2)C)CCN(C(=O)C=CCO)C(C)(C)C1 C1(C(=O)NCC(COC)(O)CO)CCN(C(=O)Cc2ccsc2)CCO1 Cc1cnncc1C(N1CCCCC1C(C)NC(=O)COCc1ccnn1C)=O C1(CCC)CN(C(=O)C(C)CC#N)CC1NC(C1CC(C)=NO1)=O c1(C(C)=O)ccnc(-n2cc(CCCCNC(=O)CC3CCCN(C)C3)nn2)c1 c1(C(N2CCC(N(C)C(C3CC3c3cccs3)=O)C2)=O)cnc2sccn2c1=O N1(C(C2CCN(C)CC2)=O)CCC2CN(CC3CCC3)CC2CC1 C1(CN(C)C(c2cc(C#N)on2)=O)COCCN1C(c1ccc(CO)o1)=O c1(CN2CCCC(C(=O)Nc3ncc(C)s3)C2)cc(S(N)(=O)=O)cc([N+](=O)[O-])c1Cl N1(C(CC2C(C)CCO2)=O)C2CCC1CN(C(c1ccc(C3CC3)nc1)=O)C2 N1(C(C2CC(CNC(C(CC)SC)=O)C2)=O)CCC12CCCC2 c1(CN2C(C(N3CC=CC(NC(C=C(C)C)=O)C3)=O)CCC2)ccc(C#N)cc1 N1(C(CC(C=C)(C)C)=O)CCC2CN(C(=O)CC(C)NC(c3ccccc3)=O)C2C1 Cc1nc(N2CC(NC(=O)CC(C)C3CC3)CC3(CC3)C2)cc(C#N)n1 C1(C(N(CCCSC)CCO)=O)CCN(C(=O)c2cccn2C)O1 c1(OCC)oc(C)nc1C(=O)N(CCC(C)NC(=O)Cn1cc(CO)nn1)C C1(C(=O)Nn2cc(CCN3CCCC3)nn2)CCC(c2nn[nH]n2)CC1 C1(CCOC)(CO)CCN(C(=NCc2ccc(F)cc2)NCC2COC(=O)N2)C1 N(C1CN(C(c2cc(CO)n(C)n2)=O)Cc2ccccc21)C(C(CC=CC)C)=O C(=O)(C(C)(C)CC(C)C)NCC(CC)NC(=O)C(N1CCCC1)C1CC1 C1(C(N2C(CC=C)CCC2)=O)CNCCS(=O)(=O)C1 c1(C(N(C(C)C)CCN(C)C(C2CCC(=O)NC2=O)=O)=O)cccc2c1OCC2 C1(NC(C(=O)N(CC(c2ccccc2)CC)CCOC)=O)CCC(=O)N1C CC(C)(CC(=O)N1CCOCC1CCNC(=O)CNC(c1ccoc1)=O)C(F)F C1(C(=O)OC)C2CN(C(C3CCCN(C(=O)C(C)SC)C3)=O)CC12 c1(OC)cc(C(N2CC(NC(=O)C(O)CF)CC(C)C2)=O)ccc1C C1(NC(CC2(C=C)CN(C(C3CSC3)=O)C2)=O)C=CC(C)(C)CC1 Cc1c(C(N2CCC(CNC(=O)C3=NOC(C)(C)C3)C(C)C2)=O)cc(O)cc1N C(CCC(F)(F)F)(C(=O)NCC1CCC(F)(F)CC1F)NC(C)=O CCC(C)C(O)C(=O)NCc1cccc(CN(C)C(c2cnc(CC)nc2)=O)c1 Cc1cc(F)c(NC(=O)CC(C(C)(C)C)NC(=O)Cc2ccoc2)cc1F Cc1c(-c2cn(CC(N3CCC3c3cccc(F)c3)=O)nn2)cccc1F C1(NC(C(C)OCC)=O)CCCCCC1C(=O)NCC(C)(C)N1CCCC1 C1(C)(C(N2CCC(C(C)NC(=O)CC3COC(=O)C3)C2)=O)CCC(F)(F)CC1 Cc1nc(C)c(C(C)NC(=O)CCN(C(c2ncccc2C)=O)CC2CC2)[nH]1 C(=O)(C1CCCc2nn[nH]c21)NCCC(CNC(C(C)SC)=O)(C)C N1(C(CN(C2CC2)CC)=O)CC2(CCCN(C(=O)Cc3cnc(C4CC4)[nH]3)C2)C1 c1(CSC(C)C(C(=O)OCC2CC2)NS(C)(=O)=O)ccc(F)c2occc12 C1(NC(CCc2onc(C)n2)=O)CCN(C(C2CC(CO)N(C)C2)=O)C(C)C1 N1(C(C(C)C#N)=O)CCC(C)(C)C(NC(c2cccc(Br)c2F)=O)C1 C(=O)(C1CCCc2nn[nH]c21)N1C(CCNC(C=CCN(C)C)=O)CSCC1 n1(CC)ccc(C(=O)NC2CC2CNC(=O)CSc2ccc(C(C)=O)cc2)c1C CC1CN(C(c2cnsn2)=O)CCN1C(C12COCC1C2)=O c1(OC)c(C(N2CCN(C(C3CC4C=CC3C4)=O)C(CO)C2)=O)cccc1Br C(CC(F)(F)F)OCC(=O)NCC1COC(CN(C(=O)C(F)=CCCF)C2CC2)C1 c1(C(=O)NC2CC(NC(C3N(C)CCCCC3)=O)CC2O)noc2c1CCCC2 c1(C(=O)NCC2(C(N)=O)CN(C(c3ccc(C(F)F)s3)=O)C2)cc(O)ncn1 C1(NC(CC(c2ccc(F)cc2)C)=O)CCC(Nc2cc(F)ncn2)CC1 n1(CC)nnc2c1CCN(C(C1CC(C3CCNCC3)C1)=O)C2 c1(C(=O)NC2CCCC(NC(C=CC)=O)C2)cccc2c(C)[nH]nc12 C(=O)(CCCS(C)(=O)=O)Nc1cnc(Nc2ccc(CC)cc2)nc1 N1(C(C)=O)CCC(NC(=O)NCCN(C)CCc2cccs2)C(Br)=C(F)C1 CC1CCN(C(C2CC(=O)N(C3CC3)C2)=O)CCN1C(C12CC1COC2(C)C)=O C1(CC(=O)NCC(CNC(c2[nH]cc(CN(C)C)c2)=O)O)CCCN(C)C1 N1(C(CCc2cc(C)sc2C)=O)CC2(C1)CN(C(=O)C(C)c1ccsc1)C2 c1(NC(C23CCC(CC2NC(C2CC(C4CC4)C2)=O)C3)=O)cccc2c1OCC2 CC1(CNC(=O)C=Cc2ccccn2)COCCN(C(c2ccsc2Cl)=O)C1 C1(CC(=O)NCCCNC(=O)C=Cc2cc[nH]n2)CC(O)C12CCC2 C1(CNCC2(C(=O)OCC)CCCC2)CCc2cnn(C)c2C1 CC1CCCCC1(CNC(c1cc(F)cnc1O)=O)NC(=O)C=Cc1cocn1 N1(C(C2(COC)CC2)=O)CCCC12CCN(C(c1sc(C3CC3)nc1C)=O)CC2 C1(CNC(C(c2cccnc2)C)=O)CCC(NC(=O)CCc2cnn(C)c2)CC1 CC1OC(C)C(C(N2CCN(C(=O)CCCCF)CC2CCO)=O)C1C CC(C)C(C(=O)NCC(O)CNC(=O)C=Cc1cc[nH]n1)C1CCCCC1 c1(CNC(C)=O)ccc(C(=O)NCC2(NC(=O)CCC=C(C)C)CCOC2)[nH]1 Cc1cc(S(N)(=O)=O)oc1C(=O)NC1(C)CC(NC(c2ncsc2C)=O)C1 C1(CC#C)(C(=O)NCCn2ncccc2=O)CCN(C(=O)COCCF)C1 c1(C(=O)NC2CC2NC(c2cccc(Cl)c2Cl)=O)cn2cc(F)ccc2n1 C(=O)(C(C(=O)NCC#CCNC(=O)CC(c1ccc(F)cc1)C)OC)OCC C1(CN(C(C(c2ccn(C)c2)C)=O)C)COCCN1C(=O)C(O)c1ccsc1 c1(C(=O)NCC23CC(NC(c4c(OC)c(Cl)sc4)=O)(C2)C3)cnc2ccnn2c1 c1(C(N2CC(C#N)C(NC(c3ccc(Br)c(Br)c3)=O)C2)=O)cccc2c1CCC2 Cc1cc(O)cc(=O)n1CC(N1CCC(C2(NC(=O)C(C)CN(C)C)CC2)C1)=O C12(C(=O)NC3CCN(C(c4ccc(Br)o4)=O)C3)CCCCC1CC(F)(F)C2 N1(C(C(C)c2ncco2)=O)CCCC(CNC(c2nn(C)nc2Br)=O)CC1 CC(CCC(C)(C)C)C(=O)NC(CC(F)F)C(=O)NC1Cc2ccccc2C1 C(CCCC(=O)NC(C)CF)n1cc(COc2cccc(O)c2)nn1.CC(N)CS N1(C(c2sc(Br)nc2C)C(=O)NCCOCC)CCN(C)CC12CCCCC2 N1(C(C(C)=C2CCC2)=O)CC(C)C(NC(c2ccc(C)nc2)=O)C(C)C1 C1(C(=O)NCCC(C=C)C)C(CC)CCN1C(c1sccc1CO)=O CCC(C)C(C(=O)NCC1CC(NC(C2(OC)CCC2)=O)C1)OC CC1OC2(C)CC1(C(=O)NCC1(C(N)=O)CN(C(c3cc(C(N)=O)cs3)=O)C1)C2 C1(CNC(C2(NC(C)=O)CCCC2)=O)CC2CC1CN2C(=O)Cc1cccnc1 CC1CC(F)(F)CCN1C(=O)C(CNC(c1cccs1)=O)C(C)(C)C N1(C(c2c(C)con2)=O)CCC(NC(COOc2cccc(O)c2)=O)CC1.C C(CN=C(NC1CC1)NC)(c1ccccc1-c1ccccc1)N1CCOC1=O.CO c1(C(N2CCCC(NC(CC(CCC)C)=O)CC2)=O)c(N)ccc(F)c1F C(CCC(=O)NOOCOC)(C(C)C)N(C(C1CCCN(CC)C1)=O)CC C1(CNC(C(c2scc(C)n2)C)=O)(NC(=O)CC2OCCC2C)CCCCC1 C1(OCCCOC)CCN(C(=NCC(C)C)NCC(c2nc(C)cs2)C)CC1 Cc1cc(=N)[nH]c(=NCc2cc(C(C)(C)C)cc(O)c2)[nH]1 Cc1ccc2c(C(=O)NC3CN(C(=O)CCc4ccn(C)n4)CC3F)n[nH]c2c1 c1(C(=O)NCC2(CNC=O)CC2)cccc(Cl)c1.C1(C2CCCO2)(CN)CCCC1 C1(CCCC)CCCC1NC(=O)N(CC(CO)OC)CC CC(O)CC(C)CN=c1[nH]c(N2CCc3cc(F)ccc3C2)nc2c1COCC2 C1(C(=O)NC2(O)CC2)C2Cc3c(Cl)cccc3C12.N#Cc1ccc(NC=O)nc1 N1(C(CC(=O)NC)=O)CCN(C(C2(COC)CCCCC2)=O)CC1CC(F)F N1(C(c2cccc(C(N)=O)c2)=O)CCN(C(c2cc(C(F)(F)F)c[nH]2)=O)C2CC12 C1(CC)CN(C(=O)CSC2CCS(=O)(=O)C2)CCN1C(C1CCSC1)=O C=CC1OCCC1C(=O)NCCN(C(=O)C(c1cccc(Cl)c1)(C)O)CC N1(C(C(C)(c2ccccc2)OC)=O)CCCC(N(C(=O)Cn2nnc(C)n2)C)C1 C(=O)(C1=CC2(CCOC2)C1)NC(C1(O)CCCCC1)C(=O)NC(C)CF C(c1ccccc1Cl)=CC(=O)N(C)CC1N(C(C2CCC(C)O2)=O)CCCC1 C(=O)(CCCCCCN=[N+]=[N-])N1CCC(C(C)NC(CC(CCC)O)=O)C1 c1(C(C(=O)NCCCSCC)N(CC)Cc2cccnc2)cccc(CC(N)=O)c1 c1(C(=O)NCCC2OCCN(C(CCC)=O)C2)nn(C)c(C(F)F)c1Cl C1(C(N(CC(C)C)CCC)=O)CC(C)CN(C(=O)CC2CCC(=O)N2C)C1 C1(NC(CCN(C)CC)=O)C(C)(C)CN(C(=O)C2=NOCC2)CC1(C)C c1(C(N(CCC)CCNC(c2ncc(F)cc2C)=O)=O)cc(S(C)(=O)=O)co1 c1(C(=O)NC2CC2NC(C2CC2(Cl)Cl)=O)cc(Cl)ccn1 c1(C(N2C(CNC(C3CCN(C)C3=O)=O)CCCC2)=O)ccc2nnn(O)c2c1 CCC(C(=O)NCC1(C(=O)N(CCCC(C)O)C)CC1)n1cncn1 c1(C(=O)NC2CC(NC(c3c(Cl)cnc(C)n3)=O)C2)ccc2c(c1)CCCCN2 C(=O)(CCC(CF)CF)NC1C(CC)CN(C(c2nnccc2C)=O)CC1 c1(CNC(Cc2ccccc2)C2CC2)cc(N2CCCC2)ncn1 CCCCC(C(=O)NCCCCC1CC1)NC(c1cnc(C2CC2)o1)=O c1(C(N(CCCCNC(C(CC)(C)F)=O)C)=O)cnn2c1NCCC2C(F)(F)F c1(C2(C(N3CC(NC(CSCC(=O)OC)=O)C(C)C3)=O)CC2)ccc(C)c(C)c1 Cc1cc(C=CC(N2CC(NC(C3NC(=O)CC3C)=O)C2)=O)ccc1OC(C)C C1(C)(NC(c2n(C)nnc2)=O)CCC(NC(=O)CSc2ccccc2Cl)CC1 c1(C(=O)NCC2CCN(C(C(C)CN(C)C)=O)C2(C)C)cn(C)c(=O)n(C)c1=O C1(CCOC)CN(C(=O)N(C)C(C2CCCC2)C)CCO1 c1(C(=O)NCC(CNC(C2(CC#C)CCCOC2)=O)C)ccc(C(C)C)nc1C C1(NC(C2(CC=C)CCC2)=O)CC2CCC1N(C(c1c(C)cc(C)nc1O)=O)C2 N1(C(C)=O)CCc2cc(C(=O)N(C(C)CNC(=O)C=CC3CCCC3)C)ccc21 Nc1c(C(=O)NCC2CC(NC(=O)C(F)C3CCOC3)C2)cc(F)cc1Cl N1(c2cc(C)c(C#N)cn2)CCC2CC(NC(=O)CCn3cccn3)CCC2C1 n1(COC)cc(C(F)(F)F)cc(C(=O)O)c1=O.C(C(C)(C)CNC(C)(C)C)NC=O C1(NC(NN(C)C)=O)CCN(C(c2ccoc2C23COC(C(F)(F)F)(C2)C3)=O)CC1 C(=O)(C(C)(C)CS(C)(=O)=O)N(C(CNC(CCSCCCC)=O)C)C1CC1 c1(C(=O)NC(CN(C(c2ccc(OCC)cc2)=O)C)C)cncc(C)c1Cl N1(C(c2nc(C)nc(=N)[nH]2)=O)CC2CN(C(=O)NC3CCC(C)CC3)CC2(C)C1 c1(OC)cc(Cl)cc2cc(C(=O)NC3CCC(NC(=O)CSC4CC4)CC3)oc12 CCC(O)CC(=O)NCC=CCNC(=O)CC(n1nc(C)cc1C)C N1(C(=O)Cc2cncnc2O)CC2CCC(C1)N2C(c1cnc(O)s1)=O C(=O)(CC(C)(C)C#N)NCC(CN(C(=O)C(F)C1CCOC1)C)(C)C C(=O)(C(CCCCN)N(C)C)NCCCCC N1(C(C(CC)OC)=O)CCC(O)C1C(=O)N(C)C.N12CCC(C1)CC2=O C1(CNC(CCCCCNC(C)=O)=O)CCC2(CN(C(c3ncc(C)o3)C)C2)O1 c1(C(=O)NCCCN(C(C(C)OCCCOC)=O)CC)ccc([N+](=O)[O-])nc1C CC1CCCC1N=c1nc(N2CCC3(CCC(=O)NC3)C2)c2cccc(F)c2[nH]1 CC1CCCCN1CC(=O)NC1CC(C)(NC(C2CC2C(F)F)=O)C1 c1(OC)ccc(C(=O)NCC2(CNC(=O)C(C)(C(C)C)OC)CC2(F)F)c(O)c1 S(=O)(=O)(c1ccc(N2CCn3ncc(Cl)c3C2)c(F)c1)NCCSCC N#Cc1cncc(CN2CC(NC(=O)CCc3ccccc3)C2)c1 CCC(C)C(O)C(=O)N1CCC(C)(NC(C2CCN(C)CC2)=O)CC1 c1(C(=O)NC2(COC)CCC2)cc(NC(=O)C(C)(O)C2CC2)ccc1N CC1CN(C(C2(C3CC3)CN(C(=O)C=CC3CCOCC3)C2)=O)CCC1CO c1(C(N(CCNC(C(COCC)C)=O)CCOC)=O)ccc(Cl)c(C)c1 CC1C(=O)CC1C(=O)N(CCCN(C)C)CCNC(=O)CC1(C(F)(F)F)CC1 c1(C(C)NC(C(=O)NC2N(C(C)=O)CC2C)=O)ccc2c(c1)n(C)c(=O)n2C c1(OC)oc(C)nc1C(=O)NCC1CC(NC(C2CCCO2)=O)CC1O C(c1cc2ccccc2o1)=CC(=O)NC1(C(=O)NCC(CCC)(C)OCC)CC1 C1(OC)(CNC(=O)CC2CC(CC)=NO2)CCN(C(=O)CCc2n[nH]c(=N)s2)C1 c1(NCC2CN(C(=O)OC(C)(C)C)C3CCN2C3)cc(F)c2ncccc2c1 c1(NC(CC)=O)ccccc1NCC(C)CN(C(=O)CCOC(C)CC(C)C)C c1(CC(N2C(C(N(CC(C)C#N)C)=O)CC2)=O)ccc(C#N)cc1 c1(C(=O)NCC2COCC2NC(=O)C(F)(F)CO)n[nH]c2c1NCCC2 CC1CN(C(=O)C=CBr)CCC12CCN(C(C1CCCC(F)(F)C1)=O)CC2 c1(OC(C2C3CN(C(=O)OC(C)(C)C)CC32)=O)cccc2cncc(F)c12 CCC1=C(C(=O)NCC2CCCN2C(c2cc3c(C)cccn3c2)=O)CCCO1 C1(CC(=O)Nc2cccc(CCC)c2)C2CCCC2N1C(=O)CS(=O)(=O)CC C1(C(N2CC(C(C)(C)NC(=O)CC3CCOCC3)C2)=O)C2CCCOC12 N1(C(c2cc(OC)n[nH]2)=O)CCOC2(C1)CN(C(c1ccc3nc[nH]c3c1)=O)C2 C=Cc1ccc(C(=O)NC2(C)CCN(C(=O)CN3CCC(=O)CC3)C2)cc1 c1(-n2c(C3CCCCN3C)nc(C(CC)O)n2)ccc(O)c(C)c1 N1(C(Cc2n(CC)cnn2)=O)CCC2(CC1)CC(Nc1ncc3ncnc-3[nH]1)CO2 N1C(=NCC2CCCC2)NCC2(CCCCC2)CC1.Cn1cnc(C(C)(C)C)n1 C1(NC(CC2C(C)CN(C(C3CC(O)C(F)C3)=O)C2)=O)CN(C)CCC1O c1(C(CC)NC2C=CCCC2)nccc(=NCc2ccc(COC)cc2)[nH]1 Cc1c(C(=O)N(C2CCN(C(c3ccn(C)c3C3CCC3)=O)C2)C)cccc1O c1(C(=O)NCC2C(CNC(C(CCC#C)O)=O)C2)cc2cccnc2o1 N1(C(C(CCC)CC)=O)CC2CCCC(CNC(=O)C(C)(C)CN(C)C)(C2)C1 CCC(CNC(=O)C(N1CCC(Cc2nc(CC(C)C)no2)CC1)=O)(CC)CC c1(CCC(=O)NC(C2CCN(C(C(C)C3CCOC3)=O)C2)C)cccnc1F n1(CC(=O)N(CC(C)NC(c2ccc(O)nn2)=O)CC)cnc2c1CCCC2 c1(CNC(C2CCC(n3cc(Cc4nn[nH]n4)nn3)C2)=O)c(Cl)cccc1Cl c1(C(N2CCC(N(C(CC=C)=O)C)CC2)=O)[nH]c(=N)ccc1C Cc1cc(C)c(C(=O)NCC2CC3CCC(C2)N3C(=O)CC(C)(C)C)c(C)c1 c1(SC)cc(NC(C2CNCCOC2CO)=O)ccc1C Cc1ccc(CC(=O)NC(C2CC2C(=O)N(C)CC2CCCCC2)C)o1 NC(=O)CCCCC(=O)NC1CCCN(C(=O)C(c2ccccc2)O)C1 c1(CC(N2CC(F)(C(=O)NCCCCOC(C)C)C2)=O)ccc(Cl)cc1 CCC(CC)CC(=O)N1CCN(C(C2CCCN(C(=O)COCCF)C2)=O)CC1 c1(CCC(=O)NCCN(C(CCC#C)=O)CC)cc(Br)cc(OC)c1OC C(=O)(CCC1=CCCCC1)N(CCC(=O)NCCCC1CC1)CCc1nncs1 N1(C(c2cc(C)sn2)=O)CC(NC(=O)COCCCF)C(C2CCCO2)C1 C1(C(=O)OC)CN(C(C2CC(F)CN2C(c2c(Cl)cccc2I)=O)=O)CC(=O)N1 C#CC1(O)CCN(C(=O)CC2(CNC(c3ccc(F)cn3)=O)CC2)CC1 c1(C(N2CCC(NC(CC(C=C)(C)C)=O)C(O)C2)=O)ccc(F)c(OC)c1F C1(NC(c2cncc(C(=O)OC)c2)=O)CC2(C1)CC(NC(=O)C(C)C(C)(F)F)C2 N1(C(c2c(C(C)C)ncs2)=O)CCC(CNC(C2(C)CCCCO2)=O)C(F)(F)C1 C(CC(CC)C(=O)NC1CCOC1C(=O)NCC(C)(O)CO)=CC c1(C(=O)OCC)cc2n(n1)CCN(C(C1CCCCCC1)C(=O)NC(C)CC)C2 C(=O)(C(O)CCc1ccccc1)Cc1cn(CCNC(C2C(C)C2)=O)nn1 c1(CC)cccc(C(=O)NC(CC2CCC2)C(=O)NCCNC(C)=O)c1 N1(C(C(C)=C(C)C)=O)CCC2(CC1)CN(C(C1CC3CCCC13)=O)CCO2 N1(C(CCCc2nc(C)sc2)=O)CCN(C(C2CC(S(C)(=O)=O)C2)=O)CC1C c1(C(=O)NC2CC(CCNC(CC=C=C)=O)C2)cnccc1-c1ccncc1 N1(C(Cc2cn(CC)nn2)=O)CC(NC(c2c[nH]c(C)c2)=O)CC(F)C1 N1(C(C(C)n2cncn2)=O)CCC2(NC(=O)CCc3ncccn3)CCCC12 c1(CNC(C2CC3CC3N2Cc2cccc(O)c2F)=O)cccc2ccccc12 C(=O)(C(CCN(C)C)NC(C1CC=CC(O)C1)=O)NC(C)Cn1cccn1 N1(C(C2(C)CC(F)(F)C2)=O)CC2(CO)CC1(C(=O)NCCc1cc[nH]n1)C2 C1(S(=O)(=O)NC(C2CCCC2)C2CCC2)(C(=O)OC)CCC1 c1(C(=O)NC(C)CCNC(C2CCC3CC3CC2)=O)cc(O)cc(F)c1F C#CCC(C(=O)NCc1ccc(C(N)=O)o1)NC(=O)CC(C)=C=C N1(c2nc(C)nc(O)c2)CC(CNC(c2cccn(C3CC3)c2=O)=O)OC(C)(C)C1 N1(C(c2c(C)ocn2)=O)CCC2CN(C(=O)Cc3cccc(N(C)C)c3)CCC12 n1(C)cc(C(C)(C)OC)nn1.C1(C(CC)NC(C2CCS2(=O)=O)=O)CCCCO1 CCCCCCCCCCNCc1ccnc(OC)c1Br c1(CCS(=O)(=O)C2C(c3nnc(C)o3)C2)ccc(F)c(F)c1 CC(C(=O)NCC(O)CN(C(=O)CCC1OCCO1)C)NC(=O)C1CC1 C1(NC(C=CC(CC)=CC)=O)CCC2(CCN(C(=O)Cc3nc(=N)[nH][nH]3)CC2)C1 N1(CC(=O)NC(c2nnc(C(F)F)o2)C)CCCN(Cc2ccccn2)CC1 C1(C(N2CCC(NC(C(c3n(C)ncc3)O)=O)CC2)=O)CCCCCS1(=O)=O c1(NC)ccc(CCC(=O)NC(C)CNC(=O)Cn2cc(Br)c(C)n2)cn1 c1(CC)c(C(=O)NC2(COC)CN(C(c3cc(C(C)(C)C)c[nH]3)=O)C2)cnn1C c1(C(N2CC3CC3(C(=O)NC3CONC3=O)C2)=O)ccc(Cl)cc1I C1(c2nnc(C(=O)OCC)s2)CCCN(C(c2nnc(C)s2)=O)C1 O=[N+]([O-])c1cccc(Cl)c1CNc1ccnn1CO c1(N(CC)CCO)ccc2sccc2c1.CCCC(O)CC(=O)OCCO C(=O)(CCC(=O)NCC1C(O)C(O)CN1C(=O)CC1CC(=O)NC1=O)NCCC Cc1cc(C(=O)NC2CC(F)CN(C(C3(N(C)C)CCCSC3)=O)C2)cnc1O CCCCCC(F)C(=O)NCC1(C(=O)N(C)Cc2cccnc2)CC12CCC2 C1(CC)(NC(=O)CCn2cc(Cl)cn2)CCCN(C(=O)C(=Cc2c[nH]cn2)F)C1 N1(C(CCCC)=O)CC2CC(NC(c3cccc(NS(C)(=O)=O)c3)=O)C(C2)C1 N1(C(c2c(N)ccc(Cl)n2)=O)CC2CCCC2(NC(c2ccn3c2CSCC3)=O)C1 N1(C(c2ncn(CC)n2)=O)CCC2(CCCN2C(=O)Cn2nnnc2C(C)C)C1 c1(OC)cc(-c2cccc(C(=O)NCCN3CCN(C)CC3)n2)ccc1[N+](=O)[O-] C(CC(=O)NC1(CO)CN(C(c2cc(=N)[nH]c(Cl)n2)=O)C1)(C(C)C)OCC c1(C(N2CC3CN(C(C4CCOC4)=O)CC32)=O)cccc2nc[nH]c12 C1(CNC(=O)CC(O)C2CC2)CC(F)CN1C(=O)COCc1ccccc1 N1(N(c2ccon2)C)CC(CC(N2CC(N3CCC3)C2)=O)CC1(C)C Cn1cc2c(n1)CCN(c1cc(NC3CN=CN(c4ccccc4)C3)ncn1)C2 CC(C)(C)S(=O)(=O)CC(=O)NCC(F)CNC(c1ncoc1CCC(F)(F)F)=O c1(CC(=O)NC(C)CNC(=O)Cc2cnns2)nccn1C c1(OC)cc(N2CCCCC2)ccc1-c1ccccc1CC(N1CCC1CO)=O n1(CCOC)ncc(C(=O)NCCC(O)CNC(C2(COC)CCOC2)=O)c1C C1(C(N(C2CS(=O)(=O)CC2O)C)=O)N(Cc2ccccc2)CCCC1(C)C c1(OC)cc(-c2ccc(C(C3CCCCC3)=O)cc2)cc2c1OCC2 N1(C(C2CCC(CC)CC2)=O)CCN(C(=O)CCC(C)(F)F)CC1C1CCC1 CC(N=c1[nH]c(=N)[nH]c(=NCC2(N(C)C)CCCOC2)[nH]1)c1nccn1C C1(C2CN(C(C3CC3CF)=O)C2)(NC(=O)C2=C(Cl)CC2)CC1 N1(C(COCCCCC)=O)CCCC1(C(=O)NCC(C1CC1)CC1CC1)COC C(=O)(CC(CC)C(C)C)N1C(C(N(CCOCC)C)=O)CCCC1 CC(C)(O)CCCNCc1ccc(CC#N)cc1 C1(NC(c2cccc(CC)c2O)=O)CCSC12CN(C(=O)C(F)CC1CCC1)C2 c1(C(=O)NC2CC(NC(c3ccc(=O)oc3)=O)C2)cc2cccnc2nc1O CC(C)C(O)CC(=O)N(C)CCN1CCN(C(C2COCC2C(=O)OC)=O)CC1 n1(C(=O)NCCc2cn(CCO)nn2)nc(C(F)F)cc1C1CC1 c1(C(=O)NC(c2ccc(F)cc2)CNC(CCC2(C)N=N2)=O)ccc(C#N)cn1 CC(C)C(O)CC(=O)NCCC1CCN(C(=O)CC(O)CN(C)C)CC1 N#CC1CCCN(C(C2(F)CCCN(C(c3csc(Cl)n3)=O)C2)=O)C1 N1(C(c2cc(CNC(c3c(C)cc(C)s3)=O)on2)=O)CC(C)C(C)C1C c1(C(=O)NCC2(F)CCC(CNC(C3(C)CC3)=O)C2)nnc(O)cc1O Cc1cc(Br)c(CN(C(c2ccnn2C(F)(F)F)C(=O)NCC2CCCO2)C)s1 C1(NC(C2(C#C)CC2)=O)C2CC3C(C2)C13C(N1CC(=O)NC(C)C1)=O C1(C(=O)NC(CCOC)C(C(=O)CCC(C)CN(C)C)=O)CC2(C1)CC2(F)F c1(CC(=O)NCC2N(C(=O)OC(C)(C)C)CC2)ccc(S(N)(=O)=O)s1 C1(C(=O)NC2(C)CC(N(C)C)C2)CCC(O)CN1C(=O)CC1(C#N)CC1 C1(OC)CN(N2CC3(CC(=O)Nc4ccc(Cl)cc43)C2)C(C)(C(=O)OC)C1 N1(C(CCSCC(=O)OC)=O)CCC(CNC(C23CCC(CC2)O3)=O)C1(C)C CCC(CC)(CCNC(=O)CCCCNC(=O)C(C)C)NC(=O)C(CO)N(C)C N1(C(C2(CC)CC2)=O)CCCC(C2CCN(C(c3cnc(C)[nH]c3=N)=O)C2)C1 N1(C(Cc2n(C)cnc2)=O)CCCCC(CNC(=O)CC2CCC(F)(F)CC2)C1 N1(C(C2C(CC)OCC2)=O)CC(C)OC2(CCN(c3nc(Cl)ncc3Br)CC2)C1 C(CC)(C(=O)N1CCCC1CCC(=O)NCC(C1CC1)C1CC1)OCC N1(C(c2c(NC)nccc2)=O)CCC2(CC2C(=O)NCc2cnc(F)cn2)C1 N1(C(CCOCC(C)C)=O)CCCCC12CC(NC(c1cnnn1C)=O)C2 N1(C(C(C)CC(N)=O)=O)CC2CCCC2(C(N2CCOC(CF)C2)=O)C1 c1(C(=O)NCC2N(C(c3c(C)oc(CO)c3)=O)CCCC2)cnc2ccccc2n1 Cc1nn(C(C)C)c(C)c1CC(N1CC=CC(NC(C2(C)CCCO2)=O)C1)=O Cc1ccc(C(=O)N(C)CCNC(c2ncc(C(C)=O)s2)=O)cc1O.C1CO1 C=CC(C)C(C)C(=O)NCCCOCCOCCNC(c1ccc(C)c(O)n1)=O C(C(C)(CC(C)C)NC(c1cnc(SC)s1)=O)NC(COCCCCC)=O c1(NC(=O)NC(C(c2ccc(Cl)cc2)OC)C)cc(C)c2n[nH]cc2c1 N1(C(CCCOC(C)=O)=O)CC2COCCN(C(c3cc(Cl)nnc3O)=O)C2C1 Cc1cc(C)c(CNC(C2CCOC2CNC(=O)Cc2cccnc2F)=O)cn1 C1(NC(CC(CCC)C)=O)CCN(C(=O)CC2OCCC2C)CCC1CO c1(C(C(=O)NCC2CC2)N(C)CC2CC(C#N)C2)cc2cccc(F)c2o1 C(CC(C(C)(C)C)NC(c1cnn(CCO)c1N)=O)N(C(C(=O)NCC)=O)C c1(OC)ccc(Br)c(CC(N2CCCC(N3CCCS3(=O)=O)C2)=O)c1 CC1=CCC(NC(C2(C)CCCN2C(=O)C(C)C)=O)CC1.C C1(CS(=O)(=O)N(C2(Cc3cccc(Cl)c3)COC2)OC)CCC2CC2C1 c1(C(=O)Nc2c(F)cc(I)cc2F)ccc2c(c1)CCN(Cc1cn[nH]c1)C2 C(CC1=CCCCCC1)N(C)C(c1ccc2cccnn12)=O Nc1ccc2c(c1)CN(C(=O)C(C1CCC(F)(F)C1)O)CCO2 CCCC(CCCNC(c1cc(C)n(C2CC2)n1)=O)NC(c1sccc1Cl)=O C1(NC(C(C=C=C)C)=O)CC2CC(C1)N(C(=O)CSc1nncs1)C2 C(CCCC(C)NC(C1CC2CC2C1)=O)NC(Cc1c(C)non1)=O Cc1ccc(C(=O)NC(C(=O)N(C(C)C(F)F)C)C2CCCC2)cn1 C12(NC(Cc3c(C)noc3)=O)CC3CCC(C1C2)N3C(C1CC(=O)NC1(C)C)=O C(CCC(=O)N(C1CCN(C(=O)Cc2csc(NC=O)n2)C1)CCO)N(C)C C1(NC(C=CC)=O)CCC(O)CN(C(C2CCN(C3CCC3)C2)=O)C1 N1(C(C(CCSC)OC)=O)CCCCC2(C1)CN(C(=O)Cn1nnc(=O)[nH]1)C2 C(Cc1ccccc1)(CCNC(=O)Cn1cc(C)cn1)NC(CC1CC(=C)C1)=O c1(CCC)nc(C(=O)N(CCCNC(=O)C(C)c2cc[nH]n2)C(C)C)co1 N1(C(C)=O)CCC2(CC1)CC2c1nnc(C(F)(F)F)s1.N12CC(=O)NC(C1)C2=O C#Cc1ccc(CNC(C2(CNC(C3CC4CCCC4C3)=O)CC2)=O)cc1 N1(C(CN(C)C)=O)CC2(CCOCC2)CC1CNC(=O)C(C)(C)C1CCOC1 Cc1cc(NC(C2CCN(C(=O)C(O)C(C)(C)C)C23CCC3)=O)cc(C)c1F C(C(CC)(CC)C(=O)N(C1CCC2CC12)C)NC(c1c(CC)n[nH]c1)=O C1(NC(C2CC(C)(C)C2C(F)(F)F)=O)CC(F)CN(C(=O)Cc2cc[nH]n2)C1 N1(C(c2cc(C)oc2C)=O)CCN(C(C2CCCCCC2)=O)C2(CC2)C1 c1(NC2C(CSCC(=O)NC(C)C)CCC2)ccc([N+](=O)[O-])s1 CCCCCC(O)CC(=O)N(CC(O)CN(C)C(c1cnc(C)cc1C)=O)C c1(C(N2C(C3(O)CN(C(c4c(C)nsc4)=O)C3)CCC2)=O)occ2c1CCC2 Cc1cc(CNC(=O)Nc2ccc(OC3(C)CC3)nc2)cc(C)c1 c1(C(C(=O)NCCCCCNC(CCC=CC)=O)(F)F)ccc(OCC)cc1 N1(C(c2cccc(COC)c2)=O)CC2(C)CC1(C(N1CCCC(C)(OC)C1)=O)C2 C(C1CCCN1C)=CC(N1C(C2(C(N(CCC#C)CCO)=O)CC2)CCC1)=O C(=O)(CCCc1csc(C)n1)NCC(CC)NC(c1ccoc1)=O.C1(=O)CN1C C(=O)(CC1=CCCC1)N(C1CN(C(=O)C(C)(C)Nc2ccccn2)CC12CC2)C C=CCCCC(C)(C)C(=O)N1CCCC1CN(C)C(C1CCC(C)(C)O1)=O CC1(C(=O)NC2CCN(Cc3cn(CCN(C)C)nn3)C2)CC(=O)CC(=O)N1 N1(C(CSc2ccc(OCC)cc2)=O)CC2(C1)CN(C(=O)C(CO)OC)CCO2 C(=O)(C(C)=Cn1ccnn1)N1CC(C(COC)CNC(C(CCC)NC(N)=O)=O)C1 N1(C(C2C(C)N(C(C3CC=CCC3)=O)CC2)=O)CCC(C)(O)C(O)C1 C1(CN2CC(C(=O)NC3(c4cc(OC)ncc4)CC3)C2)CCN(C(C)=O)C12CCC2 C1(C(C)C)C(C)CN1C=O.c1(OC)nscc1CCOC CN1CCCCC1C(=O)NC(C(=O)NCC=Cc1ccncc1)C1CC1 C1(CC=C)(NC(=O)C(C)C(C)C)CCCN(C(=O)CCCCCOCC)C1 N1(C(C2(CC)CCCN2C(c2cc(C)on2)=O)=O)CCc2nn[nH]c2C1 C(C(CCO)NC(=O)CC1CCCC1NC(=O)C(C)CC)OC N1(C(C(C)SCC)=O)CCC2C(CCCN2C(c2ccn3c(O)nnc3c2)=O)C1 c1(C(=O)NCC(C)(CNC(C2CCCC2O)=O)OC)ccccc1CO c1(C(=O)NCCCN(C(c2nc(OC)oc2)=O)C2CC2)cc(OC)ccn1 N1(CCNC(=O)C(=O)NCCc2scnc2Cl)CCC(C(F)(F)F)(C(=O)O)C1 C1(C(N(C2CCN(C)C2=O)C)=O)CCCN(C(=O)C(=O)C2CCCC2)CC1 C(=O)(C1CCCc2cncn21)N(C1CN(C(c2c(CC)nc[nH]2)=O)CC1(C)C)C c1(C(=O)NC2CCC(CNC(c3c(C)nc(N)cn3)=O)C2)cc(F)c(F)cc1F c1(CC)cc(C(=O)NCC23CC(NC(c4cnccn4)=O)(C2)C3)cc(O)n1 c1(OC)ccnc(C(=O)NCC(C)(CC(C)C)NC(c2cn(C)nn2)=O)c1OC CC(C)C(C(=O)OC(C)(C)C)C(C)NC(=O)CCC1CN(C(=O)OC(C)(C)C)C1 C1(C(=O)NCC(C)OCC#C)CCN(C(=O)C(F)=CCCF)C1CC C12(C(N3CC(OCc4cn(C(CC=C)CC=C)nn4)C3)=O)CCCN(CCC1)C2 C1(C(N(CC(=O)NC(C#C)C(C)(C)C)CCC)=O)CC2CC(=O)C1O2 N1(C(CC(C=C)(C)C)=O)CCC(C2(NC(=O)C(O)Cc3cnc[nH]3)CC2)C1 c1(C(=O)NCC2N(C(C(C)Cc3cccnc3)=O)CC(O)C2)csc([N+](=O)[O-])c1 Cc1nc2c([nH]1)C(C(=O)N1CCCC1Cn1cc(C3CCN(C)C3)nn1)CCC2 c1(C(C)C)ccc(C=CC(N2CCCC(NC(C3(C)CC4CC4C3)=O)C2)=O)cc1 C1(NC(c2c(CC)ocn2)=O)CN(C(=O)Cc2ccc(C)c(C)c2)C2CCCC12 C1(SCC2(O)CCC(NC(=O)NCCCCC(N)=O)CC2)CCCCC12CC2 C12(CNC(C3CCCCN(C(=O)CC45CCC(CC4)C5)C3)=O)CCN(CC1)CC2 N1(C(=O)CCN(C2CC2)C2CC2)CCOCC1C1CCCC1 C12(NC(C(CCC)OCC)=O)CCCC1CN(C(C1(C)CCCC1)=O)C2 c1(C(=O)NCC(C)NC(C2CC(=O)N(C)C2)=O)cc(F)ccc1Cl CCC1=C(C(=O)N2CCC(C3CC3)(CNC(=O)C(CCOC)OC)C2)SCCO1 CC(CO)CCCNC(=O)C(C1CN(C(N)=O)C1)NC(=O)C(C)(O)C1CC1 C1(C)(C(N(CC(C)NC(=O)CC2CCCN(C)C2)C)=O)CC(=O)N(C)C1 c1(OC)ccc(SCCOCCCNC(c2nnc(S)n2C)=O)cc1.C1C(=O)N1 c1(C(=O)NCC(N2CCN(C(C3C(C)=C3)=O)CC2)=O)ccc(Cl)c(C(F)(F)F)c1 c1(C(=O)NCC2N(C(c3c(C)ccs3)=O)CCC2C2CC2)cc2cccnc2o1 CCC(CNC(C1OCCC1C)=O)(CC)NC(=O)Cc1cccc(C)n1 C1(NC(C2CC3(CCC3O)C2)=O)CCCCCC1C(=O)NCC1(CC2CCC2)CC1 C1(C(=O)NCc2c(C(=O)NCCc3ccc(C)s3)occ2)CCC(F)(F)C1 N1(C(c2ccc(C)cc2C)=O)CCC2CCN(c3ccn4ccnc4n3)CC2C1 C1(NC(C2N(C(C)=O)CCC2)=O)CS(=O)(=O)CC1NC(c1ccc(CO)s1)=O C(=O)(C(Cc1ccccc1)N1CCC(CC(=O)OC(C)C)C1)NCCOC c1(C(=O)NCC(CC=C)NC(c2n[nH]cc2C2CC2)=O)nn(C)c(=O)cc1C c1(SC)ccccc1C(N1CCC1CNC(C1(C)COCCO1)=O)=O C=C=C(C)CC(=O)NC1(CNC(C2CC3CC2C3)=O)CCCC1 CC1(C)NC(=O)N(CCNC2(c3nnc(CS(C)(=O)=O)o3)CCC(=O)N2)C1=O CC1CC2(CCN(C(=O)CC3NC(=O)NC3=O)CC2)CN1C(=O)C(Cl)=CCl Cc1cnc2ccc(C(=O)N(CC(O)CNC(=O)Cc3ccoc3C)C)cn12 C=Cn1ncc(-c2cc(-c3ccc(C)o3)c[nH]2)c1N c1(NS(=O)(=O)CC2CCCCNC2)cnc(C2CC2)cn1 Cc1cccc(S(C)(=O)=O)c1NC(=O)NCC1CCCC1C#N Cc1nc(-c2ccccc2Br)sc1-c1ncc(CN(C2CC3C=CC2O3)C)s1 c1(C(N(CCCNC(=O)CNC(c2cscn2)=O)C)=O)cnc(N)c([N+](=O)[O-])c1 N1(C(C(C=C)OC)=O)Cc2n[nH]cc2C1C(=O)NCCC1CC=CC1 c1(OCCCN2CC3C(C(=O)NCc4ccnc(Cl)c4)C3C2)ccc(F)cc1F c1(C(N2CCN(C(CNC(C3N(CC)CCC3)=O)=O)CC2)=O)cccc(F)c1N c1(CC)oc(C)cc1C(N1CC2C(NC(=O)Cc3ncc(C)s3)C2C1)=O C1(C(=O)NCC2CN(C(c3c(CC)ocn3)=O)CC2C)CC2(CC2)CN1C N1(C(=O)C=Cc2cccnc2)CCC2CN(C(C3CCC3CF)=O)CCC12 N1(C(c2cccnc2Nc2cccnc2)=O)CCC2(CC1)OCC1CC21 C1(c2n(CC=C)nnn2)(NCC2CC(F)C2)CCN(c2ccncc2)CC1 c1(NC(C2N(C(C(CC(C)C)O)=O)CCCC2)=O)ccc2[nH]ccc2n1 C1(CCC)(NC(=O)CCC2CCCCC2)CCCN(C(=O)Cc2cc[nH]n2)C1 C(=O)(CCCCCC#N)N1CC(O)(C(C)NC(=O)CSCc2cccnc2)C1 C1(NC(C(CC2CC2)OC)=O)CC2CC1N(C(c1n[nH]cc1F)=O)C2 C(=O)(CCCCCC)NC1C(CNC(C(C)OCCC#C)=O)CC1 c1(C(N2CC(O)(C(C)NC(C3CC(Cl)(Cl)C3)=O)C2)=O)c(Cl)ccc(Cl)c1O c1(C(=O)NCCC2(C)CCN(C(c3c(C)snc3)=O)C2)c(O)ccc(F)c1F C1(C(NOCc2nc(C)[nH]n2)=O)(NC(=O)C=Cc2cc[nH]c2)CCC(C)(C)C1 c1(NCC2(OCC=C)CCCC2)ccc2c(c1)CCCC2(C)C C1(C(=O)NC(C)CC(F)(F)F)N(C(=O)OC(C)(C)C)CCC1(C)C Cc1ccc2c(c1)SC(C(N1CCC(C3(NC(c4ncn(C)n4)=O)CC3)C1)=O)C2 O=S1(=O)CC(C2(NCc3cccc(O)c3)CCCC2)c2ccccc21 C1(OCC)CC2CN(C(=O)CC3CC(C)N(C(=O)C(C)CO)C3)CC12 C(CCNC(c1ccc(-c2ccc(F)cc2)[nH]1)=O)(C(C)C)NC(C1C(=C)CC1)=O CCCCS(=O)(=O)NC(C)C(=O)NCC(O)CNC(c1cnn(CC(F)F)c1C)=O Cc1cn2nc(C(=O)NC34CC(CO)(C3)C4)cc2c(=O)[nH]1.C123CC(C1)N(C2)C3=O CC1(C)CC(CO)CN1C(c1cccc(Cn2cc(Cn3ccnc3)nn2)c1)=O Cc1cc(C#N)ccc1C(N1CCC(NC(=O)C(F)(F)CC2CC2)C(O)C1)=O CC1CCCCC1CC(=O)N(C(C=CC)=O)C.C1CCN(N2CCCC2)C1 C=C(C)CC(C(=O)NC(C(=O)NCC1CCC(=C)CC1)C1CC1)OC c1(C(N2CC(N(C(CC)=O)C)C2)=O)cc(S(N)(=O)=O)ccc1Br C1(C(=O)Nc2c(C(=O)OCC)cccc2)CC2(CC(NC(=O)C(C)OC)C2)C1 c1(C(N2CC3CC3(NC(C3CC3C(N)=O)=O)C2)=O)cnc(C(F)(F)F)nc1 N1(C(c2c(CCC)n(C)nc2)=O)CCN(C(C2COCC(C)O2)=O)C2(CC2)C1 CCCCC(C)C(=O)N(C(C)CN(C)C(c1ccccc1-n1nccn1)=O)C C12(NC(C(CC)NC(C)=O)=O)CC(C)(C1)OC21CN(C(=O)C(O)CF)C1 C1(OC)(CNC(c2onc(C)c2C)=O)CCN(C(c2csc(C(F)(F)F)c2)=O)C1 c1(C(=O)NCC(C)(CNC(=O)CC2CC3CC3C2)OCC)cc(C(C)C)oc1C CC1(C)CC(C(=O)N2CCC(CN=c3[nH]nc(C(C)(C)OC)s3)C2)=NO1 c1(C(=O)NC2(CNC(Cc3cccc(N)c3)=O)CCOC2)ccc(F)c(Br)c1 C12(OC)CCCCC(C(=O)NC3(CNC(C4COC(=O)O4)=O)CCOCC3)(C1)C2 c1(C(=O)NC(C)CN2CCN(C(=O)CCC3CC3C)CC2)ccc(=O)n(C)c1 c1(C(N2CC=CC(NC(CN(C3CCSC3)C)=O)C2)=O)cc2c(nn1)CCCC2 C(=O)(CC(C)CC(=O)NCC1(C)CCC(NC(c2cnc(C)o2)=O)CC1)OC Cc1noc(C(C)NC(=O)CC2CCCN2C(=O)CNC2CCOCC2)n1 C1(CNC(C2(C(=O)OCC)CCC2)=O)C(C)CCCN1C(=O)C1=CSCCO1 C1(C(N(C)CC2(CNC(C(C3CC3)OC)=O)CC2)=O)CCCN1CC(C)C C1(CNC(C(=O)N(C2CCC(C)C2)C)=O)CC(CN)C12CCC2 c1(C(N2CCC(CCC(N3C(COC)CCCC3)=O)C2)=O)cccc2c[nH]nc12 N1(C(CC(C)C(C)(C)NC(C2C3CCC(=O)C23)=O)=O)CCC2(CNC(=O)C2)C1 C1(C(N(CC#C)CC2CC2)=O)CCCN(C(=O)CCc2cncnc2)CC1 C(=O)(C(F)(F)C(O)C1CC1)N(CCNC(=O)C(c1ccccn1)C)CC C#CCCCC(C)C(=O)NC1CC(C)(NC(=O)CCCc2ccc(O)cc2)C1 C(=O)(C(F)(F)CC#N)NCCC1CCN(C(C(c2ccc(F)cc2F)(C)C)=O)C1 C1(NC(=O)Cn2cncn2)CN(C(=O)CN2CCSCC2)C2(CCCC2)C1 c1(OCCCCC)ccc(Cl)cc1CNCC1(C)CCNCC1 c1(OC)c(C(=O)NCC(C)(COC)NC(=O)CS(N)(=O)=O)csc1Cl CC1(C)CCC=C(C(=O)NCCCCCCNC(c2ccn3cnnc3c2)=O)C1 c1(C(=O)NCCC(C)N(C(CN(CC)CC)=O)C)cc(C(=O)OC)n(C)n1 C1(CCC)CN(C(=O)C(C)CCOC)CC1C(=O)NCc1ncn(C)n1 CC1CC(CNC(C2OCCOC2(C)C)=O)CCN1C(=O)C1=CCCSC1 Cc1cc(C(=O)NNC(=O)N(CCCO)CCC#N)cc([N+](=O)[O-])c1Cl c1(CC(N2C(CNC(c3cnncc3O)=O)CCC2)=O)ccc2n[nH]cc2c1 C1(NC(C(CCOC)C)=O)CC(F)(F)CC1NC(c1sc(C)nc1C)=O C1(C(=O)NC23CC(NC(C45CCCCC4C5)=O)(C2)C3)C2CCC3C(C2)CC13 Cc1ccnc2c(C(N3CC(CNC(c4ccnnc4)=O)CC3(C)C)=O)cnn12 CC1(CCNC(c2coc(C3CC3)n2)=O)CCN(C(C2CC(O)CN2C(N)=O)=O)C1 C(N=c1[nH]c(Cl)nc2[nH]ccc12)C1CN(C(c2ccno2)=O)CC12CCC2 c1(C(=O)NC)ccc(C(N2CCCC2CN(C(=O)CC(C)F)C)=O)cc1F c1(C2(C(=O)NCC(C(C)C)(C)NC(=O)C=CS(C)=O)CC2)c(F)cccc1F C1(S(C)(=O)=O)(C(N(CCNC(c2ccc(F)c(CO)c2)=O)CC)=O)CCCCC1 Cc1noc(N)c1C(=O)NC1CCC1NC(c1cnn(C(F)F)c1)=O c1(CC)noc(CCC(N2CCCC2CN(C(=O)C=CI)CC)=O)n1 C1(CCNC(CSCCN(C)C)=O)(NC(C2CCCO2)=O)CCOCC1 c1(C(=O)NCC2CN(C(c3scc(OC)c3)=O)C(C)CC2)ccc(F)c(C#N)c1 C#CC(C)(C)C(=O)N(C1CC(NC(c2nccnc2C)=O)C1)C C1(CN(CC(C)C)Cc2cccnc2)CC1C1CCC1 C1(C(N2CC(COC)(NC(c3cc(O)n(C)n3)=O)C2)=O)CCC(C2CC2)C1 C1(CC)CN(C(c2cc[nH]c(=N)c2)=O)CCC1NC(C1COCCN1C(C)=O)=O C1(C(=O)Nc2c(C)ncc(F)c2)CC2C=CC1N(C(c1nccn1C(C)C)=O)C2 C#Cc1cccc(C(=O)N(CCCNC(c2cncnc2C)=O)CCO)c1F CN1CCOCC1C(=O)NC1CN(C(C2(C)CC2)=O)CC1CC(C)(C)C C1(CNC(C2CC(CF)C2)=O)CN(C(C2(C3CCC3)CC2)=O)C2(CCC2)C1 C(=O)(C1=CC2CCC(C1)C2)NC1(CNC(C=COCC)=O)CCC1 N1(CC(=O)NCC(CC(F)(F)F)NC(c2ccc(O)cn2)=O)C(=O)CCCC1=O c1(NC2CC(CO)C2)ccc(Br)cc1[N+](=O)[O-].C12(CC1)C(=O)NC2 N1(C(C(CCC)NC(N)=O)=O)C2CCC1CN(C(C1CC1(C)CC)=O)CC2 C1(COC)(NC(C2(c3cccc(C#N)c3)CC2)=O)CCN(CCOC)CC1 C1(NC(c2cc(C)[nH]n2)=O)CC2CN(C(=O)CC(O)C(C)C)CC12 N(C1COCc2ccccc21)C(=O)CCc1nnc(Cc2ccccc2)o1 C1(CC(C)C)CCCN(C(=O)CN2CCN(CC(O)C3CC3)CC2)C1 N1(C(CSCCCC)=O)CCCC(Oc2ccccc2F)C1 c1(C(N(C)CC2C3CN(C(C(CC)C)=O)CC32)=O)ccc(=NC)[nH]c1 C(=O)(C(F)C(C)C(F)(F)F)N1CCN(C(Cc2ccc(SC)cc2)=O)C(C)C1 C1(C(=O)NC2C(CNc3nccc(C(=O)OC)n3)CCC2)CC2(CCCC2)CO1 C1(C(=O)NC2CCN(C(c3[nH]cc(C#N)c3)=O)C2C(F)(F)F)CCC=CCCC1 C(CC1CC1)(C(=O)NC(CCO)C1CCC1)NC(=O)CCc1cscn1 c1(C(=O)Nc2cc(C)sc2)cccc(CNC(=O)CCc2c(C)noc2Cl)c1 C1(C(N2CCC(C(C)(C)NC(C3CC(OC)C3)=O)C2)=O)C2CCCCCC12 CCC(=O)CCC(=O)N1CC(C)CCC1C(N1CCCC(O)CC1)=O Cc1cc(=NC(=O)C(=O)N2CC(NC(c3cc(F)cc(F)c3)=O)C3CC23)[nH]o1 N12CCC(C1)C2.c1(C(N2C(C(N(C3CC3)CC)=O)CC2)=O)occc1C(C)C c1(NC(C)=O)nc(CNC(CC2N(C(C3CC3C3CC3)=O)CCC2)=O)cs1 N1(C(c2c(CC)n(C)nc2)=O)CC(NC(=O)C(C)OCC(C)C)CC1(CC)CC C1(CCNC(c2nc(C)sc2C)=O)CCN(C(=O)C(C)SC(F)(F)F)CC1(F)F Cc1nc(NC(C2CC(F)CN(C(C3CNC(=O)C3)=O)C2)=O)ccc1C(F)(F)F N1(CC(=O)NCC2CCN(C(c3ccc(C)[nH]3)=O)C2)OC(C)(C)CC1=O n1(C(C)C)ccc(CCC(N2CC(F)(CNC(=O)Cc3cc[nH]n3)C2)=O)n1 n1(CCC)ccc(=NC(c2cc(Br)cc(OC)c2OC)c2nnnn2C2(C)CC2)[nH]1 N1(C(C=CC)=O)CCC2(CC(C(=O)NCc3ccc(Br)cc3[N+](=O)[O-])=NO2)C1 c1(C(N(CCCNC(c2cccc(CC)n2)=O)C2CC2)=O)cccc2cncn12 N1(C(Cc2ccc(OC)cc2)=O)CC2CC(C1)CN(C(=O)Cc1cncs1)C2 Cn1ncc2ccc(-c3cn(CCNC(C4CCCC(C)(C)CC4)=O)nn3)cc12 CCC(CO)C(=O)NCCOCCN(C)C(c1cc(C(F)F)[nH]n1)=O c1(C(=O)NCCCNC(CC(C)C(F)F)=O)c(O)ncc2c1CCC2 CC1CN(C(c2cnn[nH]2)=O)CC1CNC(=O)C(c1cccc(Cl)c1)(F)F C(CC(C)C(=O)NC1CN(C(=O)Cc2cnns2)CC1OC)=CCC c1(C2(OC)CCC2)ccc(C(=O)NCCCNC(C2(CO)COC2)=O)cc1 O=C(C(O)C(F)F)NC1(C(=O)Nc2ccc(-c3cnc[nH]3)cc2)CC1 N1(C(CC(C(F)F)NC(COCCC=C)=O)=O)CCN2CCCC2C1 c1(N(C)Cc2n(CC=C)nnn2)ccccc1NC(CC1(C)CCOCC1)=O C#CCCC(C(=O)O)NC(=O)C(=O)NCC(C)Oc1ccccc1Br C1(N(C(=O)C(Cl)=CCl)C)CCC(NC(=O)CN2CCS(=O)CC2)CC1 c1(C(N(C)CC2(NC(=O)C(F)CC3CC3)CC2)=O)cc(=O)n(C)cn1 c1(OC)ccc(Br)cc1C(N1CC2CC2(CNC(c2cnnn2C)=O)C1)=O c1(CC)ncc(C(N2CCOCC(O)C2)=O)c(OC(F)F)n1 C(C(CN=c1cccc(S(=O)(=O)NC(C)CN2CCCCC2)[nH]1)C(C)C)OC C1(NC(C(CCC)F)=O)CN(C(c2ccn(C(C)C)n2)=O)CC12CCC2 CC1CCCC(C(N2CCC(CNC(c3cncnc3C3CC3)=O)C2)=O)CC1 N1(C(C2(COCC)CC2)=O)CCOC2(CCN(C(=O)CC(C)c3ccco3)C2)C1 C1(C(N(C2CCN(C(c3cnn(C(C)C)c3)=O)C2)CC)=O)CC2(CCO1)CC2 C(=O)(CS(=O)(=O)C1CC1)N1CC(NC(C2N(C(CCC)=O)CCC2)=O)C2C(C1)C2 C(CC(C(=O)NC(C)(C=C)CC)NC(=O)CN1CC(C)(OC)C1)=CC Cn1cncc1C=CC(N1CCCC(CCNC(C2CC2c2ccsc2)=O)C1)=O N1(C(Cc2c(OC)cccc2)=O)CC2CCC1CN2C(c1cc(=O)cc(Cl)[nH]1)=O C1(C(N2CC3N(C(C4C(COC)C4)=O)C(C3)C2)=O)CC2CCCC(C1)C2 C1(C(N(C(CNC(C(C)C2CCC2)=O)Cc2ccccc2)C)=O)CCN(C)C(=O)C1 c1(C(=O)NC(CCNC(C(COC)(C)OC)=O)C)[nH]c(C)c(C(C)=O)c1C CC1(C)COCC(CC(=O)NCC=CCNC(=O)C(C)(C)CCF)O1 c1(C(N(CCNC(C2COCCN2C)=O)CC)=O)ccc(C)cc1Br c1(Cc2nc(C(CCC)C)nn2-c2cnnn2C)cc(C)cc(F)c1 N1(C(CCC#N)=O)CCC2CN(C(=O)CC=Cc3ccc(F)cc3)CCC2C1 CC(CNC(=O)C(N)=O)CC(=O)NCC1(O)CC2CC2C1 C(CC(C(=O)N1CCCC(C(N)=O)C1)NC(=O)COC1CC1)=CC N#Cc1cccc2[nH]cc(C(N3CCC(Cc4ccc5ccccc5c4)C3)=O)c12 c1(C(N(CC(C)NC(=O)CC(C)CCC=C(C)C)CC)=O)cc2cccc(C)c2[nH]1 C(CC1=CCN(C(=O)C(c2cc(F)cc(F)c2)O)CC1)NC(c1cc(C)ns1)=O C(=O)(CCCCCCN=[N+]=[N-])NCC1N(C(C2C(C=C)C2)=O)CC=C1 C1(N(C(=O)COC2CCC2)C)CCC(NC(=O)C(F)n2cccn2)CC1 c1(C(=O)NCC2(O)CN(C(C(CCSC)(C)C)=O)C2)cc2cc(C)ccc2o1 c1(-c2ccc(NC(=O)NC(COCCOCC)C)o2)cccc(C)c1 N1(C(CC(CC)C2CC2)=O)CC(CNC(=O)C=Cc2ccc(C)s2)C2(CC2)C1 CC(C)C(O)C(=O)NC(CNC(=O)C(C)C1CCCO1)C(C)(C)C C(C(CC(=O)NCCC12CCCC1C2)OC)NC(CCOCCCOC)=O C1(C(N(CC(C)O)CCNC(=O)C(Cl)=CCl)=O)CC12CCC(F)(F)CC2 Cc1nnc2n1CCC2(C)C(=O)NCC1(F)CN(C(=O)COC(C)(C)C(F)(F)F)C1 Cc1ccc(Cl)cc1C1CCCN1C(=O)NC1CCC(NC(=O)OC(C)(C)C)CC1 N1(C(C2C(c3cccc(C)c3)CCC2)=O)CCC(c2nnc(C(F)F)o2)C12CCCC2 C1(C(=O)NCCc2ccsc2)CSCCN1C(c1cncc(O)c1)=O C1(N(C(c2n(CC)ccn2)=O)CCF)CCCN(C(C2(C)CC2C(F)(F)F)=O)C1 C1(C(=O)NC2(COC)CN(C(=O)CCc3nncs3)C2)CCCN(S(C)(=O)=O)C1 c1(OC)cc(C)c(C(N2CC(NC(=O)CCc3ccccc3)C(F)(F)C2)=O)cn1 C1(C(N2CCC(NC(=O)Cc3cnn[nH]3)C2)=O)(CO)CCOCC1 Cc1oc(Br)cc1C(=O)NCCC(C)CCNC(c1nn[nH]c1Cl)=O c1(CC)nc(CC)sc1C(=O)NC1CCN(C(C)C)C1=O N1(C(c2ncc(NC)nc2)=O)CC(C)CCC1CNC(=O)CSc1nnnn1C C1(C2CCN(C(=O)CCC(C)(C)F)C2)(NC(C2N(C(C)=O)CCC2)=O)CC1 c1(N2C3(CN(C(=O)Nc4c(OC)cccc4)C3)CC2)ncnn2cc(Br)cc12 N(C(=NCC1=CCCC1)NCc1cccs1)C1CCC(NC(C(C)C)=O)CC1 c1(C(=O)NC2CC(N(C(=O)CC3C=CCCC3)C)C2)coc2c1C(=O)NCC2 CC(CCC(=O)NCC(F)C(C)(C)O)NC(c1c[nH]c(=N)o1)=O C1CN=C2N=C(C=C(C)N2)N1.Cc1ccc2[nH]c(=NC3CC4CC(OC)CC34)sc2n1 CN1CCN(C(=O)CSc2nc[nH]n2)C(C(=O)NCc2cc(O)ns2)C1 C1(C#N)(NC(C2CCC3(CC3)C2)=O)CCN(C(c2cn(CCN(C)C)nn2)C)CC1 C12(C(=O)OCC)CCN(C(=O)CCCCNC(N)=O)CCC1C2 c1(C(C(=O)NCC(CN(C(=O)CCCC2CC2)C)O)NC(N)=O)ccc(O)cc1 C12(C(=O)Nc3ccc(C)nc3)CCC1CN(C(=O)C(c1ccc(F)cc1)CO)C2 c1(C(CNC(N2CCC(SC)CC2)=O)=O)cnn2ccccc12 S(=O)(=O)(c1ccc(C#N)c(NC2CCCN2CC(F)F)c1)N(C(C=C)C)C C1(N(C)C)CCN(C(c2sccc2CNC(c2ccoc2C2CC2)=O)=O)C1 Cc1cnc2ncccc2c1C(=O)NC(c1nc(-c2cccs2)n[nH]1)C N1(Cc2cccc(C(C)C)n2)CC2(C)CC1(CO)N2C(=O)C(c1ccc(Cl)cc1)C C=CC(CC)C(=O)NCC1COCC1NC(C1(N(C)C)CC1)=O c1(C(=O)NCc2c(C)nns2)cccc2nnn(C)c12 CC1Cc2cc(C(=O)NC(C3CCCN3C(C3(CF)CC3)=O)C)ccc2O1 C1(CC)(NC(c2cc(C)c(C)s2)=O)CCN(C(=O)Cc2conc2C)CC1 C1(NC(CN(C(Cn2ncc(CC)c2)=O)C2CCC2)=O)CC2(C1)CC(C)(C)C2 N1(C(C2CSCCN2Cc2cccc(I)c2)=O)CCc2nc[nH]c2C1 N1(C(CCN(C(C2(C)CC(=C)C2)=O)C)=O)CC(O)C(O)C1C(=O)OC c1(C(N2CCOCC(CNC(c3cn[nH]c3)=O)C2)=O)cc2c(O)ncnc2cn1 c1(CCC(N2CC(C(C(=O)N(C3CCC3)CCSC)OC)C2)=O)cnn(C)c1 CC(C(=O)N1CCCC(O)(CNC(c2csc(-c3ccco3)n2)=O)C1)C(C)(C)O Cc1cnc2nc(C(N3CCC(C)C(CNC(c4ccc(C)o4)=O)C3)=O)nn2c1 C1(NC(COCCOC)=O)COC2(CCN(C(=O)Cc3ccc(C)cc3)CC2)C1 Cc1ccc(C(=O)NCC(CNC(=O)CNC=O)C(F)(F)F)cc1[N+](=O)[O-] CC1CN(C(=O)COCC2CCCCO2)CC1CNC(C1CC(C)(F)C1)=O c1(CN(CC(COC)O)C2CCOC2)cc(OC)ccc1F CCC(C(=O)N1CCC(O)(C(C)NC(=O)CCC(=O)NC)CC1)C(C)C Cc1ccc(Br)c(C(F)(F)C(=O)Nc2ccc(Br)c(Br)c2)c1 C1(NC(C=C(CC)CC)=O)C2COCC1CN(C(c1ccc(Cl)c(Cl)c1)=O)C2 C12(C(=O)NCCN(C(=O)C3=NOCC3)CCC)C(=O)C3CC1C2C3 C1(CNC(C(=O)OC)CCSC)CCCC(c2nn[nH]n2)C1 C1(N(C(C2ON=C(C(C)C)C2)=O)C)CCC2(CC1)CCN(C(=O)C=C1CCC1)C2 Cc1cc(Cl)ncc1CC(N1CCC(C(C)NC(=O)C(=O)NC2CC2)C1)=O C1(C)(C(N2C(CC=C)CCC2)=O)CC(O)CN1C(=O)COc1ccccc1 N1(C(c2cc(C(CC)CC)no2)=O)CCCC(CNC(=O)C2=C(C)CCC2)CC1 S1(=O)(=O)c2ccc(F)c(c2F)N1CC#C.c1(CNC(=O)OC)ccco1 N1(C(c2c(OC)ccs2)=O)CC(C(=O)N(C(C)C(C)(C)C)C)C2(CC2)C1 C1(C(N2CC(NC(c3ccc(N)cn3)=O)C3(C2)CC3)=O)CS(=O)(=O)CC12CCC2 C1(C(=O)NC(CCC=C)C)CC(O)CN1C(=O)CN1CCCCC1C N1(C(c2c(C)cc(C(F)F)o2)=O)CC2CCC(C1)N2C(=O)CCC1CCOC1 c1(CC(=O)N(CC(CC)NC(c2cc(OC)nn2C)=O)C)c(Cl)cnn1C Cc1ccc(C=CC(=O)NC2CC(C)N(C(=O)Cc3cnns3)C2)cc1 C1(C(=O)NC)CCN(C(C(=O)CCNC2CCCC2)C2CC2(C)Br)CC1 C1(C(N2CCC(N(C(=O)C(F)(F)c3cnn(C)c3)CC)C2)=O)CCCC(OC)C1 N1(C(C(C)NC(c2ccco2)=O)=O)CCOCC1CNC(C1(C)CCC(=O)N1)=O Cc1sc(C)c(C(=O)NCC2(NC(c3cc(C(F)(F)F)ns3)=O)CCCC2)c1C#N c1(C(N2CCC(Oc3ccccc3)CC2)=O)ccc2nncn2c1 C1(O)(C(=O)NCC2N(C(C(F)=CC)=O)CC2)CCSCC1 c1(C(=O)NCC2CCC(C)N(C(=O)CCc3nccs3)C2)ccc(N)c(F)c1F c1(C(N2CC(O)CC2C(=O)NCCOCC(F)(F)F)=O)c(F)ccc(O)c1F C1(OCC)(CNC(C2CC(OC)(OC)C2)=O)CN(C(=O)CCSC(F)(F)F)C1 Nc1nc(Cl)ccc1C(=O)NCC1CCCCCN1C(C1CCCC(=O)N1)=O N#Cc1ccc(=NCC(C2CCCC2)NC(c2cc(C(F)(F)F)n[nH]2)=O)[nH]c1 C1(NC(c2n(CC)nnn2)c2nnc(C3CC3)s2)CCOC(CCOC(C)=O)C1 Cc1nc(NC(c2ccc(F)cc2)=O)nn1-c1cccc(F)c1.C1CCC(=O)N1 c1(Nc2nnn(C(N3CCC(O)CC3)=O)c2C)cnc(C#N)cn1.Cc1cc(C)on1 N1(CCNC(C2(NC(C(c3cnccn3)C)=O)CC2)=O)CCCCC1C n1(CC#C)cccc1C(=O)N(CC(C)CNC(=O)CN(C)C(C)C)C C1(C(N(CCC2CN(C(C3CCC(C4CC4)O3)=O)C2)C2CC2)=O)CC2CC(=O)C1O2 C12(NC(CCCC)=O)COC(CNC(c3c(C(F)(F)F)n[nH]c3C)=O)(C1)C2 c1(NC(N2C(C)(CCC)CC2)=O)ccc(CC(=O)OC)c(OCC)c1 c1(C(=O)NCC2CCN2C(C2COCCO2)=O)cccnc1S C#CCC(CC(=O)NCCC(C)(CC)NC(=O)Cn1ccnc1C(C)C)OC Clc1ccccc1CN(Cc1ccccc1)Cc1nc(Br)n[nH]1 C12(CNC(C3OCCN(C)C3)=O)CCC(CN=c3[nH]nco3)(CC1)OC2 C1(CN(C)C(c2ccc(C(F)F)cc2F)=O)CN(C(=O)C(C)(C)C2CC2)CCO1 C1(NC(CCC#C)=O)CC(O)CN(C(c2cnn(CC(C)C)c2CCC)=O)C1 CC1CC(NC(=O)CCc2cncs2)CN(C(=O)COc2ccccc2C2CC2)C1 c1(OC)cnc(Cl)[nH]c1=NC(=O)c1nc2ccc(Cl)cc2[nH]1 C1(C(N2CCN(C(CC)C)CC2)=O)CCC(O)CN1C(c1cccc(F)c1)=O CC(C)C(O)C(C)N=c1[nH]c2ccc(S(=O)(=O)NCCC(N)=O)cc2s1 c1(OCC)cc(C)cc(NC(N2CCC3(CC2)CC3c2nn[nH]n2)=O)c1O CC(C)CCC(C(=O)NCC1COCC(C)O1)NC(c1cn[nH]c1)=O N1(C(Cc2c(C)occ2)=O)CCOCC(NC(=O)CSCC2CCCO2)C1 N1(C(c2ccc(C(N)=O)[nH]2)=O)CCCCC(C(N2CC(N3CCNC3=O)C2)=O)C1 C1(CNC(CC=C)=O)(CO)CC12CCN(C(c1coc(C(N)=O)c1)=O)CC2 c1(C(=O)NCC(CC)NC(c2c(C)nc(CCC)o2)=O)cncc(F)c1Cl C(CC(C(=O)NOCC(C)O)OC)NC(CC1C(CC)C1)=O CC1(C)CC=C(C(=O)N2C3CCC2CC(NC(=O)C2=CCCC2)C3)CC1 CC1CN(C(c2csc3ccc(Br)cc23)=O)c2c(Br)cccc2O1 C=CCC(C)(C)CC(=O)NC1(C(=O)NC(C)C(F)(F)F)CCC1 C12(C(=O)NCC3(NC(c4cc(C(N)=O)[nH]c4)=O)CCCC3)CCCC1CC2 C1(COC)(NC(=O)CCCCCSC)CCN(C(=O)C(C)(C)C#N)CC1 N1(C(C(C)OCCC=C)=O)CCCCCCC1C(=O)NCc1n[nH]cc1C c1(OC)ccc(CN2CC3(CC3Nc3ncc(C(C)=O)cc3C)C2)cc1C(=O)O C12(NC(CC3CN(C(C(C)OC4CCCC4)=O)C(C)C3)=O)CCC(F)(CC1)C2 C12CN(CCCO1)C(=O)N2.Cc1cc(Cc2cc(C)n(C)n2)ccn1 C(N=c1[nH]c(N2CCSC2)nc2cccnc12)c1c(CN(C)C)cccc1 C(C(C)(C(=O)NCC(C)(F)C(C)C)NC(=O)Cn1ncnn1)SC C(=O)(C1=NOC2CCC3(CCN(CC)CC3)C12)C(N(CC(CCCC)CC)CC)=O.N(C)C C1(NC(CC(CC)C)=O)CC2(CCN(C(c3cnc(C4CCC4)s3)=O)C2)C1 C1(NC(C(c2cnccn2)C)=O)CCC(CNC(=O)CS(=O)(=O)C(C)(C)C)CC1 C(=O)(CCCCCC#N)NC(C)CCCCNC(=O)C(C)N1CCC1 N1(C(CC(C2CC2)NC(C(=Cc2cc[nH]c2)C)=O)=O)CC(C2(C)CC2)C1 C(C(=O)N(CCCCC(N)=O)C1CC1)(C(C)C)NC(C(F)=C(C)C)=O Cc1cc(=NCC2CCN2S(C)(=O)=O)[nH]c(-c2cccnc2)n1 C(CC(C(=O)N1CC(C(=O)N(C)C)C1)NC(=O)C(C(C)C)SC)OCC.C C1(NC(c2c(C)nc(C)o2)=O)CC(F)CN(C(=O)CC(c2ccc(F)cc2)C)C1 C1(CC(=O)NCCCCC(C)NC(c2c(C)scn2)=O)CC2(CCC2)CO1 CC1(CNC(=O)CCS(C)(=O)=O)CC(F)(F)CN1C(=O)CCNC(N)=O c1(C(=O)NC(C2(O)CN(C(c3cnn(CC(F)F)c3)=O)C2)C)nccnc1N c1(C(N2CCC(Cn3cc(CC4C(=O)NC(=O)S4)nn3)C2)=O)ccc(Cl)cc1Br C=CCC(C)(C)C(=O)NCCn1cc(C(=O)N(C2CCC2C)C)cn1 CC1(C(=O)NCCOCCCNC(c2scnc2Cl)=O)CCC2CC2C1 Cc1cccc(-n2nc(C(=O)N(C)CC3(O)CCSCC3)cc2C)c1 C1(CC(N2CCC(C(=O)NC)C2)=O)CCN(CCc2cccnc2O)CC1 C1(C(=O)OC)CC(C(F)(F)F)CCN1S(=O)(=O)CC(C)c1ccccc1 n1(CC)cc(C(=O)N(CCC(N2CCC(C)(C(N)=O)C2)=O)C2CC2)c(C)n1 C1(C(N(CC(C(=O)OC)C)C)=O)C=CCN(C(=O)CC2CC=CCC2)C1 N1(C(C(CCN(C)C)NC(CC(C)C)=O)=O)CCCCCCC1C C1(C(=O)NC2CCC(N(C(c3ccc(CCC)[nH]3)=O)C)C2)CC(F)(F)C1(C)C N1(C(c2c(CC)nn[nH]2)=O)CC(F)(F)CC1CNC(=O)CCc1ncco1 CC(C)(CC(=O)N1CC(CNC(C2CC3(CSC3)C2)=O)C(C)(C)C1)C(F)F c1(C(N2CC(CNC(C3N(S(C)(=O)=O)CCC3)=O)C2)=O)cccnc1O C1(CNC(C2CC(CC(C)C)C2)=O)CCCCCN1C(c1cc2occc2[nH]1)=O N1(C(C2(NC(=O)CC3(C#N)CC3)C(C)(C)C2)=O)CC2(CC(O)C2)C1 C1(=CC(=O)NCC(CCCC)NC(=O)C=CS(C)=O)CCC(C)(C)CC1 C1(CNC(C2C(C)CCC2)=O)CN(C(c2ccc(NC(C)C)cc2)=O)CCCO1 Cc1cc(F)ccc1NC(c1cc(C)c(Br)s1)c1nnnn1C(C)(C)C Cn1cc(C(O)C(=O)NCCC2CCCN2C(c2coc(SC)c2)=O)cn1 N1(C(c2nc(C)sc2)=O)CCC2(CCN(C(=O)C(C)(C)C(C)(C)O)CC2)C(C)C1 C1(C(=O)NCC2(OC)CN(C(C3(CCCC)CC3)=O)C2)CCC(C(F)F)CC1 c1(N(CC=C)C)nnc(CC2CCCO2)n1CCC1CCCCO1 C(=O)(CCCc1nncn1C)N(CCC)CCNC(C1(n2cncn2)CC1)=O Cc1nc[nH]c1CC(=O)NCC(C)NC(=O)CNC(=O)NC1CC1 C1(C(=O)NC(C)(CNC(c2cnn(C3CC3)c2)=O)C2CCC2)CN(S(N)(=O)=O)C1 C(CCC(=O)NCCC1(C(=O)N(C2CCOC2)CCF)CCC1)OCC=C c1(C(N(CCCNC(C2CC=C(C)CC2)=O)C2CC2)=O)ccc2c(n1)NCC2 C1(CNC(C2CC(N(C)C)C2)=O)CCC(C(=O)NCC=CCl)O1 c1(C(N2C3CCC(NC(CCC=CC)=O)(C3)C2)=O)cccc2c1OCC2 Cc1cc(=O)c(C(N2CCC(CCNC(=O)C(C)CC(F)(F)F)C2)=O)cn1C N1(C(C2C(=C)C2)=O)CCC2(CC1)CCN(C(=O)CC1(C)CC1(Cl)Cl)C2 C(=O)(CC(C(C)(C)C)NC(=O)CC1COC(=O)C1)N1C(CCC=C)CCC1 C1(C(=O)OC)OC2(C)CC1(NC(=O)Cc1cc(C3CC3)no1)C2 Cc1nc(C(C)NC(=O)C(Cc2ccco2)N(C(c2cc[nH]n2)=O)C2CC2)cs1 C1(C(=O)NCC2C=CCN2C(c2cnn(C3CC3)c2)=O)COCCN1CC(F)F C1(N(C)C(C2CC2F)=O)CCN(C(=O)CC23CCCN2CCC3)CC12CC2 N1(C(C(C(=O)OCC)F)=O)CCCC(C2(NC(c3cc(OC)ccn3)=O)CC2)C1 c1(N2CCC(CCNC(c3ccnn3CC3CC3)=O)C2)cc(C(F)(F)F)nc(Cl)n1 c1(C(N2CCCC2c2cn(C3CC(O)C3)nn2)=O)c(F)ccc2occc12 Cc1nc(N2CCC2)c(C)c(C)n1.c12c(Cl)n[nH]c1SCC1(CCCC1)NC2=O C=CCC(C(=O)NCC(O)C(=O)NC(C)CN(C)C1CC1)NC(C)=O c1(C(N(C2CCC(NC(=O)C=CC(=O)OC(C)(C)C)C2)C)=O)cc(F)cc2nc[nH]c12 C1(NC(C2CN(C)C2)=O)COC2(C1)CN(C(=O)Cc1cnns1)C2 C1(OC(C)(C)C)CC2(CCC(CNC(=O)Nc3nc4ccccc4o3)CC2)C1 C1(C(N(C2CCCN(C(=O)CN3CCC(F)(F)C3)C2)CC)=O)CC12CC(C)(C)C2 CC(C)CS(=O)(=O)CCC(=O)N1CCC(CN(C(=O)CC(O)CN(C)C)C)C1 c1(CC)nccn1C(C)CC(=O)NCC#CCNC(=O)C(F)CC1CCCO1 N1(C(C2(CC#C)CCCCC2)=O)C2CCC1C(C(N1CCC(CN(C)C)C1)=O)C2 c1(C(N(CCNC(C(C=C)C)=O)CC)=O)cnn2cccnc12 C(=O)(N1CC=CCO1)C1(C)CCN(C(C(COC)(F)F)=O)C1 C1(CCNC(COCCOC)=O)COCCN1C(=O)C(C)CSC(F)(F)F C1(NC(c2cccc(COCC=C)c2)=O)CCN(C(C2(CC)CC2)=O)CC1O CCCCC(O)C(=O)N1CC2CC2(NC(c2ccc(-c3cc[nH]n3)cc2)=O)C1 C(CCN(C)C(=O)Nc1ccccc1-c1cn[nH]c1)(C(C)C)NC(C1C(=C)C1)=O c1(C(=O)NCCC2CCCN2C(c2ccc(Cl)s2)=O)ccnnc1Cl n1(CC(=O)N(C)C)cnc(=NC(=O)NC2CC3(CCC3)C(=O)N2)[nH]1 c1(C(=O)NC(c2ccc(C)c(F)c2)C)cnn2cc(C(=O)O)cnc12 CC1(C)C(C(=O)NC2CCCN(C(=O)C(=O)C(F)(F)F)C2C)CCS1(=O)=O c1(NCC(C(CC)CC)OC)ncnc(NCc2ccn(C(F)F)n2)c1C C1(COC)(CNC(c2cc3sccc3s2)=O)CCN(Cc2cc(C)no2)CC1 C1(NC(CS(N)(=O)=O)=O)COC2(CCCN(C(c3coc(Cl)n3)=O)C2)C1 C(=O)(C(CCC)S(N)(=O)=O)NC1CCC(NC(C2(C=C)CCCCC2)=O)C1 n12cc(nn1)C2C1CC1.c1nc(SC2CC2)co1 N#CC1(C(N2CCOCC(NC(c3c[nH]cc3C(F)(F)F)=O)C2)=O)CC2CC2C1 C1(NC(C(C)(C)OCC)=O)CCC2(CCN(C(c3ccc(NC)cc3)=O)CC2)C1 C12(CNC3(C4CCCN4C(=O)CCS(C)(=O)=O)CC3)CC(C1)C(C(N(C)C)=O)CO2 N1(C(c2c(C)n(C)nc2)=O)CCC2CCCN(C(=O)Cc3ccc(F)nc3)C2C1 OC12CCC1CN(N1CCC(C3OCCO3)C1)C2 C12(CCNC(C(C)OCC)=O)CCC(CC1)N(C(=O)C(CC)c1cccnc1)C2 C1(CC(=O)N(C)CC2C3CN(C(=O)CCCCCN(C)C)CC23)CC(=O)NC(=O)C1 CC1CCCCCC1NC(c1ccc(F)c(F)c1)CO CCCCCCCC(=O)NCC1CCC2(CCC2)C1NC(C1CS(=O)C1)=O c1(CC(=O)NC2CCCN(C(CSCC#C)=O)CC2F)nnc2n1CCCCC2 c1(N2CCC(C(=O)NC)CC2)nc(=N)[nH]c(=NCC2CCN(C(=O)NC)C2)[nH]1 C1(NC(CN2CC=C(C)CC2)=O)CN(C(c2ncncc2N)=O)CC12CCC2 c1(C(=O)NC2(CC=C)CN(CC3(C(=O)OC)CCOC3)C2)c(F)cccc1F CC1(C)CN(C(C2(C(N)=O)CC2)=O)CCC1NC(c1cnc2scnc2c1)=O O=C(C(O)CC(F)(F)F)NCC1C(C2CC2)CCN1C(c1cc(F)ccc1Cl)=O CCCCS(=O)(=O)NC1(C(=O)NC(C)CCNC(=O)C(C)(O)CC)CCCC1 C#Cc1cccc(NC(=O)NC2CCCC(F)C2)c1 C(C1=NOC2(CCC2)C1)C(N1C(c2cn(CC(CC)O)nn2)C(C)CC1)=O C1(CCN(C)C(C2CC2C#N)=O)CCN(C(=O)C=CCN2CCC2)CC1 N1(C(C2(c3nccc(C)c3)CC2)=O)CC2CCC1C(Nc1ncnc(Cl)c1F)C2 S(=O)(=O)(c1cccc(N2CCC(C3CC3(F)F)CC2)n1)N(CCCC=C)C c1(CN2C(C(=O)Nc3cnc(C)s3)CC2)ccc(Cl)cc1C#N CCCC(C(=O)NCc1ocnc1CC(=O)NCC1CC12CCOC2)OC C1(CNC2CN(C(=O)CC3CC3)CCO2)CCC(F)(F)CO1 C1(CC(=O)NCc2c(C)noc2C)C2CCCC2N1C(=O)C(C)CC#N CC(Cc1cnn(C)c1)C(=O)NCC1CCCN1C(C1CC(n2cnnc2)C1)=O c1(OC)cccc2sc(-c3nc(-c4ccsc4)nn3CCN(C)C)cc12 C1(C(=O)NCC2CC(NC(COC(CC)CC)=O)C2)CCC(F)C1 N1(C(CCSCC(C)C)=O)CCN(C(C2CCC2)=O)CC1C1CCC1 C(=O)(C1c2c[nH]nc2CN1C(C1SCCS1)=O)N(C)CC1CC(=C)C1 c1(C(=O)NCCC(CNC(C2CC3CCC(C2)C3)=O)OC)cn2ccccc2n1 C1(C(=O)NCc2cc(C(=O)NCC(C)(O)C3CCC3)n[nH]2)C2CCC(=O)C12 C=CC1CCCCN1C(=O)C1(C)NC(=O)N1.C(=O)(CCCSC)OCC C1(C(=O)NCc2nc(C)[nH]n2)C2CCCC2CN1C(=O)C(Cl)Cl C1(C)CCCN(C(=O)Cn2nnc(C3CC3)n2)C1.CC(C(=O)NC)c1cccs1 c1(OC)cc(Br)ccc1C(N1CC=CC(NC(=O)CN2CCCC2=O)C1)=O c1(CC(C)C)cc(C(=O)NCCNC(=O)Cn2nccn2)cc(O)n1 C1(C(=O)NC(C(CC)OC)C2CC2)C=CCN(C(C2(CC)CCOC2)=O)C1 C1(C)(CNC(CCc2c(C)ncs2)=O)CCC(NC(=O)CSC(F)F)CC1 N1(C(C(C2CC2)NC(COCCOC)=O)=O)CCCOCC1C Cc1sncc1C(=O)NCC(C1CCCCC1)NC(=O)CCn1cc(Cl)cn1 Cn1ncc(Br)c1C(=O)NC(C1(C(c2ccccn2)N)CCCCC1)=O C(=O)(CC(C)(C)C(F)F)N1C(CC(=O)NC(C)CSCc2cscn2)CCCC1 C=CCN(OC)C(=O)CCC1CC(NC(C2CCN2C)=O)C1 N1(C(C2(C)CCC2)=O)CC2CC(NC(=O)CC3CC4(CC4)CO3)C1C2 C(=O)(CC(C(F)(F)F)OC)NC(CC)CNC(c1cc(C2CC2)n(C)n1)=O c1(C2(C(=O)NC3C(NC(COCCOC)=O)CCC3)CCC2)ccc(F)c(Cl)c1 C1(CCC)CN(C(=O)CC2COCCN2C)CCN1C(=O)Cc1ccco1 c1(NC2CCN(C(=O)OC(C)(C)C)C2C(C)(C)C)cc(F)ccc1S(=O)(=O)NC C1(C(=O)NCCCCNC(=O)CCOc2cccnc2)COC2COCC12 C1CCCC(c2ccccc2)(NC2CC2)C1.[nH]1ccnn1 c1(OC)ccc(C)c(OC)c1C(=O)Nc1ccc(Sc2ncnc3ccsc23)cc1 N1(C(C(C)=O)=O)CCC2(CCC(CC(=O)Nc3cnnc(Cl)c3Cl)CC2)CC1 c1(C(N2CCC(CNC(C3(C)C(C)C3)=O)C2)=O)c(N)cc(F)cc1Cl c1(C(N(CCCNC(=O)C2=NNC(C(F)(F)F)C2)C)=O)ccc2c(c1)nnn2C N1(C(CNC(CN(C)C)=O)=O)CCC(F)(CNC(C2C3CC4C(C3)C24)=O)CC1 c1(CC)cc(C(=O)NCC2CCN2C(c2sc(C3CC3)nc2C)=O)c(C)o1 C1(NC(c2ccc(F)cn2)=O)CC2CCCC(C1)N2C(c1ncsc1C1CC1)=O Cc1cnc(NC2(C3(O)CCC3)CC2)c(S(=O)(=O)NC(C(C)C)C2CC2)c1 Cc1cc(C(N2CCC(O)(C(N3CC(CO)C(O)C3)=O)C2)=O)c(C)n1C CCCCN=C(NCCF)NCC1CCS(=O)(=O)N1C C=CC(CCC)CC(=O)NC1(CC(N)=O)CCN(C(=O)C(C)CC)CC1 CC1CCc2nc(C(N3CCC(N)CC3)=O)cc(N3CCC(O)(CO)C3)c2C1 N1(C(C(C=C)O)=O)CCC(CNC(C2(CO)CC2(F)F)=O)(COC)CC1 C(=O)(C(C)CC(F)(F)F)NCCNC(c1c(C)nsc1N)=O C(c1ccc([N+](=O)[O-])cc1)=CC(=O)NCC1CCCN(C(C(CCOC)C)=O)C1 Cc1cn(CC(N2CC(NC(=O)CSCCN(C)C)CCC2C)=O)c(=O)nc1O CC(O)C(C(=O)N1CCC(O)(CO)C1)NC(c1ccccc1)=O c1(C(N2CC(CN(C(C(CC)n3ccnc3)=O)C)C2)=O)cn2ccnc2cn1 C(C(C)(C)C(=O)NC1CC(C(=O)Nc2cccc(CCO)c2)C1)OC CCC(C#N)(CC)C(=O)N1CC=CC(NC(=O)C=CSc2nc[nH]n2)C1 c1(C(=O)NCCC2CN(C(c3c(C)nccn3)=O)C2)ccc2ccnc(Cl)c2n1 c1(C(N2C(CCNC(C=CC(n3ncc(C)c3)C)=O)CCC2)=O)cnc(N)cn1 c1(C(C)C)c(C(N2CC3CC3(C(=O)NCc3ccc(F)nc3)C2)=O)cnn1C C1(C(=O)NCC#C)(CC#C)CCN(C(=O)Cn2ccc(C)c2)C1 c1(C(=O)NCC2N(C(C(CCNC(=O)NC)OC)=O)CCC2)cnc2sccn12 C1(C(N2CC(COC)(CNC(c3cc(Cl)cnn3)=O)C2)=O)OCCOC12CCC2 C1(CNC(C2CCC(O)C2)=O)CC2CCC1N(C(c1cncc(Br)c1)=O)C2 c1(SC)cc(C(=O)NCC(O)CN(C(=O)C(C)C(=O)N2CCOCC2)C)c(C)o1 CC1CN(Cc2ccccc2)CCN1N1CCCCC(C)C1 c1(C(C)(C(=O)N(C)C)NC(C(=O)N(C)CCN2CCCC2)=O)cccc(Cl)c1 Cc1[nH]c(C(F)(F)F)cc1C(=O)NS(=O)(=O)CC1CCC(C(F)(F)F)O1 C1(C(N2C(CN(C(=O)Cc3ccnn3C)C)COCC2)=O)CCc2nnnn2C1 Cc1cc(C(N2CCC(F)(C(=O)OC(C)(C)C)CC2)=O)cc(C)n1 C(=O)(C(C)(C)C(=O)NCC1CC(F)CN1C(=O)CCCNS(C)(=O)=O)N(C)C Cc1ccc(C=CC(=O)NCC(C(C)C(C)C)NC(c2cnc(O)o2)=O)cc1Cl CCC(C#N)C(=O)N(O)Cc1cn(Cc2nn(C(C)C)cc2C)nn1 C1(NC(C(C)OC2CCCCC2)=O)CCN(C(c2cnnn2C2CC2)=O)CC1C N1(C(C2(CCC)CC2)=O)CC(O)(C2(CNC(=O)C(C)(F)F)CC2)C1 C(=O)(C1CCc2c[nH]nc21)NCC1C(NC(CCc2c(C)noc2Cl)=O)CCC1 C1(COC)(CNC(=O)C(C)NC(C)=O)CCN(C(=O)C(C)C2(O)CCC2)CC1 C1(C(N2CCC(NC(CCC=C)=O)C(CO)C2)=O)CCCc2ccccc2C1 C1(C(=O)NC(CC)CN(C(=O)Cc2cccc(C)c2)C)CCN(OC)CC1 c1(NC)ccc(C(N2CCC(NC(c3c(Cl)sc(C)c3C)=O)C(C)C2)=O)c(Cl)c1 C=CCC(C(=O)OC(C)(C)C)NC(=O)C(C1CCCN(C(C)(C)C)C1)(C)C N1(C(c2c(F)ccc(N)c2F)=O)C2CCC1C(F)C(NC(C1CCSC1)=O)C2 CC1(C(=O)NCC2(CNC(C3CCCCC3(F)F)=O)CC2)CCCCCC1 c1(NC(C(CC)C)c2nnnn2-c2ccccc2)ccc(C2CC2)c(Cl)c1 N1(C(c2cc(C(C)=O)[nH]n2)=O)CCCC1(C)C(=O)NC(c1cccc(C)c1)CO c1(C(=O)NCCC23CC(CC2)C3)n[nH]c2ccc(C(F)(F)F)cc12 Cc1ccc(CC(=O)NC(C)(C)CCCNC(=O)CCCCCF)cc1O N1(C(CC2(NC(C)=O)CC2)=O)CC(O)(C2CCN(C(c3cnn(C)c3Cl)=O)CC2)C1 Cc1cc(C(N2CC3CC(NC(=O)Cc4nncs4)C3C2)=O)cc(N)c1 c1(C(=O)NCCC(C)NC(C(c2ccc(C)cc2)C)=O)c(C)nn2c1NCCC2 C1(F)(C(N(CC(C)OC)C(C)C)=O)CCCN(C(=O)CCCCCF)C1 CC12CN(C(c3c(F)cccc3F)=O)CC1(C)CN(C(C1(C)CCCCO1)=O)C2 c1(OC)ccc(C(N2CCCC2Cn2cc(CC(C)(C)C)nn2)=O)nc1F C(CC(=O)NCCC1CCCCCC1)(CC(C)C)NC(C1(CC)CCC1)=O C(=O)(CCCC(=O)N1CC(NC(c2c(C)noc2C(C)C)=O)CC1C)NCC Cc1ccc(C(=O)NC(Cc2cc[nH]n2)C(=O)NC(C(C)(C)O)C2CC2)c(F)c1 CC1(C)OC2(CO)CC1(C(=O)NC1CN(C(=O)Cc3ccc(Cl)cc3F)CC1O)C2 C1(NC(C2C(C(N)=O)C2)=O)CCN(C(=O)C(O)Cc2ccccc2)C1C1CC1 c1(C(=O)NC2C(C(=O)Nc3c(C(=O)OC)onc3C)C2)c(C)cccc1Br C(C1=CCN(C(C2CCCC(=O)O2)=O)CC1)NC(CC=C(C)C)=O CC1CCc2cc(C#N)c(N3CCSCC3CCNC3CCCC34CC4)nc2C1 c1(C(N2CCC3(CCN(C(C(C)OCC)=O)C3)C2)=O)ccc2c(c1)C=CS2(=O)=O N1(C(C(C)(C2CCC2)NC(c2c(CCC)nco2)=O)=O)CCOC(C)(C)C1C C1(CC(=O)NC2(CNC(c3c(OC)nsc3)=O)CCC2)CCC(=O)NC1 CCC(C(=O)NC1CCC(CCC(=O)Nc2conc2C(C)C)C1)SC c1(CC)c(C(=O)NCCC2CCCCO2)cnn1C(C)(C)C N1(CCCC(=O)NC2C(NC(c3ncn(CC)c3)=O)C2)C(=O)C(=O)N(C)C1=O N1(C(CC2N(C(C)=O)CC(O)C2)=O)CCCC(CNc2nccs2)CC1 C1(NC(c2coc(-c3cccnc3)n2)=O)Cc2cscc2C1 c1(N(C(c2cc(C(F)F)no2)C(=O)NCC2CC2)CCCF)ccccc1Br c1(-c2n(C(CC)CC)nc(CCOc3ccccc3)n2)cc2cc(F)c(F)cc2[nH]1 c1(C(N(CC(C)NC(=O)CSC2CC2)C)=O)ccc2cc(F)ccc2n1 C(=O)(C(O)CC(C)(C)C)NC1CC(O)(CNC(c2c(C)n[nH]c2C)=O)C1 c1(C(=O)NC(CNC(=O)C=CCn2cncn2)C2CC2)cc(F)cc2c1NCCC2 N1(C(C(C2CCCC2)OC)=O)CCC(C2CC2)(NC(c2ccns2)=O)C1 c1(COC)ncccc1NC(C1CCN1C(=O)Cc1ccccc1F)=O C12CCN(C(C)C1)C(=O)CCNC2=O.c1(CC)occc1C(=O)NC1CCC1 N1(C(CCOCC(C)C)=O)CCC(NC(=O)C=CC2CCOC2)C(C)(C)C1 c1(C(N2CC(CN(C(c3c(C)cn(C)n3)=O)C)OCC2)=O)cc2c(cn1)OCO2 Cc1ccc(C(N2CC(NC(c3ccc(I)cc3)=O)CC(C)C2)=O)c(F)c1F n1(CC)nccc1C(=O)NCC1(C(N)=O)CN(C(C2(N3CCNC3=O)CC2)=O)C1 N1(c2n(CCOC)c(-c3cc4c(s3)CCC4)nn2)Cc2ccc(O)cc2C1 C1(NC(C(c2ccc(Cl)cc2)CC)=O)C=CCN(C(C23CC(F)(C2)C3)=O)C1 C=CCC(C(=O)NCC1CC(C)(C)CN1C(c1ccn(C)n1)=O)C(C)C C1(C(=O)NCc2cc(C)ncc2)CN(C(c2cc(Cl)cs2)=O)C(C)(C)C1 C1(NC(C(C)O)=O)CN(C(c2cc(N)c3ccccc3n2)=O)C2(CCOCC2)C1 N1(C(CNC(C=CCC)=O)C(F)F)CCN(C(c2ccoc2)=O)CC1 C1(C(=O)NCC(C)N(C(C(C)OCCOC)=O)C)C2CCC3C(C2)CC13 CC1=NOC(C)(C(=O)NCCC(C)NC(=O)CC2(C)CC2(Cl)Cl)C1 C(=O)(CN=c1[nH]c(C)cs1)NCCOC1CCN(C(C2CC3(CC(=C)C3)C2)=O)C1 C1(C)(CC)CCCN(C(C2CC(CNC(c3cncc(C)n3)=O)C2)=O)C1 C1(CNC(C(C)NC(=O)C(C)(C)C)=O)CC2(C1)CN(C(c1cocn1)=O)C2 c1(C(N2CCC(C3(NC(C4CC(CC)C4)=O)CC3)C2)=O)cnc2cc(C)[nH]c2c1 C(C(CC(F)(F)F)NC(C1CCCOC1c1ncc[nH]1)=O)NC(C=C(COC)C)=O Cc1ccc2ncc(C(N3CC(CNC(=O)CCC4(C)N=N4)C(F)(F)C3)=O)n2c1 c1(C(=O)NC(CNC(C2C(C(C)C)OCC2)=O)(C)C)cn2ccnc2cn1 c1(C(C(=O)NC(CC)(C)C)N(C2CCCCC2(C)C)C)n[nH]c2c(Cl)cccc12 Cc1cn2cc(C(=O)NCC3(C)CC(F)(F)CN3c3ccnc(C)n3)sc2n1 C1(NC(CN(C(C(C)C)=O)C)=O)CCN(C(=O)C(N2CCNC2=O)C)C(C2CC2)C1 c1(C(=O)NC(C)CC2CN(C(=O)CCCC#N)C2)ccn2c1CS(=O)(=O)CC2 N1(C(C=CC=CCCCCC)=O)CCN(C(c2cc(C)sc2N)=O)CC1 N1(C(c2ccc(COC(C)=O)cc2)=O)CCOCC(CNC(=O)CC2CC2C)C1 c1(C(=O)NCC2(F)CC(NC(CCC#C)=O)C2)ccccc1C(F)F N1(C(C(=Cc2ccncc2)C)=O)CCC2CCC(NC(c3ccncc3)=O)C12 CN1CCN(C(C2CC3COCC3C2)=O)C(CO)C1.c12n[nH]cc1CNC2=O n1(CC2OCC(C)C2)cc(C#CC(C)(C)NC(=O)Cc2cccc(Br)c2)nn1 c1(C(N2CC=CC(NC(c3coc(C4CC4)n3)=O)C2)=O)cc(F)c2cn[nH]c2c1 CCCC(O)CC(=O)NC(C1CCNC1)(C)C.c1(C(=O)OC)cc(C(F)F)on1 c1(NC(C(CCSC)NC(C2C(=C)C2)=O)=O)ccc(=O)n(C(C)C)c1 CC(C)CC(C)(O)C(=O)N1Cc2[nH]nc(C(=O)NCC3CCC3(F)F)c2C1 C(C(F)(F)C(F)F)OCCNC(C1(n2cc(CC=C(Cl)Cl)nn2)CCOCC1)=O CC(CCC(C)(C)C)C(=O)N1C2CCC1C(F)C(NC(C1(C3CC3)CC1)=O)C2 CCCCCC(O)C(=O)N1CC(OC)CC1CNC(C12CC(F)(C1)C2)=O C1(C(N(C2CCCOC2)CC)=O)CCCN(C(=O)CCc2cscn2)C1 Cc1oc(C(C)(C)C)cc1C(=O)NCC1CCCN1C(N)=O N1(C(c2ncccc2Cl)=O)CCCC(C2CC2NC(C2CC(O)(C3CC3)C2)=O)C1 C1(CN(C2CCOC(C)C2)C(CC(C)O)=O)CCC(NC(=O)C(C)(C)C)CC1 C1(C(=O)NCCCN(C(c2cnnc(C)c2)=O)CC)CCC2(CCC2)C1 Cn1cc(C(N2CC3CC3(CNC(C3(CO)CCCO3)=O)C2)=O)ncc1=O c1(N)ccccc1C=O.N1(C(=O)NCCC)CCN(CC)CC1 CC#CCCC(=O)N(C1CCCN(C(=O)C(n2nccc2C)C)C1)CC C(=O)(C(O)CC(C)(C)C)NC(CCCC)CNC(=O)Cc1ccc(CC)c(F)c1 C(c1ccc(F)c2ccccc12)=CC(=O)N(CC)CC1CC(c2ccc(F)cc2)C1 c1(N(C(CN(C)CCc2nc(-c3cccs3)cs2)=O)C2CC2)ccc(F)cc1 C(=O)(CC(C(=O)NCCCCNC(=O)C(C(C)C)N(C)C)N1CCCCC1)OC CC1CCC=C1C(=O)NCCC1CC(NC(c2ccc(CC3CC3)cc2)=O)C1 N(C1COc2cc(Br)cc(F)c21)C(=O)CN1CCCCCC1 c1(-c2cccc(S(C)=O)c2)ccc2c(C(N3CCOC(=O)C3)=O)nsc2c1 N1(C(c2c(CC)ocn2)=O)CCCC2(CCN(C(=O)C3Cc4ccccc43)C2)C1 C1(NC(C2(C)CC=CCC2)=O)CC2(CCCCN2C(=O)CCC2CC2(F)F)C1 C(C(C(=O)N1CC(OC(F)F)C1)C(C)C)NC(C=CC(CC)C)=O C=CC(CCC)CC(=O)NC1CCCCC1NC(c1cnn2ncccc12)=O C=CCC(CNC(C1C=C(C)CS1)=O)C(=O)N1CC(n2cnnc2)C1 CC1=C(C(=O)NC(c2c(C)n[nH]c2C)(C)C)CCO1.C12CCN(CC1)C2=O c1(SC)cc(C(=O)N(CCCNC(=O)CC2C=CCCC2)CCO)oc1C n1(CC(=O)NC(CN2CCN(C(CCOC(C)C)=O)CC2)C)cc(F)ccc1=O c1(C(=O)NCCOCCNC(c2n[nH]c(C)c2Br)=O)cc2cscc2s1 c1(C(=O)NCC(C)NC(=O)CCC2CCCN2C)coc2c1C(O)CCC2 c1(NC(C(=O)N(CCN(C(C(CCC)OC)=O)C2CC2)C)C)ccc(Cl)cc1Cl c1(CNC(=O)CN(C2CC2(Cl)Cl)CCO)ccc2c(c1)CCC2 C1(CCOC)CN(C(c2ncn(C(C)(C)C)n2)=O)CCN1C(=O)CCCN=[N+]=[N-] C1(NC(CCc2cccc(OC)c2F)=O)CC2CCC(C1)N2C(=O)CCC(F)F Cc1nn(CC(N2CC(CNC(C3CC3CF)=O)C(O)C2)=O)cc1Br c1(C(=O)NCC2CC(NC(C3(COC)CC3(F)F)=O)C2)ccc(C)c(F)c1 C1(NC(CCCNC(=O)OC)=O)(CO)CCN(C(C2CCSC2)=O)CC1 c1(CC)cc(C(=O)NCC2CCCC2C(=O)NCC=Cc2cccnc2)ncn1 c1(NC(C(CC)Sc2ccccc2)=O)cnc(CNC(C2CC2COC)=O)cn1 C1(C(=O)NCC(CO)NC(C2(CC#C)CCCO2)=O)CC(=O)N(O)C1 C1(C(N2CC(CN(C(CCC#C)=O)C)OCC2)=O)CCc2cnnn2C1 N1(C(c2ccc(NC(C(C)OC)=O)cc2)=O)CC2CCN(C(=O)CC(C)(F)F)C2C1 C1(NC(CC2CCN(C)C2)=O)CC2CC1N(C(=O)CCn1cnnn1)C2 c1(OC)nccc(NC(C2CCCN2C(c2cnccn2)=O)=O)n1 c1(C(N2CC3C(NC(CCc4ccc(CC)cc4)=O)C3C2)=O)ccc(Cl)c(O)c1 C(=O)(CCC1=CCCCC1)N(C1CCN(C(C(CCC)OC)=O)C1)CCC Cc1c(C=CC(=O)NCC2CCCC2NC(C2CCOC(C)C2)=O)cnn1C N1(C(CC(C)n2cccn2)=O)CCC(C2CC2)C1CNC(C1(O)CCSCC1)=O N1(C(C=CCCC)=O)CCN(C(C2CC2(C)C)=O)CC2(C)CCCC12 c1(C(=O)NCC(CSCC)(C)C)ccc(C2CC2)cc1Cl c1(CC(=O)NC2CCN(C(C(CC=CC)CC)=O)C2)nn(C)cc1[N+](=O)[O-] C(=O)(C#CC(C)(C)O)N1C(C(N(CC(CC)(O)CC)C2CC2)=O)CC(O)C1 c1(CC)c[nH]cc1C(=O)N(C)CCOCCCNC(=O)CCC1CCOC1 Cc1ccc(C(N2CCC(CCNC(=O)C(O)C(C)C)CC2)=O)c(Br)c1F CCC(CCC(=O)NC(c1cscn1)C)NC(c1ccc(C(N)=O)o1)=O C1(C(N2C(C3CCN(C(c4ocnc4C4CC4)=O)C3)CCC2)=O)CCS(=O)(=O)CC1 CCCCC(CNC(=O)CCCOC(C)(C)C)NC(c1n[nH]cc1Cl)=O NS(=O)(=O)c1cnn(CC(N2CCCC2C(C)NC(c2ccc(Cl)[nH]2)=O)=O)c1 c1(C(=O)NCC2CCN(Cc3onc(CC)n3)C2)cnn2ccn(C)c12 c1(C(=O)NCC(CN(C(CCSCCCC)=O)C)C)cnc(C(N)=O)cn1 N1(C(C2CC(C(C)C)C2)=O)CCC(CC(=O)NCC2CSCCO2)C1(C)C C(=O)(CC(F)(F)C(F)F)NCC12CCN(CC1)CC2.CC12CCN(C1)C2=O c1(C(=O)NC2COCCO2)cccc(-c2cn(CCCCCCC3CC3)nn2)c1 n1(CC(=O)NCC(CNC(=O)C#CC2CC2)O)c(=O)oc2ccccc12 C1(c2ccccn2)CCCN(CCOCCNC(CN(CCOCC)C)=O)C1 c1(NC(=O)C2CC2)ccc(F)c(C(=O)N(c2cccnc2)Cc2ncsc2Br)c1 n1(CCOC(=O)NC(C)(C)C)ncnc1NC(=O)Cc1ccco1.C12CCCC1O2 c1(C(=O)NC(CC)CNC(=O)C(C)n2ccnn2)oc(P(C)(C)=O)cc1C c1(C(N2CC(OCCNC(C)C(=O)NC3CC3)C2)=O)cnnn1C1CCCCC1 c1(CN(C(=O)C(C2CC2)N(C(=O)CCOC)C2CC2)C)cccc(O)n1 Cn1ncc(C(=O)NC2CCOCC2NC(=O)CC2CCCC2O)cc1=O N1(C(C(CCC)(C)C)=O)CCC2(CCCN2C(c2cc(F)cc(Cl)c2N)=O)CC1 N1(C(C(c2cc(OC)no2)=O)=O)CCN(C(=O)C(=O)NC2COCC2(C)C)CC1 c1(C(N2C(C)CCC2C(=O)NCCOc2ccsn2)=O)ccnc(F)c1F c1(C(N2CC(CNC(C3CC4(CCC4)C3)=O)OCC2)=O)ccc2ncsc2c1 Cc1cccc2cc(NC(C3CC4CC3CN4C(c3n[nH]cc3I)=O)=O)sc12 C1(N(C)C(C2CCCC2NC(c2nnsc2C2CC2)=O)=O)CCOCC1 C(=O)(C(CCC=C)NC(=O)CC1CCCCC(=O)N1)N(CCCCC#C)CC N1(C(c2c[nH]c(=NCC)s2)=O)CC2CC(NC(C3(n4cccn4)CC3)=O)CC2C1 C(CCO)(C(=O)NCC1(O)CC(C(=O)Nc2cnccc2CO)C1)N(C)C Cc1ccc2c(NC3C(C)CN(C(C4CCCN4C4CC4)=O)CC3C)ncnc2c1 C(=O)(CCC(=O)N1CCC(C)(C(=O)NC2(c3ncon3)CC2)C1)NC c1(CNC(CCOCC#C)=O)cccc(C(=O)N(C2CCCCC2C)C)n1 N1(C(CC(c2c(C)cccc2)C)=O)CC(NC(c2sccc2C2CC2)=O)C2CC2C1 c1(CN=C(NC(C=C)C)NCC2CC2OCC)ccc2c(c1)n(C)c(=O)n2C c1(OC)ccc(S(=O)(=O)NCCC(=O)OC)cc1OC(c1ccc(Br)cc1)C C#CCC(CC#C)C(=O)NCC(CC=C)NC(=O)COc1ccc(F)cc1F C1(O)(CNC(C(F)=CC)=O)CCCN(C(C2CC23CC(C)(C)C3)=O)CC1 CC(C(CO)NC(=O)CC1C=CCC1)NC(=O)C(c1cncn1C)N(C)C C1(C)(CNC(C2(OC)CC(C)C2)=O)CCN(C(=O)C=Cc2ccco2)C1 N1(C(CCCOC(C)C)=O)CC(NC(=O)CC2=CCOCC2)C2CCCC12 C#CCC(O)C(=O)N1CCCCC1CCNC(=O)C(N1CCOCC1)C C1(NC(c2ccc(=N)[nH]c2)=O)COC2(C1)CN(C(=O)Cc1ccc(Cl)cc1)C2 C#CCCC(C(=O)Nc1cccnc1C)NC(C1C(C)(C)C1(F)F)=O N1(C(CCOC)=O)CCC(CCNC(c2ccsc2Br)=O)CC1C Cc1ncccc1C(N1CC(NC(=O)C(c2cccnc2)C)C1)=O C(=O)(CCC(CF)CF)NC(CNC(C(c1ccccc1)C)=O)CC(F)(F)F C1(CNC(C(CCC)OC)=O)CCCN(C(c2ccc(CCO)cc2)=O)CC1 C(CCC(=O)NC(C)CCNC(C1(C(C)(C)C)CCCC1)=O)OC(C)C C1(CNC(CCOC(C)=O)=O)CN(C(=O)COc2ccc(C#N)cc2)CCC1C N1(C(CC(C)(C)OC)=O)CCN(C(C2(C)CCCCC(C)C2)=O)C2(CC2)C1 C1(N(C)C(c2cn(-c3cnnn3C)cn2)=O)CCN(C(c2ccc(Cl)s2)=O)C1 CN(C1CN(C(=O)CC(F)F)CCc2ccccc21)C(=O)CC1CC=CCN1C CN1CCn2nc(C(N3CC(C(F)(F)F)CC3CNC(=O)C(N)=O)=O)cc2C1 c1(CN2CCC(NC(CCCN(C)C)=O)C(F)C2)nnc2n1CCCC2 N1(C(c2c(C)ccs2)=O)CCC(NC(c2cnn(C)c2Br)=O)CC(C)(C)C1 CC(C)C(C)(C)C(=O)NCC=CCNC(=O)C=Cc1cn[nH]c1 c1(CC(N2CCCC(CC)(NC(c3ccc(F)s3)=O)C2)=O)ccc2occc2c1 C1(C(N2C(CNC(Cc3nnc(C)o3)=O)CC3(CC3)C2)=O)CC2CCCC(C1)C2 N1(C(C(C)OCCN(C)C)=O)CCOC(CCNC(C2CCC3CC23)=O)C1 c1(C(=O)NC2C3(CN(C(CCC(CC)(C)C)=O)C3)CC2)cc2ccc(Cl)cc2s1 C(=O)(CCCCc1cccc(O)c1)NCC1(C(=O)NC2CCC(COC)C2)CC1 C(=O)(C(C#N)=C1N=CN(CC(=O)Nc2cnco2)N1)OCC CC(C)CC(CN=c1[nH]c2ccc(Cl)cc2s1)NC(=O)CN1CCCCCCC1=O C(C(C)(C)C(=O)N1CC(CNC(C23CCC(OC(C)C)C2C3)=O)C1)NC(C)=O Cc1c(C(N2CCC(NC(c3cccc(F)c3)=O)C(F)C2)=O)ccc2c1CCC2 c1(C(N2CC3C(CNC(C4ON=C(CC)C4)=O)C3C2)=O)cc2c(cn1)CCCC2 C(C(CC(C)C)NC(c1n[nH]c(CC)n1)=O)NC(C1(C(=O)OCC)CCCO1)=O Cc1cccc(C(N2CC(CCCCNC(=O)C(C)CN(C)C)C2)=O)c1C#N C1(COC)CCCN(C2CCN(c3ccccc3Nc3nnco3)C2=O)C1 C#Cc1ccc(F)c(C(=O)NC2CN(C(C3(C(=O)O)CCSCC3)=O)CC2O)c1 C=CC(CC)CC(=O)NC1(CCOC)CCN(C(C2CCNC(=O)C2)=O)CC1 C1(C(=O)NC2(C)CC2(F)F)CCCCC1CNC(c1nccs1)=O N1(C(C(C#C)(C)C)=O)CCCC2(CCC(NC(c3cncn3C)=O)C2)C1 c1(OC)cc(C(N2CCCC(C)C2CCNC(=O)CNS(C)(=O)=O)=O)ccc1O CCCCC(CC)C(=O)NC(CNC(=O)C=CCOC)C1CCC1 c1(CC(=O)NCC2CCCN(C(=O)CCc3nccs3)C2)coc2ccccc12 CCCCC(CC(=O)NC1CCC(C#N)CC1)NC(=O)Cn1ccnn1 c1(SC)ccc(C=CC(N2CC(NC(=O)CC(C)(C)C)C(C)C2)=O)cc1 C1(OC)CCN(C(=O)CC2C3CCCC3N2C(=O)CC(F)(F)F)CC1(C)C CC1CN(C)CC1NC(c1c(CNC(=O)CCc2ccoc2)cnn1C)=O c1(C(=O)NCCCCNC(C(CC#C)C2CC2)=O)cc(C2CC2)ccc1Cl CC(C)(CC(=O)NCC1(C2CC2)CCN(C(C2CCCC(O)C2)=O)C1)C(F)F C1(NC(CC2N(C)CC=CC2)=O)CC=C(C(=O)NCCn2cccn2)C1 C1(C(N2CC(O)(CCNC(=O)C(F)n3ccnc3)C2)=O)CC2C(C1)C2(F)F c1(NC)ccc(-c2nn[nH]n2)cc1C(N1CCCC(F)C1C(F)(F)F)=O CCC(CC(C)C)C(=O)NC1(C2CN(C(c3cc(C)n(C4CC4)c3C)=O)C2)CC1 C=C(C)CC(C(=O)OC)NC(=O)CN1CCN(C(=O)NC2CCC2)CC1 N1(C(CC2(C)CCC2)=O)CCN(C(=O)CCP(C)(C)=O)C2CCCCC12 CCC(C(=O)N1CCC(C(=O)OC)C(c2ccccc2)C1)C(C)(F)F C(CC(C(=O)N1CC(N2CCOC2=O)C1)NC(=O)C1=NOCC1)N(C)C c1(C(=O)O)ccc2nc(CC(=O)NC(CC3CCOC3)CO)cn2c1 c1(C(N2CCC(N(CC#C)C(C3CC3F)=O)CC2)=O)c(C)cc(OCC)cc1F C=CC(C)(CC)C(=O)NCCC1CC(C(=O)NCCC2OCCC2C)C1 C1(CC(=O)NCC2N(C(Cc3scc(C)n3)=O)CCCC2)CCn2cncc2C1 C(C(F)C(=O)NC1(C)CN(C(c2cn(Cc3ccc(C)o3)nn2)=O)C1)N(C)CC N1(C(C(CCC)C)=O)CCN(C(c2ccc(CF)cc2)=O)C2CCCC12 c1(C(N2CC(C(C)NC(c3ccc(-c4ccco4)s3)=O)C2)=O)ncc(F)cc1F C(=O)(C1COc2ccccc21)N(CCCNC(C(CC)OC)=O)C(C)C C#CCC(C(=O)NCCC(O)CCO)NC(c1cnncc1O)=O N1(C(=O)NC(C2C(=O)CCC2)c2cccnc2)CC(F)CC1Cc1cccc(Cl)c1 C1(C)CCN(Cc2onc(-c3ccccn3)n2)CC1.C1(N)CCCCO1 N12CCCC(C1)C2=O.N1(C(=O)CCCc2ncco2)CCOCC1CO c1(-n2c(-c3cn(CCC)nn3)nc(C(CCC)C)n2)ccc(Cl)cc1OC(F)(F)F C1(CNC(=O)NCCOc2scc(CC(N)=O)n2)CC2(CCNCC2)C(=O)O1 CCC1=NOC(CC(=O)NC2CC23CC(N(C(=O)CC(Cl)Cl)CC)C3)C1 Cc1coc(C(=O)NCC(C)(C)CNC(=O)C(C)Cc2ccccc2)c1 N1(C(CC(C)(C2CCC2)N(C)C)=O)CCC(NC(=O)Cc2ccon2)C(O)C1 c1(C(C)NC(=O)NC2CC2C(C)O)cccc(F)c1Cl c1(C(=O)NN(CC(C)NC(=O)CSCC)C(C(=O)CSC)=O)cc2ccccc2o1 c1(OC)cc(Br)c(C(C)NCc2nccs2)cc1OC C(=O)(C(N)C(C)O)N(CC)Cc1cnn(CC2CCOCC2)c1 c1(NC(C2(C)CCN2Cc2cccc(-n3ccnc3)c2)=O)csc2nccnc12 C(=O)(C1CCc2cccnc21)NCC(CNC(c1c(C)cc(C)o1)=O)C C(c1ccc(F)cc1)=CC(N1C(C2N(C(c3ncn(C)c3)=O)CCC2)CCC1)=O N1(Cc2c(OC)nccc2)CCC(F)(F)C(NC(c2cc(C)ccc2Br)=O)C1 c1(CCCNC(=O)NCC(C)(C)NC(=O)OC(C)(C)C)c(F)cc(Cl)cc1F Cc1cc2cc(C(=O)NC3CCCN(C(C4CC5(CC5)CO4)=O)C3)ccc2cn1 Cc1nc(C2CC2)sc1C(=O)NCC1CC2CC2N1C(=O)Cc1cccn1C Cc1ccc(OCC(=O)NCC2CCCN2C(=O)CN(C)C(C)C)c([N+](=O)[O-])c1 c1(C(N(CC(=O)N(CCC2CC2)CC2CC2)CCC)C)cc(CC)cc(C(F)(F)F)c1 N1(C(CN(CCCCCC)C(c2ccccc2C)=O)=O)CCCCC1CF c1(C2(C(=O)NC(CSC)CCO)CC2)cccc(Br)n1 C(C)(c1ccco1)=CC(=O)NCC(CCC)NC(=O)CC12CCC(CC1)C2 c1(C(=O)NCC2(NC(C(C)OCC#C)=O)CCOCC2)cc(Cl)c2n[nH]cc2c1 C1(C2C(NC(CCC=C)=O)CCO2)CCN(C(=O)Cc2coc(C)n2)CC1 c1(C(=O)NCC(CC)NC(C2CCCC2C)=O)ccc2cc[nH]c2c1F c1(C(N2CC(CNC(C(CCSC)OC)=O)CC2(C)C)=O)ccc(C#N)nc1O c1(C(=O)NC2CN(C(CN(C)CC)=O)CC2F)cc2cc(Cl)ccc2[nH]1 c1(C(=O)NCC(C)CNC(=O)C(F)CC2CC2)nc[nH]c2nccc1-2 CS(=O)(=NCC(=O)NCCOCCC1CC1)c1ccc(Cl)cc1.C(CC(F)(F)F)O C1(C(=O)NCCSCC(=O)N(C)Cc2nnnn2C2CC2)CC(C)(C)CCO1 N1(C(=O)CSCC2CCCO2)CC2(CCC2)CC1CNC(C1CCC=CCC1)=O C1(C(=O)NC(C2CCN(C(=O)COCC(F)(F)F)CC2)CO)CC2(CCC2)CO1 c1(OC)ccc(Cl)c(CC(=O)NC2CC2NC(c2cc(OC)nn2C)=O)c1 C1(NC(=O)Cc2cnnn2C)CN(C(N)=O)CC1N(C)C.CC1C(=O)N1 C(CCC(C(=O)N1CCN(CCO)C(C)C1)NC(=O)C(O)C1CCCC1)OC CN1N=C(CC(=O)NCC2(CNC(C3CC4CCC3CC4)=O)CCC2)CC1=O C1(CCNC(COCCC=C)=O)CCCCN1C(=O)CNC(c1ccoc1C)=O c1(CC)ccc(F)c(C(=O)NCC(C(C)C)NC(C2CCCCN2N=O)=O)c1F C1(C(=O)NCCCC(=O)NC)C2CC3C(C2NC(c2nc[nH]n2)=O)C13 C(=O)(C1=CCC(C)(C)CC1)NCC(C1CCN(C(C2CC(C)(C)C2)=O)CC1)C CC1(C)CC(C(=O)NCC(C)(O)CNC(C2(N(C)C)CCCC2)=O)CC(C)(C)C1 N1(C(Cc2cc(C)ns2)=O)CCC2CC(C1)CN(C(=O)CC1CC1C1CC1)C2 CC1(NC(c2ccn(C3CCCC3)n2)=O)CCN(C(c2ncncc2Cl)=O)C1 C(=O)(C1=NOC2(CCC2)C1)N1CCC(CN(C)C(C23CCC(CC2)C3)=O)C1(C)C CCCCCCC(=O)NCCOC1CN(C(=O)Cc2cc(C)ccc2Cl)C1 C1(NC(C2(C)CC=CC2)=O)C2CCN(C(c3ccc(Cl)c(C#N)c3)=O)CCC12 CC1CC=C(C(=O)NCC2(F)CC(NC(c3nc4ccccc4o3)=O)C2)CC1 C(C(C)(CCO)NC(=O)CC1CCCN(C(c2ccnn2CCF)=O)C1)OC C(CN=c1[nH]c(=NCc2cn(C3CC3(CC)CO)nn2)[nH]c2c(F)cccc12)n1ccnc1 C(=O)(C(F)(F)C(C)(C)O)NCCOCCN(C)C(C1CC2CCC1O2)=O c1(N2CCCC(C)(C(=O)NCc3ncccn3)C2)nc[nH]c2ncnc1-2 C(=O)(CCC#Cc1ccccc1)NCC1C(CNC(=O)CC2=CCCC2)C1 c1(OC)cccc(OCC(N2CCC(CNC(=O)C=Cc3nccs3)C2)=O)c1 c1(C(N2CC(OC)CC2(C)CNC(=O)CC(C)C)=O)ccc(C)c2ncccc12 c1(NCCCc2cccs2)ccc(C2CCC23CCC3)cc1.C12CC1C(=O)O2 C1(C(N2CCC3CCC23)=O)(N(C(C(C)n2ccnc2)=O)C2CC2)CC(C)(C)C1 CCC(C)(COC)C(=O)NCC(c1cn(CC(C)Oc2cncnc2)nn1)C O=C(C(O)CNC(c1csnc1Cl)=O)NCC1CCCO1 c1(C(=O)NC(C2CCCCN2C(=O)CCc2cnc[nH]2)C)ccc(O)nn1 C1(CNC(c2cnc(C)s2)=O)CCCCN(C(c2cnsn2)=O)C1 c1(C(=O)NCCN(C2CCCC2)C(C2CC3(CCCO3)C2)=O)cnn2c1CCC2 c1(OC)ccc(O)cc1C(N1CC(F)CC1C(N1CCCC1)=O)=O N1(Cc2n(CCC)ncn2)CC(N2CCN(C(=O)OC(C)(C)C)CC2)C(C)C1 N1(CC(=O)NC2C3(CN(C(COC)=O)C3)SCC2)C(=O)CC(C)(C)C1=O CCCCC(C(=O)NC)NC(=O)COC(C)(C)CC.C12C=CC(C1)C(=O)N2 S(=O)(=O)(c1ccc(NC(C)CN2CCCCC2C)cc1Br)N1CC(OC)C(F)C1 C1(OC)(CNC(=O)Cn2nnc(C(C)(C)C)n2)CCCCCC1 C12(CNC(CN(S(CC)(=O)=O)C)=O)CC(CN1C(c1ccnn1C(C)(C)C)=O)C2 C1(NC(COCCC(C)C)=O)CCC2(CCCN(C(=O)CC(F)(F)C(C)C)C2)C1 C(=O)(C(C)(C)N=[N+]=[N-])N(C)CC1CCCC(C(F)(F)F)C1 C1(C)(C(N(CCCCCNC(C2(CC)CC2)=O)C)=O)CCSCC1 CN1N=CC(CC(N2CC(O)(CCNC(=O)Cn3ccnn3)C2)=O)C1=O C(=O)(C1=Cc2cc(F)ccc2OC1)NC(CC)CNC(C1CCC1C(N)=O)=O Cc1oc([N+](=O)[O-])cc1C(=O)N(CCCN(C(=O)C(C)CC1CCCO1)CC)C(C)C C1(C)(C(N(CC(C)O)CCNC(=O)CCc2nncn2C)=O)CCOCC1 C1(C(=O)NCCCN(C(=O)CC2(C3CC3)CC2)C)CCN(c2ncccn2)C1 C12(COCC)CCC(C(=O)NCC3CN(C(=O)CC(C)(C)C)CCCO3)(CO1)C2 CC1CN(C(=O)CCC2CCN(C)C2)CC1NC(C1CN(CC(F)(F)F)C1)=O CCC(CC)C(F)C(=O)NCC(C)(CC(C)C)NC(=O)CN(C)CCO c1(NCC2N(CC)CCC2)nccc(=NCC(OC)c2ccccc2)[nH]1 N1(C(C)C)CC(C(=O)NCC2CC2CN(C(C2CSC2)=O)C2CC2)C1.CC C1(C)(CNC(C(c2scc(C)n2)(F)F)=O)CN(C(C2CCCCC2)=O)C(C)(C)C1 Cc1nc(C(=O)N(CC(O)CNC(c2c[nH]c(=N)s2)=O)C)sc1C c1(C(N2C(C(=O)NCc3ccccc3)CCCC2)=O)ccc2cc(Cl)ccc2n1 CCC(C)CC(=O)NC1CC1CNC(c1cn(-c2ccccc2)nc1C)=O Cn1ccc(C(F)=CC(N2CC(O)(CNC(=O)CC34CCCC3C4)C2)=O)n1 c1(C(=O)NCCCOCCNC(c2cc(Cl)ns2)=O)n[nH]c2cccnc12 c1(OC)ccc(F)c(C(=O)NCC2CC2CC(=O)NC2CCN(C3CC3)C2=O)c1 C1(C(N(CCOCCN(C(=O)CNC=O)C)C)=O)CCCC2(CC2)C1 C1(NC(c2c(SC)cc(C)cc2)=O)CC2CCC(C1)N2C(=O)C(C)CCN(C)C N1(C(c2cccc3sncc23)=O)CC2CC(C2)c2ccc(Br)cc21 N1(C(c2n(C(C)C)ccn2)=O)CCC2CCC12CNC(=O)C(F)(F)C(F)F Cc1cc(C=CC(=O)NC2(N3CCOC3=O)CC2)ccc1Br c1(C(=O)NC(c2cccnc2)CNC(CC2C(OCC)CC2)=O)cc(Cl)ccc1O Cc1ccc(-n2ccnc2)c(NCc2cccnc2)c1 c1(OC)cccc(SCCCCO)c1.N12CCN(CC1)c1nccn1CC2 N1(C(CC(CC)OC)=O)CC(O)(C2(CNC(c3cn(C)nc3C(C)C)=O)CC2)C1 C1(CNC(C(C)OCC(F)F)=O)CC(O)C(O)CC1C(=O)N(CCC1CC1)C(C)C C1(CNC(c2nc(OC)oc2)=O)CCC(C(F)(F)F)CC1.c12sccc1NC2=O Cc1ccc(CC(N2CCN(C(C3CCCCCC3)=O)C3CC23)=O)cc1[N+](=O)[O-] c1(SC)ccccc1C(=O)NC1(C)CN(C(=O)CN(CC(C)(C)C)C)C1 Cc1nn(C)cc1C(=O)NCC(C)(C)CNC(=O)C(F)CC1CCOC1 N1(C(C2CCOC2)=O)CCCC2C1CCN2C(=O)CN1CCC(F)CC1 CN1CCC(C)(C(N2CC(O)CC2CNC(c2c(C3CC3)n[nH]c2Cl)=O)=O)C1 Nc1cc(C(=O)NC2CCC(CNC(C3CCCC34CC4)=O)CC2)ccc1Cl N1(C(C(CC)C#N)=O)CC2(CC2)CC1CNC(=O)CN1CCCCS1(=O)=O C1(C(C)(O)CNC(C2CCNC2=O)=O)CCCN(C(c2cncc(F)c2)=O)C1 C1(NC(c2c(OCC)nccc2)=O)CN(C(=O)CCC=C(C)C)C2(CCCC2)C1 N1(CC)CC(NC(=O)C(Cc2ccco2)NC(C2CC3C=CC2O3)=O)C(C)C1 c1(C(N(CC(C)NC(C2(S(N)(=O)=O)CCC2)=O)C)=O)ccc2ccccc2n1 N1(C(CCNC(=O)OCC)=O)CC(C)CCC1C(=O)NC1CCCC1C C1(F)(C(NOC(c2cccnc2)C)=O)CCCN(C(C2CC2C(C)(C)C)=O)C1 c1(C(N2CCC(C)(CNC(CC=C=C)=O)C2)=O)ncc(N)cc1Cl C1(CC(C)NC(C=NOC)=O)CCN(C(c2ncccc2C(=O)OCC)=O)CC1 CCC(CCC(=O)N1CCC(C#N)(CO)C1)NC(c1cnc(C)c(C)c1)=O c1(OC)c(F)ccc(Cl)c1C(=O)NNC(=O)c1cc(-c2cccnc2)[nH]n1 C(=O)(CC1COc2ccccc21)NCCC1(O)CCCN(C(C(C=C)(C)C)=O)C1 c1(CC(C)C(=O)NCC2CC(F)(CNC(C3(F)CC3)=O)C2)ccccc1Cl C(=O)(CC(C(F)F)n1ccnc1)NCC1(NC(c2c(C)nn[nH]2)=O)CCOC1 c1(C(N2CCOC(C3CCOCC3)C2)=O)ccnc2cc[nH]c12 Cc1cc(C(=O)NCC(CNC(C2(CO)CCC2)=O)S(C)(=O)=O)ncc1C#N CC1C(NC(=O)COCC2CC2)CC2CCC1N2c1ccccc1[N+](=O)[O-] CC1CCN(C(c2cc(Cl)ns2)=O)CC1CNC(c1ccns1)=O C1(CNC(c2nn(C)c(F)c2)=O)CC2CCC1N2C(C1CCCC12CC2)=O N1(C(=O)OC(C)(C)C)C2CCC(C2)C1C(N1CCN(CC(O)C(F)(F)F)CC1)=O c1(C(=O)NC(CNC(c2n(C(CC)C)ncc2)=O)CCOC)cc(C#N)on1 N1(C(CCN(CCC)C)=O)CC(NC(c2cc(C)cnc2O)=O)CCC1C C#CCC(C)(C)C(=O)NCC1CC(C)N(C(c2cc(C)n(C3(OC)CCC3)n2)=O)C1 N1(CC(=O)NC2(CF)CCN(C(C(CCC)OCC)=O)C2)C(=O)CC(C)(C)C1=O C1(OCC)(CC)CN(C(C2(F)CC(C(N3CC(C(=O)OC)C3)=O)C2)=O)C1.C=O.OC C12(C(=O)NC3(CNC(c4csc(Cl)c4)=O)CC3)COCC1C2 c1(C(C)=O)cncc(C(=O)NC(C)CN(C)C(c2sc(C)cc2OC(F)F)=O)c1 c1(NC(CSC)CC2CC2)cc(=O)n(CC(C)C)nc1Cl CC(=O)CCCC(=O)N1CCC(CCF)(C(=O)N(C2CC(C(N)=O)C2)C)C1 C(=O)(C(CCO)NS(C)(=O)=O)NC(CNC(C(C)(C)OC)=O)Cc1ccccc1 C(=O)(CCCCC(N)=O)NC1C(NC(C(C)(O)Cc2ccccc2)=O)CCC1 C(=O)(CC(C)P(C)(C)=O)NCC1(F)CCC(NC(C2CC(C)=C(C)CC2)=O)C1 C=CCC(F)(F)C(=O)NCC(C)(Cn1cccn1)NC(=O)CN1CCC1C c12cnc(F)cc1C(=O)NC(=O)COCCNC2=O.c1(NC)cc(Cl)sc1Cl C1(N(C)C(C2(n3cc(CS(C)(=O)=O)nn3)CC2)=O)CCN(c2ccccc2)C1 c1(C(N2CCC(N(C(c3cc(C)no3)=O)C)C2)=O)c(C)nc(C)n1O C(c1ccc(F)cc1)=CCC(=O)NC(CNC(c1ccn(CC)n1)=O)C(C)(C)C N(C1CN(C(=O)CCCN(C)C(C)C)Cc2ccccc21)C(CCOCCC)=O CC1(C)C(C)(C)C1(F)C(=O)NCCC(=O)NCC(C1CCCC1)O N1(C(C(C)OC)=O)CC2CCN(C(c3cc(O)ccc3C)=O)CC2C1 c1(C(C)C2CC2)cccnc1.C1(N2C(=O)CC23CC3)CCCC1 C(N=c1[nH]cc([N+](=O)[O-])c(=N)[nH]1)C1(F)CC(NC(C2C(C)CCC2)=O)C1 C1(C(CC)C)CCN(C(c2cccc(CN(C)Cc3cccs3)c2)=O)CC1 C1(C(N(C)CC2CN(C(=O)CCC3CCCN3C)C2)=O)C2CCC(=O)C12 C1(CNC(C2(C#N)CC2)=O)CC2(CCN(C(=O)COc3ccccn3)CC2)CO1 c1(C(C)C)cc(C(=O)NC23CC(NC(=O)CC#N)(C2)C3)n[nH]1 c1(C(=O)NC(CC(C)C)CNC(=O)C(C)(C)c2ccsc2)ccc(Cl)c(F)c1 C=C=C(C)CC(=O)N1CC2CC2(NC(c2sc(Br)cc2C)=O)C1 c1(COC(CC(CC=CC=C)c2ccccc2)=O)nc(C)cc(C(F)(F)F)c1C#N c1(CNC(C2CCC(C)N(C(=O)Cc3cncn3C)C2)=O)cnc2cc[nH]c2c1 CCCCCCCCNC(=O)C(=O)N(CCCCc1nccs1)CC(C)C C1(C(=O)NC2CC2)CSCN1C(=O)C(c1ccccc1)F Cc1c(F)ccc(C(=O)NC2CCN(C(c3nc(=O)n(C)[nH]3)=O)C2C)c1C C=CC1(C(N2CC3(OC(C)=O)CC2C3)=O)CCN(C(c2cncc(F)c2C)=O)C1 c1(C(=O)NC(CNC(C(C=CC)O)=O)(C)Cn2cccn2)cn(C(C)C)cc1C C1(C(=O)NC2CCC(NC(c3cnc(COC)s3)=O)CC2)CNC(=O)CCC1C C(=O)(C(CCC(C)(C)C)N1CCN(CC(C)(C)O)C(C)C1)NCCC c1(CCC)c(C(=O)NC23CC(C2)N(C(=O)Cc2sccc2C)C3)cnn1CCO C1(NC(C=C2CCC(C)C2)=O)CCN(C(c2n[nH]c3c2COC3)=O)C12CC2 C1(C(=O)NCCN(C2COC2)C(c2ccccn2)=O)CC(=O)N(C(C)(C)C)C1 c1(CNC2CC2CN(C)C)ccc(S)nc1.C(=O)(CCC1CCC1)OC C12(C(=O)NCC(C)NC(C3(C4CCCCO4)CC3)=O)CCCN(CC1)C2 C12CC(C1)NC(=O)CN(CCCOC)C(=O)C2.c1(C(=O)OC)cn[nH]c1 N1(C(C(C(C)C)(C)C)=O)CC2CC(NC(c3cnc(O)c(F)c3)=O)CC2C1 C1(CC2(C(N3C(CNC(=O)COc4ccccc4)C=CC3)=O)CC2)CCS(=O)(=O)N1 N1(C(CC(CNC(=O)C2=C(Cl)CC2)OC)=O)CCS(=O)C(C)C1 CC(C)C(CC(=O)N1CC(CNC(=O)C(C)O)C1)C(C)C Cc1nn(C)c(C)c1CC(C)C(=O)NCCN(C(c1ccc(Cl)cc1)=O)C(C)C CC1CC(=O)NCC1C(=O)N(C1(CCC(=O)N(C)CC2CC(F)(F)C2)CCC1)CC C12(NC(c3csc(Cl)c3)=O)CCN(C(=O)CCCCc3ccccc3)CCC1C2 N(C1CCCc2n[nH]cc21)C(C(C(C)OC)NC(=O)C(C)CN(C)C)=O c1(CC)cc(C(N2CCOCC2C2CCOC2)C(=O)NC(C)CC)cc(C)c1 C1(Cc2cn(CCCC)nn2)COCCN1C(c1cc(Br)n[nH]1)=O c1(C(N2CC(C)C(NC(=O)CC3CC3)C2)=O)nn(C)c(=O)c2ccccc12 C1(NC(c2c(C(C)C)noc2)=O)CC2CCC(C1)N2C(=O)C(C)C1CCCO1 N1(C(c2cnn(C(C)C)n2)=O)CC(C)CN(C(=O)C(C)c2cccs2)CC1C C(=O)(C1=NOC(CNC(=O)CSCC2CCCO2)C1)N1CC(COC)C(F)C1 c1(CC(=O)NCC2(F)CCN(C(COC)=O)C2)cccc2c(C)csc12 c1(C(=O)NC2(CO)CCN(C(c3[nH]c(CC)c(Cl)n3)=O)C2)nccc2[nH]ccc12 N1(C(CC2C3CN(C(C(CC=C)C)=O)CC32)=O)CC2CC3CC2C1C3 C1(C(N2CC3C(C(N4CCC(O)C4)=O)C3C2)=O)(CC)CCNC1=O c1(OC)ccccc1NC(=O)NCC(N1CC(NC(=O)C(Cl)=CCl)C2CC12)=O C=C1CC(CNC(=O)Nc2cnc(C3CC3)[nH]2)(CSC)C1.C1(=O)CC(=O)N1 C1(N(C(C2(C)CCOC2)=O)CCO)CCN(C(=O)C(c2ccccc2)N(C)C)CC1 c1(OC)ccc(C(N2CCC(NC(=O)Cn3nnc(C4CC4)n3)C2)=O)cc1Br C1(C(=O)NC2(COC3(CF)CCC3)CN(CCO)C2)(C(=O)O)C=CCC1.COC c1(OC)cccc(CNC(=O)CNC(=NC)Nc2cccc(F)c2)c1 c1(SCC)ccccc1C(=O)NC1CCCCC1CNC(c1nc(O)c(C)s1)=O N1(C(c2cc(CC)c(=O)n(C)c2)=O)CC(C)(CNC(c2cn[nH]c2)=O)CC1(C)C Cc1cc(C(=O)NC(C2CCN(C(=O)CSc3nccn3C)CC2)C)nc(O)n1 C1(NC(Cn2ncc(C)c2)=O)C(C)CN(C(c2cc3cnccc3o2)=O)CC1C Cn1ccc(CCC(=O)NC2CC(CNC(=O)CCC3CCC(=O)C3)C2)c1 C(=O)(C1c2c[nH]nc2CN1C(c1ccn(C2CC2)n1)=O)NCC(COCC)C CC1(CNC(=O)CCSc2nnnn2C2CC2)CC(NC(C2CCC2)=O)C1 CN1CCC2(CC1)CN(C(C1C=CCCN1C(c1ccnnc1O)=O)=O)C2 C(=O)(C(C)(C)C(=O)NCCC1CC(NC(=O)Cc2nc[nH]n2)C1)OC C(=O)(CC1=NNC(=O)C1)N1CC(C2OCCN(C(CCn3ncn(C)c3=O)=O)C2)C1 c1(CC(=O)NCC(C)CN(C)C(C2CC(C)OC2C)=O)cccnc1Cl n1(CC(CC)C)cc(CCN(C(=O)C(C)Cn2ccc(C)n2)C)nn1 C1(COC)(CNC(c2ccc[nH]2)=O)CC1C(N1CCC1CC1CC1)=O N1(C(C2N(C(C3(C)CNC(=O)C3)=O)CC=C2)=O)CCNC(=O)CC1 c1(C(=O)NC2C(CNC(C(CSC)O)=O)CCC2)cc2ccccc2cn1 CCCC(C(=O)OC)C(=O)NC1CC(C(=O)NCCNS(N)(=O)=O)C1 C1(OCC#C)CCN(C(C2CC2CNC(c2cccnn2)=O)=O)CC1 Cc1ccc(O)c(CC(=O)N(CCNC(c2ccc(NC=O)cc2)=O)C(C)C)c1 C1(NC(c2nc(Cl)cs2)=O)CN(C(c2c[nH]nc2[N+](=O)[O-])=O)C2(CCOC2)C1 c1(OC)cc(C(N2CCN(C(c3sccc3C3CC3)=O)CC2C)=O)ccc1F CC1CN(C(c2cc(Cl)cn2C)=O)CC(C)N(C(=O)CN2CCC(CO)CC2)C1 N1(CC(N2CCC(N(CC#C)C(c3cnc(Cl)s3)=O)C2)=O)C(=O)CC(C)(C)C1=O O=C1CCC2CN(C(C3CC(=O)N(C(F)F)C3)=O)CC2N1 c1(OC)ccnc(C(N2CCCC(N(CCN)CCO)C2)=O)c1OC S(=O)(=O)(c1ccc(NCC=C2CCSCC2)cc1Br)NC1CCC(SC)C1 CP(C)(=O)C(O)C(=O)N1CCC(CNC(=O)C(F)(F)CC2CCCO2)C(O)C1 c1(C(=O)OCC(=O)N(c2cncnc2)C)ccc(C#N)cc1F CC(C)CCCCC(=O)NCCCOCCN(C)C(C1(C)CCC(F)(F)CC1)=O c1(NC(CC(C)F)=O)ncccc1S(=O)(=O)NC(=O)CS(=O)(=O)C1CC1 C1(C(=O)NCC(CC(=O)NC)C)CC12CCN(C(=O)CC#N)CC2 c1(C(=O)NC23CC(CNC(c4ncc(F)cn4)=O)(C2)C3)cnc2nccn2c1 c1(CC)cccnc1-c1nc(-c2ccc(F)cc2)nn1CC(C)C CN1CCN(C(C2CCC(O)CN2C)=O)CC1CNC(c1ccc(F)cc1F)=O CCC(CC)CCC(=O)N1CCCC(NC(=O)C(n2cc(C)cn2)C)C1C Cc1cc(C(=O)NCC(C)N(C)C(c2cc[nH]c2)=O)cc(Br)c1C C(=O)(C1=CCS(=O)(=O)C1)N(C1CN(C(CC2CCCN(C)C2)=O)CC12CC2)C c1(C(N2C3CN(C(CC(CC)C)=O)CC2CC3)=O)ccc(C)c([N+](=O)[O-])c1 c1(C(N2C(CNC(CCCCCSC)=O)C(CO)CC2)=O)ccc2nccnc2n1 c1(C(=O)NCCC2(NC(c3ccoc3)=O)CCC2)cc(-c2ccco2)on1 c1(C(=O)NC(C(=O)NC(COC)CO)C2CC2)csnc1C c1(COC)nn(C)cc1C(=O)NCC(C(=O)N(CCCC(=O)OC)C)OC C12(NC(C(C3CCOC3)OC)=O)CC(NC(c3n[nH]cc3C)=O)(C1)C2 N1(CC(=O)NC)CCC(C)CC1.C12CCN(C1)C(=O)CC1CCCN1C2=O Cc1ncc(C(=O)NC(CCNC(C2CCCC23CCC3)=O)C(C)C)cc1C#N C(=O)(C(C)(C)C(F)(F)F)NCC(CC(C)C)NC(C1CCn2nnnc2C1)=O CC1CCSCCN1C(C1CCN(C(c2cc(O)cc(=O)o2)=O)CC1O)=O N1(C(C)C)CCN(C(C2CCC(NC(=O)CC(F)(F)F)CO2)=O)CC1 c1(C(N(CC(F)(F)F)CC=C)=O)cn(CC)nc1CC C1(C(=O)NCC(C2CC2)SC)CCN(C(=O)C(C)Cc2ccco2)C12CC2 Cc1ccc2cc(C(=O)N(CC(C)(C)NC(=O)CN3CCCC3C)CC)[nH]c2c1 N1(C(C(CC)=CC)=O)CCN(C(C2CC(CF)C2)=O)CC1c1ccccc1OC Cc1cc(O)ncc1C(N1CC(F)(C(=O)NC2COC3(CCC3)C2)C1)=O c1(C(=O)NC2C(NC(C3(C=C)CC3)=O)CC2)ccc(COC(C)=O)cc1 CCCC(CCC)C(=O)N1CCCC(CNC(C2CC3(C2)CC32CCC2)=O)CC1 c1(OC)nn(C)cc1C(=O)NC1CCCC1NC(c1cncc(N)c1)=O C1(NC(c2cc(=O)cc(Cl)[nH]2)=O)CCN(C(=O)Cc2ccsn2)CC(O)C1 C=C(C)CC(C)C(=O)N1CC(CN2CCN(C(c3sc(CC)nc3C)=O)CC2)C1 C1(CNC(CC=C(C)C)=O)OCCC1C(=O)NC(C1CCC1)C1CC1 C#CCCCCC(=O)N1CCC(CC=C)(C(=O)NC(c2ccsc2)C)C1 C(=O)(CC1C(=O)N1)OCC.c1(SCC2C(NCC(=O)C(C)=O)C2)nc[nH]n1 c1(CO)cc(O)ccc1C.C#CCC1C(=O)N(C)CCCC(=O)N1 C1(C(C(=O)NCc2cccn2C2CC2)F)CCN(C(=O)CCc2ccncc2)C1 C1(C)(OCCCCC(C)O)CC(F)(F)CN1C(=O)OC(C)(C)C c1(CN(C)C(C2CC2C#N)=O)nc(CNC(C2(CO)CCCCC2)=O)cc(O)n1 c1(NC(C2C(CNC(C(CCC)C#N)=O)OCC2)=O)ccn2nccc2c1 CCC(C)(C(=O)NCCOCCNC(=O)C(c1ccc(Cl)cc1)(C)F)C(F)F c1(CN2CCC(C(C)C)(CO)C2)cnc2n1CCCC2 C(c1ccc(F)nc1)=CC(N1C(C)CC(NC(=O)CCc2ccc(Cl)nc2)C1)=O N1(C(CC(C)(C)CNC(=O)CCc2nc[nH]n2)=O)Cc2ccccc2C1 Cc1cnc(NCc2cccc(NC(c3c(C)coc3C)=O)c2)nc1 c1(CC(=O)NCCC(C)N(C(=O)Cc2cn(C)nc2C(F)F)C)cccnc1O C1(CC(N2CCCC(N(C)C)C2)=O)N(C(=O)C=CCN2CCCC2)CCC1(C)C c1(C(=O)NCCC2(NC(c3ccn(CCCC)n3)=O)CC2)ccnc(OC)c1 C12(C(=O)NC3C(C(C)O)CC3)C(NC(=O)CC3CCC3)C3CC1C2C3 N1(CCCC(=O)OCC)CCC2(CC1)CC2NC(N1Cc2cccnc2C1)=O C(=O)(C(C(C)O)NC(=O)Cn1nc(C)cc1C)NC(c1nc[nH]n1)CC O(S(=O)(=O)c1c(C)nn(C)c1C)c1ccc(C(=O)OC)cc1 n1(C(C)C)cnc2ccc(NC3(CNC(=O)C4CC4)CC3)cc12 c1(OC)ccc(C(N2CCCC(CCN(C)C)C2)C(=O)NC2CCOC2)c(C)n1 C1(NC(c2cc(-c3ccc(Br)cn3)on2)=O)CC12CCN(CC1CCOC1)CC2 C1(NC(C(C2CCCC2)OCC)=O)CC(NC(=O)CCCc2ccsc2)C(O)C1 N1(C(CC2(OCC)CC2)=O)CCc2ccccc2C(NC(c2ccn(C)n2)=O)C1 c1(NC(=O)CC2CCCN(C(c3sccc3F)=O)C2)cc([N+](=O)[O-])ccc1Cl N1(C(c2c(OC)cc(Br)cn2)=O)CCC2(CCCN2C(=O)C=C2CCC2)C1 N1(C(c2cc(CC)sn2)=O)CCCC(C)(C)C1CNC(c1cc(C)on1)=O c1(C(=O)NCC(CO)NC(C2C(C)OCCC2)=O)ccc2c(c1)CCC2 c1(C(=O)NC2C(C)(C)CN(C(=O)C(O)P(C)(C)=O)CC2)cccc2cnccc12 c1(C(=O)OCC)cncc(CN2CCC(CN)C2)c1.n1(C)ccnn1 C1(NC(C(N2CCOC2=O)C)=O)CCOC12CCN(C(c1ccc(Cl)s1)=O)CC2 C(=O)(C(C)(C)C(C)(C)O)NC(CC)CCC(=O)N1CCCC1CCCO C1(C(=O)Nc2ccccc2Cl)COCCN(C(=O)C(F)OC(F)(F)F)C1 CC1N(C(c2conc2C(C)NC(=O)C=Cc2ccsc2)=O)CCOC1(C)C C1(C(N(CCCC)CC)=O)CCC(NC(=O)COC2CCCC2)C1 N1(C(Cc2ccc(C)nc2Cl)=O)C2CCC1CN(C(=O)C(O)CC(C)C)C2 C1(C=C)(CC(=O)NCc2scc(CNC(C(C=C)(C)C)=O)n2)CCOCC1 c1(C(=O)NC(C(C)NC(C2CN(S(CC)(=O)=O)C2)=O)C)ccc(Cl)c(C)c1Cl c1(OC)ccc(CC(=O)NCC2CCCCN2C(c2cccnn2)=O)c(OC)c1 c1(C(=O)NCC2(C(C)NC(C(C)OCC#C)=O)CC2)c(F)ccc(OC)c1N C1(CNC(C(CC)NC(N)=O)=O)CC2CN(C(C3CNC(=O)N3C)=O)CC12 N1(C(COC(C)=O)=O)CCCN(C(c2cc(OCCC(C)C)ccn2)=O)CC1C c1(C(=O)NCC(C)(C)CNC(=O)C2=CCCOC2)c(C(F)F)nc2ccccn12 CCC(C)(C)C(=O)C(=O)N1CC(F)(F)CC1(C)CNC(=O)Cn1cc(C)cn1 C1(NC(CCC2C(C)C2)=O)C2CC1CN(C(C1(O)CCOCC1)=O)C2 C(N=c1[nH]c(Cl)nc2c1SCC2)C1C(NC(C2N(C=O)CCCC2)=O)CCC1 C1(C(=O)OCC)CN(C(=O)CC2CCC(C)CO2)CCO1.c12cn(nn1)C2 CC(C)(CF)C(=O)N1CCC(N2CCN(C(c3scnc3C(F)(F)F)=O)CC2)C1 c1(C(N(C)CC2N(C(CC(C)F)=O)CCC2)=O)cnnc(O)c1 CS(=O)(=O)CCNCC(N1CCCC1CO)=O N1(C(C2CC(OC)C2)=O)CC2CC2(C(=O)Nc2csc(CCC(F)(F)F)n2)C1 C1(C2CCOCC2)(NC(C2N(C(C(C(=O)OC)C)=O)C(C3CC3)CC2)=O)CC1 C1(NC(C2N(C=O)CCC2)=O)CC2(CCN(C(C3C(C4CC4)C3(F)F)=O)CC2)C1 Cc1cc(N2CCN(CCNC(=O)Nc3csc(C)c3)CC2)nc(C(C)(C)C)n1 c1(CC)ccc(OCC(N2CCC(N3CCN(C(=O)CC(C)C)CC3)C2)=O)cc1 c1(OC)ccc(CCC(=O)NCC2CC(NC(C3(C4CCC4)CC3)=O)C2)cc1 Cc1nc(-c2ccc(F)cc2)oc1C(N1CCCC(CNc2ncccn2)C1)=O c1(C(N2CC(OCCNC(c3csc(CO)c3)=O)C2)=O)csc(-c2nc[nH]n2)n1 c1(C(C(=O)NC(C)C)N(C2C(C)CCCC2C)C2CC2)cc2cnccc2o1 C=CCC(C)(C)C(=O)NCCOC1CCN(C(=O)C(n2ccc(C)n2)C)C1 C12(NC(=O)COCc3nc[nH]n3)CCCC1CN(C(=O)CCc1ccncc1)C2 C(=O)(C1CCCc2cccnc21)NCCCN(C(c1cnc(CCCC)s1)=O)C C#Cc1cncc(C(N2CC(C(C)NC(=O)CNc3nccs3)C2)=O)c1 CC1(C)CC2CC(C)(CN2C(C(=O)NCC(F)F)c2cnc[nH]2)C1 c1(NC(C2CNC(=O)N2)=O)cncc(C(=O)NC2CC(C)(NC(=O)NCC)C2)c1 N1(C(CSCCOC)=O)CC(NC(c2nccn3nccc23)=O)CC2(CCC2)C1 Cc1cc(C)n(CC(N2CC(NC(c3cc(-c4ccco4)c[nH]3)=O)C(O)C2)=O)n1 Cc1oc(C(C)(C)C)cc1C(=O)NCC1CC1NC(=O)CSc1cnn(C)c1 C(CCCCN)NC(=O)C(C)OC.c1(N(C(COC)=O)CC2CCCO2)ccccc1 c1(C(=O)NCCC(C)(C)NC(c2ccc(F)o2)=O)cc2c(nc1O)CCOC2 C(C(C)C(=O)NC(C)(CNC(=O)C=CCOC(C)(C)C)CC)NC(C)=O N12CCC(F)(F)C(C1)C2.c1(NS(C)(=O)=O)ccccc1C(=O)NC(=O)COC1CC1 C(=O)(C(F)(F)c1csc(Cl)n1)NC(C)C(C1CCCCC1)NC(=O)C=CCF c1(CN(C(C(=O)OCC)c2ccoc2)CC=C)ccc2c(c1)OCCCO2 c1(CCC)ccc(CN(C(=O)CNC(=O)CC2CCC2)CC2CC2)s1 CC(C)(CS(C)(=O)=O)C(=O)NCC1CCC1NC(c1ccnc2ncnn12)=O C1(NC(C(C)c2ccco2)=O)CC2(CCN(C(=O)CC(C)(C)F)CC2)C1 CCCC(CC)C(=O)NC(Cn1cncn1)C(=O)N(C)CCN1CCCC1=O C1(C(=O)NC(C(CC)CCO)C)CCN(C(=O)CC2=C(C)OCC2)O1 C1(NC(c2ncc(OC)cn2)=O)CCC2(CC1)CN(C(C)=O)CCO2 CCCCCCCCCCC(=O)NC1(C)CCN(C(C2CC2(F)Cl)=O)CC1 N#Cc1cnc(NC(C2CC3CC3N2C(c2c(Cl)cccc2I)=O)=O)c(Cl)c1 N1(C(C2CCN(CC)C2)=O)CCCC(C(=O)NCCc2ccns2)C1C c1(NC(C2CC3N(C(CNC(C)=O)=O)C(CC3)C2)=O)ccc(Br)c([N+](=O)[O-])c1 c1(NC(CN(CCCN(C(C2CCC(C#N)C2)=O)C2CC2)C)=O)cccc(Br)c1 c1(-c2n(CC)nc(-c3ccoc3)n2)cc(C)n2ncc(Br)c2n1 C12(C)CC13CCN(CC3)C2=O.c1(NC(=O)OC(C)(C)C)ccc(C#N)cn1 N1(C(COCCC)=O)CCCC(C)C1CNC(=O)CCc1cn(C)nn1 c1(C(=O)NCC2CCN(C(CC3(CCCSC)CCCC3)=O)C2)n[nH]c(C)c1C C1(NC(=O)CONC(=O)CC2CCCOC2)CCC(CO)CC1 C1(C(=O)NC(C=C)C)COC(CNC(C2CCN2CCC=C)=O)C1 c1(CC(=O)NCC(C2CCCC2)NC(C=C(C)C(F)F)=O)ccccn1 N1(C(c2cc(OCC)no2)=O)CCN(C(=O)CC2CC(OC)C2)CC1CF C1(C(N(CC(O)CO)CC)=O)CCCN(C(c2ccc[n+]([O-])c2)=O)C1 CC(C)C(C(=O)Nc1ccc(N)cc1)NC(=O)NC1CCN(C)CC1 C1(NC(C(CCC)OCC)=O)CCC2CC1CN2C(c1nnc(S)n1C)=O c1(CNC(C2C(C(C)C)C2)=O)ccc2c(c1)CCCC2NC(=O)CC(C)(C)CF c1(C(=O)OCC)ccn2c1CN(CCC(O)c1ccco1)CC2.C1CO1 N1(C(C2(OC)CCCNS2(=O)=O)=O)CC2CN(C(=O)C=CS(C)(=O)=O)CC2C1 N1(C(C=CCN(CC(F)(F)F)C)=O)CC=CC(NC(=O)C(O)C(F)F)C1 Cc1ccc(F)c(N)c1C(=O)NCC1C2CN(C(=O)C(C)CO)CC12 N1(C(C(C)SCC)=O)CCN(C(c2onc3c2CCCC3)=O)CCC1C CN(C1CCCc2cnn(C)c21)C(=O)C(=O)NCc1c(F)cncc1Cl c1(C(=O)NC(CC2CN(C(C(=O)NCC)=O)C2)C)cnc(CC2CC2)nc1 C1(NC(Cc2scc(C)n2)=O)CCCC12CN(C(=O)Cc1cncs1)C2 Cn1nc(CC2CC2)cc1C(=O)NCCC1CN(C(=O)COCCF)CCO1 c1(OC)ccc(F)c(CNC(=O)CC2CCC2)c1.C12(CCCCC1C)CC(=O)N2 N1(C(C(C)(C)C2CCCO2)=O)CCC2CC(NC(c3cccc[n+]3[O-])=O)CCC2C1 CC1(C)OCCOC1C(=O)NC1CC(F)CN(C(c2cnccc2C(F)F)=O)C1 c1(OC)cc(CC(=O)N(CCC(C)NC(=O)C(C)NC(=O)C(C)(C)C)C)ccn1 c1(C(=O)NC2CCN(C(C(CC3CCC3)NC(C)=O)=O)C2)cnc(=N)[nH]c1 C1(CNC(C2CCC2)=O)CN(C(=O)CC2CC3(CC3)C2)CC(C(F)(F)F)O1 c1(OC)ccc(C(O)C(C)NCC(C2CC2)SC)cc1 C(=O)(C(C(C)C)N)N(CCC)C=O.c1(C2CCCO2)ccncc1 C(C(C)(C)C#CC(=O)NC1(C(=O)OC)CCCOC1)NC(C(CCCC)F)=O N1(C(c2c(C)nc(CC(C)C)s2)=O)CC(NC(=O)CCS(C)=O)C(C)(C)C1 c1(CC)nc(C(N2CCC(CCC(N3CCC(COC(C)=O)C3)=O)C2)=O)c(C)o1 N1(C(C2(CC=C)CCC2)=O)CCN(C(C2OCCCC2(C)C)=O)CC(C)C1 c1(CNC(=O)NC2CC(=O)NCC2)csc2ccc(Br)cc12 CC(C)CC(CN=c1nc(C(C)(C)C)[nH]s1)NC(c1ccc2nc(O)[nH]c2n1)=O c1(C(N(CCCNC(C2CCC(CC)O2)=O)CC)=O)cc2c(C)n[nH]c2cn1 C(CC(N)=O)(C(=O)NC1CN(C)CC1C)NC(CCC=CC)=O C1(NC(CCn2c(C)ncc2)=O)CN(C(C2(F)CCOC2)=O)C2(CCCCC2)C1 Cc1onc(C2CC2)c1C(N1CCN(CC2CN(C(=O)C(=O)N(C)C)C2)CC1)=O C(=O)(C1CCCn2ccnc21)NC(C)CNC(c1n[nH]cc1I)=O C1(NC(=O)CCOCCCOC)CN(C(=O)C(F)=C(C)C)CC1C.O(NC=O)CC CC(C)CC(CC(=O)Nc1cccc(CCO)c1)NC(=O)C(=O)CC(C)C Cc1cc(Cl)ccc1C(=O)NCC1(O)CN(C(=O)CC2CCCC2(F)F)C1 CCC(C)(C)C(C)CC(=O)N1CCC(CCCNC(=O)CP(C)(C)=O)CC1 Cc1cc(C=CC(N2CCC(C(F)C(=O)N(C)C(C)C)C2)=O)on1 C1(C2CCN(C)CC2)(C(N(CC(CN(C(=O)Cc2ccon2)C)O)C)=O)CC1 N#Cc1ccc2oc(C(N3CCC4(CC3)CN(C(=O)C(N)=O)CCO4)=O)cc2c1 C(=O)(CS(=O)CCC(F)(F)F)NCC(CNC(c1nccc(C(N)=O)c1)=O)O c1(C(=O)NCCN(C(=O)Cc2ncccc2C)CC)ccc2c(c1)C(C)CO2 C1(C(N2CC(OC)C2)=O)CC2CC1CN(C(C1CC(F)(CF)C1)=O)C2 C=C(C)c1cc(C#N)ccc1NC(=O)C(=O)NCc1cc(C)cc(F)c1 Cc1cc(F)cc(C(=O)N(CC(O)CNC(c2cnc3[nH]ncc3c2)=O)C)c1N C1(F)(CNC(CCSC(C)(C)C)=O)CCN(C2(NC(=O)C=CC3CCC3)CC2)C1 N1(C(C2(OC)CC2)=O)CCN(C(c2cncc(C(F)F)c2)=O)C(C(C)C)C1 N1(C(CN(CCOC)C)=O)CC2CC(CNC(C3C(Cl)(Cl)C34CC4)=O)C2C1 Cc1cccc2c1CCN2C(=O)C(N1CCCCC(N(C)C)C1)=O N1(C(c2c(CC)cco2)=O)CCCCC(CNC(=O)CC2OCCO2)C1 C(CCN=[N+]=[N-])OCC(=O)NCCCNC(C(c1cccnc1)OC)=O c1(C(=O)NCCNC(c2c(Br)ccc(NS(C)(=O)=O)c2)=O)cc(Br)c(F)cc1F C=CCC(C(=O)N1CCC(C)(CCNC(c2cc(Br)n(C)n2)=O)C1)NC(C)=O Cc1cnnc(O)c1C(N1CC(NC(=O)Cc2c[nH]nc2C)CC(F)C1)=O N1(C(C2N(C)CC(F)C2)=O)CCCC(O)(CNC(=O)Cc2ccon2)CC1 C1(NC(c2ccc(CO)cc2)=O)CCN(C(C2CC2C(F)F)=O)CC1C(N)=O C(CN=c1[nH]ccc(=NCC2(C)CCCC2O)[nH]1)N(N1CCCC1)C.CCO C(CC(O)C(=O)NCC1(c2ccon2)CC1)NC(C1CCCOC1)=O C(=O)(C(O)Cn1cncn1)NC(C)CC1CN(C(=O)Cc2cnsc2)C1 CCCCCC(CC)C(=O)N(C(C)CCNC(c1nn(C)cc1N)=O)C C1(C(=O)NC(CC(C)C)CNC(c2c[nH]nc2Cl)=O)CCCCC12CC2 C1(CC(=O)O)CCCCN1C(N1CCC(c2cn(C3(O)CCSCC3)nn2)C1)=O C1(NC(c2ccc(F)cc2)CC(=O)OC)CC2CCCC2N1S(=O)(=O)C(C)C N12CCCC(C1C)Oc1cnc(cn1)C2=O.C1(C(=O)OCC)CC(C)N(CC)C1 Fc1c(N2CCN(Cc3ccc(F)c(Cl)c3)CC2)ccnc1F c1(N2CCC3(C(CNC(C(C)CO)=O)C3)CC2)cc2[nH]cnc2cc1[N+](=O)[O-] N1(C(CCCNC(=O)OC)=O)CCC(C(=O)NC(c2nc[nH]n2)C)C12CC2 N1(C(CCN(C(=O)CCc2cncs2)C(C)C)=O)CCCCC1CF C1(NC(c2n(C)nc(C(F)F)c2)=O)CCN(C(C2CN3CCC2CC3)=O)CC1O N1(C(C2N(C(C(C)SCC)=O)CCOC2)=O)CCCCCCCC1 C1(NC(C=CC(CC)C)=O)CCC2(CC1)CN(C(=O)Cc1csnn1)CCO2 Cc1cc2c(cc1C)N(C(C1(C#N)CCCO1)=O)CC2 C1(NC(C2CCC23CCC3)=O)CCCCN(C(c2ccc(NC=O)cc2)=O)C1 C(CCCOC)(C(=O)NC(C)(C)C(F)F)NC(CSCCOC)=O N1(C(C(c2cccc(Cl)c2)N(C)C)=O)CC(NC(c2ccc(Cl)cc2)=O)C(O)C1 C1(c2cn(CCC)nn2)CCCN(C(=O)Cc2sccc2C)C1 c1(CC(=O)NCC#CCNC(C2(C)CC2F)=O)n[nH]cc1Br C1(C)(N(C(=O)CCOCCNC(=O)CCCC2CCCC2)C)C(C)(C)C1(C)C C(C)(C1OCCc2sccc21)OC(=O)Nc1ccccc1.CC1C(=O)N1 c1(CCC(=O)N(CC)CC2CCCN(C(=O)C(F)C(C)C)C2)ccccc1C#N C(CC(=O)NNC(=O)CCc1ccccn1)NC(=O)OC c1(C(N(CC(C)NC(=O)CC2CC2(C)C)C)=O)ccncc1F Cc1cccc(Cl)c1CC(=O)NC(C)CCCNC(=O)CC1CCCN1C C1(C(N2CCC(O)(CCNC(C3(F)CC3)=O)C2)=O)CCc2nn[nH]c2C1 Cc1nc(F)ccc1N(C1CCNCCC1C)C(=O)C(F)F C(=O)(C(C)S(C)(=O)=O)N1CCC(N(CC#C)C(C2CC(OC(F)F)C2)=O)CC1 N1(C(CN(C(C(CC)C(C)C)=O)C)=O)CCOC2COCC12 c1(C(N2C3CC(NC(CNC=O)=O)C2CC3)=O)ccc2c(c1)OCCO2 c1(C(N(CCCN(C)C(C2CCCC2(C)C)=O)C)=O)ccc2cncn2c1 CC1CN(C)CC1C1(CC(N2C(CC(=O)Nc3ccnnc3O)CC2)=O)CC1 c1(NCC2OCCN(C(C(CCC)(C)C)=O)C2)cc(C#N)ccc1[N+](=O)[O-] C1(N(C(CCOC2CN(C(CC=CCC)=O)C2)=O)C)CC(F)(F)C1 c1(OC)nc(C)ncc1C(=O)NC1(CO)CCCN(C(C2(S(N)(=O)=O)CC2)=O)C1 S(=O)(=O)(c1ccc(N(C)Cc2cc(OC)ccc2Br)cc1Br)NCC(=O)NCCC N1(C(c2ccc(Cl)cc2F)c2c(-c3nnn(C)n3)n[nH]c2)CCc2ccccc2C1 CCC(C)C(O)CNC(=O)CN(c1ccccc1OC)C(C)=O Cc1nc(SCC(=O)NCC(C)CNC(C2(O)CCC2)=O)n[nH]1 C(c1ccccc1)=CC(=O)NCC1CCN(C(=O)COCC(F)F)C1 C1(NC(C=NOC)=O)CC2CC(C1)N(C(=O)Cc1noc(C)c1C#N)C2 C1(CNCC(=O)N(C2CC(SC)C2)CCC)CCCCO1 c1(C(N2CCCC2c2ccno2)=O)cc(-c2cn(C3CC3)nn2)n[nH]1 CCCC(CCC)CCCC(=O)N1CCC1CNC(=O)CN1CC(C)(C)C1 c1(C(N2CC(O)(C(C)NC(CCCCOC)=O)C2)=O)nc(C)ccc1F N1(Cc2nnc(CCCC)s2)CCS(=O)(=O)C(CCNC(C2(C)CC2CC)=O)C1 N1(C(C2CC(C(C)C)C2)=O)CCN(C(=O)C=Cc2ncco2)C(CO)C1 C1(CCNC(CCSCC)=O)CCN(C(=O)Cn2ccccc2=O)CC1 C1(C(C)(C)C)CCC(N=c2[nH]c(=NCC3CCOC3)[nH]c3ccccc23)CC1 c1(CNC(C2CCN2C(c2cnc(O)o2)=O)=O)ncc[nH]c1=O C(CCC(C)(C)NC(C1(CC(C)C)CC(=O)C1)=O)NC(C(C)OC)=O CCCC(C)(CC)C(=O)N1CC(CNC(=O)CCCC2CC2)(OC)C1 C1(C(N2C(C)CSCC2)=O)CCOCCN1C(C1CN2CCC1CC2)=O C1(NC(c2ncsc2C2CC2)=O)CCCN(C(c2cc(-c3ccco3)no2)=O)C1 c1(NCc2c(C#N)ccs2)[nH]c(=NC2COc3ncc(Br)cc32)nc2sccc12 C1(NC(=O)CCCF)CS(=O)(=O)C12CCN(C(=O)C=Cc1ccsc1)CC2 C(C)(C)(CCCC(=O)N1CCC(N(C)C2CC2)C1)NC(c1ccc(CC)cc1)=O C1(NC(C(=O)N(C2CC(NCC)C2)C)=O)CN(c2nccs2)CC1C CC(C)(C)C(O)Cc1cn(C2(c3ccccc3)CCN(C(=O)C3=NOCC3)C2)nn1 N1(C(Cc2c(C)cccc2)=O)CCC(CCNC(=O)CO)C(F)(F)CC1 N1(C(CCC(=O)NCC)=O)CCC(NC(c2cc(C(C)C)sn2)=O)C(CC)C1 c1(-c2cn(CC(=O)N(CCCC3CC3C)CCOC)nn2)ccc(C(C)C)cc1 c1(N(CC(=O)NC2CC(Sc3ccncn3)C2)C)nccc(-c2ccnn2C)n1 N1(C(=O)Cc2ccc3[nH]ccc3c2)CCC(C(F)(F)F)n2nccc21 CC1CC(NC(c2cccnc2C(F)(F)F)=O)CN1C(=O)CCCc1cncs1 C1(C(=O)Nc2cccc(NC(c3c(C)cn(C)c3)=O)c2)C2CC3CC(C2)CC1C3 CC(CCC(=O)NC(C)(C)C(=O)NC1CC1)NC(C1COCCN1C)=O c1(CCCNC(c2ccc(C(C)(C)C(F)(F)F)cc2)=O)ccc2c(c1)CCO2 c1(CC(=O)NCC2(F)CCC(CNC(CCOC)=O)C2)cc(F)ccc1O Cc1cncc(Cl)c1C(=O)N(C)CCNC(=O)C(c1cccc(Cl)c1F)(F)F C#CCCCC(C)C(=O)N1CC2(CCCC2)C1C(=O)NCCn1nncc1C C1(C(=O)NC(C)Cn2cc(CNC(C3(CN(C)C)CC3)=O)nn2)CCCOCC1 C(=O)(CCC[N+](=O)[O-])N1C(CNC(CCCc2ccc(C)s2)=O)C(C)CC1 C1(CNC(CSc2cccc(C)c2)=O)C2CCC(C2)N1C(=O)COCC1CCC1 C=CCCC(C(=O)OC)NC(=O)CC(CC1CC1)NC(=O)C1=NOCC1 C(=O)(CCCC(C)(F)F)NC1C2N(C(c3cccc(OCC)c3O)=O)C(CC2)C1 N1(CCNC(=O)OC)CCC(C)C(NC(c2ccccc2OC)=O)C1 CC(C)C(F)(F)CC(=O)NCC1(C)CN(C2CCN(CCOCCO)CC2)C1=O Cc1ccc(F)cc1C1CC1C(N1CC(NC(=O)C2=CCN(C)C2)CC(O)C1)=O N1(C(C2CN(C(N(C)C)=O)C2)=O)CCCCC(NC(=O)CC2CCN(C)C2=O)C1 c1(CC(=O)NCC(C)N(C(C=CCC)=O)CC)csc(-c2ccoc2)n1 c1(OC)cc2ccc(CNC(C3CNCC34CCOC4)=O)cc2cn1 CCCCC(C)C(=O)N1CCN(C)C(C(=O)N(C)CC2(O)CCCC2)C1 CC(C)(C)C(=O)NCC(C1CCCC1)NC(c1cc(C(F)(F)F)n[nH]1)=O c1(CC(=O)N(CC(CN(C(CCCCOC)=O)C)O)C)cccc(F)c1F C(CCC(C(=O)NCC1(C)CCC(C)CC1)NC(c1cc(Cl)ccn1)=O)OC CC1CN(C(c2ccc3c(c2)CCC3)C)CCc2ccc(F)cc21 CC(O)C(C(=O)NCc1nocc1C(=O)NC1CCN(C)C1C)N(C)C C1(C(=O)NCC2CC(NC(C3=C(C)CCCC3)=O)C2)CCc2nnc(O)n2C1 CC(C)CC(C(=O)N1CC(C(N2CC(N(C)C)C(F)C2)=O)CC(C)(C)C1)C(C)C C1(N(C=O)CCOC)CC2CCC(C1)N2C(=O)Nc1cnc(-c2cccs2)o1 C1(C(=O)NCC(CC)C)CC(O)CN1C(C1SCC=C1C)=O N1(C(=O)Cc2ccc(O)cn2)CCCC2(C1)CN(C(c1cnc(Cl)s1)=O)CCO2 c1(C(=O)NCCN(C(C2(CC#C)CCC2)=O)CC2CC2)cc(N(C)C)ccc1N n1(CC(=O)NCCCCC(C)NC(=O)CC23CCCC2C3)nc(O)ccc1=O c1(-c2onc(CC(=O)NC3C(=C)C3)n2)cc2c(cc1OC)OCO2 N1(C(C(c2ccccc2F)C)=O)CC23CCCC2(CNC3)C1 C1(C(=O)NC(CCC)CNC(C2CC(O)(C(F)(F)F)C2)=O)CN2CCN1CC2 C1(C(N2CC(O)(C(C)NC(CCCn3c(C)ncc3)=O)C2)=O)CC12CCSCC2 c1(-c2cc(NC(C=CC(=O)NC3CC3)=O)on2)ccccc1Cl.C12CC1CNC2=O c1(C(=O)NCC(C)NC(c2c[nH]nc2-c2ccccn2)=O)ccnn1C(F)F Cc1ccsc1C(N1CCCC1CC(=O)N(C1CC1)Cc1nncn1C)=O C1(NC(N2CCN(Cc3ccc(C)c(F)c3)CC2)=O)CC(N)CCS1(=O)=O N1(C(CSC)=O)CCC(C2(O)CN(C(=O)C(C)(O)C3CCC3)C2)CC1 C(CC(C(=O)NC(c1ccccc1F)C)NC(c1cccc(CC)c1)=O)=CC CC(C)CC(=O)NCC(c1ccccc1)CNC(=O)CCc1nc[nH]n1 c1(N2CCC(n3nccc3)C2)nc(=NCc2cn[nH]c2)[nH]c2c1CCC2 c1(C(=O)NC(CC)(CNC(C2CC2(F)F)=O)CC)nn(C)c(N)c1C C1(NC(CSC)=O)CCC(N(C(C2CCNC(=O)C2)=O)Cc2ccccc2)CC1 c1(CC)nn(C)c(CNC2CCN(CCC(=O)O)C2)c1Br c1(C(=O)NC2CC(NC(c3ccc(F)s3)=O)C2)ccc(C(N(C)C)=O)s1 c1(C(=O)NCC(CC)NC(c2c(N)cc(F)cc2F)=O)cnc2scc(C)n12 c1(C(=O)NC(c2cn(CC3CCOC3)nn2)C)sccc1F c1(OC)cc(C(=O)NC2CCN(C(=O)C=CS(C)=O)C(C)C2)cc([N+](=O)[O-])c1C c1(COC)nocc1C=O.c1(NC)ccn(CCF)n1.N12CCC1C2=O N1(C(C(C)NC(=O)NC)=O)CCC2CCC(C1)N2CC(=O)NC(C)C C1(C(=O)NCC(CC)NC(c2cc(C)cc(O)n2)=O)CC2OC(C)(C)OC2C1 CC(C)(C)C(CNC(=O)NC1CCCC1CO)OC(F)F CC(C)(C)C(CNC(C1CC(=O)CCO1)=O)C(=O)N1CCC(C(N)=O)C1 C=C(CC)CN=C(NCC(=O)Nc1ccc(F)cc1)NC1CSC(C(F)(F)F)C1 C1(NC(=O)N(C2CCCC2)CCN(CC)CC)CCCC1C C(CC1=CCCCCC1)NC(C(c1nc(C)[nH]n1)N)=O C(c1cccc(Cl)c1)=C(C)C1CC1.C(C(F)(F)F)=CC(=O)N(CCN)C(C)C N1(C(=O)NCC2CCC3(CCC3)O2)CCCCC1C1CCCO1 C1(C(N(C(C#C)(C)C)C2CC2)=O)CN(C(=O)CC2CC(=O)NC2=O)CC1C1CC1 C1(c2nnnn2Cc2ccccc2)(NCCC(CC)(C)C)CC2CC1CC2(F)F C=Cc1cnn(C)c1C(=O)NCCOCCCNC(c1cnccn1)=O S(=O)(=O)(c1ccccc1Cl)NCC(=O)NC1CC2CN(C(CC=C)=O)CC21 c1(C(N2CCCCC2c2cn(C34CC(C3)C4)nn2)=O)cn2ccc(F)cc2n1 c1(N(C(=O)C(=O)NC2CON(C)C2=O)CC)ccc(F)c(F)c1 C(=O)(C(C)CC(F)(F)F)NCC(C)CNC(C1CCN(C2CC2)C1=O)=O Cc1ccn(CC(=O)NCC2(CNC(c3cc(C(F)(F)F)n[nH]3)=O)CC2)c(=O)c1 c1(C(C)C)ccoc1C(=O)N(CC(O)CN(C(=O)C(C1CCCCC1)O)C)C Cc1cccc(C)c1CC1CC1.c12ccc(cc1)C(N1CC(C)(C#N)C1)C(=O)NC2 C1(C(N(C(C2(C)CC2)C)C)=O)N(C(=O)CCP(C)(C)=O)CCC1(C)C C1(C(=O)OCCc2c(C)ncs2)CC(=O)N(C)C1c1ccc(Cl)cc1 C(=O)(CCC(C)(C)[N+](=O)[O-])NCC(C(C)C)NC(c1ccc2nc(S)oc2c1)=O c1(C(N(CCC)CCNC(=O)CC2CCCC2OC)=O)c(C)cc(C)oc1=O C1(C(N(CCNC(c2c(C)ccnc2C)=O)C2CC2)=O)CCc2c(nnn2C)C1 c1(C(N2CC3(CC)CC2(CNC(C2(O)CC2)=O)C3)=O)c2c(nn1C)CCCC2 C1(O)(CNC(CCc2cc(C)[nH]n2)=O)CCN(C(c2cnn(C3CC3)c2C)=O)C1 N1(C(c2onc(C)c2C)=O)Cc2ccccc2C(CNC(C2CC2(C)Br)=O)C1 CCCCC(CC)CC(=O)N1CC(NC(c2cncc3c2CCC3)=O)C1 Cc1ccc(F)c(-c2cc(C(=O)N(CC(C)(C)C)Cc3ccccc3)[nH]n2)c1 c1(CC(=O)NCCC2CC(OC)CN2C(=O)C(Cl)=CCl)cccc([N+](=O)[O-])c1C C1(CNC(C2C(C)CC(=O)N2)=O)CN(C(C23CCCC(CO2)C3)=O)CCC12CCC2 N1(C(Cn2c(C)nc(C)n2)=O)CCCC(F)(CNC(=O)COC2CCCCC2)C1 c1(C(=O)NC(C2CCN(C(=O)Cc3ccc(C#N)nc3)C2)C)nc2ncccn2n1 c1(C(N2CCOCC(CNC(CCCC(C)=O)=O)C2)=O)[nH]nc2c1COC2(C)C c1(CC(N2CCC(OCCNC(C(C)(C)CC3CC3)=O)C2)=O)ccc(O)c(Cl)c1 C=CCCN=C(NCCC(CSC)OC)NC1CCN(C(=O)OC(C)(C)C)C1 N(C1CCc2sc(Br)cc21)C(=O)OC(c1cccc(Cl)c1Br)=O C(=O)(C(C(C)(C)C)n1ccnn1)NCC1N(C(CCNC(C)=O)=O)CC(O)C1 C1(C(=O)NCC2OCC3(CN(C(CC=CC)=O)C3)C2)CCc2nncn2CC1 C1(C(N(C(C)CNC(=O)CC2(C)CC2)CC)=O)C2CCCCCCC12 C1(C(=O)NCCC2=CCN(C(C(CC)CC)=O)CC2)COc2ccccc2C1 CC(C)(CC(F)F)C(=O)N1CCC(C(C)(C)NC(c2cc(F)n[nH]2)=O)C1 c1(CC)ccc(C(=O)N(C2CCN(C(=O)CC34CCN3CCC4)C2)C)cc1 N1(CC(=O)NCC2N(C(C3C(C(=O)OC(C)(C)C)CC3)=O)CC2)CCCOC1=O CCCCCCC(C)CC(=O)NCC1C2CN(C(c3coc(SC)c3)=O)CC12 CC(O)C(F)(F)C(=O)NC1(c2ccccc2)CCN(C(C2CCOC2=O)=O)CC1 CC(C)CC(C)(CNC(=O)C(C)(O)C1CC1)NC(=O)COC1(C)CCCC1 n1(CC#C)cnnc1C(=O)NC1CCC(CCNC(=O)CC2CNC(=O)O2)C1 c1(C(C)(C)C)ccccc1C(=O)NCC1CN(C(C2CC23CC(O)C3)=O)CCO1 C1(NC(CC2(N(C)C)CN(C(CCCOC(C)C)=O)C2)=O)CCCCC1F c1(C(=O)NC2(CC)CC2)ccc(C)o1.C12CC(C1)C(=O)NC2 N1(C(C(C)Oc2ccccn2)=O)C2CCCC1CC(Nc1nnco1)C2 c1(OC(c2c(NCC(C)C)cccc2)=O)ccc([N+](=O)[O-])cn1 N1(Cc2c(C)nn(C)c2)CCC2(CCN(C(c3cnc(Br)s3)=O)C2)C1 C#Cc1ccccc1CC(N1CCN(C(C2CC3(C2)CC3F)=O)CC1COC)=O CCCCCC(C(=O)N1CC2CCCC1CN(CC1CCNCC1)C2)C(C)C CCC(C)(C)C(=O)C(=O)N1CCN(C(=O)C(C(=O)OC(C)(C)C)C(C)C)CC1C c1(NC(C)=O)ccc(C)c(NC(c2ncc(Br)nc2I)=O)c1 n1(CCNC(C=CCN(C(c2cc(CCC)[nH]n2)=O)C)=O)ccccc1=O c1(C(=O)NC(C2CCN(c3ccnc(OC)n3)C2)C)ccc2nc(CO)[nH]c2c1 C(CNC(=O)CC1(O)CCC1)(C(=O)N(CCC(N)=O)Cc1ccccc1)N(C)C c1(C(=O)NCC2CN(S(=O)(=O)CCCl)C2)cnn(C2COC2)c1 C1(C(=O)NC(C(C)NC(C(CC)CO)=O)C)CC2(CCC2)N1C(=O)OC C1(NC(C2C(C)N(C)CC2)=O)CCN(C(=O)C2=COCC2)C12CC2 N1(C(C(C(=O)OCC)OC)=O)CCC(C(=O)NC(C)CS(N)(=O)=O)C12CCC2 CCC(F)(F)CCOC(C1CCCC=C1Br)=O Cc1nn(CC(N2CC(F)(CNC(c3cnnn3C)=O)C2)=O)cc1Cl c1(C(=O)NC2(CC=C)CN(C(=O)C(c3cnn(C)c3)=O)C2)cccn(O)c1=O C(=O)(C(=O)CCC(C)C)N(CCC(N1CCC(N(C)C)C(C)C1)=O)CC=C Cc1nc(C)c(C(=O)NC(C)CNC(=O)C(C)(C)C2CCCCC2)o1 c1(CCC(=O)Nc2ccccc2N2CCCC2)ccc(F)c(F)c1 c1(C(N(CCC(=O)NC(c2nc[nH]n2)C2CC2)CC#C)=O)cc(O)ncn1 N1(C(CC=CCC)=O)CCN(C(c2cncc(OC(F)F)c2)=O)C(CF)C1 C(=O)(C1Cc2ccccc21)NC1C(C(=O)Nn2cccn2)C1C1CC1 c1(C(=O)NCC(C)CNC(c2cc(N)cnc2Cl)=O)cnc2n(c1=O)CCS2 c1(C(=O)NC2C=CC(CNC(C3CC4(C3)CC4F)=O)C2)ncnc2ccsc12 N1(C(C2(CC=C)CN(C(=O)CC3CCCNC3=O)C2)=O)CCC2CN(C)CC2C1 O=C(CCCC(F)(F)F)N1CC2CC(C1)N(C(=O)C=Cc1ccco1)C2 C1(C(=O)NCC(CC=C)NC(=O)CCCN2CCCC2)CC(S(C)(=O)=O)C1 N1(C(c2nc(CC)oc2)=O)CC2CC3CC2C1C3NC(=O)Cc1cccc(C)c1 N1(C(C(CC)CC2CC2)=O)CCCC2(CC2)C1.C1(C(=O)OCC)(C(=O)N(CC)CC)CC1 c1(C(=O)NCC2(c3ccccc3)C(C)(C)C2)cccnc1N=[N+]=[N-] N1(C(COC(C)=O)=O)CCN(C(C2CNC(=O)C2)=O)C(C(C)C)C1 c1(C(=O)NCC2CN(C(C3CC(C4CCC4)C3)=O)CCO2)ccc2c(c1)OCO2 C1(O)(COC)CCN(Cc2cnoc2Cc2cnn(CC(C)C)c2)C1 C1(C(N(CC)CC2CCC2)=O)C2CC(O)C(C2)N1C(c1cccc(O)c1C)=O Cc1nc2ccccn2c1SCC1CC(F)CN1C(=O)C(=O)Nc1ccccc1 N1(C(COCCOC)=O)CCC2(CC1)CC(C)N(C(c1cc([N+](=O)[O-])n[nH]1)=O)C2 C(c1cccnc1)=CC(=O)NCCCCC(=O)NC(C)Cc1ccoc1 C1(C#N)(C(N2C(C(N(CCOCC#C)C)=O)CCC2C(C)C)=O)CCCCC1 C1(NC(c2cnc(Br)o2)=O)CN(c2ncncc2I)CC(F)(F)C1 N1(CC(CN(C)C)O)CCC2C(CNC(=O)C(=O)N(C)C)C2=CC=CC=C1 C1(CCCNC(c2c(SC)ccs2)=O)CN(C(=O)Nc2cncc(C)n2)CCO1 Cn1c(C(N2CC(C)(NC(C3CCCCS3)=O)C2)=O)ccc1C#N N1(C2CC(C(=O)OCC)C2)CC(C(=O)NCc2ccsc2C)CCC1C c1(C(N2C(C)CC(NC(=O)CSC3CC3)CC2)=O)cc(C#N)ccc1O C#Cc1cccc(C(N2CC3CC2C3C(=O)Nc2cnn(CCO)c2C)=O)c1 C1(C(=O)NC2CC(=C)C2)CN(C(=O)CC(C)N(C)C)CCC1O c1(NC(=O)C(CCOCCO)NC(C2(CCOC)CCC2)=O)cnn(C)c(=O)c1 c1(CC(N2C(CC)C(NC(=O)CN3CCC(F)CC3)CC2)=O)cc(F)cc(F)c1 N1(C(C(C)OCCOCC)=O)CC2CC(C1)CN(C(c1cc[nH]n1)=O)C2 CC(O)C(C(=O)NC1CCN1C(C)(C)C)Nc1cnn(C)n1.c12cn(nn1)C2 C(=O)(C(C)CCCC(C)C)NCC1N(C(c2c(CC)ccnc2)=O)CC(C)(C)C1 C=CCC(C(=O)NC(C)CCCO)NC(c1cnn(CCC)c1)=O c1(C(N2CCOCC2C2CCC2)C(=O)NCCOC)cc(OC)c(Br)c(OC)c1 C#Cc1cc(C(=O)NCC(C(C)(C)C)NC(=O)C(CC)CCOC)cc(F)c1 C1(C(=O)NCCCNC(=O)CC2CC2)CC(C(=O)OC(C)(C)C)CCO1.CCS Cc1sc(Cl)nc1C(=O)NC(c1ccc(CNC(=O)C=Cc2ccsc2)cc1)C c1(C(=O)OC)cc(OC)cc(C(=O)NC2CN(C(=O)C=CC(C)(C)SC)CC2C)n1 C1(NC(CC(=C=C)C)=O)CCC2(CCCN(C(c3cn(CCC)nn3)=O)C2)C1 CC(C)CCC=CC(=O)NC1CN(C(C2CC2[N+](=O)[O-])=O)C1 c1(N2CC=CC(NC(CS(CCC)(=O)=O)=O)C2)cc2c(cn1)C(=O)CCC2 N1(CCNC(C2C(C=C(C)C)C2(C)C)=O)CCCN(C(=O)CCSC(F)(F)F)CC1 C(=O)(C(F)C(C)C)N1C(C(=O)NCC2(C=C)CCC2)C=CC1 C1(CNC(c2n(CC=C)ccc2)=O)CC(C)(C)CCC1NC(C1(C)CCC1)=O C(=O)(CC(C(F)F)n1cccn1)NC1C(N(C(C2CCC(=C)CC2)=O)CC)CC1 CC1CN(C(=O)C=CCF)CC(C)N1C(C1CN(CC(F)F)C1)=O CC(C(=O)OC(C)(C)C)C(=O)NCC1CC(NC(c2cc(C(N)=O)n(C)n2)=O)C1 C(=O)(C1COc2ccccc21)NC(C)CC(C)NC(c1occ2c1CCOC2)=O C1(CC#C)CN(C(c2cnn(C(C)C)c2)=O)C12CCC2 c1(CC(N2C(CNC(c3cc(C4CCC4)on3)=O)CC2)=O)ccc(Cl)cc1 c1(C(C(=O)NCC(CNC(c2c(C)cco2)=O)O)C)ccc(Br)cc1F CCCC(CNC(=O)C(C)n1ccnn1)C(=O)NCCC(C)(C)C C(=O)(C1CCc2cccnc21)NCCNC(CC(C)(O)c1ccccc1)=O C1(CCC2N(C(CC=CC)=O)CCC2)CCCCN1C(=O)Cn1ccnn1 C1(F)(CNC(c2c(C)nn(C)c2)=O)CCN(C(c2ccnn2C(C)(C)C)=O)CC1 c1(N(CCOCCCC)C)ncnc(NCc2cc(-c3ccoc3)on2)c1C c1(C(=O)NCCN(C2CCCC2)C(CN2C(C)CC2)=O)c(F)c(F)cc(F)c1F C#Cc1cnc(C(=O)N(CCCCCNC(C23CCOC(C)(C2)C3)=O)C)c(C)c1 CCCS(=O)(=O)CC(=O)NC1CC(NC(c2cnc(O)c(Br)c2)=O)C1 c1(C(N2OCC(n3cc(C(C(OC)OC)C)nn3)C2)=O)[nH]c2ccccc2c1Cl C1(NC(C(CN(C)C)O)=O)CN(C(=O)C=Cc2ccc(F)cc2)CC12CC2 C(CCC(=O)NC1CCCC1CN(C)C(c1occc1C(C)C)=O)OCCC CCC(F)(F)C(C)(C)C(=O)N1CCC(C2(NC(c3nc(C4CC4)n[nH]3)=O)CC2)C1 C1(CNC(C2(C(=O)OC)CC2)=O)CN(C(=O)Cc2ncc[nH]2)CC1(C)C c1(OCc2cc(N(CCC)C(c3ccccn3)C)ncc2)ccc(Cl)cc1C c1(CC(=O)NCC2(NC(c3on(C)c(=O)c3)=O)CCCC2)nc2ccccc2s1 C1(CNC(COC)=O)C(C)CCCN1C(c1sccc1C)=O Cc1cc(=O)c(C(N2CCOCCC2C(=O)NCCCc2ncnn2C)=O)c[nH]1 C=C1Cn2c(C(=O)NCC3(CNC(=O)Cn4cccc(C)c4=O)CC3)nnc2S1 C(=O)(N1OC2C=CC1CC2)c1noc(C(N2CCCC2)C)n1 CC(CCC(=O)NC(C)Cc1ccco1)NC(C1CC1(C)C(F)F)=O C=CCC(CC(=O)N(CC(F)(F)Cl)C)NC(=O)C(C)(C)C1CCOC1 C(=O)(C(=O)CC(C)CC)N1CCC(C(C(=O)NC(C#C)(C)C)F)C1 N(C1CN(C(=O)Cc2ccccc2)Cc2ccccc21)C(CC(C=C)C)=O N1(CCCC)C(=O)CCC(NC(=O)CC2CCN(C)C2)C1c1ccnn1C C1(NC(NC(C=C)C)=NCc2ncco2)Cc2cccc(OC)c2C1 C1(C(N2CCC(N(C(=O)CCN3CCC3)CC)C2)=O)Cc2cc(F)cc(F)c2O1 Cc1ccc(F)cc1C(N1CCC(C(C)NC(=O)CCCC(N)=O)C1)=O CN1CCC(CCNC(=O)CCN(C)C(C2CCCCC2)=O)C1=O CC1CN(CC(c2ccccc2)O)CCC1CN=c1nc(-c2ccccc2)[nH]s1 C=CC(C)(C)CC(=O)NCCC1(NC(C2COCC(C)O2)=O)CCCC1 N1(CC(C)C)CC(NC(=O)NCC2(c3nn[nH]n3)CCCCC2)CC1=O CCC(CC(=O)N(C(C)C(=O)N1CCC1C(C)O)C)C(C)(C)C c1(C(N(CCCC(=O)NC(CC)(C)C2CC2)C)=O)cc(Cl)n(C)n1 c1(C(=O)OC)cc(F)cc2c1CCN(C(C(=O)Nc1ccccc1C)c1cnn[nH]1)C2 C(CC(F)F)(C(=O)NCc1ccc([N+](=O)[O-])o1)N(C(C1C(CC)COC1)=O)C C1(NC(C(C)OCCN(C)C)=O)CCN(C(=O)CN2CCCC2=O)CC1C1CC1 C1(C(N(CC(CC)OC)C)=O)OCCC1NC(=O)C(Cc1cc[nH]n1)NC=O C(CC1=C(C)CCCC1(C)C)N(CCOCC)Cc1cccc(Br)c1 c1(C(N(CCNC(c2cc(COC)on2)=O)CCOC)=O)cncc(C(N)=O)c1 C(=O)(CCC(=O)NC(C)CC(=O)NCCN1CCC1)NC N1(C(C=C(COC)C)=O)CC(NC(=O)C(c2ccccn2)O)C(C(F)F)C1 Cc1cnc(C(N2CCC(N(C)C(c3cc(C(C)(C)C)on3)=O)C2)=O)c(Br)c1 n1(CC(N2CCC(C)C(NC(=O)C(C)(C)CN(C)C)C2)=O)nc2ccccn2c1=O C1(NC(c2c(CC)cccc2)=O)COC2(CNC(C3C4CNC(=O)C34)=O)CC1C2 C(=O)(C(CC)C(=O)N1CCC(C(=O)NCc2cccc(OC)c2)(CF)C1)OCC N1(C(c2ccc(F)cn2)=O)CC2CN(C(C3CCCC(F)C3)=O)CC(C1)O2 C1(C)(C(=O)NCc2scc(C(=O)OC)n2)CCCN1C(c1ccncc1C)=O c1(C(=O)NC(C(C)NC(C2CC23CCC3)=O)(C)C)cnc2c(c1)NC(=O)CN2C C1(O)(CNC(COCCCOC)=O)CCCN(C(=O)CCC2CC(C)(C)CO2)C1 c1(CN(CCCOC(CSC)Cc2ccccc2)C)ccc(NC(C)=O)s1 c1(CC)cn(C)nc1C1CC1.c1(NCC(=O)N(C)CC)ncnc(N)n1 N1(C(=O)Nc2cnn(CCOC)n2)CCC2(CC2c2nnc(O)o2)C1 CCC(C)C(=O)C(=O)N1CCOCC(NC(C2C=CCS2)=O)C1 Cc1nn(C)cc1-c1ccc(NC(C2CCC(NC(=O)C(C)S)CC2)=O)cc1 C=C(C)CC(C(=O)OC)NC(C1CCCCN1C(c1cnc(O)n1CC)=O)=O c1(CC)scnc1C(=O)NCCOC.C1(C(=O)NCCCO)CCC(CC)C1 N#Cc1cc(Br)c[nH]c1=NCC1CCC(CC(=O)NCC(F)F)C1 CCCCCC(C(=O)NCCCC(C)NC(c1ccnn(C)c1=O)=O)C(C)C c1(CNC(c2cccc(C(C)(F)F)n2)=O)cn2ccc(Br)cc2n1 N1(C(COCCOC)=O)CCC(C(=O)NCC2=CCCOC2)(C(C)C)C1 C(N=c1[nH]cnc(NCc2nnc3n2CCC3)c1C)c1cn(CCC)nc1C CC(CN(C)C(C1CCC1CNC(C1CCC=CCC1)=O)=O)C(F)(F)F c1(C(N2CC(O)(CNC(=O)Cc3ccccc3)C2)=O)ccc(I)cc1Br C1(C(=O)NCC2N(c3c(CC)cccn3)CCC2)CC2(C1)CC(F)(F)C2 C(CNC(c1cncc(F)c1)=O)(C(C)C(C)C)NC(C1(C(=O)OC)CC1)=O c1(C(N2CCC(CN(C(COC(CC)CC)=O)C)C2)=O)ccc2nc(O)oc2c1 CN1CC(C)(C)CC1C(=O)N(CCCCCCNC(=O)CC(O)CC1CC1)C Cc1nc(C(=O)NCC2COC(CNC(c3coc(C(F)(F)F)n3)=O)C2)nn1C C1(CC)(NC(=O)C=C2CCC(C)CC2)CCCN(C(=O)CCc2c[nH]c(=N)[nH]2)C1 c1(OC)cc(C(=O)NCCCCN(C)C(c2cccn2C2CCCC2)=O)sn1 N1(C(C23CC(NC(C4C(COC)CC4)=O)(C2)C3)=O)CCCNC(=O)CC1 n1(C(C)C)cnc(C(=O)NCC(C)NC(=O)C(C)(C)C2CC2C(F)(F)F)n1 c1(C(=O)NC(C2CCCCN2C(c2ccc(F)cc2)=O)C)cccn2nccc12 c1(NC)ncc2ccc(CNC(=O)Cc3ccnc(Cl)c3F)cc2n1 N1(C(CNC(C2C(C)C2)=O)=O)CC(C)(C(N2CC3(CCC3(C)C)C2)=O)CC1(C)C Cc1cccc(C)c1N1CCN(C(c2cn(-c3c(C)nsc3C)nn2)(C)C)CC1 N1(C(c2ccc(F)s2)=O)CC23CCCC2(C1)CN(c1ncnn2cccc12)C3 C1(C(NNC(COc2cccc(NC(C)=O)c2)=O)=O)Nc2ccccc2C1(C)C N1(C(c2c(C)ncs2)=O)CC2CCCC1C2CNC(=O)CC1(C)CC1 C12(NC(COCC(C)C)=O)CC1CN(C(C1(O)CC(CF)C1)=O)C2 C1(NC(CCCn2c(C)ncc2)=O)CCN(C(c2[nH]ccc(=O)c2C)=O)CC1F c1(CC(=O)Nc2ccc(NS(=O)(=O)CCBr)c(Cl)c2)cccc2ncccc12 c1(Sc2nnc(-c3ccccc3)s2)ccc(C(N2CCC(N(C)CC)C2)=O)cn1 N1(CC2(C)CC(C)C2)CCC2(CCCCCC2)C1.C1(C(=O)N)CCCCC12OCCO2 c1(C(=O)NCC2C=CC(NC(C(C(C)C)NC=O)=O)C2)noc2ncccc12 c1(CNC(C(C)C2CC2)=O)c[nH]nc1C(=O)N(C)CCN1CCOCC1 C1(C(=O)NCC=CCCOC)CC=CC(NC(C2CCOC2(C)C)=O)C1 C1(NC(C(C)OC)=O)CC2CC1N(C(C1CCN(OC)CC1)=O)C2 CC1CC(NC(=O)C(C)CC2CCC2)CCN1C(=O)Cn1cnc([N+](=O)[O-])n1 C1(NC(C2CC(SC)C2)=O)CCC2(CC1)CC2NC(c1cccc2nccn12)=O Cc1c(I)cc(CN2CC(C)CC2C(=O)Nc2cccc(C)c2C#N)cc1I CCCCC(CC)CC(=O)N1CCCC(NC(c2nn(CCC)cc2Cl)=O)C1C N1(C(C2OCCN(CC)C2)=O)CC(C)CN(C(c2nc(Cl)nnc2O)=O)C(C)C1 C1(C(N2C(C)(CCC)CC2)=O)CCCCN1C(=O)CC1CCCC(=O)N1 c1(OC)ccc2c(C(=O)N(C)CCNC(c3ccc(C)n3C)=O)n[nH]c2c1 N1(C(C2(CSC)CC2)=O)CCCC1CNC(C1CCCOC1)=O C1(C(=O)OCC)CCCC(NC(=O)NCCCN2CCCC2)O1 C1(C(=O)NCCC=CC=C)(OC)CCN(C(=O)Cc2csc(C)c2)C1 c1(C(=O)NC2CC(C)(C)N(C(C3CC(C4CC4)C3)=O)C2)c(Cl)ccc(Br)c1F c1(OC)cccc(C(C)C(=O)NCCCNC(=O)CC2CC3CC3C2)c1 Cc1oc2cc(C(=O)NC3CCN(C(=O)C=CC(C)C)C(C)C3)[nH]c2c1C CCC(CO)(CO)C(=O)NCc1c(C(F)(F)F)coc1C C1(CC(=O)N2C(CC)(C)CC3CC2C3)CC2(CC2)CO1.N(C)C(=O)C1CC1 c1(OC)cc(C(=O)OC(c2cc(OC(C)=O)cc(Br)c2)C)cnc1OC Cc1cc(C(=O)NC2CCC(NC(C3(C)COC3)=O)CC2)n2nccc2n1 c1(OC)cc(OC)cc(C(C)C2CC2)c1.C1CC(OC(C)C)CNC(=O)C(=O)N1 C1(C(=O)NCC2CC(NC(c3ccon3)=O)C2)CC2CCC(C1)C2=O C12(CNC(c3c(OC)scc3)=O)CC1CN(C(=O)COc1ccc(F)cc1)C2 C1(CCNC(C2(NC(C)=O)CC2)=O)COCCN1C(CC(C)C)=O C(=O)(C(C)CCCC(C)=O)N1CCN(Cc2ccc(N(CCCC)C)cc2)CC1 c1(C(=O)NC(C(=O)NCCC2CN(C)C(=O)C2)CCF)cc2cccn2cn1 Cn1nnc(=NC2CC3(CCC3)C2)[nH]1 C1(NC(C(C(C)C)NC(CCC(=C)C)=O)=O)CCC2(CC1)CC2 c1(CC(=O)NC2C(CNC(Cn3c(C(C)C)nnn3)=O)CCC2)ccc(Cl)cn1 C1(c2n(CCCOC)nnn2)(NC(c2sc(C)nc2C)C)CCCSC1 C1(NC(C(C)(C)C)=O)CN(C(c2cc(-c3ccccc3F)on2)=O)CC1O CCCCCCCCC(=O)NCCCCC(=O)N1CC(C)C1(C)C C1(CNC(CCSCCC)=O)CC(OC)CN1C(=O)C(C)Oc1ccccc1 CC1(C)C(CNC(C2Cc3nccn3C2)=O)CCN1C(N1OC(C)(C)CC1=O)=O c1(C(N2C(C3N(C(=O)CCN4CCC4)CCC3)CCCC2)=O)cc(F)nc(O)c1 c1(CC)cnc(C(=O)NCC2CCC(NC(=O)CCN3CCCCC3=O)CC2)nc1 C1(NC(c2cccc(CF)c2)=O)CN(C(C2CCSC2)=O)CC(F)(F)C1 c1(C(=O)NC(COC)C(=O)Nc2cnn(C3CCC3)c2C)ccn(C)c1C N1(C(c2nc(OC)oc2)=O)CC(CO)C2(C1)CN(C(c1cccn1C1CC1)=O)C2 C(CC(CC)C(=O)N1CC2CC(NC(=O)Cc3cc(C4CC4)no3)C1C2)=CC C1(N(C(C2(SC)CCC2)=O)C)CCC(NC(c2ccccc2N(C)C)=O)CC1 c1(CCC)cc(C(=O)NCC(C2CCCC2)NC(=O)CCn2cnnn2)nn1C c1(SCC(c2cc(F)c(Cl)cc2F)N2CCCC2)sc2cc(Cl)cc(Cl)c2c1Cl N1(C(CCOCC)=O)CCN(C(C2(CC(C)C)CC2)=O)CC12CC2 S(=O)(=O)(c1ccc(F)c(Cl)c1)N1CCC(C(F)(F)F)(N(C2CC(C)(C)C23CC3)C)C1 C1(CNC(C2C(=C)C2)=O)CCCC2(CN(C(c3cc(O)cc(Br)c3)=O)C2)O1 CCC(C(=O)NCC(O)CNC(=O)Cc1ccc(CC(C)C)cc1)C(C)(F)F c1(NC(C2(C)CCCN(C(c3cocn3)=O)C2)=O)ccc(Br)c2ccccc12 N1(C(C(C)NC(c2cscc2C(N)=O)=O)=O)CC2CCC1CN2C(c1ccoc1)=O c1(OCCNC(C2COCCN2C(c2cc(Br)c[nH]2)=O)=O)cncc(Cl)n1 C(C(C(C)C)NC(=O)C=NOC)(c1ccccc1)NC(c1ncc(CC)s1)=O c1(OCCN(CCO)CC)ccc(C)cc1.c1(CS(=O)(=O)N)cccs1 N1(C(C=CCCC(C)C)=O)CCSCC1C(=O)N(C)Cc1ncn(C)n1 N1(C(c2ccccc2Cl)C(=O)Nc2scc(OC)c2)CCCCC12CCC2 C1(CCNC(C=CSC)=O)CCN(C(=O)Cn2ccc(=N)[nH]2)CC1 C1(C#CC(=O)N2CCCCC2C(C)(C)CNC(=O)C(=O)NC(C)C)(CC)CC1 n1(C(C)C(=O)N(CCCNC(C2CC3CC3C2)=O)C)ccc2ccccc2c1=O N1(C(CC2CC(OCC)C2)=O)CCCC1(CNC(C1(OC)CCOC1)=O)CC C(CCCCCCO)NC(CCC1CC(NC(C2C(CCC)CCC2)=O)C1)=O c1(NC(C)(C)C)ccc(CC(N2CC(CNC(C3CCCO3)=O)C2)=O)cc1 C1(C2CCOCC2)(C(=O)NCC2C(C)CCN(C(c3c(C)nccn3)=O)C2)CC1 CC1OC2(C(N3CCC(CN(C)C(c4ncccn4)=O)C3)=O)CC1C2 c1(CNC2CCC(NCCS(C)(=N)=O)CC2)ccc2scnc2c1 CC1=C(C(=O)NC23CC(CNC(C4CCCCN(C)C4)=O)(C2)C3)SCCO1 N1(C(C(=O)NCC(C)C)C)CCC(CCSCN)C1.c1(C(=O)N)csc(Br)c1 c1(C(=O)NCC(CO)NC(CC(C)OC)=O)c(Br)ccc(F)c1N c1(C(N2C(C(=O)Nc3c(C(N)=O)cccc3Br)CC3CC32)=O)cc(I)cnc1Cl c1(C(=O)NC2CC(CNC(CC3CC(C)(C)C3)=O)OCC2)ccc2cnoc2c1 CC(C)P(=O)(CC(=O)NCC1(O)CCN(C(=O)Cc2c[nH]ccc2=O)C1)C(C)C Cc1cc(C(N2CCC(C(=O)N(CCF)C(C)C)CC2)=O)c(C)[nH]1 C(=O)(C(F)(F)C(O)c1ccccc1)NC1CN(C(C2CN(C(C)C)C2)=O)CC1C c1(C(C)(C)C)n[nH]cc1S(=O)(=O)NC1CCCC1C1CC1 c1(C(=O)NCC2CCC(C)CN2C(C2CCSCC2)=O)cnc2[nH]cncc1-2 c1(C(N(C)CC2CCCN2C(=O)Cc2cnns2)=O)cc2sccc2cn1 N1(C(C(C)n2ccnc2)=O)CC(CNC(C2CCN(CC3CC3)CC2)=O)C(O)C1 O=C1CCC2CN(c3cc(NCc4ccc(-n5cncn5)cn4)ncn3)CCC2N1 C(=O)(C1=CSCS1)N1CC(CC=C)(NC(c2cnc(C(C)(C)C)o2)=O)C1 c1(CCC(N2CC(C(=O)Nc3cccc(F)c3Br)C2)=O)cc(F)c(F)c(F)c1F c1(C(N(CC(CNC(CN(C(C)C)C)=O)O)C)=O)cccc2sncc12 C12(NC(CS(C)(=O)=O)=O)COCCC1CN(C(c1cnc3[nH]cnc3c1)=O)C2 n1(COC)nccc1C(=O)NC1CC1CNC(=O)COC1(C)CCCC1 C12(N)CCCC1N(C(=O)Nc1ccccc1)CC2.C(=O)(C(F)(F)F)C(=O)C1CC1 c1(C(N2CC(C(C)NC(Cc3cc(C)sc3C)=O)C2)=O)cc(C)n(C)c(=O)c1 N1(C(C(C)OCCC#C)=O)CCC2C(CCN2C(=O)COc2ccoc2)C1 c1(C(=O)NCC2C(CNC(C3(C(=O)NC)CCC3)=O)C2)coc2ccc(Cl)cc12 N1(C(C2(C)CC(C)(C)C2)=O)CCCCC(NC(c2coc(C(F)(F)F)c2)=O)C1 c1(N(CCCOCC=C)C)ccc(S(=O)(=O)N2CCC(OC)C2)c(Cl)c1 C1(NC(CCSCCCC)=O)CC2C1CCN2C(c1ccc(N2CCC2)cc1)=O c1(-c2ccc(C)nc2C)ccc2c(c1)COC21CN(Cc2cc(F)cc(Br)c2)C1 Cc1cc(C(=O)NC(C)C(C(C)C)NC(=O)CN(C)C2CC2)n(C(C)(C)C)n1 C1(O)(CN(C)C(c2coc(CO)c2)=O)CCN(C(=O)C(C)(C)CC2CC2)C1 Cc1ccncc1CC(N1CCCC1C1(NC(=O)CC2CC2C)CC1)=O O=C(C#CC1CCCCO1)N1CCC2CN(C(c3ccc4c(c3)CC4)=O)C2C1 C=CC(C)(CC)C(=O)NCC1CCCN1CC=Cc1cncnc1O N1(C(CCCOC(C)=O)=O)CCCC(c2cn(C(C)C(=O)N(C)C)nn2)C1 Cc1cc(C)c(C(N2CC3(CCC3)CC2CNC(C2CC2(Cl)Cl)=O)=O)c(O)n1 N1(C(C(C)C)=O)CCCCC1C(=O)NC(C)CN(C)C(c1cccc(F)c1)C C1(C(=O)NCCC2CC(NC(C(C(C)C)OCC(C)C)=O)C2)CCCCCCC1 N1(C(C(=O)OC)C2(OC)CCC2)CCOC(C(F)(F)F)C1C c1(C(=O)NCC(CNC(c2c(C)oc(C)c2C)=O)F)cnc2n1CCCCC2 c1(OC)ccc(C=CC(=O)N(C2CN(C(=O)C(C)CS(C)=O)C2)C)c(C)c1 N1(C(CCC(=O)N(C)C)=O)CC(CC(=O)NC(C2CCCCC2)CO)C2(CC2)C1 CCCC(C)(O)CC(=O)NC1CCCCN(C(c2ccc(F)nc2)=O)C1 N1(C(C2CC(C)CN2N)=O)CCCC(C#N)C1 c1(C(N2CC(COC)(NC(=O)CCc3cnn[nH]3)C2)=O)nc2ccccc2[nH]1 C1(CN(C(CCCOCCOCC)=O)C)CCCN(C(=O)C(c2ccnn2C)O)C1 CC(C)C(O)C(F)(F)C(=O)N1CCCN(C(=O)CCCCN2CCOCC2)C(C)C1 C(=O)(C1CCc2ccccc21)N1C(C)C(NC(=O)COC2CCOC2)CCC1 C1(NC(C2CC2)=O)CCCCC1.C(Cn1cncn1)(CO)NC(=O)COCC C1(CCNC(C23CC(F)(C2)C3)=O)(OC)CN(C(=O)CCC2CC2(Cl)Cl)C1 N1(C(NOCCN(c2cccc([Si](C)(C)C)c2)C)=O)CCCC(C2CCCCC2)C1 Cn1cc(C(=O)NCC2(F)CN(C(=O)CC3CC4CC(=O)C3C4)C2)c(O)nc1=O N1(C(C23OC(C)C(CC2)C3)=O)CC2CCC(C1)N2C(C1(C)CC(F)(F)C1)=O C=CCCCCCCCCCC(=O)NCC1CCCN1C(=O)CCc1ccco1 C1(C(=O)NCCCN(C(C2CCCCC(=O)N2)=O)CC)COC2COCC12 c1(Oc2cc(C)c([N+](=O)[O-])cn2)cnc2c([N+](=O)[O-])cnn2c1 c1(C(=O)NCC(C2CC2)NC(c2[nH]c(=N)sc2)=O)cc2ccccc2cc1F C1(OCCNC(C2CN(C3CCCCC3)C2)=O)CCN(C(=O)C(Cl)=CCl)CC1 CC1(CNC(c2csc(C3CCCO3)n2)=O)CCCN1C(=O)COCCCF c1(CCN(C(CC2CN(C(C=CNC)=O)C2)=O)C)cc2cc(Br)ccc2s1 c1(C(N(CCC)CCNC(c2nc(C(C)C)oc2C)=O)=O)cc2cnccc2o1 C1(C(N2CCC(NC(C=CC)=O)C2)=O)CCCCC1C1CC1 S(=O)(=O)(c1ccccc1)N1CC2C(CNC(c3cnnc(Cl)c3)=O)(C2)C1 C=CC(O)(C(=O)NC(CNC(c1cc[n+]([O-])cc1)=O)C1CCC1)C(F)(F)F c1(C(=O)NC(CN(C(C(CCC)C)=O)C)CC)c(C(C)C)cccc1F c1(OC)ccc(CN)cc1C(=O)COC(C)(C)C.C1(O)(SC)CCC(C)C1 N1(C(C=NOC)=O)CCC(C)(CC(=O)NCc2ccc(C#N)s2)C1 Cc1cc2ccc(C(=O)NC3CN(C(=O)C4=CS(=O)(=O)CCC4)CC3C)cc2o1 c12nc(no1)CN(CC)C2C.CCCCNCc1ccco1 N1(C(C2CC(C)(CC)C2)=O)CCC(NC(c2csc3nccn23)=O)C12CC2 N1(C(c2nc(C)sc2)=O)C2CCC1CC(CNC(c1ccnnc1Cl)=O)C2 N1(C(c2ccc(C(C)=O)o2)=O)CCC2CCCC12C(=O)NCCC(F)(F)C(C)C C1(NC(c2cccc(NC)n2)=O)CCC(CN(C(c2c(CC)c[nH]n2)=O)C)CC1 C=C(C)C1CCC(C)=CC1CC(N1CCC(C)(NC(=O)CC2CC(C)C2)CC1)=O C1(CC(=O)NCC2CN(C(c3nc(C)sc3)=O)CC2(C)C)CCn2cncc2C1 C1(CC)CN(C(=O)CC2CC(O)C2(C)C)CC1NC(c1ccc(C(C)C)s1)=O C(c1ccc(F)cc1)=CC(=O)NCC1C(NC(CN(C(C)=O)C)=O)C1 CC(c1ccccc1)=CC(=O)N(CCC(C)NC(C1(C#N)CC1)=O)C C12CN(CCC1N(C)Cc1nccs1)C2=O.C1(CC)CCN(CC)CC1 Cc1nc(CNC(c2ccc(CNC(=O)CCc3cccs3)o2)=O)no1 C1(NC(CCC#C)=O)CCSC12CN(C(c1ncc3ccccn13)=O)C2 Cc1cn2c(n1)CC(C(N1CC(C(C)NC(c3cc(Cl)sc3Cl)=O)C1)=O)CC2 Cc1ncc(C(N2CCOCC2CN(C)C(c2ccc(O)c(F)c2)=O)=O)c(O)n1 C1(C(N(CC(C)(C)NC(=O)C(F)=CCO)C)=O)CC(C(F)(F)F)CO1 N1(C(c2c(C)c[nH]c2)=O)CCn2cccc2C1.N12CC3CC1C3C2=O c1(C(N2CCC3CC23C(=O)NC2CC(O)(C(N)=O)C2)=O)ccc(F)c(F)c1 C(=O)(C(C(C)O)NC(=O)OC)N(CCCN(C(C1C(CC)CCC1)=O)C)C C1(NC(=O)C=C2CCSCC2)C2CCN(C(=O)C(c3ccccc3)F)CCC12 Cc1coc(C(C)C)c1C(N1CC(NC(C23CCC2C3)=O)C(F)C1)=O c1(C(=O)NC2CC(CNC(C3(Cl)CC34CCC4)=O)C2)c(Cl)ccc(F)c1F Cc1nn(C)cc1CN1CCSC(C(=O)NCc2cncnc2)C1 C(C)(C)(CC(C(=O)NCCc1ccc(F)cc1)OC)N(CCCF)CC c1(N(C)C)ccc(C(=O)NC2CCCCC2CNC(=O)CCNC(=O)CO)nn1 N1(C(=O)Nc2c(C#N)cccc2[N+](=O)[O-])CCc2nc(C3=CCC(O)CC3)sc2C1 C(C(=O)NC(C)(C)CCNC(C1CC=CCC1)=O)(C(C)C)NC(CC(C)C)=O c1(N2CCC(NC(C(COC)(C)O)=O)CC2)ncnc2ccc(O)cc12 Cc1c(C(N2CC3CC3(NC(c3cc(O)nn3C)=O)C2)=O)nn2ccccc12 c1(N2CCC(CC(C)NC(C3(CCC)CC3)=O)CC2)c(F)cccc1[N+](=O)[O-] C(=O)(C(=O)CC(C)CC)N(C(C(=O)NC(CCCC)C(=O)N(C)C)C)CC c1(CC(=O)N(C2CCN(C(=O)OCC)C2(C)C)C)ccc(Br)c(Cl)c1F.C(C)(C)(C)O N1(C(c2cc(CC)nn2C)=O)CCOCC(NC(C2(F)CC=CC2)=O)C1 C1(CNC(c2c(C(C)C)scn2)=O)C2CN(C(=O)Cc3c(Cl)cnn3C)CC12 c1(C(=O)NC2(COC)CN(C(C3C=CC=CC=C3)=O)C2)cc2n(n1)CCOC2 c1(C(N2CCC(C(=O)OCC)C2)C(=O)NCC(C)C)ccc(C(F)F)cc1F c1(CN(C)C(c2cc(Cl)ncc2F)=O)ccc(Br)c(Cl)c1 CCCC(O)CC(=O)NCC1(CNC(C2CC23CCOC3)=O)CC1 N1(C(CC(C)OC)=O)CCCC(C)(CNC(=O)C=Cc2ccco2)C1 S(=O)(=O)(c1ccc(C#N)cc1)N(C1CC2CCC1N2)C(c1c(C)noc1)=O C1(C(N(CC#C)CC)=O)CC(O)C(O)CC1CNC(C1CCN(C)C1=O)=O C(=O)(C(CNC(=O)C(C)S(N)(=O)=O)(CC)CC)N1CCN(C(C#C)C)CC1 C(c1cccc(Cl)c1)=CC(=O)NC(C)CCNC(=O)CC1COCCN1C C#CC1(C=C)COCCN1Cc1n[nH]cc1Br c1(OC)ccc(=NCc2ccc(NS(C)(=O)=O)c(C)c2)[nH]n1 C1(NC(=O)CCc2ncccn2)C2CN(C(=O)CCc3nc[nH]n3)CC12 N1(C(Cn2c(C)csc2=O)=O)CCCC(C)C1CNC(C1(C)CCC(F)(F)C1)=O Cc1ccc(OCCC(N2CCC(Nc3ccc(N)cn3)C(C)C2)=O)c(C)c1 c1(-c2ccc(C#N)nc2)cccc2c1CCN(Cc1cccc(O)c1O)C2 C1(NC(CCCNC(=O)OCC)=O)CN(C(c2cccc(=O)o2)=O)CC1C CCC(O)C(C)C(=O)NCC1CN(C(=O)CSCc2cccnc2)CCN1C C1(N(c2nnc(CCC)s2)CCO)CCCN(C(c2nc[nH]n2)=O)C1 C1(C(C(=O)NCC(C)N(C)C(C2(C(F)(F)F)CC(O)C2)=O)OC)CCCCCC1 C1(CCOC)CN(C(=O)CC2CCCN2C)CCN1C(=O)CC1CCCCCC1 N1(C(c2c(CCC)cccc2)=O)CC2CCOC2(CNC(c2nn[nH]c2Cl)=O)C1 c12ccc(F)c(c1)CNC2=O.c1(NC(C2CC(C(F)(F)F)C2)=O)ccc(CO)s1 CN1CCC(F)(C(=O)NC2CC23CC(COCC2(C(=O)NC(C)C)CC2)C3)C1 C12(OC)CCC(C(N3CC(NC(=O)C(C)(C)c4cscn4)C(F)C3)=O)(CC1)CC2 C(CCC(F)(F)F)(C(=O)N(CCCC1CC1)CCO)NCC N1(C(C(C)(C)C)=O)CCCN(C(C2CC3(C)CC2CO3)=O)CC1CO C1(CN(C)C(c2cc(Cl)n[nH]2)=O)CCCN(C(c2ccnc(CO)c2)=O)C1 C12CCN(C(=O)CCN3CCOC3=O)CCC1C2.C1(C(N)=O)CCN1C=O c1(C(N2CC(O)(CNC(C3(OCC)CCOC3)=O)C2)=O)cccc2c1CCCC2 C1(C(=O)OC)CCCCC1C(=O)NCCOCCCNC(c1cn(C(C)C)nn1)=O N1(C(C2(NC(C(C3CCCO3)OC)=O)CCCC2)=O)CCCC(N(C)C)C1 N1(C(CC=C)=O)CCC2(CCCCN(C(c3cnc4ncccc4c3)=O)C2)C1 c1(-n2cc(CCC(=O)N(C(C(OC)OC)(C)C)CC)nn2)cc(Br)cc2c1OCC2 C1(C(N2CCC(CNC(CC(C=C)(C)O)=O)CC2)=O)CCc2[nH]nc(O)c2C1 C=C(C)CC(C)C(=O)N1CCCCC1CN(C)C(c1occc1Br)=O CC1=C(C(=O)N2CCC2CNC(c2ccc3oc(C)nc3c2)=O)C(=O)OC1(C)C C(=O)(C(C)(C)C(=O)N1CCN(C)C(CNC(c2nc(=O)n(C)[nH]2)=O)C1)N(C)C CCC(CC(=O)N1CCC(F)(CNC(=O)C=Cc2cnccc2C)C1)C(C)(C)C C1(F)(C(=O)NC2C(CSCC(=O)NCc3ccsc3)CC2)CC2(CCC2)C1 N#Cc1ccnc(C(N2CC3C(CNC(=O)C=CCF)C3C2)=O)c1 C(CCC(C)C(=O)NC(C1CCCC1)CNC(c1cccc(F)c1C)=O)OC N1(CC(=O)NCc2c(C3CN(C(C4(C)C=CCC4)=O)C3)ocn2)CCCCS1(=O)=O CC1(C)C2CC(C(=O)OCc3ccccc3C(=O)NCc3ccoc3)CC12 C(=O)(CC1CC(O)c2ccccc21)NCCN1C(=O)CC(C(=O)OCC)C1 N1(C(C(C2CCC2)OCC)=O)CCCC1(C)C(N1CCCC(CN=[N+]=[N-])C1)=O Nc1ccc(Br)c(F)c1C(=O)NCCNC(C1C2CCCCCCC12)=O Cc1nn(C)c(CNC(c2sccc2Cl)c2nnnn2CCOCC2CC2)c1Br n1(CCC(=O)NC2(C)CC(NC(C(C)NC(=O)NC)=O)C2)ncn(C)c1=O C(=O)(C(CP(C)(C)=O)C(F)(F)F)NC(C(C)(C)C(c1cn(CCCCF)nn1)C)=O N1(C(c2cncc(OC)c2)=O)CCCC(NC(=O)C=CC2CCCCCC2)C1C CCC(COC)(CC)C(=O)NC(C)CCC(=O)NC1CC2C=CC1C2 Cc1cccc(CN2CCC(O)C2C(=O)Nc2ccc(Cl)c(F)c2)c1Br N1(C(C2(C#C)CC2)=O)CC(NC(=O)C(CC)C2CCOCC2)C(N=[N+]=[N-])C1 c1(CC)nccnc1C(=O)N(CCCNC(=O)CCC(C)Oc1ccccc1)C c1(C(=O)NC2C(C)CN(C(c3ccc(F)s3)=O)CC2)cc(Br)c([N+](=O)[O-])[nH]1 c1(OC)cc(N2CC3(CC3)CC2C(=O)NCc2ccccc2F)nc(S(C)(=O)=O)n1 N1(C(=O)CN2CCOCC2)CCn2cc(C(N3CC4(CCC4)C3)=O)nc2C1 CC12CN(C(c3ccc(N)cn3)=O)CC1CN(C(C1CCN1C1CCCC1)=O)C2 N1(C(CCOc2cccc(C)c2)=O)CC2CC(NC(=O)CC3C=CCC3)CC2C1 C1(NC(CN(C)C(=O)C2CC2)=O)COCCC1NC(C1(CF)CC1(F)F)=O c1(C(=O)NCC(CNC(C2(CC)CCCO2)=O)S(C)(=O)=O)cc2ccncc2[nH]1 C1(NC(CCOC)C(=O)Nc2cc(F)ccc2OC)CCCN(C(Br)Br)C1C Cc1ncc(C(F)(F)F)c(=NC(=O)c2scnc2Br)[nH]1 c1(C(CNC(C2C=CC(NCc3ccnc(Br)c3F)C2)=O)O)ccc(F)cc1F N1(C(c2c(C)csc2)=O)CC(C)CCC1C(=O)NCC#CC#CCO C(C)(C)(CCCNC(=O)CCC(N)=O)NC(C(C=C)OC)=O C1(CC(N2CC(C)(OCC)C2)=O)C2CCCC2N1C(=O)CCc1cnccn1 c1(C(N2CC3C(NC(C=CCCC(C)C)=O)(C3)C2)=O)ccn2[nH]c(=N)nc2c1 C(C(CC(F)(F)F)NC(C12CCC(C1)C2)=O)NC(CC1(CC)CCC1)=O N1(C(CCCCSC)=O)CCC(N(C)C(c2ccnc(CO)c2)=O)C(C)C1 c1(NC(C)C)ncccc1C(=O)NCC1CCN(C(=O)C(F)n2ccnc2)C1 c1(C2C(C#N)C2)ccc(C=O)cc1.C1(F)(C(N2CCC(OCC)C2)=O)CCCCC1 c1(CC(N2CC(C)C(NC(c3cc(CCO)on3)=O)C2)=O)ccc2sccc2c1 c1(C(=O)NC2(CF)CCN(C(CCSCC)=O)C2)ccc(-n2cncn2)c(Cl)c1 CC1=CCC(C)(C(=O)NC(CCNC(=O)CCn2ccnc2)C(C)C)CC1 C12(C(=O)NC(CCNC(c3cnc(C(=O)OC)s3)=O)(C)C)CCCN1CCC2 C(CCC(C(=O)NCc1snnc1C)NC(=O)Cc1nocc1C)OC Cc1[nH]nc2c1NC2=O.c1(CCC(=O)NCCC#C)cnc(C(=O)O)o1 Cc1cc(NC(=O)C(=O)NC2CCCOC2CCc2ccccc2)c(F)cc1Cl N1(C(C2(O)CC(C)(C)C2)=O)CCC2(CC1)OCCC2NC(C1CCC(F)(F)C1)=O c1(C(=O)NC(CCN(C(C2CC(C)C2)=O)C)C(C)C)ccc(CC=CC=C)cc1F CN1CCC(C(=O)NCC#CC(=O)NC2CCCC2C(N)=O)C1 c1(CONC(C2C3CN(C(C(CC)OC)=O)CC32)=O)ccccc1[N+](=O)[O-] c1(C(=O)NCC2(O)CCCN(C(C3CC(F)C(=O)N3)=O)C2)nccc2nn[nH]c12 c1(C(N(CCC(C)NC(c2cnc(S)[nH]2)=O)C)=O)cc2c(nc1O)CCCC2=O C1(Cl)(C(=O)NCc2cc(C#N)oc2)C2CCC(=O)C12 C1(NC(c2c(C)cc(C)o2)=O)CCN(C(=O)CCCCN(C)C)C(C)C1 Cc1cc(Cl)ccc1OCC(=O)N(C1CCN(C(C2CC2C#N)=O)CC1)CC1CC1 C(C(=O)N1CCCC(C)(NC(C)=O)C1)(C(F)(F)F)OC(C)=O C1(CNC(CCC(C)SC)=O)CCCCCN1C(=O)COC(C)C(F)(F)F N1(C(=O)OC(C)(C)C)Cc2nccn2CC(Nc2cnc(CCC(F)(F)F)s2)C1 C1(N(C(C(C)N2CCCC2)=O)C)CCCN(C(c2cnc(C(F)F)s2)=O)C1 N1(C(C(=O)NCC)=O)CCCCC(CNC(c2cnn3ccn(C)c23)=O)CC1 c1(C(N2CCCC(CC(C(CC)C)=O)C2)C(=O)N)cc(Br)cc2cccnc12 C1(C(N(CCN(C)C)C)=O)CN(C(=O)Cc2cncn2C)CC12CC2 C1(CC(N2C(CC(=O)NCCn3ncc(C)c3)CC2)=O)CCOC1(C)C c1(C(c2nnnn2C2COC2)NC(CCC)C2CC2)cc(F)cc(I)c1 c1(C(=O)NCC2CCCN(C(C(CC)n3ccnc3)=O)C2)cc2ccccn2n1 CC1CCN(C(=O)C(C)(C)C(=O)N(C)C)CC1CNC(=O)C(C)(C)F C1(C(N(CCOCCC(=O)NCCC#C)CCO)=O)CCC(=O)N(C)C1 CCCCCS(=O)(=O)CC(=O)NC1CCN(C(=O)CC(O)CN(C)C)C12CCC2 c1(C(=O)NCC(N(C(=O)C=CS(C)=O)C)C2CC2)cnc2nc(O)ccc2c1 C(=O)(CC(C)(C)C)NC(C)C(=O)NCC#CCNC(=O)CCc1cc[nH]n1 N1(C(C(F)=C(C)C)=O)CC(C(=O)NCc2ccc(C#N)cn2)C(C)(C)C1 CC1CCCC(C(=O)NCCCCCN(C)C(C2(C3CC3)CC2)=O)C1 C(=O)(C1CCc2snnc21)NC1CCC(N(C)C(c2ccc([N+](=O)[O-])[nH]2)=O)C1 CCCCC(C(=O)N1CCC(CO)C1)NC(=O)C(C)n1ccnn1 Cc1c(Br)ccc(CC(=O)N(C)C(c2cnn[nH]2)=O)c1F C(N(O)C(=O)C(C)Cc1ccccc1)c1cn(-c2ccc(C)cc2)nn1 C1(C2CC2)(OC)CN(C(=O)NCCCC2CC(C)OC2C)C1 c1(OC)nc(C)ncc1C(=O)NC1CCC(N(C(=O)C(C)(C2CC2)OC)C)CC1 C(=O)(C(C)CC(C)(C)C)NCC12C(CN(C(Cc3cc(OC)c(C)cc3)=O)C1)C2 C12(C(N3C(CN(C(=O)CCc4ccccc4)C)CCC3)=O)CCCCC1C2(F)F O=C1CCN(Cc2cc(F)c(F)cc2O)C2COCCN12 N1(C(c2n(CC)ncc2)=O)CC2CC1(CNC(c1cn(CC(F)(F)F)cn1)=O)C2 Cc1ccc(C2(CN(C(=O)Nc3ccccc3)CCc3ccccc3)CCC2)nc1 c1(OC)ccc2c(c1)C(C(=O)N1CC3CC3(NC(C3(C)CC(C)(C)C3)=O)C1)CC2 c1(NC2(C)CC(C(=O)Nc3ccc(Cl)o3)C2)ccc([N+](=O)[O-])cc1-n1cnnn1 Nc1cccc(C(=O)NCCCC2(CNC(C3CC3[N+](=O)[O-])=O)CCCC2)n1 c1(C(N2C(CN(C(c3ccoc3Br)=O)CC)CCC2)=O)cc2n(n1)CCO2 C1(NC(C(=Cc2cccnc2)C)=O)CN(C(=O)Cc2nc(=N)[nH][nH]2)CCC1(C)C c1(C(N(CCCCNC(=O)CCN2C(=O)CCC2=O)C)=O)cccc(Cl)c1F C1(NC(C2(CNC(C3CC4C=CC3CC4)=O)CC23CCC3)=O)CC2CCC1CC2 C1(C(CNC(CNCCOC)=O)OCC(=O)SCC#C)CCCSC1.CC c1(C(N2CCN(c3nc(SC)nc(C)c3)CC2)=O)ccc(F)c(Br)c1F C1(NC(C2CC(OCC)C2)=O)CC2CC1CN(C(c1coc(SC)c1)=O)C2 CCN=c1ccc(C(N2CC(O)(CN(C(=O)CCn3cccn3)C)C2)=O)c[nH]1 C=C(C)C1OCCC1C(N1CCC(NC(=O)CCOCC(C)(C)C)CC1)=O C(CC#CC(C)(C)OC)OC(C1C(C(=O)OCC)CCCO1)=O c1(C(=O)NCC2(NC(CC(C)C3CC3)=O)CCC2)cc2ccncc2s1 C(=O)(CCCC(=O)N(CCNC(c1ccc(OC(F)(F)F)nn1)=O)C1CC1)OC CC(C)(CCC(=O)NC1CCCCN(c2ncns2)C1)[N+](=O)[O-] c1(CC)cc(OC)ccc1C(=O)NCC1CCN1C(=O)C(C)(C)c1cnsc1 CC1CC(c2cccc(C(F)(F)F)c2)N(Cc2ccn(C)c2)C1 N1(C(C)=O)CCCC1C(N1CCCC1CCNC(C1C2CCCC12)=O)=O N1(C(c2nc(C)sc2C)=O)CC2(CNC(=O)CC3CCCCC3C)CC1CO2 N1(C(c2cc(C3CC3)[nH]n2)=O)CCC(CCNC(C23CCC2C3)=O)CC1 N1(C(CCC#C)=O)CCC(CC)C1C(=O)NC1(CO)CC(O)C1 C1(CNC(=O)NCCC=CC)C2CC3C(C2)C13 N1(C(c2ccc(C)s2)=O)CC(C2CCN(C(=O)C(C)N(CC(F)(F)F)C)CC2)C1 C1(CC=C)(C(=O)NC(CCOC)C(C)C)CCCN1C(=O)CC1CC(CC)=NO1 c1(C(=O)NC2CC(NC(C(C(CC)O)(C)C)=O)C2)cnc2ccccc2n1 C(CCC(C)C)(C(=O)NCCC(C)N(C(=O)COC(F)F)C)NC(=O)OC C1(C(N2CC(CCCCNC(CC3CCC(C)CC3)=O)C2)=O)CC2CCCCCC12 CC(C)CC(C)C(=O)NCCCN(C)C(C12CCC(C(F)F)(CC1)C2)=O C1(O)(CC(=O)Nc2cncc(Br)c2)CCN(Cc2cnc(Cl)s2)C1 c12ncc(cn1)NC2c1nnnn1C.c1(CC)cccnc1C(F)(F)F CCCC(C(=O)N(CCNC(c1ccnc(C)n1)=O)Cc1ccccc1)OC O=C(C1SCCc2ccccc21)NCC12CC1CN(C(=O)C=Cc1ccccc1)C2 CCCC(C)CC(=O)NCC(CC1CC1)C(=O)N(CC(F)F)CC(C)O c1(CC)nc(C)c(C(=O)NCC2CCCN2C(c2cccc(SC3CC3)c2)=O)s1 C12CCCN(C1)C2=O.c12cccc(c1)OC2.C(=O)(CC(=O)N)OC.C(C)(=O)O C1(CCC)CN(C(=O)C=CC(C)C)CCN1C(=O)CCCCC1CC1.c1csnn1 N(C(=NCC#CC1CC1)NC1CC12CC2)C1C(F)(F)CC1 CC1=C(C)CC(C(=O)NC(CCF)C(=O)NCCc2cnc(C)[nH]2)CC1 C1(CC)Cc2c[nH]cc2S1(=O)=O.c12cc(OC)cc(c1)C(=O)N(CC)C2 CC(Cc1ccc(Cl)cc1)CCC(=O)NCC1C=CCN1C(=O)CCS(C)(=O)=O c1(C(=O)NC2C(NC(c3c(C)ccc(Cl)c3)=O)CCC2)cc(Cl)c(F)c(Cl)c1 C1(CNC(c2n(CC)nnc2)=O)CC(O)CN1C(c1ocnc1C1CC1)=O c1(CC(C(N2C(C(C)(C)NC(CN(C)CC)=O)CCC2)=O)O)cc(Cl)sc1Cl c1(C(N2CCC(c3cnccn3)CC2)=O)cc(F)c(Br)cc1[N+](=O)[O-].C12CC1NC2 c1(CC)cccc(C(=O)NCCC2(O)CN(C(c3cncc(C)c3)=O)C2)n1 C1(C#N)(C(=O)NCC(CC)NC(=O)C(C)COC)CCS(=O)(=O)CC1 C(=O)(C1COCc2ccccc21)NC(C)CCNC(c1nc[nH]c2nccc1-2)=O C(N=c1[nH]c(=NCC2CC2C)[nH]c2cc(OC)ccc12)c1cc(CC)on1 c1(C(=O)OC)cccnc1NCCCC1CCCN1C(=O)Cc1ccc(Cl)cc1 N1(C(CC(C)SC)=O)CCC2CC(CNC(C3CC(C)CC(C)C3)=O)CCC2C1 c1(CC)cc(Cl)ccc1C(=O)NCCCN(C(=O)Cc1c(F)cccc1Cl)C1CC1 c1(C(=O)NCCC(C)NC(=O)CC(C2CC2)C2CC2)nn(C)cc1Cl C1(C(=O)OCC(C#C)C)CC2(CC2)C12CCC2 CCCCCC(C)CC(=O)NC1CCN(C(C2COCCN2CC)=O)CC(O)C1 N1(C(C2(C(=O)NC)CC2)=O)C2CCC1CN(C(=O)C(c1ccc(Cl)cc1)(C)C)C2 C1(CNC(C2CC(OC)C2)=O)N(C(=O)CC2CCCCC(=O)N2)CCCC1(C)C C1(=O)C2=C(CO1)N(C)C(=O)N(C)C2c1cccc(Br)c1.C1(C(=O)OC)(CF)CC1 c1(C(N(C2CCCN(C(C)=O)C2)c2ncc(CC)o2)=O)cnn2cccnc12 C1(CNC(c2cc(Cl)c[nH]2)=O)COC(CNC(C2(n3cccn3)CCC2)=O)C1 c1(C(C(=O)N(C(CNC(CC(=C=C)C)=O)C2CC2)C)O)ccc(F)cc1C N1(C(CCC(C)NC(C23CCCC2C3)=O)=O)CC2(COC(=O)N2C)C1 c1(C(=O)NCCC(C)NC(C2CC(C#N)C2)=O)cc(C2(C)CC2)n[nH]1 C1(NC(c2c(C)cc(C)s2)=O)CC(C)CN(C(=O)CC2CCCC(C)(C)O2)C1 N1(C(C2C(CCOC)C2)=O)C(CNC(c2cc3n(n2)CCC3)=O)CC2COCC12 C1(C(=O)NCC(C2CCC2)OC)CCN(C(c2cc3ccccc3[nH]2)=O)C12CCC2 c1(C(N2CCCC(CCNC(CC3(C)CCOC3)=O)C2)=O)ccc(P(C)(C)=O)o1 C1(CC)CCc2nc(O)c(C(N3CCC(C)(NC(=O)CC(C)(C)O)C3)=O)cc2C1 N1(C(C(C(C)CC)N(C(CCOCCC)=O)C)=O)CCC(C2(C)CC2)C1 c1(C(C)N(CC(CCC(C)NC(=O)NC(C)(C)C)C)C(C)=O)cc(Br)ccc1F N1(C(C(c2cccc(F)c2)C)=O)CCCCC1CNC(=O)C(O)c1ccsc1 Cc1cc(C(=O)NC2CCC(NC(C3(CC#N)CCCC3)=O)CC2)cc(C)c1Cl c1(CNC(=O)CCn2cccn2)cccc(C(N2CC=CC2COC)=O)n1 N1(C(CN(C)C)=O)CC(F)CC1CNC(C1CC1c1ccco1)=O C(=O)(C1=C(CC)OCCC1)N1CC(NC(c2c(Cl)ccc(C#C)c2)=O)C(C)C1 CN1C(=O)CC(C(=O)Nc2nnc(CC(F)(F)F)s2)NC1=O c1(C(=O)NCCN(CC(C)O)C(c2cnc(C(C)C)[nH]2)=O)cnc(Cl)c(F)c1N c1(OC)cccc(C(=O)NC(C)(CCI)c2nnnn2C2COC2)c1F C=C1C(C(=O)OC)C1C(=O)N(CCC(=O)OC(C)(C)C)C c1(CC(=O)NCC(CNC(C2C(C(C)(F)F)C2)=O)O)ccnn1C1CCCC1 N1(C(CC(CC)O)=O)CCC2CC1CN(C(c1ccc3[nH]ccc3c1)=O)C2 N1(C(C2(C#C)CCN(C(c3nccs3)=O)C2)=O)CCC2CN(C)CC2C1 c1(-c2c(COC)cccc2F)ccc2[nH]c(C(=O)Nc3cnc(Cl)nc3)nc2c1 N1(C(C(CC=C)C)=O)C2CC1CN(C(=O)Cc1ccccc1CC(N)=O)C2 CC(C(=O)NOCCCC1CC1)C(C)NC(=O)CCOC1CCC1 N1(C(C(C)CS(C)(=O)=O)=O)CCCC(C)(C)C1C(=O)NCC1CC=CC1 C1(C(C)C)CN(C(C23CC(C)(CO2)C3)=O)CCN1C(=O)CCc1ccsc1Cl N1(C(C2C(C)C2)=O)CC(C2CCCN(C(C3C4CCCOC34)=O)C2)C1 CC(C(=O)NCc1ccccn1)(C1CCCC1)NC(=O)CCc1cn[nH]c1 N1(C(Cc2c(C)noc2)=O)CC(C)N(C(=O)CN(C2CCSC2)C)CC1C C1(NC(c2c(C)[nH]cn2)=O)CCCCC1NC(C1(C)CNC(=O)N1)=O C(=O)(CCC(=O)OC)N(C(C(=O)N(CC(=C)C)CC)C)C1CCC1 Cc1cc(F)c(N)cc1C(=O)N(CC(O)CNC(=O)C1=CCCOC1)C C(=O)(C1=NNC(=O)CC1)NCC1CC(NC(C(C)c2cccs2)=O)C1(C)C c1(C(=O)NC2CC(F)(CNC(=O)CCc3ccco3)C2)ncccc1C(F)(F)F C(CCC(C)(C)C(=O)N1CC(C)(C)C1)NC(C(CC=C)NC(C)=O)=O C1(CCNC(C(CCOC)(C)C)=O)CN(c2nccc(C(N)=O)n2)CCS1(=O)=O C#Cc1ccccc1CNC(C1(CNC(C2CCC2C)=O)CC(=C)C1)=O CCCCC(CC(=O)N1CCCCC1C1(O)CC1)NC(c1ccc(C#N)[nH]1)=O c1(CCC(=O)NC23CN(C(C4CC=C(C)CC4)=O)C(C2)C3)cc(F)ccc1F C1(Nc2c(C(=O)OC)cccn2)CN(C(c2cc(C)c[nH]2)=O)CC1(F)F c1(CCSCC)nc(C2(Nc3ccsc3)CCC2)n(-c2cccc(F)c2)n1 C1(NC(C(=O)N(C2C(C)CCCC2)CC(F)F)=O)CC2CCCC1N2C CC1(C)CCC(CC(=O)NCCCCNC(=O)C(C)(C(F)F)c2ccccc2)C1 C1(NC(C2C(NC(=O)C(F)CC3CCOC3)CC=CC2)=O)CCCN2CCCC12 Cn1cc(C(N2CCC(NC(=O)CC3CCSC3)C(F)C2)=O)ccc1=O N1(CC(N2CCC(O)(CNC(C(C)C3(O)CCC3)=O)C2)=O)CCP(C)(=O)CC1 c1(CCC(N2C(CNCC3(C#N)CCC3)CCC2)=O)ccccc1Br C12(CCCCC1)C(=O)N(C(c1cnoc1C)=O)CC(F)CN2.C1(CSC)CCCO1 S(=O)(=O)(c1c[nH]ccc1=NC(C)c1cc(F)ccc1F)N(C(CC)CSC)C C1(C#N)(C(N2C(CN)CC2)=O)CCCC1.c1(C(=O)NC)scnc1CO C(CC(CC)C(=O)NCC(C)(C)CC(=O)NCCCCCCO)=CC N1(C(C2C(CCOC)C2)=O)CCN(C2CN(C(=O)Cc3cccs3)C2)CC1 N1(C(C2(C)CC(C)C2)=O)CC2CCCC2(NC(c2ccn(C(C)C)n2)=O)C1 c1(C(=O)NC2C=CCN(C(C3N(CC)CCOC3)=O)C2)cc(O)ncc1Br Cc1ncc(Cl)cc1CNC(=O)NCC(C(F)(F)F)n1cncn1 c1(OCC(=O)NCCSCC(=O)Nc2cc(F)c[nH]2)ccccc1F c1(C(=O)NC2CCCCC2NC(C2CS(=O)(=O)C2)=O)cnc2ccccn2c1=O c1(CCC(=O)N(CC2(CNC(c3c(C)c[nH]n3)=O)CC2)CC)c(C)nc(O)nc1C c1(C(=O)NC2CC(F)CN(C(=O)C(c3ccccc3)F)C2)cc2cnccc2[nH]1 CCC(CO)C(=O)NCC1CN(C(c2ccc(-c3cc[nH]n3)s2)=O)CC1N(C)C N1(C(C(C)(C)c2cccnc2)=O)CCOCC(CNC(=O)Cn2ncnn2)C1 C1(OC)CCCC(NCCN(C2(CO)CCC2)C(c2cnccc2Cl)=O)C1 C1(C)(CNC(c2c(CC)c[nH]n2)=O)CN(C(=O)C(C)CN(C)C)C(C)(C)C1 c1(C(=O)NC2(C)CCN(C(=O)C=C3CCCCC3)CC2)ccc2ncccc2n1 C(=O)(C1=CC2(CCOC2)C1)NC(CC)(CNC(C1CCCN(C)C1)=O)CC CC1(C)OCC(c2cn(CC3CC(CNC(C4COC4)=O)C3)nn2)O1 C12(NC(CCCCCNC(C)=O)=O)CCN(C(=O)CC3CN(C)C3)CCC1C2 C1(NC(c2c(C)ncs2)=O)COCCN(C(C2(C#N)CC3CC3C2)=O)C1 C12(CNC(c3c(C)[nH]nc3C(C)C)=O)CCCC1CN(C(=O)C=CC(C)C)C2 C(=O)(C1CCc2c[nH]nc21)NC1C=CCC(C(N(C2CCCCC2)CC)=O)C1 N1(CCc2nc(C)c(-c3ncc[nH]3)s2)CCC12CCCC(C)(C)C2 c1(C(=O)OCC)nc(CN2CCC(C)c3ccccc32)cc2ccccc12 c1(OC(F)F)cc2ccncc2cc1OC.c1(C2(C)C(O)CNC2)cc(F)cc(F)c1 c1(CNC(C(CSCC)NC(C2(N3CCCC3)CC2)=O)=O)ccc(C)c(O)n1 c1(C(=O)NCCC(CNC(c2c(CC)onc2C)=O)O)cccc(O)c1F C(=O)(CCC(=O)N1CC(CC=CC(=O)NCCOc2ccncc2)CC1C)NC c1(CN(C#N)CCCOC)nnc(COC(F)(F)F)n1CC1CCS1(=O)=O N1(C(c2cc(-c3ccco3)no2)=O)CCC2(CCCN2C(c2csnn2)=O)C1 C(C)(C)(CCC(=O)NCC1(CNC(=O)C=CC2CCCCC2)CCCCC1)OC N1(C(c2c(C)c[nH]n2)=O)CCC(CF)(NC(=O)C(C)Cn2cccn2)C1 C1(C(CC)C)CCC(NC(=O)CC2NC3CC2C3)CC1 Cc1nc2cc(C(=O)NCCC3CC(NC(=O)CCc4cnc[nH]4)C3)ccc2s1 N#Cc1ccc(N2CCN(C(c3ncoc3-c3cncs3)=O)CC2)c(F)c1 c1(C(N2CC(NC(C(C=C)(C)CC)=O)C(C)C2)=O)c(Cl)ccc(Cl)c1O N1(C(C(=O)NC(C)C)=O)CC(NC(C2CCC(F)CC2)=O)C(C)C1 C12COC3CN(CC13)C(=O)CC(O)CCC2.c1(C(=O)O)ccc2cccnn12 CN1CCC(C)(C(N2CCC(O)C(NC(=O)COc3cccnc3)C2)=O)CC1 c1(-c2n(C3CCC(C)C3)nc(CCCN(C)C)n2)ccc(Br)c(Cl)c1 CCCC(CC)C(=O)N1CCOCC1(C)c1cn(Cc2ccc(SC)o2)nn1 C(CCCCNC(C12COCC1C2)=O)N(C(C1CC1COC)=O)CC c1(CNC(CC2N(C(COCCOC)=O)CC2)=O)nn(C)cc1Cl Cc1cc(C(=O)NCC2CC(C)N(C(c3ccco3)=O)C2)cc(C)c1 Cc1cc(C(N2CCC(C)C(CNC(=O)C(C)(C)CO)C2)=O)c(Cl)cc1F C(C(C)(C)C(=O)NCCC1CCC(C)(C)O1)N(C(=O)Cc1cncnc1)C n1(CC)nccc1C(=O)NC1CCCC1CNC(C1(CO)CCCC1)=O C(CC(C(=O)N=c1ccn(CCN(C)C)[nH]1)N(C)C)NC(C1C(C)C2CCC1C2)=O C12(NC(C(C)C3CCCO3)=O)CC(C)(C1)OC21CN(C(=O)CC2CC=CCC2)C1 C1(C(C)(C)C)(NC(C(C)OCCSCC)=O)CCN(C(=O)CC23COCC(C2)C3)C1 c1(C(=O)NCC2CCC(NC(C3(C)CSC3)=O)C2)ccc(Cl)cc1 C1(CC)CCCCC1OCC(N1CCC(N(C(=O)C=Cc2sccc2C)C)C1)=O Cc1cc(Br)cc(C(N2CCCCC(C)C2)=O)c1C c1(NCc2ccc(OC)c(OC)c2)ccc2cc(Cl)cc(OC)c2c1 CC1=NOC(C)(C(=O)NC2(C(=O)NCC(C)(C)C#N)CC2C)C1 CC1Cc2cc(CC(=O)N(c3nc(Cl)nc(C4CC4)c3F)C3CC3)ccc2O1 c1(NC(C(C2CCC2)NC(c2ccc(SC)o2)=O)=O)cccc2nccn12 N1(C(C2CCC(C)CC2)C)CCC(C2CCCN(C(c3ccncn3)=O)C2)C1 C1(CCNC(CN(CC(C)(C)C)C)=O)CC(NC(=O)CC2(C#N)CC2)C1 c1(N(C2(C3CCCO3)CCCC2)C(=O)C2CC2)ccc(Br)cc1.C(CCC(=O)OC)NC C(=O)(C(C)(C)C(=O)NC1CC2CC1N(C(c1occc1C)=O)C2)NC N1(C(C2(C(CC)=O)CC2)=O)CCC(C(=O)NCC2CCC(C)C2)=C(F)C1 N1(C(C(C)OCC(C)C)=O)CCOC2(CCN(C(=O)CCc3ccoc3)C2)C1 C1(CNC(c2csc(-c3cn[nH]c3)n2)=O)CCCCN1C(C1CCS(=O)(=O)N1)=O CN=c1[nH]c(=NCC2CCOC2(C)C)[nH]c(=NC2CC(=O)N(C3CCC3)C2)[nH]1 C1(C(=O)OC)CCN(C(=O)Cc2cocn2)C1(C)C.CCC(C)C(=O)NCC=O N1(C(CCSCC)=O)CCCC(C(C)NC(=O)CC(c2ccccn2)C2CC2)C1 C1(C)(CNC(c2n(C)ncc2Cl)=O)CN(C(=O)CC2CCCOCC2)C(C)(C)C1 C1(NC(CC2(CC=C)CCCC2)=O)CCN(C(C2CC3CCC2C3)=O)CC1 N1(C(C2C(CC)C2)=O)C2CCC(C(=O)NCCCN(C)OC)C1CC2 CC(Cc1ccco1)N=c1nc(N2CC(F)C(F)C2)c2cc(F)cc(F)c2[nH]1 CCCC(C)CC(=O)N1CC2C(CC(=O)NCCN3CCCC(O)C3)C2C1 C1(NC(C2CCC(=O)N2)=O)CCCC(NC(=O)CC2COCCOC2)C1 c1(C(=O)NC(CC)CNC(c2cccnc2S)=O)[nH]c2ccccc2c1C1CC1 N(C1CCc2ccc(Cl)cc21)C(=O)CC1CCCCC1(F)F c1(C(N(CC(C)O)CCNC(C2COC(C)(C)C2)=O)=O)cc2n(c1)CCSC2 c1(C(=O)NCC2(C(C)NC(=O)CC3CCCC3O)CC2)nocc1Br C(=O)(C(C)CN(C(=O)CN1CC(C)(OC)C1)C)N(C(C)C(C)C)C N1(C(C=COC(N2CCC(C(=O)NC)C2)=O)=O)CCC(CC(C)OCC)CC1 N1(C(C=Cc2n(C)ccc2)=O)CCC2C(C1)CN2C(=O)C(C1CCOCC1)F C=CC(C)(C)C(=O)N(C)CCNC(c1ccccc1SCc1cccs1)=O C(c1cc(Cl)cc(Cl)c1)=CC(N1C(C(C)NC(=O)C2=CSCCO2)CCC1)=O C1(C2(c3ncc(C)o3)CCC2)CCCN(S(=O)(=O)CC2(C3CC3)CCC2)C1 CC(C)CC(C(=O)NCC1CCN1C(c1ccc(F)cn1)=O)N1CCCCCC1 N1(C(C2C(OC(C)=O)C2)=O)CCC2CC12C(=O)NCC1C(C)C1C c1(OC)cn(CC(=O)NCC2CCN2C(=O)C(C)CC(C)(C)C)c(C)cc1=O CC1Cn2nccc2CN1C(=O)N(c1ccc(Cl)cc1)CC1CC1 C(CC1CCOCC1)(C(=O)NOCC(=O)Nc1ccccc1C)OC CC(O)(CC(=O)NCC1CCCC1NC(C1(CC2CC2)CC1)=O)C(F)(F)F C1(C(=O)OCC(C2(OC)CCC2)(F)F)C2CC2C2CC12 N1(C(c2c(CC)ncs2)=O)CCOCC1CC(=O)NCCCc1nc(C)no1 Cc1nc(C(=O)O)ccc1C(=O)N.c1(C)cn(CCN2CCCCC2)nn1 CCC(C)(C)C(=O)C(=O)N1CCN(CCNC(c2ccc(C3CC3)nc2)=O)CC1 C=C(C)CCCC(=O)NCC(O)CN(C)C(c1ncccc1C(F)(F)F)=O CC(C)(C)CC(C)(C)C(=O)NC(CNC(c1n[nH]c2c1CC1CC21)=O)C1CCC1 N1(C(COC)=O)CCCC(C)(NC(N2CC(n3cccc3)C2)=O)C1 C1(C(=O)NCC2CC3CCC2O3)N(C(C2SCCS2)=O)CC12CCCC2 C1(C(=O)NCC2CCN2C(=O)CCc2cscn2)CCCOCC1 Cc1cc(C(N2CC3CC3(CNC(C3(C)CC4CC4C3)=O)C2)=O)nc(C)c1 C(=O)(C#CC1CCCOC1)N1CCCC(C(C)NC(=O)Cn2cnccc2=O)C1 c1(NC(=O)COC(=O)C=Cc2cn[nH]c2)cccc2ncccc12 N#Cc1cc(F)ccc1CN1CCC(O)(C(=O)NCc2ccco2)CC1 CC(C)(N=[N+]=[N-])C(=O)N1CCCCC(NC(=O)CC2NC(=O)NC2=O)C1 c1(C(N2CC(NC(=O)CC3CCC4CC34)C2)=O)nsc2cc(Br)ccc12 N(C(=NCCC1(O)CCOCC1)NCCN1CCCC1)C(c1ccc(C)cn1)C N1(C(CC2(C)CC2(Cl)Cl)=O)CCC(C)(NC(=O)Cc2cncc(NC(N)=O)c2)C1 N1(C(CCCC(C)=O)=O)CCCC(C2CCN(C(C3(C)CNC(=O)C3)=O)CC2)C1 C1(NC(CCC(N)=O)=O)CN(C(=O)COCC2CCCC2)CC2(CC2)C1 C1(C(=O)NCc2cc(C(=O)NC3(CCCF)CC3)n[nH]2)CCC(F)(F)C1 C1(CC)CN(C(=O)CC(C)(C)N(C)C)CCN1C(=O)CC1(C)CCCC1 C1(CNC(Cc2nccc(C)c2)=O)CCN(C(c2nccnc2N)=O)CC1(F)F C=CC(F)(F)C(=O)N1CC(CCNC(=O)C(C)CF)C1 C(=O)(C(F)(F)C1CCCCC1)OCCOCCCNCCN(CCc1ccccc1)C CC(C)(CNC(=O)Cc1cncnc1)CCNC(c1cncc(Br)c1)=O C=CCCN=C(NCC1(c2cccs2)CCCC1)NC1CSC(C)(C)C1 c1(C(=O)NC(C(CO)NC(c2c(OC)nsc2)=O)C)cc2sccc2cn1 C#Cc1cn(C)nc1C(=O)N(C)CC1(CNC(=O)CSCCOC)CC1 Cc1ccccc1C=CC(N1CC(O)(C(C)NC(C2CCC(C#N)CC2)=O)C1)=O C1(CC(NOCCC(C)C)=O)Cc2ccccc2CN1C(C1CC12CCC2)=O C(=O)(CC(F)(F)CC(=O)NCC1COCCN1C(C1CCCCO1)=O)OC CC1CN(c2ccc(CN3CC(N4CCN(C)CC4)C3)cn2)CCO1 N1(C(c2cncc(OCC)c2)=O)CCN(C(c2c(CO)n[nH]c2C)=O)CC1C N1(C(c2c(OC)n[nH]c2)=O)C2CCC(C(=O)NC3CON(CO)C3=O)C1CC2 C1(CN(C(COCCC)=O)CC)CCCN(C(C2CCC(C)(CC)O2)=O)C1 N1(C(C=C(C)I)=O)CCC(CF)(NC(c2cc(C)co2)=O)C1 C1(NC(CNc2cn(C)nc2)=O)CCN(C(c2cc(C(F)(F)F)on2)=O)CC1 c1(C(=O)NCCCC(C)NC(c2ccc(NC)cc2)=O)cc2n(n1)CCCC2=O C1(CC(=O)N(CCCCNC(=O)C(c2ccccc2)C2CC2)C)CCCCC1O C1(CN(C(c2ccc(CC)s2)=O)C)COCCN1C(C1CCCN1CC)=O C1(C(C)CNC(c2cc(Cl)ns2)=O)CCN(C(C2CNC(=O)C2)=O)CC1 c1(C(C(=O)N(C)CC2CCCCN2C(C23CC(C2)C3)=O)O)cc(Cl)cc(Cl)c1 Cc1nocc1C(=O)NC1CC(O)(CNC(c2cccs2)=O)C1 C1(O)(CNC(c2ccc(OC)cc2C(N)=O)=O)CCCC12CCOCC2 N1(C(CC(c2cccc(F)c2)C)=O)CCN(C(c2cnc(C(F)F)s2)=O)CC(O)C1 C(C(CNC(=O)C(N1CCCCC1)=O)C(F)(F)F)NC(=O)CC1CCOC1 c1(C(=O)NC2(CNC(C(C)C3CCCO3)=O)CCCCC2)cncc(O)c1Cl C1(c2c(C)nns2)CCN(C(=NCC(C)C)NCC2(C(N)=O)CCCC2)C1 C1(CNC(C2CC=CCO2)=O)CCN(C(=O)CCc2sccc2Br)CC1 N1(C(c2cc(COC)sc2)=O)CCC(NC(=O)C(C)OC2CCCCC2)C(F)C1 c1(CC=C)cccc(C(N2CC(NC(C3(SCC)CC3)=O)C(C)C2)=O)c1 C#CCCCCCCC(=O)NC1CCC(CCC(N2CCCC(C(N)=O)CC2)=O)C1 C#CCC(C)C(=O)NCC(F)CNC(=O)CCc1ccc(C(F)(F)F)cc1 c1(CN2CC(CC)N(C(c3ccnc(OC)c3)=O)CC2)cnc2snnc2c1 C1(CC(N2CC(C(F)Cn3cc(CO)nn3)C2)=O)(C(F)(F)F)CCCC1 C(CCCCC(=O)N1CCSC2CCC12)NC(c1cc(CCC)[nH]n1)=O C1(C(N(CC(CN(C(=O)C=Cc2cnn(C)c2)C)O)C)=O)CCCC2C1C2(F)F CCCCCC(CC)C(=O)NC1CC(CCNC(c2ncccc2F)=O)C1 c1(-c2cc(OC)c(O)nc2)ccc2sc(C(N3CCN(C4CC4)CC3)=O)cc2c1 N1(C(c2c(NC)cnnc2)=O)CCN(C(=O)C(=Cc2ccc(F)cc2)C)C2CC12 Cc1[nH]nc(C(N2CCC(O)(CNC(=O)CC3OCCC3(C)C)C2)=O)c1Cl C1(C(=O)NC(CNC(C2(OCC)CCOCC2)=O)CO)CC2(C1)CC(F)(F)C2 c1(C(C(=O)NCCCN(C(C(=O)NCC)=O)C)(C)C)ccc(O)cc1 c1(C(C)N(C)CC2CC(C(F)(F)F)CO2)ccc(-c2ccc(Cl)cc2)cc1 N1(C(Cc2nc(C)sc2C)=O)CC(NC(=O)C2=COCC2)C2(CC2)C1 CCCC(C)(CC)C(=O)NCCCCCCN(C(=O)C(O)Cn1cncn1)C C(=O)(CC(C)(C)C(C)(F)F)N1C(C)CC(NC(c2ccc3cncn3c2)=O)C1 N1(C(C2C(C#C)C2)=O)Cc2ccccc2CC1CNC(c1ccns1)=O c1(N2CC3(C(NC(C4C(C(C)O)C4)=O)CCS3)C2)ccc([N+](=O)[O-])cc1[N+](=O)[O-] CCCC(O)CC(=O)NCc1ccccc1CNC(C1(F)CC=CC1)=O c1(C(=O)NCC(CC)NC(c2ccc(OC)cc2C(F)F)=O)cc(Cl)cc(Cl)c1 C#Cc1cnn(CC(=O)NC2CC(NC(c3nnn(C(C)(C)C)n3)=O)CC2O)c1 C1(O)(CNC(c2c(Cl)nsc2Cl)=O)CCCN(C(=O)Cc2ccc(Cl)cn2)C1 C1(CC(=O)NC(C2CC(F)(F)C2)C)C2CCC(C2)N1C(=O)CN1CC2CC2C1 c1(OC)ccc(C)c(C(=O)NCCC2CN(C(C3(Cl)CC34CCC4)=O)CC2C)c1 N1(C(C)=O)CCN(C(C2(C)CN(C(=O)Cc3ccc(C)c(Cl)c3)C2)=O)C(C)C1 C(=O)(CCN(OC)C(=O)c1ccsc1)N1CCC(C#C)C1 n1(CCCCOC)ccc(C(=O)NC(C)(CNC(C2C(C)C2C)=O)C2CC2)n1 C1(NC(=O)C(C2CCCCC2)F)CCC2CC1CN2C(=O)CC1CCC2CC2C1 c1(CC(=O)NC(CC(C)NC(=O)C(F)(F)CN2CCCC2)C)cccnc1O N1(Cc2ccc(OC)cn2)CCC(C2CCCN(C(=O)CNC(N)=O)C2)C1 C1(N(C(C2CC2C)=O)CC)CCN(C(=O)Cc2ccccc2Br)CC1 c1(C(=O)OC)nc(Br)n2c1CN(c1noc(-c3ccc4ocnc4c3)n1)CC2 C1(C(N2C(CNC(c3nc(C)n(C)c3)=O)CCCCC2)=O)CC2CCCCN2C1 CC12CC(CC(N3CCCC(CCNC(=O)C4=CSCS4)C3)=O)(CO1)C2 Cc1ccc([N+](=O)[O-])c(C)c1C(=O)NCC(O)CN(C)C(c1c[nH]ccc1=N)=O C(c1ccc(O)cc1)=CC(=O)NCCN(CCC)C(C1CN(S(=O)(=O)CC)C1)=O c1(C(=O)NCC(C(C)C)NC(C(CCC)C#N)=O)nc2ncc(C)cn2n1 CCC(Cc1ccccc1)CC(=O)NC1CC(C)(NC(C2CN(C)C2)=O)C1 N(C(=NCCCc1cccs1)NCCF)CC(CCS(C)(=O)=O)CC(C)(O)C1CC1.OC C1(CNC(c2cnc(CC)[nH]2)=O)C2CCC(C2)N1C(c1ccc(C#N)o1)=O N1(C(C2CCOCC2)=O)CCOCC(C(=O)N(C)CC2C(c3onc(C)n3)C2)C1 c1(C(N2CC3C(NC(=O)Cc4cnc[nH]4)(C3)C2)=O)ccc2cccnc2c1F CC1CN(C(=O)CC2CCCO2)CC1(C)C(=O)NCCN1CCCCC1C c1(N2CCC(=O)NCCC2)ncc(S(=O)(=O)NC(CO)C2CC2)cc1Cl c1(C(=O)NCC2C=CC(NC(C(CCCC)O)=O)C2)ccc2c(c1)CCN2C=O C(=O)(C1CCCc2c(O)cccc21)NCC1CN(C(c2cc(C)sn2)=O)CC1O c1(-n2c(C3c4ccc(OC)c(c4)N3)nnn2)cccc([N+](=O)[O-])c1.C1(CO)CC1 N1(C(C2C(C)(C)S(=O)(=O)CC2)=O)CC2CC(NC(c3cc[nH]c3)=O)CC1C2 C1(NC(c2cc(C)no2)=O)CCN(C(C2CCC(=O)C(C)C2)=O)CC12CCC2 c1(C(N2C(C(N3CCCC3)(C)C)CCC2)=O)ccncn1.C1(C2(C(=O)NN)CC2)(CC)CC1 C1(=CC(=O)NCC2(C)N(C(CCSCC(C)C)=O)CCC2)CN2CCC1CC2 Cc1cc(C(=O)NC2(C(N3CCC(c4nn[nH]n4)C3)=O)CCSC2)cc(C)c1 CCC(CC(C)C)C(=O)NC12CC1CN(C(=O)C=Cc1nc(C)c(C)[nH]1)C2 C(=O)(CCCC(=O)NC1CN(C(C2CC2C(N)=O)=O)C(C)(CC)C1)NCC N1(C(=O)Cc2ccc(Br)cn2)CC2CN(Cc3ccccc3I)CC2C1 c1(C(N2CC(F)C(F)C2)=O)ccc(-c2cncc(N3CCCC3)c2)cc1F n1(C(C)C)cnnc1C(=O)NC1(CCC(=O)N(C)Cc2cncs2)CCCC1 C1(CNC(c2c(CC)nco2)=O)(CNC(=O)C(Br)=C(C)C)CC12CCC2 C1(CCNC(c2cocc2C)=O)(NC(C(C2CC2)SC)=O)CCOCC1 C(=O)(C(C(C)C1CC1)N1CCC(CN(C)C)C1)NCCSC C1(C(=O)NCCCNC(c2ccccc2-c2nc[nH]n2)=O)CCc2ccnn2C1 C12(C(NC(=O)CSCC3CCCCO3)C3CC3)CC1CN(C(C13CC(F)(C1)C3)=O)C2 CS(=O)CCC(=O)NC1C=CCN(C(c2cc(COC(C)(C)C)n[nH]2)=O)C1 C1(C(N2CCC(C)(NC(c3ccc(C)cc3)=O)C2)=O)CCS(=O)(=O)C1(C)C C1(N(C2CCCCO2)C(c2cc(COC)[nH]n2)=O)C2CCC1CNC2 C1(NC(c2c(C)ccs2)=O)CN(C(c2c[nH]ccc2=N)=O)CC2(CC2)C1 C=Cc1ccc(C(=O)NCC23CC(NC(c4cnn5cc[nH]c45)=O)(CO2)C3)cc1 N1(C(C)=O)CCN(C(=O)C(C)(C2CC2)N(C(=O)CCCF)C)CC1 c1(C(=O)NC(CNC(c2c(F)ccc(NC)c2)=O)C)oc2c(C)cccc2c1C C(=O)(C1=CCCCCC1)NCC1N(C(C(C)=CC2CC2)=O)CC(F)(F)C1 N1(C2CN(C(C=C(CC)C)=O)C2)C2CCC1CN(C(=O)CSc1nnnn1CC)C2 C1(CCNC(COCCOCC)=O)CCCN(C(c2ccc(C)o2)=O)C1 C1(CC(=O)N(C)CC2CCCC2F)CCN(C(=O)CC2(C)CCCCC2)C1(C)C c1(C(=O)OC)cnc(CNCC(=O)N(c2nnn(C)n2)C)o1 C(=O)(C1CCc2ccccc21)N(C(C)C(N1CCN2CCCCC2C1)=O)CC c1(CC(N2CCC(CNC(C3(COC)CCCCO3)=O)C2)=O)ccccc1Cl C1(CNC(C2C(CC)C2)=O)CC(OC)CN1C(C1CC=CCC1)=O c1(CCCC)nc(C)c(C(=O)N(C2CCC(NC(=O)COC(F)(F)F)CC2)C)s1 Cc1cncc(F)c1C(=O)NCCOC1CCN(C(c2n[nH]c(C)c2C)=O)C1 c1(C(=O)NC(CN(C(=O)CCc2cccc(C)c2)CC)C)c(C)[nH]c(C(=O)OC)c1C c1(N(C(=O)CC2CN(C(=O)CCN3CCOCC3=O)C2)CC)cc(F)c(F)cc1O N1(C(=O)NS(CC)(=O)=O)CCCC(COc2ccccc2I)C1 N1(C(C=CC(C)NC(C2(CC=C)CCC2)=O)=O)CC2(COC(=O)N2C)C1 Cc1cc(C(=O)NCC2CCC2NC(c2cn(C(C)C)cc2C)=O)c(C)c(C)c1 c1(C(=O)NC(CNC(C=C(C)C)=O)C)csc(CS(C)(=O)=O)n1 C1(CC(C)C)CN(C)CC(=O)N1.c1(OC)ncc(Nc2ccccc2)s1 CC(CCNC(c1ccc(-c2cccnc2)cn1)=O)CCNC(=O)C1=CCOC1 c1(-n2ncc(C(=O)NCC(C)(CC)NC(C(CC)O)=O)c2C)ccc(Cl)c(Cl)c1 CC1(C)NC(=O)CC1C(N1CCCC(O)(CCNC(=O)CCc2csnn2)C1)=O c1(C(=O)NC2CC(NC(C(C)NC(N)=O)=O)C2)cc(C(N)=O)cc(F)c1 C1(=O)CC(C)(C(F)(F)F)N1.CC1CN(C(=O)C(C)(C)C)CC(=O)N1 C(CCCC(=O)NCCC(O)CO)NC(c1ccoc1)=O C1(C(=O)NCCC)CCC2(CCN(C(=O)C(CC)OC)CC2)O1 CC(C)CCC(C(=O)N1CCC=C(F)C1)NC(c1cccc(CC#N)c1)=O c1(-c2cn(CC)nc2C(F)(F)F)cnc2ncc(C(=O)Nc3cncc(F)c3)n2c1 CC(C)CCC(F)C(=O)NCCCC1CN(C(c2nccc3cc[nH]c23)=O)C1 S(=O)(=O)(c1cccc(-c2c[nH]nc2C2CC2)c1)N.c1(CN(CC)C)ccc(C)o1 N1(C(C(C2CCOC2)OCC)=O)CC2(C)CC1(C(=O)NCc1ncc(C)cn1)C2 N1(C(c2c(CCC)occ2)=O)CCCC(CC)(NC(=O)C(F)C(C)C)C1 C(c1ccc(C)cn1)=CC(=O)NCCCC(C)(C)NC(C1C(CC)OCC1)=O N1(C(CCC(=O)NC)=O)CCCC2(NC(C34COC(CCO3)C4)=O)CC2C1 C1(C(=O)NCCc2noc(=O)n2C)CCN(C(C2C3CC4C(C3)C24)=O)C12CCC2 CCCC(CC)C(=O)N1CCC=C(CNC(=O)C(C)c2ccsc2)C1 c1(CC(N2CCN(C(C(=O)N(C)C)=O)CC(C)(F)C2)=O)ccc2c(c1)OCCO2 c1(CC(C)C(=O)NCC2CCCN(C(c3ccnnc3O)=O)C2)ccc(Cl)cc1Cl c1(CN(C(c2cccc(C)c2)C)C)cc(F)ccc1O c1(C(N(CC2CCN(C(C3C(C#C)C3)=O)CC2)CC)=O)cccc2c1C(=O)NC2 c1(CC(N2CCC3CN(C(=O)C(F)(F)C4CC4)CC23)=O)ccc([N+](=O)[O-])cc1Cl C1(NC(C(C)=CC)=O)CC2(C1)CN(C(=O)C(C)SCC1CCCO1)C2 N(C1c2ccccc2CC1C)C(C(=O)NCc1cc2cc(C)ncc2cc1)=O C(=O)(C1=CC2CCC1C2)N1CCC(N(C(C2CCNC(=O)C2)=O)CC)CC1 N1(C(Cc2ncn(C)c2)=O)CCCC(CO)(NC(=O)COC2CC=CC2)C1 Cc1c(N)ccc(C(=O)NCCC2CCC(NC(=O)C(C)(C)C(C)(F)F)C2)c1F c1(C(C(=O)NCC2C3CN(C(CC(C)N(C)C)=O)C2C3)(C)C)c(F)cccc1F c1(-c2nc(CC(=O)NCC3N(C(C(CSC)O)=O)CC3)sc2)ccc(C)cc1 c1(N2CC(C)C(C)(C)C2)cccc(S(=O)(=O)N2CCCC(OCCO)C2)n1 N1(C(C2(CCCC)CCC2)=O)CCCC(CNC(c2cc[n+]([O-])cc2)=O)CC1 c1(C(=O)NCCCN(C(=O)CC2CCCC2C)CC)cccnn1 Cc1cc(Cl)ccc1CC(N1CC(CNC(=O)COCc2nccn2C)C(C)C1)=O S(=O)(=O)(c1c(Cl)cc(Br)cc1Cl)N1C2CC(NC(c3cnc[nH]3)=O)CC1CC2 CC1(C)CC(NC(c2cnn[nH]2)=O)CN(C(=O)C(=Cc2c[nH]cn2)F)C1 c1(N2C(C)(C(=O)Nc3c(CC)cccc3F)CC2)ncnc2cc(CC)sc12 C(=O)(CC(C)C(C)(C)NC(c1nc(C)ccc1C)=O)NCc1c(CC)con1 N1(C(c2n(C)ncc2)=O)CCN(C(=O)CN2C(=O)CSC2=S)C(C#N)C1 N1(C(CC(C)(F)F)=O)CC(CNC(c2ccc(C3CCCO3)cc2)=O)C(C)(C)C1 C1(C(N2CC(COC)C2)=O)CN(C(=O)CCc2ccoc2)CC1C1CC1 CC1(C)CC(C(N2CCCC(F)(CNC(C3CCC(=O)N3)=O)C2)=O)CC(C)(C)C1 N1(C(=O)NCc2c(CC)ncs2)CCC(F)(F)C(S(C)(=O)=O)C1 N=c1ncc(C(=O)NCCCC2CN(C(=O)CC3CCCCCO3)CCO2)c[nH]1 N1(C(C2(C)C(C)CN(C(=O)CC3C(=O)NN=C3C)C2)=O)Cc2cccnc2C1 C(=O)(C1=CCCSC1)NC1CN(C(CN(C2CC2)CC)=O)C(C)C1 c1(C(=O)NC2CCN(C(C(CC)(C#N)CC)=O)CC2O)cccc(P(C)(C)=O)c1 C1(C)(C(N2CC(N(C(=O)CC3CC3(Cl)Cl)C)C2)=O)CCc2ccccc2C1 c1(C(=O)NC(CC=C)CNC(=O)C=CCOCC)cc(CC)oc1C c1(C(N2CC3(CC(NC(C(c4ccccc4)C)=O)C3)C2)=O)cc(Cl)c(F)c(Cl)c1 N1(C(Cn2c(C)ccn2)=O)CCC2(NC(=O)C(N3CCSCC3)=O)CC2C1 C#CCCCC(C)C(=O)N1CC(C)C(C)(CNC(=O)CCc2cccnc2)C1 CC(C)(C)CCC(=O)N1CCCC(CNC(c2n[nH]cc2F)=O)C1 CC(C)C(C)(CNC(=O)C#CC1CC1)NC(c1csc(-c2ccccc2F)n1)=O C(=O)(C(C)(O)C(F)(F)F)NC1CCN(C(c2c(OCC)nc(C)cc2)=O)C1 c1(OC)ccc(CC(=O)NC2CCCC2CNC(=O)CCC(C)(C)C)c(F)c1 C=CCC(C)C(=O)N(C1CC(C#N)C1)CC(=O)N(C)C(C)C1CC1 CC1CCC(C(=O)NCc2cc(O)ns2)N(C(C2CNC(=O)N2)=O)C1 N1(C(C(CCC)N(C)C)=O)C(C(=O)NCCNC(=O)NC)C2CC(O)C1C2 CC1(C)CC(O)CCN(C(=O)C(CC2CC2)NC(C2(C(N)=O)CC2)=O)C1 C1(NC(Cc2c(C)nc(C)s2)=O)C(C)CCN(C(=O)COC2CCCC(C)C2)C1C c1(C(=O)NCC(CN(C(=O)C(F)CC2CCC2)C)O)noc2c1CCCC2 c1(NC(C2C3(CN(C(Cc4cn(C)nc4)=O)C3)C2)=O)cc2ccccc2cc1O C1(C(=O)NC2CC(CNC(CCc3n(C)ccc3)=O)C2)CC1C1CCC1 c1(OCCOCC)ccnc(N2CC(OCC3(CO)CC3)CC2C(C)C)n1 c1(C(=O)NC2C(CNC(=O)C=CC=C(Cl)Cl)CC2)cc2nc[nH]c2cc1F c1(C(=O)NCC)ccc(=O)n(C2CC(NC(C3(CC)COC3)=O)C2)c1.S(C)(=O)(=O)N C1(NC(c2cncc(SC)c2)=O)CC(CNC(c2nn(C)cc2Cl)=O)C12CCC2 C(CS(=O)(=O)CC(=O)N(CCCOCCNC(=O)C(F)(F)C1CCCC1)C)OC C(CCNC(=O)C(CN(C)CC)Nc1ccccc1)(C(C)C)NC(C=CC(C)C)=O C1(CNC(C(=O)NC(c2ncnn2C)C)=O)CCC2(CCCC2)O1 n1(CC(N2C(CNC(COC)=O)C=CC2)=O)c(C(C)C)nc2ccccc12 CC1CCCN(C(=O)C(c2cccs2)NC(c2ncn3c2CCC3)=O)CC1 c1(OC)nc(C)ncc1C(=O)NCCC1CN(C(=O)CCc2cn(C)nn2)C1 c1(Cc2n(CC)c(N3CCC4CC4C3)nn2)ccc([N+](=O)[O-])cc1 c1(CC(N2C(CNC(C3C(CC)C3)=O)C=CC2)=O)c(C(=O)OC)c[nH]c1C N1(C(CC)=O)CCC(C(F)CNC(C2CCCN2C)=O)CC1 C1(OC)C2CN(C(=O)Cn3cc(C(c4ccc(F)cc4)O)nn3)CC12 c1(CC(=O)NC2CC2NC(C2CCCC23CC3)=O)ccccc1-c1ccccc1 CC1CCC=C1C(=O)NC1CC2(C1)CC2C(=O)NCCc1ccns1 C1(CC)(CC)CC(NC(=O)C(C)COC)CN1C(=O)CC(C)(C)OC CC1C(=O)N(CC(=O)NC23CCN(C(=O)CCc4cn[nH]c4)CC2C3)C(=O)C1C C1(C(N(C)CC2(O)CCOC2)=O)CN(C(=O)CCS(C)(=O)=O)CC(C)(C)C1 c1(N(CCOC)CCN(C)C)ncnc2sc(C(=O)N(C(C)C(C)C)C)c(C)c12 N1(C(C(c2cccc(OC)c2)C)=O)CCCC(C2CN(C(=O)CC(C)OC)C2)C1 c1(C(=O)OC)ccc(C(N2CCC(N(C(=O)C(C)N(C)C)C)C2)=O)c(F)c1 CC1CN(C(=O)C(C2CCOCC2)O)CCN1C(=O)C=CC1CCCN1C n1(CC(=O)NCC2C(CNC(C(n3ncc(C)c3)C)=O)C2)ncn(C)c1=O c1(C(=O)NCC(C2CCC2)NC(=O)CNC(c2ccco2)=O)ncc(Cl)cc1F C(c1ccc(C)cc1C)=CC(=O)NC1(CO)CCN(C(C=CCC)=O)C1 C1(NC(CCc2scc(C)n2)=O)CCC2CC1CN2C(C1CC(C)N(C)C1)=O C1(CNC(C2(C#N)CCC2)=O)CC(NC(c2cncc(F)c2Cl)=O)C12CCC2 c1(CN(C2CCN(S(C)(=O)=O)C2)C(C)=O)cccc(Cl)c1F.C12C3CN(CC13)C2 c1(C(C)=O)cccc(OCC(N2CCC(NC(=O)C(C)(C)C3CCCO3)C2)=O)c1 Cn1ncc(N)c1C(=O)N(CCNC(=O)C(C1CCCO1)C1CCC1)C1CC1 c1(C(=O)NCCNC(=O)C(=O)NCC2CCOC2C2CC2)ccc(F)cc1F C(CC(N)=O)(C(=O)NC(C)C(C)(C)CO)NC(c1c(CC)cno1)=O N1(C(C2CCC(CC)O2)=O)CC(NC(=O)COc2cccc(F)c2)C(C)C1 CC(C(=O)N1CCCC(CNC(=O)Cn2nnnc2C2CC2)C1)P(C)(C)=O C1(NC(C2C3CCN(C(C4(O)CCOCC4)=O)CC23)=O)CC(C2CCCC2)C1 c1(C(N2CCCC(C)(CNC(C3(CO)CC3)=O)C2)=O)c(F)ccc2n[nH]cc12 C1(C(=O)NC(C)CCc2cn[nH]c2)CN(C(=O)COC(C)=O)CCC1(C)C C1(C)(C(=O)NCCCOCCN(C(C2C(CC)CCCC2)=O)C)CCC2CC2C1 C#Cc1ccc(C(=O)NCCCN(C(=O)CC2CCC(=O)NC2)C2CC2)nc1 N1(C(C2N(C(c3ccc(COC)cc3)=O)CC3CC32)=O)CC2C(C1)C2(C)C C=CC1(CC(=O)NCCCCN(C)C(C2CCCC(C)CC2)=O)CCCCC1 c1(OCCC)ccc(CCC(=O)NCC2CCN2C(C2CC(F)C2)=O)cc1 c1(CNC(C2(CNC(C(C)n3cncn3)=O)CCC2)=O)ccc(F)cn1 N1(C(c2cnn(C(C)C)n2)=O)CCC2C(CCCN2C(=O)CCP(C)(C)=O)C1 N1(C(C(C)(C)n2cnnn2)=O)CCC(C(=O)NC2C(C(=O)OC(C)(C)C)C2)=C(F)C1 Cc1ccc(F)c(C(=O)N(C)CC2CCN(C(c3cn(C)c(=O)cn3)=O)C2)c1 c1(C(N2CC(NC(C(C)CO)=O)C(c3cnn(C)c3)C2)=O)ccn2ccnc2n1 C#CCCCCCC(=O)N1CCCC(CC(N2CCSCC2C2CCC2)=O)CC1 c1(C(=O)NC(c2cc(C)sc2)C)ncc(CO)cn1 Cc1ccc(S(=O)(=O)N2CCC(CN(C)C)CC2)cc1C.N12CCCCC1C2=O CN1CCN(C(=O)CC2CCOC2(C)C)C(CNC(=O)CSCC(N)=O)C1 c1(C(N2CCC(c3cn(CCNC(C(C)C)=O)nn3)C2)=O)cnc(O)nc1O CC1(O)CC(C(=O)N(C2CCN(C(=O)CC3CC(F)C3)C2)CCO)C1 N1(C(Cc2cc(C)cc(F)c2)=O)CCC2CN(C(c3n[nH]cc3C)=O)CC12 C(=O)(CCC(F)(F)F)NC1(C(N(C)CCc2cccnc2)=O)CCC1 N1(C(c2cn(C)nc2C(C)(C)C)=O)C2CCC1C(NC(=O)C1CC1)C2 c1(C(N2C(SC3(C(=O)Nc4cn(C)nc4)CC3)CCC2)=O)cc2n(n1)CCCO2 Cc1cnn(C(C)C)c1C(=O)NCC1CN(C(C2CCCC2(F)F)=O)CC1O Cc1nn(C)c(C)c1C(=O)NCC1COCC1NC(=O)Cc1cc(F)ccc1O n1(CC(N2CC(N(C(C3(CCC)CC3)=O)C)C2)=O)cnccc1=O c1(C(=O)NCC2CN(C(CCc3cc(C)no3)=O)C(C)C2)ccc(Cl)c(N)c1 C1(C(N2CC(c3cc(C4CC4)nn3C)C2)C)CC(C2CCC2)C1 C1(CC)(NC(=O)Cn2cccc(N)c2=O)CCCN(C(C23CCC2CC3)=O)C1 c1nc(O)n[nH]1.CC(C(=O)NC1(CO)CCC1)N1CCCC1.C1=CCNC1=O c1(OC)cc(C(=O)N(C(CNC(=O)C(N2CCC(C)C2)=O)C2CC2)C)cc(C)n1 c1(C(=O)NC2(CC)CN(C(c3csnc3OC)=O)C2)cc(C)c(F)c(C)c1 Cc1cc(C)c(C(N2CCN(Cc3cccc(Cl)c3Cl)CC2C)=O)cc1Br C1(NC(c2cncc(OCCOC)c2)=O)CC2CC1N(C(=O)C(CC)CC)C2 C1(NC(=O)C2=C(Cl)CC2)CC2CC1CN2C(c1cc(C(F)F)ccc1Cl)=O N1(C(C2(C)CN(C)C(=O)CC2)=O)CC2CC(F)(F)CCC2(NC(=O)C=CCO)C1 C1(c2nnnn2CCCSC)(NCc2cnc(CC)o2)CCOCC1C C1(CC)CN(C(=O)CC2OCCO2)CC1C(=O)NCC(C)(CC)CC CCCC(O)C(=O)NC1(COC)CCN(C(c2ccnc(-c3ncc[nH]3)c2)=O)C1 Cn1cnc(CNC(c2nnnn2C2CCCCC2)(C2COC(=O)C2)C)n1 CC1CCc2nc(C(C)Nc3ncccc3N3CCCCC3)c(C#N)cc2C1 S(=O)(=O)(c1csc(C(=O)NC2(C)CC(NC(=O)CC(C)OC)C2)c1)NC C1(NC(=O)Cn2cnc([N+](=O)[O-])n2)COC2CN(C(C3CC=CCC3)=O)CC12 C#CCC1(C)C(=O)N1.C1(NC(C2CCCC2OC)=O)CN(C)C(=O)C12CC2 N1(C(c2c(CC)ncs2)=O)CC2CN(C(C)C(=O)Nc3cccs3)CC2C1 C1(CCC)CCCC1CNC(C1CCN(C(c2cccs2)=O)C1)=O CCC(CC(=O)N1CCN(C(=O)CCC=CC(C)C)C(CC2CC2)C1)C(F)F c1(CNC(=O)NCC2C(C)(C)CO2)c[nH]c2cnccc12 C=CC1CCCN(C(=O)CCC(Cc2ccccc2)N2CCCC2COC(C)=O)C1 C1(N(C(CCNC(=O)NC)=O)CC(C)C)CCN(C(C2CCC(C)C2C)=O)CC1 N1(C(c2c[nH]c(=N)s2)=O)C2CCC1CC(NC(c1cccc[n+]1[O-])=O)C2 C1(NC(CC2CC(SC)C2)=O)CC2(C1)CC2NC(c1cc(C)no1)=O Cc1cnn(C)c1CC(=O)NC1CN(C(c2coc(C(F)F)c2)=O)CC1O N1(C(C(C(C)C)NC(C)=O)=O)CCN(C(=O)CCc2ccc(Cl)nc2)CC1C N1(C(C2CCCCC2)=O)CCCC(Cn2cc(CN3CCOCC3)nn2)C1 c1(NC(c2nc(CC)sc2)c2nnnn2Cc2nnn(C)n2)ncc(C)cc1Br CC1CCc2ccccc2N1CCNc1cn(C)nn1.C1(C(=O)CCC)CCCO1.C(C)(C)(C)O C12(C(=O)NCC3C(NC(C4(C5CCC5)CC4)=O)C3)CCCC1OCC2 C1(C(=O)NCCC)CN(C(c2cccc(-c3cccc(Br)c3)c2)=O)CC1(C)C C1(O)(C(C)OCCCNC(CN(CC#C)C(C2CSC2)=O)=O)CCC1 C(=O)(C1=CCc2ccccc21)NCCC1N(C(CCC(C)N(C)C)=O)CCOC1 c1(NC)cnc(C(=O)NCC2(C(=O)NC3CCCC3CCO)CCC2)cn1 C1(C(=O)NCc2occ(C(N(CCCC)C(C)CC)=O)n2)CCC2(CCC2)C1 c1(CC)[nH]nc(Cl)c1C(=O)NC1CCCN1C(=O)C(C(C)O)N(C1CC1)CC c1(CC(=O)N(C)CC2N(C(C(C(C)C)SC)=O)CCCC2)cccc2c1OCO2 S(=O)(=O)(c1cc(C(=O)NCc2csc(CCN)n2)ccc1Cl)CN(C)C S(=O)(=O)(c1c[nH]c(C(=O)N(C)C)c1)NC(C1CCN(c2ccccc2Cl)C1)C c1(CNC(=O)NCCCC2CCCCC2O)n[nH]c2c(F)cccc12 N1(C(c2cncc(CC)c2)=O)CCCC(CC)(NC(c2cc(Cl)ccc2O)=O)C1 C1(CCC(=O)NCCO)CCCCC1.C(=O)(C(F)(F)c1ncccn1)CCN(C)CC C1(C(=O)NC(CC(=O)NCCNC(C)=O)CC2CC2)CCCCC(=O)N1 C1(NC(=O)COCC2CC2)CCN(C(C23C(=O)C4CC2C3C4)=O)CC1F C(=O)(C1=NNC(=O)C1)NC1CCN(C(c2c(CC)nc(C3CC3)[nH]2)=O)C1 C1(CC)CCC(C)CN1C(C1(CNC(=O)Cc2cc[nH]c2)CC(C)(C)C1)=O C(=O)(CCCCN(C(=O)CC1CC1CC)C)NCCCOCC C1(O)(C(N(C(CC(N2CCC(N(C)CC)C2)=O)C)C)=O)CCCCC1 C=CCCCC(C)(C)C(=O)N1CC(C2(NC(=O)C(C)CC(=O)OCC)CC2)C1 C(=O)(C(F)CC(C)C)N1CCC(CCNC(CCN2CCN(CC)CC2)=O)C1 C1(C(=O)NCC2(O)CN(C(=O)C(O)CCc3ccccn3)C2)C(F)(F)C12CCC2 C1(CC(=O)NCC2CCC(C(=O)NCc3c(C)ccs3)C2)CC(=O)NC1=O Cc1onc(-c2nc(C(C)C3CC3)nn2C2CCCC2)c1I C(=O)(C(C(C)(C)C)OC(c1cc(-c2ccnc(OC)c2F)ccn1)=O)OC N1(C(c2nn(CC)c(C)c2)=O)CCN(C(=O)Cn2cc(Br)c(=N)[nH]2)C(C)C1C CC(C)C(O)C(C)(C)C(=O)NC1CN(C(=O)CN2CCCCC2)CC1C C(=O)(C1Cc2ccccc21)N(CCCNC(C1(C)ON=C(CC)C1)=O)C1CC1 c1(CCC(=O)N(C2CCN(C(=O)CN3CC(C)(C)C3)C2)CCC)ccccc1C N1(C(C(N)=O)=O)CCC(O)(CNC(=O)C(C2CCCCC2)NS(C)(=O)=O)C1 Cc1ccc(C(=O)NC2CCN(C(c3cn(C)nn3)=O)CC2C)c(C)n1 CCC(C)C(O)C(=O)N1CC(O)(C(C)NC(=O)CNC(=O)Nc2ccccc2)C1 Cc1cc(C(=O)NC23CC(CO2)N(C(=O)CC2C(=O)NN=C2C)C3)c(C)c(C)c1 c1(SCC)cc(C(=O)NC2CSC(C)C2)ccn1 CCC(O)C(F)(F)C(=O)N1CCCC(CC(=O)NC2CCN(C(C)C)CC2)CC1 Cc1nnc2n1CCC2(C)C(=O)N1CC(NC(c2ccc(C#N)[nH]2)=O)C(F)C1 Cc1ccc(OCC(=O)N(CCNC(c2c(C)nn(C)c2N)=O)C2CC2)c(C)c1 C1(C(C(=O)OCCC2CC2C(F)(F)F)F)CCOCC1 c1(CC)cc(C(N2CCCCC2C2CCN(C(=O)C(C)(C)CO)CC2)=O)ccn1 CC1OCCN(C(=O)CC2(C)CCN(C(c3cc(Cl)no3)=O)C2)C1 C1(C(=O)OCC)(NC(c2ccc[nH]2)C)CC(CO)C1 Cc1cc(CN2CCCCC2CNC(=O)Cn2nnc(=O)[nH]2)ccc1C(F)(F)F N1(C(CC2N(C(COC3(C)CCC3)=O)C3C2CCC3)=O)CC2CC(O)CC2C1 Cc1cc(N2CCC(O)C2)ccn1.c12ccccc1C(=O)N2C1CC2CNC1C2 c1(C(=O)NC2CCN(CC(=O)Nc3cccc(F)c3)CC2)ccc(C(F)F)nc1 C(=O)(CC(C)C(C)(C)NC(c1ccnc(C)n1)=O)N1CCC(O)(COC)C1 c1(CC2(O)CCCC2(C)C)ccc(P(C)(C)=O)s1.Cn1cc2c(n1)NC2=O C12(CNC(=O)C(F)CC3CC3)COC(CNC(c3cccc(C(F)F)c3)=O)(C1)C2 c1(C(N2C(C)CCC(NC(=O)C(F)(F)CC3CC3)C2)=O)ccc2oc(O)nc2n1 CC1C(NC(c2ccc(O)cn2)=O)C(C)CCN1C(c1cncc(Cl)c1)=O CCC(CC)(CCC(=O)OC)NC(C1OCCOC1C)=O Cc1ncn(C)c(=O)c1C(=O)NCC(C1CC1)N(C)C(C1CC(C)N(C)C1)=O C1(CNC(C2C3CC2N(C(C2CC4CCC4C2)=O)C3)=O)(CO)CC2CC2C1 CC(C)CC(O)C(=O)NC1CCCC1N1CCN(C(c2occc2Cl)=O)CC1 CC(C)C(C#N)C(=O)NCC=CC(=O)NC(c1ccco1)C N1(C(CCC)=O)CCCC(C)(NC(c2ccnc(OC)c2)=O)C1 C(C1C(C(=O)N(C(C)CCNC(=O)CC2CC=CCN2C)C)C1(C)C)=C(C)C C1(C(=O)NCCN2CCN(C(C3C(CC)C3)=O)CC2)CCn2nnnc2C1 C(C1CCCCCC1)=CC(=O)NC1(CN(C(=O)CC2CCCC23CC3)C)CC1 C1(NC(c2c(C)ncnc2C)=O)COC2CN(C(C3CC4(CCOC4)C3)=O)CC12 C(=O)(C(CC)CC(F)(F)F)NC(CC)CNC(=O)C(C)Cc1ccccc1Cl CN(S(=O)(=O)N=S(C)(=O)C(C)(C)C)Cc1cccs1 N1(C(c2n(C)ncc2N)=O)CCC(NC(=O)C=CC(F)(F)F)CC1c1ccccc1 c1(C(=O)NC(C2CCCN(C(CNC(=O)NC)=O)C2)C)ccc2n[nH]c(C)c2c1 c1(CC(C)NC(C23C(CN(C(C)=O)C2)C3)=O)cc(F)cc(F)c1 c1(CN2CCN(CCCNC(CC(C)(C)C)=O)CC2)c[nH]c2cccc(Cl)c12 c1(CCC(=O)N(C2CCN(C(C3CC4CC4C3)=O)C2)CC)scnc1C C1(C(N(CCSC)CC)=O)CC(C)CCN1C(c1cc(C)[nH]c1C)=O N1(C(CC2CCC(=O)N2)=O)CC2(CNC(c3ccc(F)cn3)=O)CC1CCO2 N1(C(C(C2CCCC2)OC)=O)CCOCC(CNC(C2CCCC(C#N)C2)=O)C1 C1(CCNC(C(=O)NCC(C(C)C)C(=O)O)=O)COCC2(CCC2)O1 C(=O)(C(O)C(F)(F)F)N1CC(NC(=O)CCOCCCCC2CCCC2)C1 c1(C(N2CCC(C(C)C(=O)NC3CC4(CCC4)C3)C2)=O)ccc2ccoc2c1 C(CO)(C(C)(C)CO)NCCn1ccc(COC(c2n[nH]c(C)c2Cl)=O)n1 C1(C(N(CCN(C(C(C)=C(CC)C)=O)C(C)C)C)=O)CCCCC1F c1(C(=O)NC(C)CNC(C2(C3(C)OCCO3)CC2)=O)ccc2nc(O)[nH]c2c1 C1(C(=O)NCCCC(CCC)NC(=O)CCCCF)CCS(=O)(=O)C1(C)C CC1(C)C(C(N2CC(F)CC2CNC(C2(O)CCC2)=O)=O)CCS1(=O)=O C=CCC(CC(C)C)C(=O)NC1CCCC1NC(c1cnc(C(=O)OC)s1)=O C1(NC(C(C#C)(C)C)=O)CN(C(C2CC23CCOCC3)=O)C2(CCOCC2)C1 C1(OC)CC(CC(=O)NC2C3CC2N(C(c2cocc2C)=O)C3)C1(C)C C(=O)(CC(F)(F)C(F)F)NC(CNC(c1ccc(CC)cc1N)=O)(C)CC(C)C n1(C(C)C=O)c(=O)c(F)cc2ccccc12.C1CC(=O)NC1=O C1(CC(=O)NCCC(C)NC(=O)C(C)N(C)C)SC(=N)NC1=O C(=O)(CC1=CCOCC1)NCCC(C)(CC)NC(CC(C=C)(C)C)=O C1(C(=O)NC(c2c(C)noc2C)C)N(C(=O)CC2CCC(=O)C2)CCC1(C)C c1(CCC(N2CCCC(NC(c3ncc(NC)nc3)=O)C2)=O)c(F)cccc1F c1(CC2CC(=O)N2)ccccc1F.C1(C(=O)NC)COCCN1Cc1cccs1.N Cc1csc2ncnc(N(CC(C)CNC(c3nnn(C(C)(C)C)n3)=O)C)c12 c1(NC(C2CCS(=O)C2)=O)cc(Cc2ccco2)[nH]n1 C1(NC(C(C)CC2CCCC2)=O)CC2CCC1N(C(=O)CCCC(C)(C)C)C2 c1(C(N(C2CCN(C(=O)CCCc3nncn3C)C2)C)=O)ccc(C(N)=O)c(Cl)c1 N1(C(C=C(C)C(C)(C)C)=O)CCC(C)C(N(C)C(C2CCC3(CCC3)O2)=O)C1 c1(C(N(C(C)CNC(=O)Cc2cnccc2Cl)C)=O)cc2n(n1)CCN(C)C2 C1(OC)CC(NC(=O)C(F)(F)C(F)F)CN(C(=O)CC(O)c2ccccc2)C1 Cc1cc(CN2CCC(NC(c3c(Br)cnn3C)=O)C2)c(C)cc1Br C(=O)(N=c1ccn(C)[nH]1)C1(NC(c2c(CC)ncs2)=O)CC(O)C1 Cc1ccc(C(=O)N(C)CC2CN(C(=O)CSCC(N)=O)CCO2)c(N)c1 c1(CC(=O)NC(CC(C)C)CNC(c2cnn(CCF)c2)=O)ccc(Cl)cc1Cl O=C1CCCCC(C2CN(C(=O)NC3CC3c3ccncc3)C2)N1 C(=O)(CS(=O)(=O)N1CCOCC1)NCC(C)NCCNC(=O)C(C)(C)F S(=O)(=O)(c1ccc(Br)s1)N1CCN(C(C(=O)NCC2CC2c2cccnc2)=O)CC1 C(C)(CCCCCO)NC(C1(CNC(=O)COC2CCCC2)CC(=C)C1)=O c1(N(CCNC(CN(C(=O)C#CC2CC2)CC#C)=O)CC)ccc(OC)cc1 N1(C(C#CC(C)C)=O)C(CNC(c2c[nH]c(C(N)=O)c2)=O)CC2CCCCC12 Cn1c(C(=O)NC2CC2NC(c2csc3ccccc23)=O)cc2sccc12 N1(C(CCCCCNC(N)=O)=O)CC(NC(C2CC(F)(F)C2)=O)C(C2CC2)C1 c1(C(=O)NCC(C)NC(C(CSC)c2ccccc2)=O)nn(C)c(N)c1C C1(C(N(C2CCN(C(c3sccc3-n3ccnn3)=O)C2)C)=O)CCC(O)C1 c1(C(C)NC(=O)NC(C)(C)C)c[nH]c(=NCCc2ccc(O)nc2)o1 Cn1nnc2cncc(C(=O)NC(C)(CNC(C3NC(=O)C4CC34)=O)CO)c12 C1(c2nnnn2CCC2CC2)(NCCC(C=C)(C)C)CC(C)(C)CCC1C c1(C(N2CCC(N(C(C34CC(C)C3C4)=O)CC3CC3)C2)=O)cccc2sncc12 N1(C(CC(=O)C=O)=O)CCN(C(=O)CCc2nc[nH]n2)C2CCCCC12.CNC c1(OCCN(C(C2CCCN(C(CCCC#C)=O)C2)=O)C)ccc(F)cc1C Cc1cc(Cl)nc(NC(=O)Cc2cccnc2O)n1 c1(OC)cncc(C(=O)NCC2CCCCCN2C(c2n[nH]c(C)c2Cl)=O)c1C c1(CCCOC)ccc(C(N2CC(NC(=O)C(O)CSC)C(F)C2)=O)c(O)n1 C(C)(C(=O)N(C)Cc1cocn1)(C1CCC1)NC(C(C)NC(=O)OC)=O.C1CC1 c1(C(=O)NCCNS(CC)(=O)=O)coc(COC(C(=O)NC2CCCC2)C)c1 C1(CC(=O)NCCC2(O)CN(C(C(C)CN(C)C)=O)C2)CC2(CCC2)CO1 N1(C(C2(CC(C)=O)CC2)=O)CCCC(N(C(C2CCC(C)(C)C2)=O)CC2CC2)C1 Cc1cccc(C(=O)NC(C)(C)C(C)NC(c2ccc(Cl)s2)=O)c1F N1(C(CCc2ccc(C)nc2)=O)CCN(C(c2cc(C)no2)=O)C2CCC12 N1(C(c2cncc(C)n2)=O)CCC(C2CCN(C(C3CCNC3=O)=O)CC2)CC1 S(=O)(=O)(c1cnn2ccc(=NCCC(F)F)[nH]c12)CC(CC(=O)OC)C c1(C2C(C)C2)ccc(C(=O)NC2CC(O)C2c2ccccc2)o1.C1C=CCN1 Cc1ccc(C(C)C(=O)NCCC2CC(NC(C3(N(C)C)CCC3)=O)C2)s1 C(=O)(C1CCc2nccn21)NC(C(=O)Nc1cc(CC)c(C)nc1)C(C)C N1(C(c2cc(CC)n(C)n2)=O)CC(C(F)(F)F)C(C)(C(=O)OC)C1 c1(N2CCCC(C3(C)CCCC3)C2)nccc(=NCCS(=O)CC(F)(F)F)[nH]1 c1(CSCC(=O)N)c(F)cccc1F.c1(N)nnc(-n2cccc2)o1 CCC(C)(C#N)C(=O)NCC1CCCC(CNC(c2cc(CC(C)C)on2)=O)C1 Cc1c(CC(N2CCCC2C2(CNC(=O)C(C)C3CCC3)CC2)=O)cnn1C Cn1cc(N(C(=O)CCCCC2CC2)C(=O)NC2CC2CC(C)(C)C)c(Br)n1 c1(C(N(CC(C)NC(=O)C(N2CCOCC2)C2CCC2)C)=O)ncoc1C1CCC1 C1(C(=O)NC2CC(CCNC(C3OCCN(C)C3)=O)C2)CC12CCSCC2 N1(C(C2(OC)CCSCC2)=O)CCC2(C1)CN(C(=O)CC1CC(C)OC1C)C2 c1(OC)ccc(Cl)c(CN2CCCC(CNC(c3sccc3I)=O)C2)c1F C(=O)(C(CC(C)CC)NC(=O)CCc1cnccn1)NC(CC#CC)CO C12(C(=O)NCCCN(C(COC)C(C)C)C3CC3)CCCC(CO1)C2 CCCCCCC(C)(CC)C(=O)N1CCCC(CCNC(=O)CN(C)CCC)C1 c1(OC)ccsc1S(=O)(=O)C(=O)NCC1(c2ccccc2F)CC1 CC1(C)CC(NC(=O)C(=O)NCC2(O)CCSC2)C(C)(C)O1 C1(CC(N2CCCN(CCc3c(C)noc3C)CC2)=O)CNC2CCCCC12 C(=O)(C1=NOC(C)C1)N1C(C(C)NC(CSCCOC)=O)CCC1 C1(C(N2CC(Cc3ncc[nH]3)C2)=O)CN(C(C2C(CC)C2)=O)CCO1 c1(C(=O)NC2CC(C)(CNC(C(CC)CC)=O)C2)c(OC)cc(OC)cc1OC CC(CN(C)C)CCC(=O)NC1CC1CNC(c1ccncc1)=O C(=O)(N1CCC(C(=O)N(C(C)C(=O)OC)C)O1)NC(CC(=C)C)=O C1(C(=O)NCc2cccs2)COCCN1Cc1cccc(O)c1 N1(C(C(N2CCNC2=O)C)=O)CCC(CCNC(C2CNC(=O)O2)=O)CC1 CC1(C)CCCCCN1C(=O)CN1CCN(C(=O)Nc2ccccc2)CC1 c1(NCc2cnn(C3CC3)c2)ncnc2occc12.C12CCC(CC1)C(=O)NC2 C1(C(=O)NCCN(C(C=C(C)C(F)F)=O)C(C)C)CCCS(=O)(=O)C1 N1(C(C(COCC)NC(=O)Cn2nccn2)=O)CCCC(C)(CC)C1 C1(CC)C(C(=O)NCC(C(C)(C)C)NC(=O)CCSc2n[nH]c(C)n2)CCN1C N1(Cc2c(F)c(Br)cc(OC)c2F)CCC2(CC(C(=O)NCCCCl)=NO2)C1 CCC(C)CC(C(=O)NCCCSC(F)F)NC(c1cccc(OC)n1)=O c1(N(C(C=C(C)C)=O)CCN(C(=O)CC(C)O)CCCCN(C)C)ccccc1 CC1(C(=O)NCCCCNC(C23CC2COC32CCC2)=O)CCC(F)(F)CC1 C=CC(C)(CC)C(=O)NCCC12CCC1CN(C(C13CCC(CC1)OC3)=O)C2 c1(C(N(CC(N2C(CC)COCC2)=O)CC2CC2)=O)cc(C)c(N)cn1 c1(C(=O)NC(C2(C(=O)NCCc3cccc(O)n3)CC2)C)nccn2ccnc12 C(=O)(CC(C)C(C)(C)C)N.C#CCCCCC(=O)N1CC(C2CCC(C)(C)CC2)C1 c1(CN2CCC(CNC(=O)Cc3cnccc3Cl)C2)ccc(O)c([N+](=O)[O-])c1 c1(OC)ccc2onc(CC(N3CCC(C)(NC(c4cscn4)=O)CC3)=O)c2c1 C1(C(N2CC(C(C(=O)NCC(CCC)OC)OC)C2)=O)OCC2CCCCC12 Cc1cccc(C(=O)NC(C2CCCN(C(c3ccc(C(C)(C)C)o3)=O)C2)C)n1 C1(C(=O)NCC2(C#C)CCC2)CC(CC)CCN1C(C1CCC(=O)NC1)=O CC1(C(=O)NCC2CCC(C(=O)NCc3cccnc3F)O2)CNC(=O)C1 C(CCCC(=O)NCC(Cc1ccccc1)NC(C1CCNC(=O)C1)=O)SC c1(C2(NC(CCN(C(=O)C(C3CCOC3)SCC)CC#C)=O)CC2)cccnc1Cl c1(-n2ncc(C(=O)NC(C(C)NC(CSCC=C)=O)CO)c2)nc(C)cc(C)n1 C(C(N=[N+]=[N-])C(=O)NCC1CCN(C)C1=O)OCC.C1=CCN(C)C(=O)C1 N1(C(=O)C=Cc2ccncc2)CC(F)(F)CC1C(N1CCC2(CCC2)C1)=O c1(C(=O)NCC(CC(=O)Nc2nc(C)c(C)s2)O)cccc2cc[nH]c12 c1(COC(C(n2ccnc2C2OCCC2C)C)=O)cccc(CO)c1 C#CC(C)CN=C(NCC(C)(C)C)NC1CCCCC1 N1(C(C(C#C)(C)C)=O)CC2CN(C(=O)C=Cc3cccnc3)CC2(C)C1 CC1OCCN(C(=O)C(C2CC3(CCC3)C2)NC(c2cnsn2)=O)C1CO C1(C(=O)NC2C(CC)CCC2)CCCCCCN1C(C1(C(=O)NC)CC1)=O C1(CNC(c2nc(C)oc2)=O)C2CCCC2N1C(c1ccnnc1)=O C(=O)(C1=NN(CC)C(=O)CC1)NCC(CC=C)NC(=O)CCc1c(C)noc1Cl C(=O)(C1=NOC2(CCC2)C1)NCCOCCNC(CCCc1ccc(C#C)cc1)=O C1(C(=O)NCC2C(CC)C2(F)F)(NC(c2cc(O)cc(F)c2)=O)CCC(C)(C)C1 c1(C(=O)OC)c(NC(C2C3CC2N(C(c2csc(Br)c2)=O)C3)=O)sc(C)c1C Cc1cc(C(N2CCCC2CF)C(=O)NCCOCC2CC2)n[nH]1 C1(CNC(Cc2nc(COC)sc2)=O)C(C)CCN1C(c1csnc1Cl)=O C1(C(N(C2CC(C#N)C2)CC(N2CCC(c3ncco3)C2)=O)=O)CCC(C2CC2)C1 c1(CC(=O)NCC(N(C)C(C2CCCC2(F)F)=O)C2CC2)nsc2ccccc12 Cc1conc1C(=O)NCCC(C)NC(=O)CC1(O)CCC1 c1(OC)cnnc(C(N2CCC2C(=O)NCCC2CCC(C)(C)O2)=O)c1 CC(CCN(C)C)N=c1[nH]c(N2CCC(C(F)F)CC2)nc2ccccc12 c1(CN(C2CCCC2)CC(C)C)ccc2c(c1)CCC2(C)C CCC(CCC(=O)N(CCCC(O)CO)C)NC(c1cn(C)c(=O)cn1)=O C(CC1=CCN(C(C2CC(F)C(=O)N2)=O)CC1)NC(=O)CC1CCCCO1 N1(C(C)C)CCCC(C)(C(=O)O)C1.c12ncoc1CN2 c1(C(N(CCN(C(=O)CC2CCCCC2C)CC)CC)=O)nnn(C)c1C C1(N(C)C(C2CCC(OS(C)(=O)=O)CC2)=O)COCCN(C(=O)C(N)=O)C1 c1(OC)cc(Cl)ccc1C(=O)NC1(C)CCN(c2ncc(Br)cn2)C1 N1(C(c2cc(C(CC)CC)no2)=O)CCOCC(NC(C2CC(CC)C2)=O)C1 CC1(C)CN(C(=O)CC23CCCC2C3)CC(CNC(=O)CCC(N)=O)O1 Cc1cccc(C(=O)NCC2CC2CNC(C2CN(C)CC2C)=O)c1O C(=O)(C(F)C(C)CNC(=O)C(C)COC)NCCOCC#C c1(C(C(=O)NCC2(F)CN(C(C(CC)F)=O)C2)(F)F)ccc(OC)c(OC)c1 c1(C(C)N(C)CCNC(=O)NCC2COCCN2C)cccc(C#N)c1 C(C(O)C(CC)CC)NC(CC1(N(C(c2c(CC)cncc2)=O)C)CC1)=O C1(CC)CN(C(c2cc(Cl)cnc2O)=O)CCC1NC(=O)Cc1ccoc1C CC1(C)CC(CNC(c2ccc(F)cc2F)=O)N(C(C2CCCCS2)=O)C1 C1(CNC(C(F)=CCC)=O)N(C(c2ccnn2CCC)=O)CCC1(C)C N1(CC2(C)CCC2)C(=O)CCN(Cc2cccc(-c3ccccc3)c2)C1=O C1(NC(NC(CC)CC)=NCC2CCN(C)C(=O)C2)CCN2CCC1(C)C2 CCCCC(CNC(C1CCCN(CCC)C1)=O)NC(=O)CCc1cnn(C)c1 C1(NC(C2C(OCC)CC2)=O)C2CCCN(C(=O)CCP(C)(C)=O)C2C1(C)C c1(OC)ccc(-c2ccc(O)c(C)c2)cc1CN(C=O)CC1CN2CCC1CC2 C1(C(N2CCC(c3ccncc3)C2)=O)COCCN1C1CNC1.c12csc(n1)C2 C(C(=O)N(C)CCC1CN(C)C1)(C(C)(C)C)NC(c1c(C)nco1)=O C1(C(N2CC(O)C2)=O)CN(C(=O)C(O)c2ccsc2)CCC1O C1(CC)CN(C(c2ccn(CCNC(C3C4CC(=O)CC34)=O)c2)=O)CC1O c1(C(C(=O)NCC2CC(CNC(C(CSC)OC)=O)C2)C)ccc(F)cc1 N1(C(c2ccn(C)c2)=O)CCC(C(N2CCCCC(F)(F)C2)=O)C(C)(C)C1 C1(O)(CNC(C(C)Cc2ccccc2Cl)=O)CCCN(C(C2OCCCO2)=O)C1 C1(CN(C(CC2C(CC)C2(F)F)=O)CC)CCN(C(=O)C(C)(O)COC)CC1 c1(C(N2CCC(O)(CNC(C3CC(C)(C)C3)=O)C2)=O)c(Cl)ccc(F)c1F Cc1ccc(O)c(CC(=O)N(CCC(C)(C)NC(=O)Cc2ccon2)C)c1 CCCCC(C(=O)N(C)CC1CCSC1)NC(=O)C(SC)SC C1(=O)C(C(C)C)NC2N(CC2)C(C)N1.C1(CNC(N)=O)CCCOCC1 Cc1nn(CCN(C2CCCCC2)C)c(C)c1S(=O)(=O)N(C)C C1(CC(N2C(C(=O)NC(C#C)(C)C)CC2)=O)CCC(C)(C)O1 CC(C)C(C)C(=O)N(CCCN(C(=O)C(C)OC1COC1)C)C c1(OC)cc(C(=O)OCC(c2cccc(Cl)c2)C(F)F)ccc1C#N N1(C(C(C(C)OC)N(C)C)=O)C(CC(=O)NCC(C)(O)CN(C)C)C2CCCC12 C1(CNC(c2n(CC)ncc2Cl)=O)CCC(C)CN1C(c1ocnc1C)=O CC(=O)C(C)CC(C)C(=O)N1CCCCC2(CCC2)C1 c1(C(=O)NC2(C)CN(C(C(C3CCOCC3)C)=O)C2)ccc(N)c(O)c1 N1(C(C(CCC)OCC)=O)CC(NC(C2CC(C#N)C2)=O)CC2(CCOCC2)C1 c1(NC(c2nnnn2CC2CC2)(C)CC2C=CCC2)ccc2c(c1)CCO2 C(=O)(C(N)CC(F)F)NCC1CCC(OC)CC1 C(=O)(C1c2c[nH]nc2CN1C(c1cc2n(n1)CCC2)=O)NC(C1CCCC1)C c1(NC(c2cnn(-c3ccccc3)c2)=O)nccnc1CNC(C1CCCO1)=O Cc1nn(C)c(Cl)c1C=CC(=O)NCCC(O)CNC(=O)C1CC1 c1(C(=O)NC(CC)CNC(=O)CC2CCCCO2)n[nH]c(C)c1C c1(OCC(=O)NC(C(C)NC(Cc2scc(C)c2)=O)CO)cccc(Cl)c1C Cc1cccn(CC(=O)NCCOCCCNC(C23CCC(C2)OC3C)=O)c1=O c1(C(N2CCC(C)(CNC(CC3N(C(C)=O)CCC3)=O)C2)=O)sc(C)c(C)c1C c1(CCC(=O)NC(C)CCN(C(=O)CCc2cnc[nH]2)C)c(F)ccc(Cl)c1F c1(C(N2C(C(N3CCC(C)(CO)C3)=O)CCCC2)=O)ccc(F)c(O)c1 c1(C(=O)NC(CSCC)C(=O)NC23COC(COC)(C2)C3)cncc(C#N)c1 c1(OCC#C)ccc(C(=O)NC2(CNC(C3CCOC(=O)N3)=O)CC2)cc1 C(=O)(C(C)(C)CC)N1CCC(C(C(=O)NC(CC)CSC)C)C1 C(=O)(C(C(C)(C)O)NC(=O)C(C)SCC)NC(CCC)CO c1(C(C)C)ncc(C(=O)NCCNC(c2cnc(C(N)=O)s2)=O)n1C Cc1cc(C)n(Cc2cn(CC=CC3CCCN3C)nn2)n1.N12CCCC(C1)C2 N1(C(c2c(C)cc[nH]2)=O)CCC2CCC(NC(=O)CC3CN4CCC3CC4)C1C2 CC1(C)C(CC(=O)NCCNCC2(O)CN(S(=O)(=O)C(F)(F)F)C2)CC1O c1(C(=O)O)cc(Cl)c(O)c(S(=O)(=O)NC2(CSc3ccc(O)c(O)c3)CC2)c1 C(=O)(C1=CNS(=O)(=O)N=C1C)NC(C1(O)CCN(C(C(CCCC)O)=O)CC1)C CC(C)CC(C(=O)NC1(NC(=O)C(CO)OC)CCN(C)C1)N(C)C C1(C(C)(C)O)(CNC(c2sccc2I)=O)CCCC1 C(C1COc2ccccc21)NC(=O)N(c1ccc([N+](=O)[O-])cc1)CC(O)CO CC1(C)CC(NC=O)C(=O)O1.C12(N)CC1CCN2C(=O)CNC=O CC1=NNC(=O)C1CC(=O)N(C1CN(C(=O)Cc2cccc(Cl)c2)C1)C C1(C(N(C)CC2C3CN(C(c4n(CC)nnc4)=O)CC32)=O)CCc2nnnn2C1 Cc1nc(C(N2CC3CC3(CNC(C3(C#N)CC(C)C3)=O)C2)=O)n(C)n1 c1(OCCCCC)cc(C)c(S(=O)(=O)N2CCCC2(C)CO)c(C)c1 C(=O)(C(C)(C)C(N)=O)N1CC2C(CNC(C(CC)(O)c3cccc(Cl)c3)=O)(C2)C1 C=C1CC2(C1)CC(C(=O)NC(C)CNC(=O)CC1CCNC(=O)C1)C2 c1(OC(C)C)ccc(CCN2CCCC(Nc3ncc(I)cn3)C2)cc1Br Cc1ccn2cc(C(=O)NC3(CNC(=O)C=Cc4cnc[nH]4)CCC3)nc2c1 c12ccc(cc1)[nH]c2=O.C1(N(C(C(=O)N(CCN(C)C)C)=O)C)CCC(C)(C)C1 N1(C(C(CC2CCCC2)NC(C(C=C)OC)=O)=O)CC(=O)NCC1C(C)C c1(CC)ccccc1C(=O)N(C1CCC(NC(c2cn(C)cc2C)=O)CC1)C C(C(C)(C)c1ccncc1)(c1nnnn1C)NC1(c2[nH]ccn2)CCC1 C#CCC(C)C(=O)N1CCCCC1CNC(c1cnn(CCC(C)C)c1CC)=O C1(NC(c2c(CC)cno2)=O)CCCCC1NC(=O)C=Cc1nccn1C C(=O)(C(C)SCC)NC(CN(C(=O)CC1(CO)CC1)CC)C N1(C(c2nc(C(=O)OC)sc2)=O)CCCC(N(C)C(c2oc(CO)cc2C)=O)C1 n1(CC)c(CNC(C2CCCCC2)c2ccncc2)nc2ccccc12 c1(CCC(=O)Nc2cccc(C(=O)Nc3c(C)ncn3C)c2)c(F)cccc1F C1(F)(C(N(CCCCCNC(C2C(C=C)C2)=O)C)=O)CCS(=O)(=O)C1 c1(OCC(=O)NCC2CN(C(C3C(C#N)C3)=O)C2)cc(F)ccc1Br N(C1CN(C(=O)CCP(C)(C)=O)Cc2ccccc21)C(C1(C(N(C)C)=O)CC1)=O c1(C(=O)NCC2(C)CCCN(C(C3C4CCCC34)=O)C2)c[nH]c2nccc(Cl)c12 C1(C(N(c2ccc(O)nc2)C)=O)CC2CC(C1)CN(C(=O)OC(C)(C)C)C2 CP(C)(=O)C(CC(=O)N1CCCC1c1cn(-c2cncc(CO)c2)nn1)C(F)(F)F N1(C(C(CCCC#C)C)=O)CCCC12CCCN(C(c1n[nH]c(=N)s1)=O)C2 N1(C(c2c(C)ocn2)=O)CCC(C(=O)NCC(O)C(C)O)C(O)C1 c1(C(=O)NC(C(C(C)C)NC(C=C(CCC)C)=O)C)sc2ncccc2c1Cl N1(C(COCCSC)=O)CCCC1CCC(C)(C)CNC(=O)CNC(N)=O C1(NC(C(CCCC)O)=O)CS(=O)(=O)C2CN(C(=O)C3=CCOCC3)CC12 c1(C(C(=O)NCc2cc(CCNC(C)=O)on2)O)c(C)cccc1C c1(C(=O)NCC2CCN2C(c2n[nH]c(C3CC3)n2)=O)cc2n(n1)CCCC2O c1(CC(N2CC3CC2CN3C(=O)CC2SC(=N)NC2=O)=O)c(F)cccc1Cl c1(C(=O)NCC2(CNC(C(C)C3CCCO3)=O)CC2)cc(C#N)co1 Cc1c(F)ccc(CNC(=O)NC(c2ccc(I)cn2)C)c1F CCCCC(O)C(C)C(=O)NC1(CC(=O)NC2CCC3(CC2)N=N3)CCCCC1 N1(C2(CC)C(=O)CN(C(=O)OC(C)(C)C)C2)CC(CO)CC12CCOC2 N1(C(CCCSC)=O)CCC(NC(c2cc(Cl)nnc2O)=O)C(C)C1 Cc1ccc(C(N)=O)cc1C(=O)NC1CC(NCCOC(F)(F)F)C1 c1(C(=O)NC2C(C)CCN(C(=O)CN3CCOCC3)C2)ccc(S(C)(=O)=O)cc1 CCCCCCC(C)C(=O)NC(c1ccccc1)C(=O)NC1CC2C(C1)C2(F)F C(=O)(C(C)(O)C(C)C)N(CCn1cc(-c2c(C)ncs2)nn1)C C1(NC(c2c(C)ccs2)=O)CC=C(C(=O)NCC2CCCSC2)C1 C1(CC(C)NC(=O)C(O)CCN(C)C)CCN(C(C2CCCC(F)C2)=O)CC1 C1(CC)CN(Cc2ccc(OC)cc2)C(=O)O1 C(c1cc2ccccc2o1)=CC(=O)NC1CCN(C(=O)Cc2nnc(O)s2)C1 C1(C#N)(CC(N2CC3C(CNC(CCC=C)=O)C3C2)=O)CCOCC1 C1(NC(=O)Cc2cnnc(Cl)c2)CC1C1CCCN(C(=O)CC2CC2)C1 N1(C(c2cncc(C#C)c2)=O)CCOC2(CCN(C(=O)CCC=C)C2)C1 C1(CCC)CN(C(c2ccon2)=O)CCN1C(=O)CC1CC2CCC(C1)C2 C1(C(=O)NCCN(C(C(C)(C)OCC)=O)C)CNC(=O)CC12CCOC2 c1(C(=O)NCC(C)NC(C(C(CC)C)O)=O)ccc2nc[nH]c2n1 N1(C(CCC2(C)CC2)=O)CC2CC(C1)N(C(c1ccc(C#N)[nH]1)=O)C2 CC1CC(CCNC(=O)CCC2CCOC2)CCN1C(=O)C(F)=CC1CC1 C(=O)(C1CCc2ncccc21)NCC1N(C(C(CCC)OCC)=O)C2C(C1)C2 C1(NC(CN2CC(C)C2)=O)C=CCN(C(c2ccnc(C(C)(C)C)n2)=O)C1 CC1CN2CCN1C(C(N1CC(=C(F)CNC(=O)C(O)CC3CC3)C1)=O)C2 CC(C)(CF)C(=O)NC(CNC(c1ccc(-c2ccc(Cl)cc2)[nH]1)=O)C(C)(C)C N(C(=NCC)NC1CCN(C(=O)C(C)(C)C)CC1)C(C#C)CC1CC1 N1(C(CN(C(C(C)C)=O)C)=O)CC2CCC(C(=O)NCCc3ccccn3)(C2)C1 c1(CC)cn2c(n1)CC(C(N1CCC(NC(c3ccc(Br)o3)=O)C(F)C1)=O)CC2 N1(C(=O)OC(C)(C)C)CCCC(F)(CC2CCCCN2CCNc2ccco2)C1 c1(C(N2CC3C(C(=O)Nc4ncc(Br)c(O)n4)C3C2)=O)cc(F)cc2[nH]ccc12 Cn1cc(C(C)(C)C(=O)NC2CN(C(c3n[nH]c(C(C)(C)C)n3)=O)C2)cn1 N1(C(COCC#C)=O)CCC(C#CC(=O)NCC(C)NC(=O)OC)CC1 c1(C(=O)NCCN(C(CN(C(=O)OC)C)=O)C)cnn(C2CCOCC2)c1 C(CN=C(NCc1noc(C2CC2)n1)NCC1(F)CCC1)OC CC1(C)CN(C(=O)C(O)C2CC2)CC1CC(=O)Nc1ccnnc1O N1(C(=O)NCC2N(C(=O)OCC)CCC2)CCNC(=O)c2c(Br)cccc21 C=CCC(CC=C)C(=O)N1CCC(NC(=O)C(COC(C)(C)C)N(C)C)C1(C)C C1(CNC(CC(=O)NCC)=O)CC(C)N(C(=O)C(C2CC2)C2CC2)C1 Cc1[nH]c(C(C)(C)C)cc1C(=O)NC(C)CCCNC(C12CC(C)C1C2)=O Cc1nc(C(C)C)[nH]c(=NC2CCCCN(C(c3cc(C(F)F)[nH]n3)=O)C2)c1Br C1(O)(C(C(=O)N(C(C)CO)C)NC(=O)CP(C)(C)=O)CCCCC1 CC(C)C(C)(C)C(=O)NC12CC1CN(C(C1CC1Sc1ccccc1)=O)C2 C(=O)(CC(C)(C)C(F)(F)F)N1CCC(C(C)NC(CCNC(=O)NC)=O)CC1 c1(C(C)=O)ccc(C(=O)NCC(C2CC2)N(C(=O)C(C)c2ccco2)C)nn1 CCCCCC(=O)NC(C(=O)NC1CC(CC(=O)NCCOC)C1)C1CCCC1 c1(C(CNC(=O)C=CC(C)C)NC(COCCCC)=O)cccc(Cl)c1 c1(C(N(C2CN(C(c3ccc(Cl)cc3N)=O)CC2O)C)=O)[nH]cc2c1CCC2 O=C(C1=NOC2(CCOC2)C1)N1CCN(C(C2(n3cccn3)CC2)=O)CC(O)C1 C=CCCC(N=c1cc(C)[nH]c(=NCC(COC)OC)[nH]1)C1CC1 C1(C(=O)NCCN(C(C2N(C(=O)NC)CCC2)=O)C2CC2)CNC(=O)C(C)(C)C1 c1(C(=O)NCCC2(CNC(C3C=CC(CC)C3)=O)CC2)ccnc(N(C)C)c1 C1(CC(=O)NCC(F)(F)CO)CCC(NC(=O)CC2CCCOC2)CC1 CC(C)C(C)(O)C(=O)NCCC(C)CCNC(c1ccc(C2CCOC2)cc1)=O N1(c2cc(C)ncn2)CCCC(C)(CNC(=O)Cc2coc(C(F)F)n2)C1 CC1(C)CC(NC(=O)OC(C)(C)C)CN(C(C23COCC2C3)=O)C1.C12CN(C1)C2=O N1(C(CCc2cc(C)no2)=O)CC=C(CNC(C2CCS(=O)(=O)C2)=O)CC1 CC1CCC(CO)N(C(c2coc(Br)n2)=O)C1 N1(C(CCCC(N)=O)=O)CCCC(C2CCN(C(=O)CC3(C(F)(F)F)CC3)C2)C1 c1(CC(CC)NC(=O)C(C2CCOC2)NC(=O)CSC)cnn(C)c1O N1(C(C(C)N(C)C)=O)CCOC2CN(C(c3cnn(C)c3N)=O)CC12 N1(C(=O)COC2CCC2)CCCC2C1CCN2C(c1c[nH]c2nc(F)ccc12)=O C(C)(C(C(=O)N(C)CCOCCO)C(C)C)NC(CC(C(=O)OC)C)=O C1(NC(C2N(C(C)C)CCC2)=O)CCC2CC1CN2c1ncnc2c1CCC2 c1(C(N2C3CC(CNC(C4(C)CCOC4)=O)C2CC3)=O)c(F)c(F)cc(F)c1F CCC(CCC(=O)N1CC(N(C(c2ccc(C)c(C)c2)=O)CC)C2(CC2)C1)OC C12(CNC(c3c(C)nns3)=O)CCC1CCN2C(=O)CCCc1ncco1 N1(C(C(C)N(C(C=COCC)=O)C)=O)CCC(C)(CO)C1 c1(C(N2C(C)CN(C(CCC=C(C)C)=O)C(C)C2)=O)coc2c(F)c(Cl)ccc12 c1(CCNC(C(C)C2CC2)=O)ocnc1CNC(=O)CN1CC=CC1 c1(C(=O)NCC(CNC(CN(C(=O)OC(C)(C)C)CC)=O)O)cc(O)ccc1C c1(C2C(COC)C2)ccccc1OC(=O)ON(C)C.c1(C)nccn1C c1(C(=O)NCCc2ncc[nH]2)cc(C(=O)O)cc2[nH]ncc12 C1(NC(C2COCCO2)=O)CC2CN(C(=O)CNc3ccc(Cl)cc3)CC12 C(=O)(CCCC(=O)NCC1CCCC(NC(=O)CCOC(C)C)C1)OCC Cc1ccc(C2(C(=O)N(CC(C)NC(C3CCCN3C)=O)C)CC2)nc1 C1(CN2CCCC(C)C2)CC2(C1)CN(C(C1CN3CCC1CC3)=O)C2.C1C(=O)N1 N1(C(c2nc(CCCC)sc2)=O)CCC2(CNC(=O)COC3CCC3)CCCCC12 C(=O)(C1CCc2cccnc21)NCC(N(C(CCC(=O)NCC)=O)C)C1CC1 Cc1cc(=NC2CCCc3ccc(CC(C)C)cc32)[nH]c(=NCC2CSC(C)C2)[nH]1 c1(C(N2C(CCNC(CP(C)(C)=O)=O)CSCC2)=O)cccc2c1OCCO2 CON(C)CCC(C)CCC(=O)N1CC(n2cc(CC(=O)N(C)C)nn2)CO1 c1(CC(=O)NCC2C(C)(C)OCC2)cc(C(F)(F)F)cc(F)c1 C(=O)(C1=NN(C)C(=O)CC1)NC1CN(C(C(COCC)C)=O)CC2(C1)CC2 C1(C(=O)NCCCCC2CN(C(CCSC)=O)C2)CCN(C(C2C=CCC2)=O)C1 S(=O)(=O)(c1cccc2c1OC(C)C2)NCc1c(CC)nco1 S(=O)(=O)(c1ccc(C(=O)Nc2ccc3c(c2)CCCS3)c(OC)c1)N(C(C)=O)CC S(=O)(=O)(c1cnc(NCCC2CCCC2O)c(Cl)c1)NCCC1(C)N=N1 N1(C(C2CN(C(C(C)c3cc[nH]n3)=O)CC2C)=O)CCC(O)CC(C)C1 c1(CNC(NC(CC=C)C)=NCC2CCC(C)C2)cn2ccccc2n1 C(=O)(C1c2ccccc2-c2ccccc21)N1CCN(C(CC=C=C)=O)CC1CF c1(C(=O)Nc2cc(C#N)sc2)cc2n(n1)CCCN(Cc1ccc([N+](=O)[O-])[nH]1)C2 Cc1ccc(F)c(OCC(N2CC(C(C)NC(C3CC3N(C)C)=O)C2)=O)c1 c1(C(=O)NC(C2(C(=O)NC)CCC2)C#C)c[nH]nc1OC N1(C(c2cc(Cl)cnc2O)=O)C2CCC1CC(NC(C1(O)CC3CCC1C3)=O)C2 c1(C(=O)NC(CCCNC(C(C)NC(=O)C(C)(C)C)=O)C)cccc(F)c1C#N c1(N(C)C)nc2c(C(N3CCC(NC(=O)Cc4cnsc4)C3)=O)cccc2o1 N1(C(C2(NC(c3ccncc3F)=O)CCN(C)C2)=O)CCN2CCOCC2C1 C(=O)(CC(C(=C)C)OCC)N1CCC(NC(COCC=C)=O)C1SCC N12CC(C(C)C1)C2=O.C(=O)(C(C)(C)SC)NCC(CNC(C)=O)OC Cc1cn(CC(=O)NCCN(C(C2CC(F)(F)C2)=O)CC2CC2)nc1C(F)(F)F C1(C(N(CC(CCNC(CC(CCC)O)=O)(C)C)CC)=O)CCC2(CCCC2)CC1 C1(F)(CNC(C(CC)CO)=O)CCCN(C(=O)C(C)CC2CCCCC2)CC1 N1(C(COCCNC(C(C(C)(C)C)C2CCCC2)=O)=O)CC(C2=NOCC2)C1 C12(NC(C(C=C)O)=O)CCC(NC(=O)C=Cc3cnccn3)(CC1)C2 c1(C(=O)NC(C(CO)NC(C(CC)SC)=O)C)cnn(CC)c1C1CC1 C1(NC(Cn2nc(C)c(Cl)c2)=O)CN(C(C2(CC(C)C)CCC2)=O)CC12CC2 CC(C)C(O)C(C)C(=O)NC1(C(=O)NCC2(N(C)C)CCC2)CC1 c1(OC)cccc(C(N2CCC=C(CNC(C3CCC(C)C3)=O)C2)=O)c1O c1(C(=O)NC2CCCN(C(CS(CC)(=O)=O)=O)C2)ccc2ncc(Br)n2c1 N(C(=NCCCCC1(C)OCCO1)NCC(F)F)Cc1c(C(F)F)cn(C)n1 C1(NC(CN(C(C=Cc2n(C)ncc2)=O)C2CCC2)=O)CN2CCC1(C)CC2 c1(NC(C2C(NS(C(C)C)(=O)=O)C2)=O)cccc2c(Cl)nccc12 CC1(C)CC(C(N2CCC(CF)(NC(c3occc3Cl)=O)C2)=O)CCO1 c1(CC(=O)N(CCCCNC(=O)CC2CCCCO2)C)cccc(F)c1F C1(CNC(c2cnccn2)=O)CC2CCC1N2C(c1cn(CC(F)(F)F)nn1)=O c1(N2C(CCNC(C(CC)n3cncn3)=O)CCCC2)ncnc2sc(C)nc12 N1(C(c2ccc([N+](=O)[O-])s2)C(=O)NC(C)(C)C)CCOC2(CCC(F)(F)CC2)C1 c1(C(C)C)ccc(N2CCN(C(=O)C(=O)NCC3CC4(C3)N=N4)CC2)c(F)c1 [N-]=[N+]=NC1CCC(C(=O)NCC2CC(F)(F)CN2C(C2CCNC(=O)C2)=O)CC1 c1(C(N2CCC(N(C(Cc3ccc(SC)cc3)=O)CC)C2)=O)ccc([N+](=O)[O-])[nH]1 n1(CC)nc(C)cc1C(=O)NC(C(=O)NC1CC(C)C1)c1ccoc1 CC(O)(CC(=O)N1CCCC2CN(c3ncnc(Cl)c3CO)CC12)C(F)(F)F CC(C)C(CN(C)C)C(=O)N(C1CCCN(C(c2cc(F)n(C)n2)=O)CC1)C c1(C(N2C(CNC(C3(C)CCCC3)=O)CC(F)C2)=O)cc(O)cc(F)c1F Cn1c(C(=O)NCC2(NC(C3CC4CC3C3CC43)=O)CC2)cc(Cl)c1Cl C(=O)CC1OCc2cc(Cl)ccc21.Cc1noc(C2OCCO2)n1 O=C(C1=CCCOCC1)NC1(C(=O)NCC23CCC(CO2)C3)CC(O)C1 C1(CCC)CN(C(c2ocnc2C2CC2)=O)CC1NC(c1cnc[nH]1)=O c1(CNC(C2CCCN(C(C3CC(O)(C(F)F)C3)=O)C2)=O)ccc(CO)c(Cl)c1 c1(CN(CCNC(C2CC23CC3)=O)C2CC2)csc2ccccc12 CC(C)C(C)(C(=O)N1CCC1CNC(=O)CCNC(N)=O)c1ccccc1 c1(NC(C2C3CCN(C(C(C=CC)O)=O)CC32)=O)ccc2c(c1)COC2 N1(C(C(C2CC2)OC)=O)CCCC(Nc2cnc(C#N)cn2)CC1C Cc1nc2c(s1)CCCC2C(=O)N1CCC(CCNC(=O)CC2CC=CCC2)C1 CC(=O)CC(C)(C)C(=O)N1CCC(C)N(C(=O)C(C)O)CC1 CC1(CNC(c2cccnc2)=O)CC(F)(F)CN1C(C1CCc2c[nH]nc2C1)=O N1(C(C(CC)n2nccc2C)=O)CCc2nc(CNC(=O)COCCF)sc2C1 c1(C(N2C(C(=O)NC(c3nc(C)sc3)C)C=CCC2)=O)cncn(C)c1=O C1(CNC(c2n(CCC(=O)OCC)nnn2)c2ccsc2Cl)CCC(F)(F)CC1 C(=O)(C1CCc2nnc(C)n21)NC(CCNC(C1C(OCC)C1)=O)(C)C CCCC(C)CC(=O)NCCC1CN(C(c2cncc(O)c2)=O)CCO1 C1(NC(C2C(C(=O)OC)C2)=O)(CO)CN(C(c2coc(-c3ccccn3)n2)=O)C1 C(=O)(C1=CCCCCC1)NC(CC(C)NC(C1CCC2(CCC2)C1)=O)C N1(C(c2c(C)cc(C)o2)=O)CCCC(F)(C(=O)NC(c2nccc(O)n2)C)C1 C#Cc1cnc(NC(C2CC2NCc2ccc(C(F)(F)F)c(F)c2)=O)cn1 N1(CC)CCCC(N=c2cc[nH]cc2S(=O)(=O)NCc2ncc(C)[nH]2)C1 N1(c2n(CCOCC)c(C(C)C)nn2)CCC(C)CC1C1CCC(C)O1 c1(C(N2CCN(Cc3ccncc3)CC2)=O)cnn2c1CNCC2 C(C1(C)CCOCC1)=CC(=O)NC(CNC(c1c(C)sc(O)n1)=O)CO CC1CCN(C(c2cnc(Cl)[nH]2)=O)C(C)C1NC(c1cn(C2CCCC2)nn1)=O c1(CC(N2C(C(=O)Nc3ccc(Cl)nc3)CC(F)C2)=O)c(F)c(F)cc(F)c1F Cc1cc(=NC2CCCN(C(=O)Cn3cc(C4CC4)nn3)C2)[nH]c(C2CCC2)n1 Cc1cc(=O)c(C(=O)NC2CC3CN(C(=O)Cn4nccc4N)CC23)cn1C C(CC(C(C)C)NC(=O)CCCc1csc(=N)[nH]1)N(C(C1(CCC)CC1)=O)C N1(C(C(n2c(C)ccn2)C)=O)CCCC(NC(c2cc(Cl)cs2)=O)C1 C(=O)(CCC(=O)NN(C)C)NC(C)CCCCNC(c1cnoc1C1CCC1)=O N1(C(CCc2onc(C)n2)=O)CC2CC(NC(c3csc(C)n3)=O)C1C2 CC1=C(C(=O)N2CCOC(CC(=O)NCC3CCOC3C(C)C)C2)CC1 C(CC(C)C)(CS(=O)(=O)NCC(C1CCCOC1)N(C)C)OC Cc1cc(C(N2CC(C)(CNC(=O)C(=O)c3ccco3)C2)=O)c(F)cc1Br c1(C(N2C(C(C)NC(C3CS(=O)(=O)C3)=O)CCC2)=O)cccc(CN(C)C)c1 C(C)(CCC(=O)NCCC1CCN(C)C1)NC(c1ccc(CCC)[nH]1)=O CC(C)CC(F)C(=O)NC(CNC(=O)C(C1CCCCC1)O)CO C(=O)(CC(C)(C)O)N(C1CCN(C(C2CC2C2CCCO2)=O)CC1)CC#C c1(CNC(C2CCC(C)C2)=O)nnn(C)c1C(=O)NCCc1ccnc(O)c1 c1(OC)cccc(CC(O)C(=O)NC2(CO)CCN(C(=O)CC(=O)NC3CC3)C2)c1 Cc1nc(C)n(CCC(=O)N(CCC(C)NC(=O)CCOC2CCOC2)C)n1 Cn1ncc([N+](=O)[O-])c1C(N1CC2CC1CN2C(C1CCCC(O)C1)=O)=O C(C(CC(=O)NCC(C1CCCCC1)O)OC)NC(c1cn(CCC)nc1)=O C1C(O)CC(=O)N1.C1(C(C)N(C)C)CCN(C(C2(C(=O)NC3CC3)CC2)=O)CC1 c1(CCNC(=O)NC(c2ccco2)COC)cccc(SC(F)(F)F)c1 Cc1nn(C)c(C)c1C(=O)NC1C2CC1N(C(C1SCCS1)=O)C2 CN(CCCC(=O)NC1C2CCC1CN(C(C1CC3C=CC1C3)=O)C2)N=O C1(NC(CC2(COC)CC2)=O)CCN(C(=O)C(O)Cc2[nH]cnc2C)C1C N1(CC)N=C(C(=O)N(C)CCNC(c2nn[nH]c2C(F)(F)F)=O)CCC1=O N1(C(c2cncc(C)n2)=O)CC2(CCC2)CC1C(N1CC(F)C(F)C1)=O N1(C(CSCC#C)=O)CCCC2CN(C(c3ccc(C(F)(F)F)o3)=O)CCC12 c1(CN2CC3(C(C(N(C4(C(C)C)CC4)CC)=O)C3)C2)ccc2c(c1)ncn2C C=C1CC2(C1)CC(C(=O)OCc1sc(Cl)cc1Cl)C2 Cc1cnc2ccc(NC(=O)C(=O)NCc3nnc4n3-c3ccccc3-4)cn12 N1(C(C(C(C)C)SC)=O)CCC(C(=O)N(C2CCCN(C)C2)C)=C(F)C1 N1(C(C2CCC(C(=O)OC)C2)=O)CCC(C)(CNC(=O)Cc2c[nH]nc2C)C1 c1(C(N(CC(C)NC(=O)C(C)Sc2ccccn2)CC)=O)cc(CO)ccn1 C1(C(=O)NC(C2(O)CCN(C(=O)COCC3CC3)CC2)C)CCC2(CCCC2)C1 Cn1cnc2cc(C#N)c(C(=O)NC3CN(C(C4CC4(F)F)=O)C(C)(C)C3)cc12 C(=O)(C1=CCC1)NC1CC(CNC(=O)COCCc2ccccc2)C1 C1(CNC(c2ccc[nH]2)=O)CN(C(=O)CC2(CO)CC2)C2(CCC2)C1 N1(C(C(C(C)C)N(C)C)=O)CCC12CN(C(C1CCCN1c1ccccc1)=O)C2 c1(C(C)C)ccc(F)c(C(=O)NC2C3CCN(C(c4cnsc4)=O)C23)c1 c1(NCc2cc([N+](=O)[O-])sc2)cc(-c2cccc(F)c2)nc2ccccc12 C1(CNC(c2ncc(OC)cn2)=O)(NC(=O)CC(C)C(C)C)CCCCC1C CC(C)CCN=C(NCc1ncccc1Cl)N1CCC(C(C)O)C1 C1(CNC(CSCCCC)=O)(NC(=O)Cc2ccc(C(F)F)cc2)CCOCC1 O=C(CC1COCc2ccccc21)NC1CCN(c2ncccn2)CC1 c1(C(=O)NC(CCCNC(c2c(C)ccc(=N)[nH]2)=O)C)cnc2cc(O)nn2c1 C1(CNC(C2CN3CCCN2CC3)=O)CCN(C(c2cnc(S)[nH]2)=O)CC1(F)F C1(NC(Cn2c(C)cc(C)n2)=O)CN(C(=O)CC2CCCCC2)C2CCCC12 c1(C(=O)NCC2(C(C)NC(c3n(CC)ncc3)=O)CC2)ccc2c(c1)C(C)CO2 c1(N(C)C)c(C(=O)NCCCNC(=O)C(C)(C)C(N)=O)nnc2ccccc12 C(CC(O)C(=O)NC1CCN(C(C2(c3noc(C)n3)CC2)=O)CC1)SC n1(CC)nc(C)cc1C(=O)NC(CNC(=O)CC1CCOC1(C)C)CC(C)C C1(CNC(Cc2c(C)n(C)nc2)=O)N(C(=O)Cc2cscn2)CCCC1(C)C C1(COC)CC(CNC(c2cnc(S)[nH]2)=O)N(C(=O)Cn2nnc(C)n2)C1 CC#CCC(C(=O)NCC12CC(F)(C1)C2)NC(=O)C(C)NC(C)(C)CC C1(OCCC)CCC(C(C(=O)NC2CC=CCC2)N(C)CCN2CCOC2=O)CC1 C1(O)(Cc2cccs2)CCN(C(=O)CSC)C1.C1(OCC)C(=O)N(C)O1 n1(CC)nc(CNC(=O)NC(c2ccc(C(F)(F)F)nc2)C)c(C)n1 C1(CC(=O)NCc2nccs2)CCCN(C(=O)CC2CCCCO2)C1 C1(C(N2CCC(CN3CCCC3)C2)C(=O)NCc2cccs2)(CCC)CC1(C)C c1(C(=O)NCC(CC)NC(=O)Cc2csc(C)n2)c(C)oc(C)c1C CCC1(CC)CNC(=O)N1.c1(CCN2CCCC2=O)cccc(C(F)F)c1 N1(C(C2(COC)CC(=C)C2)=O)CCCC2(CCN(C(C3SCCS3)=O)C2)C1 c1(C(C(=O)NCCCOCCCNC(c2coc(C(F)F)n2)=O)O)cccnc1 C(=O)(C(C)(C)S(C)(=O)=O)NCC1(C(C)(C)O)CN(C(C2CC(C)CC(=O)N2)=O)C1 Cc1ncc(CC(=O)NC(C)C(C)N(C(=O)CCN2CCC2)C(C)C)s1 N1(C(c2n(COC)ncc2)=O)CCC(CN(C)C(C2(n3cccn3)CC2)=O)CC1 c1(C(=O)N(C(CN(C(C2CC2c2ccco2)=O)CC)C)CC2CC2)c[nH]nc1C1CC1 n1(CCCC)ncc(C(=O)NCC2(C)CN(C(=O)CSCCC(C)C)C2)c1C C(c1ccccc1C#N)=CC(=O)NCCNC(C(N1CCCC(O)C1)C)=O N1(C(c2c(C)cnnc2)=O)C2CCCC1CN(C(c1coc3ccccc13)=O)C2 N1(C(C2(F)CCN(C(CC(C)=C(C)C)=O)C2)=O)CCc2c(C#N)cccc21 C1(N(C(=O)CCn2cc(Cl)cn2)CC)CCCN(C(=O)CC2(O)CCOC2)C1 C(CCCCCCNC(C1CCC2CC12)=O)NC(COCCOCC)=O C1(NC(C2CCCN(CC)C2)=O)CCN(C(=O)CC2CCCC2)CC1(C)C C1(O)(C(C)NC(c2nocc2C(C)(C)C)=O)CCN(C(C2COCCOC2)=O)C1 Oc1ccc(-c2noc(-c3noc(C4CC5(C4)CC54CC4)n3)n2)cc1OC(F)F C1(CNC(CC(CC)C2CCC2)=O)CCN(C(C2CCCNS2(=O)=O)=O)C1(C)C Cc1cc(=NCc2cccc(O)n2)[nH]c(=NCC2(C)CC2(F)F)[nH]1 C1(NC(CCCCCC#C)=O)CN(C(c2nn(C)c(Cl)c2Cl)=O)CCC12CCC2 c1(NC(C(CCSC)NC(C(CC=CCC)C)=O)=O)ccc(F)c(O)c1 c1(NC(C2CSCCN2C(C2CC2(F)F)=O)=O)cc(Cl)cnc1Br c1(SC)cccc(C(=O)NC2CCCC2NC(=O)Cc2csc(C)c2)c1Cl C1(C(N(CC)CC)=O)CCC1C(F)(F)F.C(CC)NC(=O)COCCF c1(C(C)=O)cc(C(=O)NC2CC(C)(NC(=O)COCCN(C)C)C2)n(C)c1 c1(C(=O)NCC2C(NC(C(CCC)OC)=O)COC2)cccc(CS(C)(=O)=O)c1 c1(C(C)C)nc(C2(C)CS(=O)(=O)C2)n(Cc2cccc(F)c2)n1 C1(CCNC(COCCC)=O)CCN(C(c2coc(Br)n2)=O)C(C)C1 C12(C(=O)NC3C(CNC(Cn4c(C)ncc4)=O)CCC3)CCC(C1)OC2 c1(C(=O)NCC2(O)CC(CNC(CSC)=O)C2)ccn(C)c1C c1(C(=O)NC2(COC)CN(C(=O)CC3CC3C)C2)c[nH]c(=N)nc1O c1(C(C)OCC)nc(C)c(C(=O)N(CCCCCNC(C2CCOC2C)=O)C)s1 c1(C(=O)NC2CC(CNC(C3(F)CC3)=O)C2)nc2n(c1Cl)CCCC2 N1(C(c2ccc(NC)cn2)=O)CCN(C(=O)CC2(C)CCCCC2)CC1C1CC1 C1(C(=O)NC2(CF)CCN(C(C(C)=C(CC)C)=O)C2)CCN(S(=O)(=O)N(C)C)C1 N1(C(Cc2cncc(C)c2)=O)CCC(C)(NC(C2CC2Cl)=O)CC1 C1(CNC(C=C(COC)C)=O)CCCCC1NC(c1ccn(CCO)c1C)=O C12(NC(C(C(C)C)SC)=O)CCOCC1CN(C(c1ccc(C)nc1O)=O)C2 C1(NC(C(C)O)=O)CC2CCC1N(C(c1cc(-c3ccco3)on1)=O)C2 c1(CC)cc(Cl)ccc1C(N1CCCC(NC(=O)CCc2cccnc2)C1C)=O c1(CN(CCCNC(=O)CC2CCCCC2(C)C)CC)nccc2ccccc12 c1(C(N2CCC(C)C2C)C(=O)NCCC#N)ncc(F)cc1F.c12ccc(cc1)n2C C1(CC(N)=O)CCCN(C(=O)C(Cn2cccn2)NC(C2CCC(O)C2)=O)C1 c1(C(N(C2CCCN(C(=O)C3=CCCSC3)C2)CCO)=O)ccc2ncnn2c1 c1(OCC(=O)NCC(CC)NC(C2COC(=O)N2C)=O)ccc(C)cc1C C(=O)(C1=Cc2cc(F)ccc2OC1)NCC1CCN(C(CC(C)O)=O)C12CC2 C1(CCOC)CN(C(=O)Cn2ccnn2)CCN1C(=O)C=C1CCC1 C1(CC(=O)OC)COC(C)CN1C(c1cccc(C(C)=O)c1)=O N1(CC(N2CCCC(N(C(C3ON=C(CC)C3)=O)C)C2)=O)CCP(C)(=O)CC1 C1(CNC(Cc2cc(OCC)ncc2)=O)CCC(C)CN1C(=O)Cn1nccn1 C1(C(=O)NC(CNC(c2ccc(C#N)cc2)=O)CO)CCC2(CCC2)OC1 c1(OC)cccc2cc(C(=O)NCCN(C(=O)CC(C)CSC)C(C)C)c(=O)oc12 C#CCC(CC)NC(=O)C(c1ccoc1)NC(=O)CCOCC(F)F c1(NC(c2c(C)ccc(C)c2N)=O)ccc(S(=O)(=O)C(F)(F)F)cc1 C1(CN(C(=O)CCCc2ccccc2)C)CCCN(C(C2(CF)CC2(F)F)=O)C1 c1(C(=O)NC2CN(C(Cc3c(C)con3)=O)C(C)C2)ccccc1P(C)(C)=O N1(C(=O)CCSc2ccc(Br)cc2)CC2(CCCC2)C1C(=O)O N1(C(CC2(C=C)CCC2)=O)CC(CNC(c2cn(CC)nn2)=O)C2(CC2)C1 c1(C(N)=O)ccc([N+](=O)[O-])cc1NC(C1CC(F)CN1C(=O)Cc1cc[nH]n1)=O Cc1ccn(C(C)C(=O)NC(CO)C(=O)NCC2(CO)CC=CC2)n1 C(=O)(CC(C)(C)C(F)F)NC(C(C)C)CCN(C)C(C1CC(C)(C)C1)=O c1(C(=O)NC2(CCOC)CCN(C(C3CCC3CF)=O)C2)cncn(C)c1=O C1(CC)(CC)CC(NC(=O)C2=CCCC2C)CN1C(c1nn(C)nc1Br)=O CCCCC(C(=O)NC1COCC(C)(C)C1)NC(=O)C(CC)CCC c1(NC(C)=O)cc(Br)ccc1NC(=O)CC1CCC(NC(=O)C=Cc2cnccn2)C1 N1(C(C23N(C(C4N(C)CCOC4)=O)CC(C2)C3)=O)CCCN(C=O)CC1 c1(N)ccc(Br)cc1O.c12cnc(nc1)N1C3CN(CC13)Cc1c-2cccc1.CS N1(C(CCNC(=O)OCC)=O)CC(F)(F)CC1CCNC(=O)COC C12(C(=O)NC3CC(N(C)C(c4ncn5c4CCC5)=O)C3)CCC(C)(CC1)CO2 CCS(=O)(=O)c1ccc(Cl)cc1C(=O)NCC1CN(C(=O)CC#N)C2CC12 c1(C(=O)Nc2ccc(C)c(I)c2)cncc2sc(-c3cccs3)cc12 CCCS(=O)(=O)C(C)C(=O)NCCN(C(=O)C(C)=C1CCCC1)CC1CC1 C1(NC(=O)CNS(=O)(=O)C2CC2)CCN(C(=O)COc2cc(Cl)ccc2Cl)CC1O c1(OC)c(F)ccc2[nH]c(C(=O)NCC3(F)CN(C(c4c[nH]cc4C)=O)C3)cc12 C(=O)(C(CC(C)CC)Nc1scnc1CC)N1CC(CCCC)N(C(C)=O)CC1 CC1CCCC=C1C(=O)NC(C)C(CO)NC(=O)Cc1ccc(F)cc1Br Cc1cc(N)cnc1C(=O)NCC1CCCC1NC(C1CCC2CC2CC1)=O N1(C(C(C)NC=O)=O)CC(C)(C)C1C(F)(F)F Cc1cc(NC(=O)CCC(=O)NC2C3CN(Cc4cnco4)CC23)c(C)cc1F Cc1ccc(C(=O)NCC2C3CCC(C3)N2C(c2n[nH]c(C)c2F)=O)c(C)n1 S(=O)(=O)(c1cnc(Cl)nc1)NCC1CCC(C(N2C(C)C(=O)NCC2)=O)CC1 C1(F)(C(=O)NCc2occ(C(=O)NCC(c3nccs3)C)c2)CCCOC1 c1(C(=O)NC2CC(C)(CC)N(C(=O)CNC(N)=O)C2)ccc2c(n1)CCC(C)C2 CC(CC(=O)N(CC(=O)NC(C)CCN1CCCC1)CC1CC1)C(F)(F)F c1(C(=O)NCC23CCC2CCN3C(c2nsnc2O)=O)cc2c(cn1)OCCO2 N1(C(CC(=C)C)=O)CC(C)OC2(CCN(c3cccc(F)c3C#N)C2)C1 C1(CCC(N)=O)C(=O)N1.C1(C(N(CCCN(C)C)CC)=O)CCNC1=O C1(C(=O)NCC(CCNC(C(CC)N(C)C)=O)OC)CC2(CCC2)CO1 C(=O)(C1=CCC(C)CC1)N(C1CCCN(C(=O)CN2CCOCC2)C1)CC N1(CC)CCc2ccccc21.c12ccc(cc1NC(CO)CC(C)(C)C)[nH]c2=O N1(C(Cc2nc(C)[nH]n2)=O)CC(NC(c2ccc(N)c(O)c2)=O)CC12CCCC2 c1(C(=O)NCC(C)NC(c2ccc3ccsc3c2)=O)cnn2c1CC(C)CC2 c1(CSC)noc(CCC(=O)N2CC(C(C)(C)NC(=O)CC3CCC(O)C3)C2)n1 C1(COC)(NC(c2cncs2)=O)CCN(C(c2cnc(S)n2C2CC2)=O)C1 C(C(N=[N+]=[N-])C(=O)NC(CC)CC(=O)NCC1CC2CCC(C1)C2)OCC N1(C(CCN(CCC)C)=O)CCC(CC(=O)N(CCC)CCC)C1 C1(C(N2CCCC(CCCO)C2)=O)CC2CCC(C1)N2C(C1CCOCC1)=O C1(NC(C2C(=C)C2)=O)COC2(C1)CN(C(c1nccc3occc13)=O)C2 C1(CNC(C2(C#N)CC2)=O)CN(C(C2CCN2C2CCCC2)=O)C2(CCC2)C1 CCN=c1ccc(C(=O)NCC2C3CN(C(=O)CCS(C)=O)CC23)c[nH]1 C1(NC(C2N(CCC)CCC2)=O)CCC(CNC(=O)COC2CCOCC2)CC1 Cc1[nH]nc(Cl)c1C(c1nnnn1CCCOC)NCC1(C)CC=CCC1.C(C)(C)C N1(C(c2c(C)nc(C)c(C)n2)=O)CCCC2(CC(NC(=O)C#CC(C)C)CO2)C1 N1(C(c2c(C)cno2)=O)CCC(NC(c2ccc(Cl)cc2C#N)=O)C(F)(F)CC1 O=C(CC(C(F)(F)F)n1ccnc1)NC1CN(C(=O)C(F)(F)CN2CCCC2)C1 N1(C(Cc2ccn(C)n2)=O)CCC2(CCCCC2NC(=O)C=Cc2cncs2)C1 c1(CSC)cccnc1C(=O)NC(C)CCN(C)C(c1ncccc1N)=O CCCCC(CC)C(=O)N(C(c1ccc(C)cc1)c1cccc(Cl)c1)CC c1(OC)cnc(Cl)cc1C(N1C2CN(C(c3cnccc3Cl)=O)CC12)=O C1(NC(C(c2ccc(Cl)s2)C)=O)CCCC(NC(C2CCC(C)(C)O2)=O)C1 c1(N2CC(COC)N(C(C3CCCCO3)=O)CC2)ncc2ccccc2n1 Cc1cc(C(=O)N(C(C)CCNC(c2cc(-c3ccns3)on2)=O)C)ncn1 C(=O)(C1=NOC(C)C1)NCC1N(C(c2[nH]cc(C(C(C)C)=O)c2)=O)CCC1 N1(C(C=C(C)C(C)C)=O)CCN(C(C2(C(c3ccc(F)cc3)=O)CC2)=O)CC1C c1(CCC(=O)N(C2CN(C(C(C)Oc3ccccc3Br)=O)C2)C)cccc(F)c1 c1(C(=O)NCCN(C(=O)C(C)Cc2ccnn2C)CC(C)O)coc(Cl)n1 c1(N(C)CC2CCCO2)nc2cccc(F)c2c(=NCC2CCCOCC2)[nH]1 N1(C(CC2(C=C)CN(C(C3CC4(CCO3)CC4)=O)C2)=O)CCOC2CCCCC12 c1(C(=O)NCC2(CNC(c3cnc(OC)s3)=O)CCCC2)cccc(N)c1O N1(C(COCCCN(C)C)=O)C2CCC1C(C(=O)NCS(C)(=O)=O)C2 C(=O)(C(C)(C1CC1)N(C)C(c1cnnn1C)=O)N(C)CC1(CO)CC1 C1(c2nnnn2C2CCCC2)(NCCCc2scc(C)n2)CN(C)CC1C C1(NC(c2c(CC)c[nH]n2)=O)CC2CCC(C1)N2C(=O)C(c1ccccc1)C CS(=O)(=O)C1CN(C(=O)CC2CCCCN2C(C2C3CCCCCC23)=O)C1 c1(CNC2CN(Cc3cc(C)cc(Cl)c3)CC23CC3)cc([N+](=O)[O-])cc(Br)c1O Cc1cccc(F)c1C(=O)NC1(C(N2CCCC(CC(N)=O)C2)=O)CC1C C(N1CCC(O)CN1C(=O)C=Cc1cscn1)C(C)=O.ON c1(C(=O)NCC2(C#N)CN(C(c3ccc(C)n3C)=O)C2)cc2ccccc2[nH]1 C(=O)(C(C(C)(C)C)N(C)C)N1CC(C(C)NC(CCN(C(C)=O)C)=O)OCC1 Fc1cccc(CCCF)c1.C1(N)CCOC1 c1(C(N(CCCN(C(=O)C=C2CC2)C)C)=O)cc2cc(F)ccc2[nH]1 C(C(CO)CC(C)C)NC(CCN(C(=O)CC1CCCC(=O)C1C)C(C)C)=O N1(C(C2C(SCC)C2)=O)CCC2CCCC2C1.c12cccc(F)c1CC(=O)N2 N1(C(CCC2CCC(NC(C3CC=C(C)CC3)=O)C2)=O)CC(O)(C2CC2)C1 c1(C(=O)NCCN(CCC)C(C2CC2CF)=O)cc(S(=O)(=O)NC)c[nH]1 CCC(C)C(O)C(=O)NCC(C1CCC1)NC(c1cnn(C)c1SC)=O c1(C2C(NC(C(F)OCC#C)=O)CC2)cc(Cl)ccc1Cl C1(NC(=O)Cc2cccc(Cl)c2)CCN(C(C23CCCC2C3(F)F)=O)CC(O)C1 c1(OC)c(Br)cc(CN2CC(C)CC2NC(c2ncc(C)c(Cl)n2)=O)cc1Br S(=O)(=O)(c1ccc(C(=O)OCc2cc(C)ccc2C)cc1)NCC N1(C(C2CCCCN(C(CCC=C(C)C)=O)C2)=O)CCC(O)CC12CC2 c1(OC)ccc(C(N2CCN(C(C3CCN(CC(C)C)C3)=O)CC2C)=O)c(F)c1 N1(C(c2coc(O)n2)=O)CCN(C2CCN(C(C3CCCC3(F)F)=O)C2)CC1 N1(C(C(=O)OC)=O)CC(CN(C2CC(O)C2)C)C2(CCC2)C1 CC1CN(C(=O)C#CCNC(=O)CCc2cnn(C)c2)CCN1C C1(NC(CSCC=C)=O)CCC(CNC(=O)C(O)Cn2cncn2)CC1 c1(CC(=O)NC2CCCC(NC(C(C)OC)=O)C2)cccc([N+](=O)[O-])c1C C1(C(=O)NC(C2(O)CCN(C(c3cnn(C)c3)=O)C2)C)CCCCCCC1 c1(SCCCC)cc2ccc(F)cc2o1.N1(C)CC(OC(C)(C)C)CC(CC(=O)O)C1 C(=O)(CCCCC(C)(C)C)NCC1N(C(C(CC=C)C(C)C)=O)CC2(CCC2)C1 O=C1CC2(CCC2)C(C(=O)NCCCNC(=O)C2=CCCO2)CN1 C1(NC(C(C)SC)=O)CC2C1CCN2C(=O)CCc1ccc(Br)cn1 CCC(F)(F)C(C)(C)C(=O)NC(C(=O)NCC(C)C(C)(F)F)C(C)(C)C C1(OC)CC2(CCC(C(=O)NCC3CC3CNC(=O)CCCCC(C)C)CC2)C1 c1(CC)ccc(CCNC(=O)N(c2ncc(-c3cccs3)s2)C)s1 c1(C(=O)NC2C(NC(C(C)SC)=O)CCC2)ccc2c(c1)N(C)CC2 C1(C(=O)NC2CN(C(c3c(C)scn3)=O)C(C)C2)CC12CCSCC2 c1(C(N2CC(C(=O)NCCCOC)C(F)(F)CC2)=O)ccc(Cl)c([N+](=O)[O-])c1 CC(O)CCC(=O)N1CC(NCC=CC2(c3ccccc3C#N)CC2)C(C)C1 C1(C(=O)NC(CNC(C(CC)Cc2ccc(N)cc2)=O)C)CN(CP(C)(C)=O)C1 Cc1c(C(N2CC3C(CNC(c4cnc(O)o4)=O)C3C2)=O)oc2ccc(F)cc12 C(C(CNC(=O)CCOC1CC1)S(C)(=O)=O)NC(C1CCC(C(=O)OC)C1)=O Cc1c(C(N2CCC(N(C(=O)CSC3CC3)C)C2)=O)[nH]c2c(C)cccc12 C=CC(C)(CC)C(=O)N(CC(O)CN(C)C(c1nc(Cl)ccc1Cl)=O)C CC1Cc2ccc(F)cc2C1NC(=O)CCCOCCCN N1(C(CC=CC=C)=O)CCCCCC1C(=O)NCC(O)CF c1(OCCC(=O)NC2CCC(NC(CC#N)=O)C2)ccccc1F c1(NC(=O)NC2CC(C(N(c3ccc(Cl)cc3)C)=O)C2)c[nH]c(=O)cn1 C1(NC(C(C)C)=O)CCCC(NC(c2ccccc2-n2ccnn2)=O)C1 C1(C(=O)NC2C3N(C(c4scc(C)c4)=O)C(CC3)C2)CCC2(CCOCC2)O1 C(=O)(C1=NN2CCCN=C2N1)NC1CC(CNC(C2(C)CCC(C)C2(C)C)=O)C1 N1(C(c2c(C)coc2C)=O)CC2=C(C1)CN(C(=O)C(C)Cc1cnc[nH]1)C2 c12cc3n(n1)CCCN3C2=O.c1(C(=O)OC)oc(C)nc1C(F)(F)F C1(C(N2CCCC(C#C)C2)=O)CC12CCN(C(C1(CCCC)CC1)=O)CC2 CC(CC(=O)NCC1C=CC(NC(=O)CNC(C2CCC2)=O)C1)C(C)(C)C C12(CNC(c3c(CC)n(CCC(C)C)nc3)=O)CC(CO1)N(C(=O)C(C)SC)C2 CC(C)CCC(C(=O)N1CCC1(C)CCO)NC(=O)C=C(C1CC1)C1CC1 n1(CC(N2C(C)(CNC(C3C(CC)N(C)CC3)=O)CCC2)=O)cnc([N+](=O)[O-])n1 N1(C(c2cccc(C(=O)NC)n2)=O)CC(C)CN(C(=O)CN2CCCC2)CC1C n1(C(C)C(N2CCC(c3ccccc3)C2)=O)cc(C(C)C(=O)O)nn1 CC1=C(C)CC(C(N2CCC(C3CN3C(=O)C(O)CC3CCCCC3)CC2)=O)CC1 c1(C(N2CCC(OCCNC(c3ccnc(O)c3)=O)C2)=O)ccc2csnc2c1 c12csc(n1)CNC(=O)c1cc(on1)CNC(=O)CS2.C1(CC)CCCCO1 N1(C(C(CCOC)NC(=O)COCC(=O)N(C)C)=O)CC2CC3CC2C1C3 c1(OC)ccccc1C(F)(F)C(=O)NCCCCCN(C(=O)C(F)C1CCC1)C N1(C(c2cc(CN(C(COC)=O)C)on2)=O)CCCC(O)C1C C=CC1CN(C(c2c[nH]c(=NC)s2)=O)CC1NC(=O)C(c1c(C)noc1C)(C)C c1(C(N2CC(C(C)NC(=O)CCCC3CC3)OCC2)=O)cc(Cl)c2n[nH]cc2c1 N1(C(c2cnn(C)n2)=O)CC2CCC1C1CN(C(=O)CCC(N)=O)CC21 c1(CC(=O)CN(CCCO)C(C2CCCCC2)=O)ccccc1Br c1(C(=O)NC2CCN(C(=O)CC3=CCOCC3)CC2O)cc2cccnc2o1 Cc1sc(N)c(C(=O)NCC2(NC(c3ccc(CO)o3)=O)CC2)c1C C(CNC(C1CCC(CNC(c2cnc(C)cn2)=O)CC1)=O)(C(F)(F)F)OC C1(C(=O)NCc2c(CC)c[nH]n2)CSCCN1C(=O)COCC1CC1 C(=O)(CC(C)(C(F)F)N(C)C)N1C(CNC(C(c2c(C)c(Cl)ccc2)O)=O)CC1 C(=O)(C(C)(NC(=O)CC1C=CC(OC)C1)NCC(N1CC(NC(C)=O)C1)=O)OC C(CC(C)(C)C)(C(=O)NC1(CN(C)C(c2sc(C)nc2C)=O)CC1)OC c1(CC)onc(C)c1C(=O)N(C)CCN(C(=O)Cc1ccccc1OC(F)F)C N1(C(c2nc(C)nc(O)c2)=O)CCC2(CCN(C(=O)C(C)CC3CCC3)CC2)C1 c1(C(N)=O)cccc(CN2CCC(C(=O)NCc3ccncc3F)C2)c1 C1(NC(C(CC=C)CC)=O)CN(C(=O)CCc2cccc(O)n2)CCC1(C)C C1(CN(C(C2CN(C(C)C)C2)=O)C)C2CN(C(C3(C)CC3(F)F)=O)CC12 C(=O)(CS(=O)(=O)C1CCOCC1)NC(C(C)NC(=O)CSc1cccs1)C C1(C)(NC(C(C)OCCC=C)=O)CCN(C(c2sccc2SC(F)F)=O)CC1 c1(NC(C(C2(O)CCCCC2)NC(C=C(CCC)C)=O)=O)ccc(N=[N+]=[N-])cc1 c1(OC)cc(C(F)(F)F)ccc1C(=O)NC1CCCCC1NC(=O)C(O)C(C)C C1(NC(c2cc(C(F)F)on2)=O)(CF)CCN(C(=O)CC2CCCO2)C1 c1(C(=O)NC(CN(C(=O)CCCN2C(=O)CCC2=O)CC)C)ccc(Cl)cc1F Cc1cc(C(N2CCN(C(=O)CCC(C)(C)C)CC2)=O)nc2ccccc12 C1(CNC(C(CCCC)F)=O)CCC2CN(C(C3(C#N)CCCOC3)=O)CC12 N1(C(CC(C)C)=O)CC(NC(C2CCN(C3COC3)C2)=O)CC12CCCC2 S(=O)(=O)(c1cnn2ccc(N3CCC(C)(N(C)C)CC3)nc12)N1C(C)C(C)CC1C N1(CC(=O)OCC)CCCC(NC(=O)CCn2cc(C(C)CC3CCC3)nn2)C1 c1(CC)nc2c(C(=O)NCC(C)CN(C(=O)C(C)C(C)COC)C)ccnc2[nH]1 C1(N(C(c2ccc(COC)o2)=O)C)CCN(C(=O)CSc2n[nH]c(C)n2)CC1 c1(C(c2nnnn2C)NCC(COC)C)sccc1I c1(C(=O)OC)ccc(C(=O)NCCCN(CCCNC(c2cnn[nH]2)=O)C)cc1Cl Cc1ccc2c(c1)C(N)C(NC(N1CCN(C(c3ccncc3)=O)CC1)=O)C2 N1(C(CN2CC(=O)N(C)C2=O)=O)CC(NC(=O)C=CC2CC2)C(S(C)(=O)=O)C1 c1(C(=O)NC(CNC(c2cnn3ccsc23)=O)CO)c(Cl)ccc(F)c1F c1(OCC(C)C)ncccc1OC(F)F.C=C1CNC1=O c1(C(=O)NC(C(N2CCC(C)(C(=O)OC)C2)=O)C2CCC2)cncn(C)c1=O C(C)(CO)(C(=O)NCCOC1CCCOC1)NC(C1ON=C(C)C1)=O N1(C(c2cc(Cl)no2)=O)CCN(C(=O)COCc2cccnc2)C2CCCCC12 N1(C(COCCOCC#C)=O)CC(NC(=O)C(C)n2cnnn2)C2(CCC2)C1 C1(C(=O)NC(CSCC)C(=O)NCC2(C)CCN(C)C2)CCCN(C)C1 C1(OC)CN(C(=O)CN2CCCCC2=O)CC1NC(=O)C(C)CN(C)C N(C(=NCC1(C(N)=O)CCCC1)N1CCC(OC)C1)C(C1CCCCCC1)CC N1(C(c2c(CC)ocn2)=O)CCN(C(=O)CCc2ccco2)C(c2cn[nH]c2)C1 c1(OC)c(OC)cc(OC)cc1CC.C12COC(C1)CN(C1CC1)C(=O)C2 c1(C(=O)NC(c2c(OC)cncc2)C(=O)O)ccc(NC)cc1Cl CC1CN(C(c2c[nH]ccc2=O)=O)CCC1NC(C1CC1c1ccoc1)=O C1(C)(CNC(CCC2CCN(C)C2)=O)CCN(C(=O)Cc2ccc(O)cc2)C1 N1(C(C2(C)CC(C)C2)=O)CCC(CCCNC(=O)CC2CCCOC2)CC1 C1(NC(c2cc(CC)no2)=O)CN(C(=O)C(C)C)CC1CN(C)C C1(N(C(C(C2CCCCC2)C)=O)CC2CN(C(=O)C(C)(C)F)C2)CCOCC1 Cc1cc(S(=O)(=O)NCCCC(=O)c2cccs2)cc([N+](=O)[O-])c1Cl c1(CNC(C2C(NC(C(C(C)C)OCC)=O)CCOC2)=O)c(O)cccc1F Cc1cc(C(=O)NCC2CC(NC(c3[nH]c(C)c(C(C)C)c3C)=O)C2)c(O)nn1 N1(C(c2ncc(NC)nc2)=O)CCC2(CCCN2C(C2CCC2C)=O)CC1 C(=O)(CCCc1ccccc1)NCCCCNC(C(c1cscn1)N(C)C)=O C(=O)(C(C)n1cnnn1)NCCCN(C(=O)C(F)n1ccnc1)C(C)C c1(OCC)ncc(C(=O)NC2CCCC(C(=O)NCCSC)C2)cn1 c1(C(C(C)NC(=O)OC(C)(C)C)NC(c2cccc(F)c2)C(=O)O)cccc(Br)c1 CC#CC1CCN(C(=O)CC2CC2CNC(c2c[nH]cc2C(C)C)=O)C1 c1(NC(=O)NCCC2C(CC)C2)cc(C)nc2[nH]nc(C)c12 c1(CC)nc(C(N2CCC(NC(C3CN(CC(F)(F)F)C3)=O)CC2)=O)c(N)s1 c1(CCC(=O)NC(C(C)C)CNC(=O)C(C)c2ncco2)ccc(C#N)cc1F c1(CC(=O)NC2(CC3CC34CC4)CC2)cccc(O)c1 CN1CCOCC1CNC(=O)Nc1oc(COc2ccccc2)nc1Cl N1(C(C(C(=C)C)(C)C)=O)CCC2CCN(c3ncnc4c3ncn4C3CC3)CC2C1 C1(C)(C(C)C)CCN1C(c1ccc(CNC(c2ccccc2)=O)s1)=O c1(C(=O)NC2CCCN(C(c3n[nH]c(C)c3C)=O)CC2)nnn2c1CCCCC2 c1(C(C)NC2CCN(C3CC3)C2=O)ccc(Cl)cc1Cl C(=O)(C(CCSC)NC(=O)Nc1ccc(F)cc1)NC1C(C(=O)OCC)CCC1 C1(CCC(=O)N(CCC)CCNC(=O)C(O)c2ccco2)(COC)CCCC1 N1(C(CN(S(=O)(=O)CC)CC)=O)CCN(C(c2cnc(O)n2C)=O)CC1C N1(C(c2ccc(CNC(c3c(CC)nns3)=O)cn2)=O)CCOC(C)C1C CCC(C#N)(CC)C(=O)N1CC(N(C(=O)C=CCF)C)C2(CC2)C1 Cc1ccnc(O)c1C(N1CCC(O)C(N(C(=O)CCOC2CCCC2)C)C1)=O CC(C)(C)CC(C(=O)N1CCCC1CF)NC(c1ccsc1)=O N1(C(N2CCC(NCC(C)CN(C)C3CC3)CC2)=O)CCc2ccccc2C1 N1(C(CN(C(C(C(C)C)SC)=O)C2CCC2)=O)CC2(CC(O)C2)C1 c1(C(N2CCC(NC(=O)COCC3CC3)C2)=O)cc(Br)c(Cl)s1 c12cc(ccn1)C(=O)N2.c1(C(N)=O)cn(C2CN(C(C3CC=CC3)=O)C2)nn1 C(=O)(CC(C)(C)C(C)(F)F)NCC1(F)CCN(C(C=Cc2scc(C)n2)=O)CC1 CCC(O)C(=O)NC(CNC(=O)NC1CC1)CCOC.C(C)(C)(C)O c1(CN(C)C(c2cc(-c3ccncc3)nn2C)=O)ccnc2ccsc12 c1(C(C)OC)nc(C(=O)NC(C)(C)CCNC(=O)C(C)CC2CC2)cs1 c1(C(=O)NC2CCCN(C(c3c(C)scn3)=O)C2C)cnn2ccn(C)c12 C(=O)(C1=CCCC1(C)C)NCCC1(CNC(C(CCC)CC)=O)CC1 C(CC(=O)NCCn1cc(C(O)CSC)nn1)(NC(COCC)=O)OCC C=CCC(CNC(c1cnnn1C=C)=O)C(=O)NC1(c2nn[nH]n2)CC1 C1(NC(c2ccc(C(C)(C)OCC)cc2)=O)C2CC1N(C(=O)C(C)C1CC1)C2C N1(C(C23CCC(OC)C2C3)=O)CCOCC(C)(CNC(C2CCN2C)=O)C1 C1(C(N(CC(=O)OCC)C)=O)CC2(CCN1C(=O)COCCOC)CC2 CC(C)C(N=c1[nH]c(Cl)ncc1N)C(=O)Oc1cccc(C(F)(F)F)c1 C1(CN(C(=O)C(c2ccccc2)NC(C2CC2(Cl)Cl)=O)C)CCCC1(C)C C(=O)(CC(C)(C)C#N)N(C)Cc1cccc(CNC(=O)CCN2CCOCC2)c1 C1(C)(C(=O)O)CCN1C(=O)CCn1cc(C)cn1.c1(CNCC)ccco1 NC1(C(=O)NCCc2ccc(CN3CCCC3)cc2)CCCS(=O)(=O)C1 C=CCCCC(C(=O)N(C)Cc1cncnc1)NC(=O)CC1(C)CCOC1 C(=O)(CCCC(C)(C)C)NC(CN(C(=O)CC1CCCC1C)C)=O N1(C(C(C)(C)SC)=O)CC(CNC(C2(SC)CC2)=O)OC(C(F)(F)F)C1 C=CCN=C(NCCCSCC)NNS(=O)(=O)CC.C1(C)C(C)(C)C1(F)F c1(-c2cccc(SC)c2)ccc2cc(C(=O)NC34CCN(CC3)C4)sc2c1 C(=O)(CC(F)(F)C(C)C)NCC1(NC(C(C)(C2CC2)OC)=O)CCC1 C1(C(=O)NC(CCC)CC)CCN(C(=O)CCc2cscn2)C(C)C1 c1(OC(C(=O)NCCN(C(C2(OC)CC2)=O)C)C)ccccc1C Cc1ncn(C)c(=O)c1C(=O)NC1CS(=O)(=O)CC1NC(=O)CCC1(C)CC1 c1(NCC(CC)(CC)NC(c2cnc(O)c(C)c2)=O)cccc(OC)c1[N+](=O)[O-] c1(CC(=O)NCc2c(CCNC(C)=O)ocn2)cccc2cnccc12 c1(N(CCCN(C(C)=O)C)C)cc(S(=O)(=O)NCC(O)C2CCC2)ccc1C#N C1(CC=C)(NC(=O)CC)CCN(C(=O)C(C(C)C)NC(c2ccccc2)=O)C1 N1(C(c2cc(CNC(C(CC#C)C3CC3)=O)on2)=O)C2CCC1CC(F)C2 C(=O)(C(CC)CCOC)N(C(C(=O)NCc1c(CC)nn[nH]1)C)C N(C1CN(C(C2(C3CCC3)CC2(F)F)=O)Cc2ccccc21)C(c1ccc[nH]1)=O c1(CNC(C2CCC(NC(=O)Cc3ccsc3)C2)=O)cc(Cl)nc(Cl)c1 CC(C)(C)C(=O)NCCCC(c1ccccc1)NC(C1(CCN(C)C)CC1)=O c1(C(C)(C)CC2CC2)[nH]c(=NC2CC(CO)C2)nc2scnc12 N1(C(C(C)SCCCC)=O)CC(F)CC1CN(C)C(c1noc(CC)c1C)=O c1(C(=O)NCC2C(NC(=O)CCc3cnco3)CCC2)cn(CCC2CC2)nn1 c1(CCC(=O)NCC2C(NC(CC3(C)OCCO3)=O)CC2)ccc(Br)nc1 N1(C(C23C(C)OC(C)(C2)C3)=O)CCCC12CCN(C(c1sccc1Cl)=O)C2 N1(C(C(c2cccc(C)c2)O)=O)CCC(NC(C2CCCN2C(N)=O)=O)C2CC12 C1(NC(C2CCC(C)C2)=O)CCN(C(c2cn(CC3CCCO3)nn2)=O)CC1F CC(CCOC(=N)O)C(=O)NCC1CN(c2ncns2)CCO1 c1(OC)ccc(C(=O)N(C)CCNC(C23CCC2C3)=O)cn1 Cc1cccc2cc(C(N3CCC(C)N(C(c4nonc4N)=O)CC3)=O)oc12 C(=O)(CS(C)(=O)=O)NCC(C(=O)NC(C)Cn1ccnc1)N(C)C N1(C(CC(=O)OCC)=O)C2CCC1CC(F)(CNC(=O)CCCCC(C)(C)C)C2 N1(CCCCNC(C(F)=CC)=O)CCCN(C(=O)C(C2CCC2)OC)CC1 C1(CCNC(C2CC(O)(CNC(CCc3n(C)cnn3)=O)C2)=O)CCCC2CC12 CN1N=C(C(=O)NC2CCC(CNC(c3cncs3)=O)C2)CCC1=O N1(C(CC(=O)OC)=O)CCC(C)(NC(c2cc(-c3ccccn3)c[nH]2)=O)C1 N12C3CCC(C3)C1CC2=O.C1(NC(CN(CC)CC)=O)COCC1C(=O)NC C(N=c1ccn(CC(=O)NC(C)CF)c(O)n1)c1ccc(OC)c(C)c1C N1(C(CCC2(CCC#C)N=N2)=O)CCC2(CCN(C(c3ccc(N)c(Cl)n3)=O)C2)C1 c1(C(N2CCC(N(C(=O)CCC3CCC(C)O3)CCC)C2)=O)cc(O)nc(Cl)c1 c1(COC(C2(CC)CC(C3OCC(CNC(=O)NC)C3)C2)=O)ccc(C)nc1 C1(CNC(c2ccn(CCOC)n2)=O)CCN(C(=O)C(C(C)C)N(C)C)CC1O c1(C(C(=O)NCCCC)N(C)Cc2cccc(Cl)c2)ccc(OC(C)C)c(Br)c1 C(C1C(=O)N1)SC.C(=O)(C(CSC)N(C)C)NC1CCC(CC=C)C1.C1=NC1 N1(C(CC2ON=C(C)C2)=O)CC(NC(=O)CC2CC(=O)C2)C(C2CC2)C1 N1(C(C(C)c2cccs2)=O)CCN(C(c2nncn2C2CC2)=O)CC1C1CCC1 CCC(C(=O)NC1CC(CCNC(=O)CCc2ccc(CO)o2)C1)n1cncn1 c1(SCC)ccc(C(=O)NCC2(OC)CN(C(C3C4CCC3CC4)=O)C2)cn1 C1(CNC(c2cc(CNC(C=C(C)C3CC3)=O)ncc2)=O)CCC(F)(F)CC1 Cc1cc(CNC(C2CC(O)C2CC(=O)NCC23CC(CCO2)C3)=O)cnc1O c1(C(N(CC(CC)NC(=O)CC2CCC(=O)N2)C)=O)ccc2ncnc(O)c2c1 C1(NC(c2n(CC)cnn2)=O)CC(C(=O)NCC(O)CSC)N(C(N)=O)C1 C(=O)(C(C)(C)c1cnn(C)c1)N(C1CCN(C(=O)C=CCOC(C)(C)C)C1)CC c1(C(=O)NCC(C(=O)NCC2(CCO)CC2)OC)ccn2cncc2c1 C1(CCNC(Cn2c(C)nc(C)n2)=O)CCN(C(=O)CS(=O)(=O)C2CC2)CC1(F)F C1(CNC(C(C)(C)SCC)=O)CCC(NC(=O)CC2CCCC(C3CC3)O2)CC1 CC1C(C(=O)N2CCC(NC(C3COC(=O)O3)=O)CC2)=Cc2ccccc21 CC(C)C(O)CC(=O)NCC(c1ccccc1OC(F)F)NC(=O)C1=CC(C)(C)C1 C(=O)(C1=NOC2(CCC2)C1)N1CCC(F)(C(=O)NC(CCCCCC)C)C1 c1(CC(C)NC(=O)C(C2CCCCC2)NC(=O)Cc2ccsc2)cccc(O)c1 C1(C(C)NC(c2cn(C(C)(C)C)nn2)=O)CCN(C(=O)C(F)(F)c2nccs2)CC1 C1(C(N2CCC(SC)C2)=O)CCC(C2CC2)N1C(c1c[nH]c(C#N)c1)=O c1(C(N(CCOC)CC)=O)ccc2c(c1)C1CCC2O1.C12CC1(C(=O)OC)CC2=O C12(CNC(C3CC(C)N(C)C3)=O)CCC(NC(=O)C(C3CCOCC3)F)(CC1)CO2 c1(C(=O)NCCN(C(CC)C)C(C2CC=CC2)=O)ccc2c(c1)NC(=O)CO2 c1(C(=O)OC)ccc(C(=O)NC2CC(CNC(c3ncsc3SC)=O)C3CC23)nc1 C(c1cc(C)ccc1Cl)=CC(N1C(C2CCN(C(CCC)=O)C2)CCC1)=O N12CC3CCCC(C1)N3C(=O)C(=O)C2=O.CCCC(C)N.C(C)(C)C c1(CC(=O)NCC(CNC(C(c2ccccc2)NC(N)=O)=O)F)ccc(O)cc1 n1(CC)nccc1C=CC(N1CC(NC(c2cc(C)oc2C)=O)C(O)C1)=O CCCCC(O)C(=O)NC1CCC(C(=O)Nc2cnc[nH]2)C1 c1(C(=O)NC2C(C)N(C(=O)CC3CC4CCC3O4)CC2)cc2ccc(F)cc2o1 N1(C(C2CCN(C(=O)NC)C2C)=O)CCCC(C(=O)NC2(CF)CC2)C1.C(COC)O Cc1cc(=NC(=O)CSCC(=O)OCC(C)C)[nH]o1.C(C)C(O)CC(F)(F)F C1(C(=O)NC2CN(C(CN(CCC#C)C)=O)CC2C)Cc2ccncc2N1 N1(C(CC(C)(C)O)=O)CCCCC(NC(c2ncnn2C2CCOCC2)=O)CC1 c1(COC)ccccc1C(=O)NC1CN(C(=O)CNC(=O)CCC(C)C)CC1F c1(C(C)NC(C(N(C(C(COC)N(C)C)=O)C)C2CC2)=O)cccc(C)c1 c1(NC(C2(CC#C)CC=CCC2)=O)ccc2sc(S)nc2c1 C#CCCC(=O)NCCN(C)C(C1CCCN1C1CCCC1)=O N1(C(CCCC=C)=O)CCC2CN(C(c3cc(CC4CCC4)c[nH]3)=O)CC2C1 CC(F)(F)CCC(=O)N1CC(NC(c2cc(=O)cc[nH]2)=O)CC(O)C1 C1(NC(C2COCCO2)=O)CC(NC(C2CC(F)(F)CS2)=O)C(O)C1 CC1CCc2c(C(N3CCCC(CO)(NC(=O)CCOC4CC4)C3)=O)csc2C1 O=C(C#CC1CCC2(CC1)OCCO2)NC1CC(NC(c2cscc2F)=O)C1 C=CC1(CC(=O)NC(c2ncnn2C)C)CN(C(c2cnnn2C2CC2)=O)C1 C1(C(=O)NC(CC#C)CC#C)CC(F)(F)CN1C(=O)CCCC(=O)N(C)C c1(C(=O)NCCCOCCCOCC)cnoc1CC(C)C.C1(C(=O)O)CC1F C1(C(=O)OC2(n3ccnn3)CC2)CN(C(C2N(C(C)=O)CCC2)=O)CC1(C)C c1(CN2CC(NC(c3cc(F)cc(Cl)c3)=O)C(F)C2)c(O)ccc(F)c1F c1(CNC(c2c(N)c(Cl)ncc2)=O)ccc2ncccc2c1 Cc1ccc(C(=O)NC2CC3(C2)CC(C(=O)NCC2C(C)C2C)C3)cc1O CCC(C)CC(C(=O)Nc1ccncc1SC)N(C(=O)C(C)NC(C)=O)C C1(C(N(C(CNC(c2nc(C(C)C)sc2)=O)C)C)=O)CC2(COCCO2)C1 N1(C(C(C)SC(C)C)=O)CCC(CNC(c2cnncc2O)=O)C(O)C1 c1(C(=O)NCC(C)N(C(c2ccccc2SC)=O)CC)cc(F)c(CC)cc1F c1(C(=O)OC)cc(Cl)cc(NC(C2CN(Cc3ccnc(CO)c3)C2)=O)c1OC C1(CNC(CN(C)CC)=O)CN(C(C2(F)CC2c2ccccc2)=O)CC1(F)F CN1CC(=O)NC(CC(=O)NC2CN(C(=O)C(=Cc3cnc[nH]3)F)CC2O)C1=O c1(OC)ncccc1CC(=O)NCC1(C)CC(NC(C23CCC2C3)=O)C1 Cc1ncc2n1CCN(C(C1COC(CNC(c3cccc4ccoc34)=O)C1)=O)C2 N1(C(CNc2ncc(C(=O)OC(C)(C)C)nc2)=O)CC2CC1CN2C(=O)C(N)=O c1(C=O)ccc2cncn2c1.C1(CC)CCN(C(=O)CC2COCC2O)CC1 c1(C(=O)NCC(=O)NC)nn(-c2ccccc2F)c2c1CCC2 N1(C(c2ccc(N)cn2)=O)CC2CC1CN2C(c1cc(SC(F)(F)F)c[nH]1)=O CCCC(CC)CCC(=O)NC(C)C(CO)NC(C1CCC(F)CC1)=O N1(C(COC(C)(C)C)=O)CC(O)(C(F)C(=O)NCC2CCOC2)C1 c1(NC(C(C2CCCN(C(c3n[nH]c(=N)[nH]3)=O)C2)C)=O)c[nH]ccc1=O CC1(C)OC(=O)CC1C(N1CCN(C(=O)CCc2nc(C3CC3)no2)CC1)=O CC(F)(F)C(F)(F)CC(=O)NCC1(C)CN(C(C2CC=CC2)=O)CCO1 Cc1cc(=O)c(C(N2CCCC2C(C)(C)C(=O)NC2(CO)CCC2)=O)c[nH]1 c1(C(N2CC(C(=O)Nc3c(C(=O)NC)cccc3)C(F)C2)=O)ccc(Br)cc1I N1(C(C(COC)(C)O)=O)CCC(F)(F)C(CNC(=O)COCc2ccncc2)C1 c1(C(N2CC(OC)(CNC(=O)C(C)(C)C3CCCC3)C2)=O)cnc(F)c(Cl)c1 N1(C(C=Cc2ccc(CC)cc2)=O)CCCC2(CCN(C(=O)CCSC)C2)C1 C(=O)(C(CC(F)F)c1ccccc1)N(CCNC(=O)CCc1nc(=N)[nH][nH]1)CC C(=O)(CCCC(=O)N1CC(F)(CNC(=O)C(c2ccc(OC)cc2)C)C1)NCC CC1(F)CCCCN(C(=NCc2ccnc(-c3ccco3)c2)NCC(F)F)C1 c1(C(N(CCNC(C(C)OCC)=O)CC)=O)ccc(F)c2ccccc12 c1(C(N2CCC(NC(CCC=C)=O)(CF)C2)=O)cc(C)nc(C)c1 C1(CNC(C2(OC)CCSC2)=O)CCCCN(C(c2cc(OC)ccc2O)=O)C1 C1(OC)CC(CNC(=O)CCCN2CCOCC2)N(C(=O)C=CC2CCCO2)C1 C1(NC(c2c(C)cc[nH]2)=O)CC2CC(NC(=O)C(F)CC3CCCC3)C2C1 n1(CC)nc(C(F)(F)F)cc1C(=O)NC(C)C(C)NC(=O)Cn1cccnc1=O CCCC(CCC)C(=O)NCC1(OC)CN(C(=O)Cn2c(C)cc(O)cc2=O)C1 C(CC(C(=O)Nc1ccc(Cl)cc1)NC(=O)CC1(C#N)CC1)=CC N1(C(c2cccc(COC)c2)=O)CCN(C(c2cc(C#N)c[nH]2)=O)C(C)C1 c1(C(=O)NC(C(C(C)C)NC(c2n[nH]cc2Br)=O)C)ccc([N+](=O)[O-])[nH]1 C1(C(N2CC(O)(CCC)C2)=O)CC2C=CC1N(C(=O)CC(C)OC)C2 c1(OC)ncccc1C(=O)NC1(CCNC(c2csc(Cl)c2)=O)CC1 C1(CC)CC(C(=O)NCCOC)CCN1C(=O)Cc1cscn1 C1(CC)CCN(C(=O)CC2CC3(CCC3)C2)C1C(=O)NCCCS(C)=O Cc1cccc(C)c1C(=O)NC1CC(F)(CNC(C23CC(CO2)C3(C)C)=O)C1 C1(CC(=O)NCC2(O)CN(C(C3C(C)(C(=O)OCC)C3)=O)C2)CN2CCC1CC2 N1(C(C=Cc2cncc(C)c2)=O)CC2(COC(CNC(=O)C(C)C3CCC3)C2)C1 CCCC(C)CC(=O)N(CCCCCCNC(=O)CCn1cccn1)C C(C(C)(CC(C)C)NC(=O)C1=NOC(C(C)(C)C)C1)NC(c1c(C)cc(C)s1)=O N1(C(C2C(OCC)CC2)=O)CCN(CCc2ccc(F)c(F)c2)C2(CCC2)C1 C#CCC(C)(C(=O)NCC1(SC)CCCOC1)NC(=O)C(COC)OC c1(C(N2CC(C(C)=O)C(C)C2)=O)cc(C)c(C(=O)O)c(C)c1 C(=O)(N=c1cc[nH]c2cc[nH]c12)C1C2(CCN(Cc3n(C)cnc3Br)CC2)C1 c1(C(=O)NC2CN(C(C(C)C3CCC3)=O)CC23CCC3)ccc(F)c2[nH]ccc12 N1(C(c2c(OC)c(Cl)ccc2)=O)CCN(C(C2CCCSC2)=O)C2CCC12 c1(CC(=O)NCCC2CCCN(C(C(C)C3CCC3)=O)C2)ccc(C#N)c(Cl)c1 N1(C(C2N(CC)CC2)=O)CCOCC1CC(N1CC2CC2C1)=O CCC(C)C(C(=O)Nc1nnc(-c2cccnc2C)n1C)N1CCCCC1=O C1(NC(CC(=O)N(C)C)=O)CN(C(=O)C=C2CN3CCC2CC3)C2(CCCC2)C1 C1(NC(CCC(C)(C)C)=O)CN(C(c2cccc3[nH]ccc23)=O)C2CCC1C2 c1(OC)ccc(Cl)c(C(=O)NCC(=O)NCC(C2CCCC2)NC(=O)CO)n1 Cc1cc([N+](=O)[O-])ncc1C(=O)Nc1ccc2c(c1)COC2 C=CC1CCCN(C(c2ccnc(CNC(c3ccsc3C#N)=O)c2)=O)C1 c1(C(=O)NC(C(N2CC=C(C)C2)=O)C)cc(F)ccc1F c1(NCc2ncc(-c3ccc(F)c(O)c3F)cc2)cccc(C2=CCCCC2)n1 c1(C(=O)NC2C(CNC(C=CC(C)(C)C)=O)C2)cc([N+](=O)[O-])cnc1N C1(NC(C2(CC)CCCO2)=O)(CO)CCN(C(=O)Cc2cnn(C)c2)C1 N1(C(CCc2cc(C)no2)=O)CCN(C(C2(O)CCOC2)=O)CC(C)C1 C(C1CCN(C(=O)CCN2CCCCC2)CC1)=CC(=O)NC1C(C(C)C)C(O)C1 c1(CNC(C2C(CCC)C2)=O)ccccc1CNC(C1CCCC12CC2)=O C1(NC(c2nc(C)oc2)=O)CC2CN(C(=O)C(CC(C)C)n3ccnc3)CC2C1 N1(C(CSCC#C)=O)CCC2(C=C(C(=O)NCC(O)CC3CCCC3)C2)C1 C1(C(=O)NCC2(C(N3CC(N(C)C)C(F)C3)=O)CCCCC2)CCC2(CC1)CC2 CC1CCC(=CC(=O)NCCC(C)(C)CNC(=O)C(c2ccc(Cl)s2)C)CC1 c1(C(N2CCC(CO)(NC(C3CCCCO3)=O)C2)=O)cc([N+](=O)[O-])n[nH]1 C1(CNC(C(CNC(C=Cc2cn(C)nn2)=O)O)=O)C2CCCCCC12 C1(NC(CC2CC(OC)C2)=O)CN(C(c2ccc(C(C)(C)C)cc2)=O)CCC1C C1(C(=O)NC2CC(CNC(C(C(C)O)C)=O)C2)CCCC2CCCCC12 C1(CC=C)CCCN1C(=O)CCC1(NC(=O)CC2(OCC)CCC2)CCC1 C1(C(=O)NCCC(C)(C)N(C)C)CC(NC(c2nccn2C)=O)C(O)C1 C(=O)(C(C(=O)N1CCC(OCCNC(=O)CCCSC)CC1)NC(C)=O)OCC Cc1cccc2c1C(NCC(O)C(F)F)CCC2 c1(CC(=O)NCCC(Cc2ccccc2)NC(C(C)C)=O)ncn2c1CCC2 Cc1cccc(F)c1CC(=O)NC1(C)CCN(C(=O)CC(C)C)CC1 N1(C(C(C)=CC)=O)CCCC2(CC(NC(c3sc(Br)cc3F)=O)CO2)C1 c1(C(C)=O)cc(C(=O)NC2CCN(C(=O)Cc3nccc(C)n3)C2)oc1C C1(NC(C)=O)CCN(C(=O)COc2cccc(C(C)C)c2)CC1C S(=O)(=O)(c1cc(C(F)(F)F)cnc1C(=O)O)N1C(C(C)C)CCCC1 c1(NC(C(C2(C)CN(C(=O)OC)C2)O)=O)ccnc(C(=O)OC(C)(C)C)c1Cl CC1C(NC(c2cc(C(F)(F)F)ccn2)=O)CCCN1C(c1cnsc1)=O CN1CCN(C(c2occc2C2CC2)=O)CC1CNC(=O)CCc1cnn(C)n1 c1(C(=O)NCC(CNC(c2ncnc(O)c2Cl)=O)F)cccc2c1NCCC2 c1(C(=O)NC2CC(NC(CSC)=O)C23CCC3)nnn2cc(C)nc(O)c12 Cn1cncc1C(=O)OC(C)(C)C.C1(=O)C(=O)C=CCCCCO1 CC1=NOC(C(=O)NCC2(C3CCCCO3)CC2)C1C CCC(C)C(C(=O)NCCNC1CCN(c2ncc(C(N)=O)cc2Cl)CC1)OC c1(C(N2CCC(O)(CN(C(=O)CC3OCCO3)C)C2)=O)ccsc1S(N)(=O)=O c1(C(=O)NCC(CC=C)NC(C2CC2C(=O)OC)=O)ccc(CC)nc1O N1(C(C(CCCC)NC(=O)CCc2ccncn2)=O)Cc2c[nH]nc2C(C)C1 C1(NC(C(N2C(CCCCC=C)CCC2)=O)=O)C=CC(=O)N=N1 c1(C(=O)NC2CC(N(C(C(C(C)C)SC)=O)C)C2)cc2cc(Cl)ccc2n1C N1(C(c2c(C)nc(O)s2)=O)CC(C(N2CC=C(CO)CC2)=O)C(C)(C)C1 C(CCC)(CCC)NC(C(CC=CC)NC(=O)Cc1cccc(O)c1)=O c1(C(N2CCC(CS(C)(=O)=O)C2)C(=O)NC)ccn(CC(F)(F)F)n1 C1(OC)CC(CNC(C2(C)CS(=O)(=O)C2)=O)N(C(=O)CCCc2csc(C)n2)C1 C1(O)(CCNC(=O)CC(O)C2CC2)CCCN(C(=O)CCCc2cnn[nH]2)C1 c1(C(N2CC3CC(C)N(C(C(CC)C)=O)C3C2)=O)cnc2sc(C)cn2c1=O C(C(C)(C)C(=O)NCC(C1CCN(C(=O)C(c2cccnc2)O)CC1)O)N(C)C C(C)(CN=c1ccnc(NC(CC(F)F)c2ccccc2)[nH]1)OC C1(O)(CNC(c2c(CCC)nns2)=O)CCN(C(=O)CCN2CCOC2=O)CC1 c1(NC(C2C3CCC(CN(C(COC)=O)C3)C2)=O)cncc2c(F)cccc12 CC(C)C(O)CC(=O)N1CCCC(CCNC(c2ccc(Cl)s2)=O)CC1 S(=O)(=O)(c1ccc(C(C)(C)C)cc1)NC(C1(C(=O)O)C(C)C1)=O CC1CCN(Cc2cn(CCCCCCC#N)nn2)C1.C(=O)(CC1(C)CC1)N c12ccc(c(Br)c1)S(=O)(=O)NCc1csc(n1)CCN2.CC1COCC(CO)O1 c1(C(=O)NC2CC3(C2)CN(C(C2CC(C4CC4)C2)=O)C3)c(Cl)ccc2c1OCO2 c1(C(=O)NC23C(NC(c4c(C)con4)=O)CC(CC2)C3)cccc2ccn(C)c12 c1(C(C)C)cccc(S(=O)(=O)N2CCC3CCN(C(C4CCC4)=O)C3C2)c1 c1(C(=O)NC(CNC(Cc2c(OC)cccc2F)=O)(C)C)csc2ccncc12 C(=O)(CCCC(=O)OC)N1CCC(N(C(=O)COC)C2CC2)C1.C#CCO C1(CNC(CCc2ccc(N)cc2)=O)CN(C(=O)COC2CCOC2)CCCO1 CC(C)CC(CNC(=O)C(C)(C)Nc1cnns1)NC(=O)CSC1CCCCO1 c1(COC)noc(C(F)(F)F)n1.c1(CC2CC3CN(C3)C(=O)N2)ccccc1 C1(NC(C2(C)CCSCC2)=O)CCC2(CCN(C(C3C=CCS3)=O)C2)C1 c1(C(=O)NCC2C(NC(=O)CCc3cnoc3)CCCC2)cc2c(nn1)OCCS2 CN1CCCC(c2cn(CC3CCN(C(c4ccc(F)cn4)=O)CC3)nn2)C1 C1(C(N2CC(C(C(C)C)O)C2)=O)CCCCCN1C(=O)CCc1nc[nH]n1 c1(C(=O)NCC(C)(CO)NC(c2cn[nH]c2)=O)ccc(-c2ccccc2)cc1Cl c1(C(N2CC3C(C2)N3C(c2ccc(F)nc2)=O)=O)cc(Cl)cnc1Br N1(C(CCn2c(CC)ncc2)=O)CC2CCC1CN2C(=O)CC1CCCOCC1 C=C(C)CC(C(=O)N=CC(=O)OC)NC(=O)C(C)CCCOC Cc1occ(C(F)(F)F)c1CC(=O)N(CCNC(C1CCCOCC1)=O)C(C)C C(CC(C(=O)NCC1CCCC1O)NC(=O)Cc1ccc(C)nc1)SC c1(CCNC(C=CC(C)NC(CSCCC)=O)=O)cn[nH]c1 C(=O)(C(C)(C)C(=O)OC)NC(CC)CNC(c1ccnc(C(N)=O)c1)=O C1(NC(C2(CC=C)CC2)=O)CN(C(=O)CCCC(C)O)Cc2nccn2C1 C1(C)(C(N(CCNC(C(COC)NC(C)=O)=O)CCOC)=O)CCc2ccccc21 N#CCCCCCC(=O)N1CCCC(NC(C2CCCOC2)=O)C1 N1(C(CCc2c(C)noc2Cl)=O)CC2CCC(C1CO)N2C(C1CC(CF)C1)=O N12CCc3sc(nc3C1)C2=O.c1(NC(C)=O)ccc2c(c1)CCCC2 C=CC(CC)C(=O)NCC(C)(O)CNC(C1CCC(=O)N1)=O C1(CC=C)(C(=O)NCC(C)O)CCN(C(C2CC(OC)(OC)C2)=O)C1 c1(C(N2CCCC2C2CCCN(C(C3CC(F)(CO)C3)=O)C2)=O)ncccc1O c1(-c2nc(C3C(C)C3C)nn2C(C)C(C)(C)C)n[nH]c2c1CC(C)(C)CC2 CCCC(CCCS(C)(=O)=O)C(=O)N1CCC2C(NC(=O)C3=NNC(=O)C3)C12 C(c1ccccn1)=CC(N1CC(C(C)NC(=O)Cn2cnc(=N)[nH]2)C1)=O c1(C(=O)NC(C2CCCC2)CNC(=O)CCN2CCCC2)nccn2cccc12 c1(C(=O)NCC2C3CN(C(C4CC45CC(O)C5)=O)CC23)cn2c(n1)CCCC2 Cc1ccc(C(=O)N(C)CCOCCNC(=O)CC(F)(F)Br)c(N)c1 C1(c2cc(CC)on2)CCCCN1Cc1ncoc1C(C)(C)C c1(C(C(=O)NCCCSCC)N(C(C)C)CC2CC2)cc(Cl)ccc1Cl CCCC(C(=O)N(CC(N1CCCC1CC(=O)OC)=O)C(C)C)OC Cc1cc(C(=O)C(N2CCCC2CCNC(C2CC2C(F)(F)F)=O)=O)cs1 N1(C(c2snc(C)c2N)=O)CCC2CCN(C(c3nocc3Cl)=O)C2C1 CC12CC(C(N3CC(=C(F)CNC(=O)CCC4CC4(C)C)C3)=O)(C1)C1(COC1)O2 c1(C(C)C)ccc(NC2CC3C(NC(=O)OC(C)(C)C)C3C2)c([N+](=O)[O-])c1 n1(CC(N2CC(NC(C=COCC)=O)C3(C2)CC3)=O)c(C)nc2ccccc12 c1(NC(C2CC(F)CN2C(c2ccccn2)=O)=O)cc(F)c(Cl)cn1 C(=O)(C1=CNS(=O)(=O)N=C1C)N1C(CCOC)CN(C(c2cncn2C)=O)CC1 CC(C)(CO)C(O)C(=O)Nc1cc(Cl)nc(C2CCCO2)n1 C1(C(N2CC(CC)(NC(=O)Cn3nccn3)C2)=O)CC12C1CC3CC(C1)CC2C3 n1(CC(=C)C)c(N2CCOC(C(N)=O)C2)nnc1-c1ccnnc1C N1(C(C2N(C(c3c(OC)nccc3)=O)CCN(C)C2)=O)CCCCC(C)(F)C1 C1(NC(C(=O)OCC)C2CC2)CCC(C)CN1C(=O)CC1CCCCCCC1 CC1OC(=O)NC1C(=O)NC1CC(O)CC1O.C1C(=O)NOCC12CC2 c1(C(N2CC(NC(c3cc(CC)on3)=O)C(C#N)C2)=O)cnc2cc(Cl)ccn12 C(N=c1ccc(Br)c(S(=O)(=O)NCc2ccccc2)[nH]1)C1(N(C)C)CCCC1 c1(C(=O)NCC2(F)CN(C(=O)C=CCF)C2)c[nH]c2ccncc12.C(C=O)=CCC C1(COC)CC(CNC(=O)CCC2(O)CCC2)N(C(=O)CCCn2cccn2)C1 c1(CC(=O)NCC(C)(C)NC(=O)CS(=O)(=O)NC2CC2)cc2ccccc2o1 c1(C(=O)OCC)cc2c(C)nn(CC)c2s1.c1(OCC)ccc(CCC(=O)O)cc1 c1(C(N2CCCC(C)C2c2cn(CCCCO)nn2)=O)noc2c1COCC2 c1(C(=O)NCC(CC)NC(c2cnn(C)c2N)=O)cc(C)c(C#N)cn1 N1(C(=O)CCCCC2CC2)CCC2CCN(c3nc(Cl)ncc3C3CC3)CC2C1 C1(NC(C=CSC)=O)CN(C(=O)CC2CCCCO2)CC1c1ccc(F)cc1 CCCC1C(=O)N1.C(CCC1CC1)(C(=O)N1CCSCC1C)N(C(N)=O)CC C1(N(C(c2n(CCC)nc(C)c2)=O)C)CC2CCC(C1)N2C(c1cc(Cl)c[nH]1)=O c1(C(N2CCN(C(CCC#N)=O)CC2)=O)cc2ccc(F)cc2[nH]1 N1(C(C2(N(C)C)CC2)=O)CC(NC(C2(C)C=CCCC2)=O)CC2(CCOCC2)C1 c1(C(=O)NC(C(C)C)CCN(C)C(c2cnccn2)=O)cc2c(F)cccc2[nH]1 CC12CC(CNC(c3ccc(F)cc3)CO)(C1)OC2C(F)(F)F C(=O)(C(CC(C)(C)C)OC)N(CCOC)CCNCC.c1(CC(=O)N)ccc(C)nc1 c1(C(=O)NCC(C2CCN(C(C3CCC3)=O)CC2)(C)C)ccc(Br)cc1N Cc1cccc2c(C(N3CC4(NC(C5CCCCC(=O)N5)=O)CC3C4)=O)n[nH]c12 CC1(NC(C2CCC2CCNC(=O)C(=CC2CCCCC2)F)=O)CCOCC1 C1(CNC(=O)CCc2cnoc2)CN(C(c2ccc(C3CC3)o2)=O)CC1O c1(C(=O)NCC2CC(CNC(C3(CC#C)CC3)=O)OC2)cnc(=N)[nH]c1 c1(C(C(=O)NCC2N(C(CCCCC#C)=O)CC=C2)CC)ccc2c(c1)OCO2 C1(NC(C2CC(C#C)(O)C2)=O)CC2(C1)CN(C(=O)Cc1cc(C)[nH]n1)C2 N1(C(C2(N(C(C(N3CCCCC3)C)=O)C3CC3)CC(O)C2)=O)CC2CN(C)CC2C1 CC1CN(C)CC1NC(c1ncoc1CNC(=O)CN1CCCNC1=O)=O C1(C)(C(=O)NCC(CC(C)C)NC(c2cccnc2)=O)CCC(C)C1(C)C N1(C(COC)=O)CC(CNC(C2(Br)CC2(F)F)=O)(OC)C1 CCCCC(CC)CC(=O)NCCCC(C)(C)C(=O)NCC(O)CC1CCCC1 CC(C(C)C(=O)N1CC(F)CC1C)NC(c1cc(C(N)=O)c[nH]1)=O C1(F)(CNC(=O)CSC2CCOC2=O)CCN(C(C2CC(O)(C(F)F)C2)=O)C1 c1(OC)cc(F)c(C(=O)NC2COCCN(C(=O)CCNS(C)(=O)=O)C2)c(F)c1 c1(CC(=O)NCC2(F)CCCN(C(=O)CCF)C2)ccc2sccc2c1 n1(CC(=O)OC)c(N2CCC(C(C)(NCc3cccc(NC)c3)OC)C2)nnc1C c1(C(=O)NCCn2cc(-c3ccc(C)cc3)nn2)coc2c1CS(=O)(=O)C2 C(=O)(C1=CC2(CCOCC2)C1)NCC1N(C(C2CC(=C)C2)=O)CCC(C)(C)C1 N1(C(C(c2c(C)n[nH]c2C)C)=O)CCCC2CN(C(C3CC(C)(C)C3)=O)CC12 c1(CN(C(c2nccc(OC)c2)=O)C2CC2)cc2ccccc2o1 c1(C(N2CC(N(C(C3CC(SC)C3)=O)C)C(C)(C)C2)=O)ccc(S(C)(=O)=O)o1 c1(NC(C2CCCN(Cc3cc(O)ccc3F)C2)=O)ncnc2[nH]c(Br)nc12 C(CNC(=O)C(CC)OC(C)(C)C)(C(C)(C)C)NC(CCOCCOC)=O C(=O)(N=c1ccn(CC2CC2)[nH]1)C1C(OC)CN(C(C2CCNC(=O)C2)=O)C1 c1(C(N(CCCC2(NC(=O)CCc3ccon3)CC2)C)=O)nn(C)cc1Cl N1(C(CC(CCC)C)=O)CC2=C(C1)CN(C(=O)C(CC)=CC)C2 CCC(CC(=O)NC1(c2nnnn2C)CC1)N(C)C(c1cc[nH]n1)=O C1(=O)C(C(F)(F)F)O1.c1(C(=O)NCC(C)N(C)C)ccccc1 C1(OC)CC(C(N2CCN(CCCCCNC(=O)CC3CC3)CC2)=O)CC1OC C(C(F)(F)C(=O)NCC(C)N(C)C(c1cccc(CC(=O)OC)c1)=O)OC CCCCC(C(=O)NC1CC(CNC(c2cc(F)cc(F)c2)=O)C1)N(C)C C1(C2CCN(C(=O)CCCc3cccnc3)C2)(NC(=O)C(=O)C(F)(F)F)CC1 C1(C(N(CC(C)CNC(c2cccs2)=O)C)=O)CNC(=O)CC1C C1(N(CCC)C(c2cc(C)co2)=O)CCN(C(=O)CCSC)C1 CN1CC(=O)NCC1C(N1CCOCC(CNC(=O)C(F)=CCCF)C1)=O c1(C(N2CC(C)C(NC(=O)CC3CC(C)(C)C3)CC2)=O)ccc2ncn(C)c2n1 C1(NC(c2nnnn2CCC2CC2)C(C)c2cccs2)C2CCCC1CC2 CCC(CC(C)CO)NC(=O)CCCNC(C1(O)CCCC1)=O c1(CCC(N2CCC(C(=O)NCC3(C(=O)OCC)CCC3)C2)=O)ccc(F)nc1 C1(CN(C(=O)Nc2ccoc2)CC)CN(C(=O)Cc2cnccc2C)CCCO1 C(C)(C(C(=O)NC1CCCC1CF)C(C)C)NC(c1n(CC)nnc1)=O c1(C(N2C(C(=O)NCCCCN(C)CC)CC2)=O)oc(C2CCC2)nc1C C1(NC(c2occ(C)c2C)=O)C2CC3CN(C(=O)C(O)C4CC4)C1C3C2 Cc1cccc(F)c1CC(N1CCC(NC(C2(C(F)(F)F)CCCC2)=O)CC1)=O C1(NC(C(CC)CC(C)C)=O)CCC2(CC1)CN(C(c1csnc1C)=O)CCO2 n1(CC(=O)NC(CC)CN(C(=O)C(C2CCCC2)OC)CC)nc(C)c(Cl)c1C C#CCC(C(=O)NCCC1(NC(c2cc(C3CC3)ccn2)=O)CC1)C1CC1 C1(C(C)C)CC(c2nnnn2C2CC2)(NCc2sc(C(N)=O)cc2Br)CS1 C1(CNC(Cc2c(C)n(C)nc2)=O)CC2(CCN(C(c3cnns3)=O)C2)CO1 C1(C(C)C)(NC(=O)NC(c2ccnn2C)C)CCN(c2ccccc2)C1=O C1(O)(C(C)NC(=O)C=C2CCCC2)CCN(C(=O)CC(C)(C)O)C1 N1(C(C(COC)COC)=O)C(C)CC2CN(C(=O)CSc3ccc(Cl)cc3)CC12 c1(C(=O)NC2CN(C(C3CC3C(N)=O)=O)C3(CCC3)C2)c[nH]c2cccc(F)c12 C1(CNC(C2(CSC)CC2)=O)CC2(C1)CN(C(c1cncc(Cl)c1C)=O)C2 Cc1nc(NC2CC2)sc1C(=O)NC1CN(C(=O)CCN(C)CCO)C1 N1(C(CCN(c2cn(Cc3conc3C(C)(C)C)nn2)C)=O)CCS(=O)(=O)CC1 c1(C(=O)NC(CC)CNC(C2(Cl)CC2(C)C)=O)ccc([N+](=O)[O-])c(O)c1 n1(CC(=O)NCCC2CN(C(c3c[nH]c(C)c3C)=O)CC2C)nc(C)n(C)c1=O c1(NC(C2C(NC(=O)CCC3CCC3)CCC2)=O)cccc([N+](=O)[O-])c1F CN(C)NC(=O)CCC(=O)N(CCCC(N1CCC(N=[N+]=[N-])C1)=O)C c1(OCC)cncc(CCC(=O)NCC2CCCCC2NC(C2OCCC2C)=O)c1 N1(C(C(C2CCN(C(C3C4CCC(F)C34)=O)C2)C)=O)CCC2CCC(C1)S2 C12(C(=O)NCC3(CNC(C4CCO4)=O)CC34CCC4)CCCC(CO1)C2 Cn1cc(C#N)cc1C(=O)NCC(C)(O)CNC(c1csc(C2CC2)n1)=O C(N=c1[nH]c(C)nc(Cl)c1C)C1OCCCN(C(C2C(OC)CCC2)=O)C1 CCCC(C(=O)OC)C(=O)NC(CC(=O)N1CC(OC(F)F)C1)C(F)F c1(C(=O)NCC2C(NC(c3cc4c(s3)CCC4)=O)C2)cccc(C(F)(F)F)c1Cl CC1CN(C(=O)CCCn2c(O)nnc2O)CC(C)C1NC(c1cocn1)=O C(CC)(CCCC(=O)N(CC(C)C)C)NC(C(C)OCCC=C)=O C1(C(=O)OC)C(F)(F)C12CC(C(=O)NCCC(C)(C)NC(c1coc(C)n1)=O)C2 C1(NC(CC=C=C)=O)CC(CNC(C2(CCN3CCCCC3)CC2)=O)C1(C)C C1(CNC(c2cc(C)c(O)nc2)=O)CCN(C(C2CCS(=O)(=O)C2)=O)CC1(F)F C(c1ccc(=N)[nH]c1)=CC(=O)NC(C)CC(C)NC(=O)C(N1CCCC(O)C1)C C1(O)(CCNC(CCSC)=O)CCN(C(=O)CC(C)c2ccco2)CC1 N1(C(C(C)=C(CC)C)=O)CCCC(C)(NC(c2cncc(OC)c2C)=O)C1 C1(CC)CCC(C(=O)NC2(C(=O)NCCC3CC(C)(C)C3)CC(F)C2)O1 c1(CC(=O)NC2CC(C(N(C)CC3(C#N)CC3)=O)C2)sccc1Cl C1(C(=O)NCC(C)=CC(=O)NC(c2cscn2)C)(OC)CCSC1 C1(C2CCCN(C(C)=O)C2)(C(=O)NC(C2CCOC2)CNC(CCC#C)=O)CC1 Cc1cnc(N(C2CCN(C(=O)CC3COCCO3)CC2)C)nc1 CC1CN(C(C2COCC2NC(C2C3CCC(F)(F)C23)=O)=O)CC(C)(C)C1 C1(NC(C(C(C)C)S)=O)CCOC2(CCN(C(=O)CC3CCC3)CC2)C1 c1(C(=O)NC2CN(C(CSCC(=O)OC)=O)CC2O)coc2cc(C)c(C)cc12 c1(-c2ccc(CC(=O)NCc3cncs3)s2)ccc(F)cc1 C1(C(=O)NCC2(SC)CC2)CCC2CCC1N2C(C1CC(F)(CF)C1)=O c1(OC)cnc(C(=O)NCCOC2CCN(C(=O)C=Cc3nnn(C)n3)C2)cn1 Cc1nn(CC(=O)NC(C)C(C)NC(c2ccc(F)c(O)c2)=O)cc1[N+](=O)[O-] c1(C(c2cncn2C)NCC(c2n(CCSC)nnn2)(C)C)cc(Cl)sc1C N1(C(=O)C=CCN2CCOCC2)CC2CCN(C(C3CCCCC3O)=O)C2C1 C1(C(N(CC(=O)NCCNC(c2ncccc2O)=O)C)=O)CC2(CO1)CC(F)(F)C2 C(C(=O)N(C)CC1CCN(C(c2sc(C(C)(C)C)nc2C)=O)CC1)(C(C)C)OC N1(C(C2CCC(C(=O)OC)C2)=O)CCC(C2CN(C(=O)C=CBr)C2)CC1 C1(NC(c2csc3nnsc23)=O)CCCC12CN(C(C1CC13CCC3)=O)C2 c1(C(=O)NCC23CC2CN(C(c2ncc(Cl)cc2Cl)=O)C3)c[nH]c2ncccc12 N1(C(C23CC(C(=O)OC)(C2)C3)=O)CCC2(CCCN(C(=O)CC3C=CCC3)C2)C1 CC1CN(C(=O)Cc2cccc(OC(F)(F)F)n2)CC1CNC(C1CC1C)=O c1(C(=O)NCCCN(C(C)C)C(C2COC(=O)N2)=O)cccnc1O CCCC(C)(CCC)C(=O)NC1CCCC(NC(=O)Cc2cc(C3CC3)no2)C1 c1(C(=O)OC)ccc(C(=O)N(C)CC2CCCN2C(C2(CC(C)C)CC2)=O)o1 N1(C(c2c(OC)cc(OC)c(Br)c2)=O)Cc2c[nH]nc2CC(C)C1 CC(C)C(C)C(CNC(C1(CC2CC2)CCC1)=O)NC(c1cc(N)cnc1Cl)=O CC(CC(=O)NC1CCCN(C(c2cnc(C3CCCCC3)s2)=O)C1)C(C)(C)C C(=O)(CCCCc1cnn[nH]1)NC1(CNC(C(N2CCC(C)C2)=O)=O)CC1 C1(C(=O)NC(c2nc(C(N3CC(C(N)=O)C(O)C3)=O)co2)C)CC2C(C1)C2(C)C C(=O)(C(CC(F)F)CN)C(=O)CC1CCOCC1.C1(CCNC(=O)CO)CCCC1 N1(C(C(C#CC)(C)C)=O)CC2CC(C(N3CCC(CC)CC3)=O)C(C2)C1 N1(C(C(C(C)C)NC(=O)Nc2ccccc2)=O)CCCC([Si](C)(C)C)C1 c12cc(Cl)c(c(Cl)c1)[nH]2.N1(C(N2CCCC(C(N)=O)C2)=O)C2CCC1COC2 C(=O)(CC(F)(F)CC)NC(CNC(C(CC)c1ccccc1)=O)(C)CO c1(OC)ccc(C(N2CC(CNC(c3nncn3C)=O)C(C)C2)=O)cc1 C=C1CC(C)(C(=O)NC2CC(NC(=O)C(O)Cc3[nH]cnc3C)C2)C1 C(C(C)C(=O)NOCCCOC)N(C(CCOCCCOC)=O)C C1(C)(C(=O)NCCCCCNC(c2cc(COC)no2)=O)CCC(C)=C(C)C1 c1(C(=O)NC(c2cn(Cc3ccccc3F)nn2)C)cnn2c1S(=O)(=O)CC2 C#Cc1c[nH]nc1C(N1CCC(NC(=O)CCc2cn(C)cn2)C1)=O N1(C(C(C)Sc2ccccn2)=O)CC2CCN(C(=O)C3=CC(C)(C)C3)CC2C1 C1(C(N2CCN(CCNC(c3ccsc3Cl)=O)CC2)=O)SC2C=CC1CC2 CC(C)(C#N)CS(=O)(=O)NCCC(c1ccc(Cl)cc1)O C(C)(CC(C)CC(C)C)NC(C)=O.c12ccc(c(C(=O)NCCOC)c1)NC(=O)N2 c1(C(=O)NC2C(C)N(C(=O)CC3CCC3)CCC2)nccc2c(Cl)cccc12 N1(C(C2(n3cc(C4CCCC4)nn3)CCOCC2)=O)CC(OCCF)C2(CC2)C1 C1(CC(=O)NC(CC)CNC(c2csc(C(F)F)c2)=O)CCCCC1F c1(CCC)noc(CCCC(=O)NCC2(O)CC(NC(C3(O)COC3)=O)C2)n1 C(C(C)CC(=O)N1CC(CO)C1)NC(c1cc(C)sn1)=O C(CC(=O)NCCC1CCCOC1)(C(C)(C)C)NC(C(=O)NCC)=O C#Cc1ccc(C(=O)NCC(O)CN(C(=O)C#CC(C)C)C)nc1 C1(NCCNC(=O)Nc2ccc(NC(CCC)=O)cc2)CCCCNC1=O C1(C(=O)NCCC2(CC)CCC2)C(C2CC2)CCN1C(c1ccnc(C)c1N)=O N1(C(=O)C=CI)CC2CC1CN2C(c1cccnc1O)=O N1(C(C2=C(C#N)CCC2)=O)CCCC12CCN(C(=O)C(=Cc1c[nH]cn1)F)CC2 N1(C(Cc2c(C)cccn2)=O)CCC2CCCC12C(=O)NC(C1CCOC1)C C1(N(C(=O)CC(=C)Br)CC#C)CCN(C(=O)CCN2CCC(F)C2)CC1 C(=O)(C(CC(C)C)NC(=O)N)OC.C1(CC)CCN(C(=O)OC(C)(C)C)C1 c1(C(N2C(CNC(C(CC=C)(C)C)=O)CC2)=O)sc2nnc(S)n2c1C Cc1c(CNC(=NCCc2ccc(F)cc2)NCC2(S(C)=O)CC2)cccc1Cl C1(CNC(C(C)OC)=O)CCC(F)(CNC(=O)C(O)Cc2ccc(F)cc2)CC1 C1(NC(c2c(C)oc(CO)c2)=O)CCN(C(c2cc(C#N)no2)=O)CCC1CO CC1(C)CN(C(C2(O)CCCCC2)=O)CCC1O.c12ccc(o1)CNC2=O N1(C(c2nnc(C)s2)=O)CC(CCNC(=O)C=Cc2ccsc2)OC(C)C1 C1(CC)CN(C(c2nnn(C(C)(C)C)n2)=O)CCN1C(c1ncc(C)cc1C)=O c1(C(N2CCC(NC(C(C)(CC3CCC3)OC)=O)CC2)=O)ccn2nccc2n1 Cn1ncc2c(N3CC4(CCC(NCc5ccc(Cl)cc5)C4)C3)ncnc12 N1(C(=O)C=CBr)CCC2(CCCCN(C(c3cccc([N+](=O)[O-])c3F)=O)C2)C1 C12(CNC(CCCCCOC)=O)CC(CNC(=O)C(=O)NCC3CC3)(CO1)C2 N1(C(c2ccc(C=C)cc2)=O)CC2(C1)CN(C(=O)CC1CC(O)C1(C)C)CCO2 C1(NC(=O)C=CC2CCCO2)CC2CC(C1)N(C(c1cc(O)nc(C3CC3)n1)=O)C2 CCC(CC(=O)OC)C(=O)N(CC(C)C#N)CC1(C)CC1.c12cc(ccn1)NC2 O=S1(=O)CCC(S(=O)(=O)N2CCC(NC(c3cc(Cl)c4n[nH]cc4c3)=O)C2)CC1 C(=O)(C1CCCn2c(C)cnc21)NC(CC)CNC(c1cc2ccoc2cn1)=O c1(C(N2CCC(N(C(=O)CC3CC3C)C)C2)=O)ccc(F)c(F)c1 C1(CNC(C2N(CC)CC2)=O)CN(C(=O)C(O)C2CCC2)CCN1C c1(C(=O)NCC(C)CNC(c2ccc([N+](=O)[O-])[nH]2)=O)cccc2c1CCCCC2 N1(C(c2scc(C(=O)OCC)n2)=O)CCN(CC)C(C(=O)NC2CCCCO2)C1 Cc1cc(C(=O)NCc2nnn(C)c2C(N2CC(C)(CF)C2)=O)c[nH]c1=N C(=O)(C(CCC)CCC)N1CC(CC(C(N2CC(C)CC(CC)C2)=O)F)C1 N1(C(c2c(C)cnn2C(C)C)=O)CCN(C(c2cscc2C)=O)CCC1C C1(C(N2CCCC(C(=O)NC3CCN(C)CC3)C2)=O)CNC(C)(C)CO1 C(=O)(CC(C)CC(F)(F)F)NCC(=C)CCNC(c1ncn(CC)n1)=O C1(NC(C(CC)C)=O)CC2CCC1N2C(c1ccc(Oc2ccccn2)cc1)=O Cc1cnc2c(cnn2CC(N2CC3CCN(C(C4CCC4(C)C)=O)C3C2)=O)c1 C(=O)(CCCCC(N)=O)N1CCC(C)C(NC(c2csc(C3CCCO3)n2)=O)C1 C(C(C)(C)CC(=O)N1CCC(O)(CN(C)C(c2cc(C)cc(Br)c2)=O)C1)OC C1(CNC(c2cccc(Br)c2)=O)CCCC2(CN(C(C3CC=CCC3)=O)C2)O1 c1(C(N2C3CN(C(C(CCC)(C)C)=O)CC2CC3)=O)cc2c(cc1Br)OCO2 C12(CNC(c3cc(CNC(C4(OC)CCC4)=O)[nH]n3)=O)CCC(C1)C(=O)N2 C1(C(=O)NC2C(F)CCN(C3C(CC)C3)C2)CCc2cccc(OC)c2C1 N1(C(C(C(C)C)SCC)=O)CC2(CC(CNC(c3ccc(F)c(C)c3)=O)C2)C1 C1(NC(C(C2CC2)OC)=O)(CNC(=O)C=Cc2ccncc2)CCCCC1C C(=O)(C(C)(C)S(C)(=O)=O)NC1CC(C)(CNC(C(CC(C)C)O)=O)C1 Cc1c(C(=O)NC2CCCC(NC(C3CCC(=O)N3C)=O)C2)c(C(F)F)nn1C N1(C(CNC(C)=O)=O)CCC(CNC(=O)COc2ccc(Cl)c(Cl)c2)C(C)C1 C(=O)(C(F)(F)C(F)F)NC(CC(C)NC(=O)CN(C)Cc1ccc(F)cc1)C C(CC(C(=O)NC1CC(O)C1OC)NC(C1CCCSC1C)=O)=CC c1(C(=O)NC2CCC(CCNC(=O)CC3CCC3)C2)ncc(Cl)cc1O Cc1csc(C=CC(=O)NC(C)CCCCNC(=O)C(c2nc(C)cs2)C)n1 S(=O)(=O)(c1cccnc1NCc1ccc(=N)[nH]c1)NC(CC)CC(C)O C(=O)(C(C)(C)CC(F)(F)F)NCC(C)N(C)C(c1cccc2c1nnn2C)=O Cc1csc(=NCC(=O)N2CC(CNC(C3CCCSS3)=O)CC2C)[nH]1 N1(C(c2cnc(C)n2C(C)C)=O)CC2CC(NC(c3c(C(C)C)cnn3C)=O)C2C1 C=C=CCCC(=O)NCCN1CCN(C(C2(C)CCC(C)C2)=O)CC1 C(=O)(C(C)CC(F)F)N1CCCC(N2CCN(C(COCCC(C)C)=O)CC2)C1 C(=O)(C1CCc2nccn21)OCc1c(C(=O)OC)cccc1F N1(CCC(=O)NC(c2ccco2)COC)CCC2(CC1)CC(O)CO2 C(C)(C)(CC(=O)NCC1CC(F)CN1C(=O)CSc1nncn1C)SC CC1CCCC1C(=O)NCCCOCCNC(c1ccnn1C(F)F)=O C1(NC(C(C)(C)OC)=O)CN(C(=O)Cc2[nH]cnc2C)CC1c1ccccc1 C(=O)(C(F)C(C)CNC(c1cccc(OCC(F)F)n1)=O)N(CCO)CC n1(C(C)C)ncc(C(N2CC(O)(CC(C)(C)NC(=O)CCOC3COC3)C2)=O)n1 C1(NC(=O)NC(c2ccc(Br)cn2)CN(C)C)CCNC(C(F)(F)F)C1 C12(CNC(c3cnc[nH]3)=O)CN(C(c3ccc(Cl)cn3)=O)CC1CCO2 CCC(O)C(C)(C)C(=O)N(CC(O)CNC(c1c(C(C)C)n[nH]c1C)=O)C C(=O)(C1=Cc2ccccc2OC1)N1CC(C)C(NC(C2CC2(C)Br)=O)C1 C1(C(N(CCNC(C2CCC(C)S2)=O)CC)=O)CCCCCC1 N1(C(c2n(C(C)C)ccc2)=O)CC2C3CCC(C2C1)N(C(=O)CNS(C)(=O)=O)C3 C1(c2cc(OC(C)=O)ncc2)CCCN(C(=NCC2CC2)NCC=C(C)C)C1 C12(C(=O)NC3(C)CN(C(C4CCC(OC)C4)=O)C3)CC(CSC)(CO1)C2 N1(C(c2cc(C)cc(Br)c2)C(=O)NCC=C)CCCC(C)(C)C1C(=O)O N1(C(CCCC=C)=O)CCC12CCN(C(c1cncc3[nH]ccc13)=O)CC2 C1(C2CN(C(=O)Cc3cc(F)ccc3Cl)C2)(NC(C2CCC=CCC2)=O)CC1 c1(C=O)ccc(OC)nc1OC.c1(CN(CC(F)(F)F)CCC)ccc(C)nc1 C(=O)(C(C(=O)NC1CCC(NC(=O)C(N)=O)CC1)c1cccs1)OC(C)(C)C N1(C(c2nc(CC)oc2)=O)CC(N(C(=O)Cc2cncc(Br)c2)C)C(F)C1 C1(O)(C(=O)NCC2(F)CC(CNC(C3N(C)CCC3)=O)C2)CN2CCC1CC2 CCC(CC(=O)N1CC(O)(CN(C(=O)CC2(O)COC(C)(C)C2)C)C1)C(F)F c1(C(=O)NC(c2cc(C)ccc2Cl)CC)cc2c(nn1)CCCC2 n1(C(CC)CC)nc(C(=O)NC2CC(CCNC(c3ccoc3Cl)=O)C2)cc1C C1(CC)(CC)CC(NC(=O)C(C)(C)n2cc(Cl)cn2)CN1C(=O)C(C)SC C1(NC(N2CCCC2Cc2cnc(Cl)s2)=O)C2CCCCCC12 C(=O)(C1CCCn2cnnc21)N1CC2OCCN(C(c3cnn(CC)n3)=O)C2C1 C1(CNC(CC2C(C)CCC2)=O)CCCN(C(C23CC(C)(CO2)C3)=O)CC1 N12CC3CC(C(C3)C1)C2=O.c1(CCC(=O)OC)ccncn1.N12CCC1CC2=O c1(CC)cccc(CC(=O)NCCN2CCN(C(=O)C(C)N(C)C(C)=O)CC2)c1 c1(C(=O)NC23CC(NC(c4cn(C5CC5)nn4)=O)(C2)C3)ncccc1CO c1(C(N(C)CC2CCN(C(=O)C(C)(F)F)C2)=O)cc2cnc(Cl)cc2s1 C1(NC(C2(C)C(C)CN(C(c3cnn[nH]3)=O)C2)=O)CC2CC1OC(=O)N2 C1(NC(=O)CCN2CCC(O)CC2)CC(O)CN(C(=O)CSC2CC(F)(F)C2)C1 C1(CNC(c2c(CC)occ2)=O)COCCN(C(c2ccc(F)nc2F)=O)C1 CC1CC(NC(C2CC(F)C2)=O)CN1C(c1ocnc1-c1nn[nH]n1)=O c1(C(=O)NC)ccc(Cl)c(C(=O)NCCCN(C(C2CC3CCC23)=O)C2CC2)c1 CC1CC(=O)NCCN1C(=O)CC1CC(C)(C)CN1C(=O)CNc1ccccn1 n1(CC)cc(C(N2CCC(CN(C)C(C3(C)CC(C)=NO3)=O)CC2)=O)c(C)n1 Cc1sccc1C(=O)NCCCC(=O)NCc1noc(C(N)=O)n1 N1(C(CNC=O)=O)CCc2cc(-c3cc(F)ncc3F)ccc2C1 CP(C)(=O)C1CCCCC(Nc2ccc(Br)c(C(F)(F)F)c2F)C1 C1(CC)CN(C(CC)C(=O)N(C(C)CCNC(c2ccnnc2C)=O)C)CCO1 c1(C(=O)NCC2C(NC(CN(CCC)C)=O)C2)cc2c(nc1O)C(C)(C)CCC2 c1(C(=O)NC2(C)CCN(C(C3C(CCC)C3)=O)C2)ccc(C2=CCOCC2)cc1 c1(CC)nc(C(=O)N(C2CCC(NC(C3(CCOC)CCCC3)=O)C2)C)co1 Cc1ccc(CN=C(NCc2c(C)noc2C)NCC2CCCCO2)c(C)c1 c1(C(=O)NC2CN(C(CC)CO)C2)ccn2ncc(-c3ccccc3)c2n1 c1(C(=O)NC2C(CNC(CSCCC(C)C)=O)CCC2)cnc(OC(C)C)cn1 S(=O)(=O)(c1ccc(Br)c(Cl)c1)N1CC(NC(=O)NCc2ccccc2F)C(O)C1 C(=O)(C1CCCc2scnc21)NCC1=CCN(C(CNC(C)=O)=O)CC1 c1(C(N2CC(N(C(CCC=C=C)=O)C)C3(C2)CC3)=O)cnn2c1CC(C)CC2 c1(CC)cc(NC(C23CCN(C(c4cccc(C)c4O)=O)CC2C3)=O)cnc1C c1(C(=O)NC2C3CN(Cc4c(C)cccc4)CC32)cccc(S(F)(F)(F)(F)F)c1 c1(C(N2CC(COC)N(C(c3ccc(Cl)[nH]3)=O)CC2)=O)cccc2c1ncn2C C1(NC(CCOC)=O)CCN(C(c2sc(C3CCCC3)nc2C)=O)CC1F c1(C(N(C2CN(C(c3c(C)nn(CC)c3Cl)=O)C2)C)=O)ccc2n[nH]cc2c1Cl c1(CC(=O)NCc2ccc(C(=O)NC(C(COC)C)C)o2)ccc(F)nc1 c1(C(=O)NCCCN(C(c2ccc(Cl)[nH]2)=O)CC)ccc(NC(C)=O)cc1F Cc1cc(C(=O)NC2CCN(C(c3cnc4n3CCC4)=O)CC2C)c(O)nn1 N1(C(CCc2c(C)noc2)=O)CC(NC(=O)C(n2cc(Cl)cn2)C)C(C)C1 C1(N(C)C)CC12CN(C(=O)Nc1nc(-c3ccn(C)n3)cs1)C2 c1(CCC(=O)O)ccnc(NCC(C2CCCCC2)=O)n1 C(=O)(C1CNC(=O)c2ccccc21)NC1CCN(C(C2(CC#C)CC2)=O)C1C1CC1 C(CCC(=O)N1CCOCC1C1CC1)(C(C)C)NC(C(C1CC1)SC)=O C1(NC(C2ON=C(C(C)C)C2)=O)CN(C(=O)C(C)(C)O)CC2(CC2)C1 CCCCC(CC(=O)N(C)CCOCCO)NC(=O)C(C)(C)N=[N+]=[N-].C(C)=O C1(O)(C(C)NC(=O)C=Cc2cscn2)CCN(C(C2(c3ncco3)CC2)=O)CC1 Cc1nc(=N)[nH]cc1C(N1C2CCC1(CNC(c1cnns1)=O)CC2)=O C1(Nc2nccc(C(C)C)n2)CN(C(=O)CCOCC2CCCO2)CCC1F c1(C(N(C2CCCN(C(c3cnccn3)=O)C2)CC)=O)cc(CCC#N)oc1C C1(C(=O)NC(C)C(C)(C)C)CCN(C(=O)C=Cc2ccccc2)CCO1 C(=O)(C1=CCCCO1)NC(CNC(CCc1onc(C(C)(C)C)n1)=O)CO N1(C(C2(CC)CCCC2)=O)CCCOC(CNC(=O)COC2COC2)C1 N1(C(C2(C)CCC(=O)CC2)=O)CC2CCN(C(C3CC3C(N)=O)=O)CC(C2)C1 N1(C(CC2(OC)CCC2)=O)CCn2cccc2C1.c12nnc(s1)NC(=O)N2 C(=O)(C1CCc2ccccc21)NCC(CC)NC(=O)C=Cc1ccc(F)c(F)c1 N1(C(CCC)=O)CCCC1C(=O)NCC(CCOC)NC1COCCO1 CCC(O)(CNC(=NCCCF)NC1CCC1(C)C)C(F)(F)F CCCCCC(C(=O)N(C)CCN(C(c1cnnc(C)c1)=O)C(C)C)C(C)C Cc1ccc(CNC(C2C=CC(NC(=O)COC3CC=CC3)C2)=O)nn1 C1(NC(c2c(CC)cco2)=O)CCC(CCC(=O)NCC(CSC)OC)CC1 c1(C(N(CCCC(=O)NCC(C)(C)N(C)C)C)=O)cnc[nH]c1=N C(=O)(C(C(C)(F)F)c1ccccc1)N(CCCCNC(=O)CS(N)(=O)=O)C c1(CC(C)C)c(C(N2CC(CN(C)C(C3CC3(F)F)=O)C2)=O)cnn1C CC1(C)CCOC1C(N1CCSCC1CCNC(c1coc(Br)n1)=O)=O N1(C(c2scc(CC)c2)C(=O)NCc2nnn(C)n2)CCOCC1C#N CCC(O)C(F)(F)C(=O)NCC1(F)CCN(C(C2CCCNS2(=O)=O)=O)CC1 CC(C)CC(C(=O)NCC1(O)CCN(C)C1)N(C)C(C1CCC(=O)CC1)=O C(=O)(C(F)(F)C(O)C1CC1)N1CCC(CNC(C(C)(C)NC(C=COC)=O)=O)C1 C=CCC(CC)C(=O)N1CC2C(N(C(=O)Cn3ncccc3=O)C)C2C1 c1(C(=O)NCC2(O)CN(C(CC3C(C)(C)C3)=O)C2)sccc1C#N CCCCCS(=O)(=O)CC(=O)N(CC)CC1CCCN(C(C2SCCCS2)=O)C1 N1(C(CCNC(=O)C2CC2)=O)CCC(CC(=O)N(C(C)CN(CCC)C)C)C1 N1(C(CCOCCOCC)=O)CCC(C)CC1C.C(c1ncc[nH]1)=CC(=O)N c1(CC(C)(C2CC2)NC(=O)NC2CC(CC(=O)OC)C2)ccc(F)cc1 C1(NC(C(CC2CC2)OC)=O)C2CC1N(C(c1ccc(Cl)cn1)=O)C2C C1(NC(=O)Cn2ccc(Br)n2)COCC1NC(C12CCC1C2)=O N1(C(C2CC(C)C2(C)C)=O)CCN(C(=O)CSCc2ccncc2)C2(CCC2)C1 C1(CC(C)C)(C(=O)NC(C)C(C)NC(=O)C(F)n2cccn2)CCC1 CCCCC(O)CC(=O)N1CC(=C(F)CNC(=O)CNS(=O)(=O)N(C)C)C1 N1(C(c2c[nH]c(=N)s2)=O)CCC(O)C(NC(=O)CC2CC=CCC2)C1 CC(C)CC(C)(C)C(=O)NCCN(C1CCCCCC1)C(C1(CF)CCC1)=O c1(C(N2CCC(NC(=O)CC3CCCCC3(F)F)C2)=O)cc(F)ccc1[N+](=O)[O-] c1(C(=O)NC23CC(C(=O)Nc4ccn(C(=O)OC)n4)(C2)C3)c(Br)cnn1C C1(F)(C(=O)NCCOCCCNC(=O)C=CBr)CC12CCCCC2 c1(C(=O)NC(c2occ(N(C(COC)C)C)n2)C)c(CO)cnc(C)c1O C1(NC(C=Cc2ncc(C)[nH]2)=O)CC2CC1CN(C(C1(F)C(C)(C)C1(C)C)=O)C2 c1(C(=O)NC2CC(C)(NC(C3ON=C(CC)C3)=O)C2)cc(F)cc(S(N)(=O)=O)c1 c1(CNC(C2CC(O)(CC#C)C2)=O)cccc(NC(C2CCN(C)C2)=O)c1 N1C(=NCC2CC2)NCc2noc(n2)C2CC(C2)C1.c1(C(C)(C)C)cccs1 Cc1cc(C(=O)NC(C2(O)CN(C(C3CN4CCN3CC4)=O)C2)C)c(C)cn1 c1(C(=O)NC(CC(C)NC(C2(C)CC(=C)C2)=O)C)ccccc1C(=O)NC c1(NCc2c(C)scc2)ccc(Cl)c(P(C)(C)=O)c1 CN1CCCC(N(C(=O)C(c2ccco2)NC(C2CNC(=O)N2)=O)C)C1 C1(NC(CCCOCCC)=O)CCN(C(c2ncccc2C(F)(F)F)=O)C(C)C1 c1(-c2cnc(OC)nc2OC(=O)C=Cc2cccnc2)ccc2c(c1)oc(=O)n2C Cc1c(C(N2CCC(CN(C(=O)C(C(C)(C)C)N(C)C)C)C2)=O)cncc1F c1(OC)cc(C)cnc1C(=O)NC1(CCCNC(C2CCOC(=O)CC2)=O)CC1 C(=O)(C1=NNC(=O)C1)N(CCCCN(C1CCCC1)C(c1c(C#C)c[nH]n1)=O)C C1(CCNC(c2n(CC=C)ccc2)=O)CCN(C(=O)CCCOC(C)=O)CC1 N1(C(C2N(C(C)(C)C)CC2)=O)CCN(C(C2CC3(C2)CC3F)=O)CC(O)C1 c1(C(=O)NC2CCC(CNC(C3(C)CC(F)(F)C3)=O)C2)ccc2ccncc2c1 S(=O)(=O)(c1c(OC(F)(F)F)cccc1OC(F)F)N1C(C)CCC1C CC1(C)CCCN(C(=O)C(N2CCC(OCCF)C2)=O)C1CO c1(CC(N2CC(CC(C(=O)Nc3cccc(SC)c3)F)C2)=O)ccc(C)c(O)c1 C1(CNC(=O)CCC2CCCC2)CCC(CNC(C23CC(CO2)C3)=O)CC1 N1(C(CC(CC)NC(C(C(=O)OCC)OC)=O)=O)CCCCC2(CCC2)C1 Cc1ccc(C(N2C(c3ccco3)CCC2c2cnn(C)c2)=O)cc1Cl c1(C(N2CC(C)(NC(C(C(C)C)OC)=O)C2)=O)cc2ccccc2o1 C12(NC(=O)C3=CCCOC3)CCN(C(=O)COc3cncc(Cl)n3)CCC1C2 C=CC1CN(C(c2csc(C3CCCCC3)c2)=O)CC1NC(=O)C#CC1CC1 C1(C(N2CC(OC)C(NC(C3(c4ncco4)CCC3)=O)C2)=O)CC2(CCCCC2)C1 N1(C(c2cn(CC)nn2)=O)CCC2(CC1)COC(CNC(c1cnc(C)nc1)=O)C2 N1(C(c2cc(C)sc2Br)=O)CCN(C(=O)CCCN(C)C)CC1CF C12(C(=O)NC(CCC)CC)CCC(CC1)N(C(C1CC3(CCC3O)C1)=O)C2 c1(OC)cc(N)c(C(=O)NC(C)C(C)NC(c2cc(Cl)sc2Cl)=O)cc1F c1(CNC(c2csc(C3CCCN3C(=O)C(F)F)n2)=O)ncc(Br)nn1 c1(CC(=O)OC)ccc(NC(C2(C(F)F)CN(C(=O)C(CSC)OC)C2)=O)s1 c1(C(c2nnnn2C)(C)NC2CCCCC2)ccccc1OCC(F)F C1(C)(C(=O)OCC)CC2=C(C(=O)N1)C(c1[nH]ccc1C)NC(=O)N2C N1(C(C2CC(CC)N(C(c3cc(C)ns3)=O)CC2)=O)CCN2CCCC2C1 C(=O)(C(C(C)(C)C)SC)NC(CNC(=O)CC1(OCC)CCC1)(CC)CC C1(C(=O)NC(c2ccc(Br)cc2)CC)COCCN1C(c1cc(C)c[nH]1)=O c1(C(=O)NCCCCCCNC(c2c(C)nc(O)[nH]2)=O)cnn2c1N(C)CC2 CC(C)CC(C)(CNC(=O)CCc1ccsc1Cl)NC(=O)CC1OCCO1 N1(C(c2n(CCC)ncc2)=O)CCOC(CNC(=O)C(O)C2CCC2)C1 C(=O)(C(C(C)(C)C)N(C)C)NCC(CC(=O)NC(Cn1ncc(C)c1)C)O c1(CCSCC(=O)OCCC(=C)C)c(Cl)cccc1Cl C12(CNC(C3CCN(C(C)=O)C3(C)C)=O)CCCC1CN(C(C1CCCO1)=O)C2 C1(C(F)(F)F)(C(=O)NCCC2(O)CN(C(c3csc(F)c3)=O)C2)CC2(CC2)C1 C12(CNC(c3cc(C(C)=O)sc3)=O)CC(C1)C(NC(=O)CCC(C)(C)C)CO2 C(=O)(CS(=O)C(F)(F)F)NCC1CC(NC(c2cn(C)nc2O)=O)C1 N12CC3CCC(C1)C3NC(=O)c1c(c[nH]n1)C2=O.C12(C)CC(F)(C1)C2.CO c1(OC)cc(N)c(C(N2CCN(C(=O)CC(C)OC)CC2CCO)=O)cc1OC CCC(C)(O)C(=O)NCC(C)(O)CNC(=O)CC(=O)OC(C)(C)C CCCCC(C(=O)NCC1CCCC1NC(c1cc(Cl)no1)=O)NC(N)=O Cc1ccc(Cl)c(OCC(=O)NC(C)(CNC(C23CC(CO2)C3)=O)CC(C)C)c1 C1(N(CCCOCc2nn(C)c(=O)n2C)C)CN(C(=O)OC(C)(C)C)CC12CCC2 c1(N2C(C)CN(C(c3ccnc4cc[nH]c34)=O)CC2)ncc(Br)cc1[N+](=O)[O-] c1(COC)ccc(NC(C2CCCCN2C(C2CC(C)(C(=O)OC)C2)=O)=O)cc1 N1(C(C2C(C(C)C3CC3)C2)=O)CC2(CO)CC1(C(=O)NCC1(C)CCC(C)CC1)C2 N=c1[nH]c(C(N2CCC(OCCNC(c3nccn3C3CCCC3)=O)C2)=O)cs1 C1(F)(CC)CCN(Cc2cccnc2O)CC1 C1(C(=O)NCCCN2CCCC2C)(COC)CN(C(=O)Cc2c[nH]nc2C)C1 C(=O)(C1=C(Cl)CC1)NC(CNC(=O)CCc1ccc(Cl)s1)CO c1(C(N2CC(NC(C(C)NC(N)=O)=O)C(O)C2)=O)ccc2scnc2c1 C1(OC)CCCCC1C(=O)N(C)CC1COCCN1C(=O)CC1CCC1 CC1(O)COCCN(Cc2cn(-c3cc(F)cc(F)c3)nn2)C1.C12CCCCN1C2=O c1(CC(=O)N(CC(C)(C)CSC)C(C(=O)OC)CC2CC2)ccc(Cl)cc1Br c1(CNC2C(C(=O)Nc3onc(C)c3Br)C2)ccc(Cl)c(F)c1 N1(C(C(c2cn(C)nc2)(C)C)=O)CC2(C1)CN(C(c1ccc(Cl)c(Cl)c1)=O)C2 S(=O)(=O)(c1ccccc1)N(C)CC1(OC)CCSC1.C(=O)(NC)NCCN C(C(O)CN=c1ncnc2[nH][nH]c(C)c1-2)NC(C(CCC)OCC)=O c1(C(N2CCC(C(CNC(CCCC=C)=O)(C)O)CC2)=O)ncc(Cl)c(N)c1Cl N1(C(c2cc(F)c(=N)[nH]c2)=O)C2CCC1CN(C(=O)CSCC#N)CC2 N1(C(C=C(CCC)C)=O)CC2CC1CCN2C(C1CCCOC1)=O c1(C(N2CCCC(C)(C(N3CCOC(C#N)C3)=O)C2)=O)cnn2cccnc12 N12CC(C)N(CC1C)C(=O)Cn1cnc(c1)C2=O.N1(CC)CCC(C(=O)OC)CC1 CCCCCC(O)CC(=O)NCC1CC(OC)CN1C(=O)CC1(CSC)CC1 C1(C(=O)NC(C#C)C)CCN(C(=O)CCC=CC)C1C(C)C CCCC(C(=O)N1CCN(C(=O)Cc2cncnc2)C(CC2CC2)C1)C(C)C c1(C(=O)NC2(C)CN(C(C3COC(=O)N3)=O)C2)cccc(C(N)=O)c1N c1(OC)ccccc1C(N1CCC(C(N2CCN(CC(=O)O)CC2)=O)CC1)=O Cc1cc(Cl)cc(C)c1C(=O)NC1CCCN(C(C2CCNC2=O)=O)C1 CC(C)C(C(=O)Nc1ccccc1F)OC(=O)CCc1cnn[nH]1 C=CC(C)(CC)C(=O)NC1CCC(NC(=O)C(C)C(F)F)CC1 c1(C(N2C(C(N3CCC3c3ccc(I)cc3)=O)C=CC2)=O)ccc([N+](=O)[O-])o1 C(=O)(C1=NOC2(CCOC2)C1)N1CCCC2(NC(C3CC34CCC4)=O)C(C1)C2 c1(C(N2C(C)CC(NC(C3CC(C)(O)C3)=O)CC2)=O)ccc2c(c1)OCCO2 N1(C(C(CC2CN(C(C(N3CCOC3=O)C)=O)C2)F)=O)CC(C2CCCCC2)C1 C1(C(C)C)(C(=O)NC2COCCC2O)CCCN1C(C12CC(F)(C1)C2)=O c1(C(N(C)CC2CCN(C(C3(C#N)CCCC3)=O)CC2)=O)ccc2nsnc2c1 N1(Cc2cncc(CCNC(=O)OC(C)(C)C)c2)CCC2(C1)CCO2 O=S1(=O)CCC(c2nc(Cc3cnc(C(F)(F)F)cn3)no2)CC1 Cc1ccccc1CS(=O)(=O)NC(c1c[nH]nc1C(F)(F)F)=O Cn1cccc(C(N2CCC(O)(CNC(=O)Cc3ccc(Cl)cc3)C2)=O)c1=O C12CCC(CC1)CCN(C)C2=O.n1(C2(NC(CN(C)CCO)=O)CC2)ccnn1 c1(C(=O)NC2(C)CCN(C(c3ncc(CC)nc3)=O)C2)ccc2scc(C)c2c1 CN1CCN(C)CC(C(N2CCC(CCNC(c3cn(C)ccc3=O)=O)C2)=O)C1 N1(C(CC(=C)Br)=O)CC2(CCCC2NC(=O)CCOC2CC2)C1 C(=O)(C(C)(C)C(=O)NC(CNC(C1(C)CNC(=O)C1)=O)C1CCC1)OCC N1(C(C(C)SC)=O)Cc2ccnn2CC(NC(c2cc(C3(C)CC3)n[nH]2)=O)C1 c1(C(=O)NCC2(CNC(C(CC)N3CCCC3=O)=O)CC2)cc(C#N)oc1C CC(C)C(C)(CNC(c1cc[nH]c1)=O)NC(=O)C(C)n1ccnc1 CCCC(C(O)C(=O)N1CC(SCC)C1)NC(c1snnc1C)=O Cc1ccnnc1C(=O)NCC1(C)CCN(C(c2ccc(F)s2)=O)C1 CCCCC(CCCC)NC(C1(C)C=CCN1C(C1OCCC1C)=O)=O CCCC(CC)CC(=O)N1CCCC1CNC(C1CCC1(C)C)=O c1(C(=O)NCC(CC=C)NC(C2CSCC(=O)N2)=O)cnc(C)cc1C C1(N(C(CC(=C)Br)=O)C)CCN(C(=O)Cc2ccc(O)cc2Cl)CC12CC2 O=C1CCC(CNC(=O)N(C2CCCC2)Cc2ccccc2Br)CN1 N1(C(C2CCC2)=O)CCC(CC2CC(OCC)(OC3(C(=O)N)CC3)C2)CC1.C(C)(C)O Cc1oc(C(C)C)cc1C(=O)NCC(C(C)(C)C)NC(c1ccccc1CO)=O N12CC(CCC1C(F)(F)F)C2.C(C(C)(C)NC(=O)C(=O)N(C)C)N(C)C C#Cc1cc(F)c(C(=O)NC2(CNC(c3cnnn3C)=O)CCCC2)cc1F Cc1cc(N2CCC3NCCC3C2)nc(=NCc2nc(C(F)(F)F)cs2)[nH]1 C1(F)(CNC(C(C)NS(CC)(=O)=O)=O)CCCN(C(c2cc(Cl)c(C)cn2)=O)C1 c1(C(=O)NC(C(CO)NC(C(CC)n2ccnc2)=O)C)ccnc2c1ncn2C N1(C(c2cc(C)sc2)=O)CCC2(CC1)CC(CNC(C1(CO)CCOC1)=O)C2 c1(CN2CC(F)CC(C(=O)Nc3c(Br)ccc(C)n3)C2)c(C)cc(Br)cc1F C#Cc1cnn(C)c1C(=O)NCC1CC(NC(=O)CNC(c2ncccc2O)=O)C1 Cc1ccc2ncccc2c1C(=O)NCCN(C)C(C1CC1(F)F)=O CCCCCC(O)C(=O)NC1C=CCN(C(c2cc(Br)cc(F)c2O)=O)C1 C(=O)(C(C)(F)C(F)(F)F)NCC(C)N(C(c1c(C)[nH]c(C)c1C)=O)C C1(NC(c2c(C)nc(C)[nH]2)=O)CN(C(=O)Cc2ccnn2C2CCC2)CCC1F C#Cc1ccc(C(=O)NCCC2CC(F)(F)CN2C(c2occc2CC)=O)cc1 C(C(F)(C(=O)NCc1c[nH]c2cnccc12)C(C)C)NC(CCSC)=O C(CC(C(N)=O)NC(C1(C)CCCN1C(=O)COCCN(C)C)=O)OC CC(C)CCC(C(=O)NC1CC(=O)NC1=O)NC(c1cnsn1)=O C12(C(=O)NCC3C4CN(CC(=O)NC5CCOC5)CC34)CCCC1C2(F)F CN1CCN(C(=O)C=Cc2cc[nH]n2)C(C(=O)NC(c2cn(C)cn2)CO)C1 C12(C(=O)NCCCC3CC(C)C3)CCC(NC(=O)CCS(C)=O)(CC1)C2 Cc1c(N(C(=O)COCCF)Cc2cccc(Br)c2)cccc1F C1(CC(=O)NCC(C)N(C)C(c2cccn2C)=O)CC(O)C12CCC2 Cn1nnc(CNC(c2ccnnc2)=O)c1C(N1CCCC(CF)C1)=O c1(CC(=O)NCC(C)N(C)C(c2cn(C)nc2O)=O)ccc2c(c1)CCOC2 n1(CCNC(=O)NC(C2(N3CCSCC3)CCCC2)C)cccc(N)c1=O c1(C(NOC(C(=O)N2C(C(C)(C)OC)CCC2)CC)=O)cc(C#N)c[nH]1 N1(C(CN2CC(C)C2)=O)CC(CN(C(=O)CCOCC(F)(F)F)C)C2(CC2)C1 c1(C(=O)NC2(C)CN(C(=O)CC3CCOC(C)(C)C3)C2)nn2c(c1Br)CCC2 c1(Cc2ccc(C(C(=O)NC3CCC3)N(C(C)=O)C)o2)c(C)cc(Cl)cc1C N1(CC)CC2CN(C(=O)CC(O)CNC(C3(CC)CC3)=O)CC2C1 CCC(C(=O)N(CC(=O)NC(CC1CC1)C(=O)OC)CC)OC c1(C(=O)NC(COC)C2CC2)cnn(CCNC(c2cnc(C(C)(C)CF)o2)=O)c1 N1(c2cc(N(CCCOCCOC)C)nc(C)n2)CCCC(C2CCC2)C1 C1(NC(c2c(OC)cccn2)=O)CN(C(C23C(=O)C4CCC2C3C4)=O)C2(CCC2)C1 N#Cc1c[nH]c(C(=O)N(C2CC2)CC2CCCN2C(c2ccc(C(N)=O)[nH]2)=O)c1 C(=O)(CCCC(C)NC(c1cc(C)cc(F)c1)=O)NC(CC)C(C)(C)O N1(C(C(C)=CC)=O)CC(CNC(C2CCC(=O)N2CCC)=O)C(CN(C)C)C1 CC1=NC(C)(CNC(=O)CC2C=CC(NC(=O)Cc3cccc(O)c3)C2)CS1 C12(CNC(C(COC)(F)F)=O)CCC1CCN2C(=O)CCCc1nc(C)no1 C(=O)(CCC(C)CCCC)N(C)Cc1ccc(CNC(CC(C=C)CC)=O)cc1 C(c1ccc(O)c(O)c1)=CC(N1CCN(C(=O)C(O)CF)C(CO)C1)=O c1(CCC(C)=O)ccc(C(N2CCSC(C(=O)OC(C)(C)C)C2)=O)cc1 c1(C(N(CCCCCCNC(c2cc(C)sn2)=O)C)=O)cccc2c1CCCN2 N1(C(C2CN(C)CC2C(F)(F)F)=O)CCCC2CN(C(=O)C(F)(F)C3CC3)CC12 c1(C(=O)NC2C(NC(CCCN(C(=O)OCC)C)=O)C2)cc2ccccc2cn1 C12(CNC(C#CC(C)C)=O)CCCC1N(C(=O)Cc1nc[nH]n1)CCC2 C1(C(C)C)CCCC1C(=O)NC(C)CC1CN(C(c2cn(CCS)nn2)=O)C1 CC1=NOC(C(=O)NOCC(=O)NCC(C)(O)C2CCCC2)C1 N1(C(c2n(CC)ccn2)=O)CC(NC(C2(n3cc(Cl)cn3)CC2)=O)C(C)C1 CS(=O)(=O)c1ccc(C(=O)NCC2CCN2C(=O)CSc2ccccn2)[nH]1 C1(OC)CN(C(c2cn(C3CC3)nn2)=O)CC1NC1(C(=O)NC(C)C)CC1 c1(C(=O)NC(C2CCN2C(=O)CN(S(C)(=O)=O)C)C)cnc2nccn2c1 n1(CC)cc(C(N2CCCC(CN(C)C(C3CC3(F)F)=O)C2)=O)c(C(C)C)n1 CC1CC(NC(c2coc(C3CC3)n2)=O)CCN1C(C12CCC(C1)OC2)=O C(=O)(C#CC(C)(C)CNC(c1occc1C1CC1)=O)N(CCCCO)CC N1(C(C(C(C)C)OCC)=O)CCC(NC(c2cn(CC(=O)NC)nn2)=O)C(O)C1 C(=O)(C1=CC2C=CC1C2)N1CCCC(CC)C1C(=O)NOCC(N)=O C(c1cnc[nH]1)=C(C)C(=O)N(C(CNC(=O)Cc1csc(C(C)C)n1)C1CC1)C C1(NC2CC(C(=O)OCC)(C(=O)OC)C2)CCN(C2CCOCC2)C1=O Cc1cccnc1C(N1CCC(CN(C(=O)CN2CCCC2CO)C)C1)=O CC1(C)CC(C(=O)NC23CC(CNC(=O)Cc4n[nH]cc4Br)(C2)C3)CO1 c1(C(=O)NCC2CN(C(COC(CC)C)=O)C(C)C2)cccc(N=[N+]=[N-])c1 Cc1ccc([N+](=O)[O-])c(N2C3CN(C(=O)N)CC23)c1.c1(C)cc(Cl)c(Cl)cc1O C1(CC)CCN(C(=O)CNc2cccnc2)C1CNC(C1CCCCC1O)=O c1(C(C(=O)NCc2cccs2)N(C(CSC)C)C)ccc(Cl)o1 C(C1=CCCN(C(c2c(C)cncc2C)=O)C1)NC(C(CC)NC(N)=O)=O Cc1cnc(C(=O)OC2CCN(C(=O)OC(C)(C)C)CC2F)cc1C CN=c1[nH]c(C(N2CCCC2(C)CNC(=O)CCC(F)F)=O)cs1 C(=O)(CC(C(F)(F)F)NC(=O)CC1CCCC(=O)N1)N1CC(C)(C)C1 c1(C(=O)OC)ccc(F)c2c1CN(C(=O)Cn1cc(-c3cnc4n3CCC4)nn1)C2 c1(C(N(CC(CC)NC(=O)CCC23CCC(CC2)C3)C)=O)ccc(Cl)cn1 CN(S(N)(=O)=O)CC(=O)NCCN(C(=O)CC1(C)OCCO1)C1CC1 c1(-c2cn(CC(=O)OC)nn2)cccc(NC(C2CCNCC2)=O)c1 C1(CC)C(NC(C23CCCCC2C3)=O)CCCN1C(c1snc(Cl)c1C#N)=O N1(c2n(CCOCCOC)c(C3(C)CCCCO3)nn2)CC2OC(C)(C)OC2C1 C1(NC(C(c2ccccc2Cl)(C)C)=O)CN(C(C2CC=CCC2)=O)CC1O C1(c2c(C)ncs2)CCN(C(c2cccc(Br)n2)C(=O)NC2CCCC2)CC1 N1(C(CSCCOC)=O)C(C(=O)NC(C)(C)CCF)CCC1C C1(NC(C2C(CNC(C(COC)(F)F)=O)CCCC2)=O)CCC2(CC1)N=N2 CCC(CC)C(C)C(=O)NC1CN(C(=O)CN(C)C(C)=O)CC1c1ccccc1 CC1CC(NC(=O)C2CC2)CN1C(=O)CCc1ccc(F)cc1 C(CN=c1[nH]nc(C)o1)N(C(COCCOCC)=O)CCOC C(=O)(C(C(CC)CC)OC)NCC1CC(F)(CNC(c2ccc(C#C)cn2)=O)C1 c1(OC)c(CN2CC(C(=O)NCC(O)CCCO)C2)cccc1F N1(CCC#C)CCN(CCCNC(=O)C(C)OC2CC2)CC1 N1(C(C(CNC(=O)C(=O)C2CCCC2)OC)=O)CCC2(C=CCO2)CC1 c1(C(=O)NC(C)CCNC(C23CCCC2C3)=O)ccc(OC(F)F)nc1 C1(C(=O)NCc2n(CC)ccn2)CC(NC(=O)C=CC2CCCC2)C12CCC2 c1(C(=O)NCC(CC=C)NC(=O)CNc2ccccn2)cccc2[nH]nc(O)c12 c1(C(=O)NCc2cc(C(N3CCCC(OC)CC3)=O)sc2)c(F)cc(N)cc1F N1(Cc2cncc(C)c2)CCC2(CC1)CC2(C)C(N1CCN(CCO)CC1)=O C(=O)(C1=C(Cl)CCCC1)NC(CCNC(C1CC(C(C)=O)C1(C)C)=O)(C)C c1(NC(CC(C=C)c2ccccc2)=O)ncnc(Cl)c1Br.C1(=O)NCCO1 C1(OC)CC(C(=O)NC(C)(CNC(=O)CCn2ccccc2=O)CO)CC1OC C1(NC(c2c(C)cco2)=O)CCC(C)N(C(c2cc(F)ccc2F)=O)C1 Cc1[nH]c2cccnc2c1CNCCC1(O)CCCCC1 Cn1nc(CNC(=O)C(=O)NC2CC2)cc1C(=O)NCC(O)C(N)=O Cc1cc(C(=O)NCC2CCC(NC(=O)C(C(C)C)C(C)C)C2)c(N)cc1F c1(CC(=O)NC2CC(CNC(=O)CCC3CCCCC3)C2)cccc(O)n1 C1(C(=O)NC(C)CC2CN(C(=O)C=C(C)C)C2)CCn2nccc2C1 C(=O)(C(CCF)NC(=O)C(c1cccs1)NC(C1CCC(=O)C1)=O)OC c1(C(=O)NC2(CO)CN(C(C(CC)(C)OC)=O)C2)ccc2sccc2c1 Cc1cc(C(=O)N(C2CC(NC(=O)CCc3ccc(F)cc3Cl)C2)C)cc(C)n1 C(C1Cc2ccccc21)NC(C1C(C)(C)CN(C(C2CC2C#N)=O)C1)=O CCCCCCCC(C)OCC(=O)NCc1c(C)cc(C(=O)O)c(C)c1C Cc1ccc(C(N2CC3CC3(CNC(=O)CN3CCOCC3=O)C2)=O)c(N)c1C C(C(=O)C1CCCc2ccccc21)OC(C1Cc2c(ccc(C#N)c2)C1)=O c1(C(N2CCN(C(C3C(=C)CC3)=O)C(C3CC3)C2)=O)cc(C)c(F)cc1Cl C1(CCC)C(O)CCCN1C(c1ccc(CC)cc1F)C(=O)NC(C)(C)CC C1(NC(C2(C(=O)NC)CCC2)=O)CCC(CN(C)C(c2c(C)nsc2C)=O)CC1 C1(NC(Cn2c(C)cnc2)=O)CCCN(C(=O)CCc2ccc(Cl)nc2)C1C Cc1ccc(OCc2cn(CC3CCCN3C(=O)C(F)F)nn2)c(Br)c1 N1(C(C2(C)CCC(=O)NC2)=O)CC2CN(C(C3CC(=O)C3C(C)(C)C)=O)CC2C1 C(C(C(=O)N1CCC(NC(c2ccoc2)=O)C(F)C1)C(C)(C)C)OCC=C CCCCC(O)CC(=O)N(CC(C)NC(c1cnc(OCCOC)c(Cl)c1)=O)C C1(C(=O)NCC(C)CNC(=O)CC2OCCO2)CCC(F)(F)CO1 C#Cc1cncc(C(=O)NC(CC(=C)Cl)C(=O)N2CC(c3ncccn3)C2)c1 c1(OCC)cccnc1C(N1CCC(C(C)NC(=O)CC2CC(=O)C2)C1)=O N1(C(C=CC(C)NC(C2CCC(N=[N+]=[N-])C2)=O)=O)CC2(CNC(=O)N2)C1 CCCCCCCCOCC(=O)N(C1CN(C(c2ncn(CC)n2)=O)CC1F)C CC1CC(NC(c2nc(Cl)nc3cnn(C)c23)=O)CC(C)S1(=O)=O c1(C(=O)NCCCN(C(C(C)OCC)=O)CC)cncc(N(C)C)c1 c1(NC(C(CCC)C)=O)ncnc(NCc2ncc(F)cc2N)c1C N1(C(CCCC)(C)c2nnnn2CCOCC)CCC(O)C(F)(F)CC1 N1(C(C(C)C)=O)CCSCC1C(=O)NC1CC1C(C)C N1(C(CCSCC(C)C)=O)CCC2CCN(C(=O)C=C(Cl)Cl)CC2C1 c1(CN2CC(C(=O)Nc3ccc(C(C)=O)nc3)SCC2)cccc(C)c1O C1(CNC(c2onc(CC)c2C)=O)CC(C)CCN1C(c1cn(CCO)nn1)=O c1(C(=O)NCCN(C)C(C2CCC2F)=O)ccc2c(c1)CCNC2=O N1(C(COCCC=C)=O)CC(n2cc(-c3ccncc3Cl)nn2)C(C)C1 C1(C(CNC(CCSC)=O)C)CCN(C(C2CCCN2N=O)=O)CC1 CCCCCC(O)C(=O)NC1CN(C(C2CC3CC3C2)=O)CC1(C)C Cn1[nH]c(=NC(=O)CN2CCCC(C(C)(O)C(F)(F)F)C2)cc1C(F)F CC(F)(F)CCC(=O)NCc1cc(C(=O)NCCCC(O)CO)n[nH]1 C1(NC(N2CCCC(CN3C(=O)CCC3=O)C2)=O)CCN(CC(F)F)CC1 Cc1cnc(CN2CCC(C(=O)Nc3cn[nH]c3)C(O)C2)c(C)c1 c1(CCC(N2CCC(C(C)NC(c3c(C)con3)=O)CC2)=O)nnc(O)nc1O C1(NC(C#C)=O)CC2(C1)CN(Cc1cc(Br)cc(I)c1)C2 CC1CCC(C(N2CCC(C)(CC(=O)NCC3CCCCS3)C2)=O)CC1 N1(C(Cc2c(C)occ2)=O)CC2CCN(C(=O)CC3(C)CCCO3)C2C1 Cc1cc(C(=O)NCC(F)CNC(=O)CCC(=O)c2cccs2)[nH]c1C C1(NC(CN(S(C)(=O)=O)C)=O)CCN(C(=O)COc2ccc(F)cc2)CC1(C)C C=CCC(C)(CC)C(=O)NCC1CCCN1C(=O)Cn1nc(C)nc1C Cc1c([N+](=O)[O-])ccc(N2CC(c3cc(F)cc(F)c3)C(O)C2)c1[N+](=O)[O-] C1(CC)C(OC)CCCN1Cc1ccc(C(=O)O)s1.CCOC c1(C2C(NC(c3n(CC=C)nnn3)C=Cc3ccccc3)C2)ccc(C#N)cc1 c1(OC)cccc(CC(=O)C(=O)NC2CC(CNC(c3cnc(C)[nH]3)=O)C2)c1 N1(CCC(=O)NCC2(NC(C(COC)C)=O)CCOC2)CCN(C2CCC2)CC1 N1(C(CNC(C(CC)C)=O)=O)C(C(=O)NC(c2[nH]c(C)nc2C)C)CCC12CC2 c1(CC)oc(C)cc1C(=O)NCCC(C)(C)NC(C1(OC)CCCCC1)=O c1(C(C(=O)N(CCCOCCNC(c2cnco2)=O)C)(F)F)ccc(F)cc1F c1(C(NC(NCC(C=C)(F)F)=NC)C)ccc(Cl)cc1Cl C1(C)(C(N2CC(SC)C(NC(c3cc(O)cs3)=O)C2)=O)CCCC1(F)F CC1(C)CC(=O)N(Cc2nc(Cc3cccs3)no2)C1=O C1(C(=O)NC2(Cc3ccc(CO)cc3)CCOC2)CCn2nnnc2C1 C(CC(=O)NCC)(C(F)(F)F)N.C=CCC(CC)C(=O)C(CNOC)=O C(=O)(C#CC1(C)CC1)NC.CCCC(C(=O)N(c1ccccc1)CCOC)OC CC(C)C(C)CC(=O)NCC(CC1CC1)C(=O)NC1(c2nc[nH]n2)CC1 Cc1cncc(C(=O)NC(CNC(=O)C(=O)N(C)C)C(C)(C)C)n1 C1(CCC(C)O)CCN(C(=O)C(c2ccncn2)C)CC1.c12cn(nn1)C2 c1(C(N2CCN(C(C=CCC)=O)CC(O)C2)=O)ccc2c(c1)nc(C)c(=O)n2C Cc1oc(-c2cccs2)nc1CC(=O)NCC1CCN1C(c1cc(C2CC2)ns1)=O N1(C(CCOCC(C)C)=O)CC2(CCC(C(=O)NC3CC3CC(C)(C)C)O2)C1 C(=O)(CCC1=NNC(=O)CC1)NC1CC(NC(c2cc(OC)no2)=O)C1 C1(C(=O)NCC2(F)CCN(C(c3cn(C)c(O)n3)=O)C2)CCC2(CC1)CC2(F)F c1(SC)ccc(C(=O)NC2(C)CN(C(C3CC(C)(F)C3)=O)C2)s1 N1(C(C(C(=O)OC)C)=O)CCC2(CC1)CC2C(=O)N(CCCCN(C)C)C c1(C(=O)NC2C(C)CCN(C(C(C)OC3COC3)=O)C2)cnc2[nH]ccc2n1 C1(c2cn(CCC3CN(C(C4(C=C)CCC4)=O)C3)nn2)CC2CCC1CC2 C1(C)(NC(CC(C)c2ccncc2)=O)CCCN(c2ccc(C(F)(F)F)cn2)C1 c1(NC(CC2CCC(=O)N2)=O)cccc(=S)n1O.C123CC1CN(C2)CCNC3=O C#CC1(NC(=O)CC2CN(C(C3CCCCN3CCC)=O)CC2C)CCCCC1 CC(C)(O)C(C(=O)NCC1(C)CCC(O)CC1)NC(=O)CCOCCCCO Cc1noc(C)c1CC(C)C(=O)NCC1CCCC1NC(=O)CSCC(F)F C1(NC(CC=C)=O)CS(=O)(=O)CC1NC(c1nn(C(C)(C)C)cc1Br)=O C=C(C)C1OCCC1CNC(=O)CC(C)(C)N(C)C(c1ccc(Cl)o1)=O Cc1nn(C)c(C)c1CCC(=O)NC1CC(CN(C(C2CC2(C)C(C)C)=O)CC)C1 C1(CNC(C2N(CC)CC2)=O)CN(C)CCN1C(=O)CSc1ccsc1[N+](=O)[O-] c1(OCC)nc(Cl)ccc1C(=O)NCC(CNC(c1c(C)ncnc1O)=O)OC C12COC3CN(CC13)C2=O.C1(c2cnc(C(=O)OCC)s2)C2CC3C(C2=O)C13 c12cn(nn1)CC1(CCC1)C2NCC1(C)CC1.CC(O)C(=O)N.C1(CC2CC2)CC1 c1(C(=O)NCC2CCCN(c3nc(C4CCCC4)ns3)C2)cnc2c(Cl)cccn12 C(C(C)(COC)NC(c1nocc1COC)=O)OC.c1(C(C)N)conc1CC c1(C(N2CCC(C3N(C(C4C(C)C4)=O)CCC3)C2)=O)cncc2c1CCC2 Cc1nc2oc1C(=O)NC2.C1(C(C2CC2)NC(=O)CCc2nccs2)CC2(CCC2)C1 C1(C(=O)NCC(C)(C)C(N)=O)(CC)CCN(C(=O)C(C)C(C)n2cccn2)CC1 c1(N2CC(CC)OCC2)ccc(S(=O)(=O)N2CCC(C)S(=O)CC2)cc1F O=C(CCCCCCCO)NC1CC(C(N2CC3(CCC(=O)NC3)C2)=O)C1 C(=O)(C(C)(C)C(C)(F)F)NCC1CC(OC)CN1C(C1(F)CCOC1)=O C(=O)(C1=NOC2COCC12)NC(CCCC)CNC(c1occc1C(C)C)=O c1(C(CCOC)(C)NCC(C2CCCC2)F)cc(Cl)cc(Cl)c1O c1(C(=O)NC2C=CC(CNC(C)=O)C2)ccc2c(c1)CC(=O)N2 C1(C(=O)Nc2cccc(O)n2)CN(C(C2CC=CCC2)=O)CC(F)(F)C1 C1(N=[N+]=[N-])(C(=O)NCC(=O)NCC)CCN(C(C2CCC2COC)=O)C1 c1(C(=O)NC(C(C)C)CCN(C)C(C2CC2C(F)F)=O)cc2cccnc2[nH]1 C1(NC(C(C(C)C)F)=O)COC2(C1)CN(C(c1ccoc1)=O)C2 C1(C)(C(=O)NCCCCNC(CCc2c(C)ncs2)=O)CCC(=O)N1 N1(C(c2c(NC)cnnc2)=O)CC(C(=O)NOCC2CCC2)C(C)(C)C1 C1(C(=O)NCC(C)NC(=O)C2=NNC(C(F)(F)F)C2)Cc2cc(F)ccc2O1 c1(C(=O)NC(CCN(C(C23CC(CCC)(C2)C3)=O)C)C)cnccc1OC C1(CCC)CN(C(C2CC3(CC3)C2)=O)CC1C(=O)N(C)C(c1cn[nH]c1)C c1(C(=O)NC2C(CNC(=O)CCC3NC(=O)NC3=O)COC2)cc(Cl)nnc1O N1(C(c2cc(OC)cc(C)c2)c2cccs2)CC(C)OC(C)(c2ccccc2)C1 c1(CN2C3CN(c4nccc(OC)n4)CC32)cc(Cl)cc(Br)c1OC C(=O)(C(C)CNC(C)=O)NC1(C(NOCCC#C)=O)CC1 c1(NC2C(NCc3cccc(OCCC)c3)COCC2)ccccc1C#N Cc1n[nH]c(C)c1CN(C)CCNC(=O)C(C)N(C(=O)C(C)(C)C)C CCCC(C(=O)NCCN(C)C(c1c[nH]nc1-c1ccnn1C)=O)OC N1(C(C(CC)COC)=O)CC(C(=O)N(CC(C)C)C(C)C)C2(CCC2)C1 N1(C(C2CN(C(C(F)=C(C)C)=O)CC2C)=O)CCC2(CCOC2)C1 c1(C(=O)NC2C3CN(C(C(C)c4ccon4)=O)C2C3)ccc2c(c1)CCN(C)C2 c1(C(N2CC(C)N(Cc3cc4ccncc4[nH]3)CC2)=O)cccc(S(=O)(=O)O)c1 C1(NC(c2ncn(C)c2)=O)CN(C(=O)C(F)(F)CC2CC2)CCC1CO C1(C2CCN(C(c3[nH]cc(CC)c3)=O)C2)CCCCN1C(C1CCC2CCC12)=O c1(SC)cc(C(N2CC(CNC(c3n[nH]cc3C)=O)C3CC23)=O)oc1C C#CC1(C(=O)NC(C)Cc2ccco2)CN(C(c2cc[nH]c2)=O)C1 c1(SCC2CC(C(=O)NC3CCN(C(COCC=C)=O)C3)C2)cc(Cl)ccc1F N1(C(C2(CCOC)CCC2)=O)CCC(NC(C2CCS(=O)CC2)=O)C(F)C1 Cc1nn(C)cc1C(=O)NC1(C(=O)NC2(CN(C)C)CC2)CC1 c1(C(=O)NCCN(C(C2C(C)C2C)=O)C)ccc(-c2cnnn2C)cc1 c1(C(=O)NC2C(NC(C3(C=C)CCC3)=O)CCCC2)cccc2[nH]ncc12 N1(C(COC2CCN(C)CC2)=O)CC2CC1CC2NC(c1cn(C)c(=O)cn1)=O n1(C(C)C)cnc2c(NC3CCC(CO)C3)[nH]c(=NC3CCCn4ncnc43)nc12 C#Cc1ccc(CC(N2CC(C(N3CC(OCC(C)C)C3)=O)C(CC)C2)=O)cc1 C1(C(=O)NCCC2(NC(c3cccnc3Cl)=O)CCCC2)CC2(C1)CC(O)C2 N1(C(C(c2cccc(O)n2)C)=O)CCC2CN(C(=O)CCC3CC(C)(F)C3)C2C1 N1(C(=O)OC(C)(C)C)CCCC1C(N1CC(C(C2CCOCC2)=O)C1C(C)(C)C)=O N1(C(C(C)=CC2CC2)=O)CC(C2CCCN(C(=O)C(CN(C)C)N(C)C)C2)C1 Cc1cc(N)cc(C(N2CCCCC2CCNC(=O)C2=CCS(=O)(=O)C2)=O)c1F C(=O)(CCCC(=O)N1CC=CC(C(=O)N(C)CCC2CCCN2C)C1)OCC CS(=O)(=O)C1CN(C(=O)C2=CCCOC2)CC1NC(=O)CNC=O c1(C(C)C)nc(NCC2(CO)CC(F)(F)C2)cc(=NC2CCn3nnnc3C2)[nH]1 C(C(=O)N(C1CN(C(c2c(Br)noc2C)=O)C1)C)(C(C)C)NC(=O)OCC C1(CCC)CN(C(c2cn(C)cc2C)=O)CC1NC(c1ccc(N(C)C)nc1)=O C#CCC(CC(=O)NCc1cc(C)sn1)NC(=O)C(C)C(C)C N1(C(C2CN(C)C2)=O)CCC2CN(C(c3cc4c(s3)CCSC4)=O)CC2CC1 Cc1ccc(C(C)NC(=O)NCc2cc(C#N)ccn2)cc1Cl C(=O)(C(C)(C)CC1CCCCC1)NC(C(C)NC(CN(C1CC1)CC)=O)CO C1(NC(c2c(OC)c[nH]n2)=O)CCN(C(c2oc(Br)nc2C)=O)CC1C c1(C(CC)N(C(c2cccnc2)C(=O)NC(C)C)C2CC2)ccccc1 CC(C(=O)NCC(C1CCCCN1C(C1CCC(O)C1)=O)(C)C)C(F)F C1(C(=O)NCC(N)=O)CCN(C(c2snc(Cl)c2Cl)=O)CC1 c1(NCC2(NC(c3cc(C4(C)CC4)n[nH]3)=O)COC2)ncnc2cccc(F)c12 CC(C)CC(CNC(=O)CC1SC(=N)NC1=O)NC(c1cc(C2CC2)on1)=O CC1CCCC1C(=O)NCC(C)(C1CCC1)NC(c1nncn1C1CC1)=O CS(=O)(=O)c1csc(C(N2CC(NC(c3cc(N)cc(O)n3)=O)C3(CC3)C2)=O)c1 n1(CCC)cc(C(=O)NC2CC(CNC(c3cc(C(C)(C)C)n[nH]3)=O)C2)c(C)n1 C(=O)(C1=CCCOCC1)N1CCC(C)(CNC(C2(F)CCOC2)=O)CC1 C(=O)(CC(C)CC(=O)NCC(C)NC(=O)Cc1cc[nH]n1)OC c1(CC2CC(OCC(=O)N(CCNC(COCC(C)C)=O)C)C2)ccsc1Cl C1(C(=O)NC(CCCNC(c2c(C)coc2C)=O)(C)C)CCCC1S(C)(=O)=O C1(CC(=O)OCCOC)CCN(C(CNC(=O)C(=Cc2ccccc2)C)=O)CCO1 C1(C)(C(N(CC(CC)NC(C2CCOC2C)=O)C)=O)CCN(CC)CC1 N1(C(C2(C=C)CCOCC2)=O)CCCC2(CCC2NC(c2cnoc2C)=O)C1 C(C(C)(O)CC(=O)N1CCC(C=CC(=O)NCCCCC(N)=O)CC1)OC CC1(C)CC(C(N2CC(CNC(C3CC(F)(F)C3)=O)C3(CC3)C2)=O)C(C)(C)O1 N1(C(CC(CC)C2CCC2)=O)CCOC(C)C1C(=O)N(C(C)C)CC1CCCO1 c1(CN(C(=O)CC2(NC(c3cocn3)=O)CCCCC2)C)cnn(C)c1O c1(OC)ccc(C=C(C#N)C(=O)N(C2CC2)C(c2ccc(F)cc2)C)cc1 C=C(C)CC(C)C(=O)N(C)CC1(NC(=O)C(F)(F)C2(OC)CCC2)CC1 Cc1ccc2[nH]c(C(N3CCC4CC4(NC(=O)C4=CCCCC4)CC3)=O)cc2c1C n1(CC(=O)N(C(CNC(C(C(CC)C)O)=O)C)C)ccc2nc(O)nc(O)c12 C(=O)(C(O)CCCNC(c1cnn(C2CC2)c1)=O)N(CCC(F)(F)F)CC C=C(C)CCC(=O)NCCCN(C(=O)C(CC)SC)CC1CCCC1 C(N=c1[nH]c2c(c(=NC(C)c3ncc(SC)s3)[nH]1)CSC2)c1c(OC)nccc1C C1(C(=O)NCC(C)(C)CC2CCC2)CCCC1C1CC1.n12cc(nn1)C2 c1(C(N2CCCN(C(CC(C=C)C)=O)CCC2)=O)cnc2[nH]c(C(F)(F)F)nc2c1 c1(C(N2CCCCC(CNC(=O)CC3CCCOC3)C2)=O)cc2ccnn2cn1 N#Cc1ccc(CNC2(c3nnnn3C3CC3)CCOC2)c2ccccc12 CC1(C)CC(NC(=O)CS(C)(=O)=O)CN(C(c2cc3c(s2)CCC3)=O)C1 C(=O)(CCS(C)(=O)=O)NC(C(C)(C)NC(Cc1ccc(C(=O)OC)cc1)=O)C c1(C(N2C(CNC(c3cnc(OC)nc3C)=O)CCC2)=O)ccc2occc2n1 c1(-c2cncc(C)c2)cnn2cc(C(=O)NC(c3ccc(Br)cn3)C)cnc12 C=C(C)CCC(=O)NCC1CC(F)(CNC(c2cccnc2CC)=O)C1 c1(CN=C(NC(CC)CC)NCC2COC(=O)O2)ccc(OC)c(S(N)(=O)=O)c1 N1(C(=O)OC(C)(C)C)CC(CC(=O)NC2C3CCCN3CCC2)OCC1(C)C C1(C(N(CCCN(C(=O)CNC=O)C)C)=O)CC2(CC2)CO1 C12(C(N(CCN(C(=O)CC3C=CCC3)C(C)C)C)=O)CCC(C)(C1)OC2 C(c1cn[nH]c1)=C(C)C(=O)NCCC(O)CNC(=O)C(C)(C)c1cscn1 c1(CC(CCCNC(=O)C(N2CC3CCCC23)=O)CO)cc(F)cc(F)c1 C12(CNC(c3c(C)nn(C)c3F)=O)CCCC1N(C(=O)C1=NOCC1)CCC2 N1(C(CC2CC(=C)C2)=O)CC(C)(C(=O)NC(C)CCSCC)C1 C1(C(N2CC(NC(C(=O)NCC)=O)(CO)C2)=O)CCC2(CCC2)CO1 c1(OC)ccc2nc(C(=O)NCC(N3CCC(O)C(F)(F)C3)=O)ccc2c1Br CCCCCC(C)(C)C(=O)N1CCCC(CNC(C2CCCCCCC2)=O)C1 c1(C(N(CC(=O)NC(CC)COC)C2CCC2)=O)ccc(C)cc1C N1(C(C2CCCC23CCC3)=O)CCCC2CCNCC12 N1(C(c2c(CC)ncs2)=O)CCC2CC2(NC(=O)C=Cc2csc(C)n2)CC1 C1(NC(=O)CNS(=O)(=O)N(C)C)CC12CCC(C(=O)NC(CC(C)C)C)CC2 CCCS(=O)(=O)CC(=O)NCC(C)CNC(c1cnn(-c2ccccc2F)c1)=O C1(C(=O)NCC(COC)O)CC=CCN1C(=O)CC1(OC)CCC1 N1(CC(=O)NC(C)C(N2CCS(=O)(=O)CC2)=O)CCc2ccccc2C(C)C1 C1(NC(C2CCCS2)=O)CC12CCN(C(=O)CCC1CC1(F)F)C2 C1(NC(C(CSC)(C)NC(c2ccsc2C)=O)=O)CCCOC12CCC2 C(=O)(CC(C(F)F)Sc1ccc(F)c(F)c1)NC1C(OC)COCC1 C1(C(N(CC#C)CC2CCCO2)=O)CCCCN(C(C2(C#N)CCCC2)=O)C1 c1(-n2c(-c3ccn(C4CC4(F)F)n3)nc(CCCOC)n2)cc(F)cc(F)c1 c1(CNC(C2N(C(N)=O)CCCC2)=O)nc(CNC(=O)CC2CC2(Cl)Cl)cc(O)n1 C1(CNC(C=C2CCC(C)C2)=O)CN(C(=O)Cc2cnn(C)c2)CC2(CCC2)O1 C1(F)(CNC(C(C)(C)C)=O)CCC(NC(=O)CN2CC(=O)NC2=O)C1 CC1(F)COCCN(C(=NCC=CBr)Nc2ccccc2)C1 N1(C(C(C)c2cccs2)=O)CC(C(=O)NC2CCC(C)(C)OC2)C2(CCC2)C1 CCCC(C(=O)NCC(c1csc2ccccc12)NC(C1CC1C#N)=O)C(C)C CN1CCCC(CC(=O)NCCC2(C(N3CCN(CCO)CC3)=O)CCC2)C1 C1(C)(C(=O)NC2(CC=C)CCN(c3cc(C(C)C)ncn3)C2)CCCCC1(F)F CN1CCC2OCCN(C(c3nc(-c4cnn(CCF)c4)cs3)=O)C2C1 C(=O)(C1=CCCCCC1)NCC1N(C(c2cn(COC)nc2C)=O)CCC(C)C1 S(=O)(=O)(c1ccc(F)c(Br)c1)N.c1(C(N2CC(C)C2CN)=O)cc(I)cn1C C1(N(C(C(=O)NCCOC)=O)CCO)CCN(C(=O)Cc2scnc2C)C1 N1(c2cc(C)nc(CO)n2)CCn2ncc(CNC(=O)C(CC(C)C)C(N)=O)c2C1 C1(NC(C(CC=CC)C)=O)CCCC12CN(C(c1cc(C(N)=O)cs1)=O)C2 c1(CC)nc(C)c(C(=O)NC2C=CC(CNC(=O)CCP(C)(C)=O)C2)c(C)n1 C=C(C)CCCC(=O)NC(C)CCCNC(=O)CSc1ccncc1 C1(NC(=O)COCCF)CC2CCC1(NC(c1csc(C3CCCO3)n1)=O)C2 N1(C(C2(CC=C)COC2)=O)CC(NC(C2CCCOC2)=O)CC2(CC2)C1 CN1CCC(C(=O)N(C2CCCC2)CCNC(=O)Cn2ccccc2=O)CC1 c1(OC)cc(CCC(N2CC(OC)C(NC(=O)CC3CC4(CC4)C3)C2)=O)ccn1 c1(N2CCCC(OC)C2)nc2ccc(Cl)cc2c(=NCC2CN(C)CCO2)[nH]1 C1(C(=O)NC(CC(CC)OC)OC)CC2(CC(C(C3CC4CCC3CC4)=O)C2)C1 N1(C(C(C)C2(O)CCC2)=O)CCCC(O)(CNC(=O)Cc2cn[nH]c2)C1 C1(NC(C(CC)NC(C)=O)=O)CCN(C(=O)C(C)CN(C)C(C)=O)C12CCC2 Cc1n[nH]c(C)c1CCNC(C1C2CN(CC(=O)NC(c3cccs3)C)CC12)=O CCC(CC)(CCNC(c1ccnc(O)c1)=O)NC(C1CCN(C(C)C)CC1)=O C(CN=c1[nH]nc(O)s1)OC1CCN(C(C2N(N=O)CCCC2)=O)CC1 CCCCCC(C)(C)C(=O)N1CCOCC(C(N2CCC(=O)NC(=O)C2)=O)C1 c1(CC(=O)N(CCCCN(C(c2c(COC)cc[nH]2)=O)C)C)ccnnc1O C1(C(=O)OCC)CCN(C(=O)C(n2cc(C)nn2)C)C12CCSCC2 CCCC(C(=O)N1CCCCC1CCC(=O)NCC1=CCCCC1)NC(N)=O C1(C(=O)NC2C(NC(=O)CSc3nc[nH]n3)CC2)CCc2ncncc2C1 C1(NC(CC(CC)(F)F)=O)CC2CC(C1)N(C(=O)Cc1ncoc1C)C2 C1(NC(=O)COCC2CCOC2)CCN(C(c2cc(CCO)on2)=O)CC1F c1(C(=O)NCCCNCc2n(C)ncn2)cccc(-c2ccncc2)c1 Cn1nc(CNC(C2CC2(F)Cl)=O)c2c1CCN(C(=O)C(C)(C)c1cccs1)C2 CCCCC(CNC(c1ocnc1C1CCC1)=O)NC(c1ccc(C2CC2)o1)=O N(C1CCCOc2cc(Cl)ccc21)CC1C(C)C1(F)F C(=O)(C(C(C)(C)C)SC)NCC12CC(NC(C(CC#C)C)=O)(C1)C2 C(=O)(C1=CCCC1(C)C)NC1(C2N(C(c3scc(OC)c3)=O)CCC2)CC1 C(C(C(C)(C)C)NC(=O)C(C)Cc1ccc(F)cc1)NC(C(CC)N(C)C)=O S(=O)(=O)(c1ccc(Cl)c(NC(NC2CCn3ccnc32)=O)c1)NCC=C c1(C(=O)OC)cc(Br)sc1CN1CCC(C(=O)NCC(N)=O)C1 c1(C(N2CCC3(NC(c4cc(SC)oc4C)=O)C(C2)C3)=O)nc(C)c(C)[nH]c1=O N1(C(C(C(CC)C)C)=O)CC2(C1)C(NC(c1ccc(CF)cc1)=O)CCS2(=O)=O C=CC1(CC(=O)NCCC(O)(CC)CC)CN(C(C2CC2C2CCC2)=O)C1 N1(C(C2(C(=O)NC)CC2)=O)CC2OCCN(C(C3SCCS3)=O)C2C1 C(c1ccc(Cl)c(Cl)c1)=CC(=O)NC1CC(C(=O)Nc2ccc(I)cc2Cl)C1 Cc1cccc(C(=O)NCC(C2CCCCC2)NC(C2COC(C)(C)C2)=O)c1 C1(C(=O)NC(CNC(=O)OC)C)N(C(=O)CCCNC(N)=O)CCC1(C)C c1(C(N(CCC)CCNC(C2(C3CC3)CCC2)=O)=O)cnc(Br)c(O)c1 c1(C(=O)NC(C)CNC(C2CN3CCCC3CO2)=O)cc(=O)c2ccccc2[nH]1 c1(CNC(CC2(C)CC2)=O)cn(CC2CNCCO2)nn1 N1(C(C(CCC)OC)=O)C(C)CC2CN(C(c3cccc4oc(=N)[nH]c34)=O)CC12 CC(CCN(C)C)C(=O)NC(C(=O)NCCCc1ccco1)c1ccoc1 C1(C(=O)NC2CC(N(C(=O)C=CC(F)(F)F)C)C2)CNC(=O)CC12CCC2 C12(CNC(c3cc(C)sc3C)=O)CCCCC1CN(C(c1csc(C(F)F)c1)=O)C2 n1(CC)cc(CNC(=O)OC)cc(Br)c1=O.C12CCCC1(C)NC2=O n1(CCC)nc(C)cc1C(=O)NCC1(O)CN(C(=O)C(C)Cc2ccco2)C1 N1(C(C2(F)CCC(=O)CC2)=O)CC(NC(C2(c3ccsc3)CC2)=O)C(C2CC2)C1 Cc1ccc(C(=O)N(CC(C)(C)NC(=O)Cc2ccnn2C)C)c(Cl)c1C c1(N2C3CCC(NC(c4cc(C)sc4C)=O)C(C3)C2)ncnc2ccc(Cl)cc12 C(=O)(CC(F)(F)Cl)N(CCN(C(C(c1ccc(CC)s1)=O)=O)C)C(C)C c1(CCC)cnnc(C(=O)N(C2CN(C(c3sccc3CO)=O)CC2F)C)c1 C1(C(N2CCC(NC(=O)C(=O)N(c3ncc[nH]3)C3CCC3)C2)=O)C(F)(F)C12CCC2 N1(C(c2c(CC)scn2)=O)CCCC(CNC(=O)C(C)Cc2cnn(C)c2)C1 c1(C(=O)NCC2CCC(CNC(c3cc(C)oc3C)=O)CC2)cc(Cl)nc(Cl)c1 N1(C(C(CC)CC(C)C)=O)CCCC2(CCCN2C(c2cc3scnc3[nH]2)=O)C1 C1(NC(c2c(COC)cco2)=O)CCN(C(=O)CS(=O)(=O)NC2CC2)CCC1CO N1(C(CC2CN(C(C)=O)C2)=O)CCC(NC(=O)COc2cnn(C)c2)C1 N1(C(C2(C)CCN(C)C2)=O)CCC(C2CCC2)(C(=O)N(C)C)C1 C1(NC(COCCCC)=O)CC2CN(C(=O)Cc3cnc(C)o3)CC12 N1(C(C(CC)O)=O)CCC2CN(C(=O)C(C)(C)c3cscn3)CC12 N1(C(C2C(C=C)CC2)=O)CCCOC(CNC(C2CCCCC2)=O)C1 c1(CC)ccc(Br)cc1C(=O)NCC(CNC(c1cc(C)ns1)=O)OC CCCC(C(=O)OC(C)C(F)F)N(CC(=O)NCc1ccccc1)C N(S(=O)(=O)NC1c2ccccc2OCC1C)C(CC(C)c1ccccc1)=O N1(C(CS(CC)(=O)=O)=O)CCOC2CCN(C(c3cc(C4CC4)ccn3)=O)CC12 C=C1CC(C(N(C2(c3nn[nH]n3)CSC2)C2CC2)=O)C1 N1(C(CC(C(N)=O)NC(N)=O)=O)CC2(NC(=O)CNC=O)CCCC2(F)C1 c1(CNCC2C(C(N3CC(C#N)C3)=O)C2)c(Br)cc(Br)c(O)c1Br N1(C(CSc2cccc(C)c2)=O)CCN(C(c2ccn(C(C)C)n2)=O)C(CF)C1 N1(C(=O)CC2CCCO2)CCCC2(CCN(C(C34CC5CC3C4C5)=O)C2)C1 S(=O)(=O)(CC(F)(F)F)NC1C(C(=O)Nc2cnc(Br)cn2)C1 C1(NC(c2cccnc2O)=O)CC2CC1N(C(=O)CCOC1CCOCC1)C2 C1(C(=O)NC(c2ncccn2)CC)C=CCN1C(c1coc(CO)c1)=O CC(CF)CC(=O)NC1(c2ccccc2)CC1.C12CN(C1)C2=O c1(OC)cc(C(=O)NC(C)CCNC(c2ccc(O)nn2)=O)c(C)cc1O C(c1cccc(F)c1Cl)=CC(=O)NC(CNC(c1c(C)oc(Cl)n1)=O)(C)C c1(CC)cc(C(=O)NCCc2ocnc2CNC(=O)CC2CC(F)C2)ncn1 C(=O)(CCC(O)C(C)(C)C)N1CC(OC)C(NC(=O)C(C)Cc2cnco2)CC1 CCC(F)(F)CC(=O)NCC1CN(C(c2cccc(CO)c2)=O)CC1(C)C c1(CCC(=O)N(CC(CNC(COCC(=C)C)=O)(C)C)C)c(Cl)cncc1Cl c1(OCC(=O)NCC2(NC(=O)CCc3cnn[nH]3)CCOC2)cc(F)cc(Cl)c1 Cc1cc(C)c(C(N2CC(O)(C(F)C(=O)NC34CCN(CC3)CC4)C2)=O)c(C)n1 C=CCC(CNC(=O)C(C)(C)C1CCC1)C(=O)NCC1CCC(=O)NC1C N1(C(CCC=C)=O)CC2COCCC2(NC(c2ncn3c2CCCCC3)=O)C1 c1(C(=O)NC(CCC)C(=O)OCc2cnccc2Cl)cc(Cl)c(C(F)(F)F)c(Cl)c1 CC1=C(C(=O)NC2(C)CC(NC(=O)C(c3c(F)cccc3F)N(C)C)C2)CCO1 c1(C(N2CC(NC(C(C)c3cccs3)=O)C(O)C2)=O)cc2cccnc2cn1 N1(C(C(C(CC)O)C)=O)CC(C2CCCN(C(=O)CCc3cncs3)C2)C1 N1(C(=O)OC(C)(C)C)CC(CNC(=O)NC2CC23CCOCC3)OC2(CCC2)C1 CCCC(CNC(=O)C(CNC(=O)C=CC1CCC1)CCC)CCO C(=O)(CC(C)C(C)(C)NC(c1nc(C)ccc1F)=O)NCCC(CC)O c1(CNC(CC2CCCN(C(=O)C=C3CCC3)C2)=O)cnc(O)nc1O C(CN=C(NCC1CCOC1)N1CCCC(NC(N)=O)C1)n1c(C)cc(C)n1 C1(C(=O)NC(CC(=O)OC)C)CCCCCN1C(=O)C(=O)N(C)C n1(CC(=O)NCC(CNC(c2c(CC)occ2C)=O)(C)O)c(C)cc(C)nc1=O C(=O)(C1CCc2ccccc21)NC1CCCCN(C(c2c(C)nncc2)=O)CC1 N1(C(CCSCC(C)C)=O)CC(NC(C2(C)CC2c2ccccc2)=O)C(C)C1 C1(CC(N2CC(CC(C#C)C)C2)=O)CCCN(C(c2ccc(OC)o2)=O)C1 CC1(CNC(N2CCc3ccc(O)cc32)=O)COCC2CCCN12 C(C(C)NC(C1(C(=O)N(C)C)CC1)=O)CC.C1(=O)CNCCN1 c1(C(=O)OCC)c(OC)cc(NC(=O)CC(C)C(C)(C)C)cc1I c1(C(=O)NCC2CN(C(C3CC(CF)C3)=O)CCO2)cccc(C#CC2CC2)c1 CC1(C)CN(C(=O)CC2CCC(=O)NC2=O)CC1NC(c1ocnc1C(F)F)=O N1(C(C(c2cn(C)nn2)NC(C#CC(C)C)=O)=O)CC(O)(C2CCC2)C1 N1(C(c2ncc(C)nc2)=O)CCC(NC(c2nccnc2Cl)=O)C(F)C1 C(C(=O)NCCC(C)(C)NC(C1(c2ccccc2)CC(=C)C1)=O)(C(C)(C)C)SC C1(C(=O)NCCc2cn(C)nc2)CC(F)CN1C(=O)C=Cc1ccco1 N1(C(C(CC)(C)O)=O)CCCC(C)(C(N2CCC(F)(CO)CC2)=O)C1 c1(C(=O)NCCCNC(CC(C=C)(C)O)=O)cc2c(F)ccc(Br)c2[nH]1 c1(C(=O)NC(CC)CN(C(=O)Cc2cocn2)C)ccc2n[nH]cc2n1 C12(CO)CCCN(C1)C(=O)C(COC)N2.C1(C(=O)OCC)CCN(C(N)=O)CC1 C1(CN(C(=O)CS(N)(=O)=O)C)CN(C(C2(c3cccc(Cl)c3)CC2)=O)CC12CC2 C1(C(=O)NC(C2CCC2)C)Cc2ccccc2CN1CCSc1ccccc1 N1(C(C(Cc2ccccc2)N(C)C)=O)CCOCC(CNc2ncc(Cl)cn2)C1 CC1=NN(C)C(=O)C1CC(=O)NCCNC(c1cc(C2CCCCC2)oc1C)=O C(C(C)(C)CCNC(C1CCCC(=O)N1)=O)NC(COCc1onc(CC)n1)=O c1(CC)nc(C(N2CC(NC(=O)CC3CCCNC3=O)CC2C)=O)c(C)o1 N(C1CCc2cccnc21)C(C1N(C(=O)CSCc2cccnc2)CC(O)C1)=O N1(C(C)=O)CCC2C(CCN2C(c2coc(CO)c2)=O)C1.C=C1CC(c2nc[nH]n2)C1 CC1CCCC12N(C(C)(C)C)C(=O)O2.c1(N)cc(C2CCCCC2)on1.C(N)=O c1(OCC)ccnc(C(=O)NC(C)CNC(=O)CSc2cccc(C)c2)n1 C1(C(=O)NCC(C2(C)CC2)NC(CSC(C)C)=O)CCCC12CC2 c1(C(=O)NC2(C)CCN(C(C3(C4CCCCO4)CC3)=O)C2)ccc(Cl)c(O)c1N C1(C(N2CC(CCNC(C(C)(C3CC3)OC)=O)C2)=O)CNC(=O)CC12CCC2 N1(C(C(CC)N(CC)CC)=O)CCC(C2CC2)(CNC(C2(OC)CC2)=O)C1 C12(C(=O)NC3(CCn4cc(CCCCC)nn4)CCOCC3)OCCCC1C2(F)F N1(C(C=CCOC)=O)CC2C(NC(=O)Nc3cc(-c4ccccc4Cl)no3)C2C1 c1(NC(COCC)C)nc(N2CC(=O)NC(C)(C)C2)c2sccc2n1 CC(CC(=O)NCCCOCCC(=O)N(CC(O)C1CCC1)C)c1ccco1 c1(C(=O)NCC(O)CC(=O)NOCc2ccnn2CCF)cnn(CCF)c1 N1(C(CSCC=C)=O)CCC(C)C(N(C)C(c2cc(C3CC3)no2)=O)C1 c1(NCc2c(C)ccnc2)cc(Br)ccc1S(=O)(=O)NCCN=c1cncc[nH]1 c1(C(N2CC(C)C(NC(C3(C(F)(F)F)CCC3)=O)CC2)=O)cc(F)c(N)cc1F c1(CC)cc2c(CC(=O)NCCCCN(C(=O)C(C)COC)C)csc2s1 N1(C(c2ccc(-c3ccccc3)o2)C(=O)NC(C)C)CCCCC1c1nccs1 N1(C(C(C(C)C)NC(C)=O)=O)CCCC(NC(=O)COCC2CCCC2)C1C C1(c2ccc(C)cc2)CC1N=c1[nH]c(=NC2CCSCC2)[nH]c2ncn(C)c12 C1(c2n(CC=C)nnn2)(NC2CC(C)(C(N)=O)C2(C)C)COC2(CCC2)C1 C1(C(=O)NC(CCN(C(c2c(CC)oc(C)c2)=O)C)C(C)C)CCC(C)(C)CC1 c1(OC)ccc([N+](=O)[O-])c(NC(=O)Nc2ccsc2OCC(F)(F)F)n1 C1(NC(c2ccc(C#C)cn2)=O)CCN(C(C2CCC(C)(C)O2)=O)CC12CCC2 O=C(CCC(F)F)NNC(=O)c1cccn1CC1CCC1 C1(C(=O)NCCOCCN(C)C(C2CCCN2C)=O)CC12CCS(=O)(=O)CC2 C(C(C)C(F)C(=O)NCCN1CCCNC1=O)NC(c1ccc(C#C)o1)=O C(CCCCC(=O)N1CCC(C(C)(C)NC(c2csc(C#N)c2)=O)C1)=CC C1(C(C)NC(=O)NCc2cnns2)CCCCO1 C(=O)(C1=CCCCC1C)NCc1nc(C(=O)NCC(C(C)O)(C)C)c(C)o1 CC1=C(C(=O)NCC2(C(C)(C)O)CN(C(=O)CC3CCCN(C)C3)C2)COCC1 n1(-n2c(Cc3c(C)cccc3)nc(-c3cccc(C)n3)n2)c(=O)oc2ccccc12 C12(C(=O)NC(C)CN(C(=O)CCSCC(N)=O)C)CC(C(C)C)(C1)C2 C12(C(=O)NC3(C)CCCN(C(=O)CCc4ccsc4)C3)CC3CC(C(=O)N1)C2C3 C(=O)(C1=NOC(C)(C)C1)NCC(CNC(c1nn(C)c(C2CC2)c1)=O)(C)C C1(F)(CNC(CCSC)=O)CCC(CNC(=O)CC2CCCC(=O)C2)CC1 Cc1cc([N+](=O)[O-])cc(C(=O)NCCC(O)CNC(=O)Cc2ccon2)c1Cl N1(C(Cn2cc(CCSC)nn2)=O)CCOCC1C.C12CC(C1)C2 C(=O)(C(O)C(F)F)C(c1ccccc1Nc1ccc(Cl)cn1)=O.C1(N)CCNC1 c1(N2CCC(NC(c3nncc(OC)c3)=O)C(F)C2)ncc2c(n1)COC2 C(CO)(CCCCNC(=O)C(O)c1ccsc1)NC(c1c[nH]nc1[N+](=O)[O-])=O CS(=O)(=O)c1cc(C(N2CCC(NC(c3ccc(N)cc3)=O)C(CO)C2)=O)co1 N1(C(c2cc(CC)no2)=O)CCC(CO)(NC(=O)CCc2csc(=N)[nH]2)C1 c1(C(=O)OCc2ccc(-n3cncn3)c(F)c2)cc2n(n1)CCNS2(=O)=O c1(NC2C3CN(C(=O)Nc4ccc(C#N)cc4)CC2C3)cc2cn[nH]c2cn1 c1(CC)nn(C)cc1C(=O)NCCCC1CCCCN1C(C1CC(=O)N(C)C1)=O C12(NC(CC)=O)CCN(C(=O)CCc3ccc(N(C)C)nc3)CC1C2 c1(CSCc2onc(C(N3CCCC(C(=O)OC)C3)=O)n2)c[nH]c2nccc-2c1 N1(C(C(C)(C)Nc2ccc(Cl)cn2)=O)CCC(C)(c2ccc(F)cc2)CC1 c1(C(C)C)cc(C(=O)NCC(CO)NC(=O)C(F)n2cccn2)ccc1F c1(C(=O)NC2(C)CCN(C(C3(C)CCC3)=O)C2)ccc(Br)c(O)n1 C1(C#CC(=O)NCC2CN(C(=O)C#CC3(C)CC3)CC23CCC3)(CC)COC1 C12(C(=O)NCc3c(OC)ccnc3)CCN(C(c3coc(CO)c3)=O)CC1C2 Cc1ccc2c(c1)SC(C(N1CCC(NC(c3cccnc3)=O)C1(C)C)=O)C2 C(=O)(CCC(=O)N1CCC(O)CC1)NC(CC(C)NC(C1(F)CCC1)=O)C c1(C(N2C3CC(CNC(C(COC)OC)=O)C2CC3)=O)cnn2c1OCCC2 c1(C(=O)NC2(C(N(C(C)CC(N)=O)C)=O)CCC2)ccc(=N)[nH]n1 N1(C(Cc2cn(C)nc2C(F)(F)F)=O)CCN(C(=O)CCC#N)CC(C)(C)C1 C(N=c1cc(C)n(C(C)(C)C)[nH]1)c1c(C(COC)C)cccc1 CC1CC(NC(C2CCCS2)=O)CCN1C(=O)CSC(F)(F)F C(CCC(=O)N1CC(CCO)C1)(C(C)C)NC(C1C(CC)N(C)CC1)=O C1(NC(c2nc(CC)oc2)=O)CCN(C(=O)CCC(C)(F)F)CCC1CO N1(C(C(CC)c2ccccc2)=O)CC(NC(=O)C2=CCCSC2)C2CC2C1 c1(OC)ccc(C(=O)NCCN(C)C(C23C=CC(CC2)C3)=O)nc1Cl c1(C(=O)NCC(CCCC)NC(c2ccc(C(F)F)o2)=O)cccc(Cl)c1OC C1(CCNC(c2cc(C)sc2)=O)CN(C(=O)C(C#N)C2CC2)CCO1 C(=O)(CC(C)C(F)(F)F)C(C=CCNC(C)C(=O)N(C)CCF)=O.CO c1(C(=O)NC2CC(NC(=O)Cc3ccccc3O)C2)ccc2c(c1)S(=O)(=O)NC2 C1(C(=O)NCC(C)(CO)CO)CC(N=[N+]=[N-])CN1C(C1CCC(=O)C1)=O c1(C(C)=O)ccc(C(N2CCC(O)(CNC(=O)C=Cc3cnccn3)C2)=O)nn1 C1(C(=O)NCCN(C(c2c(N)cncc2)=O)CC2CC2)CCc2nccn2CC1 N1(C(c2cc(CNC(c3cn(CC)nc3C)=O)[nH]n2)=O)CC2CC(C)C2C1 C#CCCCC(C)C(=O)NCC1CN(C(C2CCCN2C)=O)C1 C(=O)(CC(C)C(F)(F)F)NCC(CNC(c1nnsc1N)=O)OC C1(CC)CN(C(c2cccc(C(C)C)c2)=O)CCN1C(=O)C=C1CCN(C)CC1 CC(CO)CCCN(C(=O)Cc1csc(CN)n1)C C1(CC(=O)NC(CCN(C(CC2CC(=C)C2)=O)CC)C)CCC(C)(C)O1 c1(C(N2CC(C)N(C(C3C(C)C3C)=O)CC2)=O)cc2cc(Br)ccc2nn1 C(=O)(CCCCCO)NCC(C)CN(C(=O)C1=COCCC1)C c1(OC)ncccc1S(=O)(=O)NC(CCCO)C(C)C c1(C(=O)NCC2N(C(c3cc(C)ncc3C)=O)CCCC2)cc2ccccn2c1 Cc1sc(Cl)c(C(N2CCCCC(CNC(=O)C=CC3CCOC3)C2)=O)c1C C1(C(N2CC(Nc3ncnc(OC)n3)CC2C)=O)CC2CCCCN2C1 CCC(C)(C)C(=O)C(=O)N1CCC(OCC(=O)N(CCCc2ccco2)C2CC2)C1 CN1CCN(C(=O)CCOc2cccnc2)CC1C1CCOCC1 CCC(C)(C)C(O)C(=O)N(CCNC(=O)C=CC(C)CC)C1CC1 c1(CC(=O)NC2CCN(C(C(C(C)C)SCC)=O)C23CC3)cccc([N+](=O)[O-])c1 C1(NC(Cn2c(C)nnn2)=O)CCCCC12CCN(C(C1(O)CC(F)(F)C1)=O)C2 CC(Cl)(Cl)C(=O)N1CC(CO)(NC(C23CC(O)C2C3)=O)C1 c1(N2CCC(N(C3CCCO3)C(N3CCN(C(=O)C4CC4)CC3)=O)C2)ccccc1Cl N1(C(C(=O)NC)=O)CCC2(CC1)CC2(C)C(=O)NC(c1nccs1)C CCC(C(=O)N(CCC(C)(C)NC(=O)CC1CC1)C)n1ccnc1 c1(NC(C2N(C(CNS(CCCOC)(=O)=O)=O)CC2)=O)cncc2c1CCCC2 CCC(CC(=O)NCC1COCC1NC(c1cccc(O)n1)=O)SC c1(-c2c(CC=CCOC)cccc2C)noc(C2OC(=O)c3c(Cl)cccc32)n1 C#CC1(O)CCN(C(=O)CC2CCC(NC(=O)CC(C)CC(=O)OC)C2)CC1 C1(O)(c2cn(Cc3cccc(C)n3)nn2)CCN(C(C2CCC(=O)N2)=O)CC1 C1(NC(=O)NC2(C(=O)OC(C)(C)C)CC2)CC(CS(N)(=O)=O)C1 C(CN=c1nc(C)c(C)c[nH]1)OCc1c(F)ccc(OC)c1F c1(C(=O)NCCCN(C)C(C2(C)CCCO2)=O)ccc(N)cc1O C1(N=[N+]=[N-])(C(=O)NCC(C(CC)C)CO)CCN(C(=O)CN2CCCC2=O)C1 Cc1ncncc1C(N1CCC1(C)C(=O)Nc1ccc(I)nc1)=O CON=CC(=O)NCC(C)(Cn1cccn1)NC(C1CC(=O)C1C(C)(C)C)=O c1(CC)cc(C(=O)N2CC(=O)N3CCC3C2)n(C)n1.c1(NC)ccccn1 N1(C(C(CCSC)NC(C2CCC(C)(C)CC2)=O)=O)CCC(C)(C2CC2)C1 C(CCCS(C)(=O)=O)CCN1CCN(C)CC1.CCC(C)(C)N1C(=O)C(=O)NCC1 CCCCC(CC(=O)NCc1nnnn1CC)NC(C1(C)SCCCS1)=O C1(CC(N2CC(CCNC(C(C)OCC)=O)(OC)C2)=O)CCCCC1C(F)(F)F c1(C(N2CCN(CC3CCCC(C)C3)CC2C)=O)cnn2ccccc12 c1(C(=O)NC(CNC(C2OCCN(CC)C2)=O)C)cc(F)cc2ccoc12 C1(F)(C(N(CC(=O)OC(C)(C)C)CC)=O)CCCN(C(c2coc(C3CC3)n2)=O)C1 C1(C(N2CC(CN(C(=O)C=Cc3cnccn3)C)C2)=O)CC2COCC2C1 n1(CC(N2C(C3(O)CN(C(CC4CC(OC)C4)=O)C3)CCC2)=O)cnccc1=O N1(C(CCC(=O)NC)=O)CC(C)C(NC(c2cnn(C)n2)=O)C(C)C1 S(=O)(=O)(c1ccc(NC(=O)NCc2ccc(SC)cc2)cc1)N(C(CC)CC)C C1(CC=C)(NC(=O)CCC2CCC(=O)NC2)CCN(C(=O)COCC(=C)C)C1 C1(C(N2CC(CCNC(C3CC(N4CCCC4)C3)=O)C2)=O)CC(C(F)(F)F)CO1 C1(C(c2cnc(-c3ccsc3)s2)Nc2n(CCCF)nnn2)CCCCC1(F)F C1(C(=O)NC2C(NC(CCSCCC)=O)CCOC2)CCCCCS1(=O)=O C(=O)(C1=CC(C)CC1)NCC1(NC(Cn2c(C)c(Cl)cn2)=O)CCC1 C(=O)(CCCCC(N)=O)NC(C(C)NC(N)=O)C(C)C.CC(C(F)F)=CC=O CN1CCC(OC(=O)Cc2ccccc2)C1(C)C.C1(=O)C(=O)NOCCCN1 C1(COC)(OC)CCN(C(=O)CCCN2CCCCC2)C1.C(C1C(=O)N1)OCC CC1(CNC(=O)Cn2ccccc2=O)CCCC1NC(c1cscc1F)=O CN1N=C(CC(=O)N2CCC3CN(C(c4ccncc4)=O)CCC23)CC1=O CC1COCC(C(N2CCC(C(N3CCC(O)(CO)C3)=O)(C(C)C)C2)=O)O1 N1(C(CCCOCC)=O)CC(C)CN(C(c2ccc(C)c(F)n2)=O)CC1C C1(NC(=O)Cc2cc(O)ccc2Br)CCc2nc[nH]c2C1 c1(CCN(C)C)cccc(C(=O)NCC(O)CNC(C2(C)CCC23CCC3)=O)c1 C1(C)(CC)CCC(C(=O)NCC#CCNC(=O)C(F)(F)C2CC2)O1 c1(C(=O)NC(CCOC)CNC(c2nn(C)c(C)c2Cl)=O)c(O)nnc(C)c1C C1(C(=O)NCCCC(C=C)(C)C)CN(C(=O)CC(C)C(F)(F)F)CC12CCC2 Cc1nnc2n1CC(C(=O)N(C)CCNc1nccc(C(=O)N(C)C)n1)C2 Cc1ccc(CC(N2CCC(C)(C(=O)Nc3cccc(F)c3C)C2)=O)c(C)c1 CN1CCCC(CNC(c2ccc(CCNC(=O)CN3CCNC3=O)cc2)=O)C1 N1(C(C2CC(OC)C2)=O)CCC2(CC1)CC2CNC(=O)C1=C(C)CCOC1 C1(CCC(=O)NCCCN(C(C2(CCF)CCC2)=O)CC)CCCN(C)C1 C1(CN(C)CC2C(C)=NOC2=O)CCCCNC1=O c1(C(=O)NCCC2CCCN(C(CC3CCN(C)CC3)=O)C2)ccc(F)c(O)c1 N1(CC(n2ccc(-c3cnccc3C#N)n2)C)CC2(CCCCC2)c2ccccc21 c1(C(N2C(C(=O)NC3(C(C)C)CC3)CC=CC2)=O)c[nH]c2ncccc12 CC1(C)CN(C(=O)CC(F)(F)F)CC2(CN(C(c3ccc4c(c3)OCC4)=O)C2)O1 c1(CC)ncncc1C(=O)NCCCOCCCNC(C1CCCC(CC)C1)=O c1(C(=O)NCC(CC(C)C)NC(Cc2c(C)scc2)=O)cc(O)nc(C2CC2)n1 S(=O)(=O)(c1ccc2c(c1)nnn2C)NCC(C#C)CC1CCCC1 C12CCC(O1)CONC2=O.C(=O)(C(C1(C)CC1)CC(F)F)NC1CC1 Cc1ccc(C(N2CC(C)CC2C(=O)NCC(C)(F)C(C)(C)F)=O)nc1O CN1CC=C(C(=O)NC(CNC(=O)Cn2cc(C3CC3)cn2)C(C)(C)C)C1 c1(SC)cncc(NC(=O)CC(C)N(C)C(C2(CCN(C)C)CC2)=O)c1 c1(C(=O)NC(CNC(=O)CC2CCC3CC23)CO)ccc(F)c2[nH]ccc12 C1(C(N2CC(CC(=O)Nc3ncc(Br)cc3F)C2)=O)CCCC2CCCCC12 c1(CNC(c2occ(C(=O)NC(COC)C(C)C)n2)=O)cnc2n1CCC2 c1(C(=O)NC(CNC(C(CCSC)OC)=O)C2CC2)coc2c1NC(=O)CCC2 n1(CC(=O)NCC2(F)CN(C(C3CCC3(F)F)=O)C2)cc(Br)ccc1=O N1(Cc2cc(C)no2)CCC2(NC(=O)CCc3ccncn3)CCCC12 c1(OC)ccc(C(N2CCC(CN(C(=O)C(C)NS(C)(=O)=O)C)C2)=O)c(F)c1F N1(C(C(c2ccc(C)o2)C)=O)CCC(CNC=O)C(C)C1.O(C(F)(F)F)CCN N1(C(C2C3(CCN(C(CCOC(C)C)=O)C3)C2)=O)CC2(CCCCC2)C1 c1(NCC2(OCC)CCC2)ccc(S(=O)(=O)N2CCN(S(C)(=O)=O)CC2)cc1Br c1(CC)ccc(C(C)N(CC(O)COCc2ccc(Br)cc2)C)cc1 N1(C(c2cccn(C3CCC3)c2=O)=O)CCN(C(C2CC=CCO2)=O)C(C2CC2)C1 c1(COC)ccc(C(=O)N(C)CC2CC(F)CN2C(c2csc(CO)c2)=O)cc1 c1(C(N2CC(NC(CSc3c(C)ncs3)=O)C2)=O)cn(C)c(=O)cn1 Cc1cc(C#N)ccc1C(c1nnnn1C1CC1)NCc1ccc(F)s1 C=CCCCCCC(=O)NCC1CCN(C(c2ccc3nc[nH]c3c2)=O)CC1 C1(CC)(NC(=O)C(C)S(N)(=O)=O)CCN(C(=O)C(n2cc(Cl)cn2)C)CC1 CC(C)(C)CC(=O)NC1CCCCC1NC(=O)CCC(=O)c1cccnc1 c1(NC(C(C2CCCO2)NC(c2c(OC)scc2)=O)=O)ccc(F)cc1O c1(NCC(F)(F)F)cccc(-c2cn(CCCCC(=O)OC)nn2)c1.O=C1CN1 c1(C(=O)NCC2C(NC(CCOC(C)C)=O)CC2)nc(C(C)(F)F)cs1 C(CCC(O)CO)N(C)C(C1CC(CCNC(=O)Cc2cccs2)C1)=O Cc1cncc(C(N2CCCCC2C2CCCN(C(c3nc(C)cs3)C)C2)=O)c1 C(C)(CCCC(=O)N(C)Cc1nnnn1C)NC(C=C(CCC)CCC)=O C1(NC(C2C(CC)CCC2)=O)CN(C(=O)Cc2ccc(C#N)cn2)CCC1CO c1(C(=O)NC(COC)CC(=O)NCCC(C)CCO)ccc(C)cc1C C12(NC(C3(C(=O)OC)CC3)=O)CC1CN(C(c1occc1Cl)=O)C2 n1(CC=C)c(N2CCN(c3ccc(OC)cc3)CC2)nnc1-c1ccc(O)cc1 C(C(CC(=O)NCC12CC1CNC2=O)c1ccc(Cl)cc1)N(C)C c1(C(C)N(C)C(C2CCCN2C(c2cc(-c3cccs3)[nH]n2)=O)=O)cnnn1C CC1CCc2nc(C(N3CCCCC(CNC(c4ccncn4)=O)C3)=O)cn2C1 Cc1nn(C)c(C)c1OCC(=O)NCC(O)CN(C(=O)CC1OCCO1)C N1(C(C(CC#C)(C)NC(=O)C=C(C)C(C)C)=O)CC(C)c2ncccc21 C1(O)(C(=O)NCC2(CCC)CCC2)CCN(C(C)(C)CSC)CC1 Cc1ccc(CCC(=O)N(C(C)Cn2cc(COC3(C)CCC3)nn2)C2CC2)s1 C1(NC(c2cccc[n+]2[O-])=O)C=CCN(C(c2ccc(OC(F)(F)F)cn2)=O)C1 c1(C(=O)NCC(CC=C)NC(=O)CC(C)(C)COC)cc(C)ccc1Cl C1(NC(C2CN(C(C)C(=O)C3CCC3)C2)=O)CCCC(F)(F)C1 Cc1cccc(-c2nsc(N3CC(C4CCN(C)CC4)CC3C)n2)c1 C1(NC(CC(CC)(F)F)=O)CC2CCC(C1)N2C(C1CC(C)OC(C)C1)=O c1(OC)cc(C(=O)NCC2CC3CCC2N3c2cc(C)nc(Cl)n2)ccc1C#N C(CCCC(=O)NC(C)(CNC(=O)C(C)C(F)F)CO)OC N1(C(CCN(C(=O)CCC2CC2(F)F)C(C)C)=O)CCOCC(C2CC2)C1 C1(CC(=O)NCC(CC(=O)N2CC(SCC)C2)C)CC2(CCO1)CC2 N1(C(C2(C)N(C)CCC2)=O)CCCC2CN(C(=O)C=C3CCCC3)CCC12 C(=O)(CCCCCC(C)O)NC(CNC(c1ccc(C#C)cc1F)=O)(CC)CC c1(CC(=O)NC(CN(C(c2c[nH]nc2OC2CC2)=O)CC)C)nnc(S)n1C C(CCCCCNC(c1n[nH]c(C)c1C)=O)NC(CCN(C(CCC)C)C)=O N1(Cc2nnc(CC)o2)CCCC(CO)(NC(c2ccn(C(C)C)n2)=O)C1 c1(C(N(C2CCN(C(=O)CC3(COC)CC3)C2)CC)=O)ccncc1-n1cccn1 C1(CCOC)CN(C(=O)CC(Cl)Cl)CCN1C(=O)CCCOC(C)(C)C c1(OC)ccc(Cl)c(C(=O)NCC2CN(C(=O)C(c3cnn(C)c3)C)CC2C)n1 C(=O)(C(C)C(F)(F)C(F)F)NC(C(=O)NCC(CC=C)CC(C)C)C(C)OC c1(OC)cc(OC)c(C(=O)NC2CC(N(C)C(c3ccc(O)nc3)=O)C2)c(F)c1 c1(-c2ccc(NC(C(CCCC)O)=O)cn2)cc2ccccn2n1 N1(C(CN(CCC)C)=O)CC(N(C)C(c2cc(Cl)nnc2O)=O)C2(CC2)C1 CC(O)(C(=O)NCCn1cc(C(N2C3CSCC2C3)=O)nn1)C(F)(F)F c1(OC)ccc2cccc(NC(N3CCC(NCC(F)(F)F)OCC3C)=O)c2c1 c1(CC(N2CC(C=C)(CC(=O)NC3CCC4(CC4)C3)C2)=O)cccc(C#N)c1C n1(C(N2CC(NC(C34CC3CCC4(F)F)=O)(CO)C2)=O)nc2ccccn2c1=O c1(N(C(C(=O)NC2CCCOC2)C2CCOC2)C)cn(C(C2CC2)C2CC2)nn1 C(=O)(CCN(C(=O)CNC=O)C1CC1)N(CC(C)OC)C C1(NC(COC(CNC(COCCSC)=O)(C)C)=O)CCOCC1C C1(NC(Cc2nc(C)sc2)=O)CC2CC1CN2C(c1c[nH]nc1C(C)C)=O c1(C(=O)NCC2C(C)(C)CCN2C(=O)C=Cc2nccs2)ccn2cccc2c1 CC1CC(CNC(c2ccnn2CC(F)F)=O)CN1C(C1C2CCCC12)=O C1(NC(C(C)OC2COC2)=O)C2CN(C(c3cc(=O)cc[nH]3)=O)CC12 C1(C(=O)NCC(CNC(c2scc(COC)c2)=O)(C)C)CCn2ncnc2C1 C(C)(CC(=O)N(C1(C(=O)NC(C)C(=O)N(C)C)CCC1)C1CC1)NC(C)=O CCCCCC(O)C(=O)NC(C)C(=O)N1CCC1CF.C(c1cscn1)=CC=O c1(C(N(C)CC2CN(C(c3ncccc3CO)=O)C2)=O)cnc2[nH]c(O)nc2c1 c1(C(=O)NC2C(CNC(c3ccc(C)n3C)=O)CCCC2)cn2c(n1)CCCC2 C1(N(CCCC)C(C2CC2C)=O)CCN(C(C2CCCN2C)=O)CC1 Cc1cn2cc(CNC(c3cn(CC(F)(F)F)nc3CC3CC3)=O)nc2s1 C12(NC(C3CCC(=C4CCC4)CC3)=O)CCN(C(c3ccc(O)nc3)=O)CC1C2 Cc1cc(C(=O)NC(C)C(CO)NC(C2CC2C(N)=O)=O)cc(S(N)(=O)=O)c1C N1(C(Cn2ccc(=O)n(C)c2=O)=O)CCC2CN(C(=O)CC3CCC3)C2C1 c1(C2C(C(=O)NCCCNC(CCCC(=O)NCC)=O)C2)cccc(C#N)c1 N1(C(c2c(OC)c[nH]n2)=O)CCC(NC(c2cc(Cl)cc(Cl)c2)=O)CC1C Cc1ccc(C(=O)NCCCC(c2ccco2)NC(=O)C(C)OCCN(C)C)c(O)c1 c1(CC)cc(C(=O)N(CC(C)NC(=O)CNC(=O)OC)C)cc(N)c1 Cc1cc(C(=O)NCC(C(C)C)NC(=O)CCc2c(C)noc2C)ncc1CO c1(C(c2n(CCSC)nnn2)NCc2ccn(C(C)C)n2)ccc(Br)c(Cl)c1 CC1CS(=O)CCN1C(C1CC2CCC1N2C(c1ncccc1Cl)=O)=O C1(C)(CC(=O)N(C2CCCC2)CC=C)CCN(C(=O)CCc2cccs2)C1 C1(C(=O)NC2(C)CC(NC(=O)Cc3cnc[nH]3)C2)COCCN1C=O C(=O)(C(O)C(F)(F)F)N1CCC(C)(CCNC(c2cc(OC)ns2)=O)C1 C1(C(N2C3CC(CC(NC(c4coc(Cl)c4)=O)C3)C2)=O)CCCCC12OCCO2 Cn1ncc2cc(C(N3CCC(CCOc4ncnc(Cl)c4OC)C3)=O)sc12 N#Cc1ncccc1-c1cn(CC2CCCN2C(c2ncccc2C2CC2)=O)nn1 c1(C2(C)CNC2)cn(CCCNC(=O)CSc2ncc[nH]2)nn1 N1(CC(=O)NCc2scc(C(C)=O)c2)CCC(F)CC1.C12CCN1C2=O n1(CC(=O)NC(C)(C)CNC(c2cccc(F)c2O)=O)cc(S(C)(=O)=O)cn1 C(=O)(C#CC1CCCCC1)NC1(COC)CCCN(C(c2ncc[nH]c2=O)=O)C1 C1(C(CNC(CCSCC(C)C)=O)O)CCN(C(c2cncn2C)=O)CC1 N1(C(C(CCC=C)(C)C)=O)CC(CNC(=O)CC(C)SC)OC2(CCC2)C1 CCC(O)(CC)CCNC(C1(C)CCCN(C(c2c(C)ncn2OC)=O)C1)=O N1(C(c2sc(C)c(O)n2)=O)CCC(NC(=O)Cc2cccnc2Cl)C(C)C1 c1(CN2CC(NC(c3sccc3F)=O)C(O)C2)cnc2ccccc2c1 c1(C(=O)NC(C(=O)NCC(C)OCC=C)Cn2cncn2)cc[nH]c(=NC)c1 N1(C(c2ccc(SC)cc2)=O)CCC(NC(C2CCN(C)C(=O)C2)=O)C12CCC2 N1(C(=O)CCC2CCOC2)CCC2C(C(N3CCCC4(C3)N=N4)=O)C2C1 CCC(C)CC(C(=O)O)NCC(=O)NC(c1ccccc1)Cc1ccccc1OC c1(C(N(CC(C)N(C(=O)C(F)C(F)(F)F)C)C)=O)cccc(F)c1F C(=O)(C1=COCCO1)NC(C1CCN(C(C2(COCC)CCOCC2)=O)CC1)C C1(C(C)NC(CSCC)=O)CCCN(C(c2cnn(CCO)c2CC)=O)C1 O=S(=O)(c1cc(Br)c(Cl)s1)N1CCC(Nc2cccc(Cl)c2)CC1 n1(CC)c(=NC(=O)NNS(=O)(=O)c2ccc(Cl)cc2)n(CC#N)c2ccccc12 c1(C(N2CCN(C(C=C(C)C)=O)C(C)C2)=O)cc2ccccc2cc1O N1(C(=O)OCC(C)(C)C)CC2CC1(c1ccccc1)C(=O)N2C1CCCC1=O N1(C(CN(C(C)C)C)=O)CCC(N=[N+]=[N-])(C(N2CCC(CN(C)C)CC2)=O)C1 C(=O)(CC1=CCOCC1)NCC1C(CNC(C2CCCC(C)C2)=O)C1(F)F c1(NC(C2C(C(=O)NC(Cc3ccc(C)cc3)CO)C2)=O)nc2ccccc2s1 C1(CNC(=O)CCCc2cc[nH]n2)COCCN(C(c2cnco2)=O)C1 CCC(C)CC(=O)NCC1(NC(=O)CCc2ccc(SC)cc2)CCOC1 N1(C(C(CCC)(C)C)=O)CC2CCCC(NC(C3CCSC3)=O)(C2)C1 C1(N(C(=O)CCCc2ncco2)CC)CCCN(C(C2(F)CC=CC2)=O)C1 c1(SC)ncc(N)c(C(=O)NCCC2CCC(C)CO2)n1 C(CCN=C(NCCF)N1CCc2cc(C(C)C)ccc21)N1C(C)CCCC1 C(C)(CCCCC#N)(c1nnnn1CCc1ccccc1)NC(CCC)CSC N1(C(CC(CC)C)=O)CCC2(CC2C(N2CC3CC3C2C#N)=O)C1 c1(CC(=O)NC2CCC(NC(c3ccns3)=O)C2)ccc(F)c(Br)c1 c1(C(N(C(CCC2N(C)CCC2)=O)C2C3CNC23)=O)c(F)cccc1[N+](=O)[O-] c1(C(N(CC(C)(C)NC(C)C(=O)NC(C)(C)C)C)=O)cc(C2CC2)ns1 N1(C(c2c(CCC)onc2C)=O)CCC2(CC1)CNCC2CO c1(C(=O)NCCCCCn2cc(C(C)(C)OCC)nn2)cc2ccccc2nn1 c1(OC)cscc1CC(=O)NC1(C(=O)NCC(C)(C)NC(c2ccon2)=O)CC1 C1(CC(=O)N(C)CCNC(CCOCC#C)=O)CCCCO1 N1(C(CC(CC=C)c2ccccc2)=O)CC(CNC(=O)CCC)C(C2CC2)C1 c1(C(N2CCC(NC(C(COC)C)=O)CC2C)=O)cccc(C#CC2CC2)c1 CC(CCCNC(=O)CCc1ccccc1)NC(C1CCN1C1CCCC1)=O c1(C(N2CCC(C)C(NC(c3ncccc3F)=O)C2)=O)ccc(Cl)c(C#N)n1 CC(C)CC(F)(F)C(=O)NC1CCCC(NC(c2ccc(F)c(F)c2)=O)CC1 c1(CNC(C2CC(NC(COCCOCC)=O)C2)=O)ccnnc1 CC(C)CS(=O)(=O)CC(=O)N1CCN(C(=O)CC2OCCC2C)C(C(F)(F)F)C1 C1(C(N2CCCC(CCCC)C2)=O)COC2(C1)CN(C(c1c[nH]c(=O)cn1)=O)C2 C1(NC(=O)COc2ccccc2C)CN(CCN(C(C(C)(C)OC)=O)C)CCO1 N1(C(CCOCCOCC)=O)CC(O)C(O)C1CNC(c1cnsc1CC)=O c1(CC(=O)NC(CNC(C=CC)=O)CCOC)cc(Cl)c2c(c1)OCCCO2 c1(C(=O)NCCN(CCC)C(C2CNC(=O)C2)=O)n[nH]c2ccc(OC)nc12 C(=O)(CC(C)(CN(C)C)C(F)(F)F)NCC1C2N(C(C=COCC)=O)C(CC2)C1 N1(C(C2(C=C)CCN(C(c3ccc(SC)o3)=O)CC2)=O)CCCC2(CC(O)C2)C1 C1(C(N2CC(CC=C)(C(=O)NCCCCN=[N+]=[N-])C2)=O)CCn2nnnc2C1 c1(C(=O)NCCCCCCNC(CS(CC)=O)=O)cc2ccccc2c(O)n1 C(=O)(C(C)CC(C)(C)C)N1CC(C(C)C)C(C(=O)NCC2CCCC23CCC3)C1 C1(C(N2CC(C(C(=O)N(c3cnn(C)c3)CC3CC3)OC)C2)=O)CC2(CCO1)CC2 C1(C)(C(N2CC(CNC(c3cc(CC)[nH]n3)=O)C(C)C2)=O)CCC(O)CC1 C1(C(N(C(C(C)C)C(=O)N2CCNC(=O)C2)CC(=O)O)=O)CN2CCCN1CC2 c1(COC)ccc(CNC(C2CC(NC(C3CCCN3C(C)=O)=O)C2)=O)cc1 CC(C)C(C)C(=O)NCC1CCCC1CNC(=O)CCNC(c1cccs1)=O N12CC(OC)C(C1)C2=O.C(=O)(CS(C)(=O)=O)NC1N(CCC)CCC1 C1(NC(C2(C)C=CCC2)=O)CCCC2CN(C(c3ncsc3Br)=O)CC12 C#Cc1cccc(C(c2nnnn2C2(C)CC2)NCc2nn(C)cc2C)c1 C12(CNC(C3CCN(C(C)=O)C34CC4)=O)COCCN1C(=O)OC2 Cc1cnc2[nH]cc(C(N3CCCCC3CC(=O)Nc3cccc(Cl)n3)=O)c2c1 C(=O)(C(C)(C)S(C)(=O)=O)N1CC2C(N(C(CSCc3nc(C)sc3)=O)C)C2C1 C(c1ccc(-c2ccc(Cl)s2)nc1)=CC#N CC(CO)N(C)NC(=O)C1(C)NC(=O)OC1C N1(C(C2(CC)CC2)=O)CCCN(CCCCNC(=O)CC2(C)CC(F)(F)C2)CC1 c1(CNC2CN(C)C(=O)C2)cnc2ccccn2c1=O CON1CCC(CC(N2CC(N(C)C(c3nc(O)c(C)s3)=O)C(O)C2)=O)CC1 C(=O)(CC(=O)NCC1CC(NC(=O)CCC2CC2CC2CC2)C1)OC CCCCCCC(F)C(=O)N(C)CC1(CNC(c2ccc(CC)o2)=O)CC1 c1(C(N2CC(CNC(C(CC)O)=O)(COC)C2)=O)nnn(C)c1C(F)F c1(CCC)ncoc1C(N1CC(O)(CNC(c2ccn(CC3CCC3)c2)=O)C1)=O N1(C(COCC#C)=O)CC(N(C(=O)C=Cc2ccc(CC)o2)C)C(C)(C)C1 C(=O)(C1CCCc2cccnc21)NCCCC(C)NC(c1c(CC)oc(C)c1)=O CC1=NOC(CC(=O)N(C)CCOCCC(=O)NCC(c2ccncc2)O)C1 N1(C(c2ccc(OC)cc2N)=O)CCCN(C(C2C(C)C2C)=O)CC1C N1(C(C(C)S)=O)CC2CCN(C(c3c(Cl)ccc(Br)c3F)=O)C2C1 N1(C(C(N2CCCCCC2)C)=O)CCCC(CN(C)C(c2nnn(C)c2N)=O)C1 Cc1cc(C)c(CC(=O)N(C2CCN(C(=O)Cc3cccs3)CC2)CC2CC2)s1 N1(CC)CCC(C(=O)NC2CC(CCNC(C3(F)CC3(Cl)Cl)=O)C2)C1 C(=O)(CCCCC(C)(C)C)N1CC(NC(COC(CC)(C)C)=O)N(C)CC1 C1(N(C)C(C2CC3(C2)CC32CC2)=O)CC2CCC(C1)N2C(C1C2(CC2)C12CC2)=O C1(NC(C2(OC)CCOC2)=O)CN(C(=O)C2=C(C)CCC2)CC(C)(C)C1 CCCC(C)(C)CC(=O)NC1CC(=O)N(C2CN(N3CC4CC3C4C=O)C2)C1.OC C(=O)(C(C)C(F)(F)C(F)F)NC1C2(CN(C(c3n(CCCC)ncc3)=O)C2)CC1 Cc1ccc(C(C)CC(=O)N(CCC(C(C)C)NC(c2csnc2C)=O)C)cc1 N1(C(c2cnc(CC)[nH]2)=O)CC(NC(c2c(Cl)n[nH]c2C)=O)C(C)C1 C=CCCC(F)(F)C(=O)NCC(O)CCNC(=O)CCc1cc(Cl)no1 CC1(C)CC(NC(c2cnc(CC(F)(F)F)s2)=O)CN1C(=O)CCSCC(N)=O c1(C(N2CC(C)(CNC(CSC)=O)OCC2)=O)cnc2snc(C)c2c1 N1(C(CC(C=C)(C)C)=O)CCC(CCNC(=O)C=CCN(CC)CC)C1 C1(N(C)C)(C(N2CCCC2CNC(=O)CCCc2cncs2)=O)CCCSC1 Cc1ccc(O)c(C(N2CC=CC(C(=O)NC3CN(C)CCC3O)C2)=O)c1 C1(CC=C)(C(=O)NCCC2(NC(=O)C(O)Cc3cnc[nH]3)CCC2)CCOCC1 N1(C(c2n(C=C)ncc2)=O)CCN(C(=O)CCc2cnc(C)s2)C2CCCCC12 C1(C)(C(=O)NCCC2CCN(C)C2)CN(C(C2CN3CCN2CC3)=O)C(C)(C)C1 C(=O)(C(CC(C)(C)C)NC(c1cc(C)c(O)nn1)=O)NC(CN(CCC)CC)C C(=O)(CCN(OC)C(=O)C1CC2(CCN1C(=O)CC(C(C)C)C(C)C)CC2)OC C1(C(N(C)Cc2cnco2)=O)CCN(C(c2sccc2C(C)(C)C)=O)CC1 C1(CC=C)(NC(c2[nH]ccc2CNC(C2C(C(C)=O)C2(F)F)=O)=O)CCCC1 C1(NC(c2cc(C)c(C)s2)=O)CC2CC(NC(c3ccoc3C)=O)C1C2 S(=O)(=O)(c1cn[nH]c1)N1C(C)CCC1C(=O)Nc1cccc(C(N)=O)c1 C(C(C)NC(c1cnc(C)n1C(F)F)=O)(C(C)C)NC(COCCCC)=O C1(NC(C2(C)C(CC)CCC2)=O)COC2(C1)CN(C(C1CC3C=CC1C3)=O)C2 c1(CNS(=O)(=O)CCc2ccncc2)cc(=NC2CCC2)[nH]c(Cl)n1 N1(C(C(C)(C)C#N)=O)CCC2CCC(C1)N2C(=O)Cc1c[nH]c2cnc(Cl)cc12 c1(CCC(=O)NCCN(C(=O)Cn2cc(C#N)cn2)C)c(F)cccc1F CCCCC(C(=O)Nc1cn(CCF)nc1C)NC(c1cc[n+]([O-])cc1)=O c1(C(=O)NC2CCC(C)N(C(C3CC3C(N)=O)=O)C2)c(Cl)ccc(F)c1N c1(C(=O)NC(CN(C)C)C(=O)NCCCC2CCOC2)ccccc1O C1(CC)(NC(c2nccn2C)=O)CCCN(C(C2CC(=C(F)F)C2)=O)C1 N1(C(CC(C)n2ccnc2)=O)CC=CCC1C(=O)NCCc1cccc(F)c1 c1(C(=O)NC2C(F)CCN(C(CC(=O)OC)=O)C2)cccc2cc(Cl)ccc12 c1(CN2CCC(C(N(C(CC)C(=O)OC)C)=O)C2)ccc2ccn(C)c2c1 C(=O)(CCC(CF)CF)NCCCN(C(=O)CC1COCC(C)O1)C(C)C O=S(=O)(c1ccc(Br)cc1Nc1ncccc1F)N1CCC(C2CCOC2)C1 C1(C(N2CCCC(C)C2)=O)CCN(C(C2CC23CCCCC3)=O)C12CC2 c1(-n2cc(Sc3ccc(NC(=O)CCC4CC4)cn3)nn2)ccc(Cl)c(F)c1F c1(C(N2CCC(F)(CNC(c3coc(C4CC4)n3)=O)C2)=O)cnc2[nH]cnc2c1 c1(-n2cc(C(CC)(O)CC)nn2)cc(C(N2CC(COC)C2)=O)ccc1C C=CCC(C(=O)N1CCCC1C(=O)NCCC1CCCC12CC2)NC(C)=O c1(OC)c(Br)cc(C(N2CC3CN(C(c4csc(C)n4)=O)C3C2)=O)cc1Br N1(C(c2cc(Br)co2)C(=O)OCCNCC)CC2CCCC2(C(=O)OC)C1 CC1C(NC(=O)COCCO)C(C)CCN1C(=O)CCc1ccn(C)c1 c1(NC(C(C2CN(C(=O)C(F)CCC(C)C)C2)OC)=O)ccc(C)c(O)c1C c1(CC)ccc(C)nc1NC(C1C=CCN1Cc1nc(-c2ccccc2)cs1)=O C12(NC(c3cccc(F)c3F)=O)CCCCC1N(C(=O)N(C)C)CC2 Cc1ncc(C#N)cc1NC(C1CCN1C(C1(C#N)CC12CCC2)=O)=O N1(C(c2c(C)noc2C(C)C)=O)CC2CCC(NC(=O)CC3CCOC3)CC2C1 N1(C(C2(CC)CCOC2)=O)CC(N(C(=O)CSCCC#N)C)C2(CC2)C1 C1(Cn2cc(C3N(C(C#CC(C)(C)O)=O)C4CCC3C4)nn2)CCCCCCC1O N1(C(c2scc(OC)c2)=O)CCOC2CN(C(c3c[nH]nc3C3CC3)=O)CC12 C(=O)(CC(C1CC1)NC(=O)C(C)(O)c1cccnc1)NC c1(N(C)CC2(C3CCCO3)CC2)ccc(S(=O)(=O)Nc2ncccn2)c(Br)c1 C1(C(=O)NCC(C2CCCC2)OC)C2CC3C(C2NC(C2(C)COCCO2)=O)C13 C(C(=O)Nc1ccc(S(C)(=O)=O)s1)(C(C)C)(C(C)C)NC(=O)OC N1(C(c2c(C)oc(C#N)c2)=O)CCC2(CC1)CN(C(c1ccccc1CO)=O)C2 C1(NC(C(C=C=C)C)=O)CCN(C(=O)CSC(C)(C)C)C12CCC2 C1(NC(Cc2cn(CC)nc2)=O)CCCCC1CNC(=O)C(CO)OC C1(C(=O)NCC=C)CCC(C(=O)NC(CC(N)=O)C2CC2)C1C Cc1c(-c2ccccc2)nn(C)c1C(=O)NCC(C)NC(=O)COC1CC1 C1(NC(=O)Nc2ccc(CC)[nH]2)CCCCCC1C(=O)NCn1cc(CC)nn1 N1(CC)CCOC(C(=O)NCC2(F)CC(CNC(=O)CSC)C2)C1 c1(C(=O)Nc2cc(O)ncn2)ccc(S(=O)(=O)N2CCCCC2)cc1 Cc1oc(=NC(=O)C2(NC(=O)C(C)N3CCCC3)CCC2)[nH]c1C N1(C(C2C(=C)C2)=O)CC2(CNC(C3CCN(CC(F)(F)F)C3)=O)CC1(COC)C2 CC1(C)CCC(CC(N2CCCC2C(C)(C)NC(=O)C2CC2)=O)OC1 C(CCCC(=O)N1CC(OCC(=O)NC2COCCC2C)C1)SC c1(C(=O)NCC2CN(C(C3(C)CCC(C)CC3)=O)C2)cc2n(n1)CCNS2(=O)=O N1(C(C(CCOCC)NC(CCCC)=O)=O)CC(O)(C2CCC2)C1 Cc1ccc2c(c1)C(=O)NC1C(C1)NC2=O.C(=O)(C(O)C(F)F)NC1CC1 c1(C(N2CCCC2c2cccs2)C(=O)NC)ccccc1Br N1(C(COC(C)=O)=O)CC2CC(NC(c3cnc(C(F)F)nc3)=O)CC1C2 C(C1CC(=O)NC2(CCOCC2)C(=O)N1)OC.c1(CCCSC)ncco1 C1(NC(COC(C)(C)C)=O)CCCC1C(=O)Nc1ccnn1C1CC1 N=c1[nH]c(CCC(=O)NC2CC(NC(c3sccc3-n3ccnn3)=O)C2)cs1 N1(C(c2c(C#N)scc2)=O)CC(C2(NC(=O)Cc3cncs3)CC2)C1 CCC(C)(O)C(=O)N1CCCCC1CNC(=O)Cc1cnsc1 C(CC1CCc2ccccc21)Nc1n(-c2ccccc2)cnn1 N1(C(C2(NC(=O)C(C(C)C)NC(N)=O)CCCC2)=O)CCC(O)(COCC)C1 N1(C(C(CC)C2CCC2)=O)CC2(CC(C(=O)NCCCN3CCC3)CO2)C1 C1(C(N(C2COC(C3CC3)C2)C)=O)(NC(c2csc(C#N)c2)=O)CCCCC1 C#CCC(C(=O)NC(C)C(C)(C)N(C)C)NC(=O)C=C(C)C1CC1 C1(NC(=O)Nc2ccc(N3CCOCC3)nc2)CCc2nn[nH]c2C1 c1(CC(=O)NC(CCNC(C(CC)(C)F)=O)C)ccc(Cl)cc1F c1(C2C(C(N(CCCCN(CCC=C)C)C)=O)CC2)ccc(Br)cc1 O(C1CCCc2ccccc21)CC(=O)NC1CCC(NC(C(C)=C(CC)C)=O)C1 N#Cc1cc(C(=O)NC2CCC(C#N)C2)cnc1C(F)(F)F c1(C(C(=O)NC(C2CCN(C(c3c[nH]nc3C(C)(C)C)=O)C2)C)O)cccnc1 c1(C(N(CC(CC)NC(c2cnn(C)c2C(F)F)=O)C)=O)ccn2nnnc2c1 CCC(C)CCC(=O)NCC(C)CNC(=O)COc1ccccc1C N1(C(CCNC(CC(C)C)=O)=O)CCN(C(=O)C(C)(C)C(N)=O)CC(C)(C)C1 N1(C(C(C2(O)CN(C(CC(=O)NCC(F)(F)F)=O)C2)F)=O)CCCCC(CO)C1 N1(C(c2c(C(C)C)c[nH]n2)=O)CC(CNC(C2C3CNC(=O)C23)=O)C(C)(C)C1 C#CCC(C)C(=O)N(CC(CC)NC(=O)CNC(c1ccccc1F)=O)C C(=O)(C(F)(F)C(O)C(C)C)NC(CCNC(C1(CCOCC)CCC1)=O)(C)C C1(C(CNC(c2cc(OC)ns2)=O)(C)O)CCN(C(C2CCC(=O)O2)=O)CC1 c1(C(=O)NC2CCN(C(CCCC)=O)C(C)C2)cc(O)cc(C#N)c1 C(=O)(C(CC(=C)C)OC)N1CC(CC=C)(C(=O)NCC=C(C)C(C)(C)C)C1 n1(CCCC)ncc(C(=O)NC2CC(O)(CNC(C3CC=CCC3)=O)C2)c1C C1(CNC(COCCCC)=O)CN(C(=O)C(C)CC(F)F)CCC1(C)C C1(NC(c2onc(C)c2C)=O)CN(C(=O)COCc2nccn2C)CC2(CC2)C1 c1(C(=O)NCCOCCCF)ncccc1Cl C(=O)(C(F)C(C)(F)F)NC(CC=CC)C(=O)N1CCCCC1CC(N)=O C(=O)(CCC(F)(F)F)N1CCC(C)(CNC(C2C(=C)C2C(=O)OC)=O)C1 c1(COC)nc(CC(=O)N(C)CC2CCN(C(c3cc(C4CC4)on3)=O)C2)cs1 C(CC(C(=O)NC1CC(=O)N(C)C1)NC(C1CN(C(N)=O)C1)=O)OC c1(C(=O)NC2CN(C(=O)NC3CC3c3ccccc3)C2)c(Cl)cccc1I N1(C(CCN(C)CCO)=O)CC=C(c2cccc(Br)c2)C1 C12(CNC(C3CCC(OC)CC3)=O)CC(C1)C(NC(=O)COC(F)(F)F)CO2 c1(CC(=O)NC2C3CN(C(C4(C)CCN(C)C4)=O)C2C3)cccc(F)c1F CCC(C)(C)CCNC(=O)C(n1cc(-c2cnn(C(C)(C)C)c2)nn1)C c1(CCC(N2CC(COC)(NC(c3cc(Cl)n(C)n3)=O)C2)=O)cnc(C)nc1O C1(NC(C(C)C(C)O)=O)C(C)(C)CN(C(=O)CCC(N)=O)CC1(C)C CC1CCC(c2nnnn2C2CCCCC2)(NCc2sccc2Cl)CS1 C1(C(=O)NCC(C)CC2CC2)COCC1NC(C1CCC1)=O CCCC(C#N)C(=O)N1CC(O)CC1CNC(=O)CCc1nnc(O)nc1O CCCCC(C)(F)C(=O)NCCC1(CNC(=O)Cc2cccc(C)c2F)CC1 C(=O)(C1=Cc2ccccc2C1)NC1(CO)CCN(C(Cc2ccc(C)o2)=O)CC1 N1(C(CC(COC)(C)O)=O)CCN(C(=O)CN2CC3CC3C2)CC(C)(C)C1 C1(F)(CNC(=O)CN(C)OC)CN(C(c2c(CCC)occ2)=O)CC1C(=O)OC N1(C(C2CCC(C(=O)O)C2)=O)CC(CN)CC12CCOCC2.C(C)(C)(C)OC C1(C(=O)NC(c2cn(CC)nc2)C)CN(C(=O)CC2COCCO2)C(C)(C)C1 c1(C(=O)NCC2CCC(NC(c3ncoc3CO)=O)CC2)cc2ccncc2[nH]1 Cc1c(C(=O)NCC2C=CCN2C(C2CCCC(=O)O2)=O)nn(C)c1Br c1(C(N(CCOC)CCNC(C2C=CC(C)(C)CC2)=O)=O)nccn2ccnc12 Cc1ccc(=N)[nH]c1C(N1CCC(N(C(=O)C(C(C)C)OCC(C)C)C)CC1)=O C1(C(N(C(C)CC(=O)NC2CC(C(F)(F)F)C2)C)=O)CSCC(=O)N1 C=CCCCC(C(=O)N1CCCC(N(C)C)C1)NC(c1ncc(F)cc1F)=O c1(COC)ccc(C(=O)NC(C2N(C(C3(N(C)C)CC3)=O)CCC2)C)o1 N1(C(C(C)NC(CC)=O)=O)CCC2C1CCN2C(=O)Cc1c(C)n[nH]c1C C1(NC(CCc2cc(C)no2)=O)CCN(C(=O)Cn2nccc2C)C12CCCC2 C12(C(N3CC(CC(=O)NCc4cc(CO)ccn4)OCC3)=O)CCC(CC1)CC2 C=C1CCC(C(=O)N(CC(CC)NC(c2ccccn2)=O)CC)CC1 c1(C(N2CCN(C(C#C)C)CC2)=O)cc2c(C)cccc2o1 C(=O)(CCC(C)(C)C#N)NC(C1CCN(C(C(CC)C2CCOCC2)=O)C1)C CCC(C)CC1C(=O)NC(CCOC)C(=O)N1.C(CCF)OC c1(OC)ccnc(C(=O)NCC2C(C)CCN2c2nccc(COC)n2)c1 C1(CNC(CCSCC)=O)CC(NC(C2CC=CC2)=O)CC1O N1(C(Cc2c(C)nccc2)=O)CCN(C(c2cc(N)ccn2)=O)C(C)C1C c1(CC(C(=O)NC2CC(NC(C3CCC(C)C3)=O)C2)=O)ccc(Cl)cc1 C1(C(C(=O)NC2(COC)CCC2)F)CCN(C(C2C=C(C)CS2)=O)C1 C(=O)(CS(=O)(=O)C1CCCC1)N1CC2N(C(C(CC(C)(C)C)(C)C)=O)C(CC2)C1 c1(CNC2CCC(C(=O)NCC3C(C)CCC3)C2)ccc(C#N)s1 Cc1nn(CC(N2CC(CNC(c3cnns3)=O)CC2C)=O)cc1Br c1(C(=O)NC2C(NC(c3c(C)cc(O)cc3)=O)C2)cc(O)c2nc(C)n(C)c2c1 C=Cn1nncc1C(=O)N(C(C)C(=O)Nc1csc(Cl)c1)C1CC1 C1(CNC(C2N(CC(C)C)CCC2)=O)CCCN(C(=O)Cc2cnoc2)C1 N1(C(CCN(C(=O)CO)CCO)=O)CC(NC(=O)C(F)(F)F)C(c2cn[nH]c2)C1 N1(C(CC=CC=C)=O)CCC(C(C)C(=O)NCCS(C)(=O)=O)CC1 C#Cc1cccc(C(c2nnnn2CCCOC)NC2CNC(=O)C2(C)C)c1F c1(CC(=O)NCC(CC)(C)NC(c2ccc(C(F)F)cc2)=O)ccc(Cl)nc1 c1(CC(=O)NCCCC(C)NC(CCC)=O)ccc(F)c(Cl)c1 CC(C)CCC(F)C(=O)N1CC(CNC(=O)C=Cc2cscn2)OC(C)(C)C1 c1(C(C2CC2)NC(=O)NCCOCC=C)cnn(C)c1 CC1OCCC1CNC(=O)Cn1cc(CNC(C2CC23CC3)=O)nn1 C(=O)(C(C)C(F)(F)F)NCC(c1cccc(C)c1)NC(=O)CCCCCF C1(C(=O)NC(c2c(C)cccn2)C2CC2)(C(c2ccccc2F)=O)CCCCCC1 C1(NC(C2CSCCN2C(=O)CCCC2CC2)=O)CC12CC(O)C2 C(CN=C(NCC1(Cc2ccnn2C)CCN(C)CC1)NC1CCC1)OC CCC(CN(C(=O)C(C)SC(F)(F)F)CC)NC(=O)CC1CC(OC(C)=O)C1 C=CC1OCCC1C(N1CCC1C(=O)N(CCCC(O)CO)C)=O CC1C(C(=O)NC2CC(C(=O)NCC3(N(C)C)CC3)C2)C(O)C(=O)N1C N1(C(CC(C)(C)O)=O)CCC2(COC(CNC(=O)C(C)(C)O)C2)C1 N1(C(CC(C(C)C)C)=O)CC(NC(c2ccc(C(F)F)cc2F)=O)CC(C)(C)C1 c1(CN(C(CNC(C(C)O)=O)C)C(c2ccoc2C(F)(F)F)=O)cccnc1 C1(OC)(CNC(=O)CN2CCCCC2)CCN(C(=O)Cc2cncn2C)CC1 N1(C(C2COCCN(C(C3OCCN(CC)C3)=O)C2)=O)CC2CCN(C)CC2C1 N1(C(C2CC(=C)C2)=O)CCC(NC(=O)C=C(C)C(F)(F)C(F)(F)F)CC1C1CC1 Cc1cc(C(=O)NCC2(O)CN(C(=O)Cc3ccon3)C2)cnc1O Cc1ccc(C(N2CC3CC3C2C(=O)NCCCn2ccnn2)=O)c(O)n1 c1(C(=O)NCC2(F)CC(NC(CCOCCOC)=O)C2)ccc(Cl)cc1C C(CC(=C)Cl)(C(=O)N1CCC1(C)CC)NC(C(C=C=C)C)=O C1(C(N(CCCOC)C)=O)CCCCN1C(=O)CC(C)NC(=O)C1CC1 C1(C(N2CCN(CCO)CC2)=O)CC2(CC2)CN1C(c1cc(Cl)ncc1Br)=O C1(SC)CCCC1C(N1CCCC1CCNC(c1cc(C(C)C)[nH]n1)=O)=O c1(N2CC(CCNC(=O)C(C)C3CCCO3)(OC)C2)[nH]c(=O)n(C)c(=O)c1C#N c1(CSc2cc[nH]c2C)cnccc1C(=O)N.c1(C(=O)OCC)ccc(C2CC2)o1 CC1(C(N2CCC(O)(CCNC(c3ccccc3F)=O)C2)=O)C#CCCC1 c1(C(=O)NC2C(NC(c3cnc(CC)s3)=O)CCC2)noc(C)c1[N+](=O)[O-] N1(C(C2CCC(=O)N2)=O)CC2CC(CNC(=O)CCc3cccc(O)n3)C2C1 c1(C(N2CC(CNC(c3c(CC)scc3)=O)C2)=O)ccc(Cl)c(F)c1N c1(C(C2CN(S(=O)(=O)CCC3CCC3)C2)N)ccccc1 CN1CCC(C(=O)N(CCCNC(=O)C(C)(C)C2CCC2)C2CC2)C1=O N1(C2CC2)CCCC(C)C1.C(C1C(=O)NCC2(CCC2)COCCC(=O)N1)OC C1(C(=O)NCc2c(CCNC(C3CCC(OC)C3)=O)ocn2)C(Cl)(Cl)C12CC2 C1(O)(CCNC(C(CCC)c2ccc(Cl)cc2)=O)CCCN(C(=O)C2=CCC2)C1 C1(C(=O)NCC(=O)NC)CCN(C(C2CN(C)CCO2)=O)CCO1 c1(NC2C(C)COCC2)nc(NC2CCCc3nc[nH]c32)nc2cccc(Br)c12 Cc1c[nH]c(CC(N)=O)c1C(=O)NC1(CNC(c2[nH]ncc2C#N)=O)CCOC1 N1(C(CC=CC=C)=O)Cc2ccccc2C(NC(=O)CN2CCC(F)(F)C2)C1 C(=O)(C1CCc2c[nH]nc21)Nn1cncn1.C1(CC)CN2CCC1C1(CC1)C2=O N1(C(C2(CNC(C(CC)C)=O)CC(C)(C)C2)=O)CC2(C)COCC2(C)C1 C1(NC(c2c(OCC)nc(C)cc2)=O)CCCCCCC1OCC(=O)NCC c1(C(N2CCN(C)CC2C2CCC2)=O)noc2ccc(C(F)(F)F)cc12 c1(CC)nccnc1NC(c1cc(NC(c2cc(C)nn2C)=O)cn1C)=O CCC1=C(C(=O)N(C2CC3CCC(C2)N3C(=O)Cc2nonc2C)C)SCCO1 C1(CC(=O)NCC(C)(C)OCC(=O)NCCN(CC=C)C)COC(=O)N1 N1(C(C2CCC(=O)N2)=O)CC(NC(c2cnc(C(F)(F)F)nc2)=O)CC(F)(F)C1 C1(NC(c2c(OC)nccc2)=O)CC2CCC1CN(C(=O)Cn1[nH]cnc1=N)C2 CC1OC2(C(N3CC(CNC(C4OCC5CCCC45)=O)C(C)C3)=O)CCC1CC2 CC(=O)CCCC(=O)N1CC2CC2C1C(=O)NCC(C)(C)CC(C)C c1(NC(COCC(=O)NC)=O)cccc(CC(=O)N(C2CNC(=O)C2)C)c1 CCC(CC)C(F)C(=O)N1CCCC(N(C(c2[nH]cnc2C)=O)CC2CC2)C1 N1(C(c2cnc(C)s2)=O)CCCC(CC(=O)NCCc2cnc(C)s2)CC1 c1(C(=O)NC2CN(C(C=C(C)C)=O)CC(C)(C)C2)cc(O)nc2c1c(C)nn2C Cn1ncc2c(NCCCF)[nH]c(=NCC3CCOCC34CCCCC4)nc12 N1(C(C(F)=CCC)=O)C(C(=O)N(C(C)CC(=O)NC)CC)CC1C c1(SCCCC(=O)NC2(CCNC(C(C)NC(N)=O)=O)CCC2)ccc(F)cc1 C=CC(CCC)CC(=O)NC1(C2CCCN2C(c2oc(C(F)F)cc2C)=O)CC1 C1(CNC(c2cncc(OC)c2)=O)CC12CCN(C(=O)C=CS(C)=O)CC2 C1(F)(CNC(CCOCCC)=O)CC2CCC(C1)N2C(C1CC1(C)CCOC)=O Cc1cccc(OCC(=O)NCC2CC3(CC3)CN2C(C2CCCSS2)=O)c1C C1(C(N2CCC(NC(C3CCC(C)(CC)O3)=O)(CF)C2)=O)CC12CC(C)(C)C2 Cc1cccc2cc(C(=O)NC3C4CCN(C(=O)C=CC5CC5)CCCC34)[nH]c12 C(=O)(C1CCc2nccn21)N1CCN(C(c2c(C)c(Br)cnc2)=O)CC1 c1(NC(c2cc(-c3ccccc3-c3cnc(CO)cn3)[nH]n2)=O)cc(O)cc(O)c1 C(=O)(CC(COC)COC)NCC1C(NC(c2ccn(CC)c2C)=O)CC1 n1(CC)ccnc1C(c1nnnn1C(C)(C)C)NCC1CC1.C1CC(=O)N1 c1(C(=O)NC2C(F)CCN(C(C(n3ncc(C)c3)C)=O)C2)cc2n(n1)CCCO2 c1(CCC)cc(C(=O)N(C)CC2CCN(C(C3CC(C)(C)CO3)=O)C2)ccn1 C1(NC(Cc2c(C)noc2C)=O)CS(=O)(=O)CC1NC(c1cn(C)cc1C)=O N1(C(C(C)CC(F)F)=O)CC2CN(C(=O)C(C)(C)C#N)CC(F)(F)C2C1 C1(CNC(c2cnc(C)o2)=O)CCC(C)(C)CN1C(=O)CN1CC=CC1 C1(C(=O)OC)(C(=O)NCC(C)N(C)C(C2CN(C)CC2C(F)(F)F)=O)CCCCC1 CC(C)CCC(O)C(=O)N1CCOCC1CN(C)C(c1ccccc1O)=O CC1(C(=O)NCC2CC2C(N2CC(n3cnnc3)C2)=O)CC2CC2C1 c1(CC(=O)NC(CCNC(C(C)(C2(C)CC2)OC)=O)C)c(C)noc1C n1(CC(C)C)c(N(C2CCC2c2cccs2)C)nnc1C1CC(=O)N(C)C1 C(CC(C)C)(C(=O)NC)N(CCCC)CCCC(=O)NCC(O)CCOC CC(CC(F)(F)F)C(=O)NC1CN(C(C2CC(=O)NC(=O)C2)=O)CC1C c1(NC(C2C(CNC(C(C(C)C)OC)=O)CC2)=O)cc(C)cc(Cl)c1 C1(NC(=O)CC2CCS(=O)(=O)C2)CN(C(C23CSC(C2)C3)=O)CC1C1CC1 c1(NC(Cn2cc(C(CC)(O)CC)nn2)=O)ccc2c(c1)CCO2 c1(C(C(=O)NCC(CNC(C2(c3c(C)ccs3)CC2)=O)C)O)cccc(F)c1 c1(C(=O)NC2CCC(CCNC(C(C)(F)F)=O)C2)nncc2ccccc12 c1(COC)csc(C(c2nnnn2C2COC2)NCC(C)(C)n2cccn2)c1 CC(C)(O)C(F)(F)CNC(=O)C(Cc1ccco1)NC(c1cc[n+]([O-])cc1)=O C1(C(C)C)CN(C(C2CC(F)C(=O)N2)=O)CCN1C(=O)COC1CC1 c1(C(=O)NC(CCN(C)C)C(=O)NC2(CO)CC(O)C2)ccc2nccn2c1 C1(C(=O)NC2CC(NC(c3ccc(C(F)(F)F)[nH]3)=O)C2)CC2CCCCCC12 c1(OC)nc(C(N2CCCC(NC(c3cnc(O)nc3O)=O)C2C)=O)cc(O)n1 c1(C(N2CCC(NC(C(CCC)C)=O)C(F)C2)=O)ccc(F)c(C#N)c1 c1(-c2cn(-c3ccc(C(F)(F)F)cc3)nn2)cccc2c1sc1ccccc21 C(CCCC(=O)N(C1CCN(C(c2cncnc2C(C)(C)C)=O)C1)C)SC c1(COC(C2CS(=O)(=O)CC2O)=O)cc2cc(Cl)ccc2nc1Cl N1(C(C(CC)OCC)=O)CC=C(CNC(c2c(Br)nnn2C)=O)CC1 N1(C(c2ncc(C)nc2)=O)CCN(c2ccccc2F)CC1C NC(=NCCCF)NCCC(C)(F)F.CCCO Cc1c(F)ccc(N)c1C(=O)NC1CN(C(=O)CC2CCCCC2O)CC1(C)C C1(CC(=O)NC(C(=O)NCC2CCN(CC)C2)Cc2ccoc2)CCCC12CC2 c1(C(=O)NC2(CC=C)CN(C(=O)COC3CCOC3)C2)ccc2sccc2c1 c1(NC)cncc(C(=O)NC(C)(C)CC(=O)Nc2cnn(C)c2C)c1 C1(C(=O)OCC)CCC2OCCC2N1C(=O)Cn1cc(Cl)c(-c2ccccc2)n1 C1(C(=O)NCC(=C2CCOCC2)F)CC12CCN(C(=O)C(F)C(F)(F)F)CC2 C(=O)(CCS(C)(=O)=O)NCC(C)C(=O)N1CCC1C(N)=O C(=O)(C(C)(F)C(F)(F)F)NC1C(C)CN(C(C2(c3ccco3)CC2)=O)C1 N1(C(CC#CC)C(=O)OCC)CC(=O)NCC1C(=O)OCC.C(C)(C)(C)O C(CN1C(=O)COc2ccccc21)NC(=O)C(=O)Nc1ccc(F)c(F)c1Br CCC(C)C(C(=O)NCC(=O)Nc1ccc(CC(C)C)nc1)N(C)C C(=O)(CS(C)(=O)=O)NCC1C(CNC(C(CC)Oc2ccccc2)=O)C1 c1(-c2cc(C)no2)ccc(S(=O)(=O)NCc2cnc3c(c2)COC3)s1 C(=O)(C(O)P(C)(C)=O)NC1CN(C(c2c(C)snc2)=O)CC1c1ccnn1C C(=O)(CC(C)(C)C)N(CCNC(CCSC)=O)CC1CCCCO1 C1(F)(CNC(C=C(C)Cl)=O)CCCN(C(=O)CN2CC3CCC2C3)C1 c1(CC(C(N2CCC(COC)CC2)=O)N)cc(C)cc(F)c1 C(C)(CC(C)CC)N(C(C1(N(C(COCCCC)=O)C)CCCC1)=O)C C(C)(C(C(=O)N1CCC(C)(C#N)C1)C(C)C)NC(CCCSC)=O c1(-c2ccn(C)n2)cn2c(n1)CCC(C(=O)Nc1cc(CO)ccc1C)C2 C1(C(=O)NCCN(CCC(=O)NCCCOCCOC)CC)CN(C)CC1C C1(N(C(c2c(C)con2)=O)C)CCCN(C(=O)C=Cc2cnc[nH]2)C1 c1(CCC)nnsc1C(=O)NC(C)(C)CN(C)C(c1ccc(SC)s1)=O c1(OC)cc(Cl)ccc1C(=O)NC(C)CCNC(=O)CCCOCCC(C)C c1(CN2C(C(=O)NCCCCC=C)CC(C)C2)cc(Br)c(N(C)C)cc1C c1(C(N(CCCNC(C(n2cnc(C#N)n2)C)=O)C)=O)cc(=O)cc(Cl)[nH]1 N1(C(c2cc(C(C)(C)C)on2)=O)CC2=C(C1)CN(Cc1ccc(Cl)c(F)c1)C2 C(=O)(C(O)C(C)(C)C)NCC(CC(C)C)NC(C1C(C)(C)C1(F)F)=O C(=O)(CC(C)NC(C1(C(=O)NCC2(C)CC2(F)F)CCC1)=O)OCC CC1CCC(OCC(=O)NC2(CNC(C3COC(=O)N3C)=O)CCCC2)CC1 N1(C(C(C2CC2)OC)=O)CCCN(C(c2ccc(Br)s2)=O)CC1C Cc1coc(C=CC(=O)NC2CN(C(=O)CCC(C)N(C)C)C2)n1 c1(CC=NC(=O)C(F)CC2CCC2)c(F)ccc(S(=O)(=O)CC2CC2)c1F C1(C(=O)NCC2(NC(=O)CCn3cc(C)cn3)CCCCC2)(OC)CS(=O)(=O)C1 c1(OCC)c(C)csc1C(=O)NCCC1CN(C(=O)C(C(=O)OC)OC)C1 c1(C(C(N2CC(O)(CNC(Cc3cc(CC)no3)=O)C2)=O)(F)F)ccc(F)cc1 CON(CCC(=O)NCC1CCOC1)C(=O)CC(C)(F)F CCCCC(O)C(=O)N1CC2CC1C2C(=O)Nc1cncc(Cl)c1 N1(C(c2cc(I)cn2C)C(=O)NC(C(=O)OC)C)CC(=O)NCC1C(N)=O N1(C(c2cc(C)c(F)cc2)=O)CCC2(NC(c3cscn3)=O)CCCC12 C1(C(=O)NC(C2CCCC2O)C)CN(C(=O)Cn2c(O)nnc2O)CCN1C C1(C(=O)NC2(CC(=O)NCC(C(C)C)C)CC2)CCOC(=O)CC1 C1(NC(COC)=O)CN(C(=O)C=C2CCC2)CC1OC c1(CC(N2CC3C(NC(=O)C(F)CC4CCC4)C3C2)=O)csc2ccccc12 c1(C(=O)NC2CN(C(C(CO)NC(C(C)C)=O)=O)C2)nn(C)c2ccccc2c1=O C=CC1(C(N2CC(N(C)C)C(CNC(C3CC(C)OC(C)C3)=O)C2)=O)CCOCC1 C1(O)(CCC)CCCN(N2CCN3C(C(=O)COC)CCS(=O)(=O)CC3C2)C1=O c1(C(C2CC2)NC(CN(CC(C)C)C(=O)CC2CCOC2)=O)ccncc1F CCCC(C)(C)C(=O)N1C2CCC(C2)C1CC(=O)N(CC(C)OC)C CC1OC2CCC1(NC(C1CC(NC(c3cccs3)=O)C1)=O)C2 CCCCC(CCCC)NC(=O)CC(CC1CC1)NC(=O)C=Cc1ccn(C)c1 CCC(C)(O)C(=O)N1CCCC(C(C)NC(=O)C(C)Cc2ccnn2C)C1 CC1CCC=C1C(=O)NCC1CCCCN1C(c1cnc(C(C)(C)C)o1)=O c1(CC(=O)CCOC(C2C(C3(C)CCC3)C2)=O)csc2nc(-c3ccco3)cn12 C(=O)(C1c2ccccc2-c2ccccc21)C(=O)NCc1ccnc(F)c1Cl Cc1cc(O)ncc1C(N1CCCCCC1CNC(=O)CCC1CCOC1)=O N12CC(C(=O)N(CC(C)N(C)C)C)(C1)C(=O)OC2=O.C1(SC)CC1(C)C(C)(F)F c1(C(=O)NCC2C(C)(C)C2C(=O)NC2CC23CCC3)ncnc(O)c1F C1(C2CCN(C(C3(Cl)CC3(F)F)=O)CC2)(NC(C2=C(C)S(=O)(=O)CC2)=O)CC1 c1(C(=O)NC2CCCCN(C(CS(C)(=O)=O)=O)C2)ccc2c(c1)CCC2=O CCC(C)C(O)C(C)C(=O)NCC1(F)CCN(C(c2cc[nH]c2C)=O)C1 C1(COC)(CNC(c2cscn2)=O)CCN(C(c2ccc(C(C)C)cc2)=O)CC1 n1(CC(N2C(CN(C(C(C)OCC)=O)C)CCC2)=O)ccc(Br)cc1=O N1(C(=O)OC(C)(C)C)CC(C2CC2)C(F)(c2nc(Cn3cccn3)no2)C1 Cc1ccc2cc(C(=O)N(C(CNC(=O)CN=S(C)(C)=O)C3CC3)C)cn2c1 N1(C(c2ccc(CNC(c3n(C)c(Cl)nc3)=O)nc2)=O)CCC2(CCC2)C1 c1(N(C(C(=O)NC(CC)(C)C)c2cc[nH]n2)CC(C)C)cc(F)cc(Cl)c1 C#CCCCCCC(=O)NCC(C(=O)NCCCC(C)(C)C=C)OC N1(C(=O)OC(C)(C)C)C(C(=O)NCCC(O)C(F)(F)F)CC2CCCCC12 c1(CNC(C(C)(C)NC(C2C(C)C2C)=O)=O)cncc(F)c1 Cc1cc(Cl)ccc1-n1ccc(C(N2CCC(NC(c3csc(O)n3)=O)C2)=O)n1 C1(OC)CN(C(c2ncc(C)o2)C(=O)NCCC2(C)CC2)C(C)(CO)C1 N1(C(c2c(C)nc[nH]2)=O)CCCC(N(C(=O)Cc2ccccc2F)C)CC1 n1(CCC(=O)NCCN(C(=O)C(C)C(C)(C)C)C(C)C)cnc2sccc2c1=O c12cc(Cl)c(c(Cl)c1)C(=O)N1CC(C1)NC2=O.c1(CNC(C)=O)cccc(F)c1 CON(C)CCCNC(=O)C(C1CCCN(C(C2CC2C(N)=O)=O)C1)C C1(C(=O)NC(C(=O)NCCCCCC)C2CC2)CCCCN1C(=O)OC C1(CNC(c2ccn(CCCC)n2)=O)COCCN(C(=O)CCc2ncc[nH]2)C1 c1(OCCC)ccc(C(=O)NC(C)(C)CCNC(=O)CS(=O)CC)c(OCC)c1 CCCC(C(=O)NC)NC(=O)C(C1CCCC1)NCc1cn(C)nn1 c1(C(N2CC3(CN(C(c4cc(OC)c(Cl)nc4)=O)C3)C2)=O)cnc2occc2c1 c1(OC)ccc(CC(=O)NCCCCCN(C(=O)CSCC(C)C)C)c(OC)c1 Cc1ccc(C(N2C(CNC(C3(C4CC4)CC3)=O)CC3CC23)=O)c2c1CCCC2 c1(CC)nccn1C(C)CC(=O)NCC1(O)CN(C(C2CC3CC3C2)=O)C1 c1(OC)nccc2cc(NC(=O)NCC3(C4CCOCC4)CC3(F)F)ccc12 N1(C(CC(C=C)C)=O)C2CCC1C1CC1(NC(=O)CNC(=O)C(C)(C)C)C2 n1(CC)nnc(C(=O)NCC(C2CCN(C(=O)CN3CCCC3)CC2)C)c1C C1(C(=O)OCC)CN(C(=O)CN(C)C(C2(NC(=O)C3CC3)CC2)=O)CCC1F C1(C(=O)NCC2C(C)OCC2)CN(C)CCN1C(C1CN2CCC1CC2)=O N1(C(C(C)Cn2cccn2)=O)CCCC(C)(CNC(=O)Cc2ccno2)C1 C(CCCCCS(=O)(=O)CCO)C(=O)NC(c1ncc(C)s1)C C(=O)(C1=COCCC1)NCC1(F)CN(C(=O)Cc2ccn(C3CCCCC3)n2)C1 c1(OC)ccc(C(CNC(C2CC=CCC2)=O)NC(=O)Cc2cnoc2)cc1 N1(C(C2(CC)CCOC2)=O)CCCN(C(=O)CCn2cc(Cl)cn2)C(C)C1 c1(C(=O)NCC2(C)CCCN(C(C(CCSC)O)=O)C2)cnc2c[nH]nc2c1 CCC(C(=O)NCC1CN(C(=O)C(c2ccccc2C(F)(F)F)(F)F)C1)C(C)O Cc1cc(C(=O)NCc2ccsc2C(N2CCN3CCC2C3)=O)c(C)cn1 C(C(C)(C(=O)N(C)CC1(CO)CC1)NC(=O)CC1CCOC1(C)C)SC c1(N(C(=O)CN2CCC(CC)C2)NCC)cccc(NC(C2CS(=O)(=O)C2)=O)c1 C(=O)(CCCN1CCCCC1)NCCC(C)NC(=O)CCNC(C1CCCO1)=O C12(CNC(C(C)C(F)F)=O)CCC(NC(c3cc(C#N)ccc3F)=O)(CC1)CO2 N#Cc1ccc(N)c(C(=O)NC2CCCC(C(N3CCC(CF)C3)=O)C2)c1 c1(C(N2CCC(OCCNC(C=C(C)C(F)F)=O)CC2)=O)ccc2c(c1)CCN2 c1(C(=O)NC(C)CCCNC(=O)CCc2ccccc2Br)n[nH]c2c1COC2 CN1C(=O)c2ccccc2C1CC(=O)NC1C2CC1CN(C(=O)CS(C)(=O)=O)C2 C(=O)(C1=CCCCO1)NC1C(CNC(c2ccnc(C3CC3)c2)=O)CCC1 N1(C(CC(C)n2cccc2)=O)CCCC(C(=O)NCC2(C3CC3)CCCO2)CC1 C1(C(=O)NC2CCN(C(c3onc(C)c3C)=O)CC2O)CC(C)(C)OC(C)(C)C1 CC(C)C1=NOC(C(N2CCN(C(=O)CC3CC3)C(c3cccc(F)c3)C2)=O)C1 c1(C(=O)NCC2(NC(=O)CCC(=O)C3CC3)CCOC2)cc(Cl)c(F)cc1F C(N=c1ccc([N+](=O)[O-])c(O)[nH]1)C1C(C)CN(C(=O)CC(O)C2CCCC2)C1 N1(C(CC(=C)C)=O)CCOCC2(COCCN2C(=O)CCCCC(N)=O)C1 C1(CC=C)(C(=O)NCc2cc(C)nn2C)CCCN1C(=O)Cc1cn(CC)nn1 C1(C(=O)NOCC2CCOC2)N(C(c2cc3n(n2)CCC3)=O)CC12CCCC2 c1(CC(CNC(=O)C(C)N(C)C)NC(CC2(CC)CCC2)=O)ccccc1 C1C(C)(C)C(=O)Nc2cccc(c2)CNC(=O)O1.C(C)(C)(C)OCCOC C1(CCCNC(Cn2ncc(C)c2)=O)CCCCN1C(=O)C(C1CCC(=O)N1)C Cc1nn(C)c(C)c1C(C)C(=O)N(CCN(c1nccnc1F)C)C(C)C c1(OC)ccc(Cl)c(C(CC(N)=O)NC(C2COC3CSC3C2)=O)c1 C1(NC(CSCCC)=O)CN(C(c2scnc2C(F)F)=O)CC1OC C1(NC(C(C)C2CCC2)=O)CCC12CCN(C(=O)CCc1ccc(O)nn1)CC2 N#Cc1ccccc1OCC(=O)NC1CCC(CNC(C2NC(=O)NC2=O)=O)C1 CON1CCC(C(=O)NCCOC2CCN(C(c3cnc(C)c(N)c3)=O)C2)CC1 c1(C(=O)NCC2CC(NC(=O)Cn3ncnn3)CC2O)coc2c1COC2 N1(C(CSCC=C)=O)CCCC(N(C)C(C2CN(C)CCO2)=O)C1 CC1(C)C=C(C(=O)NCC2COCC2NC(c2cc(-c3cccnc3)no2)=O)C1 C(=O)(C(C)(O)C(F)(F)F)NCC(C1CC1)NC(c1c(C(C)C)nns1)=O CC1CCCN(C(=O)C=CCO)C1CCNC(=O)Cc1ccnc(O)c1.C1(CC)CC1 C#CC1CN(C(=O)C(O)C(C)C)CCN1C(=O)C(c1ccccn1)C C12(CNC(C3C(NC(=O)COC4CCOCC4)CCOC3)=O)CCC(F)(CC1)C2 Cc1ccccc1C=CC(=O)NCCCNC(=O)Cc1cnccn1 CC(C)(C)C#CCCNC(=O)N(C1CCOC1)CCCOc1ccccc1 C=CCCCCCCCC(=O)NC1CCN(C(=O)Cc2ccon2)CC12CCC2 C1(C(=O)NC2C=CCN(C(c3nc(C(=O)OC)oc3)=O)C2)CCC(C)(C)OC1 c1(C(C)C)cc(C(N)=O)c(O)c(CN2CC(NS(=O)(=O)CC(N)=O)C(C#N)C2)c1 C(=O)(CC(F)(F)CC(=O)N1CC(NC(C2CCN(C)CC2)=O)C(F)C1)OC c1(C(N(CCOCCN(C(c2cc(C)no2)=O)C)C)=O)cc(N)ccc1Cl N1(C(c2cc(C(F)F)cc(F)c2)=O)CCC2OCCN(C(c3cnc[nH]3)=O)C2C1 C1(C(=O)NCCN(OC)C)CN(C(C2(CC3CCC3)CC2)=O)CC12CC2 N1(C(C=CCCC=C)=O)CCC(NC(c2ccc(C(=O)CC)cc2)=O)C(CO)C1 Cc1cccc(C2(C(=O)NC(C3CCN(C(c4c(Br)cnn4C)=O)C3)C)CC2)c1 Cc1cccc(OCCOCCC#N)c1C.c1(N2CC2)sc(Br)nc1C C1(C(N2CC(COC)OCC2)=O)C2CCC(C2)N1Cc1ccc(C)nc1 Cc1ncc(C(C(=O)NC(C)(C)C)N(C2CC2)Cc2nncn2C)[nH]1 C1(NC(=O)CN)CCC1F.C(CCO)N(S(C)(=O)=O)C C(=O)(C1=NOC(c2ccccc2)C1)N1CC(COC)(CNC2CC(=O)NC2=O)C1 C1(=O)C(C(C)(C)C)CN1CCCC.C(=O)(C#CC1CCOC1)NCCOC C1(C(N2CCC(OCC(C)C)C2)=O)CCCCN(C(c2ncc(F)cc2F)=O)C1 C(C)(C)(C(=O)N(C)CCN(C(C1CC(C)C1)=O)C(C)C)OCC N1(C(COCCCCCC)=O)CCCC(CN(C(=O)C(C)C(C)C)CC)C1 C1(CC(=O)NC2CC2NC(=O)CCc2nc(C3CCCC3)no2)CCS(=O)(=O)C1 Cc1c(C(=O)NC(CO)C(=O)NCc2nc(C(N)=O)co2)cccc1O C1(C(N2CC(C(C)NC(C(CC=C)CC)=O)C2)=O)CN(C)CCN(C)C1 C(=O)(C(C(C)C)NC(N)=O)NCC1(O)CC(CNC(c2cc(CC)on2)=O)C1 C(C(C)CC(C)C)N(Cc1cc(C)no1)CC1CC(NC(=O)OC(C)(C)C)CO1 C(C(CC(F)(F)F)NC(=O)Cc1ccns1)NC(CCc1nnc(C)n1C)=O c1(C(=O)NCC(CNC(C(CC)(F)F)=O)O)cc(C(F)(F)F)cc(S(C)(=O)=O)c1 N1(C(C=CC=CC)=O)CCC(NC(c2coc(C3CCC3)n2)=O)CC1C C12(C(N(CCCC=C)CC)=O)CCC1CN(C(c1cccnc1S)=O)C2 c1(C(N2CCC3(NC(C(C4CCCCC4)C)=O)C(C2)C3)=O)c(O)cc(F)cc1F C(C)(C(C)C(=O)NCc1cn[nH]c1)NC(C1(CCOC)CCC1)=O C(=O)(C(CC1CCCCC1)C(C)C)N(CCNC(C(OC)OC)=O)C Cc1nc(C(=O)NCC(C2CC2)NC(=O)C(C)n2cncn2)c2ccccn12 Cc1cc(C(N2CC=CC2CNC(=O)Cc2coc(C3CC3)n2)=O)nn1C(F)F N1(C(Cc2cn(C)nn2)=O)CCC(CCNC(C2CC(=C3CC3)C2)=O)CC1 CC(C)(CCNC(=O)CCCCC1CC1)C(=O)N1CCC(CN=[N+]=[N-])CC1 c1(N2CCC(C(C)NC(=O)CCc3nc[nH]n3)C2)nc2ccccc2s1 C12(CCOCC1)C(=O)N2.C(C)(C(C)NC(=O)C=CC(=O)NC1CC1)SCC C1(C(=O)NCC2(C)CCN(C(CCC3C(C)=NNC3=O)=O)C2)COC2COCC12 C(CCN(C)C)(C(=O)O)n1cc(CCNC(c2scc(C(C)=O)n2)=O)nn1 C1(N(C)C(C2C=CCC2)=O)CC(O)(CNC(C2(N3CCCC3)CCC2)=O)C1 C#CC1CN(C(c2cnc[nH]2)=O)CCN1C(c1cnnc(Cl)c1)=O c1(NC(c2sccc2NC(c2nc(Cl)sc2Cl)=O)=O)nc(Br)ccc1Br c1(C(C2N(C(C=CC=CC)=O)CC3(CC3)C2)=O)cnc2n1CC(C(F)(F)F)CC2 c1(CNC(C=CC(CC)C)=O)cn(C2CCN(C(C3CC3F)=O)C2)nn1 N1(C(c2cccc(C)c2Cl)=O)CC2CCOC2(CNC(c2c(C)noc2N)=O)C1 C(C(C)(CC(C)C)NC(=O)CNC(c1ccco1)=O)NC(c1c(C)cc(C)[nH]1)=O C1(CCNC(COCC(=O)NC)=O)(OC)CN(C(c2oncc2CO)=O)C1 Cc1c(O)cc(C(=O)NC2CCC(C(=O)NCCN(C)CCO)CC2)cc1O CC(C)CC(Cc1ccccc1)C(=O)NC1CCC(NC(=O)Cc2cnc[nH]2)C1 C1(NC(C(C)C)CCN(C(=O)COC2CCCC2)C)CCC(C2CCC2)CC1 N1(N2CCC(=CC(C)(C)C)CC2)CCc2cccc(Cl)c2C1.CC(O)C=O N1(C(CCCN(C(C)=O)C)=O)CCC(C(=O)N(C2CC2)CC2CCOC2C)CC1 CC(=O)CCCCC(=O)NC1(C(=O)NC2CCN(C)CC2)CCSC1 Cc1cccc(C(=O)NC2CC3(NC(c4c(CO)noc4C)=O)COC2C3)c1O C(=O)(CCCC1CC1)NCCC(C)NC(=O)CCOCC1CCOC1 c1(C(N2C(C(N3CCCC(C)(O)C3)=O)CC(=C)C2)=O)ccc(C#N)c(Cl)c1 C1(NC(C(C)OCc2cccc(C)c2)=O)CN(C(c2cccnc2)=O)CC1(C)C Cc1c(C(N2CCN(C(=O)CN3CC(C)C3)C(CO)C2)=O)sc2cncn12 S(=O)(=O)(c1cc(C(=O)NCC(CO)NC(C2(OC)CCC2)=O)c(C)o1)NC C=CCC(CC)C(=O)NC(C)C(C)(C)C(=O)N1CCCC1(C)COC c1(C(=O)NCC2N(C(C=C(C)C(F)F)=O)CC2)ncc(F)cc1N C1(C(=O)NCC2CCCN(C(c3nc(C)oc3)=O)C2)CCC2C(C1)C2(F)F Cc1ccc2ncn(CC(=O)NCC3CCC(C)N(C(=O)C4=CCOC4)C3)c2c1 c1(CCC(=O)NCC(C2CC2)NC2C(C(N3CCC3)=O)C2)csc(Br)c1 c1(C(=O)NC(C(C)NC(CCC#C)=O)C)cc(C)nn1CCO c1(C(N(CCCNC(c2c(OC)ccnc2)=O)C2CC2)=O)cnc2[nH]ccc2n1 c1(OC)ccc(NC(C2CCc3ccccc3O2)=O)c([N+](=O)[O-])c1I C12(CO)CCN(CC1)CCn1cc(nn1)-c1nc(sc1)NC2=O.S(C)(=O)(=O)SC C(=O)(C(F)CC(C)(C)C)NC(CCN(C(CCCOCC)=O)C)C(C)C C1(NC(C=CC2CCN(C(CC3CC(=C)C3)=O)CC2)=O)CCn2cncc2C1 N1(C(CC2(C)CN(C(c3ccc(CC)s3)=O)C2)=O)Cc2cc(Br)cnc2C1 c1(NC2CC2)c(-n2cccn2)ncnc1Cl.NCC1C(=O)NCCCO1 c1(N(CCC)C(=O)N(C)Cc2nccn2C2CC2)cc(C(F)(F)F)ccn1 C1(C(C)NC(C(C)SCCCC)=O)CCCN1C(c1ccc(COC)[nH]1)=O C1(CNC(CCN(C(C(COC)COC)=O)C)=O)OC(=O)CC1(C)C C1(NC(=O)COC2COC2)CCC(NC(=O)CC2CCCO2)CC1 c1(C(C)C)ncc(Br)c(N2CC3C(C(=O)Nc4ncc(Br)cn4)C3C2)n1 Cc1n[nH]c(C)c1CCC(=O)NCCCNC(c1cnc(Cl)s1)=O C1(NC(Cc2cccc(-n3ccc(CSC)n3)c2)=O)CC2CC1N(C(C)=O)C2.CO N1(C(C(c2ccncc2)C)=O)CC2CC(CNC(c3cc(C(F)F)no3)=O)C2C1 N1(C2CN(C(C3C(=C)CC3)=O)C2)CC(Nc2cc(-c3cccs3)ncn2)CC1=O C1(COC)CCN(C(C23CC2CCN3C(C2OCCOC2C)=O)=O)CC1 C=CC1OCCCC1C(=O)NC1CC(NC(C2Cc3nccn3C2)=O)C1 C=C(C)C1CN(C(=O)C(C)(C)C2CCN(C(=O)CN(C)C3CC3)C2)CCO1 C1(C(=O)NCCN(C(CC)C)C)CC2CC1CC2NC(=O)C#CC(C)(C)C CCC(C(=O)OC)C(=O)N1CC(NC(c2cc3scnc3[nH]2)=O)C(O)C1 c1(OC)nn(C)cc1CNC(=O)CC1CC(C)N(C(=O)CC(Cl)Cl)C1 C(C(O)CC(C)(C)C)NC(C1CN(C(CC2CN(C(C)=O)C2)=O)CC1F)=O C(=O)(C#CC1CC(F)(F)C1)N1CCN(C(C=CC=CCCCCC)=O)C(C)C1 c1(CN2CCCC(C(N3CCC(O)(C(F)(F)F)C3)=O)C2)ccc(F)c(Cl)c1 C1(C(=O)NC(C)CNC(C2CCC2)=O)CS(=O)(=O)CCO1 C1(C(N(C(C2C=CC(NC(C3C(CCC)C3)=O)C2)=O)C)C)CCN(C)CC1 Cc1cccc(Cn2cc(CC(C(=O)N(C)C)N(C(=O)C(C)C(F)F)C)nn2)c1 CCC(CNC(=O)CCCC#N)(CC)NC(=O)C(C)NC(=O)CC1C=CCC1 C1(C)(NC(C2CCCN(C(CC(C=C)CC)=O)C2)=O)CN2CCC1CC2 Nc1cccc(F)c1C(=O)NC1CC2(C1)CN(C(c1ccc(CC3CC3)s1)=O)C2 C1(CNC(C2(N(C(C3CC(=C)C3)=O)C)CC2(C)C)=O)CCC(CC)CC1 N1(c2nc(C(C)(C)C)on2)CCN(C(=O)NCC2(S(N)(=O)=O)CC2)CC1.C1C(=O)N1 C(=O)(N=S(C)(=O)C1CCNC2(CC2)C1)c1cc(CC)oc1C O=C(CN=c1cc[nH]cc1)NC1CCN(S(=O)(=O)CF)CC1 c1(OC)ccc(C(N2CC(CNC(c3cncs3)=O)C3CC23)=O)c(F)c1 C1(C(N2CCN(Cc3ccccc3)CC2)=O)CN(Cc2csc(Br)n2)CCS1.OC C12(NC(CC3CC(=O)NC3=O)=O)CCCC1N(CC1CN3CCC1C3)CC2 n1(CCNC(=O)CC23COC(c4cccc(C(=O)O)c4)(C2)C3)ncc2cccnc12 c1(SC)nc(C)cc(=NCC2CCC3(CCC3)C2NC(=O)CC(C)C)[nH]1 C1(CNC(=O)C2=CCCCCC2)CCC2(CCC2)CN1C(c1cc(CO)[nH]n1)=O C12(O)CCCN(C1)C2=O.c1(N(C(CNC(C2CCC2)=O)C2CC2)C)cnc(Cl)s1 C(=O)(C=C1SCC(=O)N1C)NCC1CN(C(C(C(CC)C)OC)=O)CC12CCC2 C=CCC(COC)N=c1[nH]c(N2CCN(S(C)(=O)=O)CCC2C)nc(=N)[nH]1 C#CC(C)(C)C(=O)N1CCOC(C(=O)NCC2(C#N)CC2)C1 CC1CN(C(=O)CC(c2ccc(Cl)cc2)O)CCN1C(c1cnccn1)=O Cc1c([N+](=O)[O-])c(CC(C)NC(C2CCCCCN2C(=O)OC(C)(C)C)=O)nn1C c1(OC)ccsc1C(=O)NC(C1CCN(C(=O)CCSCC(N)=O)C1)C.C(=O)OC C(=O)(C(O)C(C)C)N.C(CO)(C(=O)N(C)CCOCCCC(C)C)OC C12(NC(C(C(C)OC)NC(C(CCC)O)=O)=O)CC1COC2(C)C C(=O)(C(C#N)C(C)(C)C)N1C(CC(=O)NCC2CCC(C)(C)CC2)CCC1 C=CC1C(=O)N(CC)CC(C)NC(=O)N1.n1(CC(=O)NCC)ccc(C(F)(F)F)n1 c1(COCn2cncn2)cc(C(N2CC(CN(CC(=O)OC)C)CC2C)=O)c(C)o1 c1(C(=O)NC(C)CCN(C)C(c2ncn(C)n2)=O)ccnc(F)c1 C1(NC(C2(C(=O)NC)CC2)=O)COC2(C1)CN(C(c1nc(Cl)c(Cl)s1)=O)C2 Cc1ccccc1C(=O)NCC1CC(NC(=O)CSCCCC(C)C)C1(C)C C(CCC(=O)N(CCCOCCC(N1CCCC1CSC)=O)C)=CCC=C N1(C(c2cc(C)on2)=O)CCN(C(c2cc(Cl)c(F)cc2Cl)=O)C2CCC12 c1(C(C(=O)NC(CN(C(COCCC)=O)C)C)(F)F)ccc(C)cc1 N1(C(C2CCCN(C(N)=O)C2)=O)CCC2(CC1)CN(C(C1CC3C=CC1C3)=O)C2 C1(CNC(c2c(C)cco2)=O)CN(C(=O)NC2CN(C3CCCCC3)C2)CC1C C1(OCC(=O)NC(C)CC2CN(C(=O)CSc3nncs3)C2)CCC(F)(F)CC1 N1(C(C)(C)NC2CCN(C(=O)OC)C2)c2ccccc2N(C)S1(=O)=O Cc1ccnc2sc(C(=O)NCCCN(C)C(C3CC(C)(O)C3)=O)c(C)c12 C(=O)(C1=NOC(C)C1C)N(C1(C(=O)NCc2c(C)nc(C)s2)CCC1)C1CC1 c1(C(N2CC3C(C2)N3C(c2cc(Br)cc(I)c2)=O)=O)ccc(I)c([N+](=O)[O-])c1 c1(C(=O)NC2(C3CCCN(C(COC(C)=O)=O)C3)CC2)cc(=O)c2ccncc2o1 Cc1cscc1Cn1cc(CC(C(=O)O)NC(=O)C(C)ON)nn1 CCC(CC(=O)NCCCN(C(=O)CC(C)N1CCCC1=O)C1CCCC1)SC c1(CC)c(C(=O)N(CCNC(=O)CC2NC(=O)NC2=O)CC)sc2ccccc12 c1(C2C(C(=O)OCC)CCC2F)ccc(COC(C2(C)CCCCO2)=O)c(F)c1 c1(C(=O)NCC(CC)NC(=O)CSCCOC)csc(-c2ccoc2)n1 C1(NC(c2c(NC)snc2C)=O)CC(O)CN(C(c2c(OC)cccc2C)=O)C1 n1(CC(=O)NCC(C2CC2)NC(C(C)C#N)=O)ccc2c(=O)n(C)c(=O)n(C)c12 c1(C(N2C(C)CC(NC(=O)CNC=O)C2)=O)ccc(CN(C)C)cc1Cl N1(C(=O)NCCC(C(=O)OC)C)CC(N=[N+]=[N-])CCC1(C)C CC1CCC(C(N2CCOC(CNC(c3cc(Cl)nnc3O)=O)C2)=O)C(=O)N1 c1(CC)ncc(C(C(=O)NCC2CC2)N(C)CC2(C(C)(F)F)CC2)s1 N1(C(Cc2cn(C)nc2)=O)CCN(C(c2cnccn2)=O)C(c2ccccc2)C1 N1(C(C2CCN(CC)C2)=O)CC(C(N2CCCC(N(C)C)C2)=O)OC(C)C1 Cc1ccc(C(=O)Nc2ccco2)c(CN(C(N2C(C3CCC3)CCC2)=O)C)c1 C1(C(N(CCC)Cc2noc(C)n2)=O)CCN(C(=O)CC2CCO2)C1 C1(C#N)(CN=[N+]=[N-])CCN(C(c2ccccn2)C(=O)NC2CCCC2)CC1 N1(C(CN(C)C)=O)CCC(O)CC1C(=O)NC1(CO)CCSC1 C1(C(=O)NC2CN(C(c3c(OCC=C)cc(Cl)cc3)=O)C2)CC1C1CCOCC1 C(=O)(C(C)(C)C(=O)N(C)CC1CN(C(=O)C(C)N(C)Cc2ccccc2)C1)OC N1(C(C2N(CC)CC2)=O)CCC(C(=O)NCCCC2(C)CC2)(CO)C1 N1(C(c2c(CC)ocn2)=O)CC2CC1CN(C(C1CCS(=O)(=O)C1(C)C)=O)C2 c1(C(=O)NC2CC(C(C)NC3CCC3)C2)c(F)c[nH]c(=N)c1C#N NS(=O)(=O)c1coc(C(N2CC3CCC3(NC(C3CC3F)=O)C2)=O)c1 CCCC(CC)C(=O)NCCC1CN(C(C23CC4CC2C3C4)=O)CCO1 C1(C(=O)NCc2cc(C)no2)CC2CCC1N2C(C1CCCN1C(=O)NC(C)C)=O C1(CN(C(=O)CC2CCC2)C)CN(C(c2cnc(CC(C)(C)C)o2)=O)CCO1 CCC(C)CN=c1nc(N2CCN(CC(=O)N(C)C)CC2)c2c([nH]1)CCC(C)C2 Cn1ccc2c(C(N3CC(NC(c4cnn5cnnc5c4)=O)C3)=O)cccc12 C(=O)(C#CC1(CC)COC1)N(C1CCN(C(c2ccc(O)nc2)=O)C1)CC c1(C(N(CC(C)O)CCNC(C2CC2F)=O)=O)cc(C(N)=O)cc([N+](=O)[O-])c1 c1(C(=O)NC2C(NC(COCC)=O)CC(F)(F)C2)ccc2c(c1)n(C)c(=O)n2C C1(NC(C2N(CCC)CCCC2)=O)CC2(CCCCN2C(C2CCC2)=O)C1 C1(CC(=O)NC2CCN(CCF)C2)(CNC(=O)CN2CC=CC2)CCCC1 N1(C(C(CCSC)N(C)C)=O)CCC(NC(c2c(C)noc2C)=O)C(O)C1 Cc1cc(C(N2CCCCC2C(=O)NCc2cccc(C(N)=O)c2)=O)nc(C)c1 c1(CC)ccc(C(=O)NC2CCC(C)(NC(=O)CCc3cnco3)CC2)cc1F C1(C(=O)NC2CCCC(NC(C3(C=C)CC3)=O)CC2)CC2CCC(C1)N2C CC(CC(F)F)C(=O)NC12CC(CNC(=O)CCC3(C)N=N3)(C1)C2 c1(OC)cc(C)c(C(=O)NCC2(O)CCN(C(C3(c4ccno4)CC3)=O)C2)cn1 CC1CN2CCN1C(C(=O)NC1(CNC(c3ccc(F)c(O)c3)=O)CC1)C2 N1(C(CC=CC=C)=O)CCCC(N(C)C(c2cc(C(C)=O)ccc2OC)=O)CC1 CC1(C)Cc2ccccc2CN1C(=O)Nc1ccccc1.C12C3CN(CC13)C2 C(=O)(C1=NN(C)C(=O)CC1)NCCOCCOCCCNC(c1c(CC)ncs1)=O c1(C(N(C2CCN(C(C3CCOC3)=O)C2)CCC)=O)csc(C(F)(F)F)c1 CCCC(CNC(=O)CCc1cccs1)NC(C12CC(C1)C2)=O C(=O)(CC1=NNC(=O)C1)N1CCC(NC(Cc2n(C(C)C)ncc2)=O)CC1C c1(C(N2CC(N(C(CCSC)=O)C)C2)=O)c[nH]c2cccc(C)c12 c1(CC(=O)N(C2CN(C(=O)CC3(C)CC3)CC2F)C)cncc(F)c1 CCCC(C(=O)OC)OCC1CCCN1Cc1ccnc(Sc2ccccc2)n1 C1(NC(CCC(=O)NC)=O)CC2CC(NC(c3cnccc3C)=O)CC12 CC(CC(=O)NCCN(C(=O)CC1(C)CCCCCC1)C1CC1)C(C)(C)C C1(C(N(CCS(C)(=O)=O)C)=O)CCN(C(=O)CC2C=CCC2)CCO1 N1(C(C2C(CNC(COC3(C#C)COC3)=O)CCCC2)=O)CCc2c[nH]nc2C1 C1(C(N(CCCCCO)C)=O)CNC(=O)CN1C(C1CC(=O)CC(=O)N1)=O N1(C(CC(C)C)=O)Cc2ccnn2CC(NC(=O)C(F)C(C)(C)O)C1 C1(NC(c2cc(C)c(Cl)s2)=O)CN(C(c2ncoc2C(C)C)=O)CC1C1CC1 C(=O)(CC(C)F)NCCCN(CCCCNC(C1C(C)C1)=O)C N1(C(C2N(CC)CCCC2)=O)CC(C)(C(N2CC3(CNC(=O)C3)C2)=O)CC1(C)C c1(C(N(C2C(C)C2)C)=O)ccc(CNC(C2OCCC2(C)C)=O)nc1 C(=O)(C1=NOC(C)(C)C1)NCC1N(C(c2cc(C)c(C)s2)=O)CC2(CC2)C1 N1(C(CCCC)=O)CCN(C(c2nc(C)nn2C)=O)C(c2cccnc2)C1 N1(C(C(C)(C)C)=O)CC(Nc2ccc(C(F)(F)F)cn2)CC(C)(C)C1 c1(C(=O)NCCCN(CC(O)C(=O)NCCOC)C)cc(Cl)c(Cl)c(Cl)c1 c1(C(=O)NCC2C(NC(c3n(C)nnc3)=O)C2)csc(Cl)c1Cl CC1(C)C=C(C(=O)N2CC(CNC(=O)CCCF)CC2(C)C)C1 N1(C(c2cc(SC)c(C)o2)=O)CCC(NC(=O)C=Cc2ccc[nH]2)C(CO)C1 c1(CNC2CCCC(C(N(CC)CC)=O)C2)cccc(-c2nn[nH]n2)c1 S(=O)(=O)(c1cccc(F)c1)N1CC2(CC(CNC3(C(N)=O)CCCCC3)OC2)C1 N1(C(C(n2ncc(C)c2)C)=O)CCCC12CCN(C(=O)C=Cc1cnc(C)s1)C2 c1(-c2cn(CC)nc2)ccc(NC2CC2C)c([N+](=O)[O-])c1 N1(C(C2(c3cccnc3)CC2)=O)CC2CCC(NC(C3(C)CCCOC3)=O)CC2C1 c1(C(=O)NCCN(C(=O)CC2CC(F)(F)C2)C)nnc(N2CCCC2)o1 S(=O)(=O)(c1cccnc1NC1CCc2nncn2CC1)NCCC(CCC)O c1(OC)cccc(C(=O)NCC(O)CCNC(C2CC2c2ccn(C)n2)=O)c1C CC(C)CCC(C(=O)Nc1cccc(O)c1F)NC(=O)C(F)n1ccnc1 c1(CC)cc(CC(=O)N(CCNC(C2CS(=O)C2)=O)CCOC)n(C)n1 N1(C(c2cc(CC)on2)=O)CCN(C(c2sc(C)nc2CC(C)C)=O)C(C)C1C N1(C(C(C)(C)C2CCCO2)=O)CC2CC2(CNC(c2ccncc2F)=O)C1 CC1(C(=O)NOCC2CCOC2)C=CCN1C(C1CCSCC1)=O C1(NC(C2C(C)(C)CC2)=O)CCC2CC1CN2C(=O)C=Cc1ccc(=N)[nH]c1 C1(NC(c2cnc(C3CC3)o2)=O)CCCC(NC(c2ccoc2C2CC2)=O)C1 c1(C(N2CC(F)CC(NC(=O)Cc3ccccc3Cl)C2)=O)ccc2nncn2c1 c1(C(=O)NC2C=CCN(C(=O)Cn3cnnc3O)C2)cc2c(=O)cc[nH]c2s1 C(=O)(C1CCCc2scnc21)NC1C(NC(Cc2c(C)ccs2)=O)CC1 C1(n2cc(-c3onc(C)n3)nn2)CN(Cc2cc(Br)no2)CC1C c1(CC)ncccc1C(=O)NCC(=O)NCC1CC1c1ccc(F)cc1 n1(CC(=O)NCCCOCCN(C)C(C2CC(CCO)C2)=O)ncnn1 Cc1nc(C(N2CCSCC2CCNC(C2(CCN(C)C)CC2)=O)=O)c(C)n1C Cc1cc(C(=O)NC(c2ccccc2)CNC(C2CCOCC2C)=O)cnc1C C(=O)(CC(C)C(C)(C)C)N1C(C(=O)NCCOC)CC(N=[N+]=[N-])C1 C1(C(N2CC(CCNC(COC)=O)C2)=O)CCN(c2cnccn2)CC1 C#CC(C(C)C)NC(c1conc1C(C)NC(c1cc(CCO)on1)=O)=O c1(-c2ccc(C(N3C(C)COCC3)C(=O)NCCC#N)o2)cc(Br)ccc1F C12(NC(=O)CC3(OC)CN(C(c4cnn(CCF)c4)=O)C3)CC(CCO1)C2 N#CC1CN(Cc2ccc(C(F)(F)F)cn2)CCN1C(c1cccc(O)c1F)=O N1(C(Cc2nc(C)sc2)=O)CC2(C1)SCCC2NC(c1cc(C)c(C)s1)=O c1(C(N(CCC)CCNC(c2cnn[nH]2)=O)=O)ccnc2ncccc12 Cc1c(C(=O)NCC(C)N(C)C(C2CC3(C2)CS(=O)(=O)C3)=O)[nH]c2c1CCCC2 C1(CC)Cc2ccccc2CN1C(C(=O)NCCC1CC1)C1=CCSC1 N1(C(c2cc(OC)c(Br)nc2)=O)CCC2(C1)CN(C(C1(F)CCC1)=O)C2 Cc1cc(=NCC2(C(F)(F)F)CC2)[nH]c(=NCC(=O)N2OC3CCC2C3)[nH]1 C(C(=O)N=c1ccn(C(C)CC)[nH]1)N(C(=O)C(CCC)N(C)C)CCC#C c1(C(N2CC3C(NC(=O)CC4COC5CC4C5)C3C2)=O)cnc(O)c2c1NCCC2 C1(NC(CN2CC(C)(C)C2)=O)CC2CC1N(C(C1(C)CC=CCC1)=O)C2 c1(-c2cn(CCC(N3CC=CC(NC(C)=O)C3)=O)nn2)cccc(C(=O)O)n1 C(CCSC)(CN=c1[nH]c(N2CC3CCCCC3C2)nc2ccccc12)OC C(=O)(C(=O)N=S(C)(C)=O)N1CCC(O)(C(C)NC(c2cc(=O)n(C)cn2)=O)C1 C1(C(N(C(C(=O)NCCCc2cnn[nH]2)C2CC2)C)=O)CC12CCOCC2 C1(NC(=O)CC(O)CNC(C2CNC(=O)O2)=O)CC2(COCCO2)C1 Cc1ccnc(C(=O)NC2CCCCC2CNC(c2snnc2C)=O)c1N c1(CN2C(CC)CN(C(=O)Cc3cc(OC)ccc3C)CC2)cc(O)c(Br)cc1O c1(N(C2CCCN2)CC)ccn2nccc2n1.c1(O)ccc(C(F)(F)F)c(OC)c1 c1(C(=O)NC(C(=O)N(C)CC2CC(F)C2)C2CC2)ncncc1Cl C(C(C)(C)C(=O)NCC1CC(NC(=O)CCc2ccc[nH]2)C1(C)C)OCC N1(CCCC)C(=S)NC(c2cnc(O)c(Br)c2)C2=C1CC(C)NC2=O c1(CC)ncc(C(N2CCC(N(C(=O)C(F)(F)COC)CC)CC2)=O)c(O)n1 c1(OC)ccn2cc(C(N3CC(C4CN(C(C5CNC(=O)N5)=O)C4)C3)=O)nc2c1 C1(C(=O)OC(C(C#C)(C(C)C)c2ccccc2)=O)CC2CN(CC)CCN2C1 C1(n2cc(CCSCC)nn2)CCC(N(C(=O)CC2CCOCC2)C)CC1 C1(C)(CC(=O)OC)CCN1C(=O)C(Cn1cccn1)NC(=O)CCN1CCCC1 c1(C(N2C(C)CN(C(=O)CCc3ccc(Cl)cc3)CC2)=O)ccnc2c1CCO2 N(C(=NCCC(C)=O)NC1CCN1c1ccc(Cl)cc1)CC(C)OC N(C(=NCc1cccc(Br)c1)NC(C1CC1)C1CC1)C(C)(C)C Cc1ccc(S(=O)(=O)NCCCNC(c2ccc(-c3cnco3)cc2)=O)cc1 C1(NC(C2C(C)CC(=O)NC2)=O)CCC2CN(c3nc(C4CC4)ns3)CC2C1 c1(C(C(N2CC3C(NC(=O)C4=CCCCC4)C3C2)=O)=O)c[nH]c2cc(F)ccc12 C1(NC(c2cnc(CCC)s2)=O)CCN(C(C2COC2)=O)CC1C(C)C c1(OC)cc(C2CCN2C(=O)NCC2CCS(=O)(=O)CC2)ccc1F Cc1cc(C)c(C(=O)NC(C(=O)NOCC(=O)N(C)C)C2CC2)o1 Cc1nc(C(=O)NC2CC(CC(=O)Nc3[nH]nc(CO)c3C(N)=O)C2)ccc1F C1(C(=O)NCCCCCNC(C2(OCC)CCOC2)=O)CCn2cncc2C1 c1(C(=O)NCCC(C)NC(=O)CN(C)CCO)ccoc1CCc1ccccc1 C1(C(N2CCN(C(CC(C)C)=O)CC2C)=O)CC2COCC(C1)C2(F)F CC1C(C(=O)NCC2(O)CN(C(=O)C(C)S)C2)C1(F)F N1(C(CN2CC(CC)C2)=O)CC2C3CCC(C2C1)N(C(c1cncc(N)n1)=O)C3 C1(OC)(CNC(C2CC(=C3CC3)C2)=O)CCN(C(=O)CN2CCCCC2)C1 c1(CNC(=O)NCCSC)ccn2nncc2c1 C(=O)(C1c2c[nH]nc2CN1C(=O)CCCn1cccn1)NCCC(=C)C Cc1nsc(C)c1C(=O)NC1CC(O)(CNC(c2ccc(C(C)(C)C)cc2)=O)C1 c1(C(=O)NC(COCCCNC(C(C)SCC)=O)(C)C)c(F)ccc(F)c1O C1(C)(C(=O)NCCC(CNC(COc2cccc(C)c2)=O)(C)C)CCN(C)C1=O C(=O)(C(F)C(F)(F)C(F)(F)F)NCC(CNC(c1n(CC)c(O)nc1)=O)(C)OC C(=O)(CS(=O)(=O)c1nnc(-c2ccccc2)n1Cc1occc1C)NC1C(CC)C1 N1(C(c2ccc(C(C)(C)C)[nH]2)=O)CC(F)CC1CNC(=O)CSC(F)(F)F C=CCC(CC)C(=O)NCC(C1CCOC1=O)NC(c1ncoc1C(C)(C)C)=O C1(C(=O)NC(CC)CNC(=O)CC(C2CCC2)C2CCC2)C(C)(C)CCCC1(C)C c1(C(=O)Nc2ccc(Br)cc2Br)cnn2c1CN(S(=O)(=O)CCCCl)CC2 CC(=O)CCCCC(=O)NCC(=O)NCC(N1CCC2(CC1)N=N2)=O N1(C(N2CCN(c3ccc(C)c(C)c3)CC2)=O)CCC2(CC1)CC2C(=O)ON(C)C N1(C(C(C)SC)=O)CCOC(CC(=O)NCc2ccc(C)nn2)C1 C(CCCN=[N+]=[N-])C(=O)NC1CCN(C(C(C)CC2CCC2)=O)C1 Cc1nc2sccn2c1C(=O)NC1CC1NC(c1cnc2cnccc2c1)=O C1(NC(c2ccc(C(N)=O)s2)=O)CC2(C1)CC(NC(c1ccc(F)cc1N)=O)C2 N1(C(CCSCC)=O)C2CCC1CC(N(C)C(C1CCCN(C(=O)CC)C1)=O)C2 c1(C(C)=O)ccc(C(=O)NCC2CCN(C(c3ccc(F)cn3)=O)CC2)cc1O C1(CC(=O)N(CC#C)CC)CCCC1C.C12(CC1)C(=O)N2 C1(OC(C)C)CCCCC1.C12CC(C)N1C(=O)CCNC2=O.C(N)(=O)N C1(C)(NC(c2cc(C)sc2Br)=O)CCCN(C(C2(c3ccno3)CC2)=O)C1 N#Cc1ccccc1CN1CC2CC2(CNC(c2ccc(CC#N)cc2)=O)C1 c12cccc(c1)S(=O)(=O)N(C)S(=O)(=O)CC2.C(=O)(C(CC1CC1)CC(C)C)NC N1(C(COCC=C)=O)CC(F)(F)CC1CCNC(=O)C(C)CC(F)F c1(C(=O)NCCCN(C(C2C(C)(C)C2(C)C)=O)CC)nn(C)c(Cl)c1Br N1(C(C(C2CC2)OCC)=O)CCN(C(=O)CCC(=O)c2cnn(C)c2)C(CC)C1 n1(CC(C)C)cc(C(=O)NCC2CC2NC(c2cc(Cl)ns2)=O)cn1 C1(N(C)C(C2(C(C)(C)C)CCC2)=O)CCCCC1NC(C1CCSCC1)=O c1(C(=O)NC(CNC(C2CCCN(C)C2)=O)CO)cccc2c1nc(O)n2C Cc1cc(=NC2CC23CCC(CO)CC3)[nH]c(N2CC3CCC(C2)N3C)n1 C1(CC=C)(NC(=O)C(F)C2CCCC2)CCN(C(c2snnc2C)=O)C1 N1(C(C2(CC(C)C)CC2)=O)CC2(CCN(C(c3n[nH]c4c3CCSC4)=O)CC2)C1 Cc1cc(C(=O)N(C(C)CN(C(=O)Cn2cnc([N+](=O)[O-])c2)C)C)ccc1F N1(Cc2ccc(CN(C)C)cc2)C2CCC1CC(NC(=O)C1=COCCO1)C2 C1(C(=O)NC2(C#N)CC2)(CNC(C(C)=CC=C)=O)CCCCC1 C1(CC(N2C(CNC(=O)C=C(Cl)Cl)CC3CC32)=O)CCn2cncc2C1 C(=O)(C1=CCCSC1)N(CCCN(C(C1(SC)CC(O)C1)=O)C)C C=CCC(C(=O)NC1CC1CNC(c1ccc(CS(C)(=O)=O)o1)=O)OC C(=O)(C1=NN(CC(C)C)C(=O)CC1)NCCC(C)NC(c1c(CC)nc(C)o1)=O C1(CNC(c2cnc(Cl)cc2Cl)=O)CCCN(C(=O)CC(O)CC2CC2)CC1 N1(C(c2c(C)n(-c3cccnc3)nn2)=O)CCc2cc(C#N)ccc2C1 c1(OC)ccc(C(=O)NC2(C)CCN(C(c3cc4sccc4[nH]3)=O)C2)c(N)c1F c1(C(N2CC(CNC(Cc3cnc(C)o3)=O)C(O)C2)=O)c(C)nc(C)n1O N1(C(CC(C)c2ccco2)=O)C2CCC1CC(CNC(C1(O)CC1(C)C)=O)C2 c1(CC(=O)N(C2CN(C(=O)CC3CC3)CC2F)C)ccc(C(F)F)cc1 c1(CN2CC(C)(C(=O)Sc3ccccc3)C2)c[nH]c(=NCC2CCS(=O)(=O)C2)s1 N1(C(c2cncc(C(C)=O)c2)=O)CC2CC1CCCN2C(=O)CC1CCCC1C C1(C(=O)NCc2cc[nH]n2)(NC(C(C)c2ccco2)=O)CCC(C)(C)C1 C1(C(=O)NC(CNC(C(c2cccc(Cl)c2)CC)=O)(C)CO)CN2CCC1CC2 c1(C(=O)NCCN(C(c2nc(COC)oc2)=O)C)ccc(O)c(N)n1 C1(N(C(=O)CC2CCC2)C)CCOCC1C(=O)NCC=C1CCSCC1 C1(OC)CC(C)CN(C(=O)CCC2CC(NC(c3c[nH]c(C#N)c3C)=O)C2)C1 Cc1cc2ccc1OC(=O)C2.c1(Cc2cccc(CO)c2)cccc(F)c1F Cc1cc(CC(=O)NCC2(O)CCN(C(c3nnc(O)cc3C)=O)C2)cc(C)c1 N1(C(=O)C2=CCCSC2)CCCCCC(NC(C2(F)CC=CCC2)=O)C1 C1(CNC(c2[nH]c(CC)c(Cl)n2)=O)CCC(C)CN1C(=O)CN1CC(=O)NC1=O C1(C(N(CCCCCC=C)C)=O)CN(C(=O)C(C)(C)O)CCC1(C)C C1(CNC(c2n(C(C)C)ncc2)=O)C2CC1N(C(C1CCSC1)=O)C2 Cc1cc(C(N2CC(O)(C(F)C(N3CCC4(CC4)C3)=O)C2)=O)nc(C)c1 c1(OC)ccc(S(=O)(=O)N(C2CC2)CC2CC3CCC2CC3)c(C(F)(F)F)c1 N1(C(c2nn(CC)c(C)c2)=O)CC2C3CCC(C2C1)N(C(=O)C(O)CSC)C3 C(=O)(CS(=O)(=O)C12CC(C1)C2)N1C(CNC(c2ccc(C)c(O)n2)=O)CC1 C1(NC(C2(CO)C(C)C2)=O)CCCC12CN(C(c1ccc(-c3cccs3)o1)=O)C2 C(CC(CNC(c1ccc(CC(C)C)s1)=O)NC(=O)C(c1ccccc1)F)OC C(=O)(C(CC(C)C)NC(C)=O)OCC.C12CCCCN1C2 C1(O)(CNC(CCOC)=O)CCCN(C(C2CN(C)CCO2)=O)CC1 C#Cc1ccc(C(=O)NCC2CCCC(NC(=O)CCCc3ncco3)C2)cc1 Cc1ccnn1CC(=O)NC1CC(NC(c2csc(Cc3ccccc3)n2)=O)C1 Nc1c(C(N2CCC3(CC(NC(=O)CC4C=CCC4)C3)C2)=O)cc(F)c(F)c1F CCCCC(=O)NC1COCC1CNC(c1ccnn1CC1CC1)=O C1(NC(=O)NC2C(C(=O)NCCC(=O)OC)CCOC2)CCCCNC1=O N1(C(C2C(C)(C)C2(C)C)=O)CC(NC(c2ccccc2Cl)=O)C(F)(F)C1 Cc1cc(C(=O)N(C2CC(NC(=O)CCC3NC(=O)NC3=O)C2)C)c(C)c(C)c1 C12(NC(C=C)=O)CCCCCC1N(C(=O)CCc1ccccc1)CC2 C1(C(=O)NCCN(C(C)C)C)CC2C=CC1N(C(=O)CCC(C)(C)C)C2 c1(C(=O)NCC(CC)NC(=O)C=CCN(CC)CC)coc(SC)c1 CC(O)CCCCCC(=O)NCC1(NC(=O)CCN2CCOCC2)CCOC1 CCC(CC(=O)N1CC(CCNC(c2ccc(C(OC)OC)o2)=O)C1)C(F)F c1(SC(C)C(=O)N(C2CCN(C(=O)CSC)C2)Cc2ccncc2)ccccn1 C(=O)(CCCCC(=O)N1CC2CC(NC(=O)C=Cc3ccc(C)cc3)C1C2)OC c1(C(=O)NCC2(O)CC(NC(CC(C)(F)F)=O)C2)cccc2c1NC(=O)CC2 C=CC1(NC(C=CCNC(=O)C2CC2)=O)CCCCC1.c12cccnc1C(=O)N2 c1(NC(C(CCC)NC(C2CC2C2CC2)=O)=O)ccc2cnccc2c1 C1(NC(c2cc(NC(=O)OC(C)(C)C)c(I)cc2)=O)CCc2cc(F)ccc2O1 c1(CNC(C)=O)sc(Cl)cc1C(=O)NCCC(O)CNC(C1(C(F)F)CC1)=O N1(C(c2nc(C(=O)OCC)oc2)=O)CC(CNC(=O)C(C)NC(C)=O)C(O)C1 C1(C)(C(N2CC(O)(C(=O)OC)C2)=O)CC(O)CN1C(C1C=CC=CC=C1)=O S(=O)(=O)(c1ccnc(C(=O)NCC2CN(C(C3CCO3)=O)C2)c1)NC C(=O)(C1=CCCCCC1)NC1CCCN(C(CCc2nc(C)sc2)=O)C1 C1(CNC(=O)C=CC2CCC2)CCN(C(C2CCCN2C2CC2)=O)CC1(F)F C1(NC(c2n(C)nnc2)=O)CCN(C(c2ccc(C3CC3)o2)=O)CC1F Cc1cccc(CC(=O)NCC2CCCCN2C(=O)COC2CCOC2=O)c1 N1(C(C(C)N(C(C)=O)C)=O)CCC(CC(C)NC(c2cc(O)ncn2)=O)CC1 N1(C(c2nccc(C)n2)=O)CC2CCCCC2(CNC(c2cnc(N(C)C)o2)=O)C1 N1(C(C2C(C=C)C2)=O)CC(NC(=O)CCOCC2CCC2)CC2(CC2)C1 C1(C)(NC(c2c(C(C)C)n[nH]c2)=O)CCCCC1C(=O)NCCCC1(O)CCC1 C1(C)(CCNC(CCOCCCOC)=O)CCN(C(c2ccncc2O)=O)C1 N1(C(CSCCN(C)C)=O)CCOC(C)(CNC(C2CCN(C3CC3)C2=O)=O)C1 N(C1CN(C(c2occc2C)=O)CCc2ccccc21)C(c1nc(C)sc1)=O N1(C(c2c([N+](=O)[O-])ccc(OC)c2)=O)Cc2[nH][nH]c(=NC(=O)c3ccc[nH]3)c2C1 CCC(C(=O)NC(C1CCCC1)CNC(c1ccc(C2CC2)nn1)=O)C(F)(F)F C1(NC(C(=O)NCC2(C)CCOCC2)=O)CCCC[Si](C)(C)C1 C1(NC(C=C(CCC)C)=O)(CO)CCN(C2CCN(C3CCCC3)C2=O)CC1 N1(C(C(C)c2cccs2)=O)CCC2(CNC(C3(CO)CCC3)=O)CCCC12 N1(C(c2c(C)ccnc2O)=O)CCCN(C(=O)CCN(C2CCCCC2)C)CCC1 N1(C(CC2(C)CNC2)=O)CCCc2c(CCN)cccc21 c1(N(C(C)CNC(=O)Cc2ccc(Cl)s2)C)ncnc(Cl)c1F C1(NC(C(C)(C)CF)=O)CC1C1CCN(C(C2CCCNC2=O)=O)CC1 CC(C)C#CC(=O)N(C(C)CNC(c1ccc(-c2ncon2)cc1)=O)C CCCC(C)(O)C(=O)NCC(O)CNC(=O)CC1CC(C)(C)CCO1 c1(C(c2ccc(O)cc2)=O)cc(N)ccc1O.C1(N(S(C)(=O)=O)C)CNC1 c1(C(=O)NC2C(C(=O)NC(C(=O)OC)CO)C2(C)C)cccc(F)c1 CC(C)C(C)(C)C(=O)N1CCOCC(C(=O)NC(c2nccc(O)n2)C)C1 C(c1c2c(nn1C)CCCC2)=CC(=O)NC1C2CN(C(CC(C=C)(C)C)=O)C1C2 c1(COC)nc(OC)cc(NCC(C2CCCC2)NC(=O)CC(C)O)n1 c1(C(=O)NCC2CCN2C(=O)CCc2ncc[nH]2)cc2c(Br)coc2cn1 N(C1COc2cc(Br)ccc21)C(c1n(CCC)nnn1)CCC1CCCC1 C(=O)(C1c2c[nH]nc2CN1C(=O)CC1=CCCCC1)N(CC(C)C)CCO c1(C(c2nnnn2C2CC2)NC2C(Cl)(Cl)C2)ccc2c(c1)OC(F)(F)O2 C1(NC(C(CC)SC)=O)CN(C(c2nc[nH]c2C2CC2)=O)CCC12CCOCC2 C1(C(=O)NCC(CC(=O)NC2(C)CCCC2)OC)(OC)CCC(C)C1 c1(C(=O)NCC2(CNC(C(C3CC3)SCC)=O)CC2(F)F)cncc(F)c1Cl c1(C(N2CCC(C(=O)NC3COCC3N(C)C)(CC)C2)=O)ccnc(C)c1C C1(OC(=O)Cn2ccc(I)nc2=O)CCCC2CCOC12 C1(NC(C(Cc2c(C)noc2C)C)=O)CCN(c2ccc(C(N)=O)nn2)CC1F C=C1CCN(C(=O)CC2CSC2)C(C(=O)NCC(CC)N2CCCC2)C1 N1(C(CC(C)C)=O)CC2(CCC2NS(N(c2ccccc2)C(=O)C(C)C)(=O)=O)C1 CCCCC(C(=O)NCCCCCNC(C1CC2CC2(CC)C1)=O)C(C)C Cc1ccc(C(=O)NC23CC2CN(C(=O)COCc2ccccc2C)C3)c(O)n1 C(=O)(C1=C(C2CCOC2)N(CC(=O)O)C(=O)NC1c1cc(Cl)cc(Br)c1)OCC c1(C(=O)NC2CN(C(=O)CCc3nc[nH]n3)C2)c[nH]c2nccc(Cl)c12 CCC(C(=O)N1CC(O)(CNC(=O)CSC2CCOC2=O)C1)C(F)(F)F C1(C(=O)NCC(CC)NC(=O)CCCn2c(C)ccc2C)C2CCC(=O)C12 C1(CNC(C(C=C)O)=O)(CNC(C2CC(OC(C)(C)C)C2)=O)CCOCC1 C=CC1(C(=O)NC2CC3(C2)CC3C(N2CCC(C)(O)CC2)=O)CCOCC1 c1(N(C)C)nc(Cl)c(C(=O)NCC(O)CCNC(c2c[nH]nc2C2CC2)=O)s1 c1(C(N2CCC(C(=O)NCCC)C(C)C2)=O)csc2c(OC)cccc12 C1(CNC(c2c(C)oc(Cl)n2)=O)C(C2CC2)CCN1C(c1coc(C(F)F)c1)=O c1(CC(C)C)ccc(CC(=O)NCCNC(=O)CSCc2ccccn2)cc1 c1(C(N2C(C)(CNC(=O)CC(F)(F)Cl)CCC2)=O)cnc(O)c2ccccc12 c1(C(=O)NCC2(O)CN(C(=O)CCCC3CC3)C2)ccc(F)c2cccnc12 C(C(O)CC(=O)N1CC(c2ccccc2)CC1CNC(C1(CF)CC1)=O)N(C)C C(=O)(CC(C)(C)OCC)NCCCC(=O)NC(COC)CCO CC(CC(N)=O)C(=O)NCCCC1COCCN1C(=O)CCC1(C)CC1(F)F c1(C(C)C)ccc(C(=O)N(C2C3CN(C(c4ccc(=N)[nH]c4)=O)CC23)C)cc1Cl N1(CCC(N2CCC(N(C(C3CCCC3)=O)CC)C2)=O)CCCCCC1 C(C(COC)CC(=O)N1CC(CN(C(=O)CC2CCCC(C3CC3)O2)C)C1)OC C(=O)(C1=CC2(CN(N(CC(c3nn[nH]n3)C)C)C2)OC1)NC(C1OC2CCC1C2)=O.C(=[N+]=[N-])CC C1(NC(CC(C)c2ccccc2)=O)CC2CC(NC(=O)Cc3ccco3)C2C1 Cc1ccc(Oc2ccc(NC(C)(CNC(=O)OC(C)(C)C)CO)cc2)cc1 C(C(C(=O)NCC(O)CN(C(=O)CCC(=O)N(C)C1CC1)C)C(C)(C)C)OCC=C c1(C(=O)NC(CN(C(=O)Cc2c[nH]nc2O)CC)C)cccc2c1C(C#N)C2 C(CCCCCNC(C1CCCCO1)=O)NC(CC1(CC(=O)OCC)CCCC1)=O c1(CC)nc(C)c(C(=O)NC(c2cccc(F)c2)CNC(=O)C(=O)C(C)C)o1 c1(N2CC(C(=O)NC(C(n3ncc(C)c3)C)=O)C2)nc2ccccc2s1 CCC(C)(C)CC(=O)NC1COCCN(C(c2nc(Cl)c(Cl)s2)=O)C1 C1(C(=O)OC)CCOC1C(=O)NCC1CC(F)(CNC(=O)C(c2cccnc2)C)C1 CCCC(C#N)C(=O)N(CCCC(=O)NCCC(O)CCO)C c1(C(N2CC(CNC(c3c(OC)nsc3)=O)C(C)C2)=O)ccc(F)cc1C CC1CN(C(c2coc(C(F)(F)F)c2)=O)CC1NC(C1(C)CCCN1C)=O c1(C(C(=O)NCCN(C(C(=Cc2cccs2)C)=O)CC2CC2)O)ccc(C)cn1 C=CCCN=C1NCC2CC(N1)C2.S(=O)(=O)(c1ccc(C)s1)NC(C)(CO)CC(C)C N1(C(CCc2cccc(OCC)c2)=O)CCC(CO)(NC(C2CC2(C)Br)=O)CC1 c1(N2CCC(OC)C(F)C2)nc(=NCC=C2CCSCC2)[nH]c2c1SCC2 C1(C(N(CCC)CCNC(=O)C(O)C(F)(F)F)=O)CC(c2ccccn2)=NO1 c1(CCN(CC=C)C(C2CS(=O)C2)=O)cccc(F)c1 N1(C(C2N(C)CC2)=O)CCC(C2(NC(c3scnc3Cl)=O)CCC2)CC1 CC1CCn2c(C(=O)N(C)CC3CCCN3C3CCN(CCF)C3=O)cnc2C1 C1(C(=O)NCC(C)NC(C2CC2C2CC2)=O)Cc2ccc(F)cc2O1 N1(C(c2[nH]c(=N)sc2)=O)CC2C(NC(=O)CNC(c3cccc(Cl)c3)=O)C2C1 N1(C(c2cn(C)nc2)C(=O)NCN2CC(N3CCCC3=O)C2)CCS(=N)(=O)CC1 c1(OC)ncccc1NC(=O)C(C1CC1)N(C)C(c1ocnc1C)=O c1(C(N(C)CC2CCCCN2C(C2CC2F)=O)=O)c(F)cncc1Cl C=CC(C)(O)CC(=O)NCCCCC(=O)NC(C)CCn1cncn1 N1(S(=O)(=O)c2c[nH]ccc2=NCC2OCCO2)CCc2ccc(F)c(F)c2C1 N1(C(c2ccc(COC)cc2)=O)CCN(C(=O)C(c2ccc(Cl)s2)=O)CC(O)C1 C1(C(=O)NC(CCOCC)C(=O)NC2CCN(CCF)C2)CC2CC(=O)C1O2 CCC(C)(CO)C(=O)NCC1CC(O)CN1C(c1nnsc1C(F)F)=O n1(CC=C)c(N2CCN(CCC#N)CC2)nnc1C1(C)OCCO1 C1(CN(C(=O)C(C2CCOCC2)O)CC)CCCN(C(=O)C(C)SC(F)(F)F)C1 C(=O)(C(C(C)C)n1cnnc1)N(C1CCN(c2snc(COC)n2)C1)CCO c1(C(=O)NC(C)CNC(=O)COCc2ccccc2)cnc2c(ccn2C)c1 c1(C(=O)NCCCCCNC(C2(C)CC3CC3C2)=O)csc2cccnc12 C1(CC=C)(NC(C2CC3(CC3)CO2)=O)CCN(C(=O)C(C(C)C)SC(C)C)CC1 C(CC)(C(=O)NCC1CC1CNC(c1cnsc1C)=O)=CCCC C(=O)(C1=NN(C2CC2)C(=O)CC1)NC(C1c2ccc(s2)N1C)=O.C1(CC)CC1 Cc1ccc(C(=O)N(C2CCCN(C(=O)C(C)OC3CCCC3)C2)C)nc1 C(=O)(C(C)(C)CCNC(=O)Cc1cccs1)NC(CCC)C(=O)NC N1(C(CCC2C(C)C2)=O)CC2CCC(C1)C(NC(C1CC1C1CCC1)=O)C2 c1(C(C)OC)nc(C)c(C(=O)NCC2CN(C(C3CCS3(=O)=O)=O)CC2O)s1 N1(C(c2nc(CCC)sc2)=O)CCCC2(NC(c3nc[nH]c3C(C)C)=O)CC2C1 C1(NC(c2c(CC)cno2)=O)COCCN(C(=O)C(C)(C(C)C)NC(C)=O)C1 Cc1cccc(CNC(C2CC(O)CN2C(c2cccc(Cl)c2C)=O)=O)c1C c1(C(N(CCNC(=O)C=Cc2nccs2)CC)=O)ccc(C)c(C)c1N c1(COC)c(C(c2nnnn2C2CCCC2)NCC2(CC)CCCC2)cccc1C C1(NC(C2CCCC3(CC3)C2)=O)CN(C(c2ncc(F)cn2)=O)CCC1CO n1(C(C)C)cc(C(=O)NCCC2CCCN(C(=O)C(C)(Cl)Cl)C2)c(Br)n1 C1(C(=O)NC(C#C)CC2CCCC2)C(O)CCN1C(=O)CCc1cccs1 N1(C(C(C)(C)OC(C)C)=O)CCOCC(C)(CNC(=O)CC(C)O)C1 CC1CN(C)CCC1N=c1[nH]c(N(C)CCN2CCCC2=O)nc2ccsc12 Cc1nn2ccccc2c1C(N1CCCC(OCCC(F)(F)F)C1)=O C1(NC(CCc2onc(CN(C)C)n2)=O)CC2CC1N(C(=O)C=C1CCCC1)C2 N1(c2ccnc(C(=O)OC)n2)CCCC(C2CC2NC(=O)C(C)(C)CSC)C1 c1(-n2c(-c3cnnn3C)nc(CCC)n2)ccc(CSC)cc1C N(C1CN(C(=O)C(C)CCCOC)Cc2ccccc21)C(C=CC)=O C=C=C(C)CC(=O)NCC1(C)CCCN1C(=O)COc1ccon1 N1(C(C(C)(C)SC)=O)CCN(C)C(C(=O)NCCC(F)(F)Cl)C1 c1(C(=O)NC(CCNC(C=Cc2c(C)ncs2)=O)C)cccc(C)c1N C1(C)(C(=O)NCC(C)N(C(=O)CC2CCOC2)CC)CCC(=O)N1 C(c1cc(OC)c(OC)cc1OC)=CCN(CC)Cc1nnc(C(C)C)n1C N1(C(C(C)C)=O)CCC2CCN(C(c3ccc4cnoc4c3)=O)CC2C1 CC1(C)C(NC(C2CCCC2(F)F)=O)CCN1C(=O)Cc1cccc(C2CC2)c1 c1(CC)ncc(C(N2CCC2C(=O)NC(CO)C2(C)CC2)=O)o1 N1(C(c2n(C)ncn2)=O)CCC2CCN(C(c3ccn4c3CSCC4)=O)CC2C1 c1(C(=O)NC2C(NC(C(c3c(C)nn(C)c3)C)=O)CCC2)cncc2c1CCC2 C1(C(=O)NC2CCCCN(C(c3ccc(CC)nc3)=O)C2)CCCCCS1(=O)=O n1(CC(=O)NC(CC2CCN(C(C=CC(CC)C)=O)CC2)C)nc(C)c(C)c1C Cc1cc(C(N2CCCC2C(C)NC(c2snnc2C2CC2)=O)=O)cc(Cl)c1 c1(NCCOCCN(C(=O)CC2(c3ccon3)CC2)C)ncnc2c1CCCC2 CC(C)(C)CCC(F)C(=O)N1CCCC(CC(=O)NOC2CCC(O)C2O)C1 c1(OC)ccc(C(N2CCCCC(NS(C)(=O)=O)C2)=O)cc1C(F)(F)F C1(CCC)(CO)CCCN1C(=O)C(CCSC)NC(c1cn(C)cc1C)=O N1(C(C(CCC2CCC2)NC(=O)C=Cc2ccco2)=O)CCCCC(CO)C1 c1(C(=O)NCC2N(C(C(C)=C(C)C)=O)CCOC2)cn(CC#N)c2ccccc12 C(C)(C(=O)N1CC2C(CNC(=O)C=CBr)C2C1)(C(C)C)NC(C)=O C12(CNC(C=CC)=O)CCC(C1)N(C(C1(CCN(C)C)CC1)=O)C2 C(=O)(C1=CC2C=CC1C2)NC(C=C)C(N1CC(O)CC1CO)=O CC1(CO)CN(C(C2CCCC2NCc2cc(Br)c(F)cc2O)=O)CCC1O c1(C(=O)NC2(COC)CCN(C(c3cncn3C)=O)C2)cc2cccc(C)c2o1 c1(OCC)nn(C)cc1C(=O)N(C1CCN(C(C2(n3cncn3)CC2)=O)C1)CC N1(C(C(C)(C)OC(C)C)=O)CCN(Cc2cnc(C3CC3)cn2)C2(CCC2)C1 C1(CN(C(C2(COC)CC2)=O)C)CCCN1C(=O)CC1(C)CCCO1 c1(C(=O)NCCCNC(C2(COC)C=CCC2)=O)cc(C)cc(Cl)c1 C1(C(=O)NCCNC(CCCC(=C)C)=O)C2Cc3cc(Cl)ccc3C12 CC(CN(C)C)CCC(=O)NCC(C)(C1CC1)NC(c1cnc(C(C)(C)C)o1)=O CCCC(C)(C)CC(=O)NCc1ccc(C(N2CCC(CNC3CC3)C2)=O)cn1 CC(F)(F)CCC(=O)NCC(F)CNC(=O)Cn1cc(F)ccc1=O C1(NC(C(C)NC=O)=O)CCCC(C(=O)NC2CCCC(O)C2)CC1 C(=O)(C(CC(C)C)NC(=O)Cc1cn(C)nc1C)NCc1ccc(CC)cc1 CC1C(=O)N(CC(=O)NC2(C)CN(C(c3cc(C(N)=O)cs3)=O)C2)C(=O)C1C c1(C(N2CCC(C#C)(C(N3CC4(CCCN4C)C3)=O)C2)=O)cc2ncccc2[nH]1 C1(CNC(CCCOCCC)=O)CC(F)(F)CN1C(=O)CCN1CCC(F)C1 Cc1ccc2c(C(=O)NC(CNC(c3cc(F)c[nH]3)=O)CC(F)(F)F)c[nH]c2c1 C1(NC(c2cc(CNC(C3(CC=C)CCC3)=O)on2)=O)CC(=O)N(C)C1 c1(OC)cncnc1C(=O)NC1CC(C(=O)NCCC=C(C)C)C1(C)C C(CNC(c1cn(C2CC2)nn1)=O)(C(C)C(C)C)NC(C1(OC)CC1)=O C(C(=O)NCCOCC)(C(C)C1CC1)N(C(c1ccc(F)cc1)C)CC N1(C(c2c(Cl)cn(C)n2)=O)CC(O)CC1(C)C(=O)NCC1(CF)CC1 C(=O)(C1=NOCC1)NC(C)C(c1ccccc1)NC(=O)COCCc1ccccc1 C1(NC(CSCCNC(c2cc(C)sc2)=O)=O)CCOC1(C)C c1(CC)ncsc1C(=O)NCC(C1CC1)N(C(=O)CC(C)C)C C(=O)(NNC(=O)c1cccc(-c2cccc(N)c2)c1)OC(C)C c1(C(N2C(C(=O)OC)CS(=O)(=O)CC2)=O)cc2c(s1)CN(C)CC2 C1(C(=O)NCCC2C(C)CN(C(c3cccc(CO)c3)=O)C2)CCCC12CCC2 C12(NC(CCC)=O)CCC(CNC(C34CC5CC(C3)CC(C)(C5)C4)=O)(CC1)OC2 c1(N(CCCOC(F)F)C)nc(N(CCCCN(C)C)C)nc2c1SCC2 C1(C(=O)NC2CCC(CC(=O)NCC(CO)N(C)C)C2)CC(C)(C)CCO1 N1(C(c2ccc(SC)cc2)C(=O)NCC=CC)CCCN(C)CC1C Cc1cc(C(=O)NC2CN(C(c3ccc(OC(F)F)nc3)=O)C3CC23)cc(Cl)c1 C(=O)(C1=C(Cl)CCC1)NC1CN(C(C2CC[Si](C)C2)=O)CC1CC1CC1 C1(C(=O)OC)CC2C(CC1C(=O)OCCc1ccc(O)c(C)c1)C2(F)F C(C(C(=O)NC1CC(F)(F)CC1NC(=O)C(F)C(C)C)C(C)(C)C)NC(C)=O N1(C(CNS(NC)(=O)=O)=O)CCC(CNC(C2CCC(C(F)(F)F)O2)=O)C12CC2 CCCC(CC(C)C)C(=O)NCC(CC(=O)NC1CCC(C)(C)CC1)OC C1(n2cc(-c3nc(C)sc3)nn2)C=CCC(C(=O)NC2CONC2=O)C1 N1(C(C=C(C)CNC(=O)COC(C)(C)C)=O)CCC(CCCO)C1 N1(C(C(CCC)OC)=O)CCCC12CCCN(C(c1c[nH]c(=N)o1)=O)C2 c1(C(N2CC(OCCNC(=O)CCn3cnnn3)C2)=O)cnc2ccnn2c1 c1(OC(C)C)cccc(CN=C(NCC(F)F)NC2CCOC2)c1.C(=O)NC c12cccc(c1)[nH]c(=O)oc1nc2cs1.c1(NC2CC2)ccccc1 C1(NC(CC(COC)NC(C2CCSCC2)=O)=O)CCN(C)C(=O)C1 C1(C(C)C)CC(C(=O)NC2CC(CN(C(=O)CN(C3CCCC3)C)C)C2)C1 C(=O)(C1CCc2scnc21)NCC1C2CN(C(C3OCCN(C)C3)=O)C1CCC2 C(C(=O)NOCC(O)CO)(C1C(C)CC1)C1CC1.C1(F)(C=O)CCOCC1 C1(C)(CNC(C2C(OC)CC2)=O)CN(C(c2cnc(N(C)C)cn2)=O)CC1C Cc1[nH]c(C#N)cc1C(N1CCC(OCC(=O)N(C(C)C(C)(C)N(C)C)C)C1)=O c1(-c2ccc(CN(C)Cc3ccc(OC)nn3)s2)ccc(OC)c(C)c1 S(=O)(=O)(c1cccc(N2CC3CC=CCC3C2)n1)NC(C1CCCOC1)COC CC1=CC(C(N2CCC2CC(=O)NCC=CBr)=O)SC1 Cc1cc(N2CCC(CC(N)=O)C2)nc(=NC(C)CCC(C)C)[nH]1.C(C(F)F)OC c1(C(N(C2CCCN(C(C(C=C)c3ccccc3)=O)C2)CC)=O)cncn(C)c1=O N1(C(C(Cc2ccco2)NC(=O)Cc2ccsn2)=O)CCC(F)(F)C(O)C1 CC1CN(C(c2nn(C(C)(C)C)cc2Cl)=O)CCN1C(C1CCCC(=O)O1)=O n1(CC(N2C(CCNC(=O)CC3(CO)CC3)COCC2)=O)ccc([N+](=O)[O-])n1 c1(C(=O)NCC2(F)CCN(C(C(CC)CC(F)F)=O)C2)nsc2ccc(C)cc12 Cc1nnc2n1CCC(C(=O)NCC1(C)CCCN1C(C1CC3(CC3)CO1)=O)C2 c1(C(=O)NC(C(C)(C)NC(CC(COC)(C)C)=O)C)cc2c(o1)CCCNC2=O C(C)(C)(CCC(=O)N1CC(C(=O)NC2C(C)C2C)C(C(C)C)C1)OC C1(C(N2CC(n3c(=N)nc[nH]3)C2)=O)CCCC2(CCN(C(=O)OC(C)(C)C)C2)O1 C1(OC)CCOC(CNC(=O)CCN(CCCO)C(=O)CC2CCCSC2)C1 c1(C(=O)NCC2N(C(CSC(C)C)=O)CC2)cncnc1C(C)C C1(NC(Cc2c(C)nc(S)s2)=O)C(C)CCN(c2ncnc(Cl)c2C#N)C1C CCC(C)CCCC(=O)N1CCCC(C)C1CNC(=O)CCc1ccncn1 CC1(CNC(=O)C(C)(C)c2ccccn2)CC(NC(=O)CNS(N)(=O)=O)C1 N1(C2(C)CC(NC(c3cc(C(N)=O)sc3)=O)C2)CCS(=O)CC1.C1(C(=O)N)(CCC)CC1 S(=O)(=O)(c1cccc(Br)c1F)N1CCCC(C(C)NC(c2cccc(CO)n2)=O)C1 C1(C(=O)NC(c2cccc(Cl)c2)C)CC12CCN(C(c1cc(Cl)ccc1O)=O)C2 c1(C(=O)NCC(CC)(C)NC(=O)C(C)CCN(C)C)cnc(O)c2cccnc12 N1(C(C2(NC(C(CC=C)CC)=O)CC(CO)C2)=O)CC(=O)NC(C)(C)C1 C12(COC)COC(C(=O)O)(CN1C(c1occc1-c1ccc(Br)cc1)=O)C2 C1(CCC)CN(C(=O)CCOC(C)C)CCN1C(=O)CCc1ccc(F)c(Cl)c1 c1(CN2CC(NS(=O)(=O)CCCCl)C(F)C2)c(Br)ccc(Cl)c1Cl C12(C(=O)NC3C(O)CCN(C)C3)CC(CCO1)N(C(=O)CCc1cccn1C)C2 Cc1nc2ccccn2c1NC(C1(O)CCN(c2ncnc3ccccc23)C1)=O CCCCC(C(=O)NC1CC2(C(=O)N(CC(C)CO)C)COC1C2)N(C)C N1(CC(=O)NCC2CCC(C(=O)NC3CCCCC3CO)C2)C(=O)CNC1=O CC(C)(C)CCCC(=O)N1CCC(Cn2cc(-c3cnccn3)nn2)C1 CC1(NC(c2cnc(-c3ccccc3)nc2)=O)CCCN(C(c2cocn2)=O)C1 c1(C(=O)OCC)cc(C)nnc1N1CC2C(NC(=O)Cn3nccn3)C2C1 c1(OC)ccc(F)c(C(N2CCC(CCNC(c3c[nH]cc(Cl)c3=O)=O)C2)=O)c1 C1(C(=O)NCC(C2CCC(=O)N2)C)CC2CCC(C1)N2C(=O)C#CC1CCCC1 Nc1cc(C(=O)NC2CC(NC(=O)CCOC3CCCCC3)C2)cc(F)c1 c1(C(=O)NCC2CC(NC(C(C)SC)=O)C2)ccc2cc[nH]c2c1 Cc1cc2c(C(=O)NC3(C)CC(NC(C4CC4c4cccs4)=O)C3)cccc2[nH]1 S(=O)(=O)(c1ccc(NC2(c3ccc(F)cn3)CC2)c(F)c1)NC1C(C)CCCC1 c1(OC)cc(Br)ccc1C(=O)C(=O)NCC1CN(C(=O)CCC2CCC2)C1 Cc1cc(C(=O)NC2(CNC(C3C4CC5C(C4)C35)=O)CCC2)sc1C c1(C(N(CCCNC(=O)CCOC2CCOCC2)C)=O)c[nH]c2cc(F)ccc12 C1(C(=O)NCC2N(C(c3nccc(N(C)C)c3)=O)CCC2)CC(C(C)(C)C)=NO1 CCCC(C)(CC)C(=O)NCCCCN(C(=O)CC(C)N1CCCC1=O)C N1(C(C(C)N(C(C)=O)C)=O)CCOCC(F)(CNC(c2nn(C)cc2SC)=O)C1 N1(C(C(CC=C)CC)=O)CCC2CN(C(=O)CN(C)C(=O)OCC)CCC12 c1(C(N(C(C)CNC(=O)CCCCSC)CC)=O)cccn2nccc12 N1(C(CCn2c(C)ncc2)=O)CCC2CCC(C1)N2C(c1ncoc1C(C)C)=O c1(C(=O)NC2C(C)N(C(=O)Cc3cncc(C#N)c3)CC2)cc(O)cc(O)n1 CC1CCN(c2ncnc(N3CCN(CCO)CC3)c2C)CCS1 C1(CC=C)(NC(CCC#C)=O)CCN(C(=O)C(c2c(C)noc2C)C)C1 C1(C(=O)NCCCC2CCCN2C(C=CC(=O)OCC)=O)CC12CCCCC2 C1(NC(CC(CC)(F)F)=O)CCC(O)CN(C(c2ccn(CC)n2)=O)C1 N1(C(Cn2cc(C(=O)NC)nn2)=O)CC2(C1)CN(C(=O)C(F)C(F)(F)F)C2 c1(C(N(CC)CC2(F)CCC2)=O)c(C)ccn1C N1(C2CCC(=O)NC2=O)CCC2CC(C(=O)NC3(c4cccc(F)c4)CC3)C2C1 Cc1ccc(C2CC2C(N2CC(N(C(=O)C(C)(C)c3cscn3)CCO)C2)=O)o1 C1(c2n(CCOCC)nnn2)(NC(C2(C)COC2)C)CCC(SC)C1 S(=O)(=O)(c1cccc2ccncc12)NCC(C(CC)CC)O N1(C(=O)CSCc2ccncc2)CC2(CC(NC(=O)C3=CCCCCC3)CO2)C1 C1(C)(C(=O)N(C2CCC2)CC2(CN(C)C(C3CC(=C4CC4)C3)=O)CC2)CCCC1O Cc1cc(F)sc1C(=O)NCC(C1CCOC1)NC(c1ccncc1N)=O c1(-c2n(C(CC)C3CCC3)nc(C(CC)CC)n2)cccc2ccncc12.CCO C1(CC)CCCCC1C(=O)N(C)CCOCCN(C)C(c1cc(F)n(C)n1)=O N1(C(C(CSC)C)=O)CCC2CCN(C(C3CCC(C)CC3)=O)CC2C1 C=CC1(CC(=O)NC2CCCC(CNC(c3cscc3C)=O)C2)CCCCC1 N1(C(c2cccc(OC(C)C)c2N)=O)CC2CC(C1)N(C(=O)C(C)CC1CC1)C2 Cc1c(C=CC(=O)NC2CCN(C(=O)C(C)S(N)(=O)=O)C2)cnn1C CN1CCC(C(=O)NCCc2ocnc2CNC(C2CNC(=O)C2)=O)C1 CCC(CC(=O)NCC1(NC(=O)C(C)(CC)OC)CCC1)C(C)C CN=c1[nH]cc(C(=O)NCC(C)O)s1.N12CCCC1(C)C2=O C1(N(C(=O)CCc2ccon2)CC)CCCN(C(=O)CCn2nc(C)cc2C)C1 C1(C(N2C(C(N(CC(C)O)C(C)C)=O)CC3CC32)=O)CCCC12CCC2 C1(CC(=O)NC(C(N2CC(C(=O)OC)C2)=O)C)CCCCC1C(F)(F)F N1(C(C2CC(OCC)C2)=O)CC(CNC(=O)CC2CC(C)OC2C)CC12CCC2 c1(C(=O)NC2CC3(CC(CNC(COCC#N)=O)C3)C2)occ2c1CCOC2 c1(COC)cc[nH]c1C(=O)NC(C)(C)C(=O)Nc1cccnc1 c1(C(N2CC(C(=O)NCCCOC)NCC2)=O)ccc2c(Br)nn(C)c2c1 C(=O)(C1=NN2CCCN=C2N1)NCC(C)NC(c1cnc(CF)s1)=O CC#CC1CN(C(=O)CN(C(=O)Cc2ccc(C)o2)C(C)C)C1 Cc1cc2[nH]c(C(=O)NC(C)CN(C)C(C3CCCC(O)C3)=O)cc2o1 c1(NC(C2CCN(CCN3C(=O)CN(C)C3=O)C2)=O)cc(Cl)c([N+](=O)[O-])cc1O C1(C(N(C)Cc2scc(C)n2)=O)CC2CN(C(c3c[nH]nc3C3CC3)=O)CC2C1 Cn1c(CN(C2CCCC2)CCNC(C(=O)NC)=O)c(OC2CC2)sc1=O.C1CC1 c1(C(N2CCC(C(C(=O)N(CC(C)O)CC(C)O)(C)C)C2)=O)cncc(F)c1 c1(C(N(C2CCN(C(=O)CCCOC)C2)CC)=O)cc2ncn(C)c2cn1 CC1CC2(CCN(C(C3(C)CCN(C)C3=O)=O)CC2)CN1C(c1nc(Cl)cs1)=O Cc1nn(C)c(C(N2CCCC2c2cnn(C)c2)C(=O)NCC2CCCO2)c1Cl c1(OCC)cc(Cl)ccc1C(N1CC2C(NC(=O)C(COC)NC(C)=O)C2C1)=O C(=O)(CCC1=NNC(=O)CC1)NC1CC(CNC(C2(C)C(C)C2)=O)C1 C(=O)(CC(C(F)(F)F)NC(c1ncc(F)cc1N)=O)N1CC(C#C)(N(C)C)C1 C1(C(=O)NC(CCO)C2CCCC2)C=CCN1C(c1cnsc1)=O N1(C(C2CCC(=O)N2)=O)CCCC(NCc2ncsc2Br)C1 C=CCCC(C(=O)NC1(C(=O)NC)CC1)NC(C1CCCC(=O)C1)=O CCCCC(CC)C(=O)NCc1ccc(C(=O)N(C)CCN2CCCC2)o1 C1(O)(C(=O)NCC(C)NC(c2cccc(C(N)=O)n2)=O)CCOC1(C)C N1(C(c2cnc(C)nc2O)=O)CCCC2(NC(c3cccs3)=O)CCCC12 C(=O)(C(C)C(C)NC(c1sncc1C)=O)NCC=CCCOC N1(C(C(C)C2CC2)=O)CCCC(C)(C(=O)NCc2c(C(F)(F)F)cccc2O)C1 c1(C(N(C2C3CN(C(=O)CCNS(C)(=O)=O)CC23)C)=O)nccnc1Cl c1(COC(C)(C)C)cccc(C(=O)NCC(F)CNC(C2CC2C(F)F)=O)c1N C1(C(=O)NC2C=CC(C(=O)NCCSC(F)F)C2)CC2CCC(C1)O2 n1(CC(N2C(C)CC(CNC(C3CC(F)(F)C3)=O)C2)=O)ncc2cccnc12 Cc1cn(C(C)(C)C(=O)N2CC(N(C(=O)CCOC3CCOC3)C)C2)cn1 c1(OC)ccc(NC(C2CCCN(S(=O)(=O)CCCCl)C2)=O)cc1Br C1(C)(C(N2CC(NC(N(CC(c3ccccc3)O)C)=O)C2)=O)CC1(F)F c12ccc(cc1)C(=O)NCCC1CCCC1CNC(=O)COCC2.COC C1(CNC(CSC)=O)CCC2(CN(C(=O)CCOc3ccccc3C)C2)O1 Nc1cc(Cl)nc(C(=O)NC2CCN(C(c3nn(C(F)F)cc3Cl)=O)CC2)c1Cl C1N=C2NC(=CS2)C(=O)N2CCOC1C2.c1(CC)ccc(OCC(F)(F)F)cc1 N1(C(C2N(C)C(=O)NC2)=O)CCCC2(C1)CN(C(=O)C(c1cncn1C)O)C2 Cc1ccc(CC(=O)NC(C2CCOC2)CNC(=O)C=CC(CC(F)(F)F)=O)o1 C(CCCn1cc(C(C)(O)Cc2ccccc2)nn1)NC(C1(C)C(C)C1)=O C12(C(=O)NCC3CCC(C)CO3)CC(CN(C(=O)C(C)(C)CO)C1)C2 C=CC1(C(=O)NC2(CCNC(C3CCCN3CC(C)C)=O)CCC2)CCOCC1 c1(C(=O)NCCNC(C2=NOC(C)C2C)=O)c(F)ccc(F)c1Br c1(CC)ncc(C(=O)N(C(CNC(=O)Cc2cn[nH]c2)C2CC2)C)o1 C1(COC)(NC(C2CC=CC2)=O)CCCN(C(=O)C(C2CCOCC2)F)C1 Cc1cc(NC(C2(NC(=O)C(C)C(F)F)CCC(C)(C)C2)=O)cc(O)c1 C=CC(C)(C)C(=O)NC(CNC(=O)Cc1cc(-c2ccco2)on1)CC N1(C(c2ccc(NC)cn2)=O)CCCC(NC(c2cn(C(C)C)nn2)=O)CC1 C1(NC(C2C(C)OCCO2)=O)C2CC1CN(C(=O)COc1cc(Cl)ccc1Cl)C2 N1(C(c2cnc(C(C)=O)s2)=O)CCCC2C1CCN2C(=O)Cn1nc(C)oc1=O C12(C(N3CC(CC(C)C)OCC3)=O)C(NC(c3ccc[nH]3)=O)C3CC1C2C3 c1(C(=O)NOC2CC2)ncoc1CO.c1(C(=O)NCC2CCCCC2)ccc(CO)o1 O=C(Cn1cc(C2C3COCC23)nn1)NNC(=O)NC1OCCC1F c1(SC(C)C(c2ccc(Br)cc2)=O)ccc(F)cc1.C1CC(=O)N1 C(CC(=O)N1OC2C=CC1CC2)(C1CC1)NC(C(C(CC)(C)C)O)=O CC1CN(C(=O)CCCc2cccc(Cl)c2)CC(C)N(C(=O)CNS(C)(=O)=O)C1 N1(C(c2ccc(OC)o2)=O)CCCC2(CCCCC2NC(c2oncc2C)=O)C1 c1(C2(C(=O)NCC3CN(C(C4CCC(C)O4)=O)C3)CCC2)ccccc1Cl C1(NC(Cc2cnc(C)s2)=O)CCC2CC1CN2C(C1CCN2CCOCC12)=O C(=O)(C(F)(F)CCn1ccnn1)NC1CN(C(c2cc(CSCC)ncc2)=O)C1 C(=O)(C(O)CC(C)(C)C)NC(CNC(c1cnc(CCC)s1)=O)CC N1(C(C2C(C(C)(F)F)C2)=O)CCC2C(C1)NC(=O)N2C1CCN(C2CCC2)CC1 c1(CC(=O)NC2CC23CC(NC(C2(O)CC2)=O)C3)c[nH]ccc1=O c1(C(C(=O)NCCCSC)N(C)CC2CCOC2(C)C)sc(Br)cc1C C12(CC)COC(C(=O)NCCOC3CCN(C(C(C)C4CCC4)=O)C3)(C1)C2.C(CF)O CC(C)(CC1CC1)C(=O)NCC1C2CC2CN1C(=O)COC(F)F.c1ccccc1 C1(C(=O)NC2CC(NC(C3CN(C(C)C)C(=O)C3)=O)CC2O)OCCN(C)C1=O C1(NC(C2CC(O)(CC#C)C2)=O)CCN(C(c2sc(C(C)C)nc2C)=O)CC1F C1(C(=O)NCC(CNC(c2nnn(C(C)(C)C)n2)=O)OC)(CC)CC(=O)C1 N1(C(=O)C(O)CC2CC2)CC2CC1CN2C(c1cc(-c2cccc(F)c2)on1)=O C(CCCCCC(=O)N1CCC(O)(CN(C(=O)CN2CCC(C)(C)C2)C)C1)SC N1(C(C(CCOC)(C)C)=O)CCN(C(C23CCC(CC2)C3(C)C)=O)CC(O)C1 c1(C(C)C(=O)NCc2nc(-c3ccco3)n[nH]2)ccc(F)cc1F Cc1cc(C(CO)N(c2ccc(COCC3CCCO3)cc2Br)C2CC2)ccc1Cl C(N=c1ccnc(N2CCOCC(C)C2)[nH]1)C1N(CC)CCC1 C1(N(C(C(N2CC(C)C2)C)=O)C)CCCN(C(c2nn[nH]c2Cl)=O)CC1 Cc1cc(C(=O)NCC2(C)CCCN2C(C2CC(F)(F)CS2)=O)cn(C)c1=O C(C(CO)CC(C)(C)C)NC(C1CCN(S(CC(C)C)(=O)=O)CC1)=O C1(NC(C2C(C(=O)NCC#C)C2)=O)CCN(C(=O)CC2=CCCC2)CC12CCC2 C1(CC(=O)NC2CC2NC(=O)CC2(O)CCOC2)CCN(C2CCC2)CC1 CC1(C)CN(C(C2CCOCC23CCC3)=O)CC(CNC(=O)CN2CC=CC2)O1 c1(C(NOCC(=O)N(CCCSC)C)=O)cc(C)c(C)nn1 S(=O)(=O)(c1ccc(C)c(C(=O)NCCOc2cccc(Br)c2)c1)NCC C1(NC(c2cc(C(N)=O)[nH]c2)=O)CCCC(NC(=O)C2=CCC2)C1 N1(C(c2ncccc2CO)=O)CCCC(N=c2nn[nH]n2Cc2ccccc2)C1 C12(C(=O)NCCN(C(=O)Cc3ccc(C)o3)CC)CCCCC1OCC2 C(C(C(=O)N(C)CC1CC1(C)C)N(C)C)NC(C(C1CCC1)OC)=O C1(NC(c2cnc(C(F)(F)F)s2)=O)C2CC1CN(C(C1CC3C(C1)C3(F)F)=O)C2 C(=O)(N=c1ccn(CCOC)[nH]1)C1C(NC(=O)Cc2cncnc2O)CC1 C(=O)(CCCC(F)(F)F)NC(C(=O)NCCC(C)(C)C(F)F)CO O=S(=O)(c1cccnc1NCCCC1CC1(Cl)Cl)NCCN1CCSCC1 C(CCCCC(=O)NC1CCN(C(c2cccc(C#N)n2)=O)CC1F)N(C)C N=c1[nH]c(C2CC2)ncc1C(N1CC=CC1CNC(=O)CCC1CCOC1)=O N1(C(CCC=CCC=C)=O)CCCCC(CNC(=O)Cc2cc(Cl)sc2Cl)C1 CCC(C)CCCCC(=O)N1CCOCC(C(N2CCC23CCSCC3)=O)C1 N1(C(C23N(C(c4c(N)cncn4)=O)CCC2C3)=O)CC2(CCC1CO)CC2 N1(C(C2C(OC)CCCC2)=O)CC2CCC(C1)N2C(C1CC(C#N)C1)=O C=C(C)CC(C(=O)Nc1ccc(C(=O)NC2CCCC2)cc1CC)OC C12(CNC(CC)=O)CN(C(c3cn(-c4cnn(C)c4)cn3)=O)CC1CCO2 CC1C(NC(C2(C3CCCO3)CCC2)=O)CCN1C(=O)CC1CCCC(=O)N1 CC(C)CC(C(=O)N1CCOCC1)NC(=O)OC(C1(C(F)(F)F)CCC1)C1CC1 C(=O)(CC(C)(C)C(=O)NC1(CN(C)C(C2CC(OC)C2)=O)CC1)OC C1(C(=O)OC)CNC(=O)CN1CCNC(C1CC1C(F)(F)F)=O Cn1ccc(C(=O)NCC2(CCCNC(=O)CC3CCOC3=O)CCCC2)n1 CCC(COC)(CC)C(=O)N1CCC(C)C(NC(=O)C(CC)C(C)(F)F)C1 O=C(C1=CCCCCC1)N1CC2(CCN2C(c2ccc(Br)c(Cl)c2Cl)=O)C1 c1(NC)ccc(F)c(C(=O)NCCC(C)(C)NC(C2CCCCC2C2CC2)=O)c1 CCCCCC(O)C(=O)N1CC(NC(=O)CCc2cnc(C)o2)CC(F)C1 CC1C2CCCCC2CN1C(=O)COCC(=O)NOCCCC1(C)CC1 Fc1ccccc1CNC(=NCC1CC1(Cl)Cl)NC1CCOCC1 c1(CN2CCN(C(C3N(C)C(=O)CC3)=O)C3C2C3)c[nH]c2cc(C#N)ccc12 N1(C(c2cc(CC)no2)=O)CC(C(=O)NCC(C)N(C)C)C2(CC2)C1 C(N=c1[nH]c(NC2CCOC2C)nc(=N)[nH]1)c1cn(-c2ccc(OC)cc2)nn1 N1(C(C#CC(CNC(C(CC=CCC)C)=O)(C)C)=O)CCC2(CC1)CN(C)C2 C1(CNC(C2CCCN(CC)C2)=O)CN(C)CCN1C(C1OCCO1)=O C1(C(=O)NC2CCN(C(=O)C=C(Cl)Cl)CC2CO)Cc2ccccc2CO1 N1(C(c2c(C)scn2)=O)CC2CC(C(=O)NCC(C)(C)C(C)C)CC2C1 c1(CCOC(C2CCCN(CC(=O)OC(C)(C)C)C2)=O)coc2c1CNC2 Cc1cnc(C)c(C(N2CCCC2CN(C)Cc2ccc(Br)[nH]2)=O)n1 CC1(C(N2CCCC(OCc3ccccc3)C2)=O)CC2CC2C1 C1(OCC)CC2(C1)CC2C(=O)N(C(C)CNC(=O)CCCN1CCCC1)C1CC1 C(=O)(CN=S(C)(C)=O)NCC1CC(OC)CN1C(C1CCCCC1C(N)=O)=O N1(C(C=CC(CC)C)=O)CCC(CN(C(=O)CN2CCCNC2=O)C)CC1 N1(C(C(C(C)C)F)=O)CCCN(C(=O)CC2CC2)CC1C C(C(C)(C)C(=O)NC1(O)CC(NC(c2ccc(N3CCNC3=O)cc2)=O)C1)OC C1(NC(CCOCCOCC)=O)CCCCCN(C(=O)C2=CCCC2C)C1 Cc1[nH]ccc1C(=O)NC(C(=O)N(C)Cc1cccnc1)C1CCCO1 C1(C(=O)NCCCC(=O)NC)CN(C(=O)C(C)O)CC1C CCCCC(O)C(=O)NC(C)(C)CNC(c1cc(C(F)F)cs1)=O CC1(C)CCC(CC(=O)NOCC(N2CCC(C3CCCC3)CC2)=O)C1 c1(NC(C2C3CN(C(CS(CC)=O)=O)CC32)=O)cn2c(n1)CC(OC)CC2 C1(CC#N)CN(C(c2cc(Br)sn2)=O)CCN1C(=O)C1=C(Cl)CCC1 c1(C(=O)NC(CCN(C(C(CCC)C)=O)C2CC2)C(C)C)c(C)oc(C)c1C C1(C(N2CC(OCCNC(C(C3CC3)SC)=O)C2)=O)CC2CC1CC2(F)F C(=O)(CC(C)CC(F)(F)F)NCC1(CNC(C(C2CC2)OCC)=O)CC1 N1(C(C2C(C)C3CCC2C3)=O)Cc2occ(C(N3CCC(C)C3CO)=O)c2C1 c1(C(N2CC(C)C(NC(=O)C(N)=O)C2)=O)oc2ccccc2c1C(=O)OC(C)(C)C C(C1CN(C(c2ccon2)=O)CC1C(=O)NCc1ccnc(OC)c1)=CC Cc1ccc(C(N2CC3CCC3(CCNC(=O)CN=S(C)(C)=O)C2)=O)c(CO)n1 N(C(=NCCSCc1nnc(C)s1)NCC(C)C)Cc1c(CC)nccn1 C(=O)(CC(C)CNC(c1cnc(C2CC2)o1)=O)NC1(CCCC)CC1 Cc1nn(C)c(C)c1CC(N1CCC(NC(c2cccc(=O)o2)=O)C(O)C1)=O C1(C(=O)OC)COC2(CCC2)CN1C(=O)Nc1[nH]nc(CO)c1C(F)(F)F Cc1ncc(CCC(=O)N(C(=O)C(O)C2CC2)Cc2ccco2)s1 C12(CNC(c3cnc(S)[nH]3)=O)CCCC1CCN2C(c1coc(C(F)(F)F)c1)=O N1(C(c2c(C(C)C)scn2)=O)CC(CNC(C2CCC(=O)NC2)=O)C(C)(C)C1 c1(CCO)ccc(NNC(=O)N=c2[nH]nc(C(C)(C)C)s2)cc1F CC1(C)CN(C(C2CC2C2CCC2)=O)CC1CC(=O)N(CCCO)CCO c1(CNC(C(=O)N(C2CCC2)C(C)C)=O)ccc2nc(O)ccc2c1 c1(C(N(C2CCN(C(=O)C=C3CCOCC3)C2)CCC)=O)ccn2c1CSCC2 c1(C(=O)NC(CCNC(CCCNC(C)=O)=O)C)ncn2c1CCC2 C1(N(C(CCC)=O)C)CCCCN(C(C)CNC(C)=O)C1 N(C(=NCCCC1CCC1)NCC1CC1)CC(c1c(C)nn(C)c1C)O CC(CC(=O)NC1CC1CNC(=O)CC1CC(C)(C)C1)C(C)(C)C N1(C(C(CC)n2cccn2)=O)CCC(C(CO)NC(=O)CN(C)CC)CC1 C12(CC=C)CCCN(C1)C(=O)CC(=O)O2.C(=O)(C(C)CC)NCC(C=C)O N1(C(C(C2CN(C(=O)CC3CC=CCC3)C2)OC)=O)CCCOCC1C c1(Cc2cn(C)nc2)cc(-c2nc(C3COCCO3)no2)ccn1 c1(C(=O)NC(C2CCN(C(C3CC(OC)C3)=O)C2)C)ccc2ncn(C)c2n1 CC(C)(CNC(c1cnc(S)nc1)=O)CC(=O)NCC1(O)CC1 Cc1cccc(CN(CCc2ccccc2)C(C2CCN(C)C2=O)=O)c1 C(C(C)(C)CC(C)C)N(CC(N1CC(F)CC1CO)=O)C(c1nc(C(C)=O)oc1)=O C1(C(=O)N(C)OC)(NC(CC2CC(CC)C2)=O)CC1(C)C CCC(CC(F)F)C(=O)NCCCCNC(=O)CCc1ccc[nH]1 c1(-n2cc(C3N(C(C4C(OC)CCC4)=O)CCC3)nn2)nc(C)c(C)n1C C(=O)(C1CCCn2cncc21)NC1(CNC(c2c(C)noc2C2CC2)=O)CCC1 CN1CC2CCN(C(C34CCC3CN(C(c3cnccn3)=O)C4)=O)C2C1 Cc1ccncc1C(N1CCC(OCCNC(=O)C(O)C2CC2)C1)=O C1(NC(c2cnc[nH]2)=O)C=CCN(C(C2(C(F)(F)F)CCOCC2)=O)C1 CCCC(CCC)=CC(=O)N(CC(=O)N(C)CC1CCOC1C)C1CC1 c1(SC)cc(C(=O)NC(C)(CNC(=O)C(C)(O)c2ccccc2)C(C)C)c(C)o1 C(=O)(C(CCCC)NC(=O)CCOCC)NC(CCCC)COC CCC(CCC(=O)NC(c1cnc[nH]1)(C)C)NC(=O)C(F)n1ccnc1 C1(NC(Cc2cn(C)nc2)=O)COC2C(NC(c3cnc(O)nc3O)=O)COC12 c1(-c2n(C(CC)C)nc(-c3ccc(C(F)F)cc3)n2)ccnc(OC)c1Br C1(CC)CN(C(c2sc(-c3ccccc3)cc2Br)=O)CC(=O)N1 N1(C(Cn2c(C)cc(O)cc2=O)=O)CC2(C)CN(C(=O)C=CCF)CC2(C)C1 C1(CCNC(c2ccc(CCC)cc2)=O)CC(F)(F)CN1C(=O)CCCN(C)C C(=O)(C(C)CN(C)CC)NCC1C(NC(COCCCC#C)=O)C1 c1(CC(N2CCOCC2CNC(C2(F)CC=CCC2)=O)=O)ccc(OC(F)F)cc1 N1(C(CC(C)OC)=O)CCOc2ccccc2C1CO Cc1ccc2[nH]nc(C(=O)NC3CN(C(c4cccc(C)c4)=O)CC3F)c2c1 C=CC1(C(N2CC3CC(F)CC3C2)=O)CCN(C(=O)CCc2ncccn2)CC1 C(CC(=O)NCCc1cc(C)ns1)(C(C)C)NC(c1c(C)n[nH]c1)=O c1(OC)ccc(C)cc1C(C)NCC1CCN1c1cnc(C(=O)OC)cn1 c1(CNC(C2(CC)CCC2)=O)ccnc(C(=O)NCC2CC2C(F)(F)F)n1 C1(C(=O)NCC2N(C(C)=O)CCC2)CC2CC1CC2NC(c1cn(C)ccc1=O)=O C1(C2CN(C(c3ccnc(C4CCC4)c3)=O)C2)(NC(c2c(C)[nH]cc2)=O)CC1 C(=O)(CC(C)OCCN(C)C)NCC=CC(=O)N(CC(=O)OC)C CCC(N=c1[nH]nc(C(C)C)o1)c1ccc(Sc2nccc(C)n2)cc1 N1(C(C2CN(C)CC2C(F)(F)F)=O)CCCC(CO)(NC(=O)C2=NOCC2)C1 C1(OC)CCC2(CCC2)C1NC(=O)C(Cc1cccc(Br)c1)c1nc[nH]n1 C(C(C)C)(C(O)C(=O)N(C1CC(NC(=O)C(C)Nc2cccnc2)C1)C)OC Cc1cnc(C(N2CCC(C3CCCN3C(=O)C(F)C3CCC3)CC2)=O)cn1 CCCC(C)(C)CC(=O)Nc1cncnc1C(C)(C)C N1(C(C(C)O)=O)CC(CNC(c2c[nH]ccc2=O)=O)C(C(F)(F)F)C1 N1(C(C=CC(=O)OC(C)(C)C)=O)CCC(NC(c2ccc(C(N)=O)s2)=O)C12CC2 Cc1ccc(C)n1Cc1cn(-c2ccncc2)nn1.C(CC=O)NCC(=O)OC C(=O)(CC(C)C(C)(C)C)N1CC(CC=C)(NC(C23CC(C)C2C3)=O)C1 c1(C(N2C(CCNC(C(C)c3cc[nH]n3)=O)CSCC2)=O)cccc(Cl)c1N Cc1cccc(Cl)c1-n1cc(C2CCN(C(c3cccc4nsnc34)=O)C2)nn1 N1(C(CCc2cc(C)no2)=O)CC2(CCC2NC(C2CCC(=O)N2C)=O)C1 C1(C)(NC(CCC(C)C)=O)CCN(C(c2c[nH]cc2Cc2ccccc2)=O)CC1 c1(C(=O)NC2CC(CNC(C3C(C)C3C)=O)C2)cc(Cl)no1 Cc1nc(CO)sc1C(=O)NCC(C1CCN(C(C2(C)COC(=O)N2)=O)CC1)F c1(C(=O)NC(CNC(CNC(CC)=O)=O)CO)nc2ccccc2nc1C C1(NC(CCn2ccc(C)n2)=O)CN(C(=O)CC(C)n2cccc2)CC(F)(F)C1 O=C(Cc1cccs1)C(=O)N1CC(CNC(C2CCC2c2nc[nH]n2)=O)C1 c1(C(=O)NC2C(CNC(CC)=O)COC2)sc(Br)c(C)c1C c1(C(=O)NC(CN(C(C2CC2(Cl)Cl)=O)CC)C)ncc(C(F)(F)F)cc1Cl c1(C(n2c3c(n(C)c2=O)ccc(Br)c3)=O)ccc2cc(S(N)(=O)=O)ccc2c1 C1(C(=O)NCC(C)NC(c2c(Cl)ccc(C)c2)=O)Cc2ccc(Cl)cc2C(=O)O1 c1(C(=O)NC(C)C(C)NC(c2cnnn2C2CC2)=O)cc(Cl)cc2cccnc12 C1(C(=O)NC(C2(O)CN(C(C(CCCC)O)=O)C2)C)CN2CCN1C(C)C2 C=CC(C)(C)CC(=O)NC1CN(C(c2ccc(=O)oc2)=O)CC1CC c1(C(NOC(C)C(=O)O)=O)ccc(=O)n(CC(F)(F)F)c1.c1(OCC)ccc(F)c(Br)c1 C1(NC(C(CC)c2ccccc2)=O)CN(C(=O)Cn2cnnn2)C(CC)(CC)C1 N1(C(C=Cc2cccc(N)c2)=O)CC2CCC(NC(=O)CC3=CCCC3)CC2C1 C(C(C)(C)C(=O)NCC1CCC(C(=O)Nc2nc(C)sc2C)C1)SC C(=O)(CCS(C)(=O)=O)O.C12(C(C)N(C3(C)CC3)C(=O)OC(C)(C)C)COC(C1)C2 n1(CC)nc(C(N2CCCC2C(C)(C)CNC(C2(C3CC3)CC2)=O)=O)cc1O Cc1ccc(CC(=O)NC(C)CNC(=O)C(=Cc2cccc(F)c2)F)cc1C#N c1(C(=O)NCC2C(OC)CC2)ccc(-c2nn[nH]n2)cc1 c1(C(=O)NC(C)CC2CN(C(=O)C(C)N(C)C)C2)ccc(Cl)c(F)c1N CC(C(=O)NC(c1cc(F)cc(Cl)c1)CNC(C1(CC#N)COC1)=O)S(C)(=O)=O c12noc(n1)CC1C(CCC1)NC2=O.c1(SC)cn(C2CC(O)C2)nn1 CC(CCCCNC(=O)C(C)(O)c1ccccc1)NC(=O)C(C)(C)CO N1(CC(=O)Nc2ccc(CCNC(C)=O)cc2)C23CCCC2(C1)C(N)C(O)C3 C(CCCC(=O)NC1CCOC(CNC(c2c(Cl)n[nH]c2C)=O)C1)OC c1(OC)ccc(C(N2CCC(NC(=O)CC3CCCN3)CC2)=O)cc1N n1(-c2cccc(OC)c2)c(C)cc(C(=O)NC2CN(C(=O)C=C3CC3)C2)c1C C1(NC(CCCOCC)=O)CC2CC(NC(=O)COCP(C)(C)=O)CC12 CN1C(=O)CCC1CC(=O)NC1CCC(NC(C2CCNC2=O)=O)CC1 Cc1c(C2(CNC(=O)CC=C(Cl)Cl)CC2)cccc1F.N12CCCC1C1(CC1)C2=O CC(C)(CC1(C2(c3cn(Cc4ccccn4)nn3)CCCCC2)CCC1)S(C)(=O)=O N1(C(=O)C2CC2)CC2CCCCC2C1.c1(O)ccnc(-c2ccco2)n1 C(CC(CC)C(=O)NCC12CC(CO1)N(C(C1(N)CCC1)=O)C2)=CC.C(N)=O c1(CC)[nH]ccc1C(=O)NC12CC(NC(C3CC(C)CO3)=O)(C1)C2 c1(CC(N2CC=C(CNC(C=COCC)=O)CC2)=O)coc2cc(OC)ccc12 c1(CNC(c2cccc(OC(C)C)c2)C)c(OC)cccc1O c1(C(C(=O)N(C2CCCN(C(C(C(C)C)O)=O)C2)C)O)ccc(Cl)c(Cl)c1 Cc1nsc(C(=O)NCCCCNC(C2(C)CC2(F)Cl)=O)c1Br C1(C(=O)NCc2c[nH]c(=N)s2)CCCC2CCNCC12 c1(-n2cc(C(=O)NCc3onc(CC(=O)O)n3)nn2)ccccc1Cl c1(OC)cc(C(=O)Oc2cccc(Cc3nncs3)c2)cc(F)c1C#N N1(C(COC(C)=O)=O)CCN(n2nnnc2CSC2CC3C=CC2C3)CC1 c1(C(=O)NC2CCC(CNC(c3nc(CC)[nH]n3)=O)C2)cc(C)cnc1C N1(C(c2c(C)nc(CC)s2)=O)CC2CC(O)C1C2NC(C1CCC(=O)NC1)=O c1(CC)sc(C(=O)NC2CN(C(=O)COc3cn[nH]c3)C2)cc1C C1(C(=O)[N+](CC2CN(C(C(F)=CCC)=O)CC2C)([O-])NC)CCC(F)(F)CO1 CC1CC(F)CN1C(=O)C(C)(C)n1ccnn1.C1CS1 N1(C(C2(F)C(C)(C)C2(C)C)=O)CC2CCC(NC(=O)CCNC(=O)CO)CC2C1 N1(CC(=O)OC)CSCC1=O.C12CC(C1)CCN(C(=O)C=C(C)C(F)F)C2C C(=O)(CC(C)(C)C(C)=O)NC(C(N1CCC(OC)C1)=O)(C)C N1(C(Cc2c(C)non2)=O)CCOCC1CNC(c1ccc(Cl)o1)=O C(CC(=O)NCc1cc(O)ccc1F)(C(F)F)NC(c1c(CC)cccn1)=O C#CCC(C)(C)C(=O)N1CCC2C(C(=O)N(C)OCC(F)(F)F)C2C1 c1(OCC)cnc(N2CCCC(CN(C(=O)CC3CCCCO3)C)C2)nc1 N1(C(CN(C(=O)OC)C)=O)CCC(NC(c2cccc(=O)n2C)=O)C(C)C1 N1(C(CCN(C)C(C2CCCOCC2)=O)=O)CC(O)CC1C(N)=O C1(C(N2CC(O)(CN(C(CCC(=O)OC)=O)C)C2)=O)CC2CC(O)CC(C1)C2 c1(C(N2CC(F)(C(=O)Nc3cnc(O)nc3)C2)=O)noc2ccc(Br)cc12 c1(C(N2CC(C)C(NC(=O)C(C)C3(O)CCC3)C2)=O)cc(Br)ncc1Br Cc1ccc(C(=O)NC(C)C(CO)NC(=O)C(C)n2cnnn2)nc1O C1(NC(C=NOC)=O)C=CCN(C(C2CC23CCC3)=O)C1 c1(C(=O)NCC(C)(O)CNC(C2(Cl)CC2(F)F)=O)nccc2c1CNC2=O N#Cc1nc(=NCCCCCCNC(c2c(C)n[nH]c2C2CC2)=O)c(F)c(Cl)[nH]1 S(=O)(=O)(c1ccc(=NCc2ccco2)[nH]c1)NCCCOC=C N1(C(C(C)SC)=O)CCC2C(NC(=O)C=CC(N3CCOCC3)=O)C12 c1(C(N(CC(CC)NC(CCSCCCC)=O)CC)=O)c[nH]c2c(C)cccc12 N1(C(CC(C=C)C)=O)CCC2CN(C(c3ccc(NCCCC)cc3)=O)CC2C1 N1(C(C2C(OC)C2)=O)CCC(C(=O)NCCn2cnnn2)C12CC2 c1(CNC(C2(CO)CC2)C)cc(C(C)(C)C)n[nH]1.c12ccnn1C2 c1(C(N2CCC(N(C)C(C3CCCN3C=O)=O)C2)=O)cc2n(n1)CC(C)(C)CO2 Cc1ccc(O)c(C(=O)NCCC(C)NC(=O)C(C)Cc2ccnn2C)c1 c1(N2CC(CCOC)OCC2)nc(NCC(C(C)C)OCC)c2c(ncn2C)n1 c1(CC)c[nH]nc(NC(COC)(CCOC)c2nnnn2C(C)C)c1=O c1(C(=O)NC(C)CC(C)NC(=O)C(C)(C)Oc2ccc(F)cc2)ccc(C#N)o1 N1(C(C2(C=C)CCC2)=O)CCC(CNC(c2cocc2C(N)=O)=O)(OC)CC1 Cc1c(C(=O)N(C)CCNC(C23OCCCC2C3(F)F)=O)ccc2c1CCC2 N1(C(C2N(CCC)C(=O)CC2)=O)CCC2CN(C(=O)CC(C)(C)O)C2C1 C(=O)(C1=CCCCCC1)N1CC(N(C(=O)Cc2sccc2Br)C)C1 C(=O)(C1=CCC(C)CC1)N1CCN(C(C2N(CC)CCOC2)=O)CC1.C(COC)S C1(CCNC(C=C(C)C(C)C)=O)CCN(C(C2(c3ncco3)CCC2)=O)CC1 N1(C(COCC(=O)OC)=O)CCC(CN(C2CCCC2)C(=O)CC2CC(C)C2)C1 C1(NC(C(C(C)C)OCC)=O)C2CC3C(C2)C13C(=O)NC1(C(=O)NCC)CCCC1 c1(C(=O)NC(CCCC)CNC(=O)CNC(=O)OCC)ccc2cnnn2c1 CC(CCNC(C1(NC(C2CC3CC3C2)=O)CCSC1)=O)C(F)F N1(C(CCC(=O)NCC)=O)CCCC(C)(CNC(C2(CF)CC2(F)F)=O)C1 C1(NC(Cc2cn(CC)nn2)=O)CN(C(=O)C(O)CC2CCCC2)CC1C c1(C(N(CCC(C)NC(=O)C2CC2)C)=O)cccc(O)n1 C(=O)(C(C)(C)CC1CCOCC1)N(CCNC(=O)C(F)C1CCOC1)CC N1(C(C2CC(C)(C)C2)=O)CCC2(CCCN(C(=O)COC(F)(F)C(F)(F)F)C2)C1 C1(NC(Cn2c(C)ccn2)=O)Cc2ccccc2C1NC(=O)C(C)C(F)F C1(CC(=O)NCC(C)NC(C2C(C(N(CC#C)C)=O)C2)=O)CC1(C)C N1(C(C(CC)Oc2ccccc2)=O)CCC2CN(C(=O)CCCF)CC2C1 c1(-n2nnnc2NC(c2cnn(C(C)C)c2C2CC2)C)cc(C)cnc1C.C1(N)CCC1 CC1(CNC(C2CCN(C(=O)Cn3cnnc3)C2)=O)CCC(=O)N1 C1(NC(c2cc(C)ncc2)=O)CN(C(c2nn(C)c(C)c2Br)=O)CCC1F N1(C(CC2C(NC(=O)CCOCC3CC3)C2)=O)CCC(c2ccon2)C1 c1(C(=O)NCC(CCNC(C2(CCOC)CCC2)=O)(C)C)cnc2[nH]cncc1-2 c1(C(N(CC=CC(=O)NC(CC)CO)C)=O)coc(CN(C)C2CC2)c1 CCC(C)C(O)C(C)C(=O)NC1(C2CCCN2C(=O)CCCC2CCC2)CC1 C1(C(N(CCC(C)O)C)=O)CCCN(C(c2ccncc2)=O)C1 C1(CNC(C(C=C)O)=O)CC(C(C)(C)C)CN(C(c2nccc(C)n2)=O)C1 c1(C(N(CC)NC(C2CCC2C(=O)OC)=O)=O)nnn2c1COCC2.CC(C)N(C)C CC(C(C)(C)O)N(C(=O)CN(C(=O)CC1CCCN1C)C1CCC1)C C1(OCC)(CNC(c2ccncc2)c2nnnn2CC2CC2)CCSC1 N1(C(C2(CC)CCCCC2)=O)CCC(c2ccccc2)C(CN(C)C)C1 c1(C(N2CCC(C)(C(=O)NCC3(C)CNC(=O)O3)C2)=O)cccc(C#N)c1 C(C)(CC(=O)NCC1CC1NC(=O)CCC1CC(NC(=O)OC(C)(C)C)C1)SC CC1CN(C(=O)CCNC(=O)CO)CCC1C(=O)NCCC1CCCN(C)C1 c1(C(=O)NCC2(F)CC(CNC(C3=C(C)OCC3)=O)C2)cnn2c1CC(C)CC2 C1(CNC(Cn2nnc(C)n2)=O)CCC12CCN(C(=O)CCCC1CC1)CC2 C(=O)(CCC(C)CN(C)C)NC(C(=O)NC(C)C(C)(C)CO)C1CCC1 N1(C(=O)OC(C)(C)C)CCc2onc(NC(N3CCC4COCC34)=O)c2C1 c1(C(=O)OC(CCSC)C(=O)OC(C)C)cc(C)c(C)cc1Cl C(CC(=O)N1CCCC1CN(C(=O)C(C)S(C)(=O)=O)C)(C1=CCCC1)OCC c1(OC)ccc(CO)cc1C(=O)NCC(c1cccc(F)c1)NC(=O)CSC C(C)(N=c1nc[nH]s1)C1OCCN(C(C=CCN(C)CC)=O)C1 C1(C(=O)NC2C(NC(CCNC(=O)NC)=O)CC2)CCc2nc(C)ncc2C1 c1(NC(C(CNC(C(CC=C)CC)=O)C)=O)cnc2[nH]cnc2c1 C(=O)(CCS(N)(=O)=O)NC1(CNC(Cc2cc(COC)no2)=O)CCC1 N1(C(C(C2CCCO2)NC(c2ccncc2)=O)=O)CCOC(CC2CC2)C1 C1(N(C(CNS(CC)(=O)=O)=O)C)CN(C(=O)C(F)n2ccnc2)CC12CC2 CC(CC1CCCC1)C(=O)N1CCCC1CN(C(=O)Cc1cnoc1)C c1(C(C)=O)cccc(OCC(N2CC3C(NC(C4CCCCN4C)=O)C3C2)=O)c1 c1(C(C(=O)NCC(CNC(CCC(=C)Cl)=O)F)C)ccc(Cl)c(Cl)c1 C1(NC(c2c[nH]c(Br)c2)=O)CN(C(c2cccnc2C(F)(F)F)=O)CC12CC2 Cc1cccc2c(C(N3CCN(C(=O)CC4CCC4)C(CO)C3)=O)cnn12 c1(C(=O)NCC2CCC(C(=O)NC(C3CC3)C3CC3)C2)cc(F)c(F)cc1I c1(COC)nc(Cl)cc(=NC2CCN(C(C3CCCC3C)=O)CC2CO)[nH]1 c1(OC)ccnc(C(=O)NCC#CC2CC2)c1OC c1(C(=O)NC(C)(CNC(c2cc(Br)c[nH]2)=O)C2CCC2)ncccc1O Cc1cc(C(=O)NC2COCC2NC(=O)Cc2ccc(C)s2)c(F)cc1F C1(NC(CCCC)=O)CCC2CCN(C(=O)COCc3cc(C)no3)C1C2 N1(C(CC(C)OC)=O)CC2(CCN(C(c3c(F)cc(C#N)cc3F)=O)CC2)C1 C1(OCC(=O)NCC2C(C(=O)NC(C3CC=CCC3)CC)C2)CCCOC1 N1(C(CC2CC(OC)C2)=O)CCC(O)C(N(C(=O)CC2CCCC(F)(F)C2)C)C1 C1(NC(C(CC=C)c2ccccc2)=O)CN(C(=O)C=CCCC=CC)CC1N=[N+]=[N-] N1(C(CCNC(C)=O)=O)C2CCC1CC(F)(CNC(C1(C(F)F)CCC1)=O)C2 N1(C(C=C(C)C)=O)CCC2C(CCN2C(=O)CN2CCCCC2)C1 CCS(=O)(=O)c1cccnc1C(=O)NC1CN(C(=O)C(F)(Cl)c2ccccc2)C1 C1(C(=O)NCC(C(=O)OC)C)CSCCN1C(=O)C(O)CN1CCCC1 C1(C)(CC)CC(NC(=O)CC(C)(C)Cc2ccccc2)CN1C(=O)C=C(Cl)Cl O(NC(=O)C(CC(CC)CC)NC(=O)C(C)C(C)(C)C)CCC=C CCCC(C(=O)NC(CNC(c1ncncc1Br)=O)C(C)C)OC C1(C(C)NC(c2cccs2)=O)CCCN(C(C2(C(F)F)CCC2)=O)C1 C12(C(=O)NC3CCC(NC(=O)Cn4ncnn4)CC3)CCCC1CS(=O)(=O)C2 C1(C(N(C(C)C)CC)=O)CCCN1N1CCc2nc(N(C)C)sc2C1 C1(C(=O)NC2C(C)CCC2C)CC2(CC(NC(=O)C=CC(F)(F)F)C2)C1 C(=O)(C(CO)N(C(=O)CN(C1CCC1)C)CC)N(C(CC)C)CC C=CC(CCC)CC(=O)N(C1CCN(C(c2ccc(OCC)nc2)=O)C1)CC(C)C C1(NC(c2c(C)nc(C(F)(F)F)s2)=O)CCCN(C(=O)Cc2ccsc2C)C1C c1(OC)c(C(=O)OC)ccc(CNC(C)Cc2ccsc2)c1C c1(C(=O)NCC2(CNC(C3CC3C3CC3)=O)CCC2)ccnn1-c1cccnc1 c1(C(N2CCC(COC)(NC(=O)C(C)C(C)C)C2)=O)ccncc1N=[N+]=[N-] O(NC(=O)CC(C)(C)NC(c1ccc(O)cc1)=O)CCC Cc1ccc(NC(N2CCCCC2C(=O)NCc2nc(C)c(C)s2)=O)cc1F c1(C(N2CC(NC(C(C)OCCC=C)=O)C(F)C2)=O)n[nH]c2c(OC)cccc12 C12(C(C)NC(=O)C(O)C3CN(C(c4cn(CCO)nn4)=O)C3)CCC(CO1)C2 O=C(CC1CCOc2ccccc21)NCC1(NC(C2CCSC2)=O)CCCC1 N1(C(CNC(CC(C)(C)C)=O)=O)CCN(C(c2cc[nH]c2)=O)CC1CO c1(CCC(N2CCC(N(C(C(C)(C3(C)CC3)OC)=O)C)C2)=O)cc(C)nc(C)c1 N#CC1=C(C(=O)N2CC(C(F)(F)F)CC2CNC(c2cccc(Cl)c2)=O)CCC1 C1(C(C)=O)C2CCC1(C(=O)Nc1ccnn1CC(F)F)C2 Cc1ncc(C(=O)NC2(CCO)CN(C(=O)Cn3cnc(Br)c3)C2)s1 C(=O)(CC(C(F)(F)F)c1cccc(F)c1)NC(CNC(c1c(C)scn1)=O)CO CCCCCC(CC)C(=O)N(CCC(=O)NCC1(CSC)CC1)CCCO C(C1CN(C(C2CCCCC2O)=O)CC1C(=O)NCCN(C(C)C)C(C)C)=CC c1(C(N2CCN(C)C(CNC(C3(CC(F)F)CC3)=O)C2)=O)cnn2ccccc12 c1(C(C(=O)NC2CC(F)(F)C2)N(C(C)COC)CC)ccc(S(C)(=O)=O)c(C)c1 CCC(C#N)C(=O)OC.c1(CC(=O)NC(C)=O)ccc(C(N2CC(C)C2)=O)cc1 N1(NC(c2n(CC#C)ccc2)=O)CC2CC2C2CC12.C1(C(=O)N)(C)CCC1 N1(C(Cc2ccn(C)n2)=O)CCCC(n2cc(CCNC=O)nn2)CC1 CC(C)C(F)(CNC(C1(C)CNC(=O)C1)=O)C(=O)N1CCC2CCC12 C(C(=O)NNC(=O)C1CCOC1C(C)(C)C)C1(OCC)CCCC1 c1(NC(C2(c3ccccc3)C(CC)C2)=O)cc2ccc(Br)cc2s1 c1(NC(=O)C(=O)NC2(C3CCCC3)CCC2)cccc2[nH]ccc12 C(C(C(=O)N1CCC(c2nn[nH]n2)C1)NC(=O)CCc1cnco1)N(C)C C1(NC(C(C)NS(C)(=O)=O)=O)C2CCCN(C(=O)CC3OCCCO3)C2C1(C)C CC1(CNCC2CC(=O)N(C(C)(C)C)C2c2ccco2)CC2CCC1C2 c1(OC)ncc(C(=O)NCC2CC(NC(=O)CC3CCCCC3)C2)c(C(F)F)n1 Nc1cc(C(=O)NC2CCN(C(C3CCCOC3)=O)C2)ncc1Cl c1(NC(=O)NC(C#CCC)(C)C)nc2ccc(N)cc2s1 c1(CC2CN(C(=O)NC3C(C)(C(C)C)C3)C2)ccc(Br)cc1 c1(CNC(CCCSC)Cc2ccccc2)nc(C(C)C)ncc1Br Cn1cc(C(=O)NCC2CCN(CC3CCCO3)CC2)c(-c2ccco2)n1 C1(NC(c2c(OC)csc2)=O)CN(C(c2cccc(F)c2N)=O)CC1(C)C N1(C(c2scnc2Br)C(=O)N(C)C)CCCCC1Cn1ccnn1 CC1(CNC(C2OCCCO2)=O)CCC(NC(c2cc(C(C)(C)C)no2)=O)CC1 C1(C(=O)NCC2(C(=O)NC3(C(=O)OC)CC3)CC2)CC1(F)F C(C(C)(C)C(=O)N1CCCC(CN(C(=O)CC2(OC)CC2)C)C1)OC N1(C(CC(CC)OC)=O)CCC2(CCC(CNC(=O)CC34CC(C3)C4)O2)CC1 N1C(=NCC#CC2CC2)NCc2ccc(cc2)C1.CS(=O)(=O)CNC1CC1 C(=O)(CCCC(F)F)NCC1OCCN(C(C2(CC)CCCC2)=O)C1 c1(C(N2CCn3c(cnc3Br)C2)C(=O)NCCC2CC2)ccc2cnccc2n1 CCC(CNC(C1CC(O)C1)=O)(CC)C(=O)N1CC(C)C(O)C(C)C1 c1(C(N(CC(C)(C)NC(Cn2c(C)ccn2)=O)C)=O)coc2c1C(O)CCC2 N1(CC2CC(=O)N(C)C2=O)C(=O)CCN(CC2CC=CCC2)C1=O C1(C(N)=O)(C(=O)NC2CC(NCCn3cc(CO)nn3)C2)CC2(CC(F)C2)C1 CCC(C#N)C(=O)NC(C)CNC(=O)CCCc1cnn[nH]1 Cc1cc(C(=O)NCC(C)CNC(C2(C#N)CC=CC2)=O)cc(C)c1C#N N1(C(C2N(C(C)=O)CC(O)C2)=O)CCC(NC(c2ccnnc2)=O)C12CCC2 C(=O)(C(C)(C)C(F)F)N1CC(C(C)NC(CCOCCOC)=O)C1 c1(C(N(CC(CNC(C2(COC)CC=CCC2)=O)(C)C)C)=O)cc(C)cc(C)c1 C(=O)(CC(O)CNC(N)=O)NCC1CN(C(Cc2cnc(C)[nH]2)=O)C1 C(=O)(CC(CCCC)NC(=O)CCCC1CCCC1)NC(C#C)CC C(CCCCSC)(C(=O)O)NC(N(CCOC)CCF)=O c1(C2(C(=O)NC3CC(NC(CC4CC(C#C)(O)C4)=O)C3)CCC2)cc(Cl)cc(Cl)c1 CCCC(CNC(C1CC(NC(C2CCOC2)=O)C1)=O)CCO CC(C)(C)CCCC(=O)NC(CC(=O)N1CCC(n2cnnn2)C1)C(F)(F)F C1(NC(c2c(C)[nH]cc2)=O)CCC2CN(C(C3CC4(C3)CC4(F)F)=O)CCC2C1 C(=O)(C(C#N)C(C)(C)C)NCCCC(C)(C)NC(=O)C1=COCC1 CC(C)C(CCc1ccccc1)C(=O)NCC(C)NC(c1ccnn1C(C)C)=O C(=O)(C1COc2ccc(Cl)cc21)N1C(C)CC(NC(c2cnoc2)=O)CC1 N1(C(C2(CCC)CC2)=O)CCOCC1CNC(=O)C(C)NC(=O)CC(C)(C)C CCC(C)C(O)C(C)C(=O)NC1CC(C)(C(=O)NCC2CN(C(C)C)C2)C1 N1(C(CSCCCC)=O)CC=CC(NC(=O)COCc2c(C)noc2C)C1 C=C(C)C1OCCC1CNC(=O)CC1CCC(NC(=O)C(CCC)OC)CC1 CC(C(=O)NC1CCN(C(=O)Cn2cnnc2)CC1O)S(N)(=O)=O C(c1ccc(C)cn1)=CC(=O)N(CCNC(C(C)OCCCCCC)=O)C1CC1 N1(C(c2n(CC=C)ccc2)=O)CC2(CCC(CNC(C3CCC4CC34)=O)O2)C1 c1(OCC)ccc(C(N2CCCC(O)(CNCS(=O)(=O)C3CC3)C2)=O)c(F)c1 N1(C(c2nc(C)sc2)=O)CC2CC1CCC2NC(c1cccc(O)n1)=O N1(C(CCNS(C)(=O)=O)=O)CC(NC(=O)CCc2c(C)noc2C)C(C2CC2)C1 C(=O)(C1=Cc2ccc(F)cc2OC1)NCCC1N(C(CSCCC)=O)CCSC1 n1(CC(=O)NCCCCNC(C23CC(C2)S(=O)(=O)C3)=O)nc2n(c1=O)CCCC2 c1(C(N(CCNC(C2(OCC)CCOCC2)=O)C(C)C)=O)ccc(F)c(C#N)c1 Cc1cnc(NCC2CCCN(C(=O)CCSC3CCCC3)C2)c([N+](=O)[O-])c1 CC(C)CCC=CC(N1CCC(N(C)C(C2(Cl)CC2(F)F)=O)C1)=O N1(C(c2ccc(C)nc2C)=O)CC(NC(C2CC(C)(O)C2)=O)C(S(C)(=O)=O)C1 C1(C(N2CC(OC)(CNC(C3(CC(C)C)CCC3)=O)C2)=O)COC2(CCC2)C1 C1(C(=O)NCC2N(C(CSCCC)=O)CCC2CC)CC2CC1CC2O C(=O)(CCCC(C)(c1nnnn1C)NC(c1ccc(C(C)(C)O)cc1)C)OC CCCCC(C)C(=O)NC1C=CCN(C(=O)CCC(=O)N2CCC(O)CC2)C1 C(CC(C)(C)C)N(C(C1CC1(C)C)C(=O)NC1CC(F)(F)C1)C(C)C [N-]=[N+]=NCCCC(=O)N1CC2CC(C1)N2C(=O)C(O)CC1CC1 c1(C(=O)NCC(C(=O)NC(C)C(C)(C)O)C)ccn(C)c(=O)c1 N1(C(C(C)OC)=O)CCC2(CC1)CN(C(C1CNC(=O)CC13CCC3)=O)CC2CO c1(C)ccc(C(F)(F)F)c(Cl)c1.N1(C(c2c(C)ccs2)=O)CCC2(C1)CN2 Cc1ccnc(CN(C)C(c2coc(C(C)NC(=O)C(C)CC3CC3)n2)=O)c1 c1(OC)ccc(C=CC(=O)NCC(C)(C)NC(C2CCCOCC2)=O)cc1 C(C)(CCC(=O)N1CCC(N(C)C(c2cc(SC)oc2C)=O)CC1)OCC C1(NC(c2c(C(C)C)occ2)=O)C2CN(CC(=O)NCC3CC3)CC12 C1(C(C)CC#C)CCCN(Cc2ccc(F)c(Br)n2)CC1.C1(C(=O)OCC)CC1 C1(NC(=O)C(N2CCC(Oc3ccccc3Br)C2)=O)CCC2(CC1)CC2 C1(C(C#C)C)CCN(C(=O)COC2CCN(C(=O)CO)C2)CC1 C(=O)(C1=CCS(=O)(=O)C1)N1CC(C(C)NC(Cc2ccc(C)nc2)=O)OCC1 N1(C(CC2(CC)CCC2)=O)CCC(O)(CNC(c2ccccc2OC(F)F)=O)C1 N#CC1(C(N2CCC(C3CCCN3c3nnn(C)n3)C2)=O)CC2CCC1CC2 Cc1ccc(C(N2C3CN(C(=O)C(C)(C)C4CC4)CC23)=O)cc1Cl Cc1cc2cccc(-c3ccc(CN4CCN(C(=O)C(=O)C5CC5)CC4)s3)c2[nH]1 C(C(C)(C)CC(=O)NC(C)(C)C=CC(=O)N(C1(OC)CCC1)CCO)OC N1(C(C(C)Oc2cccc(C)c2)=O)CCC(NC(=O)C(F)C2CCC2)C12CC2 N(C(=NCCF)NCC1(O)CS(=O)(=O)C1)C(c1noc(C)n1)CC c1(C(=O)OC)ccc(NCC2CC2)cc1OC(F)(F)C(F)(F)F N1(C(COCCC)=O)CCC(NC(=O)Cc2cc(Br)co2)C(C(C)C)C1 N1(C(CNC(C(CC)(C)C)=O)=O)CC(C2CN(C(c3ncc4[nH]ncc4n3)=O)C2)C1 C12(CNC(C(C)(C)C#N)=O)CCC1CN(C(c1cc(C(F)F)[nH]n1)=O)C2 C1(C)(NC(C(CC)CO)=O)CCCN(C(=O)C(C)Cc2ccc(C)cc2)C1 C(=O)(C(CC1CC1)NC(=O)CN1CC2CC2C1)NC(c1nccn1C)CC c1(CC)cccc(C(=O)NC2CC(N(C)C(C3CC34CC4)=O)C2)c1O n1(CC(N2CC(NC(C(C)O)=O)(CF)C2)=O)cnc([N+](=O)[O-])c1 c1(C(=O)NC2CN(C(COCCC#C)=O)CC2SC)cc2cc(F)ccc2o1 CCCC(C(=O)NC1(COC)CN(C(=O)CCC2CC2)C1)n1ccc(C2CC2)n1 N1(C(c2c(N)cc(F)cc2)=O)CC2(COC(CNC(=O)CCOC3CC3)C2)C1 CN1CCOC(CNC(C2CC(O)CN2C(=O)C(C)(C)C2CCC2)=O)C1 C12(CCNC(C(C)N(C)C)=O)CC(CO)(C1)C(C)(C)O2 c1(OC)cc(CNCC2(F)CN(C(=O)Cc3ccccc3Br)C2)cc(Cl)c1 CC#CCC(C(=O)N(C)CC1CC1C)NC(=O)CCCF Cc1c(-c2nc(CCN(C)C)nn2CCc2ccc(Br)cc2)cnc2ccnn12 CCCC(C(=O)NC1CCN(C(c2cc(SCC)cnc2O)=O)C1C)NC(C)=O N1(C(C(CC#C)C2CC2)=O)CCOCCC1C(=O)NCC(c1cccs1)C CC(CF)CC(=O)NCCCCNC(c1nc(C(F)(F)F)cn1C)=O Cc1nc(O)nc(C)c1CC(=O)NCC(CNC(C1(Cl)CCC1)=O)CO c1(N(C2CCNCC2O)C(c2ncc(Cl)cc2O)=O)ncnc2sccc12 C1(n2cc(CNC3CCc4n(C5(SC)CC5)ncc4C3)nn2)CCCC1S(C)(=O)=O N1(C(CC=CC=C)=O)C(CNC(C2CCCN2Cc2ccccn2)=O)CC2CC12 C(C(=O)N(C)OCC)(c1ccccc1O)NC(C=C(CCC)CCC)=O N1(C(C(CC(=C)Cl)NC(=O)C(C(C)C)NC(C)=O)=O)CC2(CCC(=O)O2)C1 CN1CCC(C(=O)NCCC2(C)CCN(C(=O)Cc3ccn(C)n3)C2)CC1=O CCCC(C)(C)C(=O)NC1CCC(N(C)C(C)=O)CC1 N1(C(Cn2cc(-c3cc(C)c(F)cn3)nn2)=O)CC(=O)N(C)CC1C C(C#CC(=O)NCC1(CC(N)=O)CC1)NC(CN(C(C)=O)C)=O C1(NC(=O)NC2CCC(CC#N)C2)CC2CC1CC2F C1(CC)CN(C(C23CCC(C(=O)NC)(CC2)C3)=O)CCN1C(=O)CCc1cncs1 C(C)(C)(C(C)CC(=O)NCCC1COCC1O)NC(C1CC(C#C)(O)C1)=O c1(C(=O)NCC2N(C(c3cncc(N)c3)=O)CC(F)C2)cc(F)c(F)cc1F C(C)(C(CC(=O)NC12CC(F)(C1)C2)NC(c1cc(N)cc(F)c1)=O)OC C(CCCCCNC(C1CC2CC1C2)=O)N(C)C(C1CC1F)=O C(=O)(CC(C(F)(F)F)OC)N1CCC(N(C(C2CC3(C2)CC3F)=O)CC)CC1 c1(CCCNC(=O)C(N2CCN(c3cccc(Cl)n3)CC2)=O)ccc(O)cc1 C1(CNC(C2(CC#C)CCCO2)=O)C2CN(C(C3CC4(CCC4)C3)=O)CC12 c1(C(C)C)cccc(CC(=O)NCC(C)(C)CNC(C2CCCS2)=O)c1 c1(CCC(=O)NC(C2CN(C(CCC#C)=O)C2)C)ccc(F)c(F)c1 C1(NC(C(C)SCC)=O)CCN(C(C23CCC2CC3)=O)C(C)C1 c1(C(N2CC(NC(C3ON=C(C)C3)=O)C(C)C2)=O)cnn2cc(Br)cnc12 S(=O)(=O)(c1ccc([N+](=O)[O-])c(Cl)c1)NCC(C(C(C)C)C)N CS(C)(=O)=NC(=O)c1cc(C2OCCO2)on1 N1(C(C(CC=CC)C)=O)CCCCC(CNC(c2cncn(C)c2=O)=O)CC1 C1(NC(C2(CC=C)CC2)=O)CC1C1CCCN(C(c2ccc3scnc3c2)=O)C1 N1(C(C=C(CC)CC)=O)CCSCC1C(=O)NCC(C)(O)C1(C)CC1 N(C(=NCCc1ccccn1)NCc1c(Br)nnn1C)CC(CC)(C)C N1(C(C(C)OCOC)=O)CCC(N=[N+]=[N-])(C(=O)NC2(C)CCC(=O)NC2=O)C1 c1(CC(=O)NCC(C)(C)NC(c2cc(F)cc(N)c2F)=O)ccn2cncc2c1 c1(NC(C)C)ccc(C(C)NC(C)Cc2cccc(C(C)(C)C)c2)nc1 N12CCN(CC1CCOCCON)CC2=O.C12(C(N)=O)CCCC1C2(F)F c1(OC(c2ccc(CCC)s2)=O)ccc(OCCNCC2CNCCO2)cc1 Cc1ncn2ccc(C(=O)NCC3(CCNC(=O)C=Cc4cccs4)CC3)cc12 Cc1cc(C(=O)N(CCCOCCNC(c2ccn(C)c2)=O)C)c2nccn2c1 N1(C(c2ccc(SC)s2)=O)C2CCCC1CC(NC(=O)C(C)(O)C(C)C)C2 C1(O)(CCNC(C(C)(C)c2ccccn2)=O)CCN(C(c2ccnnc2)=O)C1 C(c1ccccc1)=C(CC)C(=O)N(C(C)CSC)C c1(C(N2CCN(c3c(C#N)c(Cl)ns3)CC2)=O)ccc(F)c(F)c1O c1(C(=O)NCCN(C(=O)CCc2ccc(F)nc2)CC)cccc(F)c1COC C1(C)(CNC(CC(CC)C)=O)CC(F)(F)CN1C(=O)Cc1cc(C)nn1C c1(SCCN(C(C)(C)CC)C(C=CC=CC)=O)cc(C)cc(Br)c1F c1(N2CCC(C)(C(=O)NC)C2)ccc(S(=O)(=O)NCc2c[nH]c(=N)s2)c(Cl)c1 CN1CCC(C(=O)NCc2nocc2C(N2CCCCCCC2)=O)CC1=O C1(C(=O)NCC2CC(C(=O)NC3CC3c3ccco3)C2)CC2CCC1C2 CC1CCCc2nc(C(N3CCOC(CCCNC(=O)C(C)(C)C#N)C3)=O)cn21 c1(NC(c2nnnn2C2CC2)(CC)C2CC2)cnc(C)[nH]1 CC1CCN(C(C2CC(=O)N2)=O)CC1CNC(=O)C(c1ccc(F)cc1)F C1C(C)(CC)N1.CCC(C)OCC(=O)NCCNC(=O)OC(C)(C)C c1(C(C(C)OC)O)nc(-c2occc2C)nn1Cc1ccc(F)cc1 C(=O)(CCC(C)(C)F)NC(COC)C(=O)NCc1ccc(O)c(C)c1 Cn1nc(C(=O)NCC2CC2NC(=O)Cc2sccc2Br)cc1C(F)F C(c1nc2ccccc2o1)=CC(N1CC(C)N(C(=O)Cn2cccc2)CC1)=O c1(CC(=O)NCC2CC(NC(C3C(CN(C)C)C3)=O)C2)cccc(Cl)c1Cl CC1(CNC(=O)COc2ccc(F)cc2Cl)CN(C(C2(C)CC2(Cl)Cl)=O)CCO1 Cc1ccc2c(c1)CC(C(=O)NCC1CCCCN1C(C1CCCCCC1)=O)O2 C#CC(CNC(=O)C(C)N(C(c1scnc1C)=O)CC)CC(C)(C)C c1(C(=O)NCCC=CCCC)ccnc(NCC(O)Cc2ccccn2)c1 N1(C(c2c(CC)nccc2)=O)CCC2CC2(C(=O)NC2CCNC(=O)C2)CC1 C12(NC(c3[nH]cc(CC)c3)=O)CCCCC1CN(C(c1nocc1Cl)=O)C2 N1(Cc2ccc(CCC)o2)CC=C(CCNC(c2cc3c([nH]2)CCC3)=O)CC1 c1(C(=O)NCCCCCC(=O)NCC(C2CCCCC2)C)cccc2cncn12 c1(C(=O)NC2(C)CN(C(=O)COC3CCCCC3)C2)cc2n(n1)CCOC2 C1(CNC(C=CC(C)(C)C)=O)CCCCN1C(c1ccc(-n2ccnn2)cc1)=O c1(NC(C2C(C(=O)Nc3c(OC)ncnc3OC)C2)=O)cccc2nc[nH]c12 C12(CNC(C3C(C)=C3)=O)CCCC1N(c1ncnc3ccsc13)CCC2 c1(CC(=O)NC(c2cn(C)nc2)C(N2CCC3(CC3)C2)=O)cccc(F)c1N c1(C(=O)NC2(CO)CCCN(C(C3ON=C(CC)C3)=O)C2)nc2c(s1)COCC2 C(C(=O)N(C)Cc1ccc(C)nc1)(C(C)CC)NC(c1ccc(CC)cc1)=O c1(N2CCC(CCCC)C2)nc(N2CCC(CC(F)(F)F)C2)cc(C)n1 C=CC(C)(C)CC(=O)NC1CC(C)(NC(=O)COCC2CCCO2)C1 CC1CCCC1N=c1nc(N2CCN(CC(O)C3CC3)CC2)c2ccccc2[nH]1 CC(CC(C)NC(=O)CNCc1ccccn1)NC(=O)CC1(O)CCCC1 c1(OC)ccc(Cn2cc(CC3(O)CCSC3)nn2)cc1.c12ccc(o1)CNC2=O C1(F)(CNC(C(C)N(C)C)=O)CCN(C(=O)CN(C)Cc2ccccc2Cl)C1 CCCC(O)CC(=O)NC1CCCC1NC(c1cn(CCC2CC2)nn1)=O C1(CC=C)COCC1NC(=O)CCCN(C(=O)C(C)OCCN(C)C)C C1(NC(C=CCC)=O)CC2CN(C(c3cc[nH]c3C(C)C)=O)CC12 CC1CC(=O)CCC1C(N1CC=CC(NC(c2cc(CC(C)C)n[nH]2)=O)C1)=O C#CC1(C(=O)NOC(c2cccc(CC)n2)=O)CCN(CCCC=C)C1 CCCC(CC)C(=O)N(CCCOCCN(C)C(c1cnc(C(F)F)s1)=O)C N1(C(=O)Cc2ccc(Br)cc2[N+](=O)[O-])CCC2(CC1)OCCC2O N1(C(c2cc(Cl)c(OC(F)F)c(Cl)c2)=O)CC2CS(=O)(=O)CC2(c2nn[nH]n2)C1 c1(C(=O)OCC)c(NC(=O)N(C)Cc2ccnc(OC)c2)sc(CC)c1C C1(COC)(NC(c2cc(C(N)=O)[nH]n2)=O)CN(C(=O)Cc2ccc(Cl)s2)C1 Cc1cc(CC(=O)NC(CC2CCC2)C(=O)N(C)Cc2nnc(C)s2)on1 c1(CC(N2CCC(O)(CNC(CNC(=O)OC)=O)C2)=O)ccc2c(c1)CCN2C c1(OC)ncc(-c2ccc(N3CCN(Cc4ccc(C#N)s4)CC3)cc2)cc1C N1(CCCC(N2CC(CN)C(F)(F)CC2)=O)C(=O)Cc2ccccc2C1=O N1(C(C(C(C)C)CNC(=O)CC(C)n2ccnc2)=O)CC2(C)CCC2(C)C1 N1(C(C(CC)(C)C)=O)CCC2(CCOC2)C(CNC(=O)C2=CCC(C)CC2)C1 C1(O)(C(C)NC(CC(C)C)=O)CCN(C(c2cc(Br)co2)=O)C1 O=C(NOCC=CCl)C1c2c[nH]nc2CN1C(=O)C1=CC2C=CC1C2 CC(C)C(C#N)C(=O)NCC(=O)N(C)C(c1cccc(F)c1)C C1(O)(CN(C(=O)Cn2cnnc2)C)CCN(C(=O)Cn2cc(Cl)cn2)C1 CC(C)(CNC(c1sccc1Cl)=O)CCNC(=O)C(O)C1CCCC1 CC1COC(CO)CN1C(=O)C(CC1CCC1)NC(c1ccn(C(F)F)n1)=O C1(NCC2(C(=O)NC(C)C(N3CCNC3=O)=O)CCOC2)CC2CCCC2O1 n1(CC(=O)NCCC(CNC(Cn2c(C)ccn2)=O)O)cc(Cl)c(C)n1 c1(C(=O)NC2CCCC2CNC(C2(F)CCOC2)=O)ccncc1-n1cccn1 c1(C(CO)N)nc2ccccc2o1.N1(C(C23CC(C=O)(C2)C3)=O)CCOC2CC12 C(=O)(CC1=CCCCC1)N1CC(C(=O)NC2(Nc3c(C)c(F)ccc3)CC2)C(C)C1 c1(C(N2CC(CN(C(C(COC)C)=O)C)C2)=O)nc(-c2ccsc2)oc1C CC1(C)C2CCC1(C(N1CC=CC(NC(C3CCc4ncnn4C3)=O)C1)=O)CC2 C(C(C(=O)NCC1COCC1NC(C1CC(Cl)(Cl)C1)=O)OC)OC c1(C(C)C)nnc2n1CCCN(C(C)(C)C)C2.C12CCN1C2 c1(OC)nccc(C(=O)N(C2(CC(=O)NCCCN3CCNC3=O)CC2)C)n1 c1(C(=O)NN2C(C(=O)NCCCCOCC)CC2)cc(CC)n(CC)n1 N1(C(C2(CC)CC2(F)F)=O)CCN(C(=O)Cc2cc(C(F)(F)F)no2)CC1C c1(C(=O)NCC2CC(CNC(C(CC=CC)C)=O)C2)c(O)nnc2c1COCC2 n1(CC)cc(Cl)cc1C(=O)N(C)CCN(C(c1sc(OC)nc1Cl)=O)C(C)C C1(C(N(CC(C)(C)NC(=O)CN2CCCCC2)C)=O)CC12CCC1(CC1)CC2 C1(NC(CCC#CC)=O)CC2CN(C(=O)CN(C3CCC3)C)CCN2C1 C(=O)(C(C)(C)C(F)(F)F)N1CC2(C(C(=O)Nc3c(SCCC)cccc3)C2)C1 C1(CCNC(C(N2CCOC2=O)C)=O)CCCN1C(=O)CCSC(F)(F)F N1(C(C(n2c(C)cc(C)n2)C)=O)CC2CCC1CN2C(c1nccc(Cl)c1C)=O N(C1CCCNc2ccccc21)C(C1COCCN(Cc2c(OC)ccs2)C1)=O c1(C(=O)NCC2C(NC(C(CSC)C)=O)CCCC2)ncnc2ccsc12 CCC(CNC(C1(c2ccc(C)cc2)CCC1)=O)(CC)NC(C1CCSC1)=O Cn1c(C(N2CCC(CCNC(=O)CC3CCCC3)C2)=O)cc2ccc(O)cc12 N1(C(c2ccc3c(n2)OCCO3)=O)CCC2(CCN(c3ncncc3Cl)CC2)C1 c1(OC)ccccc1CC(=O)NC1CCC(CNC(=O)C=C(C)C)C1 c1(OC)cc(C)c(C(=O)NCCCC2(NC(C3(C)CC(F)C3)=O)CC2)cn1 c1(C(N(CCOC)CC)=O)ccoc1CNC(c1cn(CCO)nn1)=O c1(NC(C2(C#C)CNC2)=O)cc(SC2CCCC2)ccn1 c1(C(N2CCC(O)C23CCCC3)C(=O)NC(C)C)cc2ccnc(Cl)c2s1 c1(C(=O)NC(CCSC)Cc2ccco2)ccc(Br)c2c1OCCC2 N1(C(c2nnc(C)s2)=O)CCC2(CC1)CCN(CCC1CC1)C2 Cc1cc(C(C)(C)C(=O)NCC(C)NC(=O)CC(O)c2cnc(Cl)s2)cs1 CC1Cc2ccc(F)cc2C1NC(=O)Cc1c[nH]c2ccccc12 c1(NC(CNC(C(C=C)O)=O)(C)C)cc2nnc(CC)n2cn1 c1(CNC(=O)NC(C(CC)C)C)ccc(Sc2ccnn2CCN(C)C)cc1 c1(C(=O)NCC(CC)(C)NC(=O)C=C(C)C)cn2c(C)cccc2n1 C12(NC(c3c(C)oc(Cl)n3)=O)CCCC1N(C(C1COCCO1)=O)CC2 c1(NC(CCCC)c2nnnn2CC2CCOC2)ccc(-c2cccs2)cc1 C(=O)(C1=CCCOC1)N1C(C)(NC(Cc2c(CNC(C)=O)cccc2)=O)CCC1 C1(CNC(CCSC)=O)C(C)CCCN1C(c1cc(OC(F)F)cs1)=O Cc1nccc(Cl)c1C(N1CC2C(CNC(c3cc(C(C)(F)F)n[nH]3)=O)C2C1)=O C1(C(=O)NCCCNC(C(C)C)=O)CCC2(CC2)N1C(=O)CC1CCC1 C1(C(N(CCCCO)CC)=O)CC(=O)CN1C(=O)CC1CC1 C1(NC(c2c(C)nc(C)s2)=O)CC2CC(NC(c3cnoc3SC(F)F)=O)C1C2 c1(N2CCCN(C(CC#N)=O)CC2)ccc(S(=O)(=O)NC(=O)C2CC2)cc1[N+](=O)[O-] C(=O)(CCC(F)(F)F)N1CC(CC)C(C(N2CCCCC2c2cccnc2)=O)C1 Cc1cccc(Br)c1C(C(=O)N(C)CCC1CCCO1)NC(C1CC1Cl)=O c1(NC(CC(C)N(C(C2(C=C)CCC2)=O)C)=O)cccc2cc[nH]c12 C#CC1(C(=O)NCC2SCCS2)CCN(C(C2CC(=O)CCO2)=O)C1 CCC(CC)(CC)C(=O)NCC(C)(CSC)NC(N1CC(OC)C(OC)C1)=O C1(CN(C)C(=O)C2CC2)CCCN(C(=O)C(C)(F)c2ccon2)C1 Cc1cc(C)cc(C=CC(=O)NCC(O)CNC(c2cc(=O)cc[nH]2)=O)c1 C1(C2CCN(C(=O)Cc3cccc(O)c3)C2)(NC(CC2C(C)=NOC2=O)=O)CC1 C(CCN=c1[nH]c2ccc(O)cc2s1)NC(C1CCCN(C)C1=O)=O c1(SC)ccc(NC(=O)NC2CC(Nc3ccnc(C)c3)C2)cc1Cl c1(C(N2C(C(CNC(C3C(C)C3)=O)(C)C)CCCC2)=O)cc2c(cn1)COCC2 Cc1cc(C(=O)NC(CNC(=O)C=Cc2nccs2)C2CC2)cc(C)n1 C1(C(=O)NC2C(NC(CCN3CCN(CC)CC3)=O)C2)CCC(NC(C)=O)CC1 C1(F)(C(=O)NCC2(OC)CN(C(c3cnc(O)c(Br)c3)=O)C2)CCCN(C)C1 N1(C(C2N(C(c3ccnnc3)=O)CC(=O)NC2)=O)CC2CCC1C(O)C2O C=C(CNC(c1ccc(C(C2CCCC2)CC)[nH]1)=O)CCNC(c1sccc1CO)=O Cn1nc2c(c1C(N1CCCC(F)C1)=O)CN(C(=O)C1CC1)CC2 N1(C(=O)OC(C)(C)C)CCCC(O)CC1NC(=O)NCCc1ccc(O)nc1 C1(CN(C(c2ccc(C#N)s2)C(=O)NC2CCCC2)C)CC(F)(F)CO1 c1(C(N2C(CNC(C3CC4(C3)CC(O)C4)=O)C=CC2)=O)c(F)cncc1Br c1(-c2c(C3(C(N4CCC(O)C4)=O)CC3)cccc2)cc(C2CCC2)cnc1F.CC(C)NC c1(C(=O)NC(CNC(c2nccc(Cl)c2F)=O)C2CC2)ccc2c(c1)CC2 C1(NC(COC2(C)CCOCC2)=O)CN(C(C2CCOC2)=O)Cc2ccnn2C1 c1(OC)ncnc(OC)c1C(=O)NCC(C1CCOC1)NC(c1sccc1C)=O C(C(CC(F)(F)F)NC(C1CC1C1CC1)=O)NC(=O)CN1CC=CC1 c1(C(N2CCC(NC(c3c(C)noc3N)=O)C(F)C2)=O)cccc2occc12 C(C)(CC(=O)N1CCCC1Cc1cn(Cc2ccno2)nn1)OC N1(C(CC=C(C)C)=O)CC(CNC(c2cnn(CCF)c2)=O)C(F)(F)C1 Cc1cnc(C(N2CCN(C)CC2C(N2CCOC(C)(C(C)C)C2)=O)=O)cc1C Cn1ccc(CC(N2CCOCC2)=O)n1.N12CCC1C2NC(=O)C(F)=C1CCCC1 Cc1cc(F)cc(C)c1C(N1CC(NC(=O)C(C)CC(C)C)C(C#N)C1)=O C=C(C)CCCC(=O)NC1CC2(C1)CC2NC(c1cc(C2CC2)on1)=O C1(C(N(CC(C)OC)CC)=O)C=CCN(C(=O)CN2CCCNC2=O)C1 CCC(C)N(OC)C(=O)c1ccoc1NC(=O)C(=O)NC1CC1 c1(C(N(CC(C)NC(c2cc(C#N)ccn2)=O)C)=O)ccnc2c1CC(=O)N2 c1(OC(C(C)C)C)cc(CNC(C23COCC2C3)=O)ccn1 N1(C(C(COC)NC(C)=O)=O)CCC2CCCC(C1)N2C(=O)C(c1cncn1C)=O C1(NC(=O)CC2CCCCCC2(F)F)CN2CCC1c1ccccc12 CCCC(C(=O)NCC1(O)CN(C(=O)CSC(F)(F)F)C1)OC C#Cc1ccc(C(N2CC(NC(=O)CCCn3ccnc3C)CC2C)=O)o1 c1(C(N2C(CC(=O)NCC3C(C)NC(=O)CC3)CC2)=O)cnn2ccccc12 C1(NC(c2c(C)cnc(F)c2)=O)CCN(Cc2cccc3[nH]ncc23)CC1(C)C C1(CN(C(c2cnc(C(F)F)cn2)=O)CC)CCN(C(=O)CSS(C)(=O)=O)CC1 C1(CC=C)(NC(c2cnncc2NC)=O)CCN(C(=O)C(F)C(C)C)C1 N1(C(C2C(C)C2)=O)CCC(NC(C)(CO)c2ccco2)C1 N1(CC(C)NC(=O)CC2CC3CCC2O3)CCN(C(=O)C=CCO)CC1 C1(CC(=O)NCC(C(C)C)NC(c2ncsc2C2CC2)=O)CCC(C)(C)CO1 CCCC(O)C(=O)NC1CCN(Cc2nccn2CC)C1 c1(C(=O)NC2CC(N(C(C3(CC)CCCO3)=O)C)C2)onc(C)c1C CS(=O)(=O)c1ccc(C(=O)NC2CC2NC(=O)C2=CCS(=O)(=O)C2)nc1 c1(C(=O)NCC(CNC(c2cc(CC)cn2C)=O)O)n[nH]c(C(C)C)c1[N+](=O)[O-] N1(CC)CCN(C(=O)Nc2cccc3cccc(C)c23)CC12CCOC2 C1(CNc2nc(C)nc(O)c2)CC2CCC1N(C(C1(CO)CCOCC1)=O)C2 c1(CC(=O)NCCCCC2CN(C(C3CC(C)OC3)=O)C2)ccccc1[N+](=O)[O-] c1(C(=O)NCC2C(NC(C(C)C3CC3)=O)CC2)ccc2c(cnn2C(F)F)c1 C1(NC(C=C(CCC)C)=O)CN(C(=O)CC2CC(C)C2)CC12CCC2 c1(C(N2CCC(NC(CCC=C=C)=O)CC2)=O)c(OC)ccnc1OC C(=O)(C1=CC2(CCOC2)C1)NCC1CC(NC(Cc2cn(C)nc2Cl)=O)C1 C1(CNC(c2n[nH]c(C)c2C)=O)CCCC2(CCN(C(C3CCCC3)=O)CC2)O1 C1(C(=O)Nc2c(C)ccc(C)c2)CCCN1NC(=O)CN1CCCC1 N1(C(C(C)SCCCC)=O)CCCC2CN(C(C3(C4(O)CCC4)CC3)=O)CC12 C(CN=C(NCC(C)(C)C1CCC1)NCC1(C(F)(F)F)CCCCC1)SC C1(C2CCC2)CCCN1C(=O)C(C)SC.C(C)(=O)NC C(CC(=O)NC1CC2CCC(C1)N2C(c1ccc(C2CC2)o1)=O)(C(F)(F)F)OC c1(C(=O)NCC(CC=C)NC(=O)Cn2ccnn2)ccnc(OCC(F)F)c1 c1(OC)cc(C)c(C(N2CCCC2)CNCC(C)OC(C)=O)c(F)c1 N1(C(CSC(C)(C)C)=O)CC(CNC(=O)CN2CCOCC2)(OC)C1 N1(C(CC2(C)CC2(F)F)=O)CCC2(CC1)C(NC(C1CCC1)=O)CS2(=O)=O c1(C(=O)NCC(CC)NC(C2CC(=O)N(O)C2)=O)ccc2c(C)cc(O)nc2c1 C1(NC(C(C)(C)SC)=O)CC(C)N(C(=O)C(C)OC2CCCCC2)C1 c1(C(=O)NCC2CN(C(Cn3ncc(C#C)c3)=O)CC2C)cc(F)cc(C)c1O C1(NC(c2ncc(C=O)o2)=O)C2CC3C(C2)C13C(=O)NC1CCNCC1 CC(=O)CCCC(=O)N(C)CC1(O)CCCN(C(=O)CCC(=O)c2ccc[nH]2)C1 CN1CC(NC(c2ccc(CNC(=O)CCNC(N)=O)o2)=O)C2(CC2)C1 C1(C(C)C)C(C(=O)NCCn2ccnn2)CCN1C(c1csc(CO)n1)=O N1(C(c2c(CC)nns2)=O)CCN(C(c2coc(CS(C)(=O)=O)n2)=O)C(CO)C1 C#CCCC(O)C(=O)N1CC(C2(NC(=O)CCN3CCCC3=O)CCCC2)C1 CC1Cc2cc(F)ccc2N(Cc2cncnc2O)C1 C1(CNC(C2C=CCN2C(=O)CCc2cnoc2)=O)CC2(CCO1)CC2 c1(NC2CCN(C(CCSC)=O)CC2CO)ncnc2cc(OC)c(OC)cc12 CC1(CNC(=O)C(=O)NCC2CC2)CCCN1C(=O)CNc1ncc[nH]1 c1(N(C)Cc2ncc(CC)s2)nc(N(C)CCF)nc2scnc12 C(=O)(C(CO)C(F)(F)F)NC(C(=O)NCCOCC)CCSC N1(C(CSC)=O)CC(=O)CC1C(N(C)CC1CC(C(F)F)C1)=O Cc1[nH]nc(C(N2CCN(CC(=O)N(CCCF)C)CC2)=O)c1Cl c1(OCCC(=O)N(C(CNC(c2occ(C)c2)=O)C)C)cccc(C)c1C C=CCCC(F)(F)C(=O)N1CCCC1CN(C)C(C1CCC(SC)CC1)=O c1(NC(CC(=O)N(C(C)(C)C)CCN(C)C)=O)cc([N+](=O)[O-])cc(Cl)c1Cl N1(C(COCc2cc(C)no2)=O)CCC(C)C(CNC(c2cc(CF)on2)=O)C1 c1(OC)cc(C(c2ccncc2)COC)c2cccc(OC)c2n1 O=C1CCC(CC(=O)NCC2CCN(C(C3(F)CC=CCC3)=O)CC2)CN1 c1(C(N(C(C)CNC(C2(c3cccnc3)CC2)=O)C)=O)cc2n(n1)CC(F)C2 N1(C(=O)Nc2ccc(OC)cc2)CCC2(C1)CN(CC(O)CC(F)(F)F)C2 c1(CC)ncncc1C(=O)N(C1CCCC1)CCNC(=O)CC1CC1 c1(C(N2CCC(F)(CNC(COCCC)=O)C2)=O)cnc2c(C)cccc2c1 C1(NC(C(C)(C2CC2)NC(C)=O)=O)CCCCN(C(C2CC(F)C2)=O)C1 C(c1nc2ccccc2[nH]1)=CC(=O)NCC1CN(C(c2cnc[nH]2)=O)CCO1 Cc1ccc(SCCCSCC(C)C)cc1.c12nc(nn1-c1ccccc1)SC2 CCCC(C)(O)C(=O)N1CCC(C(=O)NC(CC(C)C)C(=O)N(C)C)O1 O=C1CCCC(C(=O)NC2C=CC(CNC(C3(F)CC3c3ccccc3)=O)C2)O1 N1(C(C2(CC=C)CCC2)=O)C2CCC1CC(CNC(C1CCCOC1)=O)C2 C1(N(C(C2CCCCO2)=O)CC)CC(=O)N(C(C)C2CC2)C1 CCC(C)(C)CCCC(=O)NCC1OCCC1C(=O)NCC(c1ccccc1)O Cc1n[nH]c(=NC2CC(OC(C)(C)C)C(OC)C2)cc1C1CC(C(=O)O)C1 CCC(=O)CCC(=O)NC1COCC1C(=O)NOCCOC(C)C c1(C(=O)NCC2CN(C(C(COC)OC)=O)C3(C2)CCC3)ccc(C#N)c(C)c1 N1(C(C(C2CCC2)NC(c2c(C)cc(N)cn2)=O)=O)CC(C2=NOC(C)C2)C1 CC(C)C(F)(CNC(=O)C1=CC2C=CC1C2)C(=O)NCC1(C)CC2(CC2)C1 c1(CNC(c2c(CS(C)(=O)=O)non2)=O)nc2cc(F)c(F)cc2[nH]1 N1(C(C2C(C)CCOC2)=O)CCN(C(c2ncc(F)cn2)=O)C(CC(F)(F)F)C1 c1(C(=O)NC2CCCN(Cc3cc(OC)ncc3)C2)ccc([N+](=O)[O-])o1 c1(OC)cc(C(=O)NCC2C(C)CCN2C(=O)CCCC#N)sc1Br C12(CNC(C(=O)N(C)C)=O)CCC(CNC(C3CC4(C3)CC4F)=O)(CC1)CO2 C12(NC(c3cc(CCC)ncc3)=O)CCN(C(c3nncn3C3CC3)=O)CC1C2 C1(N(C(=O)Nc2ccc(F)cc2)CCOc2ccc(Cl)cc2)CCCC12CCNC2 c1(C(=O)NC2CCC(CCNC(C(=O)NCC3CC3)=O)C2)ccc2cnsc2c1 C1(NC(=O)CCC2CC2(F)F)CC12CCN(C(C1(CF)CCC1)=O)CC2 Cc1cc(O)ncc1C(=O)N(CCCNC(=O)CCCc1cncs1)C1CC1 c1(NC(N(CCC)C(c2ccccc2OC)C)=O)cc(C(F)(F)F)ccc1F c1(NC(c2n(C(CC)C)nnn2)c2ccncc2)ccccc1SCC(C)CO C1(OC)CC(CCNC(c2cnc(CC(C)C)s2)=O)N(C(c2cccc[n+]2[O-])=O)C1 C1(F)(C(=O)NCCCOC)CCCN(C(C2(F)CC2)=O)C1 c12ccccc1C2.c1(C(C)NC(=O)C(=O)NC2CCCS2)ccccc1Br c1(OCCC(=O)NCCCCCN(C(C=C(CC)C)=O)C)cc(C)ccc1CC C(CCN=c1[nH]cncc1Br)N(C(CC1(C)CC1(F)Cl)=O)CCC1CC1 Cc1nc(C(C)C)oc1C(=O)NCCC1CN(C(c2cnc(=N)[nH]c2)=O)C1 c1(C(C)C)ccc(C2CNC(=O)N2)cc1.c1(C(N2CCCC2)=O)cc(C#N)no1 c1(C(=O)NCCC(CC)(CC)NC(CSCC=C)=O)ccc(F)c2c1CCC2 c1(C(N(CCNC(c2cnnn2C2CC2)=O)CC)=O)cc(C)n(C2CC2)c1C C1(NC(C(F)=CCC)=O)CCN(C(=O)C(Cc2ccsc2)NC=O)C(C)C1 Cc1cc(CC(N2CCOC(CNC(c3ncnc(C)c3C)=O)C2)=O)cc(C)c1 N1(C(c2cnco2)=O)CC2(C1)CN(C(C1(CC3CC3)CC1)=O)CCO2 Cc1cc(C(N2CCC(C)(CNC(C34CCCCC3C4)=O)CC2)=O)c(N)cc1F c1(CC(=O)NCCC2CCN(C(C(C)c3ccco3)=O)C2)cc(F)cc(Cl)c1 C1(C(=O)OC)CC2(CC(NC(=O)CCSC3CCCCO3)CCO2)C1 CCS(=O)(=O)c1cccc(C(=O)NC(C)CCCNC(=O)CNC(=O)C2CC2)c1 c1(NC(c2cc(C(=O)NC3CC3)no2)=O)cccc(OCCCN2CCOCC2)c1 c1(C(CC)NC(=O)CNC(=O)CNC(c2cc(COC)on2)=O)cnn(C)c1 C(=O)(CN=c1cc[nH]cc1)NC1CC(NC(C=Cc2ncn(C)c2)=O)C1 C(CCC(=O)NCCCCNC(C1(CCO)CC1)=O)NC(C)=O c1(C(N2CCC(F)(C(N3Cc4ccncc4C3)=O)C2)=O)cccc2cnccc12 N1(C(c2n(C)c(Cl)cn2)=O)CCOCC(NC(=O)C=CC2COC(C)(C)O2)C1 Cc1cc(=NCC2SCCS2)[nH]c(N2CC3CCC2C(CO)C3)n1 c1(C(N2CCC(C(N(S(C)(=O)=O)CC=C)=O)CC2)=O)cnc(OC)c(C)c1 N1(C(C(C2CCN(C(C(C3CCC3)OCC)=O)C2)F)=O)CCC=CC1CC N1(C(CSCCOC)=O)CCC(N(CC=Cc2ccncn2)CC2CC2)CC1 C12(C(N3CC4(N(C(=O)CC5(CO)CC5)CC4)C3)=O)CC3CC(CC1C3)C2 c1(C(N2CC(C(C(=O)NCCCC(C)(C)O)O)C2)=O)cc(F)ccc1O CN1CCC(C(=O)NCc2n[nH]cc2C(N2CCC(N3CC(O)C3)C2)=O)CC1 C(CNC(c1c(C)nn(CC(F)F)c1C)=O)(C(C)C(C)C)NC(CCOC)=O CCC(C)(C)CC(=O)NC(C(=O)NC1COC2(CCC2)C1)C1(C)CC1 C(C(=O)NOCC1CC1)(C1CCCO1)NC(C(CN(C)C)O)=O C(=O)(C1CCCc2cncn21)NC(C)CNC(c1cc(N)ccc1F)=O c1(C(=O)NCCCC(C)NC(=O)C(C2CCOC2)C)nc(F)ccc1Cl C(N=c1[nH]c(=NCCc2csc(COC)n2)c2ncccc2[nH]1)c1ccn(CC)n1 N1(C(CC2(NC(C)=O)CC2)=O)CCC2(CC1)CCN(C(c1ccnc(C)c1C)=O)C2 c1(C(N2CC3CC(CC(NC(CN(C)CC)=O)C3)C2)=O)cccc(S(C)(=O)=O)c1 c1(CN(CC(c2ccccc2)=O)CC)cccnc1Br Cc1ocnc1-c1cn(CC(=O)O)nn1.C123CC(C1)(C2)NC(=O)C3 C1(C(=O)NC2C(CCC)C2)(NC(=O)CC2CCOC2)CC(O)C1 C=CC(O)C(=O)NC1CC(CCNC(C2CC=CCC2)=O)C1 c1(C(c2n(CC)nnn2)NCc2cc(C)ccc2C)cc(Cl)nc(Cl)c1 c1(C(=O)NCCCC(C)NC(c2c(C(C)C)occ2)=O)ccc([N+](=O)[O-])o1 c1(CC(=O)NC(CNC(C(C=CCCC)O)=O)C(C)(C)C)c[nH]c(=N)nc1O c1(CC(=O)N(C)CCNC(C2(C#N)CC23CCC3)=O)ccc(S(N)(=O)=O)cc1 N1(C(c2c(C)ccc(OC)n2)=O)CCC2CN(C(=O)CSC3CC3)CCC2C1 C1(NC(CC=C)=O)(CNC(c2cnc(C(C)C)nc2)=O)CCCCC1C c1(C(C(=O)N(C)CC2CCCN(C(C3C(C=C)C3)=O)C2)C)nc(F)ccc1Cl c1(C(=O)NCC2C(NC(C(CC)(C)O)=O)CC2)cc(NC(C)=O)ccc1N.N N#Cc1ccc(C(=O)NCC2CCCN2C(c2ccc(S(N)(=O)=O)o2)=O)cc1F C1(C2CCC2)(C(N2C(CNC(c3snnc3C)=O)CC(OC)C2)=O)CC1(F)F C(C(F)(F)CCC(=O)NCC1CCCN1C(N)=O)n1cc(C2N(C)CCCC2)nn1 N1(C(C(c2cccnc2)SC)=O)CCC(NC(=O)CN(S(C)(=O)=O)C)C(C)(C)C1 C1(NC(CC(=O)N(C)C)=O)C2CC(O)C1N(C(=O)C=Cc1cnc[nH]1)C2 c1(C(N2CCCC(NC(c3c(C)scc3)=O)CC2)=O)ncnc2c1cnn2C C(=O)(C(F)(F)C(F)F)N1CCC(OCCNC(C23C(C(=O)OC)(CCC2)C3)=O)CC1 Cc1nccnc1C(=O)N(C)CC=CC(=O)NCC1(F)CCN(C)C1 C12(COC)CC(NC(c3cscc3OC)=O)(CN1C(C1CCCOC1C)=O)C2 C(=O)(C(C)CN(C(=O)CCc1cn(C)nn1)C)N(CCCOCC)C C1(CC(=O)NCC(CC)(C)NC(=O)CNC(c2cnoc2C)=O)CCCCN1C c1(CNC(=O)NC2CCCC(C#C)C2)cc(OC)c(O)c([N+](=O)[O-])c1 c1(C(=O)NC2(CCNC(C(F)=C(C)C)=O)CC2)ccc(Oc2ccccc2)cc1 CCC(C(=O)OC)C(=O)NC1C2CCN(C(=O)Cc3ccccc3C)C12 c1(C(=O)NC2C=CCN(C(Cc3ccc(C)s3)=O)C2)ccc([N+](=O)[O-])cc1F C1(NC(c2nc(Cl)c(Cl)s2)=O)CCCC12CN(C(C1CC3(CCOC3)C1)=O)C2 C1(O)(CCNC(CCNC(C2C(C)=C2)=O)=O)CCN(C(c2cc(C)c[nH]2)=O)CC1 C(CCC(=C)C)(C(=O)NC1CCN(CC)C1=O)NC(COCC#C)=O CCC(C)C(O)C(C)C(=O)NCC1(F)CCN(C(c2cc(C)cc(C)n2)=O)C1 CCS(=O)c1ccccc1C(=O)NCCC(C)NC(c1cncc(C(N)=O)c1)=O N1(C(Cn2nc(C)oc2=O)=O)CCN(C(=O)C(C)OCC(C)C)C(CC2CC2)C1 Cc1ccc(=N)[nH]c1C(=O)NC1(CNC(C2CC2C(C)C)=O)CCOC1 N1(C(C2CC(C)C2)=O)CCN(C)C(C(N2C3CSCC2C3)=O)C1 C(=O)(CC(O)CN(C)C)NCCCOC1CC(NC(CCCOCC)=O)C1 C1(OC)(CNC(c2csc(C(F)(F)Br)c2)=O)CCCN(C(C(C)(C)C)=O)C1 c1(C(C(=O)NCCC(=O)NCCOC)N(CC(C)C)CC#N)csc(CO)n1 c1(CC(=O)NCC2CCN(C(c3nccc(C)n3)=O)C2)n[nH]c2ccccc12 C1(CNC(C(C)(O)C2CC2)=O)CC2CCC(C1)N2C(c1cnnn1C1CCC1)=O C(C(C)CC(=O)N1CC(F)(C(=O)N(C(C)CSC)C)C1)OC c1(NCCCNS(CC)(=O)=O)cc(=NC2COc3ncc(Br)n3C2)[nH]c(C(C)C)n1 C(=O)(C1=CCCC1C)NCC(CC)NC(=O)COCC1CCCC1 C1(CCNC(c2c(OCC)scc2)=O)CCN(C(=O)C(C)OC)CC1 c1(CC)nc(C)c(C(=O)NCC2C(NC(C3SCCS3)=O)C=CCC2)o1 c1(C(N(CC(C)NC(c2n(CC)ncc2)=O)C(C)C)=O)cc(C)c(O)c(C)c1 CC1CN(C(c2cn(-c3ccc(Cl)cc3)nn2)=O)CC1NC(=O)CCC1CCC1 C1(CNC(=O)CSC(F)F)CCCC2(CN(C(C34CCCN(CCC3)C4)=O)C2)O1 N1(C2=CC(C(=O)OC)=NC=NC2)CCC(C)C(NC(=O)CCC(F)(F)F)C1C N1(C(c2c(-c3n(C)ncc3)n[nH]c2)=O)CCCOC(CNC(C2CC2C#N)=O)C1 CC1=CCC(N=c2ccnc(NCC3CC3c3ccc(F)cc3Br)[nH]2)CC1 c1(-n2ncc(C)c2)ccc(C(N2CC(N(C3CC(F)(F)C3)C)C2)=O)cc1 C(CC(C(=O)NC(c1ccc(C)s1)=O)N(C)C)OC.C12CC1NC2=O N1(c2nnc(C)o2)CCCC(C(C)NC(c2ocnc2-c2ccccc2)=O)C1 C1(C(=O)NCCNS(C)(=O)=O)(NC(C2CC23CCC3)=O)CC(O)C1 N1(C(Cc2nc(C)c(C)s2)=O)CCC2(CCCN2C(=O)CC2CCCC(=O)N2)C1 CCC(C(C)C)C(C(=O)NCCOC)N(C1CCS(=O)(=O)C1)C(C)C C(=O)(C1=NOC(C)(C)C1)NCC1CCN(C(CN(C2CCCC2)C)=O)CC1O N1(CCn2c(C)ncc2)CCn2cc(C(=O)NCc3ccc(O)cc3)nc2C1 OC1CCC(N=c2nc(N3CCC=C(Cl)C3)c3[nH]ccc3[nH]2)C1 S(=O)(=O)(c1ccnc(S(C)(=O)=O)c1)N(C(CCC(C)C)C)C c1(CNC(C2CCC(CCCC)CC2)=O)cc2ccccc2nc1Cl c1(C(N2CC(CCO)(NC(CCc3scc(C)n3)=O)C2)=O)cc(C)n(C(F)F)n1 c1(CCC(=O)NCCC2(CNC(=O)C(O)CC3CCCC3)CC2)nc(C2CC2)no1 C1(C(C)CNC(C2CCN(C)C2)=O)CCN(C(=O)CN2CCC2)CC1 N#Cc1ccc(NC(=O)NCCC(=O)OCC(O)C(F)F)cc1 C(C)(C(C(=O)NC1CC(CNC(c2cnc(C)s2)=O)C1)N(C)C)OC C(CC(C)(C)C)(C(=O)NCCC1CCCN(C(=O)C(C)=C2CCCC2)C1)OC C#Cc1ccc(C(=O)NC2CCCC2NC(=O)CCc2nnc(S)nc2O)cc1 N1(C(CSCC)=O)CCCC(C)(CNC(c2ncc(C)cc2OC)=O)C1 CCCCCC(O)C(C)C(=O)N1CC(NC(C2CCS2(=O)=O)=O)CC2(CCC2)C1 Nc1c(F)cc(F)c(F)c1C(N1CC(CNC(=O)CC2CCOCC2)C(O)C1)=O C1(C(=O)NC(CCOCCOC)=O)CCN(C(c2cc[nH]c2)=O)CC1O c1(C2(N(C(C(=O)N(c3cncc(Cl)n3)CCF)=O)C3CC3)CCC2)c(F)cccc1F c1(NC(CN(C2CS(=O)(=O)CC2O)C)=O)cc(Br)cc2c1OCO2 C12(C(N3CCCC(c4cnco4)C3)=O)COC(CF)(C1)C2 C(=O)(C1OC(=O)c2ccccc21)NCC1C(NC(CS(C)(=O)=O)=O)CCC1 N1(C(C(CCCNC(c2cncc(Cl)c2)=O)O)=O)CCc2sccc2C1 c1(C(=O)NCCC2N(C(CN(CC(C)(C)C)C)=O)CCC2)cnnc(C2CC2)c1 c1(OC)cc(=NCCOCc2ccccc2)[nH]cc1C.C12CC1C(=O)O2 C#CCC(C)(C(=O)NC1CCN(C(C)=O)C1)NC(c1c[nH]c(=NC)s1)=O c1(OCC(=O)N(C(C)CN2CCCC2)C)cc(Br)ccc1Cl C1(C)(C(=O)NC2C(NC(C=C(C)C(C)(C)C)=O)CC2)CC(=O)N(C)C1 N1(C(C=C(CC)C)=O)CCC(NC(c2cc(COC)cn2C)=O)C(CC)C1 c1(C(N2CCC(C(O)C(F)F)C2)C(=O)NCCOC)ccn(C(C)C)n1 N1(C(C(c2ccccc2)OC(C)=O)=O)CC2(CC(NC(=O)CCF)CO2)C1 C(C(=O)Nn1cccn1)n1cc(CNC(c2[nH]cc(CC)c2)=O)nn1 N1(C(C2CCC(C)(F)CC2)=O)CC2CCCC(NC(=O)Cc3cccs3)C2C1 C1(NC(c2c[nH]c(Br)c2)=O)CCCN(C(C2CC(O)CN2)=O)C1 C12(C(N3C(C(=O)NCCn4cccn4)(CC)CCC3)=O)CCC(N=[N+]=[N-])C1C2 c1(OCCOC)ccc(C(=O)NC(CNC(=O)CC2CCCC(=O)N2)CC)cc1 C1(CCNC(C2(COCC)CC2)=O)CCN(C(=O)C(=Cc2c[nH]cn2)F)C1(C)C C(C)(CNC(=O)C(C(C)C)NS(C)(=O)=O)(C(C)C)NC(Cc1c(C)non1)=O c1(NC2(CNC(c3ccc(N(C)C)cc3)=O)CC2)nc2cccc(F)c2s1 C1(C)(CNC(C2C=C(C)CS2)=O)CCCN(C(=O)C(C)NC=O)C1 C1(N(C)C)CN(C(C2CC2c2ccccc2)=O)CC1CNC(=O)CCc1ccon1 c1(Nc2cccc(-n3ncc(C)c3)c2)nccc(=NC2CNC(=O)C2)[nH]1 C(=O)(C1CCc2nccn21)N1CC(NC(C2CN(OC)C(=O)C2)=O)C2C1CCC2 CCCC(C(=O)OC)C(=O)NCCC(C)NC(c1ccc(CC)o1)=O C1(C(=O)NC(c2cc(F)ccc2F)CC)CC2(C1)CS(=O)(=O)C2 C12(CNC(CSCC=C)=O)CC(NC(C3CC3Cl)=O)(C1)C1(CCOCC1)O2 N1(CC(=O)NCC2CCN(C(CCC(=O)NCC)=O)CC2)CCCCC(O)C1=O c1(OCCOC)cccc(CO)c1N.N12CCN(CC1)C(=O)C(=O)NC(C)(C)C2 N1(C(C2CCCCS2)=O)CC(CNC(C2(c3cc[nH]n3)CC2)=O)CC12CCC2 c1(CN(C(C(N2CCC(CN3CCC(C)CC3)CC2)=O)=O)CC)cc(C)ccc1I C1(NC(C(C)(C)Oc2ccccc2Cl)=O)CC2CC1N(C(=O)Cc1ccsc1)C2 c1(OC)ccc(C(=O)NCC2CCCC(NC(=O)C=C3CCC3)C2)cc1OC CCC(C)(C(=O)NC1CCC(CCNC(C23CC(C(C)C)(C2)C3)=O)C1)OC C(CN=c1cc(C)nc(C(C)C)[nH]1)(C1CC1)NC(C=C(C)C(F)F)=O CC1=CCN(C(C2CC3CC3N2C(=O)C(C)N=[N+]=[N-])=O)CC1 CC(C)C(F)(F)CC(=O)NCC1C=CC(NC(=O)C(N2C(=O)CCC2=O)C)C1 C1(NC(c2n(CC=C)nnn2)c2ccn(CCC)n2)CCCC(C2CC2)C1 C1(NC(CCNC(N)=O)=O)CCCCC1CC(=O)N(C1CCCOC1)CCF CCC(C)(C(=O)NC(c1ccc(CNC(=O)C=Cc2cn(C)cn2)cc1)C)OC C1(CC)CCCC1(C)C(=O)NCCN(CCCN1CCCCC1C)C1CC1 N1(C(C(C(C)C)O)=O)CCCC(O)(CNC(c2[nH]ccc2C2CC2)=O)CC1 N1(C(c2ncc(CC)s2)=O)CCN(C(c2cc(Cl)ccc2F)=O)CC1CCO N1(C(Cc2c(C)occ2)=O)CCN(C(=O)CC2CCCNC(=O)C2)C(CCO)C1 Cc1cc(F)c(-c2ccccc2)nn1.c1(N)nccc(N2CCCC2)n1 c1(N(CC(COC)O)C)ccc(S(=O)(=O)NCCN(C)C)cc1F.C1CN1 C=C(C)CC(C(=O)N1CCCC(CO)C1)OC.C1(=O)NOCC12CC2 C(N=c1[nH]c(=N)[nH]c(=NCCSC2CCSC2)[nH]1)c1ccc(OC)c(C)c1 CCCCCCC(F)C(=O)NC(C)CCCCNC(C1(C)CCN(C)C1=O)=O C(=O)(C1=C(SC)CCCC1)NC(CN(C(=O)Cc1scnc1C)CC)C c1(C2(C)CC2C(=O)NCC2(C(N3CC(C#N)C3)=O)CC2)ccccc1 C1(C(=O)NCC(C)(C)NC(c2cn(CCCC#N)nn2)=O)CCCC(F)C1 C1(CC(=O)NC(COCCCOC)C(C)C)CCCN1C(=O)OC CCCCS(=O)(=O)CC(=O)NCCC1CCCN1c1nnc(CC)c(CC)n1 c1(C(N2C(C)CC(NC(CCN(CC)CC)=O)C2)=O)ccn2ccccc12 c1(NC(C=C)C)[nH]c(=NCc2cc(Cl)ccc2Cl)nc2c1cnn2C c1(N2CCC(C)C(NC(c3ccc(F)o3)=O)C2)ccn2c(Br)cnc2n1 C1(C(=O)NCC2(O)CCCN(C(C=C(C)C)=O)C2)CCc2nc[nH]c2C1 c1(C(=O)NC(C(N2C(CC(C)C)COCC2)=O)C(C)O)cn2c(n1)CCC2 Cc1cc(C(=O)NCCOCCNC(=O)C(c2ccccc2Cl)(C)C)n(C)n1 Cc1c(C(=O)NCC2(CCNC(c3c[nH]nc3-c3ccsc3)=O)CC2)ccn1C c1(C(CC)C)nccc(=NCCNc2cc(F)c(OC)c(F)c2)[nH]1 N1(C(CCCSC)=O)CC(CNC(c2cc(C(N)=O)cn2C)=O)CC(C)C1 c1(CNC(CCC=CC)=O)cccc(C(N2CCC2C2CCCCC2)=O)c1 N1(C(C(C)OC)=O)CCC(CN(C)C(C2(NC(=O)NC(C)C)CCCC2)=O)CC1 C(CCC(C)C(=O)N1CCC(O)(CNC(c2ccc(OC)cc2NC)=O)C1)OC Cc1nn(C2CCOCC2)c(C)c1N(C(=O)OC)C(c1ccccc1)n1cccn1 CCC(C)CC(=O)N1CCC(CCC(=O)NCC(O)CC(C)C)CC1 c1(C(N(CCNC(=O)CC2COC(=O)C2)CC)=O)cccc(F)c1C#N C=Cc1ccc(C(=O)N(CCCNC(C2CC2(C)C(N)=O)=O)CCO)cc1 C#Cc1cncc(C(=O)NCC2CC(C)(C)CN2C(=O)C#CC2CC2)c1 C1(NC(=O)Cc2csc(-c3ccco3)n2)CC2CN(C(=O)C(F)C3CC3)CC2C1 C(C(O)CCNC(=O)CC1CS(=O)(=O)C1)NC(COCCC#C)=O C(C(=O)N1CCC(C(=O)NOCCc2ccccc2)O1)c1n(C)cnc1 c12cccc(c1)OCCNC(=NC)NC2.C=CCOC1CC1 c1(C(N(CCC(C)NC(CCCOCCC)=O)C)=O)ccc(F)c(O)c1 c1(C(N2C3CC(NC(C4(C)CC4)=O)C(C3)C2)=O)cc2cccn2c(C(F)(F)F)n1 N1(C(c2c(C)cc(F)cc2)=O)CCC2CN(C(=O)C#CC3CCCCC3)CCC2C1 C1(C(=O)NCCC(C)NC(c2c(Cl)ccc(Cl)c2Cl)=O)CCn2cnnc2C1 C1(NC(C23CC(C)C2C3)=O)CCC(NC(=O)CSC2CCS(=O)(=O)C2)CC1 N1(C(CCCN(C(C)=O)C)=O)CC(NC(=O)C=CC2C(C)C2(Cl)Cl)CC1(C)C c1(C(N2CC3CN(C(c4c(C)ccnc4)=O)C3C2)=O)n[nH]c2c1CCC2C C1(CNC(Cc2c(C)n(C)nc2)=O)CCC2(CCC2)C1NC(c1cc(F)c[nH]1)=O C1(C(N2CC(COC)(CNC(=O)CN=S(C)(C)=O)C2)=O)CCc2nnnn2C1 C(N=c1[nH]c(=NC2CC=CC2)[nH]c2c1SCC2)C1(Br)CCSC1 CC(CCC(=O)NCC1CCCS1)NC(=O)CCC1(C#N)CCC1 C1(C)(C(=O)NC(C)CNC(c2ccnc(NC3CCC3)c2)=O)CC2CCC2C1 CC(C)(C)S(=O)(=O)CC(=O)N1CC2CC2(NC(=O)CNC(c2ccsc2)=O)C1 c1(SC)ccc(Cl)c(C(N2CCCC2CN(C)C(c2cc(C(C)=O)cs2)=O)=O)c1 C(C)(C(=O)NCC1CCC(NC(c2ccnn2C2CC2)=O)C1)(C1CC1)OC N1(C(CNS(N)(=O)=O)=O)CCOC2CN(C(c3cc(Cl)c(F)cc3F)=O)CC12 C1(NC(c2cc(-c3cccnc3)on2)=O)CC2CC1N(C(c1sccc1F)=O)C2 c1(OCCN)cccc(-c2nc(C3CCCO3)n(CCOc3ccccc3)n2)c1 N1(C(c2c(CC)scn2)=O)CCCC(NC(=O)C=Cc2ccnn2CC)C1C CCC(C)CCC(=O)OC(c1cc(O)ccc1C)C C(=O)(C(C(C)(C)C)n1ccnn1)NCC1CC(NC(c2c(OC)nccc2)=O)C1 C=Cc1cc(C(N2CC(C)CCC2CNC(c2cnsn2)=O)=O)cc(F)c1 C1(CC(N2CCC(N(CCC)C(c3n[nH]cc3Br)=O)C2)=O)C(C)(C)C1(C)C c1(CN(C(c2n(C)ncc2)=O)Cc2cc(Cl)ccc2F)cc(C(=O)O)ccc1O C(CCCC(CO)NC(c1ccc(C)cc1Cl)=O)NC(c1c(CC)nco1)=O N1(C(c2cn(C)cc2C(F)(F)F)=O)CC2(C1)CN(C(C1(C(F)F)CCC1)=O)C2 CC1CC2(CC(NC(C3CN(C(=O)CC4C=CCCC4)CC3(C)C)=O)C2)C1 C1(C(N(CC(C(C)C)C)C)=O)CC12CCN(C(=O)CNCc1nc[nH]n1)C2 c1(OC)c(C)csc1C(=O)NCC(C1CC1)N(C)C(C1CC(F)(CO)C1)=O CN1CCC2CN(C(c3ccc(C(=O)N=S(C)(C)=O)cc3)=O)CC2C1 C1(N(C(=O)CNS(C)(=O)=O)C)CCCCN(C(=O)CN2C(=O)CNC2=O)C1 C(=O)(C(C(C)(C)C)n1cc(CN(CCO)CCOC(F)F)nn1)NC(C(C)C)CCO Cc1cn2c(C)c(C(=O)NCC3(C)CN(C(=O)CNC=O)CCO3)nc2s1 c1(C(=O)OC)ccc2c(c1)OC(CNCCN1CCC(c3nncs3)C1)C2 N1(C(C(C(C)CC)NC(c2c(CC)c[nH]c2)=O)=O)CCOCC(F)(F)C1 C1(CC(=O)NC2C3(C(=O)OCC)CC3CC2)CC2(CO1)CC1(C2)OCCO1 CC(CC1CCC1)C(=O)NC1CC1CNC(=O)CCCOC1CCOCC1 Cc1ccoc1CNC(=O)C(c1cnn(C)c1)NC(C1CC1C(C)C)=O CCCC(CC)C(=O)N1CCN(C(=O)C=Cc2ccsc2)C(c2cn[nH]c2)C1 C1(CC(=O)N(CC(C)NC(C2CC(C(=O)NC3CC3)C2)=O)C)CCCCCC1 CCCC(CCC)C(=O)NCC(C)(C)OCC(=O)NCCN1CC=CC1 c1(C(=O)NCC(CN(C(=O)COCc2nc[nH]n2)C)(C)C)cc(C#N)ccc1O C(C)(C)(CC(=O)NCCn1cnccc1=O)N(C(=O)C(F)C1CCOC1)C N1(C(Cn2c(=O)sc(C)c2C)=O)CC(CO)C2(C1)CN(C(C1CCS1(=O)=O)=O)C2 CC(CNC(C1CCN(C)C1=O)=O)CC(=O)N1CCC(CF)C1 c1(C(N2C(CNC(c3ccc(Cl)o3)=O)COCC2)=O)cn2ccsc2n1 C1(C(C)C)CC(NC(=O)CCOCCN(C)C(C2C=CCCC2)=O)CO1 C(C(CO)c1ccco1)(NC(C(C)OCCC#C)=O)CNC(=O)COCCOC N1(C(C(CC)C(=O)OC)=O)CCCC2(C1)CN(C(=O)C(=Cc1ccncc1)C)C2 c1(CCC(=O)N(CC(=O)NCC)C(C)C)cc(Cl)no1.C(C)(C)(C)O N1(C(COCCCC)=O)CCC2(CCC(CNC(C3CC3(F)F)=O)OC2)CC1 c1(CC)cc(C(=O)NCCCC2CCCN2CC2CCC2)nn1CCO c1(C(N(C=O)CC2COC(C3CC3)C2)=O)cc(Br)c2c(c1)OCCO2 C1(CC(=O)NCc2c(OC)c[nH]n2)CCCCN1C(=O)C(C1CCCCC1)F CCCCC(C)CCC(=O)NC(C)(CNC(c1ncc(C#N)cc1Cl)=O)CO c1(CSCC(CO)F)cccc(F)c1I c1(CC(N2C3CCC(C3)C2CNC(=O)C(F)(F)CO)=O)cccc2nsnc12 N1(C(c2ccc(C)c(O)c2C)=O)CCN(C(C2C3COCC23)=O)CC12CCC2 CCC(C(=O)N1CC(CCOC)C1)OC.C12(CC1(F)F)C(=O)N2 c1(C(=O)OC)ccc(N(C)CCN(C(=O)Cc2ccn(C(C)C)n2)C(C)C)cc1C N1(C(CCC(C)SC)=O)CCCC(C)(CNC(C23CC2COC3(C)C)=O)C1 Cc1ccc(C(=O)NC2CCCC(NC(C3(C)CC4CC4C3)=O)C2)cc1Cl C1(NC(C(=O)NCc2cccc(CN3CCCC3)c2)=O)CCS(=O)(=O)CC1 N1(C(C2CCCCS2)=O)CC2CC(C1)N(C(c1ccnn3ccnc13)=O)C2 CC1CCC(NC(=O)CCC(=O)NC(c2ccccc2F)C)N1C C1(C(=O)NCC2(O)CN(C(C(=Cc3ccncc3)C)=O)C2)CCc2nccn2C1 C1(C(=O)N(C)C(c2ccccc2Cl)c2cn(C(C)C)nn2)(CC)CCCC1O C1(C(=O)NC2CC(C(F)(F)F)C2)CN(C(=O)CSc2ccoc2)CC12CC2 N1(C(CCC=C)=O)CC(C(=O)Nc2ccc(OC)cc2C)N2CCC1C2 C=CC(CCC)CC(=O)NCCC(O)CNC(c1c(C)nccc1C)=O CC1CC(=O)NCCN1C(C1CCCN1C(=O)COCc1ccsn1)=O C(=O)(CCCS(N)(=O)=O)N1C(C)CC(CNC(Cc2c(CC)n[nH]c2CC)=O)C1 N1(C(CSCC)=O)CCN(C(c2ccc(N)c(CO)c2)=O)CC1CF CC(C)C(CCN(C)C(C1(NC(N)=O)CC1)=O)Nc1nncn1C Cc1cncc(C(N2CCOCC2CC(=O)NCc2ccns2)=O)c1 N1(C(C(C=C)c2ccccc2)=O)CC(NC(=O)CSCCN(C)C)CC(C)C1 C=CC1(C(=O)Nc2cccnc2)CCN(C(=O)C(=Cc2ccccc2)C)C1 c1(CC(=O)NC2(CO)CN(C(CNC(C(CC)CC)=O)=O)C2)cnn2c1OCCC2 C1(CCNC(CCN(S(C)(=O)=O)C)=O)CCCN(C(C2(C)CC=CC2)=O)C1 c1(CNc2nc(Br)cc(C(C)C)n2)cc(O)ccc1[N+](=O)[O-] CCCC(CNC(=O)CCc1cnn[nH]1)C(=O)N(C)Cc1ccc(O)cc1 c1(C(N(C2CN(C(c3c(C(C)C)c[nH]n3)=O)C2)C)=O)c[nH]c2cnccc12 CC1(C)C(CC(=O)NC2(C)CC(O)(CO)C2)CCN1C(c1cc(CO)[nH]n1)=O c1(CC)ccnc(C(N2CC(OC)C(NC(=O)CSc3n[nH]c(C)n3)C2)=O)c1 c1(C(=O)NC2CCN(C(CC(C)C3CC3)=O)CC2CO)nn(C)c2c1CCC2 c1(C(C)CC(=O)N(C(C)CCNC(c2cncs2)=O)C)ccccc1F c1(C(=O)NC2C=CC(C(=O)Nc3ccc(O)c(F)c3)C2)cc2cnccc2[nH]1 Cc1oc(C(C)(C)C)cc1C(=O)NCCCNC(=O)Cc1cc(Cl)sc1Cl CN1CCCC(C(=O)NC2CC(CC(=O)N(c3nc[nH]n3)CC3CC3)C2)C1 N1(C(CN(C2CCCC2)C(=O)OC(C)(C)C)=O)CC2CC2C1C#N.C(=O)O CC(CC(F)F)C(=O)NC(C(N1CCC(F)(CO)C1)=O)C1(O)CCC1 C(=O)(C(C)(C)NC(c1ccccc1)=O)N(CC(CNC(C(F)=C(C)C)=O)C)C CC1C(NC(c2n[nH]cc2Br)=O)CCCN1C(=O)CCC(=O)c1ccc[nH]1 CCC(F)(F)CC(=O)NC1CC1CNC(c1cc(C(=O)OC)cs1)=O C(CCN=C(NCc1ccco1)NC(C1CCC(CC)O1)C)OCCS(CC)(=O)=O CN1CCCC(N=c2[nH]c(=N)[nH]c(=NCC3CC3C3CCOCC3)[nH]2)C1 N1(C(c2c(C)cn(C)c2)=O)C2CCC1CN(C(C1CC1CF)=O)C2 c1(C(=O)NCC(C(C)C)NC(C2CC(F)C(=O)N2)=O)nn(C)c(C(F)F)c1Cl N1(C(C2CCCN(C(=O)OC)C2)=O)CCCC12CCCN(C(=O)C(F)=C(C)C)C2 c1(C(N(C2CCN(C(C3CC(C)C3)=O)C2)CCO)=O)cc(C#N)ccc1O CC1(C)COc2cc(NC(c3nnnn3C3CCC3)C3CC3c3ccsc3)ccc21 O=C(C1=CC2(CCN(C(=O)C(O)Cn3cncn3)C2)C1)NCc1ccc(O)cc1 N1(C(c2cc(SC)oc2)=O)CC(C(=O)NCc2cc(C)cc(F)c2)CCC1(C)C N1(C(CC(C)OC)=O)C2COCC1CC(NC(=O)CN(C)Cc1ccccc1)C2 C(=O)(CC(C)c1cnn(C)c1)CCN(CC(CC)NCC#N)C(=O)C(=O)N(C)C C=CC1(CC(=O)NCC(O)C(C)O)CN(C(=O)CCC2CCCO2)C1 C1(C(N(CCC(c2cccs2)NC(=O)C=CCN2CCC2)C)=O)CCC(=O)NC1 c1(OC)ccnc(C(=O)NC(CO)C(C)NC(=O)CC2SCCCO2)c1OC c1(C(=O)NCC2CCN(C(C3C(C)(C)COCC3)=O)C2)cnc2[nH]ccnc1-2 CCC(C)(CCC(C)C)C(=O)NCC12CCCC1N(C(=O)Cn1cnnn1)CC2 c1(NC(=O)NC2CN(C(C(C)N(C)C)=O)CC3C2C3)cnc(O)c2ccccc12 Cc1oc(CNC(C2CC3CCC2O3)=O)nc1C(=O)NCCc1cn(C)cn1 C1(C(=O)NCCC(CCNC(CCc2c(C)noc2Cl)=O)C)CCC(C)(C)CO1 c1(C(N(CCN(C(C2C(C3C(C)C3)C2)=O)C)C)=O)cc(F)c(F)c(F)c1F c1(C(N2C(CNC(C=C(C)CCc3ccccc3)=O)CC2)=O)cnc(Cl)nc1 c1(C(N(CCCCN(C(=O)Cn2ccc(CC#N)n2)C)C)=O)ccc(CO)cc1 C1(CC(N2CC(O)(COC)C2)=O)CN(C(c2cc(OC)cs2)=O)CCC1C C1(CC(=O)NCC2CN(C(c3cnc(C)o3)=O)C2)Cc2cc(Br)ccc2C1=O CC(C)(CCCNC(c1cc(Br)no1)=O)C(=O)NCC1CC(C(F)(F)F)C1 c1(C(N2CCC(NC(C(C(C)C)C)=O)C23CCC3)=O)ccc2ncncc2c1 N1(C(c2cc(CC)n(C)n2)=O)CCN(C)C(CC(=O)N(CC)OC)C1 c1(SC)cc(C(N2CC(C(C)NC(c3ccc(O)cn3)=O)C2)=O)ccc1F C1(OCC)CCC(n2cc(CCCNC(=O)C(c3ccc(C)cc3)O)nn2)CC1 C(CCN=c1c(C#N)c[nH]c2c(F)ccc(Cl)c12)N1CC(C)(C)C(CO)CC1 CC1(C)C(NC(=O)C(=O)NCCC2CCCCC2)CCN1C(=O)CCN1CCC1 C1(O)(Cn2cc(CCCC)nn2)CCCN(C(=O)Cc2cccc(Cl)c2Cl)C1 C1(OCCONC(C(C=C)(F)F)=O)CCCCCC1C(=O)NC(C)=O C1(C)(C(=O)NCC(C)(C2CCC2)NC(=O)C(C)(C)n2cnnn2)C=CCC1 c1(C(=O)NC(CC)CNC(c2c[nH]c(C)c2)=O)cn(C)c(=O)nc1O CCCCC(C(=O)N1CC2C(C(N)=O)C2C1)N(c1ccc(C(=O)OC)c(C)n1)CC C1(NC(CC=C=C)=O)CN(C(c2csc([N+](=O)[O-])c2)=O)C2(CCOC2)C1 C1(CC)CC(C(N2CC(NC(=O)Cn3cc(Br)c(=N)[nH]3)C(C)C2)=O)CC(=O)N1 c1(OC)cc(C(N2CCC2CNC(=O)CCF)=O)cc(F)n1 C1(N(C(CC2(OC)CC2)=O)CCO)CCN(C(c2c[nH]nc2OC(C)C)=O)CC1 c1(OCC)cccc(NC(=O)C2=CCOC2)c1C C=C(C)CCC(=O)N1CC2C(CNC(c3c[nH]nc3OC)=O)C2C1 S(=O)(=O)(c1ccc(NC2(CSC)CCCC2)c(C#N)c1)NCCS(CC)=O N1(C(C(CCNC(C2COCC2C(N)=O)=O)OC)=O)CCOC(C)(C2CC2)C1 C12(NC(C3N(C(=O)NC)CCC3)=O)CCC(CC1)N(C(C1CC1C(C)C)=O)C2 N1(C(CC(C(=C)C)OCC)=O)CCC2(C1)CN(C(c1c[nH]c(Br)c1)=O)CCO2 c12cccc(F)c1OC(CC)CNC(=O)CC2.C(C)(C)(C)OC(C)=O CC(C)=C=CC(=O)NC(C)CC1CCN(C(C2CC2(c2ccccc2)C)=O)CC1 C1(NC(C(C(C)NC(c2ccsc2)=O)C)=O)CC2C(O)C(O)CC12 C(=O)(C1CCCc2c1ncn2C)N1CCN(C)CC1CNC(c1nsnc1O)=O C1(CNC(C2C(CC)C2)=O)CCCN(C(=O)CCC2CC2)CC1 c1(C(=O)NCC2CCC(C(=O)Nc3cc(Cl)cnc3O)O2)cc(F)cnc1O N1(C(C2CCC(C(C)C)CC2)=O)CCC(NC(C2CC(C)(F)C2)=O)CC1C C1(C(C)NC(C2(CCO)CC2)=O)CCCN1C(=O)C=Cc1cn[nH]c1 Cc1ccc(F)c(C(=O)NC(C)C(=O)NC(c2cccnc2)CO)n1 CCC(C)(C#N)C(=O)NCC(C)NC(=O)C(c1ccnc(C)c1)(C)C N1(C(c2cc(C)ns2)=O)CCCN(C(=O)COCC2CCCOC2)C(C(C)C)C1 C(=O)(CCCC(=O)C(C)(C)C)N1CC(CC)N(C(=O)CN2C(=O)CCC2=O)CC1 N1(C(C(c2ccc(C)cc2)=O)=O)CCC2(CCC2)C(NC(=O)CSC(C)C)C1 c1(C(=O)NCC2(CNC(=O)Cc3ccsc3)CC2)cnc(-c2ccccc2)o1 C(=O)(C(CNC(c1cnn(C)c1Cl)=O)CC(C)C)NCc1c(CC)onc1C C1(CC(=O)NC(C)CN(C)C(c2cc(C(N)=O)no2)=O)CC2(CCC2)CCO1 N1(C(c2c(CC)con2)=O)CC2CC2(C)C1 C12(CC(=O)NCC(C)(C)C)CCC1CN(C(=O)CC1(O)CCOC1)C2 C1(CC)COC(C)CN1C(=O)CC1C2CCCC2N1C(=O)C=C=C(C)C N1(C(CC2CC(=C)C2)=O)CC(NC(=O)C(C)(C)F)C(C)C1 NC(=O)CCCCC(=O)N1CCC(C(CO)NC(=O)CCCCC#N)CC1 CC(C)CCC=CC(N1CCC1C(=O)N(CCCF)C)=O N1(C(C(CC)C)=O)CC2CCC(CNC(c3ncc(F)c(OC)n3)=O)(C2)C1 N1(C(C2(C=C)CC2)=O)CCC2CCN(C(c3cc4c(C)n[nH]c4nc3O)=O)C2C1 c1(C(N2CC(C)(C(=O)NC(c3ccccc3)C)C2)=O)ccc2occc2c1 c1(OC)ccc(C(=O)NCCCOCCNC(c2ccoc2Br)=O)c(F)c1 N(C(=NCCCOC)NCCNc1ccccc1C(C)C)C(C(OC)OC)C C1C(F)(F)CCC(=O)N2CC(C)(C)C2c2cn1nn2.Cc1nn[nH]c1C(=O)O CC1CC(C)SC1CN1CCC(OCCCC(F)(F)F)CC1 c1(C(CN(S(=O)(=O)CC23CC(CCO2)C3)C)C(F)(F)F)c[nH]c2ccccc12 N1(C(=O)NC(c2ncc(-c3ccccc3)[nH]2)C(C)C)CC(F)C(F)C1 C(CC(C(C)C)NC(=O)Cc1csc(NC=O)n1)N(C(CC(=C)C)=O)C S(=O)(=O)(c1ccc(OCCN(C)C)c(F)c1)NC(=O)NCc1ccc(OC)cc1 C1(C(N2CC(c3ccc(CCO)cc3)C2)=O)C2CCCCCCC12 N1(C(c2cc(SC)oc2C)=O)CC2CCCC2(NC(c2cnc(C(C)C)s2)=O)C1 c1(CC(=O)CNC(C2(NC3COCOC3)CCCCC2)=O)ccccc1Br C(C(=O)N=c1cco[nH]1)NC(C1CN(C(c2ccnc(F)c2F)=O)C1)C C1(CC)CCC(C)CCN1C(c1cc(Cl)ncc1Br)C(=O)NC(C)(C)CC C1(CC)(CC)CCCN(C(=O)CN(CC(C)C)C(c2cc[n+]([O-])cc2)=O)C1 c1(C(=O)NC2C3(CN(C(C4CC(SC)C4)=O)C3)CC2)cc(C)c(C)nc1C Cc1cc(CC(=O)N(C)Cc2snnc2C)cc(C)c1 C1(C(=O)NCC2CCN(C(c3c(OC)cc(O)nc3)=O)C2)Cc2ccccc2S1 C(=O)(C(CC(C)(C)C)N(C)CCN1CCCCC1)NC(C)C C1(NC(C2C(CC)C2)=O)CCC2CN(C(=O)Cc3cnn(C)n3)CC2C1 C=CCCCCC(=O)NC1(CCOC)CCN(C(C2OCCOC2C)=O)CC1 Cc1sc(O)nc1C(=O)NCC(CO)NC(=O)CC1CCC(=O)CC1 C1(C(=O)NC(CNC(c2ccnc3cc[nH]c23)=O)CO)Cc2cc(Cl)ccc2O1 C1(C(N2CC(CC=C)(C(=O)NCCc3nncn3C)C2)=O)CCN(C)C1=O Cc1ccc2scc(C(=O)NC3CCN(C(=O)CCc4cc[nH]n4)C(C)C3)c2c1 N1(C(C(N2CC(C)OC(CO)C2)=O)=O)CC2CCCN2CC1C(=O)O c1(C(=O)NCC2OCCC2C(=O)NC2C3CCCC2CC3)cc2ccccc2o1 c1(CC(=O)NC(C)C=CC(=O)NCC2(C)CSC2)nocn1 c1(C(N(CCCNC(C2(COC)CNC(=O)C2)=O)C)=O)nc(OC)cc(OC)n1 C1(OC)CN(C(C2CCCN2C(=O)CCCc2cc[nH]n2)=O)CC1(C)C C1(CNC(C(c2cccc(C)c2)O)=O)CCN(C(c2ccnc(C)n2)=O)C(C)C1 C1(NC(c2ccn(CC)n2)=O)C2CCCN(c3ncncc3I)C2C1(C)C C(=O)(CC(C)CCC(=O)NCCCCCCNC(=O)CCOC1CCCC1)OC c1(C(=O)NCC(=C)CCNC(=O)CCF)cnc(C)c2c1COC(C)(C)O2 c1(C(N2CCN(C(C3CC(CC)C3)=O)CC(O)C2)=O)ncnc2c1ccn2C c1(NCc2cc(SC)ncc2)ccc(S(=O)(=O)N2CC3CC3(CO)C2)cc1Cl c1(CC(=O)NCC2C(NC(c3c(CC)ocn3)=O)C2)ccc(OC(C)C)cc1F N(C(=NCCN1CCCCCC1)NCC1CCCC1(F)F)C(C)C C1(N(C(CN(C(C)=O)C)=O)C)CN(C(=O)N(S(C)(=O)=O)C(C)C)CC1O C(=O)(C(C)(C)CCOC)NCNC(CN(C(CN)C(F)F)C(CC)(C)C)=O N1(C(C2CCC(=C)CC2)=O)CCCC(C)(C)C1CNC(=O)CC(=O)NC CCC(CC(=O)NCc1cccnn1)NC(c1nccc(OC)n1)=O C(=O)(C(CCC(N)=O)n1ccnn1)NCC1CCN(C(CC(C)(F)F)=O)C1 N1(c2nc(=N)nc(N3CCCN(N4CCCC4)C3)[nH]2)CCC2(CC1)CC2CO C=CCC(C)(C)CC(=O)N1CCCCC1CNC(c1cc(C)cc(OC)c1C)=O N1(c2nc(C)nc(C)c2F)CCC2(CCN(C(=O)CCc3ccncn3)C2)C1 C1(C(N)=O)(CNC(C=C(C)C(C)C)=O)CCCC1.C1(=O)C(F)CC2CN1C2 CC(C(C)(C)NC(=O)C=Cc1cscn1)NC(c1cc(Cl)no1)=O N1(C(c2nc(C)sc2C)=O)C2CCC1C(CNC(C1CC(C)(F)C1)=O)C2 N1(C(CCCCC)=O)CCOC2(CCN(C(c3cccnc3C)=O)CC2)C1 CCC(CC(=O)NCC1CCN(C(c2ccnn2CCF)=O)CC1C)CC(C)C C(=O)(C(C)(O)C(C)c1ccccc1)NCC(C1CCCC1)NC(CCOC)=O c1(OC)ccc(C(=O)NCC2CCN2C(=O)CCCNC(C)=O)c(F)c1 c1(C(=O)NCC2CC(F)(CNC(C3CCC(OC)C3)=O)C2)ncnc2c1CCC2 Cc1ccc(CN2CC(NC(C3CCCN(C(=O)C4CC4)C3)=O)C2)c(F)c1F C1(C(=O)NCC(CCC)n2cccn2)CCCC(NC(=O)C(C)CCOC)C1 C1(NC(CN(C(C=O)S(C)(=O)=O)CC)=O)CCCCC1.OC C1(C(N2CC(CNC(C(C)(C)N(C)C)=O)CC2(C)C)=O)CCc2ccnn2C1 c1(C(=O)NCC(CNC(C2=CCCCC2C)=O)CO)c[nH]c2cccc(C#N)c12 C1(NC(c2cc(C(C)(F)F)n[nH]2)=O)CC(CO)N(C(C2CC2c2cccs2)=O)C1 Cn1ncc(C(=O)NC2CCCCC2CNC(C2(CF)CCOCC2)=O)c1F C1(CNC(c2c(Cl)cccc2)c2ccco2)C2(CCC2)C12CCC2 N#Cc1c(N2CCCC(CCNC(c3cscc3Cl)=O)C2)ncc2c1CCC2 C1(NC(c2cc(C(C)=O)sc2)=O)CC(OC)CN(C(=O)CCCn2cncn2)C1 Cc1ccc(C(=O)NCC(C)(C2CCC2)NC(C2CC3CCC2C3)=O)nn1 c1(C(=O)NCC2C(NC(c3cnns3)=O)C2)cccc2c3c([nH]c12)CCC3 CCC(C)(C(=O)N1CCC2CN(C(c3coc(C4CCC4)n3)=O)C2C1)C(N)=O C(=O)(C1=NOC(C)(C)C1)NCC1(CC(N2C(CC(C)(C)C)CC2)=O)CC1 C(=O)(C(O)C(F)(F)F)NCC(C(=O)N(CC(CCC)C)C)N(C)C c1(C(=O)NC2CC(NC(C3N(C(C)=O)CCC3)=O)C2)c(C)ccc2ccccc12 C(C)(C(CC(=O)NCC1(OC)CCC(C)C1)NC(C1(CF)CC(=O)C1)=O)OC C(C(C)C(=O)NC(C(C)(C)O)C1CC1)NC(CC1(COC)CC1)=O C(=O)(CC1=CCOCC1)N1CCC(NC(c2cnc(C(C)O)s2)=O)C1C C1(CCC)CN(C(=O)C(ONC(=O)CSC(C)C)C)CCO1 c1(C(=O)NC2C(CNC(CC(C)C3CCCCC3)=O)C2)ccn2nnnc2c1 CCCC(CCC)C(=O)NC(C(=O)N1CC(C(C)OC)C1)C(C)(C)C c1(C(=O)NC(C)CNC(C2(C)CC(F)C2)=O)cnn2c1NCC(C)C2 Cc1ccc2[nH]c(C(N3CCC(C)(CNC(=O)Cc4cn(C)nn4)C3)=O)cc2c1 c1(NC)ccc(C(=O)NC2(CC3CC3)CCC2)cc1[N+](=O)[O-] c1(C(=O)NCC=CCNC(C2(C)CCCO2)=O)ccnc(-n2ccnc2)c1 C1(C(=O)NC(c2ccc(OC(F)F)cc2)C(C)C)(OC)CCN(CC(F)F)CC1 CC(C)(CC(F)F)C(=O)N1CCCC(O)(CNC(=O)CCC2=CCCC2)C1 CC(C)CC(C)CNC(=O)CCN(C(=O)C=Cc1ccnn1C)CCCO c1(C(N(C)CC2N(C(c3n(CCC)ncc3)=O)CCC2)=O)c(OC)cccc1F c1(N(C)CC2CCCO2)nc(N2CC=CCC(C)(C)C2)c2cn(C)nc2n1 C1(CC)CCCC1(C)C(=O)NC1(C(N2C(C(=O)OC)C2C(C)C)=O)CC(O)C1 C1(CC)CN(C(c2cc(F)n(C)n2)=O)CCN1C(C1CCC(C)(C)C1)=O CC1CCC(NC(=O)C(N2CCOCC2)C)CN1C(C1CC2(CSC2)C1)=O N1(C(c2cc(OC)c(Cl)s2)=O)CC(C2CCCCN(C(c3ccnn3C)=O)C2)C1 N1(C(c2cn(CCC)nc2)=O)CC(NC(=O)C(F)=CC2CC2)C(SC)C1 C1(NC(COCC(=O)NC)=O)CN(C(=O)CCS(=O)(=O)NC)C2(CCC2)C1 Cc1cnn2ccc(C(=O)NC3CC(NC(c4nc(Br)cnc4N)=O)C3)nc12 c1(CC(=O)NCC(C)N(C)C(c2ncc(Cl)cc2Cl)=O)c[nH]c2cc(F)ccc12 C1(C(=O)NCCN(C(=O)Cn2nccc2C(=O)OC)CC)COC(C(F)F)C1 Cc1cc(O)nnc1C(=O)NC(C)(C)C1(C(=O)NC(C)(C)CCN(C)C)CC1 C1(NC(c2nc(C)sc2C)=O)CC(CNC(c2cn(C3CC3)cn2)=O)C12CCC2 Cc1nc(NC(C2CN(C(c3csc(-c4ccccc4)n3)=O)CC2C)=O)sc1C n1(C(C)C)cc(C(=O)NC(C2(O)CN(C(=O)Cc3cnn(C4CC4)c3)C2)C)cn1 C(=O)(C(F)C(F)(F)F)N1C(CN(C2CC(O)CN2Cc2ccccc2)C=O)CC(O)C1 C1(C(N2CCC(N(C(=O)C(C)SC)CCC)CC2)=O)Cc2ccccc2NC1=O c1(C(N2CC3CC3(C(=O)Nc3ncc(I)cn3)C2)=O)cc2ncccc2[nH]1 C1(C(=O)NCC2CCCN(C(C(CC)C)=O)CC2)CC2(C1)CC1(CC1)C2 N1(C(CC(CC)(C)C)=O)CCN(C(=O)Cc2ccoc2)CCC1C C1(C(N(CCN(CC(=O)NCCCC)C)C(C)C)=O)CCCCC1C c1(C(=O)NCC(C)NC(CC2(COC)CCOCC2)=O)cc2cccnc2[nH]1 C1(C)(C(N(C(CNC(CSCCC)=O)C)C)=O)CC(C(C)C)=NO1 C1(C(=O)NCC(CO)NC(C2CC=C(C)CC2)=O)=CC2C(=NNC2=O)C=C1 CCCC(CCC)C(=O)OC.N12CCC(F)(C1)C(=O)N1CCC(C1)CC2=O C(=O)(C1=CC2C=CC(C1)C2)N(C(C)CNC(c1ccc[nH]1)=O)C C=CCCCC(C(=O)NCCOCCN(C)C)NC(c1ccsc1CC)=O c1(OCC2CC(CC(=O)OCCn3cc(Br)cn3)C2)ccc(C(=O)O)cc1F c1(CCC)cccc(C(N2CCC(OCCNC(=O)C=C3CCCC3)C2)=O)c1 C1(NC2CCN(C(C)C)C2)CCCC(c2ccccc2)C1 c1(CC(=O)NC(C)C=CC(=O)NC2(CN(C)C)CCCCC2)cccc(F)c1O N1(S(C)(=O)=O)CCCc2cc(-c3nc(-c4ccncn4)no3)ccc21 N1(c2ncnc(CC)c2F)CC2CCC(NC(=O)CS(=O)CC)CC2C1 C(=O)(C(=O)N(O)C(C)C)NC(CC=C)CNC(c1cn(C(C)(C)C)nc1Br)=O N1(C(C2CCCC(C)C2)=O)CCCOC(CNC(c2ccnc(F)c2N)=O)C1 CC1(C)CC(C(=O)N(c2ccon2)C2CC2)CCN1C(=O)CCC(=O)C1CC1 c1(C(=O)NCCCN(C(c2nc(OC)oc2)=O)C2CC2)ccc([N+](=O)[O-])cc1 N1(C(C(C2CCOC2)NC(COCC)=O)=O)CC(C)C(O)C1 c1(C(N2CCCN(C(c3onc(C)c3C)=O)C(C)C2)=O)c(F)ccc2ccoc12 N1(C(C=CCC)=O)CCN(C(c2cnn(CC(C)C)c2C)=O)C(CO)C1 Cc1cc(C(N2CCC(CCCNC(c3cnc(=N)[nH]c3)=O)CC2)=O)cc(C)n1 C=CCCN=C(NCC1CC(C)(C)CO1)NCC1CCCC1CC C1(O)(CNC(c2n(C=C)ncc2)=O)CCN(C(C2(CCCC)CCCC2)=O)CC1 C1(CC=C)(NC(c2cn(C)cn2)=O)CN(C(c2cscc2Cl)=O)C1 C12(C(=O)N)CCCC1C2.C1CC(=O)N1.c1(C(=O)NCCOCCCSC)cccs1 CCCC(C)C(=O)NC(c1ccccc1)CNC(=O)C(N)=O N1(C(CCOCCN(C)C)=O)CCCCCCC1C(=O)NCc1ccnc(O)c1 O=C(C1=CS(=O)(=O)CCC1)NCC1(F)CC(CNC(c2cc(C3CC3)[nH]n2)=O)C1 c1(NC(c2n(CCOCC)nnn2)c2cc(Cl)cs2)cccc2nc[nH]c12 c1(C(C)(C)C)nnc(Cn2cc(CNCCCO)nn2)s1 c1(N2C(CNC(c3cnc(COC)s3)=O)CC3(CC3)C2)nc(C#N)ncc1Cl c1(CN2CCN(C(c3c(CC)nccc3)=O)C3C2C3)cc(OC)c(OC)c(F)c1 C1(CNC(CN2CCc3n(C)c(Br)nc3C2)=O)CC12CCOc1ccc(Br)cc12 CCC(CN(C)C)(c1nnnn1CC1CCOC1)NC1CCSC1 C1(NC(Cn2c(C)c(Br)cn2)=O)CC2CCC1N2C(C1(O)CC(C)(C)C1)=O C(=O)(C(CC(C)C)n1ccc(C2CC2)n1)N1CCC(CNC(C(C)OC)=O)CC1 Cc1nccc2c1CCN(C(=O)NC1CCCC13CCC3)C2 c1(C(=O)NC(CC(C)NC(c2coc(C(F)F)n2)=O)C)ccc2cccnc2n1 C(=O)(CCC(C)(C)F)N1CCC(CC(C)NC(Cc2c(C)noc2)=O)CC1 C1(N(C(C(C)Cc2cccnc2)=O)C)CN(C(=O)C=Cc2ncco2)CC12CC2 C1(C)(N(C)C)CCN(C(c2cc(C(N(C)NC(C3(CCO)CC3)=O)=O)no2)=O)C1 N1(C(COC(C)(C)C)=O)CCC(OCC(=O)NC2CCNC(=O)C2)C2CCC12 Cc1cnccc1C(=O)NCCCCN(CCCNC(=O)C(C)C1CCOC1)C c1(N(C)Cc2ccc(C)o2)nc(=NC2CCC(F)CC2)[nH]c2ccccc12 C(=O)(CCC(=O)NCCCC)N(CC(N)=O)CCCc1ccccc1F.C1(=O)ON1 c1(C(N(CC(C)NC(=O)Cn2cnc(=N)[nH]2)CC)=O)noc2c1CC(C)CC2 C1(CF)COCCN(c2nnnn2Cc2nc(C3CCC3)no2)C1 CCC(CC(C)C)C(=O)N1CC(OC)C(OC)C1CNC(C1(CO)CCC1)=O C(=O)(C1=NN(CCO)C(=O)CC1)N(C1CCN(C(C2C(=C)CC2)=O)C1)CCO Cc1nccn1CC(=O)NC1CC(C)(CNC(=O)CC2CC2)C1 c1(NC(C(N2CCC(N(C(C(C(C)C)SC)=O)C)C2)=O)=O)c(C)cccc1C C1(NC(C(C)OCC=C)=O)CCN(C(C2CCC(NC(C)=O)CC2)=O)C12CC2 C(=O)C(C)(C)CF.C(=O)(C(=O)N(CC)CC)N(CCNCC)CC N1(C(c2cn(C(C)C(C)C)nn2)=O)CC23CCCC2(C1)CN(CCCCCC)C3 c1(CC)cc(CC(=O)NC2CC(O)(CNC(=O)COC3CCC3)C2)on1 c1(C(N2C(C3(NC(CCSCC)=O)CC3)CCCC2)=O)ccn(CCO)c(=O)c1 C(C)(C(=O)N(CCC(=O)NCCC1CC1)CCOC)SCC c1(NC(CNC(C(=O)OC(C)(C)C)CC#N)=O)ccc(F)c(Cl)c1 CCCCCC(O)CC(=O)NC(C)(CNC(=O)CSc1nnnn1C)CC c1(C(=O)NC2C3CN(C(C(C=C=C)C)=O)C2CC3)c(C)nc2sc(C)nn12 c1(C(=O)OC)cc(Br)ncc1NC(=O)NCCCc1ccc(Cl)cc1Br c1(CC(=O)NC(CN(C(=O)Cc2cccnc2)C)(C)C)cc(Cl)ccc1Cl C1(NC(C(C2CC2)OC)=O)CCCCCN(C(c2csc(C)c2C2CC2)=O)C1 C1(CC(=O)NC2CCC(NC(CSCCC)=O)C2)CCCS(=O)(=O)C1 c1(NC2(O)CCN(CC(=O)O)C2)cc(C(F)(F)F)nc(C2COCCN2)n1 C1(NC(C=CCCC)=O)CCCCC12CCN(C(=O)C=Cc1cnc(C)s1)CC2 c1(C(=O)NC2(CC=C)CCN(C(=O)CN(C)CCOC)C2)ccc(S(N)(=O)=O)o1 Cc1ccc(=O)n(CC(N2CCC(NC(c3c(C)cncc3C)=O)C(F)C2)=O)n1 C1(O)(CCNC(c2cnc(C3CC3)o2)=O)CN(C(C2C3CCCC23)=O)C1 C(C)(C)(C(=O)N1CC(O)CCO1)C1CCN(C(C(C)OCCC(C)C)=O)C1 c1(C(N2CCC(NC(C(CC(C)=O)C)=O)C(F)C2)=O)cc(F)cc([N+](=O)[O-])c1Br Cc1cc(C(=O)NCC(C2CCC2)NC(c2c[nH]nc2C2CCOC2)=O)n[nH]1 N1(C(c2cc(C#N)[nH]c2)=O)CC(C2(NC(=O)CSc3nncn3C3CC3)CC2)C1 c1(C(N2CC(NC(CSc3nnc(C)s3)=O)C2)=O)cc(C(F)(F)F)ccn1 C1(C(c2cn(CCCC(=O)NCC(C)C(C)O)nn2)OC)CCC(F)(F)CC1 CCCC(C)(O)CC(=O)NCCC1(NC(c2ncc(Br)cc2C)=O)CCC1 c1(NC2(C(C)NC(=O)CCCNC(=O)C3CC3)CCC2)ncc(Br)c(O)n1 N1(C(=O)CCn2cnnn2)CC2CC1CN2C(c1cc(-c2cnccn2)ns1)=O C1(S(=O)(=O)NC(c2cc[nH]c(=N)n2)C)(c2cn(CC3CCN(C(N)=O)C3)nn2)CC1 C(=O)(CC(C(F)(F)F)N(C)C1CC1)NCC1=CCN(C(CCCOC)=O)CC1 c1(C(C)NC(=O)C(n2cc(CC3CCCCO3)nn2)C)nc(CC(F)(F)F)no1 c1(C(=O)NC2CCC(NC(C(C)NC(CC)=O)=O)CC2)nn(C)c(C)c1Br N1(C(CCC(=O)OCC)=O)CCN(C(=O)C2=NNC(=O)C2)C(CC(F)(F)F)C1 C(CCCCCCC(F)(F)F)N1CCCC(C(F)(F)F)(CC)CC1 N1(C(CCC2CC(C)C2)=O)CCCC1C(C)NC(c1nccn1C)=O C1(C(=O)NC(CC)CCCO)CCCN(C(=O)CC2CSCCO2)CC1 N1(C(C2CN(C)C2)=O)CCC2CN(C(c3c[nH]nc3-c3cccs3)=O)CC2C1 CC1(CS(=O)(=O)N2CC(CC3CCOC3)C2)COC1 c1(C(N2CCN(C(C(=Cc3cccnc3)C)=O)CC2)=O)nc(O)c(C#N)cc1C CCCCCCCCN(CC(N1CCC(CC2CC2)C1)=O)C(=O)Cc1cnsc1 S(=O)(=O)(c1cc(C)cnc1NCC1(SC)CC1)NC(CCC=C)(C)C N1(CC=C)CCC(NC(=O)C(CCF)NC(=O)CC2CCC(=O)C2C)CC1 c1(OCCC(=O)NCCN(C(=O)CCn2cccnc2=O)C)cncc(Br)c1 CS(=O)(=O)c1ccc(OCC(N2CC(C(=O)O)CC(F)(F)C2)=O)cc1 C12(NC(=O)CCc3cnoc3)CC(CNC(=O)CCc3ncco3)(C1)C2 Cc1nnc2n1CC(C(=O)NC13CC(NC(=O)CC4(CO)CC4)(C1)C3)C2 C12(CN(C)C(=O)OC(C)(C)C)CCN(C1)C2=O.n1(CC(CC)O)cc(CO)nn1 CCC(CC)C(O)CNC(c1ccn(CCNC(C2CCN(C)CC2)=O)c1)=O N1(C(C(C(C)C)O)=O)CCCCC12CN(C(c1csc(Br)c1)=O)C2 c1(CCC)nc(C(=O)NCC(O)CN(C)C(C2CC(N(C)C)C2)=O)co1 c1(C(=O)NCCCC2N(C(COCC(=O)NC)=O)CCC2)ccc(F)c(C)c1Cl c1(N2C(c3ccc(NCC)s3)CCC2)ccc2cc(S(=O)(=O)NC(C)=O)ccc2n1 c1(Cc2cn(C(C(=O)OC)C)nn2)ccc2c[nH]nc2c1.C12(CCC1)C(=O)N2 Cn1nc2c(c1C(=O)NCC1(CNC(C3CC4CCC34)=O)CCCC1)CCC2 c1(C(=O)NC2C(NC(CCC(=O)OC)=O)CCC2)cc(Cl)c(Br)cc1F C12CC(C)(C1)NC2=O.C1(N(C)C)CC(O)(CNC(=O)CCC2(C)N=N2)C1 N1(C(C2CC(=C)C2)=O)CC(C2CCCCN(C(=O)CCC3C(=O)ON=C3C)C2)C1 C1(C(=O)OC)CN(Cc2ccc(C)cc2Cl)CCC1O.C12(CCCC1)C(=O)N2 c1(CC(N2CC(CCCCNC(CNS(CC)(=O)=O)=O)C2)=O)c(C)nn(C)c1Cl Cc1c(C(=O)NC(C2(O)CN(C(C3CC(F)C3)=O)C2)C)ncn1C CCCCC(CN(C(=O)CC(C(F)F)NC(=O)CN1CCOC1=O)C)CC N1(C(C2=C(C#N)CCC2)=O)CCC2CCN(C(c3cc4ccncc4o3)=O)C2C1 Cc1cnc(C(=O)NCC2(O)CCCN(C(=O)Cc3nc[nH]n3)C2)cc1Cl C1(N(C(Cn2nnc(C)n2)=O)C)CN(C(=O)COCCN(C)C)CC12CC2 c1(C(=O)NC(C)CCCNC(c2cccnc2)=O)n[nH]c2c1CS(=O)(=O)CC2 CCN=c1[nH]c(C)c(C(=O)NC2(n3cc(-c4ccc(C(=O)O)s4)nn3)CC2)s1 C1(C(C)C(=O)N2CCC2)CCN(C(=O)CN2CCSCC2)CC1 N1(C(COCCCC)=O)CCC2(C)CN(C(=O)CCC(CC)CC)CC12 c1(C(=O)NCC(C)=CC(=O)NCC(N)=O)cc(C)ncc1C N1(C(c2c(Cl)cn(CC)n2)=O)CC(CNC(c2[nH]cnc2COC)=O)CC1(C)C C1(OC)CCC2(C(N3CCC(CCNC(=O)C(c4ccccc4)F)CC3)=O)CC12 Cc1nc2cc(C(N3CCCC(CNC(=O)CC4C(C)C4(F)F)C3)=O)cnc2[nH]1 N1(C(CC(=O)OC)=O)CCC(C(C)NC(=O)CCN2CCC(F)C2)CC1 C#CCC(O)C(=O)NCCC(C)NC(c1c(C)ncn1O)=O C1(CC(=O)N(CC(=O)OCC)CC#C)CN(C(C)=O)CC1C(F)(F)F C(=O)(C1=CCCSC1)NC.c1(CC)noc2c1CC(=O)N1CCOC(C1)CC2 C1(N(c2ccccc2)C(=O)NC(C(C)NC(=O)CCC#N)C)CCCCC1(F)F c1(NC(=O)C(F)CC2CCOC2)cc(NCCOCC(=O)O)ccc1[N+](=O)[O-] C1(C(=O)NCC2CCC(C)C2)CC2(CCC2)CN1C(=O)CC1CC2CC2C1 Cc1ccc(F)c2c1CN(C(c1cccc(Cl)c1C)C(=O)NCCCF)CC2 N#CC1=C(C(=O)NC2CC(O)CN(C(c3c[nH]cc3Br)=O)C2)CCC1 C1(CC(N2CC(N(C)C(c3cc(Cl)c[nH]3)=O)C2)=O)CCCCC1O N1(C(c2c(C)nc(O)cc2)=O)CCCC(C2CC2NC(c2ccnnc2C)=O)C1 C1(C(=O)NCCO)CCC(C)CN1CCNC(CSCc1c(C)noc1C)=O c1(C(=O)NCC(CNC(c2nccn2C)=O)OC)ccc(=O)n2c1CCC2 c1(NC)c(C(=O)NC2CCC(CNC(=O)CC(C)C(C)C)CC2)cccc1F c1(C(=O)NC2C(C)CN(C(=O)Cc3cc[nH]c(=N)c3)C2)ccc2c(c1)OCCO2 n1(CC(N2C(C3CCN(C(CC=C)=O)CC3)CCCC2)=O)nc2c(n1)CCCC2 N1(C(CCc2c[nH]c(=N)[nH]2)=O)CCC(NC(=O)C2=CCSC2)C(CO)CC1 CC(CNC(=O)CSC1CCC1)CNC(C1CC1(Cl)Cl)=O C1(=O)CC(c2ccccc2)CO1.C(C(O)CNC(=O)COC(C)(C)C)N(C)C C(=O)(C(C)(O)C(C)(C)C)NC(CC)CNC(=O)CCc1csc(C)n1 c1(OC)ncc(Br)cc1CN1CC2CC2(C(=O)Nc2ccc(O)cc2C)C1 c1(C(C)NC(C(Cc2cn[nH]c2)NC(C(C)=C2CCCC2)=O)=O)ccccc1F C1(C(=O)NCC2C3CN(C(CC4(C)OCCO4)=O)CC32)CCC(C2CCCO2)O1 C1(N(C(c2n(CC(=O)OC)ncc2)=O)C)CCCN(C(=O)C(CO)N(C)C)CC1 C(=O)(C(F)C(C)C(F)F)NCCC(C(=O)NCC(COC)(C)CO)(F)F c1(C(=O)NC(C)CNC(C2(CO)CC2)=O)ccnn1C(F)(F)F O=C(C1=CCCOCC1)N1CC(OCCC(=O)NCC23CCCC2C3)C1 c1(SC(c2cscn2)=O)ccccc1.C1(C(=O)N2C3CC3C2)(CCF)CCC1 C(C(CC(=O)N(C1COC(C)(C)C1)C)NC(C1(c2cc[nH]n2)CC1)=O)OC c1(CC)nc(C)c(C(=O)NC2(C(=O)NCC3CC(=C4CC4)C3)CCCC2C)o1 c1(C(C)(C)NC(=O)NC(C(C)N2CCCC2)C2CC2)ccccc1 c1(C(=O)NCCCCCNC(C2(n3cncn3)CC2)=O)sc(Cl)cc1Cl Cc1ccn(CC(=O)NCC2CCN(C(=O)CC3CCOC(C)(C)C3)C2)c(=O)c1 C(=O)(C1=NN2CCC(C)N=C2N1)NC1CN(C(C(=C(C)C2CC2)F)=O)C(C)CC1 c1(C(N2CCC(NC(C(COC)OC)=O)C(F)C2)=O)ccc2cc(O)ccc2c1 C#CC1CCN(C(=O)CC2CN(C(=O)CCc3cn[nH]c3)CC2C)C1 c1(C(=O)NCCN(C(C2CC(OC(F)F)C2)=O)CC)ccc(Cl)c(C)c1O C(=O)(C(CCC(N)=O)NC(C1CCNC(C)CC1)=O)NCC(C)C C=CC1(CC(=O)NCCN(C(=O)CNc2ccncc2)CC2CC2)CCCCC1 CN1CCC(OCCN(C)C(C2(N(C(=O)CC3CCCC3)C)CC2)=O)CC1 C1(NC(C2CCC23CCC3)=O)CN(C(=O)C=Cc2cccc(F)c2)C2(CCC2)C1 C1(C(=O)NC2(CC#C)CC2)CC2CC1CN(C(=O)C(c1cncnc1)C)C2 CCC1CCC(=O)N2CCN(CC2CC)C(=O)CN1.C(=O)(CN(C)C(C)C)NC C1(CNC(c2ccc(C(C)C)s2)=O)C(C)CCN1C(c1c[nH]c(C#N)c1)=O C(=O)(CCCCC(C)C)N1CCC(C2N(C(C(C(C)C)NC(C)=O)=O)CCCC2)C1 CCC(CC)CCC(=O)NC(C)C(N1CCC(COC)C1)=O c1(NCC(N2C(C(N3CCC(CSC)CC3)=O)CC(O)C2)=O)ccc(C)c(C)c1 CC(C)C(C(C)NC(c1ccccc1F)=O)NC(c1ncccc1C(F)(F)F)=O CC1(C(=O)N2CCC(C3(NC(=O)CC4=CCC4)CC3)C2)CCCc2ccccc21 C(CCC(C)(C)C(=O)NC1C=CCN(C(=O)CC2(C)CC2)C1)OC CC(C)C(F)C(=O)N1CCSCC1CCNC(C1COC(C)C1)=O N1(C(C2C(CC)CCC2)=O)CC(O)(C2CCN(C(c3cnn(CC)n3)=O)CC2)C1 N1(C(N)=O)CC(O)CC1C(N1CCCC(C(=O)N(C)C)C1)=O.C1(=O)COCCN1 C1(NC(=O)CCc2cncs2)CC12CC(NC(=O)CC1COCC1O)C2 C1(C(=O)NCC2N(C(Cn3c(C)nnn3)=O)CCC2)(C(F)F)CC2(CC2)C1 C(=O)(C(F)C(F)(F)C(F)(F)F)N1CC2CC(C)N(C(C(CCCC)O)=O)C2C1 C1(NC(C(C)CN(C)C)=O)CC2(CCC(NC(=O)C(F)CC3CCCC3)CC2)C1 Cc1ncncc1C(=O)NC(C)C(C)(C)NC(C1CC(c2ccccc2)C1)=O N1(C(=O)OC(C)(C)C)CCN(C(C2CC23CN(C(=O)CCSCC(=O)O)C3)=O)CC1 N1(C(C)=O)CS(=O)(=O)CC1C(=O)N(CC(O)CN(C(=O)C#CC(C)C)C)C c1(CNC(C(C)OC(C)=O)=O)ccc(C(N2CCOCC2CN(C)C)=O)nc1 N1(C(C2N(OCC)CCC2)=O)CC(C(=O)OC)CC(C)C1 C(CCCC(=O)NC(C)(CNC(=O)Cc1cn(C2CC2)cn1)C1CCC1)SC C12(COC)CC(C(=O)NCC3(O)CC(NC(C4(CO)CCCCC4)=O)C3)(CO1)C2 N1(C(C2C(NC(C)=O)CCOC2)=O)CC2(C1)CN(C(=O)C#CC(=O)N(C)C)C2 N1(C(=O)OCC)CCC(C(C)(C)C)(OCC)C1.n12cc(nn1)NC(=O)C2C C1(CC)CCCN(c2nnc(-c3cnc(OC)cn3)n2CCOCC2CC2)C1 CC1(C2CC2)CCCN1C(=O)COCCNC(=O)Cc1nc[nH]n1 N1(C(C=CCOC)=O)CCC2CC2(C(=O)N(c2ccnn2C2CC2)C)CC1 C1(C)(C(=O)NCC(C)(C2CC2)OC)CCCN(C(c2nccc(C)n2)=O)C1 C(=O)(C(F)(F)C1=CCOCC1)N1CC(NC(c2nocc2Br)=O)C2(C1)CC2 Nc1cc(F)ccc1C(=O)NC1CC(NC(=O)Cc2c(Cl)cccc2Cl)C1 Cn1nc(C(=O)NC(CO)CCCNC(c2cncc(N)n2)=O)cc1F C1(N2CC(CN(C3CCC3)C(=O)OC(C)(C)C)C2)CCC2(CCC2)O1 C1(N(C(COCC(C)C)=O)C)CCN(C(c2n[nH]c3c2CCC3)=O)CC12CC2 C(C(C)(O)C(C)C)NC(C1C(CNC(COC)=O)CCC1)=O N1(C(C2CC(F)(F)C23CCCC3)=O)CCCC12CCS(=O)(=O)CC2 C12(CN=c3ccnc(-c4ccccc4)[nH]3)CC3CCC(C1C2)N3C1CCCC1 C1(NC(=O)CCc2cc(Br)cs2)CN(C(c2cnsc2)=O)CC1O N1(C(COC(C)C)=O)CCCC(O)(CNC(=O)COC2CCCCCC2)C1 C(=O)(CCCCCCc1ccccc1)NC(C(C)NC(CCNC(C)=O)=O)C CC1(NC(C2CC2(Cl)Cl)=O)CCN(C(C2(C(c3ccco3)=O)CC2)=O)C1 c1(NC(C(CN(CCC(=O)OCC)Cc2ccccc2)O)=O)ccnc(C)c1 NC(=O)CCCCC(=O)NCCCOCCC(N1CCCC2(CC1)CC2)=O CC1(C)C(CNC(C2CC(C3CC3)=NO2)=O)CCN1C(C1CCC=CO1)=O C(C)(C(CC(=O)NCCC1CCC(C)(C)C1)NC(C1(N(C)C)CC1)=O)OC N1(C(C(=O)NCC)=O)CCCC12CCN(C(=O)CC1(C(F)(F)F)CCC1)CC2 C1(C(=O)NCC(C)(C)OC)CCC(C(C)C)N1C(=O)C=Cc1ccc[nH]1 Cc1ccc(C)c(C(=O)NC(C(=O)NC2CCC(N(C)C)CC2)C2CCCO2)c1 C(=O)(C1=C(C#N)CCC1)NC(C1CCCCC1)C(=O)NCC(C(C)(C)O)F C1(NC(COC)=O)CN(C(C2CCCOC2)=O)CC1CO.c12cnccc1N2 C(CC(O)C(=O)NCCC(C)N(C(=O)CCc1csc(C)n1)C)SC C(=O)(CC(C)(C)CNC(c1cc(C)nc(O)n1)=O)N1C(C)CSCC1 C1(C(=O)NCC(C)CCl)CCCC12CCN(C(c1cc(F)c[nH]1)=O)C2 c1(N(CCC(=O)OC)C(C2CC(C)N2C(c2ccc(C#N)s2)=O)=O)ncncc1C c1(OC)cc(C(N2CCOCC(CNC(=O)C=CC3CC3)C2)=O)cnc1O c1(C(=O)NCC2CC(NC(c3n(CC)nc(C)c3)=O)C2)cc(F)cc(Br)c1F c1(C(=O)NC(CNC(c2cccc(SC)c2)=O)C(C)C)nc(C)ccc1Br C1(COC)(NC(c2cncc(N)c2)=O)CCCN(C(c2ocnc2C2CC2)=O)C1 N1(C(Cn2ccc(C)n2)=O)CCC(NC(c2cc(C(F)F)ccc2F)=O)C(F)C1 C(=O)(N=c1cc[nH]cc1)N(CCCN(C)CBr)C(C)C.c1cccc(Cl)c1 c1(C(N2CCN(C(c3ccc(F)cc3)=O)CC2CF)=O)ccc2ncccn12 C=C(C)CC(C)C(=O)N1CC(NC(=O)CCc2cncc(Br)c2)CC1(C)C Cc1c(C(C)NC(C2CC(C)CN2C(=O)Cc2cncs2)=O)cnn1C CC(C)CCC(F)C(=O)NC(c1ccnn1C)C(=O)NCC1COCC(=O)N1C C(=O)(C1NCc2n[nH]cc21)Nc1ccc(C(N2CCCC(C)C2)=O)cc1F C(=O)(C1=NNC(=O)C1)N1C(CN(C(C(CCC)N(C)C)=O)C2CC2)CCC1 C1(c2nc(CNC(C3C(C(C)C)C3)=O)[nH]n2)CCN(C(C23CC(C)C2C3)=O)CC1 c1(C(=O)NCC(C(C)(C)C)NC(C2N(CCC)C(=O)CC2)=O)cc(F)cc(Cl)c1 C(C(C)(CO)NC(c1cn(C(F)(F)CO)nn1)=O)NC(C(C)NC(=O)NC)=O N1(C(C(C2CN(C(C=CC(C)C)=O)C2)O)=O)CCC2(CC=CCO2)C1 C1(NC(c2cnc(Cl)s2)=O)CN(C(=O)CCc2cccnc2F)C2(CCOC2)C1 C(=O)(CS(=O)(=O)C1CC1)NC1CC(COC)C2C1C2.C1C(=O)NO1 C12(NC(c3ccc(C)nn3)=O)CCCC1CN(C(C1CC3CC3C1)=O)C2 c1(NC(C)=O)cc(C(=O)N(C2CC2)C(C)C)ccn1.N12CC3CC3(C1)C2=O n1(CCC(=O)NC2C(CNC(C3(C)CC(C)(C)C3)=O)C2)nc(O)c2ccccc12 N1(C(C(C=C)(F)F)=O)CCC2(CC1)CCN(C(C)=O)CC2C Cc1cc(N)cnc1C(=O)N(CC(C)(C)CNC(C1CC(N(C)C)C1)=O)C Cc1ncsc1CCCNC(=O)Nc1nc(-c2cccnc2)cs1 c1(C(N(CC(C)NC(c2cnc(Br)o2)=O)C)=O)csc(C(F)(F)F)n1 Cn1ncnc1CCC(=O)NCCCN(C(=O)CCCC1CCC1)C1CC1 C(C(CN=C(NCC(F)F)N1CCC(C2CCOC2)C1)C(F)(F)F)OCC N(C(=NCCCCl)NCc1ccccc1C#N)Cc1cn(CC#C)nc1 c1(C(N2C(CNC(=O)CN(C)C3CC3)CCC(C)C2)=O)coc(S(N)(=O)=O)c1 c1(S)cn2cc(Cl)ccc2n1.C1(N(S(C)(=O)=O)C)CCN(S(C)(=O)=O)C1 N1(C(C(N2CCNC2=O)C)=O)CCCCC(C(=O)NCC2CC3(C2)CC(O)C3)C1.CC C1(CNC(CCC#C)=O)C(C2CC2)CCN1C(=O)C=Cc1c[nH]c(=N)c(C)c1 CC(O)(CNC(c1sccc1C1CC1)=O)CNC(C1CC1c1ccco1)=O Cc1ccc2c(c1)CC(C(=O)N(CCCCNC(=O)C=CC(=O)N(C)C)C)S2=O C(=O)(CC(C)(O)C(F)(F)F)NCCN(C(C(C)C(C)(C)C)=O)C1CCCC1 N1(C(c2c(C)ccnc2)=O)CCC(C2(NC(C3(C)COC3)=O)CC2)C1 CCCCC(O)C(=O)NCC1CCN(C(c2cncn(C)c2=O)=O)C1(C)C CN1CCC(COC(C2(c3cncn3C)CC2)=O)CC1 N1(CCN(c2ccccc2)CC)CCCC(C)(C(=O)NCC2C(C)(C)C2(F)F)C1 CC1(C)CC(C(N2CC(F)(CO)C2)=O)N(C(c2cnc3n2CCC3)=O)C1 C(C(COC)CC(=O)N1CC(C(=O)N(CC(C)OC)C)C(C)C1)OC N1(C(CC(C=C)(C)O)=O)CCN(C(C2(C)CCCNC2=O)=O)C2(CC2)C1 C(CC)(C(=O)NCC#CC(=O)Nc1cccnc1)OCC CCCCC(CNC(=O)C=C=C(C)C)NC(=O)CNC(=O)NC1CC1 c1(C(N(C(C(=O)NCC(C)C(F)F)C2CC2)C)=O)ccc(O)nc1 c1(OC)cncc(C=CC(=O)NC(C)C(C)NC(=O)CCCc2ncco2)c1 N1(C(C)=O)CCCc2cc(NCc3c(Cl)nc(C)nc3Cl)ccc21 CCC(CC(C)C)C(=O)NCC1CC(CCNC(=O)C(C)Cc2ccncc2)C1 c1(C(N2CC(NC(C3C(c4c(C)ccnc4)C3)=O)C2)=O)[nH]ccc(=O)c1C Cn1nnc(C(=O)NC2COCC2CNC(=O)CCc2cccc(F)c2)c1N CC(C)(C)C(=O)C(=O)N1CC=CC(C(=O)NOCCC2CC2)C1 C=C(Cl)C(C)(C)C(=O)N1CCC(O)(CNC(C2CCCCO2)=O)C1 C1(COC)(NC(c2c(Cl)ccnc2C)=O)CCCN(C(c2cccc(N)c2)=O)C1 C1(C(N2C3CSCC2C3)=O)CCOCCN1C(C1CCSC1)=O C1(CC(=O)NC(c2ncc[nH]2)C)CC(NC(=O)C(F)n2cccn2)C1 N1(C(C(CCC)OC)=O)CCCC2CN(CC(Cl)=CCl)CCC12 c1(C(=O)NCC(C)NC(=O)CSCc2ccncc2)c(Br)nc2n1CCC2 C1(CC)CN(C(=O)C(C)N2CC(C)C2)CCC1N=c1[nH]nc(C#N)s1 C(=O)(C(C)(C)C(=O)NC(CNC(c1ccccc1OC)=O)C1CCC1)OCCC C1(OC)CCC(C(=O)NC2CC(CNC(=O)C=CC(C)(C)Sc3ccccc3)C2)C1 CCC(CC(=O)N1CCC(CC)C1CNC(c1cnncc1O)=O)C1CCC1 Cc1cccc(F)c1CNC(=O)C#CCNC(=O)CN1C(C)CCC1C n1(CCCNC(C2C(NC(c3cn(C)nc3)=O)CCC2)=O)ncccc1=O c1(OC)ccc(C)c(C(=O)NC2CCN(C(=O)C(F)=CCCF)CC2)c1 C1(C(=O)NCC2N(CC)CCC2)CN(C(C2(C)CCCC2)=O)CC12CC2 c1(CC)cc(C(N2CCCCC2CCC(=O)NCCOC)=O)c(C)o1 C1(C(=O)NC2C3CCN(C(c4cnc(CCCC)s4)=O)C32)CCn2cncc2C1 C1(NC(C(C)NC(C)=O)=O)(CO)CCN(C(=O)C(=O)CCc2ccccc2)CC1 C1(C(=O)NCCOCCNC(C(CC=CC)C)=O)CCC(F)(F)CC1 c1(C(=O)OC)cc(Cl)c(NCC2CC(C)N(C(c3[nH]c(C)nc3C)=O)C2)nc1C C#CCCCCC(=O)N1CC2(C)CC1(C(=O)NCCOC1CCOC1)C2 c1(N2C3CN(C(c4c(CC)scn4)=O)C(C3)C2)ncnc(C)c1C#N.C1CCCCC1 C1(CC(=O)NCCN(C(c2ccc([N+](=O)[O-])o2)=O)CC2CC2)CC(=O)NC(=O)C1 Cc1cccc2cc(C(=O)Nc3cc(Cl)c(Cl)cc3O)nn12 c1(C(=O)NCCSCC(=O)NC(C(CCC)O)CO)ccc(C#N)cc1C C1(NC(C2CC(C#C)(O)C2)=O)CN(C(=O)Cc2c(C)nn(C)c2Cl)CCC1C N1(C(C2N(C(C(C)C(F)F)=O)C3CCC2C3)=O)CCCC(C)(O)CC1 c1(C(=O)NCCOC(C)(C)CNC(=O)C2=CCCS2)ccc(C#N)nc1O C12(CNC(c3n(C)ncc3)=O)CCCC(CN1C(C1CSCC(=O)N1)=O)C2 c1(OC)cccc(C(=O)NCC(CO)NC(=O)CCc2ncccc2C)c1 N1(C(C(=O)Nc2ccccc2)=O)CCCC2(NC(=O)CSCc3ncc[nH]3)CC12 c1(C(=O)NC(CNC(C2(C=C)CC2)=O)CCC)onc2c1CCCC2 C1(CNC(C(c2cnn(C)c2)OC)=O)C2CN(C(C)C(=O)NC(C)(C)C)CC12 C#CCCCC(=O)NC(c1ccccc1)C(C)NC(C1(C)COC(=O)N1)=O c1(-c2ccc(C(=O)NC(c3n(CC)ccn3)C)o2)cccc(Cl)c1 Cc1cc(O)c(Cl)cc1C(=O)NC1(CCCNC(C2C=CCCC2)=O)CC1 C(c1cccnc1)=CC(=O)NCCC1N(C(C(CC)F)=O)CCC1 CC1(CNC(C2(C)C=CCCC2)=O)CCN(C(=O)Cc2ccc(O)cn2)C1 C1(NC(c2ccc[n+]([O-])c2)=O)CC(O)CN(C(=O)CCC=CBr)C1 c1(CC(=O)NCCN(C(c2c(CC)csc2)=O)C)cccnc1OC c1(C(=O)NCC2CCC(NC(C3(O)CC3)=O)C2)ccc2nccn2c1 Cc1cccc(C(=O)NCc2nc(SCC3CC(Cl)=NO3)n[nH]2)c1 N1(C(C2CC23CCCC3)=O)CC2(CCN2C(C2CCCC2F)=O)C1 C(=O)(CCCCCC(C)C)NC1(CCC)CCCN(C(CC2CC(=C)C2)=O)C1 C1(CC(=O)NC2(CCC(=O)N(C)Cc3nncn3C)CCC2)CC2C=CC1C2 N1(C(c2c(OCC)cccc2)=O)CCCCC(NC(=O)CC2CC(C)=NO2)CC1 N1(C(c2n(C(C)(C)OC)ncc2)=O)CC(C)C(C)(CNC(=O)CC=C(C)C)C1 C1(C(N(CCSC)CC)=O)C(C2CC2)CCN1C(c1cc([N+](=O)[O-])n[nH]1)=O N12CC3(CC(C3)C(=O)NCCC1=O)C2.c1(C(OC)OC)cnc(C(F)(F)F)s1 C1(NC(C(CC)C)=O)CCN(C(C23CC4CC2C3C4)=O)CCC1CO Cc1cc(N)cnc1C(=O)NC(C(=O)N(C1CC2CC2C1)C)c1ccoc1 N1(C(c2cc(C)c(Cl)s2)=O)CCN(C(c2cscc2Cl)=O)CC1C C1(NC)CCC2CCCC2O1.c1(CC(=O)OC)ccc(Cl)c(NC(C(=O)CC)=O)n1 N1(C(=O)NC(C(C)OC)C(C)C)CCCN(C(=O)OCc2ccccc2)CC1C C1(CC(=O)N(C2CCCN(C(=O)C=CCn3cncn3)C2)CC)C(C)(C)C1(C)C c1(CC(=O)NCC23CC(NC(C(C)OC(C)(C)C)=O)(C2)C3)cnn2ccccc12 Cc1cc2[nH]c(C(=O)NCC(C3CCCN3C(=O)CC(C)(F)F)(C)C)cc2o1 N1(C(c2cnc(C(=O)OC)s2)C(=O)NCCOC)CCC(O)(C(C)(C)C)C1 C1(C(=O)NC(C)(C)C(=O)NCCOCC2CCCC2)CCCC1C1CC1 c1(C(=O)NCC(CNC(c2c(C)c[nH]n2)=O)O)coc2c(C)cccc12 O=C(N=c1ccn(CCCO)[nH]1)C1CSCN1C(c1coc(CO)c1)=O N1(C(CS(CCCC)(=O)=O)=O)CC2CCCC2(N=c2nc(CC3CC3)[nH]s2)C1 c1(N(CC(C)NC(=O)CCC2CCC2)C)nc2cccnc2s1 N1(C(CC2CN(C)C2)=O)CCCC1CN(C)C(c1ccco1)=O c1(OCCC(=O)NCCCCC2CN(C(c3csnn3)=O)C2)cccc(Cl)c1Cl C1(OC)(CNC(=O)CC(=O)NCC(F)(F)F)CCN(C(=O)Cc2ccsc2)C1 c1(C(N(CCCCN(C)C(C2CCC(O)C2)=O)C)=O)[nH]nnc1-c1ccccc1 C1(CNC(C(CC)(F)F)=O)CC(F)(F)CN1C(=O)C(N1CCCC1)C1CC1 N1(C(=O)CC2CCCC2(F)F)CCC(CO)C(O)C1 c1(C(=O)NC2CCC(NC(C(N(C)C)C3CC3)=O)CC2)c[nH]c2ccc(F)cc12 c1(CN(CCOC)C(c2ccccc2)C)ccc(Cl)cc1 CC(C)(CNC(c1cccc(-c2ccoc2)c1)=O)CCNC(=O)CNC(N)=O C(=O)(CN=c1cc(C(N2CCCC2)C)nc(SC(C)C)[nH]1)OC c1(C(C)C(=O)NC2CC(N(C(=O)C(F)(F)C3(CC4CC4)CC3)C)C2)ccc(F)cc1F N(C1c2ccccc2CC12CC2)C(Cc1c(C)cn(C)n1)=O CCC(CC1CC1)C(=O)OC.C1(S(C)=O)(CNC(=O)C(=O)N)CC1 c1(CC)n[nH]c(=NC(=O)N(C)C(c2cccc(O)c2)C)s1 c1(NC(C(CCOCC)O)=O)ccc(NC(C2CN(C)C(=O)N2)=O)c(C)c1 C1(NC(C(C)NC(=O)NC)=O)CCSC12CN(C(c1scnc1C(C)(C)C)=O)C2 N1(C(C2CC3(CC(=C)C3)C2)=O)CCC(N=c2[nH]nc(C(C)C)o2)C(C(N)=O)C1 c1(CNC2CCC(NC(C3C(OCC)C3)=O)CC2)cc(CC)cc(OC)c1O c1(C(N(C(CCNC(CC(=O)OC)=O)C)C)=O)cccc2c1S(=O)(=O)CCC2 CCCCCCC(C)C(=O)N1CC(NC(c2cc(C3CC3)[nH]n2)=O)C(C(F)F)C1 C1(CCC)CCC(c2cn(CC(=O)OC)nn2)(NC(CCO)CC(C)C)CC1 CCC(C)CC(C(=O)N(C)Cc1ccc(C)cc1)NC(c1cc(C#N)c[nH]1)=O c1(C(CNC(c2c(CC)nco2)=O)NC(=O)CCSC)ccccc1OC CN1CC(=O)Nc2cc(C(=O)Nc3ccn4cnnc4c3)ccc21 C1(N(C(CNC(=O)C(c2ccccc2)=O)=O)C)CN(C(C)=O)C2(CCOC2)C1 C1(C(N2C(CCNC(CCC(=C)Br)=O)CCC2)=O)COC(C)(C)CO1 N1(C(C2C(CC)N(C)CC2)=O)CCC2CN(C(c3ncc(Br)cc3C)=O)C2C1 c1(-c2nc(CC(C)(C)C)nn2C2CC3CCC2C3)cc2ccccc2s1 N1(C(C(=Cc2ccco2)C)=O)CC2CC(C1)CN(C(=O)CC(=O)NC1CC1)C2 CC1CN(C(=O)CC(C)n2cccn2)CC1CNC(C1CC(O)C1)=O C1(CNC(=O)C=CCO)CC(F)(F)CN1C(c1cccc(Cn2cncn2)c1)=O N1(C(C2CN(C(c3c(C)cco3)=O)CC(F)C2)=O)CCc2ccccc2C1 CC1OC2(C)CC1(C(N1CC3CC3(NC(=O)CC3CC(C)(C)CO3)C1)=O)C2 CCC(CC)(CC)C(=O)N1CCCC(CN(C(=O)CC2CCC(C)CC2)C)CC1 C(=O)(N1CC(C)(O)CO1)C1CCN(C(c2[nH]cc(C)c2)=O)C1C1CC1 C1(NC(CC2CCN(C)C2)=O)CCN(C(=O)CC2CCCC2)CC(O)C1 S(=O)(=O)(C1CCOCC1C)NCc1cccc(C#C)c1 c1(C(=O)NCC(CC=C)NC(=O)Cc2csc(C)c2)cnc2c(cnn2C)c1N N1(C(C2(CCNC(c3cc(=N)[nH][nH]3)=O)CCC2)=O)CCC2(CCCC2)CC1 C1(C(=O)NCC#CC(=O)NCC(C)C2CC2)C2CC3C(C2=O)C13 c1(C(=O)NC(C2CCN(C(C3(C)CCCN3C)=O)C2)C)nc2ncccn2n1 N1(C(C2(C(N)=O)CCCC2)=O)CCOC(C(=O)Nc2ccc(O)cc2)C1 N(C(=NCCSC)NC1CCCC(C)(C)C1)CC1(OC)CCCSC1 N1(C(CCc2c(C)noc2)=O)CC2CCC1CN2C(c1ccc(O)c(CO)c1)=O C1(C(N2C(C)CCC(NC(c3cnc(N)cn3)=O)C2)=O)CCc2c(nnn2C)C1 C#CCC(O)C(=O)N1CC(COC)(NC(=O)CC2COC(=O)C2)C1 c1(CCNC(C2C(OC)C2)=O)ocnc1CNC(=O)CCC1CCOC1 c1(C(N2CC(N(C(C(C)P(C)(C)=O)=O)C)C(O)CC2)=O)ccc2n[nH]cc2c1 C#CCC(C)(C)C(=O)NCCCNC(=O)C(C)Cc1ccc(Cl)c(Cl)c1 C(CCCC(C)(C)NC(c1ncn2c1CCC2)=O)NC(C1C(C(C)C)CCC1)=O C(=O)(C(C)(C)CC(=O)N1CCC(O)(CCNC(=O)CN2CCCNC2=O)C1)OC N1(C(C2CC(=C)C2)=O)CCCC12CCN(C(c1ncnc3sc(C)c(C)c13)=O)C2 Cc1cc(C(=O)NCCC(C)NC(=O)Cc2cncs2)ncc1C#N C1(C(N2C(C3CCCN(C(CCNC(N)=O)=O)C3)CCC2)=O)CCC2(CCC2)O1 C1(Cn2cc(C(CC=C)CC)nn2)CCCN(C(=O)C(F)(F)CN(C)C)C1 N1(C(=O)OC(C)(C)C)CCCC2(CNc3nc[nH]c4nccc3-4)CCCC12 c1(CNC(C2N(C(c3[nH]cc(C)c3)=O)CC(O)C2)=O)ccc([N+](=O)[O-])cc1 CC1C(NC(c2cc(C3(C)CC3)on2)=O)CCCN1C(C1CS(=O)(=O)C1)=O C1(CNC(c2c(C)cc(C)[nH]2)=O)CN(C(c2cc3occc3s2)=O)CCCO1 c1(CNC(NCCOCC=C)=NC)cc(C)nc(O)c1 CC1=C(C(=O)NCC2(F)CC(CNC(=O)CC3CC3(Cl)Cl)C2)CC1 C1(NC(CNC(c2ccccc2)=O)=O)CCN(CC2C3CC4C(C3)C24)C12CCC2 c1(CCC(=O)OCC)ccc(S(=O)(=O)Nc2cc(F)cc(OC)c2Br)s1 N1(C(c2ccccc2C(F)(F)F)=O)CC2CC1CC2CNC(C1(Br)CC1)=O C1(NC(c2c(C)cc(CC)o2)=O)CCCC12CN(C(=O)CCSC)C2 C1(CC(N2CCC(CC(=O)N(CCCC)C)C2)=O)OCCC1(C)C c1(N(CCNC(c2c(C)nn[nH]2)=O)C)nc2cccc(N)c2s1 N1(C(C=NOC)=O)CC2CCN(C(c3cc4scnc4[nH]3)=O)CC12 CC(CC(N)=O)C(=O)N(C)Cc1ccc(CNC(=O)CCN2CCOCC2)cc1 C1(C(=O)NCC(C2(C)COC2)N2CCC2C2CCC2)CCC(F)C1 C1(c2ccc(C(F)(F)F)cc2)CN(Sc2nc(C)c(C(=O)O)s2)CCS1(=O)=O N1(C(C)=O)CCOCC1CC(N1CCC(C)(CNC(=O)C2=CCOC2)C1)=O C1(CNC(C2(N(C)C)CC2)=O)CC(C(C)(C)C)CCN1C(c1coc(Cl)n1)=O C(=O)(CS(=O)(=O)CCO)N1CC(OCCNC(c2ccc(N)cc2F)=O)C1 C1(CNC(C2C(C)C2C)=O)CC2CN(C(C34CCC(C(F)F)(CC3)C4)=O)CC12 c1(C(=O)NC(C)C(F)(F)F)n[nH]c2c1CCN(Cc1cc3c(cc1Br)OCO3)C2 Cc1nc(C)c(C(N2CCC(N(C(=O)CC3CCCC(C)C3)C)C2)=O)c(C)n1 c1(C(N2C(CCCC)CN(C(=O)CNC(C)=O)CC2)=O)ccc2cc[nH]c2c1 Cc1cc(C(=O)NCc2nc(C(N3CC(O)CC3CN(C)C)=O)co2)cnc1O c1(CC)occ(C)c1C(=O)N(CCCN(C)C)CCNC(=O)CN1CCSCC1 C12(NC(CC)=O)CCC(CNC(=O)COc3cccc(NC(C)=O)c3)(CC1)OC2 N1(C(=O)OC(C)(C)C)CC(C(=O)NCC#CCNC(=O)Cc2ccsn2)C1 c1(C(=O)NCC2N(C(c3c(C)nns3)=O)CCC2)ccc(S2(=O)=NCCC2)cc1 Cc1cc(C(N2CCC(NC(=O)C(C)(Cl)Cl)C(CO)C2)=O)cc(N)c1Cl C1(CNC(c2ccc(C3CC3)o2)=O)CCCN1Cc1cscn1 O=C1CC(C2(O)CC(CNc3ccc(-c4ccccn4)s3)C2)(C(F)(F)F)C1 c1(OC)cccc2c1N(C(=O)C=Cc1cnc(N3CCOCC3)s1)CCC2 c1(NCC)ccc(C)cc1C(=O)NCC12CC(CN1C(=O)COC(F)(F)F)C2 c1(C(=O)NC(CNC(C(CC(C)C)F)=O)C2CC2)nc(Br)n2ccccc12 c1(CC)cc(C#N)c(NC(C2CC(O)CN2C(C2CCC(C)(C)CC2)=O)=O)s1 c1(C(=O)NCCC2(NC(=O)CC3CCC3)CC2)csc(C(F)(F)F)c1 N1(CCC(N2C(C(N(CC(C)(C)C)CC)=O)CC2)=O)Cc2ccccc2C1 C1(CC(N2CC(C(N)=O)C2)=O)C2CCCC2N1C(C1(O)CCCCC1)=O c1(C(=O)NC2CC(C)CN(C(c3sccc3Cl)=O)C2)cccc2c1OCCN2 c1(C(N2C(C(=O)NC(C)(C)CO)CC3(CC3)C2)=O)cc2cc(Br)ccn2n1 N1(C(Cc2cnc(C)s2)=O)CC2(C1)CN(C(c1ccnc(C3CC3)n1)=O)C2 C1(NC(C2CCCN(C(C)C)C2)=O)CCN(C(C2(C#N)CC(=O)C2)=O)CCC1CO c1(C(=O)NC2C(C)N(C(=O)Cn3cccn3)CC2)ccc2c(c1)CCOC2 N1(C(c2cccnc2C(F)F)=O)CCC(F)(C(N2CCCC(CC3CC3)C2)=O)CC1 C1(C(=O)NCc2n(CC)nnn2)CC2CN(C(c3cocc3C)=O)CC2C1 C12CCC(CC1)C(=O)NC2.C1(C(=O)NCC2(COC)CCC2)COC(=O)N1 CN1N=C(C(=O)NC2(CNC(=O)CC3CC(F)(F)C3)CCCC2)CCC1=O C(N=c1[nH]c(-c2ccccc2)nc(=NC(C)CC(C)O)[nH]1)C1(C(CC)(C)C)CCC1 c1(OC)csc(C(=O)NCC2C=CCN2C(=O)C(C)CN2CCOCC2)c1OC C1(CN(C(=O)COCP(C)(C)=O)C)CCCN1C(=O)COCC1CCSCC1 C1(C(=O)NC2CC(C)N(C(=O)CC3(O)CCC3)C2)CC(C)(C)OC1(C)C Cc1cnc(C(=O)N(C2CCC(NC(=O)C(C)n3ccnc3)CC2)C)c(F)c1 c1(NCC(C)NC(C2(F)CCN(C(=O)OC(C)(C)C)C2)=O)cccc([N+](=O)[O-])c1 Cc1cc(C#N)ccc1CN(C1CCC(C(N)=O)C1)C(C)C C1(CNC(C2CCC3CC3C2)=O)CC2CCC1N2C(=O)Cc1csc(S)n1 c1(C(=O)NCC(CO)NC(c2[nH]n(C)c(=O)n2)=O)c[nH]c2cccnc12 N1(C(C2C(C=C)CC2)=O)CC(NC(c2snnc2C2CCC2)=O)CC(C)(C)C1 CCCC(C)(O)C(=O)N1CC(NC(c2[nH]cnc2C#N)c2nc(=N)[nH][nH]2)C(C)C1 C(=O)(C#CC1CCCCO1)N.N1(C(CN(C)C2CC2)=O)CCC(C2CC2)C(CO)C1 c1(C(=O)NC2C(NC(=O)CCCCCc3ccccc3)C2)ccc2nc[nH]c2n1 c1(NCCSCC)ccc(S(=O)(=O)N2CCc3ccncc3C2)c2ccncc12 N1(C(C(CC=C)(C)C)=O)CCC(C2CC2)(CNC(c2ncc(C(F)F)s2)=O)C1 C1(O)(CCNC(c2nc(C)sc2)=O)CCN(C(=O)Cc2ccc(O)cn2)C1 c1(OC)c(O)cc(CN(C(=O)Cc2ccc(Cl)cc2[N+](=O)[O-])C)cc1C#N C(N=c1[nH]cnc(NCC2(S(C)(=O)=O)CC2)c1C)c1n(CC)cnn1 C(C)(CO)(CN=C1NN(C)C2CCN1C2)OC.C1(C)CC1.C(N)=O C(=O)(C#CC1CCCOC1)C(C(C)C)CNC(=O)C(=O)NCCC(F)(F)F c1(C(C(=O)NCC2(F)CC(CNC(C3CC(=C)C3)=O)C2)O)ccccc1Cl N1(C(CC2(CSC)CC2)=O)CCC2CN(C(c3cccc(NC(N)=O)c3)=O)C2C1 c1(C(c2n(CCCCCC)nnn2)NC23CC(C2)C3)cc(Br)c(C)[nH]1 C1(CNC(=O)CC2CCC3CC23)CCCN(C(c2cc(=O)cc[nH]2)=O)C1 Cc1cccc(C(=O)NCCc2ccc(NC(C3CC3C)=O)cc2)c1C CC(C)CCCCCC(=O)N1CCN(C(=O)C(C)(C)CC2CC2)CC1CO c1(C(=O)NCC2CCN(C(C3CCC(C(N)=O)O3)=O)C2)nc2cnccc2s1 N1(C(COCC#C)=O)CC(CNC(=O)Cc2c(C)nc(O)nc2C)C2(CCC2)C1 C=C(F)C1(CC(N2CCCC2C2(C(=O)NC3CC(=O)N(O)C3)CC2)=O)CCC1 C(C(C)(C)C(=O)NOCCCCCC1CC1)N(C(C(C)SC)=O)C c1(CC(N2C(CNC(C3CC3OC(F)F)=O)CCC2)=O)ccc(OC(F)F)cc1 N1(C(c2c(CC)cncc2)=O)CC2C=CC1C(C(=O)NCC(C)(O)COC)C2 c1(N2CCCC(C(C)(C)C)C2)nc2c(c(=NC3CCCc4n[nH]cc43)[nH]1)SCC2 N1(C(C(C)(CO)OC)=O)CCN(C(c2cc3ccccc3cn2)=O)CC12CCC2 c1(C(=O)NC2C(CNC(CCCC(N)=O)=O)C2)cc2cc(Br)cnc2s1 CC(CNC(C1CC1CN(C)C)=O)(CO)NC(=O)CC=CCc1ccccc1 c1(CCNC(=O)Nc2nc(C(=O)OCC)c(CC)s2)ccc(F)c(F)c1 C(CN=c1nc2c(cnn2C)c(NC(c2n[nH]c(C)c2C)C)[nH]1)N(CC)CC CC1(CNC(=O)Cc2ccccc2F)CCOC1C1CN(C(=O)C(N)=O)C1 c1(COC(c2cnc(C(=O)OC)s2)=O)ccc(C)nc1Br Cc1cc(C(=O)NCC(O)CNC(c2cc(C(C)(C)C)n(C)n2)=O)[nH]c1C C1(C#C)(NC(N(C2CC23CC3)CC#C)=O)CC2CCCC12 N1(C(C(COC)CC(C)C)=O)CCCC2C(NC(c3cc(Cl)ns3)=O)C(C)(C)C12 Cc1nc(NCC2(CNC(c3cc(Cl)cn3C)=O)CC2)cc(C(C)C)n1 C(C(C)N=c1[nH]c2ncnc-2c(C(F)(F)F)[nH]1)N(C(C)C)C.C1COC1 N1(C(c2c(CC)cc[nH]2)=O)CC(NC(c2ccc(C(C)=O)[nH]2)=O)C(CC2CC2)C1 Cc1cccc(SCC(N2CC(N(C)C)C2)=O)c1.C1(C(=O)NCCN)CC1F c1(C(=O)NCCCCNC(C2C(C(=O)OC)COC2)=O)cc(C)cc(Cl)c1 N1(C(CCN(C(=O)Cn2cc(CO)nn2)C)=O)CCC(F)CC1 C12(C(N(CCNC(CN3C(C)CCC3)=O)C)=O)CCC(CC1)C2(C)C N1(C(c2ccn(C)n2)=O)C(CNC(c2cocc2Br)=O)CC2CC12 C1(F)(CNC(CCNC(C)=O)=O)CN(C(C2CCN(S(C)(=O)=O)C2)=O)C1 c1(C(N(CCOCCN(C(c2c(C)cc[nH]2)=O)C)C)=O)c(C)noc1C(F)(F)F N1(C(c2ccc(CNC(C(CC(C)C)OC)=O)o2)=O)CCC2CCCC2C1 C1(C(=O)NC23CCCC2CCC3)COCCN(CCOc2cccc(Cl)c2)C1 N1(C(C2(F)CCCN(C(C(C)NC(=O)OC)=O)C2)=O)C2CCC(OC)C1CC2 C1(CNC(C(C)(C)C2CC2)=O)CC12CCN(C(C13CCCN(CCC1)C3)=O)CC2 C(=O)(C(C)C(O)C(C)C)N1CCC(C(=O)N(C2CCN(OC)CC2)C)(OC)C1 C(=O)(C#CC(C)(C)C)N1C(CNC(C2CCN(C)C2)=O)C=CC1 c1(CC)cc(C(=O)NCCC(C)N(C)C(c2cncc(O)c2)=O)cc(Cl)n1 C1(NC(CN2CC(CC)C2)=O)CCN(C(=O)C(c2ccccc2Cl)C)CC1C Cc1nc(CNC(=N)NCCOC(C)C)n[nH]1 N1(c2ncc(C)cn2)CCCC12CCN(C(=O)C(c1cc(Cl)cc(Cl)c1)O)CC2 c1(C(=O)NCCN(C(C2(CC=C)CC2)=O)C)cnn(C)c1CC C(=O)(CCCCCC(C)(C)C)NCC1CCN(C(C2CC(C)=C(C)CC2)=O)C1 C1(NC(C=C(COC)C)=O)CC2CCC(C1C)N2C(=O)CCCc1cccnc1 c1(C(N2CCC(C(C)NC(C3(C#N)CC=CC3)=O)C2)=O)cnc2c(c1)CCCC2 N1(C(CCC#N)=O)CCCC(C2CC(NC(=O)COC(F)F)CCO2)C1 c1(C(N(CC(C)CNC(C2CCC(C)C2)=O)C)=O)cc(Br)n(C)n1 C(=O)(CC(C)(O)C(F)(F)F)NC1C(OC)CN(C(c2ccc(Cl)cc2N)=O)C1 C1(C(=O)NCCC(C)N2CCC2)CCC2(CC2)N1C(=O)C#CC(C)(C)C c1(C(=O)NCC(CCCC)NC(=O)CC2CN(C)C2)nc2ncccn2n1 Cc1c(C(=O)NCC2C(C)CCCN2C(=O)CC(C2CC2)C2CC2)c(Cl)nn1C C(C(=O)N=c1cc(C(F)F)[nH][nH]1)c1ccc(OC)nc1 C(CNC(C1C(C)C1C)=O)(CC(C)C)NC(CC(=O)NCC)=O c1(C(N2CC(C(C)NC(c3cncn3C)=O)C2)=O)cccc(=O)n1C N1(C(c2ccc(=NC)[nH]c2)=O)CC(C(=O)NC2(C)CCC(C)(C)C2)C2(CCC2)C1 CC1CCC=C1C(=O)N1C2CCC1C(CNC(=O)CN1CC(=O)NC1=O)C2 N1(C(CC2(CC)CCC2)=O)C2CCCC1CN(C(c1ccoc1)=O)C2 C1(C2CCSCC2)(NC(=O)NCC2CCCC2N2CCCCC2)CC1 Cc1sc(NC(N2CCSC2(C)C(=O)O)=O)c(C)c1C C1(CNC(C2CCOC(CF)C2)=O)CC2(CC2)CN1C(c1ncc(C(F)F)s1)=O Cc1sc(Br)nc1C(N1CCCCC1C)C(=O)NCC1CCCO1 N1(C(C2(C)COC2)=O)CCC2(CCN(C(C3C(F)(F)C34CC4)=O)CC2)C1 CC1(C)CCN(Cc2sc(Br)c(Cl)c2Br)CCS1=O N1(C(C=Cc2n(CC)ccn2)=O)CCN(C)C(CNC(=O)CN2CCCC2C)C1 C12(C(=O)NC3C(OC)C(O)C3)COC(C1)C(NC(c1cc(C(C)C)no1)=O)C2 C12(C(N(CCCN(C(C3(OC)CCSC3)=O)C)C)=O)CCOC(C)(C1)C2 c1(C(=O)NCC(C(C)C)F)cnc2ccsc2c1 c1(COC)nn(C)cc1-c1noc(-c2cccnc2Sc2ccc(Cl)cc2)n1 C1(CO)OCCC1(c1nnnn1CC1CC1)NC(c1ccncc1Cl)C1CC1 C(=O)(CC(O)COC)Nc1c(C(N(CCOC)CC2CCOCC2)=O)con1 CC(CCC(=O)NC(C)C(CO)NC(=O)CSCC(F)F)N(C)C C(=O)(N=c1cccn[nH]1)C1(c2ccc(-c3nccc(OC)c3)cc2)CC1 C1(C(=O)NC(c2c(C)ncs2)C)CC(F)(F)CN1C(=O)C1=CC(C)(C)C1 c1(C(=O)NC2C(NC(Cc3nc(C)c(C)o3)=O)CC2)cncc2c1CCC2 c12ccc(cc1C#N)S(=O)(=O)N2.C1(Br)(CN(CCOCCOCC)C)CC1 C1(C(=O)NCC2OCCN(C(CCP(C)(C)=O)=O)C2)CCn2cncc2C1 C(=O)(C1=CCCCCC1)N1CCCC(CNC(Cc2c(C)ccnc2)=O)C1 C1(C2CC2)(CC)c2ccccc2CN1C(=O)CC(F)(F)C(F)F CC(=O)CCCC(=O)N1CC(NC(C2CC2C2CCC2)=O)CC(C)C1 c1(CNC(C(CC)O)=O)nc2c(s1)CN(C(=O)CCCC(C)=O)CC2 c1(C(N2CCC(NC(C(C#C)(C)C)=O)C2)=O)ccc(N)c(F)c1Br C(=O)(C(C(C1CCC1)OC)N1CCC(CC(=O)OC)CC1)NC(CC)(C)C c1(Cc2nnnn2CC2CCOC2)cn(CC2CC2)nn1.CC(C)COCC(C)C C(=O)(CNCC1(CC(N)=O)CC1)N(C1(C(=O)NC)CC1)C c1(C(N2C(CNC(=O)C=CI)CCCC2)=O)ccc([N+](=O)[O-])cc1C(F)(F)F c1(-n2c(C(=O)NCCN(C(=O)C(O)C3CC3)C)ccn2)ccccc1Cl c1(C(=O)NCCC2CCC(NC(C(Cn3ccc(C)n3)C)=O)C2)cn(C)nc1O C12(NC(CCSCC)=O)CCC(C1)N(C(=O)CCC1CC1(F)F)C2 CN1CCCC(F)(CN(C(=O)CCCCN)C2CN(C(c3ccnc(Cl)n3)=O)C2)C1 C1(NC(C2CCN2C(=O)CCC2CCCCC2)=O)CN2CCC1C2 C1(C(=O)NCC2CCN(CC)C2)CC2CCC2C1.C1C(=O)N1CCC c1(C(=O)NC2C(NC(C3(C#C)CCCC3)=O)CCC2)ccc(C#C)c(F)c1 N1(C(C2N(C(C3C(OC)(OC)CC3)=O)CCCC2)=O)CC(C2CC2)C1C1CC1 C(C(CC(C)C)C(=O)N(CC(O)C(C)(C)C)CC)NC(C=C(CC)CC)=O c1(OCC=C)c(C(=O)NCC=CCNC(=O)C=Cc2cn(C)nn2)cccc1C C(=O)(C(C)(C)CCCO)NCC1C(C)CN(C(=O)CCN2CCOCC2)C1 N1(C(CC2(C)CC2)=O)CCN(C(=O)CN2CCCC2CO)CC1 N1(C(C(CC)O)=O)CC2(CCC(CNC(=O)Cc3ccccc3I)O2)C1 N1(C(Cc2c(C)occ2)=O)CC(NC(C2(n3cccn3)CC2)=O)C(O)C1 C=CCC(C)C(=O)N1CCN(CCCNC(c2ccncc2)=O)CC1 C#Cc1cccc(OCC(=O)NC2CN(C(=O)CCC(=C)C)C3CC23)c1 CC(CCc1ccccc1)CC(=O)OCC(C)(C)C.C1(=O)CO1 CCCC(C(=O)N1CCCC1C1(NC(c2ocnc2CC)=O)CC1)S(N)(=O)=O C(=O)(C(C)(C)C(F)F)NCc1cccc(CNC(C(c2cncnc2)C)=O)c1 Cc1ncc(C(N2CCN(C)C(C(=O)NC3CCC(C(N)=O)C3)C2)=O)c(=N)[nH]1 C1(NC(CCC(C)C)=O)C2CC(CN(C(c3sccc3Br)=O)C2)C1(F)F N1(C(c2cc(COC)no2)=O)CC(C)OC2(CCN(c3cncc(C#N)n3)C2)C1 C1(NC(C2C(C(C)O)C2)=O)CCCCC12CCN(C(c1ccc(C)c(Cl)c1)=O)C2 C1(NC(C2(COCC)CC2)=O)CC2C1CCN2C(c1cccc(C(F)(F)F)n1)=O C=CCC(C(=O)N1CCCCCC(NC(=O)CC=CCOC)C1)C(C)C C1(C(N(C)CCc2ccccc2)=O)CCC2(CC2)N1C(C1CC(C)(C)C1)=O c1(NCC(C(C)(C)C)OCC)cc(Br)ccc1S(=O)(=O)NC1(C2CC2)CC1 c1(C(C(=O)NC(CCNC(C=CCCC(C)C)=O)C)(F)F)cc(F)cc(F)c1 c1(C(N2CC(C(C(=O)NCC(C)C(F)(F)F)OC)C2)=O)ccnc(C)c1N CN1CC(=O)NCC1C(=O)NC1CC(CO)N(C(=O)CCS(C)(=O)=O)C1 Cc1cc(C(N2CCCC(O)(CCNC(C3CC3C)=O)C2)=O)c2cnn(C)c2n1 c1(CCC)noc2ncc(C(N3CCC(C)C3CNC(=O)CC(C)(C)F)=O)cc12 C(CCC(C)C(=O)NCCCC(C)NC(C1CCCCC1(C)C)=O)OC Cc1nn(-c2ccc(F)cc2)cc1C(N1CC(CNC(=O)CO)C(C)C1)=O c1(C(N2CCC3CN(C(C45CCC(F)(CC4)C5)=O)C3C2)=O)cnc2c(c1)CCC2 C(=O)(C(C)(F)F)N(C1CCN(C(C2CC(C(F)F)C2)=O)C1)CCC CC1CC(N(C)C(c2cc(CNC(=O)Cc3cn[nH]c3)cs2)=O)CCO1 c1(C(=O)NC(C(C)NC(C2C(C)CCO2)=O)(C)C)ccc(S(C)(=O)=O)o1 N1(C(CSC)=O)CCCC(O)(CNC(=O)CCC2(C)CC2)C1 N1(C(C=C(C)C(F)F)=O)CC2OCCN(C(=O)C(C)N3CCC3n3cnnn3)C2C1 C(=O)(C(C(C)(C)C)NC(c1ccc(CO)o1)=O)NCC(C)(O)C1(C)CC1 N1(C(C(C)CF)=O)CCC2(CCC2CNC(c2ncccc2N)=O)CC1 C12(NC(COc3cccc(CC)c3)=O)CCN(C(=O)Cc3cc[nH]c3)CCC1C2 N1(C(c2cc(OC)ncc2)=O)C2CCC(C2)C1C(=O)Nc1ccc(I)nc1 C1(C(=O)NC(CC=C)CC=C)CCC(C)(C)N(C(=O)C=CCF)C1 c1(OCC(=O)OCC2(NC(=O)CSC(F)(F)F)CCOC2)ccccc1C(F)(F)F CC1(C)CN(C(=O)CC2CCCC(F)(F)C2)CC1NC(=O)COc1ccccc1 N1(Cc2cccc(CC)c2)CCC(NC(c2ccc(Br)o2)=O)CC1C C1(CCNC(C2(C(F)F)CC(=C)C2)=O)CCCCN1C(=O)C(C)Oc1ccccc1 N1(C(C(C(C)C)C)=O)CC2(CCOCC2)CC1CNC(=O)CC1CCCN(C)C1 C1(CNC(c2cc(C(F)(F)F)cc(O)c2)=O)CC2(CCOC2)C1 c1(C(C)(C)C)cc(Cl)c(Cl)s1.C12CC(=C3CN(C3)C(=O)N1)C2 c1(OC)ccc(C)cc1NC(=O)C(CC1CC1)NC(=O)CC=C(Cl)Cl c1(C(=O)NCCCN(C(CCCNC(=O)OC)=O)C)cc(Cl)c(F)cc1OC N1(c2nc(NCCCS(C)(=O)=O)c3c(n2)ccs3)CCOc2ccc(F)cc2C1 CCC(CC(C)C)C(=O)N1CCOC(CNC(=O)C(C)=C(C)C)C1 c1(C(=O)NC2(CO)CCN(C(C3CCCS3)=O)CC2)cccc2nonc12 c1(C(=O)NCC(CNC(CCC(=O)OCC)=O)OC)nn(CC)cc1[N+](=O)[O-] C#CCC(CC(F)F)C(=O)NCC1CN(C(=O)C(C)N(C)C)CC1c1ccccc1 C1(NC(C(c2c(C)cccn2)(F)F)=O)C2CC(O)C1N(C(=O)CNS(C)(=O)=O)C2 C1CCOCC1.C1(C(=O)NC)CC(CCO)C1.C12(CC1)N(C)C2=O.C1C(=O)N1 c1(C(=O)NC(C(CC2CN(C(=O)OC(C)(C)C)C2)F)=O)cc2ccc(F)cc2s1 C1(c2n(CC(=O)OC)nnn2)(NC2CCC(F)CC2)CC2CCCN(C2)C1 c1(C(=O)NCC(CNC(c2n(CC)ncn2)=O)C)c(C)cccc1[N+](=O)[O-] N1(C(C(C)(C)OC(C)C)=O)CC2ON=C(CNC(c3ccc(F)c(F)c3)=O)C2C1 N1(C(=O)Nc2cc(C)c(NS(C)(=O)=O)cc2)CCC(C)C(C)CC1 c1(C(=O)NC(CC(C)NC(CC2(COC)CC2)=O)C)c(C)cc(Cl)cc1C CC(C)CC(C)(C)C(=O)N1CCC(C)C(N(C(=O)COCC(F)F)C)C1 Cc1ccc(CC(=O)NC2CN(C(=O)Cc3cc(F)ccc3Cl)CC2O)c(C)c1 c1(C(=O)NC(C)CNC(=O)CC2CSC2)c(O)nc(=O)n2c1CCC2 CC1(C)COCC1CNC(=O)C(c1cccs1)NC(c1ccc[nH]1)=O CC(C)CC(C)CC(=O)NC(C)(C)CN(C)C(c1cnc(C(C)(C)C)[nH]1)=O C(=O)(CC(CC)C(C)C)N(C1CCN(C(=O)Cc2ccccc2Cl)C1)CCC N1(C(COCC(OC)OCC)=O)CCOCC1C1(C(F)(F)F)CC1 c1(OC)cc(C(=O)NCCCc2nc(C3CC3)cs2)cc(OC)c1C(N)=O C1(N(C(C2CCC(=O)C2)=O)CC)CCN(C(C2(C)CCCC2)=O)CC1 c1(OC)cc(F)c(NC(C2CCN(C(c3cccs3)=O)C2)=O)cn1 C1(S(N)(=O)=O)(C(N(CCOCCN(C(C(C(C)C)OCC)=O)C)C)=O)CCCC1 C1(NC(c2ccc(C)cn2)=O)CN(C(c2c(C)cccc2F)=O)C2(CCCC2)C1 CC(C)(F)CCC(=O)NCC1CC1CNC(c1cccnc1S)=O c1(C(=O)NC(CC)CNC(=O)CCN2CCCC2)cc2cc([N+](=O)[O-])ccc2[nH]1 N1(C(=O)CC2CCOC2)CC2CC(C1)N2C(=O)CC1CC(C2CC2)C1 c1(C(=O)NCC(CNC(C(C)SCCCC)=O)O)[nH]c(C)c(C)c1C Cc1cccc(F)c1CC(=O)NC1CCCC1NC(=O)CSCC1CCCCO1 C1(F)(CNC(=O)C(O)C2CCCC2)CCC(CNC(c2cncs2)=O)CC1 C1(C(=O)NC(C(=O)NCC2(C(C)(C)OC)CC2)C2(O)CCC2)CC(=O)OC1(C)C c1(C(=O)NC(C(C)NC(C2CCS2(=O)=O)=O)C)cc(F)cc2cnccc12 C1(N(C(CN(C(C)=O)Cc2ccccc2)=O)CCO)CC(C)CN(CCC2CC2)C1 C12(CNC(c3ccc(N)cc3F)=O)CN(C(c3ccc(F)cc3)=O)CC1CCO2 c1(CNC(C2CN(C(c3ccc(O)nc3)=O)CCN2)=O)cn2cc(Cl)ccc2n1 C1(C(=O)NC(CC)C2CCC2)CCN(C(=O)Cc2c(C)cnn2C)CCO1 C1(C(=O)NC(C)CNC(c2cn(CCO)nn2)=O)CC(=O)N(Cn2cccn2)C1 c1(Cn2cc(Cn3ncc(CO)c3)nn2)ccc(F)c(F)c1.N12CCCC1C2 C(=O)(CCCCC(=O)NC1CCCCC1NC(c1ccc(C#N)[nH]1)=O)OC Cc1ccc(C(=O)NC2(CO)CN(C(=O)C(C)(C)c3ccc(Cl)s3)C2)cc1 Cc1c(NC(C2CC2NC(=O)Cc2ccccn2)=O)ccc(C#N)c1Cl N1(C(c2c(CC)c[nH]c2)=O)CCC(CNC(c2ccnc(S)c2)=O)(OC)CC1 NS(=O)(=O)C(C(=O)N1CCC(CNC(=O)C=CCF)C12CC2)c1ccccc1 n1(CCNC(=O)NCC2(OCC)CCSC2)cc(Br)c(C)n1 CC1(C)COC(CCNC(CCCCC#N)c2nnnn2CCCNC(N)=O)C1 N1(C(CC(C)N(C)C)=O)CC(C2CC2)(C(=O)NC2CC23CCCCC3)C1 c1(OCC(=O)NCCOCCNC(=O)COCc2cccs2)cccc(Br)c1 S(=O)(=O)(c1ccsc1)N1CC(c2n(CC)c(O)nn2)OCC1 C1(C(C)C)CCN(C(=NC2CCS(=O)(=O)C2)NC2Cc3ccccc3C2)C1 C1(NC(C(C(C)C)NC(C2CCC2(F)F)=O)=O)CCC2(CC1)N=N2 c1(C2(C(N(C(C3CCCC(F)(F)C3)C(=O)OC)C)=O)CC2)c(F)cccc1Cl c1(-c2ncc(C(=O)NC3C(NC(CC(CC)C)=O)CC3)s2)c(F)cccc1F C1(F)(C(=O)NC2(CNC(C(C3CCC3)OCC)=O)CC2)C(C)(C)C1(C)C Cc1cccc2[nH]cc(C(N3CCN(C(c4c[nH]c(=O)cn4)=O)C(C)C3)=O)c12 c1(C(=O)NC2CCCN(C(C(CC)n3nccc3C)=O)C2)cc(C#N)ccc1F C1(C(N2CCCC(OCCC)C2)=O)CCN(C(c2cc(C(C)=O)sn2)=O)C1(C)C CN(C(=NCCc1ccccc1Cl)NC1CC2CC1CC21CC1)CCF C1(CC(=O)NCC2OCCN(C(C3C(COC)C3)=O)C2)CCC(C(F)(F)F)N(C)C1 c1(SCC)ccc(C(N2CCC2CNC(C2ON=C(C)C2C)=O)=O)cn1 C(=O)(C(O)C(F)(F)F)NC1C(SC)CN(C(c2c[nH]nc2C(C)C)=O)C1 c1(OCC)cc2c(cc1C(N1CCC(F)(CF)C1)C(=O)NC1(C)CC1)OC(C)C2 CC1CCC(=CC(=O)NC2CCCC2NC(=O)CC2CCC2)C1 N1(C(c2c(C)occ2)=O)CC(NC(c2nccn2C)=O)C2CCCC12 N1(C(C2CCN(C(C)=O)C2)=O)CCCCC1C(=O)NC(C)(C)C(C)(C)C C(C1c2ccccc2CN1C(c1cc(C#N)ccc1N)=O)NC(C(CO)OC)=O N1(C(C2C(C3(C)COC3)C2)=O)CCC(C2CC2)C1C(=O)NOCCCF N1(C(C(C)SC(F)(F)F)=O)CC(NC(C2CC(Cl)(Cl)C2)=O)C2(CC2)C1 C(C(C)(C)C(=O)NC1CN(C(C2CCS2(=O)=O)=O)C1)OC C=C(Cl)CCC(=O)N1CCOCC1CNC(=O)CCC1CC1(F)F N1(C(c2cn3cc(C)nc3s2)=O)CCC(C2(O)CN(C(=O)C3=CCOC3)C2)CC1 CCC(CC(=O)NC1(C(=O)NCC2CC(F)(F)C2)CC(F)(F)C1)C(C)C CC(C(=O)N1CCNC(=O)C1CCO)(C(F)(F)F)NC(c1cc2c[nH]nc2s1)=O C1(C)(CNC(CSCCC)=O)CCN(C(=O)C(CC)NC(=O)OC(C)(C)C)CC1 c1(C(=O)NCCCN(CCCNC(CCCC(C)C)=O)C)ccc2c(c1)OCC2 Cc1cc(C2CC2)ccc1C(=O)NCC(C)NC(=O)C(C)Cc1c(C)noc1C C(=O)(N=c1[nH]nc(C(c2ccccc2)C)s1)NCC.N12CCC(CC1)CNCC2=O C1(OC)C=CCN(C(C2(F)CN(C(C3CC=C(C)CC3)=O)C2)=O)C1 C(N=c1nc2sccc2c(N2CCOCC(C)(F)C2)[nH]1)c1cnn(C)c1N N1(C(C2(O)CCCC2)=O)CCN(C(C2CC3CCC3C2)=O)C(CO)C1 N1(C(Cc2ncn(C)c2)=O)CCCC1(C)C(=O)NC1CC(c2ccccc2)C1 c1(C(N2C(C(N3CCC(C)C3)=O)CC(F)C2)=O)cnc2n1CCCCC2 C(=O)(C1=CCCN(C(C2CC(F)(F)C2)=O)C1)N(C1COC2(CCC2)C1)C C(=O)(C1CCc2nccn21)NC(CC)CNC(c1cnc(O)c(N(C)C)c1)=O C(CC(C)C(=O)NCC1(C(=O)NC(Cc2ccco2)CO)CCCC1)=CCC N1(C(CN(C(C)=O)CCC(C)(C)C)=O)CCN(C(=O)C2=CC(C)(C)C2)C(C)C1C C12(C(N3CC(NC(c4ccc(Cl)s4)=O)C3)=O)CCCC(CCC1)C2O C(=O)(C(C)CCCC(C)C)NC1CCN(C(c2cc(C)sn2)=O)CC1 Cc1ncc(Cl)c(C(=O)NC2CCCCC2NC(=O)C(C#N)C2CC2)n1 N1(C(CCCCCC)=O)CC2CCCN(C(=O)CCCc3ncc(C)o3)C2C1 c1(C(=O)NCC2(O)CN(C(C(C)c3ccco3)=O)C2)cncn(C)c1=O C=CC1CN(C(=O)NC(C)(C)C)CN1C(C1CN(C(=O)C=CCC)CC1OC)=O N1(C(C2CC(CC)OCC2)=O)CCOC2(C1)CN(C(c1c[nH]c(=N)c(C)c1)=O)C2 c1(C(=O)NC2CC(C)(CNC(=O)C(O)c3ccco3)C2)cccc2[nH]ncc12 N1(C(C(C(C)O)C)=O)CCN(C(c2ccccc2C(F)F)=O)CC12CCC2 CC(C)C(=O)C(=O)N1CCN(C2CN(C(c3ccon3)=O)C2)CC1 N1(C(N(c2ncn(C)n2)C)=O)CCC2(CC1)CC2c1cn(C2CCOCC2)nn1 c1(C(N2CCCC(NC(C=Cc3c(C)coc3C)=O)C2)=O)cccc([N+](=O)[O-])c1 CC1(C)CC=C(C(=O)N2CC3CC(C2)CN(C(=O)Cn2nnc(=N)[nH]2)C3)CC1 c1(C(=O)NC2C(CNC(C=CCN(C)CC)=O)CCCC2)ccc(C)c(Br)c1 C1(NC(C2C(NC(C3C(C)(C)OC(=O)C3)=O)CC=CC2)=O)Cc2ccccc2C1 c1(NC(C2C(NCc3c(OC)cccc3O)CCC2)=O)ccc2cn(C)nc2c1 C(=O)(C(C)(C)CCCNC(c1nocc1C)=O)NCC1CCN(C(C)=O)C1 c1(C(=O)NC(C2CCC2C(=O)NC2CCS(=O)(=O)C2)(C)C)ccc(N)cn1 NCCCC(O)C(=O)N1CC(n2cc(-c3ccccc3[N+](=O)[O-])nn2)CO1 c1(OC)cccc(C(=O)NCCC(O)CNC(=O)C(C)SC(F)(F)F)c1 N1(C(c2ccc(C(=O)OC)[nH]2)=O)CC(CNC(C2CCCOC2)=O)C(O)C1 C1(COC)(CNC(=O)CCCC2(OC)CCC2)CN(C(=O)C(O)C2CCC2)C1 C1(C(=O)NCCN(C(c2conc2COC)=O)CC)CCCOC1C(C)C c1(C(=O)OCC(C(CC)(C)C)=O)cc(Br)cc(S(C)(=O)=O)c1F C1(C(C)CNC(C2CCC2)=O)CCCN(C(c2ccn(-c3ccncc3)n2)=O)C1 c1(OCC)cncc(C(=O)NC2CCN(C(=O)CC3(OC)CCCC3)C2)c1 c1(OC)cc(COC(C)=O)ccc1COC(=N)O Cc1ccnc(C(N2CCC2CNC(c2ccc(CSC(F)F)o2)=O)=O)c1 C1(CN(C2N(C(CC(=C=C)C)=O)CCC2O)Cc2ccccc2)NC(=O)CC1(C)C C1(O)(CC(=O)NC(C2C(CNC(CSCC(=O)OC(C)(C)C)=O)C2)=O)CCCOC1 c1(CN(C(N2CCSC(C)C2C)=O)CC)c(O)cccc1F Cc1nn(C(C)C)cc1C(=O)N(C1CN(C(=O)Cc2cncnc2)CC1F)C c1(C(=O)NCC2(NC(c3c(C)nc[nH]3)=O)CCC2)cccc(CF)c1 CCCC(CCC)C(=O)NCC1CC(C)(C)CN1C(C1CCC1CF)=O c1(OC)cc(C)ccc1C(N1CCC(O)C(NC(=O)CN(C2CCCC2)C)C1)=O c1(C(=O)NCC(C)(CNC(C2CC2C)=O)OC)ccc(SC)cc1C C1(C(N2C(CNC(C3CC3Br)=O)CC(OC)C2)=O)CCC2(CC1)CC2 C1(C(N(CC(N2CC(O)(NC(=O)NC)C2)=O)C)=O)CCN(CC2CCC2)CC1 c1(C(=O)O)ccccc1S(=O)(=O)N1CC2(C1)CN(S(=O)(=O)c1ccc(F)cc1)C2 Cn1ccc(C(=O)NC(C2CN(C(=O)C(=O)NCC(F)(F)F)C2)(C)C)cc1=O C(=O)(C(CCCC)C(C)C)NC1C(C(N(CCCC)CCO)=O)OCC1 CC(C)(C)CC(O)CC(=O)NCC1CCCN1C(=O)CSCC1CCCCO1 N1(C(C(CC)C)=O)CCC(N(CCNC(C)=O)C(c2ccc(Cl)cc2)=O)CC1 C1(CNC(C(CC)OC)=O)CN(C(=O)COCP(C)(C)=O)C(C)(C)C1 C1(NC(C(C)OC)=O)CCN(C(c2n[nH]c(C)c2Br)=O)CC1O c1(-c2cn(C3C(N4CCC(OC)C4)CCC3)nn2)cc2occc2s1 CC(C)CCCC(=O)N(C1CCCN(C(c2cocn2)=O)C1)CCF c1(C(=O)NCC2CC(O)CN2C(=O)C2=CCS(=O)(=O)C2)cc(F)cc2ccoc12 c1(C(=O)NC2CC(CCOC)C2)ccc(NC(C)=O)s1 c1(OCC(=O)NC2C(NC(=O)CCCCCF)COC2)ccc(Cl)c([N+](=O)[O-])c1 C1(C(N(C2CN(C)CC2O)CC)=O)COCCN(CCn2ccnc2C)C1 C(=O)(C(F)C(C)(C)O)N1CCN(C(=O)NCCC(=O)OC(C)C)CC1 C1(NC)CCCN(CCC(=O)NCC(C)(C)CN(C(=O)CC2CCC2)C)C1 N1(C(C(C)N(C)C)=O)CCC(O)(CNC(c2ccc(-c3ccccc3Cl)s2)=O)C1 c1(C(N(CCCNC(C2(C)CCC2(C)C(N)=O)=O)C)=O)ccc2c(O)n[nH]c2c1 Cc1cncc(C(N2CCC(N(c3c(C(N)=O)cnn3C)C3CCCC3)C2)=O)c1 C1(NC(C2CCN(C(C3(CCO)CC3)=O)CC2)=O)CC2(CCN(CC3CC3)C2)C1 c1(C(=O)OC)ccc(NCC2CN(C(c3occ(C)c3C(F)(F)F)=O)C2)cc1 N1(C(c2ccccc2)=O)CCN(C(C2CS(=O)C2)=O)CC1CO C12(CNC(C)=O)CC1CN(C(c1ncccc1C1CCCN1C)=O)C2 c1(C(=O)NC2CN(C(c3c(C)snc3)=O)CC2F)cnc2ccccc2c1 Cc1ocnc1C(=O)NCC(=O)NC(C)CNC(=O)CCc1cnccn1 N1(c2cc(OCC)ncn2)CCC(NC(=O)C(C2CC2)OC)C(O)C1 C1(C(=O)NCC(CN(C)C(c2nnn(-c3ccccc3)n2)=O)O)COCC1(C)C CCCCC(C)C(=O)NC1(CNC(C2CCN(C)C2=O)=O)CCC1 c1(CC)ccc2cc(C(N3CCC4(CCC4NC(=O)CC(F)F)CC3)=O)[nH]c2c1 c1(C(CNC(=O)C(Cl)=CCl)NC(C2CCC(C)O2)=O)ccc(C(C)C)cc1 Cn1c(C(N2CC(OCC(=O)NC(C(N)=O)C3CC3)C2)=O)cccc1=O N1(C(Cn2ncc(C#C)c2)=O)CC2(CC(CC(=O)N(C3CCOCC3C)C)C2)C1 C1(CCCC)CCCN(C(C2(NC(=O)C(F)CC3CCOC3)CC(F)C2)=O)C1 Cc1ccc(OCCC(=O)NC(C)C(CO)NC(c2cccs2)=O)c(C)c1 C1(C(=O)NC(CC)C2CC2)(CC)CCN(C(c2cn(Cc3nccs3)nn2)=O)C1 CCCC(C(=O)N1CCC1CC(=O)NC1C(OC)CC1O)C(C)C CCC(C(=O)N1CCCC1CNC(c1cn(CCSC)nc1)=O)c1ccccc1 c1(OC(C(=O)NC2C(NC(CC=CCC)=O)CCC2)C)ccc(OC)cc1 C(C)(C(C)(C)C)=CC(=O)NC(C(=O)N(C(C(=O)OC)C)C)C1CCCO1 CCC(C(=O)OC)C(=O)NC12CC(CNC(=O)CCCN(C(C)=O)C3CC3)(C1)C2 N1(C(c2cc(C)n(C)c2C)=O)CC2(CCC2)CC1C(=O)NCCC(O)C(F)F c1(C(N2CCOCC(NC(C(CC)N(C)C)=O)C2)=O)ccc2c(c1)NC(=O)C2=O C1(NC(=O)NC(COCC)(C)C)CCCN(n2nccn2)C1 N1(C(CCCC)=O)CCCC2(NC(=O)Cc3cccc4c(C)csc34)CCCC12 c1(C(=O)NC(C)CN(C(=O)CCS(=O)(=O)N(C)C)C)cc(S(N)(=O)=O)ccc1F CC1(C)CC(C)(C(=O)NC2CCC2)CN1C(=O)C(=O)NCC(F)F C1(c2n(CC)nnn2)(NCCc2ccc(C)s2)CC2(CCC(C)(C)CC2)C1 Cc1cc(C#N)cnc1C(N1CCC2CC12C(N1CC(O)(CCO)C1)=O)=O c1(C(=O)NCC2(F)CCCN(C(C(C)(O)C3CCC3)=O)C2)ncn2c1CCCC2 N1(C(CC(C(C)C)O)=O)CC(CNC(=O)Cc2nncn2C)OC(C)(C)C1 c1(C(=O)NC2CC(NC(CC(CC)c3cccs3)=O)C2)cc(Cl)cc([N+](=O)[O-])c1 c1(NC2C(CC)CCCC2)cc(C)c(I)cn1.c12c(cnn1C)N2 c1(C(=O)NCC(CC)NC(c2nn[nH]c2C2CC2)=O)c[nH]c(=NC)s1 n1(CC)c(CC2CC2)nnc1C1CCC(=O)N1.c1(N(N2CCCC2)C)cccnc1 C(C)(C(=O)NC1CC(NC(=O)Cc2cccc(OC(F)F)n2)C(O)C1)(C(C)C)OC c1(CC(N2C(CNC(CCCCC#N)=O)C3CCC2C3)=O)cc(Cl)cc2c1OCC2 Cc1cccc(F)c1CC(=O)NCCCCCCN(C)C(C1CC(C)OC1=O)=O C1(NC(C=Cc2cnc(C)s2)=O)CC2CC(NC(=O)Cn3cc(CO)nn3)C1C2 CC1(C)CCC(CNC(C2CC2CNC(C2COC2)=O)=O)OC1 C1(CC)CN(C(=O)COC2CCC2)CCC1NC(c1c(C)nn(C)c1N)=O n1(CC(=O)NC(CNC(CCS(C)=O)=O)(C)C2CC2)cc2ccccc2n1 c1(C(=O)NCc2ccc(NS(=O)(=O)CCCCl)nc2)c(F)ccnc1Cl c1(CCC)cc(C(N2CCC(N(C(=O)COC3CCCOC3)C)CC2)=O)n(C)n1 CC1(C)C(C(=O)NCC(NC=O)C)C1(C)C.c1(C2C=NS2)ccnc(OC2CC2)c1 C12CCN(CC1)C(=O)C(=O)N2CCO.c1(OC)n[nH]c(CC2CC2)n1 C#Cc1cncc(C(=O)NC2(CC=CC(N3CCN(C)C(CC)C3)=O)CCC2)c1 c1(C(N(C2CCN(C(=O)CP(C)(C)=O)C2)CCC)=O)cc(F)cc2ccoc12 N1(C(c2c(C)nccc2)=O)CC(C)C(C)(C(=O)NCC2CC23CCOCC3)C1 C=CC(F)(F)C(=O)N1CC(O)(CCNC(c2ncccc2C2CC2)=O)C1 C=CCC(CC(C)C)C(=O)NCCC1(C(=O)NCC2(CSC)CCCCC2)CC1 CC(C)(C)C(CNC(c1ccsc1C#N)=O)C(=O)NCC1C=CCOC1 C#CCC(C(=O)NCCC(C)CO)NC(C1CC2(CSC2)C1)=O C1(F)(C(=O)NCC2N(C(=O)CCn3ccnn3)CCC2)CC2(CCC2)C1 C(N=C(NC1CCC1)N1CCN(c2ncccn2)CC1)C1C(CC)C1 C#CCC(C(=O)N1CC(OCC(=O)NC2(c3ccccc3Cl)CCC2)C1)C1CC1 c1(C(=O)NCC2CN(C(C3C(C(C)(F)F)C3)=O)CC2(C)C)coc2cc(O)ccc12 C1(C(C)CNC(=O)Cn2nnc(=O)[nH]2)CCN(C(=O)C=CC2CC2)CC1 N1(C(CC2(COC)CC2)=O)CCC(NC(c2oncc2C)=O)C(OC)C1 c1(C(C)N(C)C)cn(C2CC3(C(N4CCCC4CCO)=O)CC23)nn1 C=CCC(CC(C)C)C(=O)N1CCC(C2CCCN2C(=O)Cc2nccn2C)C1 c1(NC(C)=O)cnc(C)c(C(N2CC(CC(C)NC(c3ccn(C)n3)=O)C2)=O)c1 C1(NC(C2CCC(CC)CC2)=O)CN(C(c2cc(N)cc(N)c2)=O)CC1(C)C C1(NC(CC(C)C2CC2)=O)CC(=O)N(C2CN(C(C3(N(C)C)CCCC3)=O)C2)C1 C1(NC(C(F)=CC)=O)CCC(O)CN(C(=O)C(C2CCCCC2)O)C1 C(=O)(C(C)(C)S(C)(=O)=O)NC1CN(C(COCCC#C)=O)C(C)CC1 CC(C)C(C(=O)NCC1CC1c1ccccc1OC(F)(F)F)N1CCCCC1 c1(C(=O)NC(CC)(C)CCNC(=O)C(F)OC(F)(F)F)n[nH]cc1[N+](=O)[O-] CCCC(CCCNC(=O)CCCc1nncn1C)NC(C1(CO)CC1(F)F)=O N1(C(c2nn(C)c(Br)c2)=O)CC(C2CN(C(=O)Cc3cccs3)C2)C1 C(=O)(CCCC(N)=O)N1CC(O)(C(C)NC(c2cn(CCCCF)nn2)=O)C1 C(=O)(N1CCCc2ccnn21)c1c(CNC(c2cn3c(n2)CCC3)=O)cco1 CCCC(CC)CCC(=O)N1CCOCCC1C(=O)NC1CCCC1OCC c1(C(N2CC3CCN(C(c4c(C)nsc4)=O)C3C2)=O)ccc2c(=N)[nH][nH]c2c1 c1(C(N2CCC(CNC(c3c(C(C)(C)C)ocn3)=O)C2)=O)cnn2ccncc12 C(=O)(C(C)CS(C)(=O)=O)NCC(CCCC)NC(=O)C(CC)CC C1(CCC)CCCCN1C(C1CCCN(C(=O)C(=O)NCC(F)(F)F)C1)=O N1(C(CN(C(CNc2cn(C)nc2)=O)CCO)=O)CCN(C(C2CC2F)=O)CC1 c1(NCC(C)CC(F)(F)F)ccc(S(=O)(=O)N2CCS(=O)(=O)CC2)c(Br)c1 N1(C(c2ccn(C)n2)=O)CC=CC(NC(C2CC(=O)N(Cc3cccs3)C2)=O)C1 C1(NC(N(C2CCOCC2)C)=O)CCC(=O)N(Cc2ccncc2)C1 Cc1ccc(C(=O)NC(CCF)C(=O)NC23CCN(CC2)CC3)nc1C O=C(C#CC1CCC1)NCC(C1CCOC1)NC(=O)Cc1ccc(Cl)nc1F C12(CCCCC1)CC(=O)N1CC(O)(C1)CNC(=O)C2.c1(CN(C)C)cccn1C N1(C(Cc2cccc(C(=O)OC(C)(C)C)c2)=O)CCC2C(F)(F)C2(C(F)(F)F)C1 Cc1cnn(C(C)C)c1C(=O)N(C1CCC(NC(c2cscc2C(C)C)=O)C1)C N1(C(c2ncc(CC)cn2)=O)CCCCC(NC(c2cccc(O)c2F)=O)C1 C1(C(=O)NC2(C(C)C)CCC2)CN(C)CCN1C(C1OCCCC1(C)C)=O c1(SC(N2CCC(C(c3cn(C4CC4)nn3)C)C2)=O)cccc(C#N)c1 c1(C(N2CCC3OCC(C(=O)O)C3C2)=O)[nH]c(=NC2CCCCC2F)nc2sccc12 C1(C(C(=O)NCc2cccs2)N(CCCC(=O)OCC)C)CCOC(C)C1 C1(CN(C)C(C2CCC(=O)NC2)=O)CCCN(C(=O)CN2CCCCC2)C1 C1(CCC)(C(=O)NC(C)C#N)CCCN1C(C1CC1(F)F)=O c1(C(c2nnc(C)s2)NC(=O)Nc2ccc(OCCO)cc2)ccc(F)cc1 C1(NC(CC(=C=C)C)=O)CN(C(=O)CCC2CC(F)(F)C2)C(C)(COC)C1 N1(C(C2(C=C)CCOCC2)=O)CC(CNC(=O)CC(C)(C)C#N)C2(CCC2)C1 c1(C(=O)NC2C=CC(C(=O)NCc3cn(CC#C)nc3)C2)cnc(O)c(F)c1 N1(C(CCC(C)c2ccccc2)=O)CCC(C)C(NC(C2(S(N)(=O)=O)CCC2)=O)C1 N1(CC2OCCN(C(=O)OC(C)(C)C)C(C(F)(F)F)C2)CCC2(CC1)CNC(=O)O2 C1(CC)CCC(C(=O)NCC(C)NC(=O)C(C)(C)N2CCOCC2)CC1 C1(NC(C(=CC2CCCC2)C)=O)CCCC(NC(c2ccc(C)cc2)=O)CC1 c1(C(=O)NCC(N2CCC(C(C)NC(=O)CCCCO)C2)=O)nc(Cl)ccc1F N1(C(C(C(C)(C)C)NC(C)=O)=O)CC2(CCC(CNC(=O)CC(C)C(C)C)O2)C1 C1(NC(C(N2CCCCCC2)C)=O)CC1C1CCN(C(=O)C(C)(C)N(C)C)CC1 c1(C(c2nnnn2CCOC)NCc2cc(C)ncc2)c(O)ccc(Cl)c1Cl C=C(C)CCC(C)NC(c1cc(CNC(=O)CCN2CCCC2=O)[nH]n1)=O c1(C(=O)NCC(C)(CO)NC(c2ccon2)=O)ccc(Cl)c2c1OCCO2 C1(CC(N2CCC(CC#C)C2)=O)CC(C)N(C(C2CC(C)CCO2)=O)C1 Cc1cc(C(F)(F)F)c(SCF)cc1-c1cnn(C)c1C(F)(F)F N1(C(C(N2CCC(C)C2)=O)=O)CC2(CCCN(NC(C3CC34CCOCC4)=O)C2)C1 C1(C(N2CCC(NC(C(C3CCCOC3)OC)=O)C(F)C2)=O)CC2(CCCC2)CO1 C1(C(=O)NCC2C(C(=O)NCCOCC(C)(C)O)CCO2)CCCCC1(C)C N1(C2CN(C(CCN(C3CC3)CC)=O)C2)CC(NC(=O)C(C(C)OC)SC)CC1=O C1(NC(=O)OCC)CCC2(CCCN2C(c2ccc(COCCOC)o2)=O)CC1 C1(CC(=O)NCc2ccon2)CCCC(NC(c2cncnc2)=O)C1 CC1(F)CCCCN(C(=NCc2nnc3n2CCCCC3)NCC(F)F)C1 Cc1noc(C)c1C=CC(=O)NCC1CCCN(C(=O)COCCOCCO)C1 c1(C(C)C)ccc(C(=O)NCC2CC2CNC(=O)CC2(N(C)C)CCCC2)o1 C=C=CC(C)C(=O)N1CCC(CO)(CNC(c2scnc2Cl)=O)C1 C1(C(=O)NC2(CCC(=O)NC3CCN(CCOC)C3)CCCC2)CCCCO1 c1(CNC(COC)CC2CCOCC2)nc(C)cn1C N1(C(c2c(C)c(CO)ccc2)=O)CCC2CN(C(=O)C(C)n3cncn3)C2C1 c1(NC)cnc(C(N2CCC(N(CCO)C(C3CC(C)OC3=O)=O)CC2)=O)cn1 C#CCC(O)C(=O)NCc1ncoc1C1CN(C(c2c(SC)noc2C)=O)C1 N1(CC)CCC(C#N)CC1.c12cnccc1N1CC3C(C3C1)NC2=O c1(NCC2(COC)CCC2)[nH]c(=NCC2(S(C)(=O)=O)CCCC2)nc2scnc12 c1(OC)nccc(C(=O)NC2CC(NCc3c(F)cccc3F)C2)c1F C1(C(N(CCNC(C2(C(C)C)CCC2)=O)CCOCCO)=O)CNC(=O)N1 C(CC(C(=O)N1CCC(O)(CO)C1)NC(=O)C(C)C(F)F)=CC N1(C(CC)CC)CC(C(=O)NCCOCCNC(=O)C(F)n2ccnc2)CC1=O CC(C)CCCC(=O)NC1(C(N2CC(C#N)(CCF)C2)=O)CSC1 CCCCCCC(C)C(=O)NC(C)(CSC)C(N1CCC2CC1C(=O)O2)=O c1(C(N2CCCN(C(CC3C(C)(C)C(O)C3)=O)CC2)=O)ccn2c1CCCC2 n1(CC(=C)C)c(NCC(=C)C)nnc1C1CCCCO1 N1(C(c2cccc(C)c2F)=O)C2CCC1CC(NC(C1CC3CC1C1CC31)=O)C2 CCC(CCC(=O)NC1CCN(C(=O)CCSc2nnnn2C)CC1O)OC C(C(C)(C)CNC(=O)C(C1CCN(C(c2cnn(C(C)C)c2)=O)C1)C)OC C(C)(CSC)(C(=O)Nn1cnnc1C)NC(CC(CCCC)O)=O C1(C(C)C)CCC(C(=O)NCc2nnn(C)n2)N1C(=O)CC(=O)OC(C)(C)C Cc1cnnc(C(=O)NC2(CF)CCN(C(=O)CCOC3CCC3)C2)c1 Cn1nc(C(=O)NC(=O)C(O)C2CN(c3nnco3)C2)cc1CO N1(C(c2c(COC)non2)=O)CCC2(NC(=O)Cc3c[nH]nc3O)CCCC12 N12CCCC(C1)C2.CCCCCCN(CCCCCC1(O)CCC1)CCC#N n1(CC)c(C)nn(CC(=O)NCC(O)CCNC(C2(C)COC(=O)C2)=O)c1=O C(CCN(CC(C)C)N1CCC2(CCCN2C)C1)OC c1(SC)cccnc1C(N1CCC(C(C)NC(=O)CN2CCOCC2)C1)=O N1(C(c2csc(C)c2N)=O)CC2CCCC(NC(c3cc(C(N)=O)[nH]n3)=O)C2C1 C1(NC(=O)C2=C(Cl)CCC2)CC2(CCN(C(C3(C(F)(F)F)CCOCC3)=O)C2)C1 N#Cc1cccc(CCNC(=O)CN(C(=O)C=Cc2cccnc2)C2CC2)c1 Cc1cc(C(=O)NCC2(C(C)NC(c3cnn(C)c3)=O)CC2)cc(F)c1 c1(C(=O)NC(CCCCNC(CC2(OC)CC2)=O)C)ccc(F)cc1Cl N1(C(C(C=C)C)=O)CC(CCNC(C2(N3CCCC3)CC2)=O)OC(C)C1 S(=O)(=O)(c1ccc(C(=O)OC2CN(C(=O)OC(C)(C)C)C2)c(Cl)c1)NCCON c1(CC(=O)NC2CCCN(c3nc(C#N)cc(C)n3)C2)cccc2ccncc12 c1(C(C)NCCC(C(C)(C)C)c2nnnn2C(C)(C)C)cccnc1F CC(N=c1ccnc(NCc2cccc(N3CCCC3=O)c2)[nH]1)C1CCC1 c1(OC)ccc(C(N2CC3C(NC(c4ccn(C)n4)=O)C3C2)=O)nc1 C1(NC(c2cc(CCC)ncc2)=O)C2CCN(C(=O)Cn3ncnn3)CC12 C1(NC(=O)NCC(C(C)C)C)CCCC1(C)NCC(F)(F)F Cc1cc(C(N2CCN(C(c3n[nH]c4c3COC4)=O)C3CC23)=O)n2ncnc2n1 Cc1[nH]nc(C(=O)NC2(C)CCN(C(=O)CCC3CCCN3C)C2)c1Cl Cn1ncc(C(=O)NCCCCC2CN(C(c3cnc(C(C)(C)C)s3)=O)C2)n1 N1(c2ccnc(CNC(C3C(CCC)C3)=O)n2)CCOCC(OC)C1 CC1CN(C(C2(F)CCCOC2)=O)CC1NC(c1nccn1C)=O N1(C(C=C(C)C(C)C)=O)CCC(NC(c2cc3nnn(C)c3s2)=O)C(CO)CC1 C1(C(N2C(C(=O)OC)C=CCC2)=O)CN(C(c2nn(C)cc2C)=O)CC1(F)F C(C(F)(F)C(=O)NC1CC(C)N(C(=O)CSCCC(F)(F)F)C1)OC Nc1cccc(CCC(N2CCCC2C2(NC(=O)C=CC3CCCO3)CC2)=O)c1 C1(C(=O)OC)CCN2CCC1c1nc2nc2n1ncc2.C(F)(C(=O)NC)=CCC N1(C(C2CCC(C)(C)C2)=O)CC(NC(c2ccc(CC3CC3)s2)=O)C2(CC2)C1 C(C(C)(C)C(=O)NCC1CC(C)N(C(=O)CCc2ncc(F)cn2)C1)OC c1(C(=O)NC(c2ccnn2C)C(=O)NC(C)C(C)(C)CO)cccn2cncc12 C1(NC(C(CC)C)=O)(CC)CCN(C(C2CC(NS(C)(=O)=O)C2)=O)CC1 C(=O)(C(CN(C1CC1)Cc1nn[nH]n1)CC1CCOC1)OCC C1(C(C)(C)C)C(NC(C2CCC(=O)NC2)=O)CCN1C(=O)CNc1nccs1 C(=O)(CCCCCNC(=O)COC)NCCC1CN(C(C=CCC)=O)CC1C N1(C(Cn2c(C)cnc2)=O)CC(C2CCCCN(C(=O)C=C3CCSCC3)C2)C1 c1(NC(=O)COCSCCC2CC(NC(C3CCCO3)=O)C2)cnc(Br)o1 Cc1ncccc1C(N1CCC(C(C)(C)CNC(=O)CC(O)CN(C)C)CC1)=O C(=O)(CC(C)(O)CCC)NCc1c(CNC(COCCC=C)=O)cccn1 CN=S(C)(=O)c1ccc(C(=O)N(C(C)CNC(=O)CCn2ccnc2)C)cc1 Cc1ccc([N+](=O)[O-])cc1C(N1CC(NC(=O)C(C)C(F)F)CC1C)=O N1(C(c2ccc(C(F)(F)F)o2)C(=O)NC(CC)C)CCOCC(O)C1 c1(C(=O)NCCC(=O)NC)cc2c(s1)CCN(C(c1cc(COC)[nH]n1)=O)C2 c1(CNC(=NCC)N)ccc(C)c(N2CCN(C)CC2)c1.C1(N)CCCCC1CC C1(NC(C=C(CC)C)=O)CC2(C1)CN(C(C1(c3ccc(Br)s3)CC1)=O)C2 CC1=C(C(=O)NCC(F)CNC(C2CCCCN2C)=O)C(C)(C)CCC1 c1(C(=O)NCC2CCC(NC(c3csnc3Cl)=O)C2)ccc(=O)n(C2CC2)c1 C12(C(=O)NCCN(C(C(C(C)O)C)=O)C3CCCCC3)CC3CC(CC1C3)C2 c1(C(N(CCC(C(C)C)NC(=O)CCCCC#N)C)=O)cnc2cc[nH]c2c1 C1(CC(C)NC(CCC=CC(=O)NC)(C)C)CCC(C)(C)CC1.N1(C2CC2)CCOC1=O C1(NC(C(C2CC2)SC)=O)CCC(C)N(C(c2cccc(-n3cncn3)n2)=O)C1 c1(C(C)(C)NC(=O)OCc2cnc(C3CCC3)s2)ccc(C(F)(F)F)cc1 N1(C(c2c(CC)c[nH]n2)=O)CCCC(NC(c2cccnc2F)=O)C1C c1(C(=O)NC2CC(n3cc(C(CC)(O)CC)nn3)C2)cnc2c(c1)C(=O)CCC2 c1(C(=O)NC2CC(O)CCN(C(c3c(C#C)c[nH]n3)=O)C2)ccc2ccoc2c1 N1(C(C2(C(=O)OC)CC2)=O)CCCCC(CNC(C2(C)CC3CCC2O3)=O)C1 C1(NC(C2(CC(C)C)COC2)=O)CCCC1NC(=O)CC(C1CC1)C1CC1 C1(CNC(=O)CC2CC3(CCC3)CO2)CCC2CN(C(=O)Cc3ccsc3)CC12 C(=O)(C(C)CC(C)(C)C)NC1C(F)CCN(C(CCOCCN(C)C)=O)C1 c1(C(=O)NC2CN(C(C3CCC(C)(C)CO3)=O)CC2O)ccc2c(c1)CNC2=O Cc1nc[nH]c1CC(N1CCC1CN(C(C1CN(c2ccncc2)C1)=O)CCO)=O Cc1scc(C(=O)NC(C(=O)NCC(c2nncn2C)C)C2CCCC2)c1C Cc1cc(Cl)ccc1C(=O)NCC1CCCC1NC(=O)CC1COC(C)(C)C1 CC1(C)CC(CNC2CC3C=CC2C3)CCO1 c1(C(=O)OC)cnc(C(=O)NCC(C2CCC2)NC(=O)C(O)C2CCCC2)cn1 C1(C(=O)NC2CC(C(=O)NC(C)Cn3cccn3)C2)COc2ccccc2O1 C(=O)(CS(F)(F)(F)(F)F)NCC(CCCC)NC(c1nocc1C)=O c1(C2C(C(N3CCC(CNC(=O)CCc4ncco4)C3)=O)C2)ccccc1Cl c1(C(N(CCNC(c2ccc(F)s2)=O)CCOCCO)=O)cccnc1O Cc1cn2cc(C(=O)NC3(CCNC(=O)CC4CC4C4CC4)CC3)sc2n1 C12(CNC(N(CC(C)(C)C)Cc3ccc(Br)cc3)=O)COCCN1CCOC2 c1(C(=O)NCCCN(CCC)C)n[nH]cc1CNC(=O)C(C)N(C)C(C)=O C(=O)(C#CC1(C)COC1)N(C1CCCN(C(C=Cc2n(C)ncc2)=O)C1)CCF c1(CC)cc(C(=O)NC2CC(C)(CNC(=O)C(C)COC)C2)oc1CC N1(C(COC(CC)(C)C)=O)CC2CC(O)C1C2NC(=O)CCn1cc(C)cn1 CCN=C(NCc1ccoc1)NC(C)CC(N)=O c1(OCC)cc(C(=O)NCC=CCNC(=O)CCOCCC(C)C)cc(Cl)c1 C1(NC(c2ccc(C)c(Cl)c2)=O)COC2C(NC(=O)C(C)OCC(C)C)COC12 c1(OCC=C)c(OC)cc(C(=O)N(CCCNC(=O)C=CS(C)=O)CC)cc1OC c1(CN(C(C=CCN(C(CCSCCCC)=O)C)=O)CC)nc(C)c(C)s1 CC(=O)CCCC(=O)NC1CCCN(C(C2CCCN(C)C2)=O)C1C C1(NC(=O)NC23CC(C)(C2)OC3(C)C)CCc2ncc(Br)n2C1 C(=O)(C(C)(C)CCSC)N1C(CC)C(NC(c2csc(F)c2)=O)CC1 Cc1nnc2cnc(C(N3CC(CNC(c4cscn4)=O)OC(C)(C)C3)=O)cn12 c1(C(=O)NCC2(O)CCN(C(Cn3ncc(CC)c3)=O)C2)ccc(OC)c(Cl)n1 C1(C(N(CCN(C(=O)CC2CCCNC(=O)C2)CC)CC)=O)CCCC1C1CC1 C12(CO)CCN(CC1)CC1CCN2C1.c1(NC(=O)NCCC)nn(C)c(C)c1Br N1(C(C2CCN(C(CC3C(C)=NNC3=O)=O)C2)=O)CC(C)Oc2ccccc21 C[Si](C)(C)C1CCCC(C(N2CC(c3cn(CCCNC=O)nn3)C2)=O)C1 C(=O)(CC(C)CC(C)(C)C)NCC(N1CC2CCN(C(CNC(C=C)=O)=O)C2C1)=O c1(C(N2CCC(N(C(Cc3nnc(C)s3)=O)C)C2)=O)nc(C2CC2)oc1C CCC(CC(F)(F)F)C(=O)N1CCCC(C2CCCCN2C(C2SCCS2)=O)C1 N1(Cc2c(C)nsc2C)CCC(C2CCCN(C(c3cnn(C)c3)=O)C2)C1 N1(C(C2C(C(=O)OCC)C2)=O)CCC2CCCC12C(N1CCC(n2cnnn2)C1)=O c1(NC(C(CNc2n(C)cc(NC(C)=O)n2)(C)O)=O)ncnc2ccsc12 c1(CCC)cc(CN2CCCCC2CCOC(C)(C)C)c2ccccn12 C1(C(N(C2CCNCC2)C)=O)CCCN(CC2CCCC2(C)C)C1 N1(C(C2CCC(=C)CC2)=O)CCN(C(=O)C(C)S(N)(=O)=O)CC1C(F)F Cc1cnc(C(=O)NC(c2cn(-c3cc(F)ccc3F)nn2)C)cc1C c1(OC)ccc(Br)c(CNC2CC(C)CN(C(C3CC4C=CC3C4)=O)C2)c1 S(=O)(=O)(c1ccc(N(C)CCN(C)C)c(Br)c1)NCC1(C)CCC(C)CC1 C1(N(C(C(C)OCCOCC)=O)C)CCN(C(=O)CC2CC=CCN2C)CC1 Cc1nc(O)ccc1C(=O)NC1CN(Cc2c(C)n[nH]c2C)CCC1C c1(C(=O)NC2CCC(CC)C2)ccc2ncsc2c1 C1(CC=C)(NC(c2cnn(CCO)c2)=O)CCN(C(=O)C(C(C)C)N(C)C)CC1 Cc1ccnc2[nH]cc(CC(C3CC3)Nc3ncccc3[N+](=O)[O-])c12 CCCCC(C)(F)C(=O)N1CC(CCCCNC(c2cn3nc(C)sc3n2)=O)C1 C#Cc1cnc(C(N2CCOC(CCCNC(c3c[nH]nc3Cl)=O)C2)=O)c(C)c1 Cc1ccc(C(=O)NCC(C)CN(C)C(C2(C)CCC(C)C2)=O)c(C)n1 Cc1nnc(C(=O)NC(CNC(=O)CCC2(C)CC2)C2CC2)o1 Cc1cc2scc(CC(C)C(N3CCC4CN(C(C5(C)CC5)=O)CC34)=O)c2s1 CC1CCc2nc(C(N3CCC(NC(C4CC(=C5CC5)C4)=O)C3)=O)cn2C1 c1(N2Cc3c(=N)[nH][nH]c(=N)c3C2)ccc(S(=O)(=O)NC2(CO)CCSC2)cc1Cl c1(CCC(=O)NC(CNC(=O)CC2CC2(F)F)CO)ccc(Cl)cc1F CC(N=c1[nH]c(=NCCc2ccc(Cl)nc2)c2ncccc2[nH]1)c1cscn1 C1(CN(C(c2ccc(C)s2)=O)C)C2CN(C(=O)C(N3CCN(C)CC3)(C)C)CC12 Cc1cc(C(N2CCC(OCCNC(=O)C(C)N(C)C)C2)=O)c(C)s1 c1(C(N2CC3(CN(C(c4cccc(C(=O)OC)c4)=O)C3)C2)=O)cc2ccccc2o1 N1(C(C=CC(c2ccccc2)=O)=O)CC(NC(C2CCC(=O)N2)=O)C(F)C1 c1(NC(C(=O)NC(C)CC)=O)ccccc1C1(C)CC1(F)F.N12CC3CC1C3C2=O c1(CNC(CC2N(C(c3c(C)ccnc3)=O)CC(F)C2)=O)ccc2nonc2c1 CC(C)C(O)C(C)C(=O)NC1CCOC1C(N1CCC(O)C(F)(F)C1)=O c1(C(=O)NC(C2CN(C(=O)C3=NNC(=O)CC3)CCO2)C)ccc(Cl)c(F)c1O Cc1ncc(C(N2CCOC(CCNC(C3(C)CCNC3=O)=O)C2)=O)cc1N c1(C(=O)NCCC(C)NC(=O)CC2CCC(C)(C)C2)cncc(-c2ccoc2)c1 C(C(O)CN(C(=O)C(F)n1ccnc1)CCOC)OC(=O)C(C)OC(C)(C)C C1(CC=C)(NC(C2CC2C)=O)CCN(C(=O)C(=Cc2ccccn2)C)CC1 Cc1cc(F)c2c(c1)CCC2NC(=O)Nc1ccc2c(c1)OCC2 C1(C(=O)NC(CCC)CCC)CC2(CCN1C(=O)C(C)SC)CC2 CCC(C)(C(=O)NCC(CNC(c1csc(-c2cccc(Cl)c2)n1)=O)OC)OC c1(C(=O)NCCNC(N2C(C)COCCC2)=O)c(F)ccc(F)c1Cl N1(C(=O)CCNC2CCCCC2)CCC2C(CCN2C(C2CC2CF)=O)C1 CC(CC(F)F)C(=O)NCCN(CCOCCO)C(c1c[nH]nc1C1CCCO1)=O CCC(C)(CNC(C1(F)CCCN(C(c2cc(OC)ns2)=O)C1)=O)C(N)=O c1(OC)cnccc1C(F)(F)C(=O)NC1CC(O)(CN(C)C)C1 C(=O)(C(F)(CNC(C1(C(C)C)COC1)=O)C(C)C)NCC1(C#C)CCCC1 c1(N(CC=C)C)nc(N2CC3C(C2)C3(C)C)nc2c1ncn2C(C)C C12(NC(c3n(C(C)C)ccn3)=O)CCN(C(=O)CC3CCSCC3)CCC1C2 C1(CC)CN(C(C2(C(=O)NC)CC2)=O)CCC1NC(c1cnc(Cl)cn1)=O C(=O)(CCC(C)(C)F)NC1C(NC(C=Cc2ncn(C)c2)=O)C1 C1(NC(CC=C)=O)CN(C(c2ccc(Cl)c(OC(F)(F)F)c2)=O)CCC1(F)F c1(C(N(C(CC)CC(=O)N(C2COC(C(C)C)C2)C)C)=O)cccc(C)c1N c1(C(=O)NC2C(NC(=O)COCc3cn[nH]c3)CCC2)ccc(F)cc1C1CC1 C(=O)(C(O)CN(C)C)N(CC(CC)NC(=O)C(C)OC)C C(C)(CCC(=O)NCc1cccc(CCO)c1)OC.C12(CC1)CC(=O)NC2 c1(C(=O)NCC2CN(C(C(C(C)C)O)=O)CC2C)cccc2c1CCCC2 CC(C)(C)CCC(=O)C(=O)N1CCCC1C1CCN(C(c2cnc3n2CCS3)=O)C1 c1(CC(=C)C(=O)N(C(C)CCC)CCCC)ccc(F)cc1F N1(C(Cc2c(C)noc2C)=O)CC2CN(C(=O)C(c3cccc(O)c3)C)C2C1 c1(-c2n(C(C)C(F)(F)F)nc(-c3cncc(Br)c3)n2)ccc(Cl)cc1Cl N=c1sccn1CC(=O)NC1(CO)CN(C(c2ccsn2)=O)C1 Cc1ccc(C(=O)NCC2(C(C)(C)O)CN(C(=O)C3=NOC(C)C3)C2)cc1O CCC(C)(C)C(=O)NC12CC1CN(C(C1(c3cncnc3)CCCC1)=O)C2 c1(CC(CC)NC(c2nnc(-c3cccnc3)s2)=O)cccc(C)c1 c1(C(N2C(C)CC(CNC(CC3(C=C)CC3)=O)C2)=O)cc(C)c2[nH]cnc2c1 C1(NC(CN(C)C)=O)CCCC1NC(=O)C(CO)NC(c1ccccc1)=O c1(C(N(CCCNC(=O)C(O)COC)CC)=O)cn2cnnc2cn1 c1(OC)cc(CC(=O)NCC2CC(c3ccccc3)CO2)c(F)cc1Br c1(C(N2CCC(NC(CCCn3c(C)nc(C)n3)=O)C2)=O)ccn2c1CCCC2 CCCCCCCCCNC(=O)C(=O)NCCCC1CNC1 C1(N(C(c2c(C)nco2)=O)C)CCCCC1N(C)C(c1n[nH]cc1Cl)=O Cc1nc2ccc(F)cc2c(C)c1CCCNC(N1CC2COCC(C1)C2(F)F)=O C(=O)(C(C)(F)C(C)(C)F)NCC(CC(C)C)NC(C1CCCC2C1C2(F)F)=O N1(C(CCC(C)OCC)=O)CCC(NC(=O)CCCN(C)C)C2(CCC2)C1 CS(=O)(=O)c1ccc(C(N2CC3(C2)CN(C(=O)CC2CCC4CC24)C3)=O)o1 C1(C(=O)NC2CC(O)C2)COCCN(C(=O)NC2CCN(c3nccs3)CC2)C1 C(=O)(CC(CNC(N)=O)C(F)F)NC(CN(CC(C)C)C)C N1(C(C=Cc2n(CC)ncc2)=O)CCC(C2CC2NC(C2(COC)CC2)=O)CC1 C1(C(=O)NCCC=C=C)C=CCN(C(C2CCCC2CCC)=O)C1 C1(C(=O)NC2CCC(F)(F)C2)CC2CCC1N2C(c1cccc(Br)c1F)=O N1(C(CC(C)n2ccnc2)=O)CC2(COC(CNC(=O)Cc3ccsc3)C2)C1 N1(C(CCOCCC)=O)CC(C(=O)NC(C)CCC(=O)OC)CCC1(C)C N1(Cc2ccc(Nc3ccccc3)cc2)CCC2CCC(C1)S2 C#Cc1ccccc1C(N1CC(NC(c2cc3sccc3s2)=O)C(C#N)C1)=O c1(CC(=O)N(CC(CNC(COC)=O)O)C)cccc(Cl)c1F c1(C(=O)NCC=CCNC(c2c(CCC)occ2)=O)cc(C)nc(COC)n1 N1(C(C2CC(C)(CC)C2)=O)CCCCC(NC(c2csc(-c3cnc[nH]3)n2)=O)C1 C(=O)(CCCCCCN=[N+]=[N-])N1CC2N(C(c3c(C)cc(F)cc3)=O)C(C2)C1 c1(OCCNC(=O)NCC2CCCOC2)cncc(Br)c1 C1(C(C)NC(CC2(NC(C)=O)CC2)=O)CCCN(C(c2cc(Cl)no2)=O)C1 c1(C(=O)NCC(C(C)C)NC(C2C(OCF)(OC)CC2)=O)ccc(N(C)C)cc1 c1(C(=O)NC2(CNC(c3cn(C)nc3O)=O)CCC2)ccc(NS(C)=O)cc1Cl C(=O)(CCCCCN(C)C)NCCCCC1CN(C(C(C)n2ccnn2)=O)C1 c1(C(=O)NCCC2N(C(C3CCC(CC)O3)=O)CCC2)ccc(N)c(C(C)=O)c1 C1(C(=O)NCC2C(NC(=O)Cc3cnc[nH]3)C2)CC2(CCC2)CO1 CCCCCC(CC)C(=O)NC(C1CCCN1C(c1ccc(CC)nc1C)=O)C Cc1ncc(C(N2CC(C(N3CCC3CN=[N+]=[N-])=O)CC2(C)C)=O)c(=N)[nH]1 C1(CNC(CNC(CC)=O)=O)CC2CCC1N(C(C1(C3CC3)CCC1)=O)C2 c1(C(=O)NCC2CCC(NC(C(CC)(CC)OC)=O)C2)cnc2ccc(C)cn12 CC(C)CC(O)C(C)C(=O)N(C(C(=O)NCCCN1CCCC1)C1CC1)C C#CCC(C(=O)NCCCOCCN(C(=O)C(C1CCCCCC1)C)C)C1CC1 C1(CF)=NC(NCC2CC3(CCC3)CO2)=CC2=NC(CCOCC3=CCOC3)C2N1 C1(C(=O)NC2CC(NC(CSCCC(C)C)=O)CC2O)CCC([N+](=O)[O-])CC1 N1(C(c2c(C)ncc(Br)c2)=O)C2CCC1CN(C(=O)CC13CCCC1C3)C2 C=CC(C)(CCOC)C(=O)N1CCCN(C(=O)COCC(F)F)C(C)C1 N1(C(c2scc(C)c2)=O)CCC2(C(N3CC(c4nncn4C)C3)=O)CCCC12 C(=O)(C(C)(C)CCNC(=O)C(C)OCC1CC1)Nc1cnc(OCC)nc1 C(=O)(C1CCc2nccn21)N(CCNC(C(CC#C)C1CC1)=O)C(C)C C1(C(NOCCC(=C)C)=O)CN(C(=O)CCc2nc(=N)[nH][nH]2)CCO1 c1(C(C)SCCN2CCOC2=O)c(F)cccc1F Cc1ncc(CCC(N2CC(CNC(c3ccccc3C)=O)C3CC23)=O)c(O)n1 c1(C(N2CC(NC(c3ccncc3)=O)CC23CCC3)=O)cc2c(Cl)cccn2n1 c1(C(=O)Nc2nc(C(=O)NCCC)n(C)c2)ccc([N+](=O)[O-])c(C)c1 CC1CN(C(c2ccc(C#N)cc2)=O)CCC1NC(=O)CS(=O)(=O)CC1CCC1 c1(COC)nc(OC)cc(N2CCC(C)(Nc3cnns3)C2)n1 C1(NC(c2cc(OCC)no2)=O)CC2CCC(C1C)N2C(C1CC2CCCC12)=O c1(C(N2CC(CNC(CCCC=C)=O)C(O)C2)=O)c(C)ncnc1C C(=O)(C1(C)CCc2ccccc21)N1CC2(C(NC(C3CC(C)C3)=O)CCC2)C1 N1(C(CC2CC(=C)C2)=O)CC(NC(c2ccc(NC(C)C)cc2)=O)C(C2CC2)C1 C1(CO)CCOCC1C(N1CCC(C2OCCO2)C1)C(=O)OC C(C)(CN=C(NCc1cc(Cl)cc(Cl)c1)NC1CCN(C(=O)OC)C1)OC N1(C(COC)=O)CCN(CCN(C)C(c2nc(C)oc2OC)=O)CC1 c1(C(=O)NCCCCn2cc(C(CC)O)nn2)ccc(OC)c(F)c1CC CCC(C(=O)N1CCC(CF)(NC(=O)Cc2ccoc2)C1)C(C)(C)CC C=CC1(CC(N2CCCC(F)(C(=O)NOCCN3CCNC3=O)C2)=O)CCCCC1 N1(C(CCNC(c2nccc(N)c2)=O)=O)CCCCCC1c1ccccn1 CN1C(=O)NCC1C(N1CCC(CCNC(=O)C(c2ccccc2F)(C)F)C1)=O C1(CCCC)CN(C(=O)CC2CC(=O)NC2=O)CCN1C(c1cn(C(F)F)cn1)=O C1(CNC(C=COCC)=O)CC(C)(C)CN1C(c1cnn(C)c1N)=O Cc1c(Br)cc(Cl)c(NC(C2CCN(C(c3ccc[n+]([O-])c3)=O)CC2O)=O)c1Cl C1(NC(C2C(C)CCC2)=O)CC2CN(C(C3CCCN3C=O)=O)CC12 C1(NC(c2cn(C)nn2)=O)CCCCN(C(C2(N(C)C)CCCCC2)=O)CC1 c1(C(N2CC(OC)C(NC(c3cc(C(C)C)no3)=O)C2)=O)cc(C)ccc1F C1(CNC(CC2(OC)CC2)=O)CC(F)(F)CN1c1nc(C(N)=O)ns1 C1(C2CCN(C(c3ccncc3Cl)=O)C2)(NC(c2cc(C)c(C)nc2)=O)CC1 C1(CC(=O)NCC)CCN(C(c2cc(C(F)(F)F)on2)=O)C1(C)C c1(C(C)Nc2csc(N3CCOCC3)n2)cc(F)cc(Br)c1 c1(C(=O)NCC2N(C(C(C=C=C)C)=O)CCCC2)cc(O)nc2[nH]c(=N)ccc12 C(=O)(C(F)(F)C1=CCOCC1)N1CC2CC(CN(C(C3(C)C(C)OCC3)=O)C2)C1 c1(C(=O)NC2CC(NC(CCCSC)=O)CC2O)cc(C)c(F)cc1Cl c1(C(=O)NC(CCCNC(Cc2cc(C)nn2C)=O)C)cccc(F)c1N c1(OC(C)C)ccc(CN(C)C(c2cnn(CCc3ccccc3)c2Cl)=O)cc1 c1(CNC(C(C)NC(CC)=O)=O)n[nH]c2c1CN(C(C1CC(CC)=NO1)=O)CC2 C(=O)(C1CCCn2nccc21)NC.N1(C(C(C=C)(C)O)=O)CCC2C(C1)CN2 O=C(C#CC1CCC1)NCC1(O)CCN(CCCC2CCOC2)CC1 C1(NC(=O)CSc2ccsc2Br)CCCCC1NC(C1CNC(=O)N1)=O N1(C(C2OCCN(C(c3csc(C)c3C)=O)C2)=O)CCC(O)C(F)C1 C1(NC(c2ccc(COCCCN)cc2)=O)CCC2CCCC2C1 c1(CNC(C2CCN(C)C2c2cnn(C)c2)=O)ccc2cnccc2c1 C1(NC(CCc2onc(C)n2)=O)CN(C(c2cn(C3CC3)cn2)=O)CCC1C C1(CNC(CC(=O)NC)=O)COCCN(C(=O)C#CC2CC2)C1 c1(CNC(N2C3CN(C(c4ccccc4Cl)=O)CC23)=O)cc2cc[nH]c2cc1Cl c1(NC(C2CC2Cl)=O)cccc(NC(=S)NCc2nccs2)c1 c1(C(N(C)CC2CCN(C(c3n[nH]cc3C(F)(F)F)=O)C2)=O)cc(N)cc(O)c1 C1(C(=O)NCC(=C)F)CC12CCN(C(=O)Cc1cccnc1)CC2 C(C)(CCC(=O)NCC(CC1CC1)C(=O)Nc1cccnc1C1CC1)OCC CC(C)(C)C1=NOC(C(=O)NC(C)(CNC(C2CC3C=CC2C3)=O)CO)C1 N1(C(COCC(=O)OC)=O)CC2C3CCC(C2C1)N(C(=O)C(C)OCC(C)C)C3 C1(CCNC(C=C(C)C(F)F)=O)CC2CCC(C1)N2C(=O)C=CC(c1ccco1)=O Cc1cnccc1C=CC(=O)NCC(C)CN(C)C(C1CC1(F)F)=O c1(C(N2CCC(NC(c3c(CC)scc3)=O)C2C2CC2)=O)ccc(=O)n(C)n1 c1(OC)ccccc1C=CC(=O)NCCC(CNC(=O)Cc1cnnn1C)OC C(=O)(CS(=O)(=O)CCOC)NCC(CC(=O)NCCC1(CC)CCC1)O Cc1oc(C(C)C)nc1C(N1CC(n2cc(C(n3cncn3)C)nn2)C(C)C1)=O c1(C(N(C(CC)CNC(=O)CCSC)C)=O)ccc(C)cc1 C(=O)(C(Cc1ccco1)NC(=O)C=CC(C)(C)C)NCC(COC)C c1(CCC(=O)NC2C(CNC(c3cn(COC)nc3)=O)CC2)c(F)cccc1F c1(C(C(=O)NCCC(=C)CNC(c2nc(Cl)cs2)=O)C)ccc(OC(F)F)cc1 CC(C)C(O)C(=O)N1CCC(OCCCNC(C2(C(=O)OC)CC2C)=O)CC1 C(CCCC(=O)N(CCCC)C(C)C)NC(C1C(=C)C1)=O C1(NC(C2(N(C(=O)CCC3CCOCC3)C)CC2)=O)CCCC1CF C1(Nc2cc(OC)c(OC3CC(=O)NC3=O)cc2)CCCN2CCCCC12 c1(CCC(=O)NCC2CC2NC(c2nc(Cl)sc2Cl)=O)c(F)cccc1Cl C1(CC(=O)NCC(CNC(c2ccc(C)nc2C)=O)OC)CCC2(CC2)CO1 C(=O)(C(C)(F)C(F)(F)F)N(CCNC(c1cc(CC)oc1C)=O)Cc1ccccc1 c1(N2CCC(CCOC)C2)cc(NC(C)C)nc(C)n1.c12cc(no1)N2 C(=O)(CS(=O)(=O)CCCC)NC1CN(C(C(F)=CCC)=O)C(C)CC1 C1(CNC(CC=CCNC(CC2N(C)CC=CC2)=O)=O)CCC=CCCC1 N1(C(c2c(N)ccc(Cl)n2)=O)CCc2nc(CNC(=O)CCC3CCC3)sc2C1 C=CCC(C)(O)C(=O)N1CC2(C(=O)NCCCOCC(C)C)CC1CO2 c1(N2CCCC(CNC(C(C)OCCOC)=O)C2)nc(C)nc(O)c1C C12(NC(c3cc(C(C)=O)oc3)=O)CCCCC1CN(C(=O)C(N)=O)C2 C1(OC)CCC(CC(=O)NC(c2c[nH]cc2C(N)=O)=O)C1.C12(CCC1)CC(=O)N2 CC1CCCn2c(C(=O)NCC(O)CNC(=O)CSCc3ccncc3)cnc21 CCC(CC)C(C(=O)OC)CC(=O)NCCN(C1CCCC1)CCc1ccccc1 C1(CC)(NC(c2ncncc2Cl)=O)CCN(C(C2(Cl)CC2(F)F)=O)CC1 c1(C(=O)NC2CCC(CNC(c3ccc(Br)o3)=O)C2)ccnc(S)c1 C12(C(N3CC(C(C)NC(C4CC5(CSC5)C4)=O)C3)=O)C=CC(CC1)C2 C1(C(=O)NC2(COC)CN(C(=O)C(C)C(C)COC)C2)CC2(CCCCC2)C1 C(C)(C(CC(=O)NCC1(F)CCOC1)NC(=O)Cc1ccsc1)OC C(=O)(CC(CC(C)C)NCCc1ccn(C2CC2)n1)NCC1CCC(CC)O1 CC(C)C(C)C(CNC(=O)CCCCCF)NC(C1CC(N2CCCC2)C1)=O C(CC(=O)Nc1c(C)nn(CC)c1C)(C(F)F)NC(c1cccc(CC=C)c1)=O c1(N(C)C)ccc(C(=O)NCC2CCC(CCNC(=O)Cc3ccno3)C2)cc1 CC1CCC(C(=O)NC2CCCC2NC(c2cc(Br)sn2)=O)C1 S(=O)(=O)(c1ccc(F)cc1)N1C(CC(C)C)C(=O)N(C)CC1 C12(NC(C34CC(C)C3C4)=O)CCCC(CN(C(c3cocn3)=O)C1)C2 C1(Nc2c(CC)ccc(C(F)(F)F)c2)CCN(C(=O)OC(C)(C)C)C2(CC2)C1 C(CCCCC(=O)N(C)Cc1cnco1)NC(c1c(CC)n(C)nc1)=O c1(OC)cc(N2CCCC(C(=O)NC3(CSC)CC3)C2)ccc1[N+](=O)[O-] C12(NC(Cc3ccc(CC)cc3)=O)CCCC1N(C(C1(C)C=CCCC1)=O)CC2 c1(C(=O)NCC2(C)N(C(c3ncc(OC)cn3)=O)CCC2)ccc(C)c(Cl)c1F C1(NC(c2cn(CC=C)nn2)=O)CCCCC12CCCN(C(C1(C)CC1)=O)C2 C1(CC(=O)NC2CC(CNC(CCCOC(C)=O)=O)C2)CCC(C)(C)O1 C1(C(=O)NC(C(N2CC(=C)C2)=O)C2(O)CCC2)CCCC(=O)C1 C12(CC)COC(C(N3CC(CNC(c4ccnc(N(C)C)c4)=O)CC3C)=O)(C1)C2 N1(C(c2ccc(OCC)cc2C)=O)CC(C)CN(C(=O)COCC2CC2)C(C)C1 c1(C(=O)NCCN(C(C2(CCC)CC2)=O)CC2CC2)cccc(CC(F)(F)F)c1 Cc1nscc1CC(=O)N(CCCN(C)C)CCNC(=O)C=CBr C(=O)(CCCCc1cnc[nH]1)NC1CC(C)(NC(CCOC)=O)C1 C1(N(C(C(c2n[nH]cc2Br)N(CCC)CCC)=O)CCC2CC2)CCC(F)(F)CC1 c1(C(=O)OC)ccc(Br)c(NC(=O)Nc2c(-c3ccncc3)noc2OC)c1 c1(C(N2CC3C(CNC(C4(CO)CCCO4)=O)C3C2)=O)ccc(F)c(Cl)c1 C1(C)(CNC(C2N(C(C3C(CCC)CCC3)=O)C(C)C2)=O)CSC(C)=N1 C(=O)(C(CCOCCO)N(C1CCCC1)C(=O)CN1CCCCC1)N(CC#CC)C c1(C(N(C)CC2(NC(C3CC(CCC)C3)=O)CC2)=O)ccc(CC)cc1O N1(C(C2(CC)CC2)=O)CCC(CN(C)Cc2ccc(C)o2)C1 C(=O)(C1CCc2c[nH]nc21)NC1CN(C(c2c(F)ccc(OC)c2)=O)CC1C1CC1 c1(OC)ccc2cc(C(C)C(=O)NC(C)(C)CNC(=O)C=CS(C)=O)ccc2c1 Cc1cc(NC(=O)C(=O)NCC(CC(C)C)NC(=O)OC(C)(C)C)ccc1Cl C1(NC(c2c(CC)[nH]nc2Cl)=O)CCCN(C(c2ccn(C)c2C)=O)CC1F CC(C(=O)NC(C)(CNC(=O)C=CC(F)(F)F)C1CC1)NC(N)=O C1(NC(C(CC)OCC)=O)COCCN(C(c2coc(C(F)(F)F)n2)=O)C1 CCN=c1cc(C(=O)NCC2CC(NC(=O)C(n3nc(C)cc3C)C)C2)cc[nH]1 N1(C(CSC(C)C)=O)CCC(NC(=O)CC2(O)CCCC2)C(F)(F)CC1 c1(C(=O)NC23CC(CNC(C4CCCOC4)=O)(C2)C3)occ2c1CCCC2 C(=O)(C(O)CC(C)C)NCC1N(C(CCc2cc(C)ncn2)=O)CCCC1 c1(C(N2CC(CNC(C(n3c(C)cc(C)n3)C)=O)C(C)C2)=O)cc2n(n1)CCO2 Cn1cc(CC(=O)NCCCC2CCN(CCCC(=O)NC)C2)nn1.CO c1(C(=O)NCC2CN(C(c3ccsc3Cl)=O)CCO2)c[nH]c2nc(F)ccc12 N1(C(c2cncc(C)c2)=O)CCC(CNC(=O)C(C)OCCC(C)C)C(F)(F)C1 c1(C(C(=O)NC23CC(NC(CCC#C)=O)(C2)C3)O)cccc([N+](=O)[O-])c1 N1(C(Cc2c(C)ncc(Cl)c2)=O)CCN(C(c2cc(Cl)c(N)cc2F)=O)C(C)C1C c1(C(=O)NC2CC(NC(C3(CCOC)CC3)=O)C2)cc(Cl)cc([N+](=O)[O-])c1O N1(C(C(c2cccc(Cl)c2)CC)=O)CCC2(C1)CN(C(C1(O)COC1)=O)CCO2 C(CN=c1[nH]c(N(CC(C)OC(F)F)C)nc(=N)[nH]1)(c1ccccc1Cl)OC C1(NC(N(C)Cc2nc(C(C)OCC)sc2)=O)CCCC12CCC2 c1(CNC(Cc2nc(COC)nn2C)=O)ccc(C#N)cc1N n1(CC(=O)NC2C(OC)CN(C(CC=C)=O)C2)nc(C2CC2)n(C)c1=O C(=O)(C(C)C(C)NC(C1(CC(F)F)CC1)=O)NC N1(C(CC(C(C)C)O)=O)CC(CNC(=O)C=Cc2ncc[nH]2)C2(CCC2)C1 O=C(CCCCCCC(=O)c1ccccc1)NC1CC(NC(C2CCC(O)C2)=O)C1 N1(C(C(C2CCCC2)OC)=O)CCCC2(C1)CN(C(=O)C1=NC(=O)SC1C)C2 N12C(CCCNC(SC(F)F)=O)CCC1CCNC(=O)C2=O.C1(CO)CC1 c1(OCC)cc(N(C)C(=O)NCC2CCC(C)(C3CC3)O2)ccc1[N+](=O)[O-] c1(C(=O)NC2CC(N(C(Cc3cc(C(C)C)no3)=O)C)C2)cc2scc(Cl)c2[nH]1 CCCCC(C)C(=O)N1CCCC1(C(=O)NCc1ccccc1Cl)CC CC1CN(C(c2nc(O)nc(O)c2F)=O)CCCN1C(c1cc(O)n(C)n1)=O CC1(C)CC2(CC(C(=O)NC3COCCN(C(C4(CS(C)(=O)=O)CC4)=O)C3)C2)C1 c1(C(=O)NC(C)CC(C)NC(=O)CN2CCCC2)cc(Cl)c(N)cc1F c1(SCC)ccc(C(N2CCCCC2CNC(=O)CN(C)CCO)=O)cn1 Cn1ccc2ccc(CNC(N3CCn4cnnc4C3)=O)cc12 c1(NC2CN(Cc3ccc(F)c(CO)c3)CC2O)cccc(C(=O)OC)c1Br C1(C(=O)NC2CN(C(C3(O)CCCC3)=O)CC2F)CC2(C1)CC(O)C2 c1(OCC(N2CC(CNC(=O)CCF)OCCC2)=O)ccc2c(c1)CCCC2 C(=O)(CCCN(C)N=O)N(CCC)CCNC(c1cccn1C1CC1)=O c1(CC)ccc(OCCC(=O)N(C(C)CNC(=O)C=Cc2sccc2C)C)cc1 c1(C(N(CCC(=O)NC2CC(O)CC2O)CCO)=O)ccc([N+](=O)[O-])o1 c1(C(C)NCc2c(COC)cnn2C)ccc(OC)c(Br)c1 c1(C(=O)NC(C)CCCCNC(=O)CCCSC(C)(C)C)c[nH]c2nc(Cl)ccc12 Cc1ccc(C)c(C(N2CC(O)(CNC(c3ccnc(C(F)F)c3)=O)C2)=O)n1 N1(C(C2CC(SC)C2)=O)CCOC(CNC(c2c(CO)n[nH]c2C)=O)C1 c1(CC)nn(C)cc1C(=O)NC1CC12CC(NC(c1ccc(CO)cc1)=O)C2 C12(CNC(CN(C)S(N)(=O)=O)=O)CCC(CN(C(=O)CSCC(F)(F)F)C1)C2 c1(-c2cn(C3CCCN(C(=O)CN4CCC5CC45)CC3)nn2)ncc(Cl)cc1Cl C1(NC(COCCNC(C2(CC)CCNC2=O)=O)=O)CCCCCC1CO c1(C(=O)NCC2OCCN(c3ccnc(COC)n3)C2)cccc2ncc(C)n12 C(=O)(CCCCCS(N)(=O)=O)N(CC(CN(C(C(CCCC=C)(C)C)=O)C)O)C Cc1cc(F)c(-c2ccc(C=CC(=O)N3CCCO3)o2)cc1.C(C(=O)CC1CC1)=C N1(C(CC2(C)CC(F)(F)C2)=O)CC(NC(C2C3COCC23)=O)CC2(CC2)C1 N1(C(COC(C)=O)=O)CC(C)(C)C(NC(=O)C(c2ccc(Cl)cc2)=O)C(C)(C)C1 c1(C(=O)N(CCCO)CCCC2CCC2)cnc(-c2ccccc2)[nH]1 c1(C(N(CC(CC)NC(=O)Cc2cc(F)ccc2C)CC)=O)c(OC)ccnc1F c1(OC)ccc(NC(=O)NCc2cccc(F)c2C)c(C)c1Br CC(C(CO)NC(=O)Cn1nccn1)NC(=O)C(F)(F)C1CCOCC1 N1(C(CC(CNC(C(CCCC)F)=O)OC)=O)CC2CCC(O)C(O)C12 N1(C(c2cc(OCC)n[nH]2)=O)CCCCCC(NC(c2cccc(N)c2C)=O)C1 C1(CNC(C2CCS(=O)(=O)C2)=O)CC(F)CN1C(c1ccc(C(F)F)cc1)=O Cn1cc(C=CC(N2CCCCC2CCCNC(=O)CC2CCCOC2)=O)cn1 C1(C)(CNC(c2c(CCC)occ2)=O)CCCN(C(c2conc2C(C)C)=O)C1 C1(OC)CC(CC(N2CC(CCO)(NC(C3CCCS3)=O)C2)=O)C1(C)C Cc1cncc(C(=O)NC2CCCC2CC(N2CCOCC2C2CC2)=O)n1 C1(OC)COCCC1CC(=O)Nc1nc(C(F)(F)F)c(C)s1 c1(C(C)C)n[nH]c(=NCCCOc2ccc(C(=O)O)cc2)o1 C=C(C)CCCC(=O)N(C(C)(C(=O)NC1CCC(C)CCC1)C1CC1)C n1(CC)nc(C(=O)NC(CCOCCO)C(=O)N2CC(COC)C2(C)C)cc1O c1(C(C)OC)nc(CN(C)CC2CCN(C(c3cnco3)=O)C2)cs1 c1(NC(C23CC(NC(C4CC5C=CC4C5)=O)(C2)C3)=O)ccc2scnc2c1 c1(OC)c(C)cc(C(=O)NC2(C)CCN(C(C3(COC)C=CCC3)=O)C2)cc1C C1(N(C)C)(C(=O)NC(c2c[nH]cc2)=O)CCOC1.C12(CN)CC(C(F)(F)F)(C1)C2 C(C(F)(F)C(F)F)NC1(C(N2CC(CNC(CCSCC(C)C)=O)C2)=O)CC1 C1(NC(C(C=C)O)=O)CCN(C(=O)CCC(C)(C)OCC)CC1OC c1(N(C(C(=O)NC2CCCCC2)C2CC2C)CC)ccccc1C(=O)NC C1(NC(CSC)=O)CCOCC1C(=O)NCc1n[nH]c(C)n1 N1(C(CC=CCC)=O)CCOCC12CCN(C(=O)CCc1cnc[nH]1)C2 C1(C(=O)NCCS(CC)=O)CN(C(=O)CSC)CC12CCC2 c1(CC(=O)Nc2n(C(C)C)ncc2)c[nH]c2ccccc12 CC#CCCCC(=O)NC1C2CC1N(C(=O)Cc1ccc(F)c(F)c1)C2 C1(NC(c2cn(CCC)nc2)=O)CC12CCN(C(=O)CC1NC(=O)NC1=O)C2 C1(CNC(C2(F)C(C)C2)=O)CN(C(=O)CCc2ccc(F)nc2)CCC12CCC2 N1(c2n(CC(=C)C)c(C3(CO)CCOCC3)nn2)CCC2(CCOCC2)C1 C(=O)(C(CCCCC1CC1)N(C1(C)CCCCC1)CC)NCC(=C)C C1(CCC(C(=O)CCCc2cccs2)=O)C(=O)N(CC2CCNC2)N=C1C.CO c1(C(C)C)ccc(CNC(c2ccc(-n3ccnc3)nc2)=O)nn1 N(C1CCc2ccc(Br)cc21)C(C1CN(C(c2ccncn2)=O)CCS1)=O N1(C(c2cc(C(C)=O)on2)=O)CCC(C)C(CNC(=O)C(C)(C)c2ccns2)C1 c1(C(=O)NC(C(C)C)CCN(C)C(C2CC2C(F)F)=O)cnc2sccc2c1 c1(OC)cc2cc(C(=O)NC3(CCNC(=O)CCF)CCC3)[nH]c2cc1C(N)=O O=C(C1Cc2ccc(F)cc21)NCCCOCCNC(c1ncoc1C1CC1)=O N1(CC)CC2CN(C(C34CCC3CN(C(=O)C(n3nccc3C)C)C4)=O)CC2C1 N1(C(C(C)(F)F)=O)CCC2CCN(C(c3ccc(S(N)(=O)=O)cc3Cl)=O)CC2C1 Nc1c(F)ccc(F)c1C(N1CC2CCN(C(C3CCCCNC3=O)=O)C2C1)=O c1(C(=O)NC2C(NC(c3cc(SC)ncc3)=O)COC2)c(C)ncn(C)c1=O Cc1nc2cccc(C(=O)NC3CCCCC3NC(=O)C(C)NS(C)(=O)=O)c2s1 c1(C(CC(=O)N2CC(OCC(C)C)C2)NC(=O)OC(C)(C)C)cccc(F)c1 N1(C(=O)CCc2cc(Cl)cc(Cl)c2)CCC2(CCCN(C(C3CC3CF)=O)C2)C1 c1(CC)c(C(c2nnnn2C(C)CC)NCc2cccs2)cnn1C N1(C(CC2CC(=C)C2)=O)CCc2sccc2C1CNC(=O)Cc1ccoc1C C(=O)(C(O)P(C)(C)=O)NCCCC(C)NC(CCn1ncc(C)c1)=O C(CC(C)CC)(C(=O)N(C)Cc1ccnn1C)NC(C(C)=CCC)=O C1(C(=O)NCC(CC(C)C)NC(c2ccncc2Cl)=O)CCC2(CCOCC2)C1 c1(CNC(C(N2CC(C)C(N)C2)=O)=O)ccc2cnnn2c1 C1(C(N2CC(=C)C2)=O)C(CC=CC(C)(C)C)CCN1C(=O)C1=CCSC1 Cn1nccc1CN(C(=O)C(CC1CCCC1)NC(=O)C(F)C1CCC1)C Nc1c(C(=O)NCCNC(=O)CCC(F)F)cc(Cl)c(Br)c1F C1(CCNC(Cc2n(C)cnc2)=O)CCN(C(c2ccsc2)=O)CCC1(F)F N1(C(c2c(C)cccn2)=O)CC2CC1CN(C(=O)CC=CC(C)(C)C)C2 c1(CC(C(=O)NC2CN(C(C3(C4CC4)CCC3)=O)C2)O)cc(F)ccc1Cl c1(C(=O)NC2C(NC(c3cn(C)nc3)=O)CCCC2)c(Br)nc2n1CCC2 C(C(O)C(=O)NCCCC1(NC(C2CC(=C)C2)=O)CC1)=CCCCC CCC(CC(=O)N(C)Cc1ccnc(C)n1)NC(=O)CCCN(C)C(C)=O c1(CC(=O)NC2C(C(=O)NC3CC(=O)OC3)CCC2)ccc(O)cc1 C(CCCCNC(C1=CC=NC1C1CCC1)=O)N(C)C(C1(CO)CCC1)=O.C1CC1 C(=O)(C1CCCc2nccn21)NC1(C)CN(C(c2ccn(CC(F)(F)F)n2)=O)C1 Cc1nc2cccc(C(N3C(C)C4CC3C4NC(C3CCCCS3)=O)=O)c2[nH]1 c1ccc(C(F)(F)F)c(Cl)c1Cl.C1(CCC#C)CCCN1CO c1(OCC(=O)NCC2CC2CC(=O)Nc2sccc2Cl)ccccc1O CN1CCC2OCCN(C(c3c[nH]nc3-c3cccs3)=O)C2C1 C(C1c2ccccc2CCN1C(=O)CC1CCNC1=O)NC(c1n(C)cnc1)=O c1(C(=O)NCC(CC=C)NC(=O)C(C)Cc2ccco2)cnc2[nH]cncc1-2 c1(-n2c(C3C(c4cc(C)sc4)C3)nc(CCc3cnc[nH]3)n2)ccc(F)c(C)c1 c1(OC)cc(C(=O)NCC(O)CCNC(=O)CCC2CCC(=O)NC2)ccn1 c1(CCCN(C)C(c2nnc(C(F)F)s2)=O)nc2c(s1)CCC2 C1(C(=O)OC)CCN(C(C2C3CCC=CC23)C(=O)NCCSC)C12CCC2 c1(N(C(=O)C(C2CCN(C(=O)CSC(C)(C)C)C2)F)C)ccc2occc2c1 c1(C(=O)NCC2(NC(c3ccoc3)=O)CCC2)n[nH]c(C2CC2)c1Br C=CCCCCCC(=O)NC1CN(C(C2CCCCN2CCC)=O)CC1C N1(C(c2c(NC)cccc2)=O)CC2(CC(NC(=O)C(O)CC3CCCCC3)C2)C1 C1(C(=O)OC)CC(=O)N(C)C1C(=O)N(CC(C)NC(=O)Cc1cn(C)nc1C)C Cc1nc(CCNC(C2(F)CN(C(C3(CCF)CCC3)=O)C2)=O)cs1 CC1(C)COCC(C(=O)NC2COCCC2NC(=O)CCc2csc(=N)[nH]2)O1 C1(C(N(CCCCN(C)C)C)=O)CC2CCC1CC2NC(=O)OC(C)(C)C c1(NC(C=C(CC)CC)=O)ccc(C2CCCC(=O)N2)cc1 Cc1ncnc(C(=O)N(CCNC(=O)CCS(C)(=O)=O)Cc2ccccc2)c1C N1(C(c2cnn(CC)c2C)=O)CCCC(NC(c2ccnn2C(F)F)=O)C1C C1(SC)CC=NC1=O.C(CC(=O)OCCF)OC(C)=O C1(CC)CCN(C(=O)CCOCC2CCC2)C1C(=O)NCc1c(C)coc1C N(C1CCc2cc(F)c(F)c(F)c21)CC1CCCC(C)O1 c1(C(N2CCN(C(c3cc(CC)n(C)n3)=O)C(CO)C2)=O)c(C)cc(O)cc1O C1(C(N2CC=C(C)C2)=O)CC(C)(C)CCN1C(=O)CN1CSCC1=O C1(CC=C)(C(N)=O)CN(C(=O)C(C)COCC)C1.C12CC(F)(C1)CNC2=O C#Cc1ccc(CCCC(=O)NC2CCC(NC(=O)C(C)CC(F)F)C2)cc1 C(=O)(C1=CC2(CCOC2)C1)NC(C(C(=O)NC(c1ccnc(C)n1)C)(C)C)C c1(N2CC(OC)OCC2)cc(Br)ccc1S(=O)(=O)N1CCCC(CCF)C1 CC1CC(NC(=O)CCCCc2ccccc2)CN(C(c2ccc(F)cn2)=O)C1 N1(C(c2cc(COC)no2)=O)CC2CCCC2(CNC(C2(F)CC2(Cl)Cl)=O)C1 Cc1oc(C)c(S(=O)(=O)NC(CCCc2ccccc2)C(=O)OCCO)c1CO N(C1CCCc2ccccc21)C(CC1N(C(c2cnc(C)o2)=O)CCOC1)=O O=[N+]([O-])c1cc(F)c2c(c1)CN(Cc1snc3ccccc13)CC2 c1(NC(=O)CN2CCCCC2C(=O)NC2CNC(=O)C2)cccnc1C(F)(F)F c1(N(C(=O)CC2CCCO2)CCOCCCOC(C)C(=O)NC)ccc(F)cc1 C(=O)(C(O)CN1CCOCC1)NCC1N(C(C2C(C(=O)NCC#C)C2)=O)CC1 N1(C(C(C2(OC)CCOCC2)(F)F)=O)CC2(CCN2C(C23CCC(C2)C3)=O)C1 c1(OCC)ncc(CNC(=O)NC23CCC(OC(C)(C)C)(CC2)C3)cc1Cl N1(C(C(CC=C)C)=O)CCCN(C(=O)C2=CC(C)(C)C2)C(C)C1 n1(CC(=O)NCC(CC)(C)NC(=O)CN(C)C(N)=O)ccc([N+](=O)[O-])n1 C(c1c(Cl)cccc1Cl)=C(C(=O)NCCC(=C)CNC(=O)C(C)CC(F)F)C C1(NC(c2cccc(N)n2)=O)C2CC1CN(C(C1Cc3cscc3C1)=O)C2 c1(C(N2C(C(C)NC(c3nocc3Cl)=O)CCC2)=O)cc(C(F)(F)F)ncn1 C1(C(=O)NCC(C)NC(CCC(=C)Cl)=O)CCCN1NC(=O)OC(C)(C)C CCCCC(O)CC(=O)NCc1nocc1C(N1CCC(CCC)(CO)C1)=O CCC(CC)(C(C)C)NC(=O)Nc1ccc(F)c(C(C)=O)c1 Cc1cc[nH]c(=N)c1C(N1CCCC(NC(C2CC2C(F)(F)F)=O)C1)=O N1(C(C2(C#N)C(C)(C)C2)=O)CCC2CN(C(c3csc(Cl)c3)=O)C2C1 C1(C)(CCNC(C=C(C)C(F)F)=O)CCN(C(C2(c3ccc(F)cn3)CC2)=O)C1 C1(F)(C(=O)NC(CC)CN(C(=O)CN(C)C(=O)C2CC2)C)CCCN(C)C1 CCC(C#N)(CC)C(=O)NC(C)C(C)C(N1CCC2(CCC2)C1)=O C1(C(N(CCCCNC(c2coc(C3CC3)n2)=O)C)=O)CC2(CCOC2)C1 N1(C(C(c2ccccc2)OCC)=O)CC2(CCC2NC(c2cc(=O)cc[nH]2)=O)C1 C1(C(C)NC(C2CSCCS2)=O)CCN(CC=Cc2cccn2C)CC1 CCCCC(C(=O)NCC12CC(CN1C(C1COC(=O)N1C)=O)C2)C(C)C C1(OC)CC2(C1)CN(C(=O)C(CN(C)C)NC(=O)CC(C)(C)C)C2 C1(NC(C2(N(C)C)CCCCC2)=O)COCCN(C(c2cc(O)ncc2F)=O)C1 N1(C(C(C)NC(=O)C(F)OC(F)(F)F)=O)CC2COCC2(C)C1 c1(C(N2CCCC(F)(CNC(=O)Cc3ccsn3)C2)=O)oc2ccccc2c1Cl c1(CC)nn(C)c(OC)c1Cn1nc(-c2ccccc2)cc1C(=O)OC.C1CC1 N1(C(C2(OCC)CCN(C(=O)COCCF)C2)=O)CCC2CCCC12CO C1(C(=O)NCC(C(=O)NCC(C)C2CCC2)O)(CO)CCCCO1 c1(CC(=O)N(Cc2cn(CC(CC)O)nn2)CC)noc(C)c1C#N Cc1nc2ccccc2cc1NC(=O)NC12CC(F)C1C2 C12(NC(C3CCCCO3)=O)CCC(NS(=O)(=O)CCCCl)(CC1)C2 c1(SCC(=O)NCCCCNC(CC2(C)CC2F)=O)ccc2c(c1)CCC2 C1(C(=O)NC2(CN(C(C(n3ncc(C)c3)C)=O)C)CC2)CC1C1CCC1 C(=O)(C1CCc2cccc(=O)n21)N(CC(CNC(CCNC(=O)NC)=O)O)C C1(C(N(CCN(C(=O)Cc2cnnn2C)C)C)=O)CC2CC1C1CC21 CC(C)CC(CN=c1cc[nH]cc1C#N)NC(C1CCC(C(=O)N(C)C)CC1)=O C1(C(N2CCC(N(C(=O)C3=CCCCC3)CC3CC3)CC2)=O)CCC2CCCCN12 N1(Cc2cccc(OCC)c2)CCCCC(NC(C2CC2(C)C)=O)C1 C1(C(=O)NCC(C)CCO)CCCN(C(=O)CCN(C)CCO)CC1 C=C(C)C(C)(O)C(=O)N1CCN(C(c2[nH]c(O)nc2C)=O)C(CC(F)(F)F)C1 c1(C(c2nnnn2C2CCC2)N(C)C)c(I)cnn1C.CC1CS1 c1(CN2CC(NC(=O)C(F)(F)F)CC(C)C2)ccc([N+](=O)[O-])nc1.C1CC(=O)N1 C1(CC(=O)N(C(C)C(=O)NCCS(C)(=N)=O)CC)CCCC1C C=CC(CC)CC(=O)N1CCOC(Cc2cn(-c3c(F)cccc3Br)nn2)C1 C(C(C)(C)CNC(c1nc(Cl)cs1)=O)N(C(C12COCC1C2)=O)CC CCCC(CCCc1ccc(NC(=O)C(F)F)cc1)N=c1cc(C)nc(Cl)[nH]1 N1(C(CC(C=C)C)=O)CCN(C)CC1CNC(C12CC(F)(C1)C2)=O c1(CC(=O)NCCc2cc(O)cc(Br)c2)ccc2c(c1)OCO2 C1(N(C)C(c2nocc2Cl)=O)CCCCN(C(c2ccn(CC(F)(F)F)n2)=O)C1 c1(OC)ncc(F)cc1C(N1CCC(C)C(NC(=O)C(C2(O)CCCC2)F)C1)=O N1(CC(=O)NC2CC2CNC(=O)C(=C2CCCCC2)F)CCCNC1=O c1(C(=O)NCC(C)(C)NC(C(C)OCC)=O)cc(S(N)(=O)=O)oc1C N1(C(=O)CCN2CCC2)CCC2CCN(C(=O)CC3CC(F)C3)C2C1 CCCC(C)(CC)NC(c1c[nH]nc1CCNC(=O)Cn1cccn1)=O C(=O)(C(C)(F)C(=O)N1CC(CCO)(NC(=O)CCC=C(C)C)C1)OCC c1(C(=O)NC2CCCC(NC(CCC3CCN(C)C3)=O)C2)ccc([N+](=O)[O-])[nH]1 C1(O)(CN(C(c2cc(CCC)c(C)s2)=O)C)CCN(C(=O)C=CC(C)C)CC1 N1(CC)N=C(C(=O)N2CC(NC(=O)CCOc3ccc(F)c(Cl)c3)C2)CCC1=O CN1CC(O)CC1(C)C(N1CC2(CNC(C3CCC4CC34)=O)CC1CO2)=O C(c1ccc(Cl)cc1F)=CC(=O)NCC1CN(C(c2ccc(Cl)c(O)c2)=O)C1 C(=O)(C(CC1CCCC1)NC(=O)CCc1nnc(-c2ccco2)o1)OC(C)C C=C(F)C1(CC(=O)NCC2CCCN2C(C2(S(N)(=O)=O)CC2)=O)CCC1 c1(C(CC)C)nc(-c2cc(OC)nn2C)n(-c2ccccc2OC)n1 N1(C(CC(C)(C)SC)=O)CCN(C(=O)CC2CCC3CC23)C(CCO)C1 CC1=C(C(=O)N2CCCC(NC(c3cc4ccsc4s3)=O)C2)CCC1 Cc1cc(C(=O)NCCCCCNC(=O)CC2(n3ccnc3)CC2)co1 Cc1cncc(C(=O)NCCC2CCN(C(c3ccnc(O)c3)=O)C2)c1 N1(C(C2CC(CCNC(C(C)(C(C)C)OC)=O)C2)=O)CC2(COC(=O)C2)C1 N1(C(C2CC(OC)C2)=O)CCOC(C)(CNC(C2(Cl)CC2(C)C)=O)C1 CCCCCCC(=O)NC1CC1CNC(=O)C=Cc1cnccn1 c1(OC)ccc(C(C)C(=O)NC(CNC(=O)C=CBr)C2CCCC2)cc1OC N(C)(C(=NCCCOc1ccccc1C)NCCC(F)(F)F)CC(=O)NCCC.CC c1(C(=O)NCCCCNC(CN(C(COC)=O)C)=O)cn(C)nc1O.C(C)(=O)O C(N=c1ccnc[nH]1)C1C(NC(c2cnnn2-c2ccccc2)=O)CCC1 C1(NC(CC(=O)NCC)=O)C2CCC(C2)C1C(=O)N(CC(C)(O)C1CC1)C CC1CC(N(C(=O)C(O)C2CCCC2)C2CC2)CN(C(=O)Cc2ccns2)C1 C12(NC(C(CC)C)=O)CCC(NC(c3cscc3C(F)F)=O)(CC1)C2 N1(C(=O)NC(C(=C)C)c2nn[nH]n2)C2CCC1CN(C(=O)OC(C)(C)C)C2 CC(C)(O)CCCNC1(c2nnnn2CCCF)CCC(C(F)(F)F)C1 N1(C(=O)Cn2cncn2)CCCN(Cc2coc(-c3ccccc3)n2)CC1 N1(C(c2c(C)nsc2)=O)CCN(C(c2cncc(F)c2C)=O)CC1CC(F)F CC1CN(C(=O)CC2CC(N(C)C)C2)CC1CNC(=O)CCC1CCCC(O)C1 C1(c2ccccc2)(NC(=O)C(O)C2CCC2)CN(C(c2nc(C3CC3)cs2)=O)C1 c1(C(N2CCN(CCCC(N3CC(C)OC(C)C3)=O)CC2)=O)cn2ccccc2n1 Cc1cccc(C(=O)NCc2cccc(C(=O)NCCc3ncnn3C)n2)c1O N1(C(CS(CC)=O)=O)CCC(C)C(CNC(=O)C(C)(C)c2nccs2)C1 c1(C(n2nnnc2Nc2nc(Br)nn2C)C)ccc(S(C)(=O)=O)c(C)c1 C12(CC)CCC(C(N3CCCC(CNC(c4cnccc4C)=O)C3)=O)(CC1)CO2 c1(C(N2CC(C(C)C)N(C(C34CC(F)(C3)C4)=O)CC2)=O)cc(P(C)(C)=O)ccn1 c1(C(N2CC(C)N(C(C3CN4CCN3C(C)C4)=O)CC2)=O)ccnc2ccsc12 C1(N(C(CC)CNC(c2nocc2C(C)C)=O)C(C2CCCC2)=O)CCC(C)CC1 N1(CC)CC2CCCC(CN(C(CNC(=O)C(C3CC3)C3CC3)=O)C)C2C1 C1(CNC(c2cccc(CC)n2)=O)CCC2CN(C(=O)CCCSC)CC12 c1(COC2C(OC(=O)CSc3ccc(F)cc3)COC2)nc2ccccc2o1 N1(C(CC(=C)Br)=O)CCN(C(c2ccc(N)c(O)c2)=O)CCC1C C1(NC(CC(=O)NCCOC)=O)CC2(CCC(CNc3ccccc3C)CC2)C1 c1(C(=O)NCC=CCNC(C=CCCC)=O)cccc(OC)c1 c1(CNC(C(CNC(C2CCSC2C)=O)NC(=O)NCC)=O)cccnc1OC N1(C(C2CCC(C)CC2)=O)CC2(C1)CN(C(=O)C(F)C(F)(F)F)CC2CO C(=O)(CC(C(F)F)C(C)(C)C)NC(C(C)C)CNC(c1nsnc1O)=O C1(C(N2CCC2CNCCC(=O)OCC)=O)CCCN(c2cc(C)ncn2)C1 C(=O)(CC(C)(C)C(C)(F)F)NCC1C(C)CCN1C(c1ccc(Cl)cc1)=O C(=O)(C(C)C(O)C(C)CC)N1CCC(=C)CC1C(=O)NCC1CCOC(C)(C)C1 C1(C(N(CCOC)CCOC)=O)CC2(C1)CC(F)C2.C123CCC(C1C2)OC3=O c1(C(=O)NC2CN(C(C3C(=C)CC3)=O)CC2C)cc(Cl)c(O)cc1C CC1=C(C)CC(C(=O)N(C2C3CN(C(c4ccc(O)nc4C)=O)CC23)C)CC1 c1(C(=O)NC(C(=O)NCC2C(OCC)CC2)C2CC2)cnc(Cl)s1 Cc1cc(C)c(C(N2CC(NC(c3nccn4ccnc34)=O)C(O)C2)=O)c(S)n1 c1(C(N2CC(CC=C)(C(=O)OC)C2)=O)oc2ccccc2c1C C(=O)(C1=NOC2(CCOC2)C1)N1CCC(NC(=O)CCOc2ccc(F)cc2)C1 c1(N2CCCC(CC(C)C)C2)ccc(S(=O)(=O)NCC(c2ccco2)C)cc1Br Cc1ccc(C(N2CCN(C(c3c(C)cccc3C)=O)C3CC23)=O)cc1I c1(C(=O)NCC2CCCN(C(C(C)N(C(C)=O)C)=O)C2)ccnc(Cl)c1O Cc1cc(COCC(=O)NCC2(F)CN(C(c3cc(C(F)F)on3)=O)C2)no1 c1(-n2c(C(=O)OCC)ccn2)cccc(C(N2CCCC2c2ccc(Cl)s2)=O)c1 S(=O)(=O)(CC(=O)N1CCCC1CCCNC(C1CC(C)(C(=O)OC)C1)=O)NC C(C(C)(C)C(C)(F)F)(c1nnnn1C(C)(C)C)NCCc1ccnc(C)n1 c1(CC)nn(C)cc1C(=O)NCC1CC(NC(=O)CCn2nc(C)cc2C)C1 C1(CC)CN(Cc2csc(-c3ccoc3)n2)CCC1CO N1(C(C(CC)N(C(=O)CC(C)C2CCCC2)CC)=O)CC(C)C(O)C(C)C1 c1(C(CC)NCC(=C)C)cccc2ccncc12.c1(C)nnnn1CC1CCCO1 C1(CNC(c2ccc(CCC)s2)=O)CC2CCC1N2C(c1cc[nH]c1)=O O=C(C1=C(Cl)CCOC1)NCC1CCN(c2nnc(CO)s2)C12CC2 c1(NC2CN(C(N(CCOCCO)CC)=O)C2)ccccc1SC(F)(F)F C1(CC(=O)NCC=CCSC)CCCN(C(=O)CC2CCCNC2=O)CC1 C(=O)(CC(C(C)CC)NC(=O)C(C)(O)CC=C)N(CC=C)CC1CC1 C1(=O)CCCCCO1.c1(CC(=O)NCC(=O)OC(C)(C)C)nnc(O)o1 N1(C(c2c(CC)ccs2)=O)CC(NC(=O)C2=CCCSC2)CC1(C)C C1(COC)(CNC(C2CCSCC2)=O)CCN(C(C)=O)CC1 C1(NC(CCOCCOC)=O)COC2(CCCN(C(c3cc[nH]c(=N)c3)=O)C2)C1 O=Cc1cc(-c2cc(-c3cnn(CCC(F)(F)F)c3)[nH]n2)sc1Br C1(NC(CCc2c(C)ncs2)=O)CN(C(=O)CN2C(=O)CCC2=O)CCC1O N1(C(c2cc(CSC)c(C)s2)=O)CC2CCN(C(=O)C(C)c3ccco3)CC2C1 c1(C(N(CCCN(C)C)CC2CC2)=O)ccn2nccc2n1.C1(Cl)(C(=O)O)CC1(C)C c1(OC)ncccc1C(N1CCC1C(=O)NC(C)COc1ccccn1)=O c1(OCCC(=O)N(CCC(C)NC(CCC#C)=O)C)cc(C)ccc1Br N1(C(C(CC#C)O)=O)CC2CCCC(NC(c3ccc(=O)n(C)c3)=O)(C2)C1 C1(NC(CN(C(C)(C)CC)CC)=O)CN(C(c2c(C)cncc2F)=O)CCC1O C(=O)(C(C)(C)C1CCOC1)N(CC(=O)N(C1CC(CC)C1)C)CC O=[N+]([O-])c1cc(CNCc2c(Cl)ccc(F)c2F)ccc1N1CCCC1 C12(CNC(c3n(C)nc(O)c3)=O)CN(C(=O)COC(F)F)CC(F)(C1)C2 n1(CC=C)ccnc1C(=O)NC1CCC1NC(C1C=C(C)CS1)=O C(=O)(C(CCCCCC1CC1)N1CCOC(C)(C(=O)OC)C1)N.CCC(C)NCC C1(C(=O)NCC2CC=CCC2)CCCN(C(C2CCC(O)C2)=O)C1 C1(CNC(C2(CC)CN(C(=O)CSS(C)(=O)=O)C2)=O)CCCN(C(C)=O)C1 c1(CN2CCN(C(C3CC3c3ccc(Cl)cc3)=O)C3C2C3)ccc(Br)c(F)c1F c1(C(=O)NCC2CC(NC(C3N(CCC)CCC3)=O)C2)cnc(O)c(Br)c1 c1(CC(=O)C(C2CCC2)=O)occc1C.C(C(C)NC(=O)CN)OCC C(CN=c1[nH]c(=NCCc2cc(Br)cs2)c2ccc(C)cc2[nH]1)SC N1(C(C(C)N2CCC2)=O)CCOC2(CCC(NC(=O)C(C)n3cccc3)CC2)C1 C(CN=c1nc2sccc2c(NCC2CCCC2(F)F)[nH]1)(C1CCC1)OCC Cc1c(C(N2CCOC(CCNC(=O)C(C)C(F)F)C2)=O)ccc(Cl)c1Cl CC1(C)COC(C(=O)NC(c2ccc(F)cc2)(C)CNC(=O)CC2CCC2)C1 Cc1ccccc1NC(=O)C(N1CCC(Oc2ccc(Cl)cc2)C1)C c1(CC)csc(C(c2nnnn2C(C)CC)NCCNC(=O)N(C)C)n1 c1(C(N(CCNC(C2CCC(=O)O2)=O)CC)=O)ncc(F)cc1C C1(O)(C(=O)NCC2(NC(=O)C(=O)NC3CC3)CC(OC)C2)CCCCCC1 N1(C(C=CC(C)(C)N(c2cnns2)C)=O)C2CCC1CN(C(N)=O)C2 N1(C(C(CC=CCC)C)=O)CCCC(C2CN(C(C3CSCCS3)=O)C2)C1 C(=O)(C(C)(F)C(F)(F)F)N1CC(CNCCCCl)C(O)C1.O=C1CC2(CC2)CN1 Cc1ccc(C)c2[nH]c(C(N3CC(C)(NC(=O)Cc4ccc(O)cc4)C3)=O)cc12 C1(NC(C=Cc2cnc(C)s2)=O)CCN(C(=O)C(O)CC(N)=O)C(C)C1 N1(C(c2cc(OC)n(C)n2)=O)CC2CCC1C1CN(Cc3nonc3C)CC21 C(CC(C(=O)OC)NC(C1OCCC(NCC2(n3ccnn3)CC2)C1)=O)SC C12(C(N(CC#C)C)=O)CC(CN1C(c1cn(C)cn1)=O)C2 C1(C(C)=O)CC(C(N2CC=CC(NC(=O)CSC3CCCCO3)C2)=O)C1(C)C c1(CCC)ccc(C(=O)NCC2CC2CN(C(c2cnccc2Cl)=O)CC)cc1 c1(SC)cccc(CNC2CC(CC(=O)NC3(c4ccncc4)CCC3)C2)c1 c1(-c2cn(C(C3CCCN3C(=O)C(CCO)N(C)C)CC)nn2)c[nH]c(=N)c(C)c1 C1(n2cc(CCSCC)nn2)CCCN(C(=O)C(C)Cc2ccnn2C)CC1 N1(C(C2(C)CNC(=O)N2)=O)CCC2(CC1)CC2C(=O)NCCCn1cncn1 C1(COC)(NC(=O)Cc2cccc(NC(C)=O)c2)CCCN(C(=O)C(C)(C)C)C1 CCC(CCC(=O)Nc1ccc(O)cc1)NC(c1ncc(C)cn1)=O C(CN=[N+]=[N-])(C(=O)NCC1(C)CNC(=O)O1)NC(c1ncn(CC)n1)=O CCC(CC(C)C)C(=O)NC1CN(C(=O)C(c2cccn2C)=O)C1 C1(NC(C2CC(C(=O)OC)C2)=O)CCN(C(c2ccnc(C(F)F)c2)=O)C12CC2 Cc1cc(C(F)(F)F)ncc1C(N1CC(CC(C)NC(c2cccn2C)=O)C1)=O c1(OC(C(=O)NCC(CC)NC(=O)C(C)=C2CC2)CC)cccc(Cl)c1Cl C1(NC(=O)CC2CCN2C(c2n[nH]c(O)n2)=O)C(=O)OC2CCCC12 Cc1ncnc(C(N2CC(O)CC2CC(=O)N(C(C)CO)C)=O)c1C C(=O)(CC(O)C(C)(C)C)N1C(C(CNC(CCC)=O)(C)C)CCCC1 c1(CNC(C=CC2(C)COC2)=O)nnc2n1CCN(C(c1ccc(Cl)o1)=O)C2 c1(C(=O)NC(CCNC(c2cc(C)cc(O)c2)=O)(C)C)cc(Cl)c(F)c(Cl)c1 C(=O)(C#CC1CCCCO1)NCC12CC(NC(C(CC)C(C)C)=O)(C1)C2 Cc1cccc(C(=O)NCc2ncccc2CNC(C2CC2C2CCCO2)=O)n1 CCCCCC(C)CC(=O)N1CCN(C(C2CC(C)(F)C2)=O)C(C2CCCC2)C1 N1(C(C2(OCC)CCCCC2)=O)CCCC(CO)(NC(=O)C2CC2)C1.C(=O)(C(C)C)N C1(CNC(C(C)C2(O)CCC2)=O)COC(C)(C)CN1C(=O)CCN(S(C)(=O)=O)C c1(CCC(N2C(CNC(C(C)CC3CC3)=O)CC(F)C2)=O)ccccc1F C1(NC(CSCCOC)=O)CCC2(CCN(C(C3Cc4cccnc4C3)=O)C2)C1 c1(C(C)NC(c2ccc(OCc3ccccc3)cc2)C)nnc2n1CCOC2 Cc1cc(N2CC(C)C(C)C2)ncc1S(=O)(=O)N1CCC(c2ccn(C)n2)CC1 c1(C(C)C)nccc(N2CC(=C(F)CNC(=O)CC3CSCCS3)C2)n1 C(=O)(C(C(C)(C)C)n1ccnn1)N1CCC(OC)(CNC(C2CCS(=O)(=O)C2)=O)C1 N1(C(CNC(=O)NC)=O)CCN(C(=O)CN2CCCC2CO)C(c2nccn2C)C1 Nc1cnc(Cl)cc1C(=O)NCC(F)CNC(C1(F)CC1c1ccccc1)=O C(=O)(CC(C)(O)C(F)(F)F)NC1CCC(NC(C=Cc2n(CC)ccn2)=O)CC1 c1(N)nccn2ccnc12.C12CN(CCCO1)c1ccc(cn1)C(=O)NCC2.CO Cc1onc(C2CCCC2)c1C(=O)N(C1CN(C(=O)C#CC2CC2)C1)C Cc1cc(Cl)cc(N)c1C(=O)NCC(C)CNC(c1cnc(C(C)(C)C)nc1)=O c1(C(N2CCC(C(C(=O)NCC3(CC)CCCO3)C)C2)=O)c[nH]c2ccncc12 Cc1cc(C(=O)NCc2cc(C(=O)NCC3CCC(=O)N3)n(C)n2)ncc1N C(=O)(C1=CNC2=NCCCC2=C1)NC1CC(NC(C2C3(CC(C)(C)C3)C2)=O)C1 CCC(C)(C(=O)NCC1CC(F)CN1C(c1cc(CN(C)C)c[nH]1)=O)C(F)F C#CCCCC(=O)N1CCN(CCNC(C2CC2(C)C(F)F)=O)CC1 Cc1nn(C)cc1S(=O)(=O)N(C1CN(Cc2ccc(F)nc2)C1)C c1(C(=O)NC2(C)CC(NC(C3CN(CC(C)C)C(=O)C3)=O)C2)ccn2ccsc12 N1(C(CN(CC(C)C)C(C2CC(O)C2O)=O)=O)CC2OCC(CO)C2C1 Cc1c(C(F)(F)F)n[nH]c1C(=O)NC(C)C(C)(C)OC(F)F CC1CC(C(=O)NCC(O)CCC2CC2)N1C(=O)COc1ccsn1 C1(C(=O)NC2(CC(=O)NCC3C(C)OCCC3)CCC2)CN2CCC1CC2 C(=O)(C(O)CC(N)=O)NC(C(C)C)CCNC(=O)Cc1cnc(C2CC2)[nH]1 N1(C(CC2CC(=O)NC2=O)=O)CC2CC1CN2C(c1ccccc1)=O c1(CCOC)nc(=NCC(C)NC(=O)C(C)(C)CNC(C)=O)s[nH]1 CCCC(C)CC(=O)NCCCC(C)NC(=O)Cc1c(C)nn(CC)c1C C1(CCNC(=O)C2=CCOC2)CN(C(c2cnn(C3CCC3)c2)=O)CCS1(=O)=O c1(C(=O)NCC(CO)NC(C(c2n(C)cnc2)O)=O)scc2c1CCCC2 C1(CC(=O)NC(c2ccccc2Cl)COC)CCC2(CCC2)CO1 C=C(C)CCCC(=O)NC1(C)CCN(C(=O)C(C)N=[N+]=[N-])C1 c1(C(C(=O)NC(C2CCN(C(C)=O)C2)C)(C)C)cc(Cl)ccc1F C(=O)(CS(=O)(=O)CCOC)NC1CN(C(C2(CC=C)CC2)=O)C(C(=O)OC)(CC)C1 N1(C(CC=C)=O)CC(NC(c2cnc(C(F)F)nc2)=O)CC1C c1(NCCN(CC)Cc2ccc(OC)cc2)cncc(C(C)(C)C)c1 C(=O)(CCC(=O)c1cccnc1)NC(C)(CNC(=O)C=Cc1ncc[nH]1)CO c1(CC(C)C)ccccc1COC(=O)CSc1nnnn1C Cc1cnc(NC2CCCC2CF)c(S(=O)(=O)N2CCC3(CCCO3)CC2)c1 Cc1cnc(C(=O)Nc2cccc(NC(c3ccn(C)c3)=O)c2)nc1 N1(C(C(C)=CC)=O)CC(NC(=O)CC2CCCC(C)C2)C2(CCOCC2)C1 c1(CN(C2CC(=O)NC2=O)C(C2N(C(C)=O)CCOC2)=O)cnn(C)c1Br C1(C)(CNC(CCN2CCN(C)CC2)=O)CCCN(C(c2cc(C#N)c[nH]2)=O)C1 c1(SC(C)(C)C)cccc(NC(c2cccc(C(F)F)c2)=O)c1 c1(C(=O)NCC(CNC(=O)C=C(C)C)OC)cc(N)ccc1C c1(C(N(c2nccc(OC)n2)C(C2CCNCC2)C)=O)cnc2n1CCS2 C12(C(N(CCCCC=C)C)=O)CC(CO1)N(C(C1CCOCC1)=O)C2 C1(C(=O)NCCSC(C)C)(NC(=O)CC2CCSC2)CCN(C)C1 N1(C(c2c(C)ocn2)=O)CCC(C)(C)C1C(=O)NCC1CCCCC1(C)C CCC(C)C(C)C(=O)NC(c1ccccc1)CN(c1nc(Cl)ncc1C1CC1)C C(=O)(C(CO)C(C)(C)C)N1C(CCN(C(=O)CCc2ccccc2)C)CCCC1 c1(C(N(CC(=O)N(C)CCF)CC#C)=O)ccc(F)nc1 C12(CNC(=O)C(=O)NCC3CCCC(N)C3)CC(CN1Cc1ccccc1)C2 C(=O)(C(CC(C)C)OC)N1CCCCC1.C1(C(NOC(COC)CO)=O)CNC(=O)C1 c1(C(N(CC(C)NC(c2ccc(C)o2)=O)C)=O)cnc(P(C)(C)=O)cn1 C12CCCN(CC1)C(=O)CN(C)C2=O.O=C(COC(F)F)NC(=O)C1CC1 C=CC(CC)CC(=O)NC(C)CCCNC(c1ncccc1CC)=O c1(C(=O)NC(C2CC(F)(F)C2)C)n[nH]c2c1CN(C(c1c[nH]nc1C(F)F)=O)C2 N1(C(c2c(CC)nco2)=O)CC(OC)C(OC)C1CNC(c1cnn(C)c1N)=O C1(C(C)NC(c2ccsc2Cl)=O)CCN(C(=O)C(c2ccc(C)cc2)(F)F)CC1 CC(CCC(C)(C)C)C(=O)N(C)CCOCCCNC(=O)Cc1cnsc1 C(C1=NOC2COCC12)NC(c1c(CNC(c2cc(CC)ncn2)=O)con1)=O c1(-c2c3cc(C)oc3ccc2)csc(=Nc2cccc(F)n2)n1CC1SCCS1 c1(C(N2C(CN(C(CN(CC)CC)=O)C)COCC2)=O)csc2nccn12 C1(CNC(C2CCCO2)=O)CCCN1C(=O)CCc1cncnc1 C(=O)(CCCC(C)O)N(C(C)CNC(N)=O)C.C1(=O)CC(c2ccccc2)N1 N1(C(C(CC)C#N)=O)CCCC2(NC(C3CC4CC4C3)=O)CCCC12 c1(C(C)(C)C)ccc(C(N2CCCCC2CNC(=O)CNc2nccs2)=O)cc1 C12(C(=O)NC3C(NC(=O)COC(F)(F)F)COC3)CCC(=O)N1CCS2 C1(C(=O)NCCN(CCC)CC)(CNC(=O)Cc2cc(C)cs2)CCCO1 C(=O)(C1=CCS(=O)(=O)C1)N1CC(NC(=O)CSCc2ccc(Cl)cc2)C1 C#CCC(C)(C(=O)N(C1CC2(CC2)C1)C)NC(C1CC1Cl)=O c1(OCC(CNC(=O)NC2CC(CCOC)C2)O)ccc(Cl)cc1F Cc1ncsc1COCC(=O)NCCCCCN(C)C(c1n[nH]cc1Br)=O C1(C)(C(=O)NCCOCCC=C)CCN(C(=O)CC2CCOC2)C1 CC1=CCC(C(=O)NCC2CCN(C(=O)C(C)(C)c3cccs3)CC2)CC1 C(=O)(C1COc2ccc(Cl)cc21)NC1C2OCC(NC(CCC=C)=O)C2OC1 Cc1cc(N2CCCC(OCC(N)=O)C2)nc(NC(c2cc(F)ccc2Cl)C)n1 c1(OC)cc(C)c(C(N2CCC(CF)(NC(=O)CN=S(C)(C)=O)C2)=O)cn1 CCS(=O)(=O)C=CC(=O)N(C)CC1CCCN(C(c2cscc2C(F)F)=O)C1 N1(C(Cc2nc(CC)sc2)=O)CCC(C2CN(C(=O)C(F)n3cccn3)C2)CC1 C(=O)(C1=CCCCCC1)N1C(CCNC(=O)Cn2nc(O)ccc2=O)CCCC1 C1(NC(C(CC)N(C(c2ccnn2C)C(=O)NC)CC)=O)CC(CO)C2CC12 CC(c1cccnc1)=CC(N1CCCC(C(C)NC(c2ccc(F)cn2)=O)C1)=O N1(C(C(C)C)=O)CC2CCCC(CNC(c3ccc4oncc4c3)=O)C2C1 C(=O)(CCCCN=[N+]=[N-])N1CCC(C(C(N2CC(CC(=O)OCC)C2)=O)C)CC1 C(=O)(C(F)CC(C)(C)C)N1CCSCC(C)C1.C1CSCN1 C12(C(C)C)COC(C(=O)NCC3CCCCC3CNC(=O)Cc3cc[nH]n3)(C1)C2 c1(C(N2CC(NC(c3c(C)coc3)=O)C3C2C3)=O)cc(Cl)ccc1C(C)C C=CC(C)(O)CC(=O)NC(C)(CNC(=O)C(C)NC(=O)CC(C)(C)C)C1CC1 C1(F)(CNC(=O)CCc2ccoc2)CCN(C(=O)C(F)C2CC2)CC1 c1(C(=O)NCC2C3CN(C(C4(C)CC4(F)F)=O)CC32)[nH]nc2ncnc(O)c12 C(CNC(=O)Cc1nocc1C)(CC(=O)N(C)Cc1csc(C)n1)OC CC1C(C(=O)N2CCC(N(C(=O)CC3OCCC3C)CC3CC3)C2)=NOC1C N1(C(C=Cc2ncn(C)c2)=O)CC2(CCN(C(=O)Nc3ccc(Cl)cc3F)CC2)C1 N1(C(C=C(C)I)=O)CC2CCN(C(=O)CCc3ccccc3)C2C1 Cc1sc(=NC2CCOC3(CCNCC3)C2)[nH]c1I N1(C(C(CC#C)C2CC2)=O)CCN(C(c2cc3occc3[nH]2)=O)CC1C1CCC1 c1(C(=O)NCC(CC=C)NC(=O)C(C)CN2CCOCC2)ncnc2c1cnn2C Cc1cn2c(n1)C(C)CC(C(N1CC(NC(=O)C(C)(C)F)C1)=O)C2 c1(CNC(CC)(COC)c2nnnn2C(C)(C)C)ccc(-c2ccsc2)nc1C C1(OC)CC(CNC(c2occc2C)=O)N(C(=O)CC2(C)CCOCC2)C1 Cc1cc(C(=O)NCC2(O)CCN(C(=O)C=Cc3cn(C)cn3)C2)c(C)s1 c1(C(=O)NC2CCN(C(CCCOCC=C)=O)CC2F)nnc2n1CCCC2 C1(C(=O)NCC2(C(N)=O)CN(C(c3ccc(OCC)s3)=O)C2)COCC(C)(C)O1 c1(C(=O)NC2C(NC(CC=CC=C)=O)C2)cc(N2CCNC2=O)ccc1F Cc1noc(CCCC(=O)NCC(F)CNC(=O)C(c2csc(=N)[nH]2)=O)n1 c1(C2(C(=O)OC)CCC2)cccc(NC2CC2c2ccc(Br)s2)c1 C(=O)(CS(=O)(=O)CC(F)(F)F)N1CCC(CSCC)(NC(C2(Br)CC2)=O)CC1 Cc1nc2[nH]c(C(N3CC(CN=c4cc(C#N)nc[nH]4)C(C)C3CO)=O)cc2s1 N1(C(C2C(C)(C)C2)=O)CC(CNC(=O)CNc2ccccc2CC#N)CC1(C)C CCCC(C(=O)N1CCN(C(c2c[nH]c(C#N)c2C)=O)CC1CC(F)F)C(C)C Cc1sc(-c2nnc(CN3CCN(C(=O)C(C)(C)c4cnn(C)c4)CC3)s2)cc1Br C(=O)(C(=O)C(C)C)N(CC(=O)NC1(CC=C)CC1)C CC1CN(C(c2nc(Cl)cs2)=O)CC1NC(C1(c2cccnc2)CCC1)=O C(=O)(CCS(C)(=O)=O)N1CCC(CC)C1CNC(c1csc(=N)[nH]1)=O N1(C(CCCCC=C)=O)CCC2(CCCN(C(=O)CC3CCCN3C(C)=O)C2)C1 C1(CC)CCCN(CC(=O)NC2(CN(C)C(C3C(Cl)(Cl)C34CC4)=O)CC2)C1 N1(C(C(=O)N(CCCC(C)(F)F)c2ccccc2F)=O)CCC(O)(C(Cl)(Cl)Cl)CC1 S(=O)(=O)(c1ccc(NCCC#N)c(F)c1)NC1CC(C)(C(C)(C)C)C1 CCC1=C(C(=O)N2CCC3(CC3NC(c3cccc4sccc34)=O)C2)CCCO1 c1(CCC(=O)NCC2C(NC(C(C)SCC)=O)C2)ccc(Cl)cc1Br C1(NC(c2ccc(CCC)s2)=O)CCCN(C(c2cccc(N)c2F)=O)C1C C1(F)(C(=O)NCC(C2CCN(C(c3ncsc3C(C)C)=O)CC2)F)CCCCCC1 c1(C(N2CCN(C(CCNC(=O)NC)=O)CC2CF)=O)nn(C)c2ccccc12 N1(CC(=O)N(C2CCN(C(c3scc(C(N)=O)c3)=O)C2)CCO)C(=O)CN(C)C1=O Cc1oncc1S(=O)(=O)N1CC(N)C1.N1(C(C)=O)CCC(n2cnnc2)CC1 C12(C(=O)NS(CC)(=O)=O)C3C4C1C1C2C3C41C(N)=O.c12ccc(cc1)SC2 c1(OC)cc(O)c(C(=O)NC(C2(O)CCN(C(=O)C3CC3)C2)C)cc1Br c1(C(N2CC(NC(=O)C=CC3CCOCC3)CC(C)C2)=O)cnn2ccccc12 c1(C(N(CCOC)CCNC(=O)Cc2csc(C)c2)=O)ccc(Br)cn1 c1(C(N(CCNC(c2ccc(C(C)=O)nn2)=O)C2CC2)=O)ccc2cc[nH]c2n1 c1(C(=O)NCC2C(NC(CC3C(C)(C)C3)=O)C2)ccc(=N)[nH]c1 CCCC(CCCNC(c1cnc[nH]c1=N)=O)NC(=O)C(c1cncn1C)O c1(CCC)n[nH]cc1C(=O)NCCNC(c1coc(C2CCCC2)n1)=O C1(S(C)(=O)=O)(C(=O)NCC(CN(C)C(C2OCCO2)=O)O)CCCC1 N1(C(Cc2cnc(C)s2)=O)CCC(F)(C(=O)NCC2(O)CCCOC2)C1 C(=O)(CC(O)C(C)C)N(C1CCCCC1)CCNC(c1c(C#C)c[nH]n1)=O c1(C(NNC(CNc2cccc(-c3n(C)cnn3)n2)=O)=O)ccc2c(c1)OCO2 Cc1ccc2sc(C(=O)NCC3CN(C(=O)CN4CCCC4)C3)cc2c1 c1(C(N2C(C)CN(C(C3CC3C)=O)CC2)=O)cc2cccc(Br)c2[nH]1 C1(N(C(=O)CN(CCO)CCO)C)CCC(NC(c2cn(C(F)F)cn2)=O)CC1 C(C)(CC(F)(F)F)N(C(C(CC)NC(C1(OC)CCCCC1)=O)=O)C C1(C)(NC(c2n(CC)ccn2)=O)CCCN(C(c2ccc(OC)c(O)c2)=O)C1 C1(CNC(C2C(OCC)CC2)=O)CC2CC2N1C(c1ccnn1C1CCC1)=O C=C(C)CC(C)C(=O)N1CCC(CNC(c2cscc2C(F)(F)F)=O)C1 Cc1nc([N+](=O)[O-])cn1CCC(=O)NCC1CC1NC(C1C2CCCCCC12)=O C1(CNC(C(C)S(C)(=O)=O)=O)CC12CCN(C(C1(Cl)CC1)=O)CC2 C1(NC(C(C2CC2)SC)=O)CCC(NC(=O)CCC(F)F)CC1 C(=O)(CC(O)CCSC)NCC(C)(C)NC(c1ccc(CNC(CC)=O)cc1)=O C1(C(=O)NC(c2ccc(C(=O)OC)cn2)C)OCC2CC(=O)C1C2 c1(C(=O)NCC2N(C(CC3CC(=C)C3)=O)CC=C2)ccc(C(C)(F)F)nc1C c1(C(=O)OC(CC(=O)OC)C)cccnc1C(F)(F)F CCC(N=c1[nH]c(=NCC2CC23CC3)c2ccccc2[nH]1)c1cccc(C)c1 c1(NC(C)=O)cc(Br)ccc1C(=O)NCC1CCCO1.c12cccnc1C(=O)N2 C(=O)(C1=NN2CCCN=C2N1)N1CCC(C)(NC(C2CCCN(C(C)=O)C2)=O)C1 c1(C(=O)NC2(CC)CCCN(C(=O)CCC3CCCO3)C2)cc2cn[nH]c2cn1 C1(N(C(c2c(CC)cc[nH]2)=O)CCO)CCCN(C(c2cncc(O)c2)=O)C1 c1(C(N2CC(C)(NC(c3c(C(C)(C)C)ncs3)=O)C2)=O)cc(F)cc2nc[nH]c12 c1(C(=O)NC2CN(C(CC(=C)C)=O)CC2C)cn2c(n1)CCC2 N(C1CCc2ccc(Cl)cc21)C(CCc1cn(CCCCCC(=O)OCC)nn1)=O N1(C(c2cc(C)n(C)n2)=O)CC(NC(c2cccc(Cl)c2N)=O)CC(O)C1 c1(CC)onc(C)c1C(N1CC(N(C(c2sccc2Cl)=O)CC)C1)=O C12(CNC(c3c(Cl)cccc3Cl)=O)CCC(CC1)CN2C(=O)Cc1cnccn1 CC1=NOC2(C1)CC(C(=O)NCCCC(C)NC(C1CCC(=O)O1)=O)C2 C(=O)(C(O)CC(F)F)NCC(C)(CO)NC(=O)COc1ccc(Cl)cc1 C1(O)(Cn2cc(CS)nn2)CCCN(CC)CC1.C1(C=O)CN(C)C(=O)CCO1 c1(CCC(N2CCC(NC(C3CC4CC4C3)=O)C2)=O)cc(F)c(Cl)cc1Cl C1(C(N(C2C(C)CCC2)C)=O)CC(O)CN1C(C1CC(F)C1)=O N1(C(CCC(C2CCC(C)CC2)=O)=O)CCCC12CCN(C(=O)C(Cl)=CCl)C2 C1(C(N(CCN(C(=O)C(=O)NCC(F)(F)F)C)C)=O)CN2CCC1(C)C2 c1(C(=O)NCCC(C)N(C)C(C2CCC(OC(F)F)CC2)=O)cnc2sccn12 C1(C(=O)NC(c2ccc(C)cc2)CNC(=O)CNC(C)C)CCOCC12CCC2 N1(C(c2cc(C)[nH]n2)=O)CCCC12CCN(C(C1(F)CCCCC1(F)F)=O)CC2 C=CC(CCC)CC(=O)NC1(C(N2CC(O)(CCC)C2)=O)CC1(C)C C1(C(C)NC(C2(O)CCSC2)=O)CCN(C(=O)CC2(C)CC2(F)Cl)C1 c1(OC)ccc(Cl)cc1CC(C)(C)NC(=O)NCCC(OC)OC N1(C(c2c(C)csc2)=O)CCCN(C(C2CCCC(=O)N2)=O)CCC1 C12(CC)CC1CN(Cc1cc(O)n(C(C)C)n1)C2 C(=O)(C(=O)C(C)(C)C)NC1(C(=O)NC(c2cnccn2)C)CC(F)C1 c1(OC)cccc2cc(C(c3nnnn3CC3CC3)NCC(C)S(C)(=O)=O)oc12 N1(C(C2N(CC)CCC2)=O)CC(F)(F)CC1C(=O)N(C1CCCN1)CCO C(=O)(C1=CCCOC1)N1CC2C(CNC(c3cnn(CC(F)F)n3)=O)(C2)C1 c1(CC(=O)NC2CCCC(N(C(=O)CC3CC3)C)C2)cccc(C#N)c1 C(C)(CC(=O)NCCN1CCNC1=O)NC(CSCCC(C)C)=O c1(NC(C2CC3CC3N2C(c2ccc(O)nc2)=O)=O)cccc([N+](=O)[O-])c1Br C1(CC(=O)NCC(CC=C)NC(c2ccc(Cl)cc2N)=O)COCC(C)(C)O1 c1(C(=O)NC(C2CCC(CCNC3(CC)CC3)C2)=O)cccn2c(C)cnc12 c1(C(=O)NC2C(CNC(CCCOC(C)C)=O)CC2)cn2c(n1)SCC2 Cc1ccc(O)cc1C(N1CCC(C(C)C(=O)N(CCS(N)(=O)=O)C)CC1)=O c1(C(=O)NC(C2CCN(C(CC3C(C)OCC3)=O)C2)C)cnn(C)c1C(F)F Cn1nc(C(N)=O)cc1NC(c1ncccn1)=O.C12CCC(CC1)C(=O)NC2 c1(C2CN(C(C3CCN(C4CC4)C3=O)=O)CC2O)cc(F)cc(F)c1 C1(NC(CC(C=C)C)=O)CCC2(CCN(C(=O)Cc3ccno3)C2)C1 C1(C(=O)NCC2C(NC(c3n[nH]c(C4CC4)n3)=O)CCCC2)CC12CCSCC2 N1(CC)CCC2(CC1)OCCC2NC(c1ccc(Cl)cc1)=O c1(C(N(C)CCOCCN(C)C(C2CCCN2C)=O)=O)cc(C(F)(F)F)ncn1 C1(CC(=O)NC(=O)Oc2cc(O)ncc2F)Cc2ccc(Br)cc2C1 N1(C(c2c(C)ccs2)=O)CCN(C(=O)Cc2ccc3c(c2)OCO3)CC(CO)C1 c1(-c2nc(Cc3onc(CCCC(=C)Cl)n3)c(C)o2)ccc([N+](=O)[O-])cc1F Cc1c(C(=O)N(C2CC(CC(N3CCN(C4CC4)C(=O)C3)=O)C2)CC)cncc1Cl C12(C(=O)NCC(c3cccnc3)C)CC1CN(C(=O)C(C)Cn1cccn1)C2 C1(CCC(=O)N(CC(C)O)CCF)CCCN(C(c2cc(C(F)F)[nH]n2)=O)C1 C(CN=c1[nH]c(Cc2n[nH]cc2[N+](=O)[O-])nc(=N)[nH]1)NC(C1CCN(C)CC1)=O N1(C(C2C3(CC(N(C(c4c(CC)[nH]cc4)=O)CC)C3)C2)=O)CC(F)(F)CC1C CCCCCCC(C)C(=O)NCC(C)(CO)NC(=O)CC(C)CC(=O)OC c1(C(=O)NC(CC)CNC(=O)C(CC)N(C)CC)ccc2ncccc2c1F Cc1cccnc1CCCC(=O)NC1CCCN(C(=O)Cc2cc(Cl)cs2)C1 C1(N2CCC(C(=O)Nc3c(C)cccn3)CC2)CCS(=O)(=O)C12CCC2 CCC(CC)CCC(=O)NCC(CC1CCCC1)C(=O)NCCC1CCN(C)C1 C1(COc2c(C(=O)NCCCC)nccc2)CCN(Cc2ccccc2)CC1(F)F c1(SC)nc2ncnc(N3CCCC(NC(=O)C(C)CSC(F)(F)F)C3)c2s1 C1(C(N(CC(C)NC(c2c(SC)cnn2C)=O)CC)=O)CC2(C1)CC1(CCC1)C2 C(=O)(CC(C)(C(F)F)n1cc(C2(O)CC2)nn1)NC(C(C)C)Cc1nccn1C C1(CNC(c2ccc(CC)cc2)=O)CCN(C(=O)CCCc2ncco2)CC1C c1(C(=O)NCC2(OC)CN(C(COCCC)=O)C2)ccc(OC)c(Br)n1 c1(OC)cccc(CNCC(C2(O)CCC2)O)c1OC(C)=O c1(C(N2C(CCCNC(C(C)(C)CO)=O)CCC2)=O)cccc(O)c1[N+](=O)[O-] C1(C2CCNCC2)(c2onc(C(CCCC(C)C)C)n2)CCOCC1 C12(C(=O)NC(C(C)SC)C)CCC(CC1NC(=O)CC1(C)CC1)C2 N1(C(c2cnc(OCC)s2)=O)CC2CC3CC2C1C3NC(C1CC(F)(F)C1)=O c1(OC)ccc2c(c1)CCCC2C(=O)N1C2CCC1C(CNC(=O)C(C)(C)C)C2 c1(C(N2CCCC(N(C(C3C(C=C)C3)=O)CC)C2)=O)cc(O)nc(O)c1 c1(NC(c2n(CCC)nnn2)c2cc(-c3ccco3)on2)nc(C#N)c(C#N)[nH]1 N1(C(C2(C#C)CCCC2)=O)CCN(C(N(C)CCOCCC(=O)NC)=O)C(=O)C1 N1(C(C2C(CC)C2C)=O)CCNCC1c1ncc[nH]1 C1(C(=O)NC)C2CC(F)C(C2)N1CCC1CNCCO1 C1(COC)CCCCN1C(=O)CC1CN(C(c2ccc(CC(F)(F)F)cc2)=O)C1 CC1=CC(C)CN(C(=O)C(c2ccco2)NC(c2coc(C(C)C)n2)=O)C1 N1(C(c2n(C)nnc2)=O)CCCC(F)(C(N2CCCC3CC23)=O)C1 CCC(CC(=O)NCCN(C(=O)CC(C)COC)Cc1ccccc1)C(C)C CCC(CC)C(C)C(=O)NCC1CC2CCC1N(C(=O)C(C)(C)CO)C2 c1(C(=O)NCCC(C)NC(C2(CCC)CC2)=O)ccn2c1CCC2.N1CCCC1 CCCCC(C(=O)NCC=CC(=O)NCC1CCCC1O)N(C)C N1(C(CC2CCN(C(c3cc(C(C)=O)[nH]n3)=O)C2)=O)CCC2CC12C Cc1cc(C(=O)Nc2cccc(N(C)C)c2)c(C)n1-c1ccccc1OC(F)F C1(C(=O)NCC(CCC)=NO)CNC(=O)CN1C(=O)C(=O)NCCC(N)=O c1(C(N(CC(C)N(C(=O)C=CI)C)C)=O)ccsc1C(F)F CC(C)C(C(c1ccccc1)NC(c1cccs1)=O)NC(=O)C=Cc1ccsc1 C(=O)(C(C)(C)CC(C)C)NC(CNC(c1c(C)ccnc1C)=O)CC(C)C C1(CC(=O)NCC(CCCC)NC(c2n[nH]c3c2CCC3)=O)CCC2(CC1)CC2 c1(CNC(C(C2CCC2)NC(CCOCCOC)=O)=O)ccc(Cl)cn1 C1(NC(CCCCC)=O)CC2CC1CN2C(c1cn(C)nc1-c1ccncc1)=O c1(C(=O)NCC=CCNC(C2CC(CC)C2)=O)ccc2nc(C)cn2c1 C1(C(=O)NCc2c(C)n(C)nc2)CC2CCC(C1)N2C(C1CCCC(=O)N1C)=O C1(C(N(C2CCOC2=O)C)=O)CCC(=O)N1.C12C(C1(C)C)C(=O)NC2 C#CCCC(C(=O)N1CCCC(C)(N(C)C)C1)NC(=O)CCc1ccnn1C O=C(COC(=O)C#CCc1ccccc1)N=c1cco[nH]1 c1(C(=O)NC(C)C(C)(C)NC(=O)CC2SC(=N)NC2=O)[nH]nc2ncccc12 c1(C(=O)NC(CN(C(=O)C=CCCC(F)(F)F)CC)C)ccc(N)cc1Cl C(C(CC(C)C)NC(C1CC=CCC1C)=O)NC(C(CC1CC1)OC)=O C1(C(=O)NC2(C(N(CC=C)CC3CC3)=O)CCSC2)C(C#N)C1(C)C c1(C(=O)NCC(CCOC)NC(C2(F)C(C)(C)C2(C)C)=O)ncc(N)nc1C c1(NC(N2CC3=CC(=O)C(NC(C4CC4F)=O)(C2)C3)=O)ccc2ccccc2n1 N1(C(C(C)Oc2cccnc2)=O)CCC(NC(=O)Cc2ccon2)C1(C)C C1(NC(C2(C)CCC2)=O)CCOC2(CCN(S(=O)(=O)c3cccs3)CC2)C1 c1(C(N2C(CNC(C3(C)CCCC3)=O)C3CC3C2)=O)ccc2c(n1)NCC(=O)N2 CC1CCC(C(=O)NC(C2CN(C(=O)COC3CCOCC3)C2)C)C1 CC(C(C)(C)C)=CC(=O)NCC1OCCC1C(=O)N(CCCCN(C)C)C C(=O)(C(F)C(F)(F)C(F)(F)F)NCC1N(C(C(Br)=C(C)C)=O)CC=C1 C(=O)(C(C)(F)CC1CCCC1)NCCC(CNC(C(c1cccnc1)C)=O)O C#Cc1cnc(C(=O)NC2CC(C(N3CCS(=O)C(C)C3)=O)CC2O)c(C)c1 c1(OC)cc(C(F)(F)C(=O)NCCNC(c2cc(N)ccn2)=O)ccc1Br n1(CC(C(=O)NCC(C)(C)NC(CC(COC)C)=O)(C)O)ccc(C)cc1=O c1(C(N2CC(O)(CNC(c3c(C)c(O)ccc3)=O)C2)=O)nc2cccnc2s1 C1(NC(c2c(C)con2)=O)CCN(C(C2CC(=C3CC3)C2)=O)CC1O N1(C(CSCCC)=O)CC2(CNC(C3CCCN3N=O)=O)CCC1CC2 N1(C(C(CC)CCOC)=O)CCC2CN(C(c3cccc4c[nH]nc34)=O)CC12 C(=O)(C1=CCC2(CCOC2)OC1)NC(C(C)C)CNC(=O)C(C)(C)C1CCCC1 C12(C(=O)NCCNC(CCc3cc(C)n(C)n3)=O)CCCCC1C2(F)F Cc1noc(CCC(=O)N(CC(=O)NCCF)C)n1 c1(SC)cccc(C(=O)NC(C)CN(C)C(C2CC(=O)N(CCF)C2)=O)n1 CS(=O)(=O)CCCCNC(=O)C(=O)NCc1ccn(-c2ccc(F)c(F)c2)n1 c1(CC(=O)N(C(C)CNC(=O)CS(=O)CC)CC)ccc(C)cc1Cl C=CC1(CC(=O)NC(C)C(C)C(=O)OC)CCN(C(=O)CC2(CSC)CC2)C1 c1(C(N(C(C)CN(C(=O)CC(C)c2ccncc2)C)C)=O)cc(O)nn1C c1(C(N2CCOC(C3CCOCC3)C2)=O)cccc2ccsc12 N1(C(=O)Cc2cc[nH]n2)CCC2(CCCN2C(=O)CCCc2nccs2)C1 C(CO)(C(C)N=c1ccc(Br)c(S(=O)(=O)NCC=Cc2cccnc2)[nH]1)SC c1(-n2c(CC3C(CC)C3)nc(-c3ccc(C)c(Cl)c3)n2)cncc2ccccc12 C(=O)(C(F)CCC(C)(C)C)N1CC(F)CC(NC(C2CCCC(C)CC2)=O)C1 N1(C(C2(CC)CCN(C(c3c[nH]c4ccccc34)=O)C2)=O)CCCC(O)(C2CC2)C1 C1(NC(C2C(COC)CC2)=O)CCN(C(c2cccc(C)c2C)=O)CC1O N1(C(C=CC=CCC)=O)CCC(C(=O)NC2CC2C(C)(C)C)C1C C=CC(C)(C)CC(=O)NC(C(C)NC(=O)C=C(C)C1CC1)C(C)C C(=O)(C1=CC2CC(C1)CC2O)NCc1nc(CNC(CC2(OC)CCC2)=O)sc1 N1(C(C23C(C(=O)OC)(CCC2)C3)=O)CC2(CCN(C(C3CC4CC3CO4)=O)C2)C1 Cc1csc2cc(C(=O)NCC3CC(NC(=O)C(C)CN(C)C)C3)[nH]c12 c1(NC(CNC(C(=O)NCC(C)(C)OCC(F)F)=O)=O)cnn(CC(F)(F)F)n1 Cc1c(C(N2CC(C(N)=O)(CNC(C3(C)COCCO3)=O)C2)=O)sc2ccccc12 C1(CC#C)CCN(CCC2CC3COCC23)CC1 C1(OCCNC(C(C)SC(C)C)=O)CCN(C(=O)CNC(C2CCCC2)=O)C1 C(=O)(CC1=NN(C)C(=O)C1)NCCNC(c1c(Br)ccc(C)c1)=O N1(C(CC#N)=O)CC(F)CC1CNC(C1CCC(=O)NC1)=O c1(C(=O)NCc2cn(C3CN(C(c4cscn4)=O)C3)nn2)cccc(O)c1 c1(CC(=O)N(CCC(=O)NCCC23CCC(CC2)C3)C2CC2)cccc(F)c1 Cc1c(NCC2CCN(c3nccs3)CC2)ncnc1Nc1ncc(F)cc1F C1(NC(CCC2CCN(C)C2)=O)CCN(C(c2ncccc2CO)=O)CC1(C)C C=C(C)CCCC(=O)N1CC(C2CN(C(=O)C(C3CCOCC3)C)CCO2)C1 N1(C(CC2CCCN(C)C2)=O)CCC2(NC(C3CC4CCCC34)=O)CCCC12 C12(NC(CSCC#C)=O)CCCC(NC(c3cc(C)c(C)cn3)=O)(C1)C2 Cc1cscc1C(=O)NC1CCC1C(N1CCC(C(N)=O)C1)=O N1(C(CN(C(C=C)C(F)(F)F)C(COCC#C)=O)=O)CC(C2(C)CC2)C1 c1(CCC)nc(C(=O)NCC2(CNC(=O)COc3ccccc3)CCC2)co1 N1(C(Cc2cccc(C)c2C)=O)CCC(NC(C2(CCO)CC2)=O)C(CO)CC1 Cc1occc1CC(=O)NCC1CCCN1C(=O)CC1(N2CCCC2)COC1 C(C(CC(F)(F)F)NC(C1(C)CC(C(F)(F)F)C1)=O)NC(C(CC)SC)=O N1(C(c2cc(C)sn2)=O)CCC(C(=O)NCCC2C=CCC2)CC1 c12ccc(cc1Cl)NC(=O)N2.C12CC1C(=O)N2.C(C)(C)(C)OCCOC N1(C(C2CC(SC)C2)=O)C2CCC1CC(CCNC(=O)C=CC1CCOC1)C2 c1(-c2ccc(C(=O)NC(C(CO)NC(C(F)=CCC)=O)C)o2)ccccc1Cl N#Cc1ccc(S(=O)(=O)NC2CCCc3ccoc32)cc1 C1(NC(CN(C)S(N)(=O)=O)=O)CC(O)CN(C(=O)COc2c(F)cccc2F)C1 N1(CCS(CC)(=O)=O)CC2C(C(F)(F)F)(C1)CC2O C1(CNC(C(CCC)=CCC)=O)CCCC2CN(C(C3(C)CNC(=O)C3)=O)CC12 N1(CCC)CCC(N(C(c2cc(CC(C)C)c[nH]2)=O)C(=O)C2CC2)CC1 c1(C(=O)NCC(C)N(C(=O)Cc2cnns2)C)cc(-c2ccns2)on1 C12(CNCCNC(CCSC)=O)CCC(C(F)(F)F)(CC1)O2 C(=O)(CCCC1CCOCC1)N(CC(CNC(CCOCC)=O)O)C c1(C(=O)NCC2CCN(C(=O)C3=C(Cl)CCOC3)C2)ccc2nc(O)ncc2c1 N1(C(CC(=C)C)=O)CCC(C2CCN(C(c3cc(C4CC4)sn3)=O)CC2)C1 C(C(=O)NCC1CC(NC(=O)Cc2cc(C3CC3)no2)C1)(C(C)(C)C)SC C1(C(=O)NCCN2CCOC2=O)CC2COC(C3CC3)CN2C1 C1(C(N2C(CC(=O)NC)CC2)=O)CCCN(C(C2CC(=O)OC2(C)C)=O)CC1 N1(C(CCCC=C)=O)CCC2CN(C(C3CCCC(=O)N3)=O)CC12 c1(C(=O)NC(c2ccc(Cl)cc2F)C)cccc2c1CN(C(C1CN(C)C1)=O)CC2 c1(-c2cc(CNCCCNC(=O)OC)sc2)ccc(F)cc1 c1(C(=O)NC2CN(C(CC(CC)(F)F)=O)C(CO)C2)c(Cl)c2ccccc2n1C C1(CCC)CN(C(=O)C(C)c2ccco2)CCN1C(c1scc(C)c1Cl)=O N1(C(C2(C(CC)=O)CC2)=O)CC(C(N2CCOC(C)C2CO)=O)C(C)(C)C1 c1(C(=O)NC(C(=O)OCCCC)C(CC)CC)n[nH]c2ccc(N)cc12 c1(OCCCF)ccc(Cl)c(C)c1.CCCC(=O)N(CC(C)NC(=O)C(C)O)C(C)C c1(CN2CC(O)(C(=O)Nc3cncs3)C2)nnc2n1CCCCC2 Cn1cc(NC(c2ccn(CCNC(c3cnnn3CC(C)(O)OC)=O)n2)=O)cn1 N1(CCCOCC)CCCC(C)(NC(C2(C)CNC(=O)C2)=O)C1 C1(NC(Cc2ncc(C)s2)=O)CCCN(Cc2n[nH]c(C3CC3)c2C)C1 N1(C(CCC2CCC(=O)N2)=O)CCC(C2CN(C(C3(F)CCOCC3)=O)C2)CC1 CC1CC(C)(C)CN1C(=O)C(CNC(=O)C(C1CCCCC1)F)CC1CC1 c1(C(=O)NC2CCN(C(C3(C)CCCCO3)=O)C2)cc(N)ccc1Cl Cc1ccc(N(C(c2ncc(Cl)s2)C(=O)NCC2CCOC2)C)c(C)c1C c1(C(N2CC(C(N3CC(NC(N)=O)C3)=O)(SC)C2)=O)cncnc1C c1(-c2cc(C(N3C(Cc4cn(C(C)C)nn4)CCC3)=O)on2)ccccc1CO CC(C)C(O)C(C)C(=O)NCCc1nc(C(=O)N(C)CC2CC2)co1 c1(CN2CC(CC)N(c3nc(C(=O)OC)nc(C)c3Br)CC2)cc(F)c(F)cc1C c1(C(N2CCN(C(c3ccns3)=O)CC2)=O)cc2cccc(OC(F)F)c2o1 N1(C(C(C2CC2)SC)=O)CCOC(C)(CNC(c2nnc(Cl)cc2N)=O)C1 C1(F)(C(=O)NC(C)CCC(N)=O)CCCN(C(C2CCOC(C)(C)C2)=O)C1 c1(C(=O)NCC(=C)CCNC(=O)C(C)CCOC)cc(C#N)ccc1Cl CC(C)CC(CN=c1cc(Cl)nc[nH]1)NC(=O)C(C)(O)C1CCC1 C1(COC)CC(CNC(C2C=C(C)CS2)=O)N(C(C2CCC(C(N)=O)CC2)=O)C1 N1(C(C(C)=C(C)C)=O)CC2CCC(N(C(=O)C(c3cncn3C)O)C)C2C1 C1(NC(=O)COC2CC(NC(C3CCCNC3=O)=O)C2)CCc2n[nH]cc2C1 C1(N(C(=O)CCc2cncnc2)C)CCCN(C(c2c[nH]c(C(N)=O)c2)=O)C1 CCCC(C(=O)NCC1C2CCCC12)NC(c1cc(C(C)C)[nH]n1)=O c1(C2(NC(CCCOC)c3cccnc3)CC2)ccncc1F c1(C(N2CC3CC(NC(C4(C)CCCCO4)=O)C3C2)=O)cc(F)cc(F)c1O N1(C(CC)=O)CCC2(CCC(NC(=O)C(CC3CCC3)NC(C)=O)CC2)CC1 C(=O)(C1=CCCC(C)(C)C1)N1CC(CCNC(c2ccc(CC)o2)=O)(OC)C1 CCC(C)C(O)C(C)C(=O)N1CCOCCC1C(=O)NOC(C)C Cc1ccnn1C(C)C(=O)NC1CC(CC(=O)NCCOCCO)C1.CCCC C1(C=C)(C(N(CCCCO)CC)=O)CCN(C(c2ccc(C)[nH]2)=O)C1 O=C1CCOC(C(=O)NCC=CCC(N2CCC(F)(C(N)=O)C2)=O)C1 C1(NC(c2c(N)cccc2)=O)CN(C(c2nccn3cnnc23)=O)CC12CCC2 C12CCOCC1C(=O)N2.C1(CC(=O)NCCn2cncn2)(COC)CCC1 N1(C(Cc2cc(COC)on2)=O)CCC(C(=O)NC2CC=C(C)CC2)C1C(C)C C1(O)(CC#C)CCN(c2nnc3n2C3C2CCCC2)CC1.C(=O)(C(C)C(C)C)OC C1(C(N(CCNC(=O)C=CCc2cscn2)C2CC2)=O)CCc2ccccc2O1 C1(CC(=O)NC(c2nccs2)CC)CC2CNCC2O1 C#CC1CN(C(=O)C(CCOCC)NC(c2ccnnc2)=O)CCO1 S(=O)(=O)(c1ccc(C)cc1)N1C(C(=O)NCCNC(CCOC)=O)CCC1 c1(C(=O)Nc2occ(NC(=O)OC(C)(C)C)n2)cccc(CS(C)(=O)=O)c1 C(=O)(CC(C)CC(=O)NC1CCCN(C(=O)OC(C)(C)C)C(F)(F)C1)OC c1(C(C)(C)C)ccc(C(=O)NCCNC(c2c[nH]nc2C2CCCCC2)=O)nc1 Cc1cnccc1C=CC(=O)NCCC(O)CNC(c1ccc(Br)cn1)=O C(=O)(C(CO)C(C)(C)C)NC1C=CC(CNC(c2cc(OC)ns2)=O)C1 C(=O)(CCN(C)CCO)NC(CN(C(=O)CCC1OCCO1)CC)C C12(NC(c3cc(C)sn3)=O)CN(C(c3ccc(CO)o3)=O)CC1CS(=O)(=O)C2 c1(C(=O)OC)cc2oc(CC(C(C)C)C(C)SC)cc2[nH]1.C(C)(C)N C1(N(C(=O)CCC(=O)Nc2nccs2)C)CCCC(NC(C2OCCCO2)=O)C1 Cc1ncc(CNCCOCc2ccco2)[nH]1 c1(C(=O)NCC(CNC(C2C(C)CCO2)=O)CO)cnc(C2CC2)nc1 N1(C(c2n(CC)nc(C3CC3)c2)=O)CCC2CN(C(c3cnsc3)=O)CC2CC1 N1(C(C23CN(C(=O)CC4(O)CCCCC4)C(CC2)CC3)=O)CCC2(CCCOC2)C1 C12(C(=O)Nc3ccc(Oc4ccc(Br)cc4)cc3)CCCCC1C1C=CC21 C12(NC(CSCC#C)=O)CCCCCC1N(c1cc(O)nc(C(=O)NC)n1)CC2 c1(OC)ccc(-c2ccc(CN(C)C(c3cccs3)C)s2)cn1 CC(C(=O)NC1(CN(C)C(c2cc(F)ccc2O)=O)CC1)C(F)(F)F C#CC1CN(C(=O)COCCN(C)C)CCN1C(=O)COC C1(NC(C2C(C)C2C)=O)CN(C)CC1S(C)(=O)=O.c1(C(=O)N)cnn(CCO)c1 CC(C(=O)NCC1CCOC1C(=O)NC(C)(C)CCCO)C(F)(F)F C(=O)(CC(C)(C)CC(F)F)N1CCC(C(=O)NC(C)CC(F)F)CC1 CC1(C)CC(C(=O)NC2CC3(CC3)C2)CCN1C(C1CCC(C)(C)C1)=O Cc1ccc(C(=O)NCC(C)(C)OCCCNC(=O)Cc2nc(=N)[nH][nH]2)n1C CCC(C(=O)OC)C(=O)NCCCCCCNC(=O)CC1CCCOC1 C1(O)(CC(=O)N(CC(C)NC(c2ccoc2C(C)C)=O)CC)CCOCC1 Cc1c(C(=O)NCC(C)NC(c2cc(O)nn2C)=O)nnn1-c1cnn(C)c1 C=CCCCCC(=O)N(C1CCCN(C(=O)C=Cc2ccc(C(N)=O)o2)C1)CC C(CNC(C1C(C)(C)C1(F)F)=O)(C(C)(C)C)NC(C1C(C)CC1)=O C#CCCC(C(=O)NCC(CCC)CCO)NC(c1cc(F)cc(F)c1)=O c1(C(=O)NC2CC3(CC(NC(C4CCC(OC)C4)=O)C3)C2)cc(C)c(C)cc1C N1(C(CC)=O)CCCC(Nc2cc(NCc3n[nH]c(=N)s3)ncn2)C1 C(=O)(C1CCCc2c1ncn2C)NCC1CC(NC(c2ccn(COC)n2)=O)C1 C1(CC)CN(C(C2(c3ccccc3F)CC2)=O)CCC1NC(=O)C1=CCCCO1 c1(OCC(=O)NCCCNC(CCC2CCC(C)O2)=O)ccc(Cl)c(Cl)c1 c1(C(=O)NC(CC)CN(C)C(c2cc(CO)ccn2)=O)ccc(C=NOC)cc1 c1(OCC(N2CC(F)(CNC(c3cc(C(F)F)no3)=O)C2)=O)ccccc1Cl Cn1ccnc1SCCCOCC(=O)NC(C)(C)CC(=O)NCCNC(=O)CCF c1(NC(C)C(c2ccccc2)N(C)C)ncnc2c1nc(O)n2C N12CCCCC(C1)C2.Cc1cc(CNC(c2csnc2-c2ccccc2)=O)sn1 N1(C(c2c(N)nccc2)=O)CCCC(NC(=O)CC(c2ccccc2)C2CC2)CC1 n1(CCC(N2CC(C(C)NC(=O)CC3(C(F)(F)F)CC3)C2)=O)cnc2ccccc12 C1(NC(C(C)(C)C2CCC2)=O)CCN(C(c2cnn(CC(F)F)c2)=O)CC1 N1(C(=O)OC(C)C)CCC2(C)C(C1)C2(Br)Br.c12ccc(cc1)COC2=O c1(C(=O)NCCC(CCNC(C(C)(C)OC)=O)C)ccn2nccc2n1 C1(CC(N2CC(C3CC(NC(C4(C(N)=O)CC4)=O)CCO3)C2)=O)CCCC1(F)F C(=O)(C1=CC2(CCOC2)C1)N1CCC(C(C)(C)NC(=O)C=C2CCCC2)CC1 N1(C(C(c2cccnc2)C)=O)CC=CC1CNC(=O)CCN1CCCC1=O c1(C(=O)NCC(C2CC2)NC(C2N(C(C)=O)CCCCC2)=O)ccc2cncn2c1 C(=O)(N=c1ccn(CC(N2CCC(O)C(F)C2)=O)[nH]1)c1nn(C)c(C#N)c1 C1(CNC(C2(CC=C)CCC2)=O)(CNC(=O)Cc2cc(C)nn2C)CC12CCC2 n1(CC(=O)NCC2C3CN(C(=O)CCN4CCCC4)CC23)cnc([N+](=O)[O-])n1 c1(C(N2C(C(=O)Nc3cc(C#N)sc3)COCC2)=O)cc(F)c2cn[nH]c2c1 c1(N(CCCNC(NC=C(C)C)=O)C)ccc(Cl)cc1 N1(CC(=O)NC(CNC(C=CC)=O)Cn2cc(CC3CC3)nn2)CCC(C)(O)C1 C1(NC(C=Cc2c(C)ccnc2)=O)CN(C(=O)C(C)(C)C(F)(F)F)CC1C1CC1 CC1OC2(CO)CC1(C(N1CCN(C(c3cc4occc4s3)=O)C3CC13)=O)C2 C=C1CC2(C1)CN(C(=O)C=CCNC(c1coc(COC)n1)=O)C2 N1(C(C(C)=C2CC2)=O)CC2CCN(C(C3C4CCCC(F)(F)C34)=O)C2C1 c1(CC(=O)NCCC2(O)CCC2)ccc(-c2nn[nH]n2)cc1Cl c1(C(CNC(C(=O)NCC=C)=O)N)cc(C)no1 c1(CC)cc(Cl)ccc1C(=O)NCC(C)(CO)NC(c1ccn(CCOC)n1)=O CC1CNCCC1C(=O)N(C)Cc1ccccc1SC(F)(F)F c1(C2(O)CC(C(=O)NC(c3cncnc3)C)C2)cccc(Br)c1 C(CCCCCNC(n1ncc(NC2(C)CCN(C(C)C)C2)c1)=O)OC C1(C)(OC)CCCN(C(c2ccnc(CNC(=O)C(C)(O)C3CCC3)c2)=O)CC1 C1(NC(CN(CCC#C)C)=O)CCCN(C(=O)C(N2CCOC2=O)C)C1 N1(C(c2nc(C)oc2)=O)CC(C)(C(N2CC(C)(C)CCC2C)=O)CC1(C)C C1(C2(O)CN(C(=O)C(C)C3CCOC3)C2)(CNC(CCCC#C)=O)CC1 c1(C(=O)NC2C(CC)CN(C(=O)Cc3cccnc3O)C2)cc(C)c(O)nn1 C1(NC(CSCC)=O)CN(C(C2CC2CC)=O)CC1C(F)F c1(CC(=O)NC(C(C)NC(C=CC=CCOC)=O)CO)nc(C)c(C)[nH]1 CCCC(C)(O)C(=O)N(CC)CC1CCCN(C(c2ncc(N)nc2C)=O)C1 N1(C(c2c(C)nns2)=O)CC2C(CNC(=O)CCSC3CCCC3)C2C1 C1(NC(CCN(CC)CC)=O)CC2COCC(C1)N2C(=O)Cc1cc(Cl)cs1 C12(NC(c3ncc(OC)cn3)=O)CCCC1CN(C(=O)CCc1c[nH]c(=N)[nH]1)C2 N1(C(CC(=O)NC(C2CN(S(=O)(=O)C(F)F)C2)C)=O)CCN(C(N)=O)C(CF)C1 C(=O)(C1=NOC(CNC(C2(C3CC3)CC2)=O)C1)NCCC1C(=O)NC(=O)N1 Cc1nc(C2CC2)sc1CC(=O)NC1(C)CC(NC(C2CC(C)(C)C2)=O)C1 C12(CNC(NC3CCS(=O)(=O)C3)=NCC3CCCO3)CCC(CC1)OC2 C1(C2CC(NC(CCC#C)=O)C2)CN(C(=O)C(COC)COC)CCCO1 N1(C(c2cc(CC)n(C)n2)=O)CC(C)(C)CC1C(=O)NC1CC=CCC1 c1(NC(=O)NC2CCCN2C(=O)C2CC2)ocnc1C(=O)NCC(CNCC)F CC(CC#N)C(=O)NN1CCCC1C(=O)NC1(C2CCC2)CC1 C12(C(=O)NC)CCC(C(=O)N=c3[nH][nH]cc3C(=O)OC)(CC1)CC2 c1(C(=O)Nc2nc(C(N3CCC(C(=O)OCC)C3)=O)n(C)c2)ccc(Cl)c(O)c1 N1(C(c2c(N)ccc(C)c2F)=O)CC2CCOCC2(NC(=O)CCF)C1 c1(C(C2C(C(N(CC(CN(C(=O)C(C)(F)F)C)O)C)=O)C2(F)F)=O)cncc(F)n1 C1(CC2N(NC(=O)C(=O)NCC3CCCCS3)CC2)COc2cscc2O1 c1(-c2nnc(C)o2)cnc(N2CCCC(NC(c3coc(Br)c3)=O)C2)nc1 C1(OC(Cn2c(C(C)C)nnn2)=O)CCN(C(=O)CC2CC3(CC3)C2)CC1 CN1CCC(=CC(N2CCC(CNC(c3ccnc(Cl)c3)=O)C2)=O)CC1 c1(CC(=O)NCC2CC(NC(C3CCC4CC4CC3)=O)C2)cccc(Cl)c1F C1(NC(=O)C=CCO)(CNC(C2CCCC(F)C2)=O)CCOCC1 n1(CC(=O)N(CCCN(C(=O)CO)CCO)CCO)cncn1 CC1(NC(c2cocn2)=O)CCN(C(C2CC(C(C)(C)C)C2)=O)CC1 C12(C(=O)NCCC3(CNC(c4c(N)cccc4)=O)CC3)CCCCN1CCC2 C1(C(N2CC(OCCOC)C2)=O)CN(C(=O)CCCC2CC2)CC12CCC2 C1(O)(C(C)NC(C2CCCC2c2nc[nH]n2)=O)CN(C(C2COC(=O)N2)=O)C1 C1(NC(C(CC)F)=O)CC2(CNS(=O)(=O)Cc3cccc(C(F)F)c3)COC1C2 C1(N(C(C(=O)NCC)C)C)COCCC1N(C)C(C1CN(C(=O)OC)C1)=O c1(C(=O)NC2CN(C(C(C(C)(C)C)OC)=O)CC23CC3)nc(Cl)c(=O)[nH]c1N Cc1cc(C(=O)N(C)CCOCCN(C)C(c2ncsc2C2CC2)=O)cc(C)c1 c1(OC)cc(C(N2CC(NC(c3c[nH]c(C)c3)=O)CC2(C)C)=O)ccc1C c1(NC(C(C)NC(=O)C2CC2)=O)ccccc1Cl.C1(=O)C(=O)NCCCN1C N1(C(C2CC(CC)(CC)C2(CC)CC)=O)CCCC1(C)NC(=O)COC1CCOC1 Cc1cnc(S(C)(=O)=O)nc1N1CC(NCc2cnc(N(C)C)nc2)C(F)C1 Cc1[nH]nc2ccc(C(=O)NC34CC(CNC(C5CC5C)=O)(C3)OC4C)cc12 Cc1sc(CC(=O)OC)nc1CC(=O)N(C(C)CNC(C1CCCCC1)=O)C C#Cc1ccc(C(=O)NC2CCOCC2NC(=O)CNC(c2ccco2)=O)nc1 O=C(N=c1[nH]n(-c2ccccc2)cc1Cl)C1CCOC1Cc1ccc(Cl)c(F)c1 N1(C(C(CC(=O)OC)C)=O)C2CCC1CN(C(c1cc(CC(C)C)on1)=O)C2 c1(C(=O)NC2CCN(C(=O)C(C3CCCCC3)O)C2)ccc2c(c1)C(=O)CCC2 c1(C2C(C(=O)NCC(CC)NC(c3ccoc3CC(N)=O)=O)C2)cccc(F)c1 C1(C(N2CCC(NC(CC(=O)NCC(F)(F)F)=O)C2)=O)CCC2(CCOCC2)O1 c1(N(C)C)ccc(N=c2nc(-c3ncn(C)n3)[nH]c3c2COC3)cc1 c1(C(N2CC(CC(C)NC(C(C)OCCOCC)=O)C2)=O)oncc1C C(=O)(C(C(C)(C)C)SC)NC1C(CNC(c2nc(CCC)oc2)=O)COC1 C#CCC(CC#C)C(=O)N1CCOCC1CNC(=O)CC1(C)CCCO1 c1(C(N2CCC(CCNC(=O)CC(F)F)CC2)=O)[nH]c2ccccc2c1Br N1(C(=O)OC(C)COC(C)(C)C)CCC(C)C(NCc2ccon2)C1C C1(NC(c2cn(C)nc2)=O)COC2(CCN(S(=O)(=O)c3cccnc3Cl)CC2)C1 C1(C(=O)NC(c2cc[nH]n2)C)(N(C)C(=O)OC(C)(C)C)CC(F)C1 c1(CCC(=O)NCCCCNC(C(CC)n2cncn2)=O)ccc2ccccc2n1 C(=O)(CCCNC(C)(C)C1(CO)CCC1)OC.C(CC(C)O)N C(c1ccncc1C)=CC(=O)NC1(COC)CN(C(C=CC=CC)=O)C1 c1(NCC(C2CC2)NC(c2nnn(C(C)(C)C)n2)=O)ncnc2c1c(Br)nn2C N1(S(C)(=O)=O)CCC(NC(=O)NC(C2(O)CCCCC2)CNC(C2C=CCC2)O)CC1 C1(CNC(CCNC(c2ccncc2)=O)=O)CN(C(C2(Cl)CC2)=O)CCC1(F)F CC1CCCN(C(C2(C(=O)Nc3ncccn3)CC2)=O)CC1 C12(CNC(C(CCOC)(C)C)=O)CN(C(C3CC3(C)Br)=O)CC(F)(C1)C2 c1(N2C(C(C)(C)NC(CC(C)F)=O)CCC2)nccc(N(C)C)n1 Cc1cccc2cc(C(N3CCC(C)(NC(c4csnc4Cl)=O)CC3)=O)oc12 C=CC1OCCCC1C(=O)NCC1CC(NC(c2cnccc2N(C)C)=O)C1 C(=O)(NN=c1ccc2nncn2[nH]1)c1nc(-c2cccc(C)c2)nn1C1CCOC1 C(C)(CCCCO)NC(C)(C)C.C12(OC)CN(C1)C(=O)OC2 N1(C(C=CC(C)NC(=O)C#CC2CC2)=O)CC(=O)NC2(CC2)C1 C12(CNC(c3nc(N(C)C)oc3)=O)CC(CCO1)N(C(=O)CCn1cccn1)C2 CCCCCCn1nnnc1C(C)(CNC(C)=O)NCC1CCC(=O)O1 c1(CC(=O)NCC2CN(C(C3CC(SC)C3)=O)CC23CC3)cnc2ncccn12 CS(=O)c1ccc(-c2cn(CCCCCNC(=O)C(N)=O)nn2)cc1 C1(C(=O)OC)CCCC(C(=O)NC2CCC(NC(c3ccc(C)nc3)=O)CC2)C1 c1(C(N2CCC(NC(C3C(=C)C3)=O)C2C)=O)cnc2ccnn2c1C c1(CC(=O)NCCCOCCNC(CC(C)OC(F)(F)F)=O)cc(F)ccc1O c1(SC)ncc(Br)c(=NC(=O)C23CCC(NCc4ccc(Br)nc4)(CC2)CC3)[nH]1 C1(OC(C)=O)CN(C(=O)C(C)n2cccn2)CC1c1cn(CCOCCC#N)nn1 C1(=O)CCN=C(NCc2ccc(C)o2)NC(C)CC1=O.C(C)(C)C.CN CC1(C)CC(C(=O)N2CCC3C(NC(c4n[nH]c5c4CCC5)=O)CC23)=NO1 CC1(C)C(NC(=O)C=Cc2cc[nH]c2)CC1CNC(c1ccon1)=O C1(C(=O)NC2(CCCNC(C3(C)CN(C)C(=O)C3)=O)CC2)CC2(C1)CC1(CC1)C2 Cn1[nH]c(C(=O)NC2CCCCC2NC(C2CC2(C)C(F)F)=O)nc1=O CN(OCC(F)(F)F)C(=O)C(F)CC1CNC1.N1(CC(=O)N)CC=CC1 c1(C(=O)NCc2c(CN(C(CC=CCC)=O)C)cccc2)cc2scnc2[nH]1 N1(C(C2(C(=O)NC)CC2)=O)CC(Nc2nccc(C(=O)OC(C)=O)c2)C2(COC2)C1 c1(CN2CC3(CC(C(=O)NC(C(C)O)CO)C3)C2)ccc2c(c1)nnn2C c1(C(=O)NCCN(C(=O)C#CC2CCC2)C2CCCC2)c[nH]c(=O)c2ccnn12 C(=O)(CCCC(=O)OC)NC(C1N(C(C(COC)COC)=O)CCC1)(C)C C1(NC(=O)C2=COCCC2)CC12CCN(C(=O)Cc1csnn1)CC2 C(=O)(C(C)(C)C(=O)N(CC(C)(C)C(=O)NC(C)C)C)NC(CCC1CCN(C)C1)=O O=Cc1sc(CNC2CN(C(c3cc(Cl)cc(Br)c3)=O)CC2C#N)c(Br)c1Br C(CCCCCC(=O)Nc1cnc(F)nc1)NC(=O)CNc1cn[nH]c1 C=CC(F)(F)C(=O)NCC(O)C(=O)NCCCCN(C)C Cn1[nH]c(=NC(=O)C2CC(C)N2C(=O)C(Cl)Cl)cc1C1CC1 CC(C)CC(C)C(C(=O)NCC1CCCO1)N1CC(=O)NC(C(C)C)C1 c12ccc(cc1C)o2.N1(C(C(=O)NCC)C2CC2)CCSCC1CC#N C1(CC)CC(C)CN(C(=O)CCCCCN(C)C(c2ccsc2OC)=O)C1 N1(C(C(CSC)C)=O)CC(C(=O)NCCCn2ccnn2)C(C)C1 C1(N(c2ncc(I)cn2)C)CC2CCC(C1)N2C(=O)Cc1nc(F)c(F)cc1F C1(NC(C(C)OCCOC)=O)CC2CC(C1)N(C(C1CC3CCC(C1)C3)=O)C2 c1(C(N2CC(NC(C(C(C)C)C)=O)C(C(F)(F)F)C2)=O)ccc2nc(O)oc2c1 c1(C(N2CCC3CC(CCO)C3C2)=O)cc2nc(Br)sc2[nH]1 C1(C(=O)NC(CNC(C(c2ccccc2F)(C)OC)=O)C)C2CNC(=O)C12 N1(C(C(C(C)C)N(C)C)=O)C2CCC1CN(C(=O)C(=Cc1cn(C)nn1)F)CC2 c1(C(=O)OC)ccc(C)c(CNC(=O)C(=O)NC(c2ccc(C(C)C)cc2)C)c1 CC(C)C(CC(=O)N1CC2(CC(NC(C3OCCN(C)C3=O)=O)C2)C1)C(C)C C#CCC(CC(=O)N=c1ccn(CCF)[nH]1)NC(=O)CC1CC1(Cl)Cl S(=O)(=O)(c1ccc(NCC(C)Cn2cccn2)c(Cl)c1)NC(CC)CO c1(C(=O)NCC(CN(C)C(c2csc(C(N)=O)n2)=O)(C)C)cc2[nH]ccc2s1 c1(C(N2CCC(O)(CCNC(C3(C(=O)NC)CC3)=O)C2)=O)cc([N+](=O)[O-])oc1C C1(O)(CNC(C(CC)CC)=O)CCCN(C(C2(C#N)CC3CC3C2)=O)CC1 S(=O)(=O)(c1ccc(Br)cc1NCc1cccc(Cl)c1Br)NC(CCC)C C=CC1CCCCN1C(C12CC(CN1C(=O)C1=CCCCC1)C2)=O Cc1ccccc1NCCCC12CCCC1C2 C1(NC(c2nc(C)sc2)=O)CN(C(c2ccc(CN3CCCCC3)o2)=O)CC1C Cn1cc(C(=O)NCCCOCC(C)(C)NC(c2ccc(Cl)o2)=O)nn1 c1(C(=O)NC2CCC(C)(CNC(C3CN(C(C)=O)C3)=O)C2)c(C)nc(O)nc1C C1(C2CCC2)(C(=O)NCC2CN(C(c3cc(C)cc(Cl)c3)=O)C3C2C3)CC1(F)F N1(C(c2c[nH]c(C(=O)OC)c2)=O)CCC(CO)(CNC(c2c[nH]cc2C)=O)CC1 C(=O)(C#CC1CCCO1)NC1(CCCNC(C(CC)SC)=O)CC1 C(=O)(C1=COCCO1)N1CC(CCC)C(NC(=O)C(C)(O)Cn2cccn2)C1 c1(CNC(C(C2CC2)OC)=O)cc(C)c(C(=O)Nc2cncc(Cl)c2)o1 C(=O)(C#CC1CCCOC1)NC(CN(C(C1(O)CCOCC1)=O)CC)C.CC(C)CC C1(F)(C(N2CC(OC)C(NC(C3(SC4CCC4)CC3)=O)C2)=O)C(C)(C)C1(C)C C12CN(C1)CC(C1(C)CC1)NC(=O)N2.C1(COC)(C(=O)OC)CC1 C(=O)(C(CC(C)C)ONC(c1ccncc1F)=O)NCC(=O)NCC C1(C(=O)NCCCCCNC(C(N)=O)=O)CCCC2(CC2)C1 C(CCC(=O)NC1CCC(CNC(=O)COCC)C1)OCCOCC c1(C2C(CC(=O)NCC(CNC(=O)CC3C=CCCC3)OC)C2)ccc(F)cc1 N1(C(C(C)CC2CCCC2)=O)CCc2c(CNC(=O)CN3CCC3)cccc2C1 Cc1cc(C(=O)C(N2CCC(C)(NC(C3CC(F)C(=O)N3)=O)CC2)=O)ccc1F c1(NC(C2C3CN(Cc4c(C)cc(O)cc4)C2C3)=O)c(Cl)ncc2ccccc12 c1(C(=O)NCCC2(NC(C(CSC)O)=O)CCCC2)cccc2c1NC(=O)CO2 C(=O)(CN=S(C)(C)=O)NC(c1ccccc1)CN(C(=O)C#CC1CC1)C c1(C(N2CCC=C(C(=O)N3CCC3CO)C2)=O)cccc2c1OCCC2 C1(OC)CC(C(N2CCC(N3CCC3)C2)=O)N(C(c2cnc(OC)nc2)=O)C1 c1(OC(C(=O)NCCC2(CNC(c3cc(C)oc3)=O)CC2)C)cccc(C#N)c1 Cc1cnn(C)c1CNC(=O)CN(C)C(c1csc(F)c1)=O N1(C(C(C)=CC2CC2)=O)C2CCC1CC(O)(CNC(=O)C(C)(O)C(C)C)C2 N1(C(c2cc(C)c(F)cn2)=O)CCCN(C(c2ccc(C(N)=O)nc2)=O)C(C)C1 C1(C(=O)OC)CN(N2CCSCC2Cc2nc[nH]n2)C1 N1(C(c2n(CCC)nc(C)c2)=O)CCCCC(C(=O)O)C1 n1(CC)cc(Cl)c(C(N2CC=CC2CNC(c2cccc(C(C)C)n2)=O)=O)n1 c1(C(N(CCN(C(=O)C(n2cc(Br)cn2)C)CC)CC)=O)cccn1C c1(C(N2CCN(Cc3nc(CN)on3)CC2)=O)c[nH]c2c(F)cccc12 Cc1c(C(=O)NC2CC(C)N(C(=O)CCOCCN(C)C)C2)cnn1CCO N1(C(Cc2c(C)noc2Cl)=O)CC2CS(=O)(=O)CC2(NC(=O)C(C)(C)CC2CC2)C1 C(C)(CCCCNC(c1ncoc1C(C)(C)C)=O)NC(c1cc(C(C)C)no1)=O S(=O)(=O)(c1ccc(C(=O)NC2CCC2NC(c2cnc(C)s2)=O)cc1)NCC C(C)(CN=C(NCC(C)(C)C)Nc1ccc(OC)c(CC(F)(F)F)c1)(C1CC1)OC N1(C(CN(C(=O)OC)C)=O)CC(CCNC(C2CCCN2C)=O)(OC)C1 N1(C(CCC)=O)CC(OC)CC(CNC2(C#N)C(C#N)C2(Br)CC)C1 CC1COCC1N=c1nc2sccc2c(NCCS(N)(=O)=O)[nH]1 CCS(=O)CC(=O)N1CC(NC(=O)C(F)(F)c2ccncc2)CC1C N1(C(C2C(C)=C2)=O)CCCC2(NC(c3coc(-c4ccccc4)n3)=O)CC2C1 N1(C(CN(C)C)=O)CCN(C(C2CCOCC2(C)C)=O)CC1CC(F)F N1(CC(C)(C)NC(C2(Br)CC2(F)F)=O)CCc2ccccc2C1=O c1(NC(c2c(OCCOCCOC)c[nH]n2)=O)ccc2c(c1)C(C)C(C)C2(C)C N1(C(CC2(C)CC2)=O)CCC(N(n2cccn2)C(=O)CSc2n[nH]c(O)n2)CC1 Cc1cccc(C(N2C3CCC2C(C(N2CC=CC(O)C2)=O)C3)=O)c1C N1(C(c2cn(C)nn2)=O)CCC(C(c2cccs2)=O)CC1.C12CC13CC3CNC2=O CCCC(CC(C)C)C(=O)NC1(C(=O)NC2CCC3(CC3)C2)CC1(C)C N1(C(C(COC)NC(C)=O)=O)CCN(C(C2(CC(C)C)CCCC2)=O)C(C)C1 c1(C(N(C2(CNC(=O)Cc3ccoc3)CC2)C2CC2)=O)ccc(-c2cscn2)cc1 c1(NC(C)=O)ccc(CNCC(c2cccc(F)c2)O)cc1 CSC1=C(C(=O)NC2CCN(C(=O)C=CCOCCOC)C(C)C2)CCCC1 c1(C(=O)NC2CCC2NC(C2C=CCC2)=O)cc2c(Cl)ccc(Cl)c2[nH]1 c1(CN(c2ccn(-c3ccc(-c4ccoc4)cc3)n2)C)ccc(F)c(F)c1 C(CCC(=O)NO)NC(C(C1CCC(N)C1)(F)F)=O Cn1cnc2cc(C(=O)NC(C)(CNC(c3cc(O)cc(=O)o3)=O)CO)ccc12 Cc1c(C(=O)NCC(C)NC(=O)CC(C)N2CCCC2=O)cccc1C(F)(F)F C1(CCC(N2C(C(=O)C3CC3)CCCC2)=O)CCc2ccccc2C1=O CCC(CC)(CO)C(=O)NCCC1CC(NC(C2CCC(=O)N2C2CC2)=O)C1 CCC(CCC(=O)N(C1CCCC1C#N)C)NC(=O)C(C)n1ccnn1 c1(CC)cc(CC)ccc1NC(C1CCC(OCCF)C1)=O c1(C(=O)NCCC(C)N(C(CCc2cnc(C)o2)=O)C)ccc2c(c1)CCC=C2 N1(C=O)CC(C)(CO)CC1(C)C.Cn1nccc1C=CC1N(C(C=C)=O)CCC1 c1(NC(=O)CC2CCN(C(=O)CC3CC3)CC2)ccc(Br)cc1O c1(C(C(=O)N(CC(C)NC(C2C(CCC)CCC2)=O)C)O)ccccc1F C(=O)(C(CC1CC1)NC(=O)CONC(=O)Cn1ccnc1)OC N1(C(C2CN(C(C(C)SC(C)C)=O)CC2C)=O)CC(C(N)=O)CC(C)C1 C1(C(=O)NC2CC(NC(=O)C(C)CC3CCCC3)C2)(COC)CC=CC1 C1(CN(C(=O)CC2CC3C=CC2C3)C)CN(C(=O)CN(C)C2CC2)CCO1 C123CN(C(CNC(C4(C)CCS(=O)(=O)N4)=O)(C1)C2)C(=O)OC3.C(C)(C)(C)OC c1(C(N(C2CCC(CNC(CCN(CCC)C)=O)CC2)C)=O)cc(=N)[nH]c(Cl)n1 c1(CC(=O)N(CCNC(C(c2cccc(Cl)c2)C)=O)C2CC2)ccccc1Cl CC1CC(C)(C(=O)NC2CC(C)(NC(c3cc4n(n3)CCC4)=O)C2)CC(C)O1 Cc1nc(C(=O)C(=O)NC(C)(CNC(=O)CN(C)C)Cn2cccn2)cs1 c1(C(C)NC(N2C(CCC=C)CCC2)=O)ccc([N+](=O)[O-])cc1 C=C(Cl)C(C)(C)C(=O)N1CCCC(COC)(NC(=O)CCSCCCC)C1 C1(NC(C(CCOC)C)=O)CCN(C(c2cc(OC)cnc2F)=O)C(C)C1 C1(NC(C(=O)N(CC(c2ccccc2)O)C)=O)CC2CCC(C1)N2CC1CC1 Cc1ccc(C(N2CCC(NC(C3CC3c3cccnc3)=O)C(F)C2)=O)cc1Cl C1(C(N(C2CCN(C(c3cnn(CC)c3)=O)CC2)CCC)=O)CCCC(=O)O1 N1(C(C(C)CN)=O)C2CC1CN(C(c1ccc(Br)c(F)c1)=O)C2 CC(C)C(CCNC(=O)CC1CCCC1(F)F)NC(=O)C(C)OCC1CC1 CC1(C)COCCN1Cc1ccc(C(=O)NC2C3CC4C(C3)C24)c(F)c1 c1(CC)cc(N)c(C(=O)N(C)CC2CCCN2C(=O)Cc2ccsn2)cc1F C(=O)(CCC(F)(F)C(F)(F)F)N1C(C(C)NC(C2CCC(C)(C)CC2)=O)CCC1 C1(CNC(c2nn(CC)c(C)c2)=O)(CO)CCCN(C(C2CCC(OC)C2)=O)C1 C=CC1(C(=O)NC(C2CCN(C(c3cn(C)cn3)=O)CC2)(C)C)CCOCC1 Cc1c[nH]c(C(=O)NCC(CC(C)C)NC(=O)COc2cccnc2Cl)c1C c1(OC)cnc(C(=O)NC(C(C)NC(c2n[nH]c(C)n2)=O)C(C)C)nc1 Cc1cc(CNC(=O)COCCNC2CCC2)ccc1C(F)(F)F Cc1ccc(CC(=O)N(C)CC2CCN(C(=O)C(C)OC(C)(C)C)C2)c(F)c1 CC(C)C(CC(=O)N1CCOCC1CN(C)C(c1cnsn1)=O)C(C)C C1(C(N(CCCN(C(c2occ(C)c2)=O)C)C)=O)CCc2nnc(O)n2C1 C1(CC#C)(C(=O)NC(C)CCN(C(=O)C(O)Cc2cnc[nH]2)C)CCCC1 N1(CC(N2C(C3(NC(=O)CN4CC=CC4)CC3)CCCC2)=O)CCCNS1(=O)=O Cc1ncc(C(N2CCCC2(C)CNC(c2ncccn2)=O)=O)c(Br)c1Cl CCCCCC(F)C(=O)N1CCCC(C(=O)NCCCCc2cnc[nH]2)C1 c1(CNC(C2CN(C(=O)OC(C)(C)C)CC(C)O2)=O)cncc2ccc(F)cc12 C1(C(=O)NC(C)CC2CN(C(C3(C#N)CC3)=O)C2)CCCCCCC1 N=c1[nH]c(C(N2CCC(C(=O)NCCOC3CCCOC3)C2)=O)cs1 C1(NC(c2ccc(C)s2)=O)CN(C(=O)Cc2ccc(Cl)cc2Cl)CC2CCCC12 C(=O)(C(C(C)(C)O)NC1COCC1(C)C)NCCC1C(C)(C)CCO1 C1(C(C(=O)NC(C2(C#N)CC2)C)C)CCCN1C(=O)CN1CCOCC1 C=C(C)CC(C)C(=O)NCC1(C)CCC(NC(c2cn(CCCF)nn2)=O)CC1 CC(CCCCNC(=O)C(c1cccs1)C1CC1)NC(=O)CC1CC(=O)NC1=O S(=O)(=O)(c1c[nH]ccc1=NCCC(=O)Nc1ccccc1)CC(=O)NC c1(C(N2CCC23CCCSC3)C(=O)NCCCOC)ccc2nccnc2c1 C(C(C(C)(C)C)NC(=O)C(C)CC1CCC1)NC(CCCOC)=O CC(=O)CCCC(=O)NCCC(C)CCNC(=O)C(c1cn(C)nc1C(F)(F)F)C C(=O)(C(C)(O)CC)N1CC(C(C(=O)NC(C2CCCC2)C#C)O)C1 C1(CNC(C=CC(C)(C)SC)=O)COC(CNC(C2OCCCO2)=O)C1 C=CC1CN(C(=O)CCNC(=O)C(C2CCCC2)OCC)CCO1 N1(C(C2(CCC)CCNC2=O)=O)C2CCC1CC(NC(c1cc[nH]c1)=O)C2 N1(C(C(C(C)C)C)=O)CC2(CCC(NC(c3cc(C(N)=O)co3)=O)CC2)C1 N1(C(c2c(C)coc2)=O)CC2(c3ccccc3NC3CC(C)OC3=O)CC1CO2 CCC(CSC)C(=O)NCC(C(=O)NC(C)CCSC)N(C)C C1(NC(C)CC(F)(F)c2ccccc2)CCCC12CCC2 C(=O)(C(C(C)(C)C(N)=O)N(C)C)NCCCC(C)NC(CCCNC(=O)OCC)=O CC(C)C=CC(=O)N(CC(N1CCC1)=O)CCO.C(C)C CN1N=C(C(=O)NCCC(O)C(=O)NCCN2CCCCC2)CCC1=O C1(CNC(=NCC)NCc2ccccc2)COC2(CCCC2)O1 CC1CCC(C)(C(N2CC(CNC(=O)Cc3ccccc3F)C2)=O)C1 N1(C(c2c(OCC)n[nH]c2)=O)CCC(NC(C2(CC)CCCCO2)=O)C(O)C1 c1(C(N2CC3(CC(NC(c4cnc(SC)nc4)=O)C3)C2)=O)cc(C)c(Cl)c(C)c1 c1(C(N2CCCC(NC(=O)CC3CSCCS3)C2)=O)cc(F)cc([N+](=O)[O-])c1 C=C(C)C1OCCC1C(=O)NCC1CCC1NC(c1ccc(C(F)(F)F)nc1)=O CC1=NC(C(=O)N(CC(C)CNC(C2(N(C)C)CCCC2)=O)C)CS1 C(=O)(C(CCC(N)=O)N(C)C)NCC(C)N(C(=O)Cn1cc(CO)nn1)CC C1(NC(Cc2c(C)noc2C)=O)C2CCCN(CCOCC(F)(F)F)C2C1(C)C C=CCC(C)(O)C(=O)N1CCC(CCC(N2CCOC(CC)C2)=O)C1 C(=O)(C1=CC2CCCC12)NCC1CN(C(c2n(CC)nnc2)=O)C(C)C1 C(=O)(CCCC(C)(C)NC(c1cnc(C)c(C)c1)=O)N1CC(C)CC(CC)C1 S(=O)(=O)(c1ccccc1)NCC(=O)NCCN(C(CC(C)F)=O)C.C12CCN1C2 c1(CCC)ncc(C(c2nnnn2C2CCOC2)NCC(C)(C)OC(C)=O)[nH]1 CS(=O)(=O)c1cccc(C(=O)NC2(CO)CCCN(c3ccc(Cl)cn3)C2)c1 C(=O)(C#CC1(C)CCCO1)NCC(=O)NCC(N1C(CC)CCCC1)=O C1(N(C(C2(C(C)C)CCC2)=O)C)CN(C(c2cnsc2)=O)CC1O C(C(=O)NCC12CC(CNC(=O)C(C)CC)(CO1)C2)(C(C)C)OCC c1(C(N2CCC(C3N(C(C=CC(C)C)=O)CCC3)CC2)=O)ccn2cccc2c1 N1(C(c2ncc(C)cn2)=O)CC(C2CCN(C(=O)C3=NNC(=O)C3)CC2)C1 C1(C(=O)NCCC)CCCN(C(c2cc(OC)ns2)C(=O)NC2COC2)C1 c1(NC(=O)NC(CN2CC=C(C)CC2)(C)C)cccc2nsnc12 C(CN=C(NCc1cnn(C)n1)NC1CCN(C2CC2)C1=O)N(C(C)=O)CC C1(CNC(C(n2ccc(C)n2)C)=O)CN(C(c2csc(C)c2N)=O)CCC1(C)C c1(CC)cccc(C(=O)NCC2CCN(C(=O)CCSCC(C)C)CC2C)c1C Cc1nn(C)c(N)c1C(=O)NCC(C)(C1CC1)NC(=O)CN1CCOCC1=O C12(C(=O)NCC(C)CNC(=O)Cc3ccoc3)CCCC(C1)OC2 N1(C(c2n(C(C)C)ncc2)=O)CC2CCCC(N(C)C(C3OCCCO3)=O)C2C1 C#Cc1cnn(CC2CC2C(=O)NCC2C3CN(C(c4cnc(Cl)s4)=O)CC23)c1 N1(C(C2CC(C#N)C2)=O)CCN(C(C2CC3C=CC2O3)=O)C(C2CCCC2)C1 c1(C(=O)NC2C(CNC(CSCCC#N)=O)C2)coc2c1C(=O)NCCC2 N1(C(c2cn(CC(C)O)c(=O)cc2)=O)CC(NC(=O)CC#N)C(C2CC2)C1 C1(O)(C(CNC(COC)=O)C)CCN(C(c2ccoc2Cl)=O)C1 N1(C(C2(CC)CC2(F)F)=O)CCC2CN(C(=O)C(C)(C)C3CCCO3)CC2CC1 C1(SCC(N2CCC(CC(C)C(=O)O)CC2)=O)CCc2ccccc2C1 C(c1ccccc1F)=CC(=O)NCC(N(C(=O)C(=O)NC1CC1)C)C1CC1 Cc1cc(C(=O)N(C(C)CN(C(=O)CCCc2cc[nH]n2)C)C)sc1C c1(C(=O)NC2CCN(C(C(CC)CC(C)C)=O)C2(C)C)ccc2cnccc2n1 O(NC(=O)C(C)NC(=O)CCc1nc[nH]n1)C(C(=O)OC)C C=CC(C)(C)CC(=O)N(C1CCCC(CNC(c2c(C3CC3)noc2C)=O)C1)C N1(CCCNC(C2CC3(CCC3)C2)=O)CCN(C(c2cc(C(N)=O)[nH]n2)=O)CC1 c1(-c2cc(C(=O)NCCOC)on2)cc(F)cc(F)c1.C12(CCCC1)C(=O)N2 C1(C#N)(OC)CC(NCC2CC(=O)N(C3CN(C(=O)CCCF)C3)C2)C1 c1(C(N(CC(C)N(C(CSCCOC)=O)C)C)=O)nnc(O)nc1O c1(C(N2C(Cn3cnnc3)CC2)=O)cc(Cn2cc(CS(C)(=O)=O)nn2)ccn1 N1(CC(c2ccc(C)o2)=O)CCC(Cc2ncc(C(F)(F)F)[nH]2)CC1 N1(CC(C)(Cl)Cl)CCCCC1c1ccc(C(=O)Nc2ccccn2)cc1 N(C(=NCc1ccccc1Cl)NC1CCC(CC(=O)OC)CC1)C(CC)CC c1(CN2CC(O)(C(C)NC(=O)CC3CCOCC3)C2)c[nH]c2cccnc12 C(=O)(CS(=O)(=O)CC(F)(F)F)N1CCC(NC(C(CC)(C)C)=O)CC1C N1(C(c2c(C)nn(C)c2)=O)CC2(CC(C(=O)NOCc3cc(F)ccc3F)CO2)C1 CC(C)CCC(O)C(=O)NC1CCCC(CC(=O)NC2CCC3(CCC3)C2)C1 Cc1c(C(=O)NCC2CC3CN(C(=O)Cc4cnc[nH]4)CC23)sc2nnc(S)n12 C(CC1CC1)(C(=O)NCC(c1ccncc1)O)NC(CNC(CCC)=O)=O c1(SC)c(C(=O)N(CCCN(C)C)CCNC(C2CC3CCC3C2)=O)cnn1C CCCCCCC(CC)C(=O)NC1(CNC(=O)CCC#N)CCC(F)(F)CC1 C12(CCNC(C(C)NC=O)=O)CCC(C1)N(C(c1ccc(Cl)nc1O)=O)C2 C1(C=C)(C(=O)OCC)CCN(C(C2CC2(c2ccccc2)C)=O)CC1 c1(C(=O)NCC2(C)CCCN2C(=O)Cn2cccn2)ccnc2c(F)cccc12 c1(OC)ccc(C(C)C)cc1Cn1nc(Br)nc1C(C)NC(CO)CC(C)C CCCCCCC(C)C(=O)NC(C1CCCN1C(c1ccc(=NCC)[nH]c1)=O)C C1(NC(c2cn3c(n2)CCC3)=O)CCCCN(C(c2csc(Br)c2)=O)C1 N1(CCCNC(C2(CCC)CC2)=O)CCN(C(=O)CC(C)CC)CC1 C(=O)(C1=CC(C)CC1)NCC(CNC(c1ccc(N(CC=C)C)cc1)=O)O c1(C(=O)NC2(C)CN(C(=O)CCCc3nccs3)C2)cc[nH]c(=N)c1 c1(CCC)cc(C(=O)NCc2csc(CNC(c3cscc3CC)=O)n2)n(C)n1 C1(C(=O)NCCCCNC(C(C)NS(C)(=O)=O)=O)CC12CCCCC2 c1(C(=O)OC)cc(N2CC3C(CNC(=O)CCc4cnn[nH]4)C3C2)nc(C)n1 C(CC(C(C)(C)C)NC(=O)C(c1cncn1C)O)N(C)C(C1CCCNC1=O)=O N1(C(c2ccccc2)C(=O)N(CC(c2ccc(Cl)cc2)O)C)CCCCCC1 CC1(CNC(C2(CO)CC(F)(F)C2)=O)CN(C(=O)CCn2ccnn2)CCO1 c1(-n2cc(CNC(CN(C(c3ncc(C)nc3)=O)C)=O)nn2)ccc(Cl)cc1Cl C1(C#N)(C(=O)NCC(CNC(CC(C)CN(C)C)=O)(C)C)CCCOC1 C1(NC(C2N(CC)CCCC2)=O)CC2(CCC(CNC(=O)CN(C)C(C)=O)OC2)C1 C1(CNC(C(C)C)=O)CC(C(F)(F)F)CCN1C(c1cc[n+]([O-])cc1)=O c1(C(=O)NCC(C2CCOC2)NC(c2n(CC)ccc2)=O)nn(C)cc1[N+](=O)[O-] c12cc(ccn1)O2.c1(C2N(CC)CC2)ccc(-n2cc(-c3cn[nH]c3)nn2)cc1 C(=O)(CC(O)C(C)(C)C)NCC(CNC(C1CCN(CC(C)C)CC1)=O)C C(=O)(C(C)CC(=O)OC)NC1(C)CC(C(=O)NC(CC#CC)CO)C1 C(=O)(C1c2c[nH]nc2CCC1C)NCC1(F)CN(C(C(C)=C2CCCC2)=O)C1 N1(Cc2ccc(N(C)C)cn2)CCCC(CO)(NC(c2cc(F)n(C)n2)=O)C1 c1(OC)cc(F)ccc1C(N1CCCC(C)C1CNC(=O)Cc1ccsc1Cl)=O C1(CN(C)C(C23CCC(C2)C3)=O)CN(C(=O)CC2(C(F)F)CC2)CCO1 c1(NCCC(=O)N(CCNC(Cc2c(C)occ2)=O)C2CC2)cc(F)ccc1F C1(C(=O)NC2CC(CC=C)C2)(COC)CN(C(=O)CCNc2ncccn2)C1 CC(C)(C)CC(O)C(=O)NC1COCC1CNC(c1cc2n(c1)CCC2)=O c1(C(C)(F)F)cccc(C(N2CCOC(CNC(c3csc(C#N)c3)=O)C2)=O)c1 c1(C(=O)NCCN(C(=O)CC2SC(=N)NC2=O)CC)cc(C)cc(OC)c1C c1(C(N2C(CC)C(NC(=O)CCNC(C)=O)CCC2)=O)cc(OC)c(Br)cc1C Cc1ccc(-c2ccc(C(N3CCCC3c3ccncc3C)=O)o2)cc1 C(CCC(C(=O)NCc1cc(C)no1)NC(=O)CC1CCCCCC1)OC N1(C(CSCCCC)=O)CCN(C(=O)C=CCCc2ccccc2)CC1C(F)F c1(NC(C2CCC(Nc3c(F)cnc(C)n3)C2)=O)cc(F)c(Cl)cc1F N1(C(c2cc(CC)on2)=O)CC2CC(C1)N(C(c1ccccc1CC)=O)C2 N1(C(COCCOC)=O)CCCC(C2CN(C(=O)C(F)(F)c3ccccn3)C2)C1 C1(CNC(C(C)(C)n2cnnn2)=O)CC2(CO1)CN(C(C1CCC1(F)F)=O)C2 c1(OCC=C)nc(N2CCC(OCC3CCCO3)CC2)nc2c1CSC2 C1(C(N(CC)CC2CC2)=O)CC2(CC(NC(c3ccc(I)o3)=O)C2)C1.CC c1(C(N2CC(NC(CC(CC)SC)=O)C(C)(C)CC2)=O)cccc2[nH]cc(Cl)c12 c1(C(=O)NC(CNC(COCC(=O)OC)=O)C)cc(C)ccc1NC1CCCC1 C=CCCCC(C(=O)N1CC(OCC(N)=O)C1)NC(C1CN(C)C(=O)N1)=O N1(C(CCCOC)=O)CCN(C(c2ccnn2COC)=O)C2CCCCC2C1 C(CCC(O)CO)NC(CN(C(CNC(=O)NC)=O)CC1CC1)=O C(c1c(F)cccc1F)=CC(=O)NCC1(O)CC(NC(c2cnn[nH]2)=O)C1 C1(CC#C)(C(=O)NCCC(C(=O)NC2CCNC(=O)C2)OC)CCCCC1 CC(CO)C(=O)NCC(O)CN(C(=O)CC(c1cccs1)n1cccc1)C C(=O)(CC(C(F)F)C(C)(C)C)N1CC(C)N(C(C2OCCO2)=O)CC1 N1(C(c2c(N)csc2)=O)CC(NC(c2ccc3n[nH]cc3c2)=O)C2CCCCC12 N1(C(C2(c3cccc(-c4ccc(C)cc4C#N)c3)CC2)=O)CCCC2(CCCC2)C1 C1(NC(CCC(=C)C)=O)CC2CCC(C1)N2CCNC(C1CC1CCC)=O C1(NC(C(C(C)C)CO)=O)CN(C(c2ncccc2F)=O)CCC12CCOCC2 c1(C(=O)OC)oc(C(=O)OCC(=O)NC(c2ccccc2)C#N)nc1C N1(C(c2cnc(C)s2)=O)CC(NC(C23C=CC(CC2)C3)=O)C(O)C1 O=C1NCc2ccc(C(=O)NCCS(=O)(=O)Cc3cn(CC4CC4)nn3)cc2N1 c1(CCC(C)NC(CNS(Cc2cccc(OC)c2)(=O)=O)=O)ccc(Br)cc1C c1(C(C)(C)C)cc[nH]c(=NCCC2CCC(NC(C3(O)CCOC3)=O)C2)n1 CCC(CC(=O)N1CCCC(C)(C(=O)NC(CC)C(=O)NC(C)C)C1)C(C)(C)C CCN=C(NCCF)NCC(c1ncc(C)s1)C.n1(CC)cccn1 c1(OC)c(C)nc(C2CC2)[nH]c1=NC1CN(C(C2(C)CC2(F)Cl)=O)CC1O N(C1COc2ccc(F)cc21)C(c1cncc(N)n1)=O C1(CNC(CC(C)N2CCCC2)=O)CC(F)CN1C(=O)Cc1cc[nH]n1 CC(C)(C(=O)NCC(O)CC(=O)N1CC2CC2C1)C(F)(F)F C1(N(C2CCN(C(=O)C(=O)NCC)C2)C(=O)C2CC2)CCCC(OC)C1 C1(CNC(=O)CCC2CCC2)CC(O)C(O)CC1C(N1CC(O)(CO)C1)=O CC(C)(CCCCNC(C1(C(O)C(F)(F)F)CCC1)=O)NC(c1c[nH]ccc1=N)=O C1(NC(C(C)OCC#C)=O)CN(C(c2cc(C)cc(C)c2O)=O)CC2(CCC2)C1 c1(NC(CC2N(C(C3CCN(C)C3)=O)CCCC2)=O)ccc(Br)c(F)c1F C1(C(N2CCC(OCC(NOCC(=O)OC)=O)C2)=O)C2CCC(C2)C1C c1(C(N(CCCCCCNC(C2CC=CCC2)=O)C)=O)ccn2cccc2c1 S(=O)(=O)(c1cc(Br)ccc1Cl)N1CC2(C(C(=O)Nc3nc(C)c(Cl)nc3)C2)C1 C12(NC(C=C(CC)CC)=O)CCC(CNC(c3ccc(C)o3)=O)(C1)OC2 c1(CC(=O)NC2CCCN(C(c3occc3Cl)=O)C2)cccc2nsnc12 Cc1cc2ncc(C(=O)NCC(O)CNC(=O)C(C)N(C)C)cn2n1 S(=O)(=O)(c1cnc(Cl)nc1)NC1CCN(C(c2cc3ccccc3o2)=O)CC1F c1(C2C(C(=O)NC3(CNC(CCCOC)=O)CCC3)C2)ccc(Cl)c([N+](=O)[O-])c1 C1(CNC(c2n(CC)ccc2)=O)CCCCN(C(c2c(C)ncn2O)=O)C1 C1(OC)CC(CNC(=O)Cc2ccncc2C)N(C(=O)CSCC2CCCO2)C1 C(N=c1[nH]c(N2CCC(F)C2)nc2cc(C(F)(F)F)ccc12)c1n(C(C)C)cnn1 N1(C(CCCC(=O)OCC)=O)CCCC2(NC(=O)CCc3ccccc3)CC2C1 CC(C)CC(C(=O)NC1CCN(C)C1(C)C)ONC(c1c(F)cncc1F)=O N1(C(c2c(OC)csc2)=O)CCc2sccc2C1CNC(C1(O)CCSC1)=O N1(C(CC=C=C)=O)CCC2(CCN(C(=O)CCCC(C)CC)C2)C1 C(=O)(C(F)C(C)CNC(c1cn(CC)nc1C)=O)NC(CCC=C)C N1(C(C2(CCCC)CC2)=O)CC(NCc2cc(C)cnn2)CC(C)(C)C1 N1(C(C(=O)NC23CC(NC(c4csc(-c5ccccc5)c4)=O)(C2)C3)=O)CCCC1CO Nc1cc(F)cc(F)c1C(N1CCCCC(NC(=O)C(F)(F)c2cccnc2)C1)=O c1(OC)ccc(C(=O)NCc2csc(CNC(=O)CCNS(C)(=O)=O)n2)c(C)c1 C(N=c1nc(N2CCC(C)(F)C2)c2c([nH]1)CCCC2)c1c(CCC)nns1 CCCCCCC(C(=O)OCC)NC(=O)CC1(C)CCOCC1.C(C)(C)(C)C(=O)O C1(OC)(CNC(=O)C(C)OC2CCOC2)CN(C(=O)C=CI)C1 CCCC(CC1CCCC1)C(=O)N1CC(C(C)(C)C)CC(CNC(=O)CSC)C1 CCCC(C#N)C(=O)NCCNC(C1CC(O)(C(F)(F)F)C1)=O N(C1CC2(CN(C(c3cc(C)c(O)c(N)c3)=O)C2)n2ccnc21)C(CCOC)=O c1(C(N2CC3C(NC(C4CCCCC(=O)N4)=O)C(C3)C2)=O)ccc2ccsc2c1 CC1c2ncc(C(=O)Nc3cccc4c3OCC4)n2CCN1C(=O)CO CC1=C(C(=O)NCC(C)N(c2nnccc2C#N)C)Cn2ncnc2N1C c1(N2CC(O)(C(C)NC(CC(CCC)(C)O)=O)C2)c([N+](=O)[O-])c(CC)nn1C C(c1ccc(N(c2ccccn2)C(=O)CSN2CCOCC2=O)cc1)=CC(=O)O C1(NC(C2C(OCC)C2C)=O)C(C)CCN(C(=O)COc2ccsn2)C1C C1(N(C(c2c(C)cnnc2)=O)C)CN(C(=O)C2=NNC(=O)C2)CCC1C N1(CC(=O)N(C)CC2N(C(CCC(CC)O)=O)CCC2)C(=O)CC(C)(C)C1=O c1(C(=O)NCC2CN(C(C3CC4(CC4)C3)=O)CC2(F)F)n[nH]c2cc(Cl)ccc12 C1(CC(C)NC(=O)CNC(=O)C(C)(C)C)CCN(C(C2CC(C(C)(C)C)C2)=O)CC1 Cc1cnc2n1CC(C(N1CC=C(CNC(=O)C(F)(F)C(F)(F)F)CC1)=O)CC2 C1(OC)CC(CNC(=O)CCc2ncco2)N(C(=O)CSC2CCCCO2)C1 N1(C(c2csc3ccccc23)=O)CC2CCCC(C1)N2Cc1c(I)ccnc1F c1(C(N(C2CCCC2)CCNC(COCCN(C)C)=O)=O)cnn(C)c1C(F)(F)F CCCCC(CNC(C1(C)CCCO1)=O)NC(c1coc(OCC)n1)=O N1(CC(=O)N(C)CC)CCC(O)(C(C)NC(c2cc(-c3ccccc3)no2)=O)C1 C1(N(C)C(c2ccc(F)cc2)=O)CCCN(C(=O)C=CCN2CCCC2)CC1 N1(C(C=Cc2cncc(C)c2)=O)CCN(C(=O)CC2(C)OCCO2)CC2(CC2)C1 c1(NC)cnccc1C(N1CCCC(N(C(=O)CC2CCCC(=O)N2)C)C1)=O Cc1nc(C(=O)N(C2CCCN(C(C3CN(C4CCC4)C3)=O)C2)C)c(=O)[nH]c1C C1(NC(C(C(C)C)O)=O)CN(C(=O)CCn2cnnn2)CC2(CCOCC2)C1 C(=O)(C1Cc2ccccc21)NCC1CN(C(CCCN(C(=O)OC)C)=O)CC1O c1(C(N(CCCN(C)C)CCNC(C(C2CC2)OC)=O)=O)cn(C)c(=O)nc1O c1(OC)cc(C(F)(F)F)ccc1C(N1CC2CN(C(c3cncc(O)c3)=O)C2C1)=O N1(c2nc(C)c(Cl)cc2Cl)CCCC(C2CC2NC(=O)C(C2CCCCC2)F)C1 c1(C(C)C)cc(C(=O)NC(C2CCCC(c3ccccc3)O2)C2CC2)n(C)n1 O=C1CC(C(=O)NC2CN(C(=O)Cc3ccsc3)CC2C(F)F)=NN1 N1(C(c2cc(C)[nH]c2C)=O)CCCC12CCN(C(=O)CSC)C2.c1(C(=O)N)cscn1 C(CC(N)=O)(C(=O)NCCCC1CCC1)NC(C(CCC)NC(N)=O)=O N1(C=O)CCC(C(=O)OC)C(O)C1.C#Cc1nc(C2CC(N3CCOCC3)C2)cs1 C1(O)(Cn2cc(C(C)NC)nn2)CCN(C(=O)C(F)CC2CCC2)CC1 CCCC(C(=O)NCC(O)C1(Cl)CC1)NC(C1CCOC1C(C)C)=O c1(CC)noc(CC)c1CC(=O)N(CCCCN(C(=O)CCCCN(C)C)C)C Cc1nc(C)c(C(=O)NCC23CC(C2)C(NC(=O)CCC2CCCC2)CO3)s1 c1(CC)ccc(C(=O)NC(C)C(=O)NC2(C(O)CO)CC2)[nH]1 c1(C(N2CCC(C3N(C(CCCC)=O)CCCC3)C2)=O)cc(COC)nc(O)c1 C(=O)(C1COc2ccccc21)N1CCC(N(C(=O)C2=CCC2)CC)C1 N(C1CCc2cccc3cccc1c23)n1c(-c2c(C)cc(CO)s2)ncc1 C12=NC(=NCCOC3CCN1CC3)NC1=C2SCC1.CC(C)CCOC(F)F CCC(C)(C(=O)N1CCC(OCC2CC2)C1)NC(c1cccn1C)=O c1(C(=O)NC2C(C(=O)NCC(C)(C)CC3CC3)CCCC2)cnccc1C#N Cc1nn(C)c(F)c1C(=O)NC1CCN(C(C23CCC(C2)C3)=O)C(C)C1 N1(C(=O)CCC2OCCO2)CCN(C(C2CCCCS2)=O)C(CCO)C1 N1(C(C(=O)NCCC)C2CC(OC)C2)CCCC(n2cc(C(=O)OC)nn2)C1 c1(CC(N2C(C)(CNC(CCOC)=O)CCC2)=O)cccc(F)c1Cl C1(NC(C2CC(=C)C2)=O)CC1C1CCN(C(c2c[nH]c3cc(C)ccc23)=O)CC1 C1(NC(c2c(CCC)occ2)=O)CCC(CNC(C2CC3CC2C3)=O)CC1 C(=O)(C(C)(F)C(C)(C)F)NCC(=O)NC(C(=O)NCC(CC)OC)C(C)C c1(CC(=O)NCC(C)NC(C(c2ccc(F)cc2)OC)=O)ccccc1[N+](=O)[O-] Cc1cc(CCN=C(NCC2CCCO2)NCC23CC4CC2C3C4O)ccc1O C1(CC=C)(NC(=O)CCCOCC)CCN(C(c2cnn(CC(F)(F)F)n2)=O)C1 O=C1CC2(CCN(C(C3CC34CCNC4)=O)C2)CN1 C1(C(N(C)CC2CCCN2C(c2csnn2)=O)=O)CCn2c(O)nnc2C1 c1(C(N2CC3CCC2CN3C(C23CCCC2OCC3)=O)=O)nc2cccnc2s1 N1(C(C(C)C2CCCO2)=O)CCC(O)(CNC(=O)CN2CCC(C)(C)C2)CC1 n1(CC(=O)NC2CC(NC(C(C3CC3)OC)=O)C2)cc(C(F)(F)F)nn1 N1(C(Cc2ccn(CC)n2)=O)CC(NC(c2cc(C)nc(C)c2)=O)CC(O)C1 c1(Nc2c(CSC)cccc2)cc(S(=O)(=O)NCC2CC2(F)F)ccc1C#N CN1CCN(C(c2ncccn2)=O)CC1C(N1CC(F)(CF)C1)=O c1(C(=O)NC(C)CCNC(C2(C(F)F)CCCO2)=O)nnc2ccccc2c1O C1(CNC(C(C)OCC#C)=O)CC(CNC(c2csc(C(C)C)n2)=O)CO1 c1(C(=O)NCCCNC(C(CO)N(C)C)=O)cc(C2CC2)nn1C C1(N(CCC)C(N2CCOCC2)=O)COCCC1N(CC(=O)NC1CCCC1)C c1(-c2nc(C(CCC)C)nn2C2(C)CC3(C2)CC3(F)F)cc2cccc(F)c2s1 c1(C2C(C(=O)OC(C)(C)C)C2)ccccc1Cl.c12ccoc1C(=O)N2 N1(C(C2CCC(N(C)C)C2)=O)CCN(C)CC1CNC(=O)C=CC(N)=O C1(C(=O)NC(CC)CSC)(OC)CCN(C(c2coc(Cl)n2)=O)CC1 c1(CCOCC(=O)NCC(C)CN(C(=O)CC(O)C2CCCC2)C)ccccc1 C(=O)(C(CC#CC)NC(c1[nH]nnc1C1CC1)=O)N1C(C=C)CC1 CC1(C)CC(NC(=O)C(C2CCCO2)NC(c2c[nH]c(C(N)=O)c2)=O)C2(CC2)C1 C1(NC(CCSCC)=O)COC2(CCN(C(c3ccc(CC)[nH]3)=O)C2)C1 c1(C(=O)NC23CC(C)(C2)OC3(C)C)cccc2c1nnn2C1CCCCC1 c1(OC)ccc(CC(=O)NC2(CN(C(=O)Cn3cc(C)cn3)C)CC2)c(Cl)c1 c1(C(N2CCC3(C(NC(COC4CCC(C)C4)=O)C3)C2)=O)cc2ccsc2n1C c1(CC(N2CCN(C(CCC=CC)=O)CC2C(F)F)=O)c(F)cccc1C#N CC(O)CC(=O)N(C(C)(C(=O)NCC1(C#N)CC1)C1CC1)C c1(OC)ccnc(C(N2CCC(F)C(NC(c3ccco3)=O)C2)=O)c1OC Cc1ncnc(C(=O)NCC(C2CCC2)NC(c2cccc(N(C)C)c2)=O)c1C c1(CC)onc(C(=O)NC(Cc2cc[nH]n2)C(=O)NCC(c2ccsc2)C)c1C C(=O)(CC(F)(F)C(C)C)N1CCC(N(C(C2CC(n3cccn3)C2)=O)CC)C1 c1(N(C(C)C)C)nnc(-c2ccoc2)n1CC1CCN(CC(F)(F)F)C1 c1(CC)ncc(C(=O)N(C2CCC(NC(C3(Br)CC3)=O)CC2)C)c(C)n1 C(CCN=c1[nH]c(Cl)ncc1C)OCCNC(c1c2cccc(C)c2sc1)=O c1(C(=O)NCC2CN(C(C3CCCCC3)=O)CCO2)cc2c(O)ncnc2cn1 N1(C(c2c(C)cn(C)c2)=O)CCN(C(c2ccoc2Br)=O)C2CCC12 C1(C#N)(C(N2CCC(N(C(C(C)c3ccsc3)=O)CCO)C2)=O)CC=CC1 c1(C)cncc(F)c1Cl.C1(OC)(CNC(=O)CC)CCN(C(=O)CC2CCOC2)C1 N1(C(c2c(OC)ccs2)=O)CCCCC(NC(=O)CC2CC(OC)C2)C1 C1(CC(=O)OC)CC2(CCN(C(c3sc(Br)cc3[N+](=O)[O-])=O)CC2)CO1 c1(CNC(N2CC(C(=O)N(CC)CC)C2)=O)ccc(NC(=O)CCC(C)C)cc1 C#CCC(C(=O)NCC1(O)CCN(C(c2ccc(C(C)C)s2)=O)C1)C1CC1 c1(-n2c(C)cnn2)ccc(C(=O)N(C2C3CN(C(=O)C4=CCC4)CC23)C)cc1 C(CO)(C(=O)NC1(C2CCCN2C(=O)CCc2nc(C)cs2)CC1)OC C1(N(C(=O)CSCc2ccccc2)C)CC2CCC(C1)N2C(=O)CC1(CO)CC1 c1(C(=O)NCC(C)CNC(=O)Cc2ccco2)cc(S(N)(=O)=O)ccn1 c1(CN2CC(F)(C(N3CCC(C(F)(F)F)C3)=O)C2)nc(Br)ccc1F C(CC(C)(C)CC(=O)N1CCC(O)C1C(=O)NCC1(SC)CC1)OC Cc1c(-n2cc(C3(F)CCN(C(c4ccc(C(C)C)o4)=O)C3)nn2)cccc1Br N1(C(COCCCCC)=O)CCC2(CC1)CC2C(N1CC2CC1CN2C)=O C=CC(CC)C(=O)NCCOC(C)(C)CNC(=O)C(CO)NC(N)=O C(=O)(C(O)CC(F)F)N1CCCC(N)C1.C(C(=O)NC1CC1)NC=O c1(OC)cc(OC)c(C(N2CC(NC(C3CC(C)(C)CO3)=O)C(O)C2)=O)cc1N Cn1c(C(N2C3CCC2C(CNC(=O)Cc2cccnc2)C3)=O)cc2sccc12 C12(CNC(c3nc(C)oc3)=O)COC(CNC(C3COCC(C)O3)=O)(C1)C2 C1(NC(CN(C)C)=O)CC2CC(NC(c3cc(SC(F)(F)F)c[nH]3)=O)C2C1 Cc1ncnc(C)c1C(N1CC(C(=O)Nc2cn(CCF)nc2C#N)C(F)C1)=O Cc1onc(C(=O)NCC(C)CNC(C2CC2C(C)(C)C)=O)c1[N+](=O)[O-] C#Cc1cnn(CC(=O)N(C2CCN(C(C3(c4ccc(F)cc4)CC3)=O)C2)C)c1 N1(C(CCC=CC)=O)C(C(=O)NCc2nn[nH]c2C2CC2)CC2CC12 N1(CCNC(C2CN(C(=O)CCc3cncc(O)c3)C2)=O)CC2CCC1C2 CC(C(C)(C)C(=O)N1CC(C(=O)NCC2CC2)C1)NC(=O)Cn1ccnn1 c1(N2CCC(NC(C3(CNC(C4CC4F)=O)CC3)=O)CC2)ccc2nncn2n1 C(=O)(C(O)C(F)F)NCC(C)(C)NC(c1ccc(SC(F)(F)F)cc1)=O c1(CN)ccccc1.C(CCCNC(=O)COCCO)N(C(=O)C=CCO)C c1(C(N2CC3CN(Cc4c(C(=O)OCC)n[nH]c4)C3C2)=O)ccc(C#N)c(F)c1 C(C)(CCCC(=O)NCc1nnc(O)n1C)NC(c1c(CC)nco1)=O C1(C(N2CCC(N(CCC)C(c3cn(C)c(O)n3)=O)C2)=O)CCCCNC1=O c1(C(N(C(C)CNC(c2cn(C3CCC3O)nn2)=O)C)=O)nc(Cl)sc1Cl C1(C(C(C)C)NC(CSC)=O)CCN(C(=O)CCSc2ccccc2Br)CC1 N1(C(C2C(C)(Br)C2)=O)CCCCC12CC(NC(c1ccc[n+]([O-])c1)=O)C2 C12(NC(c3c(C)cno3)=O)CCCC1N(C(=O)Cc1nn(C)cc1Cl)CCC2 O=C(C1=C(Cl)CCOC1)NCC12CCC(CC1)N2C(=O)CCc1ccc(F)cc1 c12cc3c1cccc3[nH]2.c1(C(=O)OCC2CCCCCO2)c(CO)cccc1Cl C12(C(=O)NC(C)CF)C(NC(=O)CC3CCC=CCC3)C3CC1C2C3 C1(N(C(=O)CC2CCCCC23CC3)CCO)CCN(C(=O)C=Cc2nccs2)CC1O C12(C(N3CC(O)(CNC(c4nccc(C)c4N)=O)C3)=O)CC3CC(C(=O)N1)C2C3 C1(C(C)SCCOC)CCN(c2ccccc2)CC1.C1(SC)CCOC1 Nc1cnc(C(N2CC3(C2)CN(C(=O)CN2CCSCC2)C3)=O)c(Cl)c1 C(C)(CC(C)N=c1ccnc(CO)[nH]1)NC(c1ccc(N(CCC)CC)cc1)=O c1(NC(C2C3CCCC2N(Cc2cncs2)C3)=O)c(F)cc(CO)cc1Cl N1(C(CC2(COC)CCCC2)=O)CCN(C(=O)CCc2cc(Cl)no2)C2CC12 c1(C(c2nnnn2C2CCC2)NCC(COCC)C)ccc(CC2CC2)o1 c1(C(N2CC(NC(c3cc(CC)on3)=O)C(F)C2)=O)cc2ccccc2cc1Cl N1(C(Cc2ccc(SC)cc2)=O)CC2(CCCC2n2cc(C(=O)NC3CC3)nn2)C1 CCCCC(C)CCC(=O)NCCCNC(c1ncnc(OC)c1F)=O c1(C(N2CCC(C#N)(NC(c3cnccc3Br)=O)C2)=O)cc(Br)cc([N+](=O)[O-])c1O N1(C(c2cc(C)cc([N+](=O)[O-])c2)=O)CCCCC(N=c2ccc(C#N)n[nH]2)C1 C(=O)(CC(C)(C)CC(F)F)NC1CN(C(CC2CCCC(C)O2)=O)CC1N=[N+]=[N-] c1(C(N2CCC(NCCCCCC)C2C)C(=O)NCCCF)c(Br)c(C)nn1C C(=O)(C(=O)CC(C)CC)N1CC(C(C(=O)N(C2CC(=C)C2)C)O)C1 C1(NC(CSC)=O)CC(OC)CN(C(c2c(OCC(=O)OC)c[nH]c2C)=O)C1.C(C)=O C(C(=O)NCC1CC(F)CN1C(=O)C(C)C1CCC1)(C(C)C)NC(C)=O CC1CC(NC(C2(CF)CCC2)=O)CN(C(c2c[nH]nc2[N+](=O)[O-])=O)C1 c1(C(N2C(CN(C(=O)CSc3nncs3)C)CCC2)=O)ccn2nncc2c1 C1(CCNC(C2CCC(C(=O)OC)C2)=O)CN(C(=O)C=Cc2cc[nH]n2)CCO1 N1(C(C(CC)NC(=O)CN(C)C2CC2)=O)CC2CCN(C(=O)CCSC)CC12 CC1CC(N=c2[nH]c3c(c(=NCc4ncn(C)n4)[nH]2)CCCCC3)C1 N1(C(COCCCCOC)=O)CC2CCC(C1)N(C(=O)CCC(F)(F)C(F)F)C2 CC1CCCCC1(CNc1ncc(C(F)F)cn1)NC(C1COC(C)(C)C1)=O C1(N)CCC2(CCC2)C1O.c12ccc(cc1)CNC(=S)N2.CC(C)O N1(C(C2N(Cc3cn(C)nn3)CCC2O)=O)CCC2(CC1)CN(C)C2 c1(CN2CC(NC(c3cnc(Br)o3)=O)C(F)C2)cccc2cc[nH]c12 c1(OC)ccc(CCN2CCCC2Cc2ccccc2)c(Cl)c1OC c1(C(=O)NC2(CNC(C(c3cnn(C)c3)C)=O)CCC2)ccc(N)cc1Cl C1(CNC(C2CCN(C(C)=O)C2)=O)(CO)CCN(C(=O)Cn2cccn2)C1 C1(CC(=O)NCC2(NC(=O)Cc3cccc(Cl)c3)CC2)CC2(CCC2)C1 N1(C(c2ccn(C)c2)=O)C2CCC1CN(C(=O)CC1CCCCC1(C)C)C2 C#CCC(CC(=O)N1CCC1C1CCOCC1)NC(C1(C)COC(=O)N1)=O CC1(C(N2CCC2(C)CC(=O)NC2CC3CCC2O3)=O)COC(=O)N1 c1(CCCC(=O)NCC2(NC(c3c(C)nsc3)=O)CCC2)ccc(F)cc1 C(CC(C)CCNC(=O)C=Cc1csc(C(F)(F)F)c1)NC(c1n(CC)ccc1)=O C1(NC(CC(CCC)O)=O)CN(C(c2ccc(C)s2)=O)C2(CCCCC2)C1 CCC1=C(C(=O)NCC2(n3cccn3)CCN(C(C3CC3F)=O)CC2)SCCO1 N1(C(CC=C(C)C)=O)CC2CCC1C1CN(C(c3cnnc(O)c3)=O)CC21 Cc1ccc(NC(C)C(N2CCC(O)(CCNC(=O)CC(C)F)C2)=O)cc1OC c1(NC(C(C)N(C(C(CCCC)C)=O)C2CCCC2)=O)cnc2ncnn2c1 N1(N(C2CC2C(F)(F)F)C)CCOC(CS(=O)(=O)[N-])C1 CC1(C)Nc2ccccc2C1NCc1ccccc1C(O)C(F)F Cc1cn2c(C(=O)NCC(C)N(C(=O)CCC3CC3C)C)cnc2s1 C1(C)(CC)CC(C(=O)NCC(C2CCCC2)NC(C2CCCO2)=O)CCO1 Cc1cccc2cc(C(N3CC(NC(=O)C(=O)NC4CC4)CC3C)=O)nn12 C(c1cnccc1C)=CC(=O)NCC(CNC(C(C)SCC)=O)(C)F CCCC(CCCNC(c1cnc(S)[nH]1)=O)NC(c1occc1C(C)C)=O c1(CN2CCN(CCCCCC)CC2)cc2c(Cl)c(OC)ccc2[nH]1 c1(C(=O)NC2C(CNC(c3cnn4c3CCCN4)=O)C2)c[nH]c(=O)c2ccnn12 C1(C(=O)NC2C(=O)NC(C(=O)OCC)C2)CCCC12CCC2.c1cnc[nH]1 C1(C(=O)NCCC(C)NC(C2SCCCS2)=O)CC2C(C1)C2(C)C O=C(C1OCCc2ccc(Br)cc21)N1CC(C2CC2)(c2nn[nH]n2)C1 c1(OC)cc(C(N)C(=O)N(C(C)C(=O)Nc2ccccc2)C)cc(OC)c1OC C(=O)(C(C(=O)NC(CC1CC1)CC(=O)N(C)Cc1cccc(O)n1)OC)OC C(=O)(C1=CCN(C(C2(C3CC3)CCC2)=O)C1)NC1C(C)(C)C(O)C1 c1(C(N2CC(C)(CCC(=O)NC(C)CO)C2)=O)ccc(C#N)cn1 C1(NC(=O)CC2COCCO2)COC2(C1)CN(C(c1ccc(O)c(F)c1)=O)C2 C(C)(C(C)S(C)(=O)=O)Sc1cn(SC(CC(=O)OC)CCc2ccccc2)nn1 c1(NC(N(CCCC)C(c2ccccc2C)C)=O)ccccc1C(F)(F)F CCC(CN=C(NC1CCCC1)N1CCC2(C1)CC2(F)F)C(C)(F)F C1(NC(C2(COCC)CCC2)=O)CS(=O)(=O)CC1NC(c1cc(C)[nH]n1)=O C1(CNC(CC2(OC)CCC2)=O)(NC(C2CCNC2=O)=O)CC2CCC1CC2 Cc1nccc(C(=O)NCC(CC(C)C)NC(=O)CCC(C)(F)F)c1O C1(CCNC(C2(C(C)=O)CC2)=O)CN(C(=O)Cc2ncccc2C)CC1C N1(C(c2cnc(OC)nc2)=O)CCC2(C(=O)NC3(C)CC3)CC2C1 c1(C(N2CC(C)(NC(C3CC(C(=O)OC)C3)=O)C2)=O)cnc(S(C)(=O)=O)s1 N#Cc1cncc(C(N2CCCN(C(c3ccc(Cl)nc3)=O)CC2)=O)c1 C=CC(O)C(=O)NC(CO)C(=O)NC1(CN(C)C)CCCC1 c1(OCC)cccc(CCC(=O)NCC2CN(C(C3CC3(Cl)Cl)=O)C3CC23)c1 C1(NC(C2(CCCC)CCC2)=O)CCCCC1CNC(C1(C)CC2CC2C1)=O N1(C(c2c(CC)nns2)=O)CCCCC1CNC(C1(C)CCCS1)=O C1(C(N2CCC(CCNC(C(CC=C)CC)=O)CC2)=O)CCn2nccc2C1 c1(C(=O)NC2CCC(CCNC(c3cnc(C)[nH]3)=O)C2)nncc2c1CCCC2 C(=O)(C(CNC(c1cncc(C)n1)=O)C(C)(C)C)N(CC(COCC)O)C C(=O)(CC(C)NC(c1c[nH]c(=N)o1)=O)NCC(n1ccnn1)C CC1CCOC(C(=O)NCC(CC2CC2)C(=O)NC2(C(O)CO)CCC2)C1 C1(NC(c2cc(C)oc2C)=O)CC1C1CCN(C(=O)C(C2CC2)N(C)C)CC1 c1(NC(C2N(C(C3(C)CCN(C(C)=O)C3)=O)CCC2)=O)ccc2cccnc2c1 c1(C(=O)NC(C2CN(C(c3cc(Cl)cs3)=O)CCO2)C)ccc2ncsc2c1 C(N=c1cc(C2CC2)nc(Cl)[nH]1)C1C(NC(C(C)(C)CF)=O)CCCC1 N1(C(C2CCCS2)=O)CCC2(CCN(Cc3cccc(Cl)c3[N+](=O)[O-])C2)C1 N1(C(C(CSC)C)=O)CCCC(C2CCN(C(c3cnc(C4CC4)[nH]3)=O)C2)C1 C1(C)(CC(=O)NC(C(C)C)C(=O)OC(=O)C(F)(F)F)COc2ccccc21 C1(NC(CCOCCCNC(Cn2c(C)ccn2)=O)=O)CC2CCC1CC2(C)O c1(C(c2nnnn2CC(F)F)NCC2CC(CO)C2)cc[nH]c1-c1ccccc1 CP(C)(=O)C1CCCCN1C(=O)CC1(CC2CC2)CC1 N1(C(c2cnn(C)c2N)=O)CC(NC(c2csc(C3CC3)n2)=O)CC(C)(C)C1 Cc1nc(Cl)cc(Cl)c1C(N1C2CC1CN(C(=O)Cc1cnc[nH]1)C2)=O N12CC3CCC(C1)N3C(=O)C1(CCC1)CC2=O.c1(OC)ccc(C(F)(F)F)nc1 N1(C(C(CN(C)C)NC(C(C(C)O)N(C)C)=O)=O)CCC12CC(O)C2 c1(C(=O)NC(CC(=C)Cl)C(=O)N2CCC(C(F)F)C2)nccc2[nH]ccc12 Cc1cc(C(N2CC3CC2C3NC(C23CCOC(C)(C2)C3)=O)=O)c2c(c1)CCO2 c1(C(=O)NC2(C)CN(C(CCCC#C)=O)C2)c(C(F)(F)F)nn2ccccc12 C1(C(=O)NCC(CN(C(=O)CCc2ccc(CO)o2)C)(C)C)CCCC(C#N)C1 c1(C(=O)NC(Cn2cc(COCC)nn2)C)ccc(-c2ccco2)nc1 CCC(CCCC(=O)N1CCCCC1C(F)F)NC(C1CCN(CC)C1)=O c1(CC2N(C(=O)CC3C(F)(F)C34CC4)CCCC2)cccc(Cl)c1Cl CCC(CC)CC(F)C(=O)NCCOC(C(=O)N(CC(=O)OC)C)C(=O)OC CC(O)(CC(=O)NC1(CO)CN(C(c2ccsc2)=O)C1)C(=O)OCc1ccccc1 Nc1cc2c(cc1C(N1CC3CC1CN(C(=O)C=C1CCCCC1)C3)=O)OCO2 C1(OC)CCC2CC2C1.C12(C(=O)OC)CN(C1)C(C1CC1)c1cn2nn1 CN1CC(OCCS)C1C(=O)NC1CN(C(=O)C(O)Cc2ccccc2)C1 C1(CC)CCN(C(C2CCC2CNC(=O)COC2CC2)=O)CC1 c1(C(=O)NCC2(C)CCCN2C(=O)COCC2CCCO2)cc(=O)cc(Cl)[nH]1 c1(OC)c(C(=O)OC(C)C(=O)NO)cc(Cl)cc1C c1(C(=O)NCC2CCCN(c3snc(C)n3)C2)cnc2c(c1)NC(=O)CN2 C1(CC)CN(C(c2cc(C)nc(C)c2)=O)CCC1CNC(=O)C(O)C(C)C C1(NC(c2nc(C)oc2)=O)CN(C(C2(C(N)=O)CCC2)=O)CC1C1CC1 C(C)(C(CC(=O)N(C(C)C)CC1CC1)NC(=O)CC1CCOC1C)OC Cc1cc2c(C(=O)N(CCCCNC(c3cc(O)nc(C)n3)=O)C)nccn2n1 Cc1ncc(Cl)c(C(N2CCC(NC(=O)Cc3cc(F)ccc3O)C2)=O)n1 C1(C(N(C(CNC(COCCCC)=O)CC)C)=O)CCCCN1C c1(Oc2ccc(NC(=O)Nc3csnn3)cc2)ccc(Cl)cc1Cl c1(CN=C(NC(C)CC2(CCC)CCC2)NC2CCOCC2)ccccc1 C1(NC(=O)C=C2CCOCC2)CCCC1NC(=O)CCOCCN(C)C n1(CC(N2CC(NC(CSCCOC)=O)C(C)CC2)=O)cnc2sccc2c1=O C1(C(N2CC(CCCCC)C2)=O)COCCC1NC(c1cc(OCC)ns1)=O C1(C(N2CCCC(C(=O)OCC)C2)=O)CN(CCCN)CCC1(F)F N1(C(CNC(CC)=O)=O)CCOC(CC(N2CCC(F)(CF)C2)=O)C1 N1(C(c2nc(CCC)oc2)=O)CC(NC(c2cc(O)n(C)n2)=O)CC2(CCC2)C1 c1(C(C(=O)N(CCNC(c2c(CC)non2)=O)CCOC)O)cccc(OC)c1 C1(CCNC(C=NOC)=O)CN(C(C2CC3(CC(C)=NO3)C2)=O)CCS1(=O)=O c1(C(=O)NC2CN(C(C(C3CC3)OC)=O)CC2C)ccnc2c1ncn2C C12(NC(COC(CC)(C)C)=O)CCCCC1N(C(c1c[nH]c(=N)o1)=O)CC2 CC1CCC(NC(=O)COc2ccc(Cl)cc2)CN1C(c1csc2nccn12)=O N1(C(CCC2C(C)(C)C2)=O)C(C(=O)NC2CC3CCC2O3)CCC12CC2 Cc1nc(=NC(=O)CSC(F)(F)F)n(-c2ccc3ccccc3c2)[nH]1 N1(c2ccnc(C(C)(C)C)n2)C2CCC1CC(OC)C2.C12=CC=C(C=C1F)C2=O c1(C2(C(N3CCCC(C(C)=O)C3)=O)CCC2)ncc(F)cn1 N1(C(C2CC(=C3CCC3)C2)=O)CC2C(CNC(C3CCC4(CCC4)C3)=O)C2C1 c1(N(C)C)cncc(C(=O)NC2CCCC(NC(C3(C)CSC3)=O)C2)n1 N1(CCCNC(CCCc2cc(C)no2)=O)CCN(C(=O)C(C)N(C)C)CC1 CON=CC(=O)NC1(C2CCCN2C(=O)CSc2n[nH]c(C)n2)CC1 C1(C(=O)NCC2C(NC(c3c(NCC)scn3)=O)C2)CC12CC(C)(C)C2 n1(CC(=O)NC2C(CNC(c3c(C(C)(C)C)con3)=O)CCC2)cc(C#N)cn1 CC(C)C(C)(O)C(=O)NC1CC(O)C1CC(N1CCC(O)(CCC)CC1)=O C1(COC)(CNC(=O)CCc2cn[nH]c2)CN(C(=O)COC2CC(F)(F)C2)C1 C(=O)(CC(F)(F)CS(C)(=O)=O)N1CC(C)C(CNC(=O)CC23CC(C2)C3)C1 Cc1ccc(C(N2CCCC(N(C(=O)CCC3CCOC3)C)CC2)=O)cc1C N1(C(C=CC)=O)CCC2(CCCCN(C(c3cnc(Cl)c(C4CC4)c3)=O)C2)C1 C1(C(=O)OCC)C(C(=O)OCC)C2CCC1N2C(C1(CC)CNC1)=O N1(C(CN(C)CC)=O)CCCC(C)C1CNC(c1sccc1Br)=O CC1=CCN(C(=O)C(c2ccccc2)C2CC2)CC1.C12CN(C1)C(=O)CO2 C1(C(=O)NC(C2(O)CCCN(C(c3ccsc3)=O)C2)C)CN(CP(C)(C)=O)C1 c1(-c2cc[nH]n2)cnccc1-c1cnn(C2CCOC2)c1 C1(C(N2C(CN(C(=O)CC3CCCN(C)C3)C)CCC2)=O)CC2CCC(C1)O2 c1(C(=O)NCC(C)NC(c2cc(CC)c(F)cc2)=O)ccc2c(=N)[nH]cnc2c1 c1(-n2c(C(O)C3CC3)nc(CC)n2)ccc(F)cc1OC c1(C(=O)NC2(C(=O)NCC(CO)OC)CC2(C)C)ncc(N)cc1C C#Cc1cnn(C)c1C(=O)NCC1(CNC(C2(CC(C)C)CCNC2=O)=O)CC1 C12(C(N3CC(CNC(=O)CCc4ccncn4)C(O)C3)=O)COCC1C2(F)F c1(C(=O)NC)ccc(NC(C2CC23CN(Cc2c(Br)cnn2C)C3)=O)cc1 c1(CC)nc(C)oc1C(=O)N(C1CN(C(C2(C)CC2(F)F)=O)C1)C c1(N2CC(c3ccccc3)(NC(=O)Cc3ncccn3)C2)cnc(C2CC2)cn1 CC(C)C(C)(CNC(=O)CC1(CO)CC1)NC(c1cn(C(C)(C)C)nn1)=O N1(C(C2CCC(CC)CC2)=O)C2CCC1CN(C(C1C3CCC4C(C3)CC14)=O)C2 NS(=O)(=O)C1(C(=O)N(CCNC(c2ccc(O)nc2)=O)C2CC2)CC1 C1(NC(CCCc2n[nH]c(=N)s2)=O)C2CCC1N(C(c1cnn(C(F)F)c1)=O)C2 C(=O)(C1CCCc2ccnn21)NCC1CN(C(C2CC(=C)C2)=O)CC12CC2 N1(CC(=O)NCCCN(C(=O)C(C)Cn2ccc(C)n2)CC)CCc2sccc2C1 c1(C(C(=O)NCCNC(C=CC(=O)N(C)C)=O)C2CCCC2)cccnc1 c1(CNC(C23CCC(NC4CC4(F)F)(CC2)CC3)=O)cccc2c1OCCC2 Cc1ccc(CC(=O)NCCN(CCCN(C)C)C(=O)CC2(C)CC2(F)F)cc1O C1(C(C)NC(c2cocn2)=O)CCN(CCN2CCC2=O)CC1 CC1CN(C(c2ccc(C(N)=O)cc2F)=O)CCCC1NC(=O)Cc1cnns1 N1(C(c2cc(OC)n[nH]2)=O)CCC(C(=O)Nc2cn(C)nc2C(C)C)C1C c1(NC(=O)NCC2(N(C)C)CCSC2)c(I)cnc(Cl)c1F N#CC12C3C4C1C1C2C3C41C(=O)NCC(C1CC1)NC(C1(SC)CC1)=O N1(CCCC(N(C(C)C(=O)NC(C)(C)C2CCC2)C2CC2)=O)CCCCC1=O c1(C(=O)NCC(CNC(=O)CN2CCC(O)CC2)F)cnn2c1CCC2 c1(N2CCCC(CNC(C3C(C)(CC)C3)=O)C2)nc(Cl)ncc1OC c1(C(=O)NC2(CC=C)CN(C(=O)C=Cc3cccnc3)C2)ccc(CSC)cn1 c1(C(=O)NCC2CC(NC(c3cc[nH]n3)=O)C2)oc2ccccc2c1Br C1(CNC(CCc2ccc(C)cc2)=O)CC2CC1CN2C(=O)Cn1nnc(=O)[nH]1 N1(C(C2C(CC)C2)=O)CC(N(C(=O)CN(C(=O)COc2ccccc2)C)C)C(O)C1 CCCC1C(=O)N1.C1(CC(C)OC(C)=O)CCN(C(=O)C(C)OCC)CC1 C1(NC(C(c2scc(C)n2)C)=O)CCN(C(c2cn(CCO)nc2C)=O)C(C)C1 N1(C(Cc2c(C)nsc2)=O)CCOC(CCCNC(=O)COc2ccsc2Cl)C1 C1(CNC(C2CCCN(C(=O)C(=O)NC3CC3)CC2)=O)CN2CCCCC2CO1 N1(C(C(C)OCc2cccs2)=O)CC2CCCC(C1)N2C(C1CNC(=O)CC1C)=O c1(OC)cc(CN2CCCC2(C)C(=O)NC(C)CCO)cc(C(F)(F)F)n1 C12(NCCN(C)C)C3C4C5C3C1C5C24.C1(N)CCOC1.C1C(=O)NCCO1 C1(C(=O)NC(CC=CC)C(=O)NC(C)Cc2cn[nH]c2)CCCCC(=O)N1 c1(CC(CC)C)nc(C(O)CC)n(-c2ccccc2C(C)C)n1 N1(C(CC2CCN(OC)CC2)=O)CCCC2CN(C(c3ccc(Cl)o3)=O)CCC12 N1(C(COC(C)C)=O)CCN(C(C2CCN(Cc3cnoc3C)CC2)=O)CC1 C12(NC(CCNC(COC)=O)=O)CCC(NC(C3COCCN3C=O)=O)(CC1)C2 C#Cc1cnc(C(N2CCCC2CNC(=O)COCCC=C)=O)c(C)c1 Nc1ccc(C(=O)NCC(N2CCCC(CCF)C2)=O)nc1 CCCC(C(=O)NCCC1(O)CCN(C(c2cnc(CC)[nH]2)=O)C1)S(N)(=O)=O c1(CC)[nH]c(C(=O)NC(CNC(C2CCCNC2=O)=O)CC(C)C)nc1Cl Cc1ncccc1C=CC(=O)NCC(C)NCCO.C12(CCCCC1)C(=O)N2 C1(C(=O)OCC)CCC(C)(C)N(C(=O)CCc2ccc(C(F)(F)F)cc2)C1 C1(N(C)C(C23COC(CF)(C2)C3)=O)CCCC(N(C)C(c2ncccc2F)=O)C1 c1(C(=O)NCCCN(C(CC2CCCC(C)C2)=O)C2CC2)ccc(Cl)c(N)c1 N1(C(Cc2c(C)ocn2)=O)CC2(CNC(c3c(O)cccc3F)=O)CCC1CC2 CC1CC(C(=O)NCC2CCN(Cc3cncs3)C2)CCC1C CC(C)CCC(O)C(=O)NCC(CC1CCC1)C(=O)NC1(C2CCCO2)CC1 O=C(CCCc1ccsc1)NC1COCC1n1cc(CCCSC(F)F)nn1 c1(C2C(=O)N2)cn(CC(C)C)nn1.C1(N(C)CC)CN(CC2CC2)C1 Cc1cc(C)n(CCC(=O)NC2(C)CC(NC(c3cnoc3C3CCC3)=O)C2)n1 C1(C(=O)ONC2CN(C(CN(C)C(c3cnsn3)=O)=O)C2)CN(S(C)(=O)=O)C1 Cc1cc(C(=O)N(C)CCC(=O)C(C)C)cn1C.C(=O)(C(CO)N)N(CCO)C N1(C(C(CC2CCC2)OC)=O)CC(C(=O)NCC(C)F)C2(CC2)C1 N1(C(c2nn(CC)c(O)c2)=O)CCC(C2CN(C(C3CCC(F)CC3)=O)C2)CC1 c1(C(=O)NCC2CN(C(C(C)(C)C)=O)CC2C(F)(F)F)cc(N)cc(F)c1 c1(OCC(=C)C)cc(CCNC(CC(C(=O)O)C2CCOC2)=O)ccc1Cl N1(C(C(C(C)C)NC(C)=O)=O)CC2CCN(C(=O)CC(C)(C)C(C)(F)F)CC2C1 c1(C(N2CCC(CC(F)F)(OC)C2)=O)cc2n(c1)CCNC2 c1(CCC=C)ccc(C(=O)N(C2CN(C(=O)CC3CC3)CC2O)C)cc1 CC(C)(C(=O)NCC1CC1NC(C1COC2CCCCC12)=O)C(F)(F)F C(CC(=O)N1CCc2ncccc21)(C(C)CC)NC(C(C=C)CC)=O c1(N2CCC(C)(SC)C2)nc(=NCCC(C)c2cn[nH]c2)[nH]c2ccsc12 C1(COC)CC(OC)CN1C(=O)CCC1OCCO1.C1CCC(=O)O1 C1(CNC(CCc2nc(C)c(C)[nH]2)=O)CCCCN(C(=O)C(C(C)C)N(C)C)C1 c1(C(N2CC3C(C(N4CCC(NC(C)=O)C4)=O)C3C2)=O)cc(Cl)cc(I)c1 N1(C(C(C)c2cc[nH]n2)=O)CC(NC(c2ncoc2-c2ccco2)=O)C(C2CC2)C1 C1(NC(=O)COC2CCCOC2)CN(C(c2cnc(S)nc2)=O)CC12CC2 c1(C(N2CCC(O)(CNC(COCCC)=O)C2)=O)ccc2nc(O)cc(O)c2c1 CC(C)C(N=c1[nH]nc(C#N)s1)C(C)NC(=O)CC1CCCNC(=O)C1 C1(c2n(CC(=C)C)nnn2)(NCc2cc(Br)no2)CC2CCCC12 CC(O)(Cn1cccn1)C(=O)NCC(C1CC1)NC(c1ncccc1Br)=O N1(C(C(CCC)NC(N)=O)=O)CCOC2(CCC(NC(c3cocn3)=O)CC2)C1 C1(NC(c2ccn(CCCC)n2)=O)CCN(C(c2ncccn2)=O)CCC1CO c1(C(=O)NCC(CC)N(C(=O)CC2COCCN2C)C)cnncc1O N1(C(c2c(C)cn(C)c2)=O)CCC(CNC(C23CCCC2CCC3)=O)C1(C)C c1(CN(C)C(=O)NCC2CCN(c3nccn3C)C2)ccc(C#N)cc1 c1(CCNC(=O)C(=O)N2CC(Cc3ccccc3)C2)cc(Cl)sc1Cl C(N=c1nc(N2CCc3c(ccnc3O)C2)c2ccccc2[nH]1)C1C(C)(C)C1 c1(CCC(=O)NCC2CCCC(NC(CCNC(N)=O)=O)C2)c(F)cccc1Cl c1(NC(CCCNC(=O)Nc2ccc(N)c(F)c2)=O)csc2ccc(F)cc12 c1(C(=O)NCC(CC)NC(C2(CSCC)CC2)=O)cccc(OC(F)(F)F)c1 C(=O)(C(C(F)(F)F)C(F)(F)F)N(C1CCN(C(CN(C)CC)=O)CC1C)C C12CCCC1CN2C(C(=O)NCC)=O.C1CC1.S(C)CC N1(C(CCCOCC=C)=O)CCC(F)(C(=O)NCCCc2noc(C)n2)C1 N1(C(C2(CC)CC2)=O)CCN(C(c2cc(-c3ccc(F)cc3)n(C)n2)=O)C2CC12 N1(C(CC)CCC(C)(C)O)CCC2(CC1)OCCO2 C1(NC(CC2CCC(=O)N2)=O)CN(C(=O)CC(O)C2CC2)CC2(CC2)C1 N1(CCC2CCC(C)O2)CCC(c2nnnn2CC(F)F)(C(=O)OCC(F)(F)F)C1 C#Cc1cccc(C(c2nnnn2CC)NC(C(OC)OC)CC(C)(C)C)c1F C1(O)(C(=O)N(C(=O)CCCc2cnccn2)C2CC2)CC(c2ccccc2)C1 c1(CC(=O)NCC(CNC(C(C)CCN(C)C)=O)O)cccc2ccsc12 CC(C)CCCC(C)NC(C1C=CCCN1C(c1cnc(Cl)s1)=O)=O c1(CCN2CC(C(=O)OC)C(c3ccccc3)C2)cc(Cl)ccc1F c1(C(=O)OCC)ccc2c(c1)CCN(C(=O)NC13CCC(CO)(CC1)C3)C2 c1(C(=O)NCC(c2ccc(OC)cc2)CO)ccc2c(C)cc(Cl)nc2c1 C(CCC(=O)NCC1CC(CNC(=O)Cc2ccn(C)c2)C1)N(C)C C1(CCNC(c2c(C)n(C3CCC3)nc2)=O)CC2CCC(C1)N2C(C1CCC1)=O C(N=c1[nH]c(=NCC(C)(C)CCO)c2ncccc2[nH]1)c1cc(C)oc1C c1(C(N(C2CN(C(=O)CC3CSC3)CC2O)C)=O)cnn2ccncc12 Cc1cccc(C(C)NC(C2(NC(=O)C=CC3CCOC3)CC(F)(F)C2)=O)n1 C1(C(=O)NC2CCN(CC)C2)CCC(CC(=O)N(CC(C)O)C(C)C)CC1 C(=O)(C1=NOC2(CCC2)C1)NCC(CNC(=O)C(C)(C)C#N)OC CCCC(C)(CC)C(=O)NCC1C2CC1N(C(=O)C=Cc1cn(C)cn1)C2 c1(CNC(C2CN(CC3(C(=O)OC)CCC3)CCO2)=O)cc(OC)c(Br)cc1C Cc1cc(C(C(=O)NCSc2ccccc2)N(C2CCC(C)(C)CC2)C)ccc1I C(=O)(CCC[N+](=O)[O-])NC(CCCC)CNC(C1CCCNC1=O)=O C1(C(N(C2CCN(C(=O)CONC(=O)OC(C)(C)C)C2)CC)=O)CC1C1CC1 N1(C(=O)C2=CCCCO2)CC2CN(C(=O)CCc3ccsc3)CC2C1 CC12CC1CCN2C(c1cc(Cc2cn(Cc3ccco3)nn2)on1)=O c1(N2C3CN(C(CS(CC)(=O)=O)=O)CC32)nc(C)nc2ccccc12 c1(C(N2CC(CC#N)N(C(c3cscn3)=O)CC2)=O)c(F)c(F)c(F)c(F)c1F CC1CN(C2CCCCN(C(=O)N=c3ccc(C#N)c[nH]3)C2)c2ccccc21 c1(C(=O)NC2C3(CC(NC(=O)C4=C(Cl)CCC4)C3)C2)cc2c(nn1)CCC2 Cc1cc(C(N2CC3CC2CN3C(C2CCCC(C)(C)C2)=O)=O)c(Cl)cn1 C1(CNC(c2n[nH]cc2Br)=O)C2CN(C(C3(C4CC4)CC3)=O)CC12 C(=O)(CCCS(C)(=O)=O)N(C1CN(C(c2ccc(O)c(F)c2)=O)CCC1O)C C(=O)(C(F)C(F)(F)F)NC(C1CCCN(C(=O)Cc2cscn2)C1)C N1(C(Cc2cc(C)on2)=O)CCC2(CC(NC(C3CC3(Cl)Cl)=O)C2)C1 C(=O)(CC(C)C(C)(C)C)NC(CC1CN(C(c2sc(C)c(O)n2)=O)C1)C c1(CCC)cnnc(C(=O)NC2CCC(CNC(C34CSCC3C4)=O)C2)c1 CCC(C)(C#N)C(=O)N1CCC(CC(=O)Nc2cnn(C3CC3)c2)CC1 Cc1cccc(Cn2nc(SC(F)F)nc2-c2ccc(-n3cc(C)nn3)cc2)n1 N1(C(c2cc(C)on2)=O)CC(C)OC2(CCN(C(c3cn(CCO)nn3)=O)C2)C1 C1(n2cc(CCN(C(C)=O)CC)nn2)CON(C(=O)c2cncc(C(C)(C)C)c2)C1 CCCCCCCc1cn(CCCNC(c2ccccc2)c2ccccn2)nn1 N1(C(c2c(C)n(C)nc2C(F)F)=O)CC2OCC(NC(=O)C(C)C3CC3)C2C1 N1(C(C(C2CC2)OC)=O)CCC2(CCCCC2NC(=O)Cc2ccnn2C)CC1 c1(CC(=O)NCCC(C)NC(C2(C)CC2(Cl)Cl)=O)c[nH]c2cccnc12 C(CC(O)C(=O)NCC1CN(C(=O)CCSc2nnnn2C)CC1C)SC N(C(=Nc1ccccc1)NCC1(C)COC1)C1C(C)(C)C1 c1(C(N2C(CCNC(C(C(C)(C)O)F)=O)COCC2)=O)cc(F)c2[nH]nnc2c1 N1(CC2(OCC)CCC2)C(=O)CCN(CC2CCCC(C)(C)O2)C1=O n1(C(C(=O)NC(C2CN(C(C(C3CCCOC3)OC)=O)C2)C)C)nc(C)cc1C c1(C(=O)NCC2N(C(CC(C)n3cccc3)=O)CCC2)ccc(S(C)(=O)=O)[nH]1 c1(C(=O)NCC(CC)NC(=O)C(c2ccc(F)cc2)O)cc(C)n(CC)n1 C1(C(=O)NCC(C)NC(C2CCN(C3CC3)CC2)=O)CC(C)(C)CN1C c1(C(=O)NCC(C)CNC(=O)C(c2cnn(C)c2)O)cc(Cl)ccc1C(F)(F)F c1(CCOC)cc(C(=O)NCC2CCN2C(C2CC(C)N(C)C2)=O)cc(O)n1 N1(C(c2cc(COC)[nH]n2)=O)CCN(C)C(CNC(=O)CC2(C)OCCO2)C1 C=CC1CCN(C)CC1.c12conc1CNC(=O)C1(CC1)CNC2=O.C(C)(C)O c1(C(=O)NCCCCN(C(CN(C)C(=O)C2CC2)=O)C)ccc(F)c2occc12 Cc1cc(Br)c(Br)cc1C(=O)Nc1cc(C(N)=O)ccn1 C1(NC(=O)C=CC2CCCO2)CN(c2cnc(Cl)cn2)CC2(CCC2)C1 C(=O)(CCCCCN(C(=O)C(C1CCOCC1)C)C)N1CCC(CSC)CC1 C1(OC)CCCCC1S(=O)(=O)N1CCCC(NCc2cn[nH]c2)C1 N1(C(c2nc(OCC)oc2)=O)CC(C)CN(C(=O)CC#N)C(C)C1 c1(NC)c(C(=O)NCC2(NC(C3CCCSC3)=O)CCC2)cccc1F c1(COC)cc2ccc(-c3cc(C)cc(O)c3)cc2n1C.c12cc(c(Br)cn1)O2 [N-]=[N+]=NC1(C(N2CC(N=[N+]=[N-])C2)=O)CCN(C(c2cccnn2)=O)C1 c1(NC(=O)ON2CC3(CC3C(=O)NC(c3ccccc3)CCC)C2)cccc(Cl)c1 C12C3CC4C(C3NC1=O)C24.C(=O)(C1=C(Cl)CCC1)N1CC(=O)NCC1 C=CCC(C(=O)NC(c1ccccc1)CNC(c1ccc(O)c(F)c1)=O)C(C)C c1(OCC)ccccc1NC(=O)NCC(CCO)OC C1(NC(C(CC=C)NC(=O)CC2OCCO2)=O)CCCOC12CCC2 N(C(=NCCc1ccnc(C(=O)OC)n1)NC(C)C)CC1(CC)COC1 c1(C(C(=O)NC2CN(C(c3cnc(C)s3)=O)C2)O)cccc(F)c1 c1(OC)cc(C)ccc1CN(C(=O)C(=O)NCCc1ccc(F)cc1Br)C C(=O)(CC1CCOc2cc(OC)ccc21)N(C(C)CNC(c1cnsc1)=O)CC c1(C(=O)NC2CCN(C(C(C=C)(C)O)=O)C2)cc2nc[nH]c2cc1F CCCCC(F)C(=O)NCC1CN(C(=O)CCc2c[nH]c(C)c2C(C)=O)CC12CC2 C1(NC(c2cc(CN(C)C)no2)=O)CCCC(NC(c2cn(CCF)nn2)=O)C1 N1(C(C2OCCC(NC(C=CC(C)(C)C)=O)C2)=O)CCc2ncsc2C1 Cc1ccc2nonc2c1C(=O)N(CCCCN(C(=O)CCCCCO)C)C CC1CN(C(=O)COc2cn[nH]c2)CCC1NC(c1c(C(F)(F)F)cnn1C)=O N1(C(c2cc(C)sc2)=O)CC(NC(=O)C(C)Cn2cccn2)CC(F)C1 c1(C(=O)NCCOC2CCN(C(CC3CC(SC)C3)=O)C2)cc2c(s1)CCC2 C(C(C)(C)CC(=O)NCCN1CCCC1)Nc1cc(C)n(C)c1 C1(C(=O)NCCCCN(CC)CC)CC=CC(NC(c2c[nH][nH]c2=N)=O)C1 c1(OC)c(C(=O)NC(C)CC(C)NC(c2ncoc2Br)=O)cccc1Cl c1(C(=O)NCC(C)CNC(=O)CC2CCCCC2O)cn2cc[nH]c(=O)c2n1 c1(CNC(CC#C)COC)cccc(C)c1Br CC(C)C(CCN(C(=O)C(c1cccs1)N(C)C)C)NC(=O)C(N(C)C)N(C)C c1(C(=O)NC(c2c(OC)cccc2)C(C)(C)C)ccc(C2CC2)c(Cl)c1 CC(C)CC(CNC(C12CC(C#N)(C1)C2)=O)C(=O)NCCn1ccc(=O)cc1 C(CCC(C)C(=O)NCC(C(=O)NCc1ccns1)N(C)C)OC C1(CC(=O)NC(CN(C(COCCSC)=O)CCO)C)CCc2ccccc2C1 C1(N(C(Cc2ccn(C(C)C)n2)=O)C)CCCN(C(=O)C(C)C2CCC2)C1 N1(C(CC2(CC)CCOCC2)=O)CC2CC(NC(=O)Cc3cn[nH]c3)C1C2 c1(NC(=O)NC2(C)CCSC2)nc(N2CCCC2)sc1Cl c1(C(=O)NCC(C)N(C(c2cc(C(=O)OC)no2)=O)CC)coc2c1CSC2 c1(C(c2nnc(N3C(CCC)COCC3)n2C)=O)cc2c(OC)ccc(C)c2[nH]1 c1(CC(=O)NC2(CNC(COCC)=O)CCOC2)n[nH]c2ccccc12 N1(CC(=O)N(CCC#N)C)CC23CCCCC2(COC3)C1 c12noc(n1)NCCCN(C)C2C1CCC1.C1(CC)CCOC1 N(C(=NCCN1CCCCC1)NC1CC(N(C)C)C1)C(C)Cc1ccc(C(F)(F)F)cc1 C(=O)(C(CC)CCCCC)N1CC(CNC(C(CC(=C)C)OC)=O)CC(C)(C)C1 c1(OCC(=O)NC2CCCCC2CNC(c2ncccc2F)=O)ccc(Cl)nc1 N#Cc1nccnc1N1CCC(CNC(c2ccc(-n3cncn3)nc2)=O)CC1 C(=O)(C1=C(C#N)CCC1)NCCC1N(C(C2C(CCC)C2)=O)CCSC1 C(=O)(C1COc2ccc(F)cc21)N1CCN(C(=O)CCc2cc[nH]n2)CC1CO CCCC(CC)CCC(=O)NC1CC12CC(NC(=O)C1=C(Cl)CCOC1)C2 c1(SC)oc(C(=O)NCC2C(C)CCN2C(=O)Cc2cnccc2C)cc1C S(=O)(=O)(c1ccccc1C(=O)NC1CC1C(=O)Nc1ccc(I)cc1Cl)N(C)C C1(NC(C2(C=C)CCC2)=O)CC(OC)CN(C(c2nccn2CC)=O)C1 c1(CCCCNC(=O)CCc2cscc2Br)ccccc1Br N1(C(C(C)(C)NS(C)(=O)=O)=O)CCC(C2CCN(C(C3(O)CCSC3)=O)C2)CC1 C(C(C)(C)C1=CCCC1)NC(C(CCOCCO)NC(c1c(C)scn1)=O)=O c1(COCC(N2CCC(OC3CNC3)C2)=O)cccc(Cl)c1 c1(OCCOCC)ccc(C(N2CC(C(C)(C)NC(=O)C(C)(C)CF)C2)=O)cc1 C1(C2CC2)(CNC(Cc2c(C)ccs2)=O)CCN(C(=O)C(O)CN(C)C)C1 c1(OC)cccc(CC(N2CCCC2CN(C(=O)C(C2CCC2)OC)C)=O)c1 C1(C(N2CCCC(OCCC)C2)=O)CC2CCC(C1)N2C(c1cc[n+]([O-])cc1)=O CON1CCC(CC(=O)NC(C)CCCNC(=O)CC23CC(C2)C3)CC1 n1(CCCC(=O)NC2CCC(CNC(CC3(C)CC3(F)Cl)=O)C2)ccccc1=O n1(CC)ccc(C(N2CCC2CNC(C2(CN(C)C)CCCC2)=O)=O)n1 c1(C(=O)NC2CN(C(c3nc(OCC)oc3)=O)C(CO)C2)cc(F)c(C)cc1O c1(COC)cc(C(=O)NCC(C(=O)N2CC(C3CCOC3=O)C2)N(C)C)n[nH]1 C1(CNC(Cc2c(C)n[nH]c2C)=O)CN(C(c2ccccc2Cl)=O)CC1(F)F C1(C(=O)NCC(=O)Nc2cn[nH]c2)CC(F)(CNC(CCC)=O)C1 C12(NC(CCC(=O)NCC)=O)CCN(C(=O)CC34CCCN3CCC4)CC1C2 c1(C(N2CC(NC(c3[nH]ccc(=N)n3)=O)C2)=O)ccc(S(=O)(=O)NCC(N)=O)o1 c1(N2CCC(C(C)O)CC2)nccc(=NC(CCO)c2ccccn2)[nH]1 c1(COC)cc(C(=O)NC2(COC)CN(C(=O)CC3CC3C3CC3)C2)cs1 C(=O)(C1=CCN(C(C2(C)CC2(C)C)=O)CC1)NC(C)Cc1cnccn1 C1(CCCC)CCC(C(N2CC(NC(c3cn(C(F)(F)CO)nn3)=O)C2)=O)CC1 C#CCCC(O)C(=O)NC1C2CC1CN(C(C1CCCC1c1nncn1C)=O)C2 N(C1c2ccccc2CC1F)C(c1cc(Br)ccc1O)C c1(C(N2CCOC3CN(S(C)(=O)=O)CC23)C)c[nH]c2c(Cl)cccc2c1=O Cc1nn(C(C)C)cc1C(N1CCC(N(C(=O)CCc2ccoc2)C)C1)=O C=CC1CCCN(C(=O)C(C)(C)CNC(C2CC3CC2CC3O)=O)C1 c1(CN(C2(C(=O)OCC)CCC2)CC2CCCO2)cn(C)nc1C(N)=O c1(C(N(CCC)Cc2ccc(Cl)cc2)=O)c(Br)nc2n1CCCC2 C1(OC)(CNC(=O)CCn2ccnc2)CCN(C(=O)CC2COCC2O)C1 c1(C(=O)NCCN(CCC)C(c2cc3scnc3[nH]2)=O)ccc2cncn2c1C C(=O)(CC1=CCCC1)C(C)(C)C.n12ccc(n1)CCCCn1c(nnn1)COC(=O)N2 C#CCCC(O)C(=O)N(C1CN(C(=O)Cc2cc(Br)cs2)C1)C C#Cc1cnn(C)c1C(N1CCC(N2CCC(NC(C3(C)CCC3)=O)CC2)C1)=O N1(C(C2C(=C)CC2)=O)CC2CCC1CN2C(c1c(C)nn(CCO)c1C(F)F)=O c1(CC(=O)NC(C)(CNC(c2coc(Cl)c2)=O)C2CC2)cc(F)cc(Cl)c1 c1(CCC(C)NC(C)CC(C)N)ccccc1F c1(C(=O)NCCC(C)NC(C(C)n2cccn2)=O)cc2cccc(F)c2o1 C(=O)(CC1CN(C)c2ccccc21)NCC1(CNC(CC(C=C)(C)O)=O)CC1 C1(C)(NC(CN2CCC(C)(C)C2)=O)CCC(NC(=O)CCC2CC2)CC1 C1(C(=O)OCC)CC(C(=O)Oc2cnc(F)c(F)c2)C12CCCC2 C(C(C)(C)CCOCCN(C)C)OC(CSCC#C)=O.C1(OC)CC1 C#CC1CCCCN1C(C1(C)C=CCN1C(=O)CC1(C)CCC1)=O c1(CC)c(C(N2CC(CNC(=O)CSc3nncn3C)C(C)C2)=O)nnn1CC CC1(CCNC(C2CSCN2C(=O)CN2CC=CC2)=O)CCOC1 c1(NC(C2C(O)CCN(Cc3cc(C)c(Cl)nc3)C2)=O)nc2cc(F)ccn2n1 c1(C(N(CCCCNC(C(CC)(C)O)=O)C)=O)cc2cc[nH]c(=O)c2s1 C1(NC(C2(F)C(C)C2)=O)CCCCC1NC(c1cnn(C)c1)=O CCCCC(C)CCC(=O)NCC1CC12CCN(C(=O)C=CC(C)(C)C)CC2 c1(C(N2C(CCNC(C3C(CCC)C3)=O)CCC2)=O)ccc(N(C)C)cc1CC C(=O)(C(O)CSC)N1CC(CC(=O)N(C2(C(=O)OC)CC2)C)C1 n1(CC(N2C(CNC(=O)CC3CCCC3)CCC2)=O)[nH]cc2c(=O)ncnc1-2 O=C(CS(=O)C(F)(F)F)NC1(CO)CN(C(=O)CSCCCF)C1 c1(OC)ccc(C(N2CCC(CN(C(=O)CNS(C)(=O)=O)C)CC2)=O)c(OC)n1 C1(C(N2CCC(N(C(=O)CC=CC(C)(C)C)C)C2)=O)C2CNC(=O)C12 C(CC(C)(C)NC(=O)CCC1(NC(=O)Cc2cncs2)CCC1)=CC=C c1(C(N(CC(C)NC(C2OCCC2C)=O)CC)=O)ccnc(OCC(F)(F)F)c1 Cc1nn(CC(=O)N(CC(CO)(CO)NC(=O)C(C)n2cncn2)C)cc1Cl c1(C(N2CC(c3cn(CCCN(C)C)nn3)(O)C2)=O)cn(C)nc1C1CCOC1 CC(=O)CCC(=O)N1CC2CC2C1C(=O)NCCC(=O)NO C(=O)(C1=CCCC1)N1CCC(N(C(=O)CC2(CO)CC2)CCC)C1 CC1(CNC(c2cccnc2C(F)F)=O)CCC(NC(c2ccnnc2)=O)CC1 c1(OC)cc(C(=O)NC2CCCC(CNC(c3cccc(F)c3)=O)C2)cc(C)n1 Cc1cc(C(=O)NCCN(C(=O)C(C)CO)C(C)C)cnn1 Cc1coc(C)c1CNC1C2CN(CC(N3CCC(C)CC3)=O)CC12 CCC(C)(C)CC(=O)NC(C)(CNC(=O)CCCc1cc(O)ccc1C)C1CC1 C(=O)(CCCC#N)NC1(C(N2CCC(CCC)C2)=O)CC(O)C1 c1(C(N2CCC(C)(NC(c3ccn(C)n3)=O)C2)=O)ccc2c(c1)CCC=C2 C1(NC(=O)Cc2ccsc2)CC2CCC1CN(C(C1CCC3CC13)=O)C2 O=C(C1=CCOCC1)NCCC1(C(N2CC(O)(C(F)(F)F)C2)=O)CC1 C#CC1CCCN(C(=O)CCC2CC(NC(C3CCCOC3)=O)C2)CC1 c1(C(N2N3C(CCCC3)C(=O)NCC2)=O)cccc(C(=O)OC)c1C.CCOC CCCC(C)(C)C(=O)NC1CN(c2nnnn2C)C1 N1(C(C(CCC=C)NC(=O)C=C=C(C)C)=O)CC(C2CCCCC2)C1 O(NC(=O)CCOC1CC(NC(=O)Cc2cn[nH]c2)C1)CC=CC CC(C)C(C(=O)N1CCCCC(CNC(=O)C(F)(F)CO)CC1)C(C)C C1(c2cn(CC(COC)O)nn2)CCN(C(c2coc(CN(C)C)n2)=O)C(C)C1 CC(C)(CCS(C)(=O)=O)NCc1ccnc2[nH]ccc12 C12(C(N3CC(CNC(c4ncn(C)n4)=O)OCC3)=O)CCC(CC1)CC2 CCCCC(O)C(C)C(=O)N1CCC(NC(=O)C=CC2CCCN2C)C(C)(C)C1 c1(C(=O)NCC23N(C(c4n(CC)ncc4)=O)CCC2CC3)ccc2nncn2c1 CC(O)C(F)(F)C(=O)NC1CC(NC(C2(c3ccccc3F)CC2)=O)C1 c1(NC(c2c(NCc3c(C)ccc(C)c3)c[nH]n2)=O)cccc2c(Cl)ccnc12 c1(C(N2CCC(CNC(C3CC3C(F)(F)F)=O)C2)=O)ccncc1Br c1(N(CCCCNC2(O)CCN(C(=O)OC(C)(C)C)C2)C)cc(Cl)ncc1F C(=O)(C(F)(F)C(C)(C)O)NC(=NCCCC)NC1CCCC(C)(C)C1 CC(C)(CCNC(=O)C1=C(Cl)CCC1)C(=O)NCc1cccc(C#N)c1 CC(C)CCCC(C)NC(=O)NCC1CCN(CCc2ccccc2)C1 C1(NC(Cn2c(C)ncc2)=O)CCCN(c2ccc(C#N)nn2)C1C CC1(C)CN(C(c2cnn(C3CC3)c2)=O)CC1NC(=O)Cn1cc(Cl)cn1 C1(C(=O)NC(C)C(C)NC(c2nc(Cl)oc2C)=O)(OC)CCSCC1 C1(C=O)CCN(C(=O)C)C12CCC2.Cc1ncsc1C1CC1c1cncn1C CC(COC(C1CCC1(C)C)=O)C(=O)Nc1ccccc1 C(C(COC)CC(=O)N(C(CNC(c1cccc(=S)n1O)=O)C1CC1)C)OC C1(CNC(c2c(CC)onc2)=O)CCC(C)N(C(=O)COC2CCCCC2C)C1 CCC(C(=O)NC(CC)CCCC(=O)NCC1C2CCCC12)C(C)(C)CC C1(CCC)(NC(=O)Cc2ncccc2F)CCN(C(=O)CCN(C)CCO)CC1 c1(OC(CN(C(=O)NC(C)C)CC)C)cccc(N2CCCCC2=O)c1 N1(C(C=C)=O)CCC(C)C(CNC(=O)Nc2cnn(C)c2-c2ccc(F)cc2)C1 Cc1cn2cc(C(N3CC(NC(c4cc[nH]n4)=O)CC(F)C3)=O)sc2n1 N1(C(C2N(N=O)CCC2)=O)CC2(C(=O)NCC3CC(C(F)F)C3)CCC1CC2 CC(C(=O)N1CC2CC1(CNC(=O)C(C)(C)c1cncnc1)C2)S(N)(=O)=O C1(Cl)(C(N(CCN(C(=O)C(C(C)C)SC)CC)CC)=O)CC12CCOCC2 C(=O)(CCC(C)(C)C)NCCC1(C(N(C(C)C(N)=O)C)=O)CC1 C1(C(=O)NC2CC(CCNC(c3c(CCC)nsc3N)=O)C2)CCOCC1(C)C N1(C(c2cc(CO)[nH]n2)=O)CCC(c2ccccc2)C(Nc2ncnc(Cl)c2F)C1 C1(NC(C(C)NC(=O)NC)=O)CC(O)CN(C(=O)CSc2nnc(S)s2)C1 C1(C(=O)NCC(CNC(c2c(CCC)n[nH]c2)=O)(C)O)CCCCN1N=O c1(-n2c(C(=O)NCCNC(C(CC)N(CC)CC)=O)cnn2)ccc(C#N)nc1 c1(CC(=O)NCCOCCN(C(c2cc(C)ncc2)=O)C)ccc(F)c(C)c1 C(=O)(C(C(C)(C)C)N(C)C)NC(C(C)C)(C)CNC(=O)CCc1c[nH]c(=N)[nH]1 CC1(C)CC(C(F)(F)F)CN1CC(c1nccnc1N)=O O=NN1CCCCC1C(N1CCOC(CCNC(c2ccc(F)cc2F)=O)C1)=O N1(C(C2C(C(=O)OC)CCC2)=O)C2CCC1CN(C(C1(CO)CC1)=O)CC2 C1(CNC(C(N2CCC(C)(CC#N)C2)=O)=O)CC2(C1)CC1(CCC1)C2 c1(C(N2CCCC(CNC(C3CCC(F)CC3)=O)C2)=O)ccc(F)c(Br)c1 N1(CC(N2CCCC(C)C2)=O)CCn2ncc(CNC(c3ccsc3Cl)=O)c2C1 C1(CCC(=O)N(C(C)(C)N(CCOC=O)C)C)CCCCO1 N1(C(CC2(C)CC2)=O)CC(C)(C)C(NC(=O)CC2CCNC(=O)C2)C(C)(C)C1 CC(C)CC(C)(CN=c1ccnc[nH]1)NC(c1cnc(C(C)(C)C)o1)=O CC1Oc2cc(-c3nnc(-c4ccon4)o3)ccc2NC1=O n1(C(C(=O)N(CC(CN(C(C(C(C)C)C)=O)C)O)C)(C)C)cnc2ccccc12 N1(C(CC2CN(C(C3(C=C)CCC3)=O)CC23CC3)=O)CCCN(C)CCC1 c1(C(=O)NCC(C(C)C)NC(CCC(C)=O)=O)ccc2cnc(C)cc2c1 c1(C(=O)NCC(N2CC(N(C)C(C3CC=CCO3)=O)C2)=O)ccc(F)cc1F N1(C(C(Cc2ccccc2)OC)=O)CC2(C1)CN(C(C1CCC3(C1)N=N3)=O)C2 CCC(F)(F)C(C)(C)C(c1nnnn1C)NCCC(=O)N1CCCC1 C(CC(C)(C)C(=O)N1CC2C(C(=O)Nc3cncc(CO)c3)C2C1)SC c1(C(=O)NCCCCCNC(C2CCC2C(F)(F)F)=O)cn(CC(F)(F)F)cn1 C#CCCCCCC(=O)N1CCCC(NC(c2onc(CC)c2C)=O)C1C C1(C(F)(F)F)(C(C)C)CCN(C(c2cncc(OC(C)(C)C)n2)=O)C1 Cc1ccccc1CC(N1CC(NC(=O)C(C)(C)CN(C)C)CC1CO)=O C=C(C)C(C)(C)C(=O)N1CCCC(F)(C(=O)NCC(C)CC(F)(F)F)C1 N1(C(Cc2c(C)scc2)=O)CCCCC(N(C(=O)CC2CCCCO2)C)C1 N1(C(c2c(C#C)cn(C)n2)=O)CC2(CC(C(=O)N(CC(O)CO)CCC)CO2)C1 N1(C(CN(C)C2CC2)=O)CCCCCC(NC(c2ccnc(-c3ncc[nH]3)c2)=O)C1 N1(C(Cc2c(C)noc2)=O)CC=CC(C(=O)N(CC(C)(C)C)C)C1 CC(CCO)N=c1[nH]c(N2CCCCC(CO)C2)nc2c1CSC2 C1(CCC(=O)N(CC(O)CN(C(=O)CC2CC3(CCC3)C2)C)C)CC(C)(C)CO1 C1(CC(=O)NC(C(C)(C)OC)C)CCN(C(=O)CC2CCC2)CC1 C(CNC(C1CCC=CCC1)=O)(CC(=O)NCc1cnn(C)c1O)OC N1(C(c2ccc(OC(F)F)nc2)=O)CCOC2CN(c3ncncc3Br)CC12 C#CC1CN(C(=O)C(c2ccnn2C)NC(=O)C2=CCCSC2)CC1O Cc1cccnc1C=CC(N1CCC(NC(=O)CCC2CC2(Cl)Cl)CC1C)=O C(=O)(CCC(C)(C)[N+](=O)[O-])N(CCCCNC(=O)C1=NOC(C)(C)C1)C C=CCCCCC(=O)N1CC2CC1CN2C(c1cc(CC)[nH]n1)=O c1(NC(COCCCC#N)=O)cccc(CNC(=O)CNC(=O)CC(F)(F)F)c1 C#CCCCCCCCC(=O)N1CC(O)(C(F)C(=O)NCCC(C)CO)C1 Cc1noc(C)c1CCC(=O)NC1CN(C(c2cnccc2O)=O)CC1F S(=O)(=O)(c1c(C)cccc1Cl)N1CC(COC)N(Cc2csc(Br)c2)CC1 n1(CCOC)cc(C(=O)NCC2C=CCN2C(=O)COCCOC)c(C)n1 c1(C(=O)NC(C)CCN(C(=O)C(C)n2cncn2)C)cccc(CO)n1 n1(CC)c(C)nn(CC(N2CCC(COC)(NC(=O)C3=C(C)CC3)C2)=O)c1=O CC(C)(CC(F)F)C(=O)NCCCCN1CCCN(C(C2CC(O)C2)=O)CC1 C(=O)(C1=CCCSC1)N1CC(NC(CN(C2(C=C)CCC2)C(c2ccsc2)=O)=O)C1 C12(C(=O)NC(CC)CNC(C3CCC4(CC4)C3)=O)CCC(CO)(CC1)CC2 C12(CC(N3CCC(CN(C(c4n(C(C)C)ncn4)=O)C)C3)=O)CCC(CC1)CC2 Cc1ncnc(O)c1C(=O)NC1CC2CC(NC(C3(CF)CC(F)(F)C3)=O)C2C1 Cc1cccc(F)c1CC(=O)NC1CCN(C(=O)Cc2cnn(C)c2)CC1CO N1(CC2(CC=C)CCOCC2)CC(=O)N(Cc2cc(C)cs2)C1=O CC(CN(C)C)CCC(=O)N1CC(N(C)C(C2CC(CN(C)C)C2)=O)C2(CC2)C1 C1(OC(CCCN(C(C)=O)C)=O)CCC(NC(c2cc(CO)[nH]n2)=O)CC1 N1(C(=O)C(F)Cc2ccccc2)CCN(C(c2cnc(Cl)s2)=O)C(C2CC2)C1 c1(C(N(CCN(C(=O)CC2(N(C)C)CCC2)C)C)=O)ccc(=O)n(C)c1 CC(C)CC(O)CC(=O)N1CSCC1C(=O)N(C(C)C)C(C)C C(C)(C)(CCCCC(=O)N1CCN(C(=O)CC2=CCCC2)C(C)C1C)OC C1(NC(CCC(C)(C)NC(=O)C2=CCCCC2)=O)CCCCCCC1O C1(C(N(CCC(C)NC(CCOCC)=O)C)=O)Cc2cc(C)ccc2S1 c1(C(N2CCN(C(CSCC=C)=O)CC2c2ncc[nH]2)=O)cnc2[nH]ccc2n1 CCC(C(=O)OC)C(=O)NC1CC(C)N(C(=O)Cc2cc(F)ccc2Cl)C1 C1(CC(=O)N(CCCNC(CCC(C)C)=O)CCO)CC(=O)NC(=O)C1 N1(C(C2N(C(C(C)C)=O)CC(O)C2)=O)CCN(C(=O)C#CC(C)(C)C)C(CCO)C1 C1(NC(c2ccnc(CC(C)C)n2)=O)CC2CC1N(C(=O)C(F)F)C2 N1(C(c2c(C(C)=O)cn(C)n2)=O)CC2CC(NC(C3CC3(F)F)=O)C2C1 c1(C(=O)NCC(O)CNC(C2CCCC23CCC3)=O)ccnc2[nH]nnc12 Cc1cc(CC(F)=NCCC(=O)OC2CC2)sn1.C(CCNC=O)N(C=O)C(C)C c1(C(N(C2(CC(=O)NC(CC)Cn3cncn3)CC2)C)=O)ccc(C)nc1 N1(C(C(C2CCCC2)OC)=O)CCC(CNC(C2CN(C)C2)=O)C(O)C1 N1(C(C2CCN(C)C2=O)=O)CC2(CCN(C(=O)CSCCC(F)(F)F)CC2)C1.C(C)(=O)O C(C)(C)(CC(=O)NCC(C1CCN(C(=O)C(F)=C2CCCC2)CC1)O)OC N1(C(c2ccc(C)cc2F)=O)CCCC12CCCN(C(=O)C(C1CC1)N(C)C)C2 C(C)(CCCC(=O)NCc1cc(C)co1)NC(CCSCC)=O c1(NCC2C(NC(c3n(C)nc(CC)c3Br)=O)CCC2)ccc2cnccc2c1 c1(C(N2C(CNC(CC3C(OC)COCC3)=O)CCC2)=O)ccc(N)c(Cl)c1 c1(C(=O)NCC23C(CN(C(c4c(C)nsc4)=O)C2)C3)ccc2nnc(O)n2c1 c1(C(=O)NCCN(C(=O)CN2CCC(O)CC2)CC)nc(=N)cc[nH]1 C(C)(CN=c1ccn(C(F)F)[nH]1)(c1nnnn1CC1CCOCC1)NCC=C CCCCC(C)(F)C(=O)N1CC2(C1)CN(C(c1cccc(SC)n1)=O)C2 C#CCC(CC(=O)NCCCCC1CC1C)NC(=O)CCCC(=C)C C1(N(C(=O)CNC(=O)C2CC2)C)CCN(C(C2(C(F)F)CCC2)=O)CC1 C(=O)(C1Cc2ccccc21)NC(CNC(C(C=CC)O)=O)(C)C Cn1cc(CC(=O)NC(C)(C)CNC(=O)COC2CCCC2)c(OC(F)F)n1 c1(C(N2CC(CNC(CCN(C)CC)=O)N(C)CC2)=O)ccc2nc(S)[nH]c2c1 n1(C(C)C)cnc(CNC(c2coc(CNC(=O)CCC3CCCCC3)c2)=O)n1 Nc1cc(C(=O)NC2CCCN(C(=O)CC3CCC3(F)F)C2)cc(Cl)n1 c1(OC)ccc(C=CC(=O)NCCC(C)NC(c2ccc(F)c(F)c2)=O)cc1 c1(CC)c(C(=O)NCCOC2CCN(C(=O)C(O)C3CCC3)CC2)nnn1CC C(=O)(C(O)CC(C)C)N1C(C(N2CC(OCC(C)C)C2)=O)CC(OC)C1 N1(C(=O)C=CC2CCCO2)CC2CC1C2C(N1CC(CC2CC2)C1)=O C(=O)(C1=C(C)CCCC1)NCC#CCNC(c1cc(OC)c(OC(F)F)cc1)=O N1(OC)CCOC2(CCNCC2)C1.c1(C)nccc(=NC(=O)C2C=CCC=C2C)[nH]1 Cc1ccc(F)c(C(=O)NC(CC(=O)NC2CC3CCC2O3)C2CC2)c1 c12ccc(cc1)NC(=O)N2.N1(S(CC)(=O)=O)CCC1(CC)CC C12(C(=O)NC(C(C)C)CNC(c3coc(Br)n3)=O)CCCC1C2(F)F c1(CCC(=O)NCC2CCC2NC(C2(c3cccs3)CC2)=O)ccc2ncsc2c1 C#CCC(C(=O)NCCCc1ccco1)NC(=O)C=Cc1ccccc1 CC1CC=C(C(=O)NC2(CO)CCN(C(c3cnc(N(C)C)nc3)=O)C2)CC1 c1(CNC2CCC(C(=O)OC)CC2)cc2ccccc2nc1OC(F)F C(CC(F)F)(C(=O)N1CC(S(C)(=N)=O)C1)NC(CCC=CC)=O c1(C(N(CCNC(c2cc(C)sc2C)=O)C(C)C)=O)cc(Cl)ccc1-n1ccnc1 c1(OC(C)=O)cc(CNCC(C)C(C)(C)C)c(C)cc1C Cn1nnc(C(=O)NCCC2CC(NC(=O)CSCc3ccc(Cl)nc3)C2)c1N C(c1ccc2[nH]ccc2c1)=CC(=O)NCC(C)NC(C1(C#C)CC1)=O c1(CN)ncnn1C1CC1.C(CC(=O)N)CCCNC(C1C(=C)C1)=O c1(CNC2C=CC(C(=O)Nc3ccc(C)cn3)C2)cc(F)cnc1Cl N1(C(C(c2cn(C)nc2)(C)C)=O)CCN(C(C2CC2F)=O)C(CO)C1 O=C(C1=CCCN(c2ccnnc2)C1)Nc1c[nH]nc1-c1ccccc1 n1(CC(=O)NCCCC(C)NC(C(n2cc(C)nc2)(C)C)=O)cnc([N+](=O)[O-])c1 c1(COC)cncc(C(=O)N(C2CC(NC(c3cc(Cl)cnn3)=O)C2)C)c1 C12(NC(C(C)C3CCC3)=O)CC1CN(C(=O)CC(=O)OC(C)(C)C)C2 N1(C(CCCCNC(C2=NOC(C)C2)=O)=O)CCC2(CCOC2=O)C1 Cc1cc(C)c(C(=O)NCC(C)CNC(c2nc(C)sc2C)=O)c(C)c1 Cn1cc(C(N2CCCCC2c2cnccn2)=O)c(-c2ccc(Br)o2)n1 C1(CC=C)(NC(=O)CCNC(c2ccsc2)=O)CCN(C(=O)C=C2CC2)C1 c1(CC)cnccc1C(N1CCC1CC(F)C(=O)O)=O Cc1ccc(C=CC(N2C3CN(C(c4ncoc4C)=O)CC23)=O)s1 C1(C(C)C)CCC(C(=O)NC2CCC(CNC(=O)C=Cc3ccccn3)C2)CC1 c1(C(=O)NCCN(C(=O)Cc2cnnn2C)CC)ccc2nc(O)[nH]c2c1 C1(CNC(c2c(OC(C)C)cccc2)=O)CC2(C1)CN(C(C1CNC(=O)C1)=O)C2 c1(CC2CCC(F)(F)CC2)c(C(=O)NS(C)(=O)=O)oc2ccccc12 N1(C(C(C(CC)O)C)=O)CC2CCCN(C(c3cc(COCC4CC4)ccn3)=O)C2C1.OC CC12CC(CNC(c3nc(CC(=O)N(C4CCCC4)C)cs3)=O)(CCO1)C2 c1(NCCNC(=O)CCC2CCC2)cc2c(C(=O)O)cccc2s1 c1(C(=O)NCC2C3CN(C(C4N(C)C(=O)CCC4)=O)CC32)ccc2ocnc2c1 O=C(N=c1[nH]oc2cccnc12)C1CCCN(Cc2ccc(F)c(O)c2)C1 c1(C(N(C2CCN(C(=O)Cc3nc(C)sc3C)C2)CC)=O)csc(=NC)[nH]1 N1(C(C(C#N)C2CC2)=O)CCCCC2(CCN(C(c3ccsc3)=O)C2)C1 c1(CCC(N2CC(N(C)C(C34CCC3C4)=O)C(O)C2)=O)ccc(Br)cc1F c1(COCC)ccc(Cl)c(C(=O)OC23CC(Nc4nc(C)no4)(C2)C3)c1.OC c1(C(N(CCCNC(c2n(C)ncc2)=O)Cc2ccccc2)=O)cc(N)ccn1 c1(C(=O)NCC)oc2ccccc2c1C(C)NCc1cc(OC(C)C)ccc1F c1(C(N(CCNC(CCC(=C)Cl)=O)C2CC2)=O)cc(S(=O)(=O)N(C)C)cn1C C1(C)(c2n(C3C(c4ccc(OC)cc4)C3)nc(-c3ccc(Cl)s3)n2)CCCCCC1 c1(NC(c2cc(-c3c(C)nn(C)c3C)ncc2)=O)ccc(S(=O)(=O)C2CC2)cc1 C(C(C)(C)CC(C)NC(C1(CSc2cccc(Cl)c2)CC1)=O)OC N1(C(CCCOCCOC)=O)CC2(CCN(C(C3CC4C=CC3C43CC3)=O)C2)C1 N1(C(C)C)N=C(C(=O)NCCC2CN(C(=O)CC3CCCC(=O)N3)C2)CCC1=O N1(CC)CC2C(C(F)(F)F)CC2(C(=O)NCC(c2ccc(F)cc2)F)C1 N1(C(CNC(CCC(C)C)=O)=O)CC2CCCC2(NC(C23CC(C)(C2)OC3C)=O)C1 CC1(C)CC(NC(=O)COCC2CCOCC2)CN(C(c2cncc(N)n2)=O)C1 CCCC(CNC(=O)CC1CCN(C(C2(C3CC3)CCCO2)=O)C1)CCC c1(OC)nccc(CNC(C2C(CNC(=O)CC3(O)CCOC3)CC2)=O)n1 N1(C(C2CC(C)(C)OCC2)=O)C(C(N2CCOC(C#N)C2)=O)CC2CCCCC12 C1(CC(=O)OC(C)(C)C)CCCC12CN(C(=O)NCC(C1CCC1)SC)C2 CC1(C)CCCC(C(=O)NC2(C(=O)NOCC3(CSC)CCC3)CC2)C1 C(C(CNC(C1CC1n1cnnn1)=O)NC(C1CC1Cl)=O)OC C(C(COc1nnnn1C)C(C)C)N1CC(NC(C(COC)NC)=O)C1 c1(NC(C2CN(C(C(CC)OC)=O)CC2C(C)(C)OC)=O)cccc(Cl)c1C C1(CNC(C(C(C)C)C)=O)CN(C(=O)CCNC(C2CCC2)=O)C(C)(C)C1 C(=O)(C(C)(C)C(=O)NCC(C)(C)C(=O)NCCC(F)(F)CO)N(C)C c1(C(N(CCNC(Cn2ncc(C#C)c2)=O)CC)=O)cccc(S(C)(=O)=O)c1F c1(CC(N2C3CC(NC(C(C)n4cnnn4)=O)(C3)C2)=O)ccc2ccoc2c1 C1(NC(c2cc(C(F)F)[nH]n2)=O)CC2(C1)CN(C(c1coc(Br)n1)=O)C2 C1(C(N(C)CC2(NC(c3cn(CCC(C)C)nn3)=O)CC2)=O)CC2CC1CO2 C12(NC(c3ccc(N)cc3F)=O)CCCN(C(=O)COCCO)CC1C2 CCCC(CC)C(=O)NC1CN(C(c2scnc2C(F)F)=O)C(C)(C)C1 N1(C(c2n(C)nc(O)c2)=O)CC(CN=c2cc[nH]c(-c3nccs3)n2)C(C)(C)C1 C#CCC(C(=O)NNC(=O)CCn1ccc2cc(F)ccc12)C1CC1 Cc1cncc(CNC(C2CN(C(=O)CC#N)CCO2)=O)c1 N1(C(C(CC)C#N)=O)CCC(N=[N+]=[N-])(C(=O)Nc2cccc(C)c2C)C1 C1(C)(C(N(CC(C)NC(C2(C)CCC(=O)C2)=O)C)=O)CCS(=O)(=O)CC1 N1(C(C(C(C)(C)O)F)=O)C(C(=O)NC2COC(C(F)F)C2)C2CC(O)C1C2 c1(CC)nn(C)c(CC)c1CNC(=O)NC1(C(=O)O)CCOC2(CCC2)C1 CCCCC(C)(F)C(=O)N1CCC(COC)(NC(c2coc(OC)n2)=O)C1 CC1CCC(NC(c2ccccc2SCC#N)=O)CN1C(c1cc(Br)co1)=O c1(Nc2c(CN(S(C)(=O)=O)C)cccc2)n[nH]c2ccc(-c3ccc(O)cc3)cc12 c1(C(C(=O)NCC2N(C(CCOC(C)C)=O)CCCC2)O)ccc(Cl)c(Cl)c1 c1(N(C)C)cccc(NC(=O)NC2C=CCCC2CC(F)(F)F)c1 Cc1nc(C)n(CCC(=O)N(C23CC(NCC(=O)Nc4ccccc4Br)(C2)C3)C)n1 c1(C(CN(C)C(=O)NC2CCN2C(C)(C)C)O)ccc(S(=O)(=O)CC(F)F)cc1 N1(C(CCOC(C)C)=O)CC2CCC(C1)N2C(c1snc(O)c1Cl)=O c1(CCNC(C(=O)NCCC(c2cccc(F)c2)=O)=O)cc(F)ccc1Br c1(C(=O)NCC(CC)NC(C2(C)COCCOC2)=O)cc2n(n1)CCCC2 Cn1nc(C(=O)NC2(CNC(=O)CC3(N4CCCC4)COC3)CC2)cc1C(N)=O C1(NC(C(CC=C)CC)=O)CC1C1CCN(C(c2cnc[nH]c2=N)=O)CC1 C1(CCOC)(NC(=O)CCCn2cccn2)CCN(C(c2cc(C)on2)=O)C1 C(=O)(C1=C(C)CCCC1)NC1(CCOC)CCN(C(=O)CC2CCNC(=O)C2)C1 C(=O)(CCCCNC(=O)COc1ccncn1)N1C(C)CCC1 CC(CS(C)(=O)=O)C(=O)N1CC(CNC(c2ccc(F)cc2Cl)=O)C(C)(C)C1 c1(C(N(C2CCCN(C(C(C)SC)=O)C2)C)=O)cc(C)cc([N+](=O)[O-])c1N N1(C(CC2(C)CCCO2)=O)CC2C(CNC(=O)CCc3ccccn3)C2C1 C1(CNC(c2c(C)cco2)=O)CC12CCN(C(=O)CC1(C)CCS(=O)(=O)N1)CC2 c1(C(N(C2CCC(CNC(C3(O)CC3)=O)CC2)C)=O)cncnc1O N1(c2nc(C)nc(Cl)c2C)CC(NC(c2cn[nH]c2)=O)C(S(C)(=O)=O)C1 c1(C(=O)NC(CSCCNC(C=CC)=O)(C)C)ccc(NC=O)cc1 N1(C(C)=O)CCC(c2ncc(C(C)(C)C)[nH]2)CC1.C12CCCC1CN(C)C2=O c1(NC2C=CCN(C(CCCOCCOCC)=O)C2)cc(C(C)C)nc(Cl)n1 c1(C(N2CCC(NC(=O)Cn3cccn3)(CO)C2)=O)ccc(Cl)c(F)c1F N1(C(C(C)=C2CCC2)=O)CCCC2(CC(NC(=O)C3Cc4ccccc43)C2)C1 c1(C(=O)N)cccn2nnnc12.n1(C(C)C)nccc1NC(C1(C)CC1)=O CC1CC2CN(C(=O)C(N3CC4CCC4C3C(=O)NC)=O)CC12 C1(CNC(CC(C)SC)=O)CC(F)CN1C(=O)C(C)NC(c1cccs1)=O N1(C(C(COC)C)=O)CC(C(C2CC2)NC(=O)CN(C2CCC2)C)C(O)C1 N1(C(CC=CC=C)=O)CC(NC(c2conc2C(C)(C)C)=O)CCC1C C1(CNC(c2c(C)nco2)=O)CCCC12CCN(C(c1ccsc1C#N)=O)CC2 C(C)(CO)(C(=O)NCC(C)CN(C(=O)C=CCN(CC(F)(F)F)C)C)SCC Cc1cc(Cl)ccc1NNC(=O)N(CCCN=[N+]=[N-])C C1(CC)CCC(NC(=O)CCC2CCCN2C(c2cnco2)=O)CC1 Cc1ccc(NC(=O)C(C2CCCC2)NC(C2CCCOCC2)=O)cc1F C1(CNC(c2ccc(F)cc2)=O)CCCN(C(c2sccc2CO)=O)CC1 C(=O)(C1CCCc2c1ncn2C)NCC(C)NC(c1cc(C#C)cc(F)c1)=O C(c1ccncc1)=C(C)C(=O)NCC(C)CNC(=O)COCC1CCOC1 c1(C(=O)NC(C)C(C)NC(C2CCCC2n2cccc2)=O)ccc(Cl)c(Cl)c1 C(=O)(C#CC1(C)CCCO1)N1CCCC(F)(C(=O)NCC(C(C)C)N(C)C)C1 C1(CC(=O)N(CCCNC(C2(C(=O)OCC)CC=CC2)=O)CC)CCC(F)(F)CC1 c1(C(N2C(CN(C)C(c3cc(CCO)on3)=O)CC(F)C2)=O)cncc(Cl)c1Cl CC(=O)C(C)CC(C)C(=O)NC(c1cccc2c1OCCC2)C CCCC(C)(O)CC(=O)N1C2CCC(C2)C1C(=O)NCC1CCCCN1C C1(C2CCCCC2)(NC(C2N(C(C(CC)Cl)=O)CC(O)C2)=O)CC1 C=Cc1ccc(C(=O)N(C(CC)CC(=O)NC2CC2F)C)cc1 C#CCC(CC(=O)NCC(C)(C)COC)NC(=O)CN(CC)CCOC.OC c1(C(C)C)ccc(C(=O)NCCC(C)CCNC(C2([Si](C)(C)C)CC2)=O)cn1 c1(C(C=CC(=O)NCC(CCOC)NC(c2ccc[nH]2)=O)=O)ccc(F)c(F)c1 CCC(CC)CCCC(=O)N1CC(NC(=O)CNC(c2cscn2)=O)C2CC12 C1(NC(=O)OCC(O)CO)CCC(O)CC1 c1(CC(=O)NC2CCN(C(CCc3ccc(N)cn3)=O)C2)ccc2c[nH]nc2c1 N1(C(C(=O)NCC)C(C2CCC2)C2CC2)CCC2C(O)C(C)(C)C12 c1(CC)ncc(C(=O)NCC(=O)NCC(=O)Nc2ccccc2OC)cn1 N1(C(CC(=C=C)C)=O)C2CCC1C(C(=O)NCCC(C(C)C)OC)C2 C1(CC(N2C(C(=O)NC(C(=O)NCC)C3CC3)CCC2)=O)CCC(=O)NC1 c1(C(=O)NCC=CCNC(c2csc(Cl)c2)=O)ccccc1Oc1ccccc1 N1(C(C(CCC)O)=O)CCC(NC(=O)Nc2ccc(OC(F)F)cc2)C(C)C1 N1(C(C2CCC(CCC)O2)=O)CCC(C(C)(C)NC(c2cccc(=O)o2)=O)CC1 C1(C)(COC)CC(NC(=O)Cc2cccs2)CN1C(c1ccc(OC)nc1)=O C1(NC(CCC#CC)=O)CCCCC12CCN(C(c1ncoc1C1CC1)=O)C2 Cc1cc(C(N)=O)cc(C(=O)N(C)CCNC(C2(C#N)CC3CC3C2)=O)c1 c1(OCc2onc(-c3ccc(C)nc3)n2)c(-c2ccco2)nc2ncccn12 n1(CC)c(=O)sc2c(C(=O)Nc3cnn(CCC(=O)O)c3)cccc12 C(=O)(CC(C)C(C)C)NCCNC(c1c(C)snn1)=O c1(C(=O)NC(C(C)NC(C=CC)=O)C)cnn2c(C(F)(F)F)cc(C)nc12 c1(C(N2C(CNC(C3N(CC)CCOC3)=O)CC2)=O)cc2cc(F)c(Cl)cc2[nH]1 C(=O)(CC(C)(C)CNC(=O)CC(C)(F)F)NC(C#C)(C)CC C1(C(N2CCN(C)CC2CNC(=O)CC(C)(O)C2CC2)=O)COc2ccccc2C1 c1(C(N(CC(CN(C(CSCC=C)=O)C)O)C)=O)sc2nc(C)nc(C)c2c1C N(C1COc2cc(Br)ccc21)C(=O)Nc1cccc(SC)n1 C1(OC)CC(NC(C2OCCC2C)=O)CN(C(=O)Cn2cnnn2)C1 N1(C(=O)CC2(CO)CC2)CC2CCC1CN(C(C1(c3ccncc3)CC1)=O)C2 C=CCCCC(=O)NCC(c1ccc(F)cc1)NC(=O)Cn1nc(C)oc1=O c1(C(=O)NC2CCS(=O)(=O)C2)noc2c1CN(C(c1cc(C3CC3)[nH]n1)=O)CC2 C1(C(N2CCC(C(=O)NC3CC(C(C)C)C3)(CO)C2)=O)CC(=O)NC(C)C1 C#CC1(C(=O)NCc2cncc(C(=O)NC3CN(C)CC3C)c2)CC(=O)C1 C(CCCC(CO)NC(=O)C(c1ccc(F)cc1)F)NC(CC(=C=C)C)=O Cc1ccc(S(C)(=O)=O)cc1NC(=O)NCC1=NOC2(CCCNC2)C1 CCC(CC)C(C)C(=O)NCC1N(c2cc(C(N)=O)nc(Cl)n2)CCCC1(C)C C(=O)(C(C#N)C(C)(C)C)N(C)Cc1cc(C(N2C(CC)CCCC2)=O)ncc1 CCCCS(=O)(=O)NC(C1(C)CCN1C(=O)CNC(=O)C(Cl)(Cl)Cl)=O C1(NC(C2CCC(C)(CC)O2)=O)CC2CCC(C1)N2C(C1CCC2CC2C1)=O N1(C(C(CN(C)C)NC(=O)NC2OC(=O)CC2(C)C)=O)CCn2ccnc2C1 Cc1cc(Cl)nc(Cl)c1CNC1CC(CC(=O)Nc2cnccc2C(N)=O)C1 C=CCCC(C)(C)C(=O)NCC1CC1CC(=O)NCc1ccn(C(C)C)n1 c1(NC(=O)NCC(=O)NCC(CC)Cc2ccccc2)ccnc2ncnn12 C1(NCC(O)CN(C)C)CC(CC(=O)N(c2ccccc2)CCC(=O)OC)C1(C)C S(=O)(=O)(c1ccccc1F)N1CCCN(C(C(=O)NCC2CC2)CC2CC2)CC1 c1(C(N2CCC(CN(C)C(C3COC(=O)C3)=O)C2)=O)ccc(F)c(CO)c1 C1(NC(c2n(C=C)nnc2)=O)CCC(C)(NC(=O)CN(C)C(=O)C2CC2)CC1 N1(C(C2(CC#C)CCCOC2)=O)CCC(C)C(NC(=O)CCc2cnn[nH]2)C1 C12(NC(c3cnc(Cl)s3)=O)CCCC1CN(C(=O)Cn1ncc3ccccc13)C2 C1(NC(C(Br)=C(C)C)=O)CN(C(c2ccc(F)cc2F)=O)C2CCCCC12 c1(NC(C2(C=C)CCC2)=O)ccc(CNCCC(C)N2CCCC2)cc1 N1(C(c2ncc(CC)nc2)=O)CC(NC(=O)Cc2nocc2C(C)C)CCC1C c1(C(N(CCOC)CCNC(c2ncc(C(N)=O)s2)=O)=O)cccc(C(C)C)c1 CCCCC(O)C(C)C(=O)NCc1cnn(C)c1C(N1CCC1(C)C)=O C1(NC(C(CN(C(C2OCCN(C)C2)=O)C)(C)C)=O)CCCC(F)(F)C1 c1(NC(C2CCC2)=O)ccccc1NC(=O)COCCOC.CCC(=O)OC C1(C2CCOCC2)(C(=O)NC(C(C)NC(c2cnc(O)n2C)=O)(C)C)CC1 C(CCC(C)C(=O)NCc1cc(C(=O)NC2CC3(CC3)C2)ccn1)OC C(c1cn[nH]c1)=C(C)C(=O)N(CCC(C)NC(=O)C(F)F)C N1(C(CC(=O)NCC#C)=O)CC2CCC(C1)N2C(C1(C)CC=C(C)CC1)=O C(=O)(C1=CCCCC1)N(C1CCCN(C(=O)CC2CC3CC3C2)C1)CC c1(C(C(=O)NCC2CCCO2)N(C)CC2(OC)CCCC2)c(C)cc(C)cc1C N1(C(Cc2cc(OC)c(O)cc2)=O)CC2CCN(C(C3CC(CF)C3)=O)CC2C1 c1(C(N2CCC(CCN(C(C(C)SCC)=O)CC)C2(C)C)=O)n[nH]c(C)c1[N+](=O)[O-] C(C(=O)NC(c1ccccc1F)CNC(c1cnc(C2CC2)[nH]1)=O)(C(C)C)OC C1(CNC)CCN(C(=N)NC2CCCCC2)CC1 CC1(F)CC(C(=O)N(CCCNC(=O)CC2CCCO2)CC2CCCCC2)C1 c1(CC(N2C(CC(=O)NCC3C4CCCC34)CC2)=O)cccc2[nH]ncc12 C1(CCC(=O)NCCN(C)C(c2ccn(CCn3cccn3)n2)=O)CCC(=O)N1 c1(NC(=O)NC(C)(CO)C2CCCC2)cc([N+](=O)[O-])cnc1O N1(C(c2ccc(CC)s2)=O)CC(CO)C2(C1)CN(C(c1cscc1C(N)=O)=O)C2 c1(C(N2CCC(C)(NC(=O)CC3CCOCC3)C2)=O)cnc2c(c1)CNC(=O)N2 C=CCC(F)(F)C(=O)N1CCC(NC(C2(NC(=O)OC(C)(C)C)CC2)=O)C(C)C1 C1(CC)C(NC(c2cnco2)=O)CCN1C(=O)CCOCC(C)C C1(NC(c2c(C(C)C)ncnc2)=O)CCc2nn[nH]c2C1.C12CCC(C1)CNC2=O C(=O)(C1=CC2CC(C1)CC2O)NCC(CCCC)NC(c1cc(C(C)C)on1)=O c1(N2CCCC(NC(C(C)CSC(F)(F)F)=O)C2)ncnc2c1CCC2 c1(C(=O)NC2C(OC)CN(C(C3CCCC(CF)C3)=O)C2)c(C)cc(O)cc1C CCCCCC(CC)C(=O)NNC(C(N1CCN(CC2CC2)CC1)=O)=CCCC c1(C(=O)NCC2OCCC(NC(CCOC)=O)C2)cnn2cc[nH]c(=O)c12 N12CC(C3(CC3)C1)CC(=O)N(C)C(C)C2=O.c1(NSCC)cccn(C)c1=O CC(CCC(=O)NC1CCN(C(c2cc(C3CC3)nn2C)=O)C1C1CC1)N(C)C C1(S(C)=O)(CNC(N2C(C(=O)OC)CC2)=O)CCC1 C(N=c1nc2c(cnn2C)c(N2CC(=O)NC(C)(C)C2)[nH]1)c1n(C(C)C)cnn1 c1(-c2[nH]c(=N)sc2)ccccc1C(=O)OCc1nccc(C(F)(F)F)n1 C1(NC(C2(CNC(CCC)=O)CCC2)=O)CN(C(=O)OC(C)(C)C)CC1C c1(N2CCN(Cc3ccc(C)nc3C)C3C2C3)ccnc2ccnn12 N1(C(C(C)CC2CN(C(C3(C)CCNC3=O)=O)C2)=O)CCSC2CCCCC12 N1(C(c2cc(C)cc(Br)c2)=O)CC2CN(C(=O)C=Cc3ccc(O)cc3)CC2C1 c1(COC(c2c(Cl)ccc(F)c2O)=O)cc(F)cc2cccnc12 n1(CC)nnnc1C(C(C)Cc1ccccc1)NCCCOCCOC(C)C N1(C(CCCOCC=C)=O)CC2C(CNC(=O)CCN3CCC3)C2C1 CC1=C(C)C(N(C)CCNC(=O)NCc2ccn(C(F)(F)F)n2)CC1 N1(C(C(C=C)(C)C)=O)CC2CC(NC(=O)COCc3ccncc3)C2C1 C1(C(N(CCC=O)CC=C)=O)CCN2CCCC2C1.C(CCC(C)(C)CO)O CC(CC(=O)NCC(F)CNC(c1ccc(C(F)F)s1)=O)C1CCCC1 C=CC1(CC(N2CCC(C)C(NC(C3COC4COCC34)=O)C2)=O)CCCCC1 C(=O)(C=C1SCC(=O)N1C)NC1(COC)CCN(C(c2cnc(CCC)s2)=O)C1 CC(C)C(=O)N1CCC(C2CCCO2)C1.c12coc(c1)C2=O.S(C)(=O)(=O)NC C(CC(=O)N1CC(C)(C)CC1CO)(C(C)(C)C)NC(CC=C(C)C)=O C1(CC(=O)NCC(=O)NCCC)CCC1C(F)(F)F C(CCO)(C(C)(C)C)NC(C1CC(NC(c2cn(CCC)nc2)=O)C(O)C1)=O C=CCC(C(=O)NC1(CC(=O)N(C(CC)CO)C)CCCCC1)OC N1(C(C=CC(C)(C)SC)=O)CCC(C2CCCN2C(c2ccc(C(C)=O)o2)=O)CC1 c1(OCCN(C)C)ccc(C(=O)NCC2CC2CNC(C2CN(C)CCO2)=O)cn1 c1(SC)nc(C)c(CCC(=O)NC2CC(CNC(C3CC(O)C3)=O)C2)c(O)n1 c1(C(N(C(CNC(C2C(C#C)C2)=O)C)C)=O)ccc(O)nn1 N1(C(c2cnn(CC)c2C)=O)CCN(C(C2(C)CCCC2)=O)CC1C(C)(C)C S(=O)(=O)(c1cc(F)ccc1F)N1CC2CN(C(=O)Cc3ccccc3F)C2C1 N1(C(c2cc(OC)ncn2)=O)CC(C)CN(C(C2(C)CC3(CCC3)C2)=O)C(C)C1 N#CC1(C(N2CC3CC2(CNC(=O)CN2CCCC2CO)C3)=O)CCOC1 Cc1oc(C(N2CCC2CNC(c2ccc(CO)cc2)=O)=O)cc1S(C)(=O)=O c1(CC(=O)NCCC(C(C)C)NC(=O)CCC2CCCCC2)ccc2nsnc2c1 N1(C(C2C(C)CC2)=O)CCCC(CNC(c2csnn2)=O)C1 c1(OC)ncc(NC(N2CCC(Nc3nccc(SC)n3)C2)=O)cn1 c1(C(=O)OCC)ccc(CCNCC2COC2)nc1 C1(C(=O)NCCc2ccncn2)(NC(CC2C(CC)C2)=O)CCN(C)C1 C=CCCCCCCCC(=O)NC(Cc1cccc(C#N)c1C)C(=O)O C1(C(=O)NCCN(C(C2COCC3(CCC3)O2)=O)CC)CNC(=O)CC1C(F)(F)F C(C(C(=O)N(C)Cc1cnn(C)c1)NC(=O)CCn1ccnc1C)OCC C1(OC)CN(C(=O)C(C)OC2CCCC2)CC1NC(c1ccc(=O)oc1)=O c1(C(N2C(Cn3cc(-c4c(C#N)cccc4)nn3)C=CC2)=O)c(Cl)sc2nnsc12 C1(NC(c2n(C)cnc2)=O)CCC2CN(CC(=O)NCCn3cccn3)CC2C1 C1(CC(=O)NC(c2ccnn2C)CC)CCCN(C(c2cncc(C)c2)=O)C1 C1(C(=O)NC2(C)CN(C(=O)CN3CCCC3)C2)CC2(CO1)CC(F)(F)C2 c1(C(=O)NC2C(CNC(c3onc(CC)c3C)=O)CCC2)cc2sccc2s1 c1(C(=O)NCC(CCCC)NC(=O)Cc2csc(S)n2)cc[nH]c2nccc1-2 CC1=CC=CNC(=O)NCC1CCN1CC(OCCCO)C1=O C1(COC(c2c(CC)c[nH]n2)=O)CCC2COCCC2C1 CCC(C)(C)CCCC(=O)N1CCN(C(c2nc(C)ccc2F)=O)C2CC12 N1(C(C(=C)F)=O)CC(C(=O)NC(c2ccc(F)cc2)C(N)=O)CC(F)C1 c1(C(N(C(CNC(C2CC3CC3C2)=O)C2CC2)C)=O)csc(O)n1 N1(C(CC(CCC)CC)=O)CCN(C(c2sc(=N)[nH]c2CC)=O)CC12CCC2 N1(C(=O)C(N2CCN(CC(F)F)CC2)=O)CCCC(Cc2ccccc2)C1 C1(C(=O)NCc2occ(C(N(C)Cc3ccncc3F)=O)n2)CC2C=CC1CC2 N1(C(c2nccc(CC)c2)=O)CCC2CC2(NC(=O)Cc2ccc(F)cn2)CC1 c1(N2CC=CC(NC(C34CCC(F)(CC3)C4)=O)C2)ccc([N+](=O)[O-])cn1 C(C1CCOc2ccccc21)N(C(C(=O)NCC1CNC2(CCC2)C1)=O)CCO C1(OC)CC(CF)N(C(C2CC(O)CN2C(=O)CNc2ncccn2)=O)C1 c1(C(N(C)CC2N(C(CCC3CC(C)C3)=O)CCOC2)=O)c2c(nn1C)CCC2 N1(C(C2C(C)C2)=O)CCC(CNC(c2cc3sccc3n2C)=O)C(F)(F)CC1 c1(C(=O)Nc2cccc(C3CCCCC3O)c2)cc2cc(Cl)c(Cl)cc2[nH]1 C1(C(N2CC(CNC(C3N(CC)CC3)=O)(OC)C2)=O)CCC(F)CC1 c1(C(N2C(C(=O)NCC3(O)CCC(C)C3)C(O)CC2)=O)c[nH]c2ccncc12 Cc1ccc2ncc(C(=O)N(C)CCN(C(=O)CC(C)N3CCCC3=O)C)n2c1 N1(C(C(c2ccoc2)OCCN)=O)CC2CC2(C(C2CCC2)=O)C1.O=C1CN1 C(C(O)CN=c1cc[nH]c(-c2nccs2)n1)NC(C1C(C)OC(C)C1)=O c1(C(=O)NCC(C)N(C)C(c2csc(Cl)c2)=O)ccccc1S(=O)C(F)(F)F C1(CC(=O)NC)C2CN(C(=O)C(=O)Nc3ccccc3)CC12 N1(CCN(C(C)=O)C)CC(NC(c2nsnc2O)=O)CC12CCCC2 CC1CCc2ncc(C(N3CC4CC(N(C(=O)COCCCF)C)C3C4)=O)n2C1 N#CC1CCC(CNC(c2cc(CNC(=O)Cc3cnoc3)no2)=O)CC1 Cc1oc(C)c(S(N)(=O)=O)c1C(=O)NC1CCCC1NC(=O)COC1CCCC1 C1(C(=O)NCC(=O)OC(C)C)CCCN(C(=O)CC2CCCOCC2)CC1 S(=O)(=O)(c1ccc(=NCc2c(C)noc2C)[nH]c1)NCc1cc(C)sc1 CCCCC(O)CC(=O)N(C(C)(C)CC(=O)N(C)Cc1cc[nH]n1)C C1(CNC(C(=O)NCCC(N)=O)=O)CN(C(=O)CCNC2CCCCC2)CCO1 C1(CC(N2CCC(C(C)(C)NC(c3ccncc3)=O)C2)=O)CCC2(CC2)CO1 N1(C(c2c(C(C)=O)c[nH]n2)=O)CCOCC1CNC(C1CCCC1(F)F)=O CC(C)(C)C(CNC(c1csc(C#N)c1)=O)NC(=O)CCSCc1ccccc1 CC1CCC=C1C(=O)NC1CC(NCC(F)(F)F)C1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCC1(NC(CC=C)=O)CC1 C1(c2n(CC)nnn2)(NC(C)C)CCCN(CC#N)C1.c1(N)cccc(Br)c1 C1(C)(C(N2CC(CC(CNC(COc3cc(C)on3)=O)(C)C)C2)=O)CCC(=O)NC1 c1(C(=O)NCC(C)(C2CC2)NC(C2CCCC2c2nc(S)n[nH]2)=O)csc(O)n1 c1(C(=O)NC(c2occ(C(N(C3CCC(C)C3)C)=O)n2)C)ccccc1O c1(C(N2C3CN(C(CCCC(=O)OC)=O)C(CC3)C2)=O)cnc2ccccc2c1 C(C1CCCCCC1)=CC(=O)N(CC(CC)NC(C1CC(C(C)C)=NO1)=O)C C12(C(=O)NC3CCN(C(=O)OCC)CC3)CCCC1(F)CN(C(=O)C(C)C)C2 c1(CC(=O)NC(C2(CNC(CSCC(C)C)=O)CC2)C)ccsc1 c1(NC(C23N(C(C4OCCN(CC)C4)=O)CC(C2)C3)=O)cc(Cl)nnc1O CC1CCC(NC(C2C=CCC2)=O)CN1C(C1CCN(C)C1=O)=O C(=O)(C1=CC2(CCOC2)C1)N1CCC(NC(c2nc3ncccn3n2)=O)C(O)C1 C(=O)(CCCC(=O)NCC1(NC(=O)COC2CCOC2)CCOC1)NCC C(=O)(C(C)CS(C)(=O)=O)NCC1(NC(c2cc(C)c(C)o2)=O)CC1 C(C(CO)N=c1nc2c(ncn2C(C)C)c(NC(c2cnn(C)c2)C)[nH]1)OCC N(C1CCCOc2ccc(Br)cc21)c1nc(O)n(C)c(=O)c1 c1(C(=O)NCCN(C(=O)CCS(C)=O)C(C)C)nccc2cccnc12 c1(C(=O)NC(CN(C(CN(C2CC2)CC)=O)C)C)n[nH]cc1F C1(NC(CSc2n(C)ncc2)=O)CC12CCN(C(=O)C(=O)NCC(F)F)C2 C1(NC(C2(c3cccc(OC)n3)CC2)=O)CC12CCN(C(=O)CC(C)C(C)C)C2 CC1(C)CCC(C(N2CC(NC(c3ccc(CCF)cc3)=O)C2)=O)O1 N1(CCCCNC(C(c2n(CC)ncc2)N(C)C)=O)CCC(C)(C)C1C N1(C(C=C(CCC)C)=O)CC(NC(=O)C=Cc2nnn(C)n2)CC1(C)COC Cc1cc2ncc(C(=O)NCC34CC(CO3)N(C(C3CCC(C)O3)=O)C4)cc2[nH]1 C1(NC(C2OCCC(C)C2)=O)CC2CC(C1)N(C(C1(F)CC1)=O)C2 CCC(CC)(CO)C(=O)N1CC=CC(NC(=O)C(=Cc2cscn2)F)C1 c1(C(C)(C)C)nccc(C(N2CCC(CO)(NC(c3cn[nH]c3)=O)C2)=O)n1 C(=O)(C=CS(C)(=O)=O)NCC(c1ccccc1)CNC(C(C(C)C)F)=O c1(C(N2C(CNC(c3cn(CC(CC)O)nn3)=O)CC2)=O)ncc(OC)cc1F C(CN=c1cc(CC#N)nc(Cl)[nH]1)N(C(CCc1cnc(C)o1)=O)CCO.C=O C(=O)(C1=CSCCO1)N1C(CCNC(c2ccn(CC#N)n2)=O)CCC1 C1(C(N2CC(C(=O)OCCc3ccsc3)OC2=O)=O)CN2CCCN1CC2 Cc1ccc(Cl)cc1NC(=O)C(C1CCN(Cc2cnc[nH]2)CC1)C Cc1cc(F)c(C(=O)N(CC(C)CNC(C2CC3CCC2O3)=O)C)c(Br)c1 Cc1cc(C(N2CC(NC(c3cc(C)n(C(F)F)n3)=O)C(O)C2)=O)c(N)cc1F c1(CNC(c2nc(COC)oc2)=O)cc2c(s1)CCN(C(=O)NCC(C)(C)C)C2 C1(NC(c2c(C(C)C)noc2)=O)CCN(c2ncns2)C1C c1(NC(=O)CCCNC2CCN3CCCCC23)ccc2c(c1)OCCO2 C(=O)(C(C)(C)Cc1cccc(Cl)c1)NCC(c1ccccc1)N(C)C(C1CC(O)C1)=O c1(CC(C)C)ncc(C(=O)NCC2CC(NC(=O)CCC3CCCC3)C2)s1 C(=O)(C(C)S(C)(=O)=O)NC(CCNC(c1nn(CC)c(C)c1)=O)Cc1ccccc1 c1(C(N2CC(NC(C3CSC3)=O)(CO)C2)=O)ccc(Cl)cc1Br N(C1CCc2cc(CNC(c3ncsc3CN)=O)ccc21)C(CN1C(C)CC1)=O Cc1c(F)ccc(C(N2CCC(NC(c3cnsn3)=O)C2C)=O)c1Cl N1(C(C2(CCCC)CC2)=O)CCC(O)C(NC(=O)Cc2cn[nH]c2)C1 c1(C(N(CC(C)C)Cc2nnc3ccncn23)=O)cc2ccccc2s1 N1(C(Cc2c(C)con2)=O)CCCCC(CNC(=O)CCC2CCCCO2)C1 c1(C(=O)NCC(CNC(C=CC(=O)OCC)=O)(C)C)c(OC(F)F)cccc1Cl C(N=c1nc(O)c(Cl)c[nH]1)C1CCN(C(Cn2c(C(C)(C)OC)ncc2)=O)C1 C12(CNC(c3ccc(CCC)s3)=O)CC1CN(C=O)C2.c1ccn(C)c1CC N1(C(c2ncc(C)nc2)C(=O)NCCCF)CC2(CCC2)c2ccccc21 N12CC(N(C)C)CC1C2.C(=O)(CS(=O)(=O)NC1CC1)N.C(C=O)=CCN(CC)CC CC1(C)OCCNC1C(=O)Nc1ncc(Cl)cc1F Oc1c(F)cc(-c2cccc(CN3CCN(c4nc(Cl)ccc4Br)CC3)c2)cc1F c1(NC2CC(NCc3cc(F)c(OC)c(F)c3)C2)ncnc2[nH]cc(C#N)c12 C1(C(N2CC(CC(=O)NC(CC)CO)OCC2)=O)CCN(C)C(=O)C1 c1(OC)ccc(C(=O)NC(C)CN(C(=O)C=CCN2CCCC2)C)c(OC)c1C C1(CC)CC(C(=O)N(C)CC2CC(O)C2)CCN1C(c1cc(C)cs1)=O C1(C(N2CCC(c3cnn[nH]3)C2)=O)(CNC(c2n(CC=C)ccc2)=O)CCCCC1 Cn1nc(C(N2CCCC(CO)(NC(=O)CCC3CCOC3)C2)=O)cc1C#N N1(C(C(SC)SC)=O)CC(C)(C)CC1C(=O)NCc1nonc1CO c1(C=O)c(C(F)F)c(C(F)(F)F)nn1C.C(C(C)(C(=O)OCC)OC)OC CCC(F)(F)C(C)(C)C(=O)NCC1(C)CCC(NC(c2cnc(SC)s2)=O)C1 C(=O)(C1=CC2CCC(C1)C2)NC(C1CC=CCC1)C(=O)N(C)CCN1CC2CC2C1 C(=O)(N1CC(O)C(O)CO1)C1CCN(C(C(C)OCCC=C)=O)CC1O C1C(CC2CCCC2)C(=O)N1.C1(CNC(COCCC#C)=O)CCOC1C(C)C C12CC(C13CCC3)NC1(CC3(CC3)C1)C(=O)N2.Cc1noc(CN)n1 C(C1CC(=O)Nc2ccccc21)Nc1ccc(C(=O)NCC(N)=O)cc1 c1(OC)ncc(C)cc1NC(C1CC(NC(=O)Cc2ncccc2F)C1(C)C)=O c1(C(N2CC(NC(c3c(CC)[nH]cc3)=O)C(C)C2)=O)cc2c(Cl)cccc2[nH]1 c1(C(=O)OC)cc2c(Nc3cccc(SC4CCN5CCC4C5)c3)nccc2o1 CC(C)CC(C(=O)NC(C)CC(C)NC(=O)CC(C)(C)CC(F)F)C(C)C CC12COCC1(C)CN(C(=O)CCC1CCC(NC(c3c[nH]c(=N)o3)=O)C1)C2 C1(COC)(NC(=O)CC2(C)CC2)CCN(C(=O)CN2CC(F)(F)C2)C1 C1(C(=O)NC2CC(CC)C2)CC(O)C(O)CC1CNC(=O)CC(F)F N1(C(C2C(C=CC)CN(C(=O)CCCCCOC)C2)=O)CC2CCC1C(O)C2O CC(C)(CNC(=O)CCCOc1ccccc1Cl)CCNC(C12CCCC1C2)=O c1(C(C)C2CC2)nc(-c2cn[nH]n2)n(C2CCN(C(=O)OC(C)(C)C)C2)n1 C1(CN(C)C(c2cc(Cl)cs2)=O)C2CN(C(c3cc[nH]c(=N)n3)=O)CC12 C1(OC)CC(CSC)N(C(C2(N(C(=O)C(C3CCC(=O)C3)C)C)CC2)=O)C1 N1(C(COC(CC)CC)=O)CCC2(CC1)CC2NC(=O)CNC(c1cccs1)=O C(=O)(C(CNC(c1cc(O)ccc1C)=O)C(C)(C)C)NCCCOCC c1(C(N2C(CNC(CCCC(=C)C)=O)C(O)C(O)C2)=O)cc(S(N)(=O)=O)oc1C N1(C(C2(CC=C)CCCC2)=O)CC2ON=C(CNC(=O)Cc3cc[nH]n3)C2C1 N1(C(c2ccnn2CC(F)(F)F)C(=O)NCCCC2CC2)CCOC2CCCC12 n1(CC)nc(C(=O)N(C)CC2COCCN2C(=O)C=CSC)cc1C1CC1 C1(CCCC)CN(C(c2csc(Cl)n2)=O)CCN1C(C1(OC)CCCOC1)=O C(N=c1cc(C#N)[nH]c2ccccc12)c1ccc(OCC=C)cc1 N1(CC(=O)NC(C2CCCC2)CNC(c2ccc(=O)oc2)=O)C(=O)CCCC1=O C1(OC)(CNC(=O)COC2CCC2)CCN(C(=O)CC2CCOC2(C)C)CC1 N1(C(C2(SC)CC2)=O)CC(CNC(=O)COc2ccc(C#N)cc2)C2(CC2)C1 CCCCC(C)C(=O)N1CC(NC(c2cc(N)cnc2C)=O)C(C)C1 n1(CCCC(=O)NCC(C2CCOC2)NC(CC2CC(SC)C2)=O)nc(C)cc1C N1(C(C(CC)NCC)=O)CC=C(CCNC(C2CCCCN2C(N)=O)=O)CC1 c1(C(=O)NCC(C(C)C)NC(C(C2CCCC2)OC)=O)cnn(C(C)C(C)C)c1C CCS(=O)(=O)C=CC(=O)NC1CCC(CNC(c2cc(C(N)=O)[nH]n2)=O)C1 c1(CC)nc(=NCCC2CN(C(C)=O)C2)s[nH]1.N12CCC(C)C(C1C)C2=O C(c1ccc2c(c1)COCC2)=Cc1onc(C(C)(C)C)n1 Cc1cc(C)c(C(=O)NCC(C)CC(=O)NCCCCCCO)s1 c1(CC(=O)NCC(C)(C)N(CC(C)C)C(C2CC2C(N)=O)=O)ccccc1.CO N1(C(=O)NC(CCC=C)C2CC2)CCc2cc(C)cc(C)c21 C1(NC(=O)C(O)C2CN(C(C3CCC4(CCC4)C3)=O)C2)CC(C2CCC2)C1 N1(C(C2(CC=C)CC=CC2)=O)CC(C2(NC(=O)C(C)N(C)C)CC2)C1 N1(C(C(CC)F)=O)CC2CCC1CN2C(c1c(C)nn(C)c1-n1ccnc1C)=O C1(C(=O)NC2(C(C(C)C)O)CC2)CCCN1NC(=O)CCC(N)=O C(=O)(CCN=C(NCC(C)C(C)(F)F)NCC(C)(C1CC1)OC)NC N1(C(CCc2cc(C)on2)=O)CCC(F)(CNC(C2C3COCC23)=O)CC1 C1(NC(=O)Cc2ccc(C(F)(F)F)cc2F)CC2CN(C(=O)CSC(F)F)CC2C1 C1(CC(C)C)(C(=O)NCC2CC(C)N(C(c3csc(Cl)n3)=O)C2)CCNC1=O Nc1cc(C(=O)NC2CCCCC2CNC(c2nc(Cl)ccc2F)=O)nc(O)c1 C1(NC(c2c(CC)nco2)=O)CC2CC(C1)N(C(=O)CC1CC(C)(C)C1)C2 C1(NC(c2c(C)cncc2)=O)CC2CCC(C1)N2C(c1cc(CO)[nH]n1)=O N1(C(c2c(CNC(c3ncncc3Cl)=O)ocn2)=O)CCn2cncc2C1 CC1(C)NC(=O)CC1C(=O)NC1(CNC(c2cnc(C3CC3)s2)=O)CCCC1 c1(OC)cccc(OCCC(=O)NC2CN(C(=O)C=CCSC)CC2C)c1 c1(C(C)(C)C)cc([N+](=O)[O-])cnc1N1CCC(n2ccnn2)C(F)(F)C1 N1(C(C2(F)C(C)(C)C2(C)C)=O)CCC(C2(O)CN(C(c3cccnc3)=O)C2)CC1 N1(C(c2cc(CC)oc2C)=O)CC2CCC(NC(C3CCCCS3)=O)CC2C1 CC1C(NC(=O)Cc2cn3ccsc3n2)CCCN1C(C1CC=CCC1C)=O C1(F)(C(=O)NCC(C)F)CN(C(c2cc(C3CC3)[nH]n2)=O)C1 N1(C(C=C(CC)CC)=O)CCCC(C)(CC(N2CCC2C2CCCC2)=O)C1 c1(C(N2C3C(NC(C=C(C)C)=O)CC(C3)C2)=O)cc(C)cc2ccncc12 C1(c2nnnn2CCCOC)(NCc2cccc(OCC=C)c2)CCCC1(C)C CCCCC(CNC(C1CCCCN1C)=O)NC(=O)CC1CCCC1C N1(C(C(CCC)C)=O)CC(NC(=O)CNC(c2cccc(N)c2)=O)CC2(CCC2)C1 Cc1cc(C(N2CCC3CC2CN(C(c2ncccn2)=O)C3)=O)cc2nc[nH]c12 CC(C)CC(C(=O)Nc1cccc(F)c1)N1CCNC(=O)C1 C1(NC(CC2(CC)CCOCC2)=O)CN(C(c2cccnc2O)=O)CCC1C Cc1cc(C(=O)NCC(CC(C)C)NC(C2CC3(C2)CC3F)=O)oc1C C(=O)(C(C)(C)C(c1nnnn1C)NCc1nncn1C(C)C)OC CC1(C)CCN(C(C2CCC(=O)C2)=O)CC1CNC(c1coc(Br)c1)=O c1(COC)ccc(OCCOC(=O)C=CC(=O)NCc2ccccc2F)cc1 N1(c2nc(C)cc(C)n2)CCc2ccc(NC(c3snc(C)c3N)=O)cc2C1 c1(C(=O)OC)cc(C)nc2onc(Cc3ccccc3)c12.C1(C(F)(F)F)C(C)C(=O)N1 N1(C(C(CC)O)=O)CC(F)(F)CC1(C)CNC(=O)Cc1ccc2nc[nH]c2c1 N1(C(CCCC=C)=O)CCC(C)C(CC(=O)N(CCC)C(C)C)C1 C1(NC(C2ON=C(C)C2)=O)CCC(F)(CNC(=O)CC2(c3ccccc3)CC2)C1 C1(N(C)CC)CCN(c2nccc(NCCOc3cccc(F)c3)n2)CC1 C1(C(=O)OC2C(CNC(C3(CSC)CC3)=O)COC2)CC(=O)N(C2CCCC2)C1 C1(F)(CNC(c2cc(CCO)on2)=O)CC(CNC(C2(F)CCC2)=O)C1 CN(CCCC(=O)NCC1C=CCN1C(C1CCCCO1)=O)N=O c1(C(c2ncco2)OC)nc(C(=O)NCC2(NC(=O)C3CC3)CC2)co1 Cc1csc2cc(C(N3CCC(NC(=O)CC(C)(C)CC(F)F)C(C)C3)=O)[nH]c12 CC1CCN(C(=O)C(C)(C)C#N)CC1NC(=O)CC1CCCCC1 c1(CC(=O)NCC2N(C(C(C)SC)=O)CC2)ncc(C)o1 C1(CC(=O)NC2(CC(=O)OC)CC2)C2CCCC2N1C(c1cccc(N)c1)=O c1(NCC)scnc1C(=O)NC(C)CNC(C12CCC1C2)=O C1(C(N2CC3C(CNC(CC(C)(C)OC)=O)C3C2)=O)CCCC(=O)CC1 N1(C(c2c(C)noc2)=O)CCC(C)C(NC(c2cc[nH]c2C2CCC2)=O)C1 Cc1ccc(Cl)cc1OCC(=O)NC1CCC(C)N(C(=O)CCC2(C)CC2)C1 n1(CCNC(=O)CCNC(C2CC2(Cl)Cl)=O)ncccc1=O Cc1nn(CC(=O)NCC(CNC(C2(CC(C)C)CCC2)=O)CO)cc1Cl CCCCCC(=O)NCC(=O)NCCC1COCCN1C(=O)CSCCC N1(C(c2c(C)oc(-c3cnn(C)c3)n2)=O)CC(CNC(=O)C2CC2)C(F)(F)C1 C=CC1CN(C(C2CCC(C)CC2)=O)CC1NC(C1CC2CCC(C1)O2)=O C1(C(N2CCC(O)(C(F)(F)C(=O)O)C2)=O)C2CCC1N(CC1CCCO1)C2 C(=O)(CC(CC(=O)O)c1ccc(Cl)cc1F)NCc1cccc(COCCOC)c1 S(=O)(=O)(c1ccccc1F)N1C(COC(=O)Cc2c[nH]c3cccnc23)CCC1 Cc1c(C(N2CC(CNC(=O)C3=CCC3)C(O)C2)=O)nnn1CC1CCCC1 N(C(=NCCC(C)C)N1CCC(c2ccc(F)cc2)C1)C(C#C)CCC N(C1CCc2ccc(F)c(F)c21)C(c1n(C(C)C)nnn1)c1cn(C2CCC2)nn1 N1(C(CC2CCCN(C(C(C(C)N(C)C)N(C)C)=O)C2)=O)CC2CC=CCC2C1 c1(CC(=O)N(CC(C)O)CCNC(=O)CCC2CCCC2)ccc2oc(O)nc2c1 C(=O)(C1=CCC(NC(C2(CF)CC2)=O)C1)NCCCC1C(C)C1 C1(NC(c2ccc(Br)cc2)=O)CN(C(C2(CCF)CC2)=O)CC1n1cccn1 c1(C(=O)OCC)cc(C)nnc1NC(CNC(=O)C(C)Cc1ccncc1)CC N1(C(C(OC)OC)=O)CCC2(CCCC2NC(=O)CS(N)(=O)=O)CC1 S(=O)(=O)(c1ccc(N2CCc3sc(C)cc3C2)cc1Br)NCc1c(C)ccnc1 C1(C(N(C)C)=O)CCN(C(=O)NCC2C=CCCC2)C1 N1(C(CC(=C)C)=O)CCCC12CCN(C(C1CC(=O)N(C3CCCC3)C1)=O)C2 N1(C(C(F)=C(C)C)=O)CCN(CC2(NC(C3COC(=O)N3)=O)CC2)CC1 c1(C(=O)NCCCN(C(C(=O)NCC)=O)C2CC2)ccc(S(=O)(=O)N(C)C)o1 c1(C(=O)NCC(C)(C2CC2)NC(CC(=O)NCC#C)=O)c(C)ncnc1C N1(CC(N2C(CN(C)CCc3cccc(F)c3)CCC2)=O)C(=O)CNC1=O CC1CN(C(=O)CCn2cccn2)CCN1C(=O)CC1CC=CCN1C C1(C(=O)NC(c2nncs2)C)CCN(C(C2OCCC2C)=O)C1 c1(C(N2C(CNC(c3ccc(C)o3)=O)C(C)CC2)=O)cnn2c1OCC(C)(C)C2 C(=O)(C1=CC2CCCCCC12)NCC(C(C)C)NC(CNC(=O)OCC=C)=O C(=O)(C(C)(CNC(=O)CCn1ccnc1)CC)NC(C=C)CO Cc1cc(-c2noc(CN3CCCC3C3(C(C)C)CC3)n2)ccc1F c1(CCCC(=O)NCCC2(CNC(=O)Cc3nncs3)CC2)ccc(F)c(F)c1 NC(=O)CC(O)C(=O)NCc1ocnc1C(N1CCCC(N2CCC2)C1)=O c1(C(=O)NC(c2ccccn2)CN)ccc(SC2CCOCC2)nc1 C12(C(N(C3CCN(C(CSC4(C)CC4)=O)C3)CCO)=O)CC(CO)(C1)OC2(C)C c1(C(=O)NCCN(CCC)C(c2nnc(S)s2)=O)cc(OC(F)F)n(C)n1 Cc1sc2ncnc(NC3(C)CCC(NC(=O)C(C(C)C)N(C)C)CC3)c2c1C N1(C(Cc2ccc(CCC)s2)=O)CC2OCCCC2(C(=O)NC(C)(C)C)C1 N1(C(c2c(C)cc(CC)o2)=O)CC2CCCC1CN(C(c1cc(Cl)nn1C)=O)C2 C1(CC(C)C)CNC(=O)C(C)OC2(CCSC2)C(=O)N1.c1(COC)ccccc1 C(=O)(CCCCC(C)(C)C)NC1CC(CNC(C(C=C=C)C)=O)CC1O c1(C(=O)NC2CN(C(C3CCCS3)=O)CC2F)ccc2nccnc2c1 N1(C(c2c(C)occ2)=O)CCN(C(=O)Cc2nncn2C)C(C)C1C CC(C(=O)NCC1(CNC(=O)Cn2cc(C3CCCCC3)nn2)CC1)C(C)(C)C c1(C(c2nn[nH]n2)N(C(=O)Cc2csc(C3CCC3)n2)CCO)nc2ccccc2[nH]1 c1(OC)ccc(CC(C)C(=O)NC(C)(C)CCNC(c2cncs2)=O)cc1 C(=O)(C1CCCc2cncn21)NCc1c(CNC(C2(OC)CC2)=O)cccc1 c1(-c2cn(CC(=O)N(C(C)Cc3ncoc3C(F)(F)F)CC)nn2)cc(Cl)ccc1F C1(C(C)NCc2ccc(-n3cccn3)nc2)CCc2nnc(CN(C)C)n2C1 C1(CCOC)(NC(=O)C=CCF)CCN(C(=O)C(O)CC2CCCCC2)C1 N1(C(Cc2c(C)nc[nH]2)=O)CC2(CCC2)CC1CNC(c1cc(Br)n[nH]1)=O C#CCC(C(=O)N1CCCC1(C)CO)NC(c1coc(CO)c1)=O C(=O)(CCC1=NNC(=O)CC1)NC(C)CNC(c1cncc2[nH]ccc12)=O c1(CC(N2C(C(=O)NC3CC(CC)(CC)C3)CC2)=O)ccc(Br)cc1 Cn1cc(Br)c2c(C(N3CC(C)(C)CC3CNC(=O)C3=CCC3)=O)ncnc12 N1(C(=O)OCCC(C)C)CC2CN(C(=O)CCCc3ccc(Cl)cc3)C2C1 N1(C(c2cccc(C(C)C)c2)=O)CCC(NC(c2ncsc2C2CC2)=O)C(F)C1 N12CCC(F)(F)C(C1)C2=O.c1(C(=O)Nc2cncc(Br)n2)cc(O)ccc1O C(=O)(CCC1CCCO1)NC(C1(CC(=O)OC)CC1)=O CC1=C(C(=O)N2CCN(C(=O)C(C)C#N)CC2CC2CCCCC2)CCC1 CCCCC(C(=O)N=c1cc2ccccn2[nH]1)NC(=O)C(O)CC1CCCC1 N1(C(CCOC)=O)CC(CNC(=O)Cc2ccn(C(F)F)n2)CC1(C)C c1(C(N2CCCC(N(CCc3c(C)ncs3)C)C2)=O)c[nH]c2ccccc12 N1(CCC)CCCC(c2ccccc2)C1.N12CCCCC1c1n[nH]cc1C2=O c1(C(=O)NCC2CN(C(C3CCC(CC)O3)=O)CC2C)ncnc2c1CCC2 CCS(=O)CC(=O)NCCC(Cc1ccccc1)NC=O.c1(C(=O)N)cnc(CO)s1 c1(C(N2CC(NC(C(c3ccccc3)C)=O)C(O)C2)=O)cc(Cl)c(F)cc1F C(=O)(CCNC(c1cc[nH]n1)=O)N(CCCF)CC c1(CN2CC(C)N(C(C34CCC(CC3)CC4)=O)CC2)ccc2c(c1)OCO2 c1(C(=O)NCCC(CCNC(C(=Cc2cnc[nH]2)C)=O)C)cc(CO)ccc1Cl C1(CNC(C(=Cc2cnc[nH]2)C)=O)CCCN(C(C2CCCCC2)=O)C1 c1(C(N2CC(CCNC(c3c(C)snn3)=O)OC(C)C2)=O)ncnc2c1CCC2 C1(NC2CN(C(CN(C)CC)=O)C2)CCNC1=O C1(F)(CNC(=O)CCN2CCC2)CCC(CNC(c2cc(CCO)on2)=O)CC1 C1(CC)CC(CC(N2CC(CNC(=O)C(C)CCc3ccc(F)cc3)C2)=O)CCO1 C=Cn1nccc1C(=O)NCC(C)(C)OCC(=O)NCC1COC(CO)C1 C1(c2n(CCOCC)nnn2)(NCCCn2nc(C)nc2C)CCC(C)SC1 C(=O)(CCC(C)(F)F)N1CCCC(CCNC(COCCC)=O)C1 C(=O)(C(C)(C)CC(F)F)NCCC1CCN(C(C2(C)CCC(C)C2)=O)CC1 C1(C(=O)NCC(CC)NC(C2C(C)(CC)C2)=O)CSCCS1 C1(C(C)C)CN(C(c2scnc2Cl)=O)CCN1C(C1CCCN1C)=O c1(C(=O)NCC2C(CC)CCN2C(=O)Cc2cnn(C)c2)nnc(O)nc1O c1(C(N(CC(C)NC(C2CCN(CC)C2)=O)C)=O)cnc2c(ccn2C)c1 c1(C(=O)NC2CN(Cc3ccc(F)cc3)CCC2(F)F)cccc2nc(Cl)sc12 C(C(C(=O)N(CCCOC)CC1CC1)C(C)C)NC(c1cc(C(C)C)no1)=O C12(CNC(C3CCSC3)=O)CC1CN(C(c1cn(-c3cccc(F)c3)nn1)=O)C2 C1(CC(=O)NC2CN(C)C(CO)C2)C2CCCC2N1C(C1(n2cnnn2)CC1)=O c1(NC(C(=O)Nc2ccc(C(CC)(C)C)cc2)=O)cccc(-c2nnco2)c1C CC1COCC2(CCN(Cc3cn(-c4ccc(Cl)c5ncccc45)nn3)C2)O1 N1(C(C2CN(C(c3n[nH]c4c3COC4)=O)C2)=O)CCCC2(CCCNC2=O)C1 C(=O)(C#CC1CCCCC1)NCC1N(C(c2cc(C(C)C)[nH]n2)=O)CC1C(C)C c1(C(=O)NC2CCC(NC(CC3C(C)(C)CCO3)=O)CC2)cccc2ncsc12 CCC(C)C(C(=O)NCCCOCCNC(c1coc(C=O)n1)=O)SC.C1CC1 CC(CC(=O)NCC1CCC(C)N(C(=O)C2CC2)C1)C(F)(F)C(F)(F)F N1(C(C(CC#C)NC(=O)CC2C=CCC2)=O)CCC(C(=O)OC)(COC)CC1 C12(C(=O)NCC(C)CN(C)C(c3csc4nccn34)=O)CCCCN1CCC2 C(N=c1cc(C)nc(C)[nH]1)C1CCN(C(C(CC)Cc2ccccc2)=O)C1 C(=O)(C(C(=O)NCCCC(C)NC(=O)CN(C)C(c1ccsc1)=O)OC)OC c1(OC)ccc(Cl)c(Nc2ccnc(N3CCC(C(=O)NC)CC3)n2)c1 c1(OC)ccc(Cl)c(C(=O)N(C2CN(C(C3CCCCC3C)=O)C2)C)c1 N1(c2cc(N(C3CCC(C)(C)C3)C)ncn2)CCC12CCSCC2 c1(CC)cn2c(C(=O)NCCC3(O)CN(C(=O)CC4(C)CC4)C3)cccc2n1 O=C(N=c1[nH]nc(Cl)cc1O)C1CCc2cncn2C1 C1(NC(=O)CCF)C=CCN(C(c2ccc(C3CC3)o2)=O)C1 C1(N(CC)Cc2ccccc2OC)CC(=O)N(C2CC2)C1c1ccc(Cl)c(F)c1 N1(C(C)=O)CCCCC1C(N1CCCCC1CCNC(=O)CCn1ccnc1)=O CC(CNC(=O)CCCF)(CO)NC(=O)CCCc1ccsc1 CC1Cc2cc(C(=O)N(CC(C)(C)CNC(C3CCS(=O)(=O)C3)=O)C)ccc2O1 C(CC(C(=O)N1CC(CCNC(=O)C(C)(F)F)C1)N(C)C)SC Cc1cc(C)c(C(N(CC(C)NC(c2ccccn2)=O)C)C)o1 C1(CC)(NC(c2cc(C)n(C)c2C)=O)CCN(C(c2ncccc2F)=O)CC1 C(=O)(C(C#N)C(C)(C)C)NC(CC)(CNC(=O)COc1ccc(F)cc1F)CC c1(SC)cccc(NNC(=O)Nc2ccc(-n3cccn3)c(F)c2)c1 c1(SCC(=O)NC2CCCN(C(C3CC4(CCO4)C3)=O)C2)cc(Cl)ccc1Cl Cc1cccc(C=CC(=O)NCCCN2CCN(C(=O)C3=CCCC3C)CC2)c1 C1(C(=O)NC(C)CSC(F)F)CCN(C(C2(C)CCCCC2)=O)CC1 N1(C(C)C)CC(C(=O)N(C(C)CN(C(=O)Cc2cccs2)C)C)CC1=O N1(c2ncc(C(=O)NC3C(C4C(C)C4)C3)s2)CCCC2CN(c3ncc(O)cn3)CC12 N1(C(CC(C)C)=O)C(C(=O)NCc2cccnc2)CC2CCCCC12 C1(CN(C)C)CCN(C(C2CCC=CC2NC(c2cscc2F)=O)=O)CC1 O=C(O)C(F)(F)CNC(C1CNC(=O)CO1)=O c1(CC(N2CCN(C(c3noc(CC)c3C)=O)CC2)=O)ccc2ncsc2c1 N1(CCNC(c2cnn(CC)c2)C(=O)OCC)CCC23CCC(CC12)C3(C)C c1(C(=O)NCC2CCC(C)N(C(=O)C(Cl)=CCl)C2)ccc2occc2c1 C=CC1(C(N2CCN(C(C3CCOCC3)=O)C(C)C2)=O)CCCCC1 C(CC(=O)NCC1CC2C(C1)C2(F)F)(C(C)(C)C)NC(C(C(C)(C)C)=O)=O c1(OC)ccnc(OC)c1C(=O)NCC(O)CNC(c1cc(F)cs1)=O C1(NC(c2cnc(C(C)C)nc2)=O)CCN(C(=O)CCC2CC2(Cl)Cl)C12CC2 c1(C(=O)OCc2ccccc2)cccc(OC2CCS(=O)(=O)C2)c1Cl C1(SCC(=O)Nc2cc(Cl)ncn2)CCc2nnc(O)cc2C1 C1(C(N2CCC(NC(c3cccc(CC)c3C)=O)CC2)=O)CCc2cnnn2C1 c1(CNC(C(N2CCN3CCCC3C2)C(C)C)=O)ccc(S(N)(=O)=O)o1 C1(CC)CCN(C(=O)CCc2ccccc2C)C12CC2.N12CC(CC1=O)NC2=O Cc1cc(C)c2nc(CN3CC(c4cc5c(s4)CCCC5)C3)cn2c1 N1C(=NCc2cc(C#N)ccc2F)N2CCCC(C1CCC)C2.C=CC C1(CO)CCCOCC1.CC1CC(=O)OC2(C(=O)OC(C)(C)C)CC1C2 c1(N(N2CCC(CC(=O)O)C(O)C2)C(C2C(C)CC2)=O)cccc([N+](=O)[O-])c1 Cc1nc(C(=O)NCC2C3CN(C(=O)CCOCC(C)(C)C)CC23)nn1C CCC(CNC(=O)C(=O)NCCN(c1ccccc1)C)CO C1(NC(C(=O)NCC)=O)CC2CC1CN2C(C1CCCN1C(C)C)=O c1(OC)nc(C)ccc1C(=O)N(CCCCCNC(C1CC(C)N(C)C1)=O)C N1(C(C2(F)CCN(C(c3c(C(C)C)occ3)=O)C2)=O)CCOC(C)(C)C1C CC(CCC(C)(C)C)C(=O)NC(C)(C)CC(=O)Nc1cccc(C#N)c1 C(C)(C)(C#Cc1ccccn1)NCc1cn(C)nc1-c1cccc(Cl)c1F C1(C)(CNC(C2(OC(C)C)CCC2)=O)CCN(C(C2(C)CC2(F)F)=O)C1 CCC(C)(CNC(=O)CNS(=O)(=O)NC)NC(c1cc(C)c[nH]1)=O Nc1cc(Cl)cc(Cl)c1C(=O)NCCOCCNC(=O)Cn1ccc([N+](=O)[O-])n1 c1(C(N2C3C(NC(c4nc(CC)sc4)=O)CC(C3)C2)=O)cccc2c1ccn2C N1(C(C2(C(F)F)CCC2)=O)CCOC(CCNC(c2ccccc2F)=O)C1 CC1CN(C(=O)C(O)CNC(N)=O)CCC1N(C(=O)C=Cc1cc[nH]n1)C c1(C(N2CCC(O)(CNC(C=Cc3scc(C)n3)=O)C2)=O)cccc2oncc12 CC1CN(C(c2cc(=N)[nH]c(Cl)n2)=O)CCC1CNC(c1nocc1Cl)=O CCCCCC(CC)C(=O)N(CCC(=O)NC1CCCC(F)(F)C1)C C1(CN(C(=O)C(C#N)C2CC2)C)CCN(C(C23CC(C(C)(C)C)(C2)C3)=O)CC1 CCCCCC(F)C(=O)NC(C)C(C)NC(=O)C1=NOC(C)C1 Cc1cc(CCC(=O)N(C2CC2)CC2CCCO2)cc(C)n1.C1(=O)C(F)CC2CN1C2 N1(C(CC(=O)NCC)=O)CCCC12CCN(C(=O)Cc1sc(CO)nc1C)C2 c1(C(N(C2CCCN(C(C(c3cccnc3)C)=O)C2)C)=O)ccc2n[nH]cc2n1 CCC(Cc1cccc(Br)c1)C(=O)N1CCC(C(c2ccc(Br)cc2)=O)CC1 C1(NC(Cc2nc(C(C)C)sc2)=O)CN(C(=O)C(N2C(=O)CCC2=O)C)CC1C C1(C(N2CC(C)(NC(C3CCCC3CF)=O)C2)=O)(NC(C)=O)CCCC1 C1(C(N2C(C(=O)NCC(=O)OC)CCC2)C(=O)NC(C)C)CS(=O)(=O)CCO1 C(=O)(CCCC(=O)c1ccccc1)NCCC(C(C)C)NC(C1(COC)COC1)=O c1(NCC2(C(=O)NC(c3cncnc3)C3CC3)CC2)c(Cl)cccc1I C1(C(=O)NC(c2ccccc2)(C)C)CN(C(C2CCCC3CC23)=O)CCO1 C1(C(=O)NCC2(CN(C)C)CCCC2)CCN(C(=O)C2(C#N)CCCOC2)O1 N1(C(Cc2c(C)c(C)no2)=O)CCC(C)C(NC(C2CC(OC3CC3)C2)=O)C1 Cc1ccc(-c2nc(C(=O)N(C(C)CN(C)C(c3ccsc3C)=O)C)cs2)cn1 C1(NC(C2(O)C(C)(C)C2)=O)CN(C(C2CCN(C(N)=O)CC2)=O)CC1O c1(-c2onc(-c3cccc(N(C)C(C4CCC4)=O)c3)n2)ccc(F)c2[nH]ncc12 C(=O)(C1=CCCOCC1)N1CC2CC(C(=O)Nc3c(C)ccc(Cl)c3)(C1)C2 c1(C(=O)NCC2(CN(C(C(C(C)OC)O)=O)C)CC2)c[nH]c2cc(F)ccc12 CC1CC2CN(C(C3CC34CCCC4)=O)CC2N1NC(c1cncnc1C1CC1)=O CCC(C(=O)NC1(C(C)NC(C2CC2Cl)=O)CC1)C(C)C c1(C(N(CC(O)CNC(c2cnncc2O)=O)C)=O)cc2cccc(Cl)c2[nH]1 c1(OC)c(C(N2CC3CC2C3CNC(=O)C(C)C2CCCC2)=O)ccnc1Cl Cc1cccc2cc(C(=O)NC3CN(c4nccc(C(N)=O)c4[N+](=O)[O-])C3)[nH]c12 N1(C(n2cc(CCn3nc(C)cc3C)nn2)CC)CCC(CC2CC2(Cl)Cl)CC1 c1(C(=O)NC(C)C(=O)NCCNC(C2C(C)C2C)=O)ccc(F)cc1 c1(C(=O)NCc2ccc(C)s2)cc(CNC(=O)CC2(C#N)CC2)ccn1 CC1CCN(C(C2C3CC(=O)CC23)=O)C1C(=O)NCc1ccn(CCF)n1 C(=O)(C1=CN(C)S(=O)(=O)N=C1C)N1C(CO)CC(OC)C1.C(C)(C)(C)O C(=O)(C(C)(C)C(=O)NCCN1CCN(C(C2CNC(=O)N2C)=O)CC1)OCC c1(C(N(c2ccc(SC)cc2)C)=O)ccc2cnn(C)c2c1 N1(C(C2(SC)CC2)=O)CC(NC(c2ccc(C(F)F)cn2)=O)C2(CCC2)C1 c12cn3ccc(cc3n1)O2.Cc1cccc(COC(N2C(=O)CNC2=O)=O)c1 C1(C(=O)N(C)CC2(c3c(OC)cc(C)cc3)CCCCC2)CCN(C)C2(CC2)C1 C(=O)(CCC(C)(C)C(=O)OC)N1CC(CNC(C(C=CC)O)=O)N(C)CC1 C(=O)(C1=CCC(NC(=O)CC2CCSCC2)C1)N1CCC(NC(N)=O)CC1 C(CC(=O)NCC1(C)CC2CC2C1)(C(F)F)NC(c1c(CC)c[nH]c1)=O CC(O)C(C)C(=O)N1CCC(N(C)C(c2cc(C#N)no2)=O)C1 c1(OC)ccccc1C1(C(=O)NC(C)(C)CCNC(c2ccsc2)=O)CC1 S(=O)(=O)(c1ccnc(NC(c2coc(C)c2)=O)c1)N1CCC(SC)CC1 c1(S)cc(F)c(N)cc1F.C1(CCCC)CCCN1S(=O)(=O)CC1CCCC1 C1(C(=O)NCC(C)NC(=O)CCC2CCCCO2)CCN(CC(F)F)CC1 CN1CCC(CC(=O)NCC(F)CN(C(=O)CC(F)F)c2ccccc2)CC1 C1(NC(C2C(C=C)CC2)=O)CC2CC1CN2C(c1ccc[nH]1)=O CC1COC(C(N2CC(N(C)C(c3cc(CC4CC4)on3)=O)C2)=O)C1 C1(F)(CNC(Cc2c(C)ccs2)=O)CCC(NC(c2ccncc2)=O)C1 C=C1CC(C(F)(F)F)(C(=O)N(CCNC(=O)N=S(C)(C)=O)CC)C1 c1(C(=O)NCC2(C(F)F)CCN(C(C(C)(C)SC)=O)C2)cc2cccnc2s1 C12(NC(CCOCC#C)=O)CCC(CN(C(=O)CC(C)CC(=O)OC)C1)C2 c1(CCC(=O)NC(CC)CNC(=O)C(C)CC2CC2)nc(C)c(C)o1 C1(N(CC#C)C(c2cc(CC)no2)=O)CCN(C(C2CCCCN2CC)=O)CC1 N1(C(CSCC#C)=O)CC(NC(C2(C)CCCN2C(C)=O)=O)CC(F)C1 C1(NC(C2CCC(n3cc(CCC(F)(F)F)nn3)C2)=O)Cc2ccc(Cl)cc2S1 N1(C(COC2(C)CCOCC2)=O)CCC(C2CC2)C1CNC(c1ccc(Cl)[nH]1)=O C(=O)(C(CC)NC(=O)NCc1ccc(C2CC2)s1)NCCCC c1(C(=O)OCCc2c(N(C)C)ncnc2Cl)ccc([N+](=O)[O-])cc1S(C)(=O)=O O=C(NNCNCc1cccc2c1OCCO2)NNc1ccc([N+](=O)[O-])c(Cl)c1 C(=O)(CC(COC)N(C)C)NC(C=C)C(=O)NC1CN(C)CCO1 N1(Cc2cc(OC)no2)CC(NC(c2ccc([N+](=O)[O-])[nH]2)=O)CCC1C OC1CN(CC2CCCC2c2ccccc2)C2(CCCC2)C1 c1(C(=O)NCC(CC)(C)Cl)coc2c1CN(C(C1CCC(C#N)CC1)=O)C2 N1(C(C(C(C)(C)O)F)=O)CCCC2(CCC2NC(=O)COCC(F)F)C1 Cc1cn2cc(C(=O)NC(C)CNC(c3cnc(S)nc3)=O)cc(C)c2n1 CC(C)CC(O)C(=O)NCC1(C)CCCN(C(=O)CC(C)C2CCCO2)C1 C1(C#N)(C(N2CC(CNC(c3c(CC)occ3)=O)C(F)(F)C2)=O)CC2(CCC2)C1 N1(C(CC2CC(CC)C2)=O)CCC2CCN(C(c3n[nH]cc3Br)=O)C2C1 CCCCCCC(C)(C)C(=O)NC(C1CCCN1C(=O)CC1CC=CCC1)C C1(C(N2CC(C=C)(CC(=O)NCc3cccc(F)n3)C2)=O)CN2CCC1CC2 CN1CCC(O)(CC(=O)C2CC2CNC(=O)CN(C(=O)CC(=O)OC(C)=O)C)CC1.N c1(C(=O)NCC(C2CCN(C(=O)C#CC(C)(C)C)CC2)C)cnc2occc2c1 CCC(CC(=O)NC1CCCCC1NC(c1cc(Cl)c(Cl)[nH]c1=N)=O)C(F)F c1(OC)ccc2nccc(CNC(=O)C(CC(C)C)N3CCCC3=O)c2c1.C1CO1 c1(C(N(CCC(C(C)C)NC(C=C(CCC)C)=O)C)=O)c[nH]c2cccc(C)c12 Cc1nc(C(=O)NCCC(=O)NC2CC23CC(O)C3)sc1C c1(CC)ccc(C(=O)NCC2(NC(=O)C(C)n3cncn3)CCOCC2)c(C)n1 CC1(C)C(=O)NCCN1C(=O)C1=NOC(C2(O)COC2)C1 C1(C2C(C)(C)C2)CN(C(=O)CSCC(N)=O)CCN1C(c1cccc(C2CC2)c1)=O CC1CC2(CCC2)CN1C(=O)C(C)(CNC(c1cc2ccccn2n1)=O)CC1CC1 C(=O)(N(CCC(=O)OC)OC)C(CC)C(=O)NC(C)CC(C)(C)OC C1(NC(C2(CC)COC2)=O)CCN(Cc2snnc2C)CC1C N(C(=NCCCn1cnnc1)NCCC(C)C)CCc1c(C)n(C)nc1 C1(O)(CC(=O)N(C)CC2(N(C)C)CC2)CCCN(C(=O)C=CC2CCC2)C1 Cc1cc(N(C)C)ccc1C(=O)NC1CCN(C(c2cc[nH]c(=N)c2)=O)C2CC12 N1(C(CC(C)(C)C(F)F)=O)CCC2C(CCCN2C(c2cccc(O)c2F)=O)C1 C(=O)(C(C(C)C)C1CCC1)NCC1C(CNC(CCC=C(C)C)=O)C1 n1(C(C)C)ncc(C(N2CCC(CNC(C3CN(C)CCO3)=O)C2)=O)c1F N1(C(COCC(C)C)=O)CCCC2(C1)CN(C(C1(CO)CC1)=O)C2 Cc1cc(C(=O)N(CC(C)NC(=O)C(CO)c2ccccc2)C)n[nH]1 C(=O)(C1CCCc2nnn(C)c21)NC1(CC=C)CCCN(C(=O)CO)C1 c1(NC(C2CCCCN2C(c2cc(Cl)c(F)c(Cl)c2)=O)=O)c(Cl)ccc(O)c1Cl N1(C(C(C)NC(CC)(C)C)=O)CCC(NC(=O)C2=C(Cl)CC2)C12CCCC2 Cc1cc(-c2ccc(=N)[nH]c2)cnc1C(=O)NCc1cc(C(F)(F)F)nn1C C1(C(N2CC(F)CC(F)C2)=O)N(C(c2cc3n(n2)CCO3)=O)CC12CCCC2 C1(C(=O)NC(C(C)C)CN(C)C)CCN(C(c2cnc(S)nc2)=O)C1(C)C c1(N2CCCCC(NC(c3c(C)nc(O)cc3)=O)C2)nc(Cl)nc(C)c1F C12CCC13CCCN(C3)C2=O.c1(OC)nn(C)c(-c2ccccc2)c1Cl N1(C(c2c(C)nn(-c3cnccn3)c2)=O)CCOCC(NC(=O)C(=O)N(C)C)C1 Cc1ccc(C)c(OCC(N2CCC(NC(C3CCC(=O)N(C(C)C)C3)=O)C2)=O)c1 c1(C(N2CC(F)(CNC(c3occc3Br)=O)C2)=O)cncc(F)c1 c1(-n2c(C(COC)Nc3nc(CN(C)C)cs3)nnn2)cccc(OC)c1 N1(c2ccnc(NC3CCN(C)C(=O)C3)n2)CCCOCC12CCCC2 C=CC(CCC)CC(=O)N1CC2CC2(NC(c2cccc(C3(C#N)CC3)c2)=O)C1 C12(CNC(c3occ(C(=O)OC)c3)=O)CCC1CN(C(C1C(C)(C)C1(C)C)=O)C2 CCC(CNC(=O)CC1CCCC(C)O1)(CC)NC(=O)CCN1CCCCC1 CCCCC(CCCC)C(=O)NCC(F)CNC(=O)COC(C)CC Cc1cc(C)n(CC(=O)NC2CN(C(=O)C(C)(C)C(N)=O)CC2C)c(=O)n1 CCCCCC(CC)C(=O)NC(C)CCc1nnnn1-c1ccccc1 C1(C(N(CCCNC(c2c(C(C)C)n[nH]c2)=O)C(C)C)=O)CCCOC1C N1(C(CC23C(CN(C(CC4CC(OC)C4)=O)C2)CC3)=O)CC(OC)CC12CCC2 c1(C(=O)NCCN(C(c2ccc(C)o2)CC)CC2CC2)cc(CO)ccc1OC c1(C(=O)NC2CC(C(N3CCC(C)(C)C3)=O)OCC2)cc(O)cc(=O)o1 N1(C(N(C)C)=O)CCCC(C(=O)NCC2CCC(CNC(=O)C(F)(F)CO)CC2)C1 C(=O)(CC(C)CC(=O)NC(c1nocc1C(=O)NC1CC2CCCC2C1)C)OC CC1CC(O)CN(C(c2cccc(C)n2)C(=O)NC(C)(C)C)C1 c1(OC)cc(C(N2CCC(NC(=O)CCc3c(F)cccc3F)C2)=O)ccc1C C12(CNC(=O)Cn3nnc(=O)[nH]3)CN(C(c3cnc4n3CCS4)=O)CC1CCO2 N1(C(C(CC=C)OC)=O)CC2CC(O)C1C2NC(=O)Cn1ccc(C2CC2)n1 C1(NC(c2c(CC)onc2)=O)CCC(C)N(C(=O)C=Cc2cccc(F)c2)C1 c1(-c2cn(CC3N(C(CCC(=C)Cl)=O)CCC3)nn2)cccc(F)c1Cl c1(C(N(CCn2cc(C(C)N(C)C)nn2)C)=O)sc2cc(Br)ccc2c1Cl CC1CN(C(=O)CCCC(N)=O)CC(C)C1NC(C1(CO)CCCO1)=O N1(CC2(C(n3cc(-c4nn(C)cc4C)nn3)C)CCCC2)CC2CCC(CC2)C1 N1(C(C(CC#C)C)=O)CCC2C1CCCN2C(=O)Cc1ccon1 c1(C(=O)NNC(=S)Nc2ccccc2F)ccc2cccc(F)c2n1 N1(C(c2c(CC)noc2)=O)CC2CC1C2CNC(c1c(C)noc1C(F)(F)F)=O c1(NC(C2N(C(c3ccc(C)nc3Br)=O)CC(C)C2)=O)cc2cccnc2[nH]1 C1(C(=O)NCC2C(CC)CCN2C(=O)C=CC(=O)N(C)C)CCCCC(=O)N1 c1(COCC(=O)NC23CC2CN(C(=O)C(O)C(F)F)C3)ccc(C(F)(F)F)cc1 c1(-c2c(C)c(CO)ccc2)ccc2cc(C(=O)Nc3cncc(O)c3)cn2c1 C1(NC(C(CC)SC)=O)CCN(C(c2cnn3cc[nH]c(=O)c23)=O)CC12CCC2 CCCC(C)(CC)C(=O)NC1CCN(CCCNC(=O)CC2CCSC2)C1 C1(CCNC(=O)CCF)CC(F)(F)CN1C(=O)CC(O)C1CCCC1 CN1CC(NC(=O)C2=CCC(NC(=O)CCC3CCC(=O)C3)C2)C2(CC2)C1=O c1(C(=O)NCC2CC(NC(c3c(C)nc(C)[nH]3)=O)C2(C)C)ccc2ncnn2c1 c1(C(N2CCC(C)C2CNC(c2cc3cscc3s2)=O)=O)cc2occc2n1C N1(C(C(CC)C)=O)CC(NC(=O)CCc2ccccc2C(N)=O)C2CCCCC12 C1(C2CC2)(C(=O)NCC(C)(CO)CO)CN(C(=O)CN2CCNC2=O)C1 c1(C(N2CC(C)(CC(=O)Nc3ccc(Cl)nc3Br)C2)=O)cc(Cl)c(O)c(Br)c1 N1(C(c2cnnn2C)C(=O)NC(C)(C)C)CCn2nc(C(C)(C)C)cc2C1 c1(CC(=O)NC(CC)CNC(C2CC(F)(CO)C2)=O)ncncc1Cl C1(NC(C(CC)OCC)=O)CN(C(c2cc(C)ccc2N)=O)CCC1(C)C c1(OC)ccc(OCC(=O)NCCCCN(C(=O)C(C)(C2CC2)OC)C)cc1 CC1(C2CCN(C(=O)C(C3CCN(C(c4cnc(S)nc4)=O)C3)F)C2)CC1 C1(N(C(c2nc(C)sc2)=O)C)CN(C(C2(CNS(N)(=O)=O)CC2)=O)CC1O C1(C(NOCC(=O)OCC)=O)N(C(=O)CCS(C)=O)CC12CCCC2 N1(C(C(C(C)C)C)=O)CCC(C)(C)C1CNC(c1cc(=O)n(C)o1)=O C1(CC)(CC)Oc2ccc(NC(=O)NCC3CCOCC3F)cc2O1 Cc1ncc([N+](=O)[O-])n1CC(=O)NCC(C)(C)CNC(C1CCCC1C)=O CCCCC(CNC(=O)COc1ccc(Br)cc1)NC(C1CC2(F)CC1C2)=O N1(C(C(CCC=C)NC(=O)Cc2csnn2)=O)CCN(C)C(=O)C1C C1(CNC(CCOCC#C)=O)CC(O)C12CCC2.C12CC(CCO1)NC2=O N1(CC)CC(C(=O)NCCCCCCN(C(=O)CCC2CCOC2)C)CCC1=O Cc1ncccc1C(c1nnnn1C1CCCCC1)NCC1CC=CCC1 N1(C(CCC)=O)CCCCC1C(N1CCN(CCO)CC1)=O.C1(CC(=O)N)CN(C)C1 N1(C(C(C)n2cccn2)=O)CCN(C(=O)CN2C(=O)CN(C)C2=O)CC1C1CCC1 Cn1cnc2cncc(C(=O)NCCNC(=O)CCCn3ccnc3)c12 N12CCCC(C1C)C2=O.Cc1nn(C(C)(C)C)cc1NC(=O)CSCCC(C)C C1(O)(CN(C(=O)C(O)C(C)(C)C)C)CCCN(C(=O)C(F)CC2CCOC2)C1 C1(C(=O)OCC)CNCC12CCN(C(c1c(Cl)ccc(F)c1Br)=O)CC2 CC1=C(C(=O)NCC2(NC(c3ccc(C(F)(F)F)cc3)=O)CC2)C(=O)OC1(C)C O=C(CC1=CCCC1)NCC1(CNC(=O)C(F)(F)c2ccccc2)CC1(F)F N1(C(C(=Cc2cn[nH]c2)C)=O)CCN(C)C(C(N2CC(O)(C(F)(F)F)C2)=O)C1 C#CCC(C(=O)N1CCC(NC(c2cccnc2N(C)C)=O)C1C(C)C)C1CC1 C(N=c1[nH]cnc(Cl)c1[N+](=O)[O-])C1(NC(C2CCOC3(CCCCC3)C2)=O)CC1 c1(C(N(C)CC2COCCN2C(=O)CN2CC3CC3C2)=O)n[nH]c2c1COCC2 Cc1ccc(F)c(C(N2CCC(CNC(=O)C(C)(O)Cc3ccccc3)C2)=O)c1 N1(C(C(C)OCC#C)=O)CCC(N(C)C(C2CCC(C(=O)NC)O2)=O)CC1 N1(c2nncc(OC)n2)CC(C(=O)NCCc2cccs2)CC(C)C1 c1(COC)ccc(C(=O)NC2(NC(=O)CC3CC(C)(C)C3)CC(C(N)=O)C2)[nH]1 C1(C(=O)NC(CC)C)(NC(C2CCCN2C(=O)NC2CC2)=O)CC(F)C1 c1(OCC)ccc(C)nc1C(=O)NCC(C1CCC1)NC(=O)C(C(C)C)NC=O c1(C(N2C(CN(C(CSCC=C)=O)CC)CCC2)=O)cc(N)ccc1C N1(C(c2n(C)ccn2)=O)CC2CCCC2(CNC(c2ccco2)=O)C1 c1(CNC(=O)CC2CCCCCC2)ccc(C(=O)NC(CN(CC)CC)C)cc1 CC1CN2CCN1CC2C(=O)NC1(CCNC(=O)CC2CCCSC2)CC1 C1(CNC(c2cc(C(C)C)[nH]n2)=O)(NC(=O)C(O)C(C)C)CCC(F)(F)CC1 c1(C(=O)NCC2CCC(CNC(C(CSC)C)=O)CC2)cccc(C)c1C#N C1(NC(C2CCC(C(=O)O)CC2)=O)CN(S(=O)(=O)Cc2cccc(F)c2)CC12CC2 N1(C(CC=CCC)=O)CCOCC1CC(=O)NC(CO)C(C)(C)C N1(c2n(C)cnn2)CCCCC(c2cn(CCC=CC#N)nn2)C1 N1(C(c2ccsc2Cl)C(=O)NCc2ccccc2)C2CCC1CC(F)(F)C2 CCCC(C)C(=O)NC(C)CCN(C)C(C1CC1c1cnn(C(C)C)c1)=O n1(CC(=O)N(C(C)C)CCN(C(=O)C(O)CN(C)C)C)cnc2c1CCCC2 N1(C(C(C)SC)=O)CC(NC(c2cscc2SC)=O)CC1(C)C C1(CC(=O)NCC(CC)NC(=O)C(C)(C)CSC)SC2=NCCN2C1=O N1(N(C2(C)COC2)C)CCOCC(OCC(F)(F)F)C1.c1(C=O)ccccc1C=O N1(C(C(=O)NC(C)CNC(c2csc(C#N)c2)=O)C)C(=O)NC2(CCCC2)C1=O N1(C(c2ccn(CCCC)n2)=O)CC(C2CCCN(C(=O)C3=CCCCO3)C2)C1 C(CCCCN(C)C(c1ccn(C)n1)=O)NC(C(C)=C(CC)C)=O N1(C(C(CC)C)=O)CCC2CN(C(c3cc4cc(Cl)cnc4o3)=O)CCC12 CC(C)CC(C)(Cc1ccc(CNC(C2CC2C)=O)cc1)NC(=O)CO N1(C(c2ccnc(OC)n2)=O)C(C(=O)N(CC(C)(C)CO)C)CCC12CC2 C1(C(=O)NC2CC(F)(CNC(C3CCC3(F)F)=O)C2)CCCOC1c1cc[nH]n1 CC(C)CC(F)(F)C(=O)N(C(C)CNC(=O)CSc1ccc(F)cc1)C N1(CCC(=O)NCC(C2CC2)NC(c2c(CC)nns2)=O)C(=O)NC(C)(C)C1=O C(CC(C(=O)NOCCCOC)NC(c1csc(=N)[nH]1)=O)OC C=CC1COCC1OC.C123CC(CN1C2=O)C3 N1(Cc2cc(C)nn2C)CCc2nc(OC(F)(F)F)nn2CC1 N1(C(CC(C)OC)=O)C2CCCC1CN(C(c1cc(CC(C)C)n(C)c1C)=O)C2 c1(C(N2C(C(CNC(C3N(CC)CC3)=O)(C)C)CCC2)=O)cc2ccccc2o1 C(=O)(CCCCC(=O)NCC1(CNC(C2CC(C)(O)C2)=O)CC1)OC C1(C)(C(N(C)Cc2cccc(O)c2)=O)CN(C(C2(c3cc[nH]n3)CC2)=O)C(C)(C)C1 CC(CC(=O)N1CC2CCC1CN2C(C1CCC(=O)N1)=O)CC(C)(C)C Cc1nc(C)n(CCC(=O)NCc2ccc(C(=O)NCCC(O)CN(C)C)o2)n1 C(C)(C(=O)N1CC(C(N2CC(N(CC(C)C)C)C2)=O)C1)OC(C)=O c1(C(=O)OC)cc(O)c(C(=O)NNC(=O)Cc2cccc(Cl)c2Cl)cc1Br N1(C(C2C(=C)C2)=O)CCC(CF)(NC(=O)CNC(c2ccccn2)=O)C1 C1(C)(OCC(=O)N(CC)Cc2cnn(C)c2)CN(C(=O)C=CCF)C1 C12CC(CCO1)C2.c1(C(=O)NCC2N(C(CC)=O)CCC2)cc(C)n(C(F)F)n1 C1(N(C(C=C(CCN(C)C)Cl)=O)C)CN(C(c2csc(=N)[nH]2)=O)CC1F C(=O)(C(C)(O)C(C)C)N1CC(CC=C)(NC(=O)C(N2CCSCC2)C)C1 C1(C)(NC(CC2C(CNC(c3c(CC)cccc3)=O)C2)=O)C(C)(C)C1(C)C c1(C(N2CCC(NC(C(CC)(F)F)=O)C2C)=O)cn2c(n1)SCC2 C12(C(=O)NCC3C(C(=O)NC(C)C)CC3)COCC1C2.c1(C2(O)CCC2)nc[nH]n1 CC1(C)C(CC(N2CC=CC2)=O)CCN1C(=O)CC1CCNC1=O c1(-c2cn(CC3C(NC(CCc4cnn(C)n4)=O)CCC3)nn2)cncc(N)c1 c1(C(N2CC(NC(C(C(C)C)C)=O)C3(C2)CC3)=O)ccc2nncn2c1 c1(C(=O)NC2C(CNC(=O)Cn3nnc(C(F)(F)F)n3)C2)ccnnc1S C1(N(C(c2cc(CC)no2)=O)C)CN(C(C2(OC)CCOC2)=O)CC12CC2 c1(OC)ccc(-c2cnc(C(N3CCCC3)C(=O)NC3CC3)nc2)cc1OC C1(NC(C2CCC(C)C2)=O)C2CC1CN(C(c1ccccc1CO)=O)C2 C1(CNC(c2c(C)nns2)=O)CCN(CCN2CCC2c2nc(C)ns2)CC1C C1(C(=O)NCC(CCOC)NC(=O)CN2CC(C)C2)CCCC1(C)C CCC(C)C(C)C(=O)NC(c1ccc(F)cc1)CNC(c1ncnc(C)c1C)=O C1(F)(CNC(C2(C)CC(=C)C2)=O)CCN(C(=O)C(C)CSC(F)(F)F)C1 c1(-n2cc(CNC(C3(C(F)(F)F)CCC3)=O)nn2)ccccc1CCOCC C1(C(=O)N(C)CC2CCCN2C)(NC(Cc2c(C)n(C)nc2)=O)CCC(C)(C)C1 C=CC1(C(=O)NCC2(OC)CN(C(=O)CC(C)c3ccncc3)C2)CCOCC1 c1(C(N2CC(C)C(NCc3cc(F)c(Cl)cc3O)C2)=O)cccc([N+](=O)[O-])c1F N1(C(CCCN(C(CC(=O)OCC)=O)C)=O)CCN2CC(O)CC2C1 C(=O)(CC(C)(C)CNC(=O)CCC(N)=O)NCc1n(C)ccn1 N1(C(Cc2cc(C)sc2)=O)CCC2(NC(=O)CC3CC3C)CCCC12 N1(C(CN(C)C(N)=O)=O)CCCC1CN(C(=O)C(C)(C)n1cnnn1)C c1(OC)cccc(C(C(=O)O)NC(c2[nH]nc(Br)c2C)=O)c1C CCC(CCCC(=O)N(c1ccsc1)CC)NC(=O)C=Cc1cncs1 C1(=O)C(NC(c2cscn2)=O)CCNC(=O)OCCN1.C(C)(C)(C)OC C12(NC(c3nc(C)sc3C)=O)CCCC1CN(C(=O)CC(F)F)C2 C=CCC(C)(C)CC(=O)NCc1scc(C(=O)NCCC2NC(=O)NC2=O)c1 c1(CC)cn2c(n1)C(C(=O)Nc1nccc(=NC(=O)C3CCN3CC)[nH]1)CCC2 N1(C(c2c(C)onc2)=O)CC(C)OC2(CCN(C(c3nnn(C)c3N)=O)C2)C1 C12CCC(CC1)CNC(=O)CCOCC=CC(=O)NC2.C1(CNC)CCCCO1 CC(C)CCC(F)C(=O)N(CCCNC(C1CCC(C2CC2)C1)=O)CCO CN1C2CCCC1CC(Nc1cc(NC3CN(C4CC4)C3)ncn1)C2 N1(C(c2c(C)occ2)=O)CC(NC(=O)CCSCC(N)=O)CC1CO C(=O)(CC(C)CC(C)(C)C)NCC1(F)CCC(NC(C2(COC)CC2)=O)C1 N1(C(C2(CC=C)CCC2)=O)CCC2(CCCN2C(=O)COCC2CCCOC2)C1 c1(C(c2ccco2)NCCC2C(C)CC(c3ccccc3)CC2)coc2c1CCCC2 c12ccc(cc1F)c(=O)[nH]2.N1(Cc2n(C)ccn2)CC2CC(O)C1C2 c1(C(=O)NCC2CCC(NC(c3ccncc3)=O)C2)ccnc2ccc(F)cc12 c1(C(C(N)=O)NC(=O)C(=O)NCc2cccc(C(F)(F)F)c2)ccc(Cl)cc1F C1(C(N(CC(O)C2CCC2)C)=O)CC2CCCC2N1C(c1ccncc1N)=O C#Cc1cc(C(=O)N(C2CCN(C(C3CCSCC3)=O)C2)C)ccc1Cl N1(C(CSCC=C)=O)CC(CNC(=O)C=C(Cl)Cl)C(C)C1 C1(CCC)CN(C(C2(C#N)CCCOC2)=O)CCN1C(=O)Cc1ccccc1Cl C(CC1=CCN(C(C2CCC3(CCCC3)C2)=O)CC1)NC(C1CCNCCO1)=O c1(C(=O)OC)cnc(CNC(=O)Cn2nnc(C)n2)nc1.C12CCCN1C2=O c1(-c2nnc(CN(C)C(=O)NCc3cc(C(F)F)on3)o2)ccc(F)cc1 c1(C(NOCCCCCC(=O)OC)=O)cc(C(=O)OC2(C)CCCO2)ccc1O Cc1ccc(O)cc1C(=O)NNC(=O)CNc1cncn1C1CC1 c1(C(=O)NC23CC(NC(=O)CC4CCCOC4)C(OC2)C3)cc2ncccc2o1 Cc1cc(C(=O)NC2CC2NC(c2cncc(Cl)c2)=O)ncc1S(N)(=O)=O Cc1cc(Cl)c(C(C)NCC2CCN(C(C)C)CC2)cn1 N1(C(C(CC=CCC)C)=O)CCC(C)(C)C(NC(C2(N(C)C)CCCCC2)=O)C1 c1(C(=O)NCCC2N(C(CC(C)SC)=O)CCC2)ccc(C2(F)COC2)cc1 Cc1cc(C(N2CC(C(=O)NCc3nc(C)c(C)[nH]3)OC(C)C2)=O)c(C)nn1 C12CC3CC(C3C1)N2.c1(N(C)C)cc(N2CCC(OCCF)C2)ncn1 C1(C(N2C3CC(NC(c4nc(C)sc4C)=O)C2CC3)=O)CCCC12CCOCC2 c1(C(N2C(CNC(=O)CSc3cccnc3)CC(O)C2)=O)noc2c1CCCC2 N1(C(C2C(C)=CCS2)=O)CCCC(C(=O)NC2(C)CC2(C)C)C1C CCC(C(=O)N1CCC(N(C(=O)CCCOCC)CC2CC2)CC1)C(C)O CCCC(C)(CC)C(=O)NC1CCCN1CC1(C)CCN(c2ccccc2)CC1 O=C(CC1=CCCCC1)NC1CC(CNC(C2(Cc3ccoc3)CCOCC2)=O)C1 Cn1cc(NC(=O)CCC2CCN(C(=O)CCn3ccnn3)C2)c(C#N)n1 N1(C(=O)NC2(C(=O)NCCOC)CCOC2)CCN(C(=O)C(C)OC2CC2)CC1 N1(C(C(CCNC(C(C)(C)NC(=O)OC)=O)(C)C)=O)CC2CSCC2C1 c1(C(=O)NCC(C2CC2)NC(Cc2cc(C(=O)OC)sc2)=O)nccc(Cl)c1C C1(C(N(C(C)C2CC2)C)=O)(CNC(C2CCCC(=O)O2)=O)CCCCC1 c1(N(C)Cc2ccc(C)c(C)c2)nc(N2CCCN(C)CC2)c2c(n1)COC2 C1(NC(C2C=CCC2)=O)CCC2CCN(C(=O)Cc3nc(F)c(F)cc3F)C12 c1(CN(C2CCN(c3ccccc3F)C2)CC)ccc(F)cn1 C1(NC(C(C)(C)C)=O)CCCCC1CNC(c1ccc(-c2cc(O)ns2)cc1)=O CCCC(O)CC(=O)NCC1CC(C(F)(F)F)CCN1C(c1c[nH]nc1C)=O CCC(C)C(C(=O)N1CC2CCCC1C2)ONC(=O)c1ccco1 c1(C(=O)NC23C(CN(C(C=C(C)C)=O)C2)C3)sccc1S(C)(=O)=O c1(CNC(C2(CC#N)CCC2)=O)ncccc1CNC(c1ccsc1C(F)F)=O N1(C(C2(C(C)NC(C3CC3c3ccco3)=O)CC2)=O)Cc2ncsc2C1 C(C(=O)N=c1cc(-c2csc(C)n2)[nH][nH]1)(c1cc(OC)c(O)nc1)C1CC1 c1(N(C(C)=O)C)ccc(C(=O)N(CC(C)C#N)C2CC2)cc1 C#Cc1cncc(C(N2CC(O)CC2CNC(c2ccc(CC)cc2F)=O)=O)c1 Cn1ccc2c(C(=O)NCC(C3CC3)NC(C3CC3C3CC3)=O)ccnc12 C1(NC(CCOCCC)=O)COC2(CNC(=O)CCCCC3CC3)CC1C2 C1(C(N(C)CCOCCNC(=O)CC2(C)CCOC2)=O)CN2CCC1C2 C(C(CC(F)(F)F)NC(=O)CNC(c1cccnc1)=O)NC(C(CC)SC)=O c1(C(C(=O)NCC2CCN(C(Cn3c(NC=O)cnc3)=O)C2)(F)F)cc(Cl)sc1Cl Cc1ccc2c(c1)N(C(C1(NC(c3ccn(CCOC)n3)=O)CCCC1)=O)CC2 CCC(CC)CCC(=O)N1CCOC(C(C)NC(C2CN3CCN2CC3)=O)C1 c1(NC(c2ccnn2C)C)[nH]c(=NCCC2CCCC2)nc2c1cnn2C Cc1c(NCCCc2ccccc2Cl)nc[nH]c1=NCC12CC(C)(CCO1)C2 c1(CN2CC(N(CCS(=O)(=O)NC3CCCC3)C)C3(C2)CC3)ccc(O)c(F)c1F Cc1ccc(F)cc1CC(N1CC(CNC(=O)CCc2nc(C)c(C)o2)C1)=O Cc1c(C(N2CCC(CNC(=O)Cc3ccsc3)C(C)C2)=O)cnc2ccnn12 Nc1c(Cl)ccc(F)c1C(N1C2CCC1C(NC(c1cnc[nH]1)=O)C2)=O c1(C(=O)OC)c(C)[nH]c(C(=O)OC(C)C(C)(C)C(C)C)c1C N1(Cc2scc(C)n2)CCN(C(c2csc(CCP(C)(C)=O)n2)=O)CC1 N1(C(C(C(=O)OC)C)=O)C2CCC1C1CC1(NC(=O)C=CC(C)(C)C)C2 C1(CC(N2C(CC(=O)NCCOC(C)C)CC2)=O)CC1(C)C C=CCN=C(NCCCCC(=O)NC)NC(c1ccc(O)cc1)C Cc1csc2ccc(C(N3CC(NC(=O)C(F)=CC4CC4)CC(O)C3)=O)cc12 c1(C(N2CCN(C(C(C3CCCCC3)C)=O)CC2CO)=O)nccn2nccc12 N1(C(CCCCOC)=O)C2CCCC1CC(NC(c1cc(C(C)=O)c(C)o1)=O)C2 Cc1ccc(F)cc1C(=O)N(C)CCOCCCN(C)C(c1ccns1)=O c1(NC(N2C(n3cc(CC(C(C)C)O)nn3)CC3(CC3)C2)=O)csc(S(C)(=O)=O)c1 C=CC(F)(F)C(=O)NCC1(F)CN(C(c2cnn(CC3CCCC3)c2)=O)C1 C=CCN(CC1COc2ccccc2O1)N1CCC(O)(C(Cl)(Cl)Cl)CC1 C(=O)(C(C)(C)C(O)C(C)C)N1C(C(=O)Nc2cccc(OCC)c2)CC(OC)C1 c1(-c2cn(CC)nc2)nc(C(N2CC(O)CC2C(=O)O)=O)c(N)s1 C1(CC(=O)N(CCCN(C)C)CC)CC2CC1CN2C(C1C=CCC1)=O N12CCCCC1C2.c1(CC(=O)NCC#N)sc(Br)nc1C c1(C(=O)OC)ccc(C(=O)NC2(C(=O)O)CCC2)cc1OC c1(CC(N2C(C(=O)NCC3C(CC)C3)CN(C)CC2)=O)c(O)nc(=N)[nH]c1C c1(SC(C)C(N2CCN(C(=O)C=C(Cl)Cl)C(C)C2)=O)ccc(C#N)cc1 C1(C(c2cscc2Br)C)CCC2(CCC2)O1.C1C(O)CN1C.NC c1(C(=O)NC2CCC(Nc3ccc(C#N)nc3)CC2)cccn2c(Br)cnc12 C1(C(=O)NC(CN(CCC)C)(C)C)(NC(=O)C(C)n2cccc2)CCSC1 Cc1cccc(C(N2CCCCC2C(=O)N(C)CCn2cncn2)=O)c1C C1(CC(=O)NCCCNC(=O)NC)COCCN1C(c1cnccc1C)=O c1(-n2c(-c3coc(C4CC4)n3)nc(CCCN(C)C)n2)cc(Cl)nc(Cl)c1 c1(C(=O)NCCC(C)NC(c2cccc3ccnn23)=O)ccc(P(C)(C)=O)cn1 c1(C(C)NC(C(COC)NC(=O)C(C)c2cc[nH]n2)=O)c(C)n[nH]c1C C1(CNC(C(COC)(C)C)=O)CC2CCC1N2C(c1cncc(C(C)C)c1)=O CN1C(=O)CCCC1C(=O)NC(C)(CO)C(=O)NCC1=CCCOC1 C1(C(=O)OCC)(CNCC(c2sc(C3CC3)nc2C)(C)O)CCCCO1 N1(C(c2scc(C)c2)=O)CC2CC(NC(c3ccc4c(c3)CC4)=O)C(C2)C1 CC1(O)CCCN(C(=O)C(CC2CCOCC2)NC(C2CCC=CCCC2)=O)C1 N1(C(C=CC)=O)CCOC(C(C)N)C1.c1(C(=O)CCOC)cnccc1N(C)C S(=O)(=O)(c1ccc(N(C)C(C)C)nc1)NC(CCCC)(C)C.C1C(C)N1 C1(C(N(C(C)CN(C)C(C2(C)CCOCC2)=O)C)=O)CCN(C)C(=O)C1 CC(C(=O)N1CC(F)(CNC(C23CCC(F)C2CC3)=O)C1)S(C)(=O)=O CS(=O)CCC(O)C(=O)N1CC(O)(CCNC(c2cc(Cl)ccc2N)=O)C1 C1(C(=O)NCc2c(C)nns2)CCCC(NC(c2cc(C(N)=O)[nH]n2)=O)CC1 C1(NC(CC=CC=C)=O)CCN(C(=O)C(C)(C)C(C)C)CC1(C)C Cc1cccc(F)c1CC(N1CC2CC2(NC(=O)CCCC2CCCC(=O)N2)C1)=O N(C(=NCCc1ccc(O)cc1)NC1CCN(C(C2CCC2)=O)C1)C(CC)C N1(C(c2cnc3ccnn3c2)C(=O)NC(CC)(C)C)CCCN2CCCC2C1 C1(CC)C(NC(=O)C2=CCCSC2)CCCN1C(c1ccc(Cl)cc1)=O n1(CC(=O)NC2CC(CNC(c3n(CC)ccn3)=O)C2)nc(C)c2cccnc12 c1(C(=O)NC2(CCOC)CCN(C(c3cc(C)sn3)=O)C2)ccc(S(C)=O)cc1 N1(C(C=C(COC)C)=O)CCCC(CCC(=O)NC(CCO)C2CC2)C1 c1(CC(=O)NC2CN(Cc3c(Cl)cnc(SC)n3)CC2F)cc(Br)cc(Br)c1O n1(C(C)C)nnnc1C(C)(C1CCC1)NC1(c2cccs2)CC1 C(=O)(C1Cc2ccc(Cl)cc21)NC1C(CNC(c2c(COC)cccc2)=O)CC1 c1(SCc2nc(-c3ccn(C4(C(=O)O)CC4)n3)sc2)cc(Cl)ccc1OC(F)F Cc1c(C(N2CC3(CCN(C(c4ccnnc4)=O)C3)C2)=O)ccc2c1OCO2 NS(=O)(=O)c1cc(N2CCOCC2)c(C(=O)O)c(Br)c1 CC(CC1CCOCC1)C(C(=O)NC1CCOC1)N(C1CCN(C)CC1)C N1(C(C(C2CC2)OC)C(=O)NCC2CCOC2)CCC2(CC1)CCS2(=O)=O C#CCC(CC(=O)NCCn1cncn1)NC(=O)C(C)(C)n1ccnn1 C(c1cccnc1)=CCNC(N1CCOCC1C1CCC1)=O Cc1c(CCC(=O)N)cccc1Br.C(C)(C)(C)N N1(C(c2cnc(CC)o2)=O)CCC(C(N2CCC(OCCCCCC)C2)=O)C1CC C(CS(=O)(=O)CCN=c1[nH]c(=NCC(C)OC)[nH]c2c(F)cccc12)OC C1(C(=O)NCC2CCCN2C(c2nscc2Br)=O)CC2(CCOC2)C1 Cn1cc(C(=O)NC2CC(CNC(=O)CCNC(c3ccoc3)=O)C2)ccc1=O C=CCC(CNC(c1ncccc1Cl)=O)C(=O)NC(COC)C1CCC1 C(=O)(CC(C(F)(F)F)NC(c1coc(C(N)=O)c1)=O)N1CCCC(C)(CO)C1 Cc1ccc(C)c(CN2CCC2C(=O)Nc2ncccc2C(C)C)c1 C1(C(=O)NCC(=C)Br)CN(C(=O)Cc2nc(=N)[nH][nH]2)CCC1(C)C N1(C(CC(CNC(CN(C(C)=O)C)=O)OC)=O)Cc2ccccc2C1 C1(NC(C(C)=CC)=O)CN(C(c2ncccn2)=O)CCC1C Cn1cc(C(CO)NC(=O)COCC(F)F)cn1.C1(=O)C(C)(C)N1 N1(C(Cc2cccc(C)c2)=O)CCN(C(c2cc(O)nc(Cl)c2)=O)CC1C Cc1ncc(Br)c(N2CCC(NC(c3conc3C3CCCC3)=O)C(O)C2)n1 N1(C(CC(C2CCC2)OCC)=O)CC2(CCOCC2)C1c1cccc(C(=O)OC)c1 CCCCCCOC(C)C(=O)NCCN(C(=O)C(O)CSC)C(C)C C1(CC(=O)NC)CCN(C(=O)C(Cc2ccco2)NC(c2cnccn2)=O)CC1 C(=O)(C(CC(C)C)ONC(=O)CC(C)OC)N(CC(C#C)C(C)C)C1CC1 N1(C(C(CC)NC)=O)CCC2(CC1)CCN2C(=O)Cn1cc([N+](=O)[O-])cn1 C(=O)(C(F)C(F)(F)F)N1C(CNC(c2c(OC)noc2C2CC2)=O)CC1 c1(C(N(C2CCCC2)CCCNC(C2OCC(C)C2)=O)=O)cnc2occc2c1 N1(C(C2(c3nnnn3C3CCC3)CC(CC)NCC2)=O)CCC2(CCCNC2)CC1 Cc1c(C(=O)NC(C2CCCN2C(=O)CC2CCCC(=O)N2)(C)C)ccn1C c1(CCNC(C(=O)NC(c2cccc(OCC)c2)CCC#C)=O)cc(N)ccn1 C1(C(C(=O)NCC2CCOC2)N(CC(F)F)C(C)C)CCCC(C)C1 C(=O)(C1=CCCC1P(C)(C)=O)N1CC(C(C)NC(CCCCCOC)=O)C1 C1(C(=O)NC2C(C)(C)c3ccccc3C2)CC2(CCN1)CCOCC2 c1(C(=O)NCCCNC(=O)NCC=C)ccc(F)c(F)c1 c1(CN(C(c2c(C)cno2)=O)C)ccccc1CNC(C1CC1CC(C)(C)C)=O c1(C(=O)NC2CN(C(COCc3nnc(C)s3)=O)CC2O)nc(F)ccc1Cl N(C(=NCc1cccc(C(F)F)c1)NCC(CC(C)C)NC(C)=O)C(C=C)C C1(C(=O)NC2(COC)CCCC2)CC=CC(NC(=O)C(F)=C(C)C)C1 n1(CC(=O)NC(CN(C(c2cc(SC)c(C)o2)=O)C)C)ncc2ncccc12 N1(C(CCC(CC)C)=O)CCC(C2CC2)(CNC(c2ccon2)=O)C1 c1(OC)cc(F)ccc1C(=O)NCCC1CN(C(=O)C(C)CC2CC2)CCCO1 N1(C(c2nn(C)c(CO)c2)=O)CC2CCCC2C1C(=O)NC1CC2(CCC2)C1 c1(C(=O)NC(C(=O)N2C(CCCC)CCC2)CCOCC)ccc(C)c(O)n1 C(=O)(C1=C(C#N)CCC1)NCC1CCN(C(C(CC(C)C)C)=O)CC1C C1(CNC(C(C)NC=O)=O)CN(C(=O)CCc2cccnc2F)CC(C)(C)O1 c1(C(N(C)CC2N(C(C(COC)(F)F)=O)CCC2)=O)c(F)c(F)cc(C)c1F c1(C(=O)NC(C)C(N2CCOCC2)C)cc2cncn2c(O)n1 c1(CC(=O)NC2CCC(NC(C(N3CCOCC3)C)=O)C2)cc(Cl)sc1Cl C1(Cn2cc(C3N(C(C4CSC4)=O)CCC3)nn2)C2CC(CO)CC12 C12(NC(C3(COC)CCC3)=O)COC(CNC(C3CC3(Cl)Cl)=O)(C1)C2 C=CC(O)(C(=O)NCCCN(C)C(c1nn(C)cc1C)=O)C(F)(F)F c1(C2CCN(C(C)=O)C2)nc(C(C)CC)nn1-c1cccc(C(F)(F)F)c1 C1(C(N2CC3C(NC(C(CCCC)(C)F)=O)C(C3)C2)=O)CCn2c(cnc2C)C1 c1(C(N2C(CN(C(CNC(=O)OC)=O)C)COCC2)=O)cc2nc(Cl)ccc2s1 C1(C(=O)NC2(C)CN(C(=O)C3=CCCC3)C2)CC(c2cccc(F)c2)=NO1 c1(NC(c2n(CCOC)nnn2)c2csc(C)n2)ccc2c(c1)C(=O)N(C)C2 NS(=O)(=O)c1cc(C(N2CC(CNC(C34CC(CO3)C4)=O)C2)=O)cc(Br)c1 CC(c1ccccc1)=CC(=O)NCC1CCC(C(N2CC(S(N)(=O)=O)C2)=O)CC1 CN=c1[nH]nc(CC(=O)NCCC2CCCN(C(C3(C(F)F)CCC3)=O)C2)s1 C1(CC(=O)OCC)CCCN(C(=O)Nc2cnn(CCN3CCOCC3)c2)C1 C=CCC(C)(C)C(=O)NCC12CC(COC)(CN1C(c1cnc(C(F)F)s1)=O)C2 N1(C(c2noc(CC)c2C)=O)CCC(C2CC2)C1C(=O)NC1(C)C(C)(C)C1(C)C C1(CNC(c2c(Cl)nsc2Cl)=O)CCN(C(c2cn(CC(F)(F)F)nn2)=O)CC1 C1(CCCNC(=O)CCNC(c2cccs2)=O)CCCN1C(c1ccsc1)=O C1(NC(C(=Cc2cccs2)C)=O)COC2(C1)CN(C(c1ccc(C(C)C)s1)=O)C2 c1(C(N2CC3CN(Cc4ccc5c[nH]nc5c4)C3C2)=O)ccc2ncccc2c1 c1(C(N2CC(NC(C(CC)(C#N)CC)=O)C(O)C2)=O)cncc2ccc(F)cc12 c1(C(=O)NCCN2CCN(C(C3C(C)C3)=O)CC2)ccc2c(c1)OCCCO2 Cc1ccccc1CCNC(=O)C=CC1CCCN1C(=O)C(C)O n1(CC(=O)NC2CC(CNC(=O)C(F)(F)C3CC3)C2)ncc2ccccc12 N1(C(C=CCCC)=O)CCC2(CCCN(C(C3CC3C)=O)C2)CC1 c1(OCC)c(C(N2CCC(CCNC(=O)CC3COCCO3)C2)=O)cccc1F c1(CNC(=O)NCc2ncc(C(C)(F)F)s2)cccnc1-n1cccn1 C(C1(CC(=O)OC)CCOc2ccccc21)N1CCN(c2ncc(OC)cn2)CC1 CC1CC(C(=O)NC2(C(N)=O)CCOCC2)CN(C(C2(C3CCC3)CC2)=O)C1 C(C(=O)NCCC)(C(C1CCCC1)OC)N(CC=C)C(C1CCOCC1)C1CCC1 CCC(CC)(C(=O)NC1CCC1C(=O)NCc1ccc(F)cc1)OC C(=O)(C(C(C)C)NC(=O)C(N1CCOCC1)C)NCc1c(C)nns1 c1(CNC(C(=O)NCC(COC)O)=O)ccc2cc(C)ccc2n1 CCC(C)C(C(C(=O)NC(C)(C)C)N1C2CCCC1CC2)OC Cc1cc2c(cc1C)N(C(C1(C)CC3(CCC3)C1)=O)CC2 S(=O)(=O)(c1ccc(Br)cc1NCC1CCOC1)N1C(CC(C)C)CCCC1 c1(C(=O)NC2CN(C(CC3(C)CCCCC3)=O)C2)cc2nc(F)ccc2o1 CN1C(=O)CCC1C(=O)NC1CC1NC(C1(c2cccc(Cl)c2)CCC1)=O c1(C(=O)NCC2(NC(N)=O)CC(NC(CC(=O)NCC)=O)C2)cccc(CC)c1 Cc1nc(C)n(CCCC(=O)NC2CC(O)(CNC(=O)CC3(C)OCCO3)C2)n1 c1(C(=O)NCCN(C(=O)C(C)C2CCCC2)CC)cc(=O)c2ccccc2n1C C1(CNC(C=C(CCC)C)=O)CCCCN1C(c1cc(SC(C)(C)C)ccn1)=O N1(C(C(CCC)=CC)=O)CC(C)CN(C(=O)C(c2c(F)cccc2F)C)CC1C c1(N)ccccc1CCP(C)(C)=O.CC1Cc2cn(nn2)CCCC(=O)C1=O C(=O)(CCC(C)S(C)(=O)=O)N1CC(NC(C(OCC)OC)=O)(COC)C1 CC1CC(C)(C(=O)NC2CCN(C(=O)COCC(F)(F)F)CC2CSC)CCO1 c1(C(N2CCN(C(c3nccc(SC)n3)=O)C(C)C2)=O)c(C)cc(C)cc1O N1(C(C2N(C)C(=O)CC2)=O)CCN(C(=O)COC2CCOCC2)CC1CCO N1(C(C2N(C(CCC)=O)CCC2)=O)CC(NC(C2CCCN2C)=O)CC(F)(F)C1 C12(C(=O)OC)CCC(NS(=O)(=O)CC3CCC(N)C3)(CC1)CC2 C12CCCC1C(c1cnn[nH]1)(C)C1(CCC1)C(=O)N1C(CCC1)C(=O)N2.CCO Cc1ccccc1OCC(=O)NCC(O)CNC(c1cc(NC2(CO)CC2)cs1)=O C12(CC(=O)NC(C(=O)NCCC)C)CCC1CN(C(=O)CCn1ccnn1)C2 Cc1conc1CNC(C1CCCC1CNC(C1CCC1CF)=O)=O c1(N(C)C)ncc(C(=O)NCC2CN(C(c3ccnn3CCF)=O)CCO2)cc1Cl N=c1cc[nH]cc1C(=O)N(C1CCCC1)CC1CCN(c2ccccc2)CC1 CC1(C(N2CC(c3ccccn3)C2)=O)CCN(C(c2ccc(F)cc2)C2CC2)CC1 C(C(CC(F)(F)F)NC(C12CCC1C2)=O)NC(c1cncc(SC)c1)=O C(=O)(CC(=O)NCC(C)(C)CCNC(=O)C(C1CCCO1)c1cccs1)OCC CCC(Cc1ccccc1)CC(=O)NCC1(F)CCN(C(C2COC2)=O)C1 c1(C(CNC(=O)CN(C)C(c2ccn(C)n2)=O)OC)ccccc1C c1(C(N(C2(c3ccccc3)CN(c3nc(C4CC4)ns3)C2)C)=O)cc(O)nn1C C(=O)(CCC(CF)CF)N1CCCC(CNC(C2CCC(CCCC)CC2)=O)C1 c1(C(=O)NC2CC(CNC(C3CC3C(F)F)=O)C2)c[nH]cc1C(F)(F)F C1(NC(c2cccc(COC)n2)=O)CN(C(C2CC2C)=O)C2CCCCC12 c1(CNC(c2c(CC)cccc2F)=O)cc(Cl)cc(Cl)c1O N1(C(C2OCC(C)C2)=O)CC2CCCN(C(c3ccc(-c4ccco4)o3)=O)C2C1 CC1(CNC(C2(C#N)CC2)=O)CCC(NC(c2csc(C(N)=O)n2)=O)C1 c1(OC)cc(OC)c(F)c(NC(C2CC(=O)CS2)=O)c1 CC12CC1(C)CN(C(=O)C(=O)Nc1cncnc1)C2 c1(C(=O)NC(C)C(=O)Nc2csc(Cl)c2)ccc(O)nn1 c1(NC2CCCN(C(c3ncc(OCC)nc3)=O)C2)nnccc1C#N C(=O)(C1=CNC2=NCCCC2=C1)NCC1CCC(C)N(C(C2CC(C)(C)C2)=O)C1 C(=O)(C(C)CC(C)C)NCCC(N1C(C)(COC)C=CC1)=O CCCCCCC(C)(CCC)C(=O)N1CC(NC(c2cc[nH]n2)=O)CC(F)C1 C1(COC)CCN(C(C2(CNC(=O)C(F)=CC3CC3)CC(C)(C)C2)=O)CC1 C1(O)(C(=O)NC2C(OC)CN(C(=O)C(F)=C(C)C)C2)CCCCCC1 c1(C(N2CCCC(CC=C)(NC(C3CCC(F)C3)=O)C2)=O)c(C)cc(=O)oc1C CCC(C)C(O)C(=O)N1CC(OC)CC(NC(=O)CN(C2CCSC2)C)C1 C1(NC(CCOC)=O)CCCCN1C(C1CCN1S(C)(=O)=O)=O C(=O)(C1=COCCO1)N1CCC(OCCNC(CC(C)c2ccncc2)=O)C1 C#Cc1cc(F)c(C(=O)NCC2CC(C)(C)CN2C(c2csc(C)c2)=O)cc1F C1(CC(C)NC(CC=C)=O)CC2CCC(C1)N2C(=O)Cc1ccc(C)cc1 c1(C(=O)NC(C(C)NC(C(CC)(CC)CO)=O)C)cnn2ncccc12 C(=O)(C(C)(C)C(=O)NCC1CC(O)CN1C(C1(C(=O)OC)CC1)=O)NC C1(C(N2CCC(SC)C2)=O)CC12CCN(C(=O)C1=COCC1)CC2 C(=O)(CC(C)(C)CC(F)F)N1CC2(OCC(NC(c3c(CC)occ3)=O)C2)C1 CC1CC(C#N)(C(N2CCOC(CC(=O)NCCCc3nncs3)C2)=O)C1 CC1(O)CCN(C(C23CC(NC(c4nccs4)=O)(C2)C3)=O)CC1O C1(C(=O)NCC(=O)NCC(=O)NCC(CCC)C)CSCC(=O)N1 Cc1ccc(CN(S(=O)(=O)C2CC2c2ccc(Cl)cc2)C)c(C)c1 Cc1nccc(Cl)c1C(=O)NCC1C(C)CCCN1C(=O)C1=NOCC1 C1(CNC(c2cn(CC=C)nn2)=O)CCN(C(c2cc(Cl)c[nH]2)=O)CC1 c1(C(C)N(C2CC(NC(C)=O)C2)C)ccc(C(=O)C(C2CC(=C3CC3)C2)=O)cc1 Cn1cc(Cl)c(C(=O)NC2CCCCC2C(=O)NC(c2ccccc2)CO)n1 C1(NC(c2c(N)cccc2Cl)=O)CCN(C(=O)Cn2cc(Cl)cn2)CC12CCC2 C(=O)(C1=CCN(C(C2(CC=C)CCOC2)=O)CC1)NC(C=C)COC c1(CN2C(CC)CC2)ccncc1-c1ccccc1.C(C)(C)(C)N(C)C(=O)OC N1(C(C2C(CC(C)C)C2)=O)CC(C(=O)NC2CC(=O)N(C3CC3)C2)CCC1(C)C CC(C)CC(F)C(=O)NCC1C=CC(NC(=O)CCc2cn[nH]c2)C1 CC(C)(O)C(F)(F)C(=O)N1Cc2occ(C(=O)Nc3cccc(C(N)=O)c3)c2C1 N1(C(C(C)S)=O)CCc2[nH]nc(C(=O)Nc3cnnc(Cl)c3Cl)c2C1 c1(NC(N(C)CC2(N)CCC2)=O)cccc(N=S(C)(C)=O)c1 C(=O)(CC(C)(C)N(C)C)NCC1(OC)CN(C(=O)C(N2CCSCC2)C)C1 c1(N(CCCNS(CC)(=O)=O)C)ccc(C(F)(F)C(F)(F)F)cc1C c1(N2Cc3c(O)nccc3CC2)nc(=NCC2CC2(Cl)Cl)[nH]c2c1CSC2 C1(C(=O)NC(C)CCNC(c2cc(C(F)(F)F)c[nH]2)=O)CN2CCC1CC2 C1(NC(C(CC)OCC)=O)CCOCC1NC(C1(C2CCC(=O)O2)CC1)=O CC1CC(CCNC(=O)C=C2CCC2)CCN1C(=O)CC(=O)NC1CC1 N12CCCC(C)(C1)C2=O.c1(OC)cccnc1CNC(=O)CSCC(C)C C(CC(F)F)(C(=O)NCC1CC(C(C)(C)C)C1)NC(Cc1ccn(C)n1)=O c1(C(N2CCN(C(C3CC(=C)C3)=O)C3C2CC3)=O)cccc(C#CCO)c1 C(=O)(C1SCc2cccnc21)NC(C)CN(C(=O)COCC(F)F)C CC(C(=O)NCCCCNC(=O)C(c1ccccc1)Sc1ccnn1C)C(F)F N1(C(Cc2ccc(C)s2)=O)CCC=CC1C(N1CCC(N(C)C)CC1)=O C#Cc1cc(C(=O)NCC2CC3CC(C2)N(C(=O)CCOC)C3)cc(Br)c1 N1(c2snc(SC)n2)CC2CCN(C(c3cc4c[nH]cnc-4n3)=O)CC2C1 C1(CNC(CCN(CCCCC)C(C)C)=O)CC(F)CN1C(c1cnns1)=O C1(CC(=O)NC(CCN(C(c2c(CCC)nns2)=O)C)C)CCC(=O)N1C CCC(CCCC(=O)NCCC1CCC(=O)N1)NC(c1nccn1C1CC1)=O CCC(C)CC(=O)C(=O)N1CCC=CC1C(=O)NC1(c2cc[nH]n2)CC1 CC1Cc2c(Cl)c(Br)cc(F)c2CN1N1CCCC1c1ncccn1 N1(C(c2n(CC)ncc2)=O)CCC(CNC(c2ccn(C(C)(C)C)n2)=O)(OC)C1 N1(C(C2CCN(C(C(CC=C)C)=O)C2C(C)C)=O)CCC12CCC(C)CC2 C1(C(N(C)Cc2ccncc2)=O)CC2(CCC2)CN1C(=O)Cc1cnn(C(F)F)c1 CC1=C(C)CC(C(=O)NC2(C(=O)NCC3CC3(C)C)CCSC2)CC1 N1(C(CCCC(C)C)=O)CCC(NC(c2csc(CC(C)C)n2)=O)C(C)(C)C1 CC(C)C(CC(=O)NC(C)CN(C)C(c1cnc(S)n1C1CC1)=O)C(C)C N1(C(c2nc(OC)oc2)=O)CCC2CN(C(C3CCC=CCCC3)=O)CC2CC1 CC(C)(C#N)CCCC(=O)N1C(C(=O)NCC2(C)CC3CCC2C3)CCC1C C1(CC=C)(NC(c2coc(Br)c2)=O)CCN(C(c2cc(O)ncn2)=O)C1 C(=O)(C1=CCC(NC(c2ccccc2F)=O)C1)N(C)CC1(O)CCCC1 C(CC(C)(C)C(=O)NCCC1CCCO1)NC(c1c(C)ccnc1)=O c1(C(N2C(C)CN(C(c3cncnc3)=O)CC2)=O)cc(C#N)c(N)cc1O CC(C)CCCC(C)C(=O)NCC1COCCN1C(c1ccnn1C)=O C1(C(=O)NCCOCCC)CNC(=O)CN1C(=O)Cc1cn[nH]c1 C1(n2cc(C(CC)OC)nn2)C=CCC(C(N2CC(SC(C)C)C2)=O)C1 C1(C)(CNC(CN(C(=O)Cc2scnc2C)CCC)=O)CCC2CC2C1 CCC(C(=O)NCC(C)CN(C)C(c1ncccc1COC)=O)C(C)O N1(C(C2CCC(C)N(C(=O)CC3(C)CC3)C2)=O)CCc2c(O)noc2C1 C(=O)(CCCCC(C)(C)C)NCC(CNC(C(C(CC)C)N(C)C)=O)(C)C C1(C(=O)NC(CNC(=O)CNc2ncccn2)C2CC2)CCC2(CCC2)O1 C=CCC(C(=O)NC(Cc1cn[nH]c1)C(=O)N(C)Cc1cscn1)OC Cc1ccc(C(=O)NC2(C3CN(C(C4(C#N)CC4(C)C)=O)C3)CC2)c(F)c1Cl N1(C(C2OCCO2)=O)CC2C(=O)N(c3cccnc3)C(=O)C2C1 c1(C(=O)OC2CCCC(OC)C2)cccn(C(C)(C)C)c1=O c1(C(=O)NC2(CNC(=O)Cc3ncccn3)CCC2)ccc(F)c(CCO)c1 C(=O)(CCCCCF)NC1C(OC)CN(C(c2c(Cl)csc2Cl)=O)C1 N1(CC(CC)Cc2ccc(Cl)cc2)CCC(F)CC1(C)C CC1CCC(CC(=O)NCCn2cc(C(=O)N(C3CCC3)C3CC3)cn2)C1 C1(CSC(C)CC#N)CC(C(C)(C)C)=NO1 c1(CC)nc(C)[nH]c1C(=O)NCCC1(O)CCN(C(=O)COCC(=O)OC)C1 C1(C(C(=O)NCCC(=C)C)F)CCN(C(c2cc(OCC)no2)=O)C1 CCC(C)C(C)C(=O)NCc1cc(C(=O)NCC2(C)CCCCC2)ccn1 C12(C(=O)NCC3CN(C(N)=O)C3)CCC(CN(C(c3cncs3)=O)C1)C2 c1(C(=O)NC(CCOC)CNC(C2COCCOC2)=O)ccc(F)c(C)c1C C(=O)(C(CN(C)C)C(C)C)NCC(CCC)NC(c1c[nH]nc1Cl)=O C1(CNC(C(C)CF)=O)CCCN(C(C2(C)CC(F)C2)=O)C1 C(=O)(CS(=O)(=O)C(C)(C)C)N(CC(C)NC(=O)Cc1cc2ccccc2o1)C N1(C(c2cn[nH]c2)=O)CCC(F)(F)C(CNC(C2(F)CCCCCC2)=O)C1 N1(C(C2(C)CC(C)C2)=O)CC2(COC(CNC(=O)C(C)OCC3CC3)C2)C1 N1(c2cc(N3C4CCC3CC4)ncn2)CCCCC(S(C)(=O)=O)C1.CS(C)(=O)=O N1(C(c2c(C)nc(O)cc2)=O)CC2CCC(C(=O)N(C(CCO)C(F)F)C)(C2)C1 C1(OCCOC)C2CC1N(C(=O)O)C2.C1(C(=O)OC(C)(C)C)(CO)CC(C)(C)C1 C#Cc1ccc(N(C(c2ccc(OCc3ccccc3)c(I)c2)=O)CC)cc1Br CC(CC(=O)N(C)CC1C2CN(C(c3nccc4n[nH]cc34)=O)CC12)P(C)(C)=O C1(NC(=O)CSC(F)(F)F)C2CC(NC(C(C)c3ccco3)=O)CC12 C1(C(=O)NC(CNC(C(COC)(F)F)=O)C(C)(C)C)OCCOC12CCC2 CN1CCN(C(c2ccn(C)c(=O)c2)=O)CC1=O.c12cn(nn1)C1CCCC1NC2 N1(C(COC2(C#C)COC2)=O)CC2CN(C(=O)Cc3ccc(OC)cc3)CC2C1 c1(C(N(CCC(C)NC(C2CC2F)=O)C)=O)cn(C)nc1-c1cnn(C)c1 C(=O)(C(CCC1CC1)NC(c1cc(CSC)on1)=O)NCC(CC)C Cc1ncc(C)c(N2CCOC(CN(C(=O)CCCc3ccccn3)C)C2)n1 C1(C(N(CC)Cc2ccc(O)cc2)=O)CCN(C(c2cc[n+]([O-])cc2)=O)CC1O N1(C(C(=O)NC2C(=O)C2)=O)CC2CCCC(OCCCO)C2C1 N1(C(c2c(C(C)C)ocn2)=O)CC2(C1)CN(C(C1C3CCCC13)=O)CCO2 C(=O)(C(CN(C)C)NC(=O)C(F)CC1CCOC1)NC1(CN(C)C)CC1 C(=O)(C(C)(C)C1CCN(C(=O)C(O)CF)C1)C(COC)=O.NC c1(C(=O)NC2C(C)N(C(c3csc(O)n3)=O)CCC2)ccc2c(c1)CCCC2 c1(C(N2CC(O)(C(C)(C)CNC(=O)C=C(Cl)Cl)C2)=O)cc(C(F)F)ccc1F C1(NC(=O)NCc2c(Cl)cn(C)n2)COc2ccc(F)cc2C1 N#Cc1nc(=NC2CCCN(C(c3cc4c(F)cccc4s3)=O)C2)cc[nH]1 Cc1ccc(NS(=O)(=O)CCN2CCCCC2)c(NS(C)(=O)=O)c1 CC1CN2CCC1NC(=O)C2=O.c1(NCC2CC2)c(C(F)(F)F)ccnc1Cl C1(NC(C(C=CC)O)=O)CCC2(CCN(C(=O)C(C)CC3CCCC3)C2)C1 C(=O)(C(CC(C)C)NC(=O)OC)N(CC(CNC(c1noc(CC)c1C)=O)C)C Cn1c(NC(=O)C(F)(F)C(F)F)cc2sccc12 c1(C(N2CCC(CNC(C=CCCC)=O)C23CC3)=O)cc2cc(Cl)ccc2s1 N1(C(C2C(NC(C3(CC)CCCC3O)=O)C3CCC2C3)=O)CCC(C2(O)CC2)CC1 c1(NC(C)=O)cccc(F)c1C(=O)NC1CN(C(=O)C2CC2)CC1F C1(CC#C)CCCN(C(=O)C(CO)NC(=O)CCC=C=C)C1 CC#CCCC(=O)N1CCCC(NC(=O)CCC2(C)CC2(F)F)C1 C1(NC(C(C)S(N)(=O)=O)=O)COC2(C1)CN(C(=O)C#CC1(C)COC1)C2 N1(c2c(C#N)cncc2)C2CCC1CN(C(c1cc(CN)no1)=O)C2 C1(CNC(c2cn[nH]c2)=O)CN(C(c2cn(CC(F)(F)F)cn2)=O)CCCO1 c1(CC(=O)NC(CC)(C)C)csc(CNC(=O)CC2CCOC2)n1 Cc1cccc(OCCCC(=O)NCC(C2CCN(C(C3CCC3)=O)CC2)F)c1 c12n[nH]cc1C2(C)NC(C(C)NCC)NC(=O)OC.c1(CC)nnnn1C1CC1 c1(OC)nccc(Br)c1C(=O)NC1C=CC(CNC(=O)C(C)NC(N)=O)C1 N1(C(C2CCC(n3cc(C4(O)CCC4)nn3)CC2)=O)CCC2C(C1)C2(F)F c1(CCC(=O)NCC(=C)CCNC(c2csc(O)n2)=O)ccncc1Br c1(C(=O)NC2CCC(NC(c3ccon3)=O)C2)cc(C(F)(F)F)ncn1 C12(CNC(C3CCOC3)=O)CCCC1N(C(=O)CC(O)C1CCCC1)CCC2 c1(CC(=O)NCC2CC2F)c[nH]ccc1=O.N12CCN(CC1)CCNC(=O)C2 C1(C(N2CCCC(CN(C(C3CC(SC)C3)=O)C3CC3)C2)=O)CC2OC1C1CC21 CC1=C(C(=O)N2CCC(C)(NC(C3CCCC(C(N)=O)C3)=O)C2)C(C)(C)CCC1 c1(C(=O)NC2CC(CNC(CC(COC)(C)C)=O)C2)ccc2c(c1)NC(=O)CC2 c1(CN2CCC3(C(C(=O)Nc4c(C#C)nccn4)C3)C2)cnc2ccc(C)cn12 c1(NC(C(=O)NCC2(CC#C)CCOCC2)=O)cc(Cl)c(Br)cn1 CN(C(=NCC1CCC1)NCC1CC2CC2C1)Cc1ccccc1F C=CCCCC(=O)NC(CN(C)C(C1CC1c1ccccc1)=O)CC c1(OC)cc(C(N2CCN(Cc3cnc(Cl)cn3)C3CC23)=O)cc(O)c1O C(N=c1nc2c(cnn2C)c(NCC2(CO)CC=CC2)[nH]1)C1(N(C)C)CCC1 C12(COC)CC(NC(=O)N(CCNC(C)=O)C3CC3)(CO1)C2 C1(N(C)C(c2ccc(C#N)s2)=O)CCCN(C(=O)CCNc2cncnc2)CC1 N1(C(CCCC=C)=O)CCN(C(c2nc(C(F)(F)F)cc(C)n2)=O)CC(C)(C)C1 C1(NC(C(N2CCCC2CO)C)=O)CC12CC(NC(=O)Cn1nccn1)C2 N1(C(c2cc(CC)nc(O)c2)=O)CC2(COC(CNC(C3(F)CC3)=O)C2)C1 Cn1c(CCC(N2CCCC2(C)C(N)=O)=O)nnc1S O=C1OC2CCC1CN(C(C1CCC(C(F)(F)F)CC1)C(=O)N1CCCC1)C2 N1(C(C(CCC)OCC)=O)CCC2(CC1)OCCC2NC(c1cnccc1Cl)=O c1(OC)cc(C)c(C(=O)NCCC2(NC(=O)CC(C)CF)CCCC2)cn1 C1(OCCNC(C(C)C)=O)CCN(C(C2CC2(C)Br)=O)C1 N1(C(c2c(C)nsc2)=O)CCC2(C1)CN(C(=O)CCC1CC1(C)C)C2 c1(N2CC(=C(CNC(c3cnc(C)[nH]3)=O)F)C2)cncc(Cl)n1 N1(C(CC)=O)CCCC(O)(CNC(c2cccn(C3CCSC3)c2=O)=O)CC1 N1(C(C(=O)Nc2c(C)cccc2C)=O)CCN(C(=O)C2=CCCCC2)C2CCC12 C1(CC(=O)N(CC(C)NC(CCc2onc(C(C)C)n2)=O)C)CCCC1(F)F C(=O)(C1CCCc2nncn21)N1CCC(COC)(NC(c2csc(CO)c2)=O)C1 N(S(=O)(=O)N1CCCC1C)CCCC.c12ccc(cc1F)[nH]2 N1(C(C(CC)COC)=O)CCC2C(NC(c3ccccc3SCCO)=O)CC12 Cc1cccc(C)c1NC(c1ccc(CN2CCCC(CN(C)C)C2)s1)=O C1(C(=O)NCC2C(NC(C(C(=O)OC)(C)F)=O)CC2)CC2(C1)CC(F)(F)C2 C(=O)(CCCC(=O)NC(C1CCN(C(=O)C(C)OCC)CC1)C)NCC C1(CNC(c2nc(COC)sc2)=O)CC2(CC2)CN1C(C1(CO)CCCC1)=O CC1(O)CCC(CC(N2CC(CO)(NC(=O)CN3CCOCC3)C2)=O)CC1 C=CCC(CNC(C1CC(C(F)(F)F)C1)=O)NC(c1coc(CO)c1)=O CCS(=O)CC(=O)NCC1(CNC(c2[nH]ccc2-c2cccs2)=O)CC1 C1(NC(CCC(C)NC(C(C(C)O)NC(C)=O)=O)=O)COC2(CCC2)C1 N12CCCC1C2=O.C(=O)(CCCC1CCCC1)NCC1C(NC(CC)=O)CC1 CC(C)(O)C(F)C(=O)N1CCC1C1CCN(C(c2ccn(CCF)n2)=O)CC1 c1(OC)cnccc1C(=O)NC(C)C(C)NC(=O)C(F)(F)c1csc(=N)[nH]1 C(C(C)(C)CC(=O)N1CC(C2CCCO2)C1)NC(c1c(CC)oc(C)c1)=O C1(NC(C(CC)C)=O)C2CC3C1C3C2C(=O)NCC1CCN(CC2CC2)C1 c1(C(=O)NCCN(C(C2C(F)(F)C23CCC3)=O)CC)c(F)cccc1Br N1(C(c2c(C)c(Cl)cnc2)=O)CC2CCC(N(C(=O)C(F)CC3CCC3)C)C2C1 S(=O)(=O)(c1ccc2oc(=O)ccc2c1)C(CCn1cc(-c2cc(C)no2)nn1)=O c1(C(=O)OC)nccnc1CNC(=O)N(c1ccc(Cl)cc1)C.c12ccccc1N2 c1(C(=O)NC2(CNC(C3CCC(C)S3)=O)CCCCC2)cnn2c1CCC2 CCCCC(O)C(=O)NCC1CC2(CC2)CN1C(C1CCCN(C(C)=O)C1)=O N1(C(C(CC=CC)NC(=O)COC(C)=O)=O)CCOC2C(O)CC12 c1(C(=O)NC2CN(C(C3ON=C(C(C)C)C3)=O)CC3C2C3)ccc2c(cnn2C)c1 C(C(C)C(F)C(=O)NC(CCO)C(C)(C)O)ONC(COC1C2(C(C)C1)CC2)=O c1(C(N2C(C)CC(NC(C3CC(OC)C3)=O)C2)=O)nc(OC)ccc1Cl CCS(=O)(=O)CCCCNCCC12COC(C1)C2 c1(CC(=O)NCC2(OC)CN(C(c3cncc(C)c3)=O)C2)ccccc1SC C(=O)(C1CCc2snnc21)NC1CCCC(NC(C(C)(C)n2ccnn2)=O)C1 N1(C(CC#C)=O)CCC(CC(=O)Nc2cnn(C)c2-c2nn[nH]n2)C(F)(F)C1 C1(N(C(=O)CC2CCCN2C(=O)CC2CCCC2O)CC)CC=C(C)CC1 C(N=c1nc2sccc2c(N2CCC(CO)C2)[nH]1)C1C(O)CCCC1 N1(CCCc2cccc(OCC)n2)CCC2(CC1)CNC2c1ccccc1 c1(C(=O)NCC2CC2NC(C(C2CCCN(C)C2)(C)C)=O)c(F)cc(F)cc1F c1(N2C(C)CC(CNC(c3cc(OCC)no3)=O)C2)ncnc2sccc12 C1(CNC(=O)C(O)c2ccsc2)CCN(C(=O)CC2CCCCO2)CC1 C1(C(=O)NCCN(CCC)C(c2cc(CC)nnc2C)=O)CCn2ccnc2C1 c1(NC(=O)NC)ccncc1C(=O)NCCNC(=O)Cc1cccnc1COC C(=O)(C(O)CC(N)=O)NCCCN(C(C1CCC(NC(=O)N(C)C)CC1)=O)CC C(=O)(C(C)CC(F)(F)F)N1C(C(N(C2(C#C)CC2)C)=O)COCC1 S(=O)(=O)(c1cc(C(=O)OCC(c2ccncc2)O)ccc1Cl)NC(C)=O C(C(CO)(CO)NC(c1cc(C2CC2)nn1C)=O)N(C(=O)CC1CCCCN1C)C c1(C(N2CCC(CNC(c3ccccc3C(F)F)=O)C2)=O)c[nH]c(=O)cn1 C1(C)(C(=O)NC2C(C(=O)NCC(c3ccccc3)N(C)C)C2)CCCC1 C1(C)(C(=O)OC)CC(C(N2CCC(NC(=O)C(C)COc3ccccc3)C2)=O)C1 N(C(=NCCC(C)C)NCC1CCCC(CO)CC1)CC1(O)CCC1 C1(NC(C2CCC3(CC3)C2)=O)CCS(=O)(=O)C12CN(C(=O)CCC#CCO)C2 C1(C(=O)NCc2onc(COC)n2)CN(C(=O)CCc2ccn(C)c2)CCO1 c1(CNC(CCS(C)(=N)=O)C)cc(=O)n2ccsc2n1 Cc1nc(C(=O)NCCC(O)CNC(=O)C=CC2CCC2)cc(O)n1 N1(NC(N2COCC2(C)C)=O)CCC(O)C(Cc2ccc(C)cc2)C1.C1CO1 c1(C(C)NC(N2CCOCC2c2ccco2)=O)cc(S(C)(=O)=O)cs1 C(=O)(C1CSc2ccccc21)NC1CCCN(C(c2cc(CC)nn2C)=O)C1C N1(C(C2(C(CC)=O)CC2)=O)CC(C)CN(C(=O)CCC(C)(C)C)CC1C C12(NC(C(=O)NC(C)C)=O)CCCN(C(C3CC(=O)N(C)C(=O)C3)=O)CC1C2 c1(C(C)(C)C)ncc(C(=O)NCCn2cc(COCC(N)=O)nn2)n1C C1(NC(c2ccccc2Cl)=O)(CO)CCN(C(=O)CCC(F)(F)F)CC1 N1(C(C2(Cc3nc(CC)[nH]n3)CC2C)=O)CC2CC1C2C(=O)N.C(C)(C)(C)NC(=O)O N1(C(Cc2c(C)sc(Br)n2)=O)CC(C)c2ccccc21 Cc1cc(CC(=O)NC(CC(=O)NCC2CC2C2CC2)C2CC2)on1 C12(NC(c3coc(Cl)n3)=O)CCC1CN(C(C1CCN(CC3CC3)CC1)=O)C2 N1(C(c2cc(C)on2)=O)C2CCC1CC(F)(CNC(c1cnc(O)o1)=O)C2 CCCC(F)C(=O)N(CCN(C(=O)C(C(C)C)N1CCCC1=O)C)C(C)C CC(C)(C)CC(O)C(=O)N1CC(C2CC2)(C(N2CCS(=O)CC2)=O)C1 CC1CN(C(C2(NC(=O)CCCCN=[N+]=[N-])CSC2)=O)Cc2c[nH]nc21 c1(CC(=O)NC2C(C)N(C(C3CC3F)=O)CC2)cc2ccccc2cc1O c1(C(N2C3CC(NC(=O)CSc4cccs4)C3CC2)=O)ccc(Cl)c(Cl)c1O N1(C(c2cccc(C)n2)=O)CCC2(CC1)CN(C(C1(F)CC1C)=O)CC(C)O2 Cc1n[nH]c(C)c1C(=O)N(C1(CC(=O)NCC2CCSC2)CC1)C CCS(=O)(=O)CCN(C(=O)C=CC(C)(C)NC(=O)CC(C)n1cccn1)C1CC1 N1(C(C(C)(C)NC(=O)C(C)C(F)F)=O)CCC(CNC(C)=O)(CF)C1 N1(C(C(P(C)(C)=O)O)=O)CC2CC(NC(c3cc(Cl)nn3CCO)=O)CC1C2 N1(C(COCCOC)=O)CCC(CNC(C2(C)CCCO2)=O)C12CC2 C1(CNC(c2n(C)ncc2)=O)CC(C(=O)NOCc2ccc(F)cc2)=NO1 N1(C(C(CC)=CC)=O)CC(C)CN(C(=O)CSC)CC1C N1(C(C(=CC2CCCC2)C)=O)CCN(C(C2CCS(=O)(=O)N2)=O)C(c2cn[nH]c2)C1 C1(NC(c2c(C)nc(C3CCC3)s2)=O)CC2CC1N(C(=O)Cn1cccc1)C2 C1(C(=O)NCc2c(=O)cc(C)[nH]c2)CCc2nnn(C3CCC3)c2C1 C1(COC)(CNC(C2CC(F)(F)CS2)=O)CCCN1C(=O)C(C)NC(C)=O N1(C(CC(C)NC2CC2)=O)Cc2ccc(CNC(c3cncnc3)=O)cc2C1 C(=O)(C(CO)NC(=O)Cc1cn(C)cn1)N1CC(COC)C1 c1(C(=O)NC2(CN(C)C(C3(C(F)F)CCCC3)=O)CC2)cncc2c1CCC2 CC12CN(C(c3ccncc3)=O)CC1CN(C(C1CC(CF)C1)=O)C2 O=S(=O)(c1cncc(Br)c1)Nc1csc(Cc2cncc(Br)c2)n1 CCCC(C(=O)NC(C)CCN(C(=O)CCC1(COC)CCCC1)C)OCC Cc1ccc2c(c1)CCN(C(C1CC(=O)N1)=O)C2 C(=O)(C1=CCCC1(C)C)NCCN(CCCN(C)C)C(c1cnc(C(F)(F)F)s1)=O C(=O)(CCCC(=O)NCc1ncoc1C1CCN1C(=O)NC1CCCCC1)OC O=C1CSc2ccc(C(N3CCN(C(=O)C=CC(F)F)C4CCC34)=O)cc2N1 C(CC(C(C)C)CCOC(c1cn(C2COC2)nn1)=O)NC(C1C(=C)CC1)=O c1(C(C)(C)C)ccc(N)c(C(=O)N(C2CC3CC2CN3)c2ccccc2)c1 c1(NC(N2CCC(c3ccc(=N)[nH]n3)C2)=O)cc(O)nc2ncccc12 Cc1cc(C(=O)NC2(CO)CCCN(C(c3snnc3C)=O)C2)cc(Cl)c1 c1(C(=O)NCCOC2CCN(C(CC3CC(=C)C3)=O)C2)cc(O)ncc1Br c1(C(=O)NCC2(Nc3cc(C4CC4)nc(Cl)n3)CC2)cccc2cnsc12 CC(C(O)C(F)F)NC(c1cnn(CCNC(=O)CCc2cnn[nH]2)c1)=O N1(C(c2c(CC)nc[nH]2)=O)CCCN(C(=O)CCC(C)(C)C)C(C)C1 Cc1ncc(Cl)c(C(N2CC(NC(c3cc[nH]c3)=O)CCC2C)=O)n1 C=CC(CC)CC(=O)N1CCCCC1C(C)NC(c1cnc(C(C)C)nc1C)=O c1(OCCC)ccc(C(=O)N2CCNC2=O)cc1.N(S(=O)(=O)N(C)C)CC1CC1 C(CC(O)C(=O)NCCC1CCN(C(C2CNC(=O)C2)=O)CC1)SC c1(C(N2CCC(C)(NC(c3ncn(C)c3)=O)C2)=O)cc2cccc(Cl)c2s1 n1(CC)ncc2cc(C(=O)NCCC(C)CCNC(=O)Cc3ccco3)cnc12 Cn1ncc(CNC(c2nc(Cl)cs2)=O)c1C(=O)NC1CC(CC(F)F)C1 c1(C(=O)NCC2CC(NC(=O)COc3ccc(F)cc3)C2)ccccc1[N+](=O)[O-] c1(C(=O)NCC2C3CCC2CN(C(C2CCSC2)=O)C3)ccn2c1CSCC2 C1(N(C(C)C2CC2)C(=O)OC(C)(C)C)CCN(C(=O)C(N)=O)CC1 c1(C(=O)NCCC2C(CC)C2)c(CNC(c2ncc(F)cn2)=O)cnn1C N1(C(Cc2ccc(C#C)cc2)=O)CCC(N(C(=O)C(C2CC2)SC)C)C(C)(C)C1 S(=O)(=O)(CCCCCl)N1C(CC(=O)Nc2c(C(N)=O)cns2)CCC1 N1(C(=O)NCC(C2CCCC2)C)CCC(c2nc(=O)o[nH]2)CC1 n1(CC(=O)NC(CCNC(C=C(CC)C)=O)C)sc2ccccc2c1=O C1(CC)CN(C(c2c[nH]cc2CC)=O)CC1NC(C1CCCN1C(C)=O)=O Cn1ccn2ncc(C(N3CC4(CC(NC(c5cscn5)=O)CO4)C3)=O)c12 C1(NC(c2c(N)ccc(OC)c2)=O)CN(C(=O)C(C)C(C)O)CC12CCOCC2 C1(NC(C(n2ncc(C)c2)C)=O)CC2CC1N(C(=O)C(C)(C)C#N)C2 c1(C(N(CC(F)Cl)C)=O)cc(CCN(N2CCOCC2)C(C2CCCO2)=O)on1 N1(C(=O)Cc2ccncc2Br)CC2CC1CN2C(c1ccccc1CO)=O C1(C)(OC(C(CC(C)C)ONC(CNC(=O)OC)=O)=O)CC(C)(C)OC1=O C12(C(N3CCS(=O)(=O)CC3)=O)CCC(CC1Sc1cccs1)C2 C(=O)(CC1=CCCCC1)NCCCC(CO)NC(c1c(C)nn(C)c1C)=O c1(CNC(C2C(C(=O)Nc3cccc(CCC)n3)C2)=O)cccc(C)c1F c1(CNC(=O)C2CC2)cccc(Cl)c1.Cn1nnnc1SCCOCC(=O)NCCCS C(C(CN=c1[nH]c(=NCCC(C)OC)[nH]c2c1CSC2)OC)OC Cc1cc(CCC(=O)NCC2CCC(NC(=O)C(F)CC3CCOCC3)C2)no1 c1(C(N(CCNC(C(CC)CCOC)=O)CC2CC2)=O)[nH]nc2ncccc12 c1(CC(=O)N(CCCN(C)C(C2(C(F)F)CC(O)C2)=O)C)cnc2ccccc2c1 c1(C(N2C(C)CN(C(C3CCS3(=O)=O)=O)CC2)=O)nccc2ncncc12 C(=O)(C1CCc2ccccc21)N1CCC2(C(NC(c3cnccn3)=O)C2)CC1 n1(CCC(N2CCC3C(NC(C(C)C)=O)C32)=O)c(=O)oc2cc(Cl)ccc12 C(=O)(CCCC(F)(F)F)N1C(C)CC(CNC(c2ccnnc2)=O)C1 C(=O)(CCCN=[N+]=[N-])N1CC(CC(=O)NCC(C)SC)OCC1 C(=O)(CS(=O)(=O)CC)NC(CCCC)CNC(C1C2CCC1CC2)=O O=C1NC2CCC1CN(C(c1ccc(-n3cncn3)cn1)=O)C2 C12(CNC(c3cnc(OC)nc3)=O)CCC(CC1)N2C(C1COC(=O)N1)=O N1(C(c2c(C)c[nH]c2)=O)CCC2(C=C(C(=O)NCC(C)(O)CC(C)C)C2)C1 Cc1cccc2c1CC(C(=O)NCC1CN(C(=O)CC3CCCC34CC4)CCO1)N2 O=S1(=O)CC2CN(Cc3ccc(S(=O)(=O)NCCCO)s3)CC2C1 c1(C(=O)NCC=C(C(=O)N(C(CC)C2CC2)C)C)nccnc1N CC(CC1=CCCCC1)NC(c1cn2c(n1)CCCC2)C c1(C(c2nnnn2CC2CC2)COC)ccc(NCc2ccsc2C2CC2)cc1 N1(CCN(C(CC2(NC(C3C(C)(CC)C3)=O)CC2)=O)C)CCOCC1 c1(C(=O)NCC(CC)NC(=O)CC2(c3ccccc3)CC2)cnccc1NC(C)=O N1(C(CNC(=O)CN(C)CCOC)=O)CC=C(COCCCCC)CC1 c1(C(=O)NC2C3CCN(C(C4CC5(CC5)CO4)=O)C23)cc(Cl)c(Cl)c(Cl)c1 CCC(C(=O)NCC(=O)NCC1CCN(Cc2ccccc2)CC1)C(C)O C(CCCC(=O)NC1(C2CCCN2C(=O)CCC2CCCO2)CC1)N(C)C N1(C(CCC)=O)CC2(C1)CN(C(=O)C(c1ccccn1)O)C2 CC1(C(=O)NCC2=CCCOC2)CCNC1=O.C1C(O)C(=O)N1 N1(C(C(C)C)=O)CCCC(C(N2CCC(NC(C3CC4(C3)CC4F)=O)CC2)=O)C1 c1(CN2CC(C(=O)NCC3(CC)CCCC3)OCC2)cc2n(n1)CCC2 c1(C(=O)NCCOCC)ccc2c(c1)CCN(Cc1ccsc1Cl)C2 c1(C(=O)NCC(F)CNC(C2(C3CC3)CC2)=O)cccc(OCCF)c1 N1(C(CCCSC)=O)CC2C3CCC(C2C1)N(C(c1cc(C)n(C)c1)=O)C3 c1(C(N(CCCN(C(CN2C(C)CC2)=O)C)C)=O)cc(Br)c(C(F)F)s1 c1(N2CCC=C(C(=O)OC(=O)OC)C2)cc(C(F)F)nc2ncnn12 c1(C(N2C(CN(C(Cn3c(C)cnc3)=O)C3CC3)CCC2)=O)ccnc(CO)c1 O=C(C1Cc2ccccc21)N1CCCC(CCNC(C23CCC(CC2)C3)=O)C1 c1(NC(=O)COCC2CC2NC(=O)CCc2ccoc2)c(F)c(F)cc(F)c1F c1(C(N2CCC(O)(CCNC(=O)CCC(F)F)C2)=O)cc2ccc(F)cc2[nH]1 N1(C(c2ccn(C)n2)=O)CCCC(CC(=O)NCc2ccncc2F)CC1 N1(C(C2C(C)(C)C(NC(=O)CN3CCOCC3)C2)=O)CCCC(F)CC1 C(=O)(C1=C(F)CN(C(c2ccc(C(C)=O)o2)=O)CC1)N(C1CCC(OC)CC1)C CC(C)C(F)C(=O)N(C)CCOCCCNC(c1ccc(Cl)s1)=O c1(C(=O)OC)nn(C(C)(C)C)cc1Cl.C12(C(N(CCOC)CC)=O)CN(C1)C2 C=CCC(C)(C)CC(=O)N1CCN(C(=O)Cn2ccc(=O)cc2C)CC1COC CC1CN(C(=O)CC2OCCO2)CCC1CNC(C1CC(C(F)(F)F)C1)=O C1(NC(C=C(COC)C)=O)CC(C)CN(C(C23CC(F)(C2)C3)=O)C1 c1(C2(C(=O)NCC(C)(C3CC3)NC(CC(CCC)O)=O)CC2)cc(F)cc(C#N)c1 c1(C(=O)NCC(N(C)C(c2ncc(C)s2)=O)C2CC2)cc2ncccn2n1 N1(C(CCNC(=O)OC)=O)CC(C(=O)NCCCc2cnn(C)c2)C2(CCC2)C1 C1(C(=O)Nc2ccc(C)nc2I)CC12CCN(C(c1c(Cl)ccnc1Br)=O)CC2 C(=O)(C(C)CC(F)(F)F)N1CCC(CC=C)(NC(c2cccc(CC)c2)=O)C1 c1(CN2C(CC(=O)N(c3ccccc3)CC#C)CCC2)ccc(F)c(Cl)c1F N1(C(C2(OCC)CC2)=O)CCC(C)C(N(C(=O)C(C)=O)C)C1 c1(CNC(CC(C=C)(C)C)=O)cccc2c1CCN(C(=O)CC1CCC(O)C1)C2 c1(C(=O)NCC(CNC(=O)C2=CCCS2)O)nnc(O)c2ccccc12 C(=O)(CC(C)NC(c1c[nH]nc1CNC(c1cc(C)[nH]n1)=O)=O)NC c1(SCC(=O)N(CC(C)N(C(C=C(CC)C)=O)C)C)ccc(O)cc1 CCC(CC)C(F)C(=O)N(CC(O)CNC(=O)CC(CC)C1CCC1)C c1(C(=O)NCC#CCNC(=O)CCNC(c2cccs2)=O)ccc2nccn2n1 C1(COC)(NC(C2CCN(C(=O)Cn3[nH]cnc3=N)C2)=O)CN(C(C)=O)C1 N1(C(c2c(C)nc(C)s2)=O)CCC(C2CC2)(NC(c2cc(Cl)ccc2F)=O)C1 c1(COC(C)(C)C)cccc(S(=N)(=O)C(F)F)c1 c1(OC)cccc(N2CCC(CN(C(C)C(c3ccccc3)OC)C)C2)c1 c1(C(=O)NC2(CNC(CCC=C=C)=O)CCCCC2)cnc2c(cnn2C)c1 Cc1c(O)ccc(C(=O)NC(CNC(=O)C(CC2CC2)CC2CC2)CO)c1C Nc1c(Cl)cc(NC(C2CN(Cc3csc(Br)c3)CCS2)=O)cc1Cl CON(C(=O)C=CC(C)(C)NC(C1CC1C(=O)OC)=O)C1CCCC1 c1(C(=O)NC2(C)CCN(C(C3CCC3C(F)(F)F)=O)C2)cccc2c[nH]nc12 N12CCC(O)(CC1)NC(=O)C2C1CC1.C(=O)(C=CC(C)C)NCCC N1(C(COCCC(C)C)=O)CC=CC1CNC(=O)CCC1CC1(Cl)Cl C1(c2n(CC(=C)C)nnn2)(N(c2ccc(Br)cc2)CC(C)C)CC2OCCCC12 c1(C(=O)NCCCCC2(NC(c3n(CC#C)ccc3)=O)CC2)cnc(NC)cn1 C1(NC(c2cc(C)oc2)=O)C(C)CCN(C(C2CCCSS2)=O)C1C CC1(C(=O)NCC2CCCCN(C(C3C4CCN3CC4)=O)C2)CCC2CC2C1 C1CC2=CCN(CC2)C(=O)CN1.Cc1ccoc1CC(=O)NCc1ccoc1C c1(NC(C(CC)C(C)(F)F)=O)ccc2c(c1)CCCC2NC(=O)OC(C)(C)C N1(C(CC=C(C)C)=O)CCCN(C(=O)C(=O)C(c2ccccc2)=O)C(C(C)C)C1 C(CC)(CC)(CCNC(=O)Cc1cc(OC)ccc1F)NC(C(C)OCC=C)=O c1(C(=O)NC2(C)CC(NC(C3(COC)CC3)=O)C2)[nH]c(Cl)c(Cl)c1Br N1(C(=O)NCc2c(Br)cc(C)c(F)c2)CC2CC1CS(=O)(=O)C2 CCC(C(=O)OC)C(=O)N(C)CC1CCCN1C(=O)CNc1c(C)occc1=O c1(OC(C2CCCN2)=O)cccc(OCc2cncnc2C)c1.C12CCC1N2C C(C(CC(C)C)C(=O)NC1(C(=O)O)CC(OC)C1)NC(C(C=C)C)=O Cc1ccn(C(C)C(=O)NCc2ccc(C(=O)NCC(=O)N(C(C)C)C(C)C)o2)n1 C=CCC(CC(F)F)C(=O)NC1C=CCN(C(C2OCCOC2C)=O)C1 CC(CNC(=O)C=Cc1ccoc1)CC(=O)NCC(C)(C)F C(=O)(C(CN=[N+]=[N-])NC(=O)Cn1cncn1)N(CC(N1CCCC1)C)C C(=O)(CC(F)(F)C(F)F)N1C(C(C)C)CN(C(c2cn(CCCF)cn2)=O)CC1 S(=O)(=O)(c1cccc(=NCCS(=O)(=O)C(F)F)[nH]1)NCCS(C)=O C#CC1CN(c2nc(N3CC(CO)C(C)(C)C3)cc(C)n2)CCN1C C(=O)(C1OCCn2ccnc21)NCC1(NC(CNC(CNC(C)=O)=O)=O)CCC1 c1(C(N2CC(O)CC2CNC(C2CC2C2CC2)=O)=O)ccc(OC2CC2)cn1 CC1(C)CC(CC(=O)O)N(C(=O)CC2CCCCC2NC(=O)CC2CSC2)C1 c1(OCC(=O)NC2CC(CNC(C3(C)CC3(Cl)Cl)=O)C2)cc(Cl)cc(Cl)c1 c1(NC(C(=O)NC(COC)Cc2ccc(C)cc2)=O)cc(F)ccc1C N1(C(c2c(N(C)C)c(Br)ccc2)=O)CCC2(CC1)CC(c1ccc(Cl)cc1F)C2 c1(C(=O)NCC(CC=C)NC(=O)C=CCO)c(C)cc(C)cc1N C1(CC=C)(NC(=O)CN(CC)CC)CCN(C(c2cccc(C(C)(C)C)c2)=O)CC1 Cc1cnc(NC(C2CC(CNC(c3ccccc3C3CC3(F)F)=O)C2)=O)cn1 N1(C(c2c(Cl)ccc(C#N)c2)=O)CCC2CN(C(=O)CSC(F)(F)F)CC2C1 c1(C(C2CCOC2)NC(n2cc(C(C)(C)O)nn2)C)ccc(F)cc1 Cc1ccc(O)nc1CNC(=O)CCCC(C)NC(=O)Cc1cnsc1 C(=O)(C(CC(F)F)NC(=O)Cc1nocc1C)NCC1(COC)CCCO1 C(=O)(CC(C)(C)CC(F)F)NCC1CCN(C(c2c(CC)ncnc2)=O)CC1O Cc1nn(C)c(Cl)c1C=CC(=O)NCC1(C(N)=O)CN(C(=O)CC2COCCO2)C1 N12CCCC(C)(C1)N(C(C=CC)=O)C(C)C2=O.C(CCO)(C1CCCC1)CCCO C(CCCCCNC(c1cnc(-n2c(C)ccc2C)s1)=O)NC(C(CC)C)=O c1(CC(=O)NC2C(C)N(C(c3cnn[nH]3)=O)CC2)ccc(Br)c(F)c1 c12cc(on1)CCCNC2=O.C(=O)(C(F)C1CCOC1)N(C1CCCC1)CCO c1(C(=O)NC(CC(=O)NC2CCC=CCC2)C(F)(F)F)ccc2occc2c1 N1(C(CN(C)C2CC2)=O)CCC(CCOC)(CO)C1.c1(C(=O)NCC)cnc(S)nc1 C1(NC(Cc2c(CC)n[nH]c2CC)=O)CCN(C(=O)COCCCF)C12CCC2 N1(C(CC2CCN(C(C)C)CC2)=O)CCCC2CN(C(=O)CCC=CBr)CC12 C(C(C)CN=c1[nH]c(C(C)(C)C)nc(=NCCC(F)F)[nH]1)OC C(=O)(CC(F)(F)CC(=O)NC1CN(C(C2CCCOCC2)=O)CC1C)OC CC1=C(C(=O)NCC2(C(N)=O)CN(C(c3cc(O)ccc3O)=O)C2)SCCO1 N1(C(CS(CC)=O)=O)C2CCCC1CC(C(=O)OC)C2.c12cccc(c1)NC(=O)C2 C(=O)(CC(C)C(C)C(C)C)NC(C1(O)CN(c2cc(NC(=O)OC)ncn2)C1)C C1(C(=O)NC(CN(C(c2cccc(C(C)C)c2)=O)C)C)CCOC2(CCCC2)C1 CCCC(C)CC(=O)NC1(CC(=O)Nc2cc(CO)cc(F)c2)CC1 N1(C(C(CCCOC)C)=O)CCCCCC(Nc2ncc3ccnc-3[nH]2)C1 c1(OC)ccc2[nH]c(C)c(C(=O)NC(CNC(=O)C=CSC)C(C)(C)C)c2c1 C1(C(C)C)CCN(C(=O)CC(CNC(C2CC(=O)N(C)C2)=O)C2CCC2)CC1 c12ccc(nc1)S(=O)(=O)C(=O)NCC(OC)CNC2=O.C1(CC)(CO)CCCC1 N1(C(C2(C)CC2Br)=O)CCC2(CC(NC(=O)COc3ccccc3F)C2)C1 C1(C(=O)NC(C(C)(C)C)CNC(c2ncncc2Cl)=O)CC2(CCCO2)C1 C1(CC=C)(NC(c2cc(C)c(Br)s2)=O)CCN(C(=O)C=CC)C1 C1(CCOC(C)(C)C)CN(C(=O)OC2(COC)CCC2)CC1C C(CCC(C)C)(C(=O)N1CCCN(C)CC1C)NC(C1(SC)CC1)=O C(=O)(C(C)CC(F)(F)F)N1C(C(=O)NCCC(=O)NCC)CC(CC)CC1 N1(C(C2CC(CCC)C2)=O)CCC(O)(CNC2(C(N(C)CC)=O)CC2)C1 Cc1sc(Br)nc1C(=O)NC1CCCC1CNC(=O)C(O)CC1CC1 c1(CN(CCCC#C)c2nn[nH]n2)ccc(C(F)(F)F)o1 C(CCCC(=O)NC(C)(CNC(C1(CO)CCOCC1)=O)CO)OC(C)C Cc1ccc2c(NC(C3CN(C(=O)CNC=O)CC3C3CC3)=O)cnn2c1C N1(C(CCC(=O)OC)=O)CC2CC(NC(c3c[nH]cc(C)c3=O)=O)CC1C2 CC(C)(C)C(O)C(=O)NC1(CO)CCN(C(c2cncc(Cl)c2)=O)CC1 C1(NC(=O)CC2(O)CCCC2)C2CC(NC(=O)C(F)CC3CCC3)CC12 C(=O)(C(F)(F)F)NC1CCN(C(CSCC(=O)Nc2cc(Cl)cs2)=O)C1 C(CC(C)CC)(C(=O)NC1CN(C)CC1(C)C)NC(C(CC=C)CC)=O N1(C(c2c(C)cccn2)=O)CC(C(=O)NCCCC2CCC2)C(C)(C)C1 c1(C(N2CC(O)(C(C)NC(c3conc3C(C)(C)C)=O)C2)=O)c[nH]c(C#N)c1 c1(C(N(CC(C)NC(=O)CC2(C)CCOCC2)CC)=O)cnn2c1N(C)CC2 CC12CCC1CN(CC1CCC1c1nnnn1CC(F)F)C2.c1ccccc1 N=c1[nH]c(Cl)c(Cl)cc1C(N1CCCC(C(=O)NOC2CC3CCC2C3)CC1)=O c1(OCC)cc(NCC23CC(NC(c4cnc(S)n4C)=O)(C2)C(C)O3)nc(C)n1 CON=C(C(=O)NCC(C(C)C)NC(=O)CCCN(C)N=O)c1ccco1 N1(C(C=CSC)=O)CC2CC(NC(=O)Cc3ccc(F)cc3)C1C2 c1(C(=O)NCC(CNC(CC(=C)C)=O)C)cccc(Cl)c1C N1(C(CCC)=O)CCCC2(CCN(C(=O)CC3(O)CCCOC3)CC2)C1 N(C(=NC1COCC1(C)C)NCC(=O)NOC)C(CC)C.OC c1(N(C)C)cccc(C(=O)NCC(CO)NC(C2CCCCC2)=O)n1 CCCCCCCCc1cccc(CN(C2CN(C(=O)Cc3cn(C)cn3)C2)C)c1 CC1=NS(=O)(=O)N(C)C=C1C(=O)NCCC1(CNC(=O)C(CC(C)C)N(C)C)CC1 N1(C(C(C)C(C)(C)C)=O)CC(NC(c2cnn(C)n2)=O)CC12CCC2 CC1(C)CN(C(C23CCCC2C3(F)F)=O)CC(C)(C)C1NC(=O)Cc1cccs1 c1(Cn2cc(C(C)(C)OC)nn2)ccc(-c2ccc(Br)cc2)cc1 N1(C(C(c2ccccn2)C)=O)CC=CC(C(=O)NCCc2cc[nH]n2)C1 c1(C(N2CCC(NC(=O)Cc3cc[nH]n3)C(F)C2)=O)ccc2n[nH]cc2c1F c1(C(N2CC(C(N(C(CO)C3CC3)C)=O)C(C(F)(F)F)C2)=O)ncc(Cl)cc1F C12(NC(c3c(C)scc3)=O)CCCC1N(C(C1CCCCN(C)C1=O)=O)CCC2 CCC(C)CC(=O)C(=O)N1CCC2(CC2)CC1C(=O)NCCC1CC2C=CC1C2 N1(C(c2c(NC(C(OCC)OCC)=O)ocn2)=O)CCNC(=O)CC1 C(C)(C(=O)N1CC(CNC(C)=O)C1)N(C(C)=O)CC.C1(=O)CC2(CC2)N1 c1(C(C)C)c(C(=O)NC2CC(CNC(C3CC3(C)CF)=O)C2)cnn1C(C)(C)C C1(O)(C(C)NC(C2C(CC)C2)=O)CCN(C(C2CCCOC2)=O)CC1 C1(C(C)NC(c2cn(CC)nc2)=O)CCCCN1C(=O)C(C)(Cl)Cl N1(C(C2CCN(C)C2)=O)CCC(CCNC(=O)Cc2cc(C3CC3)nn2C)CC1 C(=O)(C(O)CCC(F)(F)F)N1CC(NC(C2C(C)OC(=O)N2)=O)C2(C1)CC2 N1(C(c2cccc(OCC)c2)C(=O)NCC2CCC2)CCOCC(CO)C1 C1(F)(C(=O)OC)COCCN(C(=O)CCCC(F)(F)F)C1 CC1(C)OCCOC1CC(=O)NCCCNC(C1CCOC1)=O c1(NC(C(C2CCCCC2)C)=O)ccnc(N2CCOC2=O)c1 CCC(CNC(=O)CCc1cscn1)(CC)C(=O)NCCCCCCCO C1(C(=O)OC)CN(C(c2nc(CO)cs2)C(=O)OC)CC1C1CCOCC1 C(=O)(C#CC1CCC(=O)CC1)NCC(C(C)C)NC(c1ncsc1Br)=O c1(C(N2CC(C(C(=O)NC3(CCO)CCC3)OC)C2)=O)ccc(COC)c(F)c1 c1(C(=O)NC2CC(C)(COC)N(C(=O)C=CCO)C2)cc(C)c(C)nc1C C(=O)(C(C)NC(N)=O)NC(C1CN(C(=O)CCN2CCC2)C1)C S(=O)(=O)(c1cc(Cl)ccc1Cl)N1CC2CCN(C(=O)Cc3nc(Cl)cs3)C2C1 N1(C(Cc2c(C)cco2)=O)CCCC(CO)(NC(=O)CC2CC(CF)C2)C1 C1(NC(Cc2c(CC)cccc2)=O)CCc2nc(NC(=O)C(O)C(C)C)sc2C1 C(=O)(C(C)(C)CC#N)NCC1CC(NC(c2c(COC)scc2)=O)C(O)C1 c1(C(N(CCNC(C(C(=O)OC)OC)=O)CC2CC2)=O)[nH]nc([N+](=O)[O-])c1Cl C1(NC(C2CC(C)CC(C)C2)=O)CCCN(C(C2CC(O)C2)=O)CCC1 CCC(CC(F)F)C(=O)NCC1CC2CCC(C1)N2C(=O)C(C)(C)S(C)(=O)=O C(CC(=O)NC1CC1NC(c1cc(Br)cnc1C1CC1)=O)(C(C)C)OCC C(=O)(C1CCCn2cnnc21)N1CCCN(C(C(C#C)(C)C)=O)CC1CO C(CCCC(CO)NC(C1(C(F)F)CCCO1)=O)NC(C(c1n(C)ncc1)=O)=O c1(OC)cccc2c(C(N3CCC3CN(C(=O)C(F)(F)F)C3CC3)=O)c(C)[nH]c12 n1(CC)nc(C(=O)N(C(CNC(=O)CCF)C2CC2)C)c(=O)c2ccccc12 C=C(C)CC(C)C(=O)NCCOC1CN(C(=O)C(c2ccc(C)s2)C)C1 c1(C(N2CC(CC(C)NC(CCCCCC#C)=O)C2)=O)cc2cc(C)ccc2[nH]1 c1(CC)ccc(C(N2CC(NC(=O)CC3(CO)CCCC3)C3(CC3)C2)=O)c(Cl)c1 c1(C(N(CCNC(=O)Cc2cccnc2)CC2CC2)=O)ccc(F)cn1 CCC(CCC(=O)NC(C)CCCNC(=O)CC(C)(C)COC(C)=O)OC c1(CC(=O)N(C)CCNC(=O)C(c2ccccc2)N(C)C2CC2)cccc(Br)c1F N1(C(CN(CC(C)Nc2ccccc2)C)CBr)CCOCC1 CC1CCCC(Oc2ccc(C(=O)NC(C)(C)CNC(=O)C(C)(C)CF)cc2)C1 N1(C(C=C(CCC)C)=O)CCC(NC(c2cccc(NC)n2)=O)CC1 c1(C(=O)NC2CCC(CCNC(C(N)=O)=O)C2)cccc(CCO)c1 N1(C(c2c(C)[nH]cc2)=O)CCC(C(=O)NCC2CCC(CO)CC2)C12CC2 c1(C(=O)NC2CC(C)(NC(=O)CCCF)C2)cccc2c1OCC2 C1(NC(C(F)=CCC)=O)CCC2CN(c3cc(C(=O)OC)cc(Cl)n3)CC2C1 Cc1nc(CC2CC2)oc1C(=O)NC1CN(C(C2CC2C(N)=O)=O)CC1O CN=c1[nH]c(=NCC2C=CCC2)[nH]c(=NCCc2cncc(Cl)c2)[nH]1 n1(CCC2CC(NC=O)C2)cc(CC23CC(C2)C3)nn1.C12(C(=O)CCC3CC3)CSCC1C2 C(CCCO)(C(F)(F)F)NC(CCC(C)OC(=O)Nc1ccccc1)=O CC#CCC(C(=O)NOC(C)CCC(=O)OC)NC(=O)C(CC)CCCCC C(=O)(C(C)S(N)(=O)=O)NCCC(C)NC(c1ccnn1-c1ccccc1)=O c1(CC)nc(C)ncc1C(N1CCOC(C(C)NC(=O)CC(C)(C)SC)C1)=O C1(C(N2C(CNC(c3nc(-c4cn(C)nc4)sc3)=O)CCC2)=O)CCCC1(C)C C(CCC(O)C(=O)N(CC(N)=O)C)NC(c1c(CC)cns1)=O C=CC(CCC)CC(=O)NC1CC2(C1)CC(C(=O)NCC(C)OC(F)F)C2 N#Cc1cc(C2(C(N3CCC4(C3)CN(C(=O)OC(C)(C)C)C4)=O)CC2)cc(Br)c1 Cc1cc(F)ccc1CNC(C1C(O)CCN(C(C(C(N)=O)C(N)=O)=O)C1)=O N1(C(C(C(C)C)NC(N)=O)=O)CCC(NC(=O)Cc2ccsc2)C2(CCC2)C1 C1(CNC(C(c2ccn(C)n2)C)=O)CCN(C(C2(F)CCC2)=O)C1 c1(OC)cc(NC(C2OCCC2CNC(C2CC(=O)NC(=O)C2)=O)=O)ccc1F N1(C(c2cc(C#N)sc2)=O)C2CCC1CC(NC(C1CC(=C3CC3)C1)=O)C2 c1(C(C)C(N2CC(O)(CNC(C3CC3c3ccco3)=O)C2)=O)cc(F)cc(F)c1 C1(C(N2CCC(C)(CCNC(c3cccc(Cl)n3)=O)C2)=O)(OCC)CCOCC1 CC(C)C(N=[N+]=[N-])C(=O)N1CCC(CC(N2CCC(C(F)(F)F)C2C)=O)C1 N1(CC2C(C)(C)OCCO2)CCOc2c(Br)cccc21 c1(CC)n[nH]c(CC)c1CC(=O)NCC1CC1NC(=O)CC(C)N(C)C c1(CC(N2CCC(OCCNC(C3CC3F)=O)C2)=O)ccn(Cc2ccccn2)n1 CCC(F)(F)C(=O)NCC1CC1NC(=O)CC1C(=O)ON=C1C C1(NC(c2cc(N)c(Cl)cn2)=O)CC(NC(c2cncnc2)=O)C12CCOCC2 c1(NC(C(C)C)=O)ccc(F)cc1NC1(c2nnnn2CC2CC2)CCC(C)C1 N1(C(C2(F)C(C)C2)=O)CCC(NC(=O)COCc2ccccn2)C1 C1(C(=O)OC)CC(C)(NC(=O)CC2(NC(C34COCC3C4)=O)CC2)C1 N1(C(CCNC(C2(COC(C)C)CCC2)=O)=O)CCC(CN(C)CC)C1 CC(CC(=O)N1CC(OCC(=O)NCCN(CC(F)F)C)C1)N(C)C C(=O)(C1=NN(C)C(=O)CC1)NCC1CN(C(c2cc(C)nc(O)c2)=O)CC1O N1(C(C2(CC#C)CCOC2)=O)CC=CC(NC(=O)Cc2coc(C)n2)C1 CC1(C)COC1C(=O)NCC(CNC(c1c[nH]nc1C(F)(F)F)=O)CO c1(C(=O)NCC(C)(C2CCC2)NC(C(F)=CCC)=O)nsnc1O C(=O)(C(O)CN1CCCC1)NC(C)(O)CNC(=O)CC1CSC1 C(=O)(C(C)(C)CC)N(CC(CC)NC(COCCC#C)=O)C.C1CC1 C1(NC(C(C)Oc2c(C)ccc(Cl)c2)=O)CC2CN(C(=O)C(N)=O)CC2C1 Cc1nonc1C(=O)N(CCCNC(=O)C(O)Cc1ccccc1)C1CC1 C12(CNC(CCOCC#C)=O)CN(C(C3(CO)CCCCC3)=O)CC(F)(C1)C2 n1(CCCOC)ccc(=NC(=O)C2CCC(NC(=O)CC(O)C3CCCC3)C2)[nH]1 C(=O)(C(C)(C)C(C)(F)F)NC(C(C)C)CCNC(=O)Cc1ccoc1 c1(-c2c(C)ccc(C#N)c2)ccc2c(c1)C1(CCN(c3ccnc(Br)n3)C1)C(=O)N2 c12cncc(c1)CNC2=O.CCC(F)C(=O)N1CC(CC(C)S(C)(=O)=O)C1 C1(C(N2CCC(CCNC(c3cnc4n3CCC4)=O)C2)=O)CCn2nncc2C1 c1(CC(=O)NCCNC(c2cc(OC)ns2)=O)cccc(S(C)(=O)=O)c1 N1(CC2N(C(C(CC)c3ccccc3)=O)CCC2)CCC(c2ccccn2)CC1 c1(C(=O)NCC2(C)N(C(c3cc(C)on3)=O)CCC2)ccc(Cl)cc1C(F)F N1(C(c2ccc(CSC)cc2F)C(=O)NC(C)C)Cc2ccccc2CCC1C Cc1cccc(C)c1NC(=O)C(N1CCOC(C)(CCO)C1)c1ncsc1C c1(C(N2CC3C(NC(c4ncccn4)=O)C(C3)C2)=O)ccc2cc(Cl)ccc2c1 C1(C(N(CCCCC)C)=O)(NCC2CCC2)CCNCC1 N1(C(C2CC3C=CC2C3)=O)CCC2(CC1)CCN(C(C1CC3(CCO1)CC3)=O)C2 C1(C2CN(C(c3ccc(Br)c(C(C)C)c3)=O)C2)(NC(CC2CC(C)C2)=O)CC1 CCCC(CCC)CC(=O)N1CC(O)CC1CNC(=O)CC1(CO)CCOCC1 c1(CN2CC(C)(CC(N3CCCC3C#N)=O)C2)cc(Br)ccc1O C1(C(C)C)CN(C(c2cn(CCCF)nn2)=O)CCN1C(=O)COC1CC1 C1(NC(C(CC)(C)CCC(C)C)=O)CCC2(CCCN(C(=O)CC(=O)OC)C2)C1 C1(C(N2CCN(C(CC=CC=C)=O)CC23CC3)=O)CCc2ccccc2C1 c1(NC(=O)NC(C(C)C)C2CCC2)nc2cc(C#N)ccc2o1 Cc1ccc(NC(=O)COCCOC)c(OC)c1.C1(CN)CCOC1 C=C1CCN(C(c2ccccc2F)=O)C(C(=O)NC2COC3COCC23)C1 Cc1c(Cl)ccnc1C(=O)NCC(F)CNC(=O)C(c1cccc(F)c1)C C1(C(=O)NCc2c(C)nn[nH]2)CN(C(C2(O)CCCC2)=O)CCN1C C(CC1CN(C(=O)OC(C)(C)C)C1)(C(=O)NCc1cnc[nH]1)SC.C1CC(=O)N1 C1(CN(CCCC(C)C)C(C2(CSC)CCC2)=O)CCCSC1.C12(CCC1)C(=O)N2 c1(OCC)ccc(C)cc1CNC1COCCN1C(=O)Cc1cccnc1Br c1(CCn2c(C(N3C(NCCCSC)CC3)CC)nnn2)c(F)cccc1Cl C1(C(N2CC(CC=C)(C(=O)N(C)Cc3cc(C)on3)C2)=O)CC(C2CC2)=NO1 N1(S(Cc2ccc(C)cc2)(=O)=O)CCC(O)(C(N)=O)CC1.C12(C)CN(C1)C2=O n1(CC)cc(Cl)cc1C(=O)NC(C1CCN(C(c2n[nH]c(C)c2Br)=O)CC1)C c1(C(N(CC(CN(C(C=C(C)C(C)(C)C)=O)C)O)C)=O)c[nH]c(C#N)c1 CCC(C(=O)NCC(C)CN(C)C(c1ccc(C(F)(F)F)o1)=O)C(C)(C)CC c1(C(=O)NCC2N(C(CSCC)=O)CCC2C2CC2)cc2c(nc1O)CCSC2 c1(CCC)cc(C(=O)NC2(C)CCN(C(c3ccc(CN(C)C)o3)=O)C2)n(C)n1 CCCCC(O)CC(=O)NCC1(CCNC(=O)C(CC)c2ccccc2)CC1 C=CC1(C2(C(=O)NCC3CC3CNC(=O)CCCC(CC)CC)CCC2)CCC1 c1(C(=O)NCC2N(C(C=C(CCC)C)=O)CC(OC)C2)ccc2c(c1)CCCCN2 Cn1ncc2c1CN(C(=O)C(CC1CC1)NC(C1C=CCCC1)=O)C2 C1(NC(c2cc(CC)on2)=O)C(C)CCN(C(=O)CCc2ccc(F)cc2)C1C N1(C(c2ccc(C=C)cc2)=O)CC(NC(=O)CC2COC3CC2C3)CC12CCC2 c1(C(N(CCCCCCNC(=O)Cc2cnc[nH]2)C)=O)occ2c1CCOC2 C(=O)(C(C(C)(C)C)NS(C)(=O)=O)NCC1N(C(CC(C)(C)C)=O)CC(F)C1 C1(C(C(N2CCC(CC=C)(NC(=O)C(C)=C(C)C)C2)=O)C)CCC(C)(C)CC1 N1(C(C2CC2Br)=O)CCOC(CNC(=O)C(F)(F)CC(C)(C)C)C1 C1(NC(c2c(C)sc(O)n2)=O)CCN(c2snc(Cl)c2C#N)CC1C Cc1ccc(C(N2CCC(F)C(NC(c3ncc(F)cc3C)=O)C2)=O)c(F)c1 C12(CCCC1)C(=O)N2.C1(CCC(=O)NCC2(OC)CCC2)CC(F)(F)C1 C12(NC(CC(C)(C)F)=O)COCCC1CN(C(C1CCOCC1)=O)C2 C1(C2(O)CN(C(c3cc(Cl)cn3CC)=O)C2)(CNC(C(C)SCC)=O)CC1 C1(NC(C=CC(=O)N(C)C)=O)CN(C(=O)C(c2ccccc2)O)CCC1O C1(C)(c2cn(CC)nn2)CCCC(SC(C)(C)CC)C1 c1(C(N2C(C3CC3)C2)=O)ccc(C)c(O)c1.C1(C(=O)OC)CC(C)(C(N)=O)C1 c1(OC)ccc([N+](=O)[O-])c(C(N2CCN(C(=O)CCCC#N)C3CC23)=O)c1 c1(C(=O)OCC)c(C(C)(C)C)csc1NC(=O)CC1(C)CC(C)=NO1 N1(CC(C2CCC(=O)C2)CC)CCC2(CCS2)CC1 C(=O)(CC(CNC(c1cc(C2OCCO2)co1)=O)Cc1ccc(Cl)cc1)OC c1(CN(C(c2cnc(C(C)(F)F)s2)=O)CC)nc(Cl)ccc1Br N1(C(=O)Nc2sc(CC)c(C)n2)CCc2c(ccnc2Cl)C1 Cc1noc2ncc(C(=O)NCC(CO)NC(=O)CC3(O)CCCOC3)cc12 C(=O)(C(F)CCC(C)(C)C)NCC(=C)CCNC(c1cccnc1OC)=O N1(C(CC(C)(C)SC)=O)CCC(C2CCOCC2)(CNC(=O)C(C)CC2CC2)C1 C1(NC(COCCCCC)=O)CC(O)CN(C(C2(CC3CC3)CCCCC2)=O)C1 C(=O)(C(=O)C(C)(C)C)N1CCC(N(C(=O)CC2CCNC(=O)C2)C)C1 CC(CC(N)=O)C(=O)N1CCCCCC1.C(CCCC(=O)O)n1ccnn1 Cc1ccc(C(=O)NCC(=O)N(C2CC2)Cc2cccnc2F)cc1[N+](=O)[O-] c1(OC)ccc(C(N2CCCC(C(N(c3cncnc3Br)C3CC3)=O)C2)=O)cc1I C1(NC(C2CCCCC(C)(C)C2)=O)CN(c2nc(C#N)ncc2Cl)C2CCCCC12 CC(C)(O)C(C)(C)C(=O)NCC(C1CCCC1)NC(=O)CC1CCCNC(=O)C1 c1(OC)ccc(C2=NOC(C(C)NC(=O)NCCc3cc(C)ns3)C2)cc1F N1(C(C(CC)N(C)C)=O)CC2(CC(NC(=O)CC3CCOCC3)CO2)C1 C1(C(=O)NC(C=C)C)C(C)OCCN1C(=O)C(CSCC)OC Cc1cncc(CCN(C(=O)C=CC(C)(C)NC(=O)C(C)c2cc[nH]n2)CC)n1 C1(CN(C(=O)CN2C(=O)CCC2=O)C)CCCC(NC(=O)CC2(CO)CC2)C1 c1(C(=O)NCC(CNC(c2nc(CC)oc2)=O)CO)ccnc(-n2cccn2)c1 C1(CCOCC)(C(=O)NCC(C2CC2)C2CC2)CCN(CC2CC(=O)N2)CC1 c1(C(=O)Nc2nc(C)c(Cl)s2)cc2c(-c3ccc([N+](=O)[O-])cc3Br)cncc2s1 N1(C(C2OCC(C)C2)=O)CCCC2(NC(=O)C=Cc3cccc(F)c3)CCCC12 N#CC1CC(N(C(=O)C(O)C2CCC2)CC(=O)NCC2CC2)C1 C1(CCC(=O)N(C2CCCC2)CCNC(C(C)C2CCCC2)=O)CCN(C)CC1 Cc1ccc(C(N2CCC(C)(NC(c3sc(=N)[nH]c3C)=O)CC2)=O)nc1O Cc1ccc(C=CC(=O)N(C)CC2CCCN2C(c2cc(C(C)C)cs2)=O)s1 c12cc(c(F)cc1[N+](=O)[O-])N(C)CC1CCN2C1.C1(COC)CCCC1OC.CO CC(CN(C)C)CCC(=O)NCCC(C)NC(C1(C(F)(F)F)CC(F)(F)C1)=O Cc1oc([N+](=O)[O-])cc1C(N1CCCC(CNC(c2coc(C#N)c2)=O)C1)=O CC1(C)CN(C(=O)C(C)(F)c2ccon2)CC1NC(C1CCCS1(=O)=O)=O Cc1cc(C(=O)NCC2CCC(NC(C3CC(C)C3)=O)C2)c2nc(C)n(C)c2n1 N1(C(=O)C2=NOC3(CCC3)C2)CC2C3CCC(C2C1)N(C(c1sccc1F)=O)C3 S(=O)(=O)(c1ccc2[nH]c(=NC(CO)CCF)ccc2c1)NCC1CCCN(C)C1 C1(C2CCCN(C(C3CC4C(C3)C4(F)F)=O)C2)(NC(C(CCSC)OC)=O)CC1 C(=O)(C(C)CC(C)CC)N(CCC)CCNC(=O)CC1(COC(F)F)CC1 N1(C(C2(C(C)O)CC2)=O)CCCC(OCC(N2CC(O)C2)=O)C1 N1(C(C(CN(C(=O)COCC2CCC2)C)O)=O)CC(CO)CC12CCC2 c1(C(=O)NCC(=O)N(C2CCC(C(=O)NCC(C)(C)C)CC2)C)cnc(S)nc1 c1(CC(=O)NC2CC(CNC(CCN(C)CC)=O)C2(C)C)c(C)nn(C)c1Cl N1(C(c2c(C3CC3)csc2)=O)CCCCC1CC(=O)N(C1CCC1)CC Cc1oncc1C(=O)NCC(N1CC(F)(CNC(c2nncs2)=O)C1)=O Cc1ccc2snc(C(=O)N(CC(O)CNC(C3(C(C)(F)F)CC3)=O)C)c2c1 c1(C2(C(=O)NC(C3(C)CCC(NC(c4cnsn4)=O)C3)=O)CC2)cc(F)ccc1F c1(C(=O)NCC(C2(O)CN(C(c3ncccc3F)=O)C2)(C)C)cc(F)ccc1F C1(OC)CCC2(C(=O)NC3CC(NC(=O)Cn4c(C)csc4=O)CC3O)CC12 Clc1cc2c(N3CCC(n4cc(-c5ccccn5)nn4)CC3)ccnc2s1 C(=O)(CCC(O)C(C)(C)C)N1CC(C2(C(O)C(F)(F)F)CC2)C(C)(C)CC1.CCO N1(C(CCc2nc(C)sc2)=O)CCC2(NC(=O)COCCCF)CC2C1 C1(NC(c2c(C#N)cncn2)=O)CN(C(C2Cc3nccnc3C2)=O)C2(CCC2)C1 c1(C(C)NC(c2cnn3ccncc23)=O)ccc2c(c1)CC(C)O2 c1(C(C(=O)NCCC)N(C(c2ccccc2Br)C)CC)cc(NC(C)=O)ccn1 c1(CC(N2CCCN(C(C(C)OC)=O)C(C)C2)=O)ccc([N+](=O)[O-])cc1F C1(NC(C2(SC)CCC2)=O)CCN(C(=O)C=C(C)c2cccs2)C2CC12 N1(C(CC2CCN(C(C(C3CC3)OC)=O)C2)=O)CC2CCCCC2C1C c1(C(C(=O)NC2COC2)N(CC(C(C)C)OC)C)ccc(-c2ccco2)cc1 N1(Cc2cn(C(C)C(=O)NC(C)Cn3cccn3)nn2)CCCCC1 CC(O)(C(=O)NC1CCC(CC(=O)NCC(O)C(N)=O)C1)C(F)(F)F c1(NCC)cc(N(C(C2CCCC2)Cc2ccc(C(C)C)o2)Cn2cc(Br)cn2)ncn1 C12(NC(c3ccccc3Cl)c3n(CCCC)nnn3)CCC(CSC)(CC1)CC2 c1(CC)nc(C)[nH]c1C(N1CCC1CNC(=O)CC1(O)CCOC1)=O C1(CNC(C(c2cn(C)nc2)O)=O)CCN(C(c2ncc(F)cn2)=O)C12CC2 C1(NC(=O)CCc2ccccc2F)C2CC1CN(C(C1CCCN1C1CC1)=O)C2 CC1CC(NC(C2(CF)CCOCC2)=O)CN1C(C1(c2ccno2)CCC1)=O Cc1nc(C(=O)NCC2C=CC(NC(=O)C(C)CC(C)(F)F)C2)c2ccccn12 c1(N2CCC(NC(c3n(CCOC)ncc3)=O)C2)ncnc2scc(Br)c12 C(CC(C(C)C)NC(c1ccnn1C)=O)N(C(C(C)NC(C)=O)=O)C N1(C(C2(C(C)C)CNC(=O)C2)=O)C2CCCC1CN(C(C1CCS1(=O)=O)=O)C2 C1(NC(=O)COCC2CC2)COCC1CN(C(=O)CC1CCCC1)C1CC1 C1(C(N(C(C)C)CCNC(=O)CN2C(=O)CN(C)C2=O)=O)CC2OC(=O)OC2C1 c1(C(N2CC3C(CNC(C=C(c4cn(C)nc4)F)=O)C3C2)=O)ccc(N)cc1O C12CCCN(C1)C2=O.C(C(C)(O)CNC(=O)CC1(C)OCCO1)NC(C=C(C)Cl)=O [N-]=[N+]=NCCCCC(=O)NCCC1CC(NC(=O)CCCCN2CCCCC2)C1 CCCC(F)(F)C(=O)NCC1OCCC1C(=O)Nc1csc(C)c1 C(=O)(C(CC(C)C)C(C)C)NC1N(C(C2CCC(OC)C2)=O)CC(F)(F)C1 Cc1cc(C#N)cc(Cl)c1C(=O)NC(C(=O)O)C1CCC1 CC1CN(C(c2cnc(-c3ccoc3)s2)=O)CCN1C(=O)CC(O)C1CCCC1 c1(C(=O)NC2(CNC(C(CC#C)C3CC3)=O)CC2)cc(F)c(CO)c(F)c1 C(C(C)C(C)NC(=O)N(C1CC1)Cc1ncoc1C(F)(F)F)OC c1(C(N2CCC(NC(COCC(=O)NC)=O)C(O)C2)=O)ccn2cnnc2c1 N1(C(c2c(N)ccc(CC)c2)=O)CC(C)CN(C(c2nc(C)n(C)n2)=O)CC1C c1(NC2(c3nnnn3C3CCCCCC3)CCCC(C)C2)ccc2c(n1)CCCC2 N1(c2cc(SC)ncn2)CCC2(CC1)CCN(C(c1cc(C)nc(C)n1)=O)CC2 C(c1ccc(C)c(Cl)c1)=C.N1(C(c2c(C)c[nH]c2)=O)CCC2C(NC(=O)CC(C)(C)C)C12 O(NC(=O)C(c1cccnc1)NC(c1ccc(CSC)[nH]1)=O)C(C=C)C c1(OC)cccc(OC)c1.N1(C(C(=O)Nc2nc(CN)cs2)=O)CCC(=C)CC1 CCCC(O)CC(=O)N1CC(NC(c2cccc(NC(N)=O)c2)=O)C2(CC2)C1 C=C=CCCC(=O)NC(C)(CNC(=O)CSCc1ccc(F)cc1)Cn1cccn1 N12CCC(CC1)OC(CC)C(=O)N(C(C)CSC)C(=O)C2.C(CF)OC.CC Cc1noc(C)c1C(N1CC(O)(C(C)NC(=O)CCCCF)C1)=O Cc1n[nH]c(C)c1SCC(=O)NCC1C=CCN1C(c1cnc(C(C)C)nc1)=O N1(C(c2c(OC)csc2)=O)CC2(CCCN(C(C3CCCC(C4CC4)O3)=O)C2)C1 N1(C(C2(OC(C)=O)CC2)=O)CC(NC(=O)Cc2csc(C3CC3)n2)CC(C)C1 N1(C(c2cc(C)no2)=O)CC2(CC(CNC(=O)Cc3cc(Br)cs3)C2)C1 c1(CCC(=O)CC2CCC2)cccc(CNC(c2ccsc2)=O)c1.N1CCC1C(=O)OC N1(C(C2(C)C(C)OCC2)=O)CCC2(CC1)CC2C(=O)NCc1nn[nH]n1 Cc1cc(F)ccc1C(F)(F)C(=O)NCC(C)N(C)C(c1ccnn(C)c1=O)=O N1(C(CCC(CC)NC(=O)C(O)CC2CC2)=O)CCC(C)(C)C(CO)C1 Cc1ccc2[nH]nc(C(=O)NCC3CCN3C(=O)C(C3CC(F)(F)C3)O)c2c1 C1(c2nc(Cc3cn(C)nc3)nn2-c2cnccn2)Cc2ccccc2N1C C1(NC(C2CCN(C(CC)=O)C2)=O)CCCC2CN(C(=O)C(C)(F)F)CC12 c1(CNC(=NC)NCCC2CCCCC2N)cccc(Cl)c1Cl C(=O)(C1=C(Cl)CCOC1)N1CC(C(=O)NCC2(C)CC(F)(F)C2)C(F)C1 N1(CC#C)CCC2CCCC(C1)N2CC(O)Cc1cccc(Br)c1 C(CS(=O)(=O)CC(=O)N1CC2CCC2(CC(=O)NC(c2cnsc2)C)C1)OC C1(C(=O)NCCC(C)CCNC(c2scnc2C(C)(C)C)=O)OC2CCC1CC2 N1(C(c2cc(COC)[nH]n2)=O)CC(C2CCN(C(C3CCNCC3)=O)C2)C1 C1(NC(c2n(C)ccc2)=O)CN(C(=O)CC=C(Cl)Cl)CC12CCC2 CC1=C(C(=O)NC2CC(C)N(C(=O)CCCN3CCOCC3)C2)CC1 N1(C(CC(C)(C)C)=O)CCC2C(NC(=O)CC3C=CCC3)CC12 C1(NC(c2cc(C)nc(O)c2)=O)CN(C(c2c(C)ccn2C)=O)CC(C)(C)C1 Cc1ccn(CC(=O)NC(C)CCCNC(=O)C(C2(O)CCCC2)F)c1 Cc1c(C(N2CCN(C)CC2CNC(=O)CC2CC2C2CC2)=O)cccc1Br C(=O)(C(C)CC(C)C)NCc1cn(C2N(C(C(CC)(C)O)=O)CC2)nn1 N1(C(CC2CCC(C)(C)O2)=O)CC2(CCCC2)C1C(N1CC2CC2C1)=O C(=O)(C1Cc2ccc(F)cc21)NC(CN(C(C(CC)NC(N)=O)=O)C)(C)C C1(N(C(Cn2c(C)ncc2)=O)C)CN(C(C2CC(CF)C2)=O)CC12CC2 N1(C(C=Cc2n(CC)ncc2)=O)CCN(C(=O)C(N2CCCC2)C2CC2)CC(O)C1 C1(NC(=O)CCc2nccs2)CC2CCC1N2C(c1cc(O)cs1)=O Cc1cccc(NC(=O)C(C2CN(C(=O)CNC(=O)C3CC3)C2)OC(C)C)c1 CC1CN(C)CCCN1C(C12CC(NC(=O)CCc3ccco3)(C1)C2)=O C1(NC(C2CC3CN(C(CS(CC)(=O)=O)=O)CC3C2)=O)CCC(C2CC2)CC1 C(CC(=O)N1CCOC2CC12)(C(C)C)NC(c1c(C)snc1)=O CC(C)C(F)(CNC(=O)C(F)n1ccnc1)C(=O)NC(c1cncnc1)C C#CCC(CC(=O)OC)NC(C1C=CC(NC(C2CCC(C(N)=O)C2)=O)C1)=O C1(CNC(C(C)N(C(C2C3CCCCCC23)=O)C2CC2)=O)CC2C=CC1CC2 Cc1ccc(F)c(Br)c1C(=O)NCCC1(CNC(C2CNC(=O)N2)=O)CC1 C1(C(=O)NCC(CNC(c2n(CC(C)C)ncc2)=O)(C)O)CCS(=O)(=O)N1 Cc1cc(C(=O)O)cc(C)c1OC(c1ccc(C(F)F)c(F)c1)N(C)C C1(NC(C(=O)OC)C)CSC(C(F)(F)F)C1 c1(C(=O)NCC(C2CCCCC2)NC(C(C)(C)C)=O)sc(F)cc1Br C(CCCCCNC(C1CCOC(=O)C1)=O)N(C)C(c1ccc(C(F)(F)F)[nH]1)=O N1(C(C(CC)(F)F)=O)Cc2occ(C(=O)NCC(C)(C)CO)c2C1 CS(=O)(=O)c1cnc(NC(=O)CC2COCCN2C(C2CNC(=O)C2)=O)c(Cl)c1 N#Cc1ccc(CN2CCC3CN(c4ncc5ccsc5n4)CC23)c(F)c1 C=CCC(F)(F)C(=O)N1CC(O)(C(C)NC(=O)COc2cncc(Br)c2)C1 C12(C(=O)NCC(CC)NC(=O)CCC3CC(C)(C)CO3)CCC(C#N)(CC1)CC2 c1(C(=O)NCC=CCNC(C2(C)CCCCO2)=O)nc(O)cc2ccccc12 CCCC(CCC)C(=O)NCC(O)CN(C)C(C1CCSCC1)=O N1(C(c2scc(OC)c2)=O)CC(OC)CC1CNC(=O)CCN1CCOC1=O C1(OC)(CNC(c2ccnc(Cl)c2F)=O)CCN(C(=O)C(=O)NC2CC2)CC1 c1(NC2CCC(CCC)CC2)ccc(S(=O)(=O)N2CCCCC2C)c(OCC)c1 C(N=c1ccc2cc(S(=O)(=O)c3ccccc3)ccc2[nH]1)C1C(C)CCC1 C#Cc1cc(C(=O)NCC(C)(CO)NC(=O)C(CC)C2CCOCC2)cc(F)c1 C1(CNC(C(=O)NCC(F)F)=O)CN(C(c2n[nH]c(C3CC3)n2)=O)CCC1(F)F C1(NC(C=C(CCC)C)=O)CC2CN(C(=O)C(C)n3cccc3)CC2C1 CN1CCCC2(CCN(C(c3cn(C4CC4)nn3)=O)C2)C1=O.c12ncc([nH]1)C2N(C)C N1(C(Cc2c(C)scc2)=O)CCN(CCNC(=O)CSc2nnc(S)s2)CC1 C1(NC(C(COC)NC(C)=O)=O)CN(CCNC(=O)CC(C)(C)C)CCCO1 C(=O)(N=c1ccn(CCO)[nH]1)C1CC(NC(CCCCCNC(N)=O)=O)C12CCC2 Nc1ccc(-c2cn(CC(F)(F)Cc3ccccc3SC(F)(F)F)nn2)cc1 c1(C(C)C)cccc(C(N2CC(Nc3cc(O)nc(C)n3)C(C)(C)C2)=O)c1F C1(S(C)=O)(C(=O)OC)CCN(C(=O)Nc2nnc3n2CCCC3)CC1 C12(C(N3CCC(NC(c4c[nH]nc4C(F)F)=O)C3)=O)CCC(CF)(C1)OC2 N1(C(c2c(CC)onc2C)=O)CCC(c2ccccc2)C(C(=O)O)C1 c1(C(=O)OC)cc(C(=O)N(CC(C)N(C)C(C2CCC3(CC3)C2)=O)C)ccc1Cl C#CCC(CC(=O)NC1(C(N2CC(CC)C(C(F)F)C2)=O)CC1)c1ccccc1 C(=O)(CCP(C)(C)=O)NC1CCC(NC(Cc2n(C)ncc2)=O)C1 c1(C(=O)NC2(C(N3C(CNC(C)=O)C=CC3)=O)CC2(C)C)ncn(C)c1C C(=O)(CC(C)CC(C)C)NC(C1(O)CCN(C(c2c(C)ncn2C)=O)CC1)C C(=O)(CCC(=O)C(C)(C)C)N1CCC(C)(C(N(C)Cc2cnccn2)=O)C1 C1(NC(=O)C(C2(O)CN(C(=O)COc3cn[nH]c3)C2)F)CC12CCCC2 C1(C(=O)O)CN(C(c2cc3cnccc3o2)=O)C2(CCCCC2)C1 c1(C2C(C(=O)NC(C(=O)OC(CC=C)CO)C(C)O)C2)ccc(OCC)c(C)c1C CCC(C)(C#N)C(=O)NC1CC(O)(CNC(c2cnccn2)=O)C1 C1(C)(C(=O)NC(c2cn(Cc3n(C)cnc3)nn2)CC2CC2)CCC2(CC1)CC2 C1(CCC)CCCN(c2nnc(CCC)n2CC(c2ccc(Cl)cc2)O)C1 C1(CC)C(NC(=O)Cn2cccnc2=O)CCCN1C(=O)CC1CCCC(=O)N1 c1(C(N2C(CNC(C(CCC#C)O)=O)CC2)=O)cc(N)c2ccccc2n1 C1(C(=O)NC(C)Cc2cnc[nH]2)C=CC(NCCC(=O)CNS(N)(=O)=O)C1 N1(Cc2onc(CC)n2)CC2C(NC(=O)CCCCN3C(=O)CCC3=O)C2C1 n1(CCSCCS(C)(=O)=O)c(C(C)(C)C)nnc1Br N1(C(CC)=O)CC2ON=C(CNC(c3cc(Br)c([N+](=O)[O-])[nH]3)=O)C2C1 C1(NC(=O)C(O)CNC(c2cccnc2CO)=O)CC(=O)N(O)C1 CN1CC(C(=O)OCC(Cl)=CCNCC(c2ccccc2)C2CC2)C(O)C1 N1(C(c2ccc(C)nn2)=O)CCC(CO)C(NC(c2coc3c2CSC3)=O)C1 c1(NC2(c3ccc(OCC=C)cc3)CCOC2)cc(OC)c(OC)c(OC)c1 N1(C(C2N(CCC)CCCC2)=O)CC(C)CCC1C(=O)NCC1CCCC1CF C(=O)(C1CCCc2cncn21)N1CC2C(CNC(CC#N)=O)(CCC2)C1 CC1CCC(=CC(=O)NC(C)(C)CN(C(=O)CSCC(N2CCCCC2)=O)C)C1 CC(CCC(=O)NCC(CC#N)NC(=O)COC1(C)CCOCC1)S(C)(=O)=O C1(C(=O)NC2CCC(CC(=O)NCCc3nc(C)cs3)C2)(COC)CCOC1 c1(OC)ncc(C=CC(=O)NC2CC3(C2)CN(C(=O)CC2CCCOC2)C3)cn1 c1(C(N2C(CCNC(C(CN(C)C)O)=O)CCC2)=O)ccc(C(F)(F)F)cc1 c1(CN(C(C(F)(F)F)C2CCNCC2)C(C2CCC(=O)O2)=O)cccc(Cl)c1O C(C(=O)N(C(C)CC(=O)NCc1ccc(Cl)cc1)C)(C(C)C)SC c1(OCC)cccc(F)c1C(=O)NCC1CC(O)CN1C(C12CC3CC1C2C3)=O N1(C(C(C)O)=O)CCC(C2(O)CN(C(c3cc(-n4cccc4)ccn3)=O)C2)CC1 C1(C(C)C)CCC(C(=O)NC2CCC2C(N)=O)N1C(c1cncc(Cl)c1)=O C1(CC)CN(C(C2CCN(C(C)=O)CC2)=O)CCC1N=c1ccc(C#N)c(C)[nH]1 C12(CNC(C3(C(C)(C)C)CCC3)=O)CC1CN(C(=O)CCc1cnn[nH]1)C2 C1(C(N2CCC(OCCNC(c3c(C)cccn3)=O)C2)=O)COC(C)(C)CO1 c1(C(N2CC(CNC(c3cc(C)cc(O)c3)=O)OCC2)=O)cnc2sccc2c1 c1(C(N2C(C(=O)Nc3c(C(N)=O)cccn3)CCC2)=O)cccc2c1NCCC2 N1(C(C)(C)C)CC(C(=O)NC2CCC(NC(C3CC3C(C)(C)O)=O)CC2)CC1=O N1(C(C(C(=O)OC)(C)F)=O)CCCN(C(c2ccc(Cl)c(O)c2)=O)C(C)C1 C(CC(C)C)(C(=O)NCC1CCSC1)NC(Cc1cc(C)n(C)n1)=O C1(C(=O)NCC(CNC(C(C)CSC(F)(F)F)=O)O)CCc2nc(O)[nH]c2C1 C1(NC(C(CO)N(C)C)=O)CCCCN(c2ncnc(=N)[nH]2)C1 N1(C(c2cc(CC)c(C)s2)=O)CCN(C(c2[nH]cnc2C#N)=O)C(C(F)F)C1 N1(C(N(C23CCC(CC2)CC3)CC)=O)CCOc2c(C)cccc2C1 N1(Cc2c(C)ncs2)CCC(NC(c2cnsc2)=O)CC(C)(C)C1 C1(C(=O)NC(CC)(C)CNC(=O)CCc2ccccn2)CCCCC1(C)C c1(OC)ccc(N)c(C(=O)N(CCNC(=O)C(c2ccncc2C)C)C(C)C)c1 c1(C(N2CC(CNC(CN(C)C(N)=O)=O)OCC2)=O)ccc(O)c(F)c1 c1(C(=O)OCC)cccc2c1CN(CCOC)C2.C1(=O)C(C2CCOCC2)CN1 C(=O)(C1CCCn2ccnc21)NC1CC2CN(C(c3ccc(N)cc3)=O)CC21 C1(NC(c2ccc(C)c(O)c2)=O)CC(NC(c2cnnn2C)=O)C12CCOCC2 C12(C(=O)NC3(CNC(C(C)CS(C)=O)=O)CCC3)CC3CC1C2C3(F)F c1(CCC(=O)N(CC(C)NC(=O)C=CSc2ccccc2)CC)ccccc1Cl Cn1ncc(=NC(=O)CC2CCN(Cc3ccc(C(F)(F)F)cc3)CC2)[nH]1 Cc1cc(C)cc(C=CC(N2CCOC(C)(C(F)F)C2)=O)c1 Cc1c(CC(=O)NCC2CN(C(=O)C(C)CO)C2)c(O)nc2ccccc12 c1(C(CNC(=O)Cc2cnoc2)N(C(C2C(COCC)C2)=O)C)ccccc1 C1(c2n(CC(=C)C)nnn2)(NCC2CC(OC)C2)CCC2COC1O2 n1(CC(=O)NCCN(C(c2c(CCC)occ2)=O)C(C)C)ncn(C)c1=O C1(O)(N2CCCC(C(N3CCC(=C)CC3)=O)C2)CCC(C)CC1 C1(CCNC(C2CC=CCC2)=O)CCCCN1C(=O)Cc1ccsc1Cl C1(C(=O)NC2CCCN(C(C(CCC)=CCC)=O)C2)CN2CCC1CC2 C1(NC(CCC)=O)CCCCN(C(c2cnc(-c3ccccn3)s2)=O)C1 C1(CNC(c2sccc2I)=O)CCN(Cc2cc3sccc3s2)CC1(F)F c1(OC)cc(C(C)NC(=O)NCC(O)C(C)(C)C)ccc1F C(c1cccc(Cl)c1)=CC(=O)NCC1CN(C(c2n(CC)ccn2)=O)C(C)C1 C1(N(C(C2CCCOC2)C(=O)NC)CCC#C)CCCCC1 N1(C(c2c(Cl)cn(CCC)c2Cl)=O)CC(NC(=O)C(F)=CC2CC2)CC2(CC2)C1 c1(CNC2CCN(C(C(CC(C)C)NC(C)=O)=O)CC2)cccc2cccnc12 C=CCC(C)(C)CC(=O)N(C1CCC(NC(=O)CCCCN(C)C(C)C)C1)C C1(C(=O)Nc2cc(SCCN3CCCCC3)cc(F)c2)CCn2cnnc2C1 N1(C(Cc2c(C)c(Cl)ccc2)=O)CCOC2(CCN(C(C3CC(=O)N3)=O)CC2)C1 c1(CC(=O)NC(C)CCNC(C2CCCC2C)=O)ccc2c(c1)ncn2C Cc1cnc2c(C(N3CC(NC(c4cnc(Cl)[nH]4)=O)C4(CC4)C3)=O)cccn12 C1(C(N(C(C)CNC(c2cc3ncccc3[nH]2)=O)CC)=O)OCCCC1(C)C C=Cc1ccc(C(=O)NC(CNC(=O)CCc2cccnc2)C(C)C)cc1 CC1CCN(C(c2cnn(CC(F)(F)F)n2)=O)CC1CNC(=O)CSC(F)(F)F N1(C(C2CCN(CC)C2)=O)CCC2(CC1)CC2(C)C(=O)N(c1ccccn1)CC C1(C)(C(=O)NC(C2CN(C(C3(n4cnnn4)CC3)=O)C2)C)CCCS1(=O)=O c1(CC(=O)NCCN(C(C2N(C(CC)=O)CSC2)=O)C(C)C)cccc(Cl)c1 c12sc(nc1C)SC(CC)CN(C)C2=O.C(C)(C(=O)NCC(C)C)NC(C)=O C12(C(=O)NC(C3CCCN3C(C3(O)CCCCC3)=O)C)C3C4C1C1C2C3C41C#N c1(C(=O)NCC23OCC(NC(CSc4n(C)ncc4)=O)(C2)C3)cc(Cl)cc(Cl)c1 c1(OC)nccc(C)c1NC(C1CC(C)N1C(C1CC2CC(=O)C1O2)=O)=O C1(CN(C)C(C2(c3ccsc3)CC2)=O)CCCC(NC(c2cnc(S)[nH]2)=O)C1 CC(C)C(COCC1CCOC1)N=c1cnc(F)c[nH]1 C1(C(=O)NCCC(C)N(C(c2nc(OC)nc(O)c2)=O)C)CCC2(CCC2)CO1 c1(C(N2C(CNC(c3n(C=C)nnc3)=O)CC(C)(C)C2)=O)oc2ccccc2c1C C1(NC(C(CC)C)=O)CCCCC12CCN(C(c1ccn(C3CCCC3)n1)=O)C2 CC1(C(=O)NC2CCN(CCCO)C2)C=CCN1C(c1cc(C2CC2)[nH]n1)=O C1(NC(=O)COC2CCCCC2)CCCCCN(C(=O)CC2CC3CC3C2)C1 N1(C(C(CCC)(C)CC)=O)CCC2(C1)CN(C(C1(C)CCCCO1)=O)CCO2 N1(C(CC2(C)CC2)C(=O)NC2CCCCC2)CCCC(n2nc(C)cc2C)C1 N1(C(C(C)OCCC#C)=O)CCN(C)C(CNC(C2(n3cccn3)CCC2)=O)C1 c1(NC(C(=O)NCC2(OC)COC2)=O)cc(Cl)ncn1 c1(C(N2CC(CN(C)Cc3ccsc3Br)C2)=O)c(I)ccnc1F C1(C(N(C2(C3CC3(C)C)CC2)C)=O)CCCCCCN1C(=O)Cc1cc[nH]n1 C(=O)(CC(C)(O)C(F)(F)F)NC1CC2CN(C(C(C)(C)C#N)=O)CC1C2 Cn1ncc2c1CN(C(=O)Cc1csc(=NCc3cccn4ncnc34)[nH]1)CC2 CCCC(CNC(=O)Cc1ncccc1F)C(=O)NCC(C)CSC C1(NC(C2C(CC)CCN2C(c2cc(CO)on2)=O)=O)CN(C)CC1(C)C CC1=C(C(=O)N2CCC2CNC(c2ccoc2C(C)C)=O)CCC1 N1(C(c2c(CC)nc[nH]2)=O)CCCC(C)C1CNC(=O)Cc1cc(C)ns1 C1(C(=O)NC(CC=C)CNC(=O)Cc2cnccc2C(F)(F)F)COCCC1(F)F Cc1cccc(NC(C2CN(C(=O)C(N3CCNC3=O)C)CC2(F)F)=O)c1C#N c1(C(=O)NC2C(CNC(C(CC)COC)=O)CC2)cc(S(=O)(=O)N(C)C)c(C)o1 C1(NC(C(C)SC(F)(F)F)=O)CC2CCC(C1)N2c1ccc(C(F)(F)F)cn1 N1(C(c2cc(C)oc2C)=O)CCCC(F)(C(=O)NCc2c(C)cccc2F)C1 C1(CC=C)(NC(c2ncccc2C)=O)CCCN(C(=O)C(C)NC(C)(C)CC)C1 n1(CCN(C)C)cc(C(=O)NC2CC2C(=O)N(C2CC=CC2)C)cn1 C1(C(N(C)CCN2CC=CC2)=O)(CO)CCCN1C(=O)CCOCC(C)(C)C N1(C(C2(C)CN(C(C3CC(=O)CS3)=O)C2)=O)CCC2C(C(N)=O)C2C1 CCCC(C)(CC)C(=O)NCCCNC(c1ccc(C#N)c(C)c1)=O N1(C(=O)C2=CCCOC2)CC2CCC1CN2C(c1cn(C2CC2)cn1)=O c1(C(=O)NCCC(=C)CNC(=O)C(O)c2cnc[nH]2)cn2c(n1)CCC(C)C2 C1(CCCNC(CCCOC)=O)CCCCN1CC(=O)N(C)C(c1ccccn1)C N1(C(C2CC(C)OC2=O)=O)CCC(C2(NC(=O)C3=COCCO3)CC2)CC1 C1(C(=O)OCC2CCN(C(C)=O)CC2)CCC2(CCNCC2)CC1 Cc1nc2cc(C(N3CC4CCCC4(NC(=O)C#CC4CCC4)C3)=O)cnc2s1 C1(C(N(C(C)CNC(C2(c3cccs3)CCCC2)=O)CC)=O)CCNC1=O C1(C(=O)NCC(C2CCC2)NC(=O)Cc2cc(C3CC3)on2)CCCC2(CC2)C1 S(=O)(=O)(c1cnc(NCc2cccc(F)c2F)c(Cl)c1)NC(C1(S(C)(=O)=O)CC1)C C(=O)(CC(C)(C)C(F)(F)F)N(C(CNC(c1c(CC)nn(C)c1Cl)=O)C1CC1)C C=CCCC(C(=O)NCc1cc(O)cc(F)c1)NC(=O)CCc1ccco1 c1(OC)ncc(C(=O)NC2C=CC(CNC(=O)C3CC3)C2)cn1 N1(Cc2cc3c(cc2)OC(C)C3)CC=C(c2ccc([N+](=O)[O-])cc2)CC1 C1(C(N(C2CCN(C(=O)C(O)Cc3cnc[nH]3)C2)CCC)=O)CC12CCOCC2 C1(OC(c2ccc(Cl)o2)C)C2CC3C(=O)OC1C3O2 N1(C(c2cnc(S)[nH]2)=O)CCN(C(=O)C2=C(Cl)CCC2)C(CCO)C1 c1(C(=O)NC2CC(CNC(c3cn4c(n3)SCC4)=O)C2)ccc2sccc2c1 c1(C(=O)NC(CNC(C(C)NC(CC)=O)=O)(C)CC(C)C)ccnc2[nH]ncc12 C(C(C(C)C(C)C)NC(c1c(Br)c(C)nn1C)=O)NC(CCC)=O C(=O)(C1Cc2ccccc21)NC1(COC)CN(C(=O)CCc2cn[nH]c2)C1 c1(C(=O)NCC(C)NC(c2ccc3cncn3c2)=O)cccc2c1COCC2 C1(CC(=O)NC)CN(C(c2c(C)coc2C2CC2)=O)CCN1C(=O)C=CC1CC1 c1(C(C)=O)ccc(NC(C2(F)CN(C(=O)C(C)Oc3ccccn3)C2)=O)c(I)n1 N1(C(CC(=O)NCC)=O)CCCC1(C)CNC(c1cn(C2CCCC2)nc1C)=O c1(NC(c2ccc[nH]2)=O)cccc(NC(=O)C(O)Cc2ccccc2)c1 Cc1cc(=NCCN2CCCC2C(C)(C)CO)[nH]c(N(C)CC2COCCO2)n1 CC1(C)CN(C(c2cnccc2C#N)=O)C(CNC(=O)CCc2cnn[nH]2)CO1 C(N=c1[nH]c(=NC2CCC=CCC2)[nH]c2c1CCCC2)C1(C)C(C)(C)C1 N1(C(C(CC=CC)C)=O)CC(C)C(C)(C(N2CCC(c3cnco3)C2)=O)C1 S(=O)(=O)(c1c[nH]c(C(=O)N(CC(C)NC(=O)C(C)(C)C(N)=O)C)c1)NCCOC C(=O)(C(C)(CNC(c1cc(C)n(C(C)(C)C)n1)=O)c1ccc(F)cc1)OC Cn1ncc2cc(C(N3CC(NC(c4csc(CO)n4)=O)CCC(O)C3)=O)sc12 C(=O)(C(C)n1cncn1)NCC1(C(C)NC(CC)=O)CC1 C1(NC(C(CO)OC)=O)CN(C(C2(C)CCOC2)=O)CC1CO CC(C)(C)CCCC(=O)N1CCOC(CC(=O)NCCN2CCOCC2=O)C1 C=CCC(C)C(=O)N1CCC(OCC2CCN(C(C3CS(=O)(=O)C3)=O)CC2)C1 C(C(C(=O)NC1CCCC1CCO)NC(C1CC1(F)Cl)=O)N(C)C c1(C(N2CC(c3ccccc3)(NC(C3C(C)CCO3)=O)C2)=O)occ2c1CCC2 c1(C(N(C(C)CCNC(=O)Cc2nc(=N)[nH][nH]2)C)=O)ncc(F)cn1 c1(C(N2CCCC(CO)(NC(C3(F)CCCCC3)=O)C2)=O)ncn2c1CCC2 N1(C(C(C=CC)O)=O)CCC(CNC(c2cn(C(C)(C)C)nc2C)=O)C12CC2 C1(NC(CN2CCN(CC)CC2)=O)CC2(CCN(C(=O)C(C)=CC)C2)C1 C=C(C)CC(C(=O)N1CC(O)CC1C(=O)NC1CCC(C)CC1)OC C1(C(N(CCN(C(=O)CCc2cscn2)C)C)=O)CC1(F)F C1(CNC(CC(=O)NCC#C)=O)CN(C(C2CCC(CC)O2)=O)CC(C)(C)C1 c1(C(=O)NC2(CN(C)C(C3(O)CCC3)=O)CC2)ccc(Br)c(C(F)F)c1 C(=O)(CC(C)C(C)(C)NC(=O)CC(C1CC1)C1CC1)Nc1ccc(OC)nc1 c1(C(=O)OC)cc(CCC(=O)NC(C)(C)CNC(C2CCC2C)=O)c[nH]1 C1(c2ncc(C)o2)CN(N(C)Cc2nccn2CC(C)C)C1 c1(OC)cc(C)cc(C(=O)NCC2(F)CCC(NC(=O)C(F)(F)C(C)O)C2)c1C c1(NC(N(CC#C)Cc2cccc(C)n2)=O)nc2cc(C)ccc2n1C Cc1c(F)cc(C(N2CC(CNC(=O)COCCF)CC(C)C2)=O)c(F)c1N C=CCC(C(=O)NC(C)(CNC(=O)Cc1ccn(C(C)C)n1)CC(C)C)C(C)C C1(C(=O)NC(C(=O)OCCC)C)CC(O)CN1C(c1cnc(S)nc1)=O C1(CCC(=O)N(CC(=O)Nc2cn[nH]c2)C)NC(=O)NC1=O CC1CCCC1(C)C(=O)N(C1CCN(C(=O)CCC(F)F)CC1)CC1CC1 N1(C(C2(NC(C(C)n3cnnn3)=O)CCC2)=O)CC2C(=O)NC(=O)C2C1 c1(NC(C2CC(N(C)C)C2)=O)cc(NC(=O)CCOCC(C)(C)C)c(Cl)cn1.CC c1(OC)ccc(-c2nc(-c3cnnn3C)n[nH]2)cc1 N1(C(C(CC)OCC)=O)CCCC(C)(C)C1CNC(c1ccc2c(c1)COC2)=O C(=O)(C1CCc2nnc(C)n21)N1CC(NC(CCC#C)=O)C(OC)C1 Cc1ccc(C(=O)NCC(F)CNC(=O)CCN2CCCC2=O)cc1C c1(C(=O)NC(C)CC(C)NC(C2(F)CCC(=O)CC2)=O)cccc2c1OCCN2 C(CC1=CCCCC1)N(C)C(C1CCC1CNC(=O)C=CC1CCC1)=O O=C(CC(C1CC1)C1CC1)NCCC1(C(=O)NCC2CCC(O)C2)CCCC1 CCC(C)(C)C(O)C(=O)N1CC2CC1CN2C(=O)Cc1cn2ccsc2n1 c1(Cn2cc(C(C3CC3C)C)c(-c3ccccc3F)n2)cn2ccccc2n1 Cc1nc(O)c(Br)cc1C(=O)NCC1CN(C(c2cnsn2)=O)CC1C N1(C(c2cn3ccccc3n2)=O)CCOC2(CCN(C(C3CC4CCC4C3)=O)C2)C1 N1(C(=O)C=Cc2ccco2)CCC(N2CCN(C(=O)CSC3CC3)CC2)CC1 C1(O)(CCC(=O)OC(C)(C)C)CCN(C(N2C(c3c(C)cccn3)CCC2)=O)CC1 CCC(CN(C)C)C(=O)NCC1C=CCN1C(c1cccc(CCOC)c1)=O N1(C(=O)OC(C)(C)C)CCC2(CCCC(C(=O)NCC(c3cncs3)O)O2)C1 n1(CC(=O)NCC(O)CCNC(c2ccoc2Cl)=O)ncn2nccc2c1=O c1(OC)c(C(=O)NCCC(C)CCn2cncn2)cccc1C.C(=O)(CN(C)CC)N c1(-c2ccc(C(N3CC4N(C)C(CCC4)C3)=O)cc2)cnc2cc(Br)ccc2c1 c1(-c2ccc(N3CCCC(NC(N(C)C)=O)C3)cc2)ncc2c(n1)CCC2 Cc1c(C(N2CCOCC(CNC(=O)C(C)C(C)C)C2)=O)c(C)n2ccncc12 C1(C(=O)NC(C)CCN(C)C(C2CC3CCC2O3)=O)CN(S(=O)(=O)N(C)C)C1 Cc1ccc(SCC2CC(NC(C3CCOC3(C)C)=O)C2)cc1.C1(C)C(=O)N1 CC1(C)CC(NC(c2csc(CC(F)F)n2)=O)CN1C(=O)CC1CC2(CC2)CO1 c1(C(C)O)cccc(CO)c1.c12cn(nn1)CCN(C1CC1)C(=O)C2.C1(C(=O)N)CSC1 c1(C(=O)NC(CC)(CNC(=O)CC2(OC)CC2)CC)cc(C)c2c(c1)CCC2 Cc1c(Cl)cnc(NCC(C)NC(c2cc3ccc(F)cc3o2)=O)c1C#N N1(C(C(CCC)OCC)=O)CC(CNC(C2(F)CC2)=O)C(C)(C)C1 Cc1cc(Cl)nc(N)c1C(=O)NCCCCCNC(=O)CN(C)CCO Cc1cc(C)cc(S(=O)(=O)N2CCC=C(C(=O)NC(C)CO)C2)c1 C(=O)(C1CCCn2nccc21)NC1(CO)CCN(C(C(C(=O)NC)(C)C)=O)C1 C1(C(=O)OCC)CCCC(C(=O)NCC(O)CN(C)C(c2conc2CC)=O)C1 N1(C(C(=O)NCC=C)C2(C(F)(F)F)CC2)C(C)CN(CC(C)(C)COC)CC1C Cn1ccnc1CC(=O)NCCCOCC(F)F.C12CC1C(=O)NC2 C1(C(=O)NCc2ccc(Cl)s2)CCN(Cc2ccco2)C1=O C#CCCCCC(=O)N1CCCCC1C(=O)NCCCSC N1(C(CC=CC=C)=O)CC2CC(NC(C3CC4C=CC3CCC4)=O)C(C2)C1 C1(NC(C(N2CCC(CCNC(=O)OC(C)(C)C)CC2)=O)=O)CC(=O)OC1(C)C Cc1nc(Br)c(CN(C)C(C2CCC(C)NC2=O)=O)n1C C1(CC(=O)OC)(NC(=O)CC2NCC23CCC3)CCOCC1 N1(C(C(Br)=C(C)C)=O)CCN(C(c2cncc(C(F)(F)F)n2)=O)CC1C C1(NC(CC(CC)C2CCC2)=O)CN(C(C2Cc3ccccc3N2)=O)CCC1C C1(C(=O)NCC2(NC(C3CC4CCC(C3)O4)=O)CCC2)CCCCC12OCCO2 N1(CC(C)NC(=O)CC2CC2)CCN(C(=O)CSc2nnnn2C(C)(C)C)CC1 CCCC(C(O)C(=O)NCCC1CC=CCC1)NC(=O)COCCF c1(C(=O)NC2C=CC(CC(=O)Nc3cncnc3O)C2)cccc2ncccc12 c1(C(=O)NCC2OCCCN(C(C(=O)NCCOC)=O)C2)ccc(C#N)cc1F c1(CC)cc(C(N2CCCC(C(C)(O)CNC(=O)CCSCC)C2)=O)ccc1C C(=O)(CS(=O)CCC(F)(F)F)N1CCC(O)(CN(C(=O)Cc2ccccc2)C)C1 N1(C(C(CNC(C(C)N(C(C)=O)C)=O)O)=O)CCC2(CC1)CC2CO C(=O)(C1=NOC(CNC(c2nccnc2OC)=O)C1)N1CCC(OCC)CC1 CC(CCC(C)(C)C)C(=O)NCC1N(C(=O)C#CC(C)(C)C)CCC1(C)C c1(-c2cn(C3CN(C(CC=CC=CC)=O)C3)nn2)cc(C)cc(F)c1 C(N=c1cc(C)[nH]c(=NCCc2c[nH]c(=N)nc2O)[nH]1)C1(CC)CCCOC1 CN1CC2CCC(C1)N2C(C1C2CCC(C2)C1NC(C1(C)CCCC1)=O)=O c1(CNC(=O)C(CC)CO)ccc(N2CCCC(C(C)OC)C2)nc1C N1(C(Cc2ccc(C)cc2)=O)CC(NCc2cccc(I)c2O)C(C#N)C1 CC1(C)OCCC1CC(=O)NCC(C1CC1)NC(C1C(C)(C)C1(F)F)=O CC1(C)COC(C)(C(N2CC3CN(C(C4CCC(F)(F)CC4)=O)CC3C2)=O)CO1 Cc1coc(C(=O)N(CC(C)CNC(c2ccc(-n3cccn3)nc2)=O)C)c1C c12cc(c(F)cc1C)C(c1n(CC)ccn1)N2.c1nnnn1C(C)C.C(C)C C1(C(N2C(CNC(CC3C(C)=NOC3=O)=O)CC2)=O)CC2CC(O)CC(C1)C2 c1(NC(C2N(CCCC#C)CCSC2)=O)cnc(C)c(Br)c1 c1(CC)c(C(=O)NC2(CN(C)C(C3CCC(F)C3)=O)CC2)cnc2ncnn12 C1(C(=O)NC(CC(C)C)CNC(=O)C=Cc2ccccc2)CCCS(=O)(=O)C1 C1(CCNC(CSCC(C)=O)=O)CCN(C(c2ccnnc2)=O)CC1 c1(OC)ncc(C(=O)NCC2CN(C(c3cccnc3O)=O)CCO2)cn1 C1(C(N(CCCOC)CCO)=O)CCCCN1C(=O)CCc1nc(C)no1 N1(C(CCC(C)NC(C(C)N(CC)CC)=O)=O)CCc2ccsc2C1 C1(CNC(CCC(C)N(C)C)=O)CCC(F)(CNC(C2CCO2)=O)CC1 C1(NC(c2cc(-c3ccccc3)cs2)=O)(CNC(C23CCC(C2)C3)=O)CCCC1 CC1CCC(=CC(=O)N(CC(=O)NCC2(C(=O)N(C)C)CCCC2)C)CC1 C1(c2n(C)ncc2)C(NC(=O)Cc2cncn2C)CC(=O)N1C(=O)NC1CC1 C=C=CCC(=O)NC(CN(C)C(c1cn(Cc2ccccc2)cn1)=O)CC N1(C(=O)C=Cc2cccnc2)CC(CNC(=O)C(F)(F)C2CC2)N2CCC1C2 C1(CC(=O)NC2(CC(=O)OCC)CC2)CN(C(c2coc(C)c2)=O)CCC1C C1(NC(C2N(C(C(C)OCC#C)=O)CC(C)C2)=O)CC2C(O)C(O)CC12 C1(NC(C=CC(CC)C)=O)CC2CCCC(C1)N2C(c1ccnnc1)=O N1(C(CN(C(C)C)C)=O)CC=C(CNC(C2CCC3CC3CC2)=O)CC1 O=S(=O)(c1nc(C2CC2)cs1)N1CCn2nnc(Br)c21 C(=O)(C1=CCCCO1)N(CC(N1CCCC(CC)C1)=O)CC#C c1(CC(=O)NC(CC)(C)CNC(=O)C(CSC)OC)cccc(SC(F)(F)F)c1 c1(NCc2c(CC)cc(Cl)cc2)nccc2c(F)cccc12 CN1C(=O)CC(C(=O)Nc2ncc(C(F)(F)F)cc2Br)C1c1nccn1C CC1(CN2CC=CC2)CCCN(C(=O)NC(=O)Cc2cnn(C(F)F)c2)C1 N1(C(C(C)O)=O)CCCCC(NC(=O)CSc2ccccc2Cl)CC1 c1(OC)ccc(NC(c2cnn(CCC(C)C)c2C2CC2)=O)cc1-c1ccco1 c1(C(N2CC(C)C(NC(C3CC(F)(CO)C3)=O)C2)=O)cc(O)nc(N(C)C)n1 c1(C(=O)NCC23N(C(C(=O)OCC)=O)CC(C2)C3)cc(OC)ccc1[N+](=O)[O-] C1(NC(C2N(CC)CC2)=O)CCN(C(c2nscc2Br)=O)CC1 c1(C(=O)NCC2N(C(c3cn(CCC)nc3)=O)CC2)cccn(C)c1=O N1(C(C2CC(C)(O)C2)=O)CC(NC(c2cccc[n+]2[O-])=O)CC2(CC2)C1 C(N=c1ccnc(C2CCC2)[nH]1)C1CCN(C(c2cc(C3CCC3)on2)=O)C1 C1(C(N(C2(C(N3CCC(C(=O)OC)C(O)C3)=O)CC2)C)=O)CCOC(C)(C)C1 c1(C(=O)NC2CCC(NC(c3nc(C)n(C)n3)=O)C2)ccc2c(O)nccc2n1 N1(C(C(c2cccnc2)OC)=O)CC2CCC1C1CN(C(=O)C(C)(C)CF)CC21 c1(C(N2CCN(C(C(CC)c3ccccc3)=O)CC2CO)=O)nsc2ccccc12 Cn1nc2c(c1C(=O)NC1CC3CC1N(C(c1ccnnc1O)=O)C3)CSCC2 C1(NC(=O)NC(Cc2ccccc2F)CO)C2Cc3c(Cl)cccc3C12 c1(C(=O)NC2C=CC(CNC(c3cc(C)oc3)=O)C2)ccncc1C(F)F CC1=NOC(C)(CNC(=O)CCOCCNC(c2cc(C)oc2C)=O)C1 C1(OC)CN(C(C2CC=CCN2C)=O)CC1c1ccc(F)cc1 Cc1nc(CC(F)(F)F)sc1C(=O)NCC1(C)CCN(C(=O)C2=CCOC2)C1 c1(OC)cc(C(=O)N(C(C)CNC(c2csc(C#N)c2)=O)C)ccc1Cl CCCCCC(O)C(=O)NCc1cccc(C(=O)NCC2CC=CCC2)n1 C1(N(C(=O)CCc2cncnc2)Cc2cc(Cl)nc(Cl)c2)COC2(CCNCC2)C1 C1(CNC(C(C)OC)=O)CC(OC)CN1C(=O)Cc1ccccc1F Cc1ccc(C)c(C(N2CC3(CO)CC2(C(=O)NCc2cccc(C)c2C)C3)=O)n1 c1(OCC)ccc(CC(N2C(CNC(C3CCC(=O)N3)=O)CC3CC23)=O)nc1 C1(NC(c2cc(C)n(C)n2)=O)CN(C(c2cocn2)=O)CCC1C C#CCCCCCC(=O)NCCOC1CCN(C(C2SCCS2)=O)C1 Cc1cccn(CC(=O)NCC2CN(C)CCN2C(=O)Cn2cc(Cl)cn2)c1=O C1(CC(=O)NCCC(C)N(C(=O)CN(c2ccncc2)C)C)CCC(=O)NC1=O n1(CC)nc(C(=O)NCC2COC(CNC(C3CCCN3C=O)=O)C2)cc1O C(CCC(=O)NCCc1nc[nH]n1)NC(C1C(C(=O)OC)C1)=O C1(CC)CN(C(=O)C(C)(C)CF)CCC1NC(c1ccn(CCF)n1)=O c1(CNC(c2cn(-c3nccs3)nn2)=O)ccccc1S(=O)(=O)c1ccccc1 N1(C(c2c(CC)n(C)cc2)=O)CCCC(C)(C(N2CCCCC2)=O)C1 N1(C(CSC(C)C)=O)CC2CN(C(=O)C(C)C(C)(C)C)CC2(C)C1 C1(NC(C2C=C(C)CS2)=O)C2CC3C(C2)C13C(=O)N(C(C)(C)CO)C1CC1 c1(C(=O)NC(C(C)NC(c2ncc(C)cn2)=O)CO)cnn2c1NCC(C)C2 C(=O)(C(C)CC(F)(F)F)NC(C1CN(C(Cc2nc(C)sc2)=O)C1)C N1(C(CC(C(=O)OC)C)=O)CCN(C(c2coc(S(=O)(=O)NC)c2)=O)CCC1C c1(NC(N2CCC(CC)CC2)=O)ccc2cnn(C)c2c1 C1(CNC(CC=C)=O)CC2CCC1N(C(=O)Cc1cn3ccccc3n1)C2 Cn1[nH]c(=NC(=O)C(CC2CC2)NC(=O)Cc2cncnc2O)cc1C1CC1 c1(CC(N2CC(CNC(c3cnc(CO)cn3)=O)C(O)C2)=O)ccc(F)cc1F C1(NC(C(CCSC)O)=O)CC2(CCN(C(C34CC(C(C)C)(CO3)C4)=O)C2)C1 C12(C(=O)OC)CCCC1(C(=O)NCCN1CCN(C(=O)C(C)CN(C)C)CC1)C2 c1(C(=O)NCC2(NC(C3CC(CC)OCC3)=O)CCC2)cccc2c1NCCC2 c1(NC(C2N(C(COC(C)C)=O)CC2)=O)ccccc1C(C)(F)F CC(C)C(O)C(F)(F)C(=O)NC1CN(C(=O)Cc2ccon2)C2CCCCC12 c1(CC)cc(C(=O)NC(CCN(C(=O)C(C)(C)F)C)C(C)C)nc(Cl)n1 Cc1ncc(NC(=O)C(CC(F)F)N(C(=O)C(C)NC=O)C)cc1Cl C1(O)(CNC(c2nncs2)=O)CCCN(C(=O)COCc2cccnc2)CC1 C1(NC(C2C(C)=C2)=O)CC2CN(C(c3sccc3F)=O)CC12 C1(CNC(C=CC=CCC)=O)N(C(=O)CCC(C)(C)C)CCC1(C)C c1(OC)cnc(Cl)nc1N1CCOC(C(C)NC(C23CCCCC2C3)=O)C1 CCC(C)(O)C(=O)NCC12CC1CN(C(=O)COc1cccnc1)C2 Nc1ccc(C(=O)NC2CC(O)CN(C(=O)Cc3ccno3)C2)nc1N C1(CC)CC(C(=O)NC2(CNC(=O)C=Cc3nc(C)cs3)CCOC2)CC(=O)N1 C#CC1(C(=O)NC(C)CC(=O)NC)CCN(C(=O)CCCF)C1 C1(CNC(C2C(CCOC)C2)=O)CN(C(c2cc(F)ccc2C)=O)C2(CCC2)C1 Cc1cc(C(=O)NC2(C#N)CCN(Cc3cccnc3Br)C2)cc(Cl)n1 CC1CN(C(=O)CC2CC2)CCC1CNC(=O)C(=O)CC(=O)c1ccsc1 C12(C(=O)NCC3C(C)CCCC3)CCC(NC(=O)CCn3cncn3)(CC1)C2 C(C(CNC(C1CCOC(C(N)=O)C1)=O)S(C)(=O)=O)NC(c1cnc(CC)nc1)=O N1(C(c2ncc(C)cn2)=O)CCCC12CCC(NC(=O)CN1CCC(C)C1)CC2 N1(c2n(C)c(-c3cc4c(cc3O)OCO4)nn2)CCOc2ccc(Cl)cc2C1 C1(C(=O)OC)CCC(C(=O)CC2(CN(C(=O)CCn3ccnn3)C)CC2)C1 N1(C(C2(COCC)CC2)=O)CC2CC(NC(=O)C=Cc3c[nH]cn3)C2C1 C(CC(CC)C(=O)NCCC1CCCN1C(=O)CSCC(F)(F)F)=CC N1(C(C(C(C)=O)(C)C)=O)CCC2(CC1)COC(C(=O)Nc1ncc(O)cn1)C2 C(=O)(CC(F)(F)CC(=O)N1CCC(C(=O)NCC2CCOC(C)C2)CC1)OC N1(C(c2cnnc(C)c2C)=O)CC2CCCC2(C(N2CC(C)(C)CC2C)=O)C1 c1(C(N2C(COC)CN(C(=O)CCCC(C)=O)CC2)=O)cnc2[nH]ncc2c1 c1(NCc2cc(C)ncn2)nc2ccccc2n1-c1ccccc1 C(c1ccc(F)cc1)=CC(C(N1CC(NC(Cc2ncc(C)s2)=O)C(C)C1)=O)=O CC#CCCCC(=O)N(CC(C)NC(C1CCCC(=O)O1)=O)C c1(-c2cc(CCC=C)c(F)cc2)cc(C)c(S(=O)(=O)NCCOC)cc1C c1(C(=O)NCC2CCCCN(C(CC3C(C)C3(F)F)=O)C2)cccc2[nH]ncc12 N12C(=O)CN(C1=O)CCC1CCCN21.Cc1ccccc1C.c1ccc(F)cc1 C[Si](C)(C)CCCNC(=O)C(C1CCN(C(=O)CC(=O)NCC(F)F)C1)F N1(C(CN(CCC)C(C2CCCC(F)(F)C2)=O)=O)CCCC(F)(F)CC1 C(=O)(C(C)Cc1cccnc1)NCCC(C)NC(C1(C#N)CCC1)=O C(C)(C)(C(=O)N(C)CC1(n2cccn2)CC1)NC(C1COC(C2CC2)C1)=O c1(C(N2C(Cn3cc(CN(C)S(N)(=O)=O)nn3)CCC2)=O)ccc(Br)cc1[N+](=O)[O-] N1(C(CC(C)CN(C)C)=O)CCCC(C)(CNC(c2cccc(Cl)n2)=O)C1 c1(C(N(C(c2cccs2)C)C2CC2)=O)ccc(Cl)c(Cl)c1 c1(CC(=O)NCC(CC)(C)NC(c2cnn(CCF)c2)=O)cccnc1O C1(C(=O)NCc2c(OC)n[nH]c2)C2CCC(C2)N1C(=O)CCc1ccsc1 CC1CN(C(=O)NC2CCCN2S(=O)(=O)Cc2ccccc2)CC(C)(C)CO1 CCC(F)(F)CC(=O)N1CCC(CC(N2CCCC2(C)CC2CC2)=O)CC1 c1(CCC(N2CC(CNC(c3c(C)snc3)=O)OCC2)=O)ccccc1[N+](=O)[O-] C1(CNC(c2n(CC#C)ccc2)=O)CCC(C)N(C(=O)CC(C)(C)OC)C1 c1(OC)cnc(Cl)c(NC(C2CCCC2NC(=O)CCC2CC2)=O)n1 N(C(=NCC1CC1)NC1c2noc1n2)CC1(OCC)CCOC1.C1CC1 C1(C(=O)NCC2CCCS2)(CNC(CCC#C)=O)CC12CCC2 c1(C(N(C2CCN(C(C3CCC(C)O3)=O)C2)CC)=O)c(C)nc2sccn12 n1(CC)cc(Cl)c(C(=O)N(C2CC2)C)n1.c1(CNC(=O)C2CC2)ccc(Cl)cc1 c1(N)ncc(Cl)nc1Cl.c1(C(=O)Nc2cccc(N)c2)ccc(Cl)cc1OCCO N1(C(C(C)C)=O)CC2CCCC2(CNC(=O)C(C)Cc2cccnc2)C1 C(=O)(C1=C(Cl)CCCC1)NC(C1N(C(c2sc(CC)c(C)c2)=O)CCCC1)C Cc1ccc(C2CC2)c(C(=O)NC2CCC2NC(=O)Cn2ccc(C3CC3)n2)c1 C(CCCC(C)(F)F)NC(CN(C(=O)Cc1ccon1)CCOC)=O C1(NC(c2cc(CCC)nn2C)=O)CCCC12CN(C(=O)CC1(C(F)F)CC1)C2 C1(C)(CNC(C(CN(C)C)N(C)C)=O)CCCN1C(c1cc(C(F)(F)F)cs1)=O N1(C(C(C)(C)C)=O)CCN(N2CCN(C34CCC(CC3)CC4)CC2)CC1 c1(C2(CC)CCC2OCc2ccc(=O)n(-c3ccccc3)c2)cc(C#N)ccn1 n1(Cc2ccc(C)cc2)cnc2c(N3CCC4OCCC4C3)ncnc12.C(=O)S C1(C2(O)CCC2)(CNC(C(C2CC(NC(c3c(C)n[nH]c3C)=O)C2)F)=O)CC1 c1(C(N2CCC(NC(=O)C=CCO)CC2C2CC2)=O)cc2ccccc2cc1F CN1N=C(CC(=O)N2CC(NC(c3ccc(O)nn3)=O)CC23CCCC3)CC1=O c1(C(C(=O)NC(c2ccccc2)C)N(CC(C)OC)C)ccc(Br)cn1 CC1(CNC(=O)CCc2cc[nH]n2)CCN(C(=O)Cc2ccccc2CO)CC1 C=CC1(CC(=O)NC2CS(=O)(=O)CC2NC(C2CC(F)(COC)C2)=O)CCOCC1 C(C1CN(C(=O)COCCCOC)CC1C(N1CCCC(O)(C(C)C)C1)=O)=CC c1(CC)ccc(Cl)c(C(=O)NC2CN(C(=O)Cn3nnc(=N)[nH]3)CC2C)c1 Cn1nc(Br)cc1C(N1CC(CNC(c2cn(CCO)nn2)=O)C(O)C1)=O CCCCCCCCCC(=O)NC1CCN(C(c2csc(C(C)=O)n2)=O)CC1O C=CC(CC)CC(=O)N1CCC(C(=O)Nc2nc(C3CC3)c(Br)s2)C1 c1(C(C(=O)NCCOCC)N(c2cc(Cl)c(Cl)s2)C)cccc(C(=O)OC)c1 CCC(C)(CCC(C)C)C(=O)N1CC(F)(CNC(=O)CN2CC(C)(C)C2)C1 CC1CCC(O)CN1CCCNC(=O)N(CCCCO)C1CC1 CC1CN(C(c2ncn(C)n2)=O)CC1NC(=O)CCn1ccnn1 CC1(C)CCN(C(c2ccc(F)o2)=O)CC1CNC(=O)C(F)(F)c1ccccc1 C1(C)(CNC(C(C)O)=O)CC(F)(F)CN1C(=O)CCc1cccnc1 CC(C)(CCCNC(c1ncccc1C1CC1)=O)NC(=O)CSCC(N)=O c1(SC)cccc(C(=O)NC2CCN(C(=O)CCc3csc(=N)[nH]3)CC2O)c1Cl c1(C(=O)NCC(CCOC)NC(C2(O)COC2)=O)cncc(Cl)c1 C1(CCCC)CN(C(C2CCCNC2=O)=O)CCN1C(=O)CC(C1CC1)OCC c1(C(=O)NC(C)CCNC(c2cc3n(c2)CCOC3)=O)cnn2c(N)ccnc12 N1(C(C(C)OCC(C)C)=O)CCC2(CC1)CC2C(=O)Nc1cncc(Cl)n1 N1(C(c2c(Br)cn(C(C)C)n2)=O)CCc2c(CCN(C)C)cccc2C1 Cc1ncc(C(=O)N(C)CCOCCNc2c(I)cnn2C)c(-c2ccccc2)n1 N1(C(c2cc(C)sc2C)=O)CC2CCCC1(CNC(=O)COc1ccon1)C2 C=C1CCC(C(N2CCC(C(=O)N(C3(CC)CC3)C)(CC)C2)=O)CC1 c1(C(C(=O)NC(CNC(C2(COC)CC2)=O)C2CC2)C)c(C)noc1C C(=O)(CC(C)(O)COC)N1CCCC(C(C(N2C(CO)CC(CC)C2)=O)C)C1 C(=O)(CCS(C)=O)NC1(C(=O)OCC)CC1(C)C c1(C(=O)NCCCC#C)ccc2c(c1)CN(C(=O)Cc1ccoc1)CC2 C1(CNC(c2c(CC)cccc2)=O)CC(C)(C)CN1C(=O)CCCn1cncn1 N1(C(C2C(=C)C2C(=O)OC)=O)CCN(C(c2cc(C)ccc2O)=O)CC1C C1(CCC)CN(C(c2cnc(C)nc2)=O)CCN1C(c1nnn(C(C)(C)C)n1)=O N1(C(C(CCCNC(CCSCCCC)=O)O)=O)CCC2(CNC(=O)O2)C1 Cn1nnc(CNC(C2CCC(=O)C2)=O)c1C(=O)NOC1CCOC1 C=C(Cl)CCC(=O)NC1CN(C(C2(COC)CCOCC2)=O)CC1C c1(C(=O)NCCC(CNC(=O)CCOC2CCOCC2)OC)cnn(C)c1N c1(C(=O)NCC2CC(F)(CNC(CN3CCC(C)CC3)=O)C2)cnn(C)c1C#N N1(C(CC=CCC)=O)CC2OCC(NC(c3cnc4ccnn4c3)=O)C2C1 c1(C(=O)NCC2(CCNC(C(C(C)O)N(C)C)=O)CC2)sc(C#N)cc1Cl c1(C(=O)NC2CN(C(CCCOCC)=O)C(C)C2)cc(C(F)F)ccc1Cl Cn1c2c(ccc1=O)C(NC1CCNCC1(F)F)CCC2 O(Nc1ncc(F)cc1Br)C(C)Cc1ccc(Cl)cc1Cl C1(CNC(CS(=O)(=O)NCC)=O)CC2(CCC2)CN1C(c1c(Cl)cnn1C)=O N1(C(CCCNC(=O)OC)=O)CCC2CN(C(C3(C(N)=O)CC3)=O)CCC2C1 Cc1ccn2ncc(C(=O)NC3CCN(C(c4nnccc4C)=O)C3(C)C)c2n1 N1(C(c2c(SC)scc2)C(=O)NC2CCOCC2)CC2CCCC(N(C)C)C2C1 N1(C(c2c(CCC)occ2)=O)CCC(C)C(CNC(C2(CCOC)CCC2)=O)C1 C(=O)(CC(C)(C)C(F)(F)F)N(C1CCN(C(c2nc(C(=O)OC)sc2)=O)C1)C c1(CN(C2(CNC(C3CC3OC(C)(C)C)=O)CC2)C)ccc(F)c(F)c1 N1(C(C(COCC=C)C(C)(C)C)=O)CCC(C2CC2NC(=O)CCC(N)=O)CC1 Cc1ccc(S(=O)(=O)N2CCC2C(N2CC(F)(F)C(F)(F)C2)=O)c(F)c1 N1(C(CCCN(C(=O)OCC)C)=O)CCCC(C)(NC(=O)CC(COC)CC)C1 C1(NC(C=CCC)=O)CN(C(C23CC4CC2C3C4(F)F)=O)C2(CCCCCC2)C1 N1(C(c2cc(OC)ncc2)=O)CCCC1C1CCCN1C(c1cnco1)=O c1(C(=O)NCC2C(NC(c3c(C)oc(Br)c3)=O)C2)ccc2sccc2c1 C12CCCCN(C1=O)CC(=O)N1CC(c3noc(n3)CC2=O)C1.CO Cc1nccc2cc(C(=O)NCC3CN(C(=O)CC(C)(C)O)CC3(F)F)[nH]c12 C1(C(N(CCCO)CC)=O)(CC)CCCN(C(C2(C#N)CC2(C)C)=O)C1 C1(C(=O)NCC(C)(C)C2CCCO2)CC(CC)C1 c1(-c2cc(C(=O)NC3CCN(C(C4C(C)C4C)=O)C3C)no2)ccc(Cl)cc1F Cc1cc(F)ccc1C(N1CCCC(C(C)NC(=O)C2=COCCC2)C1)=O C1(CC=C)(NC(c2cccc(CNC(=O)CN3CSCC3=O)n2)=O)CCCCC1 C1(C(=O)NC(CNC(CCNC(=O)NC)=O)C)CCCN1C1CCCCC1 CCC(C(=O)N(CCC(=O)N(C)CC1CCN(C)C1)C1CC1)n1cncn1 Cn1nc(C(=O)NCC2OCCC2C(=O)NC2CC(O)C(O)C2)cc1O C(=O)(CCCC(=O)NC)C(C(C(C)C)OC)=O.N1(C(CN)=O)CCOCC(C)C1 Cc1onc(C(=O)NC2CN(Cc3ccnc(F)c3)CC2F)c1C c1(C(N2CCC3(CN(c4nc(OC)c(F)cn4)C3)C2)=O)ccc2cnn(C)c2c1 c1(OCCN(CC(CN(C(CCCOCC=C)=O)C)O)C)ccccc1C C(=O)(CCCSCC(C)C)NC(=O)CSCCNC(COCCCCC)=O c1(C(=O)NCCN(C(C2C(C#C)C2)=O)CCC)cc(C)c(Br)cc1C C1(CNC(c2cc(CCC)n(C)n2)=O)CC2CN(C(=O)C=Cc3cscn3)CC12 C(=O)(CCN=[N+]=[N-])N(C1CCCC1)CC(=O)NC(C)Cc1cccs1 CCC(CC)(CC(=O)NC(=O)C(C)CC(F)F)C(=O)N1CC2CC3CC2C1C3 C1(C)(CNC(C(C(C)C)O)=O)CN(C(=O)CCc2cccc(O)n2)CCO1 C12CCC(C1)NC(=O)CC2.C1(COC)CCN1C(=O)CN1CCCC1 N1(C(c2ncc(C)nc2)=O)CC(NC(=O)CC(C)(C)C(F)(F)F)C2(CCCC2)C1 C1(CC=C)(NC(=O)C(C)C2CC2)CC2CCC(C1)N2C(=O)C=CCF C1(CCC(=O)NC2C(NC(C3(OC(C)C)CCC3)=O)C2)CCc2ccccc2C1 c1(C(=O)NC2(C3CN(C(C4CCCC(OC)C4)=O)C3)CC2)c(N)ccc(F)c1C N1(C(C(CC(C)=O)(C)C)=O)CCC2C(CCCN2C(c2coc(CO)c2)=O)C1 c1(CN2CC(CN(C(COCCC)=O)C)OCC2)ccc(F)cc1F C1(NC(C(c2cccnc2)OC)=O)CCC(NC(c2coc(C)n2)=O)C1 C(=O)(CC1OCc2ncccc21)NC(CCCNC(C=C1CCC(C)CC1)=O)C c1ccc2cc(Cl)cnc2n1.CC1CCCNC1Cn1cccn1 C(=O)(C(F)(F)C(F)F)NC(C)CNC(c1ccc(NC2CC2)nc1)=O O=C1NCC2(CO1)CN(C(=O)CC1(C)CCN1C(C1CC3CCC3C1)=O)C2 N1(C(c2c(CC)onc2C)=O)CCC2C(CCCN2C(=O)Cc2cnccn2)C1 C(=O)(C(CCCC(C)C)N1CCCC1CC(c1cnn(C)c1)O)NC(CC)C C1(CC(=O)NCC(C)NC(=O)C(C)(C)N(C)C)CC1C1CC1 N1(C(=O)NCCCC(C(F)F)c2ccccc2)CCOCC(C(F)(F)F)C1 C(=O)(C(CCC)C(=O)OC)NC1C(C(=O)NC(c2cnn(C)c2)CC)OCC1 c1(C(=O)NCC(CC)NC(=O)C(C2CC2)OC)cnc(O)c(C(C)=NO)c1 N#Cc1cccc(NC(=O)CC2CCCN2Cc2ccc(F)c(O)c2)c1Cl c1(SC)nc(NC(C2CCC2(C2CC2)NC(=O)OC(C)(C)C)=O)sc1C n1(C(C)C)nc(-c2cnn(CCO)c2)nc1C1CCN(C)C1=O CC1CN(C(=O)C(=O)Nc2ccc(CN3CCOCC3)cc2)C(C)(C)C1 C1(CNC(c2cc(C)n(C3CC3)n2)=O)CN(C(C2C=CC=CC=C2)=O)CCCO1 C1(NC(CCc2ccn(C)n2)=O)CCCCC1CNC(=O)CC1CCCCC1O C(=O)(C#CC1(C)COC1)N(CC(C)C)CC(=O)N(C)C(C1CCCC1)C Cc1nc(C)n(CC(=O)NCC2CCN(C(c3ccc(CC(C)C)nc3)=O)C2)n1 C(CCCC(=O)NC1CC1NC(=O)CC1CC2(CC2)CO1)OCC CC(CN=CC#N)NCC1CCCSC1 C(=O)(C1CCCn2nccc21)NCC(C)N(C(c1ccc(F)c(O)c1F)=O)CC C1(CNC(c2n(CC)cc(Br)c2)=O)(NC(=O)CN(C)C)CC2CCC1CC2 c1(OC(C)C)ccc(C(N2CCCC2C(C)NC(c2c[nH]nc2C)=O)=O)cc1F N1(C(=O)C2CC2)CC2CC3CC(C2)CC1C3.N1(C(=O)O)CC(N(C(C)(C)C)CCO)C1 C1(C(N(CC(C)CNC(C2CCCC23CCC3)=O)C)=O)CNC2=C1CCCC2 C1(C(=O)N(C)CC2CC(F)CN2C(=O)CCN2CCC2)CCC(=C2CCC2)CC1 N1(C(CC(=C)C)=O)CCCC2C(NC(C3CC4(CSC4)C3)=O)C(C)(C)C12 C1(NC(C2CCC(F)C2)=O)CC2(CCN(C(=O)CCc3ccc(F)cc3Cl)C2)C1 c1(C(=O)NCC(CC)N(C)C(C2CC2(C)C)=O)coc(C2CCC2)n1 C(=O)(CCC1CCc2ccccc21)NCC1(C)CCCN1C(C1OCCO1)=O Cc1cc(F)c(NC(C2(C)CCN2C(c2cc(O)c(O)c(O)c2)=O)=O)cc1Br N1(C(C2CC(=O)NC2)=O)CC(C2CN(C(=O)CC3CCNC(=O)C3)C2)C1 Cc1ncc(Cl)cc1C(=O)NC1(CO)CCN(C(=O)C2=COCCC2)CC1 CC1CN(C(C2(CCO)CC2)=O)CC(CCNC(c2n[nH]cc2Cl)=O)O1 Cc1c(C(c2nnnn2CC2CCOC2)NC2C=CCC2)cnn1C c1(C(N(C)Cc2n(CC)cnn2)C)ccc(F)c(F)c1F.c12cn(nn1)C2 C(=O)(CCCC(F)F)N1CC2C(NC(=O)Cn3cncn3)(C2)C1 c1(C(N2CCCC(C(C)Nc3nc(C)cc(C)n3)C2)=O)ccc(C)c(Br)c1C C(N=C(NCCF)NC(C)(C)C(=O)NC)C1(CC=C)CC1 c1(NC(C2(C)CCCCC2)c2n(CC)nnn2)cnnc(S(C)(=O)=O)c1 CCC(C(=O)NC(c1ccc(O)cc1)CNC(=O)COCCN(C)C)C(C)O c1(C(=O)NC(CC=C)CNC(c2cc(C)co2)=O)ncc(C2CC2)cc1F C(C(CNC(C1CCCN1CCC(C)C)=O)C(F)(F)F)NC(C(C=C)O)=O c1(C(N(C2CCC(CNC(c3cc(Cl)cn3C)=O)CC2)C)=O)cc2n(c1)CCC2 c1(C(=O)NC(C2CCN(C(c3c(C)nc(CC)o3)=O)C2)C)cc([N+](=O)[O-])oc1C c1(C(C)(C)C)cccc(C(=O)NC2(C)CC(NC(C3CCC(O)C3)=O)C2)n1 C1(C(=O)NCCc2cn(CC)nn2)C(C2CC2)CCN1C(c1n[nH]c(=N)[nH]1)=O C1(CN(C(=O)CC2(O)CCC2)C)CCCCN1C(=O)CSC(F)(F)F N1(C(c2csc(C)c2C)=O)CC2(CCN(C(=O)C(C)(C)c3sccc3Cl)C2)C1 C1(N(C(CC(C)N(C)C)=O)C(C2CC2)=CCF)CCN(C(=O)C2=CCSC2)CC1 c1(OC(CCC(=O)N(CC(CC)NC(=O)COC(C)C)C)=O)ccccc1C C=CCCCCC(=O)N(C1CCCN(C(c2csc(C(F)F)c2)=O)C1)CCF C(=O)(N=c1cc[nH]c(CCO)c1)C1SCCN(Cc2cc(C#N)cc(Cl)c2)C1 c1(C(N2CCC(C(N3CCC(O)C3)=O)C2)=O)cccc(Br)c1Br c1(C(N2CCOCC2CCC#N)C(=O)NCCC#N)cccc2c1nnn2C c1(C(N2CCC3CC3C2)=O)cc(I)c2nccnc2c1 C(=O)(C(CCOCCO)NC(=O)CCc1cscn1)N(CCOC)C CC(C)CC(CC(=O)NC1COCC1C(N)=O)NC(C1CC1(Cl)Cl)=O Cc1sc(O)nc1C(=O)NC1CC(C(=O)NC(C)CCC(C)C)C1 C(CCC(C)C(=O)N1CC(C(C)NC(C2C=C2C)=O)C1)OC C1(N(C)C)(C(=O)NCC(CO)NC(C2CC(=C3CCC3)C2)=O)CCC1 c1(OC)ccc(F)c(C(=O)NC(CNC(c2cc(Cl)cc(Cl)c2)=O)CO)c1N C(CCC(O)C(=O)NCC1(CN=[N+]=[N-])CC1)NC(c1cnn(C)c1Cl)=O C1(O)(CNC(c2cnc(C(C)OC)s2)=O)CCN(C(C2(OC)CCSCC2)=O)C1 C12(C(=O)NCCN(CCCN(C)C)C(c3ccc(F)cc3F)=O)CC1COC2(C)C N1(C(c2c(OC)ccnc2)=O)CC(C)(C)CC1CNC(=O)C(O)Cc1cnc[nH]1 CC1CN(C(c2cccc(O)n2)=O)CCC1CNC(=O)CC(C)(C)C1CC1 C1(C(=O)NCC#CCC)C(CC)CCN1C(=O)C(C)OCC(C)C C1(CS(=O)(=O)NC(CSC)=O)(Cn2nccn2)CCCC(=O)N1 C(=O)(CC1=CCN(C)CC1)NC1CN(C(C=C(COC)C)=O)C(C)CC1 N1(C(C2(C)N(C)CC2)=O)CCCC(CC(=O)NCCC2CC(C)(C)C2)C1 c1(OC)cc(C(=O)NC2(C)CCCN(C(c3ccc(C)nc3)=O)C2)cc(Br)c1 Nc1ncccc1C(=O)NCCCCCCNC(C1(CC(F)F)CCC1)=O n1(CCOC)cc(C(=O)NC2CN(C(c3csnc3C)=O)CC2O)c(=O)cc1C c1(C(N2CC(C(N)=O)OC(C)C2)C(=O)NCC)c(F)cc(Br)cc1F c1(OC)ccc(S(=O)(=O)N2CCN(C3CC4CCCCCC34)CC2)cc1C(C)C C1(NC(C2ON=C(C)C2)=O)CC2CCC(C1)N2C(=O)C=CC1CCCC1 c1(C(=O)NCCC2CCC(NC(C3CCC=CCC3)=O)C2)ccnn2ccnc12 C1(CC)CN(C(c2ccc(F)cc2)=O)CCN1C(c1cc2ccsc2s1)=O c1(CC)ccnc(C(=O)NCc2cc(NC(N)=O)no2)c1.N12CCCC(C1)C2=O CCCC(F)(F)C(=O)N(CCC(=O)NC(C(F)F)C1CC1)CC1CC1 c1(NC(C(=O)NCCC2CCC(S(C)(=O)=O)CC2)=O)cc(N)ccc1S(N)(=O)=O CC(C)CCCCC(=O)N1CC2(CO)CC1(C(=O)NCC1(O)CC=CC1)C2 c1(CC(C(=O)N(C2CCN(C(c3cnc(OC)s3)=O)C2)CC)O)ccc(F)cc1 c1(N2C(NCCNC(CC3C(=O)NC(=N)S3)=O)CCC2)ncnc2c1CCO2 C1(C(=O)NCC2CN(C)C(=O)C2)CN(C(=O)C#CC2CCC2)CC12CC2 c1(NC(C(C(C)C)NC=O)=O)cccc(C#CCO)c1.C12CN(CC1O)C2=O C1(CNC(c2ccc(Cl)o2)=O)CCCC2CN(C(C3CCC4(CCC4)O3)=O)CC12 c1(C(=O)NC(C)CCN(C)C(C2CCCCS2)=O)cccc2ccsc12 c1(CC(=O)Nc2c(C(=O)OCC)nc[nH]2)csc(=NCc2cc(F)cnc2Cl)[nH]1 C1(C)(N)CN2CCC1CC2.c1(CC)nocc1C(C(=O)CCOC1COC1)=O C=CCCCCC(=O)N(C)CCN(C)C(c1ccc(C(=O)OC)c(C)n1)=O C1(C(=O)NCC2C(NC(c3cnc(O)c(Cl)c3)=O)C2)CC(C2CC2)=NO1 C1(C(=O)NCC(C)(C)OCCNC(C(CSC)C)=O)CC(C)CCO1 C1(C)(NC(C)C(C(=O)OC(C)(C)C)N(C)C)CCC(C)(C)CC1 Cc1cc(N)ccc1C(=O)NC1CN(C(=O)CC2CCCCN2C)CC1C C=CC(C)(O)CC(=O)NCC(C)CN(C)C(c1sc(C(=O)OCC)nc1C)=O c1(C(=O)NC(C(N2CC(C(=O)OC)C2)=O)C2CCCC2)c(F)cc(Br)c(F)c1F C(=O)(C(C)N(OC)C(=O)c1ccc(CNC(c2cc(C(C)=O)c[nH]2)=O)cn1)OC CC(C)(O)C(F)(F)C(=O)NCC1(F)CC(NC(c2csc(-c3cccs3)n2)=O)C1 N1(C(c2n(CC)ncn2)=O)CC(NC(=O)CC2C=CS(=O)(=O)C2)C(C2CC2)C1 C1(C(c2ccc(OC(C)C)s2)=O)CN(C)CC(C)O1 CN=c1[nH]cc(C(N2CC(NC(=O)C=CC(c3ccccc3)=O)C(O)C2)=O)o1 C1(CC(=O)NCC=CBr)CCCC(NC(=O)CC2CCOCC2)C1 C1(CNC(=O)C(O)CCl)OCC2CCN(C(=O)C(F)F)CC12 c1(CC)ccc(CC(=O)NC(C)CCNC(c2ccc(F)o2)=O)cc1F N1(CC)CCN(C(=O)CC2C=CCN2C(C2CCO2)=O)CC1.C(=O)(OCC)O C1(NC(C2CC2C(F)F)=O)CCC2(CC1)CN(C(C1CC13CCCC3)=O)CCO2 C(=O)(C1=C(CC)OCCC1)N1C(CCC)CN(C(C2COCCN2CC)=O)CC1 CC(C)C(C(=O)NC1(CNC(C2C(Cl)(Cl)C23CC3)=O)CC1)n1cnnc1 C1(CNC(C2(C)C=CCCC2)=O)CCCCCN1C(c1ccc[nH]1)=O c1(C(C)=O)cc([N+](=O)[O-])ccc1NCCC1CC(NC(C2CC23CCOC3)=O)C1 c1(OC)cnc(F)c(C(=O)NCCCC(C)NC(=O)C(C)(C(C)C)OC)c1 C1(C(=O)OC)CN(Cc2c(C)noc2C)CC1(C)C.c1(C(=O)N)ccn(C2CC2)n1 c1(C(=O)NC2CC3CN(C(C(C)(O)C4CCC4)=O)C2C3)ccn2ncnc2c1 c1(NC)nc(OC(c2c(Nc3ccc(Cl)c(C(C)O)c3)c[nH]n2)=O)ncc1Br N1(C(c2c(C(C)C)cccc2)=O)CCCC(NC(C2CCC(=O)N2C)=O)C1C N1(C(CNC(CNC(C)=O)=O)=O)CC(NC(c2ccc(C)nn2)=O)C(F)C1 c1(C(C(=O)NCC(=C)C)N(CCC(C)C)C(C)(C)C)cc2ccnc(Cl)c2s1 C1(NC(c2nc(Cl)ccc2F)=O)CN(C(c2ccns2)=O)CC1C1CC1 C1(C(=O)NCCNC(c2cn(CC=C)nc2)=O)CC2CCC(C1)C2O C1(O)(CNC(CCOCC(C)C)=O)CCN(C(C2CCCC23CCC3)=O)CC1 C(CCC(F)(F)F)(C(=O)Nc1nn[nH]n1)NC(=O)CCN1CCCC1 C12(C(=O)NC3(CNC(C(C(C)(C)C)O)=O)CCOC3)CCC(C(N)=O)(CC1)CC2 c1(C(=O)NC(CCNC(C2(OC)CC2)=O)C)cc(Cl)cc(Cl)c1[N+](=O)[O-] N1(C(C(OCC)OC)=O)CCN(C(c2ccc(N)cc2C(F)(F)F)=O)C(C)C1C C1(C(=O)NCc2csnc2C)(NC(CN(C)CC)=O)CCSC1 Cn1nc(-c2cn(CC(N3CCC(CC4CCCC(=O)N4)C3)=O)nn2)cc1N C1(OC)CCNCC1C(=O)NCC(O)CC(O)c1ccccc1 c1(CN2C(C)(C(=O)Nc3cccc(NC(=O)OC)c3)CC2)cc(F)c(F)c(F)c1 c1(OC)ncc(C(N2CCCS(=O)c3ccccc32)=O)c2ccccc12 C(CC1CC1)(C(=O)NCC(O)CCNC(c1csc(CCP(C)(C)=O)n1)=O)OC Cc1cc(Cl)cc(Br)c1NC(C1CC(F)(F)CN1Cc1cc(Br)cc(Cl)c1F)=O C1(NC(C2CCCN(C(C)C)C2)=O)CC2(CCN(C(c3cc(=O)cc[nH]3)=O)C2)C1 C(C)(C)(CC(F)C(=O)NCC1CCCN1C(N)=O)NC(C1=NOC(C)C1)=O N1(C(C2CC(=C)C2)=O)CCOCC1CCCNC(c1cc(OC(C)C)ncn1)=O Cc1ccc(N)c(C(=O)NC2CC(O)CN(C(C34CSC(C3)C4)=O)C2)c1F C1(COC)CC(CNC(=O)C(F)C(C)C)N(C(=O)CCc2ccccc2)C1 N1(C(COCCN(C)C)=O)C(CNC(=O)Cc2cnn(C)c2)CC2COCC12 N1(C(C(C)C)=O)CCN(C2CCN(C(c3cccc(O)n3)=O)CC2)CC1 c1(OC)ccc(Cl)cc1C(=O)NC1CC2(C1)CC2NC(c1[nH]c(C)nc1C)=O CCC1CC(=O)N2CC=CC2(C)C(=O)N2CCC(CC2)C1.C1(C2CC2)CC1 N1(C(C(C(C)C)NC(C)=O)=O)CCC(C2CN(C(c3nnccc3C)=O)C2)CC1 c1(-c2n(CC)nc(-c3cc(OC)ccn3)n2)nccc2ccccc12 c1(C(=O)NCC(C2CC2)NC(=O)CC2COCCO2)c[nH]nc1[N+](=O)[O-] CC1=C(C(=O)NCC2CCN2C(c2cnc3n2CCCC3C)=O)S(=O)(=O)CCO1 c1(OC)cccc(C(N2CC(C(O)C(=O)NC3CC4C=CC3C4)C2)=O)c1 Cc1ccc(C(=O)N(C2CC(C(=O)NCc3cnccc3Cl)C2)C)cc1F C1(CC(=O)N(C2CCN(C(c3cc(C)n(C(C)C)n3)=O)C2)CC)CC2CCC1C2 CCC(CCC(=O)N1CC(CNC(c2ccc(CO)cn2)=O)(OC)C1)OC CCCC(C(=O)N1CC(CC(=O)N(CC(C)C(C)C)C)C1)OCC C1(C(=O)NC(c2ccncn2)(C)C)CCCN(C(=O)C=C2CCCCC2)C1 CC1CCC(C(=O)NCC23CC(CN2C(C2CCS2(=O)=O)=O)C3)CC1 C1(NC(c2ccn(CC)n2)=O)CN(C(C2CCN(C)C2C)=O)CC12CC2 CN(C1C(=O)Nc2ccc(C)cc21)CCNC(=O)NC1CC2CCCCN2C1 CC(CC(=O)NC1(C2CCCN2C(=O)CN2CCCC2=O)CC1)c1cccnc1 C1(OC)CC(NC(=O)CCc2ccoc2)CN(C(c2coc(C(F)(F)F)c2)=O)C1 c1(C(=O)NCC2(NC(C(CC(C)C)O)=O)CCC2)cc2c(s1)CCC2=O C(CC(C)N=c1[nH]c(N2CCCCCCCC2)nc2ncn(C)c12)OC C=CCC(C(=O)NCCCCCNC(c1ccnc(OC)c1)=O)C(C)C Cc1coc(C)c1C(=O)NCC12CC(NC(C3CC3(F)F)=O)(CO1)C2 C12(NC(c3ccc(CSCC)cc3)=O)CCC(CC1n1cc(CC(C)(C)O)nn1)C2 c1(C(N2CCCC(C(=O)NCc3ccncc3)C2)=O)c(O)c(Cl)cc(Cl)c1Cl S(=O)(=O)(c1cccs1)NC(C(c1cc(OC)ncc1)N1CCC(N(C)C)CC1)=O C#CC1CCCC(CNC(C2C=CCN(C(C3(n4cccc4)CC3)=O)C2)=O)C1 C(C(C)(C)C1=CCC(C)(C)CC1)N(C(CCC(=C)C)C(=O)NC1COC1)C N1(C(CNC(=O)OC)=O)CCC2C(C1)NC(=O)CN2C(C1CCC12CCC2)=O CN=c1[nH]c(=NCc2cc(CO)cs2)[nH]c(=NC2CC2c2cccc(F)c2F)[nH]1 c1(C(N2CC3CC(CNC(C45CC(CO4)C5)=O)C3C2)=O)c(F)ccc(F)c1F N1(C(C(n2c(C)ncc2)C)=O)CC(C(N2CC3CC3(CO)C2)=O)C(C)C1 C1(c2c(C)cccc2)CN(C(=NCC2CC2(F)F)NCC(F)F)CCO1 c1(C(=O)NCCCCN(C(C2CN(CC)C(=O)C2)=O)C)cc(COC)nc(O)c1 CP(C)(=O)c1cnn(CC(=O)NCC(C)(C2CC2)NC(c2sccc2Cl)=O)c1 C1(CNC(CSCCOC)=O)CN(C(C2CC2Br)=O)CC(C)(C)C1 c1(CC(=O)N(C(CC)COC)C)ccnc(O)c1 C(CC(C(C)(C)C)NC(c1cc2ccsc2s1)=O)N(C)C(c1cc(O)n(C)n1)=O C(=O)(C(=O)C(C)C)N1CC(OCC)(CNC(=O)C(C)O)C1 C1(NC(c2cnc(OC)s2)=O)CCC12CCCN(C(=O)CSCCN(C)C)C2 N1(C(CC2CCN(Cc3c(Cl)ccc(C)c3)C2)=O)CC(F)(F)C(F)(F)C1 C(=O)(C1=NOC2(CCOC2)C1)NC(CNC(c1ccn(C)c(=O)c1)=O)C1CC1 N1(C(C(C)c2cc[nH]n2)=O)CC2CC(C1)N2C(=O)CC1CCCSC1 c1(C(=O)NC2CN(C(c3c(C)nsc3C)=O)CC2O)cccc(Cl)c1[N+](=O)[O-] C(CCF)(C(=O)OC)NC(CSCCC)=O.C1=CCNC1=O.C1CC1 Cc1cc(=NCc2cccc(Cl)c2[N+](=O)[O-])[nH]cc1Br C#CC1(N(C)C(C2(C(C)NC(C3CCCCC3C)=O)CC2)=O)CCCCCC1 c1(NC(C2(F)CCCN(C(c3cccc(C)c3Cl)=O)C2)=O)ccc2ncoc2c1 C1(C(=O)NC2(C(N(CCCOCC(F)F)C)=O)CC2)OCCCC1O N1(C(C(CCC)C(C)C)=O)CCC2(CCCN2C(c2cn(C)nc2OC)=O)CC1 N1(C(c2nc(COC)sc2C)=O)CC2CN(C(=O)CCCC(C)C)CC2C1 CCC(C)C(C(=O)NCC(CCNC(C1(COC)CC(=O)C1)=O)OC)OC C#CCCCCC(=O)NC1CC(NC(=O)C(C(C)C)n2cnnn2)C1 C1(CC(=O)NCCN(C(=O)COc2nc(O)nc(O)n2)C)CCC2CC1C2(C)C N1(CC(C(=O)NC2C(NC(C(C)(C)F)=O)CCC2)(C)O)Cc2ccccc2C1 c1(C(=O)NCC2CCCN2C(c2cnc3sccn23)=O)noc2c1CCCCC2 N1(C(c2ccccc2)C#C)CC(CSC2(S(=O)(=O)N(C)C)CC2)CCC1=O CCC1=C(C(=O)NCCC(C)NC(=O)C(c2cc(Cl)ccc2F)(C)C)SCCO1 N1(C(C(CC)OCC)=O)CCn2ncc(CNC(=O)C(C(C)C)NC(C)=O)c2C1 C1(C(N2C(C)(C(=O)NC)CCC2)=O)CCN(C(=O)C=CCN2CCCC2)C(C)(C)C1 CC1(C(=O)NC2C=CCN(C(=O)C3=C(Cl)CCOC3)C2)CC(C2CC2)=NO1 c1(N2CC(C(C)NC(c3ccc(CCC)[nH]3)=O)OCC2)ccc2nccnc2n1 c1(CNC(C(C2CCCO2)NC(=O)OC(C)(C)C)=O)cccc(C#N)n1 CC(C(=O)NOCC(N1CCCC(CCC(N)=O)C1)=O)CC(C)(C)C CCCC(C)(CCC)C(=O)N1CCCOC(CNC(C2OCCC2C)=O)C1 C(CC(C(=O)NCC1CCOC1)N1CCC(c2cnco2)C1)SC c1(CC(C2CCN(Cc3cccc(Cl)c3)CC2)C)ccc2c(c1)CCC2 N1(C(C2(C)CCC(C)C2)=O)CC2(C1)CN(Cc1csc(O)n1)C2 O=C1CC(CC(=O)NCC(O)CNC(C2C3CC(F)(F)CC23)=O)CCCN1 C#Cc1cn(C)nc1C(=O)NC(C(=O)NOCC1CC2C=CC1C2)C1CCC1 c1(C(N2C(C)(CNC(=O)C(O)C(F)(F)F)CCC2)=O)cnn2c1OCCC2 C1CN=C2C=C(N=C(c3ccco3)N2)NC1.N1(CCSCC)CCC(C)CC1 c1(C(=O)NC(C)(C)CNC(c2ccc(Cl)o2)=O)ccc2c(C#N)c[nH]c2c1 c1(C(C)(C)C)cc2c(NC(c3cc(Cl)sc3Cl)=O)ncnc2s1 c1(OC)c[nH]c(C(=O)NCC2CN(C(=O)C(C)N(C)C(C)=O)CC2C)cc1=O C=C1CC2(C1)CC(C(=O)NCC(C)NC(=O)CC1SC(=N)NC1=O)C2 Cc1cc(N)c(C(=O)NCC2(F)CCCN(C(=O)CC(F)(F)C(C)C)C2)nc1C c1(OCCOCC)cc(N(C)CCN(C(=O)CS(N)(=O)=O)C)nc(C)n1 c1(C(=O)NC2CCCN(C(C3CC(CCC)C3)=O)C2C)sc2nnc(S)n2c1C c1(CC(=O)C(=O)C2CC2)ccc(O)cc1.C1(CC(N2CCC(N)C2)=O)C=CS(=O)(=O)C1 c1(OC)ncc(-c2cncc(C(C)C)c2)cc1-c1ccnc(C)c1 C1(NC(C(CC)C(C)O)=O)CCCCC12CCCN(C(c1cn(C)cc1C)=O)C2 C(CCC(C)CC)(C(=O)Nc1ccccc1)N1CCN(CCCC)C(=O)C1 C#Cc1ccc(C(=O)NCC(C(=O)NCC(C)(COC)CC)C(C)C)cn1 CC1C(C(=O)NC(CO)C(N)=O)CCN1C(c1nc(=N)cc[nH]1)=O c1(C(C(N2CCC(NC(CCS(C)=O)=O)CC2)=O)O)ccc(F)cc1F CC(C)CCCC(=O)N1CC(F)CC1CNC(C1CCN(c2ccncc2)C1)=O C1(NC(c2nn(C)c(C#N)c2)=O)CCC2(CC1)CN(C(C1CC1(C)C)=O)CCO2 n1(CC(=O)NCCCOC(C)C)cc(CCN)nn1.C1CC1 C12(NC(c3c(Cl)cn(C)n3)=O)CCN(C(C3(C)CCCCC3)=O)CC1C2 c1(C(=O)NCC(c2ccccc2)NC(=O)CC2(O)CCC2)nnc2n1CCCCC2 C1(C)(CCC)CCN1C(=O)CCCC1(NC(=O)OC(C)(C)C)CCC1 N(C1COc2ccccc21)C(C(=O)Nc1nc(-c2cc[nH]n2)cs1)=O c1(C(C(=O)NCC2(C)CCCC2NC(=O)CC2CC2)N(C)C)ccc(F)c(F)c1 C(=O)(CC(C)C(F)(F)F)NC(c1cc(C)on1)C(N1CCCC(C#N)C1)=O C=CCCC(C(=O)NCC1(C(N)=O)CC1)NC(c1cnn[nH]1)=O N1(C(c2c(OC)nccn2)=O)CC2(CCN(CC(O)C(C3CC3)OC)C2)C1 c1(C(=O)NC2(CCCC(=O)NCC3ON=C(C)C3)CCC2)ccc(C#N)c(C)c1 c1(C(N(CCCN(C(=O)C(F)CC2CCCC2)C)C)=O)cc(N)c(O)c(F)c1 N(C1CCCc2n[nH]cc21)C(=O)Cc1csc(N2CCCCC2)n1 CC1CCC(C(=O)NC(Cc2ccco2)C(=O)NC2CC(CO)C3CC23)CC1 N1(C(c2c(C)con2)=O)CCCC(NC(=O)C(O)Cc2ccccn2)CC1 C(C(C)C(F)C(=O)NC1CC1c1cncs1)NC(Cn1c(CC)ncc1)=O CC(CN(n1cncn1)C)N=c1[nH]c(Sc2ccncc2)nc2c1CCCCC2 c1(CC)ccc(C(=O)NC(CNC(C2(c3ccsc3)CC2)=O)C2CC2)o1 C(CCCC(=O)NCC1CN(C(c2nccn2C)=O)CCO1)OC C1(C(=O)NCC(C)NC(C(C)SC(C)C)=O)CCCSC1 c1(OC)ccc([N+](=O)[O-])c(NCCNC(=O)NC2(C)CCCO2)c1F c1(NC(CN(CC#C)C(C2(CCNC(=O)OC)CC2)=O)=O)ccc(Cl)nc1 c1(-c2ccc(CNC(C3(C)CC(OC)(OC)C3)=O)cc2)cccc([N+](=O)[O-])c1 C1(N(C(C(F)=CCC)=O)C)CCCC2CN(C(c3ccc(Cl)cc3)=O)CC12 c1(N(CCN(C(C(F)OC)=O)CCCN(C)C)C(C2CCCC2)=O)ccc(Cl)cc1 n1(CCCC)nc(C)c(C(=O)N(C2C3CN(C(=O)C4=CCCC4C)CC23)C)c1C C(=O)(C(CNC(C1CN(C2CCC2)C1)=O)C(C)(C)C)N(C)CC1(OC)CCC1 c1(C(N2CCC(C)(CNC(=O)CC3CC(F)C3)C2)=O)[nH]nc2ncc(Br)cc12 C(=O)(C(O)C(C)(C)CO)N(CCN(C)C(c1ccc(N(C)C)cc1)=O)C C1(F)(CNC(C2(C)CN(C)C(=O)C2)=O)COCCN(C(=O)C=C2CCOCC2)C1 CC(C)CCC(F)C(=O)NC(C)CCCCNC(=O)CC1CC(=O)NC1=O N1(C(C(C)N2CCC2)=O)CCCC1CNC(c1csc(-c2ncccn2)n1)=O Cc1nc(C2CC2)sc1C(=O)NCc1ccccc1CNC(C1CCC(=O)O1)=O Cc1c(Cl)ccc(C(N2CCCC2CN(C)C(c2ncnn2C)=O)=O)c1N Cc1cccc2[nH]cc(C(=O)NC3(CNC(c4nc(Cl)cs4)=O)CCOC3)c12 Cc1cccc(-c2ccc(NC(N3CC(C(=O)Nc4ccncc4F)C3)=O)nc2)c1 C1(NC(C23CCC(OC)C2C3)=O)COCCN(C(=O)C=C(C)C2CC2)C1 C(=O)(CC(CN(C)C)C(F)F)NC(C(C)NC(=O)CCc1ccon1)CO c1(C(=O)NCCC(C)NC(C2CN3CCCC3CO2)=O)oc2ccccc2c1Cl c1(C(N2C(CCNC(C34CC(OC)C3C4)=O)CCCC2)=O)ccc2n[nH]cc2c1 N1(N2CCNCC2)CCC(F)(CNC(N2CCC(C(=O)CC)CC2)=O)CC1.CS CCCCC(CC)C(=O)NCC12OCC(C(=O)OC)(C1)C2.C(=O)(C1=CC2CCCC12)N C(CCN(C)C(c1sccc1SC(F)F)=O)(C(C)C)NC(c1c(OC)scc1)=O C1(C(N2CCCC(CF)C2)=O)C2CCC(C2)N1C(c1ccc(C2CC2)cc1)=O N1(C(c2cncc(OC)n2)=O)CC(O)CCC1C(=O)NC1(C)CCCC1C C1(CC(=O)NCC2CCC(F)(CNC(c3ccc(O)nn3)=O)C2)CCS(=O)(=O)C1 N1(C(CC(CCC)CC)=O)CCC2(CCC2)C(NC(C2C(C)(C)C2(C)C)=O)C1 n1(C(C)C)ccc(=NC(c2cncc(F)c2)C2CC(c3ccccc3)C2)nc1O C1(NC(c2scc(C)n2)=O)CC2CN(C(=O)Cc3cnc(C)s3)CC12 CC1CC(NC(=O)Cn2nnn(-c3cccs3)c2=O)CN1C(c1coc(Cl)c1)=O CC(C(C)C(=O)NCCOCCOCCNC(C1CC(CF)C1)=O)S(C)(=O)=O C(=O)(C#CC(C)(C)O)N1CCC(C(C(=O)NCC(COC)(C)O)C)CC1 N(C(=NCCOCCC(C)C)NCc1ccccc1)CCSc1ccc(C)o1 C1(C(=O)NC2(C)CC(NC(Cn3ncc(C)c3)=O)C2)OC2CCC1C2 c1(COC(C(C)(C)c2cnco2)=O)ccc(I)cc1 c1(C(=O)NCCOC2CN(C(C3CC(=C)C3)=O)C2)cc(Br)c(C)s1 C1(CC(=O)NCCC(F)(F)F)(C(=O)NCCCN(CCCOCC)C)CCCC1 c1(C2CCN(C(C(=O)NC(CC)(C)C)C3CC3)C2)ccccc1F c1(C(=O)NC2CC(OCC(=O)NCC(CC)(C)O)C2)cnnc(C)c1 CC(CC(=O)NCC=CCNC(=O)C(C)Oc1ccc(Cl)c(Cl)c1)CC(C)(C)C c1(C(N2C(CN(C(=O)CN(C)C(N)=O)CC)CCC2)=O)cccc2c1nnn2C N1(C(CC(CC)C(C)C)=O)CCC2CCC(C1)N2C(=O)CN1CC2C=CC1C2 c1(C(N2CC3OCC(C(=O)O)C3C2)=O)ccc2c(c1)NCCC2 C(C(C(=O)NCCc1ccc(C)nc1)C(F)(F)F)c1ccc(OC)cc1 c1(OCC(=O)NCCN(C(=O)C=C2CCCC2)CCOC)cnn(C)c1 C1(NC(c2cnsn2)=O)CC2(C1)CC2C(=O)NCC1CC1(F)F C(=O)(C(O)C1=CCCCC1)N1CCN(C(C23C(C)(C)OCC2C3)=O)CC(O)C1 Cc1c[nH]nc1CNC(=O)CCOCCNC(=O)CNC=O.C1(C)CC1 C1(NC(=O)NC(c2ccccc2)C2(C(C)(F)F)CCC2)CCOC2(CCCC2)C1 c1(C(N2C(C)CC(CN)C2C)=O)cc(F)c2ccccc2c1 c1(C(N(C(CNC(C(C)=NOCC#N)=O)C)C)=O)ccc2cnn(C)c2c1 C1(C(=O)NCC(=O)N(CCOC)C)CC12CC2.C(=O)(CO)NCC(F)F C1(NC(=O)CCn2ccnc2)CN(C(c2c(F)cccc2Cl)=O)C2CCCCC12 Cn1ncc(C2CC2)c1C(N1CC(CNC(C2COCCO2)=O)C(O)C1)=O CCC1C(C)CN1.N1(C(C)=O)CCC(O)(C(Cl)(Cl)Cl)C1 C(O)(CCc1ncc(C)o1)(C(F)(F)F)C1N(CC2CCC2)CCOC1 N1(C(Cc2n(C)nnc2)=O)CCN(C(=O)C=Cc2nccs2)C(CC2CC2)C1 C1(NC(=O)C=CC=C(Cl)Cl)CC2(C1)CC2Nc1ncc(I)cn1 c1(C(=O)NCC(C)CN(C(=O)C(C)n2ccnn2)C)cccc(C(C)(C)C)c1 Cc1ccc(Cl)cc1NC(c1ncoc1CNC(c1cncc(Cl)c1)=O)=O C(=O)(C(C)(C)c1csc(-c2ccccc2)n1)NCC(C)N(C(=O)CSC1CC1)C CCC(CC(=O)NC1CC(CO)N(C(C2CC(CF)C2)=O)C1)C1CC1 C1(NC(c2ncc(N(C)C)nc2)=O)CC2CC1CN2C(=O)CCc1cc[nH]n1 N1(C(Cc2cnc(C)s2)=O)CCCC(NC(C2CC3(F)CC2C3)=O)C1 CC1CN(C(=O)COCCF)CC1C(=O)NC(C)(C)C(F)F C(=O)(CC1=CCN(C)CC1)N1CCN(C(C(C=CCCC)O)=O)CC1COC CC(C(C)C(=O)N(C1CC1)Cc1nc[nH]n1)NC(=O)CC1C=CCC1 c1(NC(c2n(CCC)nnn2)(C)CCCl)ccc(Cl)c(CC2CCCO2)c1 N1(C(C2CCC(CNC(C(C)C)=O)O2)=O)CC2CC3CC2C1C3 C1(CNC(=O)CC2CCC2)(NC(=O)C(F)=CCCC(F)(F)F)CCOCC1 C1(NC(C(C)SC)=O)CC1C1CCCN(c2ncnc(C)c2F)C1 c1(C(=O)NC2C(C(=O)NCCc3c(Cl)cccc3Cl)C2)cccc2sccc12 C(N=c1[nH]c(=NCC2CC=CC2)[nH]c2c1CCC2)c1cn(C(C)(C)C)nc1 C(CCC(O)C(=O)Nc1cnsc1)NC(c1c(CC)nccn1)=O Cc1c(C(=O)NCCN(C(c2cnn[nH]2)=O)C(C)C)nnn1-c1ccccc1F S(=O)(=O)(c1ccc(Cl)cc1-c1cccs1)NC(C1CCOC(C)(C)C1)CC C1(C(N(CCCC)C2CC2)=O)CN(C(=O)CC(C)CCC)CCC1(C)C N1(C(C2CCC(F)CC2)=O)CCC(C2(N=c3ccn4nccc4[nH]3)CC2)CC1 c1(C(N(CCCN(C(=O)CSc2ccc(O)cc2)C)C)=O)cnc2sccn12 N1(C(C(C)SC)=O)CC23CCCC2(C1)CN(C(c1cnc(F)c(C)c1)=O)C3 C(=O)(CCC1=CCCCC1)N1C(C(N2C(C(CC)O)CCC2)=O)COCC1 N1(C(c2c(C)nn(CCO)c2)=O)CCCC(CO)(NC(=O)CC(C)N(C)C)C1 c1(OC)cc(OCc2cccc(F)c2)nc(N2CC(C(=O)O)CC(C)C2)n1 C12(CNC(=O)CCc3cncs3)CN(C(C3COC(=O)N3)=O)CC1CS(=O)(=O)C2 Cn1cc(CNC(=O)C(C2CCC2)NC(C2CCC(=O)C2)=O)n(C)c1=O C(C)(C)(CC(=O)N1CCC(OCCNC(C2(F)CCOC2C)=O)C1)OC Cc1ccc(Cl)c2[nH]c(C(=O)NC(C)CN(C)C(c3cc(N)ccn3)=O)cc12 C(=O)(C(C(C)CC)NC)NCC(C)N(CCC)C(c1cnn(CC)c1C)=O C1(C(F)(F)F)(C(N(CC(=O)NCCNC(=O)C=C(Cl)Cl)C)=O)CC(C)(C)C1 N1(C(C(C)N(C)C)=O)CC(NC(C2C3CCC2(c2ccc(F)cc2)C3)=O)CC1C Cc1csc(C(=O)NCCn2cc(C(=O)NCCCC3C=CCC3)nn2)c1 c1(CC(CNC(C2(CC=C)CCC2)=O)(OC)OC)cc(O)c2ccccc2c1 CCC(O)(CNC(c1cn(CCNC(c2ncn(C)n2)=O)nn1)=O)CC C1(C(=O)OC)CCCCCN1C(C12CCC(NC(=O)CCNC(C)=O)(CC1)C2)=O C(=O)(C(C)(F)C(=O)NC1CC(CNC(=O)CC2(C)CCC2)C1)OCC c1(C(N2CCCC(NC(C3(NC(C)=O)CCC3)=O)C2C)=O)cc2n(c1)CCCC2 c1(CN(C(=O)NC2CC(O)C23CCC3)CC)cnc(C2CCC2)cc1C C1(C(=O)NCC2CC(NC(C3C(CC)OCCC3)=O)C2)CCCC2(CCC2)O1 CCC(C(=O)OC)C(=O)N1CCCC1(C)C(N1CCC(C(C)OC)CC1)=O N1(C(CCNC(N)=O)=O)CCC(NC(c2ccc(F)cc2)=O)C(CO)CC1 C=CCC(CC(=O)N1CC=CC(O)C1)NC(c1cc(C)oc1CC)=O C(=O)(C1=NOC2COCC12)N1CCC(C(N(CC(N2CCCC2)=O)C)=O)C(O)C1 C1(OC)CCn2cc(C(N3CCC3CNC(=O)Cn3cccnc3=O)=O)nc2C1 C1(C(=O)NCC2CC2C2CCC2)CCN(C(c2ccncc2O)=O)C12CC2 CC(C(=O)NCC=CCNC(C1(CC2CCC2)CC1)=O)=C1CCCC1 C1(C(=O)NCC(CN(C(=O)Cc2ccsc2)C)(C)C)Cc2cc(F)ccc2O1 c1(C(N2CC3CCN(C(c4c(C)ncn4O)=O)CC32)=O)ccc2c(c1)C=CCC2 N1(C(CCC=CC)=O)CCC(NC(c2cccc([N+](=O)[O-])c2N)=O)C2(CCC2)C1 c1(C(=O)NCC2(F)CC(NC(C3CC(OC)C3)=O)C2)cccc2cc(Cl)ccc12 c1(C(C)C)cc(C(=O)NC(C)(C)CCNC(c2ccccc2)=O)ccc1Cl N1(C(C(C)NC(=O)NC)=O)CCC2(CC1)CC(NC(=O)C(=O)N(C)C)CO2 C(=O)(C1=NOC2(CCOC2)C1)NCC1(C)CCCN1C(C12CC(C#N)(C1)C2)=O CC(C1CCCCC1)=CC(=O)NCC(C)(C(C)C)NC(=O)CC1(CO)CC1 CC(N=c1[nH]ccc(C#N)c1F)c1cn[nH]c1 C1(N(C(=O)C=CCc2cncs2)CCC2CC2)CCC(F)(F)CC1 c1(SC)cccnc1C(=O)NCC1CCCC(CNC(=O)C(C)SC(C)C)C1 Cc1cnc(CCN(C2(C)CCNC2=O)CCNC(=O)CCC2CCC2)nc1 c1(OC)cc(C)c(C(=O)N(CCCNC(c2c(C)nn(C)c2Cl)=O)C)cc1Cl CCCC(C)(CC)C(=O)N(CCN(c1ncno1)C)C(C)C N1(CC)CC(C(=O)N2CCC(N(C(=O)CCC(C)(F)F)C)C2)c2ccccc21 CC(CC(N)=O)C(=O)NC(C(=O)NCc1ncc[nH]c1=O)C1CCCC1 Nc1cccc(CC(N)C(=O)NC23CC(C2)C3)c1 C1(SC)CN(C(c2cc(Cl)cnn2)=O)CC1NC(=O)C(C)(C)n1cnnn1 C12CCOCC1NC(=O)C(C(C)C)Nc1cccc(c1)C(=O)N2.CCCOC O=S(=O)(c1ccc(CC(F)(F)F)cc1)NCC(O)C(F)F c1(C(=O)NC(CCNC(Cn2nnc(C)n2)=O)C)cccc2ccnn12 CC#CCCCC(=O)NC(C)C(CO)NC(=O)CCNC(=O)CC1CCCC1 CCC(C(=O)NC1C2CC3CN(C(=O)Cc4nocc4C)C1C3C2)C(C)(C)CC n1(CCC(=O)NC2CN(C(C3ON=C(C)C3)=O)CC23CC3)c(C)cc(O)cc1=O CCC(C(N)=O)(NC(=O)CC1CCN(C(=O)C(N)=O)CC1)OC c1(C(=O)NCCC2CC(NC(c3n(C=C)nnc3)=O)C2)cc(C)cc(C)c1N C1(CC(=O)NCC(CC2CC2)C(=O)N2CC(n3cnnc3)C2)CC2(CCC2)C1 Cc1cc(C(N2CCOC(C(C)NC(=O)CC(C)(C)F)C2)=O)cc(C)c1C Cc1ncc(-c2cn(C3CCNCC3)nn2)cn1.C(=O)C#CC(C)C c1(OC)cccc(C(=O)N(C2CN(C(=O)CCSC(C)=O)CC2F)C)n1 c1(OC2C(C(N3CC(N(C)C)C4(C3)CC4)=O)=CCC2)cnc2ccccc2c1 CC1OC2(C(=O)NCC(C3CCCC3)NC(=O)CC3COC(=O)N3)CCC1CC2 N1(C(c2cn(C)c(=O)cc2)=O)CC(NC(=O)CCCNC(=O)C2CC2)CC2(CC2)C1 C1(NC(C(CC)(C)C)=O)CC2CC(C1)N(C(c1csc(C(C)(C)C)n1)=O)C2 c1(C2(CC)CC(NC=O)C2)ccc(F)cc1.C(C)(CN(C(C)=O)CC)OCC C(=O)(C1CCc2c[nH]nc21)NC(CC=C)CNC(c1cc(C2(C)CC2)on1)=O c1(C(=O)NC2(C)CN(C(CCOCC(C)C)=O)C2)cccc(Cl)c1O C(=O)(C(=O)C(C)(C)C)NC(C(C)NC(C1COCCO1)=O)CO CC(C)C(O)CC(=O)N1CCC(C(F)(F)F)C(NC(C2CC2c2cccnc2)=O)C1 C1(CC(=O)NCC2CCOC2)CCN(C(C2CCCSC2)=O)C1 N1(C(CC(C)(F)F)=O)CCN(CCNC(=O)CN2CC3CC3C2)C2(CCC2)C1 S(=O)(=O)(c1c[nH]ccc1=NCC1(F)COc2ccccc2C1)N(CCC=C)CCOC Cc1nnc2n1CC(C(N1CC(NC(=O)C=Cc3cscn3)CCC1C)=O)C2 N1(C(c2c(CC)non2)=O)CCC(C)C(N(C)C(c2cccc(Cl)c2F)=O)C1 CC1(F)CN(C(c2cc(Br)c[nH]2)=O)CCN(C(c2cc(Cl)c(Cl)s2)=O)C1 CCCC(C(=O)N1CCOC(C)(CNC(=O)CCCN2CCCC2)C1)S(N)(=O)=O c1(C(=O)NC2CN(C(CCC(=C)Cl)=O)CC2O)cc2cccc(C)c2s1 c1(C(N2CC(CN(C(=O)CCCCCN(C)C)C)OCC2)=O)ccn2ccnc2n1 Cc1ccc(SCC(N2CCC(N(C)C(C3CC(F)(F)C3)=O)CC2)=O)c(C)c1 Cc1cc(C(=O)N(C(C)CNC(C2(C)CCNC(=O)C2)=O)C)cc(C)n1 C12=c3c(scn3)=NC(=NCCN1)N2.S(=O)(=O)(C1CC1)NC(COCC)COC Cc1oc(C(=O)N(CCCN(C(=O)CC(n2nc(C)cc2C)C)C)C)cc1CO C1(O)(CN(C(=O)CN(C2CCSC2)C)C)CCN(C(=O)C(C)(C)CCF)CC1 CC1CCCC(C(C(=O)Nc2ccccc2)N(C2CCCCCC2)CC2CC2)C1 c1(C(=O)NCC2CCC2NC(C2C3(CC3)C23CC3)=O)cc(F)c(F)cc1F C1(O)(CCNC(C=CCC)=O)CCN(C(=O)C(C)Cc2cnco2)C1 S(=O)(=O)(c1ccc(SC)c(F)c1)NCC1(SC)CC1.c1(S)ccc(C(C)N)c(F)c1 N1(C(c2sccc2Cl)C(=O)NCCCF)CCCCC(N2CCCC2)C1 CCC(O)CC(=O)N(C1CCCN(C(=O)C(c2cccnc2)N)C1)CC C(CCCCCC(=O)N1CCC(C)(NC(=O)C(C)Cc2cnn(C)c2)CC1)SC C#CCC(C)(C)C(=O)NCC12CC1CN(C(c1c(C)nn(C)c1Br)=O)C2 C1(CNC(C(=O)NCC)=O)CN(C(c2ccc(N)cc2O)=O)CC12CCC2 c1(C(N2CC3(C(NC(C4CC=CC4)=O)CCC3)C2)=O)ccn2c(O)nnc2c1 C(C(CO)N=c1[nH]nc(C2CCC2)o1)NC(c1c(NS(C)(=O)=O)cccc1)=O C1(NC(C2C3CC3CN2C(C2CC2C(F)F)=O)=O)CCC12CCCC2 N1(CCC)CCC(NC(=O)CCC(=O)N2CCN(C(C)=O)CC2)CC1 Cc1cc(NCC2CC3C2CCN3C(=O)OC(C)(C)C)nc(Cl)c1 c1(CC)cc(OC)cc(OC)c1C(=O)NC(C)CN(C(=O)C(C)c1ccsc1)C C#CC1CN(C(c2cnc(Cl)[nH]2)=O)CCN1C(c1cc(C#N)ccc1O)=O C1(NC(C2(C)CCCN2C(=O)C(c2ccccc2)=O)=O)CCn2cnnc2C1 c1(C(C)=O)cc(Br)c(C)cn1.C12CN(CCS1)C(=O)NC2 C(=O)(C(COC)C(F)(F)F)N1CCC(N(C(C(=O)NCC)=O)C)CC1 c1(C(=O)NCC(CNC(CC(=C=C)C)=O)O)ccc(-c2cccc(Cl)c2)cc1C C(=O)(C(C(F)(F)F)C(F)(F)F)NC1CCC(CNC(C(CCCC)C)=O)CC1 N1(C(c2ccc(C)nc2)=O)CCC2C(C1)CN2C(c1cnn2cccc2c1)=O N1(C(C(CCOC)NC(c2cc(C)[nH]c2C)=O)=O)CCCNC(=O)C1C N#Cc1ccnnc1N1CC(CCCCNC(=O)CC2CC3CC3C2)C1 Cc1c(F)cc(C(=O)NCC(CNC(C2(C)CCCS2)=O)S(C)(=O)=O)c(F)c1N C12(NC(Cc3c(C)noc3Cl)=O)CCCN(C(=O)CP(C)(C)=O)CC1C2 Cc1nc(C(C)C)oc1C(=O)NCCCN(C(=O)Cn1nnc(C2CC2)n1)C N1(C(CSCCC(C)C)=O)CCCN(C(c2ccc(CO)s2)=O)CC1 C12(NC(=O)NC3C(CCC)CN(C(C)=O)C3)CCC(C1)OC2C N1(c2nccc(=NC)[nH]2)CCOC2CCCC12 N1(C(c2c(C(=O)OC)c(C)on2)=O)CCC(NC(c2cc(C)nn2C)=O)C(C)C1 N1(C(C2=C(C)CC2)=O)CC(N=[N+]=[N-])CC1C(=O)NCC(CO)C(C)C N1(C(CCSC)=O)CCOC(CN(C(=O)Cn2c(O)nnc2O)C)C1 C1(C)(NC(c2cnc(C)o2)=O)CCN(C(c2cccc(CCO)c2)=O)CC1 c1(CC)[nH]nc(C(=O)NCC=CCNC(c2nnn(C(C)C)c2C)=O)c1Br C1(C#N)(NC(c2c(OCC)ccs2)=O)CCN(C(=O)CC(O)c2ccccc2)C1 C(C(CC(C)C)C(=O)N1CCC(C(=O)N(CC(C)O)C(C)C)C1)OC c1(C(=O)NCC2CCN(C(c3cnccn3)C)C23CC3)coc2c1C(=O)NCC2 N1(C(CN(C(=O)OC)C)=O)CC(CCNC(C2CC(O)CN2C)=O)C(C)C1 c1(CC(=O)NCCCN(C(C2CC(=C3CC3)C2)=O)CC)ncnn1C N1(C(C2CCC(C)CN2C(C2CCNC2=O)=O)=O)CC(C#N)C2(CCC2)C1 c1(CC)ccccc1CC(=O)NCC12CC1CN(C(c1ocnc1C)=O)C2 N1(C(c2cccc(C)c2N)=O)CC2CC(C)N(C(=O)CC3CCC(C)(C)C3)C2C1 N1(C(CCC=C(C)C)=O)CCC2CC2(C(=O)NC(C)(C)C(C)(C)C)CC1 C(=O)(C#CC(C)(C)O)NC12CN(C(C(c3cccs3)SC)=O)C(C1)C2 CC1CN(c2ccccc2CC2CC2)CC(C)O1.c12[nH]c(=N)[nH]c1C(=O)N2 c1(C(N2CCC(CC=C)(NC(c3ccc(C)o3)=O)C2)=O)cc2ccc(Cl)cc2o1 O=C1CCC(CC(N2CCC(NC(=O)CC3(O)CCCC3)CC2)=O)CN1 C(=O)(C(CO)C(F)(F)F)N1CC(C2CN(C(C3CCN(C)CC3)=O)C2)C1 C1(C(N2CC(NC(c3cn(CCOC)nc3)=O)C(OC)C2)=O)CC(=O)NC(=O)N1 C(CCN(C)C(C1CCCCS1)=O)(C(C)C)NC(C1(OCC)CCOC1)=O Cc1cccc2[nH]c(C(N3CCCCC3CNC(c3cccc(F)c3)=O)=O)cc12 Cc1ccccc1C=CC(N1CC2(NC(c3cc(C)n(CO)n3)=O)CCC1C2)=O N1(C(C2C(C#N)CC2)=O)CCC2(C(=O)NCCCSCCO)CCCC12 O=C(Cc1cccc(Br)c1)NNS(=O)(=O)CC1CSC1 CC(CC(=O)N1CC(F)(F)CC1(C)CNC(=O)Cc1cnsc1)C(F)(F)F c1(CC(=O)NCC(C)NC(C2CCCCS2)=O)ccc(O)nc1 N1(C(COC(CC)(C)C)=O)CC2CN(C(C3COC4COCC4O3)=O)CCC12 N1(C(Cn2ccc(=N)[nH]2)=O)CCC(NC(C2(c3ccncc3)CC2)=O)C(CO)C1 C12CC3CCC(C1C2)N3C(c1coc(CO)c1)=O.CCC=O.C1C(=O)N1 N1(C(=O)Cc2cnccn2)CC2CCC1CN2C(=O)C=C1CCCCCC1(F)F CC1CC(NC(C2(C)CCC2)=O)CN(C(c2cnc(-n3cccn3)nc2)=O)C1 c1(C(=O)NC2CN(C(c3nn(C)c(O)c3)=O)CC2(C)C)coc2c1C(=O)NCC2 CC1CCc2onc(C(=O)NC3CCN(C(c4ccnc(Cl)c4N)=O)CC3)c2C1 N(C1CCOc2c(OC)cc(C)cc21)C(=O)NC(C1CCOC1)CC C(=O)(CC(C)(C)C)N(C(C1OCC(C(N(C(C(N)=O)C2CC2)C)=O)C1)=O)C1CC1 c1(COC)ncc(C(=O)NCC2(CNC(=O)CC(C)C)CCCC2)cn1 C(C1=CCN(C(=O)C=Cc2ccc[nH]2)CC1)NC(Cn1c(C)csc1=O)=O N1(C(c2cc(CC)c(C)s2)=O)CCC2CN(C(c3ncc(Cl)cc3F)=O)CC12 C(C1=NOC2CN(C(c3cnnc(C4CC4)c3)=O)CC12)NC(c1cc(C)c(C)[nH]1)=O C1(C(N(C(CO)C2CC2)C)=O)CCCC(NC(c2cnn(C)n2)=O)C1 C1(C(=O)NC(CC)C(C)CN(C)C)CCN(C(=O)c2ccnnc2C)O1 S(=O)(=O)(c1ccc(I)cc1[N+](=O)[O-])NCCc1cc(C(C)(C)C)on1 C1(N(C)CCOC2CCOC2=O)CN(C(=O)C(F)CC2CCC2)CC12CC2 C=CCCC(C(=O)NC1CCC=CCCC1)N1CCN(c2ccc(F)cc2)CC1 c1(C(=O)NC2CCCN(C(Cn3ccc(C)n3)=O)CC2)c[nH]c(=O)c2ccnn12 Cc1cc(=NC2CCN(CC3CN(C(C4C5CC6C(C5)C46)=O)C3)CC2)[nH]c(CO)n1 C1(O)(C(C)NC(=O)C(F)OC(F)(F)F)CCN(C(c2cnn(C3CC3)c2)=O)C1 CC(CC(F)F)C(=O)N1CCN(C(C2CN3CCCC2C3)=O)CC1CCO CC1(C)CC(F)(F)CCC1NC(=O)CC1CC2CCC1CC2 C(c1ccccc1Cl)=CC(=O)NCCCNC(C12OCC(C(C)C)(C1)C2)=O N1(Cc2c(C)nc(C)s2)CCC(C)C(NC(=O)CCC2NC(=O)NC2=O)C1 n1(CC(=O)NC(CCCCNC(C)=O)C)nc2n(c(=O)c1=O)CCC2 Cc1cncc(C)c1C(N1CCOCC(CNC(=O)COc2cnn(C)c2)C1)=O c1(C(C)(C)C)n[nH]cc1C(c1nnnn1Cc1cccs1)NC1CC(CC#N)C1 CC(C(=O)NC(=O)Cn1cc(-c2ccc(C#N)cc2)nn1)(C(F)(F)F)C(=O)O CC(O)C(C)C(=O)N(CCCOCCNC(c1ccccc1F)=O)C.C(=O)C1CC1 CC(C)(C)C(O)C(=O)N1CC(NC(C2CCCC(=O)C2)=O)C(C)(C)C1 c1(CC(=O)N(CC(CC)NC(c2ccn(CC3CC3)n2)=O)C)cc(C)n(C)n1 c1(C(=O)NCCCNC(c2cnc(OC)s2)=O)ccc2c(c1)CC(C)O2 CCCCS(=O)(=O)CC(=O)NCC1(OC)CN(C(c2ccnn2CC)=O)C1 C(=O)(C(C)CC(=O)NC(CNC(=O)CC1=CCCC1)CC(C)C)OC N1(C(c2cnc(SC)s2)=O)CCN(C(c2ccon2)=O)C(CCO)C1 N1(C(C)(C)C)CCC(F)(F)C1.N12CC(C(O)C1)C(=O)NC(=O)NCC2 N1(C(C(C)O)=O)CCC(NC(c2cc(Cl)ns2)=O)C1C(C)C C1(NC(c2ccc(C(=O)OC)s2)=O)CC(O)CN(C(c2cccc(Cl)c2C)=O)C1 C1(C(=O)NCC(C)NC(=O)C(C)(C)c2cncnc2)CC(C)(C)CO1 CC(C(=O)NCC1(CCNC(=O)C(C2CCCO2)C2CC2)CC1)N(C)C c1(NC(CCOc2cccc(C(C)C)c2)=O)c[nH]c2nccc(Cl)c12 Cc1ccc(C(C)C(N2CCCC2C2CCCOC2)=O)o1 CCC(C)C(C(=O)NCC(CO)OC)N(C)C(c1cccc(C)c1N)=O C#Cc1cnn(C)c1C(=O)N(C1CCCNC1=O)C NC(=O)CCC(=O)NCc1ncoc1CCNC(=O)C1=CCC1 C=CC1(O)CCN(C(C2CCN(C(C3CC4(CC(OC)C4)C3)=O)C(C)C2)=O)C1 CC(C)(C)CCC(F)C(=O)NC12CCCC1N(C(c1cc(F)cnc1O)=O)CC2 C(CCS(C)(=O)=O)N(C(CCN(CC#C)C(c1cnn(C)c1OC)=O)=O)CC C(=O)(CS(=O)(=O)C12CC(C1)C2)NC1C2CC(NC(c3ccn(C)n3)=O)C(CC2)C1 N12C3CCC1(CC3)CC2=O.C(=O)(CC(C)(C)O)NCC1(C)CC1c1ccccc1 C1(N(CC#C)C(c2cnc[nH]2)=O)CCOCCN1C(=O)C=CC(C)CC n1(CCCSC)nnnc1C(C1C2COCC12)NCCCC(F)F CN1C(=O)OCC12CN(C(=O)CC(F)(F)c1ncccc1Br)C2 c1(CNC(CN(C)CC)=O)ncc(C(=O)NCC23COC(C2)C3)cn1 S(=O)(=O)(CCC(=O)N1CCC(C(C)C)CC1)NC.C1(C(C)OC)C(=O)N1 C1(CCC(=O)NC2(CC=C)CC=CC2)CCCCN1C(=O)CC1CCCC(C)C1 c1(C(=O)Nc2cccc(CO)c2)cnc2ccnn2c1.C12(CCCCCC1)NC2 c1(C(=O)NCC(C2CCN(C(C=CCOC)=O)C2)(C)C)c(Br)cnn1C Nc1cc(C(N2CCN(C(c3csc(Cl)c3)=O)C(c3cn[nH]c3)C2)=O)cc(F)c1 C(C)(C(=O)N(C(C)CN(C)C)CC)(C(C)C)NC(c1c[nH]c(=NC)s1)=O C12(CNC(c3c(C)nc(C(F)(F)F)cc3)=O)CC(CO)(C1)C(C)(C)O2 N1(C(C(C)CC2CCCC2)=O)CCCC(NC(C2(C)CC(F)C2)=O)C1 C(CC(C)C)(C(=O)NCCC1=CCCCC1)NC(c1cncc(NC)c1)=O Cc1ccc(C(=O)NCC2C3CN(C(c4n[nH]cc4Cl)=O)CC23)c(=O)n1C Cc1cc(O)c(Cl)cc1C(=O)NCCNC(=O)C1=NOC(c2ccc(F)cc2)C1 C=CCCN=C(NCC(N1CCOCC1)C)NCC(O)C1(C)CC1 c1(OC)cccc2c(C(N3CCC(O)(CNC(=O)CCC(C)(F)F)C3)=O)coc12 C1(CNC(c2cc(SC)no2)=O)C2C3CCC(C3)C12.C1(C)(C)C=CC(=O)N1 N#CC1CC2(CC(CNS(=O)(=O)CC3CCS(=O)(=O)N3C)C2)C1 c1(C(=O)NC2CN(C(CSC(C)C)=O)C3C2C3)cnc2cnn(C)c2c1 C#CCCC(C(=O)NCC1C=CCCC1)NC(=O)Cn1cc(C)ccc1=O CCC(CC)C(C(=O)NCCCC1CCCN1C(c1ccco1)=O)OC N1(C(COCc2cc(C)no2)=O)CCC(NC(=O)C2=CCCS2)C(CO)C1 c1(C(C)Oc2csc(C(F)Br)n2)cccc(C)c1C Cc1cccc2c1OC(C(N1CC3CC(C1)N(C(C1C4CCCC14)=O)C3)=O)C2 N1(C(c2c(OC)cncn2)=O)CC2CCC1CN2C(C1CC2(C1)CC(C)C2)=O c1(CSCC(=O)NC(C2CN(C(=O)C(F)(F)C3CCOCC3)C2)C)ccccn1 C(=O)(CCCC(C)(C)C#N)NCc1nc(CNC(Cc2c(C)cccc2C)=O)sc1 c1(C(=O)NCC(CC(F)(F)F)NC(c2cc(F)c[nH]2)=O)cccn2nccc12 N1(C(C=C(C)C(F)F)=O)CC(F)(F)CC1CCNC(=O)COC(F)F c1(C(N2CCN(C(C(COC)C)=O)C3(C2)CC3)=O)cc(OC)cc2c1OCC2 C1(NC(c2sccc2CC#N)=O)CCCC(NC(c2cnn3c2CCC3)=O)CC1 CCC(CC(=O)NCCCCN(CCCNC(c1ncsc1Br)=O)C)C1CC1 c1(C(N2CCC(C(C)NC(C(CC)F)=O)C2)=O)cc(N)ccc1O CC(CC(=O)NCC1COC(CNC(=O)Cn2nc(O)ccc2=O)C1)P(C)(C)=O CC1(C)CCCC(CC(N2CCCC(NC(=O)Cc3ccsc3)CC2)=O)C1 c1(C(=O)OCC)cccc(C(N2CCC(N(C(=O)C(C)C#N)CCO)C2)=O)c1 c1(N)c(C#N)cnn1CC.C(CCC(=O)N1CCC1CC1CC1)NC(C)=O N1(Cc2c3ncccc3[nH]c2)CC2CC=CCC2C1 N1(Cc2ccc(OC)nc2OC)CCC2CCC(C1)N2 CCC(C)C(O)C(=O)N1CCOC(C)(CNC(=O)C(=Cc2ccccc2Cl)C)C1 Cc1ccc(C(N2CCC(CCNC(c3cc(Cl)sc3Cl)=O)C2)=O)nn1 C1(C(=O)NCC(c2ccccc2)CNC(C2(CF)CC2)=O)CC2(C1)CC2F C(=O)(C(CNC(C1CC(O)C(F)C1)=O)C(C)C)NC(c1cc(C)no1)(C)C C1(C(=O)NCC(C)(C2CC2)NC(c2cnc(CCCC)s2)=O)CC12CCOCC2 Cc1nc2sccn2c1C(=O)NCC1CN(C(C2CC3CCC(C2)C3)=O)CC1C c1(C(=O)OC)ccc2c(n1)CCCN2C(c1cc2ccccc2nc1C)=O N1(C(C(N2CCOCC2)C)=O)CCC2(CCCC2NC(C2C(C)(C)C2(C)C)=O)CC1 N1(C(C(C)NC)=O)CCC2(CCCC2C(=O)Nc2ccc(-n3ccnc3)nc2)C1 N1(Cc2c(C)nn(C)c2)CCC2(CC(C(=O)Nc3c(Br)ccnc3Cl)=NO2)C1 C1(N(C)Cc2cn(-c3ccc(N=NC(N)=O)cc3)nn2)CCc2ccccc2C1 c1(OC)nc(C)ccc1C(N1CC2(CCN2C(c2cncc(Cl)c2)=O)C1)=O O(NC(=O)C(C1CC1)NC(=O)C(O)CC1CCC1)CCCC Cc1cc(=NCCC2CCC2(F)F)[nH]cc1S(=O)(=O)NCCOC(C)(C)C N1(C(C(COC)C)=O)CCN(C)CC1C(N1CC([N+](=O)[O-])C1)=O CC1CCCC1NC(=O)NCCN(C)CC1CCOCC1 C1(C)(C(=O)NC(c2ncc(C)o2)C)CCN(C(c2nnn(C)c2C)=O)C1 C1(O)(CN(C(Cc2c(C)ccnc2)=O)C)CCCN(C(C2CC2CF)=O)C1 C1(N(C(=O)Cn2ccnn2)C)CN(C)C1.C12(CC1)C(C)NC2=O c1(-n2cc(CNCCO)nn2)ccc(C(=O)NCC2(CCCO)CC2)cc1F c1(C(CC2(C)CC2)NCCCCC)nnnn1CC(=O)NCCOC c1(C(=O)NC2(CC=C)CCN(C(c3scc4c3OCC4)=O)C2)cc(Cl)cnc1C CN1CCC(CC(N2CCC(n3cc(Cn4ccnc4)nn3)C2)=O)CC1 C1(C(C)C)CN(C(c2nnn(Cc3ccccc3)c2Cl)=O)CC1N(C)C c1(C(N2CCN(C(Cc3cccc(CC)c3)=O)CC2C)=O)cnc2c(c1)NCC2 N1(C(C(c2ccnn2C)C)=O)CCC2CCN(C(C3(C)CC(F)C3)=O)CC2C1 C(CCC(N)=O)(C(=O)NC1CCCC12CN(C(C1(C)COC1)=O)C2)NC(C)=O CCCCC(C)(F)C(=O)N(C)CC=CC(=O)NC(c1ccccc1Cl)CC c1(C(=O)NCC2(NC(CCCSC)=O)CCCCCC2)c(C)cc(=O)oc1C C(C(O)(CNC(C1(C)CN(C(c2ccn(C(F)F)n2)=O)C1)=O)CO)OC c1(OC)cccc(C(=O)N(C)CC2(O)CCCN(C(c3conc3C)=O)C2)c1F C(=O)(C1CCCc2sccc21)NC1CN(C(c2c(C)cc(C)s2)=O)CC1C C1(CNC(=O)CC=C(Cl)Cl)CCCC2(CN(C(=O)C(=Cc3cccnc3)F)C2)O1 C1(C(=O)NCC2(F)CN(C(=O)COCCN(C)C)C2)SC2C=CC1CC2 N1(CCCC(=O)NC(CC)CNC(C2(C)CCCS2(=O)=O)=O)C(=O)CN(C)C1=O N1(C(CCOC)=O)CCC(NC(=O)Cc2ccccc2S(C)=O)CC(C)(C)C1 Cc1nn2c(C(=O)NC3CCN(C(C4(Cl)CC4)=O)CC3O)c(C)nc2s1 c1(C(N2CC3C(NC(=O)CSc4nccs4)(C3)C2)=O)cc(F)cc2nc(S)[nH]c12 C1(CNC(COCC(C)(C)C)=O)(NC(c2ccc(O)c(Cl)n2)=O)CCCCCC1 C1(O)(CNC(CCc2n(C)cnc2)=O)CCCN(C(=O)CN2CCC(C)(O)C2)C1 c1(C(=O)NCCOCCN(C)C(C2CCC(O)C2)=O)cccc(C(F)(F)F)c1 CC(C)C(C)CC(=O)N(CC(=O)NCCCCC(F)(F)F)C c1(CCNC(C(c2cn(C)nn2)NC(=O)Cn2ccnc2)=O)noc(=O)n1C c1(OC)cc(F)c(Br)cc1CNC1CN(C(C2CCCCC2(F)F)=O)CC1C C(=O)(C(C(C)(C)C)OC(C)(C)C)NC1(CCNC(CCC=C)=O)CCOCC1 N1(C(CCN(C)CCO)=O)CCC2(CC1)CC2(CO)CNC(=O)C1=CCCC1 C(=O)(C(C(C)(C)C)NC(c1csc(CSC)c1)=O)NCC(CCOC)(C)O C1(C(C(=O)NCCN(C)C(C2CC2(C)C)=O)Cc2ccccc2)CCC(F)(F)CC1 Cc1sc2cncn2c1CON1CCN(C2(CNS(C)(=O)=O)CC2)CC1 c1(C(N2C(CN(C(=O)C=C(Cl)Cl)C)CCC2)=O)ncn2c1CCCC2 CC(C)CC(C)C(=O)N(C1CCCC1)CCNC(=O)CC(C)(C)Cc1ccccc1 C(=O)(CCP(C)(C)=O)N1CCC(O)(CCNC(C(c2cccs2)SC)=O)C1 C1(C(=O)NCCNC(c2cccc(F)c2C(=O)OC)=O)CCn2cncc2C1 c1(C(CNC(c2n(CC)nnc2)=O)NC(C2C=CCCC2)=O)ccc(C)cc1 C1(C(N2CCC(CO)C2)=O)CCCCCN1C(c1cccc(O)c1F)=O C(C(CC)(CC)C(=O)N1CCCC(OC)CC1)NC(CCC(CC)C)=O Cc1cc(CCNC(C2CC(c3ccc(F)c(F)c3)(C(=O)O)C2)=O)ccc1F c1(C(=O)NCC2(F)CC(NC(c3cc(CC)ncn3)=O)C2)ccnc2cc[nH]c12 c1(C(N2CCN(C(CC=C)=O)CC(CO)C2)=O)ccc2oc(O)nc2c1 C1(NC(COCc2ncc(C)o2)=O)CC2CCC(C1)N2C(c1ccccn1)=O N1(C(c2c(C(N)=O)csc2)=O)CCC(CF)(NC(c2ncccc2F)=O)C1 c1(SCC)nc(C)c(CC(N2CCC(NC(c3cnn(C)c3N)=O)C2)=O)s1 c1(C(=O)NCCOCCCN(C(CCC=C=C)=O)C)ccc(C(C)=O)c(C)c1 c1(-c2nnc(N(C(=O)CNC(C(=O)O)C(C)O)C)n2C)nn(C)c2c1COCC2 N1(C(CCS(=O)(=O)NC)=O)CCC2(CCCCC2NC(c2cccs2)=O)C1 C1(CCNC(Cc2c(C)ccnc2)=O)CCCN(C(c2cncc(F)c2)=O)CC1 C1(NC(C(C=C)(C)CC)=O)CCN(CCCC2CCCCO2)CC1(C)C C1(C(=O)NCCCCNC(C2CCC(C)S2)=O)(C(F)F)CC2(CC2)C1 C1(C(=O)NCCN(C(=O)C(F)CC2CCOC2)CCC)(CO)CCOCC1 N1(C(Cc2cc(C(C)C)no2)=O)CCC(CO)(NC(C2CC=CCC2C)=O)C1 c1(NC(=O)CCSc2n(CC)c(-c3ccccc3C)nn2)cc(F)cc(F)c1 N1(C(C2(OC)CCCOC2)=O)CC(O)(C2CCN(C(=O)COC(C)=O)CC2)C1 C(=O)(C=C1SCC(=O)N1C)N1C(CCCNC(C(C)C2(O)CCC2)=O)CCCC1 N1(C(c2c(Cl)ccc(OC)c2)=O)CC2OCC(NC(=O)C(C)SC)C2C1 N1(C(S(CC2CC(CC)C2)(=O)=O)=O)CCc2c(Cl)cccc2C1C(=O)OC C(=O)(C1SCCc2ccccc21)NC1C(NC(C(C(C)C)C(C)C)=O)COC1 c1(CC)nccnc1C(=O)N(CC(CC)NC(C1(C)CC(C(F)(F)F)C1)=O)CC N1(c2cc(C)nc(C)n2)CCC2(CC1)CC=CC(=O)N2C c1(C(=O)NC2C(NC(c3csc(C(F)F)n3)=O)COC2)csc(Cl)c1Cl Cc1cccc(C(N2CCCC(N(C)C(c3cc(C)n(C)n3)=O)CC2)=O)c1F N1(Cc2ccc(OCC)nc2C)CCc2cc(OC)c(OC)cc2C1 c1(CC)c(C(N2CC(N(C)C(c3cc(C4CC4)no3)=O)C2)=O)cnn1CC C1(CCOC)CN(C(=O)C(F)(F)c2cncs2)CCN1C(c1cscn1)=O c1(NC)snc(C)c1C(=O)NCCCCCCNC(C1CCCC1(C)C)=O O=C(O)CCCCCS(=O)(=O)Nc1cnn2ccccc12 C(CC(C(=O)NC(Cc1ccco1)CO)NC(c1nc[nH]n1)=O)SC C1(C(=O)NC(C2CCN(C(C(C)=C(CC)C)=O)CC2)C)CC2(CCOC2)C1 N1(C(C2CCN(CC)C2)=O)C2CCC1CC(CNC(c1cn(C)nc1O)=O)C2 C1(C)(C(=O)NCC2C(NC(C3C(C)C3(F)F)=O)CCC2)CC(C(C)(C)C)=NO1 Cc1ccc(F)c(C(=O)C(=O)NCC2CCCN2C(=O)CN2CCC(C)C2)c1 CC1(C)CC(NC(C2CCCOC2)=O)CN(C(c2cnn3cc[nH]c23)=O)C1 C1(C(N2CC(C=C)(CC(N3CCC(C#N)C3)=O)C2)=O)C2CCC(C2)C1C O(C=C(C#N)C(=O)N1CCC(NC(c2ocnc2C2CC2)=O)C1(C)C)CC N1(C(C(C(C)C)N2CCCCC2)=O)CCC2CCN(C(=O)CC3CC3)C2C1 c1(C(=O)NCC2(NC(C3C(c4cccc(C)c4)CC3)=O)CC2)cc(C)c(C)nn1 C=Cn1ncc(C(=O)NCC2CC2C(=O)NC2CC(O)CC2O)c1N Cc1ccccc1C=CC(N1CC2(C(=O)NC3CCCC3CO)CC1CO2)=O Cc1ncc(C(=O)NCC(C)CNC(=O)CN(C)CCc2ccccc2)c(C)n1 c1(C(=O)NC(CC#C)C(=O)NCC2CCC(=O)CC2)cc(C)c(N)cn1 N1(C(C(c2cccs2)NC(COCC)=O)=O)CCC1(C)CC C(CCC(C)C)(C(=O)NCC(C)(C)NC(=O)Cc1cc(C)cs1)NC(=O)OCC C1(C(=O)NC2CC(C#C)C2)CC2C=CC1N(C(=O)C(C(CC)CC)OC)C2 C(=O)(C(COC)CC(C)C)N1CC2(N(C(C(C)SCCCC)=O)CC2)C1 CC(C)CC(F)(F)C(=O)N(C1CCN(C(=O)COCc2cccnc2)C1)CCO C1(C(=O)NCC(CC)(CC)NC(=O)CN2CCOCC2=O)CCc2cnnn2C1 C(=O)(C1=CNC2=NCCCC2=C1)N1CC2C(N(C)C(C3CCCCN3N=O)=O)C2C1 c1(C(=O)NCC2(OC)CN(C(=O)COCC(=O)NC)C2)cc(C#N)ccc1F C1(C(=O)Nc2c(OC)cc(F)cn2)CN(c2ncncc2I)CC(F)(F)C1 C1(Nc2ccc(C(=O)NC3(C)CCCC3(F)F)cc2)CCOC12CCCC2 N1(C(CC(C)OC)=O)CCCC(C)(C(=O)Nc2sccc2Cc2cccc(C)n2)C1 c1(C(c2n(CCC)nnn2)NCC(C)(C)CCO)cc2cc(Cl)cnc2o1 C12(C(N3C(COC)CC3)=O)CCCC1CCN2C(C1(O)CCCC1)=O N1(C(=O)CCC2CCC2)CCN(C(c2noc3c2CCCC3)=O)CC(O)C1 C(=O)(CCC(F)(F)CN=[N+]=[N-])NCCC1(NC(c2c(C)cc(=O)n(C)c2)=O)CC1 Cc1ccc(N(C)C(=O)NC2CCN(C(C)C)CC2C)c(C)c1 c1(C(=O)NC(CNC(c2c(C)coc2C)=O)(C)C2CCC2)ccc2c(c1)OCC2 c1(C(=O)NCC2C=CC(NC(C(C)NC(COC)=O)=O)C2)n[nH]c(C)c1Cl C1(CC(N2CC(CC(C)NC(C3(C(=O)NC)CCC3)=O)C2)=O)CCCC(C)C1 c1(OC)cc(CCC(=O)NC2CC3(C2)CN(C(=O)CC(C)C(F)F)C3)ccc1F C1(C(N(CCN(C(C(c2ccccc2O)OC)=O)C)C)=O)C2CCCCCC12 C(CC(C(=O)NCCN(C)C)NC(c1cncnc1)=O)N(C)C c1(CC(=O)NCC(C)N(C(=O)CC(C)(C)C#N)CC)coc2ccccc12 c1(C(N2CC(NC(C=C(CC)C)=O)C2)=O)c(F)cc(N)cc1F N1(C(CC(=O)NCC)=O)CCCC(C2CCCN(C(=O)Cc3cnc[nH]3)C2)C1 N1(C(c2ccc3nccn3c2)=O)CCC2CCN(C(=O)Cn3cc(Cl)cn3)C2C1 Cc1c(C(=O)NCCNC(c2cnc[nH]c2=N)=O)c(-c2ccccc2)cn1C c1(C(C)N(C2CCNCCC2C)C(C2CC2CO)=O)c(F)cc(F)cc1F N1(Cc2cn(CC(C)C)nc2C)CCCC(C)(CNC(=O)Cn2ccnc2)C1 N1(C(C2C(CC)CN(C(C3CS(=O)(=O)C3)=O)C2)=O)CCCCCCCCC1 C1(NC(c2nc(CCC)oc2)=O)CCCC(CNC(=O)OC(C)(C)C)C1 c1(C(N2CC(CC)C(NC(C3(OC)CCCC3)=O)C2)=O)cc2ccc(C)cc2[nH]1 C1(C(N(CC(C)NC(=O)COCC(F)F)C)=O)COc2ccc(Cl)cc2C1 N1(C(CCCOCC)=O)CCN(C(=O)C(C)Sc2ccc(Cl)cc2)CC1C c1(N2CC=C(C)C2)nc(N2CCN(C3CCOC3)CC2)nc2scnc12 c1(CNC(C2CCC(C(N3CC4COCC4C3)=O)OC2)=O)c(F)cccc1F C1(NC(c2c(C)nc(O)[nH]2)=O)CCN(C(C2CCC3CC3CC2)=O)CC1(C)C C1(C(=O)NCCC2(CNC(C3(C)CCC4CC4C3)=O)CC2)CN=C2N=CNN2C1 C1(CNCc2ccc(CS(C)(=O)=O)nc2)COC2(CCC2)C1 C12(OCC#CC)CCN(C(=O)C(OC)OC)CCC1C2 CC(c1ccc(F)cc1)=CC(=O)NC1COCC1NC(=O)C1=COCC1 C1(C(=O)NCC=C2CCN(C(COCC(=O)OC)=O)CC2)CN(C)CC(C)C1 c1(C(N(c2ncccc2N)C)=O)cccc(CNC(C2CC2(F)F)=O)c1 C(=O)(C(C)Cc1ccc(C(=O)O)o1)NCC1N(C(CCOCC#C)=O)CC1 N1(C(Cc2cc(C)[nH]n2)=O)C2CCCC1CC(NC(=O)C(CC1CC1)CC1CC1)C2 c1(C(=O)NC2CC(CNC(=O)C3=COCCC3)C(O)C2)cccc(C#CCO)c1 C1(C(=O)NC2CCN(C(CNC(=O)C3CC3)=O)C2)CC12C1CC3CC(C1)CC2C3 c1(CNC(=O)OC2COC(Cc3ccccc3)C2)cnn(CCF)c1 N1(C(C(COC)N(C)C)=O)CC2CC(NC(C3(C)CC=CC3)=O)CC2C1 Cc1cc2c(cc1C)OC(C(N1CC(C)(NC(c3cc(C)c(N)cn3)=O)C1)=O)C2 c1(NC(CNC(C=CC)=O)C(C)C)nc2ccc(C(N)=O)cc2cc1[N+](=O)[O-] N1(C(CSC(C)(C)C)=O)CCC2(CC2C(=O)Nc2nocc2C(=O)O)C1 CC1=C(C(=O)N2CC(CO)(NC(c3sccc3C(N)=O)=O)C2)C(=O)OC1(C)C c1(NC2C(CNC(=O)Nc3cccc(I)c3)CCC2)ncnc2[nH]cc(I)c12 CC1=CCN(CCNC(=O)NCCC2CCCOC2)CC1 Cn1ncc2ncnc(N(C)C)c12.C12CCCN(C1)C(=O)c1ccc(o1)CN2 c1(C(=O)NCC(C(C)(C)C)NC(CC2(CSC)CC2)=O)cnc2cc(C)[nH]c2c1 c12csc(n1)C(c1nnnn1C)NC2=O.C1(C(=O)NC)(C(=O)NC(C)C)CC1 N1(C(C2(C(F)F)CC(N)C2)=O)CCN(C(=O)Cn2ccnn2)CC1 c1(C(N(CC(N2CC(C)(CC(F)F)C2)=O)CCOC)=O)c(C)noc1C Cc1cc(C(N2CCC(N(C(=O)CC3CCOC3)CCO)C2)=O)cc(Cl)n1 C12(C(=O)NCC=C3CCN(C(C(C(C)OC)O)=O)CC3)CC(C)(C1)OC21CCC1 CC1(C)C(CC(N2CCN(C(=O)CCCC3CCCCC3)CC2)=O)CC1O C12(CNC(C(C)OCCOC)=O)CC(NC(c3nccs3)=O)(C1)C2 C(c1ccc(Cl)cc1)=CCNC(=O)N(CC1CC1)CC1(F)CC(O)C1 C1(CN(C)CC2CC2(F)F)CCCCN1C(C1CCC(N2CCOCC2)CC1)=O N1(C(CC2(C)N(C(=O)Nc3cccc(CC)n3)CC2)=O)CCC(C2(O)CC2)CC1 C(CC(CC)C(=O)NCCCOCCNC(=O)CC1(C)CCOCC1)=CC Cc1cc(Br)c(-n2cc(-c3cc(F)c(O)c(F)c3)nn2)cc1Cl C1(C(N(C2CN(C(c3cc(C)sc3)=O)CC2F)C)=O)CC(C)CCC1C(C)C C1(CNC(Cc2ccc(OC)cc2)=O)CC2(C1)CN(C(C1CCCC(C)C1)=O)C2 N1(C(c2cc(C)no2)=O)CCC12CC(C(=O)NC1C3CC4C(C3)C14)C2 c1(CNC(C(=O)OC)CC2CCCCO2)ncnc(OC)c1OC C1(C(N(CCC(C)NC(C2CC(OC3CCOCC3)C2)=O)C)=O)OCC1(C)C C12(CNC(Cc3c(C)cco3)=O)CCC(CN(C(=O)CCNC(N)=O)C1)C2 Cc1ccc(Cl)cc1C(=O)NCC1(NC(=O)C2=NOC(C)C2)CCOCC1 c1(CNC(C=CCOCCOC)=O)cc[nH]c1C(=O)NC1CCOC1 c1(C(=O)NCCOCCN(C(C(C=C)(F)F)=O)C)cc(F)ccc1C(F)(F)F c1(C(N2CCCC(NC(c3c(=N)cc[nH]c3)=O)C2)=O)cnn2c1OCC(F)C2 C1(C(C)(C)C)CC(C(=O)NC2(CCCCNC(=O)CN3CSCC3=O)CC2)=NO1 C(=O)(C1=CCCSC1)NC1(CCNC(C2(C)CS(=O)(=O)C2)=O)CC1 c1(-n2c(C)c(C(=O)OCc3ncc(Br)s3)cn2)cccc2cccnc12 CCC(CN(C)C)C(=O)N1CCC(CC(=O)N(C(C)COCC)C(C)C)CC1 CC1CC(=O)NCC1C(N1CC=CCC1C(=O)N(CC(C)(C)N(C)C)C)=O N1(C(C2CCCCO2)=O)CCN(C(C2CC(N3CCNCC3)C2)=O)CC1 c1(C(N2CC(N(C(c3c(C)cc[nH]3)=O)C)C(O)C2)=O)ncc(N)cc1C c1nc(-n2cccc2)nn1C1CCc2ccccc21.n1(CC)cncn1.CC Cc1cc(C#N)cnc1C(=O)NC12CCN(C(c3ccc(CO)o3)=O)CC1C2 C(=O)(C(CC(C)C)C1CCCO1)NCCC(=O)NC.C1(=O)CC(C)(C)N1C c1(CN(CC(C)(C)CS(N)(=O)=O)C)c[nH]c2cc(F)c(F)c(F)c12 C(N=c1[nH]c(=NCCC2CN(C)C2)[nH]c2c1CCC2)c1cn(CC)nn1 N1(C(C2(OCC)CCCC2)=O)CC(NC(=O)CC2(C)CC2(F)F)C(C)C1 C(=O)(CCCCC(=O)NC1C=CC(CNC(=O)Cc2c(C)nn(C)c2C)C1)OC c1(OC)cc(F)c(C(=O)NCCNC(=O)Cc2ccnc(F)c2)c(F)c1F C#CCC(C(=O)OC(C)=O)NC(c1csnn1)=O N1(CC)CCN(Cc2cccc(N)c2NC)C2CC12.c12ccc([nH]1)c(=O)n2C(C)=O N1(C(C2(F)c3cc(C)c(Cl)cc3SCC2)=O)CCCC2(CCOCC2)C1 CC1c2ccccc2CC1C(=O)NCCOCCCNC(=O)C1=CCOC1 C1(C(=O)NCC(C(C)C)NC(c2cc([N+](=O)[O-])cn2C)=O)CCn2nncc2C1 c1(CC(=O)NCCN(C(=O)CN2CCCC2CO)C)cnc(C(C)(C)C)o1 C(N=c1[nH]c2c(c(=NC3CSc4ccccc43)[nH]1)COC2)c1c(C)occ1 c1(C(=O)NC(CNC(c2c(C)nc(C)o2)=O)(C)CO)cc(C(C)(F)F)ccc1C C(=O)(C1=CCCN(C(c2ncc3ccccn23)=O)C1)N1CC(C)(CSC)C1 C=C(C)CCCC(=O)NCC1CCCCCN1C(=O)C(CC)n1ccnc1 C1(NC(C(C=C)(C)C)=O)CN(C(=O)CCNS(=O)(=O)CC)CC12CC2 N1(C(=O)CCc2nc[nH]n2)CCC2(CCCN2C(c2cc(=O)cc(Cl)[nH]2)=O)C1 C(CC(C(=O)NCCN1CCC1)NC(C1CSC1)=O)=CC N1(C(C(C)=C2CC2)=O)CCOCC(NC(c2cnnn2C2CC2)=O)C1 CC1(C(N2CCC(O)(c3cc[nH]n3)C2)=O)CCCN(c2ccncn2)C1 C1(NC(C(C)CNC(=O)C=Cc2ccncc2)=O)CCC2CC1CO2 N1(C(COC(c2ccccc2)C)=O)CC(N(C(=O)CC2CC=CC2)C)C(O)C1 C1(CC(=O)NCCNC(C(C)C)=O)C2CCCC2N1C(=O)C(C1CCOC1C)=O N1(C(CC(CC)OC)=O)C2CCC1CC(C(=O)NC(C)C(F)(F)F)C2 C12(NC(CS(=O)(=O)N(C)C)=O)CCOCC1CN(C(c1ccc(C#N)cn1)=O)C2 C1(C#N)(C(=O)NCCCNC(CCN(C)CC)=O)CC2CC2C1 n1(CC)cnnc1CCNC(=O)C(F)CC1CN(C(C2(Cl)CC2COCC)=O)C1 c1(C(=O)NC2C(CNC(c3cn(CC)nn3)=O)CC2)cccc(N2CCCC2)c1 c1(COC)cc(C(=O)NC(C)C(=O)NC2CC(n3cncn3)C2)n[nH]1 C1(CNC(C2CC2C(F)(F)F)=O)CC2COCC2N1C(=O)C=Cc1ccoc1 C(=O)(C(C#N)C(C)(C)C)NCC1(C)CCN(C(=O)CC(C)(C)C(F)F)CC1 C1(O)CCOCC1.C(=O)(C(F)CC1CCC1)CC(=O)N(CCC(C)NC=O)C C=C(C)C1OCCC1C(=O)NC12CC1CN(C(c1[nH]ccc1C)=O)C2 c1(C(N2C(CN(C(CC(CC)OC)=O)C)COCC2)=O)c(N)sc(C)c1C CC(C)C(C(C)NC(c1cnn(CCO)c1)=O)NC(=O)Cn1ccc(C2CC2)n1 c1(C(=O)NCC(CCNC(C(C)CF)=O)O)cc2c(s1)-c1ccccc1OC2 CCC(CN(C)C)CC(=O)NCC1(F)CCN(C(c2ocnc2C(F)F)=O)C1 C(C1CN2CC1C2=O)=CC.C1(C(=O)NCCOC=O)CCCCN1C c1(CC)cc(OC)c(OC)cc1C(=O)NCC(C1CC1)NC(=O)C(C)(C#N)CC CN(C)NC(=O)CCC(=O)N1CCC(CC(N2CCCC3(CC2)N=N3)=O)C1(C)C c1(SC)ccc(O)c(C(=O)NCC(c2ccc(F)cc2)NC(=O)C=CSC)c1 c1(CC(N2CC(C(C)NC(=O)Cn3cnc(Br)c3)C2)=O)ccc(OCCF)cn1 Cn1c(O)nc2cc(C(N3CCN(C(=O)CN=c4cc[nH]cc4)CC3)=O)ccc12 CC(N=c1nc2c(cnn2C)c(NCc2cc(C(F)F)no2)[nH]1)c1csc(Br)c1 C#CCC(C(=O)N1CC(c2nc(=O)o[nH]2)C1)NC(c1sccc1Cl)=O S(=O)(=O)(c1cc(C#N)ccc1F)N1C(C(N2CCC(C(=O)OC)C2)=O)CCC(C)C1 c1(C(N2CC(C)(NC(c3cc(C(C)=O)on3)=O)C2)=O)ccc(CC2CCC2)cc1 CC1(C)CC(NC(c2cocn2)=O)CN(C(=O)CC2=NNC(=O)C2)C1 CCCCC(O)CC(=O)N(CCC)CCNC(C1COCCN1S(C)(=O)=O)=O c1(-c2cc(NC(C3(C)N(Cc4occ(C)c4)CC3)=O)on2)ccc(Br)cc1 CC(C(=O)NC(C1CCCCC1)CNC(=O)CCCNC(C1CCC1)=O)C(F)F C1(NC(c2cccc(Cl)c2)=O)CCCCC1OC(F)(F)F.n12cc(nn1)CNCC2 C(=O)(C(O)CNC(=O)NC(Cc1ccccc1)C1CC1)N(C)C N1(C(C(CO)N(C)C)=O)CCC(O)(CNC(c2snc(O)c2Cl)=O)CC1 c1(C(N2C(C)CC(CNC(C34CC(C)(C3)C4)=O)C2)=O)cnc2[nH]nnc2c1 C(=O)(CCCS(C)(=O)=O)NCC(CNC(=O)CCC(=O)N(C)C)OC N1(C(c2cn(CC)nc2)C)CCN(C(C=C2CCNCC2)=O)C2CC12.C(C)=O c1(C(=O)NC(C)CNC(c2cscc2C(F)(F)F)=O)ccnc2cc[nH]c12 C=CCCCCCC(=O)NC1CC(C)(NC(=O)Cc2csc(C(F)(F)F)n2)C1 N1(C(c2n(CCC)nc(C)c2)=O)CC2CC(O)C1C2NC(=O)C#CC1CCCC1 N1(C(c2csnn2)=O)CCCC1Cc1cn(-c2cnsc2)nn1 C(CN=c1[nH]cnc(Cl)c1C#N)(C1CCCC1)NC(c1n(CC(C)C)ncc1)=O C(=O)(NNC(=O)C(C)(C)OC)c1ccc(OCC#C)c(C)c1 Cc1ccc(CNC(c2nsc(Cc3ccccn3)n2)=O)cc1 c1(C(N(C)CCNC(C2CCC23CCC3)=O)=O)cc2c([nH]1)CCCC2 c1(CC(=O)NC(CC)CN(C(=O)CCOC2CC2)C)ccc(C2CCC2)cc1 S(=O)(=O)(c1cc(C(=O)NCC2=NOC3(CNC3)C2)n(C)c1)NCC(C)C C(=O)(C(F)CCC(C)(C)C)N1CC2(C(NC(C(CCC)F)=O)CCC2)C1 C(=O)(C(C)(C)CC(=O)NCCn1cc(C(N2CCOC(C)(CO)C2)=O)cn1)OC C1(C(N2OCC(n3cc(COCC)nn3)C2)=O)CC12CCS(=O)(=O)CC2 N1(C(C(CNC(c2ccc(CO)o2)=O)N(C)C)=O)CCS(=O)(=O)CC1 Cc1cc(-n2cc(C(N3CC(COC45CCCC(C4)OC5)C3)=O)nn2)ccc1N C1(C(=O)NC23CC(CNC(C4N(C)CC4)=O)(C2)C3)CCCC1C1CC1 Cc1c(C(N2CCCC(n3cccc3)C2)=O)cc([N+](=O)[O-])cc1[N+](=O)[O-] N1(C(c2c(C)cns2)=O)CCC(C(C)(C)C)(CNC(=O)CCCF)C1 N#Cc1cccc(NC(=O)CN2CCNC(CC(F)F)C2)c1 CCCC(C)(O)CC(=O)NCC1(O)CCN(C(=O)C(C2CCCO2)C2CC2)CC1 C(=O)(CCCCCCCC1CC1)N1CCC(Cc2cc(OCC)no2)C(C)C1 c1(C(N(C(C)C)CCNC(=O)CCCCN(C)C)=O)cnc2[nH]cncc1-2 C1(OC)CC2(C1)CN(C(=O)C(CC(N)=O)NC(c1csc(F)c1)=O)C2 C1(NC(=O)C=CCO)CCN(C(=O)C=CC2CCC2)CC(O)C1 CCCC(CCC)C(C)(c1nnnn1CCOC)NCCC=CBr c1(C(c2n(CC=C)nnn2)NC2CCCC2)ccc(OCC(N)=O)c(OC)c1 c1(C(=O)NC(CNC(CC(CC)C)=O)(C)CO)c2c(nn1C)CN(C(=O)OC)C2 C12(NC(C(F)=CCC)=O)CN(C(=O)Cc3c[nH]c(=N)nc3O)CC1CS(=O)(=O)C2 C(C1=CCNCC1)NC(CC(C1CCN(C(c2ccccc2F)=O)CC1)C)=O C1(CC(F)(F)C(F)(F)Br)C(=O)N1.C1(C(C)C)CN1C.CO c1(C(N2CCN(CC3CN(C(C(CC)C)=O)C3)CC2)=O)cccc2c1OCCO2 C=C(C)CCCC(=O)N(C)Cc1cccc(CNC(=O)C(C)Cn2cccn2)c1 CC1CCc2n[nH]cc2C1C(=O)NC1CC(CCNC(c2ccc[n+]([O-])c2)=O)C1 c1(C(=O)NCCNC(C2CN(C(C3C(C)CC(=O)N3)=O)C2)=O)ccc2cc[nH]c2c1 C1(N(C(C)(C)CCOC2CC2c2ccccc2)C(C)C2CC2)CCn2ccnc2C1 N1(C(c2c(CC)nn(C)c2)=O)CC(O)(C2(CNC(c3nnc(S)n3C)=O)CC2)C1 c1(NC(C(c2cc(C)cc(Br)c2)N2CCC(O)C2C)=O)ccc2c(c1)OCO2 C1(F)(CNC(C2(OC(C)=O)CC2)=O)CCC(NC(c2cccc(C)c2)=O)C1 Cc1ccc(C(=O)NC(C)(CNC(=O)C(O)Cc2ccc(Cl)cc2)CO)cc1C N1(C(c2c(NC)nc(C)cc2)=O)CCC2CCN(C(C3CN(C)C(=O)N3)=O)C2C1 Cc1ccc(SC(C)C(=O)NCC(C)N(C)C(c2cnc(C(C)C)[nH]2)=O)cc1 C(C(=O)NCC(CCNC(=O)CNC(c1ccccc1)=O)OC)(C(C)C)SC Nc1c(C(=O)NCCCCC(CO)NC(=O)CCc2cccs2)cccc1F CCC(F)(C(=O)OC)C(=O)NCC(C)CNC(C1(Sc2ccccc2)CC1)=O c1(CNC(=O)NCc2c(C)ncc(N)n2)nccc2ncccc12.C12(CC1)C(=O)N2 C1(CNC(CC(=C)C)=O)CC2CCC1N(C(C1CC=C(C)CC1)=O)C2 N1(C(c2ncc(C(=O)OC)nc2)=O)CCOC2CN(C(=O)C(C)P(C)(C)=O)CC12 c1(NC(C(=O)N(CC(CCCC)O)CCOc2ccccc2)=O)nc2ccccc2s1 S(=O)(=O)(c1nc(N2CC3CCC(C2)C3O)ccc1Br)N(C)C c1(C(N(CCCNC(=O)CC2(OC)CC2)CC)=O)cnc2c(c1)NC(=O)CN2 C(=O)(CS(=O)(=O)CCO)N(CC(C)NC(=O)CC1CC(C)=NO1)CC C12(NC(CCCC#C)=O)CN(C(=O)CCN3CCOC3=O)CC1CS(=O)(=O)C2 c1(C(C(=O)N(C2CC23CCC3)CC(=O)NC(COC)C2(C)CC2)C)ccccc1 N1(C(C(C)S)=O)CC2CN(C(c3cccc(N4CCOCC4)c3)=O)C2C1 C(C(C)(O)CC(=O)N1CC(n2cc(-c3ccc(N)cc3)nn2)C(C)C1)OC c1(CN2CC(NC(C3CC4CC4C3)=O)C(F)C2)ccc2oc3ccccc3c2c1 C1(N(C(c2csc(Cn3ccnc3)n2)C(=O)NCC)C)CCCCCC1 c1(C(N2CC(O)(CN(C(c3n(C(C)C)ccn3)=O)C)C2)=O)cc(N)c(O)c(F)c1 C(CCCCC(=O)NC1CCCC1(C)O)NC(c1n(C)ncc1Cl)=O c1(CC)nsc(N(CCCNC(=O)C(=O)Nc2cnn(C3CC3(F)F)c2)C2CC2)n1 c1(C(=O)OCc2ccc(C)c(C)c2)nc2ccc(F)cn2c1N c1(OC)nc(N2CCCC3(NC(c4oncc4C)=O)CC3C2)nc(C)c1F c1(C(N(C(CNC(C(C(CC)C)C)=O)C2CC2)C)=O)cccc2c1CCCC2 N1(C(C(C)(C)C(F)(F)F)=O)CCOC2(CCN(C(=O)C=C3CCC3)C2)C1 C1(CC(=O)NC(C2CCCN(C(=O)Cn3ccnn3)C2)C)CCC(F)(F)CC1 c1(C(N2CC(NC(CNC(N)=O)=O)CC3(C2)CC3)=O)nnc2ccccc2n1 C1(C(N2C(COC)C=CCC2)=O)CN(C(C2CCC(O)CN2C)=O)CCN1C c1(CNN2CC(C(=O)Nc3ccn(C(C)(C)C)n3)C2)ccc(Br)c([N+](=O)[O-])c1 Cc1nn(C)cc1CCC(=O)NC1C2CN(C(=O)CNC(=O)NC3CC3)CC12 C1(C(=O)NCC2N(C(c3c(C)cco3)=O)CCC2)CC12CC(C)(C)C2 C(CC(C(=O)NCC(C)CC1CC1)NC(=O)CC1CC(OC)C1)=CC c1(C(N(C)CC2N(C(CCNC(C3C(C)C3)=O)=O)CCC2)=O)cnn2ccncc12 N1(CC(C2CCC2)OCC)CCC(NC(=O)CN2C(=O)CCC2=O)CC(C)(C)C1 N12CC3(CCCCC3)C1C2=O.C1(C(=O)OC)(OC)CC(O)C12CCC2 N1(C(Cc2c(C)ccnc2)=O)CCC(CC(=O)Nc2cnc(Cl)cc2)C1(C)C CC(CCC(=O)N1CCC(F)(F)C1)NC(=O)CCc1nncn1C Cc1cccc(C(=O)NC(C2(O)CN(C(=O)C(O)CN3CCOCC3)C2)C)c1F c1(C(=O)NC(CNC(=O)Cn2nc(O)ccc2=O)CO)cc2n(c1)CCOC2 c1(C(=O)NC(CN(C)C(c2n[nH]cc2Cl)=O)(C)C)cc(OC(F)F)cc(Cl)c1 N1(C(c2cc(C)nc(Cl)c2)=O)CCOC2(CCN(C(=O)C(F)(F)C(F)F)CC2)C1 CCC(CC(C)C)C(=O)NC1(C2CN(C(c3cncc(C)c3Cl)=O)C2)CC1 N1(C(CCC2OCC(C)(C)C2)=O)CC2CCCC2(NC(c2c[nH]c(=N)s2)=O)C1 c1(C(=O)NCC2CCN(Cc3cc[nH]c3)CC2)ccc2nc(Br)sc2c1 C#Cc1cc(C(N2CCCC2CCNC(c2cscc2Cl)=O)=O)ccc1C c1(N2CCC(CC)(CC)C2)cc(NCc2ccccc2OC)nc(C)n1 C(=O)(CC1=CCOCC1)NC(C(C)NC(CCc1cccc(C(=O)OC)c1)=O)C CC(C)(F)CCC(=O)N1CC(C(=O)NC2CCC3(CC2)CC3)CC12CC2 c1(OC)cnc(C(N2CCC(C(=O)NCC3(CCO)CCC3)(OC)C2)=O)cn1 c1(C2(C(=O)N)CC2)ccccc1Cl.C(=O)(C(CC1(C#N)CC1)N(N1CCCCC1)C)NC c1(SC)cccc(C(=O)NCCOC2CCN(C(c3cc(Cl)n(C)n3)=O)CC2)c1 CCC1CCNS(=O)(=O)c2cc3c(cc2)NC(=NC1)C=C3.C1(F)(NCC)CC1 C1(C(=O)NC(CNC(C(C(C)C)NC=O)=O)(C)C)CC(=O)NC1(C)C C(=O)(CCCC(F)(F)C(F)(F)F)NC(C)C(C)(C)NC(C1CCS(=O)(=O)CC1)=O C(=O)(CC1=CCOCC1)N1C2CN(C(C3C(C)(C)S(=O)(=O)CC3)=O)C(CC2)C1 c1(C(N2CCN(C(C(C=C)O)=O)CC(C)(C)C2)=O)ccccc1S(=O)(=O)CC C1(C(=O)NCC(CCCC)O)CC2CN(C(=O)CC(F)(F)F)CC2C1 CSC1=C(C(=O)N(C2C3CC(O)C2N(C(C2CN4CCCN2CC4)=O)C3)CC)CCCC1 C(=O)(C1=CCC(NC(C2C=CCCC2)=O)C1)NCc1n(CCC)cnc1 c1(C(C(=O)NC2CC3CC3C2)N(C)CCc2ccccc2)cc2occc2s1 CCC(CC(=O)NCC(O)CN(C)C(C1CCN(C)C1=O)=O)c1ccccc1 C1(C(=O)NC2(COC)CC2)CCC2(CC2)N1C(c1cc(CO)nn1C)=O CCCN=C(NCCC(C1CCC1)Oc1cccc(SC(F)(F)F)c1)NC(C)C c1(NC(C2CCC(NCc3cccc(OC)c3F)C2)=O)cnc2c(c1)CC(=O)N2 c1(N2CC3CC(NC(c4cc(C)oc4C)=O)C3C2)cc2nnc(C(C)(C)C)n2cn1 CC1CC(C)(C(=O)NC2CC(F)(CNC(C3(C4CCCCO4)CC3)=O)C2)CCO1 C1(NC(=O)C2=CCSC2)CC2CCC1N(C(=O)Cn1cc3ccccc3n1)C2 c1(NC(COC)C(C)OC2CCCC2)sc2ccccc2c1CSC C1(C(=O)NCC2CCCN(c3ccnc(CC(C)C)n3)C2)CC(=O)CC12CCC2 n1(CC(=O)NCCC(CCNC(C(CC)COC)=O)C)nc(O)ccc1=O N1(C(c2c(CC)cccn2)=O)CC(CNC(=O)CCC(=O)NC)C2(CC2)C1 C12(NC(CCC(=O)NC)=O)CCC1CN(C(=O)C(C)CO)C2 c1(CC(=O)NC2(COC)CN(C(CC3(OC)CC3)=O)C2)cccc2ccccc12 c1(CN2CCCC(CCNC(c3ncc(C)nc3)=O)C2)cc(Cl)c(O)c(Br)c1 C1(C)(CCOC)CN(CC2C(C(=O)OC)COCC2)CCO1.c1(S)ccccc1 C1(CC(=O)NCC(C)(C)NC(c2nocc2Cl)=O)CC2(CCCCC2)CO1 C(=O)(C(=O)CC(C)C)N(CCCNC(CCC(=O)NCCC)=O)C(C)C C(=O)(CC(CC)C(F)F)N1CC(NC(C(CC)=CC)=O)C(c2cnn(C)c2OC)C1 Cc1cncc(-c2cn(CCc3ccc(N(C(=O)C(C)C)C(C)C)cc3)nn2)c1 C12(NC(C3C=CCC3)=O)CC3CCC(C1C2)N3C(c1coc(O)n1)=O N1(C(c2c(N)sc(C)c2C)=O)CCCCC(NC(C2CCCN2C(C)C)=O)CC1 O=C(CONC(=O)C1CCSC1)N1Cc2ccccc2CO1 C(CN=c1[nH]c(C2CCCCC2)nc(=N)[nH]1)C(COC1CCCC(C)C1)=O C1(CNC(c2c(CC)c[nH]n2)=O)C2CCC(C2)N1C(C1(c2ccncc2)CC1)=O C1(NC(C(COC)NC(C(CC)N(CC)CC)=O)=O)CCCC1N=[N+]=[N-] N1(C(C2(c3ccc(C)cn3)CCC2)=O)CC2CCC(C1)N2C(=O)Cc1nncs1 N1(C(C(CC(C)C)NC(C)=O)=O)CCC2(C1)CN(C(=O)CCC(=O)OC(C)(C)C)C2 C(=O)(CCC(O)C(C)(C)C)N1C2CC(NC(C3C(C)CCO3)=O)CC1CC2 N1(C(c2nc(C)c(C)[nH]2)=O)CCCC(CCNC(c2ccncc2F)=O)CC1 C12(NC(C(CC)SC)=O)CCC(NC(=O)C(C)Oc3ccc(Cl)cc3)(CC1)C2 N1(C(C(C2CC(F)(F)C2)OC)=O)CCC(CN(C(=O)CC2CC=CC2)C)C1 c1(CC2N(C(=O)Nc3ccnn3-c3ccccc3)CC=C2)ccc(F)c(Br)c1 c1(CNC(CC(=O)O)C2CCCCC2)cncc(Cl)c1Cl Cc1cc(C(N2CCC(C)C(NC(=O)COc3ccon3)C2)=O)c(C)nc1C Cc1ccc(C(C)NC(C2CC23CC(NC(c2csc(C)c2)=O)C3)=O)cc1 C12(CC(=O)NCC3(F)CC(NC(CP(C)(C)=O)=O)C3)CCC(CC1)OC2 C1(C(=O)NCC(C=C)(C)C)N(C(=O)C2=CCCOC2)CCCC1(C)C N1(C(Cc2c(C)cccc2)=O)CC2CN(C(c3n[nH]c(C)c3[N+](=O)[O-])=O)CCC12 N1(c2cc(C3C(C)C3)[nH]n2)CCN(C(C2CCC(Cl)CC2)C(=O)NCCF)CC1 C1(C(=O)NC(c2ccc(C)cc2)CC(=O)OC(C)(C)C)CCOC(=O)CC1 c1(CN2C(C(N3C(CC(=O)OCC)CCCC3)=O)CC(O)C2)cc(F)ccc1O c1(OC)ccc(C(C)NC2CC2)cc1OC.C12CCN(CC1)C(C1CC1)C(=O)N2 N(C(=NCCCCc1ccccc1)NC1CCC1)C1CCN(Cc2occc2)C1 c1(CC(=O)NCC2C(CNC(COCC)=O)C2)cccc(C#N)c1 N1(C(c2nccc(C(N)=O)c2)=O)CCC2(CNC(=O)C#CC3CC3)CCCC12 C(=O)(C(CO)C(C)(C)C)N(C(CC(=O)OC)C)Cc1ccccc1 n1(CCC)nc(C)c(C(=O)NC2CN(C(c3cncnc3CC)=O)C3CC23)c1C C1(NC(CC(=O)NC)=O)CN(C(=O)C(C)OCCOC)CC1C c1(OC)ccc(SC(c2sc(C(C)=O)nc2C)=O)cc1 c1(CC)cc(C(=O)NCC23CCCN(C(c4ncn(C)n4)=O)C2C3)c(C)nn1 c1(C(C)C(=O)NCC(CO)NC(C23CCC(CC2)CC3)=O)cc2ccccc2o1 Cc1cc2ccc(C(N3CCC(O)(C(C)CNC(=O)CCC(N)=O)C3)=O)cn2c1 C1(C)(NC(C(N2CC(C)C2)C)=O)CCCC1NC(c1ccc(CCO)cc1)=O CC(CN(C)C)CC(=O)NCC12CC(CN1C(=O)Cc1ccc(C(F)(F)F)cc1)C2 c1(C(=O)NCCC2CCN(C(C3COCCO3)=O)C2)cccc2c1CCCCC2 N1(C(=O)Cc2cc(C(F)(F)F)ccc2Cl)CCSc2c([nH]c3ccccc23)C1 Cc1scnc1C(=O)NC(C)C(C)NC(=O)C=CCN1CCCC1 C(C1C(C(N2CCCC2CC(=O)NCCC2CCCC2)=O)C1(C)C)=C(C)C N1(C(CC(CCC#C)O)=O)CCCC12CCCN(C(c1nn(C)cc1Br)=O)C2 C1(NC(c2n(C)cnc2)=O)CCN(C(C2CC3(C2)CC3(F)F)=O)CC12CCC2 C(=O)(CC(C)C(F)F)N(C1CCCN(C(C2C(C(C)=O)C2(C)C)=O)C1)CC1CC1 c1(C(=O)NCCN(C(=O)C(C)(C)C2CC2)C(C)C)ccc2c(c1)NC(=O)CCN2 c1(NCC(C)(C)C(F)(F)F)nc2ccccc2nc1NCc1ccc(F)cn1 Cc1ccc2c(c1)CCC(C(=O)NCC1CCCCN(c3ncc(O)cn3)C1)O2 C(=O)(CN=c1[nH]c(N2CCN(CC(F)(F)Cl)CC2)nc2c1CCC2)NCCC C1(NC(=O)CC(C2CC2)C2CC2)CN(C(C2CCC(=O)N2)=O)CCC1O c1(COC)nc(C)c(C(=O)NC2CC(NC(C3(CC4CC4)CC3)=O)C2)s1 CC1CCN(CC(N2CCCC2CN(C(C2(F)CC=CC2)=O)C2CC2)=O)C1 c1(OC2CC(CS(N3C(CSC)CC(OC)C3)(=O)=O)C2)ccc(C#N)nc1 N1(C(c2c(C)nc(C3CC3)s2)=O)CCCC(C)(NC(C2CCCC(C)(C)O2)=O)C1 N1(C(C=C(C)c2ccsc2)=O)CC2(CCCCN2C(=O)CC2CCOC2)C1 c1(OCCNC(=O)NC2CC23CC3(F)F)cccc(F)c1F C(CC(C)C)(C(=O)N1CCC(CNC(C2(OC)CCC2)=O)CC1C)OC C#Cc1ccc(C(N2CCCC2C(C)(C)C(=O)NCC2CCC2C)=O)cc1 Cc1nn[nH]c1C(=O)NC(C)(C)CNC(=O)CCC1CCCC1O c1(C(N2C3C(CNC(CCC(C)SC)=O)C(C3)C2)=O)coc2ccc(Cl)cc12 c1(-c2nc(C(N3CCN(c4cccc(Cl)c4)CC3)C)on2)ccc(Cl)c(F)c1 O(NC(=O)C(CNC(=O)C(C1CCC1)OC)C(C)(C)C)CCCCC C1(C2CN(C(CCCn3cc(C4N(C)CCC4)nn3)=O)C2)OC(=O)CC12CCC2 Cn1c(O)nc2cccc(C(N3C(CNC(c4cnn[nH]4)=O)CC4CC34)=O)c12 C(CC(=O)NC(c1snnc1C)C)(C(F)(F)F)NC(c1ccn(CCC)n1)=O c1(N2CCC(NC(c3ccc(CCC)cc3)=O)C(F)C2)ncc(C#N)cc1F C1(O)(CNC(CC(C=C)CC)=O)CCCN(C(c2ccnn2CCC)=O)CC1 N1(C(c2n(C)nnc2)=O)CCC(C(N2CCOC3CC23)=O)CC1(C)C N1(Cc2ccc(C)cc2)CCC(F)C(NC(c2ccnc(CCO)c2)=O)C1 Cc1nc(-n2nc(Cc3cnn(C)c3)nc2-c2cnn(CC(C)C)c2C)n(C)n1 CON1CCC(C(=O)NCCCN(C)C(C2CCC(C3CC3)C2)=O)CC1 C1(CC(=O)NCC(=C)Cl)CC(O)CN1C(=O)CN1CCCCCC1 CC1(C(=O)NCC2CC(F)(F)C2)CCN(C(=O)COCc2cccnc2)CC1 C1(CNC(C2(COCC)CC2)=O)CC2CC(C1)N(C(=O)C#CC(C)(C)C)C2 c1(CCC)ccc(C(N2CCC(N(C)C(c3sncc3C)=O)C2)=O)cc1N C1(C(N2CCC(CNC(C3CCCNS3(=O)=O)=O)C2)=O)CC2(COC(=O)N2)C1 C1(C(=O)NCC(C)N(C(CCOc2ccc(C)cc2)=O)C)CCCC(F)(F)CC1 c1(C(N2C3CCC2CN(C(C2CC2C2CC2)=O)C3)=O)ccc(F)c(F)c1Br C1(C(N2CC(C(C)NC(=O)CC3CCC(C)(C)O3)C2)=O)OCC2CCCC12 C(=O)(C(CC)C(=O)NC1COCC1C(=O)NCc1nn(C)c(=O)n1C)OCC CN1CCN(C(C2CCC3(CC2)CC3)=O)CC1CNC(=O)C1=CC(C)(C)C1 c1(CC)cccc(C(N2CCCC2CF)C(=O)NC2CC2)n1 N1(Cc2cn(CCCCC(=O)O)nn2)CCC2(CCCO2)CC1 N1(C(C(C)C2CCCC2)=O)CC(N(C(=O)Cn2ncnn2)C)C2(CC2)C1 C1(CNC(C2CC(C)(C)OCC2O)=O)CC2(CCN(C(C3(C)CCC3)=O)CC2)C1 CC(C)CC(O)CC(=O)NC1CCN(C(=O)Cc2cc(Cl)cc(Cl)c2)C1 c1(NC2C(OC)COCC2)nc(=NCC2CC3C(C2)C3(F)F)[nH]c2c1COCC2 N1(C(C2C(C)=CCS2)=O)CCC(C(N2CCSC3CC23)=O)CC1 C1(C)(CC(C)C)CN(Cc2cccc(C(=O)N(C)Cc3cccnc3)c2)CCO1 c1(C(C(=O)NCCOC2CCN(C(C3(C(C)C)CCC3)=O)C2)C)ccc(F)cc1 c1(C(=O)NC2CC(CCNC(C3(C)CS(=O)(=O)C3)=O)C2)cccc2[nH]c(=N)oc12 c1(NC(C)=O)ccc(C(=O)NC2CCN(Cc3nc[nH]n3)C23CC3)c(F)c1F c1(N2CCC(C(=O)OCCOCC)CC2)nc2ccccc2o1 c1(C(N(C)CC2COCCN2C(=O)C2=CCCS2)=O)nn(C)c(Cl)c1Cl n1(CC(=O)N(CCNC(c2c(C)coc2)=O)C2CC2)nnc2ccccc2c1=O C1(C(C(=O)N(CCCCC)C(C)C)C)CCCN(C(c2ccn(CC)n2)=O)C1 C1(NC(=O)CCn2cnnn2)CCOC(C(=O)NCC2(CO)CCCC2)C1 C(CC(=O)NCc1cn(C)cn1)(C1CC1)NC(CC=C)=O c1(CCC(CO)NC(C)Cc2ccc(F)cc2)ccc(Br)cc1 N1(C(c2c(C)ncs2)=O)CC2CCC(NC(c3cc(C4CC4)[nH]n3)=O)CC2C1 N1(C(c2c(CC)csc2)=O)CCN(CC(C)NC(=O)C(C)CC2CC2)CC1 CC1(C)CC(NC(=O)CC2(C)CC2(Cl)Cl)CCN(C(c2nc(Cl)cs2)=O)C1 C1(C(=O)Nc2ccc(C)nc2)CN(C)CCN1C(=O)C=Cc1nccs1 C1(C(N(CCC(CC)NC(=O)Cn2nccc2C)C)=O)CCN(CCF)CC1 C12(CNC(CCC(CC)OC)=O)CCN(C(=O)COC3CC3)CCC1C2 c1(C(N(C(CC)CNC(C2CC(C(F)F)C2)=O)C)=O)oc(SC)cc1C Cc1nn(C)c(C)c1C(=O)NCC1CCN(C(c2cc[nH]c2C2CC2)=O)CC1C N1(C(C2(CC(C)C)CC2)=O)CCC2(CC1)C(NC(c1nccn1C)=O)CS2(=O)=O N1(C(Cc2ncc(C)s2)=O)CCCC(NC(=O)C(C2CCCC2)C2CCCC2)C1 CCCCC(C(=O)N(C1CCCCC1)CCNC(=O)CCN(C)CCO)C(C)C C1(C(N2CCC(C(CNC(C3CCCCC3F)=O)O)CC2)=O)CCC(F)(F)CC1 Fc1ccc(C(c2nnnn2CCC2CC2)NC2(CCO)CCOC2)c(F)c1 c1(C(N2CCC(C#N)(C(=O)NCCc3c(C)ncs3)C2)=O)n[nH]c2c1CCCC2 C(CCCCC(=O)NCC1CC1NC(C1CC(c2ccc(C)cc2)C1)=O)OC C#Cc1ccc(C(=O)NCC(CC=C)C(=O)N2CCOC(COC)C2)c(C)c1 c1(OCC(=O)NC2CC(O)CN(C(c3ns[nH]c3=O)=O)C2)ccc(F)c(Cl)c1 CC1(O)CCN(C(=O)CC2(C)CCCN2C(=O)C(F)=CC2CC2)CC1 c1(C(c2nnnn2C2CC(F)(F)C2)NC(c2nccs2)CC)cnc(O)s1 C1(CC(N)=O)(NC(C(C)SCC)=O)CCN(C(C2(C)CCC(C)C2)=O)CC1 c1(OC)cccc(OCCCN2CCC(C(=O)NCC3(CC(=O)N)CC3)C2)c1 C1(C(=O)NC2CCC(NC(C(CC)SC)=O)C2)CCC2(CC1)CC(=O)C2 CCC(C)(CCNC(=O)CCOCC1CCC1)NC(=O)C(c1ccccc1)C c1(N(C)C)ccccc1SCCCC(=O)N1CCCC1C(=O)NC1CCC(O)C1 CC(C)C(CCN(C)C(C1CCNC(=O)C1)=O)NC(=O)Cc1cc[nH]c(=N)c1 C(CCC(O)C(=O)NCC1CCCCS1)NC(C1CC(C#C)(O)C1)=O c1(C(N2CC3CN(C(c4c(C)cco4)=O)CC32)=O)c[nH]c2cc(Cl)ccc12 O=C(C1=CCCN(C(=O)CCC2CC(OC)C2)C1)NC1COC2(CCCC2)C1 c1(OC)ccc(C)cc1C(N1CCN(C(=O)C=CCSC2CCCCO2)C2CC12)=O CC1CN(C(c2cnc3n2CCC3)=O)CC(C)N(C(=O)C(c2ccccn2)O)C1 N1(C(Cc2c(OC)cccc2)=O)CCN(C(c2cn(C)nc2O)=O)CCC1C C(=O)(C1=NOC(C)C1)NCCNC(C(C(C)O)NC(=O)C1CC1)=O C1(c2cn(Cc3scc(C)n3)nn2)(NC(C2CC23CC3)=O)CC2(CC2)C1 Cc1ccc(C(N2CCCC(N(C)C(C3(C(N4CCSCC4)=O)CC3)=O)C2)=O)cn1 C1(Cc2cc(CNC(=O)NN=c3cncc[nH]3)on2)CCC2(CCOCC2)C1O C1(CNC(C(C)N2CCC2)=O)CN(C(C2CCOC3(CCC3)C2)=O)CCC1(F)F C(CCN(C(=O)C(N1CCOC1=O)C)C)(C(C)C)NC(C(C)SC)=O N1(C(C(=O)Nc2cc(NC3CCC3)cc(OC)c2)C)CCOCC(C2CCC2)C1 C1(C(=O)N)CCC(CCOC)NC1=O.C1(CC#C)(C(=O)NC)CCOCC1 CN1CCC(=CC(N2CCC(CCNC(C3C=CCCC3)=O)CC2)=O)CC1 N(C1CCCc2n[nH]cc21)C(C(CC)NC(C)=O)=O CC(C)(C(=O)NN=c1[nH]c(Cl)c(Cl)nc1Cl)N1CCCCCC1 CC1CC2CN(C(=O)CNC(=O)CCCF)CC12.C12CN(C1)C2=O N1(C(CCc2ccc(C)o2)=O)CCC2(CC1)CC2C(=O)NCc1c(C)n[nH]c1C c1(NC(N2CCC(CCC3CCN(C(C)=O)CC3)C2)=O)cc2c(s1)CCCC2 N1(C(Cc2c(C)nc(-c3ccc(Cl)cc3)s2)=O)CC(C(=O)O)CC(F)(F)C1 CCCCS(=O)(=O)N1CCC(N2CCC(Oc3ccc(Br)cc3)CC2)CC1 c1(C(=O)NCC2CC(OC)CN2C(=O)CCNC(C2CCC2)=O)cncn(C)c1=O N1(C(C2CCN(C)C2=O)=O)C(CC(=O)NCc2ccc(Cl)c(O)c2)C2CCCC12 C1(C(N(C)CCc2cnccn2)=O)CCN(C(=O)c2cncc(Cl)c2)O1 C1(NC(CC2(CN(C)C)CCC2)=O)(CF)CN(C(=O)Cc2cn(C)nn2)C1 c1(COCC(=O)N(C2CC(NC(C(C)=C)=O)C2)C)ccccn1.C1(C)CC1 C1(COC)(NC(C2(O)CCC2)=O)CCCN(C(=O)Cn2nnc(C)n2)C1 CCC(C)(C(F)(F)F)NC(c1cccc(-n2nnnc2O)c1)=O C1(C(F)(F)F)(C(N2CC(CNC(c3scnc3Cl)=O)OCC2)=O)CCCCCC1 C1(C(N(CC(CC)OC)C)=O)(NC(C2COCCO2)=O)CCC(C)(C)C1 Cc1cccc(C)c1C(=O)NCC(C)CN(C(=O)C(C)(C)c1ccccn1)C CN1CCN(C(C2COCC2C(=O)NC2CC(C)(C)CCO2)=O)C(CCO)C1 C1(C(F)(F)F)(C(=O)OC)CC(C)(C)C1.C12CCN(C1)C(=O)C1(CCC1)NCC2=O N#Cc1cscc1C(=O)NCC12CC(C(N3CCCC(CN(C)C)C3)=O)(C1)C2 C(=O)(CC(O)CC(C)C)NCC1(C(=O)NC(C2CCOCC2)C#C)CC(C)(C)C1 c12ccc(c(OC)c1)OCC(=O)N2.CCC(CNC(=O)NC=O)(CO)OC c1(C(=O)NCCN(C(C2CC(F)(F)CS2)=O)CC)ccccc1-n1ccnn1 C1(NC(Cc2c(C)con2)=O)CCCCC12CCN(C(c1ccc(O)cc1)=O)C2 CCCCC(O)C(=O)N1CCC(CO)(CNC(C2(N(C)C)CCC2)=O)C1 C1(CNC(=O)Cc2ccc(F)cc2)CCCCCC1NC(=O)CC1CC2CC2C1 C(CC(=O)NC(CO)C1CCC1)(C(F)(F)F)NC(CN(C(=O)OC)C)=O C(=O)(C(CC(C)C)N(C)C(c1cnc(O)cc1C)=O)NCC(C)OCC=C N(C1CCCS(=O)(=O)c2ccccc21)C(N1CCOC(C2CCCOC2)C1)=O CCCCC(C)(F)C(=O)N1CCC(CN(C(c2cnsc2)=O)CC)CC1 C1(C)(COC)CC(NC(c2ccnn2C(C)C)=O)CN1C(=O)COCC1CC1 CC(C)S(=O)(=O)CC(=O)NC1CCCCC1CNC(C1CCCC12OCCO2)=O CCCCC(CO)NC(C1CN(C(=O)Cc2cscn2)CC1F)=O CCCCC(=O)C(=O)NC1C2CCN(C(=O)Cc3csc(C)c3)CC12 Cc1oc2ccccc2c1CNC(c1cc2ccccc2o1)c1nnnn1C1CC1 N1(C(c2n(CCC)ccc2)=O)CCCC2CN(C)CC12 CCC(C)(C)C(=O)N1CCN(C2CCCN(C(=O)CC3CCNC3=O)C2)CC1 S(=O)(=O)(c1ccc(C#N)c(NC(C2COCCO2)C)c1)N(C(C=C)C)C c1(C2C(NC(=O)Nc3cc(Cl)ccn3)C2)cn2ccccc2n1 C(=O)(CCCCCCN=[N+]=[N-])N1CCC(N(C)C(c2cc(=O)n3nccc3[nH]2)=O)C1 n1(CC)nc(C(=O)N(C)CC2CCN(C(C3CC4CC3C4)=O)C2)cc1C N1(C(C2C(C(=O)OC)C2)=O)CC(CNC(=O)C(F)(F)CC2CC2)CC1(C)C C1(C(N2CC(CC)C2)=O)CCC2CCC1N2C(=O)CS(C)(=O)=O c1(CO)ccc(Br)cc1C(N1CC(C)C(NCc2c[nH]ccc2=N)C1)=O C1(C(C)(C)O)(CNC(CCNS(C)(=O)=O)=O)CN(C(=O)CCCF)C1 N1(C(c2nc(OCC)sn2)=O)CC2CC(C)N(C(C3(OC)CCCCC3)=O)C2C1 Cc1[nH]c(C)c(C(=O)NC(C2CCCN(C(c3ccc(Cl)nc3O)=O)C2)C)c1C CCC(CNC(=O)C(CC(C)C)NC(=O)OC)N=c1nc(C(C)(C)C)[nH]s1 C1(CC#C)CCC(CNC(=O)COC2(OC)CCOCC2)CC1 C1(CC(N2CCOCC(NC(C(C)=C(C)C)=O)C2)=O)CCc2sccc2C1=O C(CN=c1[nH]c2cc(F)cc(F)c2o1)C1CN(C(C23C(C)OC(CO)(C2)C3)=O)C1 C12(C(N(CCNC(=O)C(C)Oc3cccnc3)CC)=O)C3CCC(CC13)C2(F)F Cc1ccc(O)cc1CNC(=O)COC(C)(C)CNC(C1CC2CCCC2C1)=O N(C(=NCCNS(C)(=O)=O)NCC1CCC(C#N)CC1)CC(C)C C(CC(CNC(=O)CO)NC(=O)C(C)(c1ccccc1)Oc1ccccn1)OC C(=O)(C1=NN(CCO)C(=O)CC1)N1CCC(N(C(C2CC(C)OC2=O)=O)C)CC1 C1(CCC)(NC(c2nc(Cl)sc2Cl)=O)CCN(C(c2cn(C(C)C)nn2)=O)CC1 c1(CNC2CCC(C(=O)NCC(O)CO)C2)cc(Cl)nc(Cl)c1 N1(C(CCC=C=C)=O)CC(C2CC2)(C(=O)Nc2cncc(C(N)=O)c2)C1 C(CC(C)C)(C(=O)N1CCN(C(C2CC2OC)=O)C(C)C1)CC.CC(=O)NC Cc1cc(C=CC(N2CCC(CN(C(=O)CCc3cnc[nH]3)C)C2)=O)c[nH]c1=N C(=O)(C1=CCCCC1)N1CC(C(C)NC(C2CCC(C)O2)=O)C1 C(N=c1cc(C)[nH]cc1C#N)C1CCN(C(CSSC)=O)C1 Cc1ccc(C(c2nnnn2C2CCCC2)NCc2ccc(Cl)o2)cc1[N+](=O)[O-] N1(C(C=CC)=O)CCN(C(c2ccc(C3CCCCC3)cc2)=O)C2CCCC12 N1(C(c2ccc(NC(C)=O)cc2)C(=O)NCC(C)C)Cc2nn(C)c(N)c2C1 c1(OC(C(N2C(CNC(CCC=C)=O)C=CC2)=O)C)cccc(C#N)c1 N1(C(C(C)(C)OC(C)=O)=O)CC(NS(=O)(=O)c2ccccn2)CCC(O)C1 C1(C(=O)NC2CC(N(C)C(C34CCN(CC3)C4)=O)C2)CC2CC1C1CC21 c1(-c2ccc(C(N3CC4CCCC3CC4)=O)c(F)c2)cc(F)c(C)c(F)c1.CNC Cc1ccccc1C(=O)NCC(=O)NCC12CC1CN(C(C1(O)CC(F)(F)C1)=O)C2 C1(C(N2CC3C(N(C(CCCSC)=O)C)C3C2)=O)CCC2(CC1)CNC(=O)C2 c1(NC(C)C)cccc(C(N2CC3CC3(CNC(C3(O)CC3)=O)C2)=O)c1 N1(C(C(C)(C2CC2)OC)=O)CCC(C2CC2)(NC(c2ccc(S(N)(=O)=O)s2)=O)C1 N1(C(CCC2(C)N=N2)=O)CC(OCc2ccccc2)C2(CC2)C1 C12(CC=C(CCC=C(C)C)C)CN(C(=O)OCc3ccccc3)CC1CCO2 c1(CC)ccc(C(=O)NC2CC(NC(C3(C)CCC3)=O)C2)cc1[N+](=O)[O-] c1(C(N)CO)cncc(N(CC(O)CF)C(=O)NCC(F)(F)C(F)F)c1 c1(OC)cccc(Cl)c1C(=O)NC1CC1CNC(c1ccc(C(C)(C)C)[nH]1)=O.CN C(=O)(CCS(N)(=O)=O)NCC(CCCC)NC(C1CCC1CF)=O N(C1CCc2cc(F)cc(Br)c21)CC(N1C(=O)C2CCCCC2C1=O)C1C(=O)CCC1 C1(CC)CCN(C(=O)Cn2ncccc2=O)C1CNC(C1CC(F)(F)C1)=O c12ccc(cc1)C(=O)NC(C)(C)CCNC(=O)c1ccc-2s1.C1(CO)(SC)CC1 CCCCC(O)CC(=O)NCCOCCN(C)C(C1(COC)CC1(C)C)=O c1(CCC(=O)NCC2CCCN(C(C3(OC)CC3)=O)C2)cccc(Br)c1F C(=O)(CCN1CCCC1)NCC1C(NC(CSCC#C)=O)C1.C1(=O)CC2(CC2)C1 C1(C(C)(C)C)CC2CCC(C1)N2C(=O)NCC1CCCC1c1nc[nH]n1 C(CC(C)C)(C(=O)N(CCNC(=O)Cc1cc(C)no1)C1CC1)OC CN1CCC2CCN(C(c3ccc(O)cc3Br)=O)C2C1 CC1(C)CC(CC(N2CCC(NC(C3CNC(=O)N3)=O)C2)=O)CC(C)(C)O1 c1(C(=O)NC23CCCC(NC(CC(C=C)C)=O)(C2)C3)cn2nc(C)cc2[nH]c1=O c1(N(C)CC2CCCN2C(=O)C(O)C2CC2)cc(OCCO)ccc1[N+](=O)[O-] C(=O)(C(F)(F)CO)N(C1CN(C(=O)C=C2CCC(C)C2)CC1O)C CC(C)(C)C(O)C(=O)NCC1CN(C(c2cccc(C(F)(F)F)c2F)=O)CCO1 c1(C(N2CCC(NC(CCCOCC)=O)C2)=O)cnnc(O)c1 c1(OC)cc(C)c(C(N2CC(C)(NC(c3cnc[nH]3)=O)C2)=O)cc1OC Cc1cc2c(cc1Br)CN(C(CO)CC(O)c1ccccc1)CC2 c1(C(N2CC(NC(C(CC)n3cncn3)=O)C(C)C2)=O)cc([N+](=O)[O-])n[nH]1 CC(C)CC(O)C(=O)NC(C)(C(=O)NCC1(O)CC1)C1CCC1 c1(NC(C2C3(CN(Cc4ccc(C#N)cc4F)C3)C2)=O)c(F)c(F)nc(F)c1F N1(C(CC2CCCN(C(C)C)C2)=O)CCC(CO)C(F)(C(=O)O)C1 C#CCC(CC(=O)NCC1(C#C)CCCC1)NC(=O)COc1ccsn1 C1(C(=O)NCC(C)NC(c2c[nH]c3nccc-3c2)=O)CCOCC12CCCCC2 C1(CNC(c2cc(C)sc2)=O)CC(NC(=O)CCNC2CCCC2)C(O)C1 c1(CC)ccc(C)cc1NC(=O)C(C(C)C)NC(C1(C#N)CCCOC1)=O C12(CNC(c3oc(C)c(Br)c3)=O)CCC(CC1)N2C(C1CC2CCC1C2)=O N1(C(COCC(=C)C)=O)CC2(CCN(C(=O)C(C)c3ncco3)C2)C1 C(C)(C)(C(C)CC(=O)N1CCCCC(C)(F)C1)NC(C(C)SC)=O c1(C(=O)NC(CC=C)CNC(=O)C(O)Cc2ccccc2)cc2occc2s1 C1(N(C(CC=C=C)=O)CC)CCCN(C(c2ccn(C)c2-c2ccccc2)=O)C1 N1(C(C2(COC)CCCC2)=O)CC2CC(C(=O)N(C3CCCC(C)(C)C3)C)(C2)C1 N1(CC)CCOC(C(=O)NCC2(CSC)CCN(C(=O)COCCC(C)C)C2)C1 N1(CC(C)N(C)C)CCC(C)(C(N2CCN(c3ccccc3)CC2)=O)CC1 CC(C(=O)NCCOCC(C)(C)NCC1(Cl)CC1(F)F)C(C)(C)C c1(C(=O)NCCCN(C(c2cnc(SC)s2)=O)C)cc2cncn2c(O)n1 C1(NC(c2ccon2)=O)CCN(CC2C(Cc3ccccc3)C2(F)F)CC1O CCC(C)(C#N)C(=O)N1CCC(C(N2CCOCC2)=O)C1.C12CC(C1)CNC2=O C(=O)(C1=CCCN(C(c2ncn3ccccc23)=O)C1)NCc1ccc(C)nc1 N1(C(CCC(=O)OC)=O)CCC2(NC(C3CC3c3ccccc3)=O)CCCC12 O=C(C#CC1(C(F)(F)F)CC1)NC1CCC1NC(c1ccn(CC(F)F)n1)=O N1(C(Cc2ccc(C(=O)OC)cc2Cl)=O)CC2OCCN(C(C3CCCS3)=O)C2C1 c1(C(c2n(C(C)C)nnn2)NCC2(C)CC2(Cl)Cl)cn(C)nc1-c1ccc(Cl)s1 c1(NC2CCN(C(C(c3cccc(F)c3)C)=O)C2)ncnc2sc(C(F)(F)F)nc12 CC1CCCCN1C(=O)CN1CCCC(CCNC(=O)CCn2ccnc2)C1 C1(C(=O)OC)CC2(CCNCC2)CN1C(=O)CN(C)C(=O)C1CC1 C1(COC)(CNC(C2(C)CCOCC2)=O)CCCN1C(=O)C(c1cccnc1)F C1(CC(N2CC3CC3(C(=O)NCC=Cc3ccncc3)C2)=O)CN2CCC1CC2 Cc1cc(C(N2CCC(NC(=O)CSCC(F)F)C(CO)CC2)=O)cc(=O)n1C N1(c2nnc(CC)s2)C(CNC(=O)CC(=O)NC2CC2)CC2COCC12 c1(C(N(CCN(C(c2nnn(CC)c2C)=O)C)C(C)C)=O)cc(C)c(C(N)=O)cn1 C(=O)(C1CCCc2ccnn21)NC(CN(C(c1cc(C(F)F)[nH]n1)=O)CC)C Cc1cccc(NC(=O)COc2ccc(Br)cc2)c1F.C1CCC(=O)N1 C1(NC(CN(CC#C)C(c2csc(S)n2)=O)=O)CCCCN1C(=O)CC CC(CC(N)=O)C(=O)N1CC(C(C)NC(c2cc3c([nH]2)CCC3)=O)C1 C1(CO)(NC(c2nnnn2CCC2(C)CC2)CCC2OCCO2)CCCCC1 CC1CN(C(c2cccc(F)c2C2CC2)=O)CCCN1C(c1sccc1C#N)=O C1(CCC=C)NC(=O)N(c2cnn(C(=O)NCC3C(COC)CC=CC3)c2)C1=O C1(O)(C(=O)NC(CN(C(CC(CC)(C)C)=O)C)C)CCCC(C)(C)C1 c1(C(N(C(CCNC(c2ccc(C)[nH]2)=O)C)C)=O)csc2cncn12 C=CC1CN(C(=O)CCCCCOCC)CC1NC(=O)Cc1cc(F)cc(C)c1 N1(CC(=O)N(C2CCN(C(C3CC(C4CC4)=NO3)=O)C2)C)C(=O)NC(C)(C)C1=O O=C(CCCCC(F)F)NCCC1CC(F)(F)CN1C(c1cnc(S)nc1)=O Cc1cnn2c1CN(C(C1COCCN(c3nccnc3N(C)C)C1)=O)CC2 c1(SC)ncc(N)c(C(=O)NC(CNC(c2csc3cncn23)=O)C(C)C)n1 C1(C(=O)NC(C(=O)NCCc2onc(CC)n2)C2CC2)CC(F)CN1C C(C)(CCCN=c1[nH]cnc(C)c1OCC(F)F)Nc1c(C)ccc(C(=O)NC)c1 CCCCC(F)C(=O)NCCC1(C(=O)NCC(C)CO)CCC1 c1(C(=O)NCCC(C(C)C)NC(c2nn[nH]c2Cl)=O)ccc2c[nH]nc2c1 C1(C(=O)NC(CC)CO)C2CC1N(C(=O)CN1CCC(C)CC1)C2 N1(C(C(C)(F)c2ccon2)=O)CCCC2(C1)CN(C(C1CCC(C3CC3)C1)=O)C2 C#CCCCC(C)C(=O)NCC(C1CCC1)NC(c1cc(F)c(F)c(F)c1)=O N1(c2cc(C)nc(Cl)n2)CCC(C2(NC(=O)C3=NOC(C)(C)C3)CC2)CC1 CC(CSC1CCCO1)C(=O)N(CCNC(=O)C(C)OC(C)(C)C)C1CC1 c1(C(=O)OC(c2ncccn2)C)ncn2c1CCCCC2 c1(C(=O)NC2COCCC2NC(C2CC23CC3)=O)nc(Br)c2n1CCCC2 N1(C(C(C)c2ccco2)=O)CCOCC1CC(=O)NCCCN1CCOC1=O Cc1ccc(S(=O)(=O)C2CCCCC2CC(=O)NCC(CC2CC2)C(=O)O)cc1 N1(C(COCCOC)=O)CC2(C(N3CCC4(C3)CN(C)C4)=O)CC1CCO2 CC1(O)CCCC1CN1CCC(CS(C)(=O)=O)C1 N1(C(CCOCCCNC(C(CC)=CC)=O)=O)CCCC1(C)C(C)(C)C c1(N(C(C)=O)C)ccc(Cl)c(C(N2CCC(CNC(C34CCC3C4)=O)CC2)=O)c1 CC1CCCC(C)N1CCC(=O)N(C1CC(NC(=O)CN2C(=O)CNC2=O)C1)C C1(CC(=O)NC(CCC(=O)NC(C=CC(=O)OC)C)C)C(C)(C)C1(C)C C(CCC(CCC)NC(c1sccc1CC#N)=O)NC(CCSCCC)=O CCC(CC(=O)N1CCC(NC(C2(Oc3cnn(C)c3)CC2)=O)C1)C1CC1 c1(CC)[nH]nc2ccc(C(=O)NC3CC(NC(C4CCC4CN(C)C)=O)C3)cc12 C(CN=c1[nH]c(CC(=O)NC2CCCOC2)cs1)c1cccc(OC)c1 C12(NC(C3N(C(C)=O)CC3)=O)COCCC1CN(C(c1cc(C)co1)=O)C2 c1(C(=O)NCC=CCNC(=O)C(c2ccccc2F)(F)F)cnccc1Cl N1(C(c2c(C)snn2)=O)CCCC2CN(C(c3cccc(Cl)c3Cl)=O)CCC12 C12(CC(=O)NC(COC)CC)CCC1CN(C(=O)CCc1ncc(C)[nH]1)C2 C1(C(N2CCC(NC(CN3CC(CC)C3)=O)C2C(C)(C)C)=O)CCC2(CCC2)O1 C1(N(C(=O)CCc2ccc(F)cc2)CC(F)(F)F)CCN(CC(F)(F)F)CC1 CCCCC(C(=O)N(CCCCCCNC(C1C2COCC12)=O)C)N(C)C c1(C(N2CCC(NC(C3CC=C(C)CC3)=O)C2)=O)ccccc1S(=O)(=O)C(C)C C1(C(N(CCNC(c2c(C)csc2)=O)C2CC2)=O)CC2(C1)CC(F)C2 C=CC1CCCN1CC(=O)NC1CC(OC(C)CC)C1 Cc1ccc(CNC(C2(CNC(c3cc(Cl)ns3)=O)CC23CCC3)=O)c(O)c1 c1(CC)cccc(F)c1C.C1(C(N2CC3(C2)C(=O)NC3)=O)NC(=O)OC1(C)C C(CCC)(C(O)C(=O)N(C)Cc1cn(CC)nn1)NC(C(C=C)(F)F)=O C(=O)(C1=CC2C=CC(C1)C2)N1CC(CNC(c2c(N(C)C)cccn2)=O)C(O)C1 CCCCCC(C)(C)C(=O)NCC(C)(O)CNC(C1CC1(C)C)=O c1(C(N(C(CNC(C(CC=C)CC)=O)C)C)=O)ccc2c(c1)nc(O)n2C N1(c2c(C(C)=O)cccn2)C2CCC1CN(C(C1CC1C1CC1C)=O)CC2 c1(C(N(CC(=O)NCC)C)=O)cc(CNC(=O)C(C)N=[N+]=[N-])nn1C N1(C(C2(c3c(C)cno3)CC2)=O)CCC(CNC(=O)CN2CCNC(=O)C2)C(C)C1 N1(C(=O)NCc2cc(O)cc(O)c2)CCCC2(CCCCO2)C1 n1(C(C2CCOCC2)C)cnc2c(N(C)CCF)nc(N3CC4CCC4(C)C3)nc12 c1(C(=O)NCC#CCNC(C(CC=CC)C)=O)c(C)[nH]c2ncccc12 c1(C(=O)NC(C23CCC(CC2)C3)CNC(C(COC)C)=O)ccnnc1O N1(C(COCCC#C)=O)CC2CCN(C(c3cc4nc(C)sc4[nH]3)=O)C2C1 c1(CN(C(=O)C(=O)NCCc2cccnc2)C)ccc(Cc2ccc(Cl)s2)cc1 N1(C(CCC=C)=O)CC(CNC(c2cccc(F)c2C(C)C)=O)C(F)(F)C1 N1(C(C(C2CC2)SC)=O)CCC(C)(CCNC(c2cc(F)c[nH]2)=O)C1 C1(CNC(c2ccnc3[nH]ncc23)=O)CN(C(C23CC(C2)C3)=O)CCC1(F)F C1(NC(c2cc(OC)no2)=O)CN(C(=O)Cc2cnoc2)CC2CCCC12 c1(NCC)ncnc2c1CCC2.N1(C(=O)C=CCn2cncn2)CCC(C)CC1 N1(C(c2ccc(NC=O)cc2)=O)CCC2C(NC(=O)COCC3CCOC3)C2C1 CCC1=NOC(C(=O)NC2(C(=O)NCC(F)Br)CC2)C1 C(=O)(CC(O)CC(C)C)N1C(CNC(=O)CC2(CO)CC2)CC(OC)C1 CCCCC(CNC(=O)C=CS(C)=O)NC(=O)Cc1ccc(C)o1 c1(C(N2CC(NC(C3C(OCC)C3)=O)C3C2C3)=O)cc(C(C)(C)C)ccc1N CC(C)C(C)(O)C(=O)N1CC(C(C)(C)O)(CNC(c2c[nH]cc(F)c2=O)=O)C1 Cc1cc(CNCC2CCN2C(C2CCCOC2)=O)c2ccccc2n1 c1(C(N2CCCC(F)(CO)C2)C(=O)NC(CC)C)nc2c(s1)CC(C)(C)CC2 C1(NC(CC2(C)CC2(Cl)Cl)=O)CCN(C(=O)COC2CC(F)(F)C2)C12CC2 C1(CC=C)(NC(C(COC)OC)=O)CN(C(C2CCCN2C(=O)NC(C)C)=O)C1 c1(C(N(CCCN(C)C)CCNC(C2CC2(C)C)=O)=O)cn2cccc(F)c2n1 CCCCC(O)C(C)C(=O)N1CCC(C(N2CC(c3cc(O)no3)C2)=O)C1 S(=O)(=O)(c1ccc(NCCC(C(C)C)SC)c(C#N)c1)N1CCC(OCC=C)C1 c1(C(=O)OC)cc(C(=O)NC23CC(CNC(=O)C(C)N(C)C)(C2)C3)cn1C c1(C(=O)NC(C)CCN(C(=O)C(C)n2cccn2)C)ncc(F)cc1N CC(C(C(=O)NCC1CC1)N1CCCC1C(N1CCCC1)=O)C1CC1 Fc1cc(Br)cc(-c2noc(C34CCCCC3C4Br)n2)c1F C1(CNC(=O)CCOCC2CC2)CCN(C(=O)CN2CCC(=O)CC2)CC1(F)F Cc1ccc(C(=O)NC2CCCC2(C)CNC(c2nsnc2O)=O)cc1C C1(NC(C(C)(O)C2CC2)=O)CC(F)CN(C(c2sccc2C2CCC2)=O)C1 C(=O)(CCCC(F)(F)F)NC(CCN(C)C)C(N1CCC(=C(F)F)CC1)=O C1(C(=O)NCC(O)CNC(C2CCN(c3ncccn3)CC2)=O)(CC)CCOCC1 C(CCCCC(=O)NCC(C)OC(F)F)NC(C=C(C)C(C)C)=O N1(C(C2(C#N)CC2)=O)C2CCC1CC(CCNC(=O)Cn1cc(CO)nn1)C2 Cn1cc2cccc(C(=O)NC3CC3CNC(c3cccc(N)n3)=O)c2n1 CC1CCC=C1C(=O)N1CCN(C(=O)CCC(=O)OC(C)(C)C)C(C2CC2)C1 Cc1c(C(=O)NC(Cc2cn[nH]c2)C(=O)NCC2CC(=O)N(C)C2)cccc1O C(N=c1nc2c(cnn2C)c(NC2CC(=O)N(C)C2)[nH]1)C1C(CC)C1 C(=O)(CCCS(C)(=O)=O)N1CC(NC(C(COCC)(C)C)=O)C(CC(=O)OC)CC1 CS(=O)(=O)c1ccccc1CC(N1CC(O)(CNC(C2(F)CCCOC2)=O)C1)=O C1(N(C(C(C)SCC)=O)C)CCCN(C(=O)Cn2cc(C(F)(F)F)cn2)C1 c1(-n2c(C)ncc2)ccc(C(N2CC(C)(C(=O)Nc3nc(O)cs3)C2)=O)cn1 C1(NC(CCC(=C)Cl)=O)CCC(C)(C)CC1CNC(C1(F)CCCC1)=O c1(-n2ncc(C)c2)cnc(Nc2ccccc2CC(C)(C)NS(C)(=O)=O)nc1O CC1=C(C(=O)NC23CCCC2CN(C(C2CC4CCC2O4)=O)C3)CCCC1 C=C(C)C1OCCCC1C(=O)NCC#CCNC(C1CCCCC1n1cccc1)=O C1(C(=O)NC2(C3CC3)CCN(C(C(C)OCC)=O)C2)CN2CCN1CC2C C(=O)(C1CCSc2ccccc21)N(CC(C)NC(C1CCN(CC)CC1)=O)C N1(C(Cc2c(C)[nH]c(=N)s2)=O)CCC(O)c2cc(Cl)ccc21 c1(CN(C(c2nc(OC)oc2)=O)C)ccccc1CNC(c1cc(Cl)n(C)n1)=O N1(C(c2ccc(Cl)c(F)c2)=O)CC(N=c2[nH]nco2)C1 c1(C(C(=O)NCC2CCN(C(CC(C)F)=O)C2)O)cccc(Cl)c1 N1(C(CC2(OC)CCCC2)=O)CCCC(CCNC(=O)C(O)C(C)C)C1 C1(C(N)=O)CCC(NC(=O)CC(CNC(=O)C2CC2)c2ccon2)CC1 N1(C(CNC(=O)NC2C(OCC)C2)=O)CCCC2(CCCO2)CC1 CN1CC2CC1CN2C(C1COCCN1C(C1CCC2(CCC2)O1)=O)=O C1(C)(NC(CN(C(CCc2ccn(C)n2)=O)C2CCC2)=O)CCC(=O)N1 N#Cc1cccc(CC(N2CCCC(NC(c3cc[nH]n3)=O)C2)=O)c1 c1(NC(c2n(CC=C)nnn2)c2ccc(COC)s2)cccc(CCC(N)=O)c1 C(=O)(C(CCC(C)C(C)(C)C)N1CCC2CCC(CSC)C2C1)NCCOC C1(NC(C2C(C)CCN2C(=O)Cn2cc(C#N)cn2)=O)CCC(C2CC2)C1 C=C=CC(C)C(=O)NCC1(OC)CCN(C(c2cc(CC(C)C)nn2C)=O)C1 c1(CC)[nH]ccc1C(=O)NCCCC1CCCN1C(C1CSCCS1)=O CCC(C#N)C(=O)N1CCC(N2CCN(c3ccncn3)CC2)C1 N1(c2ccnc(NC(C3(N4CCOCC4)CC3)=O)n2)CCC(N2CCCC2)C(F)C1 c1(C(N(CC(C)NC(=O)C(O)C2CCC2)C)=O)c[nH]c(C(F)(F)F)c1 Fc1ccc(N2CCOCC2c2nnc(-c3ccn(CC(F)(F)F)n3)o2)cc1 c1(C(N2CCC(NC(C3CC(CC)C3)=O)CC2)=O)c(F)ccc2c1OCC2 C1(C(=O)NCC(C)N(C(CC2C(C)=NNC2=O)=O)C)CC2(CC(N(C)C)C2)C1 C12(C(=O)NC3(C(=O)NC4CC=C(C)CC4)CC(O)C3)CCN(CC1)CC2 C1(C(C)NCC2CCC2C(F)F)CN(C(=O)OC(C)(C)C)CC12CC2 C=CCC(CC(F)F)N(C(=O)C(C)(C)C1CCCN1C(c1ncncc1N)=O)CC C1(C(NOCCCC)=O)CN(C(c2nocc2Cl)=O)CCO1 C(=O)(C(F)(F)C(F)(F)Cl)NC1CCC(CNC(c2c(C)snc2)=O)CC1 C(CCC(C(=O)Nc1cccc(CCO)c1)NC(C1CCOC(=O)CC1)=O)OC N1(C(C(C)=CC2CC2)=O)CC(N(C(=O)CCC2CCCCO2)C)C(C)(C)C1 C1(C)(CC(=O)NCCN(C(C(C2CC(F)(F)C2)OCC)=O)C2CCCC2)CCCC1 Cc1cc(=NC2CCOC3(CCOCC3)C2)c2cc[nH]c2[nH]1.C1CO1 n1(C(CC)CC)nc(-c2ccccc2)nc1CCCC1CCCCO1 c1(CCN(C)CC2CN(CC(F)(F)F)C2)c(Cl)cccc1Br CC(C)C(C)(CNC(=O)CCOC1CC1)NC(c1ccc(CO)cn1)=O CC(C)(C)CC(O)C(=O)NC(C)(C)CC(F)C(=O)N1CCCC(C)(CO)C1 C1(CNC(=O)NCC(=O)OC)COCCN1c1ccc(C(F)(F)F)nn1 C1(C(=O)NC2CN(C(=O)OC)C2)CCCN(C(=O)Cn2ccnn2)C1C C1(NC(c2scc(C)c2)=O)CCN(C(c2ccc(C(F)(F)F)cc2)=O)C1(C)C N1(C(CNC(CC)=O)=O)C2CCC1C(NC(=O)C(F)n1ccnc1)C2 N1(C(C(CN(C(c2cncc(C)c2)=O)C)C)=O)CC2CCC(CC2)C1 C1(OCCC)CCCN(C(=O)CC2CCCN2C(=O)CC2C=NN(C)C2=O)C1 N1(C(C)=O)CC(C)(C)CC1C(=O)NCC(C)N(C)C(C1C(C=C(C)C)C1(C)C)=O C1(CNC(=O)CCc2cnoc2)CCCC(NC(=O)C(C2CCOCC2)F)C1 c1(C(=O)NC(C2CCN(C(CC=C=C)=O)CC2)(C)C)cc2c(n1C)CCOC2 N1(C(CC(CC)CC)=O)CCC2N(CCOC)CC2C1 CCC1(CC)CN(C(C)=O)c2ccccc21.C12CC(C1)NC(=O)C2 Cc1ccc(SCC(=O)NC2CN(C(=O)CCc3ccco3)C2)cc1C CC1CN(C(C2(C(=O)N(C)C)CC2)=O)CCC1NCC1CCC(F)(F)CC1 c1(CSc2c(C)cc(-c3nn[nH]n3)cc2)nnc2cc(C(F)(F)F)cc(C)n12 C12(C(N(C)CCNC(c3cc(=O)n(C)cn3)=O)=O)CCC(CC1(F)F)C2 c1(C(=O)NC(CCCNC(C(N2CCNC2=O)C)=O)(C)C)cnn2c1N(C)CC2 c1(C(C)NN2CCN(C(=O)CC(C)C3CC3)CC2)ccc(-c2nn[nH]n2)cc1 N1(C(C(COC)C)=O)CCC(CNC(c2cnc(OC)nc2)=O)C12CCC2 C(=O)(C(C(C)(C)C)OC)NCCC(C)(C)NC(C(CC)CC1CCCCC1)=O C1(CN(C(c2csc(=N)[nH]2)=O)CC)CCCCN1C(=O)CN(C1CC1)CC.C1CC1 c1(C(N2C(CN(C(=O)C=CCO)CC)CCC2)=O)oc(CO)cc1C c1(C(c2nnnn2C(C)(C)C)NCC(C)C(F)F)cc(C(=O)N(C)C)cc(Br)c1 CC(CCN=c1[nH]c(N(C)Cc2nccs2)nc2c1COC2)CC(F)(F)F CCC(C)(CNC(c1coc(-c2cnn(C)c2)n1)=O)NC(=O)Cc1cc[nH]n1 N(C1CCCn2nccc21)C(C1CCN(C(c2ccn(C3CC3)n2)=O)C1)=O C(=O)(CS(=O)(=O)C(C)(C)C)NC1(COC)CCN(C(=O)CC2(O)CCCC2)C1 C#CC1CC2(CC(OC(=O)NCCCS(=O)(=O)NC)C2)C1 N1(C(CC2(C=C)CCC2)=O)CCC(NC(C2CCCN(CCC)C2)=O)C(O)C1 C#CCCCCC(=O)N1CC(CNC(C2C(C)OC(C)C2C)=O)C1 CC1C(NC(c2ccc(OC(F)F)cn2)=O)CCN1C(c1c[nH]cc(Cl)c1=O)=O c1(CC)sc(C(=O)N(CCNC(=O)CC(C)F)C2CC2)cc1Br C1(C(N2C(C3CCCN(C(c4cnoc4)=O)C3)CCCC2)=O)CCCC2(CC2)C1 c1(NC(C(F)=CCC)=O)ccc(Nc2cc(-c3ccccc3)ncn2)cc1C CC1(C)CN(C(=O)C2=NOC(C(C)(C)C)C2)C(CNC(c2cc[nH]c2)=O)CO1 CC(C)CCC(O)C(=O)N1CCC(CNC(=O)C=C2CCC(C)CC2)C12CC2 C(=O)(C1=CCC(C)(C)CC1)NCC1N(C(CC2CC(=C)C2)=O)CC2(CC2)C1 Cc1ncc(N)cc1C(N1CCCC1CCNC(=O)C(C)C(F)F)=O C1(C(=O)NCCN(C(CC2CCN(C)C2)=O)C2CC2)CCCNS1(=O)=O S(=O)(=O)(c1ccc(NCC2CSCCS2)c(C#N)c1)N1CCc2c(nc(C)s2)C1 CCCC(C(=O)NC1CC(F)(F)CC1NC(C1CC(OC2CC2)C1)=O)C(C)C C(=O)(C(O)CC(F)F)NC(CNC(Cc1cccc(OCC=CC)c1)=O)C(C)(C)C N1(C(C2(CNC(C(COC)NC(C)=O)=O)CC2)=O)CCC(C(N)=O)C(O)C1 N1(C(=O)C=CC(F)(F)F)CC2(CCN2C(c2ccc(COCCCCl)cc2)=O)C1 N1(CC2(OCC)CCCOC2)CCC2(CCCC2)CC1 Cc1ccnc(C)c1C(=O)NC(C1CCN(C(c2cn(C)c(=O)n2C)=O)C1)(C)C c1(C(=O)NC2CN(C(CCCC)=O)CC2c2ccc(F)cc2)cc(Cl)cnc1O N1(CCNC23CCCC2C3(F)F)CCCN(C2CNC2=O)CC1.C(COC)OC C#CC1(NC(=O)Nc2ccc(Cc3ccco3)cc2)CCC(C)(C)C1 C1(NC(c2cc(OC)no2)=O)C2CCC(C2)C1C(N1CCCCC1CC(N)=O)=O C=CC(C)CC(=O)N1CCC1C(=O)NCC=CCOC Cc1ccc(CCNC(c2ccc(-c3cn[nH]c3)cn2)=O)cc1 c1(C(=O)NC2CCC2c2cccc(-c3nn[nH]n3)c2)cccc(F)c1F Cc1cnccc1C=CC(=O)NC1(CNC(=O)CCCOc2cccnc2)CC1 C1(CNC(CCCn2c(C)cc(C)n2)=O)CCC(C)N(C(c2csnc2C)=O)C1 C1(CC(=O)N(CC(=O)N(C2CCCO2)C)C)CCC12CN(C(=O)OC(C)(C)C)C2 CC(C)CC(C(=O)N1CC(CCNC(=O)C(C)N(C)C)C1)c1ccccc1 C1(C(N(C)CC2CN(C(c3cn(C)nn3)=O)CCO2)=O)CS(=O)(=O)CC12CCC2 c1(C(=O)NCC2(NC(C(C)SC)=O)CCCCC2)ccnc2c1ncn2C c1(C(=O)NC2C(NC(CSCC)=O)C2)cc(N2CCOCC2)ccc1F CC(CS(=O)(=O)N1CCC(N(C)Cc2ccc(Cl)cc2F)CC1)C(C)(F)F N1(C(C2CC(OC)C2)=O)CC(NC(=O)COc2cc(C)ccc2F)CC1(C)C Nc1c(C(=O)NC2CC(CNC(=O)C(C3CCCO3)C3CC3)C2)ccc(Cl)c1F c1(C(=O)NC(CC(C)NC(c2c(OC)n[nH]c2)=O)C)ncc(Br)cc1OC c1(CC)[nH]nc(C(=O)NC(C2CCOC2)CNC(C2CCCN2C(C)=O)=O)c1Cl c1(NC(C2C(NC(CCc3cccc(C)c3)=O)C2)=O)cc(F)c(Cl)cc1Cl N1(C(c2cc(OCC)ncn2)=O)CC(CCNC(=O)C2=C(C)OCC2)OC(C)C1 N1(C(C2C(C)N(C(=O)CN3CCCC3)CCC2)=O)CCC2(C1)CN(C)C2 CCC(CC)CCCC(=O)N1CCN(C(=O)CCCNC(C)=O)C(C2CCC2)C1 C1(CCNC(C2CC3CC3C2)=O)CN(C(=O)CC2CC3(CC3)C2)CCS1(=O)=O c1(C(=O)O)cncc(-c2csc(C(C3CC3C3CC3)=O)c2)c1 CCCC(C)(C)C(=O)NCC(c1ccc(C)cc1)NC(=O)COCC1CC1 c1(CC)ccc(F)c(C(N2CCC(NC(C3(F)CCOC3)=O)C(O)C2)=O)c1 N1(C(C=CC(C)(C)C)=O)CCCC(CCCCNC(c2cnns2)=O)C1 C(C(=O)NOCCCC1CC1)(N(C)C)OCCCN(C(C)=O)C.C(C)C N1(C(CCn2ncc(C)c2)=O)CCCC(NC(=O)CCNC(N)=O)C(F)C1 C1(NC(CS(=O)(=O)NC)=O)COCCN(C(c2cnc(C(F)(F)F)s2)=O)C1 CCC(CCCC(=O)N(C1CCCCC1)CC)NC(=O)C(C)N(C)C(C1CC1)C CC(CC(=O)NCC1(F)CC(CNC(=O)CC2OCCC2(C)C)C1)C(F)(F)F c1(CCNC(C=CC)=O)ccc(CNC(c2cnn(C3CCCC3)c2C)=O)cc1 C1(C(=O)NCCC(C)N(C(c2cnc(C)s2)=O)C)CCc2nn(C)cc2C1 c1(C(N2CC(NC(c3cc(F)ccc3CO)=O)C2)=O)cc(Br)cc2[nH]ccc12 c1(C(=O)NC(CC(=C)Cl)C(=O)N(C)CCN(C)C)ccc2[nH]ccc2c1 CC1(C)CN(C(C2CCC3C(C2)C3(F)F)=O)CCC1NC(=O)Cc1ccccn1 n1(CC)c(=N)[nH]c2cc(C(=O)NCC(=C3CN(c4ccncn4)C3)F)ccc12 c1(C2(C(=O)NCCOC)CC2)cncc2c1CCNC2=O.C12(N)CCOC(C)(C1)C2 C(=O)(C1CCCc2cncn21)NC1(C)CCCN(C(=O)CCc2cnccn2)C1 N1(C(c2cc(C)nc(C)c2)=O)CCC2(CC1)CC(NC(=O)C(C)N1CC(C)C1)CO2 C1(CCNC(C(C)NC(COC)=O)=O)CCCCN1C(C1(c2nc[nH]n2)CC1)=O c1(NC(N(CCCN(C)C)Cc2cnccn2)=O)cc(C(C)(C)C)ccn1 C(CCC(O)C(=O)NCC#CC(F)(F)F)NC(C1CC(O)C(F)C1)=O c1(C(=O)NCC2CCN(C(c3ccc(OC)cc3Cl)=O)C2)cc2sc(C)cc2s1 C=CC1N(C(c2sc(C(=O)OC)c(C)c2OC)=O)CC1(C)C Cc1ncnc(C(=O)NCCCC2CN(C(C3(C)CC=CCC3)=O)CCO2)c1C c1(OC)ccc(-c2cc(CN=C(NC3CCCC3)NC3CCC3)no2)cc1 n1(CC=C)cc(NC(C2C=CC(NC(=O)CCSCC(C)C)C2)=O)cn1 c1(C(N2CC(O)(CCNC(CC3CCC(C)CO3)=O)C2)=O)cc2ccccc2[nH]1 C1(NC(c2cccc(Br)c2)(C)C)CCCCC1C1CCCC1 c1(CC)ccc(C(N2CCC(C(F)F)(CNC(=O)C(C)C(C)C)C2)=O)cn1 C1(C)(CNC(C2C3(CC(OCC)C3)C2)=O)CC(F)(F)CN1C(=O)CC1(C)CCC1 c1(C(C)(F)F)ccc(C(=O)NCC2(F)CC(CNC(C3CCOC3C)=O)C2)cc1 c1(C(CC)C(C)NC(=O)CCc2cnccn2)nccc(=NCCCC(C)OC)[nH]1 C(=O)(C1CCCn2nccc21)NC(CNC(C(C(C)C)NC(=O)OC)=O)C C1(NC(CN2CCN(C)CC2)=O)CCN(c2cc(=O)n(C)cn2)CC(C)(C)C1 N1(C(C2(CCOC)CCC2)=O)CCCC(n2cncn2)C1 C(=O)(CS(=O)c1ccc(Cl)cc1)NCCC1CC(NC(C=CC=CC)=O)C1 N12CCC(CO)(C1)NC(=O)c1cc(no1)C2=O.C1(C)(OC)CC(C(=O)OC)C1.COC N1(C(C2CC2NCc2cncnc2)=O)CCC(F)(F)CC1 c1(C(C(=O)Nc2c(C)cccc2)N(C2CCC2)C2CC2)c2c(nn1C)CCCC2 C(=O)(C1CCCc2nncn21)NC(C#N)CO c1(C(N2CC(N(C)C(c3ccnn3CCF)=O)C2)=O)cc(Br)n(C)c1 CC1C(NC(C2CCS(=O)(=O)N2)=O)CCN1C(=O)C(N1CCC(O)CC1)C C1(C(=O)NCCC2CC(C(N(C3CCSC3)C)=O)C2)CC2CCC1C2 c1(OC)nc(NC2CCCC2C(N2CCCCC2c2ccccc2F)=O)ncc1C C1(OC)CCC(C(=O)NCc2cc(C(=O)NCc3nnn(C)n3)n[nH]2)CC1 N1(C(C2N(C(C3CCC(=O)C3)=O)C3CCC2C3)=O)CCn2ccnc2C1 N1(C(c2c(CC)nco2)=O)CCCC(C)C1CCNC(c1cc(C(F)F)no1)=O c1(CC)nocc1C(N1CC(C(=O)NCCO)C1)=O.C(=O)(CC)N(C1CC1)CC Cc1cnc2nccc(C(=O)NC(C)CCNC(c3cnc(C)n3C)=O)c2c1 C1(C(N2C(C(=O)NCC(C)(C)SC)C=CC2)=O)C2CC(=O)CC12 O=C(NN1CCOCC1)C1CC1CNC(=O)CC1CC1 S(=O)(=O)(c1ccc(Cl)c([N+](=O)[O-])c1)CC=CCNC(C1(C#C)CCCCC1)=O c1(COC)cc(C(N2CCC(OCCNC(=O)CC3(O)CC3)C2)=O)on1 c1(C(=O)OCC)c(C)oc2nc(CNC(C#N)CC3CCC3)nc(N)c12 N1(C(C(CCCC)NC(c2nnsc2N)=O)=O)C2C=CCC1CCC2 c1(C(N2CCC(O)(C(C)NC(C3ON=C(C)C3)=O)C2)=O)cncc(Br)c1C Cc1ccc(C(=O)NCC2CC2NC(c2cc3sc(Cl)cc3[nH]2)=O)c(O)c1C c1(C(=O)NCC(CNC(C(CC)(C)C)=O)O)[nH]c2ccccc2c1C1CC1 N1(C(C=CSC)=O)CCC2(CCCCC2NC(c2ccsc2C(F)F)=O)C1 Cn1nc(C(=O)NCC2CCC(C(=O)NCC3CCCCC3)CC2)cc1Cl C1(S(N)(=O)=O)(C(=O)NCC(CNC(C2(C)N(C)CCC2)=O)O)CCCC1 C1(CCNC(CCC(=O)OCC)=O)CCN(C(=O)Cc2cnc(C)[nH]2)C(C)C1 C1(C(=O)N(C2(CN(C)C)CCCCC2)C2CC2)C(N)C2CCCCC12 C1(CC#C)(C(=O)NCC(CC(C)C)NC(=O)CCOC2CCOC2)CCOCC1 C1(CCNC(=O)COCC2CC2)CC2CCCC2N1C(=O)C=Cc1ccc[nH]1 C(=O)(CCCCCCCCCO)NC1(CNC(C(CC)SC)=O)CCCCC1 Cc1cc(O)ncc1C(=O)NC1(C(=O)NCCCC(C)(F)F)CC(CO)C1 CC(C)C(C)C(=O)NC(CNC(c1ccc(-c2nnc(C)o2)cc1)=O)C1CCC1 C1(O)(CNC(c2n(C=C)ncc2)=O)CCN(C(c2ccc(CC)c(F)c2)=O)CC1 c1(-c2occ(C(N(CC(C)NC(CN(C(C)C)C)=O)C)=O)n2)ccccc1Cl C1(C)(C(=O)NC2C(NC(C(COC)(F)F)=O)CCCC2)CC(C2CC2)=NO1 C(=O)(CC1=CCCC1)N(CC(C)CNC(C1(c2ccccc2)CCOCC1)=O)C C1(C(C)NC(c2nc(OC)oc2)=O)CCN(C(C2CCCC2C(C)C)=O)CC1 C(=O)(C(C(C)C)NC(=O)Nc1ccccc1)NCC1(O)CN(C(CC(C)C)=O)C1 CCCCC(O)CC(=O)N1CC(NC(=O)COC(C)C)C(C)(C)C1 c1(C(N(C2CCCNC2)Cc2cn(CCOC)nn2)=O)cccc2c1OCC2C C12(C(=O)NCC3(CC)CCC(=O)N3)C(NC(=O)CC=C(Cl)Cl)C3CC1C2C3 CCCC(CC)CCC(=O)N1CC2CC(NC(c3cc(C)nn3CC)=O)CC2C1 C1(C(CNC(c2c(CC)csc2)=O)(C)C)CCCCN1C(=O)Cc1c(C)cnn1C N1(C(C(C)CC2CCCC2)=O)CCC(C2CC2)C1C(=O)NC1(C)CCSC1 c1(CC)cn2c(C(=O)OC(C)(C)C)cccc2n1.C1(C2CC2)CNC(=O)N1 Cc1cc(NNC(=O)C2CCN2C2CCOCC2)ccc1F CC#CCCCC(=O)NC1C=CC(C(=O)NCCN2CCC(OCC)C2)C1 C(=O)(C(C)(C)S(C)(=O)=O)NCC12C(CN(C(C3(CC(C)C)CC(=O)C3)=O)C1)CC2 Cc1[nH]c(C)c(C(=O)NCCC(C)CCNC(=O)C(c2ccc(F)cc2)=O)c1C C1(C)(OC)CCCN(c2nc(N3CCCC(C(C)C)C3)cc(C)n2)C1 N1(C(c2nn(C(CC)CC)c(C)c2)=O)CCC2(CC1)CC2NC(=O)C(CC)SC Cn1nccc1-c1n[nH]cc1SC.c12ccn-1n2.C1(C)CC1 S(=O)(=O)(c1ccccc1Cl)N1CCC(C(=O)Nc2cnon2)CC1 N(C1COc2ccccc21)C(CC1(CNC(c2c(C)ccc(O)c2)=O)CC1)=O N1(C(C(N2CCC(O)CC2)C)=O)CCC2(CC1)CN(C(=O)Cn1nccn1)C2 c1(C(N(CCNC(c2cc(OC)n[nH]2)=O)CC)=O)cc(C)c2c(O)n[nH]c2n1 C1(CC)CCN(C(N2CCN(c3ccccc3)CC2)=O)C1Cc1ccccc1Cl c1(CC(=O)NC2CCC(NC(=O)Cc3cncs3)C2)ccc2nc[nH]c2c1 C(CCC(C)(C)NC(C1CC1C(F)F)=O)NC(CC1C(CC)C1)=O c1(C(=O)NC2CC(CNC(C(CSC)O)=O)C2)ccnc2ccc(Cl)cc12 CCCCCC(O)CC(=O)NC1(C)CCN(C(=O)Cn2cnc([N+](=O)[O-])n2)C1 C1(CC=C)CCCCC1NC(=O)C(C)N(C(=O)C=Cc1nccs1)C C(CC)(CO)N(C(CN(C(C1C(CCC)C1)=O)CCOC)=O)C1CC1 C1(Cl)(C(N2CC(OCCNC(CC3C(C)C3)=O)C2)=O)C2CCC(=O)C12 C1(CCCC)CN(C(c2cc(C)c(C)[nH]2)=O)CCN1C(C1C2COCC12)=O c1(C(N(C(CCNC(CCC(=C)Cl)=O)C)C)=O)cc(C#N)c2n1CCCC2 N1(C(c2c(C)coc2)=O)CC2(CCN(C(=O)CCS(C)=O)CC2)C1 C1(C(N(CCNC(C(COC)(C)O)=O)CC2CC2)=O)CCCCS1(=O)=O c1(C(=O)NC2CC(N(C(CSCC=C)=O)C)C2)cn(CC(F)F)cn1 N1(C(C2C=CCCN2C(=O)Cc2ccns2)=O)CCCN2CCCC2C1 c1(OCC(N2C3C(CNC(C4C(CC)C4)=O)C(C3)C2)=O)ccc(Cl)c(C)c1 O=C(C1=CC2(CCOC2)C1)Nc1cccc(S(=O)(=O)N(CCO)C2CC2)c1 CCC(F)(F)C(=O)N1CCC(OC(=O)CNC(=O)C(C)(C)C)C1 CC1C(C(=O)N(C)CC2CCCN2S(C)(=O)=O)CCN1C(=O)OC(C)(C)C c1(C(=O)NCC(C)(C2CC2)NC(C(C)OCCC(C)C)=O)c[nH]nc1C1CC1 c1(C(N2CC(C)N(CCNCc3ccco3)CC2)=O)cc(F)ccc1C#N CCC(CCCC(=O)N1CCOCC(NC(c2cn(C3CC3)nc2C)=O)C1)OC c1(C(=O)NC(C(C)C)CNC(c2coc(C(F)(F)F)c2)=O)c(Cl)ccnc1F C(=O)(CCCCCOC(C)(C)C)NCC(C(C)(C)C)NC(=O)CCCC1CC1 c1(C(=O)NCC(CNC(CCCC=C)=O)C)ccc(C)cc1Br c1(C(=O)NCCOCCC(=O)NCC2CC=CCO2)ccc2ccncc2c1 N1(CNC(N(c2ncccc2O)C)=O)CCN(c2ccccc2Cl)CC1 N1(C(C=Cc2ccc(C)o2)=O)CC(NS(=O)(=O)CC#N)CC(F)C1 CC(CC1CCCO1)C(=O)NC1(CCNC(=O)CC2(C)CC2)CC1 N1(C(CCCOC)=O)CC2CCOCC2(NC(c2cc(C(C)=O)cn2C)=O)C1 N1(C(C=C(C)CONC(c2cc[nH]c(=N)n2)=O)=O)CC2(CCOCC2)C1 N1(C(C(=O)NC(C)C)CC2CCOC2)CCOC2CS(=O)(=O)CC12 C1(C2(C)CC2)C2CN(C(=O)COCC3CCCCN3)CC12.c12cc(cs1)NC2=O C#CCN(OC)C(=O)C1C2CN(C(C3CCN(C)C3)=O)CC12 C12(NC(CCN(CC)CC)=O)CCCCC1N(C(=O)C(c1ccccc1)=O)CC2 C(=O)(CC(CNC(=O)CCCSC)OC(C)C)NCC(CC)(C)Cl Cc1n[nH]c(C)c1S(=O)(=O)N1CCC(O)C(Nc2ncnc3ccccc23)C1 N1(C(COC2(C)CCCC2)=O)CC2CC2(CNC(=O)CCCC#N)C1 CCCC(C)C(=O)NC1CN(C(=O)Cc2ccnc(OC)c2)CC1C C(=O)(CCP(C)(C)=O)NC1C(C)CN(C(c2ccc(-c3ccc(Cl)cc3)[nH]2)=O)C1 C12(CNC(c3cc(=N)[nH]cc3)=O)CN(C(=O)Cc3ccoc3)CC1CS(=O)(=O)C2 c1(NC(C2CC(F)CN2Cc2ccc(O)cn2)=O)c(F)ccc(Cl)c1F C1(NC(C(C)NC(C)=O)=O)CCN(C(C2CCCN2C(C)C)=O)CC1O c1(OC)cnccc1CCC(N1CCCC1C1(NC(=O)CC(C)(F)F)CC1)=O C1(C(=O)NC(C)Cc2cccs2)C=CC(NC(=O)C(CO)N(C)C2CC2)C1 C1(N(CCc2c(C)ccnc2)C)CCc2cc(Br)ccc2C1 c1(C(=O)NCC2C(C)(C)N(C(C3CC34CC4)=O)CC2)cccc(S(N)(=O)=O)c1 C(C(CC(C)C)C(=O)NC1CC12CC(NC(c1cccc3[nH]ncc13)=O)C2)OC c1(C(N2CC(C(N3CCCC(O)CC3)=O)C2)=O)ccc2ccccc2n1 c1(CN(CCN(CCC(c2ccccc2)C)C)C)c[nH]c2cccnc12 N1(C(c2c(C)sc(O)n2)=O)CCC2(CCCCC2NC(=O)CC2(N(C)C)CCC2)C1 C1(CC=C)(NC(c2nc(CC)oc2C)=O)CCN(C(c2ccc(CO)o2)=O)CC1 C(=O)(C1=CCCCO1)N(CC1CCN(C(C(CC)OC)=O)C1)Cc1ccccc1 Cc1cc(C(N2CC(NC(=O)CCCCBr)C(O)C2)=O)nn1C C1(CNC(c2cc(CCCO)on2)=O)CC(O)CN1C(C1COCCO1)=O CC(C)C(F)C(=O)NC(C)(C)CNC(C1OCCO1)=O c1(C(N2CC(C)(C)C2C(F)(F)F)=O)nn(C)c2c1CCC2.CN1CCNC1=O C1(C(N(C2CCS(=O)(=O)C2)CC(CC)OC)=O)CCCCC1C(C)(C)C N1(C(c2cnn(C)c2C#N)=O)CC=C(CC(=O)NC2CCOC2=O)CC1 c1(CNC(CN(C(CCC2CCC(C)O2)=O)CC(C)C)=O)ncccc1Cl C1(C)(C(=O)NCC(CN(C(=O)CCn2cccc2)C(C)C)O)CCCN1C N1(C(CC2(COC)CCOCC2)=O)CC(C)(C)CC1CNC(c1n[nH]c(C)n1)=O c1(CC)ccc(CC(N2CC(NC(C3C(COC)CCC3)=O)C(SC)C2)=O)cc1 C=CCC(CC)C(=O)NCCOCCNC(=O)Cc1c(C)ncnc1C C(=O)(C(C)CC(C)C(C)=O)NCC(CC(=O)NC(CC)CCO)O C=CCC(C(=O)NC(C)C(C)NC(C1CCC(CCC)CC1)=O)C(C)C C(C)(CCCCN=c1[nH]cncc1I)NC(C1CC2CC(OC)C2C1)=O N1(C(c2n[nH]c(CC)c2Cl)=O)CCC(C)(C)C(NC(c2cnc(O)cc2C)=O)C1 C1(NC(CCS(C)=O)=O)CC2CC(NC(c3ccc([N+](=O)[O-])[nH]3)=O)CC12 C1(CC(=O)NC2CCC(NC(C3C(COC)C3)=O)CC2)CCC2(CCCC2)CC1 Cc1ccc(NC(=O)CN(C)C(C2COC(C)C2)=O)c(C)c1 c1(C(N(C(CN)C2CC2)C)=O)ccc(CNC(=O)CCn2cnc(=N)[nH]2)nc1 c1(C(=O)NC2CC(N(C(=O)C(O)CC3CC3)C)C2)c(F)cccc1[N+](=O)[O-] O(N1CCC(NC(=O)CNC(c2sccc2CC)=O)CC1)CC C1(O)(CC#C)CC(C(=O)NCCN(C)C(=O)Cc2ccc(C(=O)OC)s2)C1 C12CC(F)CN1C(=O)C(O)CONC2=O.c1(CC(=O)OC)ccoc1 N1(C(Cc2nnc(C)o2)=O)CCC(NC(c2ccc(F)c(Cl)n2)=O)C(F)C1 C1(NC(CCC(=O)N(C(C)C)C)=O)CC(F)(F)CC1NC(C1CC2(CC2)CO1)=O N(C(=NCC(F)F)NCc1ccnn1C1CCCCC1)CC1(C(C(C)C)O)CC1 c1(C(N2CCC(NC(C3C4COCC34)=O)CC2)=O)cc2nccc(Cl)c2s1 n1(CC(N2CC3CC(NC(C=NOC)=O)CC3C2)=O)cnc2c(N)ncnc12 C(=O)(CC(C)(O)C(F)(F)F)N1CC(C)(C)OCC1CNC(=O)CCNS(C)(=O)=O C(c1ccc(C)o1)=CC(=O)N(C(C(=O)NC(C(=O)OCCC)C)c1ccoc1)C c1(C(=O)NC2C(CNC(c3ccc(CO)c(F)c3)=O)C2)ncnc(O)c1Cl Cc1[nH]nc(C(=O)NC2CCC(NC(=O)C(C)C(=O)N3CCOCC3)CC2)c1F N1(C(C2(COC)CC2(F)F)=O)CCOC(CCNC(C2CC=CC(O)C2)=O)C1 C1(C(N2C(C(F)(F)F)CC(C)(C)C2)=O)CC12CCN(CC(=O)O)CC2 c1(C(C)=O)cc(C(=O)NC(c2nocc2C(=O)NCCCC2CCCC2)C)n[nH]1 n1(CC(N2CCOCC(NC(c3nc(CC)oc3)=O)C2)=O)c(C)cc(O)cc1=O C1(NC(C2CCC(=O)NC2)=O)CCCCCC1C(N1CC(N2CCOCC2)C1)=O C1(C(=O)NC(c2cnn(C)c2)C)CCN(C(=O)Cn2c(C)ccc2C)C1(C)C C(=O)(CC1=CCN(C(=O)C(C)(CC)CO)CC1)NC(CCC=C)C1CC1 c1(-c2nnc(N(C)C(C3(C)CC(N)C3)=O)s2)ccc(F)cc1 c1(NNCCOCC(C(=O)C(C2CCCO2)NC(C2CCOC2)=O)=O)cc(Cl)ns1 CCC(CC(=O)N1CCC(CC=O)C1)CC(F)(F)F.C1CCC1 S(=O)(=O)(c1cccc(=NCCC(C)CCCC)[nH]1)NCCOC c1(CC)nccc(=NC(=O)C2CC23CCN(C(=O)C(C)n2cccn2)CC3)[nH]1 c1(C(=O)NCCCN(C2(Cl)C(C(=O)OC)=CC=C2Cl)CC)cc(Cl)cnc1O C1(N(C(COCCCC(C)C)=O)C)CC2CC1N(C(c1cc(Cl)ns1)=O)C2 C1(CNC(c2cc(C)c(C)nc2)=O)CC2(CO1)CC(F)(F)C2 N1(C(CN(CC(C)C)C(C2CCN(C3CC3)CC2)=O)=O)CCN(CCO)CC1 C12(CNC(C(n3ccc(C)n3)C)=O)CC(CNC(=O)Cc3c[nH]nc3O)(CO1)C2 C1(CNC(C(C=CC)O)=O)CCN(C(c2nc(C)ccc2C)=O)C1(C)C C12(NC(C=COCC)=O)CCN(C(=O)C(C(C)C)c3ccc(Cl)cc3)CC1C2 c1(OC)cc(F)c(F)cc1CN1CCC(O)(C(=O)Nc2c(C#N)cnn2C)C1 Cc1cc(N)cc(C(=O)NC2COCC2NC(C2(OC(C)C)CCSCC2)=O)c1F C1(C(=O)NCC(F)Cl)CCCCCCN1C(=O)Cc1cnoc1 C=CC(O)C(=O)NCCCN(C1CCCC1)C(c1cnn(C2CCCC2)c1)=O C1(CC)CCC(C)N(C(c2ccc(C3CCC3)cn2)C(=O)NC2CC2)C1 C1(CC)CCN(C(c2ncc(F)cn2)=O)C(C(=O)NC(CSC)CCC)C1 c1(C(=O)NC2CCN(C(=O)CCOC3CCCC3)C2)ccc(C2=CCCC2)cc1 C1(CCC)CC(OCC)CN1C(=O)C1CC1.C(=O)CCCn1cccn1 N1(C(CCN(CC)CC)=O)CCCC(N(C(C2(F)CCC2)=O)CC)C1 N1(C(C(CNC(=O)CCc2ccco2)OC)=O)CCC2OCCC2C1 c1(C(N2CCC(C)(CNC(C3(OCC)CCCC3)=O)C2)=O)c(C)nn(CC)c1C C(=O)(CS(=O)(=O)CCO)N(C1CCC(NC(C(COC)N(C)C)=O)CC1)C C1(NC(C2(OC(C)C)CCC2)=O)CCCC(CNC(C2CC(OC)C2)=O)C1 n1(CC)nc(C(=O)NC2CN(C(C3(CC(C)C)CC3)=O)CC2O)ccc1=O C=Cc1cnn(C)c1C(=O)NCC1(F)CCN(C(C2CCC(=O)C2)=O)C1 N1(C(=O)Cn2cc(Cl)cn2)CCC2C(CCN2C(c2cn3cccnc3n2)=O)C1 c1(CNC(C23CC2CN(Cc2cncs2)C3)=O)cccc2ncccc12 N1(C(CCCCC)=O)CCN(C(c2nc(C)ccc2OC(C)C)=O)C(COC)C1 CC(C)CC(CNC=O)CC(=O)NC1CN(C(c2ccc(C3CC3)s2)=O)CC12CC2 c1(OC)ccc(C(=O)NC2COCC2CNC(=O)CCSC)cc1N C1(NC(c2sc(C)c(O)n2)=O)(CNC(c2cnc(N)c(Cl)c2)=O)CCCCC1C N1(C(c2onc(CC)n2)=O)CC(CNC(=O)CCc2cnc(C)o2)CCC1C C1(F)(C(=O)OC(C)(C)C)CCC(CNC(=O)C(=O)NC2CCOC2)C1 CC1CCc2[nH]c(=NCC3(C)CCOC3)[nH]c(=NCCOc3ccncc3)c2C1 N1(C(c2nc(C)oc2)=O)CCC(C2CCN(C(=O)C(c3cccnc3)C)CC2)C1 N1(C(c2c(COC)ccs2)=O)CCN(C)C(CNC(=O)CCC(N)=O)C1 CCC(C)C(C(=O)NC(C)CNC(=O)CCCc1nnc(C2CC2)o1)OC c1(OC)ccc(C(=O)NCC(C)N(C(=O)Cc2ccc(Cl)nc2)C2CC2)cc1O Cc1cc(C(N2CCCC2CC(N2C3CCC2CC3)=O)=O)cc(C)c1C N1(C(CCSCCCC)=O)CCC2C(CCCN2C(=O)CCN2CCCC2)C1 c1(NCC(CC)CO)ncc(C)cc1S(=O)(=O)N1CC2(CCCC2)CC1C C(=O)(CC(C)(C)C(=O)NCC(c1ccccc1F)NC(C1(O)CCOC1)=O)OC C(=O)(CCC(=O)NCC(F)(F)CN(C(=O)COCC1CCCC1)C)NCCC c1(C(=O)NC2CCN(C(=O)Nc3cccc(F)c3)C2)cc(NC2CC2)nc(Cl)c1 CCC(C)C(C(C(=O)NC1CCCCC1)N1CCCC(CCC(=O)OC)C1)OC C1(C)(OC)CCCN(C(=O)C(CNC(=O)Cc2ccsn2)C(C)C)CC1 CS(=O)c1cccc(C(N2CC(F)(F)CC2CNC(c2nc(Cl)cs2)=O)=O)c1 C(CCN(C)C(c1cc(C)cs1)=O)(C(C)(C)C)NC(C(CCSC)O)=O N1(C(Cc2cn(CC)nc2)=O)CCC2(CC1)CC2NC(c1cnc(C2CC2)s1)=O c1(C(=O)NCC(CC=C)NC(=O)CCCCOC)cncc(Cl)c1 c1(OC)ccccc1-c1cnc(C2CCCN2c2nc(C(=O)O)ns2)[nH]1 c1(C(N2CC(CNC(CCC#C)=O)C3C2C3)=O)cnc2[nH]ccnc1-2 C=C1CC(C(=O)N(C(C)CC)C)(CN(C(=O)C(C)=CCO)C(C(C)=O)C2CC2)C1 c1(C(N2CCCC(NC(c3n[nH]c4c3CCC4)=O)CC2)=O)ccc(Cl)c(Cl)c1O N1(C(c2nn[nH]n2)CC)CCC(CSC)CC1 N1(C(CC(CN(C)C)O)=O)CCC(O)CC1C(=O)NCC(C)(C)C1CC1 S(=O)(=O)(c1ccc2c(c1)CCCN2)N1CC(C2CC(=O)NC2)OCC1 N1(C(c2c(CC)n(C)cc2)=O)CCC2(C(=O)N3CC(O)CO3)CC2C1 S(=O)(=O)(c1ccc(CCC(=O)OCCC2CCCC2)cc1)NC C1(N(C(C(CC#C)C)=O)C)CCCCN(C(c2ccc(OC)nc2Cl)=O)C1 C1(CCC(=O)NCCOCCC)CCCCN1C(c1[nH]ccc1CC)=O c1(CNC(C(C)Oc2ccccc2CNC(=O)C2CC2)=O)ccc2c(c1)NC(=O)C2 N1(CC(=O)NC2CN(C(=O)Cc3csc(Cl)c3)C3C2C3)CCCCCC1=O N1(C(CCOc2c(C)cccc2)=O)CC(CO)C2(C1)CN(C(=O)CSC(=N)N)C2 c1(CC)cnc2ccccc2c1C(N1CCC(O)(CN(C(=O)C(F)F)C)C1)=O CC(C)CC(CNC(=O)C(C)(C)C1(O)CCOC1)NC(=O)Cc1cncc(F)c1 N1(C(c2cnc(SC)s2)=O)CCC2(CC1)CC(NC(=O)C1=CCCCC1)CCO2 C1(CNC(CCc2cn(C)nn2)=O)CC12CCN(C(c1sccc1Cl)=O)CC2 CC1CCC(C)(CNC(C2C(C#N)C2(C)C)=O)CC1 C(=O)(C1CCCc2ncccc21)NCCCCN(C(=O)CCC(C)(C)C#N)C CCC(F)(F)C(=O)NCCC1(NC(c2cccc(=O)o2)=O)CCC1 C12(CNC(Cc3ccc(C)nc3)=O)CN(C(C3CC(F)(F)C3)=O)CC1CCO2 c1(C(=O)NCC(CNC(=O)C=C(Cl)Cl)C(F)(F)F)cc2ccccn2n1 Cc1sc(C(=O)NCC(C)NC(=O)C(C)Oc2ccc(F)cc2)cc1Br n1(CCCC)nccc1C(=O)NC1CCCC1NC(C1(COC)CCCC1)=O CCC(CC(=O)NCC1CC1CNC(c1cn(C)c(=O)o1)=O)c1ccccc1 C1(CC)CCCC(C(N2CCC2CC(=O)NC)=O)N1 C1(NC(c2nnnn2C2CCCCCC2)(C)C2CCC2)C=CS(=O)(=O)C1 c1(-c2ccc(NCc3ccc(OCC=C)c(O)c3)c(F)c2)ccc(F)c(F)c1C c1(C(N(CC(=O)NCC(C)(CO)CO)CC2CC2)=O)ccc2nccn2c1 c1(SCCC(=O)NC2C(NC(CN3CCC(C)CC3)=O)CC2)ccc(F)c(F)c1 Cn1cc(C(N2CC3CC3(NC(c3scnc3C(F)F)=O)C2)=O)c(=O)n(C)c1=O C12(C(N3CCCC(CCC(=O)N(CC=C)C)C3)=O)CC(C)(CCO1)C2 c1(OC)nn(C)cc1CNC(=O)C(Cc1ccoc1)NC(=O)C(C)CSC C(=O)(C(F)(CNc1cc(C)oc1C)C(C)C)NC(CC)(C)COc1nnnn1C.OCC C1(CC#C)(C(=O)NC2COCC2SC)CCN(C(c2cncs2)=O)C1 C1(CC(=O)NCC(C)(CO)NC(C(N2CCOCC2=O)C)=O)CC(=O)NC1=O c1(C(N(C2CN(C(=O)C(C)(C)C3CCCO3)CC2O)C)=O)cccc2cnsc12 c1(N2C(=O)CC(C(=O)NC(C(=O)OCC)CC)C2)cc(C)ccc1OC N1(C(COc2cn(C)nc2)=O)CC2C(CCNC(=O)CC3CCOC3)C2C1 Cc1ccnn1C(C)C(=O)NCC1(C(=O)NC2(CF)CCC2)CCCO1 C1(C(=O)NCCC(=C)CNC(=O)C(F)CC(C)C)CC2(CCCCC2)S1(=O)=O CCCCC(O)CC(=O)NCCCCNC(=O)CCc1ccc(C(N)=O)cc1 NC(=O)CC(C(=O)N1CCC(CF)C1)NC(C1C2CCCOC12)=O CN1CCC2(CCN(C(C3(NC(C4C5(CC5)C45CC5)=O)CC(O)C3)=O)C2)C1 N1(CCNC(N2C(C(=O)OCc3cnc(Cl)nc3)CCC2)=O)CCCS1(=O)=O CC#CCCCC(=O)NC1CCC(NC(c2cn(C3CCOCC3)cn2)=O)CC1 c1(SCC(=O)NCC(C2CC2)NC(C(F)=CCC)=O)nnc(S)s1 C1(COC(=O)Cc2ccc(N3CCOCC3)o2)CCc2cc(I)ccc2O1 CCC(C(=O)NC(C)COC1CC1)N1CCCC1=O CC(C)(CO)C(C1CC1)NC(=O)CN(C(c1ccc(F)cc1)=O)CC1CC1 C1(OCC)(OC)CC(C(=O)N(C)CCN(C(C)C)Cc2cscc2Br)C1 Cc1cc(C(=O)NC2CCCN(C(C3(C)CC4(CC4)C3)=O)C2)ccc1Br Cc1cccc(CC(=O)NCCNC(c2n[nH]c3c2COC3)=O)c1F Cn1nc(C(=O)NCC2CCN(C(=O)CN3C(=O)CCC3=O)CC2)cc1C(F)F c1(C(N(C(CN(C(c2c(C)cc[nH]2)=O)C)C)C)=O)ccc(C(N)=O)nc1 C(=O)(C#CC1CCCCO1)N1C(CCOC)CN(C(c2cc(C)sc2C)=O)CC1 CCC(C)C(CC(=O)NCCC(C)C(C)(C)C)NC(C1(CC)CCC1)=O c1(OCC)c(CN=C(NCc2nc(C3CC3)n[nH]2)NCCSC)cccc1C c1(C(N2CCC(NC(CN(CCC)C)=O)(CF)C2)=O)nc(C)ncc1C Cc1ccc(Br)cc1S(=O)(=O)N1CCC(O)(C(=O)N(C(C)C)CC2CC2)CC1 c1(C(=O)NCCCN(C(=O)CNC(C)=O)CC)sccc1C(C)=O N1(C(C(CCO)N(C)C)=O)CC(C)(C)OCC1CNC(c1cc(C(F)F)no1)=O c1(CN(C(c2cc(CC)no2)C(=O)NC(c2ccsc2)C)C)cccc(C)c1 C1(NC(c2cc(C)no2)=O)CCC(C)N(C(=O)CCOc2ccc(F)cc2Cl)C1 CC1(C(=O)NC2CC2NC(=O)CN(C2CCC2)C(C2CCCC2)=O)C=CCCC1 C(C(=O)NC1CC(C)(NCC)C1)(C(C)NC(C)(C)C)NC(CNC(C(CC)C)=O)=O c1(C(=O)NCc2ccc(Br)c(O)c2)ccc2occc2n1 c1(CNC(C(C)N(CCOC)CCN(C)C)=O)oc2ccc(Cl)cc2c1C C1(NC(c2cccc(CC)n2)=O)CCCN(C(=O)CCc2cn[nH]c2)C1C C(=O)(CCS(C)=O)N(CC(C)NC(=O)C(=CC1CCCC1)C)CC C(=O)(C1=CCS(=O)(=O)C1)NCCCN(C(=O)C1=NOC(C)C1C)C(C)C c1(CCC(=O)NC(CNC(C2(C)C(C)(C)C2)=O)C2CC2)ccc2c(c1)OCO2 N1(C(COCCOC)=O)CC(C(=O)NC(C)(C)CCNC(=O)OC)CC(C)C1 C1(C(=O)NCC2N(C(c3n(C=C)ncc3)=O)CC(O)C2)CN2CCN1CC2C C(=O)(NNc1ccc(F)nn1)c1c(C)nn(C)c1C N1(C(C(Cc2cc[nH]n2)NC(C=COCC)=O)=O)CC2CCC(CO)(C2)C1 c1(CN2CCC(CNC(C3CC4C=CC3C4)=O)CC2)ccc(O)cc1F c1(C(=O)NC2(C)CN(C(C(C)CF)=O)C2)ccc(N2CCCC2)cc1 CC(c1cccs1)=CC(=O)NCCC1CSCCN1C(C1CCC(F)CC1)=O Cc1cccc(C(=O)NCC2CN(C)CCN2C(C2CC3CCC2C3)=O)c1N N1(C(C(C)NC(CC)(C)C)=O)CCC(CO)(NC(=O)CN2CCOCC2=O)CC1 N1(C(Cc2c(OC)cccc2)=O)CCC(NC(=O)CC(C)(C)F)C(C)(C)C1 c1(C2(C)CC2)cc(C(=O)NC2CCCC2CNC(=O)Cc2cc[nH]n2)no1 N1(C(c2cnccn2)=O)CCN(C(=O)CSC2CCOC2=O)C(CC(F)(F)F)C1 c1(C(=O)NC2C(CC)N(C(C3CC3F)=O)CC2)cnc2ncccn12 C#CCCC(C(=O)NCC(C1CCC1)OC)NC(C1CCCC(=O)C1)=O C1(C(N2CC(C(=O)NC(C(=O)OC)Cn3cccn3)(CC)C2)=O)CCCCN1N=O N(C1c2ccccc2CC1Br)C(c1cccc2nsnc12)=O c1(NC(N2CCC(C)(C)C2CC(=O)O)=O)cc(Br)cc2cc[nH]c12 C=CC1(CC(=O)NC2CN(C(=O)C(C3CC3)C3CC3)CC2C)CCCCC1 N1(C(c2ccc(C#N)s2)C(=O)NCCCCCC)CCN(c2ccccn2)CC1 C#CC1(NC(C2CC2C(C)NC(=O)C(C)(CO)OC)=O)CC(F)(F)C1 CC1CN(C(=O)Cc2ccccc2C(F)(F)F)CCN1C(C1CN(C)C1)=O c1(OC)cccc2cc(C(=O)NCC3CCN(C(=O)CCOCCN(C)C)C3)oc12 Cc1cccc(CN(C(=O)C(C)C)Cc2cccs2)c1 Cc1ccc(N(C(=O)C(C)CN(C(=O)C(C)n2cncn2)C)C)cc1C C1(C(=O)NCCN(C)C(c2cnn(C(F)F)c2)=O)CCCCC1P(C)(C)=O [N-]=[N+]=NC(CCC(N)=O)C(=O)NCCC(F)(F)Br C1(NC(CC(CC)N(C)C(C2CCCC2O)=O)=O)CCCCCC1C N1(C(c2cc(I)ccc2Cl)=O)CCCC2C1CCN2C(=O)CCn1ccnc1 c1(-n2c(C)cnn2)ccc(C(=O)NC(C)CCNC(=O)C(C)n2cncn2)cc1 Cc1cnc(Cl)cc1C(=O)NC1C2CC1N(C(c1snnc1C(C)C)=O)C2 N1(C(C(n2cc(CCCCC)nn2)C)=O)CC(O)CC1Cn1nc(C)cc1C n1(CC)nc2c(c1C(=O)N(C)Cc1nc(=N)[nH][nH]1)CCCC2 Cc1ncc2n1CCC(C(N1CC(C)(C(N3CCCN(C4CC4)CC3)=O)C1)=O)C2 Cc1cc(I)c(F)cc1NC(C1CCCC(NCc2cccc(CO)n2)C1)=O c1(CC(C(=O)NC2CCCC2CNC(=O)CCc2cnc[nH]2)O)ccc(O)c(F)c1 C=CC(CC)CC(=O)NCC1CCCCN(C(=O)CN2CCN(C)CC2)C1 C12CCC(C)(CC1)C1C=CCN(C1)C(=O)CN2C.C(C)(C)(C)OC(=O)NC1CC1 N1(C(c2c(-c3[nH]c(=N)sc3)c[nH]n2)=O)CCC23CCCCC2(C1)C3(F)F c1(-c2c(C(N(C)CCNC(C3CC3F)=O)=O)cccc2)cccc(C#N)c1 C1(C(=O)NCc2ccnc(F)c2)C2CC(O)C(C2)N1C(C1COCCOC1)=O C1(C(=O)Nc2ccc(CC)cc2)CN(C(=NC)NCc2ccccn2)CC1CC C(=O)(CC(C(C)C)C(C)C)N1CC(NC(c2c(C)nc(COCC)s2)=O)C1 c1(C(=O)OC)cnc(N2CCC(C)C2CNC(c2cccnc2)=O)nc1 C=CCC(CCCCC)C(=O)NC1(CCOC)CCN(C(=O)CC(C)C=C)C1 c1(CC(N2CCC(N(C(=O)CCN3CCOC3=O)C)C2)=O)ccc(F)nc1 N1(C(C2(CNC(C(C3CC3)SC)=O)CCCC2)=O)CCCCCC1C CC1CN(C(C2(CC(F)F)CC2)=O)CC(CCNC(=O)CC2CCCC3CC23)O1 N1(C(C(C)SCCCC)=O)C2CC1CN(C(=O)C=Cc1cn(C)nn1)C2 C1(CCC(=O)C(=O)COC(CN2CCCC2)CO)CN(C(=O)COC(F)F)C1.NC c1(C(N2C(C)CN(C(c3nncn3C)=O)CC2)=O)c(Cl)ccc(O)c1N c1(CCC(=O)NC2(C)CN(C(C=CCCC)=O)C2)c(C)nn(C)c1C C12(CNC(CC3(C)N(C(C4CC(C(C)C)C4)=O)CC3)=O)CCC(CC1O)C2 N1(C(c2cn(C)nc2C2CCOC2)=O)Cc2n[nH]cc2CC1C(=O)O C1(C(N(CC)Cc2ccccc2C(C)C)=O)C=CCNCC1 c1(C(N(C(C)CNC(=O)CCP(C)(C)=O)C)=O)sc2cc(F)ccc2c1Cl N1(C(c2ccc(F)c3c2CNC3)=O)CCS(=O)(=O)CC12CNC2 CC1=NN(C)C(=O)C1CC(=O)NC1(C2CCCN2C(c2sc(O)nc2O)=O)CC1 c1(C(=O)NC(C(C)NC(c2cc(O)nc(O)n2)=O)CO)cn2c(n1)CCCN2 C(=O)(C1=C(C#N)CCC1)NCCN(C1CCCCCC1)C(CC(C)=C(C)C)=O c1(OCCCC(=O)NC(C)CCNC(C2CCCCS2)=O)ccc(F)cc1F CCC(CC)C(F)C(=O)N1CC=CCC1C(=O)N(C)OCC(F)(F)F CN1CCC(CC(=O)NCCOCCCNC(=O)CO)C1=O C12(CNC(C=CCCC)=O)CN(C(C3(C)CC(=O)N(C)C3)=O)C(CO)(C1)C2 c1(N2CC(O)(CCNC(c3cc(OC)n[nH]3)=O)C2)ncnc2cnccc12 c1(N(CC(C2CC2)OC)C(=O)CSc2cc(C)on2)ncnc2sc(C)c(C)c12 CCCC(C(=O)NC1CC2CN(C(=O)CCSC)CC2C1)C(C)C c1(C2CCCN(C(C(CC)CC)=O)C2)cc(F)ccc1F CCCC(CC)CC(=O)NCCC(C)NC(c1nccc(OC)c1O)=O C1(C(=O)NCCSCCCC)CC2(CCC2)CN1C(=O)CN1C(=O)CCC1=O C1(C(=O)NC(c2cccc(C)n2)C)CC2(CC2)CN1C(c1csc(C)c1)=O C#CCC(O)C(=O)N1CCC(N(C(=O)C(C#N)CC)C)C1 c1(C(CNC(=O)CC2(O)CCCC2)NC(=O)C=CCF)cccc(Cl)c1 CC1CN(C(=O)CC2CC(F)(F)C2)CC(C)N1C(C1CC2(CCC2)CCO1)=O CC1CN(C(=O)CNc2cccnc2)CCC1N(C)C(c1coc2c1CSC2)=O c1(C(N(CC)CC2CCCN2C(=O)Cc2cc[nH]n2)=O)csc2ccc(F)cc12 C1(NC(c2cn3c(n2)SCC3)=O)COC2(C1)CN(C(c1cscc1F)=O)C2 c1(C(=O)NCC(CNC(C2CC(N(C)C)C2)=O)O)ccc(C2CC2)nc1 C(=O)(CCCCCC)NCC(C(=O)NC(C#CCC)(C)C)O C(N=C(NCC(C)(C)C1CC1)NCC1CCCO1)C1(CC)CC1 N1(C(CCC=C)=O)CC2CCC1C(NC(c1cc3n(c1)CCSC3)=O)C2 N1(CC(=O)NC(COC)C)CCCC(N(C(=O)CCC(C)(C)C)C)C1 c1(C(=O)NC(CCC)CNC(=O)C(C)CCOC)nc(C)ccc1F N1(C(CCCCOC)=O)CCC2(CCC2)C(NC(c2sccc2OC(F)F)=O)C1 C(C1=NOC2CN(C(c3cccc(N)n3)=O)CC12)NC(c1ccc(CCC)s1)=O C1(C(=O)NCCC2CCCOC2)CC2(CCC2)CN1C(=O)CCCCC1CC1 c1(C(=O)NCC2(NC(C=CCOC)=O)CCOC2)[nH]nc(OC)c1Cl c1(C(=O)NCCCCCN(C)C(c2cn(C)nn2)=O)ccnc2c1nnn2C S(=O)(=O)(c1cccc(=NC(C)c2cc(C)cc(C)c2)[nH]1)NC(C)CF c1(OC)cnncc1C(N1CCCC(C(C)C(=O)N(C)Cc2scnc2C)C1)=O C(=O)(CC(C)CC(F)(F)F)NC1CN(C(CC2(CC(=O)OC)CC2)=O)CC1N=[N+]=[N-] CON=CC(=O)NC(C)(C)CNC(=O)Cc1cncn1C CCC1=C(C(=O)N2CCC(C(=O)NCCN=S(C)(C)=O)C2CC)CCCO1 N1(CC(=O)NCC(CO)NC(=O)CN2CCC(F)C2)CCCCCCC1=O CC1=CCC(C)(C(N2CCCC(CO)(NC(C3CCCS3)=O)C2)=O)CC1 c1(C(N(CCC(=O)NCC(C)(C2CCC2)OC)CC2CC2)=O)ncc(N)cc1C N1(C(C(COC)OC)=O)CCCC(O)(CNC(c2c[nH]nc2Br)=O)CC1 C1(C(=O)NCCCN2CC=CC2)CCCN(C(=O)CCCF)C1 C(=O)(C(CC(C)C)ONC(C1CCS(=O)(=O)C1)=O)NC c1(C(=O)NCCN(C(CC(CC)C2CCC2)=O)C(C)C)coc2c1CCCC2 Cc1ccc(Br)c(CC(=O)NC(C)CCNC(C2CCC(C)(C)CC2)=O)c1 c1(C(=O)NCCCNC(CCCOCCOCC)=O)cc(CC)ccc1Cl C1(C(=O)NCCCCCN(C(CN(C(C)=O)C)=O)C)C2CCC1(c1ccco1)C2 C1(C(=O)NC(C#C)(CO)CO)CN(C(c2ccccc2F)=O)CC1C1CC1 n1(CCCSC)nnnc1C(c1cnn(CC(F)(F)F)c1)NCC1C2COCC12 C1(CNC(c2cc(CC)nn2C)=O)CC(F)(F)CN1C(c1sc(F)cc1C)=O N1(C(C2(COC)CC2)=O)C2CCC1CN(C(c1cc(C3CCCCC3)cn1C)=O)C2 CCCCCCCC(C(=O)NC(C)=O)N(C1CCOCC1)Cc1ccc(O)cc1 C(=O)(C(F)CC(CC)CC)NC1CCC(NC(CNC(CC)=O)=O)CC1 c1(C(=O)NCC2C(CNC(c3cnc(C)[nH]3)=O)COC2)[nH]nc([N+](=O)[O-])c1Cl C12(CNC(CCSC)=O)CCCC1CCN2C(c1c(N)sc(C)c1C)=O C1(NC(c2cc(C3CC3)[nH]n2)=O)Cc2ccccc2C1NC(C12CCC1CC2)=O c1(CC)cccc(S(C)(=O)=O)c1.C12CN(CCC1NC(C1CCC(=O)N1)=O)C2=O CC1CN(C)CC1NC(C1OCCC1CNC(c1ccn(C)n1)=O)=O C1(C(N(C2CCCCC2)CCNC(C=CC=CCC)=O)=O)CCn2nccc2C1 c1(C(N2CCCC(CC)(NC3CCC(F)CC3)C2)=O)cc(C)cc2nc[nH]c12 N1(C(CCC(C)C)=O)CCc2nc(O)cc(C(=O)NCC(C)C3CC3)c2C1 n1(CC(=O)N(CCNC(C2(C)COC2)=O)CC)ncc2ccccc2c1=O c1(CC)cc(C(N2CC(O)CC2CNC(=O)CSCCC(C)C)=O)c(C)nn1 c1(C(N(CCC(=O)NCCC2CCCOC2)CC2CC2)=O)ncnc(O)c1F c1(C(=O)NCCCN(C(c2cc(C(C)C)no2)=O)CCO)ccn2c1CCCC2 c1(C(N2CC(OC)C(NC(=O)CN3CCCCC3C)C2)=O)cnn2c1CCC2 C(C(C)(C)COC)(c1n(CCCC)nnn1)NC1CCCCC12CC2 NS(=O)(=O)c1cccc(S(=O)(=O)NCc2c([N+](=O)[O-])ncn2-c2ccccc2)c1 C1(CN(C(=O)NCCNC(=O)OC(C)=O)C)CC2(CCOCC2)CO1 N1(C(C2(CCOC)CCC2)=O)CCC(C2CCN(C(=O)CC3CCCC3)CC2)C1 c1(C(=O)NCCC(CNC(C(CC#C)C2CC2)=O)O)csc2ccc(OC)cc12 C(=O)(C1=NOC2COCC12)N1CCCC(NC(c2c(C)cnn2C)=O)CC1 c1(C(=O)NC(CNC(C(C(C)C)(C)C)=O)C2CCC2)n[nH]c2c1CCC(C)(C)C2 c1(C(C)OC(C2CC(CO)C2)=O)cccc2cccnc12 CN=c1[nH]c(=NCC(=O)N(CCC(C)(C)C)C)[nH]c(=NC(C)c2nc(=N)[nH][nH]2)[nH]1 C1(C(N2C(C(=O)NCC3CN(C(C)C)CCO3)CC(C)C2)=O)CCCCC(=O)C1 C(=O)(C(C)(C)C(F)(F)F)NC(CN1CCN(C(C=CC)=O)CC1)C C1(C)(C(=O)NCCCN(C(=O)COCC2(F)CC2)C)C2Cc3ccccc3C12 C1(CCNC(c2nc(CCC)oc2)=O)C(OC)C(OC)CN1C(=O)CC(C)SC C(CC(N)C(C)(C)C)N1CCN(c2c(CC(=O)OC)ccnc2)CC1 Cc1cc(C(=O)NCC(CO)NC(=O)C#CC(C)(C)C)n2ncc(C#N)c2n1 n1(CCCOCC#N)c(N2CCCC(N3CCCC3)C2)nnc1C1CC12CC2 C1(C(N2CCCC(NC(=O)C=Cc3cc[nH]n3)CC2)=O)CCc2cncn2C1 c1(NC(C2CCCC(NC(c3cc(C)c(F)nc3)=O)C2)=O)cccc(C#N)c1Cl C(CN=C(NCC1CC1)NC1CC(=O)N(C(C)C)C1)c1ccc(C)cc1 CC1CC(C(=O)NCC2(C)CCN(C(=O)C(F)(F)C3(O)CCC3)C2)=NO1 Cc1ccc2[nH]c(C(N3CC(CNC(=O)COCCF)C(F)(F)C3)=O)c(Cl)c2c1 Cc1cn2c(n1)C(C)CC(C(=O)NCC(CO)NC(c1cc(C)sc1C)=O)C2 Cc1cc(C(N2CCCC(NC(=O)C(C)Sc3nncn3C)CC2)=O)c[nH]c1=N C#CCCCCC(=O)N1CCC(N(CCO)C(C2CC3C=CC2C3)=O)C1 C1(CNC(CCCC=C)=O)CN(C(c2cccn2C)=O)CC1(F)CO Cc1ncc(C(N2CCCCC2C2CCCN(C(c3ccno3)=O)C2)=O)n1C C1(NC(c2c(CSCC)cccn2)=O)CC(C)CN(C(C2CCC2CF)=O)C1 C1(O)(CCOC)CCN(c2nnc(CC3CCCCC3)n2Cc2cocn2)CC1 Cc1ncc(C(=O)NC(c2cc(Cl)ccc2Cl)c2nn[nH]n2)cc1C#N c1(OC)nc(=NCC2CCCCN(C(=O)C(=O)NCC(F)F)C2)nc(OC)[nH]1 N1(C(C(C)=C2CC2)=O)CCC(F)(CNC(c2cc(-c3cccc(F)c3)no2)=O)C1 C1(NC(C2N=C(C)SC2)=O)CCN(C(c2cc(C)ccc2O)=O)C1(C)C N1(C(C2N(Cc3c(F)ccc(OC)c3)CC(O)C2)=O)Cc2cc(Br)cnc2C1 C=CC1(C(=O)NC2C=CCN(C(=O)C(c3cccc(OC(C)C)c3)C)C2)CCCC1 C1(C(=O)NCc2scc(CNC(=O)Cc3cnco3)n2)CC2(CC2)CO1 C(=O)(CC(C)(C)CCOC)NCC(CC(=O)N(C1CCCOC1)CC)O n1(CC)ccc(CNCC2CCCC2)c1.c1(C2CCC2)nnnn1CC1CCCO1 c1(OC)ccc(NC(c2ccc(C(F)F)cc2)c2nnnn2C(C)C(=O)OC)cn1 c1(CC(=O)NCC(CN(C(C(COC)COC)=O)C)O)cc(Cl)ccc1Cl C1(NC(c2ccc(COC)o2)=O)CC12CCN(C(=O)C(C)N(CC(F)(F)F)C)C2 C1(CNC(=O)C(N2CCCC2N2CCC2)=O)CC(CNC(=O)C2CC2)C12CCC2 C12(C(=O)O)CCCN1C(=O)N(C(=O)c1nnnn1CC(F)F)c1cccc(Br)c12 CCC(C#N)C(=O)NC(C(=O)NCCOCC)c1cccs1 C1(C(N2CCCC(COC)C2)=O)N(C(=O)CC2CC3(CC3)CO2)CCCC1(C)C C12(NC(C3CCCCCC3)C(=O)OC)CC3(C)CC(C)(C1)CC(C)(C2)C3 N1(C(c2c(CC)con2)=O)CC2COCC(C1)C2NC(=O)CN1CC=CC1 C1(C(=O)NCCCCN(C)C2CC2)CNC(=O)CN1C(=O)CC1CCCO1 C1(CNC(c2n[nH]cc2[N+](=O)[O-])=O)CC2CCC1N(C(c1ccc(CO)o1)=O)C2 c1(Nc2c(C(=O)NCC#N)n[nH]c2)c(F)cc([N+](=O)[O-])cc1Br Cc1ccc2c(c1)SC(C(=O)NCC1CC1NC(=O)CS(=O)(=O)CC(C)C)C2 N1(C(C2(OCC)CC2)=O)CCC(C)C(CNC(C2(C)CC=CCC2)=O)C1 c1(N2CCCC(C#C)(C)C2)ncnc2c1ncn2C(C)C(O)C(F)(F)F.C1CO1 c1(C(=O)OC)nnc2ccccc2c1NCC1CCN1C(=O)CC(C)CC CC(C(=O)NC(C1(CNC(c2cccc[n+]2[O-])=O)CC1)C)C(F)F S(=O)(=O)(c1ccc(C(N2CC3CCC(NS(C)(=O)=O)C3C2)=O)cc1)NC(C)=O c1(OC)nc(C(N2CC3CC3C2)C(=O)NCC2CCCO2)sc1C C(=O)(CS(=O)CC)N(CCC(=O)NC(C#C)(C)C)CCCO C(C(c1cccs1)=CC(N1CCC(C)(NC(=O)CCc2cncc(F)c2)C1)=O)OC C1(CNC(c2c(C)n(C3CC3)cc2)=O)CC2(CC2)CN1C(C1C(C)C1C)=O c1(CC)nscc1NC(=O)CCN(C(c1cc(C(C)C)no1)=O)C(C)C C(=O)(CC(F)(F)CC)N(CC(N1C(C)(CCC)CC1)=O)C(C)C Cn1nc(C(=O)Nc2ocnc2C(=O)N(C2CC3CCC2O3)C2CC2)cc1C(N)=O N1(C(C(C)OCCOCC)=O)CC2CCN(C(c3cc([N+](=O)[O-])n[nH]3)=O)C2C1 CC(C)(C)CCC(=O)N1CC(NC(=O)CCN2CCOCC2)CC(O)C1 C1(CCNC(C(N2CCC=C(C)C2)=O)=O)CCC(C)C(C)C1 C12(C(=O)NCCc3c(C)nsc3)CC(CN(C(C3CCC(=O)N3)=O)C1)C2 C(CCC1CC1)(C(=O)N(c1ccncc1)CC)NC(CCC)=O c1(C(=O)NCC2OCC(CNC(=O)Cn3nnc(=O)[nH]3)C2)cc(F)cc(Cl)c1 S(=O)(=O)(CCCS(=O)(=O)C(F)(F)F)NC(c1cccc(CCC)c1)=O N1(C(CC2CC(=C)C2)=O)CCCC(C(=O)NC2CC2CC(C)(C)C)C1CC c1(C(N2C(CNC(=O)C=Cc3cc[nH]c3)COCC2)=O)ccc(F)c2occc12 Cc1cc(C)c(CN2CCCC2(C)C(=O)Nc2ncc(F)cn2)[nH]1 CS(=O)(=O)CC(C(=O)Nn1cc(Br)c(O)nc1=O)ON Cc1scnc1C(=O)NCC(C)(O)CNC(=O)C(C)(C)OC(C)C N1(c2ccccc2)CCCC(Cc2ccoc2CNCC2CCCCC2)C1 c1(C(N2CCC(NC(c3cc(C)c(Cl)s3)=O)C2C)=O)cc2c(ccn2C)[nH]1 N1(C(=O)CC2CCC2)CC23CCCC2(C1)CN(C(c1ccc(Cl)c(O)c1)=O)C3 C(=O)(C(O)C(F)(F)F)N(CCCNC(c1ccn(-c2ccncc2)n1)=O)C1CC1 C1(NC(C(C)O)=O)CCOC12CCN(C(c1cc(Cl)cc([N+](=O)[O-])c1N)=O)CC2 C(CCC)(C(=O)N1CCCC1CN(C(=O)CC1CCCO1)C)=CCC C(C(O)C(=O)NC(C)(C)CNC(c1cn(CCC(C)C)nn1)=O)=CCCC C(C(O)C(=O)NCC(O)CNC(=O)C=C1CC1)=CC(C)C c1(C(=O)Nc2n(C)nc(C)c2CC(=O)O)cn2cccc(C)c2n1 S(=O)(=O)(c1ccsc1CO)NC(=O)Nc1ccccc1NC(C1CCC(F)(F)C1)=O C#CCCCCCC(=O)N(CCC(=O)NC(CC)C(C)(C)C)C C1(C(N(C(C#C)C)C)=O)(CNC(=O)CC=C(Cl)Cl)CC2(CC2)C1 C1(N(C)C(c2csc(C(F)(F)F)n2)=O)CCN(C(c2cncnc2)=O)CC1 c1(C(N(CCNC(c2c(C)ncn2C)=O)CC)=O)ccc2cn(C)nc2c1 c1(C(C(=O)NCCOCCNC(=O)C(c2ccc(F)cn2)(F)F)O)ccccc1F N1(C(C(C)=C2CC2)=O)CCC(NC(=O)CCc2cn[nH]c2)C(C(N)=O)C1 N1(C(C(CC(=O)OC)C)=O)CC(N(C)C(c2ccc(F)c(C)c2)=O)C(C)(C)C1 C1(C(=O)NC2(CCC(=O)NC3CN(C(=O)OC)C3)CCC2)CCCC1C C1(NC(COCCC=C)=O)CC=C(C#CC(=O)NC2CCOC2=O)C1 c1(C(NC)=O)n[nH]c2c1CN(C)CC2.C(CC(C(=O)NCCSC)N1CCCC1)SC CC(CCC(=O)N1CCCC1)NC(C1CCN(C(c2ccccc2)C)CC1)=O Cc1ccc(CNC(c2cccc(CNC(=O)C(C)(C)C(N)=O)n2)=O)cc1O c1(OC(C)(C)C)ccc(-c2noc(CS(C)(=O)=O)n2)cc1 CC1(CC(=O)NCCC2CCCN2C(=O)CC2CC3CC3C2)CCCO1 N#Cc1cc(F)c(C(=O)NC2COCCC2NC(=O)CC2CCCCC2)c(F)c1 c1(C(=O)OCC)cc(CN2CCC(c3ncc[nH]3)C2)no1.c12cnn(c1)c(=O)[nH]2 Cc1cccc(C)c1NC(=O)NC(C)C(=O)NCC1CC(=O)N(C)C1=O N1(C(CCSC(=N)N)=O)CCC(C2(NC(C3CCCC3)=O)CCC2)CC1 c1(C(=O)N(C2CC2)Cc2cccc([N+](=O)[O-])c2)c(O)c(Cl)cc(Cl)c1Cl N1(C(CCOC)=O)CCCCC1CCC1CCN(C(=O)CSc2nc[nH]n2)CC1 C(=O)(CC(C)(C)C#N)N1C(C)CC(NC(COCCCC(C)C)=O)C1 c1(C(=O)NC2CCN(C(c3c(Cl)cc(C)c(C)c3)=O)C2)ccc2c(c1O)CCC2 N1(C(C2(SC)CC2)=O)CC(O)(CNC(C2CCN2C(C)C)=O)C1 C1(=O)CCCCN1.C1(=O)C(CO)N1.C(C(OC)OC(C)C)OC.OC C(=O)(CCC(=O)NN(C)C)N1C(C)CCN(C(=O)C(CN(C)C)N(C)C)CC1 N1(C(c2c(O)ccc(N)c2)=O)CC(NC(c2cc(C(N)=O)[nH]n2)=O)C2CCCC12 c1(C(=O)NCCN(C(C=CC=CCC)=O)CCCO)cnc(O)c2cccnc12 c1(C(=O)Nc2ccccc2)cc2n(n1)CCCO2.N12CC3C(C3C1)CN(C)CC2=O N(C1CCc2ccccc21)C(C12CN(C(C3(C#C)CC(=O)C3)=O)C(C1)CO2)=O C12(CNC(CNC(CC)=O)=O)CC1CN(C(=O)C(C(C)C)n1ccnc1)C2 CC1CCCCC1(C)NC(=O)C=CC1CCN(C(=O)C(C)C(F)(F)F)CC1 S(=O)(=O)(c1cc(Br)c(Br)s1)N1CCN(C(c2c(OC)nc(Br)cc2)=O)C2C1C2 n1(CC(C)O)cc(C(=O)NCCN(C(N)=O)C2CC2)ccc1=O.C1(=O)CN1 C=CC(C)(C)CC(=O)N1CCC(C)(NC(c2cccc(NS(C)(=O)=O)c2)=O)C1 N1(C(c2nnn(C)n2)=O)CCN(C(c2sccc2F)=O)CC1CS(C)(=O)=O C(=O)(CCCCC#N)N(CCC)CCNC(c1ccc(C(C)F)cc1)=O c1(CC)cnc(C(c2nnnn2CCCOC)NCC=C(Cl)Cl)s1 C(C)(C(=O)NC1CCCC1C(=O)NCc1ccoc1)(C(C)C)OC C(=O)(C1=NN2CCC(C)N=C2N1)N(C(CCNC(c1cc(C)sc1C)=O)C)C CS(=O)(=O)C1CCCN(C(C23CC(NCc4cncnc4)(C2)C3)=O)C1 n1(CC#C)cccc1C(=O)N(CC(=O)N(CCCF)CC)C c1(C(=O)NCC(C)N(C(CCC(C)O)=O)C)ccc(O)c(Cl)n1 c1(C(=O)NCC(C)N(C(=O)Cn2cccc2)C)cnc2ccsc2c1 C1(CC(=O)NCCN(C(c2cc(F)cc(Cl)c2)=O)C2CC2)CCCCC12CC2 c1(C(=O)NC(C2CCN(C(C3CCC(F)C3)=O)C2)(C)C)cc(CC(F)(F)F)[nH]n1 C1(O)(CNC(C2CC23CC3)=O)CCCN(C(c2cscc2Br)=O)C1 C1(CC)CN(C(=O)C(C)C(C)(F)F)CCN1C(=O)Cn1nc(C(F)(F)F)cc1C c1(C(=O)NC(c2ccc(C)cc2)CNC(=O)C2=CCC2)c(N)ccc(F)c1F C(N=c1[nH]c2c(c(=NCCCN3CCOCC3)[nH]1)CC2)c1ccc(Cl)o1 C1(C)(CN(C(c2ccc(Cl)cc2Cl)C)C(=O)NC2CC2)CC2(C1)CC(F)(F)C2 c1(C(=O)OCC)cc(Br)sc1NC(C12CC1CN(c1ncccn1)C2)=O N1(C(c2cc(OC)cc(Cl)c2)=O)CCN(C(C2CCCN2N=O)=O)CC(CO)C1 C1(C(=O)NC2(CNC(c3c(C)oc(C#N)c3)=O)CCCC2)CCS(=O)(=O)C(C)C1 Cc1cc(CC(=O)NCCC2COCCN2C(=O)CCN(C)C)n(C)n1 c1(C(=O)NCC2CCC(NC(c3n(OC)cnc3C)=O)C2)cc2cccnc2o1 CC1(C)CC(C(=O)N2CCOCC2CNC(c2nc(Cl)ccc2F)=O)=NO1 C1(C(C)(C)NC(C(CC)OCC)=O)CCCCN1C(c1csc(CC)n1)=O C1(C(=O)O)(CO)CCCN(C(c2cccc(=S)n2O)=O)C1.CC(C)(CC(=O)OC)C1CC1 C1(CCC2(CO)C(CCCC(=O)OCC)NCCCS(=O)(=O)N2)CCCC(F)(F)C1 c1(C(C)(C)NC(=O)N(C2CC(CS(C)(=O)=O)C2)C2CC2)ccc2ocnc2c1 c1(C(=O)NC2C(NC(CC(C)SC)=O)CCC2)coc2c1COC2 c1(C(N2CCN(CC(C)C)CC2)C(=O)NCC2CCCO2)ccc2n[nH]cc2c1 N1(C(CSC)=O)CCC(NC(c2cc(C)ccc2OC(F)F)=O)C12CCC2 C(=O)(C#CC1(C)COC1)NCCCC(C)NC(CSc1c(C)ccc(C)c1)=O C1(NC(C2C(C=C)OCC2)=O)CCN(C(c2oc(C)nc2C)=O)C12CCC2 c1(C(C(=O)NC2CC2NC(c2ccnnc2O)=O)OC)ccc(F)cc1F c1(OC)ccc(S(C)(=O)=O)cc1C(N1CC(N(C)C(C2(F)CCC2)=O)C(F)C1)=O N1(C(CP(C)(C)=O)=O)CC(CCNC(C2CCC3(CCC3)C2)=O)CC1(C)C C1(CNC(C(CSC)O)=O)CC2(CCN(C(c3cc(C)cc(Cl)c3N)=O)CC2)C1 C12(n3cc(CC(C=C)O)nn3)CCC(C(=O)NCC3CCCC(C)CC3)(CC1)C2 c1(OCc2nnc(SC)n2-c2ccccc2Cl)cc(Br)cc(F)c1F Cc1nscc1CC(=O)NCCNC(=O)CCc1cncs1 CCCCCCCC(=O)N1CCN(Cc2ccc(Br)s2)CC1CC#N C1(C)(C(N2CC(CNC(c3cncc(C)c3)=O)C(C)C2)=O)CC2CCC(C1)S2 C(=O)(C(C)(C)Cc1ccccc1)NCC1N(C(C2C(=C)CC2)=O)CC1 c1(SC)cc(C)ccc1C(=O)NC1(CF)CN(C(C2C3CCC(F)(F)C23)=O)C1 c1(C(N2CC3(C(NC(CC(C(C)C)O)=O)CCS3)C2)=O)cc2nn[nH]c2cc1F Cc1cncnc1C(N1CCCC(CCNC(=O)CCc2csc(=N)[nH]2)C1)=O N1(C(C2C(C)(C)CCCC2)=O)CCN(C(c2ccc3cnsc3c2)=O)CC(O)C1 c1(CC)ccc(C(=O)NCCC2CN(C(=O)Cc3nc[nH]n3)C2)cc1Cl c1(OCC)ccc(C(=O)NCCN(C(=O)CC2CCSCC2)CC)nc1 C1(NC(C2CCN(C(c3n[nH]cc3Cl)=O)CC2)=O)CCn2cnnc2C1 N12CCC(CC1)C2.n1(C2CN(C(C(C)OCCOC)=O)C2)nnc(=O)[nH]1.C(=O)(C)N C1(NC(c2cn(CC(N)=O)nn2)=O)CC2CN(C(C3CCOC3)=O)CC12 c1(C(N2CCOCC(C)(CO)C2)=O)noc2ccc(Br)cc12 C(=O)(C1=C(C)OCC1)NCC(CN(C(C1COCC(C)O1)=O)CC)(C)C N1(C(c2c(C)cncc2)=O)CCCN(C(c2ccccc2S(C)=O)=O)CC1C N1(CC(C)C)CCC(C(=O)NC2(CNC(C3CCN(C(C)C)C3)=O)CC2)C1 C1(CC(=O)NC2CC(C)(NC(=O)CNC(C3CCCC3)=O)C2)CCS(=O)(=O)C1 C(=O)(C1=NNC(=O)CC1)N1CC(CNC(C2=C(C)CCC2)=O)C(O)C1 Cc1ncnc(C(=O)NC(C)(CNC(=O)C(C)(C)C2CCCO2)C(C)C)c1C c1(C(N2CC(NC(c3ccc(C=C)cc3)=O)C(F)C2)=O)c(F)ccc2ccoc12 c1(NC(C2(CN3CCC(C(=O)N)C3)CC(=C)C2)=O)cc(C)c(C)c(C)c1 N1(C(CC2(NC(C)=O)CC2)=O)CCN(C(C2CNC(=O)C2)=O)C(c2ccccc2)C1 C1(C#N)(C(N(CC(C)NC(c2cnsc2)=O)C)=O)CC1(C)C C1(CN(C(C=C(CC)CC)=O)C)CN(C(c2oc(C(C)C)nc2C)=O)CC12CC2 c1(C(=O)OC)cnc[nH]c1=NCCCCCCNC(=O)C(C)CF N1(C(C(n2cc(C(N3CCCCC3)(C)C)nn2)C)=O)CC2(CC(O)CNC2=O)C1 c1(C(N(C2CCN(C(N3CCCC3)=O)CC2)C(C)=O)=O)cn(C)c(=O)n(C)c1=O c1(NC(C2C(NC(c3cc(OC)cc(Br)c3)=O)C2)=O)cc(Cl)c(Br)cc1[N+](=O)[O-] c1(C2(NC(N3CCC(NC(CC(C)F)=O)C3)=O)CC2)cc(Br)ccc1Br C(CC1CCCC1)(C(=O)NC(c1ccoc1C(N)=O)C)NC(=O)OC.C12(CC1)NC2 Cc1ccc2c(c1)ncn2CC(=O)NC(C)CCNC(C1(C)COC1)=O c1(C(=O)NCCCC(C)=O)cccc(-c2sc(C)nc2C)c1 Cc1cccc(C)c1NC(=O)C(Cn1cccn1)NC(C1CCOC1(C)C)=O c1(C(N2CC(C)N(C(=O)C(CO)N(C)C)CC2)=O)cc2cccnc2o1 N1(C(C2(C#C)CN(C(c3nc(O)sc3C)=O)C2)=O)CCC(O)(C#C)C1 Clc1ccc(CC2CN(C(=O)NC(C3CCCOCC3)c3ccoc3)C2)cc1 CON1CCC(C(N2CCC(N(C(=O)CC3CC(F)C3)C)CC2)=O)CC1 c1(C(=O)NC(CC)CN(C)C(C2CC=CCC2)=O)nccc(OC)c1F N1(C(c2cc(Cl)c(Cl)s2)=O)CC(NC(C2(C3CC3)CCCO2)=O)C(O)C1 O=C1CN(C(c2nc(C(=O)C3CC3)n(-c3ccccc3F)n2)=O)C(=O)CN1 N1(C(c2cccc(NC)n2)=O)CC2CCCC2(NC(c2nc(C3CC3)cs2)=O)C1 N1(C(=O)CC(C(F)F)c2ccc(F)cc2)CCOc2c(Br)cncc21 c1(OCC(=O)NC2CCC2CNC(C2CC(n3cnnc3)C2)=O)cncc(Cl)n1 CCCCC(CN(C(=O)C(C)Oc1ccccc1C)CC)NC(c1cccs1)=O c1(CC(N2CCC(C)CC2)C(=O)NC(C)(C)C#N)c[nH]c2ncccc12 c1(C(C(=O)N(CCNC(C2C(OC)CC2)=O)C)=O)ccc(OCC)c(O)c1 N1(C(c2cc(C3CC3)[nH]n2)=O)CCOC(CCCCNC(CC(C)C)=O)C1 C(=O)(N1CC=CCO1)N1CC(O)CC1.CN(C)C(N)=O c1(C(N(CCNC(C2NCSCC2C)=O)CC)=O)ccc(C#CC2CC2)cc1 c1(C(N(CCCNC(C2CC(=C)C2)=O)C2CC2)=O)ccc(SC)c([N+](=O)[O-])c1 N1(C(C(C)=CC)=O)CCCCC(C(=O)OCC)C1.C1(=O)CC(C)N1C C(=O)(CCCC(F)(F)F)N1C(CN(C(C(CC=CCC)C)=O)C)CCC1 Cc1cc(CNC(C2(CF)CCN(C(=O)CNC(=O)CN(C)C)C2)=O)ccc1F c1(NC(C2CCCC2NC(c2ccnc(Cl)c2)=O)=O)cccc(C2CC2)c1Cl C(=O)(C(F)C(F)(F)F)NC1(CC(=O)NCC(C2(C)CC2)=O)CC1 CCC(CC)CC(=O)NC(C)CN1CCN(C(=O)CCc2cnccn2)CC1 C1(CNC(=O)C(F)OC(F)(F)F)CCC(C(=O)NCc2noc(C(N)=O)n2)O1 N=c1nc(C(F)F)[nH]c(=NC2CN(C(=O)Cc3ccon3)CCC2C(F)(F)F)[nH]1 c1(CC(=O)NC(CC)CNC(=O)C(C)N2CCCC2)cc2ccccc2nc1O NC(=O)C1=NOC(CNC(C2CCN(C(=O)C=Cc3ccsc3)CC2)=O)C1 c1(C2C(=O)N2)c(C)cnn1C.C1(N(C)Cc2ccccc2)(CC)CCOC1 c1(C(N(CCN(C(=O)C(F)(F)c2cccnc2)C)C)=O)ccnc2ncccc12 CC1(C(N2CCCC(CO)C2)=O)CCN(C(=O)CC23CCCC2C3)CC1 Cc1nn2cc(C(N3CCC(N(C(=O)Cn4cncn4)C)C3)=O)nc2s1 C1(CNC(CN(CC)CC)=O)CN(C(=O)COC2(C)CCOCC2)CC1(C)C CC1CN(C(=O)CC2CSC2)CC(C)N(C(=O)C=CSc2nc[nH]n2)C1 N1(C(C(C)C#N)=O)CCC(C)(C)C(NC(c2ccc(C3CCC3)nc2)=O)C1 c1(C(N2CC(NC(c3ccc(C)c(C)c3)=O)C(O)C2)=O)cc([N+](=O)[O-])ccc1C c1(C(c2nnnn2C)NC2CN(CC)C(=O)CC2)cc(Cl)c(C)cc1Br C(=O)(C1CCC2(CC1)CC2Br)NC1(CNC(C2(C)CCCC2)=O)CCC1 Cc1noc(C2(NC(c3nc(CNC(=O)CC4CC4)cs3)=O)CC2)n1 C(=O)(C(C)C(F)(F)F)NCCCOCCC(=O)NCCSCC#C C(c1ccc(F)cc1)=C(C)C(=O)NC1(CNC(c2coc(C(F)F)n2)=O)CCC1 C1(C(=O)NC(C2CC3(CC3)C2)C2CC2)CC2(CC2)CO1.C12(CC=CC1)C(=O)NC2 c1(OCC)ncccc1C(=O)NC(C1(O)CN(C(C2CC2(C)CC)=O)C1)C C1(C(=O)NCC(CNC(c2cn(-c3ccccc3)nn2)=O)OC)CCCCC1O c1(C(=O)NC(C)CCCCNC(c2cnc(N)cn2)=O)c[nH]c2cccc(F)c12 c1(N2CCC(CNC(C3(COCC)CC3)=O)C2)ncc(Cl)c(C)c1C#N CCC(CNC(=O)CCc1cncnc1)N=c1[nH]c(Cl)nc(C)c1F C=CCC(C)(C)CC(=O)N1CC(C(=O)NC(C)CCN2C=C2C(=O)OC)C1 c1(C(=O)NC2CC3(CC(NC(C=CC(C)C)=O)C3)C2)ccn2ncccc12 N1(C(C2(CC#C)CCC2)=O)CCC(CCCCNC(C2CCC(=O)N2)=O)CC1 C1(N(CC(C)C)C(c2cnco2)=O)CCN(C(C2CCC(O)CC2)=O)CC1 C(=O)(C(C(CC)CC)OC)N1CC(C=C)(CC(=O)Nc2ccc(C)cc2)C1 c1(Cc2onc(-c3n(C)ncc3Br)n2)ccc([N+](=O)[O-])cc1[N+](=O)[O-] C1(NC(C2CN3CCN2CC3)=O)C2CC1CN(C(C1CC=CCC1)=O)C2 N1(C(CCc2onc(C)n2)=O)CCC2(CCCN(C(=O)CCC(C)N(C)C)C2)C1 c1(C(=O)NCC(C)=CC(=O)NCC2CCCC2C2CC2)nc(C)ccc1C C1(CC(=O)N(C)CCn2cnnc2O)CC(F)CN1C(c1cccc(F)c1)=O C1(NC(C2(NC(c3c(CC)c[nH]n3)=O)CC2(C)C)=O)CCCC(C(N)=O)C1 C(=O)(CCC1=CCCCC1)N1CCC(C)(C(=O)NC2CC3CCCCN3C2)CC1 C1(CNC(c2c(C)occ2)c2nnnn2C2CCC2)COc2ccccc2C1 N1(C(C2N(C(=O)OCC)CSC2)=O)CCC(C2(NC(c3coc(Br)c3)=O)CC2)C1 c1(C(=O)NCC(CC)N(C(=O)C=CC2CC2)C)cc(C)n(CCN(C)C)c1 N1(C(C#C)C)CCCN(C(C(=O)NC2CCC2)C(C)C2CCOC2)CC1 C12(NC(C=CCOC)=O)CC(C)(C1)OC21CN(C(c2nn(C)cc2SC)=O)C1 C1(C(=O)NC(C(=O)NCCc2n(C)ncn2)Cc2cn[nH]c2)Cc2nccn2C1 c1(CN(C)CC2(c3cnn(C)c3)CCCO2)cccc(C(N)=O)c1 C(=O)(C(=O)N=S(C)(C)=O)NC(CCCC)CNC(=O)C(c1cccnc1)O N1(C(Cn2cc(CNC(C)=O)nn2)C)CCCN(C(=O)C(C)c2ccsc2)CC1 C(C(C)(O)C(=O)N1CC2CC2(NC(C2CC(C(C)C)C2)=O)C1)OC Cc1ccc(-c2nc(CC3CCCO3)n(CC3CCCOC3)n2)cc1Br C1(NC(C=C(C)C)=O)CCC(C)N(C(c2cn(-c3nonc3C)cn2)=O)C1 Cc1sc(C(=O)NCCCCC(C)NC(=O)C=CBr)cc1Br Nc1cc(Cc2ccc(CONC(C3CCN(CCCCO)C3)=O)cc2)cnc1Cl c1(C(N(CCC(=O)Nc2c(OCC)nccc2)C)=O)cccc(C)c1F Cc1ncn(C)c(=O)c1C(=O)NCC(C)NC(=O)CCc1ncco1 C1(CC=C)(NC(=O)C(F)(F)c2ccccc2)CCN(C(=O)CC(=O)N(C)C)C1 CC(C)CC(O)C(=O)NC1(CCCNC(=O)CSC)CC1.C(=O)(N(C)C)O CC1(C)C(C(=O)NCC2(CNC(=O)CCCCc3cnn[nH]3)CC2)C1CS(C)(=O)=O Cc1ccc(NC(c2sccc2NCc2ccc(O)c(Cl)c2)=O)c(C#N)c1 CC1(C)COCCC1NC(=NCCc1cccnc1O)NCC(F)F C(=O)(C(C)(C)C=O)O.S(=O)(=O)(CCN(C)CC1CC1)NC CC(C)C(CCN(C)C(C1(C)C=CCCC1)=O)NC(C1(CC(F)F)CCC1)=O C1(C(=O)NC2CC3(CN(C(c4c(SC)nn(C)c4)=O)C3)C2)CC(=O)N(C)C(=O)N1 N1(C(C2(C)C=CCCC2)=O)CCCC(CCNC(=O)Cc2cnoc2)CC1 CP(C)(=O)CN1CCOC(C(=O)NC2CN(C(=O)Cc3cnccn3)C2)C1 CP(C)(=O)C(O)C(=O)NCCCC1(O)CCN(C(c2ccc(CO)s2)=O)CC1 C(=O)(CC1OCc2ccccc21)NCC(C)(C)CNC(c1ncn2c1CCC2)=O Cc1cccc(C(=O)NCC2(F)CC(NC(c3c[nH]c(=O)cn3)=O)C2)c1[N+](=O)[O-] C=CCCC(CC(C)C)C(=O)N(C)CCN(C)C(C1CC2CCCCN2C1)=O N1(C(C2C(C)(CCCc3ccccc3)C2)=O)CCCC1(c1cccs1)C(F)(F)F CCCCCCCCC(=O)NCC(O)CNC(=O)COc1ccccc1Br CN1CC(F)CC1C(=O)NCCNC(=O)C(=O)NCc1ncc[nH]1 CC#CCCCC(=O)N1CCC(NC(=O)C2CC2)C1C N1(C(c2n(CC)nnc2)=O)CCC(C(C)C(=O)NC(c2cccnc2C)C)CC1 C1(NC(C2CC(SC)C2)=O)CC(CNC(=O)CCc2cn(C)cn2)C1(C)C C(=O)(CC(C)(O)C(F)(F)F)NCC(C)NC(c1cccc2nc(C(F)F)sc12)=O c1(C(=O)NC2(CC=C)CCN(C(=O)C(COC)CC)C2)ccnc2ccsc12 n1(CC)nncc1C(c1nnnn1C1CC1)NCCOCCOC Cc1cncc(C(=O)NCC2CC(O)(CNC(c3cnn(C)c3Cl)=O)C2)n1 N1(C(c2cnc(C)[nH]2)=O)CCN(CC(C)(C)NC(=O)C2=CCCC2)CC1 N1(C(C(C)OC)=O)CCC(O)C(N(C(=O)CC2CNC(=O)C2)C)C1 c1(C(N2C(CC)C(C(=O)NCC3CCN(C)CC3)CC2)=O)cccc2[nH]ncc12 C(c1cccc(C#N)c1)=CC(=O)NCCNC(c1cncc(SCC)n1)=O C(CCC)(C(O)C(=O)N(C)CCN(C)C)NC(c1c(C#C)c[nH]n1)=O N1(CCN(C)C)N=C(C(=O)N2CC(CC3CC3)C(F)C2)CCC1=O.C1(=O)CCN1 N1(C(C(CC)NC(C)=O)=O)CCCC(C2CC2NC(c2cc3scnc3[nH]2)=O)C1 C(CCCC(=O)NCCCCCCNC(c1sccc1C)=O)N(C(C)=O)C C1(C(N2CCC(C(=O)OC)CC2)=O)CCN(C(=O)COCC(C)(C)C)C(C)C1 N1(C(c2cc(SC)nn2C)=O)CCCC12CCN(C(C1CC3OC1C1CC31)=O)C2 C1(CC)CN(C(=O)C=CC2CCC2)CCN1C(c1sc(Br)cc1F)=O c1(C(N(C(C(=O)NCCC2CC3C=CC2C3)C2CC2)C)=O)cc(O)ccc1F c1(N2CCC3(C(C(N4C(C)C(O)CCC4)=O)C3)CC2)cnc2c(Cl)cccc2n1 C1(C(=O)NC(CNC(C(C)CCc2ccccc2)=O)(C)CO)CCc2c[nH]nc2C1 c1(OC)cc(C=O)c(Cl)cn1.n1(CCN2CCNC2=O)cc(CC2CCCNC2)nn1 C1(CNC(C(C)CC2CC2)=O)CCN(C(C23CC(CF)(CO2)C3)=O)CC1 c1(NC(C(CNC(C=CC)=O)OC)=O)cnc2ccnn2c1 C(=O)(C(O)C(C(C)C)OC)N(CC)CC1CCCN1C(=O)C(F)C(F)(F)F C1(CC)CN(C(=O)C(O)C2CCC2)CCN1C(C1CCC2(CC1)CC2)=O C1(C(N(CC(C)NC(=O)Cc2ccccc2F)C)=O)CCn2cncc2C1 N1(C(c2cccc(-c3cccc(C)c3)n2)=O)CCc2c(cnn2C)C1 c1(C(=O)NC(C(C(C)C)NC(=O)Cc2cnc[nH]2)C)cccc(C(F)(F)F)c1F C(C(C)(CC)C(N)=O)NC(C(CC#C)NC(=O)CSC(F)F)=O CC(O)C(F)(F)C(=O)NCC1CC1NC(C1(c2ccc(F)c(F)c2)CCCC1)=O C(=O)(C(C(C)(C)C)OC)NCCN(C(c1cnc(O)c(Br)c1)=O)CC C1(C(=O)OCC2C(OCC)CC2)CCCN(C(C2CC(F)(F)C2)=O)C1 c1(C(N2CC(CN(C(C(CCC)(C)C)=O)C)OCC2)=O)ccc2nnc(O)n2c1 C#CCC(O)C(=O)NCCC1CCCCN1C(c1c(Cl)n[nH]c1C)=O C1(OC(C)C)CCCCCC1CNC(=NCCF)NC(c1cccc(C#N)c1)C N1(C(CC(C)c2ccco2)=O)C(CNC(=O)CC2CCCC2)CC2COCC12 c1(C(=O)NC2(CC)CCCN(C(c3occc3CN(C)C)=O)C2)ccc(C#N)cn1 C1(C(=O)NCC(C)NC(CCc2c(C)n(C)nc2)=O)CCC2CCC1O2 C(=O)(C1=CCN(C(c2nc(C#N)cs2)C(=O)OC)C1)NCCOCC1CC1 C1(CCNC(=O)C(c2ccc(I)cc2)F)(OCC)CCOCC1 c1(C(CC)C(=O)NCC2(O)CC(C(=O)NC)C2)ccc(OC(F)(F)F)cc1.C(C)(=O)O C1(COC)CN(C(=O)C(C)Sc2nncn2C)CCN1C(c1ccn(CC)n1)=O c1(C(N2CCC(O)(NC(CC=C)(C)C)C2)=O)cc(Cl)ccc1OCC C1(C(=O)NC(C(=O)OCC)C)CN(C(C2(C)CCNC2=O)=O)CCC1(C)C c1(C(c2onc(-c3ccn(C(C)(C)C)c3)n2)c2nccs2)cccnc1Cl c1(NCC=C(C)C)nc2ccccc2nc1NC1CCC(C)(C)CC1 Cc1cccc(C(=O)NC2CC23CCN(C(=O)C(C)Cn2ccnc2)C3)c1N Cc1cc(CNC(=O)C(F)OC(F)(F)F)cnc1F.C1(=O)CCCC2(CCC2)N1 N1(CC(=O)NCCC)CCN(C(c2ccc(OCC)nc2)C)CC1 C1(C)(C(=O)NC(C)Cc2cn[nH]c2)CCN(C)C1.N12CCC(C1)C2=O C1(NC(c2c[nH]nc2-c2cccnc2)=O)CCSC12CN(C(c1cc[nH]c1)=O)C2 C(C)(C(CC(=O)N(C)CCN1CCOCC1)NC(C1CC1(C)C)=O)OC N1(C(c2ccc(CC)s2)=O)CCC(C(=O)NCC(C)Cc2cn[nH]c2)C1(C)C c1(NC(=O)CNCCSC(c2ccccc2)COCCO)ccncc1Cl c1(C(=O)NC2(C)CCN(C(c3cnn(C)c3N)=O)C2)cccc([N+](=O)[O-])c1 C1(C(=O)NC2(CC)CC2)CC(=O)N(C)C1.[nH]1cc(C(N2CC(CC)C2)=O)cn1 N1(C(c2c(C)sc(O)n2)=O)CC2CC1CN2C(=O)CC1CCCNC(=O)C1 c1(C(N(C2C3CN(C(=O)CC(C)(C)C4CC4)CC23)C)=O)ccc([N+](=O)[O-])o1 c1(C(=O)NC2(CC)CCN(C(=O)CCOC)CC2)ccn2ncccc12 Cc1cccc(CC(N2CC(C(=O)NC(c3ccccc3O)C)(CC)C2)=O)c1C C12(OC(C)=O)CC(C(N3CCC(CN(C(=O)C=CC(C)(C)N(C)C)C)C3)=O)(C1)C2 C1(CN(C(CCC)=O)C)CN(C(=O)C(=O)NOC)CCO1 CS(=O)(=O)C1(C(=O)NCC=CCNC(c2cnn(C3CCCC3)c2)=O)CCCC1 c1(C(=O)NCC2(O)CCN(C(C(C)(C)OC)=O)CC2)c(C)nc(C(C)C)nc1O C(CN=c1[nH]c(N2CCC(CCCO)C2)nc2ccccc12)C1CS(=O)(=O)C1 C(CO)(CO)(C(=O)O)NC(C1CCN(Cc2ccccc2)C1=O)=O C#CC1(C(=O)NCc2ccccc2CN(C(=O)C(CSC)OC)C)CCCC1 c1(N2C(C3CCN(C(C(c4n(C)ncc4)(F)F)=O)C3)CCC2)ccn2ccnc2n1 Cc1c(C=CC(=O)NCC(C)(C2CCC2)NC(=O)C(O)C2CCC2)cnn1C CC(O)C(F)(F)C(=O)NC1COCC1CNC(=O)Cn1cnc(=N)[nH]1 c1(C(N2CCCC(N(C(=O)CC3CSCCS3)C)C2)=O)ncc(N)cc1Cl n1(C(C)C)ccc(=NC(=O)C2CCC(C)CN2C(C2CC3CCC3C2)=O)[nH]1 c1(C2(C)CC2)ccccc1C(=O)NCC(C)NC(=O)CC1CCCC(=O)N1 N1(C(c2n[nH]c(C)c2Cl)=O)CC(CNC(C2CC2F)=O)OC2CCCC12 CCC(CC)C(C(=O)N1CC(C(N2CCC3(CO)CCC3C2)=O)CCC1(C)C)OC C(=O)(C1=C(C)OCCS1)N1CC(CCNC(c2cc(C)cc(C)n2)=O)(OC)C1 C(C(C)(C)C#CC(=O)N(CC(C)(C)C)CCO)NC(CCCCN(C)C)=O C1(c2ccccc2)(C(N(C2CN(C(c3cccs3)=O)C2)C)=O)CCCO1 Cc1ccc(CSCC(=O)NC2CN(C(=O)C(C)(C)C)CCO2)cc1 c1(C(=O)OCC)n[nH]c(=NC2CC(CCNC(=O)CN=S(C)(C)=O)C2)s1 N1(C(C(CN=[N+]=[N-])NC(C2C(C)(C)C2)=O)=O)CCOCC2(CCC2)C1 CCCC(CCC)C(=O)NC1CCCCC1NC(=O)CC1CCOC1=O C1(NC(C(CNC(CCc2cc(C)[nH]n2)=O)O)=O)CN(C)C(C)(C)C1 c1(C(=O)O)c([N+](=O)[O-])cnc2ccc(NC(=O)C=CCC3CCOCC3)cc12 Cc1cc(C)n(CC(=O)NC2CCNCC2F)n1 c1(NC(CC)C(=O)ONC2CCC(F)CC2)ccccc1Cl CN=c1[nH]c(C(=O)NC(CNC(=O)C(c2cccc(Cl)c2)C)C(C)(C)C)cs1 C1(NC(c2cnn(CCN3CCCCC3)c2)=O)CCc2ccccc2C1 C1(N(C(CC(CC)C2CCC2)=O)CC)CN(C(C2C3(CC3)C23CC3)=O)CC1(C)C c1(C(N2CCCC(CNC(C3C4CCCC34)=O)CC2)=O)cnc2ncccn12 C12(C(N3CCC(C)(CNC(=O)C(F)(F)C(F)F)C3)=O)CCC(=O)N1CCS2 Cc1cccc(F)c1CC(=O)NCCC1(CNC(=O)C=CCN2CCCC2)CC1 N1(C(C2C(OC)C2)=O)CCC(C)(CNC(c2ccccc2OCC(N)=O)=O)CC1 C(CC(C(=O)N1CCC(CO)(OC)C1)NC(=O)COC(C)C)OCC C(C(C)(CC(C)C)NC(=O)C(c1cccnc1)O)NC(COC)=O Cc1csc(=O)n1CCC(=O)N1CCC1CNC(c1cnn(C2CCC2)c1)=O C12(NC(CC=CC)=O)CCC(CNC(C3CC34CC4(F)F)=O)(CC1)OC2 CCCC(O)C(=O)N1CC(NC(c2cc(-n3cccc3)ccn2)=O)C(SC)C1 N1(C(c2occ(C)c2)=O)CC2CC(C1)CN(C(=O)Cn1cnnc1O)C2 c1(CC(=O)N(C)CCNC(=O)CC2CC2(Cl)Cl)cc(F)cc(Br)c1 c1(C(N2CC(NC(C3(C)CCOC3)=O)C2)=O)cc2occc2s1 CC1(C)OCCC1C(N1CCC(NC(=O)CSCc2ccccn2)C1)=O.C1CO1 c1(SCC(=O)NC2CN(C(CSC)=O)C(C)(C)C2)ccc([N+](=O)[O-])cc1 C1(CNC(CC(C)SC)=O)CCCCN(C(c2cnc(C(C)C)n2C)=O)C1 C1(NC(=O)NCCCN2CCCc3ccccc32)Cc2nc3ccccc3n2C1 N1(C(Cc2cc(C)no2)=O)CCOCC1C(C)NC(c1nccnc1C)=O Cc1ncc2c(n1)CCC(NC(=O)C(c1ccc3c(c1)OCCO3)(C)C)C2 c1(C(N2CC(C)C(NC(=O)CC(C3CC3)C3CC3)CC2)=O)cnn2c1CCCC2 CC(C)(C)C(CNC(C1CCCC12CCC2)=O)C(=O)N1CCC(C#N)C1 N1(C(C(CC=C)OC)=O)CCC(NC(=O)C(CC)OC)CC(O)C1 c1(OCCC)nc(C)ccc1C(=O)NC1CC(NC(=O)C=CCF)C1 N12CCC(C)(C)CC1C(=O)N1CCCC1SC(C(=C)C)CC2=O.S(C)CC N1(C(c2cc(OC)ncn2)=O)CCC2CC2(NC(=O)CC2CCC=CCC2)CC1 N1(C(CNC(=O)OCC=C)=O)C(C(=O)NCCCC(=C)C)CC1C C1(NC(c2c(CC)scc2)=O)CC2CC(NC(=O)C=Cc3sccc3C)CC12 N1(C(C2(N(C)C)CCCC2)=O)CCC2(C=C(C(=O)N3CC(O)CC3C3CC3)C2)C1 C1(OC)CCN(c2ncnc3c2cnn3C(C)(C)C)C2CCCCC12 Cc1cc(Cl)c(C(=O)NCCOCCNC(C2CCC3(CC2)CC3)=O)cc1F Cc1cnc(NC2CCN(C(=O)CCCN3CCCCC3)CC2)nc1C N1(C(C(CC=C)NC(c2ccncc2CC)=O)=O)CCCC(O)(CC=C)C1 C=C(Br)CC(C)(C)C(=O)N1CCC2(CC1)CC2C(=O)NCCOC Cc1[nH]nc(C(N2CC3CC(NC(C4CCOCC4)=O)CC3C2)=O)c1[N+](=O)[O-] c1(OC)cc(C(=O)OCCn2cnc([N+](=O)[O-])n2)c(N)c(OC)c1 c1(C(=O)NCc2c(C3CCN(C(C=CCOC)=O)C3)n[nH]c2)nn(C)nc1Br C1(CCC)CCCCN1C(=O)C(O)CNC(=O)C(c1ccn(C)c1)C Cc1ncc(C(N2CC(NC(=O)COC3CCOC3)CC(F)C2)=O)c(O)n1 C1(NC(C(C)NN2CCOCC2)=O)(CNC(c2cc(C3CC3)on2)=O)CCCC1 Cc1c(C(F)(F)F)n[nH]c1C(=O)NCC(CC(C)C)NC(=O)CN1CCC(O)CC1 C1(C(=O)NCC23CCC(CC2)N3C(C2CC23CCC3)=O)CC1C1CCCCC1 C1(NC(C=CCC)=O)CCOCC1CNC(C1(c2ccn(C)n2)CC1)=O c1(C(=O)NCC2N(C(C(CCC)C)=O)CC2)ccc(OCc2cccc(C)c2)cc1 c1(C(=O)NCCN(C(c2cocn2)=O)CC)cnn2cc(C(N)=O)cnc12 c1(C(=O)NC2CCC(CNC(CSCCOC)=O)C2)ncccc1Cl N1(C(C(=O)NCCC2CN(C)C2)=O)CCC2CN(C(=O)OC(C)(C)C)CC2CC1 C1(C(=O)NCC(C=C)(C)C)C2CC1N(C(c1c[nH]nc1OC)=O)C2 NC1CC2(CCC(C(=O)NCC(N3CCCCC3)=O)CC2)CO1 C(CCCCCCO)N.C(=O)(C(C)(C)C)C(C(C)NC(C1CCC(C)O1)=O)=O CC(=O)NCCNC(=O)N(C1CC1)CC1CC1.CCOC C(N=c1[nH]c2c(c(=NC3C=CCC3)[nH]1)CC(C)CC2)c1cnc(COC)[nH]c1=N c1(CC(=O)NCCOC2CN(C(=O)CCOCCF)C2)cccc(Br)c1F C(C(C)(C(F)F)NC(=O)CC1CCCC12CC2)OC c1(CN(C(Cc2ccccc2)CO)CC)ccc(CC(=O)NC)cc1 c1(C(=O)NC(C)(C)CNC(=O)COC2CCCCCC2)cc(N)ccc1OC(F)F O=C(CCC(F)(F)F)NCc1c[nH]nc1C1CCN(C(c2ccc(=N)[nH]n2)=O)C1 C1(NC(=O)NC2CCN(C(c3c(OCC)ccs3)=O)C2)CC2(CNC(=O)C2)C1 C1(NC2C(C)(C)CNC2)CCn2ccnc2C1 C1(CC=C)(NC(C2OCCC2C)=O)CN(C(=O)C(C)(C2CC2)N(C)C)C1 C1(CNC(C2COC(=O)O2)=O)CCC(F)(CNC(C2CCC(C(N)=O)C2)=O)C1 c1(CC(N2CC3C(NC(CC=C(C)C)=O)C(C3)C2)=O)cc(F)c(F)cc1F c1(C(N2CCC(NC(C(C)OCC#C)=O)C2C2CC2)=O)cc(C#N)ccc1F N1(CC)CCOC(C(N2CC(O)(C(C)NC(=O)Cc3cscn3)C2)=O)C1 c1(C(=O)OC)c[nH]c2cc(CNCCC(F)=C(F)F)ccc12 N1(C(CC2C(CC)C2)=O)CCC(CO)(NC(=O)CSc2nnnn2C)C1 Cc1cccc2nc(C(=O)OCc3ccc(N(C)Cc4ccccc4)cn3)cn12 c1(C(N2CC(N(C)C(c3scnc3Cl)=O)C2)=O)ccc2c(c1)C(=O)CCO2 C1(C(=O)NC(C2CN(c3cncc(Cl)n3)C2)C)CC(C(N)=O)C1(C)C C12(C(=O)NC3(CC=C)CCC3)CCCC1CCN2C(=O)Cn1cc(CO)nn1 c1(C(N2CC(N(C(C(C(=C)C)(C)C)=O)C)C2)=O)cnc2c(c1)ncn2C C=C(C)CCCC(=O)NCCN(C)C(c1ccncc1NC)=O c1(NC(=O)NC(C(C)C)Cc2ccccc2F)ccc2nnnn2c1 c1(C(C)Sc2c(C)cccc2)cc(CNC(C)(C)C)nnc1C c1(N(C(=O)CN2CCc3ccc(Cl)cc3C2)CC)cnc2cccc(Cl)c2c1 C(CCC(C)C(=O)N1CCC(N2CCC(NCc3sccc3Cl)CC2)C1)OC c1(CC)occc1C(=O)NCC(CO)NC(=O)Cc1cn(CC)nn1 CC1(C)C(C)(C)C1(F)C(N1CCN(C(c2ccc(F)c(C3(C)CC3)c2)=O)CC1)=O CC(=O)C(C)CC(C)C(=O)N(CC(C)(C)NC(=O)C1=CC(C)(C)C1)C CC1(C(=O)NCCC2CCCC2NC(=O)CSCc2cscn2)CC1(F)F N1(C(c2cc(OC)nc(Cl)c2)=O)CCCCC(N=c2cc[nH]cc2[N+](=O)[O-])C1 N1(C(C=COCC)=O)CCC2C(C1)CN2C(c1ccc(-c2cnn[nH]2)cc1)=O CC1=C(C(=O)NCC2CCCCN(C(=O)Cc3nc(=N)[nH][nH]3)C2)C(C)(C)CCC1 N1(C(C2CCC(C(=O)OCC)C2)=O)CCC(F)(CNC(c2ncn(C)n2)=O)CC1 n1(CCOC)nc(C(=O)NC2CCN(C(=O)C(C)(C)CF)CC2C)ccc1=O C1(CC=C)(NC(c2nocc2C)=O)CCN(C(c2cc(F)c[nH]2)=O)C1 N1(C(CCCCC)=O)CCCC(C)C1CNC(C1(N2CCOCC2)CCC1)=O S(=O)(=O)(c1ccc(Br)cc1NC1CSc2ccccc21)NC1CC(CC)N(C)C1 C1(CN(C(C2(N(C)C)CCCC2)=O)Cc2cc(C(=O)OC)[nH]c2)CC2CCC1C2 C1(NC(C2ON=C(CC)C2)=O)CC2(NC(=O)COC(C3CCCC3)C)COC1C2 Cc1c(C(=O)NCC2(O)CN(C(=O)C=Cc3ccn(C)c3)C2)cnn1CC(C)C C1(NC(C2(C)CCCS2)=O)CC2(C1)CC(NC(c1ccc(C(N)=O)nc1)=O)C2 c1(C(N(C)CC2CCCC(Nc3nccc(C)n3)C2)=O)c(F)cc(C)cc1Cl C(=O)(CCS(=O)(=O)C1CCCC1)NC1C2(CC(NC(=O)C=C3CC3)C2)C1 C1(OC)CN(C(=O)CCCNC(C)=O)CC1NC(c1cc(CC2CC2)on1)=O c1(C(=O)NC2CCC(NC(=O)CCC3CCOC3)C2)ccn2c1CCCC2 c1(C2CC(C(=O)OCCCn3nccn3)C2)cccc(F)c1 Cc1nc(O)[nH]c1C(=O)NCC1(C(F)F)CCN(C(C2(C)CC(C)C2)=O)C1 C1(CC(N2CCCC(N(C(=O)CCSC)C)C2)=O)(CC=CC)CCOCC1 C12(COC)CC(NC(c3cc(C)ns3)=O)(CN1C(=O)C(c1cccnc1)C)C2 c1(C(=O)NCCOc2c(C#N)cccc2F)cc2cncc(Br)c2s1 CC1(CCNC(C2CCC2)=O)CCN(C(c2scnc2C(=O)O)=O)C1 C1(C(=O)NCCn2c(C)ncc2)CN(C(=O)CCCN2CCCCC2)CC1(C)C c1(COC)cccc(F)c1C(=O)N(C1CCCCC1)Cc1ccc(F)cc1 C(=O)(C(C)S(C)(=O)=O)N(CCCCCCNC(C=C(C)c1ccco1)=O)C N1(C(C2(CC)CCC2)=O)CCN(C(=O)CC2C=CCCC2)C(c2ccccn2)C1 c1(C(=O)NCCN(C(C(C)OC)=O)CC(C)O)cc(O)c2sccc2c1 Cc1n[nH]cc1C(=O)N(C(C)C(=O)NCC(O)C1CCC1)C C1(C(=O)Nc2cnc(CCC)nc2)CN(C(C2CCC(C)(C)OC2)=O)CCN1C c1(C(=O)NC2CCN(C(=O)C(C3CCOCC3)F)CC2F)cccn2nnnc12 Cc1ccc([N+](=O)[O-])c(C(N2CCC(NC(=O)Cc3conc3C)C(C)C2)=O)c1 CCC(C)(O)C(=O)NCC(F)CNC(c1c[nH]c(Br)c1)=O c1(CC)[nH]nc(C(=O)NCCOC2CCN(C(c3cc(F)c[nH]3)=O)C2)c1Cl c1(C(=O)NCC(N(C(C(C)NC(COC)=O)=O)C)C2CC2)c(F)cccc1Cl C12(C(=O)Nc3c(C(=O)OC)n[nH]c3)CCN(C1)C2.C1(C(=O)OC)CC(C)CCO1 CCCCC(CC)C(=O)NC(CC)CCCC(=O)NCCOCCCC Cc1ncc(C=CC(=O)NC(C2(O)CN(C(=O)CC3CCS(=O)(=O)C3)C2)C)s1 Cc1cc([N+](=O)[O-])ccc1N1CCC(C)C(NC(C2CC2(C)CC2CC2)=O)C1 C1(C(C)C)CN(C(C2CC(O)CN2C(C)C)=O)CCN1C(c1ncccc1N)=O C1(NC(=O)COC2CCCCO2)CN(C(C2CCCCN2CC(F)F)=O)CC1O C(CN=c1[nH]cnc(C)c1C#N)NC(CN(CCCCCC)C)=O.C(N)=O C1(NC(C2CC(C(C)C)C2)=O)CN(C(C2CC(O)C(F)C2)=O)CC1n1ccnn1 CCN=c1[nH]cc(C(=O)NC2CCCN(C(=O)C(O)Cc3cn(C)cn3)C2)s1 N1(C(CCc2nc(C)sc2)=O)CCC2CN(C(=O)CSC3CC3)CCC12 C1(CNC(c2n(C)ccn2)=O)CN(C(=O)C=C2CCOCC2)CCCO1 c1(NC)ccc(OC)c(N)c1C(=O)NC1CC(F)(CNC(=O)C(C)C(C)(C)C)C1 C1(C)(COC)CCN(C(=O)C(CN(C)C)NC(c2cscn2)=O)C1 C(=O)(C1=NOC(c2ccc(F)cc2)C1)N1CCCC(NC(CN(C)CC)=O)C1 C1(C(N2CC(C)(NC(CC3CC(NC(C)=O)C3)=O)C2)=O)CC12CCCCCC2 CCC(CC(=O)NC(C)(CNC(=O)C(c1cccnc1)O)CO)CC(C)C C1(CNC(=O)C(O)c2ccsc2)CCN(C(C2CCS(=O)(=O)C2)=O)C12CC2 CC1CCc2sc(C(=O)NC3(CF)CCN(C(C4CSCC(=O)N4)=O)C3)cc2C1 Cc1ccc(Cl)cc1C(=O)NCCCC(C)NC(C1(C2(O)CCC2)CC1)=O C=C(C)CC(C)C(=O)NCCC1CCN(C(=O)CCc2cnn(C)c2C)C1 C1(NC(C2CC(C#C)(O)C2)=O)CCN(C(C2CC2C#N)=O)CC12CCC2 S(=O)(=O)(c1cnn(C)c1)NCC(=O)NC(CNC(CC(C)(C)OC)=O)(C)CO C1(CC)CN(C(C2CCN(C)CC2)=O)CCN1C(=O)CC(O)C(C)C C(=O)(CC1=CCCCC1)N1CCCC(CN(C)C(C2COCCOC2)=O)C1 N1(C(c2cc(C)ncc2)=O)CC(NC(c2csc(Br)c2)=O)CC(C)C1 C1(C)(C(N(C2CN(C(CNC(C(CC)C)=O)=O)CC2O)C)=O)C(C)(C)C1(C)C C=CC(CC)CC(=O)NCC(CC(=O)NCC(c1ccccn1)C)OC c1(CCN(C(N(C2CCN(C)CC2)CCO)=O)CCO)c(S(N)(=O)=O)cnn1C c1(COC)nc(C)c(C(N2CC3CC3(CNC(c3ccnc(OC)c3)=O)C2)=O)s1 N1(C(C2N(C)CC(C)(C)C2)=O)CCC(C(N2CCCC(F)(F)CC2)=O)C12CCC2 C1(NC(CC2C(C)=NOC2=O)=O)COC2(C1)CN(C(C1(CO)CCCCC1)=O)C2 c1(COC)nc(C(=O)N(CCCN(C)C)CCNC(=O)C(C)=C(C)C)cs1 C(C(C)(C)CC(=O)N1CCC(C)C1CNC(=O)CCc1cccc(C#N)c1)OC Cc1oc(Cl)nc1C(=O)NC(C)(C)CNC(=O)CCC1CC1C c1(C(N(C2(C(N3CCN(CC#C)CC3)=O)CC2)C)=O)cc2ccccc2[nH]1 N1(C(C2(CCC=C)CC2)=O)CCN(C(=O)C(CNC(C)=O)N(C)C)C(C)C1 c1(CC)nnc(CNC(C2CC2N(C)C(C2(NC(C)=O)CCC2)=O)=O)o1 C1(C)(OC(C)(C)C)CC(NC(c2ccc(Cl)cc2Br)=O)C1(C)C c1(C(N2CCC(CNC(C(C)Cc3cnc[nH]3)=O)C2)=O)noc2c1CCCCC2 N1(C(c2cc(C)c(F)cc2)=O)CC2COCC2(C(N2CCCCC2C#N)=O)C1 C1(NC(CCOCCCOC)=O)CC2CCC1CN2C(c1n[nH]cc1C)=O c1(CC(=O)NC2C(NC(c3c(C)snn3)=O)CCC2)nnc2n1CCCC2 c1(C(=O)NCCC(C)(C)NC(C2CCCOC2)=O)ccc2oc(=N)[nH]c2c1 c1(CCC)cccc(C(=O)NC(C2CCN(C(=O)C(C)SCCN(C)C)C2)C)c1 C1(C(C)NC(C2(C)C=CCC2)=O)C2C3CC4C1C1C2CC3C41.C12CN(C1)C2 C1(NC(c2n(CCOC)ncc2)=O)CCCN(C(C2CCC2OC)=O)C1C(C)C C1(c2n(CC)nnn2)(NCC2CC2)CCCC(NC2(C3CCC3)CC23CCCC3)CC1 Cc1cnc2cc(C(=O)NC(CNC(c3cc(C(N)=O)ccn3)=O)CO)ccn12 C(=O)(C1=CCCCCC1)NC1CCN(C(c2cn(CC(N)=O)nn2)=O)CC1CO C1(NC(C(C(C(C)C)O)C)=O)CS(=O)(=O)C2CN(C(C3CCC3)=O)CC12 C1(C(N2CCC3(C2)CN(C(C2CC4CCC(C2)O4)=O)C3)=O)CN2CCCN1CC2 C(=O)(C(=O)N=S(C)(C)=O)NCc1cn(C2CC3(Cc4c(OC)cncc4)C2C3)nn1 Cc1ccn(C)c1C(=O)NCC(C)NC(c1cc(-c2ccco2)no1)=O CC1(CNC(=O)COCC2CCCO2)CCCN1C(=O)CSc1n[nH]c(O)n1 C1(CC)CN(C(=O)C(CC(C)C)OC)CCN1C(c1ccc(=O)n(C(C)C)c1)=O c1(C(N2CC(CNC(CCC=C=C)=O)C3C2C3)=O)ccc(OC)c(F)c1F N1(C(c2cc(C)nn2C(C)C)=O)CCC2CCN(C(c3cnoc3)=O)CC2C1 C1(C(=O)NCCC(C)NC(c2nc(C)oc2)=O)CCCC(CF)C1 C1(CN(C(c2c(C(C)C)nns2)=O)C)COCCN1C(C1CCCCC1)=O c1(N(C(CN)=O)CC2CCC2)ccc(I)cc1 C12(NC(CC3N(C(CCC(C)CN(C)C)=O)C4C3CCC4)=O)CC3CC(CC1C3)C2 C#Cc1ccc(Cl)c(C(=O)NCC2CCN(C(C3COCCN3C)=O)C23CC3)c1 C1(C(=O)OC)CCN(C(=O)C(=O)NC(C2(O)CCN(CC(F)(F)F)C2)=O)C1C N1(C(c2cc(OC)n[nH]2)=O)CCCC(O)(CCNC(C2CC3CCC2O3)=O)C1 C1(C(=O)NCc2cccc(NC(C(n3ncc(C)c3)C)=O)c2)CCN(C)C(=O)C1 c12c[nH]cc1C2.C12CC(C1)C(=O)NCCOCCN(C)C(=O)C2.CCC.C1(O)CC1 CC(O)CCCCCC(=O)N1CC(=C(F)CNC(=O)C=C2CCN(C)C2)C1 C1(C(N(CC(CN(C(=O)CCC(=O)OC)CC)(C)C)CC)=O)C(Cl)(Cl)C12CC2 c1(N2C(CCNC(c3cnc(C)s3)=O)COCC2)cc(C(N)=O)nc(Cl)n1 C1(CC(=O)NC2CC(CNC(C=C(COC)C)=O)C2)NC(=O)CN(C)C1=O CC1(C)CC(C(=O)NCC2(C)CC2(C)C)CN(C(C2(C)CC3CC3C2)=O)C1 c1(NC(C)C2CC2)ccc(S(=O)(=O)N(C2CCNC(=O)CC2)C)cc1Cl CC1(C)CC(CC(=O)NC2CCC(=O)NC2=O)N(C(=O)CC2CC=CC2)C1 c1(-c2cc(C=O)c(F)cc2)c[nH]c(=NCC(C)CN(C)C)c(C)c1.CCC1CC1 CC(C)CCCCCC(=O)N1CC(NC(=O)CS(N)(=O)=O)C(C2CC2)C1 C1(C(=O)OC(C)(C)C)CC2CN(c3nc(NC(C(C)(C)C)=O)ns3)CC2C1 c1(C(=O)NCCC(=C)CNC(c2ccc(C)nc2)=O)ccccc1SC(F)F c1(OC(F)F)cncc(NC(c2cccc(Oc3cccc(N)c3)c2)C)c1.CO C1(NC(C(c2ccccc2Cl)(C)C)=O)CN(C(c2cnc(N)cn2)=O)CC1(C)C CC(C)CC(C)C(=O)N1CCCC(CCNC(c2nn(C(F)F)cc2Cl)=O)C1 C12(C(=O)NC(CCC)CC)CCC(CC1)N(C(C1CC3C=CC1C3)=O)C2 c1(C(=O)NC2C(C)N(C(=O)Cn3cnccc3=O)CC2)cc(F)cc2ccoc12 c1(NC(C2C(C(N3CCN(C4CCC4)CC3)=O)C2)=O)cccc(C2CC2)n1 N1(C(c2c(OC)ccs2)=O)CCC(CNC(c2ncc(N)cc2Cl)=O)C(F)(F)C1 N1(C(c2c(C)scc2)=O)CC(NC(=O)C(C)CSCc2ccccc2)C(O)C1 N1(C(C2(COC)CC2)=O)CC2(CCCC2NC(=O)CC(C)P(C)(C)=O)C(C)C1 N1(C(CC2CCCN(C)C2)=O)CCC(C(=O)NC2COC(=O)C2)C12CCC2 c1(C(=O)NCC2C(C(=O)NC3(CCC)CCC3)CC2)cnn(C)c(=O)c1 C(=O)(C(=O)N=c1ccn(-c2ccccn2)[nH]1)NC1CN(CC(C(C)(C)C)=O)C1 c1(NC)ccc(C(N2CCCCC2CNC(C2(NC(C)=O)CC2)=O)=O)nc1 CC(=O)CCCCC(=O)N1CCCC1CNC(=O)CCC1(C)CCC1 N1(C(c2cc(Br)ccn2)=O)CCC(F)(C(=O)N(CCn2ccnc2)C2CC2)C1 Cc1cnn(C(C)C(N2CC(C(O)C(=O)N(C)C(C3CC3)C3CC3)C2)=O)c1 n1(CCCNC(C(=O)NC(C)CC2CC2(Cl)Cl)=O)nnnc1C(C)(C)C C1(CCNC(c2c(CC)csc2)=O)CC(F)(F)CN1C(=O)CCN(C)CCO N1(C(C(=O)NC(c2ccccc2)C)C2CC2(Br)Br)CCN(c2nncs2)CC1 C=CCC(CNC(=O)CCCOC)NC(C1(C(N)=O)CC1)=O C1(CNC(C)=O)CN(C(c2nn(C)cc2C(F)F)=O)CC2(CCC2)O1 c1(-n2cc(C(N(C)C=CBr)CCn3ncc(C)c3)nn2)cccc2[nH]ncc12 C1(NC(C2CCCO2)=O)CS(=O)(=O)C12CCN(C(=O)C=CC1CCCO1)CC2 C1(CNC(c2cnc(C)s2)=O)CC2(CC(NC(=O)C(C)c3ccsn3)C2)C1 c1(NC(=O)NC(c2ccc(C)s2)C)ccc(-c2cnco2)cc1.C12CCCN1C2 c1(C(=O)NCC2C(CNC(c3ccc(O)cn3)=O)C2)cc(Br)cc(F)c1F N1(C(C2(CNC(C3COCCO3)=O)CC=CC2)=O)CCN(C2CC2)CC1 Cc1sc2nc(C(C)NC(=O)Nc3cnn(CC(C)C)c3C)nc(O)c2c1C Cc1cccc(C(N2CCC(O)C2C(=O)NCCN(C)C)=O)c1F N1(C(CC2C(C)CCC2)=O)CCC(N(C)C(c2cn(CC3CC3)nn2)=O)CC1 C=CCC(C(=O)N1CCC(C)N(C(=O)CC(C)(F)F)CC1)C(C)(C)C C(=O)(C(F)(CN(C(=O)C(C)NC(N)=O)C)C(C)C)NCC(COC)OC N1(C(c2cc(OCc3cccs3)ns2)C(=O)NCC)CCCC(CNC(C)(C)C)C1 c1(C(=O)NC(C)CNC(=O)C=CCN2CCCC2)cccc2nccnc12 c1(OC)cc(Cl)c(CS(=O)(=O)Cc2nnc(-c3ccc(Cl)cc3)o2)cc1F C12(OC)CCC(C(=O)N(C3CCCN(C(=O)CN(C)C(N)=O)CC3)C)(CC1)C2 C(=O)(CC1=Cc2ccccc2C1)NCC1CC(OC)CN1C(C1CCC(O)C1)=O N1(C(C(=O)NC)=O)CC(CNC(c2cnc(C)c(N(C)C)c2)=O)OC2(CCC2)C1 N1(C(C(c2c(F)cccc2F)C)=O)CCCC2CN(CC3CN(C)C(=O)N3)CC12 c1(OC)nc(=NC2CCC(NC(=O)CSC(C)=O)CC2)[nH]cc1C Cc1cc2cc(C(N3CCN(C(C4CCC(CO)CC4)=O)C4CC34)=O)ccc2o1 c1(CC(=O)NCCC2CCN(C(c3cc(C)c(C)o3)=O)CC2)cn2ccsc2n1 CC(C)C(C)(CNC(c1ccon1)=O)NC(=O)C(=Cc1cn(C)cn1)F C(=O)(CC(C(F)(F)F)c1ccccc1)NCC(=O)NCCC CC(C)(C(=O)NCc1nocc1C(=O)NCC1(F)CC1)c1ccno1 c1(CC(=O)NC(CNC(C2(COC)C=CCC2)=O)C2CCC2)cccnc1C N1(C(c2n(CC)cnn2)=O)CC2(CCN(C(=O)CC3CCCNC3=O)CC2)C1 C(=O)(CC(C)(C)C(=O)N(CCCNC(=O)Cc1nc2ncccn2n1)C)OCC C(CC(C)C(=O)NCC1CN(C(C2(Nc3ccccc3)CC2)=O)C2CC12)=CCC Cn1ncc(C(N2CCC(CCNC(=O)CCc3c[nH]c(=N)[nH]3)C2)=O)n1 Cc1ncsc1C=CC(=O)N(CCCCCNC(c1cc(Br)n(C)c1)=O)C C1(C(C)(C)C)CCN(C)C(=O)C2(CCOC2)C(=O)N1.c1(C2(CC)CC2)cc[nH]n1 C1(CNC(C2(C)CC2Br)=O)CCCCN(C(=O)CN2CCC2)C1 C1(C(N2CC(NC(c3ccn(C)n3)=O)C(CO)CC2)=O)COc2ccccc2C1 C(c1ccccc1)=CC(=O)NC1CC1.C(=O)(C(C)=CC)N(CC=C)CCOC N1(C(c2n(CC)c(O)nc2)=O)CCC2(CCCN2c2cc(O)nc(O)n2)C1 N1(C(C=CC)=O)C2CCC1C(NC(=O)CCCn1ccnn1)C2 c1(C(=O)NC(CC)CNC(=O)COCC(F)F)cnn(-c2ccccc2F)c1N N1(C(CCN(C)CC)=O)CC2CCC(N(C)C(c3cc(C)cc(Cl)c3)=O)C2C1 c1(C(=O)NCC2C3N(C(CNC(=O)NC)=O)CC(CC3)C2)cc(F)cc(C)c1N c12cccc(n1)NC2=O.CCC(C(=O)N(C)CC1(OC)CCC1)NC(N)=O c1(CC)ncccc1C(=O)NC(C)(C)CCNC(=O)C(C)C(C)C C(=O)(C1=NOC(CNC(C2(C#C)CC(=O)C2)=O)C1)N(C(C)CCNC)CC#C C1(CC(N2C(C)(CC(=O)N(C)CC3(O)CCC3)CC2)=O)CC2CCC1O2 Cc1ncc(NCC2CCCN(Cc3cc(Cc4ccccc4)on3)C2)nc1C c1(C(N2CCC(N(S(C)(=O)=O)C)C2)C(=O)NCC2CCOC2)sc(Br)nc1Cl c1(N(c2cc(OC)ncc2C(F)F)CC2CNC2)ncnc2cc[nH]c12 c1(NC(c2n(C(CC)C)nnn2)c2cn(CCCl)nn2)cccc(OC(C)C)c1 C1(CNC(CCCOCCC)=O)CCN(C(c2c(C)noc2CC)=O)CC1(F)F C(c1cccnc1)=CC(=O)N(CC(CC)NC(=O)C(c1cccs1)SC)C C1(CNC(CC(C)(F)F)=O)C(C2CC2)CCN1C(=O)Cc1nc(C2CC2)n[nH]1 n1(C(c2nc(C3CCCOC3)cs2)=O)nc(C(F)F)cc1C1CC1 CC1(C(=O)NO)CCCN(C(=O)CC2CCC(=O)CC2)C1.N12CCC(O)(C1)C2=O C=C=CCCC(=O)NCC(c1ccccc1)N(C(=O)COCC1CCCCO1)C C1(CN(C(C(C)N(C(=O)COCC(C)(C)C)CC)=O)C)CCN(C)CC1 c1(N(CCC)C)ccc(C(N2CCCCC2CCNC(=O)C2=CCSC2)=O)cc1 N1(C(CC2(SC)CC2)=O)CCN(C(=O)C[SH](CCC(F)(F)F)C(C)C)CC1 CCC(CC)C(C)N=c1cc[nH]cc1S(=O)(=O)NC1CC2(CCCO2)C1 N1(C(Cc2c(C)cccn2)=O)CCCC(C(=O)NCc2cc(O)ncn2)CC1 CC12CC(C(=O)O)(C1)C1(CCN(C(=O)N(CCO)CC3CCCO3)CC1)O2 FC1(F)CCCC(NC2(c3nnnn3C3CCCC3)COC(C3CC3)C2)CC1 C1(C(=O)NC2CCN(CCC)C2)CCN(C(C2CC23CCCCC3)=O)C12CCC2 C(=O)(C#CC1(C)COC1)N(C)CC1CCN(C(=O)CC23CCC(C2)C(=O)N3)CC1 Cc1cc(C(N)=O)cc(CCNC(c2cc(Cl)c(Br)[nH]2)=O)c1 C#CC1(CC(C2CNC(=O)C2)=O)CCCC1.C1=CC(=O)NC(C)(C)C1 C1(CC)CC(C(=O)NCCCN(C(=O)CC2CC3CC3C2)C(C)C)CCO1 N1(C(C(CC)CO)=O)CC2CCN(C(C3CC=CCC3)=O)CCC2C1 O=c1n(CC(O)COC(=N)O)nc2ccccn12.N1CCOC1=O c1(C(=O)NCCC2(NC(C=CC)=O)CCCC2)cc2sccc2s1 N1(C(Cc2ccc(OC)cn2)=O)CC2CS(=O)(=O)CC2(NC(c2cscn2)=O)C1 c1(NC(C2N(C(Cc3cc(C)no3)=O)CC(C)C2)=O)ccc2c(c1)CNC2=O C1(CNC(Cc2ccc(C)nc2)=O)CCC(C)N(C(=O)C(n2nccc2C)C)C1 C12(C(N3CCC(C(C)(C)NC(CC(CC)OC)=O)C3)=O)CCC(C#N)(CC1)CC2 C#Cc1ccnc(C(=O)NCC(C)(C)CNC(c2cccc(CC=C)c2)=O)c1 CCC(CCCC(=O)NCCC1(OC)CC1)NC(=O)C(C)(C)C1CCOC1 C(=O)(C1=C(F)CN(C(=O)CCCC(C)=O)CC1)NC(CCC)CC C1(NC(C2C=C(C)CS2)=O)CC(C(=O)NCc2ccc(C)cc2O)C12CCC2 c1(C(N2C(C(=O)NCC3CCNC3)CCC2)=O)cccc(O)c1 N#Cc1c(Cl)nsc1NCC1CCCCC1NC(C1CC12CCCC2)=O C1(C)(C(N2CC(CC)(NC(=O)Cn3ncnn3)C2)=O)Cc2ccccc2NC1=O C=CC(C)(O)CC(=O)N1CCC(N(C)C(c2ccc(CO)cc2F)=O)CC1 c1(C(=O)NC2C(C)N(C(C3CC4CCC3CC4)=O)CC2)cncc(F)c1Cl Cc1ccc(C(N2CCCN(C(=O)C=Cc3ccccn3)CC2)=O)cc1O N1(C(C2N(C(C(CCC(C)C)F)=O)C(C)C2)=O)CCc2cnccc2C1 N1(C(CCCCCSC)=O)CCC2CN(C(=O)CCC3CCOCC3)C(C)C12 c1(C(=O)NCC(C(C)(C)C)NC(C(CC#C)O)=O)ccc(OCC)nc1F N1(C(C(C=C=C)C)=O)CCN(C(C2(CC)CC2)=O)CC1C C1(C(=O)NCC(CCc2ccncc2)OC)C=CC(NC(c2ccccc2)=O)C1 N1(C(C(CC)=CC)=O)CCN(C(c2cc(C)c(N)cn2)=O)C2CCCCC12 c1(OC)ccc([N+](=O)[O-])cc1NC(C1CCN1Cc1cnc(Cl)c(Cl)c1)=O C1CC2C(=O)N(C)CC(=O)N2C1.CC1=C2CN=C(N1)S2.c1ccc(N(C)C)cc1 Cc1cc(C(N2CCC(N(C)CCN(C)C)C2)C(=O)NC2CC2)c2c(c1)CCC2 C(=O)(C(C1=CCSC1)N1CC(C)(C)OCC1CCO)NC(c1ccccc1)C c1(CC)cccc2[nH]c(C(N3CCC4C(C3)CN4C(C3COCCO3)=O)=O)cc12 C(=O)(C(CNC(c1cc(C)cc(C#N)c1)=O)C(C)(C)C)NCCC(=C)C C(CC1=CCN(C(=O)CCc2cnco2)CC1)NC(c1cn(CC)nc1)=O C1(C)(C(N2CC(CCNC(C3CCN(CC)C3)=O)C2)=O)CC=CCC1 [nH]1cc(C(C(=O)NC2CC2)N(CCN)C)c(C)n1.C1(CC)CC2CCC1C2 N1(C(c2cc(C)sc2C)=O)CC(=O)NC2CN(C(=O)CC(C)C3CC3)CCC12 c1(-c2ccc(NC(C)=O)cc2)cc2nc(C)oc2cc1OC(c1cscn1)=O Cc1noc(C)c1CC(=O)NCCNC1(n2cc(CC(O)C3CC3)nn2)CC1 C1(CC(=O)NCC(CC)NC(=O)Cc2csc(C(=O)OC)c2)COC2CC1C2 CC(O)C(C(=O)NCCCNC(C1(C)CC(F)(F)C1)=O)NC(=O)OC(C)(C)C N1(C(CC(C)(C)C)=O)CC(NC(C2CC(=O)N(O)C2)=O)CC2(CCOCC2)C1 N1(C(CCCOCCCCCC)=O)Cc2[nH]cnc2CC1C N1CCCC1C1(C(N2CC(C3CCCO3)C2)=O)CC1.C1(OC)CC(OC)C1 N1(C(Cc2c(C)nc(C)s2)=O)CCC(NC(=O)CC2CCCO2)C(F)C1 C1(C2CCCN(C(=O)C=Cc3ccc(F)c(OC)c3)C2)(NC(C=COCC)=O)CC1 Cc1nc2cc(Cl)cc(C(=O)NC(CNC(C3CC=CCC3C)=O)C3CC3)c2[nH]1 CC1(C)NC(=O)N(CC(=O)NCCC2CCCN2C(C2(C)COC(=O)C2)=O)C1=O C12(C(=O)NCCN(C(CC3CC(=C)C3)=O)CCC)CCCCC1OCC2 c1(CC)cccc(C(=O)NC(CC2CC2)C(N2CCOC(C(N)=O)C2)=O)n1 N1(C(c2n(C(C)C)ccn2)=O)CC(O)CC1CNC(=O)C=CC1CCOC1 C1(C(=O)NC2CN(C(C(CC#C)(C)C)=O)CC2(C)C)CCn2cnnc2C1 C1(NC(c2ccc(N)cn2)=O)CC2CCCC(C1)N2C(C1CC12CC2)=O N1(CC(=O)NC2C3N(C(C(C(CC)C)C)=O)C(CC3)C2)CCCCCCC1=O N1(CC(=O)NC(CCOC)CNC(=O)Cc2cccc(F)c2)CCCCC(O)C1=O C123CCC(C1C2)NCC3.c1(CCCC)csc(C(=O)O)n1 C(=O)(CS(=O)(=O)CCOC)NCC(CC)NC(c1ccc[n+]([O-])c1)=O N1(C(CN(C)C)=O)CCC(NC(c2ccccc2OCC#N)=O)C(CO)C1 c1(C(=O)NCC2N(C(CCCCCOC)=O)CCC2C)cccc2nsnc12 C1(CNC(C2(OC)CCC2)=O)CCC(C)N(C(=O)CCCC2CCCC2)C1 C1(C(N2C(C)(C)CCC2)=O)CC2(CC2)CN1C(c1ccc(F)o1)=O N1(C(C(=O)N(CC(CC)NC(=O)Cc2ccccc2F)CC)C)C(=O)CCC1=O N1(C(CCOCC#C)=O)CC(NC(c2cc(CCC)oc2C)=O)C2CC12 c1(C(N2CC(C)C(NC(=O)CC3C=CCCC3)C2)=O)c[nH]c2c(C#N)cccc12 c1(C(N2CCC(C(CNC(c3c(CC)occ3)=O)F)CC2)=O)cccc(F)c1C C1(C(=O)NCCCOCCNC(C(n2ccc(C)n2)(C)C)=O)CCC2C1C2(F)F c1(Cn2ccc(NC(N(C(C)CN3CCOCC3)CC)=O)n2)cccc(F)c1C c1(NC(C2CN(C(=O)CSCC#N)CCO2)C)ccc([N+](=O)[O-])c(OC(F)F)c1 Cn1ncc(C(N2CCCC2CC(=O)NC(C2(O)CCC2)(C)C)=O)c1N N1(C(c2c(=O)ccn(C)c2)=O)C(CNC(=O)CC(O)C2CC2)CC2COCC12 N1(c2c(C)cncn2)CC2CC1CN2C(c1ccn(-c2cccc(F)c2)n1)=O c1(C(=O)NC2CC(CNC(C3C(C(N)=O)CC3)=O)C2)csc(S)n1 N1(C(c2cc(SC)oc2)=O)CCCC2CN(C(c3cc(=O)cc(Cl)[nH]3)=O)CCC12 C(=O)(CCCC(F)F)N(C(C)CCNC(=O)CSC(F)(F)F)CC(Cl)=CCl C1(CC(=O)NCCN(C(=O)Cc2sccc2C)CCC)CC(C)=NO1 C1(NC(C2CN(C(C)=O)C2)=O)CCN(NC(c2cn(CCO)nc2C)=O)C1C1CC1 c1(C(N(CCNC(=O)CC23CCCC2C3)CC2CC2)=O)ncnc2ccsc12 CC(CN(C)C)N=c1[nH]c(=NCc2cc(Cl)nc(Cl)c2)[nH]c2ccc(Cl)cc12 C1(NC(CC2ON=C(C)C2)=O)CCN(C(=O)C(=O)NCC(F)F)C1(C)C C1(N(C(=O)COC(F)F)C)CCCC(NC(C2(C#N)CCC2)=O)C1 N1(C(CN2CC(CC)C2)=O)CCC2(NC(=O)Cc3nnc(C)o3)CCCCCC12 C1(C)(CNC(CCCOCC)=O)CCN(C(=O)C(C2(OC)CCCCC2)(F)F)C1 C1(NC(C(C(C)O)C)=O)C2CC3CN(C(=O)C(O)Cc4cnc[nH]4)C1C3C2 c1(OC)ccc(CO)cc1C(=O)NC(C1CCCCN1C(C1CC(F)C1)=O)C Cn1cncc1-c1cn(C2CCN(C(=O)C(F)C3CCOC3)C2)nn1 c1(OC)cnccc1C(N1CCC(C)C1CNC(=O)Cc1ccc(C)s1)=O C(=O)(CCCN=[N+]=[N-])NC(CCCNC(c1n(C)ccc1)=O)(C)C Cc1ccc(C(C)CC(=O)N(CCn2cc(CN)nn2)CCF)cc1 C1(C(=O)OCC)CCCC1S(=O)(=O)N(CCO)CC1CC1 N(C(=NCCc1cccs1)NCc1ccnn1C)Cc1ncc(C)nc1 N1(C(C(C)=C2CC2)=O)CCCC(C2(NC(C3(C)CCOCC3)=O)CC2)C1 C12(CCOCC1)C(=O)N2.C1(CC(=O)NC2(C(C)(F)F)CC2)CCCC(=O)O1 C1(NC(C=C(CCC)C)=O)CCC2CCN(C(c3cc(C)ns3)=O)C1C2 CC1(CF)CCN(C(C2(NC(c3cccs3)=O)CC(F)(F)C2)=O)C1 CCC(C)C(O)C(=O)NCCCCCCNC(=O)C(C)n1ccnc1 C(C)(CCNC(C1CC1CF)=O)NC(COCCC)=O C1(C(=O)NCCCC(C)C)CCCCCN1C(=O)CP(C)(C)=O Cc1cc(C(N2CCOC(CCCNC(=O)CC3C(C)C3(F)F)C2)=O)nc(O)c1 c1(C(N2CC(C)C(NC(=O)CN(C3CCC3)C)CC2)=O)ccn2c1CCCC2 C=C(C)CC(C(=O)N(CCOC)CC)NC(c1n[nH]c(C)c1O)=O c1(SCCNC(c2n(C(C(=O)OC)C)nnn2)=O)cccnc1Cl C1(C(N(C2CCC2c2nc[nH]n2)C)=O)CCN(C(=O)Cn2cnnn2)C1 N1(C(C=C(C)C)=O)CCC(CCC(=O)N2CC(C(C)CC)C2)CC1 C1(C(N(C2CCC2)C)=O)CN(C(=O)C=Cc2cocn2)C2(CCC2)C1 c1(N2CCC(CN(CC)CC)CC2)cc(N2CCC(C(=O)NOC)CC2)nc(C)n1 C1(C(C(=O)N(C(CCO)C2CCCC2)C)F)CCN(C(c2ns[nH]c2=O)=O)C1 C1(COC)CCCC1C(=O)N(C(c1ccccc1)CNC(c1cc(Cl)c[nH]1)=O)C CCS(=O)CC(=O)NC(CCN(C(=O)C=Cc1cn[nH]c1)C)C(C)C C#Cc1ccc(F)c(NC(C)CCN(C)C(=O)OC(C)(C)C)c1 c1(CNC(CC2C(CNC(c3c(CC)ncnc3)=O)C2)=O)ccc(F)c(O)c1 N1(C(Cc2ncc(C)[nH]2)=O)CC(CNC(=O)C=Cc2cccc(O)c2)C(C)(C)C1 c1(CC(=O)NCC(CC)NC(=O)CCc2cc(C)on2)ccc(S(N)(=O)=O)s1 N1(CCC(=O)NC2C(CNC(C3OCC(C)C3)=O)C2)CCC(O)CC1 c1(CC)ccc(C(N2CC3C(CN(C(=O)C(C)(CO)NC(C)=O)C)C3C2)=O)cc1 Cc1cc(OCC(N2CCN(C(c3n[nH]c(O)n3)=O)CC2CCO)=O)cc(C)c1 N1(C(C2COCCN2C(=O)CCc2ccoc2)=O)CCC2(CCCNC2=O)CC1 N1(C(Cc2c(C)non2)=O)CC(NC(=O)CCS(C)(=O)=O)CC12CCCOC2 c1(NC(C23CC(NCC(=O)NC4CC4)(C2)C3)=O)ccc([N+](=O)[O-])cn1 C1(NC(c2nc(C)sc2)=O)CC2CN(C(=O)CC(C)F)CCN2C1=O C1(C(=O)OC)CC(C(F)(F)F)CCN1C(=O)C(Cc1ccccc1)C(C)OC C(=O)(CN=c1cc[nH]cc1)N1CC2C(NC(C3CC34CCC4)=O)C(C2)C1 C1(CC(=O)OCC)CN(C(C2CCC3(CC3)C2)=O)C1C(F)(F)F c1(NC(CCN(C(C(CN(C)CCO)O)=O)CCO)=O)ccccc1N C1(NC(Cc2c(C)occ2)=O)CC2CN(C(=O)CCn3ccnc3)CCN2C1=O CC1=C(C(=O)N2CCOCC(NC(=O)Cn3cnc(C(F)(F)F)n3)C2)CCO1 N1(C(C2(CC#C)CCC2)=O)CC(NC(C2CCCC2C2CC2)=O)C(SC)C1 N1(C(C2COCC(C)O2)=O)CCN(C(c2sccc2F)=O)C2(CC2)C1 Cc1cn(C)nc1C(=O)NC1CCC1NC(=O)Cc1nccc(OC(F)F)n1 N1(C(c2cc(C)n(C(C)C)n2)=O)CCC2OCCN(C(C3CCC(C)O3)=O)C2C1 N1(C(C(C)SC)=O)CC(NC(=O)C(C2CCOCC2)F)C2(CCCC2)C1 C(=O)(C1=C(C#N)CCC1)NC(CNC(C(CC#C)O)=O)CC(C)C C1(NC(Cc2c(OC)cccc2)=O)CC2(CCC(NC(C3CC3CF)=O)CC2)C1 C1(CC(=O)NCC2(C)CCN(C(C(C)(C)CC#N)=O)C2)Oc2ccccc2NC1=O Cc1nc[nH]c1CC(=O)NC1CC(C)(NC(=O)C(C)OCCC(C)C)C1 c1(C(=O)NC2C3(CN(C(CC4(C)CC4)=O)C3)SCC2)ccc2c(c1)N(C)C(=O)C2 C(C(O)CN=c1cc(F)nc[nH]1)NC(C(CC)SC)=O CC1CCCCN(C(c2cn(CC(F)(F)F)nn2)C(=O)NC2COC2)C1 Cc1cn2cc(CC(N3CCOC(c4ccc(F)cc4F)C3)=O)nc2s1 C=CCCC(CC(C)C)C(=O)N1CCCC(C(=O)NCc2ccnc(F)c2N)C1 C1(C(=O)NCC2CC(NC(C3CCS3(=O)=O)=O)C2)(CCc2cc[nH]n2)CCCC1 Cc1ccn(CC(=O)NCC(C)CN(C(=O)CCCc2cnn[nH]2)C)c(=O)c1 c1(C(=O)NC2CCN(C(C3C(C=C)C3)=O)C2CC)sc2cc(Cl)ccc2c1Cl C12(C(=O)NCC(=O)NC3C(C)CCC3)CC(NC(=O)COC(C)(C)C)(CO1)C2 C(=O)(CC(C)(C)CC(F)(F)F)NCCCC(C)NC(CCc1c(C)n(C)nc1)=O Cc1nc2n(n1)CCN(C(=O)C(N1CC3(COC3)C1Br)=O)C2 n1(CCC)nc(C2CCCC2)nc1-c1cccc(C)c1 CCCCCC(C)CC(=O)NCC1CCCC2(CN(C(=O)C(O)COC)C2)O1 Cn1cnc2cc(C(=O)NCCCCNC(C3CNC(=O)C3)=O)ccc2c1=O C1(C(=O)NC2C(NC(c3c(C)con3)=O)C2)CCc2c[nH]nc2C1 C12(C(N(C(CNC(=O)C(F)C3CCCC3)C3CC3)C)=O)COCC1C2 C1(N(C)C(c2cnnc(O)c2)=O)CC2CCC(C1)N2C(c1cnc[nH]1)=O N1(CC(=O)O)CCCC(n2cc(-c3c(C)ocn3)nn2)C1.C(=O)(CCOCC1CC1)O N1(C(CC(C=C)(C)O)=O)CCC(C(N2Cc3cncnc3C2)=O)CC1(C)C N1(C(c2cnc(OC)s2)=O)CCC2CN(C(=O)C=Cc3ccncc3)CC12 c1(NC(=O)CC(F)F)cncc(C(N2CCC2CC2(C)CC2)=O)c1 C1(NC(C(C)CF)=O)CN(C(C2(C#N)CCCCC2)=O)CC2(CC2)C1 CCCCC(O)C(C)C(=O)NC1(COC)CN(C(=O)C=Cc2cnccc2C)C1 n1(CC)ncc(C(=O)NC(c2ccnn2C)C(N2CCC=C(Cl)C2)=O)c1C c1(OCC)cc(C(=O)N(C2CCCCC2)CCOC)oc(=O)c1.C1(=O)CC(C)N1 c1(CC(C(=O)NCCN(C(=O)C(C)N2CC(C)C2)C)OC)ccc(F)cc1 C1(CC(=O)NC2CCN(CCCNC(C3(CC(F)F)CCC3)=O)C2)CC1C1CC1 C(C(=O)N1CC(N2CCC2)CCO1)C(COCC)(C)C(=O)OC(C)(C)C C1(CC(=O)NC(CN(C(c2ncn(CC)n2)=O)CC)C)CCCC(=O)N1 Cc1cc(C(=O)NC2COCC2NC(c2c[nH]nc2C2CC2)=O)cnc1C(F)F N1(C(C)CNC(c2ccnnc2)=O)CCN(C(C2(F)CCCC2)=O)CC1 c1(CNC(CC2C(C)(C)C(NC(=O)CC3CSC3)C2)=O)cccc2c1CCC2 N1(C(CC(C(C)C)(F)F)=O)CC2CCC(C1)N(C(=O)C=CC1CCOCC1)C2 N1(C(C2COCCN(C(c3c(CC)c[nH]n3)=O)C2)=O)CC2CCCCC12C N1(CC)CCCC(C(=O)NCCn2cc(NC(=O)CC(C)N(C)C)nn2)C1 C=C(Cl)CCC(=O)NC(CCOCCO)C(=O)Nc1cccc(N(C)C)c1 C1(NC(c2c(C)cccn2)=O)CCN(C(=O)CCN2CCCCCC2=O)CC1F CC(=Cn1ccnn1)C(=O)NCCCCNC(C1SCCS1)=O C1(CCC)(NC(C2CCN(C3CC3)C2=O)=O)CCN(C(=O)CCS(N)(=O)=O)CC1 C1(C(=O)NCCCN(C)C(C23CCCN2CCC3)=O)C(F)(F)C12CCC2 C=CC(F)(F)C(=O)NC1CC(NC(c2csc(O)n2)=O)C1 n1(CC(N2CCC(NC(C3C(C)C3)=O)C2(C)C)=O)nnc2c1CCCC2 C1(NC(C(C)=C2CCCC2)=O)CC2(CCN(C(C3(C#N)CCOC3)=O)C2)C1 c1(CC=C)ccnc(C(=O)NC2(C(=O)NC(C)C=CC)CC2(C)C)c1 c1(C(CC)C)ccc(OCC(=O)NC2CCC(NC(=O)CC3CC3)CC2)cc1 CCC(CC)C(C(=O)NC1CCC(C(=O)N(CC(C)O)C2CC2)C1)OC C#Cc1cccc(CC(=O)NC2CC(NC(C34CC(C)(CO3)C4)=O)C23CCC3)c1 Nc1ccc(C(=O)NCC2CN(C(C34CC(CN3C3CC3)C4)=O)CCO2)cc1O C1(CONC(C(C2(O)CCCCC2)NC(c2nc(C)sc2)=O)=O)CC2C=CC1C2 CP(C)(=O)CCC(=O)C1C2C(C1)N(C(Cc1c(O)cccc1F)C(=O)N(C)C)CN2 CCC(C)CCCCC(=O)N1CC(C)(C)CCC1CNC(=O)CSCC(F)(F)F C1(C)(NC(c2cccc(NC(c3c(C)cc(O)nc3)=O)c2)=O)CN2CCC1CC2 C1(CC(=O)N(C)C)CC(NCCc2cn(CCN(CC)CC)nn2)C1(C)C Cc1ccc(O)c(C(=O)NCC=CCNC(c2ccc(C(C)(C)C)nc2)=O)c1 c1(C(=O)NCCN(C(c2ncccc2C(C)=O)=O)CC)ccccc1OC CCCC(C(C)C)c1nc(C2CCOC2)nn1-c1ccncc1C Cc1ccc(CC(=O)NC2CN(C(=O)CSc3n[nH]c(=N)s3)CC2(C)C)c(F)c1 S(=O)(=O)(c1c[nH]c2c(Br)cccc12)NC(c1ccc(N2CCOCC2=O)cc1)=O c1(C(=O)NCC2=CCN(C(C3CC34CCOC4)=O)CC2)c(O)ncc2c1CCC2 C1(CN(C(C)C)C(C2CC2)=O)CCCN(C(C2CC(N3CCOCC3)C2)=O)C1 CC(c1ccco1)=CC(=O)NCCCC1CCCN1c1ccnc(C2CC2)n1 c1(OCC)cccc2c1OCC(C(=O)N(C1CCCN(C(=O)C=CCF)C1)C)=C2 c1(C(=O)NCCC(O)C(=O)NCCc2ccccc2)ccc2cc[nH]c2c1 N1(C(C2CC3CCC2CC3)=O)CC2CC(NC(C3(n4nccn4)CC3)=O)CC2C1 C1(C(N2CC=CC(C(=O)NC(COC)(C)C)C2)=O)CCCC12CCC2 C1(C(C(=O)NCCNC(C2C(CC)OCC2)=O)O)CCCCCC1 CCC(C)C(O)CC(=O)NC(CC)CCCC(=O)NCc1cnn(C)c1 C1(NC(c2c(CCC)nns2)=O)CCC(C)(CNC(c2ccc[nH]2)=O)C1 Cc1cc(C)nc(N2CCN(Cc3cccc(O)c3Cl)CC2CO)n1 c1(C(N(CC(O)CN(C)C(C2COC(C)(C)CO2)=O)C)=O)cc(S(N)(=O)=O)c[nH]1 c1(CN(C)CCC2CCCCN2C(c2cc(CO)on2)=O)ccc(F)c(O)c1 C12(NC(C(CC)F)=O)CC1CN(C(c1cncc(-c3ccccn3)c1)=O)C2 N1(C(=O)CCc2nc(C3CC3)no2)CC2CC(C1)N(C(c1cocc1Br)=O)C2 Cc1nn(C)c(C)c1CN(C(=O)C(c1cnn(C)c1)O)CC.c12ncnn1C1CN2C1 N1(C(C(COC)(C)OC)=O)CC2(CCC2)CC1CNC(c1ccoc1Br)=O C=CCC(C(=O)NCCCNC(=O)C(CCCC)Oc1ccc(Cl)cc1)C(C)C n1(CCCC)nnnc1C(C)(CCC1CCC1)NCCCCCC1CC1 C1(NC(c2ccn(CCF)n2)=O)C2CN(C(C3(F)CCCOC3)=O)CC12 c1(C(=O)N(CC2C(NC(CCCCOCCC=C)=O)C2)CC)c(N)cccc1F c1(C(N2CC(C(=O)NC(CCO)C3CCC3)(CC)C2)=O)cc2ccccc2[nH]1 N1(C(C2(OC)CCN(C(=O)CSC3CC3)C2)=O)C2CCCC1COC2 c1(N2CC(C)C(F)C2)nc(=NC2CCCN(CCOCCO)C2)[nH]c2cc[nH]c12 Cn1nc(Cl)c(C(N2CCC(OCCNC(c3cc4occc4[nH]3)=O)C2)=O)c1Cl c1(OC)c(Cl)ccc(Cl)c1CC(N1CC(NC(C2CC(F)(CO)C2)=O)C(F)C1)=O CN1Cc2ccc(C(=O)NC(CNC(C3CCNC3=O)=O)C3CC3)cc2C1 CCC(CC(=O)Nc1cnccc1C(C)C)N(C)C(c1cc(C)[nH]n1)=O C=Cc1cc(C(N2CCC3(C2)CN(C(c2ccnc(OC)n2)=O)C3)=O)cc(F)c1 CCCCCCC(CC)C(=O)NC(C)CNC(c1cncc(NC)c1)=O C1(CC=C)(C(=O)NCCC2(O)CN(C(c3cc(C(C)C)on3)=O)C2)CCOCC1 N1(C(C2(F)C(C)C2)=O)CCC(n2cc(CNC(C3(C)CC3)=O)nn2)C1 Cc1ccc(NC(=O)NC23CCC(CN4CCCCCC4CO)(CC2)C3)c(C)c1 C1(CC(=O)NC2C(C(=O)NCCCOCCCC)C2(C)C)OCCC1(C)C C(=O)(C(CCC(N)=O)N(C)C)N1CCC(NC(C(C)OC)=O)CC1 C(C(F)(C(=O)NC1C(C)C1(C)C)C(C)C)NC(C=C(C)C(C)(C)C)=O Cn1cc(NC(C2COCC2CNC(=O)CC(C)(C)C2CCCCC2)=O)c(C#N)n1 C1(C)(COC)CC(NC(C2(CSC)CC2)=O)CN1C(c1oc(C(C)C)nc1C)=O C(C)(C(C(=O)NCC1OCCC1(C)C)C(C)C)NC(c1c(NC)nccc1)=O C(C)(C)(CN=c1[nH]c(N2CCC(C(C)C)CC2)nc2c1CCCCCC2)N(C)C c1(C(=O)NC(CNC(C(CC)CN(C)C)=O)CO)ccc(C)c(C)n1 c1(NC(C2CC(N)C2)C)nc(Cl)ccc1O Cc1ccc(CN2CCC(NC(c3oc(C(C)C)nc3C)=O)C(F)C2)c(O)c1 c1(OC)cnc(C(N2CC(CN(C)C(C3CC(O)C3)=O)C3(CC3)C2)=O)c(F)c1 C#CC1(O)CC(C(=O)NCC(CC(=O)N(CC(O)CNC(N)=O)C)C2CCC2)C1 C(=O)(C(F)C(C)CNC(C1CC(F)C1)=O)NCC(C(=O)OC)C CC1CCCC(N(C(=O)C(C)(C)C)C2CCC2)C1.C12(CC1)C(=O)N2 c1(C(=O)NCCC(=O)Nc2c(CC)cccc2)nccc(C#N)c1Cl C=C(C)CC(C)C(=O)NC1(CF)CCN(C(c2cc(Br)n(C)n2)=O)C1 CCCCC(O)C(=O)NC1CCCC1NC(=O)CCc1ccon1 c1(C(=O)NCC(C(C)C)NC(c2ccc(C(=O)OC)s2)=O)ccc(CC(C)C)cc1 Cc1c(CC(N2CC(CN3CCCC3)CC2C)=O)cnn1C.C12(CC1)C(=O)N2 C1(C(N2CC(CC)(OC)C2)=O)CN(C(=O)C(C)N=[N+]=[N-])CC1O C1(NC(CCC(=C)Cl)=O)CC2CC(C1)N(C(c1cccc(N)c1F)=O)C2 Cc1cn(C)cc1C(=O)NCCN(CCCN(C)C)C(c1ccc(C(N)=O)o1)=O C(Cc1cc[nH]n1)(C(=O)NCC1(O)CCOC1)NC(=O)Cn1cnnc1 C1(NC(c2nc(C#C)sc2)=O)CCCN(C(C2CC2(F)F)=O)CC1 c1(C(N(C(C)C)CCNC(C2(C(F)(F)F)CC2)=O)=O)ccc2c(n1)CCC(C)C2 c1(C(=O)NCC(C)CNC(=O)Cc2cnccn2)ccc(C(F)F)c(Cl)c1 c1(C(N(CCN(C(=O)Cc2sc(O)nc2O)CC)CC)=O)ccc(F)c(F)c1F N1(C(c2c[nH]c(=NC)o2)=O)CCC2(CC1)C(OC)CC2NC(c1ccc(C)o1)=O c1(C(N2C(CNC(CCOC(C)=O)=O)CCC2)=O)cc(C(C)C)nn1C c1(C(=O)NC(CN(C(=O)CC2(C)CCOC2)CC)C)ccc(NC)cn1 C1(CC)CN(C(=O)C(=Cc2c[nH]cn2)F)CCN1C(C1CC1c1sccc1C)=O Cc1sccc1CC(=O)N(C)CC=CC(=O)NCC1(CC(C)C)CCC1 O=C(C1Cc2ccc(F)cc21)NCC1CCN(c2nnc(CO)s2)C1 C(=O)(C(C(C)C)N1CCC(C)CC1)NCCCCNC(CCNS(CC)(=O)=O)=O C1(NC(=O)Oc2ccccc2)CCC(OCC2CCCCO2)CC1 C(CNC(c1cnn(CCCOC)c1)=O)(C(C)(C)C)NC(C(CC)OC)=O c1(NC)cc(Cl)ccc1C(=O)NCCC(C(C)C)NC(c1cc[nH]n1)=O C1(NC(C2(C#C)CC2)=O)CC2CC1CN(C(C1CCC(O)CN1C)=O)C2 C(=O)(CC(C)CNC(=O)CC1CC(OC)C1)NC1(C)CC(C(=O)OC)C1 c1(CCN=C(NCC(C)C)NCC(C)OC(F)F)ccc2c(c1)OCCO2 CCCC(C)(C)C(=O)NC1CCC(N(C)C(c2cnn(CCO)c2CCC)=O)C1 C(=O)(C(C)C(O)C(C)C)NC(C(C)C)C(=O)N(CCCOCCC1CCCC1)C Cc1ccc(C(=O)NCCCOCCCNC(=O)C=CCN2CCCC2)[nH]1 C1(NC(c2cccnn2)=O)CCN(C(C2(O)CCSC2)=O)CC1CO N1(C(C(CCC)Cl)=O)CCC12CCCN(C(c1cccc(CC)c1)=O)C2 C1(C(N2CC(C(C)NC(=O)Cc3cc(C4CC4)no3)C2)=O)CCc2c[nH]nc2C1 C(=O)(C1=NOC2CCN(C(c3ccco3)=O)CC12)NCCCCOCC C1(CNC(c2scnc2-c2ccc(C(=O)O)cc2)=O)CCn2nccc2C1 C1(NC(c2c(CC)onc2)=O)CC2CC(NC(=O)CCCc3csc(=N)[nH]3)CC12 c1(-c2nnc(CN(CCCn3c(=O)oc4ccccc34)C)o2)cc(F)c(F)c(F)c1 C(c1ccn(C)c1)=CC(=O)NCCNC(c1c(SC)ccs1)=O N1(C(CCc2n(C)ncn2)=O)CCC2(CC(NC(=O)C=CC3CC3)C2)C1 CCCCC(C(=O)O)OC.c12ccc(nc1)-n1cc(nn1)C(C1CC1)NC2=O C=Cc1ccc(C(N2CCOC(C(=O)NCCOCC3CC3)C2)=O)cc1 S(=O)(=O)(c1cnc(NC(C2CCN(C(=O)OC(C)(C)C)C2)=O)s1)NCC N1(C(c2scnc2C2CC2)=O)CC2CCCC(C1)N2c1nccc(C(F)(F)F)n1 C1(NC(=O)CN2CCN(Cc3ccsc3)CC2)CCc2c[nH]nc2C1 c1(C(=O)NC(CN(C(C2CCC(=O)N(C)C2)=O)CC)C)cnc2c(C)nsc2c1 C1(C(=O)NCC23OCCC(C(=O)N)(C2)C3)CC2CCC(C1)N2C.C1(COC)CC1 c1(C(=O)NCCc2ccn(CC)n2)cc(F)c(C)cc1Cl Cc1coc2c(NC(=O)NCC3(C)COCCO3)cccc12 Cc1ccc(C(=O)NCC2(C)CCCN(C(C3CC(C)(C)CCO3)=O)C2)c(O)n1 c1(SC(C)C(=O)NCC(CO)NC(c2cnc(O)s2)=O)ccccc1Cl N1(C(=O)CN2CCOCC2=O)CC2CCN(C(c3ccc4nsnc4c3)=O)C2C1 C1(c2cn(CCCC)nn2)CCCN(C(=O)CCCCOC2CCOCC2)C1 c1(C)cccc(C(=O)O)c1.n1(CCSCC)cc(C2CCOC2)nn1 n1(CC)nc(C(N2CCC(C(C)(O)CNC(=O)C=CS(C)=O)CC2)=O)ccc1=O C(C(C)(O)COC)N(C(CNC(CCOCC#C)=O)=O)CC c1(NC(C2CC(NC(c3ccnc(F)c3Cl)=O)C2)=O)c(Cl)cnnc1Cl CS(=O)(=O)c1cc(C(N2CCC(NC(=O)Cc3c[nH]c4ncccc34)C2)=O)co1 N1(C(C=CCC)=O)CC2COCC2(C(=O)NCc2c(C)cccc2C)C1 C(=O)C(O)CC(C)(C)C.C(C)(C(=O)NCCCOCCOC)SC N1(C(C2CC(C)CC(C)C2)=O)CCOC2(CCN(C(=O)CN3CC=CC3)CC2)C1 c1(CNC(C2(c3cc(F)cc(Cl)c3)CCC2)=O)csc2c1CCCC2 C1(NC(C(CN(C)C)OC)=O)CN(C(=O)C=CS(C)=O)CC1C C12(CNC(C(C)=C(CC)C)=O)CC1CN(C(c1cnn(CC)c1C1CC1)=O)C2 c1(C(=O)NC(C(C)NC(c2cnc(SC)s2)=O)C)cc2ncccc2o1 c1(OC)cc(C(=O)NC2(C)CCN(C(=O)C(F)C3CC3)CC2)c2ccccc2n1 CC1CN(CC(N)=O)CCN1c1cc(C(=O)NC2(C3CCCO3)CC2)ncn1 N1(C(C(CC)C#N)=O)CCCC2(CCN(C(C3CCC4C(C3)C4(F)F)=O)C2)C1 C1(C[SH](=O)=O)CCN(CCN(C)CCOC)C1.C1(NC(=O)NC(C)(C)C)CCCS1 N1(C(c2cncc(NC(C)C)c2)=O)CCCCC(NC(=O)C(C)n2cncn2)C1 c1(OC)cc(C(=O)NC2(C)CCN(C(c3cccc(F)c3Cl)=O)C2)cnc1O c1(C(N2C(C(=O)Nc3ccno3)CC(F)C2)=O)cccc2cnccc12 S(=O)(=O)(c1cccc(F)c1F)NCC(=O)NC(CC(N)=O)C(=O)O C1(C(=O)NC(c2ccc(C)nc2)C)CCOCCN1C(c1nnc(S)n1C)=O c1(C(=O)NCC(C2CC2)NC(CCCOC(C)=O)=O)nc2cccnc2s1 c1(OC)ccc(S(=O)(=O)N2CC3CN(C(c4cc(C#N)ccc4Cl)=O)C3C2)cn1 C1(C(=O)NC(C2CCOC2=O)(C)C)CCCN(C(C2CC2(F)F)=O)CC1 S(=O)(=O)(c1ccc(N2CC(N(C)C)C(C)(C)C2)c(Br)c1)NC(c1nnc(C)s1)C N1(C(C2(CCNC(C=CC(CC)C)=O)CC2)=O)CCC2(CCCO2)C1 C(=O)(C1CCCc2n[nH]cc21)N1CCC(NC(CCC(C(C)(C)C)O)=O)CC1C c1(CC)ccc(C)c(C(N2CCN(C(=O)Cc3[nH]cnc3C)C3CC23)=O)c1 CCC(C)CC(=O)NC1C2CC1N(C(=O)C(C1CCCO1)OC)C2 C1(NC(c2ccoc2)=O)CCCC1NC(c1sccc1Cc1ccccc1)=O c1(CC(=O)NCC(C)=CC(=O)NCCN(C)C2CC2)cnn(C)c1C c1(C(N2CCC(NC(c3ccc(COC)s3)=O)C2C)=O)ccc(F)c(F)c1 C1(CC(=O)OCC2(Oc3cc(C)sc3)CC2)CC2(C1)CC1(CCC1)C2 CC1=C(C(=O)NC2CC(NC(=O)CCC(F)(F)C(F)F)CC2O)S(=O)(=O)CCO1 C12(C(=O)NC(CC)COC(F)(F)F)CCC(n3cc(CN(C)C)nn3)(CC1)C2 CC(C)C(CNC(=O)Cc1nccn1C)NC(c1ccoc1C(F)(F)F)=O N1(C(=O)C(F)C2CCOC2)CC(F)(F)c2ccccc21 c1(C(N2CCC(F)(F)C(Nc3ncccn3)C2)=O)coc2cc(O)ccc12 c1(N2CC(C)(NC(CC(C)(C)SC)=O)C2)cc(=O)n2ccncc2n1 c1(C(N2CC(CNC(C3N(CC)CCC3)=O)(OC)C2)=O)cn2nccc2nc1C C1(C(=O)NC(CN(CCCC)C)C)CCC(O)CN1C(C1CCC(=O)CC1)=O N1(C(C2(c3ccc(Cl)c(F)c3)CC2)=O)CCC2(CC1)OCc1ccccc12 Cc1cc(F)c(C(N2CCOC3(CCC3)C2)C(=O)NC2CCOC2)nc1Br c1(C(=O)NCC(C(=O)NC(COC(C)=O)CO)C)c(C)nn(C)c1N N1(C(C)C)CC(OCC(N2CCN(C(=O)CN3CC=CC3)CC2)=O)CC1=O CCC(C)CC(C(=O)NCCCN1CCCC1=O)NC(=O)CSCC(F)F C(C)(C)(C(=O)NC1CC(CNC(C2CC2c2cccnc2)=O)C1)OC(C)C C1(C(N2CC(NC(C(N)=O)=O)C3(C2)CCC3)=O)Cc2ccc(F)cc2C(=O)O1 N1(C(C)CN(C)C)CCC(C(=O)C(C)(C)C)CC1 CC1(C)C(C(N2C3C=CC(C3)C2C(F)F)=O)CCS1(=O)=O CC1CCC(C)(C(N2CC(C)(NC(=O)CC(C)(F)F)C2)=O)C1 C1(CC=C)(NC(=O)CCCCCC)CC2CCC(C1)N2C(c1n[nH]c(C2CC2)n1)=O c1(C(C(=O)NCC)NC(CCN2CCN(CCC#C)CC2)=O)cccc(F)c1F C(C(CC(=O)N1CC(F)(C(=O)OC)C1)OC)NC(C(CC)SC)=O N#CC1(C(=O)NC2CCCCC2CNC(=O)CC(F)(F)F)CC2CCC1CC2 CC1(CC(=O)NC2CC(F)(CNC(=O)CC3CC(CF)C3)C2)CCOCC1 C1(NC(c2cc3c([nH]2)CCCC3)=O)C2CC3CN(C(=O)CCCCCF)C1C3C2 C1(CNC(C2(CC=C)CCC2)=O)CC2COCC2N1C(c1ccc(N)cc1Cl)=O CCC(C)(C(=O)NCn1cc(CCC(=O)OC)nn1)OC.c1(C)ccccc1 C1(CCC#C)CCCN(c2ccnc(NC3CCOC3)n2)C1 C1(C(N2CCCC(N3CCCCC3)C2)=O)(OCC)CCSCC1 c1(CC(N2C(CN(C(c3oc(C)cc3C)=O)CC)CCC2)=O)ccc(F)cc1 Cn1cc(CC(=O)NCCn2cc(CNC(c3csc(F)c3)=O)nn2)nn1 Cc1cc(C(=O)N(CC(C)(C)NC(c2csc([N+](=O)[O-])c2)=O)C)c2nccn2c1 c1(CCC)c(C(=O)NCCCN(CCO)C(C2CC3(CCC3)C2)=O)nnn1C C1(C)(C(N2C(CNC(c3[nH]cc(C(C)=O)c3)=O)CCC2)=O)CCCCNC1=O N1(C(C(CCCC)O)=O)CC2CCC(C1)N2C(C1(C)CC2CCC(C1)S2)=O N1(C(CCNC(=O)NC)=O)CCC(NC(c2cc(Cl)ccc2O)=O)C(C)(C)C1 C1(CNC(c2ccc(CC)cc2)C(F)(F)F)CCC2(CCC2)OC1 Cc1ccc(I)c(C)c1NC(C1CCC2(CN(C(=O)Cn3cccn3)C2)O1)=O CN1CCCC(CC(=O)NCC2CCC2C(=O)NC2CC23CCC3)C1 C(=O)(C(C)CCC(C)(C)C)NCC(C)CN(C)C(c1ncn(C(C)(C)C)n1)=O CC1CN(C(=O)C=CC2CCCC2)CC1CNC(=O)CSc1cccc[n+]1[O-] c1(C(=O)OCC(=O)NCC2(C(=O)OC)CCCC2)[nH]nc([N+](=O)[O-])c1Cl CC1(C)C(NC(=O)C=Cc2ccncc2)CCN1c1ncc(C(F)F)cn1 N1(C(c2nc(Cc3ccccc3)no2)C)C2CCC1(CCO)CC2 C1(C(=O)Nc2cc(Cl)ccc2O)CC(F)CN(C(=O)CCN2CCCCC2)C1 c1(C(=O)NCC2C(CNC(C3(COC(C)C)CC3)=O)C2)ncc([N+](=O)[O-])n1C c1(CC)cc(OC)ccc1C(N1CC(OC)C(CNC(=O)C(F)CC2CC2)C1)=O c1(C(=O)NCC2(CN)CC2)coc(NC2(CCCC)CC2)n1 C(=O)(C1CCCn2nccc21)NC1CC2(CCCN(C(C(C)NC(C)=O)=O)C2)C1 N1(C(C2=CCC(NC(c3n(CC)nnc3)=O)C2)=O)CC(C)(C)OC(C)(C)C1 N1(C(C2(CC)CCC2)=O)CC(CNC(=O)C=CC=C(Cl)Cl)CC1(C)C C(=O)(C#CC(C)(C)CNC(=O)Cc1cnn(C)c1)N(CC(CC)(C)OC)C c1(N2C(C3(CO)CC3)COCC2)cc(C2CC2)nc2c(Cl)cnn12 C12(OC)CCC(C(=O)NCC3CCN(C(=O)Cc4ccno4)CC3C)(CC1)C2 c1(SC(C(=O)NCCC(CNC(CNC(CC)=O)=O)O)C)ccc(C)c(C)c1 C1(C(N2CCC(O)(CN(C(CC(C)C3CC3)=O)C)CC2)=O)OC(C)(C)OC1(C)C C1(NC(c2ccc(CC)s2)=O)CC(NC(=O)CN2CSCCSC2)C(O)C1 CC1=C(C(=O)NC2C3CCN(C(c4nn(C(F)F)cc4Cl)=O)C23)SCCO1 C1(C)(C(=O)NCC2(C)N(C(c3cc(OCC)n[nH]3)=O)CCC2)CCN(C)CC1 C1(NC(=O)NCC=CCCC)(CO)CC2CC2C1 c1(CS)ccc2c(c1)OCCNC2=O.O=C(C=CC(=O)N(CCO)CCl)COCC1CC1 CCC(C)C(O)CC(=O)N1CCC(C(=O)NC(C)C(=O)N(C)OC)C1 c1(C(N(CCCN(C(=O)Cn2[nH]cnc2=N)C)C)=O)nn(C)cc1Cl C12(C(=O)NCCc3ccc(Cl)cc3)CC1CN(C(C1C=CCN1)=O)C2 C(C1c2ccsc2CCN1C(=O)CSc1cn[nH]c1)NC(=O)Cn1nccn1 N1(CCCNC(C2CC2NC(=O)CCC2CCC2)=O)CCN(CC(F)F)CC1 N1(C(Cc2ccc(C)o2)=O)CCC(O)(CNC(=O)CCOCC2CC2)CC1 c1(C(=O)NC2C3CN(Cc4c(OC(C)C)nccc4)C2C3)cc(C(N)=O)cc(F)c1 C1(C(=O)NC2CCC(NCc3ccc(OC)c(O)c3)C2)CC(=O)CC12CCC2 c1(C(C2CC(OC)C2)NC(=O)C(=O)NC(C)C)nnnn1C1(C)CC1(Cl)Cl c1(CCCCC)ncc(C(=O)NC(C2CCCC2)CNC(C2(CCC)CC2)=O)o1 c1(CC)ccc(C(=O)NC2CC(CNC(=O)CC(C)(F)F)C2)c(F)c1 C(=O)(C(F)(CC)C(=O)OC)NC1(CCCNC(c2ccc(COC)o2)=O)CC1 N1(C(=O)NCc2ccn(-c3ccc(F)cc3)n2)CCC12CCC(C(=O)O)CC2 C=CC1(Nc2cccc(OC)c2C(c2nnnn2CCOC)CC)CCCCC1 C1(CNC(C2C(C)C2C)=O)COC(C)(C)CN1C(c1cnn2cnnc2c1)=O CC1CC(C(=O)NCC(C)(C2CCC2)NC(=O)CCOCCN(C)C)=NO1 N1(C(CC(C)C)=O)CC2CCCCC2(C(=O)CCC(C)(F)F)C1 N1(C(c2c(C)ccc(C)c2)=O)CC(C)CN(C(c2ncc(Cl)cc2Cl)=O)CC1C C(CO)(C(C)N=c1nc(N2CCN(CCS(N)(=O)=O)CC2)c2c([nH]1)CSC2)SC N1(C(CC(CC)O)=O)CC2(CCCC2N=c2scc(C)n2CCC(=O)OCC)C1 c1(N(C)C)cccc(C(=O)N(C2C3CN(C(=O)C4CC4)CC23)C)c1 C(=O)(C#CC1CCCCC1)N1CCC(N(C(=O)CN(C2CC2)CC)CCC)CC1 N1(C(c2conc2C)C(=O)NCCSC)CCN(C)c2ccccc2C1 N1(C(C2C(CCC)C2)=O)CCCCCC1C(N1CC(CO)C(CCO)C1)=O C1(C(N(CC(C)SC)C)=O)CC(N=[N+]=[N-])CN1C(=O)Cc1csnc1C c1(OC)cc(C(=O)N(CC(C)O)CCNC(C2CC2C)=O)cc2c1OCCO2 c1(C(=O)NCC(CO)NC(C(c2scc(C)n2)(F)F)=O)cccc2c1nnn2C C(=O)(C1CCCc2nnn(C)c21)NCC1CC(NC(C=C(C)C)=O)C1 c1(N(CCC)CCC2CCCCO2)ccc([N+](=O)[O-])cc1S(=O)(=O)CC(=O)OC N1(C(CN(C)C)=O)CC2CC1C2NC(C1CCCN1C(C1CCCCN1C)=O)=O CC1Oc2c(C(=O)NCC=CCNC(C3(C#N)CCOCC3)=O)cccc2C1C C1(N(C(CCCc2ccc(C)s2)=O)CCO)CCN(C(=O)COCCF)CC1 c1(C(N2CCC3C(C2)CN3C(c2ccc(Cl)nc2O)=O)=O)ccc2ocnc2n1 CCC(CO)CN=c1[nH]c(=NCC(C)(C)N2CCOCC2)[nH]c2c1COCC2 Cc1ccc2c(c1)CCC2NC(=O)NNc1ccccc1F C=CCC(C(=O)NCC(C1CCC1)NC(=O)CCSCC)C(C)C c1(OC)cc(OC(C23CCC(F)C2CC3)=O)ccc1F c1(CN(C(CC)Cc2ccccc2)C(c2cncc(F)c2)=O)ccc(SC)cc1 C(C(C)(C(=O)NC1CCN(C(=O)C(C)(C)C2CCC2)CC1)OC)OC C1(C(N2CC(C)(NC(C3C(C(C)C)OCCC3)=O)C2)=O)CN2CCC1CC2 C12(C(=O)NC(C3CCCCN3C(c3ccc4c(c3)CC4)=O)C)COC(CCO1)C2 C1(NC(c2cc(C3CC3)cnc2Cl)=O)CC2CCC(C1)N2Cc1cncc(Cl)c1 C1(NC(c2ccc(C(F)F)cc2)=O)CC(O)CN(C(c2[nH]cc3c2CCC3)=O)C1 C1(Nc2nccc(CC#N)n2)CN(C(c2cccc(Cl)n2)=O)C2(CCOC2)C1 c1(C(=O)NCCN(C(C2(S(N)(=O)=O)CC2)=O)CC)ccnc2ncc(C)cc12 c1(C(=O)NC(CC)CNC(C2(Br)CC2)=O)cc([N+](=O)[O-])ccc1N1CCOCC1 Cc1[nH]nc2ncc(C(=O)NC3CCC(C)N(C(=O)CCC4CCCC4)C3)cc12 c1(NCC(N2CC(NC(C3CN(C(C)=O)C3)=O)C2)=O)c(C)cc(C)cc1Cl.C(C)=O c1(C(=O)NCCC2(NC(C3CC3Cl)=O)CCOCC2)c[nH]cc(Cl)c1=O c1(CCC(=O)N(C2CN(C(c3cscc3F)=O)CC2F)C)ccc2c(c1)CCO2 C(C)(C(=O)NC1CC2CCC1N2C(c1csc([N+](=O)[O-])c1)=O)(C(C)C)OC C1(NC(c2cc(CCCC)oc2C)=O)CCCCN(C(c2cnn(C)c2F)=O)C1 C(CN=c1[nH]c(=NC2CCCS(=O)(=O)C2)[nH]c2c1SCC2)(c1ccoc1)N(C)C C1(OCCOCC)CCC(C)N(C(c2cn(CCC3CC3)nn2)=O)C1 N1(CC)CC(C(=O)NC2CCCC(N(C(=O)CCc3cnc[nH]3)C)C2)CCC1=O N1(C(C(C)(C)SC)=O)Cc2[nH]nc(C(=O)NCc3cc(C)co3)c2C1 Cc1csc2ncnc(N3CCC3(C)C(N3CCCCCC3c3ccccc3)=O)c12 Cc1ccn(CC(N2CCC(CCNC(=O)C(O)C3CC3)C2)=O)c1 CC(C)(CCC(=O)NCCc1ncccc1F)NC(C1CCCC2(CC2)C1)=O N1(C(Cc2c(C)nn(C)c2C)=O)CCN(C(c2ccns2)=O)C(C)C1C C1(CC)CCN(C(=O)C(Cc2ccoc2)NC(c2cc(OC)cs2)=O)CC1 C1(C(N2CCOCC(F)(F)C2)=O)CN(Cc2cc(Cl)c(F)c(Cl)c2)CCC1(F)F N1(C(C(CCC)O)=O)CCN(C(c2ccn(C)n2)=O)CC1C(C)C C=C=C(C)CC(=O)NC(CNC(C1(N(C)C(=O)OC(C)(C)C)CC(O)C1)=O)CO C1(C(=O)OCC)C=CCCN1C(c1cc(CC)on1)=O N1(C(c2cccc(C)c2N)=O)CCC2(C1)CN(C(C1(C)CC1(F)Cl)=O)CCO2 C(=O)(C(C)(F)C(=O)NC1CCN(C(C2CCN(C3CC3)CC2)=O)C12CC2)OCC CC(C(=O)NCc1cccnc1NC(=O)C(Cc1cnc[nH]1)N(C)C)S(C)(=O)=O C(C(C(=O)N(CC(C)N(C(=O)C1=CCC1)C)C)NC(C)=O)OC(C)(C)C C1(C(=O)OC)CN(Cc2c(C)cc(Cl)cc2C)CCC1(C)C c1(NC(C23CC(CN(C(C4CCC(OC)C4)=O)C2)C3)=O)c[nH]c2nccc-2c1 C(CCCCCNC(c1cccnn1)=O)N(C(C1C=C(C)CS1)=O)C C(C)(N=c1[nH]c(=N)[nH]c(=NC(C)CCC2CCCC2)[nH]1)c1cccc(SC)c1 C12(C(=O)NCC3N(C(c4n(C)ccn4)=O)CCCC3)CCOC1CC(=O)NC2 N1(CC(C)(C)C)CC(N=c2ccc(F)c(C(=O)OC(C)(C)C)[nH]2)C1 N1(C(CC2(OC)CCC2)=O)CC(CNC(=O)CC2(C)CC2)CC(C)C1 N1(C(CCc2ccc(C#C)cc2)=O)CCC2(CC1)CN(C(C1CCC(C)C1)=O)C2 N1(C(C(CCCC)C)=O)CC2CCN(C(=O)CNS(=O)(=O)CC)CC2C1 N1(C(C(CN(C)C)N(C)C)=O)CC2(C)CC1(C(=O)NCCC1COCCO1)C2 C=CC1(C(N2CC3C(CNC(c4cccc(C)c4Cl)=O)C3C2)=O)CCCCC1 n1(CC(=O)N(CC(CO)(CO)NC(C(F)=CC)=O)C)c(CC)nc2ccccc12 C(C(C(=O)NCc1cccnc1C)C(C)C)NC(C(C=C)(C)O)=O c1(CC(C(=O)NCC2C(NC(c3cn(CCOC)nc3)=O)CC2)C)ccc(F)cc1 CC(C(C)C)=CC(=O)NC(C)(C)CNC(=O)CCC1CC1(F)F c1(CC)nc(C)ccc1NC(C1CCCC1C(=O)Nc1nc(Cl)c(Cl)s1)=O c1(C(=O)NC(C(=O)N(C)CC2(O)CCC2)Cc2cn[nH]c2)ccc2c[nH]nc2c1 Cc1cnc(Nc2ccc(C)c(C(N3CC(N(C)C)C3)=O)c2)nc1C n1(CC(N2C(CCNC(COCC#C)=O)CSCC2)=O)ccc(=O)c([N+](=O)[O-])c1 N1(CC2(CN=c3n(C)ncc4cccnc43)CC2)CCS(=N)(=O)C2(CCC2)C1 Cc1ncc(Cl)c(C(N2CC3CC3(CNC(=O)C(C)CC(C)C)C2)=O)n1 Cc1sc(N)c(C(N2CC3C(NC(C4NC(=O)CC4C(F)(F)F)=O)C3C2)=O)c1C c1(C(C(=O)NCCC2(NC(=O)CCC3CC3(F)F)CC2)O)ccc([N+](=O)[O-])cc1 CC1(C)COC(=O)C1NC(=O)CCCn1cc(C2CCCCO2)nn1 c1(C(=O)NCCn2ccc(C(=O)NC(c3nc(C)sc3)C)c2)cncc(C#N)c1 c1(C(=O)NCC2(OC)CN(C(CCC)=O)C2)ccccc1CNS(C)(=O)=O C=C(C)CCC(C)NC(=O)CC1CCC(NC(=O)CCC2CCC2)C1 Cc1ccc(C)c(C(=O)NC2COCCN(C(=O)C(c3ccc(O)cc3)=O)C2)n1 N1(C(c2nc(NC(C)=O)sc2)=O)CC(NCc2c(F)cccc2Cl)CC(F)(F)C1 Cc1cccc(C(=O)NC2CC2NC(c2cn(C3CC3)nc2C)=O)c1C c1(N2CCCC(NC(C3C(C)OC(C)C3C)=O)C2C)cc(C#N)ccc1[N+](=O)[O-] N1(C(c2c(C)nc(CC)o2)=O)C2CC=C(C(=O)NC(C)COCC3CC3)C1CC2 N1(C(c2c(OC)nn(C)c2)=O)C(CC(=O)NCCNC(C)=O)C2CCCC12 Cc1cccc(CC(=O)NC2CCCC(NC(c3cc(C)oc3C)=O)C2)c1 c1(SC)ccc(CNC(=O)Cc2sccc2C)o1.N12CC(c3ccccc3)(C1)C2=O N1(C(COCC(=O)NC)=O)CC2CCC2(CCNC(c2cnc(C)cc2Cl)=O)C1 c1(C(C)C)noc(CC2CC(C(=O)N(c3ccncc3)C)C2)n1 CCCC(CNC(C1CC1[N+](=O)[O-])=O)C(=O)NCC(=O)NOCC Cc1ccnc(C(N2CC3CC3(CNC(=O)CN3CCCCC3)C2)=O)c1O C(=O)(C1=C(C)S(=O)(=O)CC1)NC1(COC)CCN(c2nc(CC)nc(=N)[nH]2)CC1 N1(C(c2ccc(CC(C)C)o2)C(=O)Nc2cccc(F)c2)CC2(C)CC1CCO2 N1(C(c2nc(CCC)sc2)=O)C2CCC1C(NC(c1nncn1CC)=O)C2 C#CCCCCC(=O)NCc1occc1C(=O)NC1CCOC(C)(CC)C1 Cc1c(C(N2CCN(C(c3ncn(C)n3)=O)CC2C)=O)ccc2c1CCC2 N1(C(C2CN(C(C)=O)C2)=O)CCCC(CNC(c2cccc(Cl)c2C)=O)CC1 c1(C(=O)NC(C)CCC(=O)N2CC(CC(N)=O)C2)ccc(Cl)c(O)c1 N1(C(CCC(C(C)C)NC(=O)CCC2CC2C)=O)CCCC12CCOCC2 c1(NC(=O)NC(c2ncc(Cl)s2)CC)ccsc1C(=O)NCCSC c1(CC)ccc(CN(CCNCc2cc(C)[nH]n2)C2CC2)o1 C1(C(=O)OC)CCCCC1C(=O)NC1CCC(NC(C2(CCO)CC2)=O)CC1 C1(CNC(C(CC)NC(N)=O)=O)CCN(C(=O)CC2CCC(=O)N2)C1(C)C C1(c2occ(C)n2)C=CCN(CC(=O)Nc2ccc(C(C)(C)C)cc2)C1 C1(C(N2CCC(C)N(C(C3CC4CCC3O4)=O)CC2)=O)CCc2ccccc2C1 C(=O)(N=c1[nH]c(Cl)ncc1O)C1CCCN(Cc2c(C)nc(Cl)cc2)CC1 N1(C(C(C(C)C)O)=O)CCC2(CCN(C(c3cncc4nc[nH]c34)=O)C2)C1 C1(COC)CNC(=O)CN1C(=O)C(C1(C)CC1)NC(=O)CNC(=O)C1CC1 c1(CCC(=O)NC2CCC(Nc3ncccn3)C2)c(Br)cncc1Br C1(OC)CN2CCCC2(C(N2CCOC(C(C)NC(C3CC3(C)C)=O)C2)=O)C1 C1(C(N2CC(NC(C=CC(C)(C)SC)=O)CC2(C)C)=O)CC(C)(C)OC(C)(C)C1 Cc1noc(N)c1C(=O)NCCCOCCNC(c1ccc(C(C)C)o1)=O c1(C(N2C(C(C)(C)NC(c3cnns3)=O)CCC2)=O)cc2cc(Cl)ccn2n1 C1(C(=O)NCCNC(C2CCC2)=O)CC(=O)N(C)C1.n1(CCCOC)cnnc1 N1(C(c2ccc(COC)cc2)=O)CC2CCC2(CNC(C2CC(C)=NO2)=O)C1 C1(CNC(C2CC3CCC2O3)=O)CN(C(c2ncc(C(F)(F)F)s2)=O)CCO1 C1(NC(CC2C(C)=NN(C)C2=O)=O)CCN(C(c2cn(C)[nH]c2=N)=O)CC(O)C1 CC(CNC(C1CN(C(N)=O)C1)=O)C(=O)NCC1CCC1 CC1CCN(C(C)C(=O)NCC(O)COC2CCOCC2)CC1 c1(C(=O)NCCCCC2CN(CC=Cc3ncc[nH]3)C2)ccc(-c2ccsc2)cc1 CC1(C)CCOC1CNC(C12CC(NC(c3cnn[nH]3)=O)(C1)C2)=O C(=O)(CC1=NN(C)C(=O)C1)N1C(CNC(CCNS(CC)(=O)=O)=O)CC(C)CC1 c1(C(N2CCC(N(C(=O)CN3CC4CC4C3)C)C2)=O)cccc2scnc12 c1(COC(c2n(C)nc(C3CCCOC3)c2)=O)cc(Br)ccc1F c1(C=O)cc(N2CCOCC2)ncn1.C1(C(=O)NCC(N(C)C)C2CC2)CCN1C c1(CC)nc(C(=O)NCC2(CCNC(=O)C(C)C)CC2)c(-c2ccccc2)s1 c1(N(CCc2onc(C(C)C)n2)C)nnc(-c2ccc(Cl)nc2)n1CC(C)CO N1(C(=O)CCN2CCOCC2=O)CC2CC(C1)CN(C(C1CCCS1(=O)=O)=O)C2 CC(C(=O)NCC(c1ccccc1)CNC(=O)CCC(=O)c1ccc[nH]1)C(F)F N1(C(CCSCC)=O)CC(NC(=O)Cn2cnc(C(N)=O)n2)C(C)(C)C1 C1(CN(C)C(c2cc[n+]([O-])cc2)=O)COCCN1C(=O)CCOc1ccccc1 N1(C(CNC(c2c(CC)c[nH]c2)=O)=O)CC(C)(C)CC1C(=O)N(C(C)CO)C N1(C(C(CC)C(C)O)=O)CCCC(C2CCN(C(C3CCC(F)CC3)=O)C2)C1 c1(C(=O)Nc2ccc(NC(c3ccc(F)cc3F)=O)cn2)c(Cl)cccc1Br N1(C(=O)Cc2sccc2Cl)CC(NC(C2(c3cnccn3)CC2)=O)C(O)C1 C1(OCC(=O)NC2CC(n3cc(C(C)(C)OC(=N)O)nn3)C2)CCS(=O)(=O)N1 c1(C(=O)NC2C(NC(CSCCOC)=O)C2)cc(NC(C)=O)c2occc2c1 CC1CCOC1C(=O)NC(C)(C)CCNC(=O)C(F)(F)c1nccs1 c1ccc(C)cc1CN(S(=O)(=O)c1cccs1)CC.C12CC1NC2C N1(C(C)=O)CCC2(CC1)CC(NC(=O)CCSC1CC1)CCO2 c1(C(N2CCC(N(C(=O)C(=C3CCCCC3)F)CC)C2)=O)cccc2nsnc12 C1(CC(=O)NC(C2CN(C(c3cc(C#N)on3)=O)CCO2)C)CCC(=O)NC1 c1(SC)nc2ncnc(NC(C3(C(=O)NC4CC(N(C)C)C4)CCCC3)=O)c2s1 Cn1nncc1CC(=O)NCC1COCC1NC(c1scnc1Cl)=O c1(CC(N2CCCC(CC(=O)Nc3cnccc3Br)C2)=O)ccc(O)c(O)c1 c1(C(=O)NC(C2CCN(C(=O)CS(=O)(=O)N(C)C)C2)C)csc2ncnc(O)c12 N1(C(C2C(COC)C2(C)C)=O)CC2=C(C1)CN(C(=O)CCc1cccc(O)n1)C2 C=CCC(F)(F)C(=O)NCCCN(C(C1CCCC1(F)F)=O)Cc1ccccc1 c1(CNC(N2CC(C)(OC)C2(C)C)=O)nnc2c(Br)cccn12 C(C(=O)N(C)CC=CC(=O)OC)(C(C)C)NC(C(CC)OC)=O c1(C(=O)NC(CNC(C2(C)CCCCCC2)=O)C2CCC2)ccc2cnoc2c1 c1(C(=O)NCCCOCCNC(C(C2CCCOC2)OC)=O)nc(O)c(C)s1 CCC(C)CCC(=O)NC1CN(c2nc(C(F)F)nc(=N)[nH]2)CC1(C)C c1(C2C(C(N3CCC(NC(C4CC(F)C4)=O)CC3)=O)C2)ccc2c(c1)OCO2 N1(C(C2CCCC(=O)C2)=O)CCC2CN(C(=O)C(F)(F)c3cccnc3)CC12 Cc1cnn(C)c1C(=O)NCC1C=CCN1C(C1CC2CCC2C1)=O c1(NC(=O)CCn2cc(-c3ccncc3)nn2)nc2c(s1)Cc1cc(Br)ccc1-2 C1(C(=O)NC2CCCCC2NC(=O)COCc2nccn2C)(OC)CS(=O)(=O)C1 C1(C(N2CCCC(C(=O)NC3CC(C)(C(N)=O)C3)C2)=O)CCOC(=O)CC1 C1(OC(C)(C)C)CCCN(C(=NCCC2CC2)NC(c2ccccc2Cl)C2CC2)C1 C1(C(=O)NC2(CCOC)CCN(C(C3C(F)(F)C34CC4)=O)C2)CN(C)CC(C)O1 c1(C(=O)NCC(=O)NCC(COC)NC(=O)C2CC2)scc2c1OCCO2 n1(CC(=O)N(CC(C)O)CCNC(C(CCC)C)=O)c(=O)cnc2ccccc12 C1(C(N(CCCCC)CC)=O)CCCCC1(C)NC(c1ccccc1F)=O Nc1cncc(C(=O)NCC(C2CCCCC2)NC(c2csnc2Br)=O)c1 c1(CC(N2C(CCNC(C=NOC)=O)COCC2)=O)cn2ccccc2n1 CC(C)C(O)C(C)C(=O)NCC1(F)CCCN(C(c2ccc(CO)nc2)=O)C1 CCCC(C(=O)N(CCCCNC(=O)Cc1ccnn1C1CCC1)C)OC c1(OC)ccnc(C(C)NC(=O)NC(c2cc(OC)ccn2)C(F)(F)F)n1 N1(C(COCC(=O)OC)=O)CC2CC(C(N3CC(O)(C(N)=O)C3)=O)C(C2)C1 N1(C(C(c2cccnc2)C)=O)CCCC(n2cc(CNC(C3(F)CC3)=O)nn2)C1 C1(CCOC)(NC(c2cnc(O)s2)=O)CCN(C(=O)Cc2cc(C)on2)C1 C1(NC(c2scc(CNC(C(C)OCOC)=O)c2)=O)CCCCCC1(C)C CN1CCC(C)(C(=O)NCC2(F)CN(C(=O)CN(C)C3CC3)C2)C1 c1(C(N(C2CCCN(C(=O)CN3CCCCC3C)C2)CC)=O)scc(C)c1C C(=O)(CC(C)C(F)(F)F)NCC1(C)CCN(C(CC(C(C)C)O)=O)CC1 CN1CCOc2cc(CNC(C3CCCC3OCc3cccnc3)=O)ccc21 Cc1nc(CO)sc1C(N1CCOC(CCNC(C2CCCC2O)=O)C1)=O C(=O)(CC(C(F)(F)F)NCc1nnnn1-c1ccccc1C)NCCCOC N1(C(CCC(CC)OC)=O)CC2CC1CCN2C(c1cnn(CC)c1C1CC1)=O c1(C(N2C(CC)C(NC(=O)C(C)OC(C)(C)C)CCC2)=O)cc2n(c1)CCCC2 c1(C(=O)NC2C=CCN(C(c3cc(OC)nn3C)=O)C2)ccc2c(n1)CCC2 C12(NC(c3ccncn3)=O)CCC1CN(C(c1ccc(SC(F)(F)F)o1)=O)C2 c1(C(=O)NC2(CC=C)CCN(C(c3ccc(C)[nH]3)=O)C2)cc2sccc2[nH]1 C(=O)(C(=O)NCC1(C(=O)NCCN(C(=O)CO)CCO)CC1)N(C)C CCCC(F)(F)C(=O)NC(C)C(C)(C)NC(c1ccccc1)=O.C12CC(C1)OC2 C1(NC(C2CCC2(F)F)=O)Cc2ccccc2C1NC(c1ncsc1Br)=O c1(C(N2CCC(NC(c3c(CC)cno3)=O)C2)=O)ccc(=O)n(CC(F)(F)F)c1 c1(CNc2ccc(-c3c(C#N)ccnc3)cn2)cc(Cl)ccc1[N+](=O)[O-] c1(C(N2C(C(=O)Nc3cnc(Br)nc3)CC(O)C2)=O)ccc(F)cc1[N+](=O)[O-] C1(C(=O)Nc2cnc(Cl)[nH]2)CC2CCC1N(C(c1cnon1)=O)C2 C1(CN2CCC(N3CCCCCC3)(C(F)(F)F)CC2)CCC2COCCC2C1 CC1(NC(=O)Cn2cnc(C#N)n2)CCCCC1C(=O)NCCC(=O)N1CCCC1 C(=O)(C1=NNC(=O)CC1)NCCN(C(C1Cc2cc(C)ccc2S1)=O)CC C1(C)CCC2(CCC2)C1CNC(=O)CNC(c1nnnn1C1CC1)=O.C(=O)(C1CC1)OC C1(CN(C)C(c2cc[nH]c2)=O)CCN(C(C2CCC(C(C)(C)C)CC2)=O)CC1 C(c1c(C)noc1C)=CC(=O)NC(CNC(CCc1nc(C)c(C)[nH]1)=O)CC(C)C C1(=CCNC(C(c2cccc(Cl)c2)C)=O)CCN(C(C2(F)CC=CC2)=O)CC1 Cc1c(C(=O)NCCC(O)CNC(c2cccc(CO)c2)=O)nn(C)c1Br Cc1cc(NC(c2cccc(NC(c3cn[nH]c3)=O)c2)=O)c(C)n1C(C)C C(=O)(C1CC(C)(C)Oc2ccccc21)N1CC2C(CNC(C3(C=C)CC3)=O)(C2)C1 N1(C(C(CC)n2ccnc2)=O)CC(CO)C2(C1)CN(C(c1cc(N)cs1)=O)C2 c1(C(CCC)O)nnc(N2CCOC(c3ccccc3)C2)n1CC(C)C N1(C(c2cn(CC)nn2)=O)CC2CCC1C(NC(=O)CNC(C)=O)C2 c1(C(=O)NCC2CC(NC(C3CCCC(C)(C)O3)=O)C2)cnc2nccn2c1 N1(C(C(C)n2ccnc2)=O)CCCC12CCCN(C(=O)CC1(C(F)(F)F)CC1)C2 c1(C(=O)NC(C(=O)NC(C#C)(C)C2CCCC2)C2CC2)cc(C(F)F)[nH]n1 N1(C(CC=CC)=O)CCC(C2CC2)C1CNC(=O)C(c1cccc(F)c1)(C)C C(N=c1[nH]c(CN2CCN(c3c(F)cccc3Cl)CC2)cs1)c1c(C)noc1C C=CC(CCC)CC(=O)NC(CCC)CC(=O)NC(CCOC)C(N)=O Cc1ccc2[nH]c(C(=O)NC3CC4CCC3N4C(c3ccn(C)n3)=O)cc2c1C CC1(C)CCC(C(=O)NC(CC2CC2)C2CC2)CN1C(c1c[nH]c(=S)cn1)=O N1(C(C(C)OC2CCCC2)=O)CC(NC(=O)CCOCCCN(C)C)C(O)C1 C1(C(=O)NCc2cn[nH]c2)CC2CC1CN(C(c1coc(CO)c1)=O)C2 N1(C(=O)OC(C)(C)C)C(C(=O)OC2CC(F)(F)C2(F)F)C2CC(F)C1C2 c1(C(=O)NC2CC(NC(C(C)OCCC#C)=O)C2)c(C)nc(C)n1O C1(NC(C2CN(C(C3CCC(C)O3)=O)C2)=O)CC(C)(C)C12CC2.CO C(C(C)(C(=O)N(CC(n1ccnn1)=O)CC1CC1)NC(c1ccncc1)=O)SC C1(O)(C(C)NC(c2cn(CC(F)F)cn2)=O)CCN(C(=O)CCc2cscn2)C1 C1(COCc2cncc(Br)n2)CN2CCC1CC2 C1(C(N(CCCNC(c2c(C(C)(C)C)con2)=O)CC2CC2)=O)CCS(=O)(=O)C1 c1(C(=O)NC2CC(NC(C(CC)(C)COC)=O)C2)cc2cc(C)cc(C)c2[nH]1 CP(C)(=O)c1ccc(C(N2CCCC(NC(=O)CCC3CCC3)CCC2)=O)nc1 C(=O)(N=c1[nH]nc(CC2CC2)s1)N1CC(C)N(c2ccccn2)CC1 C1(C(=O)NC2CCCC2C#N)(CC)CCN(C(C2CC(O)C(F)C2)=O)C1 CC(C)(C)CCC(=O)NCCOCCNC(C1CC1c1ccccc1Cl)=O c1(C(=O)NCC2(C)C(C)CN(C(C=NOC)=O)C2)cnc(S(C)(=O)=O)s1 c1(N2CCC(CNc3n(C)nc(C4CC4)c3)C2)ccc(Br)cc1C1OCCO1 c1(CNC(C(C)N(C(COCCOC)=O)C)=O)cc(C)no1 c1(C(=O)NC(C)CCc2ccnn2C)cc(O)c2ccsc2c1 CC1CC(NC(=O)CCc2cnccn2)CCN1C(c1ccc(F)nc1F)=O c1(C(C)NC(c2n(C(C)C)nnn2)c2cscc2F)ccnc(F)c1 c1(C(N2CC(NC(CCOCCOC)=O)C2)C)nnc(-c2ccccc2)o1 c1(OCC)ccc(C)nc1C(N1CC(C(C)NC(=O)Cc2ccc(Cl)nc2)C1)=O c12cccnc1NC(=O)c1cn(nn1)CC(C#C)NC(=NC)NC2.C(C)OC C1(O)(CNC(CNC(CCC)=O)=O)CCN(C(C2(c3ccno3)CCC2)=O)C1 Cc1c(F)cc(-c2cnc(C(F)(F)F)cc2C(=O)NCC2CCC(F)C2)cc1F N1(CC(=O)NC(c2n(CC)ncc2)C)CCN(C(=O)CCN2CCOC2=O)CC1 c1(C(=O)Nc2cn(-c3cn(C)nc3)nc2)c(NC(=O)CN)sc2c1CCCC2 C1(C)(CC)CC(NC(C2CN(C(c3ncccn3)=O)C(C)(C)C2)=O)CCO1 C1(C(=O)NC2CCC(OC)C2)CC2CCC1N2C(=O)CCc1cnc(C)o1 C1(C(=O)Nc2c(OC)ncnc2)CCN(C(c2ccc(F)cn2)=O)CC1O C1(OC)CN(C(C2CCC(=O)N2C)=O)CC1NC(c1conc1C)=O N1(C(C=Cc2n(CC)ncc2)=O)CC(CNC(=O)CC2CCC2C)C2(CC2)C1 C1(C(N(C(C)C)CCNC(=O)CC2CCOC2)=O)CCOC(C(C)C)C1 N1(C(=O)NC(C)C2CC2)CCC(C(=O)NCCCCN2CCC2)C(F)(F)C1 c1(OC)ccccc1C(C)C(=O)NCCCCNC(c1sccc1Cl)=O Cc1ccc2cc1C(=O)N(C)C2.C(=O)(C(F)OC(F)(F)F)NC1(C(C)(F)F)CC1 C1(C(=O)NC(CNC(C(C)NC(=O)OCC)=O)(C)CC)CCNC(=O)C1 N1(C(CCOC(C)C)=O)CC(C)(C)CC1CNC(C1CC1c1ccccn1)=O c1(C(N2CCCC(N(CCF)C(C3CC(O)C3)=O)C2)=O)cc2ccc(Cl)cc2[nH]1 c1(OC(C)C)ccc(C(=O)CNC(=O)C(c2ccc(F)cc2)N(C)C)cc1 C1(CNC(c2ccn(CC)n2)=O)CC(C(=O)N2CCCCC2C)=NO1 c1(CC(C(=O)NC(C2(C)CCCN2C)c2nc(C)[nH]n2)O)cc(Cl)cc(Cl)c1 N1(C(C=C(C)C)=O)CCC2CC12C(=O)NC(c1nc(=O)o[nH]1)C c1(C(=O)NCC(C(C)C)NC(C(CC)N(C)C)=O)ccc(C(=O)OC)cc1SC N1(C(c2cc(C#N)on2)=O)CCC2(CC1)CC2(CO)CNC(=O)C1=CCCOC1 C(C)(C(C(C)C)NC(C)=O)NC(=O)CCc1ccc(Oc2ccccc2)cc1 N1(C(=O)Cc2c[nH]ccc2=O)CCC2CN(C(=O)Cn3cnnc3)CCC2C1 C1(C(=O)NCCCCCN(C(C=C(COC)C)=O)C)CCCC(C(C)C)C1 N1(C(C2(C)CCCC2)=O)CC2CC(NC(c3cnn(CC(F)F)c3)=O)CC2C1 C1(NC(CCCOC(C)C)=O)CC(NC(=O)C(C)CC2CCCC2)CC1O c1(C(=O)NC(C)CNC(=O)Cc2ccoc2)cncn1-c1cnn(C)c1 C1(CNC(c2n(CCC)ccc2)=O)CN(C(=O)C=Cc2cnc[nH]2)CC1O C1(CNC(C)Cc2cc(Cl)cc(Br)c2)CCc2ccccc2O1 CCCCC(O)C(=O)N1CCOC(CCNC(=O)CC(C)(C)SC)C1 c1(NC(C2CC(NC(c3cccc(OC)n3)=O)C2)=O)csc2nccnc12 C(=O)(CC1=CCCCC1)N(CC(CC)NC(c1ncc(C)cn1)=O)CC Cc1cccc(C)c1NC(=O)CNC(CN1CCCS1(=O)=O)C(C)C c1(OC)nc(C(=O)NC(C)(CNC(C2CC2F)=O)C2CC2)sc1C C1(C(=O)OCC)(N(C(=O)C(C2C3CCCC23)c2ccccc2)C2CC2)CCOCC1 c1(C(=O)OC)cc(C(=O)NCCOCCSC)cn1C.C12CN(CCO1)C2=O C1(C(=O)NCC2CC(F)C2)(CC)CCCN1C(c1cc(C(C)C)on1)=O c1(C(N2CC3C(C2)N3C(c2ccc(I)cc2Cl)=O)=O)ccc(F)c(F)c1F N1(C(c2c(C)nc(C)s2)=O)Cc2ccccc2C1C(=O)N1CCN(C)C(=O)C1 C(=O)(C1Cc2ccccc21)N1CC(NC(c2c[nH]c(Br)c2)=O)C(O)C1 C(=O)(CC(C)(C)CSC)N1CC=CC(NC(C(C2CC2)SC)=O)C1 c1(C(=O)NC(C)CN(c2ncc(C#N)cc2Cl)C)ccc2c(n1)CCCN2 C1(C(=O)NCC2CCCO2)CC12CCN(C(c1cn(C3CC3C3CCC3)nn1)=O)CC2 Cc1cc(Cl)c(C(N2CC(NC(c3nc(O)sc3C)=O)CC(O)C2)=O)cn1 C1(NC(Cn2nc(C)c(Cl)c2)=O)COC2(C1)CN(C(c1ccc(O)nn1)=O)C2 c1(C(N2C(CN(C(=O)C(F)C(C)(C)O)CC)CCC2)=O)cnc2cc(C)nn2c1 n1(CCC(=O)NCC(N(C(C(C)NC(C)=O)=O)C)C2CC2)c(C)csc1=O Cc1ccnc2c(C(N3C4CCC3CN(C(C35CCC(C3)C5)=O)C4)=O)cccc12 C(=O)(C1=CC=CN2CCS(=O)(=O)N=C12)NCC(C)NC(c1cccc(=O)o1)=O c1(CC(C)C)nnc(C(=O)NC(C2CCN(C(=O)COCCN(C)C)C2)C)s1 C1(C(N2CC(C)C(C)(CNC(c3cnncc3O)=O)C2)=O)Cc2ccccc2O1 c1(C(N2C(C(C)NC(C3N(CCC)CCC3)=O)CCC2)=O)cccc(Cl)c1O c1(C(=O)NCCCNC(=O)Cc2ccc(Cl)cc2)ccc(O)cc1C(F)F O=C(C1=NOC2(CCC2)C1)NC1CCN(C(=O)CC23COCC(C2)C3)C12CC2 c1(OC)ccc(C(C)C(=O)OC)cc1OCn1nc(C)cc1CC(CC)CC(C)C N1(C(C(C)C2CCOC2)=O)CCCC(C2CN(C(C3(C4CC4)CCC3)=O)C2)C1 N1(C(C(C)OCC(C)C)=O)CCN(C(=O)CCCC(N)=O)CC2(CC2)C1 Cn1nc(C(=O)NC2(C3CN(C(C4CCCCN4C)=O)C3)CC2)c2c1CCCC2 CCC(C)(COC)C(=O)NCC1(F)CC(CNC(=O)CC23CCCC2C3)C1 CCC(c1ccc(Cl)cc1)=CC(N1CC(C(=O)O)CC(C(F)(F)F)C1)=O C1(C(N2CCC(C(N)=O)C2)=O)COCCN1C(c1nc[nH]n1)=O C1(C(N2CCC(C3(NC(C4CC4(F)F)=O)CC3)C2)=O)CCc2ccccc2CC1 C12(CCC)CCCN(C1)C(=O)CC(=O)C2=O.c1(C(CN)OC)cccnc1.O(C)CC C1(C(=O)NC2CCN(C(CNC(C)=O)=O)C2)COC2(CCC2)CO1 N1(C(CC(C=C)(C)O)=O)CC2(C1)CN(C(=O)C(c1cncc(F)c1)C)CCO2 C(C)(C(C)(C)NC(c1cc[nH]c1C1CCC1)=O)NC(C1(CC=C)CC1)=O C(=O)(C(C)(C)C1CCCN1C(=O)Cn1cc(CO)cn1)NCC=CC(C)(C)C CC1(C)C(C(=O)NCC2CCN2C(=O)CC2(N3CCCC3)COC2)C1(F)F C12(NC(c3c(C)cn(C)c3)=O)COC(C1)C(NC(c1cc(Cl)cs1)=O)C2 N1(CC(=O)NC2(C)CN(C(=O)C3=C(C#N)CCC3)C2)C(=O)NC2(CCCC2)C1=O c1(CC(=O)NC2C(NC(CC(CCC)(C)C)=O)CCC2)ccc(S(C)(=O)=O)cc1 c1(C(=O)NCC(C)(C(C)C)NC(CNC(C)=O)=O)c(C)[nH]c(C2CC2)nc1=S.C(=O)O CCCCCCC(C)C(=O)NC(COCC)C(=O)N(C)CCSC Nc1nc2c(cc1C(N1C3CC1CN(C(=O)C=Cc1ccoc1)C3)=O)CCC2 Cc1ccc(C(C)(C)CC(=O)OC(c2cc(O)ccn2)C)cc1 c1(C(N2CC(CNC(c3nc(Br)c[nH]3)=O)OCC2)=O)cn2ccnc2s1 C1(NC(C2(C)CCC(=O)NC2)=O)CC2CC(C1)N(c1cc(C(N)=O)ncn1)C2 C1(CNC(C=CC2N(C)CCC2)=O)CC2(CC2)CN1C(C1CC2(CCO1)CC2)=O N1(C(C(C(CC)O)C)=O)CCN(C(c2cnn3cccnc23)=O)C2CCCC12 N1(C(Cc2ccc(C)s2)=O)CCOC2CN(C(=O)C(O)CCC(C)C)CC12 CCC(C)C(O)C(=O)N1CCC(CNC(=O)C(CCO)N(C)C)C12CC2 C12(C(=O)NC3CCC(NC(=O)CC4CC5CC5C4)C3)C(=O)C3CCC1C2C3 Cc1cn2c(n1)CCC(OC(c1cccc(OCc3ccccn3)c1)=O)C2 N1(C(c2cc(NC)n[nH]2)=O)CCC(CNC(c2cccc(COC)n2)=O)CC1C c1(-c2nn(CC3(C)CCC3)c(C3CC34CCOC4)n2)ccc(F)c(Cl)c1 CC#CC1CCN(C(C2(C3CCCN3C(c3cccn(C)c3=O)=O)CC2)=O)C1 Cc1c2ncnc1N1CCC(C1)N2.C(CC(C)C)N(C1CCCC1)C1CC1 N1(C(c2csc(C)c2C)=O)CC(C)(C(N2CC(S(C)=O)C2)=O)CC1(C)C c1(OC)ccc2nc(N3CC(NC(c4scnc4Cl)=O)C(C)(C)C3)sc2n1 c1(C2(C(=O)NCCCNC(C(C)(C)C3CC3)=O)CC2)cccc(C(F)(F)F)c1 c1(CC(=O)NC(CN(C(CCc2cc(C)on2)=O)C)C)cccc([N+](=O)[O-])c1 N1(C(c2ccc(CCC)[nH]2)=O)CCOC2(CCN(C(=O)CS(=O)(=O)C3CC3)C2)C1 C1(F)(CNC(C2CC2(Cl)Cl)=O)CN(C(=O)C(CN2CCCC2)c2ccccc2)C1 n1(CC(C)O)cc(C(=O)NCCCCCNC(c2ccc[n+]([O-])c2)=O)ccc1=O S(=O)(=O)(CCC(=O)N1CCC(NC(C2CCC(C3CC3)C2)=O)C1)N(C)C C1(CNC(c2cc(C)[nH]n2)=O)CC(NC(c2cnc(S)nc2)=O)C1(C)C N#Cc1ccc2c(c1)CCC(NC(c1cc(C3CC3)no1)c1nnnn1CC)O2 CCCC(=O)N(CCCOCCNC(=O)C(C)NC(C)=O)C Cc1cnc(N(C(CN(C)C)C(C)C)C)c(S(=O)(=O)N2CC(C)(C)CC2CO)c1 C1(NC(C(CN(C)C)O)=O)COC2(C1)CN(C(c1csc(=N)[nH]1)=O)C2 C(CC(C(C)(C)C)NC(c1cn(C)c(=O)n1C)=O)N(C)C(C1CC1C(F)(F)F)=O CCCCCCCCNC(C1CCCCN1C(=O)N(C)CCc1cn[nH]c1)=O N1(C(C2CCCN(CC(C)C)C2)=O)CC2CC(C1)N(C(=O)CCSC(F)(F)F)C2 CN=c1nc(C(N2CCC(NC(=O)CC3CCC(=O)NC3)C(F)C2)=O)cc(C)[nH]1 N1(C(C(COCC)C)=O)CCc2sccc2C1CNC(c1ccc(Cl)c(N)c1)=O CC(C)CCCCC(=O)N1CCCC(CNC(=O)CC2CCN(C(C)C)CC2)C1 N1(C(=O)CCc2ncco2)CCC(CNC(CCN(C)CC)=O)CC1 CCC(C)(C)C(C)CC(=O)NC(C)C(CO)NC(c1cc(=O)c(OC)c[nH]1)=O N1(CC(COC)C)C(=O)C(CC(=O)NC2(CCF)CCC2)SC1=Nc1ccccc1 Cc1ccncc1CNC(C1CCCCN1C(c1cc(C2CC2)no1)=O)=O Cc1cccc2c(=O)c(C(=O)NC3CCN(C(=O)C(N)=O)CC3F)c[nH]c12 C1(CNc2cc(OC)ncn2)CCCCN(C(=O)CSc2cccc[n+]2[O-])C1 c1(C(N2CC(N(C(C3N(C(C)=O)CCOC3)=O)C)C2)=O)c(N)cc(Cl)cc1Cl N(C1c2ccccc2OCC1O)C(C(=O)Nc1ccc(CCC)cc1C#N)=O c1(C(=O)NCc2ccc(CCNC(C(CCC)C)=O)cc2)scc2c1OCCO2 c1(CC)cc(C(=O)NC2CCCCC2NC(c2ccc(N)c(N)n2)=O)cc(Cl)c1 N1(C(C2C(C)(C)C2(C)C)=O)CC(NC(=O)CCCOC2CCOCC2)CC(O)C1 C1(C(=O)NC(C)C(F)(F)F)(COC)C=CCN1C(c1sccc1Cl)=O C(=O)(CCC(=O)NCCCCNC(C1CCCN(C(=O)C(C)C)C1)=O)NC N1(C(C(C)(F)F)=O)CCOC(CNCC2CC(=O)N(Cc3ccccc3)C2)C1 C1(C(N2C(C)CN(C(=O)C(F)(F)C3CC3)CCC2)=O)COc2cc(F)ccc2C1 N(C(=NCc1csc(C(F)(F)F)n1)NC(C)C1CC1)CC(C)(CO)OC c1(C(=O)NCC(CC(=O)NC(c2cccnc2)CC)O)ccc(O)nc1C c1(C(=O)NCC2C(CNC(CCc3cccc(C)c3)=O)C2)cc(Cl)ncc1F C(CC1=CCCCC1)N(C)C(c1ccn(CCNC(=O)Cn2cnc(C#N)n2)c1)=O c1(C(N(C2CCCN(C(c3ccc(CO)cn3)=O)C2)C)=O)cncc(C(N)=O)c1 C1(OC)CC2(CCC(C(=O)NC(C3CCCN3C(=O)C(C)SC)(C)C)CC2)C1 N1(C(CSCC=C)=O)CCC(C)C1CN(C(=O)CCCOc1cccc(Cl)c1)CC C1(NC(C(CC=CC)C)=O)CC=C(C(=O)N(C2CC2)Cc2cnn(C)c2)C1 C=CCCC(C)(C)C(=O)N1CCCC(N(CCF)C(c2ccc(CC)cc2)=O)C1 c1(C(N2CCCC(CNC(CCOCC)=O)(COC)C2)=O)ccc(C)c(F)c1F Cc1sc2ccccc2c1C(=O)NCC(C)CN(C)C(C1(F)CCCCCC1)=O c1(N(C)C)cnc(C(=O)NCCC2CCCN(C(c3nocc3Cl)=O)C2)nc1 N1(C(C2(F)CCCC2)=O)CC2CCC1C1CN(c3nc(-c4ccoc4)ns3)CC21 N1(C(C(CCCOC)C)=O)CCCCC(CNC(c2ncoc2C)=O)CC1 n1(CC)cc(CN(C(C(=O)NCc2cc(C)on2)C2CCOC2)C)c(C)n1 C1(CC(C)C)CC(CCNC(=O)N(CC(C)(C)CO)C(C)C)CCO1 Cc1cc(N(C(c2cccnc2)C(C)C)C)nc(N(C)CC2CCCCO2)n1 Cc1nccn1CCC(=O)NCCOC(C)(C)CNC(=O)Cn1cnnn1 c1(C(N2CC(C)(CNC(C3CNC(=O)N3)=O)OCC2)=O)cc(F)c(F)c(Cl)c1F Cc1nc(CN2CCC(O)C2C(=O)NCC(C)O)c(C)s1 C(=O)(CCCC(F)F)NCC(CC)NC(=O)C(C1CC1)N(C)C C1(C)(CNC(N2CCC(C)C(N3CCOCC3)C2)=O)CCS(=O)(=O)N1C C1(CNC(C(=Cc2ccco2)C)=O)CCCCC1NC(C1CC(=O)N1)=O C1(CC(=O)NCC(CC)N(C(=O)CC2CCC(=O)NC2)C)NC(=O)NC1=O C(=O)(C(CNCC1(c2ccccc2)CC2(CC2)C1)C(C)C)N(CCCCCC)CC N1(C(C2(CC)C=CCC2)=O)CCCN(C(=O)C(C2CCCCC2)OC)CC1 N1(C(C2CCCC(OC)C2)=O)C2CCC1C1CC1(NC(=O)C=CC1CC1)C2 C1(NC(c2ccn(C(C)C)n2)=O)CC=CCC1C(=O)NCC1(O)CCCOC1 C(F)(C(F)(F)F)(C(F)(F)F)c1c(C(N2CCCC(c3cn(C)nc3)C2)=O)scc1 CC(CC(=O)NCC12CCC(NC(=O)C(F)=C3CCCC3)(CC1)CO2)C(C)(C)C N1(c2cc(N(C)CCc3ccc(F)cc3F)nc(C)n2)CC(C)S(=O)CC(C)C1 c1(C(C)=O)ccc(C(=O)NC2CCCC2NC(=O)C(C)C(C)C)cc1F C12(CNC(C(C3CCCO3)NC(C(CCC)F)=O)=O)CCN(CC1)CC2 c1(C(=O)NC(CC)CNC(=O)Cc2cc(C)ccc2C)n[nH]c2ccc(F)cc12 C(=O)(C1=Cc2ccccc2C1)NC(C1CCN(C(c2c(CC)nc(C)o2)=O)C1)(C)C c1(NC)ccccc1C(=O)NC(C)C(C)NC(C1C2CCCCC12)=O N1(C(C2(COCC)CC2)=O)CC2(C1)CN(C(C1CCCC(C)(C)O1)=O)CC2CO c1(C(=O)NC2CC(OC)CN(C(=O)C(F)C(C)C)C2)c(C)cc(C)oc1=O CCC(O)CCN=c1nc(N2CCOC(C)(C(=O)N(C)C)C2)cc[nH]1 N1(C(CSCC=C)=O)CC(O)CC1CC.C12CC(O)C1CC(=O)N2 C1(NC(c2onc(C)n2)=O)CN(C(C2CC(C#N)C2)=O)CC1C C1(CC)(NC(=O)CC2COCCO2)CCN(C(=O)C(C)(C(C)C)OC)CC1 NS(=O)(=O)CCC(=O)NCC1(CNC(C2CCCCC2F)=O)CC12CCC2 C12(COC)CC(NC(=O)CC(=O)N(C)C)(CN1C(c1cnc(O)c(OC)c1)=O)C2 C12=CCNC(=O)C(=O)N(CC1)CC2.C1(CCC)(C(=O)NCC(F)F)CC1 C1(CNC(C(C(C)C)(C)O)=O)CCC2(CN(C(=O)CCn3cnnn3)C2)O1 c1(C(=O)NCC2(OC)CN(C(=O)C=C(Cl)Cl)C2)cnc2nccn2c1 CC(C)C(C(=O)N1CC(CCNC(C2CCO2)=O)C1)N1CCCCC1 C1(NC(c2cc(C(F)(F)F)n[nH]2)=O)CCN(C(C2CCC=CCC2)=O)CC1O N1(C(CC)=O)CCCCC1C(=O)NCC(C)NC(C1(Br)C(C)C1C)=O c1(C(N2CCC(C(C)(C)NC(=O)C3=C(Cl)CC3)C2)=O)cc2c(cc1Cl)OCO2 C1(NC(C2(OCC)CCC2)=O)CC2CC(NC(c3ccoc3C(C)C)=O)C1C2 Cc1cc(C)c(C=CC(=O)NCC2CC2NC(=O)CC(C)(C)CC(F)F)c(C)c1 C(C1=CCN(C(c2ccn(C)c2C2CCC2)=O)CC1)NC(CCSCCCC)=O C1(OC(C(c2cccc(O)n2)C)=O)CCN(c2ccc(Cl)cc2)C1=O c1(C(N2CC(F)(C(=O)NC3(CC)CCCC3)C2)=O)sc(C)nc1CC(C)C C1(C(=O)NCCCCC2CN(C(C3(C(=O)OCC)CCC3)=O)C2)CNC(=O)N1 CC1(C)CC(NC(c2ccc(C(C)(C)C)nc2)=O)CN(c2cnc(C#N)cn2)C1 CC(N=c1[nH]c2cc(Cl)c(S(=O)(=O)NCCF)cc2s1)c1ccccn1 C1(NC(=O)Cc2cscc2F)CCCC(CNC(C2OCCO2)=O)C1 CC1(C)CCC(CNC(c2sc(F)cc2Cl)=O)N(C(=O)COCC2CCC2)C1 Cc1cc(C)n(CCC(=O)NC2CCC(C(=O)NC3CCC(F)(F)C3)C2)n1 C1(SC)CCCC1NC(C1CCC(n2cc(CCCOCCO)nn2)C1)=O c1(C(=O)OC)ccc(CNC(CN(C(=O)CN2CCCCC2)C)CC)c(OC)c1 Cn1cnc(N2CCC(OCCCNC(c3nc(Cl)ccc3F)=O)CC2)cc1=O C(=O)(CS(=O)(=O)C1CC1)N(CCn1cc(Cc2ccc(Br)nc2)nn1)CC N1(C(C(C)CCO)=O)CCC(C(=O)NCC(c2nn[nH]n2)C)C1.C(C=O)=CC CC(C)C(CNC(C1Cc2nnc(C)n2C1)=O)N=c1cc(Cl)nc(S(C)(=O)=O)[nH]1 C(c1scnc1C)=CC(=O)NC1C(NC(C(C)(c2cccs2)N(C)C)=O)COC1 N1(C(C(C)=CC2CC2)=O)CCC(C)N(Cc2nnnn2C)CC1 N1(C(CC2C(C(N(CC(=O)OC)CC#C)=O)CCC2)=O)CCCC(O)C1 C1(C(=O)NCC(C)OCC=C)(CNC(c2nnsc2N)=O)CCCCC1 c1(OCC(=O)NCC(CO)NC(c2cnn(C3CCC3)c2)=O)ccccn1 c1(C(N2CCC(NC(Cc3cnc(C)[nH]3)=O)C2)=O)cnncc1C N1(C(C2(NC(CC(C)OC)=O)CCN(C)C2)=O)CCn2nc(C)cc2C1 Cc1nc(C(N2CC(NC(C3CC34CCSCC4)=O)C(O)C2)=O)c(C)n1C1CC1 N1(C(C=C(C)C)=O)CCC2(CC1)CC(NC(c1cc(Cl)n(C)n1)=O)CO2 c1(NC(C2C3CN(Cc4cn(CC(C)C)nc4)C2C3)=O)cc(O)cc(O)c1 c1(C(N2C3CC(CNC(CS(CC)(=O)=O)=O)C2CC3)=O)c(O)nnc2c1CCC2 CCC(CC(C)C)C(=O)N1CCC(NC(=O)C=C(Cl)Cl)C(CO)CC1 c1(CN(S(=O)(=O)CC)CCNC(C(CNCC)OC)=O)ccc(CO)cc1 C1(NC(C(Cn2ccnn2)NC(C2C=CCS2)=O)=O)CC2CCCC(C1)C2 CC1CCN(C(c2cc[nH]c(=N)c2)=O)CC1CNC(c1nscc1Br)=O c1(CC)cc(C)c(C(=O)NC2(C(=O)NC3CCNC(=O)C3)CCOCC2)o1 c1(C(=O)NCC2(F)CN(C(c3c(C)con3)=O)C2)sc(C)c(C)c1C Cc1nc2ccccn2c1C(N1CCN(C(c2ncn3c2CCCC3)=O)CC1)=O C1(CC(N2CCOC(CNC(C3(C4CCCO4)CC3)=O)C2)=O)NC(=O)NC1=O C#CC1(NC(C2CCCN2C(=O)C(C)CCC)=O)CCCCCC1 C=CCCCCCCCOC(C1CCCCC1N)=O S(=O)(=O)(c1ccc([N+](=O)[O-])cc1C(=O)O)N1CC2CCN(C(C(C)(C)F)=O)C2C1 C1(C(=O)NC)CC(C2CC2)=NO1.N12CC(C(C)C1)C(N(C)C)c1n(nnn1)C(C)C2=O C(CCC(N)=O)(C(=O)N1CCCC1)n1cc(CC(C=C)O)nn1 CC(C)C(CNC(=O)CN(C1CCCC1)C)C(=O)N(C1CCN(C)C1)C N1(C(CNS(NC)(=O)=O)=O)CC=CC(NC(c2c[nH]nc2OC(C)C)=O)C1 C(C(O)CC(=O)N1CCC(OCCN(C)C)C1)NC(C=C(C)C(F)F)=O C(=O)(CS(=O)(=O)CC)NCCCN(C(CC(CC)C)=O)C1CC1 Cc1ccc(CCN2CCCN(c3ncc4c(n3)CCOC4)CC2)cc1[N+](=O)[O-] N1(C(c2c(CC)nns2)=O)CC(CCNC(C2(c3cc(C)on3)CC2)=O)OC(C)C1 c1(C(=O)NCC2C(NC(Cc3ccc(C)nc3Cl)=O)CC2)csc2cc(C)sc12 n1(CCN=C(NC(C)CN(C)C)NCC2CC2)cc([N+](=O)[O-])c(O)nc1=O C(=O)(C(C)(C)C(C)(F)F)N(CC(C)CNC(=O)C(F)CC1CC1)C c1(NCC(=O)NCCCCC(C)NC(=O)CC2CC2)ccccc1[N+](=O)[O-] c1(CNC(C2CN(S(C)(=O)=O)C2)=O)c(F)cncc1F c1(C(N(CCCNC(c2cncs2)=O)C(C)C)=O)nccn1C N1(C(c2c(C)ccnc2)=O)CCCC2CCN(C(c3cn4ccnc4s3)=O)CC12 N1(C(CC)=O)CCN(C(C2(c3ccccc3)CCCC2)=O)CC1CC(F)F c1(C(=O)OCC2CC(=O)C23CCCCC3)cc(S(=O)(=O)CC)ccc1F N1(C(C(CNC(c2c(CC)nccc2)=O)O)=O)CCC2CCCC12 C(=O)(CC1CN(C)c2ccccc21)N(CCN(C(C(CC)SC)=O)C)C N1(C(CC(C)NC(=O)C(C2CCCCC2)F)=O)CCn2cnnc2C1C N1(C(CC=CC)=O)CC2CCC1C1CN(C(c3c(C)noc3C(F)(F)F)=O)CC21 C1(NC(c2nnc(O)nc2O)=O)CN(C(=O)CCCn2cccc2)CCC1CO C1(NC(c2cccnc2C)c2n(CCCSCC)nnn2)CCCN2CCCC12 Cc1ccc(C(=O)NC2CCC(CNC(C3CCC(N(C)C)C3)=O)C2)o1 C1(C(N(CCOCCN(C(C(CCC)(C)OC)=O)C)C)=O)CN2CCC1CC2 S(=O)(=O)(c1cccc(Br)c1)NC(C)C(N1C2CCC1CC2)=O N1(CC)CC(C(N2CCC(O)(CNC(c3cnn(C)c3Br)=O)C2)=O)CC1=O CC1(C)C(NC(=O)Cn2cc(C3CC3)cn2)CC1CNC(=O)Cc1sc(O)nc1O C12(NC(c3cc(Cl)cs3)=O)CCC(CN(C(C3CCCS(=O)(=O)N3)=O)C1)C2 N1(C(C2N(C(C3C(COC)CC3)=O)CC2)=O)CC=CC1C(N)=O N1(C(c2ccn(C)c2)=O)CC(O)CCC1C(=O)NCc1cnn(C)c1O N1(C(CNC(CN(C)C)=O)=O)CCCC(NC(c2coc(C(F)F)c2)=O)C1 O=C(N=c1[nH][nH]c2c1CCCC2)c1n[nH]c2c1CCN(C(C1CC1(F)F)=O)C2 CCC(CC)(CCC(=O)OC)NC(=O)Cc1c(C)cc(Cl)cc1C C(CN=c1nc(CC2CC2)[nH]s1)=CCNC(=O)CC1CC2(CCC2)C1 N1(C(CCC#C)=O)CC(C2CCCN(C(C3CCCCN3N=O)=O)C2)C1 Cc1occc1CC(=O)NCC12CC(NC(c3ccn(C4CCC4)n3)=O)(C1)C2 CN1CCCC1C=CC(=O)NCC1CCN1C(c1ccc(C#N)s1)=O N1(CC)CCN(CCCC(N2CCC(NC(=O)CC(C)F)C2C)=O)CC1 Cc1csc(CC(=O)NCC(C2CCCC2)NC(=O)Cc2csc(C)n2)c1 C1(CC(N2CC(OC(C3(CCCC)CC3)=O)(CNC(C)=O)C2)=O)COCCN1CC N1(C(CCCOCC=C)=O)CCC(CO)C(NC(=O)CN2CC3CC3C2)C1 C1(C(=O)NCC(CN(C)C(c2ccc(CC#N)cc2)=O)(C)C)CCCCC1CO C(=O)(CCCC(C)(C)NC(c1ccccc1OC)=O)NCC#C c1(OC)cc(C(=O)NC(CNC(C2(O)CCOCC2)=O)CC(F)(F)F)cc(F)n1 N1(C(c2ccc(=N)[nH]c2Cl)=O)CCC2(CC1)CC2NC(c1ccoc1C1CC1)=O c1(SCC)cccc(C(N2CC(C(N)=O)(CNC(C3CCC(C)(C)O3)=O)C2)=O)c1 C1(C(=O)NCC(c2cccs2)C)CCN(C(C2CC2C(C)(F)F)=O)CCO1 C(=O)(C(CC)(CC)CCO)N1CCC(O)(CNC(Cn2ncc(C#C)c2)=O)CC1 N1(C(c2ccc(COC)[nH]2)=O)CCOCC1CCNC(=O)CN1CCSCC1 c1(C(=O)NCCCNC(c2c(C)nc[nH]2)=O)c(C)nsc1C Cc1ccc(NC(=O)C(=O)NC2CN(C(=O)C(N)CN)CC2O)cc1C CCC(C(=O)N1CCC(C)N(C(=O)CN2CSCCSC2)CC1)C(C)(C)CC c1(CC)nc2ncnc(N3CCCC3C(=O)Nc3cc(C)n(C(F)F)n3)c2s1 C(C(C)(C(=O)NC(C12CCC(CO1)C2)C)NC(=O)C(C)N(C)C)SC Cc1nncc(C(=O)NC2(CO)CN(C(C3CCC4(CCC4)O3)=O)C2)c1C CCCCC(O)C(C)C(=O)N1CCC(CCNC(c2cnc(OC)nc2)=O)CC1 CC1C(NC(=O)COC2CCOCC2)CC2CCC1N2C(C1CCN1C)=O CC1(C)CN(C(=O)C=Cc2ccoc2)CCC1C(=O)NCCn1cnnc1 N1(N(CCC(=O)OC)CC=C)CC2(CC(CO)CO2)C1.C1(C=O)CC2(C1)OCCO2 n1(C(=O)NCC2CCN2C(c2ocnc2C2CCC2)=O)cnoc1=O C1(C(=O)NCC(CCCC)O)CC(C)CCN1C(=O)CC(C)CN(C)C C1(OCC)CCN(C(c2cnn(CCO)n2)C(=O)NCCC#N)CC1 c1(-n2cc(C(=O)NC3(C4CCCO4)CCC3)nn2)ccc(Cl)cc1Cl C(=O)(CC(C)(C)N(C)C(C1(C)CCOC1)C)NC1CC(COC)C1 c1(C(=O)N(CC2(CNC(c3csc(C(F)F)n3)=O)CCC2)C2CC2)cccc(=O)o1 c1(C(=O)NCC(CN(C(c2c(CCC)n[nH]c2)=O)C)O)cccc([N+](=O)[O-])c1Cl C(=O)(C(C(C)NC(c1coc(CO)c1)=O)C(C)C)NC(CC(=O)OCC)C N1(C(C2(C)C(C)(C)C2)=O)CCN(c2ccc(CNC(=O)C(F)OC(F)(F)F)cn2)CC1 c12ccc3c(n[nH]c3c1)-c1cccc(c1)OC(=O)C(CC)NC2=O.C(CF)OC c1(C(N(C2CCN(c3nc(O)c(C)s3)C2)CCC)=O)cc(O)nc(C)n1 C=CCCCC(C1CC1)NC(=O)C(C1CCN(C(C2CCC(=O)NC2)=O)CC1)C C(N=c1nc2sccc2c(N2CC(=O)NC(C)C2)[nH]1)C1(C(C)C)CCCC1 c1(C(=O)NCC(CO)NC(C2CN(C3CC3)C2)=O)cc(F)c(O)c(F)c1 C=CC1(CC(=O)NCC2CCN(C(C3C4CCC(=O)C34)=O)C23CC3)CCCCC1 N12CC3CC1CN3CC2=O.C(CCC(F)F)NC(=O)CSc1ccccn1 N1(C(c2ccc(C)cc2)=O)C2CCC1CC(NC(c1c(C)noc1C)=O)C2 C1(C(N2C(C(=O)NCc3occ(C)c3)CC(C)C2)=O)CN(C)CC(C)O1 c1(NC(C#CCNC(c2ccc(OC)nn2)=O)=O)cccc(C#N)c1C C1(C(C)(F)F)(C(=O)NCC2C(NC(C=C(CCC)C)=O)CCC2)CCOCC1 c1(CC(=O)NCCCN(C(=O)C(c2ccc(C)cc2)=O)CC)cc[nH]c(=N)c1 N1(C(C2CC23CC3(F)F)=O)CC(O)(C2CC2)C1 Cc1c(C(=O)NC2(C)CN(C(=O)C(C(C)C)NC=O)C2)ccc(F)c1F C1(NC(c2cc(C(C)(F)F)n[nH]2)=O)C=CCN(C(=O)Cc2cn[nH]c2)C1 O(N1CCC(CC(=O)NCCCNC(c2noc(C)c2C)=O)CC1)CC c1(OC)ccc(F)c(N)c1C(=O)NCC(CNC(=O)C=Cc1nc(C)co1)OC CC1CN(C(C2CCC(O)CC2)=O)CCCN1C(=O)CCc1cncn1C c1(C(=O)NCCC(C)N(C)C(c2ccc(C(F)F)nc2)=O)cnc(N)c(O)c1 C(=O)(C(CC(F)F)SC)NCC(CCCC)NC(c1nn[nH]c1C(=O)OC)=O c1(C(=O)OC)csc2cc(C(N3CC(NC(C4CCC4(F)F)=O)C(C)C3)=O)[nH]c12 c1(C(=O)NCCCOCCNC(C2CC2Cl)=O)ccc(CO)cn1 CC1CCC(=CC(N2CC(NC(c3cnn(CC(F)F)c3)=O)C2)=O)C1 C1(CSC2(C(=O)Nc3ncc(OC)c(C(F)(F)F)c3)CC2)COc2ccccc2O1 C(C)(C(=O)N(CC1CCC1C(=O)NC(CC)CC)CC1CC1)OCC CCCC(CCC)CC(=O)N1C(C(=O)NC(CC2CC2)C(=O)OC)CC2CCCC12 C12CC(CO)N(C1)C(=O)C2N(C)C.C1(C(C)(C)N)CCCCO1.C(=O)(C(C)OC)OC CC1CC(NC(c2c[nH]ccc2=N)=O)CN1C(c1cc(C2CC2)oc1C1CC1)=O CC1CCC(C(=O)NCCc2csnn2)CN1C(=O)COCC(F)F C(CC(C)(C)C(=O)NCC1CC1CNC(c1nocc1Cl)=O)OC C1(C(F)(F)F)(CNC(C2(NC(C3(C)CC3C(F)(F)F)=O)CC2)=O)CNC(=O)C1 Cc1oc(S(C)(=O)=O)cc1C(=O)NCC(C)(O)CNC(=O)CC1CC1 C1(CC(N2C(C(C)NC(=O)COc3cccc(F)n3)CCC2)=O)CCOCC1(C)C c1(CC)nc(Cl)ccc1C(=O)N(C)CC1CCCN1C(=O)C(=Cc1cnc[nH]1)C C1(CC)C(C)CCN1C(c1ccc(C2(C#N)CCC2)cc1)=O c1(C(=O)NCCC2CC(NC(C3(CC)CCC3)=O)C2)oc(CO)cc1C C(CNC(=O)CC1CCSC1)(CC(=O)N1CC(C)(C(=O)OC)C1)OC c1(C(=O)NC(C2(O)CCN(C(C(C)NC(=O)NC)=O)C2)C)ccn2ccnc2c1 C(=O)(C(CC(F)F)NC(=O)CN1CSCC1=O)NCC(C)CCO Cc1nc(N2CCSCC2)sc1C(c1ccc(CC(C)C)cc1)=O Cc1c(CC(N2CCCC(CNC(c3cc(Cl)no3)=O)C2)=O)sc2ccccc12 CCC(C)C(O)CC(=O)NCc1n[nH]cc1C(=O)NC1CCS(=O)CC1 N1(C(c2nc(COC)oc2)=O)CCN(C(C2CC3CC3CC2C)=O)C2(CC2)C1 S(=O)(=O)(c1cccc(=NCCOc2ccccc2)[nH]1)N(C1CCCOC1)C c1(CC(C)C)cc(=NC(=O)C(=O)NCC2CCCC(C(F)(F)F)C2)cc[nH]1 N1(C(C2N(CC)C(=O)CCC2)=O)CCC2CN(C(C34CC(CN3C3CC3)C4)=O)C2C1 C=CC(CC)C(=O)NCC1(CNC(c2cnn(CCO)c2)=O)CC12CCC2 C1(NC(C2(N3CCN(C)CC3)CC2)=O)CN(C(=O)CC2CCC2)CC2(CC2)C1 N1(C(c2ccc(N)cn2)=O)CCCCCC1CNC(C1(F)CCCCCC1)=O CC1(O)CCC(C(N2CC(C)(C(N3CCCCC(CO)C3)=O)C2)=O)CC1 C(=O)(CC(C(F)(F)F)OC)N1C(CNC(c2ncc(CC)cn2)=O)CN(C)CC1 N1(C(CCC(C)SC)=O)CCCCCC1C(=O)NCCC1CCC(=O)N1 C1(C(=O)NCCCNC(c2c(C(F)(F)F)oc(C)c2C)=O)CCc2ncnn2C1 CC(C)CCCC(=O)NCCCOC1CCN(C(C2CCCCCN2C)=O)CC1 S(=O)(=O)(C1CC2(CC2)C1)C(CN1CCCC(n2cc(-c3c(C)con3)nn2)C1)=O N1(C(C)=O)CCN(C(=O)Cc2ccc(F)cc2C)C(C)C1C CCC(CC(=O)NCC=CCNC(=O)C(F)(F)c1csc(C)c1)SC C(C)(C)(CC(=O)N(C)CC1CN(C(C2(C#N)CCCO2)=O)CCO1)OC c1(CC)ccc(C(=O)N(C)CC2CCN(C(=O)Cc3ccc(C)o3)C2)cc1F c1(-c2cn(C(CC=C)CC=C)nn2)cccc(C#N)c1.c12oc(cc1C)SC2 c1(C(N(C(CC)CC(=O)NC2(CNC(N)=O)CCCC2)C)=O)cc2cccnc2[nH]1 c1(C(=O)NC(c2ccncc2)CC)coc(CNC(C2CC3(CC3)C2)=O)c1 Cc1cc(C(=O)NCC(C)(C)CNC(c2[nH]c(C)nc2C)=O)c(N)c(C)c1 C1(NC(C(C(C)C)O)=O)CCC(C)N(C(=O)CC2CCC(C3CC3)O2)C1 Cc1nn(-c2ccncc2)cc1CN(CC(O)C(C)(C)C)C C1(O)(C(=O)NC2C(N(C)C(c3cnn(C)c3F)=O)CCCC2)CN2CCC1CC2 CCC(C(=O)NOC1CCCC1)N(C)C(C1CN(CC)CC1C)=O C1(NC(c2nccc(OC)c2)=O)CN(C(=O)C(C)NC=O)CC12CC2 N1(C(c2c(OC)csc2)=O)CC(CNC(=O)CC(C)CF)C2(CCOCC2)C1 N1(C(c2c(CC)nn[nH]2)=O)CCN(CCNC(c2ccnc(C)n2)=O)CC1 N1(C(CC(C)(F)F)=O)C2CC1CN(C(c1cc(C(C)(F)F)ccn1)=O)C2 c1(OC)cc(C(c2nnnn2C)NCC(C)(F)F)cc(Br)c1 C(C(=O)N(CC(C)(C)NC(C1CCN(C)CC1)=O)C)(C(C)C)NC(C)=O CC1(C)CC(CNC(c2nnnn2-c2ccccc2Cl)C2C3COCC23)CNC1=O C12(C(N(C)CC3C(C)C3)=O)CCC(CC1NC(c1cc(F)c[nH]1)=O)C2 CCC(C#N)(CC)C(=O)NCC(C1CC1)NC(C1(C)CC(C)(C)C1)=O C1(C2CC2)(CNC(COC)=O)CCN(C(=O)C(c2cc(C)ncn2)(F)F)C1 N1(C(C2CC2c2cc(I)c[nH]2)=O)CCC(c2ccccc2)NC1=O c1(C(=O)NC(C2(O)CN(C(C3CC(OC)C3)=O)C2)C)sc(Cl)cc1Cl C1(NC(C2C(=C)C2)=O)CCN(C(=O)CCc2csnn2)C12CCC2 N1(C(C(CC(C)C)NC(c2cc(C)nn2C)=O)=O)CCC(C)(C2CC2)C1 Cc1ccc(C(N2CCCC2CCc2cccs2)C(=O)NCC2CCC2)o1 CCC(CC(=O)N(C)Cc1ccsc1)NC(=O)Cc1csnc1C C1(NC(CC2CCN(C(C=C(C)C(C)C)=O)CC2)=O)CCOC12CCOC2 N1(C(CN(C)C(N)=O)=O)CCC(C2CCN(C(c3cc(C4CC4)ccn3)=O)C2)C1 c1(N(C(C(c2cccnc2)NC(CC)=O)=O)CC(N2CCCC2)C)ccncc1F C12(NC(=O)CCCF)CCCN(CC(F)(F)F)CC1C2.c12cccc(n1)NC2=O c1(C(N(CC(C)N(C)C(c2nnn3c2CSCC3)=O)C)=O)csc2c1CCCC2 c1(OC)nc(-c2nc(-c3nccs3)nn2CCN2CCCC2)cc(O)n1 N1(C(C)=O)CCCC12CCN(C(=O)C(C)OCC(C)C)C2 C1(C(N(C2COCC2(C)C)CC)=O)CCN(C(=O)CC2CCCN2C)C(C)(C)C1 N1(C(CC2ON=C(C)C2)=O)CCC(N(C(=O)CC2(O)CCOCC2)CCO)CC1 N1(C(c2cccc(C#N)c2)C(=O)Nc2cccc(C)c2)CCC2CCCC12 c1(C(=O)NC(CN(C(C(C)C2CCCC2)=O)C)(C)C)ccc2c(c1)nnn2C c1(C(=O)NCCCN(C(CCC(C)=O)=O)CCO)cnc(N)c(Cl)c1 C(=O)(C1=NNC(=O)CC1)N(CCCNC(C1CC(C)(C)C(=O)NC1)=O)CCO c1(CC)cc(NC2CN(C(c3n[nH]cc3C)=O)CC2C)nc(C)n1 CCC(C)(CCNC(=O)Cc1ccc(O)nc1)NC(=O)C(=Cc1cccnc1)F c1(CC)ccc(NC(C2CC(OC)CN2C(=O)CCN2CCCCC2=O)=O)cc1 Cc1cc(Cl)cc(N)c1C(N1CCC(C(C)(C)C)C1)=O CC(C)C(C)CC(=O)NC1(CNC(c2ccc(Cl)cc2Cl)=O)CCOC1 c1(C(N(CC)Cc2cccnc2)=O)cnc2n1CCN(C(C1CCCO1)=O)C2C C1(F)(CNC(c2n(C(C)C)ccn2)=O)CCN(C(C2CCC(C)(F)CC2)=O)CC1 c1(C(=O)NCCC(=O)N(C(C)C(=O)NCC(F)F)CC)c(F)cncc1F c1(C(=O)NC(C(C)NC(=O)CCc2ccoc2)(C)C)cccc(S(N)(=O)=O)c1 N12CCC(C)(C)C(C1)C2=O.Cc1nc(O)ccc1C(=O)NCC=CC(C)(C)C Cc1occc1C(N1CCCC1CCNC(C1CC1(C)C(F)F)=O)=O S(=O)(=O)(c1ncc[nH]1)NC1CC(CC(=O)OC)C(O)C1 C1(C=O)CN2CCC1(C)CC2.CC1(C)CCCC(C2(c3cn(C)nn3)CCC2)O1 S(=O)(=O)(CC(=O)NC(C)CN(C(=O)Cc1ccc(F)cc1)C)NCC C(=O)(C#CC1CCCCC1)NCC1CCCCN(C(CCC2N(C)CCC2)=O)C1 c1(C(=O)NCCC2(OC)CN(C(=O)COC(C)C)C2)cc2cccc(Cl)c2cn1 Cc1ccnc(C(=O)N(C)CC2CN(C(=O)C(n3ccnc3C)C)CCO2)n1 c1(C(=O)OC)cc(C)ccc1S(=O)(=O)Oc1cccc(NC2CCC2)c1 N1(C(c2cccc(C)c2)=O)CC2(CCCC2NC(C2CC3CCC2C3)=O)C1 C=CC1(C(=O)NC2CC(n3cccn3)C2)CCN(C(=O)C(C(C)O)N(C)C)C1 N1(C(c2c(C(=O)OC)ccs2)=O)CC2(NC(c3cc(C4CC4)ccn3)=O)CC1C2 N1(C(c2c(C)nc(Cl)cc2)=O)C2CCC1CC(CC(C)NC(C1(C)CC1Br)=O)C2 c1(C(=O)NOCCCC2CCCN2)ncnc2sc(Br)cc12 C1(NC(CNC(=O)OC)=O)CC2CC1CC2C(=O)NCC(F)C1CCC1 N12CC3C(C1C(=O)Nc1cc([nH]n1)C2=O)C3(C)C.C1(COC)(CO)COC1 CC1CN(C(=O)Cc2n[nH]cc2Br)CC1CNC(=O)C(C)(C)F c1(CCC)cc(=NC2CN(C(C3CC(C)CO3)=O)CC3(CCC3)C2)[nH]c(Cl)n1 c1(CCCC(=O)NC2CC(C)(NC(C3CC(C(F)F)C3)=O)C2)cccc(Cl)c1 S(=O)(=O)(c1cc(C(=O)O)c(F)cc1Br)N1CCCN(C(=O)OC)CC1C Cc1cc(C#N)sc1C(=O)NCC12CCC1CN(C(=O)Cn1cccn1)C2 c1(CC)cccc(NC(=O)C(CC(C)(C)N)NC(=O)OC(C)(C)C)c1 c1(C(=O)NCC2CN(C(C(C)CC(C)(F)F)=O)CC2C)cccc2c1ccn2C C(=O)(CCCC(C)(F)F)NC(C(C)C)(C)CNC(c1ccsc1C(F)F)=O CCCC(O)C(=O)NC1CCN(C(=O)COCCOCC)C1 Cc1cc(C(=O)N(C)CCN(C)C(C2CCC(O)(C(F)(F)F)C2)=O)c(C)s1 CCCCCC(O)CC(=O)NCC1(C)CCCN(C(=O)CCOCC)C1 c1(OCC)ccccc1C(=O)NC(C1CN(C(=O)CC(C)(C)OC)C1)C N1(C(C2C(OC)CC2)=O)CC(F)(CNC(c2cnc(C3CCCO3)s2)=O)C1 N1(C(CCC2(C)CN(C(C(C(C)C)O)=O)C2)=O)CCCC(C)(C#N)C1 Cc1cnn(C)c1NC(c1ccc(CNC(C2C3CC4C(C3)C24)=O)cn1)=O C1(C(=O)Nc2ccc(C(C)C)o2)CN(C(=O)CC(C)N(C)C)CCC1O c1(C(=O)NCCC2CC2)c[nH]c2ncccc12.Cc1ccns1.C12(CCC1)C(=O)N2 C=C(C)C(C)(C)C(=O)N1CCCC(N(C)C(C2CCN(C)C2=O)=O)CC1 c1(NC(C2(NC(C)=O)CCC2)=O)cccc2c1C1CCC2N1C(=O)C=C(Cl)Cl N1(C(CCSC)=O)CCCCC1COC.C1(C)(C)CC=CC(=O)N1 N1(C(C)C)CCC(C(=O)NC2CCCC(N(C)C(c3cn(C)nc3Cl)=O)C2)CC1 c1(SC(C)C)ccc(C(=O)NC2C(NC(CCC)=O)CC2)cc1.C1(=O)CN1 C1(OC)CN(C(=O)CC2CCCOC2)CC1NC(c1ccc(SC(C)CO)o1)=O N1(C(CCC(CC)NC(C2CC23CCCCC3)=O)=O)Cc2cnn(C)c2C1 Cc1nc(C(=O)NCC2CCC(NC(=O)CCNc3ccccc3)CC2)ccc1Br CCCCC(C)CCC(=O)NC(C)C(C)(C)C(=O)N1CCCC1C c1(C(N2CC(C)C(NC(=O)CC3CC=CCC3)C2)=O)cc2scnc2[nH]1 C1(COC(c2cc(F)n[nH]2)=O)CCCC1(C)NC(=O)CC1CC(OC(C)(C)C)C1 N1(C(c2c(C)nco2)=O)CCN(C(=O)CNC(c2c(C)n[nH]c2C)=O)CC12CC2 C12(C(=O)NCC(CNC(CN3CC(C)(C)C3)=O)O)COC(CC3CCCC3)(C1)C2 N1(C(C(C)OCC=C)=O)CCCCC2(C1)CN(C(=O)C=Cc1ccc(C)cc1)C2 CCCCC(O)C(C)C(=O)N1CCC(F)CC1C(=O)N(C)CCC(CC)C=O c1(C(=O)NC(CCNC(C2CN(CC)C(=O)C2)=O)C)cnc2n(c1=O)CCS2 C(=O)(CCCCNC(c1cnn(CC)c1C)=O)NC(C#C)CC c1(CC(=O)N(C2CCN(C(=O)C(C)SC)C2)CC)cccnc1Br C#CCC(C)(C(=O)N(CCC(=O)N1CCOCC(C2CC2)C1)OC)OC N1(C(C(C)Cc2cnco2)=O)CC2CCC(C1)N2C(=O)C(F)(F)c1nccs1 CN=c1nc(N2CCCCC(C)C2)[nH]c(=NCC2CSCCS2)[nH]1 Cc1cc([N+](=O)[O-])cc(C(N2CCN(C(=O)C(C)C)CC2c2ccncc2)=O)n1 S(=O)(=O)(c1ccc(NCCSC(F)F)c(Cl)c1)NCC1CC(COC)OC1 c1(C(=O)NCC2(CCNC(C3(COC)CCCC3)=O)CC2)c(Cl)cccc1Cl C1(C(C)Nc2cccc(C(=O)NC(C)(C)C)c2)CC(C(C)(C)C)=NO1 c1(C(=O)NC2CC3(C2)CN(C(C2CCCS2)=O)C3)ncc2n1CCCC2 C(=O)(C1=CCC(F)(F)CC1)N1CCC(NC(c2cn(C)[nH]c2=N)=O)C12CC2 C1(CC(N2CCN(C3CCN(C(=O)CC4CC4)C3)CC2)=O)C2CN(CCCO)CC12 CCCCCCCCNC(=O)C(N1CC(O)CC1CNC(=O)CSCC(N)=O)=O C(=O)(C1=NN(CC(C)C)C(=O)CC1)NC(CNC(C(CC)CC)=O)(C)C(C)C C1(C(=O)NC2CCN(CCNC(c3ccc(CC)[nH]3)=O)CC2)CCCCC1C1CC1 C=CCCC(F)(F)C(=O)N(C)CC1CCCN1C(=O)C=CSC c1(C(=O)NC(CN(C(C(CC#C)O)=O)CC)C)oc2c(C)cccc2c1C N1(C(C(CCOC)C)=O)CC(C(=O)NC(C)CC(C)(C)CO)CC1(C)C C1(C(C)C)CCCCC1NC(C1(CNC(=O)C(=Cc2cscn2)F)CCCC1)=O c1(-c2c(C(=O)NCC(CNC(CC(C)(C)F)=O)(C)O)c[nH]n2)c(F)cccc1F N1(C(C2(c3ccc(Cl)nc3)CC2)C)CCCCC(Cn2cc(COC(=N)O)nn2)C1 CCCC(C)(C)C(=O)N1CCC(C(F)CNC(=O)C(C)(O)c2ccccn2)CC1 C1(CNC(CC2(C=C)CC2)=O)CN(C(=O)COCCCOC)CCC12CCOC2 C1(NC(=O)CN(C2CCC2)C(c2ccc(O)nc2)=O)CCOC12CCOC2 c1(C(=O)NCC2C(NC(c3cncc(OCC)c3)=O)C2)ccnc2nnn(C)c12 C1(F)(C(=O)O)CN(C(=O)O)CC1SCCCn1cnccc1=O.c1(C)ccccc1 NS(=O)(=O)C1(CSCC(=O)Nc2cncc(-c3cc[nH]n3)c2)CC1 c1(C(=O)NC2C(NC(C(C=C)(C)CC)=O)C2)ncn2ccccc12 C1(O)(C(C)(C)C)CC(CN=c2cc(Cl)nc(-c3cccc(C(F)(F)F)c3)[nH]2)CCO1 c1(OCC)cc(F)ccc1CN1CC2(CC2)CC1C(=O)NCc1ncccc1F c1(C(N2C(C)CCN(C(C3CC=CCO3)=O)CC2)=O)cnc2c(c1)C(=O)CCC2 c1(CC(=O)NC2(CNC(CC(=O)NCC)=O)CCC2)ccc(C)nc1Cl c1(CCC)c(NC(=O)NCC2CC2C(=O)OC(C)(C)C)nsc1OCCC N1(C(c2cc(C)ns2)=O)CC2CCC(NC(C3CCN(C)C(=O)C3)=O)CC2C1 C(C(=O)NCC1(F)CN(C(=O)CCC2CCCCN2C)C1)(C(C)(C)C)SC C(C(C)(C)C1=CCOCC1)NC(CCCCC)c1n(CC=C)nnn1 N1(CC(=O)NC(CNC(C(C)OCC#C)=O)(C)CO)C(=O)CCC1=O Cc1nc(O)ccc1C(=O)NCCCCC1CCCN(C(=O)Cn2cnnc2)C1 C(=O)(C1=CCCN(C(C2CC(=C3CCC3)C2)=O)C1)NCc1cc(C)cc(Cl)c1 C1(C(C)C)CN(C(c2ccn(CC(F)(F)F)n2)=O)CCC1NC(c1nccs1)=O Cc1ccccc1N1CCC(C(=O)NCC2(N)CCCC2)C1=O c1(C(N2CCC(C)(CCNC(C3(C)CC3)=O)CC2)=O)ccc2sccc2c1 C1(NC(C(C)C2CCCO2)=O)CCC(CNC(C2CS(=O)(=O)C2)=O)C1 CC1(C)CN(C(C2CCCCC2)=O)CCC1NC(c1ccccc1OC(F)F)=O CC1CCCC=C1C(=O)N1CC(O)CC1CNC(c1ccc(Br)cn1)=O C=CC1CN(C(c2ccc(SC)cc2)=O)CC1NC(=O)CC1(CC(=O)OC)CC1 CCC(C)CC(C)C(=O)NCC1COCCN1C(=O)Cc1cc[nH]c1 O(N(C)C(=O)CN=C(NC(C)COC)NC1CCC(C(F)(F)F)CC1)CC N1(CC(N2C(CNC(c3cccn3C)=O)CC(OC)C2)=O)C(=O)CC(C)(C)C1=O c1(Cn2cc(CN3C(CCC(C)O)CCCC3)nn2)noc2c1CCC2 N1(CCC(=O)N(CC(=O)N(C)C)C(C)C)CCOCC1.C12CC1C(=O)NC2C Cc1noc(Cl)c1COC(C1CC(=O)N(C(C)(C)C)C1)=O C(C)(C(=O)NCCCCN(C(=O)C(C1CCCC1)C1CCC1)C)N(C(C)=O)C C1(CCNC(C(n2c(C)ccn2)C)=O)CN(C(c2csc(F)c2)=O)CC1C c1(CC)sc(C(=O)NC2CC(F)(CNC(=O)CCC3CC(OC)C3)C2)cc1C N1(C(c2c(O)ccc(SC)c2)=O)CCC(C)N(C(=O)C(C)C(F)F)CC1 C=CCC(O)(CNC(=O)Nc1ccccc1SCCN(C)C)CC=C CCCCS(=O)(=O)CC(=O)NC(C)(C)CCNC(c1cnc(COC)cn1)=O c1(OC)cc(Br)c(F)cc1S(=O)(=O)N1CCCC1NCCCOC(F)(F)F C(CCCCCN=[N+]=[N-])NC(C1CCCC1)CC c1(C(=O)NC2C(C)CN(C(C3CCCC3)=O)C2)ccc(-n2ccnc2)c(F)c1 C(=O)(C(CCC)C(C)C)NC(CC#C)CC(=O)NC(C)C(=O)NC1CC1 Cc1cc(C#N)cnc1C(N1CCCC1(C)C(=O)NC(C1CCCCC1)C)=O C1(C(N(C2C3CN(C(=O)C(c4cccc(F)c4)F)CC23)C)=O)CCC2(CCC2)C1 C(=O)(C(=O)C(C)(C)C)NCC(C)N(C(=O)Cc1c[nH]nc1C)CC CC(C)(C)C(C(=O)NCCCc1ccco1)c1ccccc1 c1(CC)cscc1C(=O)NC(C)C(C)(C)NC(c1[nH]nnc1COC)=O C12(CNC(=O)Cc3cccnc3)CCCCC1N(C(c1ccc(F)cn1)=O)CC2 N1(C(C=CC)=O)CCN(C(c2cc(C)co2)=O)CC1C1CCCC1 c1(OC)ccccc1-n1nc(Cc2csc(C)n2)nc1-c1ccc(C)nn1 c1(CC(N2CC3CC3(C(=O)NCc3ncc(Cl)cn3)C2)=O)nc2ccccc2s1 C(=O)(CCS(=O)(=O)CC(C)C)NCC1(CNC(c2cccc(C)n2)=O)CC1 C1(O)(CCNC(C2N(C)CCC2)=O)CCCN(C(=O)C=Cc2cnn(C)c2)C1 CCC(CCC(=O)N1CC(=O)NCC1C(C)C)NC(=O)C1=CCCC1C c1(OC)cc2c(cc1Br)C(NCC(=O)Nc1ccc(C)c(Br)c1)CC2 N1(C(C=CCCC)=O)C2CCC1CN(C(c1cc(O)nc(C)n1)=O)C2 C(C(=O)NCC1CC1CNC(=O)Cc1ccnnc1O)(C(C)(C)C)N(C)C Cc1cc(Cl)c(C(=O)NCC2CCC(C)CN2C(=O)CN2CSCC2=O)cc1F CCC(CNC(C1CCC1CNC(c1cc(O)cc(F)c1)=O)=O)(CC)CC c1(C(=O)NC(CCCOCCC)c2ccccc2)c(SC)cnn1C c1(C2(C(=O)NCC3N(C(C(CC)N(C)C)=O)CCC3)CC2)cccc(OC)c1 N1(C(C2C(OC(C)=O)C2)=O)CC2CN(C(C3CC(=O)N(C(C)C)C3)=O)CCC12 c1(CC(N2C3CN(C(CCCCOC)=O)CC2C3)=O)c(C)nc2ncnn2c1C N1(C(c2ncn3c2CCC3)=O)CCC(O)C(NC(C2(CO)CCCCO2)=O)C1 c1(CN2CCC(N(C(=O)CC3(C4CC4)CC3)C)C2)cnc2n1CCOC2 c1(CC(C)C(N2CCCC(C(N3CC=CC3)=O)CC2)=O)ccc(F)c(F)c1 C(c1ccsc1[N+](=O)[O-])=CC(=O)N(CC(C)NC(CCCOC(C)C)=O)C O=C(CC1=Cc2ccccc2C1)NCc1cc2cccc(Br)c2o1 c1(C(=O)NCC(CO)NC(=O)CCCN2CCCCC2)cnc2c(c1)CCC2 CCC(C)CCCC(=O)NC(C(=O)NCc1cc(C)ncn1)C1CCC1 c1(C(COC(C(=O)OC)C)=O)ccc2c(C)ccnc2c1 c1(C(N(C2CCN(C(c3ncc(CC)nc3)=O)C2)C)=O)cnc2cc(C)ccn12 c1(-c2cn(CC3N(C(c4cc(C(F)(F)F)co4)=O)CC3)nn2)cnc(Cl)c(Cl)c1 N=c1ncc(C(=O)Nc2ccccc2C(F)(F)F)c[nH]1 c1(C(=O)NCCO)cc2cccnn2c1.N12CCC3CC13C(=O)NCC2=O C1(C(C)(C)NC(c2cc(C(C)C)[nH]n2)=O)CCN(C(C2CC(N=[N+]=[N-])C2)=O)CC1 C(=O)(CCC(C)S(C)(=O)=O)NCC1N(C(CC(C=C)(C)C)=O)CC2(CC2)C1 CC(C)C(CC(=O)NCC(C)(C)C(C)O)NC(=O)CC1CCC(=O)N1C C(c1ccc(C)cc1)=CC(N1CC(CC)C(C(=O)NC2COCC2O)C1)=O C#Cc1cn(C)nc1C(=O)N(C1(CC(=O)NCCCCC)CCC1)CC Cc1sccc1CC(=O)N(C1CN(C(C23CC(c4ccccc4)C2C3)=O)C1)C C1(C(=O)NC(C)CCNC(=O)C(F)CC2CC2)CCN(c2cccc(F)c2)CC1 C(=O)(CC(C)(C)COC)N(CC(C)NC(C1CCC(=O)NC1)=O)CC C(C(C)(C)C(=O)N(CC)OCC)C(=O)NC(C(CCC)O)=O C1(CC(=O)NCC(CN(C(CC(C)F)=O)C)(C)C)CC(C)(C)CO1 CN1CCC(n2nccc2-c2ccc(N)cn2)CC1.C1(=O)C=CCO1 c1(OC)nc(Cl)ccc1C(=O)NCC1CCN(CCOC)C1.c1(C)nc(C(C)C)no1 CC(C)(C)CCC(=O)NC1CCCC(NCc2ccccc2F)C1 c1(N2C(CNC(c3ccc4nn[nH]c4c3)=O)CCC2)ncnc2cnccc12 N1(C(CCNS(CC)(=O)=O)=O)CCCC(C)(C)C1CNC(C1CCCCC1O)=O C1(CN(C(C(CC)C)=O)C)CCN(C(c2cncn2C2CC2)=O)CC1 C1(CCCC)CN(C(=O)C(O)CC(N)=O)CCN1C(=O)Cc1ccc(C)cc1F N1(C(C2CC(=O)C2)=O)CC(C(=O)NC2CC3(C2)CC(O)C3)C(F)(F)C1 C(=O)(C(CC)C(=O)NC(CNC(c1ccc(F)cc1SC)=O)C(C)C)OCC c1(C(N2CC(C)C(CNC(c3[nH][nH]c(=N)c3Br)=O)C2)=O)cnc2n1CCOC2 C(=O)(C1=CCCN(C(c2cn3c(n2)CCC3)=O)C1)NC1CC(C)(C)OCC1 C12(CC(N3CCC(COC)(NC(=O)C=C(C)Cl)CC3)=O)CCC(CC1)C2(C)C C12(C(=O)Nc3c(OCCCC)ccc(F)c3)CC(C)(C1)OC2(C)C c1(C(=O)NCC(CC)Nc2cc3nnc(C)n3cn2)cc2ccc(OC)cc2[nH]1 C(CSC)(C(=O)N1CC(F)(C(=O)NC(CC2CCCC2)CO)C1)OC c1(CNC(C2(F)CCCN(C(=O)CC3CC4CCC3C4)C2)=O)cc(F)cc(F)c1 N1(C(c2ccn(CC)c2C)=O)CCN2C(=O)C(NC(c3cc(C)c[nH]3)=O)CC2C1 C(N(C)N1CCCCC1c1nnc(-c2ccccc2C(F)F)o1)c1c(C)n(C)nc1 c1(C(N2C(CN(C(C3C(COC)C3)=O)C)CCC2)=O)ccc(F)c(C(F)F)c1 c1(C(N(CCN(C(=O)CSCc2cccs2)CC)CC)=O)n[nH]c2c1CSCC2 c1(C(N2C(CN(C(C(COCC)(C)C)=O)C)COCC2)=O)c(F)cc(C)cc1F c1(OC)ncc(-n2cc(N3CC(OC)CC3C(N3CC4CC4C3C=C)=O)nn2)cn1 C(=O)(C(C)P(C)(C)=O)NC(C)CCN(C)C(C1(c2ncccc2F)CCC1)=O c1(CN(CCc2nc(C(C)C)on2)C)cc2n(n1)CCCC2 n1(CCC)ccnc1CN(C(C1CCC(C)C1)C(=O)N(CC(F)F)CC)C c1(C(=O)NCC(CO)NC(=O)C(O)CF)ccc2c(c1)OCC2 C#CCCCCC(=O)NCCCNC(c1cc(C2CCC2)no1)=O c1(C(=O)NCCN(C(c2ccnc(S)c2)=O)CC)ccnc(SC)c1 C(=O)(C#CC1CCC2(CC1)OCCO2)NCC1N(C(C2(CC)CC2(F)F)=O)CC1 C1(C(=O)NCC2CCCO2)CSCCN1C(c1ccc(C2CC2)o1)=O CC(C)C(C(=O)NCCCCCNC(c1ccnnc1S)=O)NC(N)=O C(C(C)(C)CNC(=O)CC1CC=CCC1)NC(C(C1CCC1)OCC)=O N1(C(C2(COC)CCC2)=O)CCC(CN(C(=O)C(C)CF)C)CC1 C1(C(=O)NCC2CC(=C)C2)CC(F)(F)CN1C(=O)Cc1ncc(F)cc1F CCCCCCCC(=O)N1CCCC1(C)CNC(=O)Cn1nnc(=O)[nH]1 n1(CCCC)ncc(C(N2CCCC2CCCNC(C2(C)C=CCC2)=O)=O)c1C CN1CCC(F)(CNC(C2CN(C(c3c[nH]cc3C3CC3)=O)CCO2)=O)C1 c1(C(=O)OC)cc(C(=O)NC(C(F)(F)F)C2CC2)ccn1.N12CC(=O)CC1C2=O C1(O)(CC(N)=O)CN(C(=O)C(Cc2ccoc2)NC(C2CCCC2O)=O)C1 N1(c2ncc(C)cn2)CCC(C2CCCN(C(c3nc(Cl)ccc3F)=O)C2)C1 C1(C(N(C)CC2CCSC2)=O)C2CCN(C(C3CCCC(C)(C)C3)=O)CC12 C1(C(=O)Nc2cnc(F)nc2)(COC)C=CCN1C(=O)C(CO)NC1CC1 C1(C(=O)NC2CCN(C(=O)C(F)F)C2)CC(O)CN1CC(F)(F)F c1(C(=O)NC)cnn2c1CN(C)CC2.c1(C(=O)NCCN(CC)CC)cccc(CO)c1 C1(C(=O)NCC(=O)N(C2CCN(S(C)(=O)=O)C2)C)CCOC1C(F)(F)F n1(CC)ccc(C(=O)NC(C(=O)NCC(C)C(F)F)C2CCCC2)c1C c1(C(N2CC(CNC(c3cnc4cc[nH]c4c3)=O)C2)=O)c[nH]c2cccc(Cl)c12 N1(C(C2N(CC#C)CCC2)=O)CC(CCNC(c2nccc(N)n2)=O)C(C)C1 c1(C(N(CCCN(C)C2CC2)C)=O)coc(C(F)F)n1.C(=O)(CCOCC(F)F)N N1(C(c2ccsc2C(F)(F)F)=O)CCCC1C1CCCN1C(c1cnns1)=O C(=O)(CC(C)(C)CC(F)F)NC1C=CCN(C(c2cc(C)nn2C2CCC2)=O)C1 C(=O)(C1=CCCCCC1)NCC(c1ccccc1)N(C)C(C1CCCC1CF)=O c1(C(N2CC(CCCCNC(C(CC)F)=O)C2)=O)ccc(-c2cnn(C)c2)nc1 CC1(CNC(C2CCCOC2)=O)CC(NC(c2c[nH]nc2-c2ccccc2)=O)C1 N1(C(CS(=O)(=O)NC)=O)CCCC(CO)(NC(=O)C(C)Oc2ccc(F)nc2)C1 C1(NC(c2cc(C(C)C)no2)=O)CN(C(C2CC3(CC3)CO2)=O)CC1C n1(-c2ccn(C)n2)cc(C2CCCN2C(c2cnn3c2OCC3)=O)c(O)nc1=O C(C)(C)(CCC(=O)NCCC(O)CNC(C1C2CCCCCC12)=O)N(C)C C1(C)(C(=O)N(CCOC2CN(C(CC(C)c3ccncc3)=O)C2)CC)C=CCCC1 N1(C(C=C(CCC)C)=O)CC(C(=O)NCCC(=O)N(C)C2CC2)C(F)(F)C1 C1(CC)CCC(C(N2CCCC(N(CCF)C(C3CC(N(C)C)C3)=O)C2)=O)CC1 CC1CC(NCc2cn(C3COC3)nn2)(CO)CC1(C)C c1(OC)ccn2c(C(=O)NCCC3(NC(c4cnco4)=O)CC3)cnc2c1 c1(CC)nc2c(C(N3CCN(C(c4cn(CC)cn4)=O)CC(O)C3)=O)ccnc2[nH]1 C1(NC(C(c2ccc(OC(C)=O)cc2)CC)=O)CCN(C(C)=O)CC1O c1(CNCC2C3CCC(CO)C23)ccc2nncn2c1 N1(C(c2cc(C)no2)=O)CCCC(CC(=O)NC2CC2c2ccccc2)CC1 CC(C)(C)C(C)(O)C(=O)NC1(CNC(C2CC(n3cnnc3)C2)=O)CC1 CC(C)CC(C(=O)N(CCNC(=O)C(C)(C)C(C)C)CC1CC1)N1CCCCC1 c1(C(=O)NCC(C)NC(c2nscc2N)=O)nn(C)c(Cl)c1Cl CCC(CC)(CCNC(=O)CCc1ccc(O)cc1)NC(C1CCC(C)CC1)=O c1(C(=O)NC2CC(NC(C3CCOC3c3cc[nH]n3)=O)C2)cccc(C(F)F)c1 CCC(C(=O)Nc1ncccn1)n1ccc(COC(C2CCCSC2)=O)n1 c1(-c2n(-c3c(C)cccc3)nc(CCCO)n2)ccc2ccccc2c1 c1(-n2cc(CC(C)(C)CSc3cn(-c4ccccc4)cn3)nn2)cccc(Cl)c1 c1(NC(=O)NCCc2nnc(C3CC3)s2)cc(N2CCCC2)cc(Cl)c1 c1(C(C(=O)NCCN(c2cccc(F)c2)C(=O)CO)(F)F)ccc(Br)nc1 N1(CC)CCCC1CC(=O)NC1CC1CNC(c1sncc1Br)=O C1(C(CC)C)CCC(CNC(=O)NC(C)C2CC2)CC1 N1(C(Cc2[nH]c(=N)sc2)=O)CCOC(CNC(C2CCCC2(F)F)=O)C1 C1(CNC(C(CSC)N(C)C(C)=O)=O)CCCCC1c1nc[nH]n1 C(CCCc1ccccc1)(C(=O)NC1CCCCC1)N(CC(=O)OCC)C C12(CC13CCC3)C(=O)NC2.c1(SC)ncc(C(N2CC(c3nc(C)no3)C2)=O)s1 C(=O)(CCC(=O)N1CCC(CNC(c2cccc(CS(C)(=O)=O)c2)=O)C1)NCC C1(C(C)NC(=O)CN(C)C(N)=O)CCCN(C(=O)C(C)SCC(F)F)C1 c1(OC)ccc(C)c2[nH]c(C(=O)OCCOc3ccc4c(c3)CC4)cc12 C1(C(CO)NC(c2cc(Cl)ns2)=O)CCN(C(=O)Cc2nc(C3CC3)cs2)CC1 C(=O)(C1Cc2ccccc21)NCC1N(C(C=CC(=O)OCC)=O)CCC(C(C)C)C1 N1(CC(N2CC(C)N(C(=O)CSc3nc[nH]n3)CC2)=O)CCc2sccc2C1 Cc1nn(C(C)C)c(NCC2(F)CC(NC(C3CCC3(C)C)=O)C2)c1[N+](=O)[O-] c1(C(=O)NCCN(C(C2CC3(CCCO3)C2)=O)C2CC2)coc2c1CS(=O)(=O)C2 c1(C(N2C(C(=O)NCC3N(CC)CC3)C=CC2)=O)ncnc(O)c1F n1(C(C)C(=O)OCCCC23CCCCC2C3)c(C2CC2)nc2ccccc12 N1(C(c2cc(OCC)n[nH]2)=O)CCC(O)(C(C)NC(C2(CO)CCCC2)=O)CC1 N1(C(C2(Cc3ccccc3)CCOC2)=O)CCC2(CC=CCO2)CC1 c1(C(C)N=c2[nH]c(C(F)(F)F)cs2)ccc2nn[nH]c2c1O c12cn(nn1)CC1CN(C1)C2CC.c1(C)conc1C(C)(C)C.N(C)C CCC(C(=O)OC)C(=O)NCC1(C)CCN(C(C2CC(C)(C)CN2C)=O)CC1 Cc1cc2[nH]c(C(N3CCCC(NC(C4(Cl)CC4(C)C)=O)C3)=O)cc2o1 Cc1cccc(C(N2CCN(C(=O)CCF)C(C)C(C)C2)=O)c1[N+](=O)[O-] C(=O)(C(C)CCC(C)(C)C)C12C(NCC1)CN(CCC)CCC2 c1(N(C2CC(OCCCC)C2(C)C)C)ccc(I)c(F)n1 c1(CC(=O)NC2(CCCNC(=O)Cn3ncnn3)CC2)ccccc1O N1(C(C2CCN(C(C3CCN(C(C)=O)C3)=O)CC2)=O)CCN(C)C(C(C)C)C1 c1(C(=O)NCCOCCNC(c2[nH]cc(CC)n2)=O)ncn2c1CCCC2 c1(N2C(CCNC(c3c(CC)ncs3)=O)CCC2)ncnc2c(Br)cccc12 N1CCN2C(=O)CCC2C1.CCC(C)CN(CCCOC)C N1(C(Cc2cccc(C)c2F)=O)CCC2C1CCN2C(c1cccc(F)c1)=O C(C(C(=O)NC1CC(CC)C1)n1cc(CN2CCCC2)nn1)OCC C1(C(N2C(C)CN(C(c3ccc(Cl)nn3)=O)CC2)=O)CCC2(C1)CC2(F)F c1(CC)cncc(C(N2CC(NC(=O)CN3CCN(c4nccs4)CC3)C2)=O)c1 C(C(C)(C)CC(=O)NC(c1cnn(C)c1C)C)NC(C1CC(C#C)(O)C1)=O C1(C(N(CCCC(=O)NCC(=C)Br)C)=O)C(C)(C)C1(F)F c1(N2CCC(CC=C)(NC(C3C4CC5C(C4)C35)=O)C2)ncnc2sc(C)nc12 c1(CC(N2CCCC(NC(c3ccc(=N)[nH]c3)=O)CC2)=O)n[nH]c2c1CCCC2 C1(C(=O)NC(CC)CO)CC(F)(F)CN1C(c1ccnc(C)n1)=O C1(C(=O)NC(C(=O)N(CC=C)CCO)C2CC2)CC(C)(C)CO1 Cc1ccc(C=CC(=O)NC(CNC(C2CCC(CO)CC2)=O)C2CCC2)nc1 Cn1cc(NC(=O)CC2CCCC2)nc1C(=O)NCCc1ccc(F)nc1 C(=O)(C(CO)C(F)(F)F)NCc1c(C(=O)NCC(C)N(C)C2CC2)con1 N1(C(c2ncn(C(C)C)n2)=O)CCCN(C(c2coc(N(C)C)n2)=O)CCC1 c1(C(N(C)CC2CCCCN2C(c2cn[nH]c2)=O)=O)cc(F)c(F)cc1O C1(C(N2CCN(CCOC)CC2)=O)CCCCCN1C(=O)Cc1ccnn1C N1(C(C(C)NS(CCCC)(=O)=O)=O)CC2(CCN(C(=O)CN3CCOCC3)C2)C1 C1(NC(C2(CCOC)CC2)=O)CN(C(c2ccoc2)=O)CC(C)(C)C1 O(NC(=O)CCCCC(C)C)C(C(=O)NCC=C(C)C)C c1(CC(=O)NC2CN(C(C=Cc3c(C)cccc3)=O)C2)cccc2[nH]ncc12 C1(C(=O)NCC(CNC(C=Cc2cn(C)nn2)=O)(C)C)CC2(C1)CC(O)C2 c1(C(=O)NCC(CCNC(CCCC(C)C)=O)O)coc(S(=O)(=O)N(C)C)c1 c1(C(=O)NCCCOCCNC(c2cnc(C)s2)=O)cc(Cl)c(Cl)n1C Cc1cc(C(C)C(N2CC3CC(NC(=O)CC4CC45CC5)C2C3)=O)cc(F)c1 C(=O)(C1COc2ccccc21)NCC1(CNC(c2cc(C)nc(O)c2)=O)CC1 C(=O)(NNC=O)NC(C)(C)C.Cn1ccnc1C1CC1 N1(C(=O)Cc2ccsc2)CC2CCN(C(C3Cc4c(F)cccc4O3)=O)CC2C1 C(=O)(CCCC(C)(F)F)N1CC2C(NC(CSCC=C)=O)(CC2)C1 N1(C(CC2OCC(C)(C)C2)=O)CC2(CCCC2NC(c2coc(N(C)C)n2)=O)C1 N1(CC)CCCC(NC(=O)CC2(NC(C3CCOC3(C)C)=O)CC2)C1 CCCC(C(O)C(=O)NC(CC)C1CC1)NC(c1cn(C)cn1)=O c1(NCCCC(C)NC(C2CC(c3ccncc3)C2)=O)cc(C(F)(F)F)ncn1 CC1(C)OCCC1C(N1CC2C(C(=O)NCCNS(C)(=O)=O)C2C1)=O C(=O)(C1=CCCCC1C)NCC(CCC)C(=O)NCCC(O)CCO c1(OCC)ncc(C(N2CC(NC(=O)C(C)OCCC(C)C)C(C)C2)=O)cn1 C1(C(=O)NC(CNC(c2cc(C)ncc2)=O)(C)CO)CC2CCC(C1)N2C(C)C c1(C(=O)NCC2C3CN(C(CCCOCC)=O)C(C3)C2)nccc2n[nH]cc12 C=CCC(CC(C)C)C(=O)NCCCCCC(=O)N(CC)CC CCCCC(CC(=O)NCCCC(C)(C)OC)NC(=O)C1=C(Cl)CC1 C1(C)(C(=O)NCCC(CCC)C)CCN(C(=O)COC(F)(F)F)CC1 C12(COC)CN(C(C3COCCN3C(C3CC(CF)C3)=O)=O)C(COC)(C1)C2 Cc1cc(CNC2CCC(C(=O)NCCc3ccc(Br)cc3)C2)c(C)cc1O C1(C(N(CC#C)CC=C)=O)CN(C(=O)CCOCCCN(C)C)CCN1C N1(C(C23C(CN(C(c4ccc(CCO)cc4)=O)C2)C3)=O)CCN2CCCC2C1 C(C(C)(C)C(=O)N1CCC(OC2CCC2)C1)N(C(C(C)SC)=O)C C#CCCCCCC(=O)N1CC(NC(C2(C)CCNC(=O)C2)=O)CC12CCC2 c1(-c2cn(CCNC(CCN(C(CCC)C)C)=O)nn2)cc(F)ccc1NCC N1(C(C2N(N=O)CCC2)=O)CC2CC(C1)CN(C(=O)CCc1ccco1)C2 C(c1cccc(Cl)c1)=CC(=O)NC12C(CN(C(c3n(C=C)nnc3)=O)C1)C2 C1(NC(C(C)(C)N2CCCC2)=O)CC2C(NC(=O)Cn3cnnc3O)C2C1 c1(OC)ccc(Br)c(C(=O)NC(C2CCCN(Cc3ccc(F)c(C)c3)C2)C)n1 Cc1ccc(C(N2C(CON)C(CC(C)C)CC2)=O)c(-n2cc(CCO)nn2)c1 c1(C(=O)NC(CNC(CC2C(CC)C2)=O)CO)cncc2c1CCNC2=O C(=O)(CCCC(F)(F)CO)N1C(CCN(C(CCC(CC)OC)=O)C)CCCC1 Cc1cc(F)cc(C(N2CCC(CO)(CNC(=O)CN3CC4CC4C3)C2)=O)c1O c1(C(N2C(CNC(C3(COC)CC(=C)C3)=O)CCC2)=O)ncc(C)cc1C c1(CC(=O)NC(C(C)NC(CN(CCC)C)=O)C(C)C)ccc(F)c(OC)c1 CC1OC2CCC1(CNC(Cc1ncnn1C)C(=O)O)C2 C#Cc1ccc(C(=O)NC2CC(OCC(=O)N(CC3=CCCOC3)C)C2)c(C)c1 C1(NCCCN(CCC(=O)OCC)CC(F)(F)F)CC2CCC1NC2=O C(C(CC(C)C)C(=O)NC1COCC1CO)NC(c1c(C)n[nH]c1C)=O c1(NC(=O)CC2(NC(C3C4CC5C(C4)C35)=O)CCC2)cc(F)cc(F)c1 Cc1cccc2c(=O)c(C(N3CCCC(CO)(NC(=O)CC(C)F)C3)=O)c[nH]c12 C1(CC)CCC(CNC(=O)CN(C(=O)CCCSC(C)C)C2CC2)O1 n1(C(C(=O)NC(CN(C(c2cnn(C(C)C)n2)=O)C)C)C)cnc(C#N)n1 N1(C(C)C)CC2(CCN(C(=O)OC(C)(C)C)CC2)CNC1=O Cc1cc(F)cc(C(=O)NC2(CO)CCCN(C(C3CCNC(=O)C3)=O)C2)c1O CCC(C)C(C(=O)N1CC2(CCC2)C1)NC(c1cccnn1)=O C=CC(C)CC(=O)NCCCN(C(=O)C1=CSCS1)Cc1ccccc1 C1(C(=O)NCC=CCNC(CCCCC(=O)NC(C)C)=O)CS(=O)(=O)CC(=O)N1 Cn1c(C(N2CCC(CCNC(=O)CC(C)(C)C3CC3)CC2)=O)nnc1S CC(C)CC(=O)C(=O)NCC(C)(C1CC1)NC(=O)CCC1CCC(=O)NC1 Cn1c(C(N2CC(F)(F)CC2C(=O)Nc2cnn(C3CC3)c2C)=O)cccc1=O c1(C(=O)NC2C(CNC(C(C)NC(CC)(C)C)=O)C2)n[nH]c2cc(OC)ccc12 N1(C(C(CC)=CC)=O)CCCC(O)(CNC(c2cnn3c2CCC3)=O)CC1 C1(C(NOCc2cccc(C)n2)=O)CCCCCN1C(C1CN(C)C1)=O c1(C(=O)NCC(CNC(c2cncc(C)c2)=O)F)c(C)nc2sc(C)nn12 C1(NC(=O)C(=O)c2ccco2)CCC(c2ccccc2)C1 c1(NC(CC2CCN(CCNCc3ccc(SC)s3)C2)=O)ccc(C)nc1C N1(C(c2c(C(C)NC(c3c(C)nc(CC)o3)=O)noc2)=O)CCC(C)CC1CC C1(CNC(C(C)(C)OCC)=O)CC(F)CN1C(C1CC(C)CO1)=O Cc1nn(C)c(C)c1OCC(=O)NC1CCOCC1NC(C1CC2C=CC1O2)=O CC(F)(F)C(F)C(=O)NCC1CCN(C(=O)C(C)(O)C2CCC2)CC1 N1(C(c2c(CC)occ2)=O)CCN(C(C2OCCOC2(C)C)=O)CC1C(C)(C)C C(c1ncc(C)[nH]1)=CC(=O)NCC1CC(F)(CNC(C(C)N(C(C)=O)C)=O)C1 c1(C(N2C(CNC(c3cc(Cl)cnc3O)=O)CC2)=O)cc2c(s1)CCOC2 Cc1ccc2cccnc2c1C(=O)NCC1COCC1NC(=O)CSCC(C)C CC(C)(CCCNC(c1coc(C2CC2)n1)=O)C(=O)NCC1(C)CCCO1 N1(C(c2c(SC)ccc(N)c2)=O)CC2(CCN(C(c3cc(Br)n[nH]3)=O)C2)C1 C1(CN(C(C(N2CCOCC2)C)=O)C)COCCN1C(C1CCCN1C1CC1)=O C1(C#CC(=O)N2CCC(NC(=O)C(C(C)O)N(C)C)CC2C)(CC)CC1 c1(C(=O)NCCCC(=O)N(CCC(=O)OC)CCO)ccn2cncc2c1 CC1CN(C(C2(CNC(c3ccc(Br)cc3F)=O)CC2)=O)CC(C)O1 C(=O)(C1=NOC(C)(C)C1)N1C(C(=O)NCC2(CC)CCOC2)CCCC1 N1(C(c2c(C)cco2)=O)CCCCC1CCN(C)C(C1CC(F)(CO)C1)=O N1(C(c2c(C)[nH]cc2)=O)C2CCC1CN(C(c1cnc(C(C)C)n1C)=O)C2 c1(C(=O)NCC2CN(C)C2)ccn2ncc(Nc3ccn(C)c3)c2c1 N1(CC)CC2OCC(CN(CC(F)(F)F)C(C3CC(O)CN3)=O)C2C1 CC(C)C(O)CC(=O)N1CCC(NC(=O)CCCc2cccnc2)C1C C1CC(C)(C)CN=C(NC(CO)CC(C)(C)C)NC(C)=CC=CC=C1CCCC CC1(C(=O)NCC2(CCNC(=O)C(F)(F)c3csc(Cl)c3)CC2)CC=CCC1 c1(N2C(C)C(NC(=O)CC(C)Cc3ccccc3)CC2)cc2c(cn1)C(=O)CCC2 Cc1c(-c2cn(CC(CC(C)C)NC(c3cccc(F)c3)=O)nn2)ccn1C c1(OC)cc(OC)c2cc(CNC(=O)NCC(C3CC4(CCC4)C3)O)[nH]c2n1 C(c1cccc(F)c1)=C(C(=O)NCCN(C(c1c(CC)nc[nH]1)=O)C1CC1)F Cc1cnc(Cl)[nH]c1=NC1CN(C(c2cc(C)n(C(F)F)n2)=O)CC(C)(C)C1 C1(CCNC(Cc2n(C)ccc2)=O)CCN(C(=O)CCc2cncs2)CC1 Cc1cncc(C(=O)NCCN(CC(C)O)C(c2ncc(F)cn2)=O)c1Cl C(=O)(C1CCCc2c1ncn2C)N1CC(O)(CNC(c2n(CC)cc(Cl)c2)=O)C1 S(=O)(=O)(CC(=O)NCC1CCN(C(N)=O)C1)NC.c12ccc(o1)[nH]c2=O c1(C(=O)NC(CNC(C2CCN(CC)C2)=O)C(C)C)cncn(C)c1=O N1(C(c2ccc(SC)s2)=O)CC2(CCCCN2C(=O)COc2ccsn2)C1 Cc1nc(CC(=O)NC(C)(CNC(=O)CC(O)C2CCCC2)C2CC2)co1 C1(NC(C(CC)CC)=O)CC12CCN(C(=O)CCC1(C)CC1(F)F)C2 C1(NC(C(C)Cc2cnc[nH]2)=O)CN(C(=O)Cn2cncn2)C2(CCCC2)C1 N1(C(COC)=O)CCN(C(=O)C(C2CCCCCC2)O)CC1CC(F)(F)F C1(C(N2C(CC(=O)NCCN(C)CC)CCCC2)=O)CC2(CCCO2)C1 C1(NC(C(C)C)=O)CC(C)N(C(c2ccnc(Cn3[nH]cnc3=N)c2)=O)C1 C1(NC(C2CC(N(C)C)C2)=O)CCN(C(=O)CNC(c2ccsc2)=O)C1C N1(C(CC2ON=C(C)C2)=O)CC(C2(NC(c3n[nH]c(C)n3)=O)CC2)C1 C(=O)(C(C)(F)C(F)(F)F)NCCCC(C)NC(=O)CCc1ccccc1Br C1(NCCn2cc(C(=O)NC3C4CCC(F)C34)nn2)CCCC(C2CC2)C1 n1(CC(=O)NCc2c(C(=O)NC(C)CC3CC3)occ2)cnc(C#N)n1 C1(CCN(C(CCOCCC)=O)C)CCCCN1C(=O)C(=Cc1c[nH]cn1)F c1(OC)ccc(O)c(C(=O)NCc2nc(-c3ccc(N(C)C)cc3)no2)c1 n1(C(CC)C)nc(C(=O)NCC(C(C)C)NC(c2ccc(C)s2)=O)cc1C c1(C(N2CC(CC)N(C(=O)C(O)C(C)(C)C)CC2)=O)cc(N(C)C)cc(C#N)c1 N1(C(C=C(CC)CC)=O)CCCC(C2CCN(C(=O)Cn3cnc(=N)[nH]3)CC2)C1 C(=O)(C(F)(F)C(C)(C)O)NCC(C(C)(C)C)NC(C12CCC(N=[N+]=[N-])C1C2)=O C(=O)(C(O)CC(N)=O)N(C(C(N1CC(C)(COC)C1)=O)(C)C1CC1)C c1(CC(=O)N(CCNC(COCCC=C)=O)C(C)C)cn[nH]c1 C1(OC)CN(C(c2sccc2-c2cn[nH]c2)=O)CC1NC(=O)CCF CC1=C(C(=O)NCCN(C)C(c2c(OC(F)F)cccc2Cl)=O)CCCC1 N1(Cc2c(CC)ocn2)CC2(CC(NC(c3c(C)ncnc3C)=O)CO2)C1 c1(C(N(CC(O)CNC(=O)CSC2CCS(=O)(=O)C2)C)=O)cncc2c1CCC2 c1(CNC2C(c3ccc(C)c(Cl)c3)CCC2)cc(F)c(Br)cc1F c1(C2C(NC(c3n[nH]c(-c4cccc(C)c4)n3)=O)C2)ccc2c(c1)OCO2 C=C(F)C1(CC(N2CCC3CC23C(=O)NC(CO)C(C)(C)C)=O)CCC1 N1(C(Cc2cc(C)on2)=O)CCC(NC(=O)C(N2CCCC(C)C2)=O)C(CO)C1 c1(SC)ccc(Br)c(CNC(=O)NC(c2ccccc2)C(C)N(C)C)c1 C(C(CNC(C1(C)CC(NC(=O)CCC2CCOC2)C1)=O)CO)OC Cc1noc(C(C)C)c1C(=O)N(C)CC1(NC(C2(C(C)(C)O)CCC2)=O)CC1 c1(C(=O)NC2C(CNC(c3c(C)cno3)=O)C2)ccc(F)c(C(F)(F)F)c1 C(=O)(C1CCCc2cccnc21)N(C1CCN(c2cc(C(N)=O)nc(Cl)n2)C1)C Cc1nc(Cl)c(NC(C2CC2C(=O)NCc2ccc(F)cc2Cl)=O)c(Cl)n1 Nc1sc2c(c1C(N1CC3CC1(CNC(C1CSC1)=O)C3)=O)CCC2 Cc1cc(C(=O)NC2CCCC(NC(c3cccc(Br)c3Cl)=O)C2)cc(C)n1 c1(C(=O)NCC(C)N(C(CCCOC(C)=O)=O)C)cc(OC(F)(F)F)ccn1 c1(C(CC)=O)ccc(NNC(=O)C2CCCN(C(=O)C3CC3)C2)cc1 C(=O)(C1=NN(C)C(=O)CC1)NCCC1OCCN(C(C2C(C)C3CCC2C3)=O)C1 C1(C(=O)OCc2n(CC(C)C)c(-c3ccco3)nn2)SC2CCC1CC2=O CC(C)C(C)S(=O)(=O)N=S(=O)(N(C)C)N(C)CC1CC(F)(F)C1 C(C)(C(C(=O)N1CC(F)CC1C(=O)NCc1nccn1C)N(C)C)OC N1(C(CC2(C)CC2(F)Cl)=O)CCN(C(=O)COC2(C)CCCC2)C(CCO)C1 Cc1cc(C(N2CC(NC(C3CC4(C3)CC4F)=O)C(C(F)F)C2)=O)c(C)o1 C1(C(=O)O)(N(CCC=CBr)C2CC2)CCOC1 O=C1CCc2cccc(C(=O)NCCC3CCCN3C(=O)C(=O)NC3CC3)c2N1 c1(C(=O)NC2CCCC(NC(C3CSCCS3)=O)C2)ccc(O)cc1F c1(C(=O)NCC2CN(C(c3cc(C(C)(C)C)n[nH]3)=O)C2)c(C#N)cnn1C c1(C(=O)NC2CCN(C(c3c(N(C)C)coc3)=O)C2)ccc(O)nc1 C1(O)(CNC(=O)CCN2CCCC2=O)CCN(C(c2cn(CCO)nn2)=O)CC1 CN1C(=O)Cc2cc(C(=O)OCC3CCC(F)C3)ccc21 N1(C(CCC2C(C)(C)C2)=O)CCOC2(CCN(C(c3ncsc3C3CC3)=O)C2)C1 c1(N2CC(CNC(c3c(O)nc(C)c(C)n3)=O)OCC2)c([N+](=O)[O-])cnn1C C(=O)(C(CC(F)F)NC(=O)C(O)C1CCCC1)NCC1CCN(C)C1 CC(C)CC(C)CC(C)C(=O)Nc1cncc(-c2cn(CCOC3CC3)nn2)c1 C=C1CC(C)(C(=O)N(CCCCN(C)C(c2cnoc2C)=O)C)C1 c1(CN2CC(C(=O)Nc3cccc(OC)c3)CC(F)(F)C2)c(O)cc(Br)cc1F CC1CCCC(CC(=O)NCCCCn2cc(-c3ncccn3)nn2)C1 C1(CCC)CCC(O)(C(=O)NCC2(F)CN(C(c3cc(OC)n(C)n3)=O)C2)CC1 c1(OC)cccc(F)c1CC(=O)NCC(C(C)C)NC(c1ccc(=O)n(C)c1)=O C1(C(N2C(COC)CN(C(=O)C=C(C)C)CC2)=O)CCc2nc(O)[nH]c2C1 N1(C(CC2CCC(C#N)C2)=O)C2CCC1CC(C(=O)NC1CC3(CC3)C1)C2 C1(C(N(CC(C(=O)OC)C)C)=O)CCN(C(C2CC3CCCC3C2)=O)CC1C C1(C(N(C)Cc2cncn2C)=O)CCC2(CC2)N1C(=O)C#CC1CC1 c1(C(N(C(c2n3cc(C)sc3nc2)=O)C2CC2)=O)cnc2c(ccn2C)c1 CCCCCCC(=O)N(C)CC1CCN(C(c2cnc(C(C)=O)s2)=O)C1 C12(CNC(c3c[nH]nc3C(F)F)=O)CC1CN(C(C1CC13CC(O)C3)=O)C2 Cc1ccc(C(N2CC3CC(NC(C4C(C)C4C)=O)C3C2)=O)cc1C#N C(CC(C(=O)NCC(O)C(N)=O)NC(C)=O)=CC.C12(CC1)CCN2 c1(CCC)c(C(=O)N(CC(O)CNC(=O)Cc2ccnc(C)c2)C)cnn1CC S(=O)(=O)(c1c[nH]c2nc(F)ccc12)N1CCC2(CCCS(=O)(=O)C2)C1 C1(NC(c2nc(C)sc2)=O)CN(C(c2cccc(C#N)c2F)=O)CCC12CCC2 c1(CCNC2(c3n(CC(=C)C)nnn3)CC(C(N)=O)C2)ncc(F)cc1F Cc1cccnc1C(c1nnnn1CCCC1CC1)NC1CCCC(CO)C1 C#Cc1cc(C(N2CC(NC(=O)CN(C)C(C)C)C(C=C)C2)=O)ccc1C N1(C(C2C(CCC)C2)=O)CC2CC2(CNC(c2c(-c3cccs3)noc2C)=O)C1 Cc1ccccc1C=CC(=O)NCC(C1CC1)NC(=O)CSCC1CCCO1 C(=O)(C(CC(C)C)NC(=O)CNC(=O)CNC(=O)C(C)(C)C1CCC1)NC.C(C)(=O)N c1(CC)nc(C(C)NC(=O)C(=O)N(CC)Cc2csc(C)n2)cs1 c1(CC(=O)Nc2c(C(N3CCC(=C)CC3)=O)scc2)ccc(F)cc1Br C1(OC)CCC(C)(C(=O)NCC(C2(O)CN(C(c3sccc3C)=O)C2)(C)C)CC1 Cc1ccc(C2CC2)c(C(=O)NCC(C)(C)NC(=O)CC2CC(=O)NC(=O)C2)c1 C(C1=NOC2CC12)(c1nnnn1C1CCC1)NC1CCC(OCCOC)C1 CC(C)(C)C(C)(C)C(=O)N1CCCC(NC(=O)CN2CCCNC2=O)C1 Cn1ccc2cc(C(N3CCC(NC(=O)C(N)=O)C(C(N)=O)C3)=O)cnc12 CC1(C)CN(C(=O)C=CCC)CCC1CN(C(C1(C2CCC2)CC1)=O)C1CC1 N1(C(CCCc2ncc(C)o2)=O)CC(NC(c2sccc2C(F)F)=O)CC(C)C1 C#Cc1ccc(F)c(C(=O)NC2CCCC2NC(c2cncc3sccc23)=O)c1 C=CCC(F)(F)CNC(=O)CCCCNC(=O)CNc1ncccn1 N1(C(C(COC)C)=O)CCC(C2CN(C(=O)Cc3cc(C)ns3)C2)CC1 C#CCCCC(=O)NCC(C)(O)CNC(=O)C(C)(C)NS(C)(=O)=O c1(C(N2CCC(CC=C)(NC(C3CC(C)(O)C3)=O)C2)=O)ccc(OCC)cc1Cl c1(C(N2C(CCNC(CSCC)=O)COCC2)=O)nn(C)c2c1CCCC2 C1(C)(CNC(C2(SC)CCC2)=O)CCN(C(=O)Cc2nocc2C(C)C)C1 C(=O)(C1c2c[nH]nc2CN1C(=O)CN1CCC(OC)C1)N1CC2C(CC)(C2)C1 C(CCCOC)(C(=O)NC(CO)C(C)CCC)NC(CSCCCC)=O C(=O)(C(C(C)C)C(C)C)NC1(CNC(c2cccc(COC)c2)=O)CC1 c12cnc(cn1)[nH]c2=O.C1(N(C)C2CC2)CN(C(C2(Cl)CC2C(=O)NC2CC2)=O)C1 CC(C)CC(C)CN=c1nc(N(CCC(F)(F)F)C)c2c([nH]1)COC2 CCC(CNC(=O)C(=O)Nc1cccnc1-n1cncn1)C(C)C n1(CC#C)cc(C(=O)NCC=CCNC(c2cc(C(F)F)cs2)=O)nn1 Cc1ccccc1CCC(=O)NCC1(C(N)=O)CN(C(=O)C(F)F)C1 N1(C(C(C(C)C)S)=O)CCOC2(CCCN(C(=O)Cn3cc(C4CC4)cn3)C2)C1 C(C(C)(COC)C(=O)N(CC(=O)O)CCc1cn(Cc2nc(C)cs2)nn1)OC N1(C(CCC)=O)CCN(Cc2ccccc2)CC1.C12CCC(CC1)NC2=O C(=O)(CC(CNS(C)(=O)=O)C(F)F)NCC1(NC(C(C=C)C)=O)CC1 N1(C(C(C(=O)N2CCCC2c2cc(Br)cn2C)OC)=O)CCc2ccccc21 N1(C(C2C=CCN(C(C(CC)CC)=O)C2)=O)CCC2(CC(F)C2)C1 C1(C(N(C)CCNC(c2cn(C(C)(C)C)cn2)=O)=O)CCCCC1O C1(CCNC(C=CC=CC)=O)C(C)CCCN1C(c1cc(CSC)on1)=O Cc1cc(C(=O)NCC2(C)CCCN2C(C2CCC2(C)C)=O)c(C)n1C N1(C(c2cccc(Br)c2C)C(=O)NCCCCCC)CCc2oc(C)nc2C1 C=CC1(C(=O)NCCCOCCN(C(=O)C(F)C(F)(F)F)C)CCCCC1 C(CCN(C)C)(C(=O)NC1CCN(C)C1C)NC(C1C(OC)CCC1)=O C(c1ccncc1)=C(C)C(=O)NCC(C)NC(c1ccc(C)n1C)=O C1(CC)CCCC1(C)C(=O)N(CC(C)(C)CNC(c1ccc(C(F)F)cc1)=O)C c1(C(=O)NCC(c2ccsc2)O)ccc(C2CC2(F)F)cc1 c1(C(=O)NC2(C)CCCOC2)coc2c1CN(C(=O)C(C)(C)NC(C)(C)O)C2 N1(C(c2nnn(C)n2)=O)CCN(C(=O)CCc2ccccc2Cl)CC1CCO Fc1ncccc1C1(NCC2CCC(C(F)(F)F)O2)CCOCC1 C(C)(N=c1nc(Cl)[nH]c(C)c1C#N)C1N(C(C2=CC(C)(CC)C2)=O)CCCC1 c1(CN2CC(C3(NC(C(CC)NC(C)=O)=O)CC3)C2)cn(C)c2ccccc12 c1(C(=O)NC23CN(C(CN(CC)CC)=O)C(CC2)C3)cc(C)c(F)cc1F CCCCCC(O)C(C)C(=O)NC(C1CCN(C(=O)CCC)CC1)C c1(C(=O)NC(Cn2cc(-c3[n+]([O-])ccc(OC)c3)nn2)=O)ccc2nsnc2c1 c1(C(N(C(C(=O)N(C(c2cnnn2C)C)C)C)C)=O)ccc(C2CC2)cc1 c1(SC)ccc(Cl)c(C(=O)NCC2(CNC(C3(C#N)CC3)=O)CC2(F)F)c1 N1(C(=O)OC)C(CNC(C)=O)CC2COCC12.N(C1CC1)CC C(=O)(CCCC(F)F)NC1CCN(C(C2CN(c3cn(C)nc3)C(=O)C2)=O)CC1 c1(C2OCCN(C(C(c3ccc(F)c(Br)c3)N)=O)C2)ccc(Br)cc1F N1(C(C23C(C)(C)OC(CO)(C2)C3)=O)CCc2nc(CNC(=O)COC3CC3)sc2C1 N1(C(Cc2cc(C)ncc2)=O)CCC(O)(C(=O)N(C)CC2CCOC2)CC1 c1(OC)cc(Br)cc(NC(N2CCN(C3CC3)CC2)=O)c1OC C1(C(N(CC(C)NC(c2cc3[nH]ccc3s2)=O)C)=O)CC2(CCOC2)C1 C1(CC)(CC)NC(=O)N(CC(=O)NCC2CN(C(C3CC3C)=O)C(C)(C)C2)C1=O Cc1[nH]nc2ccc(C(N3CC(C)(NC(=O)CC(C4CC4)C4CC4)C3)=O)cc12 N1(C(Cc2cn(C)nc2)=O)C2CCCC1CN(C(c1ccnc3ccnn13)=O)C2 n1(CC)ncc(C(=O)NCC2(NC(=O)C(C)CC3CCCC3)CCCCC2)c1Cl c1(C(=O)NCC(CN(C(CC(C)N(C)C)=O)C)O)cc(F)c(Cl)cc1F c1(C(=O)NCc2csc(C)c2C)coc2c1CN(C(C1CCC(C)O1)=O)C2 N1(C(=O)Nc2ccc(-c3cncnc3)cc2)CCc2cccc(NC(=O)OC)c21 N1(C(CCCCC)=O)CC2CCCC2(CNC(=O)C2=COCCC2)C1 CCC(CC)CC(F)C(=O)NC12CC(NC(c3cc(C(C)C)no3)=O)(C1)C2 c1(C(=O)NCC(CC(=O)N2C(CC(C)C)CCC2)C)cccc([N+](=O)[O-])c1 C(=O)(C(C)(Cl)Cl)NC1(C(=O)NCC2(C(=O)NC)CCC2)CC1 C1(NC(C(N)=O)=O)CN(C(=O)C(c2cccc(Cl)c2)N2CCCC2)CC1O.C1CN1 N1(C(c2ccc(OCC)cc2)=O)CCCN(C(c2ccon2)=O)C(CO)C1 n1(CC(=O)NC(C2CCCC2)CNC(C(C)OC(C)=O)=O)cnc2c1CCCC2 c1(C(N2CC(NC(C3CCC(OC)C3)=O)C2)=O)c[nH]c(C)c(Br)c1=O N1(C(C(CO)N(C)C)=O)CC(C(=O)NC2Cc3ccccc3C2)CC12CCC2 C1(CNC(C2(C=C)CC2)=O)CN(C(=O)CCCC(C)(F)F)C2(CCOCC2)C1 N1(C(C=COCC)=O)C2CCC1CC(CNC(=O)CC1COC(C)(C)CO1)C2 CCCCC(C(C(=O)O)Nc1nc(C(C)C)no1)NC(=O)NCc1ccc(C)cc1 CCCCCC(CC)C(=O)NCC1(C(=O)NC2(COC)CCCCCC2)CCC1 c1(CN(CC(CNC(c2ccon2)=O)OC)C(=O)C(F)C2CCC2)cccc(Cl)c1 CC1CC(NC(C2(CF)CC3(CCC3)C2)=O)CN(C(c2nn[nH]c2Cl)=O)C1 C1(NC(N(C)Cc2ccoc2)=O)CCSC(c2cnccn2)C1 c1(C(N2CCN(CC(C)NC(=O)C(N)=O)CC2)=O)ccnc2c1CC(=O)N2 c1(C(N2CCC(N(C(C3CC3F)=O)CC)C2)=O)cc2cc(Br)cnc2s1 C1(OCC)CS(=O)(=O)N1C1CCCS1.c1(CCN(C)C)cnn(C)c1 C1(CC(=O)N(CC(=O)NCc2ccncc2)C)CCCC(=O)N1 c1(SC)ccc(NC(c2ccccc2NCC(C)NC(=O)C(O)C(C)C)=O)cc1 c1(OC)ccc(Cl)c(C(=O)NCC(O)CN(C(=O)Cn2cncn2)C)c1 c1(C(N2C(C)(CNC(C3(OCC)CC3)=O)CCC2)=O)cc(OC)c(O)c(CC)c1 CCCC(CC(=O)N1CCCC1c1nnc(C)o1)NC(=O)OC C1(n2cc(C(CC)(C)O)nn2)CON(C(=O)c2cc(Br)ccc2OC)C1 Cc1ccc(C(N2CCN(CC(N3CCOC(C(N)=O)C3)=O)CC2)=O)cn1 CC(C)(C)CCC(=O)NC1CCCC(Nc2cc(O)nc(O)n2)C1 C1(F)(CN)CCN(CC(=O)Nc2cccc(OC(F)(F)F)c2)CC1 C(=O)(C1=CCCSC1)CC.N1(C(c2cc(COC)on2)=O)CCC(F)(c2cn(C)nn2)C1 CC1CC2CN(C(=O)C3=CC(C)(C)C3)CC12.C1(C2CCNC2)CCCCN1CCC c12csc(n1)N(CC1CCCO1)N(CC)C(=O)C2.C#CC(C)C c1(CN=C(NC(C#C)CC2CCC2)NC(C)CC)cc(OC)c(OC)cc1Br c1(C(=O)NCCC(C)NC(c2ccnc(C(F)(F)F)c2)=O)ccn2nnnc2c1 N1(C(c2sc(C)c(Br)c2C)=O)CC2CN(C)C(C(=O)O)C2C1 O=C(CCCc1ncco1)OC1CN(c2ncc(Br)s2)C1 C1(C(=O)NC2C(CNC(c3c(C)[nH]cc3)=O)CC2)CCc2c(n[nH]c2C)C1 O=C(CCCc1cccs1)NCCNc1ccccn1 N1(C(C2(CC(=O)OC)CCCC2)=O)CC(n2cc(CCN)nn2)C(C)C1 c1(C(N2CC(F)(C(N3CCOC4(CC4)C3)=O)C2)=O)cc(F)c2cc[nH]c2c1 N1(C(C(CC(N)=O)O)=O)CC(O)(C2(CNC(=O)CCn3ccnn3)CC2)C1 CC(CC(=O)NC1CC2CC(C1)N(C(=O)CSc1cnn(C)c1)C2)CC(F)(F)F c1(C(N(C2CC3CC2N(C(C2CC2C2CCC2)=O)C3)C)=O)cc(F)cc(Cl)c1 N1(C(C(C)OC2CCCC2)=O)CCC(CNC(c2ccnn2C(C)(C)C)=O)CC1 c1(CNC(=O)NC2(C(F)F)CC2)ccc(=O)n(CC(N2CCCC2)=O)c1 Cc1ccc(F)c(C(=O)NC2(C)CCCCC2NC(=O)C(C)N=[N+]=[N-])n1 CN(C)NC(=O)CCC(=O)N1CC2CC2(CNC(C2CCC(C3CC3)CC2)=O)C1 c1(C(C2CSCCO2)NCc2n(CC)nnn2)ccc(C2(OC)CC2)cc1 CCCC(O)CC(=O)NCC(c1cccc(Cl)c1)NC(c1nnn(CC)n1)=O CC(C)CC(C#N)C(=O)N1CC(NC(=O)CC23COCC(C2)C3)C2(CC2)C1 C1(C(=O)NC(C(CO)NC(C(C)OCCOC)=O)C)CCN(OC)CC1 C=CC(C)(CCOC)C(=O)NCCN(C(=O)COCc1nnc(C)s1)CCC CC1c2c[nH]nc2CCC1C(=O)NCC1CCN(C(c2csc(CO)n2)=O)CC1 C(=O)(C(C)(C)C(C)(F)F)NC12OCC(NC(CCCCCCCCC)=O)C(C1)C2 C(=O)(C(O)C(C)(C)C)NC1CC(NC(Cc2c(C)nc(C3CCC3)s2)=O)C1 C1(CCC2N(C(CCOC(C)=O)=O)CCC2)CCN(C(C2(C)CCCS2)=O)CC1 CC(N=c1ccc([N+](=O)[O-])c(O)[nH]1)C1CN(C(=O)CCc2cnccn2)CCO1 c1(C(=O)NC(C(C(C)C)NC(c2c(C)ncnc2C)=O)C)cc2cccn2cn1 CC1CC(NC(=O)Cc2nc[nH]n2)CCN1C(c1ccc(C2(C)CC2)cc1)=O C1(CC)CN(C(c2ccsc2)=O)CCC1NC(c1cnc(C)nc1)=O c1(CC(=O)NC2CC3CC(NC(C(CC)C)=O)C3C2)cc(F)c(F)cc1F Cn1cc(C(N2CC3CC(N(C)C(C4CC4F)=O)C2C3)=O)n2cncc2c1=O CCC(CC(F)(F)F)C(=O)NCC(C)N(C(=O)CC(C(F)(F)F)OC)CC c1(NC(CC(C(F)F)NC(C(C2CC2)OCC)=O)=O)ccc(O)c(=O)cc1 N1(C(C2C=CCN2C(=O)Cc2ccns2)=O)Cc2ncsc2C1 c1(OC)nc(C)ccc1C(N1CCCN(C(=O)C(C2CCCCC2)C)CC1)=O C1(NC(C2CCC(NC(c3ccc(C)nc3)=O)C2)=O)CCCCC1C1CC1 c1(C(N2CCC(CCF)(NC(=O)COC3CC3)C2)=O)cn2ccc(CO)cc2n1 N1(C(c2[nH]cc(C#N)c2)=O)C2CCCC1CN(C(C1CCCS1(=O)=O)=O)CC2 C(=O)(C(O)CC(C)C)NC(C(=O)NCC1CCC(=C)CC1)C1CC1 N1(C(c2cn(C)nc2)=O)CCC(C)(C)C(C(=O)NCc2cnc(O)c(F)c2)C1 c1(C(=O)NCC2CCCN(C(CC)C)C2)ccccc1[N+](=O)[O-] C1(COC)(NC(=O)C(n2ccnc2C)C)CN(C(=O)CN(C)C(C)C)C1 c1(C(C)=O)ccc(C(=O)NC2CC(NC(=O)CC3(C#N)CC3)C2)nn1 c1(C(=O)NC2CC(CN(C)C)C2)ccc(-n2ccnc2)cc1 c1(C(=O)NCC23C(CN(C(C(C(=C)C)(C)C)=O)C2)CC3)cc2nc(Cl)ccc2s1 Cc1nc(C#N)c(C(=O)OC(C)(C)C)o1.c12ncc(cn1)CCOCCCN2 c1(CC(=O)NC2CN(C(c3cnc(O)s3)=O)CC23CC3)ccc(Cl)c(Cl)c1 C1(NC(CNC(=O)OCC)=O)(CO)CCN(C(c2cccnc2C(C)(F)F)=O)C1 CC(C(=O)N1CC=CC1(C)C(N1CCCN(C2CC2)CC1)=O)S(N)(=O)=O C1(NC(C2(CC#C)CC2)=O)CC2(C(=O)NCCC3CCC(C)CC3)COC1C2 c1(COC)cccnc1C(N1CC2CC2(NC(=O)CC23CCCC2C3)C1)=O C1(C(=O)NC2(CNC(CCN(C)CCO)=O)CC2)CC2(C1)CC21CCC1 CC1CN(C(c2cnc(O)n2C)=O)CC1NC(c1cnns1)=O C(CCNC(C1(CC2CC2)CCC1)=O)(C(C)C)NC(C(C)NC(C)=O)=O C(=O)(C1=C(Cl)CCC1)N1CC(C(C)NC(=O)C(Cl)=CCl)OCC1 N1(C(C(C)NC(=O)OC(C)(C)C)=O)CCCC(O)(C(=O)NCC2(CO)CC2)CC1 N1(C(CCC#C)=O)CCC(C)C(NC(c2ccc(NCCO)cc2)=O)C1 c1(-c2cc(OCC)c(OC)cc2)ccc2cc(NCC(=O)OC(C)C)ncc2c1 N1(C(C2CN(C)C(=O)N2)=O)CC(CNC(c2cccc(F)c2F)=O)C2(CCC2)C1 c1(CCCC(=O)NCC(C2CCCN(C(CC#C)=O)C2)(C)O)cc(F)ccc1F N1(C(COCCCCC)=O)CCC(C(C)(C)C)(CNC(c2cn(CC)nn2)=O)C1 C(=O)(C(C)(C)CC(C)C)NCC1(F)CCC(NC(C2C(C(=O)OCC)CC2)=O)C1 N1(C(C2(C)CSC2)=O)CC2CC(NC(c3cccnc3N)=O)C1C2 C(=O)(CCP(C)(C)=O)NCCO.C1(CCC2N(C)CCC2)CCN(C(=O)CO)CC1 c1(C(N(CC(=O)NCC(CC)O)C(C)C)=O)cc(C(C)=O)c[nH]1 C1(CNC(CCc2ccc(OC)nc2)=O)CN(C(=O)CCS(C)=O)CCC1(F)F C1(NC(c2c(CC)con2)=O)CC(F)CN(C(=O)C(Br)=C(C)C)C1 C1(C(=O)NC2(C)CCCN(C(c3n(CC)nnc3)=O)C2)Cc2nc(C)cn2C1 C(CCCC(C)NC(=O)C(CCC)Oc1ccccc1)NC(CCC#C)=O CC1CC(c2ccccc2)N(C(=O)C(=O)NC2CC2C2CC2C)C1 N1(C(C(CC)N(C)C)=O)CC2CCN(C(c3cn[nH]c3)=O)C2C1 C[S+](C)CCC(O)C(=O)NCC1C2CN(C(=O)C3=CCSC3)CC12 c1(CCC(N2CCC(N(C(c3c(CC)ncs3)=O)C)C2)=O)ccc(OC)cc1 CCC(C(=O)NCC(C)(CC)NC(=O)CC1CCCO1)Oc1ccccc1 C1(C(N2C(CC)CC(O)C2)=O)CC(F)CCN1C(=O)CCN1CCCC1 C(=O)(N1CCC(C(N2CCC(CC(C)(C)C)C2)=O)O1)c1c(C)scn1 N1(C(CC(C#C)(C)C)=O)CCOC2(C1)CN(C(C1CCC(=C)CC1)=O)C2 C1(CNC(COC2CCCC(C)C2)=O)N(C(=O)CCC2CC2)CCCC1(C)C c1(SCC(=O)NCCC2(NC(CCCC#C)=O)CC2)ccc(F)c(F)c1 N1(C(c2c(C)occ2)=O)Cc2nccn2CC(NC(C2Cc3nccn3C2)=O)C1 C#CC1(C(=O)Nc2cccc(C)c2Br)CCN(C(=O)CN(C)CCOC)CC1 c1(CC(N2CCC(CNC(c3ccc(C)o3)=O)C(C)C2)=O)ccc2nonc2c1 c1(CN2C(C(N3CCOCC3C)=O)CC(=C)C2)c(F)cc(C)cc1F C1(N(C(C(C)SC(F)(F)F)=O)C)CN(C(C2CCN(CC3CC3)CC2)=O)CC1O C1(C(N2CC(CN(C(C3(SC)CCC3)=O)C)C2)=O)OCCC1CCc1ccccc1 c1(OC)nccc2c1CN(C1CC(CS(N)(=O)=O)C1)CC2 CC(C)(Cc1ccccc1)C(=O)N1CCC(CNC(c2nnncc2N)=O)CC1 c1(C(=O)NC2CCC(NC(CC3(OC)CC3)=O)C2)cccc(-c2ccncc2)c1 c1(CC(=O)NCC(CCC)NC(c2ccccc2OC)=O)c(C)cnn1C N1(C(COCCC#N)=O)CCc2ccc(C(=O)NCC3CCCCO3)nc2C1 N1(C(C2(N3CCCCC3)CCN(C)C2)=O)CCOC2(CCC2)C1 c1(C(=O)NC2C(CNC(CC)=O)CCC2)nnn(C)c1N.N12CCC(C1)C2=O c1(C(=O)NC(C2N(C(c3cc(SC)oc3C)=O)CCCC2)C)ccnc(C)c1C c1(C(N2CCC(OCCNC(c3ccc(F)c(Cl)c3)=O)C2)=O)ncnc(O)c1F N1(C(C(C(C)C)O)=O)CCN(C(c2cncc(N(C)C)n2)=O)CC1c1ccncc1 c1(-c2cc(C(N(CC)Cc3cccc(F)c3CC)=O)c(C)o2)cccc([N+](=O)[O-])c1 C(=O)(C(O)C(C)(C)C)N1CC(CC(C)NC(C=Cc2nnc(C(C)C)o2)=O)C1 C1(NC(CC(C)OC)=O)COC2(CCN(C(C3(CO)COC3)=O)CC2)C1 C(=O)(C1CCc2snnc21)N1CCN(C(Cc2nc(C)oc2)=O)CC1CCO Cc1nn(C)c(C)c1OCC(=O)NCC1(F)CC(NC(=O)CCSCC(C)C)C1 c1(CC(=O)NCCN(C(c2c(CC)c[nH]c2)=O)C)cccc(N2CCCC2=O)c1 Cc1cc(C(N2CCCC2CCCNC(C2CC3(CC3)CO2)=O)=O)ccn1 c1(CCCC(=O)NC2CCN(C(=O)C=Cc3nccs3)C2)cc(F)ccc1F N1(C(C(=O)NC2CCCCC2)C2CCCC2)C2CCC(O)C1CCC2O S(=O)(=O)(c1cc(Cl)sc1C(=O)NC1CC(C)N(C(=O)CCCC2CCC2)C1)NC N1(c2sc(C(=O)OC)c(Cl)n2)CC2CC(NC(=O)CCCCC(C)C)CC2C1 c1(C(=O)NCC2CN(C(c3cc(OC)ns3)=O)C(C)C2)cnc(O)c(C)c1 c1(C(=O)NC2CCN(C(c3cnc(OCC)s3)=O)C2)ccc(Cl)cc1[N+](=O)[O-] c1(C(N2C(CN(C)C(C3CCC=CCCC3)=O)CCC2)=O)cnn2ccccc12 CCCCCC(O)C(=O)NCC1(C)CCN(C(c2nnsc2C)=O)C1 c1(OC)cc(C(N2CCC3(NC(=O)CSC)CCCC23)=O)cc(Br)c1OC C1(C(N2CCC(C(C)(C)NC(c3cc(OC)no3)=O)C2)=O)CCCCC(F)(F)C1 N1(C(CCCC(=O)NCC)=O)CC2=C(C1)CN(C(=O)C(C)(O)CC(C)C)C2 C1(C(=O)NCc2c(C)noc2C)CC(C)CN(C(=O)CSc2ccccn2)C1 c1(CN(C)C(=O)OCCNC(=O)CS(N)(=O)=O)ccc(-n2ccnn2)cc1 C12(CC)CC1CN(C(=O)Nc1c(NC3CC3)onc1)C2 c1(C(=O)NC(CC(C)NC(c2c(CC)c(C)sc2)=O)C)cccc([N+](=O)[O-])c1 C(=O)(C1=CCCC1C)N(CCC(=O)NCC1(COC)CC1)CCCN(C)C C1(C(=O)NC2(CNC(c3c(C)n(C(C)C)cc3)=O)CCOC2)COCC(C)(C)O1 C(=O)(C(O)CC[S+](C)C)N(C(C)C)CCN(C)C(C1(C#N)CCSCC1)=O CP(C)(=O)C1CCCCC1C(=O)NC1CC(C)(NC(=O)Cc2cncnc2O)C1 Cc1cnn(C)c1CC(=O)NC1CC(C)(CNC(=O)CC(C)n2cccn2)C1 c1(OC)ccc(C(=O)NC2CC2NC(=O)CC2(C)CCCC2)c(Br)c1 N1(C(CC(CC)C(C)(C)C)=O)CCC2(CC1)CN(C(=O)CCC(N)=O)CC2CO c1(Nc2nccc(C)n2)cc(OC(F)F)c(N)cc1F N1(C(C2N(CCC)CCC2)=O)CCC(C(=O)N(C)Cc2c(C)noc2C)=C(F)C1 C1(CNC(CC=CC=C)=O)CCC2(CCC2)CN1C(C1COCCN1C)=O CCC(F)(C(=O)OC)C(=O)N1CC(C2(NC(=O)CCc3cncs3)CC2)C1 c1(C(=O)NCC(C)N(C(=O)C(C2CCOCC2)C)CC)cc2cccnc2[nH]1 C=CC(C)(C)CC(=O)NC1CC(OC)CN(C(=O)CN2CCCC2CO)C1 c1(C(N2C(CC)C(NC(=O)Cc3ccco3)CCC2)=O)cnc2sccc2c1 c1(OCC(C)C)ccc2cc(C(=O)NC(C)C(C)NC(=O)CC(C)SC)[nH]c2c1 N1(C(c2cc(COC)no2)=O)CC(NC(C2CCS2(=O)=O)=O)CCC1C C1(NC(C=CC2(C)COC2)=O)CCCCN(C(C2CC(O)C2)=O)C1 c1(-c2nc(-c3c(OC)cccc3)on2)ccc2sc(C(F)(F)F)nc2c1 C1(C(=O)NC(CO)C(C)NC(C2C=C(C)CS2)=O)(OC)CCOC1 Cc1cc(CC(=O)NCC(CNC(=O)C(C)Cc2cscn2)CO)n(C)n1 N1(C(c2nnc(C(C)C)o2)C)CCC2(CCN(C(=O)CC3CCS(=O)(=O)C3)C2)C1 c1(NC2CC(C)N(C(C3CCCOC3)=O)CC2)ncnc2sccc12 C(=O)(N=c1[nH]sc2ncccc12)C1C2COCC12.CC12CCCN(C1)C2=O O=C(CCCCC(F)F)NCCC1CCCCN1C(c1cc2sccc2cn1)=O N1(C(CNS(CC)(=O)=O)=O)CCOCC1C(N1CCCCC1C(N)=O)=O C1(C(=O)NCC2CCC(=O)NC2)(CC)CCN(C(=O)CCn2ccc(C)n2)C1 C1(CCC)CC1N=c1[nH]c(N(CC(C)(C)OCCOC)C)nc2c1CC(C)CC2 C1(NC(CCSc2nc(C)[nH]n2)=O)CCN(C(=O)CC=C(Cl)Cl)CC12CCC2 N1(C(C(CO)N(C)C)=O)CC2CCCC(CNC(=O)C3=C(Cl)CC3)C2C1 N1(C(C(C)SCCCC)=O)CC(C2CCCCN(C(=O)COCC3CCC3)C2)C1 Cn1ncc(C(=O)NCC(F)(F)Oc2ccc(F)cc2)c1N CC1(CNC(C2(CF)COC2)=O)CC(F)(F)CN1C(=O)Cc1nc([N+](=O)[O-])n[nH]1 c1(C(N(CCNC(C2CCC(C)S2)=O)C2CC2)=O)ccc(N)c2c1CCCC2 CCCCC(O)C(=O)N1CCC(CNC(=O)CCCc2ccc(C#N)cc2)CC1 c1(C(=O)NC(C(=O)N(CCC2CC2)CC)CO)ccc(C#N)[nH]1 C1(c2nnnn2CC(F)F)(NCCC(=O)NC)CN(C)CC1C N1(C(C(C)NC(CC)(C)C)=O)CC(NC(=O)CC2(C)CCC2)CC2(CCC2)C1 C(=O)(CC(C)CC(C)(C)C)N1CC(C)N(C(c2coc(CO)c2)=O)CC1 C1(C(=O)NC(C2CCN(C(CC(C)(F)F)=O)CC2)(C)C)CCC12CCOCC2 C=C(C)C(CC(=O)N(C)CC=CC(=O)Nc1cc(C)ccc1CO)OCC c1(CN(CCNC(C2C3CN(CC(F)(F)F)CC23)=O)CC)cc(F)c(F)cc1F CC(=O)CCCC(=O)N1CC(F)CC1CC(N1CCC(CN(C)C)CC1)=O c1(C(=O)NCc2cccc(CN(C(CSCC#C)=O)C)c2)cccc(C#N)c1C C(C(C)(C)C(=O)NCC(C)(CO)NC(c1coc(C(F)(F)F)c1)=O)SC C(=O)(CCN1C(=O)NCc2ccccc21)NC(C)CN(C(=O)C1=CCSC1)C N1(C(Cc2cc(C)[nH]n2)=O)CCC(C(=O)NC(c2nc[nH]n2)CO)C1(C)C N1(C(C(C)(C)CF)=O)CCCCC(C2CN(C(c3ccc4ccsc4c3)=O)C2)C1 N1(C(C2CC(OCC)C2)=O)CC=C(CNC(=O)CCc2nc(C)no2)CC1 CCC(C)(COC)C(=O)N1CCCC(CN(C)C(c2cc(C3CC3)nn2C)=O)C1 c1(OC)ccc2nccc(C(N3CC4C(N(C)C(c5cc[nH]n5)=O)C4C3)=O)c2c1 C(=O)(CCCCC#N)N1C(CN(C(CSc2n(C)nnn2)=O)C2CC2)CCC1 c1(N2CCC(F)(F)C2)nc2c(c(=NC3COc4cccc(Cl)c43)[nH]1)CSC2 N1(C(CC2(C=C)CC2)=O)CC2CC2(CNC(c2ccnc(C(F)F)c2)=O)C1 CN1CC2(CCCN(C(=O)C(N3CCC4C(C3)C4(F)F)=O)C2)CC1=O c1(C(=O)NC2(C)CCCN(C(=O)COC3CCC3)C2)cccc2c1OCCN2 C1(C(N2CC(O)(CN(C(c3c(C)scn3)=O)C)C2)=O)CCC2(CCC2)O1 C1(SC)CN(C(=O)CC2(CO)CCC2)CC1NC(C1CCC1C)=O Cc1ccc(F)c(C(N2CCCC(CN(C(=O)CC3CCCCN3C)C)C2)=O)c1 N1(Cc2ncc(C)cn2)CCC(CNC(C2(c3ccccc3O)CC2)=O)C(C)C1 C=CC(O)C(=O)N(CCCNC(=O)Cn1[nH]cnc1=N)Cc1cccnc1 N1(C(C(C)(C)NC(C2CC(=C)C2)=O)=O)CCC(O)(CF)CC1 Cc1nnc(CNC(c2ccn(CCF)n2)c2nnnn2CC2CCCO2)o1 C1(C(=O)NC2(CNC(CS(C)(C)OC(F)F)=O)CCC2)CCCC12CC2 N1(C(C)C)C(=O)COCC1C(=O)NC1CC(F)(CNC(C2CC=CC2)=O)C1 c1(C(=O)NC2(CCCNC(CC(C=C)C)=O)CC2)ccc(OC)nc1Cl C(C)(CCC(C)(C)C)NC(C(CCOCC)NC(C12CCC(C1)C2(C)C)=O)=O C1(CNC(C=C(CC)CC)=O)CCC2CN(C(c3cccc4[nH]ncc34)=O)CC12 C(=O)(C(F)(F)CCc1ccccc1)NCC(CC)NC(c1nccc(C)c1O)=O Nc1c(F)ccc(Cl)c1C(=O)NCC1(CCNC(C2(F)CC=CCC2)=O)CC1 CC(C)CC(C(=O)NC1CN(C(C2(C)CCC(C)CC2)=O)C1)n1ccc(C2CC2)n1 C(=O)(C(C)(C)CC(F)F)N1CC(OC)C(NC(c2cncc3c2CCC3)=O)C1 O=C(N=c1nc2cc(Cl)ccn2[nH]1)N1CCC(c2ccc(O)cc2)C1 c1(OC)ccc(C(N2CCC(N(C(=O)CCOCC3CCCC3)C)C2)=O)c(F)c1 Cc1cc(C)c(C(=O)NC2CCCC2NC(c2ccncc2Cl)=O)[nH]1 CCCCC(CC)C(=O)N1CCN(C(C2(F)CCCC2)=O)C(COCC)C1 C1(C(=O)NC2CCCCCN(C(CC=C)=O)C2)CC(=O)c2cc(Cl)ccc2O1 N1(C(c2c(C)occ2C(F)(F)F)=O)CCC(C2CCCN(C(=O)C3CC3)C2)CC1 c1(C(=O)OC(CC#C)C)ccccc1 c1(N(CC#CCOC)C)nn(CC)cc1Br c1(CC(=O)NC2CC(NC3CC3)C2)nc(C(=O)NC(=O)C(C#N)C2CCCO2)cs1 C1(C(=O)NCCCCCn2cc(CN(C)C)nn2)(CCO)CCOCC1 c1(C(N2CC(CC(C)NC(=O)CC3CCC(=O)NC3)C2)=O)cccnc1S c1(NC(C(c2csc(C(C)(C)C)c2)N(C)CC2(C)CCCC2)=O)ccccc1Cl C12(C(=O)OCC)CCC(NC(=O)Nc3cc4n(n3)CC(F)C4)(CC1)CC2 c1(CC)cccc(C(=O)NCC(C2CC2)N(C(=O)C(C)c2cccs2)C)c1F c1(C(=O)NCC2(COC)CN(C(c3cc4sccc4s3)=O)C2)cncn(C)c1=O O(C1CCc2ccccc21)C(c1cc(F)cc2c1CCC2)=O N1(C(c2n(CCC)ncc2)=O)CCC(C(=O)Nc2cc(C)cc(O)c2)C(C)(C)C1 c1(C(N2C(CNC(C3CCCO3)=O)CC(OC)C2)=O)cc2c(C)ccc(F)c2[nH]1 CCC(C)CCCCC(=O)NC1C=CC(C2CCCN2C(=O)Nc2nccs2)C1 c1(CNC(C2C(COC)C2)=O)ccc(CNC(=O)C(F)(F)c2cnnn2C)cc1 c1(C(N(CC(C)N(C(C=CC)=O)C)C)=O)ccc(C)c(OC)c1 CC1C(C(=O)NCC(=O)N(C)O)CCN1C(=O)CCCCC1CC1 c1(OC)cnc(C(=O)NC2CCOCC2C(N2CCC(CC(N)=O)CC2)=O)cn1 c1(C(=O)NCC(C)(CO)NC(C2CCCS2)=O)nc2c(s1)COCC2 c1(C(N(C(CC)C)CC(=O)OC)C)ccc(NC2CCOCC2)cc1 N1(C(c2c(C)cncc2C)=O)CCC2CC1CN(C(=O)CN(C)C)C2.O(N)CC c1(C(=O)NC2C3(CC(NC(C(CC)=CCCC)=O)C3)C2)cc2n(n1)CCCN2 c1(CC(N2CC(C(=O)NC(CCOC)COC)(OC)C2)=O)cccc(C)c1C c1(C(N2CCC3CN(S(=O)(=O)c4ccncc4)CC23)=O)ccc(Br)c(F)c1F C(N=c1cc[nH]c(C2CC2)n1)c1c(CNC(C(n2cc(CN)nn2)C)=O)cccc1 n1(CC(CC)O)ccc(C(=O)OC)n1.C12(n3cc(CC(C)O)nn3)CN(C1)C2=O C(=O)(C(C)C(C)NC(=O)C(c1ccco1)NC(c1cc(Cl)n(C)n1)=O)OC c1(OC)cccc(C(=O)O)c1NC(c1cnc(C2CC2)nc1C)=O c1(C(=O)NC2(CCNC(CC(CCC)O)=O)CCCC2)cc2cnccc2o1 N1(C(c2cc(C)nnc2O)=O)CCC2(CCCN2C(c2c(C)csc2Cl)=O)C1 N1(C(C(CC)CO)=O)CCN(C(c2ccccn2)=O)CC(O)C1 c1(OC)cccnc1C(O)C(=O)NC1CC1c1cn(-c2ccc(Cl)cc2)nn1 CC1CN(C(=O)CC(C)F)CC2(CCN(C(c3ccnnc3O)=O)CC2)O1 Cc1cc(NC(C2=CC=C(C)C2)=O)ccc1NC(C1CC12CCOC2)=O CC1CCCN(C(=O)Cc2cccc(OC(F)F)c2)C1CNC(=O)COCCF c1(CNC(C(CNC(=O)COC2(C)CCC2)N(C)C)=O)ccc(F)cc1F N1(CC)CC(C(=O)NCCCCNC(c2cc(OC)no2)=O)CC1=O c1(C(=O)NCC(CNC(CCC2(C)CC2(F)F)=O)F)ccc(N)cc1C(F)(F)F C(C)(CCCCNC(c1ccc(F)cn1)=O)NC(Cn1c(C(C)C)nnn1)=O C1(CNC(c2n(C=C)ncc2)=O)C(O)C(O)CN1C(=O)C(C1CCCCC1)F CN1CCn2cc(C(=O)NCCCN(C(C3CCO3)=O)C3CC3)nc2C1=O C(CCCC(=O)OC)NCC(c1ccc(C(F)(F)F)cn1)N(CCCC#C)C N1(C(CC(=C=C)C)=O)CCCCC12CN(C(=O)C(c1ccccc1C)C)C2 C1(C(=O)NCC(CO)NC(c2c(C(C)C)noc2)=O)CCc2nccn2C1 Cc1cc(C(=O)N(C2CN(C(=O)CC3CNC(=O)C3)C2)C)cc(Br)c1 Cc1cc(C#N)ccc1C(N1CCN(C)CC1CNC(C1(F)CCOCC1)=O)=O C1(NC(C(C)OC(C)C)=O)CCC2(C1)CN(C(=O)Cc1cc(F)ccc1F)C2 C1(O)(CNC(C2CC(N(C)C)C2)=O)CCCN(C(c2ccc(Cl)c(N)c2)=O)CC1 c1(C(N2CCC(CNC(c3ccnc(C(F)(F)F)n3)=O)C2)=O)cc([N+](=O)[O-])c[nH]1 N1(C(c2cc(C(C)C)n(C)n2)=O)CC2CCC(NC(=O)Cc3cncs3)CC2C1 C(=O)(CC(C)(C)N1CCOCC1)NC(CCNC(C1C(COC)C1)=O)C Cc1cncc(C(=O)NCCCC(C)(C)NC(c2ccc(C(F)F)cc2)=O)n1 N1(C(COCC(C)C)=O)CCCN(C(c2ccc(F)cc2C(F)(F)F)=O)CC1 C=CCC(CC(C)C)C(=O)NCC(=C)CCNC(c1ccc(C(F)(F)F)cn1)=O c1(C(n2cc(C3CCCN(C(CC(CC)O)=O)C3)nn2)C)ccc(C)c(C)c1 c1(CCC(=O)NCC=CCNC(C2CCC(C)CC2)=O)cc2ccccc2o1 n1(CC(C)NC(=O)CC(C)C(F)F)ccc(=NC(=O)Cc2cnn(C)c2)[nH]1 N1(CC)CC2CN(C(C3CN(C(=O)C(C(C)C)OC)CCN3C)=O)CC2C1 CC(C)(C(=O)N1CC(CNC(c2ccns2)=O)C(C(F)(F)F)C1)S(=O)(=O)C1CC1 C1(NC(c2c[nH]nc2C2CCC2)=O)CCC(NC(C2(CC3CC3)CC2)=O)CC1 N#CC1=C(C(=O)N2CCC(C(=O)NC3CNC(=O)NC3=O)CC2)CCC1 N1(C(COC)=O)CCN(CCCCCC2CCCN(C(=O)C=CC(N)=O)C2)CC1 C1(C(C)NC(C2(F)CCC2)=O)CCN(C(=O)Cn2cnnc2O)C1 CCC(CC(=O)NCCC(C)NC(C1CC(C)(O)C1)=O)OC C1(C)(C(N(CCc2ccc(C)s2)C)=O)CC12CCN(CC(=O)NC(C)C)CC2 c1(C2N(C(C(=O)NC(C(=O)OC)C)C3CC3Cl)CCCC2)ccc([N+](=O)[O-])cc1 CC1=C(C(=O)NC2CC3CCC2(NC(C24CC(C)C2C4)=O)C3)CCO1 C#Cc1cccc(C(=O)NC2CC(C)N(C(C3CCC4C(C3)C4(F)F)=O)C2)c1F c1(-c2nc(CCCCCC)nn2-c2ccc(OC)nc2)cn2ccccc2n1 C1(NC(C(C)NC(C)=O)=O)CC12CC(NC(=O)CCc1ccnc(C)c1)C2 C(=O)(C1=Cc2cc(F)ccc2OC1)N1CCC(Nc2ccnc(C)n2)C1 N1(C(c2cncc(SC)c2)=O)CC(F)(F)CC1C(=O)NCc1ccccc1C C1(CNC(C(CC)SC)=O)(NC(c2cnn(-c3nccs3)c2)=O)CCCCC1 N1(C(C(CC2CC2)NC(c2cc(Cl)cs2)=O)=O)CCCC2(C1)N=N2 C(CCC(=O)NC(CN(C(=O)CCC1(N(C)C)CCCC1)C)CC)=CC CN1CCC(CN(C2C3CCC2(c2ccccc2)C3)C)CC1 N1(C(CCN(C)CCO)=O)CCC2CCCC12CNC(c1ccoc1Cl)=O C1(C(=O)NC2COCC23CCC3)Cc2ccccc2S1(=O)=O N1(C(C23N(C(C(C(CC)C)N(C)C)=O)CC(C2)C3)=O)CCOC2COCC12 C1(C(=O)NCC2(CC)CC2)CC(F)(F)CN1C(=O)C(F)CC1CCOC1 N1(CC(=O)NCC(C)(C)OCCNC(COCCCC#C)=O)CCCNS1(=O)=O n1(C(CC)C)ccc(=NC(=O)C2=CCCN(C(=O)COCCCN(C)C)C2)[nH]1 c1(N2CCC(C3(C)CC3)C2)nc2ccc(Cl)cc2c(=NCC2(C)CCCCC2)[nH]1 CS(=O)(=O)c1ccc(C(N2CC(O)CC2C(=O)NCCc2ncc[nH]2)=O)cc1Br c1(CN(CCOC)C)cn(C2CCC(C(=O)NC3CS(=O)(=O)C3)C2)nn1 Clc1cccc(CNC(C2CCCCO2)Cc2ccccc2I)n1 c1(C(C)C)ccc(OCC(=O)NCC(CO)NC(=O)CCCCN(C)C)cc1 N1(C(C2C3C(=O)C4C(C3)C42)=O)CCOC(C(N2CC(n3ccnn3)C2)=O)CC1 CC(C)(C)CC(=O)NCC12CC(NC(=O)CC3CCCC(O)C3)(C1)C2 C1(CC)CCC(C(=O)NCC2(NC(C3(CC)CC(C)(C)C3)=O)CC2)CC1 C1(C(=O)O)CCOCC1C(c1cc(CNCC2(N3CCCC3)CCCC2)on1)=O c1(C(N2CC(CNC(C(C)n3ccnc3)=O)C2)=O)cccc(OC(C)C)c1N CC(C)(C)CCC(=O)C(=O)NC1CCCCN(C(c2cnc3[nH]ccc3n2)=O)C1 C1(C(N2CC(C)C(NC(C3CCOCC3(C)C)=O)C2)=O)CCC(=O)N(C2CC2)C1 c1(OCCCC)ccc(CCN(C2CCN(C(=O)C(C)CC)CC2)C)cc1 c1(C(=O)NC2CC(O)(CNC(C3(OCC)CCC3)=O)C2)cc(C)c(C)cn1 C1(OC)CN(C(c2conc2C2(C)COC2)=O)CC1NC(C1CC2C=CC1C2)=O N1(C(C=NOC)=O)CCOCCC1C(=O)NC(C)CN(C)C(C)C C(C)(C)(CC(=O)NC1CC1c1ccsc1)N(C)C(c1cc(C#N)c[nH]1)=O N(C1CN(C(c2ncc[nH]c2=O)=O)Cc2ccccc21)C(C(CCC)N(C)C)=O N1(C(=O)CCCc2cccs2)CCC2(CCCN(C(=O)CCc3cnn[nH]3)C2)C1 Cc1cnc(F)cc1CNC(C1CCCN1C(=O)COc1ccsn1)=O C12(CNC(CCc3c[nH]c(=N)[nH]3)=O)CCC1CN(C(c1ccc(Cl)cc1Cl)=O)C2 c1(-c2ccc(CC(=O)NC(=O)NCCCOC)cc2)ccc(C(C)C)c(F)c1 CCCCC(C)CCC(c1nnnn1-c1cc(C)ccc1C)(NCCOC)OC C1(C)(NC(C(CC)C)=O)CCN(C(c2ccc(CCC(N)=O)cc2)=O)C1 C#CCC(C(=O)Nn1cnnc1C)NC(=O)CC(C)(C)C=C c1(OC)cncnc1C(=O)NC1(C(=O)NCC(C2CCCCC2)O)CCC1 C1(OCCC)CCN(C(C2CCN(C(=O)C(C)C3(O)CCC3)C2)=O)CC1 Cc1c[nH]nc1C(=O)NC(C)CC(=O)NCCCN(C)C(C)C C1(CCCC)(NC2(CC(=O)NCC(C3CC3Cl)=O)CCC2)CCC1 C(=O)(C(C)(C)C#N)N1CC(c2cn(C(C(=O)NCCCOC(C)C)C)nn2)(F)C1 C(=O)(C(C)C(C)c1ccccc1Cl)OCC(=O)NCCCCCC C1(NS(=O)(=O)Cc2ccc(C(F)F)cc2)CCCC2CNCCC12 C1(NC(c2c(C(C)C)con2)=O)CCC2(CC1)CN(C(=O)CSCCN(C)C)C2 c1(C(N2CCN(C(C3CC(SC)C3)=O)C3(C2)CC3)=O)cc2c(C)cccn2n1 CC1(C)COCCC1CC(=O)NCC1CCCCCN1c1nc(C(F)(F)F)ns1 CC(C)(CS(C)(=O)=O)C(=O)N1CC2C(C(=O)NCC3(OC4CCOCC4)CC3)C2C1 C(=O)(C1=CC2C=CC(C1)C2)N(CC1(NC(C(C)C(F)(F)F)=O)CCCCC1)CS(=O)(=O)CC N1(C(c2ocnc2C(=O)NC)=O)CCC(C)(CO)C1.C(C)(C=O)SCC c1(NC(C2(NC(C3CC(C)C3)=O)CC(O)C2)=O)ccc(Cl)cc1C c1(C(N2C(CC(=O)NC(CCC)CO)CC2)=O)snc(C)c1N N1(C(c2c(CC(=O)OC)occ2)=O)CC2(CCCC2NC(=O)CCCC(C)O)C1 Cc1ccc(CCCCC(=O)NCC2C=CCN2C(C2C3CNC(=O)C23)=O)cc1 C=C(C)CCC(=O)N(C1CCCCC1NC(=O)Cc1nc(C)sc1Cl)C C(=O)(CC(C)(C)C1CC1)NCC(C)=CC(=O)NCC1CCCN1C C1(C(=O)NC2C(NC(CCC=C=C)=O)CC2)(OC)CCCCCC1 C1(CNC(c2ccc(O)nc2)=O)CC2CCC1N2C(=O)CCC1CCC1 C1(C(CNC(=O)Cc2nc[nH]n2)F)CCN(C(=O)CCc2nncs2)CC1 C1(NC(=O)CC2CSC2)CCN(C(c2cnnc3ccccc23)=O)CCC1CO C(=O)(C1Cc2ccc(Cl)cc21)N1C(CO)CC(NC(CC(C)C)=O)C1 N1(C(c2c(CC)csc2)=O)CCN(C(c2ncn(CC(F)(F)F)n2)=O)C(C)C1C c1(C(=O)NC(C)(C)CCNC(C2CC2Cl)=O)cc2c(cc1N)OCO2 N1(C(C(C)OCCC=C)=O)CCC(NC(c2ncc(F)cc2F)=O)C(O)C1 C12(CNC(C3CC(CCC)C3)=O)CC1CN(C(=O)Cc1cncc(C)c1)C2 c1(C(=O)NC(CNC(C(C)OCCCC)=O)C(C)C)cccc2nc(C)cnc12 C1(CC(=O)NCC=CCNC(C2CC2c2ccncc2)=O)CC2CC2C1 C1(NC(=O)NC(CCCC)CF)CC2c3ccccc3CCC12 CCCC(C(O)C(=O)N(C)CCc1ncon1)NC(C1CC(F)(F)C1)=O C1(C(=O)NCC(Cl)Cl)CCN(C(c2cc(=O)cc[nH]2)=O)C12CC2 c1(NCC)ccccc1C(=O)NC1(CNC(=O)C(F)F)CC1 C1(NC(CN2CCC(C)CC2)=O)CC(O)C12CCC2.N12CCCC1CC2=O C(=O)(C1=NNC(=O)CC1)NC(C)Cn1cc(CNC(c2nscc2Br)=O)nn1 c1(C(N2CCCC(c3cncn3C)C2)C(=O)NC)ccc(C2CC2)cc1F C1(C)(C(=O)NC2CCCN(C(C)=O)C2)CN(C(=O)C(C)C2CCCC2)C(C)(C)C1 Cc1ccc(CS(N2C(C(N3CCCOCC3)=O)CC2)(=O)=O)c(F)c1 C(C)(C(CC(=O)N(CCC(O)CO)C)NC(=O)CC1CC(C)=NO1)OC C(=O)(C1=NOC2COCC12)NCC1CCC(NC(c2[nH]cc(CC)c2)=O)CC1 c12ccc(cc1)CC(=O)NCC2.C1(CC)(NC(C2(CSC)CC2(F)F)=O)CCCC1 n1(CC)cc(C(N2CCC(CF)(NC(=O)C(C(C)C)n3cncn3)C2)=O)c(C)n1 CC(C)C(CC(=O)O)NC(C(=O)N1CC(c2ccc(Br)cc2)C1)(C)C c1(C(=O)NCC(N(C(CC(=C=C)C)=O)C)C2CC2)sc2cccc(F)c2c1COC C1(C(C(=O)OCC)CNc2cc(C3CCC3)nn2C(C)C)CC2CCC1C2 N1(C(C(=O)NC2C(C)(C)CNC2)=O)CCOc2cccc(F)c2C1 C=C=CC(C)C(=O)NCCCN(C(c1cc(C)n(-c2ccc(Cl)cc2)n1)=O)CC N1(CCCC(=O)NC2CC(O)C2)C(=O)CCC1=O C(=O)(C1=C(F)CN(C(C2CCCCNC2=O)=O)CC1)NC1(CO)CCC(C)C1 c1(C(C)C)nc(NCC2CCCC(F)C2)cc(=NCC(C)(C)CCO)[nH]1 C1(N(C(c2ccc(C(N)=O)[nH]2)=O)CCSc2cnc[nH]2)CCCCCC1 CC1(C(=O)NCCOCCNC(=O)CP(C)(C)=O)COC(=O)C1 n1(COC)ccc(C(=O)NCCN(C(=O)Cc2ccsn2)C(C)C)n1 N1(C(C2CC(C(=O)OC)C2)=O)CCCC2(CCCN2C(c2cc(N)c(Cl)cn2)=O)C1 C(CN=c1[nH]c2c(c(=NCC3CCS(=O)(=O)C3)[nH]1)SCC2)c1cccc([N+](=O)[O-])c1 c1(CC(=O)NCC2(O)CCN(C(COCCC(C)C)=O)C2)c[nH]c2cccnc12 N=c1cc2c(n[nH]1)CCN(CC(=O)N(C(C1CCC3CC13)=O)C1CC1)C2 C1(C(=O)NCC(C)N(C)C(C2CC3CCC(C2)C3O)=O)CC(C)(C)OC(C)(C)C1 Cc1ccc(F)cc1C(=O)NCC(C)NC(c1cc(O)ccc1F)=O c1(NC2CC(CNC(Cc3nc(C)sc3C)=O)C2)cc(C)c([N+](=O)[O-])cc1Br c1(NC(c2c[nH]c(=N)o2)=O)ccc2c(c1)CCCC2 N1(C(C(C)C2CCC2)=O)CCC2(CCCC2NC(c2nccc(Cl)c2F)=O)CC1 C(CC(C)(C)C(F)(F)F)OC(CS(=O)(=O)N1CC(C)C1)=O C1(NC(c2ccc(CC)cn2)=O)(CNC(=O)Cc2c[nH]nc2C)CCCCCC1 C(=O)(CCC1CCCC1)NC1(C)CC1.C12(CC1)C(=O)N2.COC Cc1cnc(C(=O)NC(C)CCN(C)C(C2CC2CF)=O)o1 C1(C(=O)NCC2(C(=O)OCC)CCC2)CN(C=O)CCO1.C1(CCC=C)CC1 C=CC(C)(CC)C(=O)NC1CC(C)N(C(c2ccc(C3CC3)s2)=O)C1 N1(S(CCOCC)(=O)=O)CCC(NC(=O)C(=O)NC)C(NC(C2CCC2)=O)C1 N1(C(C(CC)C)=O)CC(OC)CC1C(=O)NCC1CCCC1N(C)C N1(C(C(c2ccc(N)cc2)C)=O)CCC(CCN(C)C(C2CC=CC2)=O)CC1 C1(OC)(CNC(C2CCCN2C)=O)CCN(C(=O)C(C)(C)C2CCCC2)C1 C1(CNC(CSCC(C)=O)=O)C2CN(C(C3(C)CC3c3ccccc3)=O)CC12 c1(NC(c2cn(CCNC(C3CCC(F)S3)=O)cn2)=O)ccc(O)c(Cl)c1 C1(OC)(CNC(c2ccsn2)=O)CCN(C(c2cnc(Cl)cn2)=O)C1 c1(OC)cc(CN2CCC2(C)C(=O)Nc2cc(C)cnc2Br)c([N+](=O)[O-])cc1O C1(C(=O)NCCOCCCN(C(=O)C(C)(C)CF)C)C2CCC1(c1cnco1)C2 C(=O)(C(C1=Cc2ccccc2OC1)N1CCc2nc(Br)sc2C1)NCCCCCC CCC(C)(CO)C(=O)N1CCC(C)(CNC(C2(c3cccc(OC)n3)CC2)=O)C1 n1(C(C)(C)C)nnnc1C(C1CCCCC1)(C)NCC1(CSC2CCCC2)CC1 O=C(C1=CCCOC1)NC1CN(C(c2cscc2Cl)=O)CCC1CO c1(C(N(C(CC(=O)OC)C)C)=O)n[nH]c2c1CN(C(C1CC1C(C)C)=O)C2 c1(N(CC(C2CC2)OC)C)nc(=NCCC(C)(C)C)[nH]c2c1COC2 c1(C(N(C(C)C(=O)NCCc2cc(C)ns2)CCC)=O)ccc(C)cc1F C(CCCCCNC(C1(F)CC=CC1)=O)NC(C(C)CF)=O CCCC(C#N)C(=O)N1CCC(C(=O)NC2CC(CO)(CO)C2)C1(C)C C1(N(C(C(C)NC(N)=O)=O)C)CCCN(Cc2ccc(CN)s2)CC1 C(=O)(C#CC1CCOCC1)NCC1(C2(O)CN(C(C(CCCCC)O)=O)C2)CC1 N#CC1CCN(C(c2cncc(NC(=O)Cc3cc(Br)cs3)c2)=O)C1 CC1CCCN(C(C2CCCN(C(C3CCOC3)=O)C2)=O)C1CN Cc1oc(-n2cccc2)cc1C(=O)NC1CC(C)(NC(=O)CCCC2CC2C)C1 Cc1cc(F)c(C(N2CC(NC(c3cc(O)nc(Cl)c3)=O)C(F)C2)=O)cc1F c1(C(=O)NC2C(C(=O)Nc3n(C(C)C)ncc3)CCC2)ccc2nccn2n1 C1(CC)CN(C(=O)C(C)S(C)(=O)=O)CCC1NC(C1CC(O)CN1C(N)=O)=O N1(C(CC(C)C)C(=O)N2CC(C(C)(F)F)C2)CCc2ccccc2C1 CC12CC(C1)C(C(N1CCC(c3cccnc3N)CC1)=O)CO2 c1(CN2CCC(NC(=O)Cc3ccn(CCF)n3)C2)c(Cl)cccc1I C1(F)(C(=O)NCC2(OC)CC2)CCCN(C(=O)Cc2c(C)cnn2C)C1 Cc1c(C(N2CCC3CN(C(=O)C=CC(=O)N(C)C)CC23)=O)sc2cc(F)ccc12 CCCCC(C(=O)NCCC1CCN(C(=O)C(C)(C)C2CCOCC2)CC1)N(C)C n1(CC(=O)NCC2(F)CN(C(C3=C(C)OCCC3)=O)C2)ccc2ccc(Cl)cc12 c1(OC)cc(Cl)cc(Cl)c1CN1CCOC(C(N2CCC(C)(C(N)=O)C(O)C2)=O)C1 c1(C(=O)NC(C)CNC(c2ccn(C)c2)=O)cc2cc(F)c(F)cc2[nH]1 CC1CC(CNC(C2(C(=O)NC3CC3)CC2)=O)CN1C(c1ccc[n+]([O-])c1)=O C1(NC(c2cnc(C)n2C)=O)C(C)CN(C(C2(c3cc[nH]n3)CC2)=O)CC1C C=CC1CN(C(c2c(C)nn(CCO)c2C)=O)CC1NC(=O)CCCNC(C)=O c1(CN(C)C(c2ccnc(C3CCCC3)n2)=O)cccc(Cl)c1Cl n1(CC)cc(Cl)c(C(=O)N(C)CCN(C)C(c2nccn2CC)=O)n1 C1(C(N(CCCCCCNC(C(CCC)C)=O)C)=O)CC2CCCCC12 C1(CNc2cc(N(C)C(C3CN(CC)C(=O)C3)=O)ncn2)CCCC2(CCC2)O1 N1(C(c2cccc(C)c2)=O)CC(NC(C2(c3cccc(Cl)c3)CC2)=O)CC(O)C1 C(N=c1[nH]c(=NCCS(C)=O)[nH]c2c1CSC2)C1C(CCC)CCC1 c1(C(=O)NC2CN(C(C(C)SCC)=O)CC2N=[N+]=[N-])c[nH]c2cccnc12 c1(OC)ccc(C)nc1C(=O)NCC=CC=CCNC(C1CCOC1C1CC1)=O CC1(CNC(C2CC3C=CC2O3)=O)CN(C(=O)CC2(O)CCOCC2)CCO1 CCC(C(=O)NC(C)CNC(c1ccn(-c2ccccc2F)n1)=O)C(C)(C)CC CC1(C2CCC2)CCCN1C(=O)N(C1CC=CCC1C(F)(F)F)C1CC1 c1(C(=O)NCC2CCCN2C(=O)Cc2cnoc2)coc2c1CSC2 CC1C(NC(=O)CC(O)C2CCCC2)CCN1C(=O)CSc1ccccc1Cl c1(C(N2CC(C(=O)NCCN)OCC2)=O)ccccc1[N+](=O)[O-] C1(C(=O)NC(CN(C(C(n2ccc(-c3cccs3)n2)C)=O)C)(C)C)C2COCC12 c1(CC)ncc(NC(=O)CCN(C(C2SCC=C2C)=O)C2CC2)cn1 C(CNC(c1cn(C)nn1)=O)(CC(F)(F)F)NC(CCN(CC)CC)=O C1(C(=O)NCC(C)(CO)NC(C(C)C#N)=O)CN2CCN1CC2C CC(C)(C(=O)N(CCS(=O)(=O)Nn1cncn1)C1CC1)c1cncnc1 N1(C(C2C(COC)C2)=O)CC2CC2(CNC(=O)Cc2cnc(-c3ccsc3)s2)C1 N1(CC)CCN(CC(=O)NCCC2(OC)CN(C(C3CCCC(=O)O3)=O)C2)CC1 C(=O)(C(C)(C)C1CCCN1C(c1cc(Cl)cs1)=O)NCCCN(CCC)C Cc1ncc2ccc(C(N3CCC(O)C(NC(C4CC=CCC4)=O)C3)=O)cn12 Cc1nnc(O)c(C(=O)NCC2(CNC(=O)CC(C)C(F)F)CCCC2)c1C N1(C(c2n(CCC)ncc2)=O)CC(CCNC(C2(CO)COC2)=O)OC(C)C1 C1(CNC(C(Cc2ccccc2)OC)=O)CCN(C(c2cn(C)c(C)n2)=O)C1(C)C CC1Cc2cccc(C(=O)NC3CC4C3CCN4C(=O)C=Cc3ncc[nH]3)c2O1 c1(CN(C(CC2(C)CC2)C(=O)NC2CCOC2)C)ccncc1 n1(CCNCCCCC=CC)cnccc1=O.C(=O)OCC N1(CCC)CC(NC(C2CC(O)(CNC(=O)C(C)CO)C2)=O)CC1=O C(c1cccn1C)=CC(=O)NC1CC(CNC(CC2N(C(C)C)CCC2)=O)C1 C(C1=CCN(C(c2ccn(C)c2-c2ccccc2)=O)CC1)NC(CC=C)=O c1(NC(N2CCC23CCC(CO)CC3)=O)ccc2cc(Cl)ccc2n1 c1(C(=O)NC2CCN(C(c3cnnc(Cl)c3)=O)C2)cc(O)nc(O)n1 c1(C(=O)NCC2(O)CN(C(c3c(C)ccc(OC)c3)=O)C2)ccc(O)c(F)c1F S(=O)(=O)(c1cc2ccccc2s1)N1CCC(C(C(F)(F)F)NC(C=CC)=O)CC1 C1(C(=O)NC(C)(C)CCF)C2CCC(C2)C1NC(c1ncncc1Cl)=O C1(CNC(COCCC=C)=O)CCC(C)N(C(=O)CCC(N)=O)C1 C1(OC)CC(NC(c2cc(C)n(C)n2)=O)CN(C(C2CCCN2C=O)=O)C1 C12(C(N3CCC(F)(C(N(CCCCCO)C)=O)C3)=O)CCC(CO)(CC1)CC2 c1(C(N(CC(C)CNC(=O)C(C)(C)CN(C)C)C)=O)ccc2nccnc2n1 C(=O)(C(CNC(C1(C2(C)CC2)CC1)=O)C(C)C)NC(c1ccc(C)s1)C N1(C(C2C3COCC23)C(=O)NCCSC)CCOC2(CCOCC2)C1 Cc1c(C#N)sc2ccc(NC(N3CCC(C(C)CO)CC3)=O)cc12 C(=O)(CCCC(=O)NCC12COC(CNC(C3CC4CCC4C3)=O)(C1)C2)NCC Cc1ncc(C(=O)NC(CCOCCO)C(N2CCCC(C)(F)C2)=O)c(C)n1 c1(C(N(C2C3CN(C(C4(C(=O)OCC)CC4)=O)CC32)C)=O)cccc2cnsc12 Cc1nc2ccccn2c1C(N1CCC2CN(C(=O)CN3CCC(C)C3)C2C1)=O CN=c1[nH]c(=NCCc2cccc3ccccc23)[nH]c(=NCCCCC(N)=O)[nH]1 N#Cc1cncc(C(=O)NC2(CCNC(=O)CC3CC4(CCC4)CO3)CCC2)c1 C1(CCC)(C(C)C)CCN(C(C2(OC)CCN(C(c3ccoc3CC)=O)C2)=O)C1 c1(C(=O)NC2CCCN(C(C=Cc3c(C)coc3C)=O)C2)cccc2nccn12 CCCCC(F)C(=O)N1CC2CC(C(=O)NCCc3[nH]cnc3C)(C2)C1 Cc1[nH]c(C)c(C(=O)NCC(C2CC2)NC(=O)CCCCN(C)C)c1C N1(C(CCCC(CC)NC(c2c(C)n[nH]c2C)=O)=O)CCC2CCN(C)CC12 c1(CCC(=O)NC(CC=C)CNC(C2CC(OC)C2)=O)ccc(Cl)c(OC)c1 c1(OC)cc(C(N2CCN(C(c3cnn(C(C)C)c3)=O)C(CO)C2)=O)ccc1O c1(C(=O)NCC2(O)CN(Cc3ccc(C)cc3F)C2)cc(F)c(F)cc1O C(=O)(C(C)CCCCCC)NCCNC(C1CC(OCC)C(NC(C)(C)C)C1)=O CC1CN(C(C2C3CN(C(=O)C4CC4)CC23)=O)CC(C)C1C(=O)OC(C)(C)C c1(C(=O)NCC(F)CNC(c2ccc(CO)s2)=O)cc(F)c2ccccc2c1 c1(OCCC)ccc(N(C)C(c2[nH]cc(C(C)=O)c2C)=O)cc1 C12(C(=O)NCCCCN(C(c3cnc(CC)s3)=O)C)CCC(C)(C1)OC2 N1(c2n(CCOC)c(C(=O)NC(C)C)nn2)CCn2c(C(C)(C)C)nnc2C1 N1(C(C=Cc2n(C)ncc2)=O)CCOC2(CCCN(C(c3cnc(Cl)s3)=O)C2)C1 c1(CC2N(C(c3c(C)scc3)C(=O)NC3(C)CC3)CCCC2)cccc(Cl)c1Cl C1(c2n(CCC)nnn2)(Nc2cn(C)nc2SC)CCC2CN(C)CC12 CC(O)(CNC(C1(NC(=O)COCCCN=[N+]=[N-])CCSC1)=O)CCO C1(N(C(c2cc(C)n(C)n2)=O)CC)CC(C)CN(C(=O)CC2CCNC2=O)C1 N1(C(=O)C(N2CCC3C(C2)C3(F)F)=O)CCc2ccc(F)cc2C1 O=C(CCCS(=O)(=O)c1ccc(Br)cc1)Nc1cc(OCC(F)F)cc(F)c1 CCCCC(C)NC(=O)C(=O)NCc1ccc(C(N2CCOCC2)C)o1 C1(C(=O)NC2C(C)CN(C(=O)Cc3cc[nH]n3)C2)CCC(C)(C)CC1 c1(C(=O)NC2(CC=C)CCN(C(=O)CCOCC)C2)ccc2ccnc(C)c2c1 CC(C)C(C(=O)Nc1nnc(C2CCCO2)s1)Sc1ncccn1 c1(NCc2cc(OC)ncn2)nccc(=NC(C)c2ccc3c(c2)OCO3)[nH]1 c1(C(C(=O)NCC(CC)NC(=O)CN2CSCC2=O)C)cc(C)cc(F)c1 C(=O)(C(O)C(C)c1ccccc1F)N1CCC(CC(=O)Nc2c(CC)n[nH]c2)C1 C1(C(N(C2CCN(C(=O)COC3(C)CCC3)C2)C)=O)CCc2nnc(O)n2C1 c1(CC(C)C)ccc(C(=O)NCCN(C(=O)C2=CCC2)C(C)C)s1 C1(NC(CCc2n(C)ccc2)=O)CCCCC1C(=O)NC1CCC=CCC1 N1(C(c2c(C)nn(C)c2)=O)CCCC(C(=O)NCC(C)(O)C(C)C)CC1 C1(CC)CN(C(c2n[nH]c(C)n2)=O)CCC1NC(C1CCCN1C1CCCC1)=O c1(N(C)C)cncc(C(N2CCCC2(C)CNC(=O)C(F)F)=O)c1 C1(C(=O)NC(C)C(C)(C)C)C=CCCN1C(=O)C(=O)N(C)C c1(N(C)C)nc(CC(=O)NC2CCC2CNC(C2(n3nccn3)CC2)=O)cs1 N1(C(C2(C(C)C)COC2)=O)CC2C3CCC(C2C1)N(C(=O)COCCCO)C3 CC1COCC(C(=O)N(CCCCN(C)C(C2CC(F)(CO)C2)=O)C)O1 N1(C(c2cc(C(=O)OC)c(F)cc2)=O)CCC(NC(=O)C(C)SC)CC12CC2 c1(CN(c2cccc(OC)c2)C(=O)C(=O)NCCO)ccc(NC)c(N(C)C)c1 CC1CCCCC1C(=O)NCCCOCCC(=O)NCCC1CC1 C(=O)(C(CCF)NC(c1cnsc1)=O)N1C(CCC#C)CCC1 C1(CC)C(NC(=O)C(C)SCC2CCCO2)CCCN1C(=O)C1=CCCC1 C1(C(=O)NCC(CC)N(C)C(c2nnsc2C)=O)C2CC3C(C2)C13 c1(OC)cc(NC(c2nnnn2C2COC2)(C)CC2CCCCO2)cc(F)c1 c1(C(=O)NCCC(C)N(C)C(C2(C#N)CC2(C)C)=O)ccc(Cl)c(F)c1 CC1CN(C(=O)CN2CC3CCC2C3)CC2(CCN(C(=O)C(C)CC3CC3)C2)O1 C1(CN(C(C2CC(OC)C2)=O)C)COCCN1C(C1CCC(OC)CC1)=O CC(C)C(C)CC(=O)N1CCC(C)(CNC(=O)C=CC(F)(F)F)CC1 O=S(=O)(c1ccc(=NCCN2CCC2)[nH]c1)N1CCC2(CC1)CC2NC1CC1 Cc1cc(N)ccc1C(=O)N(C(C)CNC(c1cccc(OC(C)C)c1F)=O)C c1(CC(N2C(C(C)C)CN(C(=O)C(O)C(C)(C)C)CC2)=O)ccc2[nH]ccc2c1 CC(C(=O)NCc1ccoc1)N(C(=O)CCNC(N)=O)CCCN1CCCC1 c1(NC(C2CCC(NC(c3cc(CC)nn3C)=O)CO2)=O)cc(O)c(Cl)cc1Cl c1(C(N(CC(C)(O)CNC(C2(c3cccs3)CC2)=O)C)=O)ccc(CO)cc1F CC1CCC(C(=O)NC23CC(NC(=O)COc4ccsc4)(C2)C3)O1 N1(C(C(C)N(CC)CC)=O)CCC(NC(=O)N(C2CCCC2)C)C(O)C1.[SH](C)(=O)=O C1(NC(C=CCN(C)CC)=O)CCCC(NC(C2CCOC(C(F)(F)F)C2)=O)C1 Cc1c(CN2CCC(CNC(C3CNC(=O)O3)=O)C2)cnn1C c1(NC(=O)CCCC2CCC2)cnc2c(c1)CN(C(=O)CCc1nncs1)CC2 n1(CCOC)nc(C(=O)NCc2cn(C3Cc4ccccc4C3)nn2)ccc1=O c1(C(N(C2CCN(C(C3CCC4CC3C4(C)C)=O)C2)C)=O)cc2n(c1)CCOC2 N1(C(c2c(C)cc(C)s2)=O)CCC(C)(C)C(NC(=O)Cc2cn(C)nc2C)C1 Cc1cnc(C)c(NC(C2CC2C2CN(C(C3(c4cc[nH]n4)CC3)=O)C2)=O)c1 N1(C(C2N(CC(C)C)CCC2)=O)CC(NC(c2cn(C)c(=O)n2C)=O)CC(C)C1 C1(CC(=O)NCCN(CCCC)C)CC(NC(=O)Cc2cccs2)C1(C)C N1(C(CC(=O)OC(C)(C)C)=O)CC2CCCC2(C(N2CC(NC(N)=O)C2)=O)C1 S(=O)(=O)(c1ccc(OC)c(Sc2cncc(F)c2)c1)NC1(C(=O)OC)CC=CC1 C1(CC(=O)N(CCNC(=O)CC(C)C(C)C)CC)SC2=NCCN2C1=O N1(C(C(C(CC)O)C)=O)CCn2ncc(CNC(C3CS(=O)(=O)CCO3)=O)c2C1 C(=O)(C(C)C(CC)CC)NC(CC#C)CC(=O)NCC(c1ccccc1)F C1(C(=O)NC)CCCCCN1C(=O)CCN(C(=O)CN1CCCC1)CCO C=CCC(CC=C)C(=O)NC(C1(C(N2CCC3(CNC(=O)N3)C2)=O)CC1)C n1(CC(C)C)nc(-c2cccc(N(C)C)n2)nc1C1CCCC(F)C1 N1(C(Cc2c(C)scc2)=O)CCCC(CNC(=O)CC(C)(C)C2CC2)C1 CC1(C(=O)O)CCCCC1NC(C1CC1CN)=O Cc1cccc(C(O)C(=O)NC2CCCC2C(=O)NCCCCC2CC2)c1C Cc1cc(O)c(F)cc1NC(=O)CCC1(NC(=O)Cc2ccoc2C)CCC1 N1(C(C(C2(OC)CC2)CC=C)=O)CC(O)(N(C(=O)COCCCC(C)C)C)C1 C(=O)(C1=CCC(C)(C)CC1)N(CC(C)O)CCNC(c1cnc2ccsc2c1)=O C1(N(C)C(c2cnc(OC(C)C)s2)=O)CCCC(NC(c2ccsc2C(F)F)=O)C1 C(=O)(CC(F)(F)C(F)F)N(C(C)CNC(=O)CC1CCOC1)C Cc1csc2c(N3CCC(CNC(C4CC5(CC(=O)N5)C4)=O)C(C)C3)ncnc12 C1(C)(C(=O)NC(CNC(c2n(CCC)ncc2)=O)COC)CCCCCC1 C1(C2CC2)(C(N(CC=C)CCO)=O)CN(C(=O)Cn2ccnn2)C1 c1(C(N(C(CNC(Cc2cc(C)[nH]n2)=O)C)C)=O)cc(C)c(Cl)c(N)c1 C(C(C)(C)C(=O)N1CCCC(NC(c2c(C3CC3)cnn2C)=O)C1)SC c1(C(=O)NCC2N(C(CN(C(COC)=O)C)=O)CCC2)cc(Cl)cc([N+](=O)[O-])c1 N1(S(CC=C)(=O)=O)CCC2CN(C(c3ccc(CN(C)C)s3)=O)CCC12 Cc1cccc2cc(C(N3CCC(F)(CNC(C4CCCC4O)=O)C3)=O)nnc12 C1(C(=O)NC(C2CCN(C(=O)C(F)(F)C(C)O)CC2)C)Cc2cccnc2C1 Cc1nc(-n2cccc2)sc1CNCC(O)COC(F)(F)F c1(NC(C2(CC)CCCN2C(=O)C(C)OCOC)=O)cc(C)c(F)c(C)c1 N1(C(c2n(C)ccc2)=O)CC(NC(=O)Cc2cc(F)ccc2F)CC(C)(C)C1 C1(n2cc(C(C)(C)N(C(=O)CCCN(C)C)C)nn2)CCCC(NS(C)(=O)=O)C1 C1(N)CC(=O)N(c2ccnn2-c2ccccc2)C1.CC(C)CC(=O)N1CCCC1 CC1(CC(=O)CC(c2scc(Nc3cccc(Br)c3)n2)=O)CCC(=O)N1 C12CC(=NO1)C(=O)NC2.C1(C(=O)OCC)(Oc2cncnc2)CCOC1 CS(=O)(=O)c1cc(CNC2C=CC(C(=O)Nc3c(Cl)cnnc3Cl)C2)ccc1F c1(CC)cccc(C(N2CCC(Cn3cc(-c4nccs4)nn3)C2)=O)n1 c1(C(=O)OC)cccc2c1CCC2NCc1ncc(C(F)(F)F)[nH]1 c1(NC(C2CCN(C3CCCC3)CC2)=O)cnc(Br)c(I)c1.C12COCCN1C2 N1(C(C2CCN(CC)CC2)=O)CC2CC(C1)C2N=c1cc(Cl)nc(C2CC2)[nH]1 c1(CC(=O)NC(CNC(C(C)(C2CCC2)OC)=O)(C)C)ccc([N+](=O)[O-])c(N)c1 O=C(CNC1CC1)NNc1ccc([N+](=O)[O-])cc1OC(F)F.c12cccc(c1)OC2 c1(NC(=O)NCC2N(C(N3CC4CC4C3)=O)CC2)ccc(C)cc1.CCOCCO CCC(CC(=O)NCC(C1CCCCC1)NC(=O)CC1COCCO1)C1CC1 C=C(CNC(=O)Cc1cnn(-c2ccccc2)c1)CCNC(C1CCC(F)C1)=O C1(CC(=O)OC)CCCN1C(C1OCCC1N(C)C)=O.c1(S)ccccc1 C1(NC(c2c(C)ocn2)=O)C(CNC(=O)Cn2cccn2)CCC12CCC2 CC(C)CC(C)CNC(C1CSCN1C(C1CCN1C)=O)=O N1(C(C2C(C(=C)C)OCC2)=O)CC2CCC1CN2C(c1cncc(C(F)F)n1)=O c1(OC)cncnc1C(=O)NC1N(C2(CNC(=O)OC(C)(C)C)CC2)CC2CC21 c1(C(=O)NC2(C(N(C)CC3C(C)C3)=O)CC(F)(F)C2)cncc2[nH]ccc12 c1(C(=O)NC2CCN(C(C(C(=C)Cl)(C)C)=O)CC2)[nH]c2cccc(F)c2c1Cl C1(NC(C2CCSC2)=O)CCC2CN(C(c3cnn4c3NCCC4)=O)CC2C1 c1(C(N2CC(NC(C=Cc3cnc(C)s3)=O)C3C2C3)=O)ccc([N+](=O)[O-])cn1 c1(N2C(C)CN(C(=O)CCCN3CCCC3)CC2)nc2cc(F)ccc2o1 c1(C(N2CC(NC(CSCC=C)=O)CC3(C2)CC3)=O)ccc2c(c1)CCN(C)C2 C12CC(CN1C(C)=O)ONC2=O.C1(C(N2CC(O)(CC)C2)=O)CCCCS1 c1(C(N2CC(NC(Cc3nnc(C)o3)=O)C3C2C3)=O)cc(S(N)(=O)=O)cnc1C C1(NC(Cc2nc(NC=O)sc2)=O)CCCN(C(c2cc(C3CC3)on2)=O)CC1 C1(C(=O)NCc2cc(C)sc2)CC(=O)CC12CCC2 CCC(C)(COC)CNC(=O)CCC(C)NC(C1CC1(Cl)Cl)=O c1(C(=O)NC(C)CN(C)C(c2cnoc2)=O)nc(=O)cc(N)[nH]1 N1(C(C2C3(CCN(C(CSCC)=O)C3)C2)=O)CC2NC(=O)OC2C1 C(CCC1CC1)(C(=O)N(C(CO)C1CC1)C)NC(CCCOCC(C)C)=O CCC(F)C(=O)N1CC(O)(CCN(C(C2CCCC2)=O)Cc2occc2C)C1 c1(CNCC2(O)CCS(=O)(=O)C2)ccc(F)c2cccnc12 c1(OC)cccc2c1OC(C(=O)N(C1CN(C(c3cc(F)ccc3O)=O)C1)C)C2 N1(C(C(CC)O)=O)CC2CC2C1C(=O)NCCc1ccncn1 N1(C(CCCOCC)=O)CC(NC(C2CNC(=O)N2)=O)C(C)(C)C1 C#CCC(CC(=O)NCc1nc(C(N)=O)co1)NC(=O)C(C)(O)C(C)C C1(CC=C)(NC(c2cncc(CC)c2)=O)CCN(C(c2nnc(S)n2C)=O)C1 N1(C(C2CC(O)(CC#C)C2)=O)CCC(NC(=O)CC2CCCN2CC)C12CCC2 C1(NC(=O)CC2CC3CC3C2)CCC(NC(=O)CCc2cnc(C3CC3)o2)CC1 c1(OC(C(c2n(CC)ccn2)N(C(C)(C)C)C)=O)ccccc1OCCC(C)C c1(NC2CC(CNC(c3cc(C(F)(F)F)on3)=O)C2)nc(Cl)[nH]c2ncnc1-2 N1(C(c2c(C)nc(C)s2)=O)CCOCC(C(=O)NCC(C)(C)C2(O)CCC2)C1 C(C1OCCc2sc(-c3ccccc3)cc21)NC(c1cc2ccc(F)cc2s1)=O CCCC(CCCNC(=O)C(CC)OC)NC(c1cc(C)ccc1NCCO)=O c1(C(N2CC(NC(c3c(CC)n(C)nc3)=O)(CO)C2)=O)cccc2c1CCCC2 CC1CN(C(c2cncc(NS(C)(=O)=O)c2)=O)CCN(C(=O)NC2(C)CC2)C1 C1(c2ccc(OC)nc2)NC(=O)N(C)C(C2CC2)=C1C(=O)OC c1(C(=O)NC(C)CNC(=O)CCCc2ccc(Cl)cc2)cc(CO)ccc1Cl C1(C(N2CC(C)C(NC(N)=O)C2)=O)CN(S(=O)(=O)Cc2cccc(Cl)c2)CCC1O N1(C(C(CC)C2COC2)=O)CCCC(c2nc(N3CCOCC3)no2)C1 c1(C(=O)NCC(CNC(Cc2ccn(C)n2)=O)(C)O)ccc(N)c(F)n1 N1(C(c2ccccn2)=O)CC2CC(CO)C(C2)C1 C1(O)(CN(C)C)CCN(C(=O)NCCc2cccc(N3CCOCC3)n2)C1 CC(C)(O)C(F)C(=O)NCC1CN(C(=O)C2=CCCCO2)CC1C(F)(F)F C12CN(C(c3sc(Br)nc3C)=O)CCN1C2.c1(CC)ccc(OC(C)C)nc1 N1(CC(N2C3C(NC(c4n(CCC)ncc4)=O)C(C3)C2)=O)CCn2ccnc2C1 c1(C(N2CC(CC(C)NC(C(CSC)O)=O)C2)=O)noc2ncccc12 COC1c2ccccc2CC1NC(=O)NCC(c1cccc(C#N)c1)(C)O Cn1ncc(C(=O)NC2CCN(C(=O)Cc3nnn(C(C)(C)C)n3)C2)c1C1CC1 C1(CC(=O)NCC2CCCC(C)O2)CC2(CC2)CN1C(=O)CN1CCCC1 C1(C(C)C)CCC(C)CC1C(=O)NCC1(F)CC(NC(=O)CC2CCCC2)C1 C1(NC(=O)Cc2ccsn2)CNC2(CCCC2)C1.CCS(=O)(=O)N1CCCC1 C1(NC(CSCC(C)C)=O)CC2CN(C(C3CCC(C)(C)OC3)=O)CC2C1 C12(NS(=O)(=O)CCc3ccccc3Br)CCC(CF)(C1)OC2 C1(NC(=O)NCCn2ncccc2=O)CCC(C(F)(F)F)NC1=O Cc1ccc(Cl)c(C(=O)NC(C)CCNC(=O)CCc2ccoc2)c1 C1(C2CCC2)(C(NC(=NCC2CC(F)(CF)C2)NC)C2CC2)CCC1.C1(CC2CC2)CC1 C(=O)(CCCCCCC(C)=O)N1CCC(C)(NC(CC=C)=O)C1 CCCC(CCC)CC(=O)N1CCCN(C(c2ccc(C)c(C)c2O)=O)CC1C N1(Cc2cc(OC)c(F)cc2)CC2C(C1C(=O)NC(CO)C(C)O)C2(C)C N1(C(c2ccc(CC)[nH]2)=O)CCN(C)CC1CNC(=O)C(c1c(C)n[nH]c1C)C C1(CC(=O)NCC(CNC(C2C(CC)C2)=O)O)(CO)CCCC1 CC1(C)COCCC1C(=O)NCCC1(NC(c2cc(Cl)ccc2Cl)=O)CC1 c1(C(=O)NCC2(COC)CCCN2C(c2ccc(O)nc2)=O)cn(C)c(=O)n1C C1(F)(CNC(COCCC)=O)CC(N=c2nc(Cl)[nH]c(C)c2C#N)C1 C(=O)(CC1=CCCCC1)N1C2C(CNC(c3c(CC)c[nH]n3)=O)C(C2)C1 C1(F)(C(N2CC(CC)C2)=O)CN(C(=O)Cc2cnc(C)s2)C1 CC1CC(CNC(=O)C2CC2)CN1C(c1cc(C2CCCOC2)[nH]n1)=O C(=O)(C(CCC)C1CCCC1)N1C(C(NOCCCC=C)=O)CCC1 Cc1ccc(C(=O)NC2CCCC(C(=O)N(C(C)C)Cc3cccs3)C2)cc1C c1(C(=O)NCC(N(C)C(C2SCCS2)=O)C2CC2)coc(C(F)(F)F)c1 c1(C(N(CCCCN(C(C2(CSC)CCC2)=O)C)C)=O)cc(C2CC2)cs1 CC(CCCCc1ccccc1)NCCCCF N1(C(CCCc2onc(C(C)C)n2)=O)CCCCC(NC(C2CCOC2=O)=O)C1 C(CCCCN=[N+]=[N-])NC(CCN(C(=O)C(O)C1CCC1)C)=O C=CC1CN(C(=O)C(C)(C)C=C)CC1NC(=O)C(CC)N1CCCCC1 CC(C(CO)NC(=O)CCCNS(C)(=O)=O)NC(=O)C(O)c1ccsc1 C1(CC(=O)NCC(CC)NC(=O)CCC2CCCCC2)COc2ccccc2O1 c1(C(=O)NCC(CNC(C(Cc2c(C)noc2C)C)=O)O)cnn2cnnc2c1 Cc1ccncc1C(N1CCC(C(=O)NCCC2(C)CC2(F)F)(CF)C1)=O n1(CC)cc(C(=O)NC2CCCCC2NC(=O)C(C)NC(C)=O)c2ccccc12 c1(C(=O)NCc2cc(C(N(c3ccccn3)CC)=O)n(C)n2)cc(C#N)oc1C N#CC1CCN(C(=O)C(C2CC=CCC2)NC(C2CCC3(CC3)C2)=O)CC1 O=C1CCC(NCC(N2CCC(CCC(=O)O)(C(F)(F)F)C2)=O)CN1 c1(C(=O)NC(CNC(c2c(C)nc(CO)o2)=O)CO)cc(S(C)(=O)=O)cnc1O CCC(C)(CCC(C)C)C(=O)N1CCC(F)C(NC(=O)CCN2CCCC2)C1 Cn1c(CC(N2CCOCC2C(F)(F)F)=O)nc2ccccc12 CC1=C(C(=O)NCC2(O)CN(C(c3cn4c(n3)CCC4)=O)C2)CCCO1 C1(NC(C(C)(C)OC)=O)CCCCC12CCN(C(c1cc(O)cc(=O)o1)=O)CC2 N1(C(C(c2ccccc2)OC)=O)CCCCC1CCNC(c1cscc1F)=O N1(C(C(C)NC(=O)Cc2ccc(-c3ccccc3)cc2)=O)CCOC2(CSC2)C1 c1(C(N2CCC(O)(CNC(C34CC(OC)C3C4)=O)C2)=O)cscc1S(C)(=O)=O c1(C(=O)NCc2scc(C(=O)NCCCCCC=C)c2)ccnc(O)c1F C1(CC)CN(C(=O)CC(c2ccc(C(F)(F)F)cc2)O)CCN1C(=O)C(F)F c1(C(N2CC(CNC(c3n[nH]c(C)c3C)=O)C3C2C3)=O)cnc2ncccn12 N1(C(c2cn3c(n2)CCC3)=O)CCCC12CCN(C(C1(C(F)(F)F)CCCC1)=O)C2 Cn1cc(Br)c2c(C(=O)NCc3ccc(C(=O)OC(C)(C)C)cc3)ccnc12 c1(SCC)cncc(C(N2CCC(CF)(NC(=O)C(F)CC3CCC3)C2)=O)n1 C12(NC(COCC(C)C)=O)CC(NC(c3ccoc3)=O)(C1)C2 N1(C(CCCc2onc(C)n2)=O)CCN(C2CN(C(C3C(C)C3C)=O)C2)CC1 N1(C(c2c(CC)ncs2)=O)CC(C)(C)OCC1CNC(=O)C(F)OC(F)(F)F N1(C(C2(C)C(C)(C)C2(C)C)=O)CC2(CC(C(=O)N(CCF)CCO)CO2)C1 C1(OCC2(CNC(=O)CN3CCC(O)CC3)CCC2)C#CCCCCC1.O=C1CO1 CC(C)C(C)(O)C(=O)NCC1(NC(=O)C(c2cccnc2)n2cccn2)CC1 c1(N2CCN(C(c3ccc(CN(CC=C)C)cc3)=O)CC2)cncc2nnnn12 Cc1ccc2[nH]c(C(N3CCC(CNC(=O)CC4CCN(C)C4)C3)=O)c(C)c2c1 C1(NC(CCCOCC(=O)OC)c2nnnn2C2(C)CC2)CCN(C)CC1C CN1CCCC(CCC(=O)NCC(C2CCCC2)NC(=O)C(F)=C2CCCC2)C1 C1(CN(C(c2nc(COC)oc2)=O)C)C2CN(C(=O)C(Br)=C(C)C)CC12 C(=O)(CC(C)C(F)F)NC(CCOCC)C(=O)NC(C)Cc1nncn1C N1(C(c2cc(C(=O)NCC#CC3CC3)[nH]n2)=O)CC(C(N)=O)C2(CC2)C1 C(=O)(C1n2ncc(CO)c2NC1)NC1CN(C)C(=O)CC1 C(CC(C)(O)C(F)(F)F)NN1CCCC1.c12cccc(c1)NC(=O)C(=O)N(C)C2 C12C3CN(CC13)C2.C1(C(=O)C2CC2)CCN(CCO)CC1.c12cc(c[nH]1)CNC2 C(=O)(CC1CCCN(C)c2ccccc21)NC(CCN(C(C(CC)CC)=O)C)C C=CCC(C)(C)CCOCC(=O)Cc1cccc(N(C)C)c1 C(CC(CC)C(=O)NCCNC(=O)NCc1ccccc1)=CC.n12cc(nn1)C2 Cc1cc(O)nc(CNc2cccc(C(=O)NCC3(C)COCCO3)c2)n1 N1(CC(=O)NCCOCCN(C(c2c(CC)[nH]cc2)=O)C)CSCCSC1 N1(C(c2ccc(SC)s2)=O)CC(NC(c2cnncc2O)=O)CC1CO C=CC1(C(N2CC3CCC2C(O)C3)=O)CCN(C(=O)CCCC=O)CC1.OC CC1CC(NC(C2CC(C)(C(C)(C)C)C2)=O)CN1C(C1CC(C)(C)C1)=O c1(C(=O)NC2C(NC(C(CN(C)C)N(C)C)=O)CCOC2)cnn2ccccc12 c1(C(=O)NCCOCCNC(=O)C2=C(Cl)CCC2)ccc(F)cc1F c1(C(N2CC=CC(NC(C(C3CCCC3)OC)=O)C2)=O)ccc2cn(C)nc2c1 CCS(=O)(=O)NCC(=O)NC1CC(CNC(=O)C(C)SCC(C)C)C1 c1(NC(C(=O)NCC2CC(CCC)C2)=O)cn2ccc(Br)cc2n1 N1(C(c2cc(C)[nH]n2)=O)CC(C(=O)NCC(C)C(F)(F)F)OC(C)C1 c1(C(=O)NC23CN(C(C4(CC=C)CC=CC4)=O)C(CC2)C3)ccc(F)cc1C#N C(=O)(CC(C(F)(F)F)n1cccn1)OCC(O)COc1ccccc1.O=CCNCC1CC1 c1(C(c2n(CC(=C)C)nnn2)NCCC2(C)CCCO2)cc(C#N)n(C)c1 Cc1c(C(F)(F)F)n[nH]c1C(=O)NC(C1CCN(C(C2(C)CCCC2)=O)C1)C c1(C(N(CC(C)NC(C2C(C)C2(F)F)=O)CC)=O)nnc2ccccc2n1 C1(NC(C2C(C)C2)=O)CCCN(C(=O)C(O)Cc2cn(C)cn2)C1C Cc1cc(O)nc(C)c1C(=O)NCC(C)NC(C1(C)CCCCO1)=O Cc1sc(-c2ccco2)nc1C(=O)NC1CCCC(CNC(c2cc[nH]n2)=O)C1 C#Cc1ccc(CCCC(=O)NCCN(C)C(c2ccc(SCC)cc2)=O)cc1 N1(C(c2ccc(C)o2)=O)CC2CCC2(CC(=O)NCCC2(C)CC2)C1 c1(C(N(C2CN(C(C(C=C=C)C)=O)CC2(C)C)C)=O)cc2ccccc2cc1F C(=O)(CCCN=C1NS(=O)(=O)c2ccccc21)NCC(C)(C)NC(C(C)N(C)C)=O C1(C(C)C)CN(C(=O)C=Cc2cc[nH]n2)CCN1C(=O)Cc1cc[nH]c1 C(C(CC)CCO)NC(C1(F)CC(NC(CCNC(COC)=O)=O)C1)=O C1(C(N)=O)(CNC(=O)CC2CCCN(C(c3cccnc3S)=O)C2)CC12CCC2 C1(C(=O)NCCN(C(C(CC)N(C)C)=O)C2CCCCC2)CCN(C)CC1 Cc1cn2cc(C(=O)NCC3CN(C(=O)C=Cc4cccs4)C4CC34)ccc2n1 c1(C(C(=O)OC)N(C(c2cccc(I)c2)C(=O)NCCCOC)C)cccc(Cl)c1 c1(CNC(CCN(C(CC2ON=C(CC)C2)=O)C2CC2)=O)[nH]ccc(=O)c1O C#Cc1ccc(C(N2CCN(C(c3cnc(C#N)s3)=O)C(CCC)C2)=O)c(F)c1 c1(C(=O)NC2C(NC(C3(CCOC)CC3)=O)CCCC2)c(O)cccc1O C1(CNC(CCC)=O)CC(NC(=O)CCSCc2ccccn2)C1(C)C CCCC(F)C(=O)NCC1(CC(=O)N(CC(F)F)CC)CC1 C1(CC)CC(CC(=O)N(C2CCN(C)CC2)CCCN2CCCCCC2)CCO1 c1(-c2nnn(C)n2)ccc(-c2cccc(C(N3CCNCC3)=O)c2)cc1 C(=O)(C1Cc2ccccc21)N(CCC(=O)NC1CCCC1NC(C)=O)CC=C C(CCN=c1nc2sccc2c(NC2CCc3cccnc32)[nH]1)SC N1(C(C(C(C)C)(C)C)=O)CCC2CCN(C(=O)Cc3cnn(C(C)C)c3)CC2C1 c1(CC)cc(C(=O)O)sc1C.C1CCCCNC(=O)C(=O)N1 C(c1c(C)coc1C)=CC(=O)N(C1CCN(C(c2cc(CC)ncc2)=O)CC1)C CC1=NN(C)C(=O)C1CC(=O)N(C1CN(C(c2ncccn2)=O)CC1O)C Cc1cc(=NC(=O)N(CCC2CCc3ccccc32)C)[nH]n1C c1(C(N(CCC)CCNC(=O)CCC2CC2C)=O)nsc2ccccc12 C1(CC#C)(C(=O)NCCCC(=O)NCCC)CCN(C(=O)CC2CCOC2)C1 N1(C(c2c(C(C)C)scn2)=O)CC2CCCN(C(c3cc(CO)ccn3)=O)C2C1 C1(C(N2C(CO)CC(NC(Cc3c(C)nc(C)s3)=O)C2)=O)CCOCC1(C)C c1(CCC(=O)OC(C(C(=O)O)C2CCC2)C)cccc(OC(F)(F)F)c1 Cn1c(C(N2CCC(C)(NC(C3CC3C#N)=O)C2)=O)c(Cl)c2ccccc12 C1(NC(Cc2ncc(C)nc2)=O)CCN(C(=O)Cc2cc(C3CC3)no2)CC1C Cc1cc(C(F)(F)C(=O)NCCC2(CNC(C3SCCC3C)=O)CC2)cs1 N1(C(CSC)=O)CC2CCCC2(NC(=O)Cc2ccc3c(c2)OCO3)C1 c1(CNCc2cn(CCCO)nn2)noc2c1CCCCC2 c12cccc(F)c1NC2=O.N1(Cc2cn(CCC)nc2)CCOCC(O)C1 N1(C(C(C)NC(=O)CN(C2CCC2)C)=O)CCCC(C)(C)C1C C1(NC(c2[nH]nc(OC)c2Cl)=O)CCCCC12CCCN(C(c1cnsc1)=O)C2 C(=O)(C1c2c[nH]nc2CN1C(C1CC2(C1)CC(O)C2)=O)N1CC(CC(=O)OCC)C1 C(=O)(CC(=O)NCC1(C(=O)NCCOC(F)F)CCC1)OC C(=O)(C(CNC(=O)CCN=[N+]=[N-])CC(C)C)NCC1(C#C)CCC1 C1(C(N(CCN(C(CC(C)F)=O)C)C)=O)CCCC1(C)C C(=O)(C1=CC(O)CCC1)N(C)CC1CN(C(c2cscc2C(F)F)=O)CCO1 CCCC(CC)C(=O)NC1(CCCC(=O)NC2CCC(C3CC3)C2)CCC1 C1(NC(c2ccn(C)n2)=O)C2CC1N(C(C1CCC(OC(F)F)CC1)=O)C2 c1(C(C)C)cncc(C(=O)NC2CCCC2CN(C)C(c2ccc[nH]2)=O)c1 c1(C(=O)NC2CCN(C(CN(CCOC)C)=O)CC2O)ccc(F)c2occc12 N1(C(CC2N(C)CCCC2)=O)CCC(C2CN(C(C3(C)CC=CCC3)=O)C2)CC1 N1(C(c2ccc(CC)cc2N)=O)CCC2(CC1)CN(C(C1CCCN1CC)=O)C2 C1(C(N2CCC(C(C)(C)NC(=O)C=CC3CCCCC3)C2)=O)C2CCC(F)(F)C12 C1(C(=O)NC2(CF)CCN(C(C(C)SCCCC)=O)C2)CCc2nccn2C1 CC(=NO)C1CC(C(=O)NC2CCCCCN(C(=O)C#CC3CCC3)C2)C1(C)C c1(NCCCN(S(=O)(=O)CC)C)[nH]c(=NCCSC(C)(C)C)nc2c1cnn2C C(=O)(CCCCOCCC(C)=O)NCCCOCCCNCC(C)(C)NC(CC)=O Cc1n[nH]c(=NCc2ccc(-n3cncn3)cc2)o1 C1(NC(Cc2n(C)nnc2)=O)C2CCN(C(c3ccc4c(c3)OCO4)=O)CCC12 C1(NC(c2cnc(CC)[nH]2)=O)CC(OC)CN(C(c2ccc(C(C)=O)[nH]2)=O)C1 c1(C(N(C(CCNC(Cc2cc(C)nn2C)=O)C)C)=O)cccc(P(C)(C)=O)n1 C1(N(C(CN(c2ccncc2)C)=O)C)C2CN(C(c3cnc(N)cn3)=O)CC12 N1(C(=O)Cc2ccccc2)CCS(=O)CC1CO c1(OCC(N2C(C(CC)C)CCC2)=O)cccc(C)c1 C1(OCC#C)CC(N(C)N2CCOC(c3ccccc3Br)C2)C1 C#Cc1ccc(Cl)c(C(N2CCC(C3CC3)C2CNC(=O)CCOCC=C)=O)c1 Cc1cc(C)nc(N2CCC(C(=O)NC(=O)CCc3ncc(Br)cn3)C2)n1 C(CC(=O)NC1(C)CN(C(=O)Cc2ccoc2)C1)(c1cccs1)NC(C)=O N1(C(CC2N(CC)CCOC2)=O)CCN(C(c2cc[n+]([O-])cc2)=O)CC(O)C1 C1(C(N2CCC(CCNC(c3cn(C)c(O)n3)=O)C2)=O)OCC2CCCCC12 C#Cc1cc(F)c(C(=O)N(C2CN(C(C3CC4(CCCC4)CO3)=O)C2)C)c(F)c1 C(=O)(C(C(C)(C)C)NC(c1ccc(C#N)s1)=O)N(CCOCCOC)C S(=O)(=O)(c1cccc(C(=O)NCCc2n[nH]c(CO)n2)c1)N1CCN(CC)CC1 c1(C(=O)NC2CC3CN(C(C4(C)CS(=O)(=O)C4)=O)C2C3)cnn2cccc(Cl)c12 c1(C(=O)NC(C)C(c2ccc(F)c(Cl)c2)O)cnc2c(cnn2C(C)C)c1 C1(C(=O)OC)(NC(C(=O)OCCOC)=O)CC1(F)F.CCCCO.C1CO1 c1(OC)cc(Br)ccc1CNCC1CCCN(C(c2cc(Br)no2)=O)C1 c1(NC(=O)NC(CC(C)=O)C)c(F)cccc1Br CC1CCC(NC(=O)Cc2cncnc2)CN1C(=O)COc1cccc(C#N)c1 N1(C(CC2ON=C(CC)C2)=O)CC2(C1)CN(C(c1ccnc(Br)c1)=O)C2 C12(CC(N3CC(CNC(C4CSCC(=O)N4)=O)C3)=O)CCC(CC1)OC2 C1(C(=O)Nc2cncc(C(=O)OC)c2)C(C)CCCN1C(=O)Cc1csc(Cl)c1 c1(C(N2CCN(C(=O)C(N)=O)C3(CCC3)C2)=O)c(F)c(C(=O)OC)cc(F)c1F CCC(CC)CCC(=O)NC1CC1CNC(=O)CSc1ncnc2[nH]cnc12 C(c1ccccc1)=CC(=O)NCCOCC(=O)Nc1ccnn1CC1CC1 N1(C(C2(CCNC(=O)CC(O)C3CCCC3)CCC2)=O)CC2C=CCC(C2)C1 C1(C(N(CC(O)CN(C)C(C2(C3CCCO3)CC2)=O)C)=O)CCCCN1C(N)=O c1(N2CC(CN(C)CC3CCN(c4cnccn4)CC3)OCC2)cnc(C#N)cn1 CN1Cc2ccccc2C1C(=O)OC(c1cnc(C2CCc3ccccc3C2)s1)=O c1(C(N(CC(C)NC(C2(CC)CCCO2)=O)C)=O)cc2scnc2[nH]1 N1(C(=O)Cc2csc(S)n2)CCC2(CCCN(C(C3CCC4CC4CC3)=O)C2)C1 c1(CN(C(c2cnc(C3CCC3)s2)C(=O)NCCOC)C)ccc(C#N)cc1F CCC(C)(C#N)C(=O)N1CCC(CCNC(c2ncccc2CSC)=O)C1 c1(OC)ccc(C2(NC(C3(c4ccc(F)cn4)COC3)=O)CCC2)cc1 C(N=C(NC1CC1)N1CCOC2(CCCCC2)C1)C1CCC(C(=O)OCC)O1 N1(C(C=C(C)C(F)F)=O)CC(C2(NC(C3CC(c4ccc(C)cc4)C3)=O)CC2)C1 N1(CC(=O)N(CCNC(CCN(C)CCO)=O)CC2CC2)CCCNC1=O C=CCCN=C(NCc1cscc1C)N1CCC(C(=O)NC)CC1 C#Cc1c[nH]nc1C(=O)NCC(CCOC)NC(=O)C=Cc1sccc1C C1(C(=O)O)CCC(C(N2C34CC(C3)C(COC4)C(CCCC=CBr)C2)=O)CC1 Cc1ncc(C=CC(=O)NCC(C2CCCN(C(C3(CO)CCC3)=O)C2)(C)O)s1 C1(NC(C2(CC#C)CCOC2)=O)CCN(C(c2sc(CCC)nc2C)=O)CC1C C1(C(=O)OC)CC1C1CCN(C(c2cccc3o[nH]c(=N)c23)=O)CC1 N1(C(CCCOC(C)=O)=O)CC(CNC(c2cn(C)cn2)=O)CC1C C1(C)(C(N2CCC(C(C)NC(C(CC)SC)=O)C2)=O)CC(C(C)C)=NO1 C=C(F)CN=C(NC1CCCC1)N1CCC2C(C1)NC(=O)N2C c1(CNC2CCN(C(c3cc(C)c(O)cc3)=O)CC2F)cc(Br)cc(F)c1O C1(O)(CC(=O)NC(C(=O)OC)C)CCN(C(C2CC2(F)Cl)=O)CC1 c1(OC)cc(NC(C2CC3(C2)CN(c2ncc(F)c(NC)n2)C3)=O)cc(Br)n1 C(=O)(C1=CCC(C)(C)CC1)NC(CCOC)C(=O)NCc1cncn1C1CC1 C1(C(=O)NCC2(S(C)=O)CC2)CN(C(c2ccccc2F)=O)CC12CCC2 c1(CC)cc(C)c(C(=O)NCCCNC(C2(CC(F)(F)F)CC2)=O)o1 C1(C(N2CCC(OCc3cccnc3)CC2)C(=O)NCC)CC2C(C1)C2(F)F n1(CC(=O)NC(C)C(CO)NC(C2(CCF)CCC2)=O)c(O)nc2ccccc12 C1(C(=O)NCC(N2CCCC2)C)CN(C(c2ccc3c(c2)CC3)=O)C2(CCC2)C1 N1(C(CC2CCN(C(C)=O)CC2)=O)CCCC(NCCc2ccc(C)cn2)CC1 c1(C(=O)NC2CN(C(C3C(OC)C3)=O)CC2C)cc2sccc2[nH]1 N1(CC(=O)NCC2C(C(N(C)CC3(O)CCCC3)=O)C2)CCOCC1=O c1(C(c2cnccn2)C(=O)N(CCNC(=O)C(C)NC(C)=O)CC)cccnc1 c1(C(N2CCCC3(NC(C(CSC)C)=O)C(C2)C3)=O)cn(C)c(=O)n(C)c1=O Cn1c(=O)oc2c(C(=O)NCC3CN(C(=O)Cc4ccccc4O)C3)cccc12 C#CCC(CC#C)C(=O)NC1CC(CNC(C2COC(=O)O2)=O)C1 Cn1nc(C(=O)NC2CCC(CNC(=O)CC3CSC3)C2)c2cc(F)ccc12 n1(CCC(=O)NCC(CC=C)NC(=O)CCC=CBr)cccnc1=O CCC(CNC(C1CCOCC1NC(=O)CC1CC=CCN1C)=O)C(C)(F)F C1(N(C(=O)C(F)C2CCC2)CC)CCN(C(=O)CNC(=O)OC)CC1 c1(C(=O)NC(C2CN(C(=O)C(C)Sc3ccccc3)C2)C)ccc(C2CC2)cc1 C1(C(N2C(C)(C)C(CNC(=O)C3=CCCOC3)CC2)=O)CCC2(CCOCC2)O1 C=CCCCC(C(=O)NOCC)NC(=O)CC(=O)NC1CC1 c1(C(=O)NC23C(CN(C(C4ON=C(CC)C4)=O)C2)C3)ccc(C)c(S(N)(=O)=O)c1 C(=O)(CC(C)C(F)F)N1CCCC(C(=O)NC(c2nnc(C)o2)C)C1 c1(NCC2CCC(N(C(=O)CC3(C4CC4)CC3)C)CC2)c([N+](=O)[O-])cnn1C n1(CCNC2CCSC2)nnnc1C(COC1CC1)NC1CC(OC)C1 N1(C(C(C)CC(F)F)=O)CCC(N=[N+]=[N-])(C(=O)NCC2C(C)(C)C2(C)C)C1 C(=O)(C(CO)C(C)(C)C)N1C(Cn2cc(-c3nccc(C)n3)nn2)CN(C)CC1 Cn1cc(C(N2CCCCC2C(N2CCC(F)(C(N)=O)C2)=O)=O)ncc1=O CCC(C)CCCC(=O)Nc1nc(OCCC(F)Cn2cc(C(C)O)nn2)c(C)s1 C=CCCC(O)CNC(C1(N(C(c2ccn(CCC)n2)=O)C2CC2)CCC1)=O C12(NC(C3C(C=C(C)C)C3(C)C)=O)CCC(CN(C(=O)C3=C(Cl)CC3)C1)C2 C(=O)(C1=CS(=O)CCC1)N1CCC(N(C(c2n(CC)ncc2)=O)C)CC1 C(=O)(CCC(C)(C)C(=O)NCCC1CCN(C(=O)Cn2nccn2)C1)OC C1(C(C)NC(=O)C(F)=C2CCCC2)CCN(C(C2CC2c2cncn2C)=O)C1 N1(C(CC2C(CC)C2)=O)CCC(NC(c2ccsc2C(F)(F)F)=O)C1(C)C c1(COC(=O)NC(CCOC)C(N)=O)ccc(S(=O)(=O)NC(C)(C)C)s1 C1(C(=O)NC(C)C(C)(C)C)CCCCCC1NC(=O)C(C)(C)CC#N c1(CCC(=O)N(C(C(CCC)F)=O)CC2OCC3CCCC23)cc(C)cc(C)c1 C1(OC)CCCC12CCN(C(=O)C(C)CO)CC2.C12CN3CCCC3(C1)C(=O)N2 CC1CC(C(=O)Nc2cccc(C#N)n2)CCS1(=O)=O CCC(F)(C(=O)OC)C(=O)NC1CC(C)CN(C(c2cnn(C3CC3)c2C)=O)C1 CC(F)(F)CCC(=O)NC(C)(C)CCNC(=O)Cc1c(Cl)cccc1Cl N1(C(C(C(C)C)=O)=O)CC2(C(=O)NCCNS(N)(=O)=O)CC1CCO2 C1(NC(=O)Cn2ncccc2=O)CC2(C1)CN(C(=O)Cc1ccccn1)C2 C1(NC(C2(C)CC2)=O)CC2(C1)CC(NC(C1CC1c1ccc(Cl)s1)=O)C2 N1(C(CC#N)=O)CCCC(C2(NC(c3noc4c3CCCC4)=O)CC2)C1 C1(CNC(C(CC)=CC)=O)(CNC(C2CCC(C(=O)OC)C2)=O)CCOCC1 C1(F)(CNC(c2cc(C)[nH]n2)=O)CCN(C(c2nc(Cl)sc2C)=O)CC1 CCC(C(=O)NC1COCC1n1cc(C(C)OC)nn1)c1cccnc1 C(=O)(C(F)C(F)(F)F)N1C(CNC(Cn2c(C)cnc2)=O)C(C)CC1 C1(CNC(C2N(C(Cc3c(OC)cccc3)=O)CSC2)=O)CC2(CCC2O)C1 CCC(C)(COC)C(=O)NCc1c(Br)sc(C)c1C CN1CC=C(C(=O)N2C3CCC2C(CNC(=O)CCc2cncs2)C3)C1 N1(C(c2n(CC)ccn2)=O)CCC2CCC(C1)N2c1nc(C(F)(F)F)cc(C)n1 N1(C(CCn2cc(N(CC)CC)nn2)=O)CCC(C(C)O)CCc2ccccc21 C(=O)(C(CCC1CCCO1)N(C)Cc1c(C)noc1C)NCCOC C1(C(N2C(CNC(=O)COc3ccc(F)cc3)C=CC2)=O)CCC2(CCC2)CO1 C(=O)(CC(C)C(C)(C)C)NC(C(=O)N(CCCC(CC)CC)C)CCOCCO c1(OC)cc(-c2csc(C(N3C(C(=O)NS(C)(=O)=O)CC(O)C3)=O)n2)ccc1F C1(C(N2CCC(CNC(CC3C(=O)NC(=N)S3)=O)C2)=O)CCC2(CC1)CC2(F)F C(=O)(C(C(C)(F)F)c1ccccc1)N(CCC(C)NC(C1CCCCC1)=O)C N1(C(CC(C)CC(C)(C)C)=O)CCC2(CCC(NC(=O)C3=COCCO3)C2)CC1 c1(C(=O)NCC(C)N(C(c2cnsn2)=O)CC)ccnc(OCCO)c1 CC(F)(F)C(F)C(=O)N1CC(O)CC1CNC(=O)CC1CCCOC1 N1(C(c2cc(C(C)=O)on2)=O)CCCC(CNC(=O)CCc2ncccn2)(OC)C1 C(=O)(C(C)(C)COC)NC1CCN(CCCNC(c2c(CC)nc[nH]2)=O)C1 C1(NC(C(C)=C(C)C)=O)CCN(C(c2ccc(-c3ccccc3)nc2)=O)C(C)C1 C1(C(=O)NCC(COC)(O)CO)CCCCCCN1C(=O)CC1(C)CCOC1 c1(CC)cc(C(=O)NCC(C)(C)CNC(c2c(C)coc2C(C)C)=O)cc(Cl)c1 c1(C(=O)NC(C2(O)CCN(C(Cc3c(C)cco3)=O)C2)C)cc(C#N)ccc1C CC(C)C(C(C)NC(=O)C(=O)NCCc1ccc(F)cc1)NC(=O)CCCC#N n1(CC(=O)NC2CCN(C(CCC(=O)OC)=O)C2C2CC2)ccc([N+](=O)[O-])n1 Cc1ccc(CN2CC3C(C2)N3C(=O)C(=O)c2ccco2)c([N+](=O)[O-])c1 Cc1c(O)nc2ccccc2c1C(N1CC(NC(=O)CC(C)F)CCC(O)C1)=O CC(N=c1[nH]c(=N)[nH]c(=NCCc2ccc[nH]2)[nH]1)c1ncc(F)cc1F c1(C(=O)NC2CCC(NC(CC(C=C)C)=O)CC2)cccc2oc(C)nc12 c1(NC)ccc(C(=O)NC2CCCN(C(=O)CN3CCCCC3C)C2)nc1 Cc1cccc(NC(=O)COC(C)C(=O)NCCN(C)C(C)C)c1 C(=O)(CS(C)(=O)=O)N1C(CNC(C(CC2CCC2)NC(C)=O)=O)CCCC1 c1(C(=O)NC2C(NC(c3n(C)c(S)nc3)=O)CCC2)cnn(C)c1C#N S(=O)(=O)(c1cccc(Br)n1)NC1CCN(Cc2c(C)c(F)c(F)cc2)CC1(F)F Cc1nc(Cl)[nH]c(=NC2CCCCC2NC(C2(C)CCN(C)CC2)=O)c1[N+](=O)[O-] N1(C(CC2CC(C)OCC2)=O)CC2(CC(NC(C3CC4(C3)CC3(CC3)C4)=O)CO2)C1 C1(N(C(c2ccc(C#C)cc2)=O)C)CCCC2CN(C(=O)C(COC)CC)CC12 c1(N2C3CN(C(=O)Nc4c(C)c(Cl)cnc4)C(C3)C2)ncnc2ccsc12 C=C(C)CN=C(NCc1nc(Cc2ccnn2C)n[nH]1)N1CCS(=O)(=O)CC1 c1(C2CCCN2C(=O)CN(C(C)C)C(C)=O)ccc(F)cc1Cl.Cc1ncsc1C(=O)O c1(OC)cccc(NC(=O)C(C)(C2CCC2)NC(=O)CCCN=[N+]=[N-])c1F C1N=C(N2CC=C(c3cccs3)CC2)NCN2CC1CC2=O.C(C)(C)CC N1(C(c2cnc(C3CC3)s2)=O)CCC2C(CCCN2C(=O)CCc2cnc[nH]2)C1 c1(NCC(CCC)OCC)ncccc1S(=O)(=O)NC(C)COCCO c1(C(N2C(CCC(=O)NCc3nc(C4CC4)n[nH]3)CCC2)=O)ccc(O)cn1 CC(C)CCC(=O)C(=O)N1CCC1CN(C(=O)COc1cccc(F)c1)C(C)C N1(C(C(C)Cc2ccco2)=O)CC(C2CN(C(c3ccc(CC4CC4)s3)=O)C2)C1 CS(=O)(=O)c1cc(C(N2CC3(CC(NC(C4CCC45CCC5)=O)C3)C2)=O)cs1 N1(C(C2(C)COC2)=O)CCOC(CNC(c2cccc(C(C)(C)C)c2)=O)C1 C1(C(N(C2CCS(=O)(=O)C2)CC(C)C)=O)CC=CC(SCC(C)(C)C)C1 C1(NC(=O)Cc2c(Cl)cccc2Cl)CCCN(C(C2CC=CC2)=O)CC1 C1(C(N(c2ccccc2)CCNC(C2(C#C)CC2)=O)=O)CCOCC1C c1(C(=O)NCC(CN(C(C(N2CCNC2=O)C)=O)C)O)cc2sccc2s1 C1(C(=O)NC2CN(C(C(CC)CO)=O)CC3(C2)CC3)CCc2nnc(O)cc2C1 C(C(=O)NCC1CCCCO1)(C1=NOC2CC12)N(C)CC1(C)CC1 C1(CNC(=O)COCCF)CN(C(c2cncs2)=O)C2(CCC2)C1 c1(CNC2C(C)CN(CC)C2C)c(C)nc2cc(Cl)ccn12 C(=O)(CC(CCC)NC(c1ccnc(C)c1)=O)NC(CC#C)CCOC C(=O)(C(C)(C)C)NCCC(=O)NCC1C(NC(CC2CC(=C)C2)=O)C1 S(=O)(=O)(c1cccnc1NC1(CNCCO)CCCCC1)N1C(CO)CCC(C)C1 c1(C(=O)NCC2CN(C(C3CCC(F)(F)C3)=O)CC23CC3)ccc2sncc2c1 c1(ON2CCC(OCC)CC2)nc(=NCc2ncc[nH]c2=O)[nH]c2ccsc12 c1(C(N2CCCC(NC(CCOCC#C)=O)C2C)=O)cc(C)c(F)c(C)c1 c1(C(N2CCC(CCNC(C(C)c3cccs3)=O)C2)=O)ccnc(OCCO)c1 C1(C(=O)Nc2ccsc2)CC2OC1C1CC21.C12CCN(CC1)CCNC2=O N1(CC)CCOC(C(=O)NCC(CNC(c2ccnc(C(F)F)c2)=O)CO)C1 C(=O)(C(O)(CN(C)C)C(F)(F)F)NC1(CNC(CC(CC)CC)=O)CCOCC1 c1(SC)cc(C)c(C(=O)NCC(C2(O)CCN(C(=O)CCc3cn[nH]c3)C2)C)o1 C1(CCC(=O)N(C2(CCNC(CCSCCOC)=O)CC2)C2CC2)CCCOC1 c1(C(N2CCN(C(C(C(C)(C)O)F)=O)CC(O)C2)=O)c(F)ccc2ccncc12 c1(C(=O)NC(C(C)NC(CS(=O)(=O)NCC)=O)C)cccc(C)c1N CC1CCN(CC2(C(=O)NCc3c[nH]nc3C3CCN(C(N)=O)C3)CC2)CC1 C1(C(=O)NCCC2N(C(C=C(COC)C)=O)CCCC2)CC(C2CC2)=NO1 Cc1[nH]nc2ncnc(N3CCC(CF)(NC(=O)C=CSc4ccccc4)C3)c12 c1(NC(c2ccc(NC(C(CC)(F)F)=O)cc2)=O)cnc2c(c1)CNCC2 c1(C(N2CCN(C3CCN(C(c4ccsc4)=O)C3)CC2)=O)ccc(Cl)cc1F C1(C(=O)NC(C(=O)OC)CC(C)CF)CCN(S(=O)(=O)N(C)C)CC1 C1(CNC(C(n2cc(C(C)(C)C)nn2)C)=O)COCC1C(F)(F)F C(CN=c1[nH]cnc2c1COC2)N(C)C(C1CCCC(F)(F)CC1)=O c1(C(N2CCCC(CN(C(c3cc(OC)ncc3)=O)C)C2)=O)cccc(C)c1C c1(C2(C(N(CCC)C)=O)CNC2)ccccc1C N(C1CC2(CN(C(c3ns[nH]c3=O)=O)C2)n2ccnc21)C(c1cncc(Cl)c1)=O c1(C(=O)NCC23N(C(C=CCOCC#C)=O)CCC2CC3)cccc2ncccc12 c1(C(=O)NCCC(C)NC(c2cc(SC)oc2C)=O)cc(F)cc2nccnc12 C1(CC(N2CC(=C(CNC(C3CCCC3(F)F)=O)F)C2)=O)CC2(CCC2)C1 c1(C(=O)NCC2CCN(C(c3ccc(C)s3)=O)C2)cnc2ncnn2c1C CCCCC(O)C(=O)NCC12CC(CO1)N(C(=O)C=Cc1ccnn1CC)C2 c1(CC(N2C(C(=O)NCCCC(C)(C)C)CCCC2)=O)cccc(Br)c1F CN1CCN(C(=O)Cn2cc(C3CCCCC3)nn2)C1=O CC1(C(=O)NC2CCC(CCO)CC2)CC(O)CN1C(C1CC2(CCC2)C1)=O c1(C(=O)NC(CC(C)C)CN(C)C(C2CCCCO2)=O)[nH]nc([N+](=O)[O-])c1Cl C(=O)(C(CCC1CCC1)NC(C1CC=CCC1)=O)N(CC(C)C)C1CC1 C(=O)(C(Cc1ccc(O)cc1)C(F)(F)F)NCC(C)NC(CC=C=C)=O N1(C(C(c2cccc(Cl)c2)CC)=O)CCC(NC(=O)Cn2cc(Cl)c(C)n2)C(F)C1 Cc1ccc(C(=O)NCC2=CCN(C(c3snc(Cl)c3Cl)=O)CC2)nc1C N1(C(CCc2cc(OC)no2)=O)CC2CCC(C1)N2Cc1ccnc(C)n1 C(=O)(CC(CC#C)N(c1oc(C)nc1CC)Cc1ccccc1)OCC#C Cn1[nH]c(=NC(=O)C2CN(C(c3cscn3)=O)CCO2)cc1Cl C1(C(=O)NCC(CCNC(c2occ3c2CCCC3)=O)O)COC2CCCCC12 C#Cc1cncc(C(N2CCN(C(=O)C(C)OCC3CCCO3)C(C)C2)=O)c1 N1(C(C(C)OCC=C)=O)CCC2CCCC(C1)N2C(=O)CSc1ccccc1 C1(C)(C(N(CCNC(C2C(c3n(C)ccn3)C2)=O)C2CC2)=O)CC(C)(C)C1 C1(NC(CC2CCCC(C)C2)=O)CCN(C(=O)C(c2ccccc2)=O)CC12CCC2 c1(C(=O)NCC2CCCN(C(CN(C3CC3)CC)=O)C2)ccc2ncn(C)c2n1 C1(NC(CC(=O)NC)=O)CC2CC1N(C(=O)CC(C)c1ccccc1)C2 C(=O)(C(C)C(O)C(C)C)N(CCC)CCNC(c1ccc(C(F)F)cn1)=O CC1CC(CNC(=O)COc2ccccn2)CCS1 C1(C(=O)NCC2CC(OC)CN2C(C2CCCC2(C)C)=O)CN2CCN1CC2C C1(C(=O)NC(C)CN(C)C)(CNC(c2cnc(O)o2)=O)CC12CCC2 Cc1cccc2[nH]cc(C(N3CC(NC(c4csnc4Cl)=O)C4CC4C3)=O)c12 C12(C(=O)N)CCCC1CN(C(C1(O)CC1)=O)C2.C1(COC(=N)O)(C)CCC1 C(=O)(C(C)(C)C(C)(F)F)N1CC(CC(C(N2CCC(NC(=O)OC)C2)=O)F)C1 C1(C2CCCO2)(C(=O)NCC(CNC(c2cccc(C#C)c2Cl)=O)C)CCCO1 c1(-n2c(-c3csc(C(F)F)n3)nc(CC)n2)cc(C)nc(C)c1 C1(C(C)(C)NC(C(C)OCCCC)=O)CCN(C(=O)Cc2ncc(CC)[nH]2)C1 Cc1cccc(C(N2CC(O)(C(C)NC(C3CCN3S(C)(=O)=O)=O)C2)=O)c1C C12(C(=O)NCC3(C)CC(CNC(C=C(CC)CC)=O)C3)CC(C(F)(F)F)(CO1)C2 c1(OC)c(Br)cc(CC(=O)Oc2cc(C(N)=O)cc(Cl)c2)cc1Br c1(C(N2CCN(C(C(C)(C)C)=O)CC2CC(F)F)=O)ncn2c1CCCC2 C(=O)(CS(=O)(=O)CCO)N(C1CCN(C(c2csc(=N)[nH]2)=O)CC1)C N1(C(c2scc(C)c2C)=O)CC(CC(=O)NC(C2CCCCC2)CO)CC1(C)C c1(CC)[nH]c(=N)sc1C(=O)NCC1(CNC(=O)C=Cc2cnc[nH]2)CC12CCC2 c1(OCC(=O)NCC=C2CCN(C(C3C(C(C)O)C3)=O)CC2)ccc(F)c(F)c1 C=C(C)CCC(=O)NCC1(CNC(C2(CNN3CCN(C)CC3)CCCC2)=O)CC1 N1(C(CC(c2c(C)noc2C)C)=O)CC2(CCCN(C(C3CCCS3)=O)C2)C1 C=CCN=C(NCC1COCCN1CC)N1CCC(O)C(C)(C)C1 CC(C)C(C)(CNC(=O)CCC(F)F)NC(=O)CCc1cccnc1F N1(C(C2N(C(C)=O)C(=O)CC2)=O)CCC2(CC1)CN(C(C1(C#N)CCCC1)=O)C2 N1(CC(C(C)C)NC(=O)OC(C)(C)C)CCOCC2(COCCN2C)C1 N1(C(=O)CCc2ccncc2Br)CCC2(NC(=O)COC3CCOC3)CC2C1 CC(C)C(O)C(=O)N1CCC(CN(C)C(C2CCN(C(=O)C3CC3)CC2)=O)C1 Cc1cc(C(=O)NC(C2CCN(C(=O)C(c3cncn3C)O)C2)(C)C)nc(O)c1 C1(CNC(C(C)NS(CC)(=O)=O)=O)CC2(CCC2)CN1C(=O)Cn1cncn1 C1(CC)CCN(C(C2CCCCS2)=O)C(C(=O)NCCc2ncccn2)C1 C#CC12CCC(C(N3CC(CC=C)(NC(c4scc(C)c4Cl)=O)C3)=O)(CC1)CC2 Cc1cc(P(C)(C)=O)oc1C(c1ccc(F)c(Br)c1)N1CCOCC1c1nn[nH]n1 C1(C(=O)NC(C2CCCN(c3snc(COC)n3)C2)C)CCCCCCC1 C(c1ccc(SC)cc1)=CC(N1C2C(CNC(C(C)OCCOC)=O)C(C2)C1)=O N1(C(C2(C(C)C)CCC2)=O)CC(C(=O)NC2CCN(C)C(=O)C2)CC(C)(C)C1 c12ncnc3ccc1cc23.C1(CC(=O)OC)CCc2ncncc2C1 CC1C(=O)CCC1NC(=O)CC1CCN(C(=O)COC2CC2)CC1 CCCC(CNC(C1CCC(=O)N(C)C1)=O)C(=O)N1CCC(c2ccon2)C1 C(CC(C(C)C)NC(=O)C(CNC(=O)COCCCCC)CC1CC1)OC C1(C(=O)NCC(CNC(c2c(COC)nn[nH]2)=O)O)COCC2(CCC2)O1 C1(CNC(c2nc(Cl)cs2)=O)COC(CC2CCC2)C1.C12(CC1)C(=O)N(C)C2 CC1=NOC(C(=O)NCC(O)CCNC(=O)COC2(C)CCCC2)C1C C(=O)(C(CNC(CN(CCOC)C(=O)OC(C)(C)C)=O)Nc1nnsc1N)OC CCCCCC(=O)N1CC=CC1C(N1CCC(NC(=O)OC(C)(C)C)CC1)=O c1(OCC)nc(N2CC(C)(C)CC2CN(C(=O)C(CC)n2cncn2)CC)ncc1C O=C1OC(C(=O)NC2COC3(C2)CN(C(=O)CCC(F)F)C3)Cc2ccccc21 C(c1cnc[nH]1)=C(C)C(=O)NCC(C)CNC(C1(c2ccno2)CC1)=O c1(CC(N2CCC(OC)(NC(C(CO)OC)=O)C2)=O)ccc(Cl)c2cccnc12 C(=O)(C#CC1CCCCC1)NC(CC=C)CNC(=O)Cc1cncnc1 C12(CNC(C(CC)SC)=O)CCC(CC1NC(=O)Cn1cnccc1=O)C2 C(CCCCC(=O)NCCCN1CCN(C(C23C=CC(CC2)C3)=O)CC1)SC CC1CC(C(=O)N(CC(N)=O)CC(N)=O)N(C(=O)CCCn2cncn2)C1 C1(NC(CCNC(C)=O)=O)CCN(C(=O)CSc2cnn(C)c2)CC(O)C1 C1(O)(CC(N2C(C(C)NC(c3csc(Br)n3)=O)CCC2)=O)CCCCC1 Cc1cc(CCCC(=O)NCCC2CCN(C(=O)C(C)N(C)C)C2)on1 c1(C(=O)NCC(O)C(=O)NCc2cnns2)ccc(F)c(O)c1 C1(CCC(=O)NCc2cc[nH]c2C(=O)N(CCCO)C2CC2)CCCOC1 CC(C)(CS(C)(=O)=O)C(=O)NC1(C2CN(C(C3CC(C(F)(F)F)C3)=O)C2)CC1 C=CCCC(C)(C)C(=O)NCC1C=CC(NC(=O)CCN(C2CC2)CC)C1 c1(C(N2CC(NC(CCCOCC)=O)C(C)C2)=O)csc2c1CCCC2 CC(C)C(C(=O)N(CC(C)NC(C1(F)CC1c1ccccc1)=O)C)N(C)C c1(C(=O)NC(C(CO)NC(CC2CCN(CC)C2)=O)C)cccc(OC(F)F)c1 Cc1cnc(C(=O)N(CC(=O)NCCS(C)(=N)=O)CC(C)C)c(F)c1 c1(CNC(CCN(C(=O)C(O)C=C)CC#C)=O)cccc(C)c1C c1(N2CC(CN(C)C(c3csnc3Cl)=O)OCC2)ncc([N+](=O)[O-])cc1C(N)=O CCCC(C(=O)N1CC2(NC(=O)Cc3cc(SCC)nn3C)CC1C2)NC(N)=O c1(OCCCC)ccc(C(C)NC(c2ccccn2)C)cc1OC C(=O)(C(C(C)(C)O)NC(=O)C(C)N1CC(C)C1)N(C1CC(C#N)C1)CC#C N1(CC(N2C(CNC(C3CC3(F)F)=O)C=CC2)=O)CCCC2(CC2)S1(=O)=O N1(C(c2c(CC)nns2)=O)CCC(O)(CCNC(c2ccc(CSC)cn2)=O)C1 c1(OC)ccc(C(N2CCN(C(=O)COC(C)(C)CC)C(C)C2)=O)c(C)c1 C1(N(C)C(c2cccc(OC(C)(C)C)c2)=O)CC12CCN(CC1CCNC1)CC2 C1(CNc2occ(CC)n2)CN(C(c2cnn(CC3CC3)c2)=O)CC1N(C)C N1(c2ncc(C)c(C)n2)CC2CCCN(C(=O)CCc3ccccn3)C2C1 C(=O)(C(CNC(=O)Cn1ccc(C)n1)C(C)C)N(C(COC)C)C N1(C(CN(C(=O)C(n2nccc2C)C)CC#C)=O)CCC(F)(C(=O)OC)CC1 N1(C(C=Cc2c(C)ncs2)=O)CCCC(NC(C2(O)CC2)=O)C1C C=C(Br)CCC(=O)NC1COCCC1NC(=O)CN1CCCCC1 c1(CN2C(CC(=O)Nc3cc(OC)c(O)cc3)CCC2)cc([N+](=O)[O-])ccc1F CC(C)(C)C(O)C(=O)N1CCCC1(C)CNC(=O)C(C1CCCCCC1)O CCC(C)(C)CC(=O)NCC(C)(C(C)C)NC(=O)Cc1ncc(Cl)s1 C(CC(C)C)(C(=O)NCC1NC(=O)NC1=O)ONC(C(c1cc(C)[nH]n1)C)=O c1(C(=O)NCC(CNC(C(COC)OC)=O)(C)F)cc(C)c(C)c(C)c1 N1(C(CCc2onc(C)n2)=O)CC2CC1CN2C(=O)C(C1CCC(=O)N1)C c1(C(=O)NCCCC(CO)NC(C2(c3ccsc3)CC2)=O)cccc([N+](=O)[O-])c1 c1(OC)ccnc(OC)c1S(=O)(=O)N1CCC(S(N)(=O)=O)CC1 c1(C(=O)NC2CN(C(CCOC(C)=O)=O)CC(O)C2)[nH]c2ccccc2c1Cl c1(C(N(C)CC2(O)CCCN(C(=O)COCC(N)=O)C2)=O)cc(S(N)(=O)=O)c[nH]1 C1(CN2C3CN(C(=O)CC4=CCCC4)CC2C3)CCc2cncn2C1.c12cn(nn1)C2 C1(F)(CNC(C2(C)CCC(C)C2)=O)CCCN(C(C2CC3(C2)CC(O)C3)=O)C1 N1(C(C2N(CC)CCCC2)=O)CCC(NC(=O)CC2(N(C)C)CCC2)C(F)C1 C1(NC(C2CCCS2)=O)CCC2(CC1)CN(C(C13CCCC1(CO)C3)=O)CCO2 N1(C(COCCC)=O)CCC(C)N(C(=O)CC(O)C(C)CC)CC1 c1(C(C(=O)NCC2CCN(C(CC=C)=O)C2)(F)F)ccccc1Cl N1(C(C(C)C2CC2)=O)CC(N(C)C(c2ccc(CN3CCOCC3)o2)=O)C(F)C1 C1(C(=O)NCC(=O)N(CCC(N2CCCCC2C2(SC)CC2)=O)C)CN2CCC1C2 C1(C(=O)Nc2cnc(OC)c(Br)c2C)CC1N=c1ncc2c(O)n(C)cc2[nH]1 C1(C(N(CCNC(c2c(C(C)C)ccs2)=O)CC2CC2)=O)CCCC1S(C)(=O)=O c1(C(=O)NC)cc(C)cc(S(=O)(=O)N2CCN(C(C3CCCCC3)=O)CC2)c1 C1(NC(C2(COC(C)C)CC2)=O)CC(O)CN(C(=O)CCCC(C)=O)C1 c1(C(c2cc(CC3CCCC3)on2)=O)cccc(C2(CO)N=N2)c1 c1(C(=O)NCCC2CN(C(C(CC)OCC)=O)CC2C)c[nH]c2cc(F)ccc12 CC(C)C(CNC(=O)Cc1cc[nH]n1)NC(c1c[nH]nc1-c1ccco1)=O Cc1cc(C(=O)NC2COCCC2NC(C2CC2C)=O)nn1-c1cccc(Cl)c1 CCC(CCCC(=O)N1CC(C)=CC(C)C1)NC(c1cn(CC)nn1)=O Cc1cc(C)cc(C=CC(=O)NC(C)C(C(C)C)NC(c2nscc2N)=O)c1 C1(C(=O)NCCN(C)C(c2ncccc2N)=O)CC2CCC(C1)S2(=O)=O c1(C(=O)NCc2nc(CNC(=O)C=C3CC3)nc(O)c2)cnn2cc[nH]c(=O)c12 c1(C(N(C)CC2(O)CN(C(CCC#CC)=O)C2)=O)cc([N+](=O)[O-])oc1C C#CCC(C)C(=O)NC1(CN2CCN(C(C3(O)CC3(C)C)=O)CC2)CC1 C1(N(C(C2N(CCC)CCC2)=O)C)CCC(CNC(c2ncccc2Cl)=O)CC1 c1(C(N(C2CCN(Cc3ccn(C)n3)C2)CC)=O)c(F)cccc1F C1(c2nnc(N3CC(=O)NC3=O)o2)CC2CCC(C1)N2C(=O)C(O)(C1CC1)C1CC1 N1(C(c2c(CC)c[nH]c2)=O)CC(NC(c2ccc(CSC)o2)=O)CC(C)C1 CCC(C)(C(=O)NCC1CCCCN1C(=O)COCc1ccncc1)C(F)F CONC(=O)C(=O)N1CC(=O)CC1C(=O)NCc1c(F)cncc1F C1(OC)CCC2(CCN(C(C3CCSCC3)C(=O)Nc3c(C)cccc3C)C2)C1 S(=O)(=O)(c1cccc(Br)n1)N1CCC2(C(C(=O)Nc3cncc(Br)c3Cl)C2)C1 N1(C(C(C=C)O)=O)CC(NC(=O)CSc2ccc(F)cc2)C2(CCC2)C1 C(N=c1[nH]cnc2c1COC2)C1CN(C(CC2(CC=C)CCCC2)=O)CC1C CCC(CCCC(=O)NC1(c2ncc[nH]2)CC1)NC(=O)C=CC1CCOC1 c1(C(N2CCC(F)(C(=O)NCC=CCCC)CC2)=O)ccc2c[nH]nc2c1 C1(CC(=O)N(CCC(=O)NCCCSC(F)F)CCCO)CCC(=O)O1 C1(CNC(=O)CCCCOC)CN(C)CCN1C(c1sc(C(=O)OC)c(N)c1)=O c1(-c2c(N(CC)CSC)cc(NCC)cc2)c(C)nc(C(C)(C)C)nc1C C1(=O)C(F)CC2CC(C2)N1.C1(C(CC)NC(=O)C(F)C2CCC2)CCCOC1 C(=O)(C1(C)CCn2c(C)nnc21)NCC(CN(C(C(C=C)O)=O)C)(C)C N1(Cc2ccc(OC)nc2)CCC2CN(C(c3cccnc3)=O)CCC12 C1(CC(=O)N(C2CC(CNC(=O)CCCOc3cccnc3)C2)C)CCC(=O)N1 c1(-c2n(NCCSC)c(N3CC4CCC3C4)nn2)cnn2c1CCCC2C Cn1ccc(C(N2CCN(CC(N)=O)CC2)C(=O)NCc2ccco2)c1C1CC1 CC1CC(NC(=O)Cn2[nH]cnc2=N)CN(C(C2(N(C)C)CCCCC2)=O)C1 C(c1cccc(Cl)c1)=CC(=O)NC(CC)CN(C(=O)CCC(=O)N(C)C)C n1(CCCOC)cc(C(=O)N(CC(CC)NC(=O)C(C2CC2)C2CC2)C)cn1 N1(C(COC(C)C)=O)CC2(NC(=O)C(c3cc(F)cc(Cl)c3)=O)CCCC2(F)C1 c1(C(=O)NCCCCCNC(C2(CN(C)C)CC2)=O)cnc(O)c2ncccc12 N1(C(C(CCOC)OC)=O)CCC2CCC(C1)N2C(=O)Cc1ccn(C(C)C)n1 C(=O)(C(CNC(=O)CCc1cccs1)CC(C)C)N(CCC)CC1CC1 c1(C(=O)NC(CNC(C2C(C(=O)OC)C2)=O)C2CC2)cc2cc(Cl)cnc2[nH]1 CCCCC(CC)C(=O)N1CCCCC1CN(C(=O)COC)CC N1(C(C=CC)=O)CCCCC1CN(C(=O)CC1CSCCS1)C CC12CCC(C(=O)NCC3CC(NC(c4[nH]ccc4C4CC4)=O)C3)(C1)OC2 N1(C(C(CC)COC)=O)CCC2(CCC2)C(NC(c2cccc(CF)c2)=O)C1 CC(CNC1CCC1)C(=O)NCC1CC(NC(c2cnc(CC3CC3)s2)=O)C1 c1(CC)ccc(C(=O)NC(CO)CCCCNC(C2CC(C3CC3)C2)=O)c(C)c1 C(=O)(CC(C)(C)COCCOC)NC1(CC)CCN(C(=O)CCn2ccnc2)C1 Cc1cn2nc(C(N3CCC(NC(=O)C(C)CC4CC4)CC3)=O)cc(C)c2n1 CC(C)C(C(=O)N(C1CN(C)C1)C(C)C)NC(=O)Cc1cscn1 c1(C(C)OC)nc(C)c(C(=O)NC2CCN(C(=O)CCC(C)OC(C)C)C2C)s1 C(=O)(C1=CC2CCC(C1)C2)N1CCC(C)(NC(c2cc(OC)no2)=O)CC1 N1(C(C2C(C)=C2)=O)CCC(N(C(=O)CC2(C(F)(F)F)CC2)C)C1 c1(NC(C2C(COC)CCCC2)=O)ccc2c(c1)N(C)C(=O)CO2 C(N=c1[nH]c(=NC2CCC(CO)CC2)c2sccc2[nH]1)C1C(C)(C)CC(=O)N1 N#Cc1nc(Cl)ccc1NC(C1CC(F)CN1C(=O)CCN1CCCCC1)=O C1(NC(c2cncs2)=O)CCN(C(=O)NOC2CCC2)O1 C1C(C)C(=O)O1.C(C)(CCNC(N(CCOCCC)C)=O)OC(C)(C)C c1(C(=O)NCCCN(C(CC2CC(OCC)C2)=O)C2CC2)ccc2cncn2c1 c1(NC(C)=O)cccc(F)c1C(=O)NC1CC1NC(=O)C=Cc1cnn(C)c1 C(=O)(C1Cc2ccccc21)N1CCCC(CCNC(c2[nH]c(=N)sc2C)=O)C1 O=C1CC(CC(=O)NCC2CCCCN2C(=O)CNC(c2cnc[nH]2)=O)C(=O)N1 Cc1nc(C(N2CCC=C(C(=O)N(C)CP(C)(C)=O)C2)=O)ccc1C#N c1(C2C(C(=O)NCCCN(CCC#C)CC)C2)cccnc1OC N1(C(CNC(COCC#C)=O)=O)CCC1CF C1(NC(C2(C3CCCC3)CCNC2=O)=O)CC1C1CCCN(C(C2SCCS2)=O)C1 c1(C(=O)NC(CNC(c2[nH]cc(C)c2)=O)C(C)C)nnc(O)nc1O c1(SC(C)COCc2noc(C(F)(F)F)n2)ccccc1Cl CC(C)CC(C(=O)NCC(C)NC(c1ccc(C2CC2)o1)=O)C(N)=O CC1OCCC1CC(=O)NCC(=O)NCC1CCCS1 c1(SC)ccc(O)c(C(=O)N(C)CC2CN(C(c3n[nH]c(C)c3C)=O)C2)c1 Cc1cc(Cl)cc(C)c1OCC(N1C2CCC1CC(NC(=O)CCC(C)C)C2)=O c1(C(=O)NC2C(C(=O)NCC(C)F)C2)ccc2cnn(C)c2c1 N1(C(C=CSC)=O)CCC(C)C(CNC(=O)Cn2nnnc2C2CC2)C1 Nc1cc(C(N2CCCCCC2CNC(=O)C=CCO)=O)cc(Cl)n1 C(=O)(CCCCc1ccc(F)cc1)N1CC(CC(C)NC(C2CC2C)=O)C1 c1(C(=O)NCC2CC(OC)CN2C(c2ccsc2)=O)ccc([N+](=O)[O-])[nH]1 c1(OC)nc(C)ncc1C(=O)NC(CNC(C12CC(F)C1C2)=O)C(C)(C)C C1(CC)CCN(C(=O)C=NOC)C1CNC(=O)CNc1cccnc1 c1(C(C(=O)N2CC(N(C(C3CC(OC)C3)=O)C)C2)(C)C)ccc(Cl)c(Cl)c1 C1(N(C)C)CC2(CCC(C(=O)NC3CC(C)(NC(C4(N(C)C)CCC4)=O)C3)CC2)C1 c1(C(C)NC(N2CCCC(CO)C2)=O)nccc(O)n1 Cc1cnc(C)c(C(=O)NCC2CN(C(=O)CCOC3CCOCC3)CCO2)c1 C(=O)(CCC(CF)CF)NC(C(=O)N(C)Cc1snc(C)n1)(C)C1CCC1 c1(SC=CC(=O)NCCN(C(c2cn(CCOC)nn2)=O)CC)cccc(C#N)c1 N#Cc1cccc(OCC(=O)NCCN(C(=O)C=CC2CCCO2)CC2CC2)c1 c1(C(=O)NCC2C(C)CN(C(=O)CN3CCOCC3)C2)cc(C(N)=O)cc(F)c1 N1(C(C(C)SCCCC)=O)CCOCC2(COCCN2C(c2coc(O)n2)=O)C1 n1(CCC(=O)N(C2C3CN(C(C(CCC)O)=O)CC32)C)ccc(O)nc1=O C1(C(=O)NC(c2ccccc2)C#C)CC(C(=O)O)N(C(=O)OC(C)(C)C)C1 CC1CCCC=C1c1ccc2[nH]c(C(N3CCCCC3C(C)(C)O)=O)cc2c1 c1(OC)ccc(CN2CCC(C)CC2)c(C)c1C.c12ncccc1CN2 C1(CC(=O)NCC2(C)CN(C(Cc3cnc(C)s3)=O)C2)CCCCC1(F)F C#CCC(CC(=O)N(C)OC1CCCC1)NC(=O)C(=O)N(C)C c1(NC)cc2c(cc1S(=O)(=O)NC(C1CCN(CCOC)CC1)=O)CCC2 CN1N=CC(CC(=O)NCC2CC(C(=O)NC3CCCC(CO)C3)CO2)C1=O Cc1cc(C#N)sc1C(N1CCC(N(C(=O)Cc2cocn2)C)C1)=O CC1(C)COCC1(CO)Nc1ccc(-c2ccccn2)nc1 c1(OC)ccc(C(=O)NC(CNC(c2csnc2C)=O)C2CC2)c(F)n1 N1(C(C(C)=CC2CC2)=O)CC(CNC(c2nccnc2N)=O)C2(CC2)C1 CC1(C)OCC2CC12CN.c1(O)ccccc1Cl Cc1nc(N)cnc1C(=O)NCC1CCCC(CNC(c2csc(C#N)c2)=O)C1 N1(C(C(C#N)=CC(C)C)=O)CCC(C)(C)C(CNC(C2CCOC(C)C2)=O)C1 C#CCC(CC#C)C(=O)N1C2CCC1CC(N(C)C(C1CC(F)C(=O)N1)=O)C2 N1(C(c2n(C(C)C)ccn2)=O)CC(C(=O)NCC(O)C(F)F)CC(C)C1 CC1(C#CC(=O)N2CC(O)CC2C(=O)NCC2CC2(F)F)COC1 CC(C(=O)NCC1CCC1NC(=O)CCC1CC1)c1cc[nH]n1 c1(C(CCO)Nc2c([N+](=O)[O-])cccc2)ccc([N+](=O)[O-])cc1Cl N1(C(CC#C)=O)CC(C(=O)NOCc2cc(Cl)n(Cc3ccccc3)n2)C(F)C1 N1(C(C(c2ccc(OC)cc2)C)=O)CCC(NC(=O)C(C)=C(C)C)C(C)(C)C1 C1(CNC(C(C2CC2)SC)=O)CCN(C(=O)Cc2cnc(Cl)s2)C1 c1(C(N2CCC(NC(C(Br)=C(C)C)=O)C2(C)C)=O)cc(O)cc(C#N)c1 C#CC(C1CCc2ccccc21)NC(=NCCCCl)NCCC1(O)CCOC1 C1(CNC(C(C)OCC(C)C)=O)C2CN(Cc3ncnn3C)CC12 C1(CN(C(c2c(C)cns2)=O)C)C2CN(C(c3c[nH]nc3C3CCCO3)=O)CC12 C12(C(=O)Nc3c(C)nsc3)CC(CO1)N(C(=O)Cn1cc(C#N)cn1)C2 c1(OC)ncnc(OC)c1C(=O)NCCC1CN(C(c2cnsn2)=O)CC1C c1(C(=O)NCC(c2ccccc2)CNC(C=NOC)=O)ccc2nccnc2n1 c1(C(N2CCC(CN(C(C(C3CCC3)OC)=O)C)C2)=O)cc(Br)n(C)c1 Cc1cccc(C(N2CC=CC(NC(=O)Cc3ccoc3C)C2)=O)c1N C(=O)(C(F)(F)C(F)F)N1C(C(=O)NC2CC(Cl)(Cl)C2)CC2CC21 n1(CC)cnc2nc(=NC(C)c3ccccc3Br)[nH]c(N3CCC(C)(CCO)C3)c12 O=C(C1=CC2(CCOC2)C1)NCn1cc(C(=O)NCC2CC2)nn1.C1CCCC2CC12 C1(COC)CN(C(c2cc(N)ccn2)=O)CCN1C(c1sncc1C)=O [N-]=[N+]=NCC(F)(F)CCC(=O)N1CCC2(CC1)CC(CO)C2 c1(NC2C(C(N3CC(C)OC(C)C3)=O)CCCC2)nc2c(cc1C#N)CCC2 C1(C(=O)NCC(C)(C)CNC(C2CCCSC2)=O)COCCN1CC1CCC1 N1(C(C(CC)=CCCC)=O)CCC(O)(CN(C(=O)C=CCN2CCCCC2)C)C1 C1(NC(C(CSC)C)=O)CC2(C1)CC2NC(=O)CCC(=O)c1ccncc1 C1(CCOC)CN(C(C2CCS(=O)(=O)C2)=O)CCN1C(C1CS(=O)(=O)C1)=O c1(C(N2CCC(C(=O)NC3CCNC3=O)(OC)C2)=O)nnc(O)nc1O C12(C(=O)NCC3CN(C(c4c(C)ncs4)=O)C3)CCC(CC1)C(C)(C)O2 c1(C(N2CCC(O)(CNC(Cn3c(C)ccn3)=O)C2)=O)ccc2ncn(C)c2n1 C1(O)(C(C)NC(=O)C2=CCSC2)CCN(C(c2cc(C3CCOC3)[nH]n2)=O)CC1 CCCC(C)(C)C(=O)N1CC2CC2(CNC(c2cc(C)ccc2SC)=O)C1 C#CCCN=C(NCC1CC2CCC1CC2)NC1CCCCC1C c1(C(N2CC(CC)C(NC(=O)C(C)SC)C2)=O)cc(C)c2n[nH]cc2c1 C(=O)(C1=C(Cl)CCC1)NCC(CC)NC(=O)C(Cc1ccccc1)N(C)C Cc1[nH]nc(C(=O)N(CC(O)CNC(C2CC2c2ccn(C)n2)=O)C2CC2)c1C Cc1c(C(=O)NC2CCCC2CNC(=O)CC=CC(C)(C)C)sc2ccccc12 c1(OC)ccc(C(=O)NC2(C3CN(C(c4ccnc(C)n4)=O)C3)CC2)c(F)c1N N1(C(C(NOC)=O)=O)CC2(C=C(C(=O)NCCC(C(C)C)OC)CO2)C1 N1(C(C2(C)CCC2)=O)CC=C(CNC(C2Cc3nnsc3S2)=O)CC1 CCCC(C#N)C(=O)NCC1CN(C(=O)C=C(Cl)Cl)CC1C CC1(C)COCCC1CNC(C1CC(=O)CN1C(=O)CN1CCSCC1)=O C(=O)(CC(C)(O)CCC)NC1CCC(CNC(C(C)SCCCC)=O)CC1 C1(NC(C2(C)CC=CCC2)=O)CCN(C(c2cc(O)ccc2Cl)=O)CC1F N1(Cc2nc(C)[nH]n2)CCC2CN(C(=O)Cc3cccc(Cl)c3)CC2C1 C1(N(C)C(c2cc(C3CC3)ns2)=O)CN(C(C2(N(C)C)CCOC2)=O)CC12CC2 C1(OC)CCC(C(N2CCSCC2C(=O)Nc2cccnc2SC)=O)CC1 c1(C(=O)NCC(CNC(c2ccc3scnc3c2)=O)O)cc2c(Cl)ccnc2s1 c1(C(=O)NCCC2(O)CN(C(c3cnc(C(C)(C)C)s3)=O)C2)ccc([N+](=O)[O-])o1 S(=O)(=O)(c1ccc(C(=O)NC2CCCC2NC(=O)COC2(C)CCCC2)o1)NC C(=O)(C(C)(O)C(F)(F)F)NCCCC1N(C(C2CCN(CC)C2)=O)CCCC1 c1(C(=O)NCC#CCNC(C(CC=C)C)=O)cc2c(=O)[nH]c(C)cn2n1 N1(C(CC(=O)NCC)=O)CCC2(NC(=O)Cc3cc(F)ccc3O)CC2C1 C1(NC(c2cccc(C(=O)NC)n2)=O)CCCN(C(C)C(=O)NC)CC1 C12(OC)CCC(C(=O)NC(C)(C)C(C)NC(C3C4CCCOC34)=O)(CC1)C(=O)C2 N1(C(c2cnc(COC)s2)=O)CCC2(C1)CN(C(c1ccno1)=O)CCO2 C1(CC(=O)NC2(CCC)CCNC2=O)CN(C(c2c[nH]nc2CC)=O)CCC1C N1(C(C(N)=O)=O)CCC(CC(N)=O)(NC(C2CCCNC2=O)=O)CC1 C(=O)(CCCS(=O)(=O)N1CCCC1)NC.CC1CCC=C1C(=O)NC1CN(C(=O)C)C1 C1(NC(CNC(CCC)=O)=O)CCCC12CN(C(C1(C(F)(F)F)CC1)=O)C2 C1(CNC(CC)=O)CC(F)(F)CN1C(=O)C(C)C(F)(F)F Cc1ccnc(C(N2C(C(=O)N(C)Cc3cccc(O)n3)CCC2C)=O)c1F n1(CC(=O)NCC(CNC(CC2C(C)(C)C2)=O)O)ccc(C(F)F)n1 N1(C(C=CC)=O)CC(C)(C)OCC1CC.c1(N2C3(CC3)C2=O)ccc(C)c(C)c1 C1(C(N(CCCCC=C)CC)=O)COC2(CCC2)C1O CC1CCN(C(c2ns[nH]c2=O)=O)C1C(=O)NCCc1cocn1 CC(C)C(C)(CNC(c1cc(C2CCC2)no1)=O)NC(C1CC(F)(F)C1)=O CC(CCNC(C1CCN(C(c2ncccn2)=O)C1(C)C)=O)C(C)(C)C c12cccc(c1)NCCN2c1ccc(C)cc1.c1(C(=O)OCC)cc(C)cs1 C1(N(C(C=CCCC)=O)CC)C2CCCN(C(=O)CC3(C(F)(F)F)CC3)C2C1(C)C c1(C(=O)NC(CCOC)C(=O)NCCN2CCC2)c(C)cncc1C C12(CCC(=O)OC)CC3(CC(C3)CC3C(CCCC3)N1)C2.c1(SC)nnc(C)n1C Cc1cccc(CC(=O)NC2CCC2NC(C23CC(F)(C2)C3)=O)c1Br C=CC1CN(C(=O)C(C)(CC)CO)CC1NC(c1c[nH]ccc1=O)=O C(=O)(C#CC1(C)CCCO1)N1C(CNC(C#CC(C)(C)C)=O)CC(OC2CC2)C1 C(CCC(C(=O)NC1CCCCCC1C)NC(=O)Cc1ncn(C)c1C)OC c1(NC(C=CC)=O)ccc2c(c1)C1CN(C(c3sccc3Cl)=O)CC1NC2=O c1(NC(C2(F)CCN(C(CCSC)=O)C2)=O)c(C#N)cnn1-c1ccc(Cl)cc1 Cc1ccc(CCNC(c2nnnn2C)(C2CCOC2)C)c(F)c1 C1(C(N2CC(NC(c3c(OC(C)C)ccnc3)=O)C2)=O)C2Cc3ccccc3C12 Cc1nc(NC2CCCCC2NC(=O)CCF)c2c3c(sc2n1)CCCCC3 CC1CCN(N2CCCC2CC#N)CC1OC(F)(F)F c1(C(C)=O)cc(C(N2CCC(C)C2c2cn(Cc3cocn3)nn2)=O)ccc1C C1(C(=O)NC2CN(C(c3c(OC)scc3)=O)CC2F)CC2(C1)CC(CO)C2 C#CC1(O)CCCN(C(=O)CNC(=O)CN(C(=O)CCC2CCCOC2)CC)C1 c1(N2C(C3(NC(C4C(OC)(OC)CC4)=O)CC3)CCCC2)cc2nncn2cn1 C1(C(N2CCC(NC(c3n(CC)c(O)nc3)=O)C2C(C)C)=O)COC(C)(C)CO1 c1(CNC(c2ccn(CCNC(c3csnn3)=O)c2)=O)cnc(C2CC2)nc1 N(C(=NCCCn1cncn1)N1CCC(Oc2ccncc2)C1)CCF c1(C(=O)NC(CC)(C)CNC(=O)CCNC(C)=O)ccc(C(F)(F)F)cc1C CCC(CC)C(C(=O)N1CC(F)CC1CC(=O)NCc1nc(C#N)cs1)OC c1(NCCNC2CCCN(C(c3cc(C)c(O)nc3)=O)C2)cn(C)c(=O)cc1C Cn1nccc1C(=O)NC1CCN(N2CCCC2)C1.c12cn(nn1)CC(=O)N2 C1(C(=O)NCCN(C(c2c(CC)oc(Br)c2)=O)CC)CC(C)CC(C)(C)C1 N1(C(C2CC(CF)C2)=O)CCN(C(=O)CCC2CC2(F)F)C(CC(F)F)C1 C1(C(=O)NCC2C(CNC(=O)Cc3cnoc3)C2)CCCCC1(F)F C1(CNC(C2C(C)(C)C2C(=O)NCCCCc2nccs2)=O)CCC(O)CC1 c1(C2C(C(N(CCC)CCNC(C3C=CCC3)=O)=O)C2)ccc(Cl)cc1 N1(C(=O)OCC)CC2C=CC1C(C(N1CC(O)(COCc3cc(CC)no3)C1)=O)C2 C(=O)(C1=C(Cl)CCOC1)NC(CNC(C1CC2C(C)(C)C2C1)=O)(C)C1CCC1 S(=O)(=O)(c1ccc(Cl)c(O)c1)N1C(C)(C)COC(C(F)(F)F)C1 c1(C(=O)OCC)ccc(C(=O)NCCCCCNC(c2cn(C)nc2C)=O)nc1 c1(C(=O)NC(CC(=O)NC(CC)CSC)(C)C)cc(O)cc(F)c1 c1(C(N(C)CC2(O)CCCN(C(CCN(C)CC)=O)C2)=O)c(C)ccc(Cl)c1F C1(CC(=O)NCC(C)(CO)NC(CC(CC)C)=O)CCN(OC)CC1 C(C(=O)NCCC1CCCN1C(c1cc(C)c(Br)o1)=O)(C(C)(C)C)OC C1(C)(C(=O)NCC(C)C(=O)NCC2(O)CC3C=CC2C3)CC(C#N)C1 N1(C(c2cc(C)ncn2)=O)CCC2CN(C(=O)Cn3cc(C4CCC4)nn3)CC12 N1(C(CC2(C=C)CC2)=O)CCC(F)(CNC(=O)C(F)(F)c2cccnc2)C1 C(=O)(C1c2c[nH]nc2CN1C(=O)CC(CC)C1CC1)N(CCOCC)CC C=CCN=c1[nH]cc(C(N2CC=CC2CNC(=O)CCCOC)=O)s1 c1(CC(C=O)NC(C)=O)ccc(Br)cc1.C(C(N)C1CC1)NC(N)=O O=C(NN1CCCC1C(N1CCC2CC1C(=O)O2)=O)c1ncc(F)cn1 Cc1cc(C(=O)OC2CN(Cc3cnn(-c4ccccn4)c3)C2)c(Cl)cc1F C1(CNC(Cc2cccc(C(C)C)c2)=O)CN(C(=O)CC2CC2C)CCC1C C=CCCCCCCCCC(=O)NC1CCC2CC1CN2C(=O)CCC(=C)Cl C#CCCC(C(=O)NCCC1CCCO1)NC(=O)CCOC(C)C CCC(C(C)(F)F)NC(c1conc1C(C)NC(=O)CCc1ccccc1)=O c1(C(=O)NC(CNC(CCCCC#C)=O)(C)CC)cc2cc(F)ccc2[nH]c1=O c1(OC)ccc(Cl)c(C(N2CC(O)(CCNC(=O)C(C)CN(C)C)C2)=O)c1N C(=O)(CS(=O)(=O)C1CCCC1)NC1CN(C(C=C(C)C(C)C)=O)C2C1C2 C12(C(=O)NCC(CN(C(C=C(C)C(C)C)=O)C)O)CCN(CC1)CC2 C12(C(=O)NC3(CC=C)CCN(C(C4C5CC(=O)CC45)=O)C3)CCN(CC1)CC2 N1(C(CCC2CC(CC)C2)=O)CC(CC(=O)N(CCC(O)CO)C)CC1(C)C c1(C(=O)NC2CN(C(c3cc(CC)nn3C)=O)CC(O)C2)cc2ncccc2s1 Cc1cc(C)c(C(=O)NC(C)C(C(C)C)NC(c2[nH]nnc2C)=O)o1 C1(NC(C2(OC)CCSC2)=O)CC(NC(=O)C(=O)NC2CC2)C(O)C1 c1(C(=O)NC2(C)CCN(C(C3(SC)CC(O)C3)=O)C2)ccc2cnoc2c1 CCC(F)(F)C(=O)NC1CC1CNC(=O)CCCOc1ccccc1Br C1(C(=O)NC2CCC(NC(CCNC(c3ccccc3)=O)=O)C2)COCCOC1 Cc1cccc(C(O)C(=O)NC(C2CCN(C(C3(C4CC4)CC3)=O)CC2)C)c1F N1(C(C=C(C)C)=O)CC(NC(c2c[nH]c(=N)o2)=O)CC1C N1(C(COCc2nnc(C)s2)=O)CCC(C)(C)C(CNC(=O)O)C1.n1(CC)cncn1 C1(Cc2c(-c3onc(C(C)C)n3)cc(Br)o2)CCCC1P(C)(C)=O CCCC(O)(CCC)CC(=O)NC1CN(C(c2oc(CC)cc2C)=O)CC1CC Cc1ncnc(C)c1C(=O)N(CC(C)(C)NC(C1CS(=O)C1)=O)C c1(C(C)NC(c2cc(C(=O)O)cc(Cl)c2)C)ccc2c(c1)CC(=O)N2C C(c1cc(Cl)sc1Cl)=CC(c1nc(CC2CCCC2)no1)(C)C C#CCCCCCC(=O)NC1CC(C)CN(C(C2CCCN2C(N)=O)=O)C1 CCC(C)(CC)C(=O)NC1CCCN(C(=O)C(C)SCc2ccccn2)C1 c1(N2CCC(NC(C3=CCN(C)C3)=O)C(C)(C)C2)ncnn2c(Br)ccc12 C(=O)(CCC(C)(C)F)N(CCC(C)NC(C1(C)CC2CCC1O2)=O)C c1(CC)ncc(C(N2CC(=C(F)CNC(C3CC(OC)C3)=O)C2)=O)s1 C1(O)(C(=O)NCCN(C(=O)C(C)CC2CCC2)CCOC)CCCCCC1 c1(N(C2CC23CC3)C(=O)NCCCN(S(C)(=O)=O)C)ccccc1 c1(C(=O)NC(CC=C)CNC(=O)Cc2c(C)n[nH]c2C)cc(C)ccc1[N+](=O)[O-] CCC(C)(CNC(=O)C(C)(C)CCNC(c1cn(CC)cc1C)=O)C(C)O C(=O)(C(F)(F)C1=CCOCC1)N1CCCN(CCNC(C(C)(C)C(N)=O)=O)CC1 S(=O)(=O)(c1cnc(N(CC(C)C(F)(F)F)C)c(Cl)c1)NC(C(CC)C)CO N1(C(COCCOCC)=O)CC(NC(=O)C(c2ccc(F)c(Cl)c2)O)CC(F)C1 c1(NC(CC)=O)ccccc1NC(C1CN(C(c2ccncc2Cl)=O)CCO1)=O C(=O)(C1=C(C2CC2C)N(Cc2ccccc2)C(=S)NC1c1cnn(C)c1Cl)OC c1(-c2cc(CN3CC(O)(C(C)NC(C4C(C)C4)=O)C3)[nH]n2)cccc(Br)c1 CCCC(C)(C)CC(=O)NCCCCc1cn(-c2cc(Br)nc(Br)c2)nn1 c1(C(=O)NCC(C2CCC2)NC(=O)Nc2n(C(CC)C)ncc2)cc(O)nn1C C1(F)(CNC(C(C2CC2)NC(C)=O)=O)CCCN(C(=O)C(C)OCC(C)C)C1 c1(CNC(C(=O)NCCC(=O)OC)=O)cncc(OCC(F)(F)F)c1 c1(C(N(C(CC2CCCCC2)C(=O)NCC2CCOC2)CC)C)cccc(Br)c1 C1(C(=O)NC2CCOC2=O)(CF)C=CCN1C(=O)C(COC)OC C1(NC(c2cc(C)[nH]c2)=O)CC2CC(NC(C3CC4CC4C3)=O)C1C2 c1(C(N(C)CCOC2CCN(C(=O)CC3(C)CC3F)CC2)=O)ncc(F)cc1F C1(C(N2CC(CC(C)NC(CNC(C)=O)=O)C2)=O)CC2(C1)NC(=O)NC2=O C1(NC(=O)C=Cc2ccccc2F)CCC2CCN(C(=O)C=CC=C(Cl)Cl)C1C2 C1(NC(C(C)C)=O)CC2CN(C(=O)C(c3cc(F)cc(F)c3)C)CC2C1 C1(CNC(c2n[nH]c(C)c2C)=O)CC2(CCC2)CN1C(=O)C=Cc1csnc1C C1(C(=O)N(CCOC2CCN(C(c3c(C)nco3)=O)C2)C(C)C)CC(C)CC(C)C1 C1(NC(COC(CC)(C)C)=O)CS(=O)(=O)CC1NC(=O)C(F)(F)c1nccs1 CC(C)(CCCNC(=O)CNC=O)Nc1cc(NC(C2CCCC2O)=O)ncc1 c1(N2CCC(C(=O)Nc3n(C)nc(C)c3C(N)=O)C2)ncc([N+](=O)[O-])cc1F Cc1cc(S(=O)(=O)N2CCC(C(c3ccccn3)O)CC2)c(C)cc1[N+](=O)[O-] C=C1CON(C(=O)c2cc(-c3ccccc3)ns2)C1 C1(C)(CNC(C2C(CC)C2)=O)CCN(C(=O)CCC2CC2(C)C)C1 C1(C)(C(=O)NCCCCCC#C)CC(O)CN1C(c1cc(C)co1)=O c1(OC(C)C)ccc(-c2ccc(N3CC(C)(NC(=O)CC(C)Br)C3)cn2)cc1 c1(CC)onc(C(=O)N(CC(O)CN(C(=O)C(c2ccc(C)s2)C)C)C)c1C CC1(CNC(C2(C3CC3)CCC2)=O)COCCN(C(c2cccc(Cl)c2F)=O)C1 c1(NC(NC)=NCc2cnc(CC(C)(C)C)o2)nc2ncccn2n1 N#Cc1c[nH]c(C(=O)N(CCOCCCNC(=O)Cc2nncs2)C2CC2)c1 C1(F)(CNC(c2c(C)nc(CC)s2)=O)CCN(C(C2CCCC(C)(C)C2)=O)CC1 c1(-c2cn(C(C(=O)OCC)C)nn2)ccc2[nH]ccc2c1 C12(CNC(=O)Nc3ccc(Cn4cccn4)o3)COCCN1C(=O)COC2 C1(CCOC)(C(=O)NC2(C)CC2C)CCN(CCC2NC(=O)NC2=O)CC1 C(C(C(=O)N(CCO)CCO)NC(C1CCNC1=O)=O)OCC N1(C(S(CCN(CCC)C)(=O)=O)=O)CCC2NC(=O)OCC2C1 C(=O)(CC1=NN(C)C(=O)C1)NC(CSC)(C)C(=O)NC1(C(O)CO)CCC1 C1(N(C(=O)OCC)C)CC2(CCCO2)C1.C1(=O)C(C2(C)CC2)O1 C1(C(=O)NC(CSCCc2c(OC)cccc2)=O)COCCC1(F)F C(=O)(C(CCF)NC(C1CC(=O)CCO1)=O)N1CC(C#C)C1 C1(NC(C(C(=C)C)(C)C)=O)CN(C(=O)COCC(=O)NC)C2(CCCOC2)C1 C(C(=O)N1CC(CNC(=O)CCc2cncs2)CC1C)(C(F)(F)F)OC(C)=O C12CCC(CC1)N2.Cc1cnn(C2CN(C(=O)N(c3ncccn3)C(C)C)C2)c1 Cc1cc(C(=O)NC2(CNC(C3CCOC(=O)CC3)=O)CCCC2)c(F)cc1N c1(C(N(CCOCCC(=O)N(C)Cc2cccc(O)n2)C)=O)cc([N+](=O)[O-])n[nH]1 Cc1nccc(C(=O)NCCCN(C(=O)C(O)C(C)C)CCO)c1N C(=O)(C1CCSc2ccccc21)N1CC2CN(C(C=CCOC)=O)CC2C1 C(=O)(C(C)(C)CC(=O)N1CCCCC1CC(=O)NCc1cc(C)nc(O)c1)OC c1(OC)ccnc(C(N2CCCCC2CN(C(c2coc(Cl)n2)=O)C2CC2)=O)c1 Cc1cc2[nH]c(C(N3CC(C4CN(C(=O)Cn5[nH]cnc5=N)C4)C3)=O)cc2o1 c1(C(=O)NCC2=CCN(C(C(C)SC)=O)CC2)cccc2c1OC(C)C2 C(CCC(C)C(=O)NC(C)(C)CNC(c1cnc(C)c(CC(C)C)c1)=O)OC N1(C(c2c(C)cc(C)s2)=O)Cc2ccnn2CC(NC(=O)C(O)C(F)F)C1 C1(NC(c2cccc(C)n2)=O)CN(C(C2CC3(COCCO3)C2)=O)CC2(CC2)C1 Cc1ccc2c(c1)SC(C(N1CCC(CF)(NC(C3CC4CC4C3)=O)C1)=O)C2 c1(CC)cc(F)ccc1C(=O)N(C1CN(C(C2CCCNC2=O)=O)C1)C c1(C(=O)NC2C(CNC(c3ccccc3O)=O)COC2)cnn2c1CCC2 c1(C(N2CC3CC3(CNCc3ccncc3Br)C2)=O)cc([N+](=O)[O-])cs1 Cc1[nH]c2ncccc2c1C(=O)NCCCN1CCN(C(=O)CC(C)N(C)C)CC1 CCCCCC(C)(CC)C(=O)NCCCCCNC(c1cnn(C2COC2)c1)=O C1(OC)(CNC(=O)CNC=O)CN(C(=O)C(F)(F)c2cccnc2)C1 C(=O)(C(C)CC(C)C)NCC1(OCC)CN(C(C2CCCCC2O)=O)C1 C1(C(=O)NC2CN(CCC)C(=O)C2)CCCCCCN1C(c1ocnc1C)=O c1(NC(CCn2cc(-c3cc(N)c(F)cc3)nn2)=O)cccc2nc(O)ccc12 N1(C(C2C(CC)C2)=O)CC2CC(NC(=O)Cn3nc(C)ccc3=O)CC1C2 Cn1c(C(=O)NCC2(O)CCN(C(C34CSCC3C4)=O)C2)cnc1S N1(C(CN(CC)CC)=O)CCCN(C(=O)COCc2nc(C)no2)C(CO)C1 n1(C(C)C)ncc(C(=O)NCCOC2CCN(C(=O)CCCF)CC2)c1N C1(CC(=O)NCc2c(C(=O)NCC=CC)occ2)CCC(C)CO1 C1(C(N)=O)CCCC(C(=O)NCCCCNC(=O)CCF)CC1 c1(CC(=O)NCC2CC(CC3CC3)C2)ccccc1-n1cc(C(F)(F)F)nn1 C1(N(C(C(F)OC)=O)CC)CCC(NC(c2n[nH]cc2-c2ccon2)=O)CC1 N1(C(N2CCC(C)(COC)C2)=O)CC(C)CCCC1C N1(C(c2nc(C)sc2)C(=O)NC2CCOCC2)CCOCC1CCC(F)(F)F C1(CN(C)C)(NC(c2[nH]nc(Br)c2Cl)=O)CCOCC1 CC1CCc2ncc(C(=O)NC3CCC3C(=O)N(C(=O)Cn3cccn3)CC)n2C1 C1(C(N(CCC(C(C)C)NC(c2n(CC)ncn2)=O)C)OC)CCCCC1(C)C N1(Cc2c(C)cccn2)C(=O)CCN(Cc2cccc(Cl)c2Br)C1=O CC1C(C(=O)N(c2ncccn2)CC2CC2)CCN1C(=O)C=Cc1ccncn1 CCCCC(O)C(=O)N1CCC(C(C)NC2(C(=O)OCC)CCCC2)C1 c1(C)cccc(OC)c1.C12(C(N(CCN(C(=O)COC)CC)CC)=O)CCCC1CC2 Cc1cc(C(=O)NCC(C2CC2)NC(c2snnc2C2CC2)=O)cc2ccoc12 CCC(C(=O)NCC1CCC(NC(=O)CCC=CC(C)C)C1)C(F)(F)F c1(COc2c(CN(C(=O)Nc3ccccc3)C3CC3)cccc2)ccncc1Cl C1(N(C(c2cc[nH]n2)=O)CC)CCC(N=c2[nH]c3ccc(F)cc3s2)CC1 N1(C(C(CCCC)CC)=O)C2CCC1C(CO)N(C(c1cc(OC)ncn1)=O)C2 N1(C(C(CCCC)F)=O)CCC2CN(C(C3CCc4nccn4C3)=O)C(C)C12 N1(C(C(C(=O)OC)C)=O)CCC(CCNC(C2CN(S(C)(=O)=O)C2)=O)C(F)(F)C1 c1(OC)ccc(C(=O)NC2CCN(C(C3(CCF)CCC3)=O)C2)c(F)c1 C1(C(=O)NOC2CCC2)(CN(C)C(C2CCC(C)(C)C2)=O)CCCCC1 CC1OCCC1(F)C(=O)NCCN(C(c1coc(O)n1)=O)CC1CC1 C(C(=O)NNC(=O)C(=O)OC(c1nccn1C)C)c1ccc(OC)cc1 c1(CC(=O)NC2C(NC(c3c(C)cn(C)c3)=O)CC2)ccc2n[nH]cc2c1 n1(CCC)cc(CNC(=O)C(C2CC2)NC(=O)C(C)O)nn1 Cc1noc2nc(C(N3CCN(C(c4cccnc4S)=O)C(C)C3)=O)ccc12 C1(NC(C(c2csnn2)N(C2CCOC2)CCOC)=O)CCOCC1 C1(NC(C(C)=CC)=O)CC2CCC1C(NC(=O)CC(C)CN(C)C)C2 Cc1nsc(NCC2CN(C)CCN2C(=O)C2=CS(=O)CCC2)c1C#N c1(NC(=O)CCCC2CCOCC2)cccc(NC(c2occc2Br)=O)c1 CC1(C)CN(C(C2CCCN2C=O)=O)CCC1NC(=O)CN1C(=O)CCC1=O N1(C(C2(CO)CCN(C(COCCCN(C)C)=O)C2)=O)CCCOCC1C c1(-n2nccc2)ccc(F)c(Cl)c1.CC(C(=O)N(C)C)NC(=O)NCC C1(NC(c2nc(C)nn2C)=O)CCN(C(c2cnc(C3CC3)s2)=O)C1(C)C C(CCCCCC(=O)NCC1CCOCC1)NC(c1c(C)c(F)cnc1)=O c1(C(=O)NCCC2OCCN(C(CC(CC)C)=O)C2)c(O)cc(Cl)cc1F C(c1ncc(C)[nH]1)=CC(N1CC(C(=O)NC(COC(C)C)CO)(CC)C1)=O c1(C(N2CCC(C(CO)NC(C(C(C)C)(C)C)=O)CC2)=O)ccnc2cc[nH]c12 C1(C(=O)NC(CC)C2CC2)CN(C(c2cc(CO)oc2C)=O)CC1C(C)C C1(C2CCN(C(c3ccc(C(N)=O)[nH]3)=O)C2)(NC(c2c(CC)nccn2)=O)CC1 c1(OC)ccccc1C(C)C(=O)NC(c1cc[nH]n1)C1CCCC1 C1(CCNC(c2n(CCCSC)nnn2)c2cnn(C(F)F)c2)CCC(C)(C)O1 CCCC(C)(O)CNC(C1CCC1CNC(c1cc(CO)ccn1)=O)=O c1(C(=O)NC2CCCN(C(CC(C)C3CC3)=O)CC2)cccc2[nH]c(=N)oc12 c1(OC)cccc(C2(C(=O)NCC(c3ccnn3C)O)CC2)n1 c1(C(N2C(C)(C)C(NC(=O)CNC=O)CC2)=O)cnc(O)c2cccnc12 CCC(C)CCCC(=O)NC1CC2(C1)CN(C(C1CCC1c1nncn1C)=O)C2 C1(C(=O)NC(CC)CNC(C2CC2C2CCCO2)=O)CC(=O)NC(=O)C1 C1(C(=O)NC(C)CCSC)(OC)CCN(C(c2nccnc2N)=O)C1 c1(OC)ccc(C(N2CCCC2CNC(C2CCC3(CC2)CC3)=O)=O)nc1OC n1(CC)nnc2c1C(C(=O)N1CC(C(C3(O)CCC3)O)C1)CN(C(=O)C(C)C)C2 c1(C(N(CCN(C)C(c2cnoc2-c2ccoc2)=O)C)=O)snc(O)c1Cl C1(CC(=O)N(CCC(=O)NCC2CSCCO2)CC)CCCN(C)C1 c1(C(C(=O)NC2CC(CNC(=O)CC3CCNCC3)C2)O)cccc(Br)c1 N1(C(Cc2c(CC)cccc2)=O)C2CCC1C(NC(C1(COC)CC1)=O)C2 C(C(=O)N(C1CCCCC1)CCNC(=O)CCn1cccnc1=O)(C(C)C)SC N1(C(c2ccc(OC)nn2)=O)CCCC(N=c2nc(CC3CC3)[nH]s2)CC1 C(C(C)(CC)C(=O)NCC(C)(C)C#N)NC(c1n(C=C)ncc1)=O N(C)(C1CCc2ccccc21)CC(C(=O)Cc1n[nH]cc1C)=O.CCCCN N1(CC(CC)C)CCCC(F)(COC)C1 c1(C(N2CC3C(NC(C(C)(C(C)C)NC(C)=O)=O)(C3)C2)=O)cnc2scnc2c1 N1(C(CC2CC(=C)C2)=O)CC(C)CCC1CNC(c1ncc(OC)cc1F)=O c1(OC)ccc(C(=O)NC(C)(C)CNC(C2SC3C=CC2CC3)=O)cc1C c1(COC)cc(C(=O)NCC(C)=CC(=O)NCCNC(C2CCC2)=O)n[nH]1 C12(CNC(C(CC)COC)=O)CN(C(C3SCCS3)=O)CC1CCO2 N1(C(c2c(CC)noc2)=O)CCC(C)(CC(=O)NCC2(O)CC2(C)C)C1 C(=O)(C1=C(SC)CCCC1)NC1(CCOC)CCN(C(C(CC)(C)OC)=O)C1 CC1(C)CCC(C(=O)NCC23CC2CN(C(c2ccncc2F)=O)C3)OC1 C1(NC(c2c(C)cc(C3CC3)cc2)=O)CN(C(=O)C2=NOC(C)C2)CC2(CC2)C1 N1(C(c2ccc(OC)o2)=O)CCC(C)(NC(C2CCN(CC3CC3)C2)=O)CC1 c1(C(N(C2CCCC(NC(c3cnccc3Cl)=O)C2)C)=O)ccnc(S)c1 c1(C(N2CC(O)(CN(C(C(c3cnn(C)c3)OC)=O)C)C2)=O)cncc(Cl)c1C C(=O)(C1CCCn2nccc21)NC1CCN(C(CSc2nc(C)[nH]n2)=O)C12CC2 C=C(C)CC(C(=O)OC)NC(=O)C=C(C)CNC(C1CCN(C)C1CC)=O CCCC(CC)C(=O)NC1C=CCN(C(=O)CSc2ccc(OC)cc2)C1 C1(C(=O)Nc2ncc(C(C)C)[nH]2)COC2(C)CC1C2 CCN=C(NCC(c1ccccc1)OC)N1CCn2c(C(=O)OC)nnc2C1 c1(SC)cccc2c1CCC2NC(=O)C(C)(C)n1cc(-c2ccc(C(=O)O)s2)nn1 c1(C(=O)NCC(CNC(CCc2ccc(C(=O)OC)[nH]2)=O)O)cnc(C)nc1O C1(CCC(=O)NC(C=C)COC)CCCCN(C(=O)C(CO)N(C)C)C1 C=C(C)C(C)(C)C(=O)NCc1nocc1C(=O)NCCC1CC2CC2C1 c1(C(N2CC(CNC(=O)C(O)C3CCCC3)C2)=O)cc2cccnn2c1 c1(CN(C)C)ccc(C(=O)NC2(C)CCN(C(=O)C(O)CN3CCCC3)C2)cc1 C1(NC(CCC(N)=O)=O)CCCOC12CCN(C(=O)C(c1cccnc1)O)CC2 c1(N(C(c2cccnc2)N2CCOC2=O)CC)n[nH]c(C)c1Br.n1(C)cc(C)nn1 N1(C(CN(C)C)=O)CC2CCCCC2(NC(c2cccc(C(N)=O)c2N)=O)C1 CCCCCC(C)CC(=O)N1CCCC(NC(c2c(C)ccc(Cl)c2N)=O)C1 C1(CC=C)(C(N2CC(C(N)=O)(OC)C2)=O)CCN(C(=O)C(C(C)C)SC)C1 C(C(C)C)(C(O)C(=O)NC(C)C(CO)NC(c1cc(C)ccc1O)=O)OC C1(C)(C(=O)NC2(CC)CC2)CCN(C(=O)C=CC2CCOCC2)CC1 c1(C(N(C(C)CNC(C2CCC3(CCC3)O2)=O)C)=O)coc2cccc(O)c12 N1(C(COCC=C)=O)CC2CCCCC2(NC(c2cc(C3CC3)nn2C)=O)C1 c1(NC(c2ccccc2)=O)ccncc1SN1Cc2cnn(CCO)c2C1 c1(C(N2CC(C(=O)NCC3CC4CCC4C3)(CC)C2)=O)cc(O)cc(F)c1 C(=O)(CCN(C=O)C(C)C)N(CCN(C(=O)OC(C)=O)C)C.CN C(=O)(C(O)CCc1ccc(F)cc1)NCC1CCN(S(C)(=O)=O)CC1.O=C(CCl)S(=O)N c1(C(N(CC(CNC(C(c2cccs2)SC)=O)O)C)=O)cc(C(F)(F)F)n(C)n1 N1(CC(=O)N(CC(C)N(C(=O)CN(C)C)C)C)CCC(C)(O)C1 C1(N(CCCNC(C2CC2F)=O)C(C2CC2F)=O)CCCC1 c1(OC)cc(C(=O)NCC(O)CN(C)C(C2CCN(C)C2C)=O)cc(N)c1OC C12(C(=O)NCC3CCCC(NC(c4cccc(=S)n4O)=O)C3)CCC(=O)N1CCS2 C1(C)(NC(C2(COC)CCC2)=O)CN(C(=O)CNC(c2cncnc2)=O)C1 N1(C(C2CC(OC)C(OC)C2)=O)CCCC(C)(CNc2nccc(C3CC3)n2)C1 C1(CNC(C2CN(C(=O)NC)C2)=O)COCCN(C(C2CCCS2)=O)C1 c1(OC)ccc([N+](=O)[O-])cc1CNC(C1(C)CCCN1S(=O)(=O)CC#N)=O c12ccc(cc1)c(=O)[nH]2.C(=O)(C(C)(C)C)NC(CCC)c1nn[nH]n1 N1(C(c2cc(C)n(C)n2)=O)CCC2(CCC(NC(C34CCCC3(C(N)=O)C4)=O)C2)C1 N1(C(CCC=CC)=O)CCC(C(F)F)(CNC(=O)CCc2ncccn2)C1 C(=O)(CCC(=O)N(C)C(C)C)NC1N(C(C2CC(O)(CC#C)C2)=O)CCC1 C1(NC(C=C(CCC)C)=O)CN(C(=O)C=Cc2c(C)coc2C)CCC1F c1(-c2c(OC)cc(OC)cc2F)ccn2c(CO)cnc2c1 C1(NC(C(C=C)O)=O)CN(C(=O)C(C)(C)OC)CCC1(C)C c1(C(=O)NC)cccc(NCC(=O)NC2CCCN2C(=O)NC(C)C)c1 Cc1ccc(C(=O)NC2(Cn3cc(C4OCCO4)nn3)CCCCC2C)c(C)n1 C(=O)(C(C)P(C)(C)=O)NCCCCNC(C1N(S(CCC)(=O)=O)CCC1)=O C(CC(C)C)(C(=O)NC(C)CS(C)=O)N(C(CN(C(CCC)=O)CCC)=O)C C1(CC(=O)NCCC2(OC)CN(C(C=C(COC)C)=O)C2)COC(C)(C)C1 C1(C(C(=O)NC2(C)CC2)N(CCOC)CC2CC2)CC12CCOC2 C1(C(=O)NC(CCSC)C(=O)N2CC(CO)C(CO)C2)CCCC12CCC2 n1(CC(=O)N(C2CC(NC(C3C(CCC)CCC3)=O)C2)C)cc(C#N)cn1 CCC(C)CC(=O)N1CC2CC2(CC2CCCCC2)C1.C1(=O)C(C)(C)CN1 N1(C(C2=C(C)OCCS2)=O)CCC2CCCN(C(=O)C=Cc3ncc[nH]3)C2C1 Cc1cc(C#N)cnc1CC(=O)N(CCCCNC(=O)C(F)CC1CCCC1)C Cn1cc(Cl)c(CC(N2CCCC(CCNC(=O)CC3CCCC3O)C2)=O)n1 C1(CNC(C2(C)N(C(C3CC(=C)C3)=O)CC2)=O)CCC(=O)NC1 C(CC(=O)NNC(=O)c1ccccc1)NC(C1CCS(=O)(=O)N1)=O N1(C(CCCCC)=O)CC2(CCC2NC(c2ccc(Cl)c(F)c2)=O)C1 CCCCC(O)C(=O)NC12CC(C(=O)NOCCOC(C)C)(C1)C2 c1(C(=O)Nc2ccc(C3CCN(S(=O)(=O)C4CC4)CC3)cn2)cnn2ccccc12 N1(CC(=O)NCC(O)CNC(=O)Cn2ccc(C(F)F)n2)C(=O)CNC1=O C1(CC(N2CCN(C(c3ccc(F)c(Cl)n3)=O)CC2CO)=O)CCC(F)(F)CO1 N1(C(C(COC)Oc2ccc(OC)cc2)=O)CCN(C(=O)CCC(N)=O)CC1C C1(C(=O)NC2CCC(NC(c3cncs3)=O)CC2)(COC)CCOCC1 c1(C(N2CCC(N(CC#C)C(c3c[nH]nc3CCC)=O)C2)=O)nnccc1C c1(C(N2CCCC2C(=O)Nc2cccc(OC(F)F)c2)=O)ccncc1.OCF N1(C(C(C2CN(C(C3C(C)CCOC3)=O)C2)O)=O)CCC(F)(F)CC1 c1(NC(C(C)NS(CC)(=O)=O)=O)cccc(NC(=O)CC2CCC23CCC3)c1 N1(C(CCC(=O)OCC)=O)CCC(CNC(C2CC(O)C2)=O)C12CC2 N1(C(COc2cccc(C)c2)=O)CCN(C(=O)C(C)c2ccon2)CC12CC2 c1(C(N2CCC(N(C(=O)C=C3CCOCC3)CCC)C2)=O)cc2sccc2n1C N1(C(C(CC)F)=O)C(CNC(=O)CNc2nccs2)CC2CC12 Cc1cc(C(N2CC(CNC(C3(c4ccc(Cl)c(F)c4)CC3)=O)C2)=O)ccc1Cl Cc1[nH]c2ccccc2c1C(=O)N(C)CC1CCN(C(C23CC(C)(CO2)C3)=O)C1 CC1=CC(O)CN(C(c2ncoc2CNC(C2(C#N)CC23CCC3)=O)=O)C1 Cc1cc(C)n(CC(=O)NC2CC(C)(NC(C3CCCC(F)C3)=O)C2)n1 C(=O)(C1=CC2CCCC12)NCCNC(c1cccc(C(=O)NC)c1)=O c1(OC)c(C(=O)N(C2CCCN(C(=O)CCC3CC(C)(C)CO3)C2)C)csc1C CCC(C)C(C(=O)N1CC2C(C1)C2(F)F)N(C)C(C12CC1CNC2=O)=O N1(C(c2nccc(C)c2N)=O)C2CCC1CC(CNC(c1ccnc(F)c1)=O)C2 c1(C(=O)NCC(C)CNC(C2CCOCC2)=O)c[nH]cc1C1CC1 C(=O)(C1CCCc2c1ncn2C)NCC(CNC(Cn1c(C)ccn1)=O)CO Cn1ncc2cc(CN3CCC3CNC(c3cccc(F)c3)=O)ccc12 C#Cc1ccc(F)c(C(N2CCC(C)(CNC(=O)CC(C)(O)COC)C2)=O)c1 c1(CC(=O)N(CCCNC(=O)CC2CC(=O)NC2=O)C)csc2nccn12 C(C(COC)C(=O)NC1CCC1C(=O)NCC(C)CC1CC1)OC c1(C(N2CCCC(CNC(c3cc(Cl)ccn3)=O)C2)=O)cnc(O)nc1O C1(C(=O)NCc2cc(C)oc2)Cc2ccc(F)cc2C(=O)O1 c1(C(N2CCN(C3CN(C(C4(C(=O)OC)CC4C)=O)C3)CC2)=O)nnc(O)cc1C c1(OC)ccc(F)cc1CCC(=O)NC1(CCNC(=O)CNC(C)=O)CCC1 C(CS(=O)(=O)C1=NOC(C)(C)C1)NC(c1n(CC)nnn1)(CC1CC(OC)C1)CC c1(OC)cc(O)ncc1C(=O)N(CCCCNC(C1(C)CCCC1N=[N+]=[N-])=O)C c1(NC(c2cn(CCN(C)C)nc2)=O)ccccc1Cl.C12CC1C(=O)N2C1CCC1 O=C(N=c1ccn(C2CC2)[nH]1)C1CC(O)CN1C(C1CCCOCC1)=O C=CCN=C(NCC(F)(F)C1CCC1)NCC(C)(F)F C1(CCNC(c2nc(C)sc2)=O)C(C)CCCN1C(C12CC(C)(C1)OC2C)=O S(=O)(=O)(CC(=O)NC1CCC(CC(=O)N(CCCCO)C)C1)NCC C1(NC(CCSCCOC)=O)CN(C(=O)CSc2nncs2)CCC12CCC2 c1(C(=O)NCc2c(F)ccc(C)c2Br)cnc2c(Br)cncc2c1 O(NC(=O)C(C)(CO)NC(c1cnc2cc[nH]c2c1)=O)CCCC C1(F)(C(N(C2CCN(C)CC2)C)=O)CCCN(C(C2CC3(C2)CC32CC2)=O)C1 CCCCC(O)C(=O)N1CC(C(N)=O)(CNC(c2sc(C(N)=O)nc2C)=O)C1 CC1=C(C(=O)NC2CC3CC2N(CC2CC4(CCC4)C2)C3)SCCO1 c1(C(=O)NC2C(C(=O)NC(C(=O)NC)C(C)(C)C)C2)cccc([N+](=O)[O-])c1Cl Cc1ccc2c(c1)SC(C(N1CCC(CNC(c3cc(N)ccc3Cl)=O)C1)=O)C2 C=CC1(C(=O)NC2CCC(CCC(N3CCC(COC)C3)=O)C2)CCCCC1 C1(CC(N2CCOCC(NC(C3(COC)CCC3)=O)C2)=O)CCC2(CCC2)CO1 C1(C(=O)NC2CN(C(CCC(=O)N(C)C)=O)CC2O)CC(c2ccccn2)=NO1 CC(C)C(O)C(=O)NC(C)(C)C(C)NC(=O)CCCC1CCCC(=O)N1 n1(CCC)nnnc1C(c1csc(Cl)n1)NC(C)C(C)SC1CCCCC1 n1(CC)cc(CCNC(=O)COC2(C)CN(C(=O)CC3COC(=O)C3)C2)cn1 C1(CNC(C2CC2c2cccc(Br)c2)=O)CN(CC2CNCCO2)CCO1 c1(C(=O)NCc2ncn(C)c2)ccc(-c2ccc3ncsc3c2)c2c1OCO2 C1(NC(CC2CC(=C)C2)=O)C2CC3C1C3C2C(=O)NCC1CC2(CCC2)CO1 Cc1cc(NC(=O)NCC2CCN(C(=O)NC3CC3)CC2)c(Br)nc1C c1(CC(C)(C)C)cn(CCCOC(C)(C)CN)nn1.C12(CC=O)CC(C1)C2 c1(NC(C2N(C(CCOC)=O)C3C(C2)C3)=O)cc(F)c(Cl)cn1 CC1CN(C(c2sc(N(C)C)nc2Cl)C(=O)NCC2CCOC2)CCS1=O Cc1c(CC(=O)NC2CCCC(C(N3CCC(CO)C3)=O)C2)cnn1C CCC(C)(C)C(C(=O)NC(C)CNC(=O)CC1CCC(F)(F)CC1)OC c1(CC)ccc(C(=O)NCCC(C)N(C(=O)C(c2ccc(Cl)nc2)(C)C)C)nc1 C1(C(=O)NC2(CSC)CC2)C2CCCC2CN1C(=O)CC1C=CCC1 C1(CNC(=O)Cc2cnn(C(F)F)c2)CC2(CCC2)CN1C(C1CCCSC1)=O C#Cc1ccc(C(N2CC(NC(=O)CC(=O)N(C)C)C3(CC3)C2)=O)nc1 CCCC(O)CC(=O)N1CC(CNC(c2cc(CC3CCC3)c[nH]2)=O)C(O)C1 C(=O)(C1=NN(C)C(=O)CC1)NCCOCCN(C)C(C1CCCC1(F)F)=O C(=O)(CCC(C)(C)C#N)NC(C(=O)N(C)Cc1ncc(C)o1)Cc1ccco1 Cn1nc(C(=O)NC2(CCNC(=O)CC3CCNC(=O)C3)CC2)cc1C(F)F C1(C2(NC(C(C3CC3)SC)=O)CC2)CCCCN1C(=O)CC(C)(F)F C12(C(C(=O)NCC(F)F)N(C3CC3)Cc3onc(N(C)C)n3)CCC(CC1)O2 CN1CCCC(C)(C(=O)NCc2ocnc2C(N2CC(C(=O)N(C)C)C2)=O)C1 N1(C(Cn2c(C)cnc2)=O)CCOC(C(C)NC(c2ccn(CCCF)n2)=O)C1 CC(C)(CS(C)(=O)=O)C(=O)N1CCN(CC(C)(C)NC(C2CCOCC2)=O)CC1 N1(C(c2cnc(COC)s2)=O)CC(C2CCCCN(C(C3(C)CCCC3)=O)C2)C1 CCC(O)C(C)C(=O)N1CC(C)(NC(c2cccc(SC)n2)=O)C1 N1(C(CNC(CC(C)C)=O)=O)CCC(C)(NC(=O)CC2CC(F)C2)CC1 Cc1ccnc(O)c1C(=O)NC(C)CC1CCN(C(=O)C(C)C2CCC2)CC1 N1(C(CC(C)S)=O)CC2(CCN(C(=O)C=CCOC(C)=O)CC2)CC1C.C(C)(C)(C)O C=C1CC2(C1)CN(C(=O)CN(C(=O)C(C)(C(C)C)OC)C1CCC1)C2 C(CC(O)CC(=O)NCCN(C(C1CCO1)=O)Cc1ccccc1)SC N1(C(C(C2CCCO2)NC(CCCOC)=O)=O)CCCCC1C(=O)OC C1(C(=O)Nc2n(CC)cc(Br)c2)CC2CCC(C1)N2 N1(CC)CCC(NC(C2CC(=O)CN2C(=O)CC2CCCOCC2)=O)CC1 c1(C(N2C(CCNC(C3C(C)OCC3)=O)CSCC2)=O)cccc(P(C)(C)=O)c1 Cc1cc(F)ccc1N1CCCN(C(C2(c3ccc(Cl)cc3)CC2)=O)CC1 C1(CN(C)C(C2CC(OC(C)(C)C)C2)=O)CCCC1(C)NC(C1CC(F)C1)=O c1(C(=O)Nc2nc(C(=O)Nc3cc(C)cc(C)c3)n(C)c2)cc(C)c(C)cc1C c1(C(N2CCN(C(C(c3ccccc3)C)=O)C(CF)C2)=O)c(Cl)ccc(F)c1N N1(C(c2ncc(NC)nc2)=O)CCCC2(CCN(C(C3CCCC(C)C3)=O)C2)C1 N(C(=NCCC(C)SC)NCc1cc(Cl)ccc1C)Cc1c(C)cccc1 N1(C(c2cc(CN(C(C3(CCC)CCCC3O)=O)CC)oc2)=O)CCC(O)C(C)C1 C(=O)(C(F)(F)C(C)(C)O)NCCCCC(C)NC(C1C=CCCC1)=O C=CC(C)(C)C(=O)NOC(CC(C)C)C(=O)N1CCC(C2(C)N=N2)C1 c1(OC)ccccc1CC(=O)N(CCNC(c1ccnn1C1CCC1)=O)C1CC1 N(C1CCCc2ccoc21)C(C1CC(O)(CNC(CN(C)C(N)=O)=O)C1)=O c1(CN2CCN(C(C3=CC=NC(=O)C3)=O)C3C2C3)cccc(Br)c1[N+](=O)[O-] C#CCCCCC(=O)N1CCCC(C)(NC(=O)C(N2CCSCC2)C)C1 c12ccc(cc1)CC(=O)NC2.C1(C(=O)NCCOCCN(C)C)CCCC1C#N CCCCC(CNC(C1C(Cl)(Cl)C12CC2)=O)NC(c1cnn(CC)c1)=O N1(C(C2N(C(C(=C)F)=O)CCC2)=O)CCOC(C(F)(F)F)C1 c1(C(=O)NC2CCCC(NC(c3cn(C)nc3)=O)C2)cc(N)c(Cl)cn1 c1(C(=O)NC2CCN(C(c3[nH]c(=NCC)sc3)=O)C(C)C2)cc(C)c(Cl)cc1C N1(C(=O)CSc2nnc(S)s2)CC2CCC(C1)N2C(=O)CCN1CCOCC1 N1(C(CC2CC(CC)C2)=O)CC(NC(=O)CNC(=O)OC(C)(C)C)C(C(F)F)C1 c1(C(N(CC(CC)NC(=O)C2=NOCC2)CC)=O)cc(OC)ccc1Cl N1(C(C(C)OC)=O)CCCC2C1CCN2C(=O)Cc1cc(C)cc(F)c1 N1(Cc2c(C)cc(C)cc2C)CCCC2C(NC(C3CC3F)=O)C(C)(C)C12 C(=O)(CCOC1CN(C(=O)C(C)OC2CC(OCC(C)N(C)C)C2)C1)OC CC(C)CCC(O)C(=O)N1CC(C)(CCC(N2CCNC(=O)C2)=O)C1 c1(C(=O)NCc2ccccc2C#N)cc(C)c(C)cc1Cl.C1(OC)CC2N(C1)C2=O Cc1[nH]nc2c1CN(N1CCCCC1CC1CC1)CC2 c1(C(C(=O)N(C(C)C)CCNC(C2COCCO2)=O)C)ccc(C(N)=O)cc1 Cc1ccc(C(=O)NC2CC(F)(F)CC2NC(=O)C(O)CN(C)C)c2c1CCC2 C1(NC(C(CC)=CCCC)=O)CC2(CCC(NC(=O)CCS(=O)(=O)NC)CC2)C1 C1(OC)CCN(C(=NCCc2ccc(OC)nc2)NCc2cncnc2)CC1 CCC(CC(=O)N1C2CCC(C2)C1CNC(c1ccncc1C(F)F)=O)C(C)C Cc1cccc(C(C)(C)C(=O)NC(CNC(C2CC(=C(F)F)C2)=O)C(C)(C)C)c1 N1(C(C=CCOC)=O)CC2CCC(C1)N2C(c1cc(C(C)(C)C)n[nH]1)=O C(C(C(=O)NCC)Nc1ccc(CC)o1)SCC=C Cc1nn2cnnc2c(C)c1NC(c1cc(Cl)ccc1-c1nn[nH]n1)C1CCC1 CC1(C)CC(C(=O)NCC2(NC(C3CCC(O)C3)=O)CCOC2)CC(C)(C)C1 N1(C(c2cc(F)c(I)c(F)c2)=O)CCC2(CCN(C(C3(F)CC3)=O)C2)C1 C1(N(C(=O)CCc2cc(O)no2)CCCNC(C)=O)CCC(C)C1.CO C1(NS(CC2C(C)(C)CCO2)(=O)=O)CN(C(=O)CSC2CC2)C(C)(C)C1 c1(C(=O)NC2(CNC(C(C)SC)=O)CC2)ccc(NS(C)(=O)=O)nc1 c1(-c2ccc(C(=O)NC(CN(C(=O)COCCCF)CC)C)s2)cccc(F)c1 c1(C(C(=O)NC2C(CNC(C(c3cn(CC)nc3)=O)=O)C2)C)ccc(C)cc1 N1(C(c2c(C)occ2)=O)CCCC(NC(=O)CCc2ccc(Cl)cc2Cl)C(F)C1 CCCC(C(=O)OC)NC(=O)CC1CCC(NC(=O)C(F)CC2CCOC2)CC1 C1(CN(C(=O)C(O)Cn2cncn2)C)CCCN(C(=O)C(CCN(C)C)N(C)C)C1 Cn1ncc2c(O)nc(=NC3CN(C(c4ccc([N+](=O)[O-])c(Cl)c4)=O)C3)[nH]c12 c1(NC(CC2CCCN(C(C(C)C(F)(F)F)=O)C2)=O)cnc2c(c1)CCC2 N1(C(c2cc(SC)c(Br)cc2)C(=O)NCC2CCOC2)Cc2cc(O)nnc2C1 C1(NCc2nc(CCC(=O)NC)on2)CCC(N2CCCC2=O)CC1 CC1(C)CC(CNC(=O)CCc2cnco2)N(C(C2CCC2(C)C)=O)C1 C1(C(=O)OC)CCC(C(N2CC(CNC(=O)CNC(N)=O)C2)=O)C1 N1(C(C2CC(C(C)C)C2)=O)CC(O)CC1C(=O)NC1CCCCC1F C(=O)(C(C(=O)N1C(C(N2CCC(C(C)C)(CO)C2)=O)CCC1C)OC)OC Cn1cc2ccc(C(=O)NCC(c3ccccn3)N3CCOCC3)cc2n1 N1(C(C(C=CC)O)=O)CC2(CCN(C(c3cccc(O)n3)=O)C2)C1 Cc1cc(Br)c2c(c1)CN(Cc1ccc(OCc3ccccc3)c(F)c1)CCO2 C1(CC=C)OCCC1(c1nnnn1CC1CCCO1)Nc1cccc(C(N)=O)c1 C1(C(N(C(=O)CNC=O)C)=O)CC(CC)CCO1.C12C=CC(C1)NC2=O C1(C(=O)NCCC(C)NC(=O)Cc2cncc(Br)c2)CCCC(=O)N1C C(=O)(CS(=O)(=O)CCO)NCC1CN(C(c2c(OC)cc(Cl)cc2)=O)C2C1C2 c1(OCC=C)ccc(CC(N2CCC(NC(c3nc(=O)n(C)[nH]3)=O)C2)=O)cc1 c1(C(=O)OC)cc(C)nn1CC(=O)NC1CCC(CNC(=O)C=CC2CC2)C1 N1(C(C(CC)C(C)O)=O)CCC(C2(NC(=O)C=Cc3ccc(C(F)F)o3)CC2)C1 c1(OC)cc(N)ccc1NC(=O)C(=O)NCC1(C(F)(F)F)CCCCCC1 C(C(=O)NOCCOC)(c1ccccc1)NC(CC1C(CC)C1)=O C1(C(=O)NC(C#C)(C)C2CCCC2)C2CC3C(C2NC(=O)C(C)CC(F)F)C13 C1(C(N(CCN(C(c2c(CC)ocn2)=O)C)C)=O)CC(=O)N(C(C)(C)C)C1 N1(C(C(N2CCCCC2)C)=O)CCCC2(NC(c3ccncn3)=O)CCCC12 C12(CCNC(CCC(C)OC)=O)CCC(C1)N(C(c1cnn(CCOC)c1)=O)C2 C1(C)(CNC(C=C(C)C(C)C)=O)CN(C(=O)Cn2cc(F)ccc2=O)C(C)(C)C1 n1(C2CN(C(CCOC(C)(C)C)=O)C2)cccnc1=O.C12CCC1NC2 C1(c2nc(CNC(c3ccc(C)o3)=O)[nH]n2)COCCN1C(=O)C(C#N)CC1CC1 Cc1cccc(CCC(=O)NC2CCOCC2C(=O)NCc2ncccc2C)c1 c1(N2NCCC(=C)C2)nc(=N)[nH]c(=NC(C)Cc2ccnc(O)c2)[nH]1 c1(CCC)n[nH]cc1C(=O)NCC1CC(C(=O)NCC2CC(CN=[N+]=[N-])C2)CO1 c1(CC(=O)NC(C2(CF)CCN(C(c3coc(Cl)n3)=O)C2)C)c(O)ncnc1O C1(NC(CC(C)(C)O)=O)CS(=O)(=O)C12CCN(c1nc(C(F)F)nc(=N)[nH]1)CC2 C=C=CC(C)C(=O)NC(C)(C)CCNC(c1cc[nH]n1)=O Cc1nc(C(C)(C)C)nc(O)c1C(=O)NC(C)C(CO)NC(=O)C#CC1(C)CC1 C1(C(N(C(C(=O)O)C(C)C)CC(OCC)OC)=O)Cc2nccn2C1 N1(C(Cc2c(C)noc2)=O)CCC(NC(c2ccc(C(C)C)c(Cl)c2)=O)CC1C C1(NC(CN(C(C=C(CC)CC)=O)C)=O)CC(C)(C)C12CCC2 O=S(=O)(c1cccc(=NCCC2CCC3CC23)[nH]1)NCCC1(C)CC1 C(c1ccc(C)cn1)=CC(N1CC(O)(CCNC(C(CC)n2ccnc2)=O)C1)=O N1(C(c2c(OC)nn(C)c2)=O)CCC2C(CCN2Cc2ccc(N(C)C)s2)C1 C=C=CCC(=O)NCCCC(=O)NCCOC(C)(C)C C(C(C)(C)C(=O)NCC(CC)NC(=O)COCC1CCCO1)NC(C)=O CCCCCCC(C(=O)N(C)C)n1cc(C2COCC2O)nn1 C1(NC(CCC=C)=O)CS(=O)(=O)CC1NC(c1cnc(N(C)C)c(Cl)c1)=O Cc1cccc(C(C)C)c1C(=O)NC(CO)C(C)NC(=O)CCC1CCC1 C(CC(=O)N=c1ccn(C)[nH]1)OCCNC(C1C(OC)CCC1)=O C(=O)(C1CCCc2nccn21)N1C(C)CCN(C(c2cc(CC)c(C)s2)=O)CC1 c1(OC)cc(NC2CC(NC(C3(C)CC3Br)=O)C2)ccc1[N+](=O)[O-] C1(C)(CC(=O)Nc2c(CC)cccc2)CCN(C(c2ccnc(C)c2)=O)C1 C(=O)(C(O)(C(F)(F)F)C1CC1)N1CCC(OCCNC(=O)C2=CCCSC2)CC1 Cc1nc(-c2nc[nH]n2)sc1C(=O)NCC(C)(C1CC1)NC(c1ccnnc1)=O c1(NC)cccc(C(=O)N(C=O)CCN(C(=O)CSCCC(F)(F)F)C)c1 c1(C(=O)NCCN(CCOC)Cc2cc(C)[nH]n2)nccc2ccccc12 c1(C(N(C2CC2)CC2CN(C(CC(C)n3cccn3)=O)C2)=O)cccc2c1CCC2 c1(C(N2C(CN(C(C(CC)N(CC)CC)=O)C)CCC2)=O)cc2c(ccn2C)[nH]1 CC1CCCN1CC(=O)NC1CC(CNC(c2nocc2-c2ccccc2)=O)C1 N1(C(Cc2nc(NC(c3c(C)ccc(OC)c3)=O)sc2)=O)CC2(CCOCC2)C1 Cc1nnc(CC(=O)NCC2(C)CCN2C(=O)CCCC2CCCCC2)n1C c1(C(N2CCC(O)(C(C)NC(=O)COC(F)F)C2)=O)n[nH]c2c1CCSC2 C1(C(=O)NCC2N(C)CCN(C(C(C)n3ccnc3)=O)C2)CCC(C2CC2)CC1 CCC1=NOC(CC(=O)NCC=CCC(=O)NCCOCC(F)F)C1 C(=O)(CC1=CCCC1)N(C(C)C)CCNC(=O)C(c1ccc(O)cc1)C CC1Cc2c[nH]nc2CC1NC(=O)N(C)Cc1ccc(C(F)F)o1 C(c1ccc(F)cc1)=C(C)C(=O)N(CCC(O)C(C)(C)C)C.c1nn[nH]n1 Cc1coc(C=CC(N2CCC(CF)(NC(=O)CCCN(C)C)C2)=O)n1 C1(NC(CCc2ncn(C)c2)=O)CN(C(=O)COC(=O)CO)CC1N=[N+]=[N-] N1(C(C2CC(C#N)C2)=O)CC2CC(NC(c3cc(F)cc(F)c3)=O)C1C2 c1(OC)ccc(C(=O)C(=O)NC2CC(F)(CNC(c3cnc(S)[nH]3)=O)C2)cc1 CC1CC(C(=O)NC(C)CCNC(=O)C=CC2CCCC2)CCS1(=O)=O N1(C(C(C)(C)c2ccns2)=O)C2CCC1CN(C(=O)COCC(F)F)C2 c1(OC)ccc2cc(O)c(-c3ocnc3C(N3CCCCNC(=O)CC3)=O)cc2c1 CC(C)C(C(=O)NC1CCC1NC(c1cnc(Cl)[nH]1)=O)c1cnn(C)c1 C1(CCNC(C(C)(C)N(C)C)=O)CCN(C(c2ccc(C(F)(F)F)cn2)=O)CC1 Cc1cc(C(N2CCC3(NC(c4cnc(C(F)F)nc4)=O)CC3C2)=O)c(C)n1C Cc1cnn(C(C)C(=O)N2CCC2CC(=O)NC)c1.C1(C=O)CCN(C2COC2)C1 C(C(C(=O)N(C1CCC1C)C)NC(=O)CCC1CC1)OC(C)C c1(CN(C(=O)N(CC(O)CO)Cc2ccc(F)cc2)CC)nc(Cl)oc1C C#Cc1ccc(F)c(C(=O)NCC(CNC(=O)C(C)C2CC2)S(C)(=O)=O)c1 N1(C(C2CC(CC)(CC)C2)=O)CCC(=CCNC(=O)C(C2CC2)N(C)C)CC1 C(=O)(C(=O)CC(C)CC)N1CCC(OCC(N2CCCC(CC)CC2)=O)C1 C12(C(N(CC=C)C)=O)CC(CN1C(=O)CC(C)OC)C2 C1(C(=O)NCCC2(C(C)(F)F)CC2)CCCN1C(C1CC1C1CCCC1)=O CC1C2CCC(C2)C1C(=O)N(CCCC(=O)NCCOCCCF)C C1(C(N2CCC2CF)=O)CCC(NC(=O)C(O)c2ccsc2)CC1 C1(C(N(CCCNC(c2coc(Cl)n2)=O)C)=O)OCCOC1(C)C c1(C(N2CCCC(CN(C(C(CC)C#N)=O)C)C2)=O)c(C)ncnc1C C(=O)(C1CC(=O)c2ccccc21)NC12CC(NC(C=CC(C)C)=O)(C1)C2 CC(C)CC(C)CC(=O)NCC1(O)CCN(C(=O)C(F)(F)CO)C1 C(=O)(C1=CCOCC1)N(C)CC1CCN(C(c2nn(CC)c(C3CC3)c2)=O)C1 N1(C(c2c(C)ccc(C)n2)=O)CC2(CC(C(=O)NC(CO)CC(C)(C)C)CO2)C1 C1(OC(C)C(=O)NC2CCC2CNC(c2ccc(=N)[nH]n2)=O)CCCCCC1 Cc1cccc(CC(N2CCCC2Cn2cc(CC3CC4CCC3O4)nn2)=O)c1 c1(C(CO)NC(C2CCN(Cc3cnccc3Cl)C2)=O)ccc(Cl)cc1 N1(C(c2cccc(CC)c2N)=O)CCC2(CC1)CC2NC(=O)C1=CCCC1C c1(CN2CCN(C(=O)C(Cl)(Cl)Cl)C(CO)C2)c[nH]c2c([N+](=O)[O-])cccc12 CC(C(=O)N(C1CN(C(=O)C(C)OC)C1)C)OC.C1(C(=O)OC(C)(C)C)CCC1 N1(C(C2(C)COC2)=O)CCC2CCCN(C(=O)CS(C)(=O)=O)C2C1 C(c1ccccc1C)=CC(=O)N(C1CCN(C(C(C2CCC2)OCC)=O)C1)CC c1(OCCCC(=O)N(CC(C)NC(=O)C(C)OC)CC)ccc(C)cc1Br c1(OC)ccc(C(N2CC3C(NC(C4(NC(N)=O)CC4)=O)C3C2)=O)nc1 c1(CC(N2C(CN(C)C(c3cnn(C(F)(F)F)c3)=O)CCC2)=O)cccc(F)c1 N1(C(C2(OC)CCSC2)=O)CC2(CC(NC(=O)Cn3nnnc3C3CC3)CO2)C1 C(N=c1cc(NCCNC(=O)C(F)(F)F)nc[nH]1)C1(OC)CCSC1 CCCC(C(=O)NCCCNC(c1c(C(C)C)cnn1C)=O)C(C)C C(=O)(CCC(C)C)NCC1CC(F)(CNC(C(F)(F)C2(OC)CCC2)=O)C1 CC1(C)CCC(CNC(=O)C=Cc2ccccc2)(NC(=O)C(O)C(F)(F)F)CC1 N1(C(CCS(=O)(=O)N(C)C)=O)CCC2(CC(NC(C3C=CCCC3)=O)C2)C1 N1(C(CC(C)(C)C2CC2)=O)CC2CCCC(C1)N2C(=O)CCN1C(=O)CCC1=O C(=O)(CC(O)CCCCC)NC(CC=C)CNC(=O)CNC(C)=O C1(NC(=O)OCC)CCN(C(C2C3CNCC23)=O)CC1 Cc1cc(Cl)c(C(=O)NC2CCN(C(c3ccc(C)c(N)c3)=O)CC2O)cn1 c1(C(N2CC(N3CCN(C(C4C(C)CC4)=O)CC3)C2)=O)cc2cccc(Cl)c2s1 C1(C#N)(C(N2CCC(O)(CNc3ncc(C)cn3)CC2)=O)C(C#N)C1(C)C C12(NCC3(CC)CCOC3)CCC(C(=O)NC3(C)CCC3)(CC1)CC2 c1(C(N(CC(C)NC(C2(SC)CC2)=O)C(C)C)=O)nc(Cl)c(COC)[nH]1 C1(F)(C(N2CC(OC)C(NC(=O)C(C)c3cccs3)C2)=O)CCN(C)CC1 N(C1Cc2ccccc21)C(C1N(C(C2(C#N)CC2)=O)CC(F)C1)=O C1(C(=O)NC(C)CNC(C2CC(=O)N(O)C2)=O)CCc2cnnn2C1 N(C1CCCc2c1cnn2C(C)(C)C)CCc1ccc(C(C)(C)C)cc1 C(=O)(CC(C)(C)C1CCCCC1)N(CC(C)NC(=O)C=Cc1ccncc1)CC c1(C(N2CCC3CN(C(C4C(CN(C)C)C4)=O)C3C2)=O)cc([N+](=O)[O-])cnc1O C1(C(C)C)C(=O)N1.C(C(=O)N(CCn1cncn1)C1CC1)(C1CCCO1)OCC N1(c2c(C)c(N3CCC4(CCC4)C3)ncn2)CCC2(CC1)NC(=O)C(C)O2 c1(C(N2CC(=O)NCC2CC)C(=O)NC)ccc(OC)cc1C C1(C2CCN(C(=O)CCP(C)(C)=O)C2)(NC(C(C)OCC=C)=O)CC1 N1(C(c2cn(CCC(C)(C)C)nn2)=O)CCC(F)(CNC(C2CCOC2=O)=O)C1 CCCC(C)(C)C(=O)N1C(CNC(=O)Cn2c(C)c(C)sc2=O)CC2CC12 N1(C(Cc2nc(C)sc2)=O)CCCC(C)(C)C1CNC(C1(C)CCNC1=O)=O Cc1nc(C)c(CC(=O)NC2CCC(C(=O)NC3CC3c3ccn(C)n3)CC2)s1 c1(C(=O)NC2CCC(N(C(c3c(C)cccn3)=O)C)C2)cc(N)cc(O)c1C C1(N(CCCC)CCO)CCCN(C(=O)NCCNC(C2CC3(N)CC2C3)=O)C1 N1(C(c2scc(C)c2)=O)CC2(CCNC(c3ccc(Cl)cc3)=O)CCC1C2 Cc1noc(CCNC(C2(C(=O)NCCCN(C)C(C)C)CC2)=O)n1 C1(C(N2CC(NC(=O)CC(F)(F)F)CC(OC)C2)=O)CCc2cnnn2C1 CCCCC(CN=c1[nH]c(C)cc(Br)c1[N+](=O)[O-])NC(C1CCN1C(C)(C)C)=O Cc1ccc(C(N2CC(C(N3CC4CC4C3)=O)C(F)(F)C2)=O)cc1C#N N1(C(C(Cn2ccc(C)n2)C)=O)C2CCC1C(C)C(NC(=O)CC1CN(C)C1)C2 c1(C(=O)OCC)ncc(CNC(C)C(C)O)cn1 Cc1cc(Br)sc1C(=O)NCC(C)NC(=O)CCc1ccco1 CCCC(CCC)C(=O)N1CC(CNC(c2ccnc(NC(C)=O)c2)=O)CC1C N1(C(Cc2c(C)cccn2)=O)C2CC=C(C(=O)N3CC(O)(CC4CC4)C3)C1CC2 c1(OC)cc(N(C)C(c2c(C)noc2C)=O)cc(OC)c1 NS(=O)(=O)c1coc(C(=O)NC(CNC(c2cnn(-c3nccs3)c2)=O)CO)c1 c1(C(N2CCC(N(C(=O)CC(C)SC)CCCC)C2)=O)cccc(F)c1Cl c1(C(=O)OC)cocc1C(=O)NC1CCCC1C(N1CCC1C(=O)N(C)C)=O c1(C(=O)NCC(c2c(C)ncs2)C)c(-c2ccccc2)nn(C)c1Cl c1(OC)cccc(Cl)c1C(N1CC(O)(C(C)(C)CNC(C2CC(SC)C2)=O)C1)=O C12(OC)CCCC(CC(NC(=O)Nc3ccc(SC)nc3)C1)C2 N1(C(COC(CC)(C)C)=O)CCC(NC(c2c(Br)nnn2C)=O)CC1 N1(C(c2c(OC)cnnc2)=O)CC(C)CN(C(c2cncnc2C)=O)CC1C C=CCCC(C)N=c1[nH]c2c(c(=NC(C)c3ccc4ncccc4c3)[nH]1)CCC2 C1(CNC(CCSCCC)=O)CC2CCC(C1)N2C(=O)C(CO)NC(N)=O C1(C(=O)Nc2cn(COC)nc2)C2CC1N(C(c1ccc(Cl)cn1)=O)C2 c1(C(=O)NCCCOCCCNC)cc(S(C)(=O)=O)c(C)o1 c1(C(C)C)ccc(C(N2CC(NC(c3cc(C4CC4)ccn3)=O)CC2C)=O)cc1 c1(C(=O)NC2CC3C2CCN3C(c2csc(O)n2)=O)ccc2c(c1)CCNC2=O N1(C(c2cn(CC=C)nc2)=O)CCN(C(c2csc(Cl)n2)=O)CC(O)C1 C=C1CCC(C(N2CC=CC(NC(=O)C(C3CCC3)OC)C2)=O)CC1 C1(C(=O)NCC(CN(C)C)(C)C)CCCCN(C(=O)C=Cc2ccco2)C1 c1(C(=O)NCCC2(O)CN(C(C3CCC(C)(C)CC3)=O)C2)ccc2cnoc2c1 C1(C2N(C(c3ncc(CC)s3)=O)CCC2)CCN(C(=O)CN2CCN(C)CC2)CC1 C1(C(=O)NC(CNC(c2c(OC)cc(CO)cc2)=O)C)Cc2ccc(F)cc2O1 Cc1cc[nH]c1C(=O)NCCCCCNC(=O)C(C)NC(c1ccccc1)=O N1(C(Cn2c(C)nnn2)=O)CCC(C2CCCN2C(C23CC(CN2)C3)=O)CC1 CCC(CC(=O)N1CCCC(NC(=O)Cc2ccn(CC)n2)CC1)C(C)C C1(C(=O)NC2CC(NC(C(C)NC(=O)C3CC3)=O)CC2O)CCCC12CCC2 C1(C)(CNC(=O)COC(C)(C)C)CN(OCCNC(=O)C(N2CCOCC2)=O)C1 Cc1nc(C(C)C)sc1C(N1CCC(CNC(c2c[nH]nc2F)=O)C1)=O n1(CC)nc(C)c(CC(N2CCOCC(NC(=O)CC(C)O)C2)=O)c1C N1(c2c(Cl)ncc(OC)c2)CC2(CN(C(=O)CC3(O)CCC3)CCO2)C1 CC(CF)C(=O)NC(C)CCNC(=O)CCNC(c1ccco1)=O c1(C(N2CC(C)C(NC(=O)C(C3CCOCC3)O)C2)=O)ccc(O)c(N(C)C)c1 C1(NCc2cccc(-c3n(C)c4c(n3)cc(F)cc4)n2)CCCCC(P(C)(C)=O)C1 C=CCC(C)(CC)C(=O)NCCOC1CCN(C(c2ncccc2C)=O)C1 C(=O)(C(CCC)OCC)NCC(CNC(C1(C=C)CC1)=O)CO CCCCC(CC(=O)NCCCC1CC=CCC1)NC(c1cccc2ccoc12)=O N1(CC)CC(C(=O)NCCC2(CNC(c3cnn(CC(F)F)n3)=O)CC2)CC1=O N1(CCC(=O)NCC(=O)NCc2cn(C(C)(C)C)nn2)C(=O)CCC1=O N1(CC(=O)NC2CC(c3ccn(C)n3)C23CCC3)C(=O)C2CCCCN2C1=O Cc1onc(-c2ccc(F)cc2)c1C(=O)OCC1CCC(C2CC2)O1 c1(C(=O)NCC(O)CNC(C2(F)CC3CC2C3)=O)cncc2sccc12 C1(NC(c2cnc(SC)s2)=O)CCC(C)(CNC(=O)CCc2cccn2C)C1 N1(C(c2c(C)[nH]nc2C(F)(F)F)=O)CCCOC(CCNC(C2CC2(C)C)=O)C1 Cc1ccc(C(N2CC3C(CNC(C4(C)CCC(=O)NC4)=O)C3C2)=O)c(F)c1C c1(NC(C2(F)CCN(C(Cc3nc(C)on3)=O)C2)=O)cc(C)cc(Br)c1F N1(C(c2c(C)cc(Br)o2)=O)CCN(C(=O)C(O)C(C)(C)C)C(C)C1 C(CN=c1[nH]nc(C(C)(C)C)s1)=CCNC(C(n1ncc(C)c1)C)=O C1(C(N(C(C)CCNC(c2ccc(F)nc2)=O)C)=O)C2C3CCC(C3)C12 C1(C(=O)NCC(CC(C)C)C)C2CC(O)C(C2)N1C(=O)C(C)CC1CCC1 C1(NC(c2ccco2)=O)COCCN(C(=O)Cc2cccc(F)c2Cl)C1 c1(NC(C(C)N(C(C)=O)C)=O)cccc(NC(=O)C(C)(C)CN(C)C)c1 C(CC(F)F)(C(=O)NC1CC(C)(C)C12CC2)N(C(Cc1c(C)n[nH]c1)=O)C Cc1ccc(CC(=O)NCCC2CCC(NC(=O)C(=O)NCC(F)(F)F)C2)s1 c12cc([nH]n1)C(=O)N(CC1CC1)C1CCN(C1)C(=O)CO2.C12(CO)CC(O)C1C2 N1(C(C(CC)COC)=O)CCN(C(C2CC3(CC(OC)C3)C2)=O)C(C)C1 CC1(C)CCCCC(C(=O)NCCNC(C23COCC2C3)=O)C1 CCC(C)(CCC(C)C)C(=O)N(C(CNC(=O)CCCC1CCCC1)C1CC1)C C1(NC(CC(C)C)=O)CC1C1CCCN(C(c2cn(C)nc2C2CCCC2)=O)C1 N1(CC(COC)NC(=O)C(=O)NC(C)C(c2csc(=N)[nH]2)=O)CCOCC1 c1(C(=O)NCC2CC(NC(C34CC(C)(C3)C4)=O)C2)cc2n(n1)CCNC2=O c12cc(n[nH]1)C(=O)NC2.C1(C(CO)NC(COCCOC)=O)CCOC1 c1(C(N(CCCCN(C(c2cnc(C)s2)=O)C)C)=O)cccc(-n2cncn2)c1 N1(C(C2C(CCOC)C2)=O)C2CCCC1CC(NC(C1CC=CCC1)=O)C2 CC1(CC(=O)NCC(O)CCNC(=O)CCSc2ccccn2)OCCO1 C=CC(C)(C)CCCNC(C1CCCN(C(C2(SC)CC2)=O)CC1)=O CC(C)(F)C(C)(F)C(=O)NCCC1CC(NC(=O)CC2(C#N)CC2)C1 Cc1cc(-c2noc(CN3CCCC3c3nnc(C)s3)n2)on1 c1(NCCS(CC)=O)ccc(S(=O)(=O)Nc2ccc(OC(F)(F)F)cc2)cc1F C1(OC)CCN(CC=O)C1.C1(c2ccoc2)C(=O)NCC2(CC2)CC1.CO CC(O)C(C)CNC(=O)CCOCCN(C(=O)C(C)(C)n1ccnn1)C(=O)N(C)C N1(C(C(C(=O)OC)C)=O)CC(CNC(=O)Cc2ccccc2Cl)C2(CCC2)C1 N1(C(COCCCCC)=O)CCC(C(=O)NOC(c2cnn(C)c2)C)CC1 CCC(CC)C(C)C(=O)N1CC2CCCC2(Nc2cnc(C#N)cn2)C1 c1(N2CCCN(C(CC)=O)CC2)ncccc1S(C)(=O)=O.C(C)(C(=O)NC)OC=O c1(SC)cccnc1C(N1CC(O)CC1CNC(=O)C=CCF)=O C(=O)(C1=NOC(C)C1)NC1C(CCC)CN(C(C2CCC=CCC2)=O)C1 C1(CCOC)(NC(=O)C=C(C)Cl)CCN(C(=O)CCC2C(=O)NN=C2C)C1 C(=O)(CC(O)C(C)C)N(C)CC1CCN(C(C2(CCOCC)CCC2)=O)CC1 C1(CNC(C(C(C)C)O)=O)CCC2(CO1)CC(NC(=O)Cc1cc[nH]n1)C2 c1(C(=O)NC(C2CCN(C(C3N=C(C)SC3)=O)CC2)C)c(Cl)ccc2ccoc12 c1(CN2CC3C(C(N4CCSCC4)=O)(C3)C2)cccc2c1CCC2 C(=O)(CS(=O)CCC(F)(F)F)NCC1CCN(C(Cc2cn(C)nc2)=O)C1(C)C c1(CC(C(=O)N(C(C#C)C)C)NC(=O)CC2(OC)CCC2)ccc(Cl)cc1Cl N1(C(C2(OCC)CCOCC2)=O)CC2CCC(NC(c3n[nH]cc3Cl)=O)CC2C1 C(=O)(C(CCC)CC(C)C)NC(CC)CNC(=O)Cn1cc(C(=O)N(C)C)nn1 c1(CC)ccccc1C(=O)N(CC1C(CNC(=O)C(O)CC2CCCCC2)C1)CC C1(CNC(c2c(C)ccs2)=O)CN(C(=O)C(C(C)C)C2CCC2)C(C)(C)C1 N1(C(c2ccc[n+]([O-])c2)=O)CCC2(CCNC2)CC1 c1(C(=O)NC2CN(C(=O)C#CC3CCCCC3)C2)cc2c(nc1O)CCCC2=O N1(C(C23CC(CSC)(OC2)C3)=O)C2CCC1CN(C(C1CC3(CC3)CO1)=O)CC2 CC(C)CS(=O)(=O)CC(=O)N1CCCC(N(C)C(C2CC3C(C2)C3(F)F)=O)C1 C(=O)(C1CCc2c(F)cccc21)C(CCc1c2ccc(C)cc2[nH]c1)=O N1(C(C23CCC(OC)C2C3)=O)CC(C)C(C)(C(=O)NCC2CC(=O)N(C)C2)C1 Cc1noc(CNC(=O)NCc2nc(C(C)O)n[nH]2)n1 C(c1ccccc1OC(F)F)=CC(=O)NCCC1CC(NC(C2(C)C(C)C2)=O)C1 C(C(=C)C1CCOCC1)NC(CCC1CC(NC(COCCCC#C)=O)C1)=O c1(OC)ccn2ccnc2c1C(N1CCCC(N(C(C2CCSC2)=O)CC)C1)=O c1(C(N2C3(CN(C(c4cc(C(=O)OC)sc4)=O)C3)CC2)=O)cc2scc(Cl)c2[nH]1 CC1CCN(C(=O)CNC(=O)CS(C)(=O)=O)CC1N(C(=O)CCCCO)C Cn1nccc1C1CC1C(N1CCC(NC(=O)COCCOC2CC=CC2)C1)=O N1(S(CC)(=O)=O)CCCCC1C(=O)NCCCNC(=O)CCCc1ccccn1 N1(C(C2N(CCC)CCC2)=O)CCCCC1CNC(c1ccc(OC)cc1)=O C1(NC(CC2(C)CC2(Cl)Cl)=O)CCN(C(C2Cc3cscc3C2)=O)CC1F C1(N(C(CC(c2cccc(F)c2)C)=O)C)CCC(NC(=O)COCC(F)F)CC1 CN1CCCC(O)(CC(=O)NCCNC(C2(CF)CC2)=O)C1 C(=O)(C(C)CS(C)(=O)=O)NCC(c1cccc(C)c1)NC(C1(O)CCCC1)=O CN1C(=O)CCC1C(=O)NC(C(=O)NCCCOCCO)C1CC1 c1(C2CCN(C(C3CC4OCCC4N3)=O)CC2)cc(F)ccc1[N+](=O)[O-] CCC(CC(=O)NC(C(=O)N1CCC1(C)C(=O)NC)C(C)C)SC C1(C(=O)NC(CC)CNC(C2CC(C#N)C2)=O)COc2ccc(Cl)cc2C1 N1(C(CC(=O)OCC)=O)C2CCCC1CC(NC(c1cnn3ncccc13)=O)C2 S(=O)(=O)(c1cc(C(N2CC(NC(c3cnn(C)c3)=O)C(O)C2)=O)n(C)c1)N(C)C C1(NC(c2cccc(CNC(C(C(C)C)(C)O)=O)n2)=O)CC2CCC(C1)C2O c1(C(N2CCC(NC(Cc3c(C)n[nH]c3C)=O)C23CC3)=O)cccc(S(C)=O)c1 C(CCCCCCCCCO)N(C)CC1CCOC1 S(=O)(=O)(c1cccc(C(=O)NC(CNC(C2CC(CF)C2)=O)C2CC2)c1)N(C)C Cn1cc2cc(C(N3C4CN(Cc5c(O)cccc5O)CC34)=O)ccc2n1 N1(C(c2c(OCC)nccc2)=O)CC2CN(C(C3CC(O)CN3C(C)=O)=O)C2C1 C1(OC)(CNC(C2(c3cccnc3)CC2)=O)CCCN(C(=O)CC(C)C(F)F)C1 C1(CNC(C2(CC#C)CC2)=O)CC(C)(C)CN1C(c1csc(C)c1C)=O C1(CNC(COCCCC)=O)CC2(CCN(C(=O)CN3CC=CC3)CC2)C1 C(=O)(CC(=O)NCC)OC1(C(=O)NOCC2CCN(C3CC3)C2)CC(C(N)=O)C1 CCCCC(F)C(=O)N1CCCC(CNC(=O)CC(C2CC2)OCC)C2CC12 C1(NC(C2N(CC)CC2)=O)CC2CN(C(=O)CCC3CCCN3C)CC12 c1(CC(=O)NC(C(C)NC(C2CCC(=O)N2C)=O)(C)C)cccc2ccccc12 N1(C(C(F)=CC)=O)CCN(C2CCCN(C(c3nncs3)=O)C2)C(=O)C1 C12(NC(CONC(=O)Cc3ccc(O)cc3)=O)CCC(CC1)OC2 C1(C(N2CCOCC2)=O)CC(O)CN1Cc1ccnc(-c2cccc(F)n2)c1 c1(C(=O)NC(CC)CNC(c2ccnn2C(C)(C)C)=O)cn(C(F)F)c(C)n1 C1(NC(c2[nH]cc(C)c2)=O)CCC(CC(=O)N(C2CCOC2=O)C)CC1 C1(C(=O)NCC2CCC2)CCCC12CCN(C(c1cc(I)ccc1F)=O)C2 c1(C(N2CCCCC(NC(C3CC(=O)N(O)C3)=O)C2)=O)cc2cnccc2[nH]1 c1(OC)cc(F)ccc1CC(N1CC(O)CC1C(=O)NCC1CN(C)CCO1)=O c1(SC)cc(C(N2CCCC2CN(C)C(C2CCO2)=O)=O)c(Cl)cc1Cl CC(CNC(=O)C(C1CCC1)NC(c1ccns1)=O)CCCO Cn1c(CC(=O)NC2COCC2C(=O)Nc2cnccc2CO)nnc1S c1(N(C)C)ccc(F)c(C(=O)NC2CC3CC2CN3C(=O)C2=CCCC2)c1 N1(C(COCC(=O)NC)=O)CCN(CCNC(=O)C(C)Cc2c(C)noc2C)CC1 C1(C)(C(=O)OCc2c(COC)cccc2)CC2CCC1CC2=O c1(OC)ccc(-c2ccc(-c3nccn3CCC(=O)O)s2)cc1Cl N1(C(CCC(=C)Cl)=O)CCC(C)C(N(C)C(c2ccc[nH]2)=O)C1 C1(C(=O)NCC=C(C)C)C(C)CCN1C(c1cccc(C)n1)=O C12(C(N)=O)C3C4C1C1C2C3C41C(N1CCCC(C)(CNC(=O)C2=CCCC2)C1)=O C1(N(CCOC)C(C2C=CCCC2)=O)CCN(C(c2snnc2C)=O)CC1 Cc1cc2nccnc2cc1C(=O)NC1CCC1NC(C12CC(C)(C1)OC2C)=O C(=O)(C1=NOC(CNC(c2cnnn2C)=O)C1)NCc1nnc(C)n1C Cc1cccc(C)c1CNC(=O)Oc1cnccc1CO C1(CC(=O)NC2CCCCC2NC(c2nnc(C3CC3)o2)=O)C=CS(=O)(=O)C1 C1(C(=O)NCCC(C)NC(=O)CCc2csc(Br)c2)NC(=O)OC1C N1(C(c2cccc(CCC)c2)=O)CCCCC(NC(=O)C(CCO)N(C)C)C1 n1(CC)ccc(C(=O)NCC2CN(C(=O)C(C)NC(=O)OC(C)(C)C)C2)cc1=O C1(C(C)=O)CC2(CC(NC(=O)CN3CCSCC3)C2)C1.C12(CC1)C(=O)N2 N1(C(CCN(CCCCC)C)=O)CCC(C#N)(C2(C#C)CCCC2)CC1 Cn1ncc2c1CN(C(c1cc3c(c([N+](=O)[O-])c1)OCO3)=O)C2C(=O)O c1(C(N2CC(CCC)C(NC(C3CC(O)(C#N)C3)=O)C2)=O)noc(C)c1[N+](=O)[O-] N1(CC(CN(C2C3CC=CCC23)C(=O)OC(C)(C)C)O)CCP(C)(=O)CC1 C(=O)(C1CCc2cc(OC)ccc21)NCC(=C)CCNC(C1(CO)CCC1)=O C(c1cc(C)cc(C)c1)=CC(=O)NCC1(O)CN(C(COCCC#C)=O)C1 C1(CNC(c2cc(I)sc2)c2nnnn2C2CCC2)COCC2(CCNC2)O1 C(=O)(C1=C(CC)OCCC1)NCC(c1ccc(C)cc1)NC(CCC)=O c1(OC)c(C(=O)NCC2CCCN2C(c2nnc(C)s2)=O)oc2ccccc12 N1(C(C(=O)OC)=O)CCN(CC=O)CC1.N1(CCCCS)CCCCC1 c1(CC(=O)NC2(CC=C)CCN(C(=O)C#CC3CCC3)C2)cc(OC)ccc1Cl c1(N2CCC(N(C(=O)CCCCCF)CCC)C2)ncn(C)c(=O)c1Br c1(C(=O)NC2CCC3(C(NC(=O)C=C4CCC4)C3)CC2)coc2c1C(=O)NCC2 c1(C(N2C(CN(C(=O)CNC(=O)C(C)(C)C)C)CCC2)=O)ccc(N)cc1F C1(C(=O)NCC2CC3CN(C(c4ncncc4Cl)=O)CC23)CCc2nc[nH]c2C1 N1(C(c2n(C)nnc2)=O)CCCCC1CC(N1CCC1c1ccccc1)=O C1(NC(C2C(C)CCN2C(c2nc(=N)cc[nH]2)=O)=O)CCCC(O)C1O C12(NC(C(CCC)OCC)=O)CCC(C1)N(C(c1cnn(C)c1Br)=O)C2 Cc1ccn2c(C(N3CCC3CNC(C3C(F)(F)C34CCC4)=O)=O)cnc2c1 C#CC1(C(=O)NCCCCNC(C2CCNC2=O)=O)CCC1 CCCCC(O)CC(=O)NCC1(Nc2ncc(C(=O)OC)cc2Cl)COC1 C(N=c1nc(N2CCC(COC(C)(C)C)C2)c2c([nH]1)CCS2)C1(CCC)CCC1 N(C(=NCC(C(F)(F)F)Nc1c(C)ccc(C)n1)NCC1CCCC1)C(=O)N(C)C c1(C(=O)NC2CC(CCNC(=O)C(F)C(F)(F)F)C2)cccc2c1OCCCO2 C1(NC(C2(C)CC=CC2)=O)CS(=O)(=O)CC1NC(c1ncc(F)cc1N)=O C1(C(=O)NCCCn2cc(CO)nn2)CC=CCN1C(=O)CC1CCCO1 Cc1nc(NCC2CCCCO2)cc(=NC(C)c2cccc(O)n2)[nH]1 C1(CNC(CCCSC)=O)CC2(CCN(C(C3Cc4nncn4C3)=O)CC2)CO1 c1(OC)cc(C)sc1C(=O)NCC1CCCC1NC(=O)C=CSC Cc1ccc2cc(C(=O)NCC(C)NC(c3cc4ccsc4[nH]3)=O)ccc2c1 N1(C(CCn2ncc(C)c2)=O)CCC2(CCC(NC(=O)C(C)S(N)(=O)=O)C2)CC1 c1(C(=O)NC2C(NC(=O)C(F)(F)c3cncs3)CC2)cncc(N2CCCC2)c1 N1(C(Cc2c(C)noc2)=O)CC2CCC1C1CN(C(=O)C(C)(C)N(C)C)CC21 C(=O)(C1=C(Cl)CC1)N(CCNC(C(n1ccc(C)n1)(C)C)=O)Cc1ccccc1 N1(C(c2cc(OC)no2)=O)CCCC2(CNC(C3C(C)C3C)=O)CCCCC12 c1(C(=O)NC(C2CCN(C(c3c(CC)nns3)=O)C2)C)cccn2cc(C)nc12 c1(C(c2nnnn2C2CCOCC2)NCC(COC)C)cn(C)nc1I c1(NC(C=C(C)C(F)F)=O)ccc(OCCC(N)=O)cc1.C12CCN1C2=O C1(CNC(C2(SC)CN(C(c3cn(C)nc3O)=O)C2)=O)CCCC12CCC2 n1(CC(N2CCC(CCNC(CCC(C)(C)F)=O)CC2)=O)ccc2ccccc12 C=CC1(C(=O)NCC2CN(C(c3ccc(CC)o3)=O)CC2C)CCCC1 N1(C(CCN(CCCCOC)C)=O)CCC(C)(CCNC(=O)CCC(C)OC)C1 Cc1cc(CNC(=O)NCC2COCC(C)(C)O2)nc(Cl)c1Br c12ccc(cc1)c(=O)[nH]2.C1(C(N(CCN(C(=O)C(C)(C)C)C)C)=O)CCCC(O)C1 CCC(C)C(C(=O)N(C(C(N)=O)C1CC1)C)NC(C1CC2(CC(=O)C2)C1)=O c1(C(N2CCCC2c2ncc(Br)cn2)=O)nc(Cl)nc2c1CCOC2 C1(CNC(c2ccn(C)c2)=O)CCCCN(C(=O)Cc2cccnc2N)C1 CC1CN(C(c2cc(C(F)F)nn2C)=O)CC(C)C1NCc1cc(C2CC2)no1 C(=O)(C(C(C)C)NC(C)=O)NCC1(OCC)CN(C(=O)C(F)C2CCCC2)C1 CCCCCCCCC(=O)NCC1(C)CCCN(C(c2cnccc2SC)=O)C1 Cc1ncnc(C(=O)NCc2ccc(C(=O)N(C)Cc3cnc[nH]3)cn2)c1C CC(C)C(C)C(=O)NC1CN(C(c2csc(C(F)F)n2)=O)CC1C N1(C(CCCCC#C)=O)CCC2CCN(C(c3noc(C)c3Br)=O)CC12 Cc1c(C(N2CCCC(O)(CNC(C3CC4CC3C4)=O)C2)=O)ccc(Cl)c1Cl Cc1cc(O)ncc1C(N1CCCC(N(C(=O)COc2cnn(C)c2)CC)C1)=O C1(C(=O)NCCN(C(=O)COc2ccn(C)n2)C)C2CCC12c1ccccc1 CC1CC(NC(c2ccnc(C(F)F)c2)=O)CN(C(=O)CC2CCCCC2)C1 N12CCn3c(nnc3C1)C2.c1(CC2CC=CCN2)cnc(C2CC2)cn1 C1(C(=O)NC(CCC)C2CCCC2)(NC(=O)CNC(C)=O)CC1(C)C C(C)(CCCC(=O)NC1CN(C(=O)NCC)C1)NC(c1c(C)nc(CC)o1)=O Cc1nn(C)c(=O)c(C(=O)NCC(C(C)C(C)C)NC(c2ccc[nH]2)=O)c1C c1(CC)cncc(CNC(C2CC23CC(NC(c2cnc(O)n2CC)=O)C3)=O)c1 c1(C(N(CC(=O)Nc2c(C(C)C)nsc2)C2CCC2)=O)cnn2c1CCC2 C(C(C)(C(=O)N1CCCC(C(F)F)C1)NC(=O)CN1CCC(O)CC1)SC Cn1nc2c(c1C(=O)NC1CCCC1CNC(=O)CN(C)CC1CC1)CSCC2 C#CCC(C)(C)C(=O)NCC(O)CNC(c1cnnn1Cc1ccccc1)=O c1(C(N2CC(NC(c3ccc(O)nn3)=O)C3C2C3)=O)cc2nccnc2cc1F c1(OCC(=O)N(C(Cc2cn(C(C)C)nn2)C(N)=O)C2CC2)cccc([N+](=O)[O-])c1 c1(C(C)C)cnc(C(=O)OCCSc2nc[nH]n2)c(C#N)c1 C12(CC(=O)NC(CN(C(C(C=C)C)=O)C)C)CCC(CC1)C2(C)C c1(C(C)OC(c2nc(C)n(Cc3ccccc3)n2)=O)cc(F)c(F)c(F)c1 C1(C#N)(C(N(CCCNC(C2CCC(C(F)F)CC2)=O)C)=O)CCS(=O)(=O)CC1 C(=O)(CCCN(C)N=O)NC1(COC)CCN(C(C2CC(C#C)(O)C2)=O)C1 c1(C(N(CCC(N2C(CCCC)CCC2)=O)C)=O)ccnc(C)n1 C1(NC(C2N(C(C)=O)CCC2)=O)CCCN(C(=O)CCO)C1.c1(CSC)cn(CC)nn1 c1(C(C)C)ccc(S(=O)(=O)NC2CCN(S(=O)(=O)c3cnn(C)c3)CC2)cc1 C12(CNC(=O)C=Cc3ccco3)CCCCC1CN(C(c1cnsn1)=O)C2 n1(CCCC(=O)NCC2(F)CC(NC(C3C(C)(C)C3(C)C)=O)C2)c(O)nnc1O C(=O)(C(CO)NC(=O)C(c1cccnc1)N)OC c1(C(=O)NCC2(C(N3CCCC(CCF)C3)=O)CC2)cnc(C(F)(F)F)nc1 N(C1CCCn2ccnc21)C(CC(CNC(C1(C)CC(F)(F)C1)=O)OC)=O c1(C(=O)OC(C)(C)C)cc(C(=O)NCCCNC(=O)C=Cc2ccc[nH]2)cs1 C1(NC(Cc2[nH]c(=N)sc2)=O)C2CC(O)C1N(C(=O)Cn1nc(Cl)ccc1=O)C2 C12(CNC(C3(CC)CC3)=O)CC(CO1)N(C(=O)Cc1ccccc1CC(C)C)C2 C(CO)(C1CCc2ccccc21)N(C(CCCNC(=O)OCCC(C)C)=O)CCO C(=O)(CCN(OC)C(=O)C1(C)CCCN(C)C1)NCC#CC CC(C)CS(=O)(=O)CC(=O)NCCN(CC(C)O)C(c1ccc(=O)n(CCF)n1)=O C(=O)(CCCCCC(C)O)NCC1(C)CCCN(C(CCC(=O)NCC)=O)C1 C1(C(=O)NCC2CC3CCC2N3C(C2CCCN2C2CC2)=O)CCc2ccnn2C1 C1(COC)CCC(C)N(C(=O)CC2CCN(c3cc(C(F)(F)F)nc(Cl)n3)C2)C1 C1(NC(C(CCNC(C23OCCC(C)(C2)C3)=O)O)=O)CCCCC12CCC2 c1(-c2ncc(C(N(CCCNC(=O)C=Cc3nccs3)C)=O)s2)ccccc1F C(C(C(=O)N1CC(CNC(C2CC2)=O)C1)N(C)C)OC.c1(CNC=O)ccccc1 c1(N2CCC(CCO)C2)nccc(N2CCC(c3ncncc3F)CC2)n1 N1(C(C(C)Oc2ccccc2)=O)CC2CC1C2NC(c1c[nH]c(C(N)=O)c1)=O C(=O)(C(CC(C)C)c1ccccc1)NCC(C)N(C(c1c(OC)csc1)=O)C C=C1Cn2c(C(N3CC(C)CCC3CNC(c3c(C)[nH][nH]c3=N)=O)=O)nnc2S1 CN(C)NC(=O)CCC(=O)NC1CCCCC1NC(c1cc(C(F)(F)F)c[nH]1)=O C12CC3CCC(C1)N3Cc1cncc(c1)C(=O)N2.N1(CC)CCCC1CO C(=O)(CC(CC)C(C)(C)C)N1CCC(OCCC)C1.N12CCC(CC1)SCCC2=O C(CC)(C(C)CN(C)C)NC(C(CNC(c1c(C)nns1)=O)N(C)C)=O Cc1nnc(CCC(=O)NC(CO)C(C)NC(=O)CC2CC2(C)C)n1C C1(CNC(C2N(C)C(=O)NC2)=O)CC2COCC2N1C(c1csc(Cl)c1)=O CCCCCCn1nnnc1SC(=O)CC1C2COCC12.C1(CCO)CN1 c1(C(C)NC(C)Cc2ccccc2Cl)ccc2nc[nH]c2c1 Cc1cc(CNC(=O)Nc2cn(CC3(C(=O)O)CCCO3)nn2)sn1 Cc1cccc(C(=O)NC(CNC(C2CC3CCC2O3)=O)CC(C)C)c1 c1(C(N2C(CNC(C=CS(C)=O)=O)CC(O)C2)=O)cccc(Br)c1F Cc1ccc(F)c(S(=O)(=O)NCCC(C)NC(=O)C=CC2CC2)c1.C1C(=O)O1 S(=O)(=O)(CCC(C)C(F)F)NCC1(C=O)CC1.Cc1ccc(O)cc1 C1(C#N)(OC)CC(C(=O)NCCN2CCC2c2cc(C)[nH]n2)C1 S(=O)(=O)(c1ccc(NC2CCCSC2)cc1Br)N(CCOC)CC1CCCO1 c1(N(CC(F)(F)F)C(CC2CCN(C(C(=O)OCC)=O)CC2)=O)ncc(C#N)cn1 C1(C)(CNC(C(CSC)NC(c2ccc(C(C)=O)o2)=O)=O)CC=CCC1 C(CC(C(=O)NCC1CCCCS1)NC(c1cnc(=N)[nH]c1)=O)N(C)C N1(C(c2ccc(C=C)cc2)=O)CCN(C(=O)O)CC(C)C1.C(C)(C)(C)N(C1CC1)CCCCl c1(C(N2CC(CNC(C3CN(C(C)=O)C3)=O)C(F)(F)C2)=O)c([N+](=O)[O-])c(C)nn1C c1(C(=O)NC(CC)(F)F)nc2ccccc2n1-c1cccc(Cl)c1 N1(C(C(C)(C)CF)=O)CCC=C(C(=O)N(C2CC2)CC2CCOC2)C1 C(=O)(C(CNC(=O)C(F)=C(C)C)CC1CC1)NC1(C(C)OC)CC1 C(=O)(CC(C)CC(F)(F)F)NC1C2(CN(C(c3c(CC)cccc3)=O)C2)CCC1 C#Cc1cccc(C(=O)NC2CC(C)(NC(c3cc(C)nc(C)c3)=O)C2)c1C N1(CCOC)CC(NC(=O)NCC2CCC(C(F)(F)F)O2)CCC1=O c1(OC)ccccc1CC(C)CC(=O)NC(CNC(=O)CCNS(C)(=O)=O)C1CC1 c1(C(=O)NCC(CO)OC)c(F)ccc(NC(c2cccc(Cl)c2)=O)c1F c1(C(c2n(CCC)nnn2)NCC(C)(CC)C(=O)NC)ccc2occ(C)c2c1 C(=O)(C(CC(C)C)NC(c1ccc(C)nn1)=O)N1CC(C(=O)OC)(SC)C1 N1(C(C=Cc2c(C)ncs2)=O)CCCC2CN(C(=O)CCCC(C)O)CC12 C(=O)(CCC(C)(C)[N+](=O)[O-])N1CC(OCCC(=O)NCCCCCCOC)C1 S(=O)(=O)(c1cccc2c(Cl)nccc12)N1C2CCN(C(CC)=O)CC2CC1 C1(NC(=O)CCN(CCCO)C(c2ncccc2Cl)=O)CC2CCC1O2 c1(C(=O)NCCc2cc(C(N(C)Cc3nc(C)on3)=O)no2)cccnc1S c1(C(N(CC(O)CN(C)C(C2CCOC2)=O)C)=O)ccc(C(C)(C)C)s1 c1(C(=O)NCC(C2CCCC2)NC(CC2(C)CC2(Cl)Cl)=O)cccc(C2CC2)c1 C(CCNC(C1CCCCC1n1ccnc1)=O)(C(C)C)NC(c1cc(C)[nH]n1)=O N1(C(C(COC)(F)F)=O)CCC(C)(C)C(CNC(C2(SC)CC2)=O)C1 c1(C(=O)Nc2ccc(C(F)(F)F)cc2)cc(Cl)ccc1NC(CCC)(CC)CC C(=O)(C(F)C(F)(F)F)NC1(CNC(c2c(OCC)c[nH]n2)=O)CCOC1 N1(C(C2C(C(=O)OC)C2)=O)CCCC(N(C(=O)CCn2cnnn2)C)C1 c1(SCCC(=O)N(C)CCNC(C2CCCC2n2cccc2)=O)cccc(Cl)c1 Cc1ccc(C(=O)NC2CN(C(c3cc4ccccn4n3)=O)CC2F)c([N+](=O)[O-])c1 C1(C)(CN(C(=O)CC2(NC(=O)CCc3nncs3)CCC2)C)CCOC1 c1(C(=O)NC2C(OC)CN(C(=O)Cc3cnn(C)c3)C2)cc2c([nH]1)CCOC2 CN=c1nc(N2CCC(C)(N(C)C)C2)[nH]c(=NCC2(F)CCOCC2)[nH]1 N1(C(Cn2ncc(CC)c2)=O)CC2CCCC2(CNC(C2CC2OC)=O)C1 c1(C(=O)NC(C(C)C)C(=O)Nc2ccccc2C2CC2)cccn2ccnc12 CCCCC(CNC(c1cnn(Cc2ccc(Br)cc2)c1)=O)CO C(=O)(CC1OC(=O)c2ccccc21)N(C)CCNC(C1Cc2ccc(F)cc2C1)=O C(=O)(C1=CCS(=O)(=O)C1)NC1C2CC(NC(=O)CCc3ncccn3)CC21 N1(C(c2c(C)c(Br)cnc2)=O)CCN(C(=O)Cc2ccnn2C)CC2(CC2)C1 N1(C(CC2C(C)OCC2)=O)CCc2nc(O)cc(C(=O)Nc3cccnc3F)c2C1 C(=O)(C1=CC2(CCN(C(=O)C=CC3CC3)C2)C1)Nc1ccc(C(C)C)nc1 C(C(C)(C)C(=O)NC(CC1CC1)C(=O)OC)N(C(C(C=C)OC)=O)C C(=O)(C(O)C(C)(C)C)N1C(CN(C(c2nc(OC)nc(O)c2)=O)C)COCC1 O=C(CC(F)(F)c1ccccc1)NC1CCCCC1CNC(c1cccnn1)=O N1(C(c2cnc(C(C)OC)s2)=O)CCN(C(C23CC(F)(C2)C3)=O)C(CO)C1 N1(C(C(Br)=C(C)C)=O)CC2(COC(CNC(C3CCCC(O)C3)=O)C2)C1 C(C(C)C(C)(C)C)N(C(c1ccccn1)C)Cc1ccc(OC)o1 c1(C(=O)NCC2CN(C(C34CCC(CC3)O4)=O)CCCO2)ccc2nc[nH]c2c1 C1(NC(C(CC)c2cccnc2)=O)C=CCC(C(=O)N(C2(COC)CC2)C)C1 C(C(=O)N1CCN(C2CCN(C(=O)CC(C)(O)COC)C2)CC1)(C(C)C)OCC CC1C(C(=O)NC2CN(C(C3CCC3)=O)CC2Cc2ccccc2)CCN1C c1(C(N2CCCC2CCCO)C(=O)NCc2ccccc2)ccc(O)cc1Cl C(=O)(CCCCNC(C)=O)NC(CCN(C(c1cnc(SC)s1)=O)C)C c1(OCCCC(C)NC(=O)Nc2cc(Cl)c(Br)cn2)ccc2c(c1)OCO2 N1(C(c2n(C)ccc2)=O)CCCOC(CNC(=O)CC2CCN(CCF)CC2)C1 C1(=O)CCCCO1.c1(C2CCN(CC)C2)ccccc1F.N12CCCC1C2=O c1(C(=O)NC(C(C)NC(c2ccoc2Cl)=O)C)cc2ccc(F)cc2nc1O NC1CN(C(=O)CC2C=CCCC2)C2(CCC2)C1 Cc1ccc(C(N2CCCN(C(=O)CC3(CO)CCCC3)CC2)=O)cc1CO N1(C(C(CC=C)C(C)C)=O)CC2(C1)CN(C(=O)CSCc1ccccc1)CCO2 N1(C(C2=CC(C)(CC)C2)=O)CC(C2CCCN(C(c3cnc(Cl)cc3Cl)=O)C2)C1 C(=O)(CCC(F)F)NCC(C)CC1CN(C(=O)Cn2cc(C#N)cn2)C1 C(C(=O)NCC1(CO)CCN(C)C1)(C(C)O)OC.C12CC1C(=O)NC2 C1(NC(CCSC)=O)(CNC(=O)C(C)(C)CC2CC2)CCCCC1C N1(C(COC)=O)CC2CN(C(=O)CCCn3cccn3)CCC12 C(CC(O)CNC(=O)CCOCC1CC1)OC.C1(=O)CCCN1C Cn1c(C(N2CCN(C(=O)C3=CCC3)CC2CF)=O)cccc1=O Cc1c(C(=O)NCC(CNC(=O)C#CC(C)(C)C)CO)cncc1Cl N1(C(c2ncc(C)cc2O)=O)CCC2(CCCN2C(=O)CCCF)C1 C#CC1CN(C(C(=O)NC2CCCCC2)C(C)CC2CCOCC2)CCO1 CC1(C(=O)NCC2CN(C(=O)COC3CCOC3)C2)CC2CCC1C2 Cc1cc(C(=O)NC2CC(CNC(c3ccc(CO)o3)=O)CC2O)c(Cl)cc1F c1(CC(C(=O)OC)NC(=O)Cc2c(C)nn(C)c2C)cccc2c1OCCO2 Cc1cc(=NC(=O)CN2CCN(C(C3(C)CCC(=O)N3)=O)CC2)[nH]o1 c1(C(=O)NC2CCN(C(C(C)C)=O)C(C)C2)ccc2c(c1)C(=O)CCC2(C)C C12(CNC(CSC(C)C)=O)CCCC1CN(C(C1CCC3(CCC3)CO1)=O)C2 N1(C(C2C(SC)CCC2)=O)CC(F)(F)CC1(C)CNC(c1snnc1C1CC1)=O C(=O)(C(=O)N1CCC(C(=O)NC(C)C(C)(C)O)O1)N(C)C c1(C(=O)NC(C(C)NC(=O)CSC2CC2)CO)cc2sccc2cn1 C1(C(N2CCCC(OC)C2)=O)CC2CCC(C1)N2C(=O)CCn1ccnc1C c1(OC(C)C)cc(NC(=O)NC(c2ccccn2)CCc2ccccn2)nn1C n1(CC)ncc(Cl)c1C(N1CCC(C(C)NC(C2(C#N)CC2(C)C)=O)CC1)=O c1(C(=O)NC2CC(O)(CNC(CC(CC)C3CCC3)=O)C2)nc2ncccn2n1 C12C(CCN1C(=O)CNS(=O)(=O)N(C)C)N2.CC1CC(C(=O)N(C)C)C1 C1(CC=C)(C(=O)NCC(C)(O)C2(C)CC2)CN(C(=O)C(F)OC(F)(F)F)C1 c1(C(=O)NCCCC2OCCN(C(c3cnn(C)n3)=O)C2)cnc2[nH]ncc2c1 c1(OC2CCC(N(C)C)CC2)ccc(-n2nnnc2Nc2ccc(Cl)cc2)cc1 N1(C(Cc2c(C)nc(S)s2)=O)CCC(NC(=O)C=CC(=O)NC2CC2)C(CO)CC1 N1(C(CCNC(=O)NC)=O)CCc2sc(CNC(C3CCCN3C=O)=O)nc2C1 Cc1coc(C(=O)NCC(=O)NCc2cn(-c3cnn(C)c3C)nn2)c1C C1(CC(N2CC(COC)C2)=O)CC(NC(c2ccnc(C)c2)=O)C1(C)C C(=O)(C1=NOC(C)(C)C1)NC(CN(C(c1scnc1Br)=O)CC)C C12(NC(Cc3cccc(C)c3)=O)CCCC1N(C(c1ccc(F)cc1Cl)=O)CC2 c1(C(C)O)ccc(C(=O)NC2COCC2C(F)(F)F)cc1.c12ccc(nc1)[nH]2 c1(C(=O)OC)c[nH]c(=NCC(C)CNC(C23CCC(CO)(CC2)CC3)=O)s1 c1(C(N2CC(C3N(C(c4n(C)ncc4)=O)CCC3)(O)C2)=O)cnn(C)c1C(F)F C1(C(N(C)CC2(CNC(C3CCC(=O)N3)=O)CC2)=O)CNS(=O)(=O)C1 C1(NC(CCCCOC)=O)CC2(C1)CN(C(=O)CCOC)C2 c1(C(=O)NC(CC=C)CNC(=O)OC(C)(C)C)c(C)[nH]c(-c2nn[nH]n2)c1C c1(C(=O)NC(C)CCNC(C2CC(=O)N(C3CC3)C2)=O)cccc(Cl)c1F Cc1nc(NCC23CC(CN2C(C2CCCCN2C)=O)C3)cc(O)n1 c1(C(N2CCC(NC(=O)CCc3cccs3)(CO)C2)=O)ccn2c(O)nnc2c1 c1(N(C(CO)C2CC2)C=O)ccc(OC(C)(C)C)cc1.C1(N)CCCC1(C)C1CCC1 Cc1cccc2oc(C(N3CC(N(C(=O)CCC4(C)CC4)C)C4(CC4)C3)=O)cc12 C1(C(=O)NC(CCNC(C(C=C)OC)=O)(C)C)CCOC1C=C C1(CC(=O)NC(C)CCN(C(=O)CN(S(C)(=O)=O)C)C)OCCC1(C)C CC(c1ccccc1F)=CC(=O)NCC1CN(C(=O)C(F)C2CCC2)CCN1C c1(N(CC(=O)Nc2cc(F)cc(Cl)c2)C)nc(NC2CCC2)c2ncsc2n1 c1(C(C(=O)NCCC)N(CC(F)(F)F)CC2CC2)ncc(C)cc1OC c1(CC)cccc(C(=O)N(CCCNC(=O)CCNC(=O)CN2CCCC2)C)c1 C1(C(=O)NC2CC(N(C(C(C)Cc3cnco3)=O)C)C2)CC12CCCCC2 N1(C(c2cccc(C)c2)=O)CC2CCN(C(c3ccc4c(c3)COC4)=O)CC2C1 N1(C(Cc2ccn(CC)n2)=O)CCCC12CCN(C(c1csc(C(N)=O)n1)=O)C2 c1(C(=O)NCC2(CNC(CN(C(C(C)C)=O)C)=O)CC2)nc(-c2cc[nH]n2)cs1 c1(C(=O)NC2C(NC(C3N(CC)CCOC3)=O)CCC2)n[nH]c2ccc(Cl)cc12 NC1CS(=O)(=O)CC1CN1CCC(c2nccn2C(F)F)CC1 C#CC1(O)CCCN(C(C2CC(CNC(C3CCNC3=O)=O)C2)=O)C1 C1(NC(C2N(C(c3nc(C)sc3)=O)CC=C2)=O)CCCC2(CC1)CC2 c1(SC)ccnc(N2CCC(NC(c3ccnc(O)c3)=O)C2)n1 C(=O)(C(O)C(C(C)C)OC)NC1CCN(C(c2ccc(C#C)cc2)=O)C1C(C)C N1(C(CN(C(c2cnc(C)o2)=O)CCO)=O)CCN(C(=O)C=CC(C)C)CC1 c1(CC(=O)NCCN2CCN(C(=O)COC(F)F)CC2)cccc2ccoc12 CP(C)(=O)c1ccc(C(=O)NC2CC(CNC(C3CC4COCC4C3)=O)C(O)C2)o1 N1(C(C=CC2(C)COC2)=O)CCC2CN(C(=O)CCC3CCCO3)CC12 CCC(N=c1[nH]c2c(c(=NCCCCCCO)[nH]1)SCC2)c1ccccn1 C1(C(=O)NCC(CO)NC(CCC#C)=O)CCC(=O)N(CC(F)(F)F)C1 C1(C(=O)Nc2c(C)n(CCN(C)C)nc2)CCN(C(c2c[nH][nH]c2=N)=O)C12CCC2 c1(OC)ccc(O)cc1-c1cn(C(C)CNC(c2ccc(C(N)=O)[nH]2)=O)nn1 CC1(C)CC(C(=O)NCCC(=O)NCc2ccc(N3CCOCC3)cc2)CO1 N1(C(C2C(OC)CCCC2)=O)CC2(C1)CN(C(c1coc(C)c1)=O)CCO2 C1(CCNC(C2(C)COC2)=O)CCCN1C(=O)CC1COCCO1 C1(C(=O)NC2C(CC)CNC2)CC2CSCC(C1)C2 C1(NC(CN(CCOC)C)=O)CCC2(CCCN2C(=O)C2=NOC(C)C2)CC1 C(=O)C#CC1(C(F)(F)F)CCCCC1.c1(N(C(CCOC)C)CC)cccc(C#N)c1 C(c1ccccc1)=C(C)C(N1CC=CC(NC(C2CC2c2ccncc2)=O)C1)=O c1(C(=O)NC2CCN(C(c3cccc(Cl)c3)C)CC2)cccc2nsnc12 N(n1c(C2CCN(C(=O)C=C(C)C(C)(C)C)CC2)noc1=O)C(C)=O c1(CC(=O)NCCN(C(c2ccc(OC(F)F)cc2)=O)CC)ccnc(F)c1F c1(C(=O)NC2CC(O)(CNC(c3c(C)n(C)cn3)=O)C2)ccc(O)nc1Cl c1(C(N2CC(F)CC(C(=O)NCCS(C)(=O)=O)C2)=O)cc(O)cc([N+](=O)[O-])c1 c1(C(=O)NC2C(CNC(c3ccnnc3)=O)CC2)nc2ccc(Br)cn2n1 C1(NC(Cn2cc(-c3ccc(C)c(C(F)(F)F)c3)nn2)=O)CC12CCCCCC2 C(C(C(F)(F)F)N1CCN(C(C2CCCCS2)=O)CC1)NC(C=C(COC)C)=O c1(C(=O)NCC(C)(CO)NC(c2ccc(C#C)cn2)=O)cccc2c1CCC2 C1(CNC(C2C(C)C2C)=O)CCC2(CCN(C(c3cnc(S)[nH]3)=O)CC2)CO1 N1(C(Cc2c(C)ncs2)=O)CCCN(C(=O)CCOCC2CC2)C(C)C1 C1(C)(C(=O)OC)CCCC1O.C12(CN(CCC(C)O)C1)n1cc(nn1)C2 N1(C(c2c(C)cns2)=O)CCC(C)(CNC(c2ccc(O)c(N)c2)=O)CC1 c1(C(N(CC(C)(C)CNC(=O)CC2CC23CC3)C)=O)[nH]cnc1C#N N1(S(=O)(=O)c2ccccn2)CCc2cc(C(=O)NC(CO)CO)cnc2C1 c1(C(=O)NC(CN(C(=O)CCN2C(=O)CCC2=O)C)(C)C)cnn2c1N(C)CC2 C1(CNC(c2ccnc(OC)n2)=O)(CO)CC12CCN(C(c1cnn[nH]1)=O)CC2 N1(C(C2(OC)CCC2)=O)CCCCC(C2CN(C(C34CC3CCC4(F)F)=O)C2)C1 CCC(C)(C(=O)NCC(C)(O)CNC(=O)C(c1ccc(F)cc1)F)C(F)F CC(C)(C)C1=NOC(C(=O)NCCCNC(=O)CCCN2CCCC2)C1 C1(C(=O)NCC2CC(C)N(C)C2)(CC)CCN(C(=O)C(C)CCN(C)C)CC1 C(=O)(C1=C(Cl)CCOC1)NCC1(C)CC(NC(C(C)c2ccsc2)=O)C1 c1(C(N2CC(C)C(NC(C3CCC(=O)N3)=O)CC2)=O)cccc(N=[N+]=[N-])c1 CCCCC(C(=O)NCC(C)(C)OCCNC(c1csc(C(F)F)c1)=O)OC CC1CCC(F)(C(N2CCN(C(=O)C(=O)c3cccs3)C(C)C2)=O)CC1 C#CCC(C)(CNC(=O)NC1(C(=O)OC)CCOC1(C)C)CO N1(CCOCCc2n(C)cnn2)CCCCC1c1n[nH]c(C(F)(F)F)n1.C=O c1(CC(=O)NCCN(C(=O)C(C)c2ccsc2)CCC)ccn(C)c1 c1(NC(C2CCC(NC(c3c(Cl)cc(Br)cc3Cl)=O)C2)=O)cnc2n[nH]c(Br)c2c1 N1(C(C(C(CC)C)=O)=O)CCC(C2CC2)C1C(=O)Nc1cncc(C)c1 C1(C(c2ccco2)C)CCCN1C(=O)NCc1c[nH]nc1C1CCC1 c1(C(N2C(C)CC2C(N2CC(F)(F)C2C2CC2)=O)=O)cn2ccccc2n1 C1(NC(c2coc(CO)c2)=O)CN(C(c2ccoc2C2CC2)=O)CC12CCC2 c1(N2CCC(OCCNC(c3ccc(CO)nc3)=O)C2)nc2cccc(F)c2o1 c1(NC(C(CC)NC(=O)C=Cc2ccc(C)o2)=O)ccc(C)c(F)c1F N#Cc1ccc(Br)cc1CN=c1[nH]c(C(=O)Nc2ccc(C3CC3)nc2)cs1 c1(C(N(C)CC2N(C(C3CC(=C)C3)=O)CCCC2)=O)cnc2nc(C)oc2c1 c1(NC(C2(NC(CNC(CC(C)C)=O)=O)CCC2)=O)cnn2ccccc12 c1(C(=O)NCCCCNC(=O)CN2CCSCC2)cc(Cl)c(Cl)cc1Cl Cc1cn(CC(N2CC3(NC(c4csc(Cl)c4)=O)CCC2C3)=O)c(=O)n1C C=C1CCN(C(C2(C)CN(C(c3scc(C)c3Cl)=O)C2)=O)CC1 C(=O)(C1=NN(CC(=O)O)C(=O)CC1)N(C(C)CNc1ccc(C(=O)O)cn1)C C12(NC(c3cc(C)c(C)s3)=O)CCC1CN(C(=O)CNC(=O)CN(C)C)C2 CC1OOC(=O)NC1C(=O)NCC(C)(C1CC1)NC(=O)Cc1cc(C2CC2)no1 C1(C)(COC)C=CCN1C(=O)CC(CNC(c1ccnc(CO)c1)=O)C1CCC1 C1(NC(c2c(Cl)cn(CCC)n2)=O)(CNC(c2ccoc2Cl)=O)CCCCC1C CCC(C)CCCC(=O)NCC1CC(NC(=O)CCOc2ccc(Cl)cc2Cl)C1 C1(CCCC)CN(C(c2sc(OC)nc2Cl)=O)CCN1C(=O)C(C)c1cccs1 CC1(C)CN(C(C2(O)COC2)=O)CC2(CN(C(=O)C(C3CC3)C3CC3)C2)O1 N1(C(c2ccc(CCCCCC)s2)=O)CC2CCCN(C(=O)C(N)=O)C2C1 c1(CC)cncc(CNC(=O)CSCCNC(C23CCCC2C3)=O)c1 c1(OC)ncc(C(N2CCC(CF)(NC(=O)CCCC3CC3)C2)=O)nc1C C1(C(=O)OC)CCn2ccnc2C1.c1(OCCC)cccnc1NC(C)C c1(CC)ccc(Cl)cc1S(=O)(=O)Nc1n[nH]c2c1CN(C(=O)C(C)OC)C2 c1(NC(CC)CO)ncc2cccc(Br)c2n1.c12nc(cs1)CC(=O)N2 C1(CC(=O)NCC(C)(CO)NC(CCCC(C)C)=O)CCc2sccc2C1=O c1(C(=O)NC2CN(C(c3cnc[nH]3)=O)CC2CC2CC2)cc2c(=O)cc[nH]c2s1 c1(CNC(CCC=C)c2nnnn2C2COC2)cnn(C2CCN(C)CC2)c1C C1(CC(N2CCC(N(C(=O)CN(C(=O)C(C)C)C)CCC)C2)=O)CC(=O)NC1=O c1(N2CCN(C(CC3C(C)=NN(C)C3=O)=O)C(C)C2)nc2cccc(C)c2o1 C=CC(CC)CC(=O)N1CCC(N2CCCC2)C1.C1C(=O)NO1 CCCC(C)(C)C(=O)N1CC2C(C(=O)NCc3ccccc3OC)C2C1 c1(C(=O)NC2CN(C(=O)CN3CCNC3=O)C3CC23)ccc(C(F)F)c(Cl)c1 CCC(C)CC(=O)C(=O)N1CCCC1C(C)(C)C(=O)Nc1cncnc1O CCCCN=C(NCC1CC1CC)NC1CC(C#N)C1 c1(C(N2CC(C)OCC2C)=O)ccc2nonc2c1.c12ccc(cc1)C(CN)N2 C1(ONC(C2CC23CCC3)=O)(C(N2CCC(F)C2)=O)CCCCC1 C1(n2ncc(C)c2)CCCN(C(c2ncoc2C)C(=O)NCC2CC2)C1 CC1(C)C(NC(c2n[nH]c(=N)s2)=O)CCN1C(=O)C=Cc1cccc(F)c1 CC(CN1CCN(C)CC1)N=c1ccnc(NC(c2ccc([N+](=O)[O-])cc2)C)[nH]1 C=CCCCC(C(=O)NCCc1cn(C)nn1)NC(C1C=CC1C(=O)OC)=O CN1C2CCC1CC(C(=O)NC1CC(CNC(=O)CN3CC(=O)NC3=O)C1)C2 c1(N(CCO)OC)ccc(S(N)(=O)=O)cc1.C(=O)(NNC=O)C1C(C)C1 N12CCCC(C1)N(C)CC1C(C1)C2=O.c1(CCC)noc(CCCC(=O)OC)n1 C(=O)(CC(C)(C)CC)N(C1CCN(C(=O)CCC2CCC(C)O2)CC1)CC#C C(=O)(C(C)(C)C(C)(C)C)N(CCNC(C(C1CC(F)(F)C1)OCC)=O)C1CC1 c1(CCC(=O)N(C(CNC(c2cccnc2O)=O)C2CC2)C)ccc(O)nc1 c1(C(=O)NC2CC(C)(NC(CC3C(C)CCC3)=O)C2)cnc2n1CCCC2 c1(OC(CC)Cc2ccc(N(C)C)cc2)ccc(Br)c(C(F)(F)F)c1 c1(OC)noc(C(N2CC(CNC(=O)Cc3n[nH]c(C)n3)C(O)C2)=O)c1Br c1(OCCC(=O)NC(CC)CN(C(=O)CSCCC#N)C)cccc(C)c1 c1(N(C)Cc2nnc(O)o2)nc(=NC2CC3CC3C2)[nH]c2c1COCC2 CC(C)CCC(=O)NC(C)(C)COCCCNC(c1cnn(C2CC2)c1Cl)=O n1(CCCC)ncc(C(=O)NC(CO)C(C)NC(C2(C)CCCOC2)=O)c1C c1(N2CCC(COC)C2)nc(N2CCC(F)C2)nc2c(F)cccc12 c1(C(N2CC(CNC(CCCC#C)=O)C(C)C2)=O)cc(C#N)ccc1C C12(CNC(C(c3ccccc3)SC)=O)CN(C(=O)CCC3CC3)CC1CCO2 C=C(Cl)CCC(=O)N1CCC(CF)(NC(=O)CCNC(C2CCCCC2)=O)C1 C1(C(=O)Nc2ccc(OC)c(C)c2)CN(C(C2(CO)COC2)=O)CC1C1CC1 c1(C(N2CCCCC2=O)=O)cccc2c1OCC2 C(=O)(CC1=CCCCC1)N(c1nnc(C2CCS(=O)(=O)C2)n1CCCC1CC1)CC C12(CC(=O)NC(CNC(CC=CCC)=O)(C)CC)CC3CC(CC(C3)C1)C2 c1(CC(=O)NCCC2CCCN2C(=O)CCc2ccc[nH]2)cnc(C2CCC2)s1 N1(CC)CCC(c2nnnn2CC)(N)C(NC(C2CCOC2)C)C1.OC c1(N(C2CCNCC2(C)C)C(c2nccc(C)c2)=O)ncnc2cccnc12 C(=O)(CC(O)Cc1ccccc1)N1CC(NC(CN(C)C)=O)C1 C(=O)(C#CC1CCOC1)NC1CC(C)(NC(c2cc(C(F)(F)F)c[nH]2)=O)C1 CC1(CNC(C2COCC2C(N)=O)=O)CCN(C(=O)CNC2CCCC2)CC1 C1(C)(C2CN(C(CSC(C)(C)C)=O)C2)C(=O)N1.C(C1CC1)(C1CC1)C(N)=O c1(C(N2CC3CC(CNC(C(C(=O)OC)C)=O)C3C2)=O)cc2ccccc2n1C C(C(=O)N1CCC(C(=O)N(c2cnn(C)c2)CC)CC1)(C(C)C)OCC Cc1ccc(=O)n(CC(N2CC(N(C(=O)Cn3nnnc3C)C)C(O)C2)=O)n1 C1(NC(c2ccnn2C(F)F)=O)CCN(C(C2CCC=CCC2)=O)CC1 c1(OC)c(F)cc(C(=O)N(C2CN(C(C3(C)CCCC3)=O)CC2F)C)cc1F C#CCCCC(=O)N(C1(C(=O)NC2CCOC(C3CC3)C2)CC1)C c1(OCC=C)c(C(=O)NCC2CCN2C(=O)C(C(C)O)NC(C)=O)cccc1C N1(Cc2c(C)nc(C)o2)CCC(F)C(Sc2ccccc2)C1 CC(C)CC(C)(O)C(=O)NC1CCN(C(c2c(O)cc(Br)cc2F)=O)CC1 c1(C(=O)NC2C(Cn3cc(C(CC)(O)CC)nn3)C2)cc(C)nc2c1cnn2C c1(C(N2CCCC(NC(c3c(C)cncc3)=O)CC2)=O)nc[nH]c2ncnc1-2 Cc1nc(CO)oc1C(=O)NCC1CCCC(NC(=O)COc2ccn(C)n2)C1 C1(C(=O)NCC2(CNC(C(C=C=C)C)=O)CCOCC2)CC2(CCOCC2)C1 c1(C(=O)NCC2N(C(C3OCC3(C)C)=O)CCN(C)C2)ccnc2ccnn12 C1(O)(C(C(=O)N(CCN(C(C)C)C(C2(C#N)CC2C(F)(F)F)=O)C)F)CCCC1 c1(OCC(=O)NCCCC(CO)NC(C2CCCSC2)=O)ccc(F)nc1 C1(CC(=O)N(CCCN(C(=O)C=C2CCC2)C)C)CC(=O)c2ccccc2C1 C1(C(=O)NC2(CNC(COC(CC)(C)C)=O)CCCCC2)CCN2CCCC2C1 CCC(C)C(C(=O)NC(CC(=O)N(C)Cc1cccc(OC)c1)C(F)F)OC Cc1cc(=O)ccn1CC(N1CCC(C)C1CNC(c1cccc(CO)n1)=O)=O C1(CC(N2CC(NC(C3CCN(C(=O)NC)CC3)=O)C2)=O)CCN(OC)CC1 C1(OC)CC(NC(C2(C)COC2)=O)CN(C(C2(n3cncn3)CC2)=O)C1 c1(CCC(=O)N(C)CCOCCNC(C2CC2C(F)(F)F)=O)ccc(F)c(F)c1 N1(C(C2=C(C)CCOC2)=O)CCC2(CC1)CC(NC(C1CC1C(C)O)=O)C2 C1(CNC(C2N(C(C)=O)CCC2)=O)CC2CCC(C1)N2c1cc(F)ncn1 CC(CC1CCCO1)C(=O)NCC(O)CNC(=O)CCNC(=O)C=CCl C(=O)(C(C)(C)C(C)(C)O)NCCC(C)CCNC(=O)C=C1CCCCC1 N1(C(CNC(CC)=O)=O)CCC2(CC(NC(=O)C(C)(C)N(C)C)CO2)C1 N1(C(CN(C)S(N)(=O)=O)=O)CCC(O)(CNC(=O)C(C)CC#N)C1 c1(N2CCCC(C=O)C2)nc(N2CCC3CC3C2)nc2c1COC2.C(C)(C)NC C=CCC(C)(C)CC(=O)NCC1CNC(=O)CO1.c1(COC)nc[nH]n1 C1(n2cc(CCC(=O)NC3CC3)nn2)CCCN(C(C2(C(=O)O)CCC2)=O)C1 N1(C(c2c(C)nc(CC)s2)=O)CCCC12CCN(C(=O)C(C)SC(C)C)C2 C1(CN(C(C(CC)(C)OC)=O)C)CC(F)(F)CN1C(=O)C(COC)OC c1(CC)ccc(CCC(=O)NCC(CNC(C2C3CCN2CC3)=O)OC)cc1 N1(C(c2ccc(C(F)F)c(F)c2)=O)CC2CCC1C(Nc1ncnc(Cl)c1Br)C2 c1(C(=O)NC2C(CNC(CN(C)C3CC3)=O)CC2)nc2ccccc2[nH]1 N1(C(C(C)O)=O)CCN(CC2CCN(C(=O)CC3CCOC3)CC2)CC1 C(C1c2ccccc2CCN1C(=O)Cc1cnn(CC)c1)NC(C(C#C)(C)C)=O N1(C(=O)NCC(c2ccc(Cl)cc2)C2CCC2)CCOC2CCCC12 c1(C(N(C2CCN(C(=O)C(COC)OC)C2)CCC)=O)oc(Br)nc1C c1(C(=O)OC(C)(C)C)ccc2ccn(CC(N3CC(CS(N)(=O)=O)C3)=O)c2c1 c1(C(=O)NCCN2CCN(C(C(C)(C3CC3)OC)=O)CC2)ccc2ocnc2c1 C12(C(=O)NCC3N(C(C4C(=O)NCC4)=O)CCSC3)CCC(CC1)CO2 CN1C(=O)OCC1C(=O)NCC(CC(=O)N1CC[Si](C)(C)C1)N(C)C c1(OCC)c(CC(=O)NCCN(C(=O)CC2(O)CCCC2)CC)cccc1Cl n1(C(C)C)cc2c(n1)C(C(=O)N(C)CC1CCCN(C(=O)CC3CC3)C1)CCC2 N1(C(C2(C(N)=O)CCC2)=O)CCN(C(c2ccc(OC(F)(F)Cl)cc2)=O)CC1 c1(C(N2CC(n3cc(COC)nn3)C2)=O)c(F)cc(Br)c2c1NCCC2 C(=O)(CC1=CCN(C)CC1)N1CC(CN(C)C(C2CCC(N(C)C3CC3)CC2)=O)C1 C1(CC(=O)N(CCOCC#C)C)C2CN(C(=O)C(C)CSC)CC12 C1(C(=O)NC2CCCC(NC(c3ccncc3O)=O)C2)CC2CCC(C1)S2 c1(C(=O)O)cccnc1N1CCCC(CNC(C2(C(F)F)CCCO2)=O)C1 c1(C2N(S(=O)(=O)C3CCC3F)CCC2)cccc2ccccc12.C1CSCCS1 C1(CNC(C23CC(COC)(OC2)C3)=O)CC(C)(C)CN1C(=O)CC1CC(C)=NO1 C1(CCC(N2C(CC(C)O)CCC2)=O)CCCN(C(c2scnc2Cl)=O)C1 C(c1ccc(Cl)cc1F)=CC(=O)NC1CC1NC(c1cnc2n1CCCC2)=O c1(C(C(=O)NCC(C)(C(C)C)NC(CC=CC)=O)C)ccc(F)cc1F N1(C(CCC)=O)CC(NC(=O)C(C)(C)Cc2ccccc2)CC2(CC2)C1 C12(C(=O)NCC(CNC(CCc3n(C)ncc3)=O)O)CC(C)(C1)OC2(C)C c1(COC)c(C(N2CC(OCCNC(C3CC=CC3)=O)C2)=O)sc2ccccc12 c12ccc3c(c1)C(NC2=O)CC3.c1(OCC)cccc(OC(C)(C)C)c1 Cc1c(Br)ncc(F)c1CNC(=O)Nc1cccc(C(C)O)c1 c1(C(=O)NCC(CNC(C2ON=C(C)C2C)=O)O)c([N+](=O)[O-])cnn1C Cc1cccc2c(C(N3CCN(C(c4ccoc4C(C)C)=O)CC3C)=O)c[nH]c12 N1(C(C(C)OCCC=C)=O)CC(O)(C(C)NC(c2cc(Cl)n[nH]2)=O)C1 c1(C(=O)NCCN(C(=O)CC2CCC(=O)N2C)CC)ccn2c1CS(=O)(=O)CC2 N1(C(CC(C)OC)=O)CCOCC(F)(CNC(=O)CCc2cnc(O)[nH]2)C1 C1(C(=O)NC(C)Cn2cccn2)N(C(c2cc(O)ccc2F)=O)CCC1(C)C c1(N2CCC(C(C)NC(=O)NC3CCC(=O)NC3C)C2)nc(C(C)(C)C)nc(=N)[nH]1 Cc1c(NC(=O)CCCNC(=O)C=CC2CCCC2)cccc1C#N Cc1ccc(C)c(OCC(N2CC3(CCC3NC(c3[nH]c(O)nc3C)=O)C2)=O)c1 N1(C(c2cc(C(C)(C)C)no2)=O)CC(NC(c2nccnc2N)=O)C2(CC2)C1 C1(CNC(C(OC)OC)=O)CC(NC(c2cc(C)ccc2C2CC2)=O)C12CCC2 N1(C(Cc2c(C)scc2)=O)CCOC(CNC(=O)Cc2ccc(O)cc2)C1 c1(C(N2C(c3nnc(C)o3)CCCCC2)=O)cc(F)c(F)c(Cl)c1F c1(C(=O)NC2CCCC(NC(C3CCC(F)(F)C3)=O)C2)cnc2cccnc2c1 c1(C(=O)NCC2(CNC(=O)CC(F)(F)F)CC2)cc2cc(Br)ccc2[nH]1 C12(NC(C(CSC)OC)=O)COC(C1)C(NC(C1(CF)CCC1)=O)C2 C1(NC(C(c2c(CC)cccc2)(F)F)=O)CCCCCC1NC(c1cnc[nH]1)=O N1(C(C(C)c2ccsc2)=O)Cc2ccccc2C1CNC(=O)C(F)OC(F)(F)F CCC(C(=O)N1CCC(CNC(c2cccnc2OC(C)(C)C)=O)CC1)C(C)C C1(OC)CN(C(=O)C(n2ccc(C)n2)C)CC1NC(=O)C=Cc1nccs1 c1(C(=O)NC(CCOC)C(=O)N(C)C(c2nc(C)no2)C)ccc(C)c(O)n1 C1(C(=O)NCCOCCCNC(Cc2c(C)n[nH]c2C)=O)CC2(C1)CC(C)(C)C2 c1(CNc2nc(C)c(C(N)=O)s2)cc(O)ccc1N.N(C)(C)C c1(C(=O)NCC(CNC(C2C(C(N)=O)C2)=O)F)n[nH]c2ccc(F)cc12 Cc1nc(NC2CCCN(C(C3CC(C)CO3)=O)CC2)c(C)c(O)n1 N1(C(c2ccc(OC)cc2)=O)CC(=O)NC2CN(C(c3ns[nH]c3=O)=O)CCC12 c1(C(=O)NC2C3CN(C(c4cc(C)nn4C)=O)CC32)c(C)ccc2c[nH]nc12 Cc1ccc(F)c(C(C)NC(N2CC(C(F)(F)F)OC(c3ccc(F)cc3)C2)=O)c1 N#Cc1cc(F)ccc1C(N1CCC=C(C(=O)Nc2cccc3nsnc23)C1)=O C=CC1CCCN(C(=O)Cc2coc(-c3ccc(Br)cc3)n2)C1 Cc1noc2ncc(C(=O)NCC34CC(NC(C5CC6CC6C5)=O)(C3)C4)cc12 C1(C(=O)NCCn2cc(C)nc2)(NC(C23CC(F)(C2)C3)=O)CCCCC1 N1(C(C(C(F)(F)F)OC(C)=O)=O)CCC2(CC1)CN(C(=O)C1=NOCC1)C2C(C)C C(C(C)(C)CN=c1[nH]c(=NCC(C(C)C)N(C)C)c2cccc(F)c2[nH]1)OC C1(N(C(C(C)N(C(C)=O)C)=O)C)CCC(CNC(C2(C)CC=CCC2)=O)CC1 OC1CC2(CCN(c3nccc(=NCCOCC(F)F)[nH]3)CC2)OCC1O c1(C(=O)OCC)ccc(C(N2CCC(CCNC(C3CC3(C)C)=O)CC2)=O)cc1 c1(CCC)nnsc1C(=O)NCCC(C)NC(=O)Cn1nnc(C)n1 CN1CCN(C(=O)OCC(c2ccccc2)c2ccoc2)C(c2cccc(F)c2)C1 C1(SCCNC(N)=O)CCC(C(=O)Nc2cn(C3CCCC=C3Br)nn2)CC1 C12(C(=O)NCC(C)NC(c3ccnc(C(F)(F)F)n3)=O)COCC(C1)C2 c1(C(C)NC2CCN(C(c3ncc(F)cn3)=O)C2)c[nH]c2c(Cl)cccc12 C(=O)(C1=CCCCCC1)N1CCC(O)(CCNC(C2CC3CC2C3)=O)CC1 c1(C(=O)NCC(C(C)O)C)nnc2ccc(Br)cn12 c1(NC(C(c2ccncc2)N(CCC)C)=O)ccc(C(=O)OC)cc1C.CCC#N CCCC(C)CC(C)(c1nnnn1CC(F)F)Nc1cncc(-c2ccoc2)c1 Cc1cc(CNC(C2CN(C(=O)CCC3CC(F)(F)C3)C2)=O)cc(C)c1 CC1CN(C(C2CCCCN2C(c2ccc(Sc3cnc[nH]3)cc2)=O)=O)CCO1 c1(C(N2CCC(N(C(=O)CSC(F)F)C)C2)=O)cc(F)c(F)c(O)c1F c1(C(=O)NCCCCC(C)NC(C(C#C)(C)C)=O)cc(C)cnc1Cl C1(OC(CC)=O)CCc2c(NC(c3ccc(C(F)(F)F)nc3)C)cccc2C1 C12(C(N3CCCC(CCC=C)C3)=O)CC(CCO1)N(C(=O)CC1CC3CC3C1)C2 c1(C(N2CC(OCCNC(CN(C)C3CC3)=O)C2)=O)ccc(F)c(Cl)c1N C(C1CCc2ncnn21)NC(Cc1cc(C)ns1)=O.C12CC(CC1)NC2=O N1(C(c2cc(CC)[nH]n2)=O)CC(NC(c2cnoc2C(C)C)=O)C(C(F)(F)F)C1 CC(C)C(F)(CNC(=O)CN(CCCF)CC)C(=O)NC(c1cccnc1)C c1(C(N2CCC(C)(CNC(C34CC(C)(C3)C4)=O)C2)=O)ncc2c(F)cccn12 CC(C)CC(C)(CNC(=O)CCC(=O)NC1CC1)NC(=O)COC.C1(S)CCCCO1 C1(C(=O)NC2C3CN(C(c4c(CC)cno4)=O)CC2C3)CCc2ccccc2C1 O=C(C(F)(F)C(O)C1CC1)NCC1C2CN(c3ccc(Cl)nn3)CC12 Cc1cc(F)c(C#N)cc1OC(C1CCCN(c2ncccn2)CC1)=O CCC(C(=O)N(CC(C)(CC)OC)C)N(C(=O)C(C1CCCCC1)F)C C1(C(N2CCN(C(C(n3cc(Cl)cn3)C)=O)C(C)C2)=O)(CF)CCC(F)(F)CC1 Cc1ccc(CC(N2CCCC2c2cn(CC3CCC(=O)NC3)nn2)=O)c(C)c1 C1(CN(c2cc(N3CCCCC3)ncn2)C(C2CNCCC2O)=O)NC(=O)NC1=O C1(C(=O)NCC2CC(F)(CNC(=O)C(C)CO)C2)(CSC)CC(F)(F)C1 c1(C(=O)NC2(CCOC)CCN(C(C=CC)=O)C2)cc2n(c1)CCSC2 Cc1c(C(N2CCCCC2CN(C)C(C2CC(F)C2)=O)=O)cnn1CCN(C)C c1(C(=O)NC(CC)CNC(=O)Cc2ccc(Cl)nc2C)ccc(N)c(F)c1F CC(C)(CC(=O)NCCOC1CN(c2ccn3c(Br)cnc3n2)C1)C(F)(F)F c1(C(=O)NCC(CN(C(c2cn(CC(CC)O)nn2)=O)C)O)cc(=O)n(C)o1 CC1CCC(NC(=O)C=CC2CCC2)CN1C(=O)C(N1CCOCC1=O)C C(=O)(CCCC(C(C)C)NC(=O)CC(C)C1CC1)OC C=CCCC(O)CNC(=O)CC(C)(C)N(C(=O)CN1C(=O)CNC1=O)C c1(C(=O)NC2CC(CO)N(C(C3CC34CCOCC4)=O)C2)ncc(Cl)cc1F CC1NC(=O)CCC1NC(=O)C(Cc1ccoc1)NC(=O)CNC(C1CC1C)=O CC(C)CC(F)(F)C(=O)NC1(C)CCCN(C(C2CN(C(C)C)CCO2)=O)C1 CCCCS(=O)(=O)CC(=O)NC(C1CCCC1)CNC(=O)CC(C)N(C)C c1(CC)ccc(C(=O)N(C)CC2COCCN2C(c2occ(C)c2C)=O)nc1 N1(CC)CCC(NC(=O)C(O)Cc2ccccc2)c2ccccc21 CC(C)(C)CC(=O)NC1COCC1CNC(=O)Cn1cc(CO)nn1 c1(N2CC3N(CC)CC(CC3)C2)nc(=NCC(CSC)OC)[nH]c2c1CC(C)CC2 c1(CN2CCOCC(C(=O)NCCOC(C)(C)C)C2)c[nH]c2ncc(Cl)cc12 N1(C(c2nocc2C)C(=O)Nc2ccc(OC)cc2)CCSc2ccc(C)cc21 C1(NC(CC)=O)CCN(C(C2(CNC(=O)CCOC3CCCC3)CCCO2)=O)C1 C1(NC(CCCCC)=O)CC12CCN(C(C1CCC(=O)N1CCC)=O)CC2 C1(C(=O)NCC2(C)OCCN(C(CC3CC(OC)C3)=O)C2)CCn2c(C)nnc2C1 C(CN=c1[nH]c2c(c(=NCCC=CBr)[nH]1)CC(C)CC2)c1cc(C)oc1C c1(C(N2CC3C(CNC(C=C4CCN(C)CC4)=O)(C3)C2)=O)cc2ccccn2c1 N1(C(CCCOC)=O)CCC(C)C(NC(=O)COCC2CC2)C1C C(=O)(C1=NNC(=O)C1)N1CC(CNC(c2c(C)nc(CC3CCCC3)o2)=O)C(C)C1 c1(C(C)C)noc(CCC(=O)NC(CNC(C2COCCO2)=O)CO)n1 CC(C)(O)C(F)C(=O)NC1CCCC1NC(=O)Cn1cc(F)ccc1=O Nc1cc(C(=O)NC2CCC2CNC(=O)C(c2ccccc2)F)ncn1 CC1OC(C)C(C(N2CCOCC(NC(C3(S(C)(=O)=O)CCC3)=O)C2)=O)C1C N1(C(CCC(N)=O)=O)CCC2(CCOC2)C(CNC(=O)CC2CCNC2=O)C1 c1(NC(CC)C(C)(C)C)nccc(=NCC2CCC(NC(N3CCCC3)=O)C2)[nH]1 c1(OC)nc(C)ccc1C(=O)NCC1CCCN1C(=O)CCc1ccc(C)nc1 c1(-n2cc(CN(C(c3c(OCCC)cccc3)=O)O)nn2)ccc2c(c1)OCO2 Cc1cncc(C(=O)NC(C)C=CC(=O)NCCCCCCC2CC2)n1 c1(SCC(=O)N(CCCN(C(=O)COC2CCOC2)C)CCO)ccc(N)cc1 c1(C(=O)NC2CC3CCC2O3)cc(F)ccc1-c1cn(Cc2cccc(Cl)c2)nn1 N1(C(C(C=CC)O)=O)CCCN(C(C2CC(C(C)(C)C)=NO2)=O)CCC1 C12(CC(F)(F)C1)C(=O)N2.c1(C(C)NC(=O)NC)cnn(C)c1 C=Cc1cnn(C)c1C(N1CCC(NC(c2ccccc2Cl)=O)C(C(C)C)C1)=O C1(c2cccnc2)(C(=O)NCC2C(NC(=O)CCOC3CCOC3)C2)CCCC1 C(=O)(C(C)CCC(C)(C)C)NCC(C(C)C)NC(=O)C(C)(C)CNC(N)=O N1(C(C(C)NC(COC)=O)=O)CC(O)CC1Cn1cc(-c2ccc(F)nc2)nn1 C(c1cccc(Cc2ccccc2)c1F)=Cc1nccn1C.OCCC=C N1(C(C(CC(C)=O)(C)C)=O)CC(C2CCCN(C(=O)Cc3cnsc3)C2)C1 N1(CCNC(Cn2c(C)ccn2)=O)CCN(C(=O)C(C)CN(C)C)CC1 N1(C(C(=O)N(C)CC2(O)CCCNC2)=O)CCC(C2(N)CC2)CC1 N1(C(CCC2CC(OC)C2)=O)CC2CCC1CN2C(C1CC2CC2C1)=O C(c1ccc(F)cc1)=CC(N1CC=CC(NC(Cc2c(C)nc[nH]2)=O)C1)=O Cc1c(Br)ccc(-n2cc(CCCSC3CC3)nn2)c1C.c1(N)nnnn1CCCF CC1=C(C)CC(C(=O)NCC23CCC(CC2)N3C(=O)CC2CCOC2=O)CC1 C1(CC(=O)NCCCN(C(=O)Cc2csc(C)c2)CCC)CCCC(C)(C)C1 Cc1coc(C(C)C)c1C(=O)N(C1CCCC1)CCCNC(c1coc(Br)n1)=O Cc1[nH]nc(Cl)c1C(=O)NCC1(F)CC(NC(=O)CC2(C)CCCO2)C1 C1(C(=O)OCC(c2ccccc2N2CCOCC2)=O)CCC(C2CCCO2)O1 C1(O)(CC(=O)NC2CN(C(=O)C(O)CF)C2)CCOCC1 C(CC(C(C)(C)C)NC(=O)Cn1ncc(O)nc1=O)N(C)C(C1CC1(C)C)=O CC(CC(=O)NC(C1CCCC1)CNC(=O)CNS(C)(=O)=O)C(C)(C)C c1(OC)ccc2c(c1)CC(C(=O)NC1CC3C1CCN3C(=O)Cc1ccsn1)O2 c1(C(N2CCCC(OC)C2C)=O)c(Br)nc2n1CCC2 C1(C(=O)NC(c2cnn(C)c2)C)CCCN(C(=O)CC2COCC(C)O2)C1 C(C(CC(C)C)C(=O)N1CCC(C)(NC(=O)C(O)CCC(C)C)CC1)OC C1(CNC(C2CC(C(=O)OCC)C2)=O)CC(O)CN1C(C1CC1Br)=O O(N(C(=O)C1COCC1NC(C1C=CC1C(=O)OC)=O)C(C)C)CC C(N=c1nc(N2CCC(c3cc[nH]n3)C2)c2c([nH]1)COC2)c1snc(C)n1 C1(C(C(=O)N(CCO)Cc2ccco2)F)CCCCC1 c1(C(=O)NC2C(N(C)C(C3(c4cccc(Cl)c4)CCC3)=O)CCC2)ccc(=N)[nH]c1 C1(NC(c2c(C#C)c[nH]n2)=O)COC2(C1)CN(C(C1(CC=C)CCOCC1)=O)C2 CC(C)C(C(=O)NCc1ncsn1)C(C)NC(C1CC2CC(=O)C1O2)=O N1(C(C(C)c2cncs2)=O)CCC(O)(CNC(c2coc(C(N)=O)c2)=O)C1 CC1(C)COC1C(N1CC(O)(CCNC(c2ccc(-c3cccs3)s2)=O)C1)=O c1(OC)c(CN2C(C(=O)NCc3cc[nH]n3)CC(F)(F)C2)cccc1F C(=O)(C(F)CCC(C)C)Nc1cc(C(=O)NCCN(C(=O)C2CC2)CC)c(Cl)cc1 c1(CCC)cccc(C(=O)NCCC2CN(C(c3c(C)ncn3O)=O)CCO2)n1 C(=O)(C(C)(C)CCC#N)NC1(C(N2CCC(CC(C)C)C2)=O)CC(O)C1 c1(CC(=O)NCCc2n(CCC)cnn2)ccc(OC2CCCC2)cc1Br c1(OC)cc(NC(C2COCCN2C(c2cc(C)ccc2F)=O)=O)nc(Cl)c1 C1(C(=O)NC2(CC=C)CN(C(=O)CC3CSCCO3)C2)CCCNC1=O N1(c2ccnc(NCCCc3nc(=N)s[nH]3)n2)CCC(C2CC2(F)F)C1 C(CCCS(=O)(=O)CCCCO)Nc1c(C)nn(-c2ccccc2)c1 c1(C(=O)Nc2ccc3nc(C(F)F)oc3c2)cc(O)nc2ncccc12 N(C1CCc2cc(F)cc(Br)c21)C(=O)C1=CC2CCCCC12 c1(C(N(CC(=O)N(C2(C(=O)OC)CC2)C2CC2)CCC)=O)nccc2[nH]ccc12 n1(CC(N2CCCN(C(C(CO)OC)=O)CC2)=O)ccc2ccccc12 c1(C(=O)NC(CC=C)CO)cc(C)ccc1CCCNC1COC1 C(=O)(CCC(=O)N(CC)CC1CN(C(=O)CCC2CC2(Cl)Cl)CC1C)N(CC)CC C(c1ccc(O)cc1)=C(C(=O)NCCOCCOCC)C.C1CCCO1 C1(C(=O)NCCNC(=O)C(O)CN2CCCC2)OCCOC12CCC2 C1(C(N)=O)CCC(NC(=O)Cn2cc(CCc3ccccn3)nn2)C1 CCCCCC(=O)NC1CCOC(CNC(=O)CCc2cc(C)[nH]n2)C1 c1(C(=O)NC2C(C(=O)NCc3n(C)ccn3)C2)ccc(-n2cncn2)cn1 C1(C(=O)NCCC(C)OC)CCN(C(=O)CCc2cccnc2)C1C N1(C(=O)CO)CCN(C(=O)C(c2ccccc2)NCc2ccc(Cl)cc2)CC1 c1(C(=O)NCC2OCCCN(C(C(CC)N(C)C)=O)C2)c(C)ncn(C)c1=O c1(C(N2CCC(CNC(CS(CC)=O)=O)C2(C)C)=O)ccc2cccc(O)c2c1 C1(C(=O)OC)CN=C2N=C(CCC3CCC(c4n[nH]c(C5CC5)n4)O3)NN2C1 CC1CN(C(C2COCCO2)=O)CC1CNC(=O)CN(S(C)(=O)=O)C c1(SC(C(c2n(C)nnn2)NCC2CCCO2)(C)C)ccncc1F N1(C(c2n(C(C)C)nnc2)=O)CC2(NC(=O)C(C)CSC(F)(F)F)CCC1CC2 C1(N(C(Cc2c(C)cccc2)=O)C(C)(C)C)CCN(C(C)C(=O)NC(C)C)C(C)C1 C(C)(C(=O)NCCOC(C)(C)CNC(C1CN(C2CCOC2)C1)=O)=CC C1(C(=O)NCC(CC)NC(=O)C(C)(O)CC)CCCC1(F)F Cc1c(C(=O)N(C)CC2CCCN2C(C2(C)CC(O)CN2C)=O)cc(O)cc1N c1(SC)c(C(=O)NCC2CC(NC(c3cnc(C)[nH]3)=O)C2(C)C)cnn1C C1(COC)CN(C(=O)CCC2CC2CSC)CCN1C(=O)CN1CCN(C)CC1 CC(C)(C(=O)N1CCC(CC(=O)NCC2CCCNC2=O)C1)C(F)F CC(CC(=O)NCC#CC(=O)N(C)CC1(C#N)CCC1)N(C)C c1(C(N(C(C)C)CCNC(c2ccnc(C(F)(F)F)c2)=O)=O)csc2nccn12 C(=O)(CCCCCCBr)N1CCCC(NS(CCOC)(=O)=O)C1 c1(CCCNC(=O)NCC2(O)CCC(C)C2)nccc(Cl)c1O C(=O)(C(O)(C(F)(F)F)C1CC1)NCCCN(C(C1(OCC)CCC1)=O)CC N1(C(c2ccn(CC(C)C)n2)=O)CC(NC(C2CC3(CCC3)C2)=O)CC12CCC2 c1(C(=O)OCC)cnc(NCC2CCCN2C(=O)CC2CCC(C)(C)O2)c(C)c1 N1(C(c2cc(OC)no2)=O)Cc2ccccc2C(NC(c2c(C)n[nH]c2C)=O)C1 c1(N(C)C)noc(CCC(=O)NC2(CNC(=O)CNC(N)=O)CCOC2)n1 C1(n2c(C)nc(C(N3CCCC3CC3CC3)=O)n2)CCS(=O)(=O)CC1 C12(CCCCO1)CC(=O)N1CCN(CC1)CC2.C12(CC(=O)OC)CCCC1C2 c1(C2C(C(C)NC(c3nc4cccc(Br)c4[nH]3)=O)C2)ccc2c(c1)OCCO2 CCCC(C(=O)NCC(CCCC)NC(=O)CC(=O)N(C)C)c1ccccc1 C(=O)(CC(C)CC(C)(C)C)N1CCC(CC#C)(NC(=O)CC(=O)NCC)CC1 Cn1ncc(NC(c2cc(Cl)n(C)n2)c2nnnn2C)c1-c1cn[nH]c1 Cc1ccc(SCC(N2CCN(C(c3sc(C)cc3Cl)=O)C3CC23)=O)c(C)c1 N1(C(Cc2n(C)ccn2)=O)CCC2(NC(c3cn4ccsc4n3)=O)CC2C1 N1(C(C2C(CC)C2)=O)CC2(CCN(C(c3ccc(OC)cc3I)=O)CC2)C1 c1(CCC(=O)NC2CCN(C(C3=C(C)CCC3)=O)C2C)nc2ccccc2s1 c1(C(=O)NC2(CC)CCCN(C(C3(O)COC3)=O)C2)cnc2ccc(C)cn12 N1(C(CC2CC(OC)C2)=O)CCC2C(NC(=O)C=CCN(C)CCO)CC12 Cc1cc(C2CCC2)ncc1C(N1CC(F)CC1CNC(c1cscc1Cl)=O)=O C1(C(=O)NC2CN(C(C)=O)C2)CC2CC1CN(C(c1coc(C)n1)=O)C2 C1(NC(C(c2ccccc2)SC)=O)CCN(C(=O)CC(C)(C)C2CC2)CC12CCC2 CC1CN(C(C2(C)CC3CC3C2)=O)CC1NC(=O)C(c1ccccc1)F C1(S(C)(=O)=O)(C(N2CCC(C(CNC(C(CC(C)C)O)=O)O)CC2)=O)CCCC1 CCCC(CCC)CCCC(=O)N(CCC(C)NC(=O)CC1CC(OC)C1)C C1(C(N(C2(C(=O)NC3CCCCC3(F)F)CC2)C)=O)C2CCCCCC12 CCC(CC)C(C)C(=O)N1CC(O)(CN(C)C(c2cc(C)ccc2NCC)=O)C1 C1(CC(=O)NC(C)(CNC(=O)C=Cc2ccsc2)C2CC2)CCCC12CC2 C1(NC(c2c(CCC)nco2)=O)COC2CN(C(=O)C3=CCCCO3)CC12 C12(C(N3CCCN(C(c4cc(CC)[nH]n4)=O)CC3)=O)CCCN(CCC1)C2 CN1CCOCC1CC(N1CCC(C)(CNC(C2CC2CC(C)(C)C)=O)C1)=O CC1CC(NC(c2ccns2)=O)CN1C(=O)CC1CCC(CN(C)C)O1 CCC(C)C(O)CNC(c1coc(C(C)NC(c2ccc(C#N)o2)=O)n1)=O c1(CC)cccc(NC(=O)CC2C(NC(c3c[nH]c(=NC)o3)=O)CC2O)c1F c1(OC)cc(OC)c(C2CC2C(=O)NCC2(c3ccc(Br)s3)CC2)c(OC)c1 N1(C(c2csc(C)c2C)=O)CCC2C1CCN2Cc1nnc(-c2c(C)cccc2)o1 CN1C(=O)NCC1C(=O)NC1CC(C)(NC(=O)COc2ccc(F)cn2)C1 c1(C(=O)NC2C(CNC(c3ccoc3)=O)CCC2)nnn2c1C(=O)NCC2 C1(CC(=O)N(CCC)CCN(C)C)CCN(C(c2ccnn2CCF)=O)C1 c1(C(=O)NC(CCCN(C(=O)C(C)(C)c2cscc2Cl)CC)C)ccc(NC)cc1 C(=O)(C(F)CC(C)(C)C)NC1C2OCC(C(N3CCC=C(C)C3)=O)(C2)C1 c1(C(=O)NC(CNC(C(c2ccc(F)cc2)OC)=O)C)cc(C(N)=O)ccc1F c1(CC(=O)NCCC(C)NC(=O)C(C)(C)CC2CC2)c[nH]c2cccc(F)c12 N1(C(CCc2c(C)cccn2)=O)CCC(C)N(C(=O)Cn2cc(CO)nn2)CC1 c1(C(=O)NCCN(C(C(C=C=C)C)=O)C2CCCCC2)ccc2c(O)ncnc2c1 CC1CCN(C(C2(CO)CCC2)=O)CC1CC(N1CCCC1CF)=O.C1CC1 N1(C(C(C=CC)O)=O)CC(NC(=O)CCSCc2ccccc2)C(C)(C)C1 C1(C(C)NC(=O)COc2ccsc2)CN(C(=O)COCP(C)(C)=O)CCO1 N1(C(=O)COC2CCCOC2)CCC2CCN(C(c3cccc[n+]3[O-])=O)C2C1 c1(OC)cnnc(C(=O)NCC(c2ccc(C)cc2)NC(C2CCCSC2)=O)c1 C(C(O)C(C)(C)C)OC(c1ccc(CNC(=O)OC(C)(C)C)s1)=O c1(SC)cn(C)nc1C(=O)NC1CC(C)(NC(=O)CC(c2cccs2)N(C)C)C1 C1(O)(CC(=O)NCC(=O)OC)CN(C(=O)COC(C2CCOCC2)=O)C1 C1(C)(C(=O)NCCN(CC(C)O)C(c2ccc(C(C)(F)F)cc2)=O)COCCO1 C1(CNC(c2n(CC=C)ccc2)=O)CN(C(=O)C(CC)OCC)CC12CC2 C1(C)CC(=O)N1.C(=O)(CCCN1CCCCC1)NCCOCCOCCSC N1(C(c2nccc(OC)c2C)C(=O)NCCC)CCC2(CC1)C(=O)NCC2C#N Cc1ccc(C=CC(=O)NCCCCC(C)NC(=O)CCCc2nccs2)cc1 N1(C(=O)Nc2csc(C(F)(F)F)n2)CCc2cccc(CO)c2C1 c1(C(=O)NCC2(F)CN(C(CC)=O)C2)ccc(C)c(S(=O)(=O)CCO)c1 C1(C(N(CCC)CCC)=O)CNC(=O)CN1C(=O)CCN(C1CC1)CC Cc1cc(C(N2CCN(C(=O)C(C)OC(C)(C)C)CC2CCO)=O)ccc1Cl C(=O)(CC1OCCc2sccc21)N(C1CC(C(=O)OC)C1)C1CC1 Cn1nnc2ccc(C(N3CCC4CCC(C3)N4c3nc(C#N)c(Cl)s3)=O)nc12 C1(C(=O)NC2CC(NC(CCCN(C(C)=O)C)=O)C2)CN2CCC1CC2 C12(CNC(=O)Nc3cc(C(F)(F)F)ccn3)CCN(CC1)CC2 N1(C(CN(CC)CC)=O)CC2CC(NC(=O)C=CSc3ccccc3)C(C2)C1 c1(CN(C(=O)C(F)(F)F)CC(=O)NCC(O)CF)noc(C(F)F)n1 C1(NC(COCC(=O)NC)=O)CCCN(C(=O)CCc2ccc(Cl)cc2)CC1F c1(C(=O)OC)ccc(C(=O)NCC(CNC(=O)CN2CCSCC2)OC)s1 Cc1cccc(C(N(C)CC2CC2CNC(=O)CC2CCCN2C)=O)c1C C(CC(C(C)C)NC(=O)COC1CCCOC1)N(C(C(CC)SC)=O)CC c1(C(=O)NCC(CC)(C)NC(c2nn(C)cc2C)=O)ccc(N)cc1S(N)(=O)=O c1(NC(C(=O)NC(C2CCCO2)C)=O)ccccc1F.C(CSC)NC(=O)C1CC1 C12(NC(C=CC3N(C)CCC3)=O)CCC(CNC(=O)CC3CC=CC3)(CC1)OC2 c1(C(=O)NC2CCN(C(CS(=O)(=O)NC)=O)C23CC3)cnc2cnn(C)c2c1 N1(C(c2c(C)c[nH]c2)=O)CCN(CC2CCN(C(=O)C(O)C3CCC3)CC2)CC1 C(=O)(CCCCCCS(N)(=O)=O)NCCC(C)NC(=O)C(C)(O)C1CCC1 c1(C(=O)NC(C)C(=O)NCCC#CCO)ccc([N+](=O)[O-])[nH]1 c1(C(=O)NCCC2(O)CCN(C(C3(C#N)CC=CC3)=O)C2)nc2ccccc2[nH]1 C(=O)(C1Cc2ccc(Cl)cc21)N1CC(C)(C)C(F)(C(=O)O)C1.C(CN)SCBr C1(CC(=O)N(CCCCCNC(c2c(C(C)C)con2)=O)C)COCC1(C)C c1(C(N2CC(NC(c3cnc(OCF)cn3)=O)C(O)CC2)=O)cc(Cl)c(Cl)nc1Cl C1(CCC)C(=O)NCCN1C(=O)CCNC(=O)C1=CCCSC1 Cc1nc(-c2ccc(C(F)(F)F)cn2)sc1NC(N1CC(CO)C1)=O c1(C(=O)NC2CCN(C(CC(C)O)=O)CC2O)ccc2c(Cl)ccnc2c1 CS(=O)(=O)c1sccc1C(N1CC(CNC(=O)COCCF)C1)=O Cc1ccc(C(N2CC=CC2C(=O)Nc2csc(C3CC3)c2)=O)cc1C#N Cc1nc2nc[nH]n2c(=O)c1CCC(=O)NC(C)C(C)NC(C1CC1F)=O C(=O)(C(O)CC(C)(C)C)N1C(c2ccc(CC3N(C(C)=O)CCC3)s2)CCC1 C1(C(N2CCN(CC#C)CC2)=O)(NC(=O)CSC)CCC(C)(C)C1 C(=O)(CC(C)C(F)F)N(CCN(C(CC1CC(C(=O)OC)C1)=O)C)C(C)C c1(C(=O)NCc2nc(C)[nH]n2)ncccc1NCc1cccnc1C(F)(F)F N1(C(c2cnn(C)c2C(C)C)C(=O)NC)CC(CO)OC(C)C1.C(=O)(CCC(C)C)N Cc1ccc(S(=O)(=O)NC2(c3nnnn3CC3CC3)COC3(COC3)C2)c(C)c1 C(c1ccccc1)=CCCN1CCC(N(C(Cc2nc(C(C)OC)sc2)=O)C)C1 c1(C(=O)NCC2(O)CCN(C(COCCC=C)=O)C2)c(C)sc2ccc(F)cc12 N1(C(C2C(CCC)CCC2)=O)CCCC2CN(C(=O)CC34CC(C3)C4)CC12 C1(NC(C(Cc2ccco2)NC(C(C=C=C)C)=O)=O)CC2CCC(C1)N2C Cc1cccc(CC(=O)NCC(C)(O)CNC(=O)Cc2ccn(C(C)C)n2)c1Cl n1(C(=O)NCC2CCCCN2C(=O)CC2CCOC2)nnc2c1CCCC2 N1(C(C2N=C(C)SC2)=O)CCC(CNC(c2n[nH]cc2Cl)=O)C(F)(F)CC1 C=CC(C)(O)C(=O)NCCN(CCC)C(C1CC(C)CCO1)=O c1(C(N(C(C)CN(C)C(C2CC23CCC3)=O)C)=O)cn(C)nc1-c1ccoc1 c1(NC(C2C3C(=O)OCC23Br)=O)cc2c(s1)COCC2 C(=O)(C(C)S(N)(=O)=O)NC1(CF)CCN(C(C2CC(C(=O)OC)C2)=O)C1 c1(C(=O)NC(CNC(Cc2cnc(C)o2)=O)C)cc(C)n(-c2cccc(Cl)c2)n1 N1(C(C2CCN(C(c3c(C)nccc3)=O)C2)=O)CC2CCC(C1)N2C N1(c2cnc(SC(C)=O)c(C)c2)C(=O)C2CC(CC(O)CN2)C1=O c1(C(N(C2CCN(C(C(C)C3(O)CCC3)=O)CC2)C)=O)ccnc2[nH]ncc12 c1(C(C(=O)N(C(CNC(C(C)SCC)=O)C2CC2)C)(F)F)ccc(F)cc1F c1(CC)c(C(=O)NC2(C)CC(NC(=O)C3=CS(=O)CCC3)C2)sc2ccccc12 c1(C(N2CCCC(CCNC(C3COCCO3)=O)CC2)=O)ccc2cccnn12 C1(N(C(c2nc(OC)c(C)s2)=O)C)CCCC2CN(C(=O)CCF)CC12 Cc1sc(=O)n(CC(=O)NC2CN(C(=O)CSCc3cccs3)CC2(C)C)c1C c1(-c2nc(CC(CC)C)nn2C(C)C2CC2)cccc(S(=O)(=O)CCO)c1 C1(C(=O)NC2(CO)CCN(C(C3(c4cc[nH]n4)CCC3)=O)C2)COCCC1(F)F C1(C(=O)NCCNC(C)=O)(CF)CN(C(=O)Cn2cccn2)C1 C1(CNC2(c3cccc(OC)c3)CC2)N(C(=O)C#CC(C)(C)C)CCC1(C)C N1(C(COCC)=O)CCN(C2CCCN(C(=O)CSc3n[nH]c(O)n3)C2)C(=O)C1 CCCCC(O)C(C)C(=O)NCC1CCN(C(c2ccc(COC)o2)=O)C(C)C1 N1(C(c2c(C)n(C)nn2)=O)CCC2(CCCCC2NC(=O)Cc2csc(Cl)n2)C1 C1(NC(=O)CC2CCNC2=O)COCC1CNC(C1(F)CCCC1)=O C(CC(C)C(=O)NCc1cncc(C(=O)Nc2ccc(C(C)C)cc2)c1)=CC c1(N(C(CF)C2CC2)C)nc2cc[nH]c2c(=NC2CC(c3cc[nH]n3)C2)[nH]1 S(=O)(=O)(c1cc(C)cnc1NCC(C)OC)N(CC(c1ccc(OC)cc1)O)C S(=O)(=O)(c1cnccc1NC(C)CCS(C)(=O)=O)NC(C)CCOC(C)C c1(C(=O)NC2CN(C(CC3C(C)(C)CCO3)=O)C2)ccc(C#N)c(C(F)(F)F)c1 CC1CN(C(=O)C=Cc2cncs2)CC1(C)CNC(=O)CCCN(C)C C12(C(N3C4CC(C(=O)O)(C4)C3)=O)C3C(=O)C4C5CC(C14)C2C35 N1(C(C2(COC)CC2(F)F)=O)CC2CC1CN2C(c1cccc(Cl)c1Br)=O c1(NC(C)=O)ncc(C(=O)NCC2C3CC=CCC23)cn1 N1(C(c2cc(C)nc(O)n2)=O)CC(C2CN(C(c3nc(Cl)sc3Cl)=O)C2)C1 N1(C(C2(OC)CCS(=O)(=O)C2)=O)CCC2CC(NC(=O)CCC(N)=O)CCC2C1 O=C(N=c1ccn(C(F)(F)F)[nH]1)C12CC(C1)C2.c1(CNCC)cnccn1 c1(CC(=O)N(C2CCCN(C(=O)COCCF)C2)C)ncc(Br)cc1C N1(C(c2nccc(OC)c2)=O)CCN(C(=O)C(=Cc2ccccn2)C)CC1CO c1(C(=O)NCC(C(C)(C)C)NC(=O)C(O)C2CC2)ccc2c(c1)OC(C)(C)C2 CC1CN(C(c2ccnn2CCF)=O)CCCN1C(=O)CCC1CCC(=O)NC1 N1(C(C(C=C)(F)F)=O)CC(CNC(=O)CCc2cn[nH]c2)C2(CCC2)C1 Cc1cc(C)c(C(N2CC3(CNC(C4CCN(C)C4=O)=O)CC2CO3)=O)c(C)c1 CS(=O)(=O)c1ccccc1CN1CC2C(Nc3ncnc4sc(Br)cc34)C2C1 C1(C(=O)NCCC(C)N(CCC)C)C=CCN(C(=O)C(C)C2(O)CCC2)C1 C(c1ccnc2ccccc12)=CC(=O)NC1CCCC(N(C)C(c2ccns2)=O)C1 C1(NC(C(C)OCOC)=O)CCOC(C(=O)N(C2CCC(CO)CC2)C)C1 c1(NC(CCC(C)(C)NC(CCc2n(C)ncc2)=O)=O)cccc2c1CCC2 c1(NC(C2(NC(C3CCN(C4CC4)C3=O)=O)CC(O)C2)=O)cccc(O)c1 C(=O)(CCC(=O)N1CC(NC(=O)C(CO)NC(N)=O)C(O)C1)OC C1(NC(C2CCC(NC(C(CCC)F)=O)C2)=O)CC2CC(O)C1C2 c1(CC)nc(C)c(C(=O)NCC2CN(C(c3c[nH]c(=O)cn3)=O)CCO2)s1 C12(C(=O)NCC3CC(NC(CN=S(C)(C)=O)=O)C(O)C3)CCC(O)(CC1)CC2 C1(C(N2CCC(C(C)(C)NC(c3c(CC)csc3)=O)C2)=O)CCC(=O)NC1 c1(CN2CCOCC(NC(c3cnc(C)c(Cl)c3)=O)C2)cccc2ncccc12 C#CC1CCCC(CNC(=O)CCCC(C)NC(=O)C(F)(F)C2CC2)C1 C(=O)(C1Cc2ccccc21)OC.N12CCOC(C1)CN1CC(=C(C)C2=O)C1 c1(C(=O)NCCCCNC(C(C(CC)O)(F)F)=O)cc(S(C)(=O)=O)ccc1C c1(NC(C2C(NCc3c(OCC)cccc3)CCC2)=O)ccc(O)c(C)c1 CCCC(C(=O)N1CCCC1(C)C(F)(F)F)NC(=O)CSc1ccncc1 C(c1ccccc1C#N)=CC(=O)NCC1(O)CN(C(C2C(C(C)(C)C)C2)=O)C1 C1(CNC(=O)CCc2nncnc2O)CC2(CCC2)CN1C(c1cnc[nH]1)=O N1(C(C2CN(C(C(C)=C(CC)C)=O)CC(C)C2)=O)CCC(F)(F)C(F)C1 C#Cc1ccc(C(=O)NC2CCC(NC(=O)C(c3cscn3)N(C)C)C2)cc1C N1(C(C(C)C2CC2)=O)CCCC(NC(=O)COCCCF)CCC1 S(=O)(=O)(c1cc(Cl)cc(Cl)c1)N1CCCC(C(=O)Nc2cc(C)nn2C)C1 c1(C(N(CCNC(=O)C=Cc2ccsc2)CC)=O)c(F)cc(O)cc1F CC(C)C(C)C(C)CC(=O)N1CC(CNC(C23CC=CC(C2)OC3)=O)C1 Cn1nc(C(N2CC3CC3C2C(=O)NCCCOCCO)=O)cc1C#N C1(C)(CNC(c2cc(O)n(C)n2)=O)CN(OC)CCO1.C12CCC(C1)C(=O)NC2 n1(CCC)ncc(C(=O)NCC(C(C)(C)C)NC(c2coc(Cl)n2)=O)c1C N1(Cc2c(C3OCCO3)nc(Cl)s2)CC=CCC2(CCOCC2)C1 C(=O)(CCC(=O)NCC(F)(F)Cn1cc(-c2cccc(F)n2)nn1)N(C(C)C)C c1(C(C)NC(=O)Nc2cccc(C3CC3)c2)ccc(Cl)c(F)c1 C1(C2CCOCC2)(C(=O)NCCCOCCNC(CCC2N(C)CCC2)=O)CC1 N1(C(C=Cc2nnn(C)n2)=O)CCC(CO)(CNC(=O)CCc2ccoc2)CC1 C1(C2CCN(C(=O)CS(N)(=O)=O)CC2)(NC(c2c(C)n(CCO)cc2)=O)CCC1 C(CC(=O)NCC(=O)NCC(CO)NC(=O)CC1CC1(C)C)NC(C)=O c1(C(C(=O)NCCN(CCC)C(c2cncn2C)=O)O)ccc(O)c([N+](=O)[O-])c1 CCCC(C)(O)C(=O)NC1CC1NC(c1ccc(N2CCCC2)nc1)=O C1(C(=O)NC2C(CCN(C(COC)=O)C(C)C)CC2)(OC2CCC2)CCCC1 c1(CCC)nc(C)c(C(=O)NCCN(CCC)C(c2oc(C(C)C)nc2C)=O)o1 C(C(C(=O)NCCCCSC(=O)CC)NC(=O)COCCF)OCC.OC N1(C(C)=O)CCN(C(c2cnn(C3CC3)c2)=O)C(CF)C1 N1(C(C2C(CC)C2)=O)CCC(CCNC(=O)C(O)CC2CCCC2)CC1 C1(C(NNC(C)=O)=O)CCN(C(=O)OCC(C)(C)C)CC12CCC2 c1(CC(=O)NCCC(O)CNC(=O)CC2CCC2)cc(-c2ccco2)no1 CC(CC#N)C(=O)NC1CCCN(C(=O)C(C)(F)F)C1 C(=O)(C1=NOC(CNC(=O)CC(C)(C)C#N)C1)NCC(CC)(C)O N1(C(C23CC(C)C2C3)=O)CCCC2(CCN(C(c3cnc(Cl)c(F)c3)=O)C2)C1 C12(NC(C3CN(C)C3)=O)CCCC(NC(=O)CCS(C)=O)(C1)C2 C(=O)(C1(C)CCn2ccnc21)N1CC(CNC(c2oc(CC)c(C)c2)=O)C1 C1(C(=O)NOc2ccccc2)C=CCCN1C(c1csnn1)=O c1(C(N2C3C(NC(C4CC5CC5C4)=O)C(CC3)C2)=O)cccc2nn[nH]c12 S(=O)(=O)(c1c[nH]c(C(N2CC(NC(C3CC3OC)=O)CC(C)C2)=O)c1)NC c1(Nc2ccncn2)cccc(F)c1C(N1CCC(C)CC1)=O N1(C(c2nccc(N)c2)=O)CC2CCC(NC(=O)C(c3ccccc3)F)CC2C1 N1(C(C(C2CC2)OCC)=O)CCC(C2CC2)C1C(=O)NCc1cccn(C)c1=O N1(C(C(CCC#C)NC(c2cnsc2C)=O)=O)CCCC(C)(C)C1C n1(CCSC)nnnc1C(c1occc1C(C)C)NCc1cc(C)cs1 CC(C)CCCCC(=O)NCC1CC1CNC(=O)COc1ccccc1O c1(C(N2CC(C(N(CC)CC3CCCOC3)=O)C(C)C2)=O)cc2ncccc2[nH]1 C(=O)(C1=CCCCO1)NCCCN(C(C(n1cc(C)nc1)(C)C)=O)CC1CCCC1 c1(CN2CCC(O)(C(N3CC(=O)NCC3)=O)C2)ccc(F)c([N+](=O)[O-])c1 N1(C(CCC#CC)=O)CCN(C(=O)C(F)(F)c2nccs2)CC1COC N1(C(C(c2cccs2)SC)=O)CC2CC2(CNC(=O)CN2CCC(C)CC2)C1 C#Cc1cncc(C(=O)NCCC2(NC(=O)C(O)(C)C3CCC3)CC2)c1 c1ccc(C=CC(=O)NC23CC(NC(=O)CSCCOC)(C2)C3)s1.CC=C C1(c2n(CC=C3CCCCC3)nnn2)(OCC)CCCCC1NCCS(N)(=O)=O c1(CC(=O)NCCCNC(c2nc(CC)sc2Br)=O)cccc(C)c1F c12ccc(cc1)-c1cn-2nn1.C1(CCC(=O)NCCCC(C)O)CCCCN1C N1(C(C(C)OCC)=O)CCC2CC(CNC(c3n[nH]c(C)c3Cl)=O)CCC2C1 C1(NC(=O)CCC#N)CN(C(c2ccccc2)=O)CC1OC.CC1C(=O)NC12CC2 c1(C(=O)NCc2ccc(C(=O)NCC(CC3CC3)OC)s2)nccc(C)c1F c1(C(=O)NC(CC(C)C)CNC(=O)CC(C)N(C)C)ccc2c(c1)C(=O)NCC2 N1(C(CC2CCC(=O)N2)=O)CC2CCCC(C1)N2C(c1cccc(=S)n1O)=O N1(C(c2ccnc(SC)n2)=O)CC2CCC1CN(C(=O)CCc1ccsc1)C2 N1(C(C(C)O)=O)CCOC(c2cn(CC3CC4CC4C3)nn2)CC1 Cc1cc(C#N)cc(C(=O)NC2CCC(CNC(=O)C(F)(F)F)CC2)c1N c1(OCCC)ccc(CCNC(C(c2ccccc2C)CF)=O)c(OC)c1 c1(C(=O)NC(C)C(C)(C)NC(=O)C=CC2CCOC2)cc(N)ccc1Br N1(C(CCOC(C)=O)=O)CCCN(C(=O)C(F)c2ncc[nH]2)CC1 C1(C(=O)NC2(CNC(Cc3cccc(OCC)c3)=O)CC2)Cc2nccn2C1 c1(C(CNC(=O)C=CC(=O)OC(C)(C)C)SC)ccc(F)cc1 CC1C(C(=O)NCC(C)(C)CC(N2CCC3(CC2)CSC3)=O)=NOC1C c1(OC)cc(OC)cc(CN2CC3(C(=O)Nc4coc(C(F)F)c4)CC2CO3)c1 c1(CN(C(C(=O)N(C(CC)CO)CCc2ccccn2)=O)C)cc(Cl)ccc1Cl N1(C(c2c(C)nc(C)[nH]2)=O)CC2CN(C(c3ccn4nccc4n3)=O)CC2(C)C1 C1(N(C(=O)C(CSC)OC)CC)CCCN(C(c2n[nH]c(C)c2Cl)=O)C1 c1(C(N2C3C(NC(CC(C)NC(N)=O)=O)CC(C3)C2)=O)cccc(C#CCO)c1 N1(C(C(CC(C)C)CNC(=O)Cn2cncn2)=O)CCCC(C2CC2)CC1 N1(C(COCCCOC)=O)CC(C)(C)CC1CNC(=O)C(F)(F)c1nccs1 Cc1nc2ccc(C(N3CCN(C(=O)CC4(C)CC4)CCC3C)=O)cn2n1 C1(CC(=O)NCC2CCCO2)COCCN1C(c1ccc(SC2CCOC2)s1)=O N1(C(CN2CC(CC)C2)=O)CCC2(CC1)C(OC)CC2NC(=O)CSC(F)F N1(C(c2c(OC)noc2C(F)(F)F)=O)CC2CC(C1)N(C(=O)Cc1ccoc1)C2 O=C1N(CC(O)CNc2cnn(-c3ccc(F)cc3)c2)C(=O)C23CC(CN12)C3 Cc1cc(NC(=O)C(=O)NCC(C)(C(C)C)NC(=O)CC(C)O)nn1C CCC(C)(CC)C(=O)NCC12CC(NC(c3nnc(C)s3)=O)(C1)C2 CC1(C)CC(C(=O)NC2CC3CCC2C3)CN1C(=O)CCc1ccc[nH]1 c1(CNC(C2N(C(COCCOCC)=O)CCC2)=O)ccc(C)nn1 C1(CC=C)(NC(c2nc(O)c(C)s2)=O)CCN(C(=O)CCN2CCC(F)C2)CC1 C1(NC(c2csc(C(F)F)c2)=O)CC(F)(F)CC1NC(C1CCOC1)=O C1CC(NC(=O)Nc2ccccn2)CC(=O)N1.C1(COC)CCN(C(C)(C)C)C1 N1(C(CCNC(C)=O)=O)CC2(C1)CN(C(=O)CC1CC(C)OC1C)CCO2 c1(CC(=O)NC(CN(C(=O)CCC2(N(C)C)CC2)CC)C)ccc(C)cc1F C1(CC)CNC(=O)CN1C(=O)CC(C(F)F)NC(=O)C(C)c1ccco1 C(c1ccccn1)=CC(=O)NC1CCN(C(C(C)OCc2ccccc2)=O)C1 Cn1nc(C(=O)NC2CCCN(C(c3cccc(=O)o3)=O)C2)c(Br)c1Cl N1(C(c2c(OCC)cccn2)=O)CC(CO)C2(CCN(C(=O)CS)CC2)C1.OCC C1(C(N2C(C3CCN(C(c4cccc(O)c4)=O)C3)CCC2)=O)CCCC2(CCC2)O1 CC1CN(C(C2C3CN(C(=O)COc4ccccc4C)CC23)=O)CCC1=O c1(C2C(NC(=O)NCC(=O)NCc3ccncc3)C2)ccnc2ccccc12 C12(NC(c3cn(CCC)nn3)=O)CCC(CC1)N(C(c1ncoc1CC)=O)C2 C1(C(=O)NCCOCC#C)(NC(C2CC3CCCC3C2)=O)CCC(C)(C)C1 C1(NC(=O)CCCc2ccccn2)CN(C(C2CC3CCC3C2)=O)CC12CCC2 c1(-c2cn(CC3C(CNC(C(C)SC(C)C)=O)C3(F)F)nn2)ccc(F)c(F)c1 N1(C(c2cnc(O)o2)=O)CCCCC1C1CCN(C(c2ncccn2)=O)C1 C(=O)(CC(O)C(Cl)(Cl)Cl)NC(CCNC(C1(CC#C)CCOCC1)=O)C C1(OC)CN(C(C23CSCC2C3)=O)CC1C(=O)NCc1cncnc1 N1(C(c2n(CC)ccc2)=O)CC2C(NC(C3CCN(C)CC3)=O)C2C1 C(=O)(C(C(C)C)n1ncc(N)n1)N(C(CNC(CCc1cnc(C)s1)=O)C)C C(CCC(N)=O)(C(=O)N1CC2CC1C2NC(=O)C(C1CCOCC1)F)N(C)C Cc1ccc2c(N(C3CC4CNC3C4)Cc3c[nH]c4ncccc34)cccc2c1 CCCCCC(O)C(C)C(=O)N(CC(C)(C)CNC(c1c(C)ncnc1C)=O)C c1(-c2cn(CCC(=O)OC(C)C)nn2)cc(Cl)c(Cl)cc1Cl C1(NC(c2c(F)ccc(C)c2)=O)CC2CCCCC2N1c1ncnc(Cl)c1Br Cn1cc(NCC2=CCN(c3ncncc3I)CC2)c(O)nc1=O NS(=O)(=O)C1CCN(c2cc(N3CC4CC3CS4)ncn2)C1 C=CC(C)(CC)C(=O)NC1CC(C(=O)NC(c2ccnn2C)CC)C1 CCCC(CC)(c1nnnn1C(C)C(=O)OC)NCc1ccsc1Br N1(C(CCNC(=O)NC)=O)CC(C2CN(C(=O)Cn3c(C)c(C)sc3=O)C2)C1 CN1CCCC(C(N2CC3C(CNC(=O)Cn4ccnc4C(F)F)C3C2)=O)C1 N1(C(CCn2ccc(C)n2)=O)CC(C)CN(C(c2csc(F)c2)=O)CC1C N1(C(c2n(CCCC)ncc2)=O)CC(NC(=O)Cc2cnnn2C)CCC1C N1(C(C2(CC(=O)NC)CC2)=O)CCC(CCN(C(=O)COCC(F)F)C)CC1 N1(CC(=O)NC(C)(CNC(c2ocnc2C2CC2)=O)CO)CCCNC1=O Cc1ccc(C(N2CCCC(CN(C(=O)C(C)CC(F)F)C)C2)=O)c(C)n1 CCCCCCC(F)CN1CCC(c2ccc(C(=O)OCC)cc2)C1 N1(C(C(CC)C)=O)CC2CC(CNC(c3cnn(CCN(C)C)c3)=O)C2C1 c1(C(=O)Nc2n(C)nc(-c3ccccn3)c2)cccc([N+](=O)[O-])c1O O(NC(=O)C(NC(=O)C(C)n1cncn1)SC)CC(=C)Cl CC1(NC(c2[nH]ccc2C2CC2)=O)CCCCC1C(=O)NCc1ncon1 N1(C(CNS(NC)(=O)=O)=O)CC(NC(=O)C=Cc2cccs2)C(C)C1 c1(NCC(N2CCC(NC(COCCCC)=O)C(C)C2)=O)cc(C)c(Cl)c(C)c1 N1(C(C(C=C)O)=O)CC2CCC1C1CN(C(C3(n4ccnn4)CC3)=O)CC21 c1(NC(CCCC(=O)N(C)C)=O)ccc2c(c1)C(=O)NC2.C1CN1 C1(N(C(c2cc(C)n(C)c2)=O)C)CC2CCC(C1)N2C(=O)C=C1CCC(C)CC1 Cc1cc(C(N2CC(N(C)C(c3nnn(C)n3)=O)C(C)(C)C2)=O)c(N)cc1F C1(CC(N2CCC(CC(=O)O)C2)=O)OCC2CN(c3ccncn3)CCC12.CC=O c1(C(=O)NC(C)CNC(C2CCCC3(CC3)C2)=O)cc2ncccn2n1 c1(CNC(CNC(=O)COCCNC(C(C2CC2)OC)=O)CC)ccc(Cl)cc1 C(=O)(C(CC=C)C(C)C)NC1CC(NC(CC=CC=C)=O)C(O)C1 N1(C(CC(=O)OCCC(C)C)=O)CCC2(CCN(C(C3(C)CC(=O)N(C)C3)=O)C2)C1 c1(CCC)cc(C(=O)NC(CC(N)=O)CO)no1.n12cc(nn1)COCC2 N1(C(C)=O)CCC(NC(=O)CC(CNC(=O)CCOCCF)C2CCCC2)CC1 CCCCC(C(=O)N1CCCC1CCNC(=O)C(C)NC(N)=O)NC(N)=O Cc1ccc(C(C)C)c(OC(C)C(=O)NCCCCN(C(=O)CNS(N)(=O)=O)C)c1 c1(C(N2CC(CNC(C(CC)(F)F)=O)CC2(C)C)=O)ccc2c(C)noc2c1 CCCC(C)(CC)C(=O)C1=CSC=C2CC(C1)CO2 C1(CO)(NC(=O)CN2CCC(CNC(C3(F)CC=CC3)=O)CC2)CC2CCC1C2 C=C(C)CCC(C)NC(c1cnc(CNC(=O)CC(C)(F)F)nc1)=O c1(C(N2C(C)(C(N3CC(C)(C)C(O)C3)=O)C=CC2)=O)ccc2cccnn12 Cc1cccc(C2(C(=O)NCCC3CN(C(c4cscc4C)=O)C3)CCCC2)c1 C(=O)(C1=CC2(CN(C(=O)CC3C(=O)NN=C3C)C2)OC1)N(CC(F)F)CCOC C12CN(C3(CCC3)C1)C2=O.c1(OC)ccc(CC(=O)NC2CC2C(C)C)cc1F c1(C(C(=O)NCCCF)N(C)CC2CCCO2)cccc(S(C)(=O)=O)c1 C1(NC(c2ncc(C)cc2C)=O)CN(C(=O)CCCCN(C)C)C2CCCC12 C1(NC(C2C(CCC)CN(C(c3ccccn3)=O)C2)=O)CC(O)C12CCC2 S(=O)(=O)(c1ccc(Cl)s1)NCC(=O)N(CCCN(C(C(C(C)OC)O)=O)C)C c1(C(=O)NCC(CCC)NC(=O)C2=CCCCO2)c(C)cccc1O C(N=c1[nH]c2c(c(=NC3CC4(CCCC4)C3)[nH]1)CCCCC2)c1nc(C)c(C)s1 N#Cc1cc([N+](=O)[O-])ccc1CNC1CC(CF)C1 C(c1ccc(F)c(Cl)c1)=CC(=O)NCC(CN(C)C(c1cn2c(n1)SCC2)=O)O C(c1cc(F)cc(F)c1)=CC(=O)NCC1CC2(CN(C(CNC(C)=O)=O)C2)C1 C#CCCCCCC(C(=O)NC1(C)CC1)N1CCN(c2ncccn2)CC1 C(=O)(C1CCCc2sccc21)N1CC2CC(CNC(C(C)(C)C)=O)C2C1 C(=O)(C(F)CCC(C)(C)C)NC(C(C(=O)N1CCC(OC)C(F)C1)C(C)C)C CCC1C(=O)N2CCCC2C(=O)N1C.c1(CC)sccc1C C1(NC(CCOCCC)=O)CCC2CN(C(c3ccnc(F)c3OC)=O)CC2C1 c1(C(CN2CC(SCC(O)C3CCC3)C(O)C2)OCC)ccc(F)c(C)c1 C=CCCCC(C(=O)NCC=CC1CC1)NC(c1cc(C#N)n(C)n1)=O N1(C(C2CN(C)C(=O)C2)=O)CC(C(=O)NC2CC2CC(C)C)CC1(C)C c1(CNC23CC(C(=O)NCCC)(C2)C3)nccnc1C n1(CC)ncc2c(NC(C)CCNC(C3CC34CCC4)=O)ncnc12 C1(C(C)NC(=O)CC2(C)CC2)CN(C(c2ccc(C(F)(F)F)cc2)=O)CCO1 N1(C(=O)NCC(CC2CCCC2)OC)CCN2C(CNS2(=O)=O)C1 C(=O)(C(C)C(C)O)NCCN(CCOC)C(c1sccc1C(F)F)=O c12c(n[nH]c1CC)CNC(=O)C2.C1(C)C(=O)N(CC)CC(C)N1.C(C)(C)SC C(=O)(CC(=O)NC(Cc1cn[nH]c1)C(=O)NCCCNC(N)=O)N(C)C c1(NC(c2c(C)ocn2)=O)cnc(F)cc1C(=O)Nc1nc(-c2ccc(Cl)s2)cs1 C12CCON1C(=O)NCC#CCNC2=O.C(C)(C(=O)OC(C)(C)C)OCC c1(SCCOC(c2c[nH]c(C(=O)NC3CC(F)(F)C3)c2)=O)c(F)cccc1F C1(CCC(=O)NCC2(Nc3cc(-c4cn(C)nc4)no3)CC2)CCCCCC1 c1(C(N2C(CNC(CCc3c(C)ncs3)=O)CCCC2)=O)cc(C#N)ccc1Cl N1(C(C(CO)NC(c2cncc(CO)c2)=O)=O)CC2CC3CC2C1C3 N1(CCc2ccn(CC)n2)CCCC(NC(c2cc(C)ns2)=O)C1 C1(CCNC(C2(OC)CC2)=O)CN(C(C2(C)CNC(=O)C2)=O)CCO1 CC(CO)CCCNC(=O)CCC1CCCN(C(C2COCCC2C)=O)C1 c1(C(n2cc(CC3CCCN3)nn2)C#N)nccc(OC(F)F)n1 c1(CC)oc(C(N2CC=CC2CNC(C2C3CCN2CC3)=O)=O)cc1C C(=O)(CC(=O)NC(Cn1cccn1)C(=O)NCCCc1n[nH]c(C)n1)NCC C1(CC)CC1N=c1[nH]c(=NC(C)c2cccc(CO)n2)[nH]c2c(F)cc(F)cc12 C=CC(CCC)CC(=O)NC1(C(=O)NCC2(F)CCC2)CC(CO)C1 N1(C(c2cnc(CNC(C(CC(C)C)O)=O)nc2)=O)CCC2(CC1)CSC2 c1(C(=O)NCCC(C)NC(c2cc(C(C)C)c(F)cc2)=O)cccc2nsnc12 c1(OC)cccc(N2CCCC(C(C)NC(c3coc(C)c3)=O)C2)c1[N+](=O)[O-] Cc1nc(N)c(CC(=O)NC(C)CCCNC(c2ccn(C)c(=O)c2)=O)c(O)n1 N1(C(C2(NC(c3[nH]cc(C)c3)=O)CCCC2C)=O)CC(CO)OC(C)C1 CCC(CC)C(C)C(=O)N(C1CN(C(=O)COc2ccc(CO)cc2)CC1O)C C=CC(CCC)CC(=O)N(C)CCN(C)C(c1cc(C(F)(F)F)n(C)n1)=O C#CCC(C)(C(=O)NCC(C)(O)CN(C)C)NC(C1CC2(CCC2O)C1)=O C(C(C)(CO)NC(c1ccn(C(F)F)n1)=O)NC(CNC(C)=O)=O C(N=c1[nH]c(=NCCc2ncccc2F)[nH]c2c1CSC2)c1n(CC)c(C)nc1 c1(NC(=O)NC(c2c(C)cc(Br)cc2)(C)C)ncc(S(=O)(=O)N(C)C)cc1Cl C(=O)(C1=NOC(C)(C)C1)NC1C(CNC(C(c2ccc(OC)cc2)=O)=O)COC1 c1(C(N(CC(C)CNC(=O)CNC(N)=O)C)=O)cccc2[nH]ccc12 Cc1oc(-c2cccs2)nc1CC(=O)NCC1C2CN(C(=O)CSC(C)C)CC12 C1(CNC(C(C)NS(CC)(=O)=O)=O)COC(CNC(=O)Cc2n[nH]c(C)n2)C1 c1(C(N2CC(CC)C(NC(c3cn(C)cn3)=O)C2)=O)cccc2c1CCS2(=O)=O N1(C(C(F)=CCC)=O)CCC2CN(C(=O)CC(C)SC)CCC12 c1(OC)cc(Cl)cc2[nH]c(C(N3CCC(NC(=O)C(C)OC)C(O)C3)=O)cc12 C(CCCC(=O)N1CC(OCCCNC(c2ncccc2N(C)C)=O)C1)=CC CCCC(C)CC(=O)N1CC2CC1CN2c1ncc(C)c(O)n1 N1(C(C(=O)NCc2nnc(OC(C)C)s2)=O)CCC2(CCCNC2)C1 c1(C(N2CCC(CCOC)(C(=O)OC)C2)=O)cccc(S(=O)(=O)CCO)c1 C1(CC(=O)NC(COCC)CO)CC(C)(C)CN1C(=O)C(C)CCN(C)C C1(CC)(NC(C2CCC(F)C2)=O)CCN(C(=O)CC2=CCCC2)CC1 N1(C(Cn2ncc(C(=O)OC)c2)=O)CCC2CC1CN(C(=O)C(F)C1CC1)C2 CC1CN(C(=O)CC2(N(C)C)CCC2)CC1NC(C1CCC(C)(C(=O)O)O1)=O C=C(C)C1OCCC1C(=O)N(C)CCOCCC(=O)NC1CCCN(C)C1C n1(CC(=O)NC2CC(CCC(=O)NC(c3cn(C)cn3)C)C2)cc(C#N)cn1 C(=O)(C(C)(C)S(C)(=O)=O)NC(C1CCCCC1)CNC(CCN(CCC)C)=O N1(C(c2c(OC)cncc2)=O)CCC2CN(C(=O)C(C)CC(C)C)CC2C1 N1(OCCCNCc2nc(C)sc2)CC(C(=O)Nc2ccccc2)CC(F)(F)C1 CC(C(=O)NCC(C)NC(c1csc(C(F)F)c1)=O)C(C)(C)C c1(C(=O)NC2CCC(CNC(c3ccsn3)=O)CC2)ccnc2ncccc12 N1(C(Cc2c(C)ccnc2)=O)CCCCC2(CCN(C(=O)CN3CSCC3=O)C2)C1 N1(C(Cc2c(C)n[nH]c2C)=O)CC(O)(C2(CNC(=O)C3=CCCCC3C)CC2)C1 c1(C(=O)NCC2C(C)(C)CN(C(C3(CO)CCCO3)=O)C2)cc2c([nH]1)CCCC2 C=CC(CCC)CC(=O)NC1(CNC(=O)CC(=O)OC)CC(C(F)F)C1 N1(C(C2C3(CC(C#C)C3)C2)=O)CCC(C)N(C(C2CC3CCC2CC3)=O)CC1 N1(Cc2c(F)ccc(C)c2F)CC2C(CC1(C)C)C2(F)F C1(C(=O)NCC23CCCNC2C3)CCN(C2CCCCC2)C1=O c1(OC)ccc(C(=O)NCC=C2CCN(C(C3CC(O)C(F)C3)=O)CC2)c(F)c1 O=S1(=O)CCN(C(=NCCF)NCCOCCO)CC1 CC1(C)C(=O)CC1C(N1CC(O)CC1C(N1CC(n2cccn2)C1)=O)=O c1(C(N(C)CC2COCCN2C(=O)C(O)C2CC2)=O)c(F)cc(F)cc1Cl N1(C(=O)CCN(C)CCO)CCC(C)(C(=O)NOC(c2c(C)scc2)=O)C1 C1(C(=O)NCCCC(C)NC(c2c(C)c(Br)no2)=O)CCC(N=[N+]=[N-])CC1 c1(CNC(C2C(OC)CC2)=O)ccnc(N2CCN(C(c3cc[nH]c3)=O)CC2)c1 c1(CCC)cccc(C(=O)NC2CC(NC(c3c[nH]nc3OC(F)F)=O)C2)c1 c1(C(=O)NCCCN(C(C2(OC)CCC2)=O)CC)cccnc1C C(=O)(C(F)(F)C(C)O)NC1(C)CC(NC(CCCc2nnc(C)n2C)=O)C1 C1(CC=C)(C(=O)NC(CN(C)C(C2CCCCN2CCC)=O)CC)CCOCC1 N1(C(C(C)P(C)(C)=O)=O)CCCN(C(c2ccc(N)c(N)n2)=O)CCC1 N1(C(=O)Cc2cccc(Cl)c2)CCC2CN(C(=O)C3=C(Cl)CCC3)CCC2C1 C1(CNC(=O)CO)CC(F)CN1C(=O)NCCC1CC2(CC2)CO1 N1(C(COc2cc(C)on2)=O)CCCCC1C1CCCN1C(=O)CC(C)(C)C#N N1(NC(C2N(C(CC(CC(=O)OC)C)=O)CCC2)=O)CCC2(CCOCC2)C1 c1(C(=O)OC)cnc(C)[nH]c1=NC(C)CN(C)C(c1csc(S)n1)=O c1(C(N2CCCC(CNC(c3n[nH]c(C)c3Cl)=O)C2)=O)ccc2[nH]c(=N)sc2c1 N1(C(CC2N(C)C(=O)CC2)=O)CC2(CCC(C(N3CC4CC4C3)=O)CC2)C1 n1(CC)nc(C)c(C(=O)NC2CCOC(CO)C2)c1C(F)F c1(COC)cccc(CC(N2CCCC(NC(=O)C(C)NC(=O)OC)C2)=O)c1 C(CC(=O)N(CC(N)=O)CCC)(C(F)F)NC(C(CC#C)O)=O N1(C(C2C(CC)C2)=O)CCC2(CCCC2CNC(C2CCCC(CF)C2)=O)CC1 C1(C(C)C)CCCCC1.N1CC(C(O)C(=O)N2CC(N3CCCC3)C2)C1 c1(C(N(CCCNC(C2CC23CCOCC3)=O)CC)=O)cc2c([nH]1)CCOC2 c1(C(=O)NCC2(NC(C(CC#C)O)=O)CCC2)ccc(S(=O)(=O)NC)o1 c1(C(=O)NCC(CNC(c2cnn(CC)c2C)=O)CO)c(F)ccc(O)c1F C1(NC(=O)C=CC(=O)NC2CC2)CN(C(=O)CC2C=CCCC2)C2CCCC12 C(=O)(C1CCCc2cccnc21)NCC(C1CC1)NC(c1occ(C)c1C)=O C(=O)(CCS(N)(=O)=O)NCc1c(C(N2C3(C(=O)OC)CC3CC2)=O)occ1 c1(CC)c(C(=O)N(C(C)CCNC(=O)C=Cc2cn(C)nn2)C)nnn1CC C1(C(C)C)CN(C(=O)C=CC=C(Cl)Cl)CCC1NC(=O)CC12CCCN1CCC2 CCC(CC)(CC)C(=O)N1CCC(NC(C2CC(=O)N(O)C2)=O)C1 c1(NCC(CCNC(C(F)N(C2(C#C)CC2)C)=O)O)ocnc1C(=O)OC C#CCC(C)(C(=O)N1CCC(C)(O)C1)NC(=O)CCN(C)CCC C=Cc1cncc(C(=O)N(c2cn[nH]c2)CCN(CC(C)O)C2C(CC)C2CC)c1 n1(CC)cnc2c(NCCc3nnc(CSC)s3)[nH]c(=NC(C)CC(N)=O)nc12 C1(O)(CNC(CCCOC(C)C)=O)CCN(C(C2OCCCO2)=O)CC1 C(c1ccc([N+](=O)[O-])s1)=CC(N1CCN(C(C=NOC)=O)C(CCOC)C1)=O c1(C(=O)NCCN(C(=O)CSCC(F)F)CC2(F)CC2)ccoc1 C1(NC(Cc2c(C)occ2)=O)CC=C(C(=O)NCc2cnccn2)C1 C1(CNC(c2nc(C)c(C)s2)=O)COCCN(C(C2Cc3nncn3C2)=O)C1 n1(CC(NNC(N2CC(C)C(O)CC2)=O)=O)cnc2ccccc12 C1(NCc2cn(CC(=O)NCC(=O)OC(C)(C)C)nn2)CCCCC1O C(=O)(C1=COCCO1)NC(C)CCN(C)C(c1ccc(C2COC2)cc1)=O CN=c1nc(N2CCCCC2)[nH]c(=NCCCOCCC(C)C)[nH]1 C(=O)(C(C)(C)CN(C)C(c1ncc(F)cn1)=O)NCc1nc(C(C)C)sc1 c12nc(n[nH]1)NC2C.C(CC(C)(C)c1ccccc1)NC(C(=O)OC)=O CN1CCOC(C(=O)NCCN(C(C2CC3CC3C2)=O)Cc2cccnc2)C1=O Cc1ccc(CNC(=O)C#CC(=O)Nc2cn(C3CN(CC(=O)O)C3)nn2)nc1 Cc1cc(C(=O)N(C2CN(C(=O)CCCn3ccnc3C)CC2F)C)oc1C C12(CNC(c3c(CC)cno3)=O)CCC1CN(C(c1cccn(C)c1=O)=O)C2 C1(F)(CNC(Cc2c(C)nc(C3CCOC3)s2)=O)CCCN(C(=O)C(Cl)=CCl)C1 CCCCS(=O)(=O)CC(=O)NCC1C(C)CCCN1C(=O)Cc1ccoc1 c1(CN2CCN(C)C(CC3(c4ccccc4)CC3)C2)n[nH]c2ccc(F)cc12 C(=O)(CCCCCN(C)C(C1(C)CC1(C)C)=O)NCc1nnc(CC)o1 Cc1ccc2sc(C(N3CC(NC(=O)CCOC4CC4)C(C)(C)C3)=O)c(C)c2c1 N1(C(=O)Cc2cnccn2)CC2(CCN(CC3CCCC3C(F)(F)F)CC2)C1 C1(NC(c2cnn(-c3ccncc3)n2)=O)CCCCN(C(c2ccsn2)=O)CC1 c1(C(=O)NC2(C3CC3)CCN(C(=O)COC3CCC3)C2)cnc2c(c1)CCCC2 CC1CC(NC(=O)COC2CC=CC2)CN1C(c1cnc(C(N)=O)cn1)=O c1(C(N2CC(CC(=O)NCC3(F)CN(C)C3)(OC)C2)=O)cc(N)cc(F)c1 Cc1cnc(C(=O)NC(c2ccnn2C)C(=O)NCC2=CCOCC2)c(C)c1 C1(NC(CC=C)=O)CC(C)CN(C(=O)C=Cc2ccc(C)o2)C1 CC1CCCN(C(C2CCCC23CC3)=O)C1CNC(c1ccc(C2CC2)o1)=O CC1(CNC(=O)CCC(=O)c2ccc(Cl)cc2)CN(C(c2ccoc2)=O)CCO1 C(=O)(CC(C(F)F)C(C)(C)C)N1CC(CC(C)NC(C2=C(C)OCC2)=O)C1 C1(NC(CC2C(C)(C)C2(C)C)=O)CN(C(c2cc(F)cc(Cl)c2N)=O)CC12CCC2 CCCCCCCCC(=O)N(CCNC(C1CCC(O)C1)=O)CC c1(C(=O)NCCCC(C)NC(C2(C)ON=C(C)C2)=O)ccc(=O)n(C)n1 c1(CC(N2CC(CC)N(C(=O)C3=CSCS3)CC2)=O)ccc(OC)cc1[N+](=O)[O-] N1(C(C)CC(N2CC3(C2)CN(C(=O)Cn2cnnc2)C3)=O)CCc2ccccc21 N1(C(c2ncc(CC)s2)=O)CCN(C(c2cccc(C(C)(F)F)c2)=O)C(CC)C1 C(=O)(CCS(C)=O)N(CC(C)=CC(=O)NC(=O)C(C)C(C)O)CC(C)C Cc1ccn2c(C(N3CCC3CNC(c3sccc3F)=O)=O)cnc2c1 c1(NC(=O)OC)ccc(C(=O)NC2CC(NC(C3CNC(=O)N3)=O)C2)c(Cl)c1 c1(CN2C(C(=O)Nc3nc(C)c(Br)nc3)CCC2)cc(F)c(F)c(Cl)c1F c1(C(N2CCC(CC)C2CNC(=O)COC)=O)n[nH]c2c1CCC2 C(=O)(C1=CCCCC1C)NC1C(NC(c2snc(C)c2N)=O)CCC1 Cc1c(C(N2CCCC(NC(c3cn4c(n3)SCC4)=O)C2)=O)cccc1N c1(C(=O)NCCC(C)(C)NC(C2(c3cc[nH]n3)CC2)=O)cc(Cl)cc(Cl)c1F N1(C(c2n(C)nc(O)c2)=O)CCC(CNC(=O)CC2(C)CC2(Cl)Cl)C12CCC2 Cc1ccncc1C=CC(=O)NC1CN(C(=O)CO)CCC1c1ccccc1 c1(OC)cc(C)cc(Cl)c1CN(Cc1ccccc1)Cc1ccc(Cl)cc1Cl c1(C(=O)NCCCCNC(C2C(C)(Br)C2)=O)ccc2c(c1)C(=O)OC2 c1(NC(c2ccc(NC(=O)OCC)nc2)=O)nccc(Cl)c1F CC1(C#CC(=O)NC2CCN(C(c3cc4n(n3)CCO4)=O)C23CC3)CCCO1 Cc1snnc1C(=O)NCC1C=CC(NC(=O)CNC(=O)C(F)(F)F)C1 C(C(C)C)(C(O)C(=O)N1CCCC(CO)(NC(=O)CCc2ccncn2)C1)OC c1(C(=O)NCC2CCCC(CNC(c3n(C)ncc3Cl)=O)C2)cccc(F)c1N c1(C(=O)NCC(C)(C2CC2)NC(c2ccc(Br)o2)=O)cncc(O)c1 Cc1ccc(C(=O)NC(C(=O)N2CCCCC2C)C(C)O)n1C C1(NC(C(CSC)O)=O)CC(C)N(C(=O)CSc2nnc(S)s2)C1 C12CCN(CC1)C2.C1(C(=O)NC2(N(C)C)CC2)CN(C(=O)CCNS(C)(=O)=O)C1 N1(C(C(CO)OCC(C)C)=O)CC2CC(NC(=O)C(C)(C)C#N)C(C2)C1 c1(C2(CNC(C3(CNC(c4cnc(I)cn4)=O)CC3)=O)CC2)c(O)cccc1F c1(C(N2C(CNC(C3=NOC(C)C3)=O)COCC2)=O)cnc2cc(O)ccc2c1 N1(C(c2c(OC)nccc2)=O)CCCC12CCN(C(=O)CC1CC13CC3)C2 C12(CC3(CCC3)C1)C(=O)NCCN(CC)C2=O.c1(CF)cccc(F)c1F Cn1ncc(S(C)(=N)=O)c1-c1cn(C23COCC2C3(F)F)nn1 N1(C(c2c(CC)ocn2)=O)CCC(C(C)NC(=O)COCCF)CC1 Cc1cc(C(=O)NCC(O)CNC(=O)CC2CCSCC2)nn1C(C)C c1(OC)csc(C(N2CCC(CNC(c3ccnc(O)c3)=O)C23CC3)=O)c1OC c1(C(=O)NCC(CC)NC(=O)CCc2nncs2)ccc(F)c(Cl)c1 N1(Cc2cc(C)cc(-c3cnn(C)c3)c2)CC(C(N)=O)CC(F)(F)C1 C1(CN2C(n3ncc(C(C4CCS(=O)CC4)=O)c3)CCCC2)CCc2nncn2C1 c1(C(N2CCC(NC(=O)Cc3cc[nH]c3)C(F)C2)=O)ccc2c(c1)S(=O)(=O)NC2 C(=O)(C1CCCc2cncn21)NC(C)CCN(C)C(c1cc(Cl)ccn1)=O c1(CC)cccnc1C(=O)NCC1(C)CCN(C(c2cc(C)nn2CC)=O)C1 n1(CC(=O)N(C(C)C)C2CC2)cc(CNC(c2ccon2)=O)nn1 N1(C(Cn2c(C)csc2=O)=O)CC2(CCC2)CC1CNC(c1cn(C)c(O)n1)=O c1(-c2sc3c(n2)CN(C(C(CCCCC)C)=O)CC3)cc(C2CC2)cc([N+](=O)[O-])c1 C1(C(N(C)CC2N(C(C(C(C)C)SC)=O)CCC2)=O)CCC(C)(C)OC1 N1(C(CSCC=C)=O)CC2CC(NC(=O)CCNC(=O)CC)C(C2)C1 C1(NC(C)=O)CCCN(C(C2CN(C(C3CN(C)CCO3)=O)CC2C)=O)C1 c1(OC)ccc(CC(N2CCC(NC(C3CCC(=O)NC3)=O)C(O)C2)=O)c(Cl)c1 Cc1cc(C(F)(F)C(=O)NCC(C)NC(=O)CCCC2CC2)cnc1Cl c1(C(=O)NC(C)CCCNC(=O)C(=O)N(C)C)cc2ccccc2cn1 C(=O)(CCCCC(N)=O)N(C1CCCN(c2ccnc(C(F)(F)F)n2)C1)C C1(C(N2CCC(CN(C)C(c3ccncc3)=O)CC2)=O)Cc2cccnc2C1 c1(C(=O)NCC2OCCCN(C(C=C(C)C)=O)C2)cnn2ccccc12 c1(C(N(C2CC(NC(=O)C(F)CC3CC3)C2)C)=O)cc(Br)ccc1Cl C=CC(C)(O)CC(=O)NC1CCN(C(=O)CCC(=O)NCC)CC1 N1(C(C(=O)c2ccco2)=O)CCCCC1C(N1CCC2CC12)=O c1(C(N(CC(CN(C)Cc2noc(C3CC3)n2)O)C)=O)cc2ccc(Cl)nc2s1 c1(C(=O)NC(CCC)CO)ccc(F)c(-c2cnc(OC)c(OC)c2)n1 C1(NC(C2CCCC(F)C2)=O)C=CCN(C(c2ccc[n+]([O-])c2)=O)C1 N1(C(C2CC(OCC)C2)=O)CCCC(C2CCN(C(c3nocc3C)=O)CC2)C1 c1(C(N2CCC(C)(CCNC(C3(COC)CC3)=O)C2)=O)cc2c([nH]1)CCC(C)C2 c1(C(N(C)CCNC(C2CC(O)CN2C)=O)=O)ccccc1[N+](=O)[O-] N1(C(C(C)(C)OCC)=O)CCCC(Cn2cc(CCCOCCS(N)(=O)=O)nn2)C1 CC(CCNC(=O)C#CC(C)(C)CNC(c1nn(C)cc1Cl)=O)CC(C)(C)C c1(CC(COC(C)=O)NC(=O)C(Cl)=CCl)ccc(C)cc1 C(CC(C)CCNC(=O)CN1CCC(C)(C)C1)NC(C(C)C1(O)CCC1)=O N1(C(CC2(C=C)CC2)=O)CCCCC2C1CCCN2C(C1CCC(F)(F)C1)=O C1(NC(C2CCC(CC)CC2)=O)CCN(C(=O)C(C)CN2CCCC2)CC(O)C1 c1(C(N2CC3CN(C(C=C4CCC(C)C4)=O)CC3C2)=O)cccc2oc(O)nc12 C1(NC(c2cc(F)cs2)=O)CC2(CCCCN2C(C2Cc3ccccc3O2)=O)C1 c1(C(N(CC(O)CNC(c2cc3c(s2)CCC3)=O)C)=O)nc(O)nc(O)c1F CC1CN(C(c2nccnc2Cl)=O)CCC1CNC(c1ncc(Cl)cc1Cl)=O c1(C(=O)NCCN(C(=O)CNC(c2cccs2)=O)C)cnc(O)c2cnccc12 Cc1cc(F)c(NC(c2ccc(CNCCc3cccs3)s2)=O)cc1Cl c1(C(=O)NC(CC(C)NC(=O)CC2CCC3CC23)C)ccc(Br)cc1 c1(C(=O)NCCC2CC(NC(C(C)(C)C#N)=O)C2)cc2ccc(Br)cn2c1 Cc1nc(NCC(C)OC(F)F)cc(=NCc2noc3ccccc23)[nH]1 Cc1cc(C)n(C(C)C(=O)NCC2CCCN2C(c2ccnn2CC#N)=O)n1 c1(OC)cccc(C(N2CC(CCNC(=O)C(C3CCOC3)OC)C2)=O)c1F C(=O)(CC1CNc2ccccc21)NCCCC1C(N)C1 N1(C(C(C)C)=O)CC(CNC(C2CC2F)=O)C2(CCOCC2)C1 C1(CC(N2CC=CC(NC(c3c(C)nccn3)=O)C2)=O)CC(C)(C)CCO1 C1(NC(c2n(CC=C)nnn2)(C)CSC)CC2(C1)CC(C)C2 C1(CNC(C2(CNC(C)=O)CCCC2)=O)CN(C(c2cncc(C)c2)=O)CC1O C(=O)(C(C)S(C)(=O)=O)NCCN(CCC)C(c1ccc(CO)cn1)=O c1(CC(=O)NCC2(F)CCN(C(c3c(C)c[nH]n3)=O)C2)ccc2sccc2c1 C=CCC(F)(F)C(=O)NC1C2CC1CN(C(c1cccnc1OC)=O)C2 C1(NC(c2c(C)nco2)=O)CC(NC(c2nc(Cl)ccc2C(C)C)=O)C12CCC2 c1(CN2CCC(CC(=O)N(N3CCN(C)CC3)CC=C(C)C)C2)ccc(C)c(F)c1 S(=O)(=O)(c1cccc(NC(C23CC(C)(CN2C(=O)OC(C)(C)C)C3)=O)c1)N(C)C C#Cc1ccc(F)cc1C(=O)NCC(C)CNC(c1cc(CC)ccc1F)=O C1(NC(C2CCC(F)(F)CC2)=O)C2CCC(C2)C1C(=O)Nc1cc(CO)ccn1 C1(CC(=O)NCCCN(C(C2CCN(S(C)(=O)=O)C2)=O)CC)CCCC1(F)F C=CCCN=C(NCc1ccc(C)cc1OC(C)C)NCC(C)(O)C(F)F N1(C(C(C=C)(C)CC)=O)CC2(CCN(CCNC(=O)C(C)CC)C2)C1 c1(C(=O)NC(C(C)NC(C2(C#C)CCCC2)=O)C)nc(SC)n2ccccc12 C1(NC(C(c2n(CC)ncn2)Nc2cnn(CCO)c2C)=O)CCC(F)(F)CC1 CC1CCN(C(=O)CCOc2ccccc2Cl)C1c1cn(C2CC2)nn1 C1(CNC(CC(COC)NC(c2ccc(OC)s2)=O)=O)CC(C)CC(C)C1 C=C(C)CC(C(=O)NC1C=CC(CNC(c2cc(C3CC3)no2)=O)C1)OC C=CCCC(C)(C)C(=O)NC1CC2CCC1N(C(=O)C(F)(F)C(O)C1CC1)C2 c1(Nc2c(C#N)cncn2)ccc2c(c1)CCN(S(=O)(=O)CCC(F)(F)F)C2 c1(OC(C)C)ccccc1CC(=O)NCCC1CC(NC(C2CCC2F)=O)C1 N1(C(C(=O)Nc2c(C)nsc2)=O)CCN(C)CC1C1CC1 c1(CC)ncccc1C(=O)NC1CCN(C(c2cc[nH]c2C2CC2)=O)C1C1CC1 c1(CC)cc(F)ccc1C(=O)NC1CC(C)(NC(c2ccc(NC=O)cc2)=O)C1 C1(C(=O)NCCOCCN(C(C(C)CO)=O)C)(CF)CC12CCC2 Cc1cn2nnc(C(=O)NCCCN(C(C3C4CC(=O)CC34)=O)C3CC3)c2c(O)n1 c1(C(c2n(CCCSC)nnn2)NC2(C3CCCO3)CC2)cc(S(C)(=O)=O)co1 C(=O)(CC(CC(C)C)NC(=O)CC1CCCN1C)N1CCC(=C)CC1 C1(NC(C(C)OCCC)=O)CC2CCC1N(C(c1ccnnc1C)=O)C2.C(=O)(C)OC C12(NC(C(C)c3cccs3)=O)CCC(NC(c3ccnn3C)=O)(CC1)C2 C(=O)(C(CNC(c1ccsc1Cl)=O)N(C)C)N(C1CCN(C)C1)CCC C12(NC(C3CC(F)(F)C3)=O)CCC1CN(C(=O)CCN1CCCCC1=O)C2 C(=O)(C(F)CC(CC)CC)NC(CCCC)CNC(c1ccccc1F)=O C(=O)(C(C)(C)N=[N+]=[N-])NCC1C(C)CN(C(c2ccnnc2)=O)C1 C1(C(=O)NCC2C(CNC(CSc3cn(C)nc3)=O)C2)CN=C2N=CNN2C1 c1(C(=O)NC(CNC(C(c2ccn(C)n2)C)=O)CO)cc2c(nc1O)CCSC2 CC1CC(C)CN(CCN(C(=O)C(O)CCn2cc(C3CCC3)nn2)C2CC2)C1 c1(-c2cn(CCOC)nn2)ccccc1OC(=O)CCCSC C1(CNC(c2nc(Cl)cs2)=O)CC(NC(C2(C(F)(F)F)CCOCC2)=O)CC1O N1(C(CCCC(=C)C)=O)CC2CC(C)N(C(c3ccc(N(C)C)cc3)=O)C2C1 N1(C(=O)OC(C)(C)C)CC(COCCl)CC12CCC2.c12ccc(o1)C(=O)N1CC2C1 C1(C(N2CCC(C(C)C(=O)NCC=C(Cl)Cl)CC2)=O)CN(C)CCN1C CC1CCc2nc(Cl)nc(N3CCCC4(NC(C5CN(C)C5)=O)CCCC34)c2C1 c1(C(C)=O)c[nH]c(C(=O)NCC(C)CN(C(=O)C=CCN(CC(F)(F)F)C)C)c1 c1(OC)ccc(C(=O)NCC(C)NC(=O)Cc2cc(C)ccc2F)n2nccc12 c1(NC(c2cc(OCC)ncc2-c2cnc(C)nc2)=O)cccnc1[N+](=O)[O-] n1(CCOC)ccc(C(=O)N(CCCNC(=O)C=Cc2ccsc2)C)n1 C(=O)(CC(F)(F)C(F)F)NCC1C(C)CCCN1C(C1CCCN1C(N)=O)=O c1(C(N2CC(NC(c3c(Cl)cnc(CC)n3)=O)C2)=O)ccc2c(c1)CCN(C)C2 C1(c2n(CCOCC)nnn2)(NCc2nc(C(C)(C)C)oc2C)CCC2CC12 N1(C(C2CCC(C)O2)=O)CCC(C2(NC(C3(C)CC(C4CC4)=NO3)=O)CC2)CC1 Cc1cccnc1NC(=O)NCC(N1CCC(CN(C)C(c2cccs2)=O)C1)=O CC(=O)CCCC(=O)NC1(CF)CCN(C(c2cccnc2CO)=O)C1 C(=O)(CCCN(C)N=O)NCCC(CNC(C(CC=C)C)=O)OC C(=O)(C1=C(CC)OCCS1)N1C(CCCC)CN(C(=O)C(F)C2CC2)CC1 C=CC(C(=O)NCC(C)(CNC(=O)CC1(C(F)(F)F)CC1)OC)c1ccccc1 C(c1cncnc1O)=CC(=O)NC1C(OC)CN(C(=O)CC2(O)CCCOC2)C1 Cn1nccc1CNC(c1cc(CNC(=O)C=CCN2CCCC2)no1)=O N1(C(C(COC(C)C)N(C)C)=O)CC2(C1)OC1(C)CC2(n2ccnn2)C1 CC(CS(C)=O)C(=O)NC(C1CCN(C(C2CC=CC2)=O)CC1)CO c1(C(=O)NCC2CN(C(Cc3cccc(N)c3)=O)C2)nnn2c1COCC2 N1(C(CC(=C)C)=O)CCC2CCCN(C(c3ncn4ccc(C)cc34)=O)C2C1 N1(C(c2cc(C)cc(O)c2)=O)CCCC1C1CCCN1C(c1ncc(F)cn1)=O c1(C(=O)NCC2CC(NC(c3cc(C)ncn3)=O)C2)ccc(N)c2ncccc12 N1(C(c2nccc(CNC(C(C(CC)O)(C)C)=O)c2)=O)CCOC2CN(C)CC12 C(CC(C)(C)CC(=O)NCC12CC1CN(C(c1cn(C)cn1)=O)C2)OC c1(OC)ccc2c(N(CCCC3CCC3)C)nc(N3CCCC(C#N)C3)nc2c1 c1(C(=O)NC(C(C)NC(c2c(OCC)cccn2)=O)CO)nsc2ccccc12 C(=O)(CCCC(C)(F)F)N(CC1CCN(C(CC(=O)OCC)=O)C1)CC c1(C(N(CCNC(CC2CCC(C)O2)=O)C2CC2)=O)ncnc2c1ncn2C1CC1 N1(CC)C(=O)NC(c2ccc(N)c(Br)n2)C2=C1C(C)CN(C)C2=O N1(C(Cn2c(C)ccc2C)=O)CCC2CCN(C(c3ccn4ccsc34)=O)CC12 C=CCC(CC(C)C)C(=O)N1C(CNC(=O)C(N)=O)CC2CCCC12 CCC(C(=O)NCC(O)CSC)N(C)C(C1SCC=C1C)=O C1(NC(=O)CC2CCCO2)COCCN(C(c2cccc(-c3ccncc3)c2)=O)C1 c12cc3n(c1)CCN(C3)C2.C(CO)(C(C)c1ccccc1)N(C)C(=O)O.C(C)(C)(C)S CC(C)C(CC(=O)N1CCCCCC1)NC(=O)C(CO)N(C)C O=C1NC(=O)C(CC(N2CCC(n3cc(CCC(O)C4CC4)nn3)CC2)=O)N1 CC1C2C(CCN2C(C2CC(C)(O)C2)=O)CN1C(=O)C1=COCC1 C1(C(=O)NC2(C(N3CC4C(C)(C4)C3)=O)CCCCC2)CC2CC(=O)C1O2 C1(CC(N2CCC2(C)C(C)C)=O)(OC)CN(C(=O)Cc2cc(C)on2)C1 N1(C(c2ccc(CC(C)C)nc2)=O)CCC(O)C(N(C(=O)C(F)C2CCC2)C)C1 N1CCC2(CC1)CC(n1cc(CC(N)=O)nn1)CCO2.CC(C)(C)OC(=N)O C(=O)(C(CC(C)C)NC(C1CC(=O)CCO1)=O)NCc1scc(C)n1 c1(OC)ccc(F)c(CN2C(C(=O)N(C)CCC3OCCO3)CC3CC23)c1F N1(C(c2cccc(-c3nc(C)on3)c2)=O)CC2CCCC2(NC(=O)CC(F)F)C1 CN1CC=C(CC(=O)N2CCC3CCC(C2)N3c2nc(C3CC3)nc(Cl)c2Cl)CC1 N1(C(Cc2scc(C)c2)=O)CCCC(O)(CN(C(=O)Cc2ccns2)C)C1 C(=O)(C1=CCC(NC(C2CCCN2C=O)=O)C1)NCC1NC(=O)OC1 CC1CN(C(c2cnsc2)=O)CCC1CNC(C1CC1c1ccc(F)cc1F)=O CON(CCC(=O)NCC=CCSC)C(=O)C(C)N1CCCC1=O C1(C(=O)OC)CC12CN(C(=O)C(C)(C)CN(C)C(c1cn(C)cn1)=O)C2 c1(C(N2CCCC(C(=O)NCC3CCCO3)C2)=O)ccc(C2CC2)nc1 c1(CCNC(C2C(CC)NCC2)=O)cc(C)ccc1C C1(O)(CCC)CCN(C(C2CC(F)CCN2C(C2CCSC2)=O)=O)CC1 c1(CCCC(=O)NC(CC)CNC(=O)C=CCOC)ccc(C)c(C)c1 c1(N2C(CNC(CNC(=O)NC)=O)CCC(NCC)C2)ncnc2sc(C)nc12 C(=O)(C(C)CC(C)C)NCC1CN(C(c2c(CC)n(C)nc2)=O)CC1C c1(C(=O)NC(C2CC2(C)C)CC)ccc(CNC(c2cnc(CO)s2)=O)cn1 CC(CCN=c1[nH]c(N2CCOC(CC(N)=O)C2)nc2cc[nH]c12)C1CCC1 C1(CC)C(C(=O)NC2CC3(CC(OC)C3)C2)CCCN1C(=O)C(F)C1CCC1 N1(C(C(C)(CO)NC(C(=O)N(C)C)=O)=O)CCOC2CCC12 C(=O)(N=c1[nH][nH]c2ccc(OC(F)(F)F)cc12)N1C(c2n(C)ccn2)C(C)(C)C1 C1(NC(CC(CCC)O)=O)CN(c2ncnc3sc(C)c(C)c23)C2CCCCC12 c1(CN(C)CC2CCCN2C)cc(O)ccc1Cl CC(C)(CO)CCCNC(=O)CC1CCC(NC(C2(C#N)CCCOC2)=O)CC1 C1(CC=C)(C(=O)NC2CCC(NC(C3(COC)CCCO3)=O)C2)CCCC1 Cc1cc(C#N)ccc1C(=O)NC1CN(C(=O)CC(C)(C)C(F)F)CC2(CC2)C1 N1(C(CSC)=O)CC=CC(NC(c2ccn(C(C)(C)C)n2)=O)C1 N1(C(C(COC)C)=O)CCCC(C(C)NC(c2cnn(C)c2C)=O)C1 N1(C(C(C)n2ccnn2)=O)CC2CCCC(C1)N2C(=O)CC1CCN(C)CC1 N1(C(C(CSC)C)=O)CCC(O)(C(C)CNC(=O)CC=C(Cl)Cl)C1 c1(C(=O)NC(CNC(CC(C=C)(C)C)=O)(C)C2CCC2)ccc(N)c([N+](=O)[O-])c1 C1(C)(CNC(C2(SCC)CC2)=O)CN(C(=O)CC2CCCOC2)CCO1 C12(NC(C(N3CCCCC3=O)C)=O)CC1CN(C(=O)CCc1cc[nH]n1)C2 C12(NC(c3cc(Cl)ccc3F)=O)CCN(C(c3conc3C3CC3)=O)CC1C2 N1(c2ncnc(NCC3(CCCC)CC3)c2C)CCCN(C)C(=O)C1 c1(C(c2ccc(CCCC(F)F)s2)NCOC)ccc(F)cc1.N N1(C(c2cc(C)oc2C)=O)CCC(NC(=O)Cc2cc(F)ccc2O)CC1C c1(C(=O)NCC(C)(C2CCC2)NC(=O)C(F)=CCF)ccc(F)cc1 Cc1[nH]c2ccc(C(=O)OCCc3ccc(Cl)c(Cl)c3)cc2c1C C(CC1=CCN(C(=O)CC2CCCCC23CC3)CC1)NC(C1(C)CCOCC1)=O CC(C)(C)C#CC(=O)N1CC2CC(C1)C2NC(c1ccc(C2CCOC2)cc1)=O C1(O)(C(=O)NCCCN(C)C(c2ccc(CC#N)cc2)=O)CC2CCC1C2 C1(C2CCN(C(c3nn[nH]c3Cl)=O)C2)(NC(C2CC2c2ccsc2)=O)CC1 c1(OC)ccc(Cl)c(CC(N2CCN(C3CCC3)CC2)=O)c1F.C(C(O)CO)C=O c1(CCC)nc(C)c(C(=O)NC2C=CC(CNC(c3cscc3COC)=O)C2)s1 C(=O)(CC(C)(C)C)N1CCC(N(CCC)C(c2cnn(CC(F)(F)F)n2)=O)C1 C(=O)(C(O)CC(N)=O)N1CCC(NC2(C(=O)NCNC(C)=O)CCOCC2)CC1 N1(C(c2ccc(NC(C3(C)CC(=C)C3)=O)nc2)=O)CC2(CCCCCC2)C1 c1(C2C(C(N(CCCNC(C3(NC(N)=O)CC3)=O)C)=O)CC2)c(Cl)cccc1Cl C=CCCCC(C(=O)OC)NCCc1cnc(OC)nc1 c1(C(N(CCS(C)(=O)=O)C)=O)ccnc(-n2cccn2)c1 N1(C(c2c(C)noc2)=O)CC2(C1)CN(C(C1CC1c1cccs1)=O)CC(C)(C)O2 CCC(CC)C(F)C(=O)N1CCN(C(c2cccn(C)c2=O)=O)C(CO)C1 c1(C(CC)CC)n[nH]c(=NCc2noc(-c3ccsc3)n2)o1 C(C(C(=O)NCC(O)C(=O)NCCCC1CCCC1O)N(C)C)N(C)C c1(OC)ccc([N+](=O)[O-])cc1CNC(c1ccc(I)cc1)(C)C c1(CNC(c2c(CS(C)(=O)=O)cccc2)=O)n[nH]c(=Nc2cccc(F)c2)s1 c1(C(=O)OC)cccc(C(=O)Nc2ccc(C(N3CCCC(C)CC3)C)s2)c1O c1(CC)ncc(C(=O)NCC2CC(F)(CNC(=O)CCCC#N)C2)c(C)n1 c1(SC)nc(C)c(CCC(=O)NC2CCN(c3nccc(C#N)n3)C2)c(O)n1 N1(C(=O)NCc2c(C)nc(C)s2)CC(NC(=O)OC(C)(C)C)C(C)(C)C1 Cc1cc(C(=O)NCCCNC(=O)CCC#N)ccc1F C1(NC(C(CC)N(CC)CC)=O)COC2(C1)CN(C(=O)CC1CCCC1)C2 c1(OCC(CNC(c2nc(-c3ccsc3)cs2)=O)O)ccccc1 Cc1cn(C)nc1C(=O)NC1CCC1NC(=O)CCSc1ccccc1 c1(C(=O)NC2CN(Cc3cccc(C(=O)OC)c3)C2)ccc2c(c1)CCCC2 c1(C(=O)NC2CC3(CCN(C(=O)CCC4CCC4)C3)C2)cc2cc(Cl)cnc2o1 Cc1ccc(C(C)C(N2CCOC(CN(C)C(c3cc(Cl)cn3C)=O)C2)=O)cc1 N1(C(C2CCC(C)O2)=O)CC2(C1)CN(C(=O)Cc1cn(CCO)nn1)CCO2 C(=O)(CCC(C)C#N)NC12CC(CNC(c3cncc(OC)n3)=O)(C1)C2 c1(C(N(C)CC2CCN(C(COCC=C)=O)C2)=O)ccc(OC)c(F)c1F CS(=O)CCC(=O)NCCC1(NC(c2cc(C(=O)C(F)(F)F)c[nH]2)=O)CCC1 C1(NC(C2CC3(CCC3)CO2)=O)CC2(CCCN(C(c3ccc(Br)o3)=O)C2)C1 c1(C(=O)NCC=CCNC(CC2(O)CC(C)(C)OC2)=O)cc2ccc(O)cc2[nH]1 C1(CC)CCCCCN1C(=O)Cn1cc(-c2cccc(OC(F)(F)F)c2)nn1 c1(C(=O)NCCCN(C(=O)Cc2cnccc2OC)CC)[nH]nc([N+](=O)[O-])c1Cl Cc1cc(F)c(C(=O)NCC2=CCCN(C(C3(Cl)CCC3)=O)C2)c(F)c1 c1(OC)cncnc1N(C)C(C1CCN(C(=O)C(n2ccc(C)n2)C)CC1)C C1(CNC(CN(CCOCC)C)=O)CCCC(NC(=O)COC(C)(C)C)C1 C1(NC(c2ccc(-c3ccccn3)o2)=O)CCC12CN(C(=O)CC1OCCO1)C2 c1(C(=O)NCC2(OCC)CN(C(=O)C=Cc3ccccn3)C2)cc(C#N)c[nH]1 C1(C(N(CCCNC(CS(CC)=O)=O)C)=O)CCc2nc(C3CC3)ncc2C1 C(=O)(CC(C)C(C)(C)C)N1CC(NC(CCCOCCC)=O)C(n2ccnn2)C1 C(N=c1[nH]c(CC(=O)Nc2ccccc2C#N)cs1)c1ccc(CN(C)C)nc1 c1(C(=O)NC2CC3CN(C(CCN(C(C)=O)C)=O)CC32)cccc2ncnn12 C1(NC(c2c(C)nccc2)=O)CC2CCC1N2C(C1(C(C)(C)C)CCCCC1)=O c1(OC)cc(C(=O)NC2CN(C(=O)Cc3nc[nH]n3)CC2C)cnc1Cl C1(CC)CN(C(c2cc[nH]c2C2CC2)=O)CCN1C(C1CCC(=O)N1)=O N1(C(=O)CCCc2ccsc2)CCC2(C1)CN(C(C13CCC(F)C1CC3)=O)C2 C(=O)(C(F)CCC(C)(C)C)NCC(C(=O)NC(C)C1CC1)CC1CC1 C1(CCNC(C(C2N(C(Cn3ccc(C)c3)=O)CCC2)(C)C)=O)CCCCCC1 C(CS(=O)(=O)NCc1cc(OC(F)F)ns1)(C1CC1)OC C(N=c1[nH]c(=NCC2SCCS2)[nH]c2cccnc12)c1nnc(C)n1C C12(C(N(CCC(C)NC(c3ccn(C(C)C)n3)=O)C)=O)C3C4C1C1C2C3C41C N(C1c2ccccc2CC1NC(=O)Cc1cnoc1)C(C(C)c1ccsn1)=O c1(CC(N2C(C)CCC(NC(=O)C(F)(F)F)C2)=O)ccc(Br)c(C#N)c1 O=C(C1=COCCC1)NC1CCN(C(=O)CCOc2ccccc2)CC1F N1(C(CCc2[nH]c(=N)sc2)=O)CCN(C(=O)CC2CC2)C(c2ccc(F)cc2)C1 C(=O)(C(C)(C)CNC(=O)Cn1cc(Cl)cn1)NC1C(OC)COC1 CC1CC(C)(C(N2CC3CC(NC(=O)CSCCN(C)C)C2C3)=O)CC(C)O1 C1(CNC(C(C(C)C)NC(=O)OCC)=O)CCN(C(c2ccoc2)=O)CC1C n1(CC(=O)N(CC(CC)NC(c2cc(C)sn2)=O)C)nnc2cc(C)ccc12 C1(CC(N2CCCC(NC(C3(C#N)CCC3)=O)C2)=O)CN2CCC1CC2 n1(CC(=O)NCC)cc(CCN(C(C2CCCC2C)=O)CC)nn1 C12(CCCC1)C(=O)N2.C1(F)(C(=O)OCC)CC1C(=O)NC(C)CCN1CCCC1 CC1CCC(O)C(C(=O)NCCSCC(=O)Nn2ccc(-c3ccccc3)n2)C1 C1(C(=O)N(C2C(NC(C3C(CC)N(C)CC3)=O)CCCC2)CC)CC2CCC(C1)C2 N1(C(COCCNC(C2(C)CCC(=O)N2)=O)=O)CCC(CSC)CC1 C1(C2CC2)(C(=O)NCC2(OC)CN(C(C(CC)N(C)C)=O)C2)CCOCC1 c1(C(N2CCC(OC)(CNC(C)=O)C2)=O)cc2c(Br)c(F)ccc2[nH]1 N1(C(c2cccc(NC(C)=O)c2)=O)CC(NC(c2occc2F)=O)CC(F)C1 CC(C)CS(=O)(=O)CC(=O)N1CCC(CNC(c2cc3c(ncn3C)[nH]2)=O)C1C c1(CC)cc(C)nc(NCC2(OC)CCN(C(C3CCOC3)=O)CC2)n1 C(CC1CC1)(C(=O)NC(CC1CCC1)C(=O)N1CC(OCCN(C)C)C1)OC c1(C(=O)NCCC(C)N(C(c2c(CC)ccs2)=O)C)ccc(C(C)C)c(C)c1 c1(C(N(CCN(C(CCC(=O)NC)=O)C)C)=O)nc(C(C)C)ncc1Cl CCS(=O)c1ccccc1C(=O)NCCC(=O)C(C)n1cncn1.C(CCSC)O C(C(C(=O)NC(C)CN(C(=O)Cn1nnnc1C1CC1)C1CC1)NC(C)=O)OC C1(C(=O)NNC(C2CC3CCCC(C2)N3)=O)CCOCC12CCC2 C(=O)(C1=C(COC)N(C2CC2)C(=O)NC1c1cc(I)c(Br)cn1)OCC C(C1CCOCC1)=CC(=O)NCC(CC=C)NC(c1cc(C)nn1CC)=O N1(C(c2n(C)nc(C)c2Cl)=O)CCC(C)(C)C(NC(=O)C=CS(C)(=O)=O)C1 N1(C(c2c(C(C)=O)ccs2)=O)CCCC(C)(NC(=O)COCc2cccnc2)C1 c1(OCC)ccc(C(N2CCCCC2CN(C(C)C(N)=O)C)=O)cc1OC C1(NC(CC2(CSC)CC2)=O)CCCCC1NC(C1CCCN1C(C)=O)=O CCCC(CCCNC(=O)C(C1CCC1)OC)NC(=O)C=CC=C(Cl)Cl C(=O)(N=c1c(Br)c[nH]cc1Br)c1nc(-c2ccc(CC)cc2O)c(F)cc1 C1(C(=O)NC(CCC=C)C2CC2)CC2(CCN1C(c1ccc(CC)o1)=O)CC2 C#CC1(C(=O)NCC(C)(C)CN2CCCC2)CCN(C(=O)C(C(C)C)SC)CC1 CC1CN(C(c2ccco2)=O)CC2(CCN(C(=O)C(C)NC(C3CCC3)=O)C2)O1 C(CC1=CCN(C(c2ccc(Cl)s2)=O)CC1)NC(C1OCC(C)C1)=O c1(OC)cc(C)c(C2CCN2C(=O)Cc2cncs2)cc1OC N1(C(c2cnc(OC)o2)=O)CCc2cc(C(N3CCCC(O)C3C)=O)ccc2C1 CN1CCC(C(N2CCC(C(C)(C)C(=O)NCCC3OC(=O)NC3=O)C2)=O)CC1 N1(C(C2N(C(C)=O)CCC2)=O)CCC2C(C1)CN2C(=O)Cn1nnnc1C1CC1 N1(C(C(CC)C)=O)CCc2ccccc2C(NC(C2Cc3ccncc3C2)=O)C1 CCC(CC)(C(=O)N(C1CCN(C(=O)COC2CC2)CC12CC2)C)c1ccccc1 c1(CNc2c(C(N3CCC(OCC)C3)=O)[nH]cc2)ccc(NC(=O)C2CC2)nc1 Cc1cn2cccc(C(=O)NC(C)CNC(c3ccc4c(c3)N(C)CC4)=O)c2n1 c1(CCCC(=O)NCCNC(=O)CC2CCC3CC23)ccc2c(c1)CCO2 c1(NCC2(SCCC=C)CC2)[nH]c(=NCC2CCO2)nc2c1ncn2C N1(C(c2ccc(COC)cc2OC)=O)CCC2(CC1)CN(CC#C)C2C(F)(F)F c1(Cc2c(C)cco2)nc(-c2nccs2)nn1-c1ccc(Br)cc1 c1(OC)ccc(CC(C)C(=O)NC(c2conc2C)C)cc1OC CC1CCC(=O)CC1.N1(C(c2ccc(C(=O)NOCC)o2)=O)CC(N=[N+]=[N-])C1 C#Cc1cnc(NC(C2CC23CCN(C(=O)CC2CCCC2)C3)=O)cn1 c1(CC(=O)NCC(=O)NC(C)C(=O)NCC=CCC2CC2)ccn(C)c1 Cc1cc(C2CC2)ncc1C(=O)NC(C)CCNC(=O)Cc1csc(Cl)n1 C1(NC(CS(C)(=O)=O)=O)CC2(C1)CN(C(=O)Cn1ncc(Br)n1)C2 C(CO)(CCCCNC(c1ccc(=O)oc1)=O)NC(C1OCCN(C)C1)=O CCCCCC(O)C(=O)NCC1(O)CCN(C(c2cc([N+](=O)[O-])sn2)=O)C1 c1(C(=O)NC2CC(O)(CNC(C3CCCC3F)=O)C2)ccc2n[nH]cc2c1 C1(NC(C(CC=C)NC(=O)C=C(C)C(C)C)=O)CC2C=CCC(C1)C2 CCC(C(=O)N1CCOCC1CC(=O)Nc1csnc1OC)C(C)(C)CC c1(NC(=O)NCC(c2ccccc2OC(F)(F)F)O)ccc(C(=O)O)cc1 C(=O)(CS(=O)c1ccc(Cl)cc1)NC1CN(C(C2CC(C)(O)C2)=O)CC12CC2 c1(C(=O)NC2(CNC(C(CCC)(C)O)=O)CCOC2)ccc(C)c(OC)c1F C1(C(=O)N(CCCNC(C2(C)CCOC2)=O)C)(COC)CCOC1 N1(C(C2(C(=O)OC)CC2)=O)CCC(CCNC(C2CC2C(N)=O)=O)C1 c1(OCC)ncc(C(N2CC(NC(c3ccoc3)=O)C(O)C2)=O)cn1 C1(C(=O)NCC23C(CN(C(C(COC)(C)C)=O)C2)CC3)CCC2(CC1)CC(O)C2 Cn1nccc1C(C(=O)NC1CCC1O)NC(=O)CC1(N(C)C)CCC1 C(=O)(CCC(C)(C)OC)N(CC(=O)NCC(F)C1CCC1)CC CCCC(C(O)C(=O)N1CC(CO)CC(C)(C)C1)NC(=O)C(CC(C)C)OC C1(C(N(C2CC(NC(=O)C(F)C3CC3)C2)C)=O)Cc2nocc2C1 N1(C(C2(CC)CC2(F)F)=O)CCN(C(c2cc(C#N)c(Cl)s2)=O)C(C2CC2)C1 C(=O)(C(F)CC(C)(C)NC(=O)Cc1cc[nH]n1)NC(CCC)(C)CC C1(C(C)C)CN(C(=O)C(CNC(=O)CCn2ccnc2)CC2CC2)CC(=O)N1 C(=O)(C(C(C)(C)C)NC(N)=O)NCCN(CC(C)O)C(c1c(C)ocn1)=O N1(C(COCCC(C)C)=O)CCOC(CNC(=O)COC2CCOC2)C1 c1(CNC(C2CC23CCN(Cc2ncccc2F)C3)=O)cc(O)nc(Cl)c1 c1(C(CC)C(=O)OC)nc(C(C)OC)nn1-c1cccc(OC)c1.C(C)NCC C1(C(=O)NC(C)C(C)NC(c2cc(=N)[nH]c(Cl)n2)=O)CC12CCSCC2 C(C)(C)(C(C)CC(=O)N(C(C)CN(C)C(C)=O)C)NC(c1c(C)cc(C)o1)=O C1(NC(C=NOC)=O)CCC(C)(CNC(=O)C(C)N(C)C)CC1 C12(C(=O)NC(CNC(C3N(C)CC(F)C3)=O)C3CCC3)CCOC(C)(C1)C2 C=CC(C)(O)CC(=O)NCC(CC1CCCC1)C(=O)NCCC1CCOCC1 N#Cc1csc(C(N2CCN(CC3CN(C(c4cccc(I)c4)=O)C3)CC2)=O)c1 C12(C(=O)OCC)CC(N)CC1CN(C(c1nncn1C1CC1)=O)C2 C(C(CC(C)C)NC(=O)C(F)(F)c1cnn(C(C)C)c1)NC(c1ccc(C)s1)=O C(CN=c1nc(N2CCC(CC3CCC3)C2)c2sccc2[nH]1)C1(C)CCC(=O)N1 CC1CCNCCC1N(c1ccc(F)nc1)C(C1(c2cccc(Cl)c2)CC1)=O C(=O)(C#CC(C)(C)O)NC1CC(CNC(C(C(C)C)OC)=O)C1(C)C C1(CC(=O)N(CC(CC)NC(=O)CN2CCOC2=O)CC)CCOC1(C)C c1(C(=O)NC(CN(C(C2(C(C)C)CCC2)=O)C)C)csc2c1C(C)(C)CCC2 C(=O)(CS(=O)(=O)CCO)N1C(C(C)(C)NC(C(C)SCC)=O)CCC1 C(=O)(N1CCCc2ccnn21)c1c(CNC(C2(C)C(C)CCC2)=O)cco1 C(=O)(C(C)(C)C(C)NC(C1CCC2(CC1)CC2)=O)N(CCC)C C12CCCC(C1)NC1CCN(C1)C2=O.C(CCC(=O)NC1COC1)=CC C1(C(N2CCC(N(CCC)C(C34CCC3CC4)=O)C2)=O)CCCC2(CCC2)O1 C12(CCC1)C(=O)N2.c1(CCNC(C=CCC)=O)cc[nH]n1 c1(C(N(C)CC2CCN(C(c3ccc(C(C)C)s3)=O)C2)=O)cc2occc2s1 C1(C(=O)OC(CNC(Cc2cc(C)no2)=O)=O)CCCC(C)CC1 c1(C(=O)NC(C2CCCC2)CNC(C2CC2C(F)(F)F)=O)ncn2c1CCC2 C1(C2(NC(=O)CCC=CBr)CC2)(C(=O)OC)CCC1 c1(C(=O)NC2CC(N(C(C(C)SCCCC)=O)C)C2)cnn2c1OCC(C)(C)C2 O=C(C1=CS(=O)(=O)c2ccccc21)NCC1CCCC(NC(C2(O)CC2)=O)C1 C1(CNC(Cn2ncc(C)c2)=O)CC2CN(C(c3c[nH]c(=N)nc3C)=O)CC12 c1(CC(=O)N(CCNC(C2CCOC2COC)=O)CC)cncc(F)c1 CC1CC2(CC(C(=O)NC(CC(=O)NCCC3CCCOC3)C(C)C)C2)C1 N12CCC(C1C1CC1)C2=O.C1(CC)(CC)CC(NC(=O)CCc2ccco2)C1 N1(C(C2N(C(c3ccc(C#C)nc3)=O)CC(F)(F)C2)=O)CC2(CCOC(=O)N2)C1 c1(-c2nnc(SC3C=CCN(Cc4ccc(OC)cc4)C3)o2)ccc(C)c(Br)c1 CC#CCCCC(=O)NCC=CCC(=O)NCC(O)C1CC1 C1(NC(Cc2cn(C(C)C)nc2)=O)CN(C(=O)CCc2ccc[nH]2)CCC1CO c1(C(=O)NC2C(CNC(c3cnn(C)c3Cl)=O)C2)cc(Cl)cc(F)c1N c1(OC)ccc(C)c(C(=O)NCC(C2CCCC2)NC(=O)CC(CC)SC)c1 c1(OC)ccccc1C=CC(=O)NCC1CC(NC(c2ccnn2C(C)C)=O)C1 O=C1CN(C(=O)C2=CS(=O)CCC2)C2CCN(C(=O)Cc3c[nH]nc3O)CC2N1 C1(C(C)NC(=O)C(C)n2cncn2)CCCN1C(=O)Cc1cnsc1 CCCC(CNC(=O)Cc1cncs1)C(=O)NCC1(O)CC(O)C1 C1(C(N(C2CC(O)C2(C)C)C)=O)CNCC(O)C1.c1(C)ccccc1 CCC(C(=O)NC1CC2CC(C1)CN(C(C1(OC(C)=O)CC1)=O)C2)C(C)(C)CC c1(C(N2CCCC2CNC(C2(OC)CC2)=O)=O)ccncc1Br.C(C)(=O)N C(=O)(C1CCCc2sccc21)N1CC(C)CN(C(c2cccc(C)c2Cl)=O)C(C)C1 C(=O)(CC#Cc1ccc(Cl)cc1)NC1C(C(C)C)NCC1 N1(C(CC2C=NN(C)C2=O)=O)CCCC(C2(NC(c3ccc[n+]([O-])c3)=O)CC2)C1 C1(CCCC)CN(C(c2cc3n(n2)CCC3)=O)CCN1C(c1cnc(C)nc1)=O C1(CC=C)(NC(C2CCOC2)=O)CCCN(C(=O)CC=CC)C1 C(C(CC(C)C)C(=O)N1CCCC(C(C)(C)C(=O)NCc2nc(C)cs2)C1)OC N1(C(c2c(C)onc2)=O)CC(C)C(NC(=O)CCC2CCC(=O)NC2)C(C)C1 n1(C(C)C)ncc(C(N2CCCC2CN(C)C(c2ccn(C3CC3)n2)=O)=O)c1Cl CC(C)CCC(=O)N1CCN(C(CNC(C2(Br)CC2)=O)C(F)F)CC1 CC1(C)CCC(N(C)C(C2(NC(C3C=CCS3)=O)CCC(C)(C)C2)=O)CC1 C(N=c1ccn2nccc2[nH]1)C1CN(C(CCC2CCC(C)O2)=O)C1 C1(OC)(CNC(=O)C(O)CN(C)C)CCN(C(=O)CSCc2ccc(Cl)s2)C1 C#CCCCCC(=O)NCC1CCC(NC(C2(O)CCCC2)=O)C1 CCC(C(=O)NCC(C)(CC)C(=O)N1CCOC(CC)C1)C(F)(F)F c1(C(N(CCN(C(C2CCN(C(C(C)C)=O)CC2)=O)C)C)=O)ccc(O)c(F)c1F c1(OC)cc2c(cn1)N(C(C1CC1c1ccccc1Br)=O)CC2 N1(C(c2c(CC)c(CC)c(C)[nH]2)=O)CCCC(N=c2ncc3cc(F)cc(Br)c3[nH]2)C1 c1(C(C(F)(F)F)OC(C(c2ccc(Cl)cc2)(C)O)=O)ncc(Br)cn1 N1(C(CCC=CC(C)C)=O)CCN(C(=O)C2=CCCCC2)CC1CC1CC1 C(=O)(C#CC1CCCCO1)NCC1CN(C(C(n2c(C)ccn2)C)=O)CC1C c1(C(=O)NCC2(O)CCCN(C(=O)C=CCF)C2)cc2nccnc2[nH]1 C(CCCC(=O)NCC12CC1CN(C(c1cccn1C1CCCC1)=O)C2)N(C)C CC1CCCC(C)N(C(C2CC=CCC2NC(C2COC(=O)N2)=O)=O)C1 N1(C(CC(C)C(F)F)=O)CC2CCC1C(CNC(C1CCC(F)(F)C1)=O)C2 C[Si]1(C)CCCCN(C(C2N(C(=O)CSc3cccnc3)CC23CCCC3)=O)C1 Cc1cccc(-c2cccc(NC(=O)NCC3CC3N3CC(C)C3)c2)c1 c1(C(=O)NC2CC(CNC(=O)CNc3ncccn3)C2)ccc(F)c(O)c1 C1(CC)CN(C(c2cnccn2)=O)CCC1NC(c1cc(O)nc(O)n1)=O N(C(=NCc1cnnn1C)NCC1C(C)(C)C1(C)C)C(c1cccs1)C c1(N(CCCNC2CCCCO2)C)nc(=N)nc(N2CC3CCC(C2)O3)[nH]1 c1(C(N(C2CCCN(C(C3(CO)CCCCO3)=O)C2)CC)=O)cc2occc2[nH]1 CN1N=C(C(=O)NCC(C)(C)OCCNC(=O)CCCCC2CC2)CCC1=O c1(CCOCCCOC(C(C)(C)C2CCCO2)=O)c(Cl)cccc1Cl N1(C(C(c2ccc(OC)cc2)O)=O)CC=C(CNC(C2CC2C(C)O)=O)CC1 CC1CC(CNC(C2(C)CCCCCC2)=O)CCN1C(c1cnc(C(N)=O)s1)=O Cc1cc(CNC(C2CCC(n3cc(CCCCCO)nn3)C2)=O)cnc1O C1(CC(N2C(CCNC(c3c(CC)cno3)=O)CCC2)=O)CCCC12CC2 c1(C(=O)NC2CC(C)(C)N(C(=O)CC#N)C2)occ2c1CCOC2 C1(NC(CCCC#C)=O)CC2CCC1N(C(=O)CCc1cnoc1)C2 c1(C(=O)OC)cc(CC(=O)NCCN(C(=O)C(n2cnnn2)C)C)ccn1 C12=CC(=NCCNC1=O)NC(C)=N2.c1(C(C(=O)OC)F)ccccc1 O=C(C1=CCC(NC(C2CC3CCCC3C2)=O)C1)NCC1COC(=O)N1 Cn1ccc(C(=O)NCCOCC(=O)NCC2COC(CC3CC3)C2)n1 CC1(C2CC2C(=O)NC2CCC(CNC(c3cccc(F)c3)=O)CC2)COC1 CCC(C)(COC)C(=O)NC1CN(C(c2nccc(C(F)(F)F)n2)=O)CC1SC C=CCCCCCCC(=O)N(C1CN(C(=O)C(C2CCOCC2)C)CC1(C)C)C C1(CNC(C2C(CC)OCC2)=O)CCCCN1C(c1ccc(Br)o1)=O C(CCC(=O)NCCN(C1CCCCC1)C(C1(C)CC12CC2)=O)OCCOC C1(C(=O)NC(c2nccs2)C)CCN(C(=O)c2cc3n(n2)CCC3)O1 N1(C(CN(N2CCC2C)C)=O)CCC(SCCOC)C12CC2.C(C)(C)(C)OC=O Cc1cc(OCCC(=O)NCC2CCN2C(C2COC(=O)O2)=O)cc(C)c1 C=C=CC(C)C(=O)NC(C1(C(=O)NC(C)CO)CC1)C c1(C(C)NC(CN(C(C)C)C(C2CCC2C(C)(C)C)=O)=O)ccncn1 c1(CN2C(CC(C)C)C(=O)NCC2)cc(=O)n2nccc2[nH]1 C#CC1(C(=O)N(CCC(=O)NC(C)(C)C)CC)CN(C(=O)C(O)CCSC)C1 Cc1nc(N(C)CCN(C)C(c2ccnc(CO)c2)=O)c2cnn(C)c2n1 c1(C(N(C2CCCC(NC(CC(C)C)=O)C2)C)=O)ccn(C)c(=O)c1 C1(N)COCC(C)(C)C1.C(C(C)(C)C(=O)N1CC2(C1)CC(=O)N2C1CC1)OC C1(OC)CN(C(=O)CN2CCCC2=O)CC1C(=O)NC(c1cnn(C)c1)(C)C C1(CNC(Cn2c(C)ncc2)=O)CCC12CCN(C(=O)C(C1CC1)C1CC1)CC2 c1(C(CC)NC(N2CCCC(N(C)C)CC2)=O)nc2ccccc2[nH]1 N1(c2cc(SC)ncn2)CC2(C)CN(C(c3cccc(F)c3)=O)CC2(C)C1 n1(CCCC(=O)NCCN(C(=O)Cn2ccnn2)CC2CCCC2)ccccc1=O c1(C(=O)NCC(CN(C(c2c(CC)c[nH]n2)=O)C)C)cc(Cl)cnn1 CC1C(NC(c2ccncc2C2CC2)=O)CC2CCC1N2C(=O)CC1CC1(Cl)Cl CCCCCCCC(=O)N1CCCC(NC(c2cncc(OCC(F)F)c2)=O)C1 c1(C(=O)NC2(CNC(C3CCC(C)(C)O3)=O)CCCCC2)cnc2[nH]cnc2c1 Cc1nc(NC(C2CCN(C(C3CN(C(C)C)C3)=O)C2)C)c(C)c(C)n1 Cc1cc(-c2cnc(CNC(c3ccc(F)cc3Cl)=O)nc2)cnc1F c1(C(C(N2CC(N(C(CC3C(CC)C3(F)F)=O)CCO)C2)=O)O)cn(C)nc1C CN1CCN(C(=O)CC2CC(F)(F)C2)C(CNC(=O)COC2CCC2)C1 C1(F)(C(=O)NC(c2ncnn2C)CC)CCCN(C(=O)C2=C(C)CC2)C1 CCC(CC(=O)NCC(C1CCCC1)NC(=O)CCC1NC(=O)NC1=O)C(C)C C(=O)(C#CC(C)(C)C)N1CCC(CC)C1CNC(c1ncn2c1CCC2)=O N1(C(CN(S(C)(=O)=O)C)=O)CCC(CCNC(C2NC3CCC2C3)=O)CC1 CC(CC(=O)N1CC(C(=O)NC2(c3ccccc3F)CC2)C2CC12)C(F)F C1(CC(=O)NCCN(C(=O)Cc2ccc(C(C)C)cc2)CC)CCOC1(C)C C1(NC(C2CCc3c[nH]nc3C2)=O)CC2CN(C(=O)CCn3cnnn3)CC2C1 C1(C(=O)NCCC(C)O)(CO)CCN(C(=O)CCc2ncccn2)C1 c1(C(=O)NCC2(CNC(C=CSC)=O)CCC2)cnc2cc(O)ccc2c1 C1(NC(c2c(C)cc(N)cc2)=O)CCN(C(C2CC(O)C2)=O)CC12CCC2 CCC(C)(C)C(O)C(=O)NCCC1=CCN(C(=O)CCC2CCC(=O)NC2)CC1 C1(CNC(CCCSC(C)(C)C)=O)C=CCN1C(=O)CCn1cnnn1 c1(CN2CCC(Nc3cc(C(=O)OC)ncn3)CC2)cc2c(SC)cccc2s1 CN1C(=O)Cc2ccc(NC(N3C4CCCC(O)C3CC4)=O)cc21 CC1C2CCC(C2)C1C(=O)NCC(O)CC(=O)NCCc1cnn[nH]1 CC1(C(=O)NC23CCC(NC(c4ccc(F)cc4)=O)(CC2)C3)CCCCNC1=O CCC1=NOC(C(=O)N(C2(C(=O)NC(c3ccncn3)C)CC2)C)C1 c1(C(C(=O)NC(CC)C)N(CCc2ccccc2)CC)cc2cccc(OC)c2o1 CC(=O)CCCCC(=O)NCC(O)CCNC(c1cn(CC(N)=O)nn1)=O N1(C(C2(C=C)CCC2)=O)CCCC(N(C)C(C2CCC(CCC)CC2)=O)C1 c1(OC)cccc(C(=O)NCC2CCCN(C(C3C(C)OC(C)C3C)=O)CC2)c1C C1(CCC)CN(C(c2ccc(N)cn2)=O)CCN1C(c1cn(C2CC2)nc1C)=O C12(C(N3CC(CC)(OC)C3)=O)CC(C)(CN1C(C1CN(C3COC3)C1)=O)C2 C1(C(C(=O)N(CC(C)NC(Cn2c(CC)ncc2)=O)CC)C)CCC(C)(C)CC1 C1(C(=O)NC(CC=C)CNC(c2ccon2)=O)CCCCN1C(C)=O C1(CNC(C(=O)NCCNC(C2CCN2C2CCCC2)=O)=O)CCCCCC1 CC1(C)CCN(C(=O)CC2CCSC2)C1CNC(C1CC(=O)NC(=O)C1)=O N1(C(C=CCC)=O)CCCC(C)C1CCNC(c1cncc(C(N)=O)c1)=O N12CCC(CC1(C)C)N(C(=O)CCOC1CCOC1)C2=O.C1(OC)CC(CC)C1 S(=O)(=O)(c1ccc(=NCCCNc2c(C)csc2C)[nH]c1)NCC Cc1c(C(N2CCCC(NC(C3(C)CCCN3C)=O)C2C)=O)cnc2ncnn12 c1(C(=O)NCC(CC)NC(c2cccc(C)c2)=O)nc2n(c1C(C)C)CCCC2 CC1CCN(C(=O)COc2cccc(N)c2)CC1CNC(c1cccs1)=O C1(CCNC(C2(CC#C)CCCC2)=O)CN(C(c2cccc(NC)n2)=O)CC1C c1(C(=O)NCCC(CNC(c2c(C)c[nH]n2)=O)O)nnc(O)cc1O c1(OC)cn(CC(=O)NC2(C)CCN(C(C3(Cl)CC34CCC4)=O)C2)c(C)cc1=O Cc1cc(CCCNC(C2(C(C)C)CCN(C(=O)CCCC#N)C2)=O)nn1C N1(C(N2CC(CSC)C2)=O)CCn2nccc2C12CCNC2 N1(C(C(CC(C)C)F)=O)CCCN(C(=O)CNC(N)=O)C(C)C1 N1(C(c2c(C)noc2C2CC2)=O)CCCC2(CC(NC(=O)C(C)SC3CC3)C2)C1 N1(C(c2ccn(CC)c(=O)c2)=O)CCC(CNC(=O)CCOC(C)C)C(F)(F)C1 N1(C(C(n2cc(-c3cc(C)cc(N)c3)nn2)C)=O)Cc2cccc(Cl)c2C1.C(=O)(CO)N C1(CC(=O)N(C)CCOC(C)(C)C)CCCC1.C(CC(=O)NCC(=O)N)SCC c1(C(=O)Nc2cnc3n2CCCC3)noc2c1CN(C(C1CC1(F)Cl)=O)CC2 N1(C(c2ncc(OC)cn2)=O)CCC2CN(C(C3(C)CCN(C)CC3)=O)CC2C1 C(=O)(C(C)C(F)(F)F)N(C1CCN(C(C2(F)CCC(=O)N2)=O)CC1)CC N1(C(CC2C(C)CCO2)=O)CCC2(C1)CN(C(=O)CCC1(C)CCC(=O)N1)C2 CN=c1cc(OC)cc[nH]1.C1(O)(C2CNC2=O)CCN(C(=O)COc2cccnc2)C1 c1(C(N2CC(N3CCN(C(C4OCCO4)=O)CC3)C2)=O)c(F)cccc1Br C(=O)(C(C)(F)C(C)(C)F)N1CCCC(CN(C(C(CCC)NC(N)=O)=O)CC)C1 CC1CCN(CC(=O)NC(C(=O)NCCCS(C)(=O)=O)c2cccs2)CC1 Cc1cc(F)c(C(N2CCOC(C(C)NC(=O)CCCC(F)F)C2)=O)c(Cl)c1 C1(C2CC2)(CNC(c2ncc(C)nc2)=O)CCN(C(=O)CCCC2CC2)C1 C(=O)(C(C)CC(C)(C)C)N(CCCNC(C1(OC)CCS(=O)(=O)C1)=O)CC Nc1cc(C(=O)NC23CCC(NC(=O)C=CCOCC(F)(F)F)(CC2)C3)cc(F)c1 C1(CNC(=O)C(N2CCCC2c2ccc(Cl)cc2Cl)=O)CCC2(CCOCC2)C1 c1(NC(CCC)=O)cccc(N2CCN(C(C3(CC)CCNCC3)=O)CC2)c1 CCCC(CC(=O)OC(CN1C(C)CCCC1C)CC)OC(=O)NC.c1(CC)ccccc1 C1(C(=O)NCC2(CCC)CC2)C2CCCOC12.C12CCCC1CC(=O)N2 CC(CS(C)(=O)=O)C(=O)NC1CCN(c2nc(C(C)(C)C)ns2)C12CCC2 C1(C(=O)NCCOC2CN(C(=O)CCC3CCOC3)C2)CCCC2C1C2(F)F Cc1nc(N2CC(CNC(C3CCCO3)=O)CC2C)cc(C(C)C)n1 c1(C(N(CC(C)(C)NC(c2ncc(CC)cn2)=O)C)=O)cccc2cnsc12 CC(C)CC(C(=O)NC(c1ccn(C)n1)C)NC(c1ccc(C#N)[nH]1)=O N1(C(C=CC(=O)N(C)C)=O)C2CCC1C(C(N1CCCCC1c1cccnc1)=O)C2 c1(CC)ccc2cc(C(=O)NCC34CCC(C3)N(C(=O)C(C)CC)C4)[nH]c2c1 C(CCCCC(=O)NCc1cccc(OC)c1)N(C(C(C=C=C)C)=O)C C1(NC(c2c(C)ncnc2)=O)CCN(C(c2sccc2F)=O)CC1C(C)C C#Cc1cccc(C(=O)NC(CCF)C(=O)NCC(C)OCC=C)c1 C=CCC(CC(F)F)C(=O)N1CCN(C(c2cnc(CO)nc2C)=O)C2(CC2)C1 c1(NC(C(C)N(CCC)C(c2ncccn2)=O)=O)cccc(F)c1O C1(NC(CCCNC(=O)OCC)=O)CC(C)N(C(c2ncncc2F)=O)C1 c1(C(=O)NC2C(NC(c3[nH]nnc3C3CC3)=O)CCCC2)cccc2cc[nH]c12 c1(CN2CC(CNC(C(C=C)(C)O)=O)N(C)CC2)cc(=O)n(C)c(=O)n1C N1(C(c2ncc(C)s2)C(=O)NC)CCC(n2cc(Cl)cn2)CC1 c1(C(=O)NCC(C2CCC2)NC(C2CCCOCC2)=O)ccn2c1CCCC2 C1(C)(NC(C(CCSC)NC=O)=O)CCN(C(c2ccc(Cl)c(N)c2)=O)CC1 CON=C(C(=O)NCC1CCN(C(c2cc(C)c(C)c(N)c2)=O)C1)c1ccco1 N1(C(CC2(OC)CC2)=O)C(C)CC2CN(C(C3OCCC3C(C)C)=O)CC12 c1(C(=O)NC2CCC(C)(NC(C)=O)C2)cccc(CO)n1 C#CCC(CC(F)F)C(=O)NCC(C)N(C)C(c1ncn2c1CCC2)=O C1(C)(C(N(CCC(=O)N(CCCN(C)C2CC2)N)C)=O)CC(=O)N(C)C1.C(=O)(C(C)OC)OC.CC C1(C(=O)O)(COCCC(=O)NC(C2CCCCCC2)C2CC2)CCCCO1 C(=O)(CC(O)C(C)C)N1CCC(F)(CNC(C2(CCC=C)CC2)=O)C1 C1(NC(c2occ(C)c2C)=O)CCN(C(=O)C(C)N2CCC2)CC1CO c1(CN2CC3N(C(c4cnc(OCC)nc4)=O)C3C2)ccc2cc[nH]c2n1 N1(c2snc(C(=O)OC)n2)CCCC2CN(C(=O)CCC3CCOC3)CCC12 c1(COCCOCCOC)cc(NC(C2CC(O)C2)=O)ccc1Cl Cc1cnc(C(=O)NCC(C)NC(C2(C)CCNC(=O)C2)=O)cc1C N1(C(C(C)c2cc[nH]n2)=O)CCC2(C1)CN(C(=O)CCC(F)(F)F)CCO2 C1(O)(CC(=O)NCC(CNC(C(C)N(C)C)=O)(C)O)CCOCC1 N1(C(C2(SCC)CC2)=O)CCC(CCC(=O)NC(C)CC2CCCCO2)CC1 c1(SC)cccc(C(=O)N(C)CC2CCN(C(=O)C=NOC)C2)c1 CC1CCCC(OCC(=O)NC2CC(O)(CNC(=O)Cn3cnnc3O)C2)C1 C=CC1CCCCN1C(c1ccc(F)cc1C)=O.C12CCCC1CONC2=O C(=O)(N=S1(=O)CCC2(C1)NC(=O)NC2=O)c1ccc(CNC(C)=O)cc1 CCC1=C(C(=O)NCC(O)CNC(c2cc(C)c(F)cn2)=O)CCCO1 C1(C(=O)NC23CC(C2)N(C(c2ccccn2)=O)C3)CCc2nnc(O)cc2C1 N1(S(CC2(C(=O)Nc3ccc(C4CC4)cc3)CCC2)(=O)=O)CC2CCC(C1)N2 C(=O)(C#CC1(C)CCCC1)NCc1ccc(CNC(C2CC(C(C)C)C2)=O)cc1 c1(C(N(C)CC2N(C(C3(C=C)CCC3)=O)CCC2)=O)cnc2[nH]ccc2n1 c1(CCC(N2CCOCC(NC(C(C)C(F)(F)F)=O)C2)=O)cnc2n1CCOC2 Cc1ccc(CC(=O)NC(C2CCCN2C(c2coc(C)c2)=O)C)nc1 C1(NC(C=C(C)C)=O)CCCC(NC(c2cc(CF)on2)=O)CC1 CCCC(C)(O)C(=O)N1CC(F)(C(=O)NCCCc2cnn[nH]2)C1 C(=O)(C(C)S(=O)(=O)C1CCOCC1)NC(C1(C)CN(C(C)=O)C1)c1ccccc1 N1(C(c2c(C)nn[nH]2)=O)CCCC2(CNC(c3cc(C)n(C(C)(C)C)n3)=O)CC12 c1(NC(C)CC(=O)N2CC(OC3(C)CCC3)C2)ccc(C#N)cc1[N+](=O)[O-] c1(OC)ncc(F)cc1C(=O)NCC1CCCCN(C(=O)Cn2cnnc2)C1 N(C(=NCCn1ccnc1)N1CCC(Nc2ccccc2)C1)Cc1n(C)ncc1 C(=O)(C(C)(C)CSC)NC1(CO)CC(NC(CCCOC)=O)C1 c1(CC)c(C(=O)N(CC(CC)NC(=O)C(C)NC(=O)C(C)(C)C)C)cccc1C C12(NC(CN(S(N(C)C)(=O)=O)C)=O)CCCC1CN(C(C1CC3CC3C1)=O)C2 CC1(C)CCCN(C(=O)CCn2cccn2)C1CNC(C1CC12CCC2)=O C(=O)(C(CCNC(=O)CC1COCCO1)N(C)C)NCC(C1CCC1)OCC n1(CC(=O)N(C2CCCCN(C(=O)CC3CC=CC3)C2)C)cc(S(C)(=O)=O)cn1 C12(C(=O)NC(CC#CC)CO)CCCC1CCN2C(=O)CS(=O)(=O)CCOC c1(CCC(=O)NC(CCNC(c2nc(C)nn2C)=O)(C)C)cnc2ccccn12 C1(C(=O)NC(C)CN(C(=O)CSC2CC2)C)CN2CCCCC2CO1 Cc1cc(=NC(=O)CC(O)C2CCCC(O)C2)[nH]n1-c1ccc(Br)cc1 Cn1nnc(C(=O)NC2CC(CCNC(=O)CS(N)(=O)=O)C2)c1N c1(C(=O)OC)cccc2c1CCCC2NC(=O)NCC1CC1CO c1(OC)nc(C(=O)NCCCNC(C2(C)CC=CCC2)=O)sc1C C1(NC(C(Cc2ccsc2)NC=O)=O)CC2CC(NC(=O)CC3OCCO3)C1C2 c1(NC(N(c2nccc(OC)n2)C2CCCNCC2)=O)cccc(Cl)c1F C(C(N=c1ccnc[nH]1)c1ccccc1)NC(CC1N(CC)CCOC1)=O C(=O)(C(C)CC(C)(F)F)NCC(CC)NC(c1ccc(C)c(Br)c1)=O C(=O)(C1(C)Cc2c[nH]nc21)NCCCN(C(C(N1CCCCCC1)C)=O)CCO S(=O)(=O)(c1ccc(C#N)cc1)NC(C(=O)NC1CN(C(C)=O)CC12CC2)C(C)O CCCCC(O)C(=O)N1CC(CC(=O)NCC(C)(C)n2cccn2)C(C)C1 C=C(C)C1CN(C(=O)C(C)(C)C2CCN(C(c3cccn3C3CC3)=O)C2)CCO1 C1(C(N2C(C(C)C)CN(C(=O)CN3CCCCC3)CC2)=O)CCC2(CCCC2)C1 C1(C(=O)NCCC(=C)C)CCCCCC1NC(c1cc(C(C)C)[nH]n1)=O C1(CNC(C2(C=C)CC2)=O)CC2(C1)CN(C(=O)OC(C)(C)C)C2 C12(CNC(=O)NC3CCN(C(CN(C(C)C)C)C)CC3)CCCC1OCC2 N1(N2C(CCCC)CCC2)CCCCCC1C=C(C)C C(=O)(CC(C)(O)C(F)(F)F)NCC1(O)CC(NC(c2c(C)ccc(Cl)c2)=O)C1 CC1CCC(NC(c2ccc(CNC=O)cc2)=O)CO1.C1CCOCC1 c1(C(C)C)nnsc1C(=O)N(CCCN(C(=O)Cc1ccon1)C)C N1(CC)CCC2(CCC(N3CCN(CC#N)CC3)CC2)C1.C1(=O)C(C(=O)OC)O1 CCC(C)(O)C(=O)N1CCC(O)(CNC(=O)CCCc2cncs2)C1 CCCCCCCCC(C)C(=O)N1CCN(C(=O)Cc2ccns2)CC1CO CN1CC(C(N2CCN(C(c3ncccc3-n3cccn3)=O)CC2)=O)CC1=O c1(C(=O)NC2(CC=C)CN(C(=O)C(C)NC=O)C2)nccc(OC)c1F CC(C)CC(C)C(=O)N1CCOCC1CN(C)C(c1cc(F)c[nH]1)=O O=[N+]([O-])c1cc(Cl)cc(Cl)c1OC(F)F.N12CCCCC1C2 C(=O)(C(C)(C)C(N)=O)N1CC(O)(CCNCc2cc(C(=O)OC)no2)C1 C1(N(C(=O)Cc2csc(Br)c2)CC#C)CCN(C(=O)C=C(C)C)CC1 c1(CC(c2ccccc2)N(C2COC(=O)C2)CCC(=O)O)ccc(F)cc1 Cc1ccc(Cl)c(F)c1C(N1CCC1CNC(C1CCC2CC12)=O)=O c1(NC(C(CNC(C2CC(O)CN2C)=O)OC)=O)cc(C)c(F)cc1C c1(OS(CC)(=O)=O)ccc(C)c(NC(=O)C2=CCCC2C)c1 CC1CCN(CC(=O)NCC2(O)CN(Cc3cccc(Cl)c3)C2)CC1 O(NC(=O)CC(C)(C)COc1ccccc1Br)C(CC(C)C)CO C1(C(=O)NC2COC3(CNC(C4CCCO4)=O)CC2C3)CCn2c(O)nnc2C1 C1(CSCc2c(-c3ccc(F)cc3)n[nH]c2)COC2CCCC2O1 c1(C(=O)NC(C2CCCN2C(=O)CCC2CCCOC2)(C)C)n[nH]cc1Br N1(C(C(C(C)C)OC)=O)CC2(C1)CN(C(=O)C(N1CCCCCC1)C)CC2CO N1(C(C(c2cn(C)nc2)=O)=O)CC(NC(c2ocnc2C(F)F)=O)CC12CCC2 c1(C(=O)NCC2CN(C(C(C)C(F)(F)F)=O)C(C)CC2)c(N)cccc1[N+](=O)[O-] C(=O)(C(C1=C(C)C=CCC1(C)C)N(C(C)C)Cc1ccccc1C)NCCSC N1(C(c2c(C(=O)OC)cco2)=O)CC(NC(=O)Cc2ccccc2)CCC1C c1(CN2CC(=O)NCC2)cc(I)ccc1C(=O)Oc1ccc(CC(=O)N)cc1.[nH]1cccn1 C(=O)(N=c1ccn(C2CN(C(C)(C)C)C2)[nH]1)NC1(c2nccs2)CC1 N1(C(C2N(CC=C)CCC2)=O)CCC(O)C(C(N(N2CCCCC2)C)=O)C1 c1(C(C)C)cc(C(=O)NCC2(O)CN(C(=O)C(CCO)N(C)C)C2)n2ncnc2n1 c1(C(N2C(C)CCC(CNC(CCCCC#C)=O)C2)=O)n[nH]c2ccc(Cl)cc12 c1(OC)c(CN2CCOC(CO)C2c2ccnn2C)cc(C)cc1C CC1(C)CCCCC1C(=O)NC1CCCCC1NC(C1(C#N)CCC1)=O C(CN=C(NCc1nnc(CC(C)C)s1)NCC1CCCCC1C)OCC c1(C(=O)NC2CC(CNC(C3(C)N(C)CCC3)=O)C(O)C2)cc(S(C)(=O)=O)co1 C1(COC)CN(C(=O)C=Cc2nccs2)CCN1C(c1cnn(C)c1N)=O n1(CC(=O)NC(CN(C(=O)CC(C)F)CC)C)nc(C)c(C=NO)c1C CCCCC(C(=O)N(C1CCCN(C(=O)Cc2csnn2)C1)CCO)C(C)C C(CCC(N)=O)(C(=O)N1CCC1C1CCCC1)n1cc(CCN(CC)CC)nn1 N1(C(c2n(C)nc(C3CC3)c2)=O)CC2OCCN(C(=O)C3=CS(=O)(=O)CCC3)C2C1 C1(C(=O)NC2C(CNC(CN(CCC#C)C)=O)CC2)CCCCNC1=O N1(C(c2cc(OCC)n[nH]2)=O)CC(CCNC(=O)COCCF)C(C)C1 c1(C(N(CCN(C(c2ccc(OCC)c(C)c2)=O)C)C)=O)ncc2n1CCCC2 N1(C(C(CNC(C2C(CC)OCC2)=O)CC(C)C)=O)CCC2(COC(=O)N2)C1 c1(C(=O)NCCC(C)N(C)C(c2occc2F)=O)cccc2ncnc(O)c12 n1(CC(=O)N(CC(C)NC(=O)C(C)CSC)CC)cnc([N+](=O)[O-])n1 CCC(C)C(C(=O)N1CCN(C)CC1)N(C(=O)C(CN(C)C)CC)C CC(C)(C)S(=O)(=O)CC(=O)N1CCC2CN(C(c3ccc(F)cc3F)=O)C2C1 N1(C(Cc2cc(C)ns2)=O)CCC(C2CCN(C(C34CCCC3C4)=O)CC2)CC1 N1(CC=CC(N2CC(CNC(C3C(C)CC(=O)N3)=O)C2)=O)CCc2sccc2C1 c1(N2C(C)COC(C)(C)C2)ccc(Br)c(Cl)c1F CCCCCC(=O)NCC(N1CCCC1CCNC(c1cccc(NC)n1)=O)=O C1(C(=O)NC(C#CC)(C)C)CCCCN(C(=O)CCc2nncs2)C1 CCC(CC)CCC(=O)N(CCCC(=O)Nc1cc(C#N)ccc1OC)C S(=O)(=O)(c1ccc2c(c1)OCCO2)N1CCCC(CNC(CN(C)C)=O)C1 c1(C(=O)NC(CNC(c2c(CC)csc2)=O)C2CC2)cc(N(C)C)cc(C#N)c1 C12(CN(C(C3CCCO3)=O)CC)CCC(CC1)N(C(=O)CC1CCCNC1=O)C2 C(=O)(C1=CCC(C)CC1)NCC1(OC)CCN(C(=O)Cn2nc(C)cc2C)CC1 C1(CCC)CCN(C(=O)CC2(N(C(=O)C(F)=C(C)COC)C)CC2)CC1 C1(C(=O)OC)COC2(CCN(S(=O)(=O)c3cc(C(=O)OC)sc3Br)CC2)C1 c1(C(=O)NCCCC(C)(C)NC(c2c(CC)c[nH]c2)=O)cc(F)ccc1C C1(C(=O)NC(CC=C)CNC(c2ccsn2)=O)CCc2nnnn2CC1 C1(C)(C(=O)NCCC2CCN(C(C(C)NC(=O)C3CC3)=O)C2)CCCN1C C1(C(N(C(c2cccnc2)C)CC)=O)CC=CCC1C c1(C(=O)NC(CC=C)CNC(c2ccn(C)c(=O)c2)=O)cnc2onc(C)c2c1 C(=O)(C(C)(C)CC(F)F)NCCCC(C)NC(C(C(C)C)C)=O C(CCCC(=O)NC1CCC1C(=O)NC(C)C(O)C(C)C)OC C1(N(C(=O)CSCC(F)(F)F)C)CCCN(C(C2(F)CCOCC2)=O)C1 C1(NC(c2c(Cl)cn(C)n2)=O)CC2(C(N3CCOCCC3C3CC3)=O)COC1C2 CCC(C(=O)NCCCOCCC(N1CC=CC1(C)CO)=O)C(C)(C)CC C(CCC(C)(C)C(=O)NCC(CC(C)C)NC(C1C2CNC(=O)C12)=O)OC C(C)(C)C(CNC1CC1)C(=O)N1CCN(c2ncnc(O)c2F)CC1 CCC(C(=O)NCC1CC2(C1)CN(C(=O)C(c1cc(F)ccc1C)=O)C2)C(C)C C(=O)(CC(C)NC(C1CC1CNC(=O)C(C)CC1CC1)=O)OCC c1(NC(CCNC(C(C2CCCCC2)OC)=O)=O)cc(F)ccc1O CN(CCCC(=O)N1CC(NC(=O)CC(O)Cc2ccccc2)CC(C)(C)C1)N=O CN1CCC(CO)(CNC(=O)C=CCN(C)C(c2cncnc2)=O)C1 N1(C(C(CCC)O)=O)CC2(CCC(CNC(C3(n4ccnc4)CCCC3)=O)O2)C1 c1(C(=O)NCC2(COC)CCCN2C(c2coc(C)n2)=O)ccc(C)c(Cl)c1F C1(C2CCN(C(c3cscn3)=O)C2)(NC(c2c(C)cc(C)s2)=O)CC1 c12ccc(cc1)CN2NC(NCC)=NC.C1(NS(C)(=O)=O)CCN(S(C)(=O)=O)C1 CC1(CNC(=O)C2=CCOC2)CN(C(=O)Cn2cnc(C(N)=O)n2)CCO1 C1(CC)(NC(=O)CC(F)(F)F)CCCN(C(=O)COC)C1 Cc1oc(CO)cc1C(=O)NC1CC(=O)N(C2CN(C(c3cc[nH]c3C)=O)C2)C1 C1(NC(C(C)OCCN(C)C)=O)CCC12CN(C(=O)CN1CCCCCC1)C2 N1(C(C2C(NC(CCCCCC)=O)CCOC2)=O)CC2(CCC(=O)NC2)C1 c1(C(=O)NC(CNC(CCOCC#C)=O)C(C)(C)C)ccc2nc(CO)[nH]c2c1 C1(C(=O)NCC(CC)NC(C2(CC)CCC2)=O)COCCOC1 N1(c2ccc(C(=O)OCC)cn2)CCC(C)C(NC(c2ccn(C)c2)=O)C1 c1(C(=O)NCC(CCCC)NC(c2cc(C)oc2C)=O)c(C)nc2sccn12 Cc1cn(C(C)C)cc1C(=O)NC1CC(CNC(=O)CCN2CCCCC2C)C1 N1(C(Cc2nc(C)sc2)=O)CCOCC1CN(C)CC1CCC(=O)NC1 Cc1nn2c(c1CNC(=O)CCCc1cccs1)CN(C(=O)C(O)C(C)C)CC2 N1(C(C(C)(C)NC(=O)OC)=O)CCC2(CC1)CN(C(=O)CN(C)C1CC1)C2 C(C)(C)(CCCCNC(=O)CCC1CCCCC1)NC(C(CSC)C)=O C=CCC(C)(C)CC(=O)N(C)CCNC(=O)CN(C)Cc1nnc(C)n1C N1(C(CC(CC)O)=O)CCC2(CCN(C(=O)C=Cc3ccncn3)CC2)C1 C1(C(=O)NCCC(C)(C)OCC)N(C(c2c[nH]cc2C(C)C)=O)CCC1(C)C c1(C(=O)OC)ccccc1N(C(c1cn(-c2cnn(C)c2)cn1)=O)C(C)C c1(C(N2CC(NC(C3C(C(=O)OC)CC=CC3)=O)(CO)C2)=O)cc(Cl)ccc1Cl CN(OCC(F)(F)F)C(=O)C(Cc1cn[nH]c1)NC(C1CC12CC2)=O C1(C(=O)NCC2(F)CCC(NC(CCCC)=O)C2)COc2cc(F)ccc2O1 C1(NC(CCC2(NC(CC3CCCN(C)C3)=O)CCC2)=O)CCCCNC1=O N1(C(C2C(C3C(C)C3)C2)=O)C2CCC1CC(CNC(C1CC13CCOCC3)=O)C2 CC1=C(C(=O)NCC2CCN(C(C3(CCN(C)C)CC3)=O)C2)CCS1(=O)=O c1(C(=O)NCCN(C(C(CC)CC(C)C)=O)CC)cc(=O)oc2ccc(O)cc12 c1(OCCNC(C2N(C(C(CC)O)=O)CCC2)=O)ccc(Nn2cccn2)cc1 CCC(C)C(C(=O)N1CCC2(CC1)CC2)N(C)C(C1C(C)C1C)=O N1(C(C(CC(=C)C)Nc2cc(F)c[nH]2)=O)CCCN(C(=O)OC(C)(C)C)CC1C N1(C(c2c(C)nccc2)=O)CC2CC(C(N3CC(F)CC3C#N)=O)C(C2)C1 CC(C)CC(F)C(=O)N1CC(C2CCCCN2C(=O)CCCOc2cccnc2)C1 c1(N2CC3CN(C(c4ccncc4Cl)=O)CC32)ncnn2cccc12 c1(OC)ccc(C(N2CCC(C)(CNC(C3C=C(C)CS3)=O)CC2)=O)cc1N c1(C(=O)NC2(C(=O)NCCCCCC3CC3)CC(F)(F)C2)cnn2ccccc12 Cc1cc2c(C(=O)NC3CCC(NC(=O)Cn4ncnn4)C3)cccc2o1 C(=O)(C1=CCC(C)(C)CC1)NC(C1CCCN(C(=O)CSCc2cscn2)C1)C CC1CC(C(=O)NOC(CCF)CF)N1C(C1CCC1)=O c1(CN(CC(c2ccccc2)C)C(C2CC2C(C)C)=O)cnc(Br)cn1 c1(CN2CC3(CN(C(=O)CCc4cccc(Cl)c4F)C3)C2)ccc2occc2c1 N1(CC=C)CCCN(C(=O)CCN(C(c2cc(C3CC3)on2)=O)CC)CC1 Cc1cc(C)c(CNC(C2(F)CCCC2)=O)c(C)c1.N12CCCC(C1)C2 C(=O)(CN1C(=O)CCCc2sccc21)N(CC(CC)NC(c1ncn(C)n1)=O)C N1(C(C(=O)OCC)=O)CCCN(C(c2ccc(F)cc2C#N)=O)C(C)C1 N1(C(c2nc(CC)oc2C)=O)CC2CCC2(CCNC(=O)CCC#N)C1 C1(C(=O)NCCOCCn2cc(CC(=O)OC)nn2)CN2CCC1(C)CC2 C1(OC)CC(CNC(C2CC(O)C2)=O)N(C(=O)CC(F)F)C1 c1(C(N2C(CNC(c3cnc(C)[nH]3)=O)CC(C)(C)C2)=O)ccc(S(C)=O)cc1 N1(C(=O)OC(C)(C)C)CCC2(CCC2C(=O)NCC(=O)NC2CCC2)CC1 c1(OCC(N2C(C(C)NC(CC(=C)Br)=O)CCC2)=O)ccccc1C(F)F c1(C(N(C2C(N(C)C(C3CCCS3(=O)=O)=O)CCCC2)C)=O)ncn2c1CCC2 c1(NC(C(c2ccc(Cl)s2)N(CC(=O)NCC)C2CC2)=O)cccc(OC)c1 c1(OC)cc(Cl)ccc1CC(=O)NC(C)(CNC(c1ccns1)=O)CC(C)C Cc1[nH]c2c(CNC(C3OCCC3F)=O)cccc2c1C c1(NC(=O)CCC(CNC(C(C)C2CC2)=O)F)ccc(OC2CC2)cc1 C(C1=CCCOC1)N(C(=O)C(Cc1cccnc1)C1CCCC1)C(C)(C)C CC1C(=O)CCC1CC(N1CC=CC1Cn1cc(-c2cnc(C(C)(C)C)o2)nn1)=O C1(C(=O)NCCC)CC2CCN(Cc3c([N+](=O)[O-])cnn3C)CC12 C1(C(C)NC(CN(CCOC)C)=O)CCCN(C(c2ccc(C(C)F)cc2)=O)C1 C(=O)(C1SCCc2ccccc21)NCC=CCNC(=O)CC1COCCO1 C1(N(C(CCOCCNC(c2snc(C)c2N)=O)=O)C)CN2CCC1CC2 C1(C)(C(=O)NCc2onc(CC)n2)CN(C(=O)CC2(O)CCOC2)C(C)(C)C1 C1(OCC)CC(NC2CN(C(=O)Nc3nnc(O)nc3O)C2)C12CCC2 c1(CN(C(c2ccnn2CC(C)C)C(=O)NC(CC)(C)C)C2CC2)nnn(C)n1 Cc1cccc2c1ccn2CC(=O)NC1C=CCN(C(=O)C=CC(F)(F)F)C1 C1(C)(CC(=O)N(CC(CC)NC(=O)C(c2ccccc2F)C)CC)CC(F)(F)C1 C1(F)(CNC(C(C2CCOCC2)C)=O)CCN(C(c2c[nH]ccc2=O)=O)C1 N1(C(C2N(C(C)=O)CCOC2)=O)CCC(F)(F)C(CNC(c2cscn2)=O)C1 N1(C(C2(CCC)CCOC2)=O)CCN(CCCCCn2cc(COC)nn2)CC1 N1(C(c2c(Br)ccc(N)c2)=O)CCCC12CCN(C(=O)Cc1ccccc1)CC2 N1(C(CCCC=C)=O)CCN(C(c2ccc(Br)o2)=O)CC1CC N(C1c2ccccc2CC1NC(=O)CCc1nncn1C)C(C(C)C1CC1)=O C1(N(C(CCNC(C(=O)CN)CC)=O)CCN(C)C)CC(F)C1.C(C)(C)=N.CC=C Cc1cnc2ccccc2c1C(=O)NCCC(C)NC(=O)C(C)CF S(=O)(=O)(c1ccc(NCCCOc2ccccc2F)cc1Br)NCC(C)OC C1(C(C(=O)NC)N(c2c(F)ccc(OC)c2)C)CC2(C1)C(F)(F)C21CCC1 c1(C(=O)NC(CN(C(c2c[nH]c(=N)s2)=O)CC)C)sccc1C1CC1 CC1(C)CC(CNC(c2ccccc2)(C)Cc2c(F)cccc2F)OC1=O Cc1ccn2ncc(C(=O)NC(C)CC3CN(C(C4(C)CCCC4C)=O)C3)c2c1 C1(C(C)C)C(=O)NCc2cn1nn2.c1(CCC)nn[nH]n1.C(C1CC1)(C1CC1)SC N1(C(c2nccc(OC)c2)=O)CCCN(C(c2nc(C3CC3)oc2C)=O)CC1 CC(C)S(=O)(=O)C1CCN(c2nccc(-n3c(=O)oc4ccccc34)n2)C1 N1(C(C(c2ccn(C)n2)C)=O)CCC(C)(C)C1CNC(c1c(O)cccc1F)=O N1(C(CNC(c2cncs2)CC)CC(=O)NC)C(=O)c2ccccc2C1=O C1(NC(C2(O)CN(C(CNC(C3CN(c4nncs4)C3)=O)=O)C2)=O)CCCCS1 N12CCC(C(C)C1)NCC2=O.c1(CCCCCOCC#C)ccccc1Cl c1(C(N2CC3(C(NC(C(CCC)OC)=O)CC3)C2)=O)nc(O)nc(O)c1F C#CCCC1C(=O)N1.C(=O)(CCCCC=CC)NCC(C)(F)C(C)C C1(C2CN(C(C34CC(F)(C3)C4)=O)C2)(NC(c2cn(CC)nn2)=O)CC1 CC1(OCCc2c(-c3ccccc3)noc2Cc2ccccc2)CC(O)(C2CC2)C1 c1(CCC(=O)N(C2CCN(C(=O)OC(C)(C)C)CC2C)CCC)ccc(F)cc1Cl N1(C(C(CC=C)OC)=O)CCOCCC1C(N1CCC(O)C(C)C1)=O CC1CN(C)CCC1N=c1cccc(S(=O)(=O)N2CCC(OC(F)F)CC2)[nH]1 CC(C)(C(=O)NCc1cn(-c2cc(C(=O)O)cc(F)c2)nn1)S(C)(=O)=O C1(N(C)C)CCCN(C2CC2)C1.C12CCC(O1)NC2=O.C12(CCSC1)C(=O)N2 c1(C(CC#C)NC(=O)C(C)c2cccs2)ccc(OCCc2ccccc2)cc1 c1(C(N2CCC(O)(CNC(C(C)c3ccsc3)=O)C2)=O)ccc(=O)n(O)c1 c1(C(N(C)CC2CCN(C(C(N3CCOC3=O)C)=O)C2)=O)ncc(Br)cc1F C12(CNC(C(C)Cc3ccncc3)=O)CCC(CC1)NC2 C(=O)(C(CC(F)F)C1CCC1)N(CC(CNC(c1cn(CC)nc1)=O)C)C C#CCCC(C(=O)Nc1cnc(C(=O)OC)nc1)NC(C1C2CC3C(C2)C13)=O CN1CCN(C(c2cnn(C(F)F)c2)=O)CC1CNC(c1cnc(C(N)=O)s1)=O N1(C(c2cnc(C3CC3)s2)C(=O)NCCC2CC2)CCS(=O)C2(CCC2)C1 O=S(=O)(c1ccc(NCCC2CC3(CCC3)C2)c(F)c1)NC1CC2CCC(C1)C2 CC1CCNCCC1N(C(=O)CC1CCCCO1)CC1CCOCC1 C(=O)(C(C)(C)C(N)=O)NCCCN(C(=O)CN1CC2CCC1C2)CC C1(CNC(C2(CC)CC2)=O)CCN(Cc2ccc(Br)[nH]2)CC1O C1(C(N2CCCC(n3cc(SCC)nn3)C2)=O)COc2c(OCC)cccc2C1 c1(C(=O)NC(C(C)C)CNC(C2CCCCN2C(C)C)=O)ncnc2ccsc12 C1(F)(C(=O)OC)CC(C(=O)NCCCNC(=O)CC2CC(F)(F)C2)C1 C1(CNC(c2cccc(C(N)=O)c2)=O)CN(C(c2cscn2)=O)CCCO1 N1(C2CCN(c3ccc(C)cc3)C2=O)CCn2c(cc3c(Cl)cccc23)C1 c1(C(N(CCNC(=O)C(Cc2ccco2)CC)CC)=O)nccc2ncn(C)c12 c1(C(=O)NC23CC2CN(C(=O)CN2CCSCC2)C3)cnc2ccsc2c1 c1(C(=O)NC2C(NC(C(CC)n3cncn3)=O)C2)oc2ccccc2c1C CC1(C)C(C)(C(=O)NCC2(F)CCC(NC(=O)CCc3ncc[nH]3)C2)C1(C)C C=CCCCC(C(=O)NCC1(C)CCCOC1)NC(=O)Cc1c(C)noc1C c1(CNC(c2c(CC)cco2)=O)nc(C(=O)NCC(C)(C2CC2)OC)c(C)o1 N1(C(C2C(C)N(C)CC2)=O)CC(C(N2CCN(C)CC2CO)=O)C(F)(F)C1 c1(C(=O)NCC#CCNC(C2CCC(C)(CC)O2)=O)cc2ccccc2nc1O CCCCCCCC(=O)NCC1COCC1NC(c1ccc(Cl)o1)=O c1(SC)ccncc1-c1nc(-c2nccs2)nn1CCOc1ccccc1 CCCCC(C(=O)NCCn1ccc(C(=O)NC2CCCC2C#N)c1)C(C)C C1(C(=O)NC2C(NC(C3CSC3)=O)COCC2)Cc2nnsc2S1 C1(N2CCCC2C(N)=O)CNC(=O)C1.c1cc(C2CC2)nn1C.CO CN1CC(O)CC1C(=O)NCC=CCNC(c1cnc(N(C)C)nc1)=O c1(NC(C2CN(C(Cc3c(C)n[nH]c3C)=O)CC(F)C2)=O)cccnc1[N+](=O)[O-] C12(NC(c3c(C)nc(C(C)OCC)s3)=O)CCCC1N(C(C1(SC)CC1)=O)CC2 c1(C(N2CC(CC(C)NC(C3C(CC(C)C)C3)=O)C2)=O)ccoc1C(F)(F)F C1(NC(C(CN(C(CCC2(C)N=N2)=O)C2CC2)O)=O)CCCC(F)C1 C1(CCOC)CN(C(c2ncoc2C2CCCO2)=O)CCN1C(=O)CP(C)(C)=O c1(C(N2CC(C)N(C(=O)C3CC3)CCC2)=O)cn2ccc(Cl)cc2n1 CCCCC(CNC(c1cncc(-n2cccn2)n1)=O)NC(=O)C(C)N1CC(C)C1 C(=O)(C1=C(c2ccccc2)SCCO1)NC(CCNC(c1cc(C)nn1C)=O)C c1(C(=O)NC2(CO)CCN(C(CCNC(C)=O)=O)C2)cc(NC(C)=O)ccc1F O(NC(=O)C(O)CNC(=O)CC1CCCC1O)CC(CC)C Cc1cc(Br)ncc1NC(C1CCN(C(=O)C2CC2(C)C(F)F)O1)=O Cc1cnc(N(C(c2cscn2)C)C)c(S(=O)(=O)NC(CO)C2CC2)c1 N#CC1(C(=O)NC2CCC(NC(C3(C(F)F)CCCO3)=O)CC2)CCOC1 C(C)(CNC(=O)CN1CCCC1C)(CC(C)C)NC(CCc1ccc(C)o1)=O C1(NC(=O)C(CO)N(C)CC)CCN(C(C2(OC)CCCC2)=O)C1.C(=O)(OCC)N c1(C(=O)NCC(CNC(c2ncc(Br)cn2)=O)OC)cnc(O)n1C C(C(C)(C)CC(=O)NCCC1CC(NC(c2ccc(Cl)nc2OC)=O)C1)OC Cc1ccc(C(C)C(=O)NC2CC(NC(c3ncncc3Br)=O)C2)cc1 N1(C(c2nc(CC)sc2)=O)CCCN(C(c2ncnc(OC)c2OC)=O)C(C)C1 C12(NC(COCCC)=O)CCCC1N(C(=O)Cn1cc(C)cn1)CCC2 c1(C(CC)(C)C)cccc(C(=O)N(C)CCN(C)C(c2cccnc2F)=O)c1 C(CC(C(=O)N1CCC(C#N)C1)NC(=O)CCCOC)OCC C12CCC3(CC1)CC(C3)N2.C1(C(=O)NCCC)CN(C(=O)OCC)C2CC12 S(=O)(=O)(c1c[nH]ccc1=NCc1ccc(Cl)cc1)NC(CCC)(C)CO CCC(C(=O)NC(CNC(c1cccc2cnsc12)=O)C1CC1)C(F)(F)F c1(OC)ccc(CCCC(=O)NC2COCC2NC(=O)C(C)C(C)O)cc1 N1(C(C(C)SC)=O)CC2(C1)CN(CCc1ccc(NC(=O)C=COCC)cc1)C2 C1(C(=O)Nc2n[nH]cc2C2CC2)CN(C(=O)COc2cccc(O)c2)CC1CO N1(C(C(CC=C)C)=O)CC2CCC1CC2NC(=O)C(F)(F)C1(O)CCC1 c1(C(=O)NCC(=O)N(CCC(=O)NCC(=O)NCC)C)cn(C)cc1C C(CCCCC(=O)NCC(c1cncn1C)NC(=O)Cc1ccc(F)c(F)c1)OC N1(CC(CSc2c(OC)cccc2)O)Cc2c(C(=O)O)ccc(F)c2C1 N1(C(CCN(C)CC)=O)CCC2(CC1)CCN(C(=O)CC1CCC(C)O1)C2 c1(CC#C)c(C(F)(F)F)n[nH]c1C(=O)NCC1(C)CCN(C(=O)CC2CCCO2)C1 C(=O)(C1=C(F)CN(C(C2C3CCC(C)(C3)O2)=O)CC1)N(CC(C)O)C C1(CNC(C2(CS(C)(=O)=O)COC2)=O)CC2CC(C1)N(C(c1cnn(C)n1)=O)C2 C1(CC)(NC(=O)Cc2cccc(C(F)(F)F)c2)CCN(C(=O)C(N)=O)CC1 C(=O)(C(C)(C)COC1CC1)NC(c1n(CC)ccn1)Cc1ccccc1NCC C(=O)(CCCCC(C)C)NC(C(C)NC(c1n(CC)cc(Br)c1)=O)C C(=O)(C(CCCOC)NC(c1nccn1C)=O)Nc1c(CC)nsc1 c1(NC2CCN(C(C(CCC)C)=O)C(C)C2)nc(C)c(C#N)cc1Cl c1(CCCC(C)SC)nc(CCN(C)C)nn1-c1cnn(C)c1 c1(C(=O)NC(C(=O)NC(CC)(C)C(N)=O)C2(O)CCC2)cc2occc2[nH]1 O=C1NC(Cc2ccc(F)c(Cl)c2)C(=O)N1Cc1cccc(-n2cncn2)c1 C(=O)(C(C)(CO)Nc1ncccn1)NCC(N1C(CC)CC1)=O CCC(C(=O)N(CCN(C)C(c1cnn(C2CC2)c1)=O)C(C)C)OC1CCCC1 N1(c2cc(C)nc(N3CCC(C#N)CC3)n2)c2ccccc2CC(C)C1C c1(CNC(=O)NCCNC(c2ccncc2)=O)ccc(C2CC2)cn1 c1(OC)nc(C(=O)NC(c2ccc(C)cc2)CNC(=O)C(C)N(C)C)sc1C c1(C(=O)OC)ccc2c(-c3ccc(Sc4ccc(CC)c(C#N)c4)nc3)n[nH]c2c1 C1(N2C(CN(C(=O)CC3CC=CCC3)CC)CCC2)CC2CCCCC2NC1=O C1(NC(=O)C=CC(F)(F)F)CC(O)CN(C(c2cc(C3CC3)cc(F)c2)=O)C1 C1(C(N2C(C)(CCO)CC2)=O)CC2(CCN1C(c1cccs1)=O)CC2 N1(C(CC=C)=O)CCC(NC(c2ccc(NC3CCCC3)nc2)=O)CC1C CC(C)CCCC(=O)NCCC1CN(C(=O)CCCn2ccnn2)CC(C)O1 C1(C2CN(C(=O)CCCC(N)=O)C2)(NC(c2c(C(=O)OC)csc2)=O)CC1 C(=O)(C(C(C)(C)C)n1ccnn1)N(CC(CNC(CN1CCC(C)CC1)=O)C)C c1(C(c2cn(C3CCN(C(=O)CC4CCC4)CC3)nn2)=O)ncc(Cl)cc1O C=C(C)CC(C)C(=O)N(C1CCN(C(c2oc(C)nc2CC)=O)C1)CCO c1(OCC(N2CC(CS(N)(=O)=O)C2)=O)ccc([N+](=O)[O-])c(F)c1 C1(NC(COCCOCC#C)=O)CCCC1NC(=O)Cn1cc(CO)nn1 C1(N(C(C)(C)C(=O)NCC)C(C)(C)CC)CC2CNC1C2 N1(C(=O)OC(C)(C)C)CCC(C2(C(=O)NC3C4COCC34)CCOCC2)CC1 C1(C(=O)NC2C(NC(Cc3c(C)non3)=O)CCC2)Cc2ccccc2S1(=O)=O c1(C(N2CCC(NC(CC3(C)CCC3)=O)C2)=O)cccc2ncsc12 N1(C(CCSCCCC)=O)CCC(C)C(NC(=O)CCCCCN(C)C)C1 c1(N(CC(F)F)C)nc(=NCCc2ccsc2Cl)[nH]c2c1CCCCC2 c1(C(=O)OC)cccc2c1CCC2NC(=O)Nc1c(I)ccnc1OC c1(C(=O)OCC)cc(=NCC2CN(C(c3coc(Cl)n3)=O)CC23COC3)[nH]cc1C C1(NC(Cn2nc(C)oc2=O)=O)CN(C(c2ncccn2)=O)CC1C1CC1 c1(OC)cncc(CN2CCC(NC(c3cc(CN4CCCC4)c(C)s3)=O)C2)c1 CC1(NC(c2cc(CN(C)C)on2)=O)CCN(C(C2(c3ccncc3)CC2)=O)CC1 c1(C(=O)NC2C(NC(C(C(CC)(C)C)O)=O)COCC2)cnc2onc(C)c2c1 c1(C(=O)NC2CCC(NC(C3(COC)CCCCO3)=O)C2)ccc(P(C)(C)=O)o1 C(=O)(CCC(C(=O)O)Oc1ccc(F)cc1C(F)(F)F)OCC C(=O)(C(=O)C(C)(C)CC)N1C(CCC)CN(C(=O)Cn2cc(C)ccc2=O)CC1 c1(C(=O)NCCCCC(=O)NC(C(=O)OCC)C2(C)CC2)cn(C)c(=O)cn1 C12(CNC(C(C)(C3CC3)OC)=O)CCC(CC1)N2C(C1CN(C(N)=O)C1)=O C1(C(N2CC3C(C(=O)OC)(C3)C2)=O)(CC)CCCN(C(=O)C(C)(C)N(C)C)C1 c1(OC)cc(NC2(CCC(F)(F)F)CCC2)cc(OC)c1O C1(C(N2CC(CC(C)NC(c3n[nH]c(C4CC4)n3)=O)C2)=O)COC(=O)C1 c1(CC)ccc(C(=O)NC2CCN(C(=O)C(C)CNS(C)(=O)=O)CC2F)cc1Cl C(=O)(C1=CCc2ccccc21)NC1C(NC(CC(C(N)=O)NC(C)=O)=O)CC1 C1(Nc2cc(NC3CC(N(C)CC)C3)ncn2)CCCC1S(C)(=O)=O C(=O)(C(F)(F)C(C)O)N1CCC(NC(CCCc2ccc(SC)cc2)=O)CC1 N1(C(C(C(C)(C)O)F)=O)CC(CNC(=O)CC23COC(C2)C3)Cc2ccccc21 N1(C(=O)Nc2c(OC)ncnc2OC)CCc2ccc(C#N)cc2C1 CC(C)(CCCNC(=O)C(N1CCCCC1)O)NC(C1CCCN(C(N)=O)C1)=O c1(C(=O)NC2CCC(NC(C(COC)C)=O)C2)cc2c(Cl)cccc2s1 N1(S(C)(=O)=O)CC(C(=O)NCCCCNC(C2(CC3CCC3)CC2)=O)C1 C1(NC(=O)CC2CCCC(O)C2)CC2(C1)CC(NC(C1CC13CCCCC3)=O)C2 C1(CNC(=O)C(N2CCC(F)(F)CC2)=O)CCCCC2CN(CC(F)F)CC12 C1(C(=O)NC(C(=O)NCC)C)CSCCN1C(=O)CCN1CCCC1 c1(CC)ccccc1C(=O)NC1CCOCC1NC(=O)CCCc1csc(C)n1 CC1CCC(CC(=O)NC2CCC(CNC(=O)CC(C)CN(C)C)CC2)OC1 CCC(C)C(O)C(=O)NCCN(C1CCCC1)C(=O)CSc1ccccc1 c1(OC)n[nH]c(C(N2CC3CC3(NC(=O)CC3CC=CCN3C)C2)=O)c1Cl Cc1nc(C(C)(C)C)ncc1C(N1CCCCC1CNC(c1cnoc1C)=O)=O C(C(=O)OC(C)(C)C)(C(C)C)N(N1CC(c2cn[nH]c2)(c2ncc[nH]2)C1)C=O N1(C(C(C)NC(CCCCC)=O)=O)CCC(C2CCN(C(N3CCCC3)=O)C2)C1 N1(C(C(=C(C)C2CC2)F)=O)CC(CNC(C2(n3cncn3)CC2)=O)C(C)(C)C1 CC1=NN(C)C(=O)C1CC(=O)NCC1CCCC(CNC(C2CC=CCC2C)=O)C1 N1(C(C(CC(C)C)OC)=O)CCC(Nc2nccc(S(C)(=O)=O)n2)C(F)(F)CC1 N1(C(Cn2c(C)c(Br)cn2)=O)CC(N(C)C(=O)OC(C)(C)C)C(C)(C)C1 C1(C(=O)NCC(CNC(CN(C)C(N)=O)=O)C(F)(F)F)CCn2ncnc2C1 CS(C)(=O)=NC(=O)C(=O)NCC1CN(C(c2c[nH]nc2C2CCOC2)=O)CC1O c1(OC)cc(C(N2CC(F)CC2CNC(=O)C(F)OC(F)(F)F)=O)ccc1Cl c1(OC)ccc(C(C)N(C)C(C2CC2C(=O)Nc2cn(C)nc2C)=O)cc1 N1(C(c2ccc(C(C)(C)C)s2)=O)CC(NC(C2CCCO2)=O)CC(O)C1 c1(C(N(CCNC(Cc2cc(C)sc2)=O)C)=O)ccccc1C.N(C)(C1CC1)N.CC.S Cc1ccc(F)cc1C(=O)NC1CN(Cc2cscn2)CC1(F)F N1(C(CC(=O)NCC#C)=O)CCC(C)N(C(=O)CC2CNC(=O)C2)CC1 c1(SCC)ccc(CC(=O)NCC2(NC(C3CCCCC3CC)=O)CCC2)cc1 c1(CNC(=O)NC(=O)CCc2cccc(COC)c2)ccc(C)cc1C N1(C(C(C(=O)OCC)F)=O)CCCC(NC(=O)C(C(C)CC)N(C)C(C)=O)CC1 c12ccc(cc1)CNC(C(C)C)CS2.c1(CC)cccc(NC)c1 C1(C(N2CCCC(C(=O)NCC3(SC)CCC3)C2)=O)CCCC(F)(F)C1 c1(NC(CC2(O)CCN(C(C=C(CCC)C)=O)C2)=O)cc(Cl)cc([N+](=O)[O-])c1 C(=O)(C1=Cc2ccccc2OC1)N1CC2N(C(c3ccc(C)nc3)=O)C(CC2)C1 C(=O)(CC(C)(C)C)NC(C)CNCCN(C(=O)C=CCCc1ccccc1)C CC1(C)COC(C(=O)NC(CNC(c2ccccc2OCCF)=O)C2CCC2)C1 C(=O)(C1=NOC2(CNC2)C1)N(C1CN(C)CC1O)C CCCCC(C)CCC(=O)NCC(O)CN(C(=O)CC1(N(C)C)CCC1)C C1(NC(c2cc(CC)on2)=O)C2CC3CN(C(=O)CC4CC(C)(C)CCO4)C1C3C2 C(CO)(CCCCNC(=O)CCC(N)=O)NC(CC1CC(C)C1)=O C1(CC(=O)NCCCC)CC2C=CC1C2.C(=O)(COC)N(C(=O)C)CC#C CC(C)(C)CCC(=O)NCC1(NC(C2CCC(C3CC3)C2)=O)CC1 C1(CCC)COCCN1C(CCC1C=CCCC1)C(=O)Nc1ccc(OC)cc1 c1(C(C(=O)NC2C=CCN(C(c3cnc(SC)n3C)=O)C2)C)ccc(F)c(Cl)c1 C(C(=O)NC(C)CCn1cncn1)(C(C)(C)C)NC(C=Cc1c(C)n[nH]c1)=O C1(C(=O)OC)CCN(C(C2(OC)CCC2)C(=O)NC2CCOC2)CC1N(C)C C#Cc1ccccc1C(N1CC2CN(Cc3ccn(-c4ccccc4)c3)C2C1)=O C1(CC(=O)N(C)CC2(F)CCC2)C(NC(c2ocnc2C2CC2)=O)CC1O CC1(C)CC(CC(=O)NCCCCNC(c2ccn3c2CCC3)=O)C(=O)O1 C1(NC(=O)NC(C(C)(C)C)c2ncccn2)CCc2nn[nH]c2C1 c1(C(=O)NC2CCCCN(C(C3(C)CCCO3)=O)C2)cccn2nncc12 C(=O)(C(=O)N=S(C)(C)=O)NC1C(OC)CN(C(=O)COc2ccsn2)C1 c1(C(N(CC(C)NC(C2CC3(CSC3)C2)=O)CC)=O)[nH]c2ccccc2c1Cl c1(C(N2C(CNC(C3CC(F)(F)C3)=O)CC3CC32)=O)cc2cccn2cn1 C1(C)(c2ccc(C)cc2)CCN(CC(c2ccc(F)cc2C)=O)CC1 CCCCCC(C(=O)N1CC(COC)(NC(=O)C(C)(F)C(=O)OC)C1)C(C)C c1(OC)cc2[nH]ncc2cc1NC(=O)CCC1CCCN1Cc1cnc(Cl)nc1 C1(NC(c2cc(C)sn2)=O)C2CCC(C2)C1C(N1CCCC1C(=O)N(C)C)=O Cc1cncc(S(=O)(=O)N2CCN(c3cc4cnccc4s3)CC2)c1 c1(C(N2CCOCC(NC(C(C(C)C)C3CCC3)=O)C2)=O)ccc2c(c1)CCO2 N1(C(C(C)=CC(C)(C)C)=O)CCCC(C(C)(C)C(=O)NCCCCF)C1 C#Cc1ccc(C(=O)NCC2(OC)CCN(C(=O)Cc3c(Cl)cnn3C)C2)nc1 C(=O)(CC(C)CCC(=O)Nc1cnn2c1OCC(NC(C)=O)C2)OC c1(OC)ccc(N)c(C(N2CC3(CC3)CC2CNC(C2SCCCS2)=O)=O)c1 Cc1cnc(C(=O)NCCOC2CN(C(C3(C)CCCCC3C)=O)C2)cc1C#N c1(OC(C)C)ncc(-c2nc(-c3cc[nH]n3)nn2C(C)C(C)C)cc1Cl C(CN=c1[nH]c(=N)[nH]c(=NC2CC3CCCCCC23)[nH]1)c1scc(C)n1 N1(C(C(C=CCCC)O)=O)CCC2(CC(NC(c3ccc(Cl)c(O)c3)=O)C2)C1 Cc1ccc2[nH]c(C(=O)NCC3(F)CN(C(c4cnc(C)s4)=O)C3)cc2c1F N1(C(C(C(=O)OC)C)=O)CC2CCC2(CNC(=O)CC2(C#N)CCOCC2)C1 C1(F)(CNC(CC2(C=C)CC2)=O)CCC(NC(=O)Cc2cncn2C)C1 O=C(C1=C(Cl)CCCC1)NCCOC1CN(C(c2nc3c(s2)COCC3)=O)C1 N1(C(C2(NC(CCCN(C(C)=O)C)=O)CCC(C)(C)C2)=O)CCC(=O)N(C)CC1 C(C(C)(C)CCCC(=O)OC(C)=O)NCCOC FC1(F)CC(c2nc(-c3nnc(Cn4cc(Br)cn4)o3)no2)C1 C1(NC(c2c(CCC)nns2)=O)CCN(C(=O)CCn2ccccc2=O)C1(C)C c1(CC(=O)NCCC2CCCN2C(=O)C(O)C(F)F)ccc(F)cc1 N1(C(C2ON=C(C)C2)=O)CC=C(CCNC(C2CC2(F)F)=O)CC1 Cc1cc(Cl)c(O)c(Br)c1C(N1CCCCC1c1ncc[nH]1)=O N1(c2n(NC(=O)OC(C)(C)C)nnn2)CC(c2ccccc2)C(c2ccnn2C)C1 c1(C(N(CC(CNC(C(CC=CC)CC)=O)O)C)=O)cnc2ccnn2c1C CC1CCCC1(C)C(=O)NCCN(C(=O)COc1nn(C)cc1Br)C c1(NC(c2n(CC=C)nnn2)C2CCOC2C(C)(C)C)cnc(Br)c(C#N)c1 C(CCCC(CO)NC(=O)C(c1ccccc1)N(C)C)NC(c1scc(C)c1)=O Cc1noc(C)c1CC(C)C(=O)NCC1CCC(F)(CNC(=O)CCF)C1 c1(C(N(CCCNC(C2CC23CC3(F)F)=O)CC)=O)nccc2ccsc12 c1(C2C(C(=O)NCC(CN(C(CN(C)CC)=O)C)C)C2)ccncc1 C(=O)(CS(C)(=O)=O)NCC(=C)CCNC(=O)CC1(S(=O)(=O)CC)CC1 C(C(CC1CC1(F)F)C(=O)N(C)CC1CCC1)NC(C(C)OCCOC)=O C#CCC(C(=O)N1CCC(C(C)CNC(=O)C=Cc2cocn2)CC1)C1CC1 N1(C(C=Cc2cc(C)no2)=O)CCCC(C)C1CCNC(=O)C1=CCCCC1 C1(C(CNC(C(C)OCCC=C)=O)(C)NC(C2CC(F)C2)=O)CCCCC1 C1(NC(CCOC)=O)CC2CC1CN(C(c1cccc(NC(C)=O)n1)=O)C2 C(=O)(CCCC(F)(F)C(F)(F)F)NCC1CCC(NC(C(C)(O)C2CC2)=O)CC1 c1(C(N2CC(NC(CN(C)C(N)=O)=O)C(C)(C)CC2)=O)cc(F)cc2nn[nH]c12 C(CC1C(=O)N1)OC.c1(C(CN2C(NC(=O)OC(C)(C)C)CC2)C)ccc(F)cc1 c1(N(C)C)cc(C(=O)NC2(CO)CN(C(C3COC(C)(C)C3)=O)C2)cc(Cl)n1 C1(CNC(c2n[nH]c(C)c2C)=O)CC(C)CN(C(=O)C=CC2CCOC2)C1 C=C(C)CCC(=O)Nc1cccc(CNC(=O)C(C)NS(C)(=O)=O)c1 N1(Cc2c(C)ccs2)CC(CO)C(N)C1 C(=O)(C1CCCn2nccc21)NC1CCCN(C(CCCCCOCC)=O)CC1 CCC(CNC(=O)Cc1nc(=N)[nH][nH]1)(CC)C(=O)NCC1CCC(C)C1 C(=O)(C(=O)C(C)(C)C)NC(CCNC(CSC(C)C)=O)(C)C C1(CC)CCCN(C(=O)CC(CC)CC)C1C(=O)NCc1cnc(C)[nH]1 Cn1nc(CNC2CCC(C(=O)N(C)CC#N)C2)c2ccccc12 C(=O)(C(F)(F)C(O)CC)N(CCNC(c1nc(C(C)OC)oc1)=O)C CC1(C)CC2(CC(C(=O)NCCC3=CCN(C(=O)C(C)CC(N)=O)CC3)C2)C1 c1(C(N(CC)Cc2ccsc2)=O)ccc(F)c(-c2cccc(SC(F)(F)F)c2)n1 N1(C(CN(C)C)=O)CCOCC(F)(CNC(C2CCCN(c3nccs3)C2)=O)C1 C(=O)(CC(C)CC(C)C)NC(CNC(c1c(CC)cccc1F)=O)(C)CC N1(C(C=Cc2cc(C)c(OC(C)C)cn2)=O)CC=C(c2cccc(F)c2)CC1 C(=O)(C(F)(F)C(F)(F)C(F)F)NC1C(NC(C2CCC(C)(C)O2)=O)CCC1 N1(c2c(C)cc(C#N)cn2)CC2(C1)C(NC(c1ccsc1)=O)CCS2(=O)=O N1(C(C(c2cccc(C)c2)=O)=O)CCC(C)(C)C1CNC(c1csc(C)n1)=O C1(NC(c2ccc(C#C)o2)=O)CC2CCC(C1)N2C(=O)CCCCC(C)C C(=O)(C1=CC2CCC(C1)C2)NCC(C)CC(=O)NC1CCCC1CCO CCC(C)C(C(=O)NC12CC(C(=O)NCc3cnn(C)c3O)(C1)C2)OC N1(C(C2(C#C)CN(C(=O)CCCCC)C2)=O)CC2(CCC2)C12CCC2 C(C(O)CC(F)(F)F)NC(C(C)N(CCC)C(C1CC2CC1CC2=O)=O)=O c1(C(N(C(C)CNC(c2cnc(O)c(F)c2)=O)C)=O)cccc(S(=O)(=O)CF)c1 c1(C(N2C(C)CN(C(C3CCCC3O)=O)CCC2)=O)cc2c(nn1)CCCC2 c1(C(=O)NCC=CCNC(CC2(O)CCCN(C)C2)=O)cc2cccnn2n1 c1(C(C)(C)NC(C(=O)NCC2CCC(C)C2)=O)ccc(Cl)cc1 c1(CC(=O)NC2(C)CC(NC(COCC(=O)OC)=O)C2)nc2c([nH]1)CCCC2 c1(C2(O)CC(NC(=O)NCCCc3n(C)cnn3)C2)ccc(I)cc1 C1(C(=O)NCC=C(C(=O)NCC2(CO)C(C=C)C2)C)CC2(CC2)CO1 N1(C(C2(COC)CC=CC2)=O)CC(N(C)C(c2nncs2)=O)C2(CC2)C1 c1(N(C)Cc2cc(O)ns2)cc(Cl)ccc1Oc1ccc(Cl)c(Cl)c1 C1(C)(C(=O)NCC2CN(C(C(c3c(C)noc3C)(C)C)=O)C2)CCCNC1=O Cc1nc2cnn(C)c2cc1C(N1CC(C(N)=O)OC(C)C1)=O Cc1cnc(C(=O)NC2CCC(CNC(C3(F)CCCOC3)=O)C2)cn1 N#Cc1ccc(CN2CCC2C(=O)Nc2cccc(C(F)F)c2)cc1Cl CCC(CC)C(C)C(=O)N1CCCC(CC)(NC(c2cn(C3COC3)nn2)=O)C1 N1(C(CCOCC#C)=O)CC2=C(C1)CN(C(c1occc1CSCC)=O)C2 c1(CC(=O)NCCCN(N2CC(N)CC2=O)C(C23CCC2C3)=O)ccc(F)cn1 N1(C(C(Cc2c(C)nc[nH]2)O)=O)CC2=C(C1)CN(C(=O)CSC(C)C)C2 c1(N(CC(C)NC(C2COCC(C)(C)O2)=O)C)ccnc2ncnn12 c1(C(=O)NC2(CNC(c3ccc(CC#N)cc3)=O)CC2)cc(Cl)cc(Cl)c1O c1(C(=O)NC2CCN(c3nccc(C)n3)CC2F)cccc2c1CC(=O)N2 C1(C)(CNC(C(CC)=CC)=O)C(C)CCN1C(=O)CCCc1cc(C)sc1C C(=O)(CC(C)C(=O)NCC(C)CNC(c1ccnc(NC(C)=O)c1)=O)OC N1(C(C2C(C=C)OCCC2)=O)C2CCC1CC(CNC(=O)CCOCCOC)C2 C1(C)(C(=O)NCCC)CN(C(C2CCCN(C)C2)=O)C(C)(C)C1 C(N=c1[nH]c(=NC(C)c2ccc(F)cn2)c2sccc2[nH]1)C1N(CC)COC1 Cc1noc(C)c1C(c1nnnn1C)Nc1cccc(CC2CC(=O)NC2=O)c1 c1(CN(CCOC)CCNC(c2cc(CC(C)C)[nH]n2)=O)c(O)cc(Cl)cc1F Nc1ccccc1C(=O)NCC1C=CCN1C(c1cc(-c2cccc(F)c2)no1)=O C1(NC(C2CCSC2)=O)CCC(n2cc(CSc3ccccc3)nn2)C1 c1(C(=O)NCCCC2N(C(C3CC(N(C)CC)C3)=O)CCC2)cc(Cl)ccc1F C=CC(C)CC(=O)NC(CO)C(C)NC(=O)C(C)OCOC c1(CC(=O)NC2(CCCCNC(C3(OC)CCCC3)=O)CC2)cncc(Br)c1 C1(C(=O)NC(CC(C)NC(=O)CN(C)C)C)CCN(C2CCCC2)CC1 c1(C(N2CCC(CCN(C(C3C(C=C)C3)=O)C)CC2)=O)cc(C)cc(OC)c1O N1(C(C(CC=C)N(C)C)=O)CC2CN(C(C3(CCOC)CCCC3)=O)CC2C1 Cc1ncccc1Cn1cc(CCC(N)CC2CCCCC2)nn1 C(=O)(C1=CCCS1)N(C(C)C)CCNC(C1CC(=O)C1C(C)(C)C)=O N1(C(C2(C)CCN(C)C2)=O)CC2CN(C(c3ccn(C4CC4)n3)=O)CC2(C)C1 N1(C(CC(CC)CC)=O)CC(NC(=O)COC(=O)CO)CC12CCCC2 N1(C(C(CN(CC)CC)F)=O)C(CNC(c2cncc(C)n2)=O)CC2CC12 N1(CCC(=O)NNC(=O)c2ccccc2Br)CCc2n[nH]cc2C1 CCCCC(CC)CC(=O)NC1(C)CCCCC1C(N1CC(F)CC(F)C1)=O c1(C(C)(C)C)cccc(C(N2CCOCC(CNC(c3ccon3)=O)C2)=O)c1N Cc1cc(C(=O)NCC(C2CC2)NC(c2cn(C(F)(F)CO)nn2)=O)co1 CCN=C(NCc1ccn(C)c1)NC1CCOc2ccccc21 Cc1nc[nH]c(=NCC2CCCN2C(c2nc(-c3cccn3C)cs2)=O)c1Br C1(F)(C(=O)NCC(C(=O)NCc2ccn(COC)n2)N(C)C)CC=CCC1 C1(C(=O)NCCCOCC#C)CCC2(CC2)N1C(=O)C(C)S(N)(=O)=O C1(NC(CCCOCC)=O)CCN(C(C2CCC(=O)N2)=O)C1C(C)C CCCC(C(=O)NCc1ncoc1C1CN(C(=O)C(c2csc(=N)[nH]2)=O)C1)OC C1(CC=C)(NC(=O)CCc2ccccc2)CCCN(C(=O)C(C)NS(C)(=O)=O)C1 C1(CNC(CC2C(OC)COCC2)=O)CC12CCN(C(c1cc(Br)co1)=O)CC2 c1(C(=O)NC2CCC(NC(=O)CNc3cccnc3)CC2)cnn2ccncc12 CC(CC1CCCO1)C(=O)NCCCCNC(=O)C(C)C1(O)CCC1 C1(CNC(c2ccc(C)nc2)=O)CC2(CCN(C(c3nnccc3C)=O)C2)CO1 C1(NC(CCc2cc(C)no2)=O)CC(C(=O)NC2C3CCC2CC3)C12CCC2 C(=O)(C(O)C(F)(F)F)N(CC(CN(C(c1cccc(OCC)c1)=O)C)O)C c1(OCC)ccc(N2CCOCC2)c(C#N)c1.c12ccc(C)nc1[nH]c(=O)[nH]2 c1(-c2nc(-c3cc(OCCCC)ncc3)nn2C(C)C)ccc(N(C)C)nc1C c1(Cn2cc(CC3(O)CCNCC3)nn2)ccc(I)c(Cl)c1 c1(C(=O)NC(C(C)NC(C(CCOC)C)=O)(C)C)ccc2[nH]c(=N)n(C)c2c1 N1(C(C(F)=CCC)=O)CC(NC(C2CC(C)(C)CO2)=O)CC1(C)C N1(C(CC(=C)C)=O)CCC(O)(C2CCN(C(C3CN4CCN3C(C)C4)=O)CC2)C1 Cn1ncc2c1CCCC2N=c1[nH]c(N2CCC3(CNC(=O)C3)C2)nc2ccsc12 N1(Cc2n(C)ncn2)CC2CN(C(c3ccc(OC(F)(F)F)nc3)=O)CC12 C1(NC(Cc2nc(C)sc2)=O)CC1C1CCCN(C(=O)CN2CCCCCC2)C1 c1(C(=O)NCCC(C)NC(c2ccnc(OC(C)C)c2F)=O)n[nH]c2c1CC1CC21 N1(C(c2nc(C)oc2C)=O)CC2CCN(C(=O)C=CSc3nc[nH]n3)CC12 c1(C(=O)NC(CC=C)CNC(=O)C(C)c2ccsn2)cc(C)c(F)cn1 C1(CNC(C(C)c2ccco2)=O)CN(C(=O)CC2CCC(F)(F)CC2)CCC1(F)F Cc1cc(C(F)(F)F)nc(=NCCOCCNC)[nH]1.c1(CN)csc2nnsc12 C1(NC(c2ccc(SC(F)(F)F)s2)=O)CCCCC1c1ccccc1 Cn1ccc2[nH]c(C(=O)NCCC3CCCN3C(c3cccn(O)c3=O)=O)cc12 c1(C(N2CC(N(C(c3c(CC)occ3C)=O)C)C(F)C2)=O)ccc(C)c(N)c1 C12(NC(=O)C=CBr)CCCC1CN(C(c1cccc(CN3CCCCC3)c1)=O)C2 C(C)(CCC(=O)NCCN(C)C(c1cc(OC)cnn1)=O)OC C1(C(=O)N(CC2CN(C(CNC(c3ccccc3)=O)=O)C2)C2CC2)COCOC1 C1(NC(c2cc(CNC(C3C(C)SCCC3)=O)no2)=O)CC2(CCC2)C1O O=C(C1=CCOC1)NCC(O)CCNC(=O)C(O)(C1CC1)C1CC1 c1(C(N(CCCN(C)C)CCNC(=O)CC2CCC(O)C2)=O)[nH]nc2ncccc12 Cn1cc(C(=O)O)c(Cl)n1.n12cc(nn1)C1(CCCC1)NC(=O)CC2 N1(Cc2nccc(C)n2)CCC(=O)N(CCOCCN2CCOCC2)C1=O C1(NC(CN(C2CC2)CC)=O)CCCN(C(=O)CC2CCOC2=O)CCC1 c1(-c2scc(CC(=O)Nc3n[nH]c(C4CC4)n3)n2)ccc(F)c(Cl)c1 C1(C(=O)NCC(c2ccccc2F)NC(c2n(CC)ccn2)=O)(OC)CCCOC1 N1(CCC(CCC)(C)O)CCCC2(C1)CCCN2C.C(=O)(C(C)C)N Cc1c(C(N2CC(C)(C(=O)Nc3cnn(C4CC4)c3)C2)=O)cccc1S(C)(=O)=O N1(C(C(CC)Cn2cncn2)=O)CC2CN(C(c3cc(F)ccc3F)=O)CC2C1 CN1CCCCC1CC(N1C(CNC(c2csc(C(F)F)c2)=O)CC2CC12)=O c1(CC(=O)NCC2(n3nccn3)CC2)cc(C)nc(O)c1.CCC1CC(=O)N1 C1(C(=O)NCc2c(C(N(CC(F)Cl)C)=O)con2)C2CC3C(C2=O)C13 c1(OC)cc(NC(C23CC2CN(C(C2(C)CCCN2)=O)C3)=O)cc(F)c1 Cc1nc(N)cnc1C(=O)NCC1CCN1C(=O)C=CC1CCC1 N1(C(c2cnc(C(C)OC)s2)=O)CCCC(C)(NC(=O)CCCCOC)C1 c1(-c2c(C(=O)NCC(CC=C)NC(=O)C(C)O)nco2)ccc2c(c1)OCCO2 c1(SC)cncc(NC(C2CC(C)N2C(=O)CC2CCC(C)(C)C2)=O)c1 CN1CCN(C(=O)CC2CCCCN2C(c2ncn(C)n2)=O)CC(O)C1 c1(CN(C2(CC=O)CC2)C)cc(Cl)c(Br)c(OC)c1[N+](=O)[O-].CN c12noc(c1C)C(=O)C2=O.C1(CC)(OCc2cn(C3CC(N)C3)nn2)CCOC1 N1(C(CCC(Sc2c(=N)c(=N)[nH][nH]c2)C2CC2)=O)CCC2(CC2)CC1C(F)(F)F c1(N(C)C)ncccc1C(=O)NC(C)(C)CCNC(C1CCC(C(N)=O)C1)=O CCC(CC)C(C(=O)NC12CC1CN(C(C1(c3ccno3)CCC1)=O)C2)OC c1(OC)cccnc1C(=O)NC12CC(CNC(=O)C(COC)N(C)C)(C1)C2 c1(C(N2C(C)CCN(C(c3ccc(Cl)o3)=O)CC2)=O)cncc(S(C)(=O)=O)c1 C(=O)(C1=NOC2(CCC2)C1)NCCCCCN(C(=O)C(C)N1CCC1)C(C)C C1(C(N(CCN(C)C)CC)=O)COC2(C1)CN(C(=O)C(C)(C)C(C)C)C2 N1(C(c2ccc(OC)nn2)=O)CCC2CCN(C(=O)CC(O)C3CCCC3)CC12 c1(C(=O)NCCOCC(=O)NCCC=CCC)cnn(CCC)c1 c1(CC)ccc(OC)c(C(N2C3CC2CN(C(=O)COCC2CCCO2)C3)=O)c1 Cc1cc(Cl)nc(N)c1C(=O)NCC(O)CNC(=O)CCc1cncs1 c1(OC)cc(NC(C2CC(C)CN(C(=O)Cn3ccc(C)c3)C2)=O)cc(F)c1 c1(CC)cc(C(N2CCC(CCC(=O)N(CC)CC3CC3C)C2)=O)n[nH]1 c1(C(N2CC(NC(C3CN(C)C3)=O)CC(C)(C)C2)=O)cnc2ccc(C#N)cn12 C1(OC(C2CCC(CC)O2)=O)CCCCC1CNc1cnc(F)cn1 c1(SCC)noc(C)c1-n1nc(CCOC2CC2)nc1-c1ccccc1F CCC(C)C(C(=O)NC(Cc1ccco1)C(=O)NCC(CC)C(C)C)N(C)C N1(C(c2cc(CC(C)C)nn2C)=O)CCCC2(CCN(c3cc(O)ncn3)C2)C1 C1(NC(CCC=C(C)C)c2nnnn2C2CCOC2)COC(C)(C)C1 C(=O)(CC1OCc2ccccc21)NC(C)CNC(c1coc(CO)c1)=O c1(C(=O)NCC(C)N(C(C=CCCC)=O)C)c(C)cc(C)nc1OCC N1(C(C=CCNC(c2ccccc2)=O)=O)CCC12CCCOC2 C1(C2(F)CN(C(=O)CN(C)C(C)C)C2)(NC(CC(C(=O)O)NC)=O)CC1 C1(NC(CC(CCC)C)=O)CN(C(c2cccnc2)=O)CCC12CCCC2 N1(C(COC(C)C)=O)CC(CN(C)C(c2nn(C)cc2Cl)=O)C2(CC2)C1 CC1(NC(=O)CCCCNC(=O)C(F)F)CCCCCC1 N1(C(CCCC#CC)=O)CCC2CN(C(=O)CCCCCc3cccs3)CC12 C1(CCC)CN(C(c2ccsc2)=O)CCN1C(c1nc(C)ccc1C)=O C(=O)(C#CC1(C)COC1)NCC1(F)CCN(C(C(C)C)=O)C1 c1(-c2cn(CS(C)(=O)=O)nc2)cc(C(=O)NCCS(C)(=O)=O)c2nccn2c1 c1(C(=O)NC(c2ccc(C(F)(F)F)cc2)C)cnn(CCN2CCOC(C)C2)c1N C(=O)(C1Cc2ccccc21)N1CC(C2(NC(c3scc(C(C)(F)F)n3)=O)CC2)C1 N1(C(CCN(C(C)C)C)=O)CC(O)CC1CNC(C1CCN(CC2CC2)CC1)=O CC(CSC(F)(F)F)C(=O)NC(CNC(c1ccco1)=O)CO Cc1cn(C)cc1C(N1CCC(n2cc(C3CCC(C(C)C)CC3)nn2)C1)=O n1(NC(C(C(C)C)OC(C2CCSC2)=O)=O)c(=O)oc2ccccc12 C1(NC(Cc2n(C)cnc2)=O)CCCN(C(=O)CCOCc2ccccc2)CC1 c1(C(N(CC(CC)NC(=O)CC2CCC(=O)N2)C)=O)ccc(O)nc1Cl C(=O)(C(C)(C)CCCNC(=O)CC1CCC(C#N)C1)NCCOCCN(C)C C1(CNC(C(N2CCNC2=O)C)=O)COCCN(C(=O)C(c2ccccc2)C)C1 Cc1ccc(F)c(CC(=O)NC(C)CC2CN(C(c3cc([N+](=O)[O-])sn3)=O)C2)c1 c1(C(=O)NCC23N(C(c4c(C)nccc4)=O)C(CC2)CC3)c(Cl)sc2nnsc12 C1(CC(=O)NC(CCC2N(C(CSC)=O)CCCC2)(C)C)CC2(CCC2)CCO1 n1(CC(=O)NCC(C)NC(=O)C(F)(F)c2cnn(C)c2)nc2n(c1=O)CCOC2 c1(CC(=O)N(C)CC2C(NC(c3c(C)csc3)=O)CCC2)cc(Cl)n(C)n1 Cn1cc(C(=O)NCc2cc(C(=O)NCC3(O)CCCOC3)n(C)n2)n(C)c1=O C1(CNC(C2(OC)CCCC2C)=O)CC(C)CN(C(=O)Cc2cnsc2)C1 C1(C)(C(=O)NC2C(C)CN(C(c3ncccc3Br)=O)C2)CCCCCC1 C(CC(=O)NCCNC(c1cc(CO)c[nH]1)=O)(C(C)(C)C)NC(=O)OC(C)(C)C c1(CC)nc(C(=O)NCC(C(C)C)NC(c2cc(CC(C)C)on2)=O)co1 C(=O)(C1=Cc2ccccc2OC12CCC2)NCCN1CC(C)N(C(=O)C2CC2)CC1 C1(NC(COCCOC)=O)CS(=O)(=O)C12CCN(C(C1CC3C=CC1C3)=O)CC2 C12(CNC(c3cc(C)n(C)n3)=O)CCCCC1N(C(=O)C(C)C(C)C)CCC2 c1(C(=O)NCCC(CNC(C=C(C)C(C)C)=O)O)ccccc1SC(F)F C1(NC(CCNC(C)=O)=O)CN(C(C2CCN2C(C)(C)C)=O)CCC1(C)C C1(O)(CC(=O)N(CCCOCCNC2CC2)C)CCCCC1.n1(CC=O)cccc1 CC1(CNC(=O)CC2CC2(Cl)Cl)CC(F)(F)CN1C(c1cc(O)cc(O)n1)=O C1(C#CC(=O)N2CCCC(CN(C(=O)C(F)(F)C(F)F)C)C2)(CC)CC1 N1(C(c2cccc(C)c2C)=O)CCCN(C(=O)CC(F)F)C(C)C1 C(C1c2ccsc2CCN1C(=O)Cn1cnnc1O)NC(C(=O)NCCSC)=O C(=O)(C(CO)C(C)(C)C)NCC1CN(C(Cc2ccc(C)cc2)=O)C1 N1(C(CCC=C)=O)CCOC2(CCN(C(C3(c4ccc(Cl)nc4)CC3)=O)C2)C1 N1(C(CC2(CCC#C)OCCO2)=O)CC(CNC(=O)CC2CC2C2CC2)CC1(C)C C1(CC)N(C(=O)CC2CCCN(C(=O)CNC(C)=O)C2)CC12CCCC2 CC(C)(C)C(CNC(c1cccc(C2CC2)n1)=O)NC(c1cnc(C2CC2)s1)=O C=C1CC(C(=O)NCCCCN2CCC2)(CNC(C2CCCCO2)=O)C1 C12(C(=O)NCC3(O)CN(C(C4CC(C(F)(F)F)C4)=O)C3)CCCCCC1OCC2 O=C(N=c1ccn(C(F)F)[nH]1)C1CC(=O)CN1C(c1cccc(F)c1)=O C(=O)(C1=CCCSC1)NC1C2CC(NC(C(CC)C#N)=O)CC21 c1(C(=O)NCC(CCOC)NC(c2c(CC)noc2C)=O)cccc(C=C(F)F)c1 Cc1cc(CNC(=O)NCC2CCCN(C)C2C)ccc1Cl Cc1ccc(OCCC(=O)N2CC(NC(=O)CNC3N(C(=O)C4CC4)CC3)C2)cc1 n1(CC=C)cc(C(=O)NC2(C3CCCN3C(=O)CC3(CO)CCCC3)CC2)cn1 c1(NC(=O)NC2C3CCC2CN(C(C2(C4CC4)CC2)=O)C3)ccccc1[N+](=O)[O-] C1(C2CCN(C(c3ccc(Cl)c(C(F)(F)F)c3)=O)C2)(NC(C2C(C)(C)C2)=O)CC1 C(CN=C(NCC1CC12CC2)N1CCCC(CC(C)C)C1)OCC#C N1(C(c2cccc(-c3ncc[nH]3)c2)=O)CCC2(CC1)CN(C(C13CCC1C3)=O)C2 N1(C(CCC(C)c2ccccc2)=O)CCCN(CCNC(=O)COCCF)CC1 C1(C(=O)NCC(C)(C)C(=O)NCCCn2cnnn2)CCCC12CCC2 Cc1cc(C(N2CC(F)(C(=O)Nc3cc(Br)ncc3C)C2)=O)ccc1O CC(C)C(C)CC(=O)N1CCCC1Cc1ccccc1 c1(C(N2CCC(N(C(=O)C=NOC)CC)C2)=O)cc([N+](=O)[O-])c(N)cc1F Cc1nc(NC2CC(NC(C3CC4CC4C3)=O)C2(C)C)c2scc(C)c2n1 N#Cc1cnc(C(=O)NCC2CN(C(C3CCCS(=O)(=O)C3)=O)C2)c(Cl)c1 C1(C(=O)NCC2CN(C(c3c(COC)ccs3)=O)C2)CCc2ccc(F)cc2O1 N(C(=NCCC(C)(C)O)NCCc1ccncc1)C(C)CSC1CCCCC1 C1(CCC(=O)NC(CC)CN(C(C2(CC)CC2)=O)C(C)C)NC(=O)NC1=O N1(C(c2cc(C)[nH]n2)=O)CC2CCCCC2(CNC(=O)Cc2nonc2C)C1 N1(C(CN(c2ccncc2)C)=O)CCC2C(NC(=O)CCC(=O)NC3CC3)C12 C1(CCNC(C2(CC)CC(=O)C2)=O)CCCN(C(=O)C=Cc2cncs2)CC1 N1(C(CCN(C)CC)=O)CC2C(CNC(C3(C)CC(F)(F)C3)=O)C2C1 c1(OC)ncnc(C)c1C(N1CCN(CC2CC(OCC3CCCC3)C2)CC1)=O C1(CNC(=O)CCOC2CC2)CN(C(c2cc(C(O)C(F)(F)F)ccn2)=O)CCO1 C(=O)(CCCCCF)N1CCC(N(C(C=CC(CC)C)=O)CCO)CC1 C12(C(=O)NC3(C)CC(NC(C(C)CS(C)=O)=O)C3)CC1COC21CCC1 CC1CC(NC(C2CC(=O)N2)=O)CCN1C(c1nc(Cl)sc1Cl)=O CS(=O)(=O)CCCC(=O)N1CCCC(CO)(NC(=O)CCc2cscn2)C1 c1(C(=O)NC(C(=O)OCC(C)C)C)ccc2[nH]cc(-c3cncn(C)c3=O)c2c1 C(=O)(C(Cn1cncn1)NC(=O)C=Cc1ccco1)N(C1CCCC1)C C1(NC(c2c(CCC)nco2)=O)CC2CC1N(C(C1CC1COC)=O)C2 C1(C(=O)NCCc2cc(CC)on2)CCCN(c2cc(C=O)nn2C)CC1 c1(C(N2CC(OC)(CNC(C3CNC(=O)C3)=O)C2)=O)cnc(N)c(N)c1 CC1CN(C(=O)C(=O)Nc2ccccc2I)CCN1S(C)(=O)=O CC1(C)C(C(=O)NCC2CCCCC2)CCN1C(C1CC(F)(CF)C1)=O N1(C(c2c(Cl)cn(CC)n2)=O)CCN(C(c2cccc(F)c2Cl)=O)CCC1C Cc1cc(CCC(=O)NCC2CC2NC(c2c[nH]cc2C)=O)c(C)s1 c1(C(=O)NCC2N(C(C(CCCOC)C)=O)CC(F)(F)C2)ccc2c(c1)CCC2 N1(CCC(=O)NCC(C)CNC(c2c[nH]c(C(N)=O)c2)=O)CCP(C)(=O)CC1 c1(C(=O)OCC)cccc(O)c1F.C12CC(C(SC)C1)NC(=O)C(=O)N2 C1(NC(CCCCCC)=O)CC2CC1CN(C(C1OCCCC1(C)C)=O)C2 C12(NC(C3(C(F)(F)F)CC=CC3)=O)CCN(C(=O)C=CC=C(Cl)Cl)CC1C2 n1(C(CC)C)ncc(C(=O)NC2COCCC2NC(c2ccncc2O)=O)c1C C1(NC(c2c(C(F)(F)F)ncn2O)=O)CCC2CCN(C(C3CCOC3)=O)C1C2 N1(C(c2cc3cccc(C)c3[nH]2)=O)CCCC(C2CN(C(=O)C(C)(C)C)C2)C1 c1(C(N2C(C)CC(CNC(C3C(C)(C)C3(C)C)=O)CC2)=O)ccn2ccccc12 C1(OC)(CNC(C2(C(=O)NC)CC2)=O)CCCN(C(=O)C(F)(F)CC2CC2)C1 CC1(CNC(=O)NCC2(OC)CC2)CC2(C1)CC(F)(F)C2 C(CC(CC)C(=O)N(CCCNC(c1cc(OC)n(C)n1)=O)CC)=CC C1(NC(C=C(CCC)C)=O)CC12CCN(C(c1ccc(NC(C)C)nc1)=O)CC2 c1(OC)ccc(C(=O)N(CCCCNC(=O)CCCC2CC2C)C)cc1N Cc1cc(Cl)ccc1OCC(N1CCC(NC(=O)C2=CCC2)C(C(C)C)C1)=O CC(F)(F)CCC(=O)NCc1ccc(C(=O)NCc2nccn2C2CC2)o1 C=CCN=c1[nH]c(NCC(C)(F)F)nc2cc(OC)ccc12 c1(CN(C(=O)CCC2CCCN2C(c2ccoc2Cl)=O)C)cccc(F)c1 c1(OC)ccc(OC)c(C2CN(C(=O)NCCF)CCN2CCO)c1 N1(C(c2ncccc2Cl)=O)CCC2(CC1)CN(C(C1CC13CC3(F)F)=O)C2 c1(C(N2CC(CNC(CCC(C)(F)F)=O)C3C2C3)=O)ccc2c(=N)[nH]cnc2c1 C1(C(N(C)CCC2CCNCC2)=O)C2CN(S(=O)(=O)CC3CCS(=O)(=O)C3)CC12 C12(NC(c3c(C)con3)=O)CCC(CNC(=O)C=CC(C)C)(C1)OC2 C(=O)(CC(C)CCC=C(C)C)N1CCC(C(C)NC(C2(OC)CC2)=O)C1 CC1CC(F)(F)CCN1C(C1(CNC(=O)CC2(N(C)C3CC3)CCC2)CCCC1)=O N1(C(Cc2cc(C)[nH]n2)=O)CC2CC1(c1cn(Cc3cc(C(F)F)on3)nn1)CO2 c1(C(=O)NC2C(NC(C(C)(O)CCc3ccccc3)=O)C2)cccc(F)c1F c1(C(=O)Nc2cc(-c3cnc(C)s3)ncc2)cccc(S(C)(=O)=O)n1 C1(N(C)CC)CCN(C(C2CCN(C(=O)C(F)n3ccnc3)C2)=O)C1 C1(C(C)C)CC(NC(=O)C(CN(C)C)NC(=O)CC2(O)CCC2)CCO1 c1(C2(C(N3C(CN(C(=O)CC4CC4)CC)CCC3)=O)CC2)ncccc1F C1(CNC(CC2(OC)CN(C(c3cc(=O)n(C)cn3)=O)C2)=O)CCC(=O)NC1C O=C(C1=NOCC1)NC1CCCC(NC(c2cc(C(F)(F)F)ns2)=O)C1 C1(C)(CNC(CC2N(C)CCCC2)=O)COCCN(C(=O)CC2CC3(CC3)C2)C1 C(=O)(CC(C)(C)C(F)F)NCCC(CNC(c1ncc(C)cc1F)=O)O C1(CC(=O)N(CCC(=O)NCCCN(C)C)CC=C)C=NN(C)C1=O N1(C(c2nc(C)oc2)=O)CC(C)CN(C(c2ccc3c(c2)COB3O)=O)C(C)C1 Cc1ccc(C=CCNC(C2CCC(n3cc(-c4scnc4C)nn3)C2)=O)s1 Cc1ccccc1N=c1[nH]nc(CC(=O)NC2CCC3CCC23)s1 C1(OC)C=CCN(C(=O)CC2CC(C)N(C(C3CCSCC3)=O)C2)C1 C1(C(=O)O)(CC)CCCN1CC(C)CC1CCCC1 C(=O)(C(C)(O)C(C)(C)C)N1CCC(n2cc(CCC(=O)OC)nn2)CC1 O=C(C1=NOC2(CCC2)C1)NCCC1CN(C(=O)C=CCn2cncn2)CCO1 C1(NC(CCNC(c2n(C)ccc2)=O)=O)CCN(C2CC2)CC1 c1(C(N2CCC(NC(C(CC)CC)=O)C2)=O)cc(=O)oc2ccc(O)cc12 N1(C(C2(CC#C)CCOCC2)=O)C2CCC1C1CC1(NC(c1snnc1C)=O)C2 c1(NC(C2CCN(Cc3cc(C)c(Cl)cc3)CC2O)=O)cc(C#N)cnc1C CN1CCCC(CN(CCN(C)C)C(=O)C2CC2)C1 Cn1ccc2cc(C(N3CC4CC(C3)N4Cc3cc(I)c[nH]3)=O)ccc12 c1(C(=O)NC(CN(C(C(COC)N(C)C)=O)C)C)cc(Cl)nnc1O N1(C(C(C=C)(C)O)=O)CC2CCCC(NC(=O)CN3Cc4ccccc4C3)C2C1 C1(NC(c2cnc(CC)s2)=O)CN(C(=O)Cc2nc(C)no2)C2(CCCOC2)C1 C1(C(=O)NCC(C)CC(=O)NCC2CC2(C)C)CC2(CCO1)CC2 C=C(C)CC(C(=O)N1CCC(NC(c2[nH]nc(C(F)(F)F)c2C)=O)C1)NC(C)=O c1(C(N(CCNC(C2(C)CC=CCC2)=O)CC)=O)ccnc2ccc(OC)nc12 S(=O)(=O)(c1cnn2ccc(N3CCc4oc(C)nc4C3)nc12)NC(C(CC)C)C c1(C(=O)OC)c(C)[nH]c(C(=O)COC(=O)CC23COC(CC)(C2)C3)c1C C(=O)(C1=COCCC1)NCC1C(CNC(c2n(CC(=O)OCC)ncc2)=O)C1 N1(C(C23CC4CC2C3C4)=O)CCC2CN(NC(C(C)(F)F)=O)CC2C1 n1(CCC(=O)NCCCN(C(C2(CC)CCCCC2)=O)CC)cnccc1=O C1(C(=O)NC2CCN(C(C(C)C#N)=O)CC2)CCc2ncc(Br)n2C1 CC1=NOC(=O)C1CCC(=O)NCCC1CCN(C(=O)COCCCF)CC1 C(C(C)(O)C(C)(C)C)NC(CCC1CC(NC(C(C)N=[N+]=[N-])=O)C1)=O C(C)(CNC(=O)C(=O)NCC(F)(F)F)(C(C)C)NC(c1cc(C)on1)=O O=C1COC(CNCc2cccc(-n3ccnn3)c2)CN1 C(=O)(C(CC(C)C)C1CCCCC1)N(CCCCNC(C=CCC)=O)CCC N1(C(c2c(OC)ccc(Br)c2OC)=O)CCCC(C2CN(C(C3(C)COC3)=O)C2)C1 C=CCC(CNC(=O)CC1COCC1O)NC(=O)Cn1nnc(-c2cccs2)n1 C(CN1C(=O)CCc2ccccc21)NC(C1CCCN(C)C1=O)=O Cc1cccc(N)c1C(N1CCCC(NC(c2c(Br)cnn2C)=O)C1)=O C(=O)(C(C)C(O)CC(C)C)N1CCC(C(C(=O)NC(CCOC)(C)C)F)C1 N1(C(C(C=C)CC)=O)CC(C)CN(C(=O)CCCc2ncco2)CC1C N1(C(c2c(C(=O)OC)cccc2)=O)CCC(F)(F)C(CNC(=O)C(C)N(C)C)C1 C(=O)(C(CC)C(C)O)N(CC(C)NC(CC(CC)O)=O)C C=Cc1ccc(C(=O)NCCC2CN(C(=O)COc3ccsc3Cl)CC2C)cc1 c1(C(=O)NC2CN(C(c3cnc(N(C)C)s3)=O)CC2C(F)F)ccc(F)c(N)c1 c1(C(N2CCN(CCOC)CC2)C(=O)NCc2nnn(C)n2)cc(C)cc(C)c1 C1(C(CNC(C(C)OCC(C)C)=O)(C)C)CCN(C(=O)C(F)=C2CCCC2)CC1 C(=O)(C(C(C)C)C(C)C)N1CCCC(NC(C2N(C(CC)=O)CCCC2)=O)C1 C(=O)(C(CC(C)C)NC(c1csc(CNC(c2ccoc2C)=O)c1)=O)NC N1(C(c2nc(C(C)(C)C)oc2C)=O)CCCN(CCNC(=O)Cc2csnn2)CC1 c1(N(C)Cc2cc(COC)no2)[nH]c(=NC2CC2C(C)C)nc2c1cnn2C C1(C(=O)NC23CC(CC(=O)OC)(C2)C3)CC(=O)N(Cc2ccccn2)C1 Cc1nccn1CCCN.N1(C(=O)CN2CCOCC2)CCC(CCCO)C1 C1(NC(=O)CC=C(Cl)Cl)CC(NC(c2ccc(Br)cc2)=O)C12CCC2 C=CC1CN2CCC1CC2=O.C1(C(=O)NC)CCCOC1 C1(NC(=O)CCn2cccn2)CCC2(CC1)CC(NC(=O)C(O)Cn1cncn1)C2 c1(C(=O)NC(C2(CNC(CCC(CC)C)=O)CC2)C)cc2c(F)cc(F)cc2o1 N1(C(C2CCC(CC)C2)=O)CCC2(CC1)CN(C(C1CC(=C)C1)=O)C2 C12(C(N(C3CCN(C(C(C=CCCC)O)=O)CC3)C)=O)CCC(CO)(CC1)CC2 C12(CNC(=O)Nc3ccc(-c4ccc(Cl)cc4)cc3)CC=CCN1CCC2 c1(C(N2CC(N(C(C(C)CC(N)=O)=O)C)C2)=O)cc(C(F)(F)F)ncc1[N+](=O)[O-] c1(C(=O)NC2CN(C(C=C(C)c3cccs3)=O)C3C2C3)c(C)cccc1F c1(N2CCC(CNC(C3(C)CCC(C)C3)=O)C2)ncccc1C#N C1(NC(C=CC(C)(C)C)=O)CCCC12CN(C(=O)Cn1nc(O)ccc1=O)C2 c1(C(=O)NC(C(C)NC(C(C(C)C)OCC)=O)(C)C)cnc2ccncc2c1 C=C1CCC(C(=O)NC2COCCC2NC(=O)C(C(C)C)NC(N)=O)CC1 c1(C(N2CCC(CCNC(CCCCC)=O)C2)=O)ccc(Cl)c(O)c1N N1(C(CCc2ccc(=N)[nH]c2)=O)CCCCC(CNC(c2nc(Cl)sc2Cl)=O)C1 CCC1=NOC(CC(=O)NCC(CNC(=O)CCc2ccc(Cl)cc2)CO)C1 C1(C(=O)NCCC2CCCC3CC23)CC2(CCC2)CN1C(=O)C(O)C(F)(F)F c1(C(=O)NCC2(F)CCC(NC(C(C)OCC)=O)C2)nccc2c(F)cccc12 c1(C(=O)OC)ccc(S(=O)(=O)N2CCC(N(S(=O)(=O)CCOC)C)C2)n1C N1(C(c2cc(C)[nH]c2)=O)CCC2(NC(=O)CC3CCNC(=O)C3)CCCCCC12 C1(CNC(C2(OC)CCOCC2)=O)CN(C(c2ns[nH]c2=O)=O)CCC1C C1(F)(CNC(C=CC(C)(C)SC)=O)CCN(C(c2c(Cl)nsc2Cl)=O)CC1 CC(CCCC(=O)N1CCOC(CCCNC(=O)CCn2cccc2)C1)N(C)C O(S(=O)(=O)c1ccc(C(F)F)nc1)c1ccc(OCCCC)cc1 C=CCC(Cc1ccccc1)C(=O)NCC(C1CC1)NC(C1(CO)CCCC1)=O Cc1cc(NCC2CC(F)(F)CO2)ncc1S(=O)(=O)NC(C)(C)CF c1(C(c2nnnn2CC=C)NCc2cn(CC#C)nc2)ccc(OC(F)F)cc1 C1(O)(CCS(=O)CC2CCCN(c3ccccn3)C2)CCOCC1 c1(C(CCN(CCOCCOCCNC(CSC)=O)C)=O)cnsn1 C1(O)(CCNC(C(C)(C)OC(C)(C)C)=O)CCN(C(=O)Cc2nnc(O)s2)CC1 c1(CN(C2C(CC)CCCC2)C)cc(C)c2nccn2c1 C(C(CC(F)(F)F)NC(=O)C(C)NC(C)=O)NC(C1(OC)CC1)=O.C(C(C)C)S N1(C(C2C(C)CCOC2)=O)CCCN(C(c2cc(Cl)ns2)=O)CC1 C(C)(C(C)(C)O)N(C(CSCCNC(C(C)n1cncn1)=O)=O)C c1(C(N(C2CCN(C(c3csc(C(C)(F)F)n3)=O)C2)CCC)=O)ncccc1N c1(OC)ccc(CN=C(NCC2CCCCS2)NC2CCC2)c(F)c1 c1(NCC2(NC(C3C(=C)C3)=O)CCCC2)cc2nnc(COC)n2cn1 CCCCC(C)CCC(=O)N1CC(NC(=O)C2=NOC3(CCC3)C2)C2(CC2)C1 N1(CCNC(=O)C=Cc2nccs2)CCN(C(=O)CC2COC(=O)N2)CC1 c1(C(=O)NCC(CC)NC(=O)C#CC(C)C)cc(S(N)(=O)=O)ccc1O CCCC(C(O)C(=O)N1C2CCC1(CO)CC2)NC(c1nn(C)cc1C)=O N1(C(C(CN(C)C)NC(=O)CCc2cnn(C)c2)=O)CCCN2CCCC2C1 CC1CCCCC1C(N1CCN(CCCNC(=O)C(F)F)CC1)=O C(=O)(C1=CCCCC1)N(CC(=O)OC)C.C12(CC1)C(=O)N2 C(=O)(C1=C(C)CCCC1)N1CC2(CC(NC(c3[nH]c(=NCC)sc3)=O)C2)C1 N1(C(Cc2c(C)ocn2)=O)CC(F)CC1CC(=O)NCC1(O)CCOC1 c1(C(N2CCN(CC(=O)NC(C#C)C(C)(C)C)CC2)=O)cccc(F)c1F CC(CC(C)NC(=O)C=Cc1cn[nH]c1)NC(=O)C(C)(C)Nc1ccccc1 c1(C(N2CC(CNC(CCNC(=O)NC)=O)C(C)C2)=O)ccc2c(c1)CCO2 CC1CCN(C(c2cncc(OC(F)F)c2)=O)CC1NC(c1cccc(O)n1)=O c1(C(=O)NC2CCCC(NC(CCCC=C)=O)CC2)cc(C)cc([N+](=O)[O-])c1 c1(C(N(C2CC(F)(F)CC2N)C)=O)cc2cc(F)c(F)cc2[nH]1 C1(C(N2CC3(CN(C(COCC)=O)C3)OCC2)=O)Cc2ccc(F)cc2O1 N1(C(CC(=C=C)C)=O)CC2(CNC(C3(C4CCCCO4)CC3)=O)CC1CO2 N1(C(C(C)NC(C)=O)=O)CCCC12CCN(S(=O)(=O)c1cc(Cl)ccc1Cl)CC2 CC(C(C)(C)C(=O)NC1CON(CC)C1=O)NC(c1cc(Cl)c[nH]1)=O CC(C)C(O)CC(=O)NC1CN(C(c2ccnn2CCN(C)C)=O)CC1C c1(C(N2CC(CC)N(C(c3n[nH]cc3Br)=O)CC2)=O)cc(F)c(F)c(F)c1 c1(C(=O)NC2CCC(N(C(c3c(C)cno3)=O)C)C2)cc2n(n1)CCN(C)C2 C(C)(C(C(C)C)NC(=O)C(=CC1CCCCC1)F)NC(COCCCOC)=O c1(C(=O)NC(CNC(C=CCOC)=O)(CC)CC)ccc(OC)c(N)n1 C(CCN=c1[nH]nco1)OCC(C)C.c12cccc(n1)C(=O)N2 Cc1cn(C)cc1C(=O)NC(C)(C)CNC(c1ccc(SC(F)F)cc1)=O C1(C)(CC(=O)N(CCN(C(=O)C(C)n2cnnn2)C(C)C)C)CC1(F)Cl Cc1noc(Cl)c1CC(=O)NCC1CCC(NC(=O)Cc2cccc(Cl)c2)C1 Cc1ccc(C2(C(=O)NCC(C)NC(=O)CCC(C)(C)C)CC2)cc1Cl c1(-n2c(SCC(N3C(C)(CC)CC3)=O)nnn2)ccc(OC)cc1 c1(C(N2CCC(O)(CNC(C3CC34CC4)=O)C2)=O)cc2c(s1)CCCCCC2 S(=O)(=O)(c1cc(C(=O)NC2(C(=O)O)CCCCC2)n(C)c1)NCc1cccc(C)c1 C12(CNC(C(C)OCC3CCCO3)=O)CC(CN1c1ncnc(=N)[nH]1)C2 c1(COC)n[nH]c(CNC(C2(Nc3ccccc3)CCC2)=O)n1 c1(CSCC(=O)NCCN(C(=O)Cc2nnc(C)s2)CC)cccc[n+]1[O-] C(C)(CO)(C(=O)NCc1cc[nH]c1C(=O)N(C)Cc1ccoc1)OC C1(C(N(CC(C)O)CCO)=O)(CNC(=O)CC2CCCCC2)CC=CC1 c1(CC(N2CC3CC(CCNC(=O)C=O)C2C3)=O)ccc2c(c1)COC2.C(=O)(C1CC1)N CC(C)CCC(O)C(=O)NC(c1ccc(Cl)cc1)CNC(=O)CN1CCCCC1 c1(CC)cc(NC(CNC(=O)CC2(C)CCCC2)CC)ncn1 c1(C(N2CCC(CC(=O)Nc3c(OC)cccc3)C2)=O)cc2cc(Br)ccn2n1 C1(C(=O)NCC=CCOC)C2CC3C(C2NC(C2CC2C(N)=O)=O)C13 c1(NCc2cc(O)cc(F)c2)cccc(NC(C)=O)c1O.C12(CCC1)CC(=O)N2 c1(CC)ccccc1CC(=O)N(C1CCCCC1NC(C1(C)CC1)=O)C c1(C(=O)NCCc2c(CNC(C=CSC)=O)nco2)ccc(CO)c([N+](=O)[O-])c1 c1(C(=O)N(C2CC3(C2)CC(O)C3)CC)cc2c(nn1)CCOC2 Cc1ccc(F)c(C(=O)NC2C3CC2N(C(c2cc(C4CCC4)nn2C)=O)C3)n1 Cc1cc(C(N2CCN(C(c3ccnnc3C)=O)CC2C)=O)c(C)n1C C12(NC(=O)Cc3cc[nH]n3)COC(C1)C(NC(c1cnc(C3CCC3)s1)=O)C2 S(=O)(=O)(c1ccc(F)cc1)N1C(CNC(c2cc(Br)cs2)=O)COCC1 c1(Nc2c(NC(=O)NC3C(OC)CC3)cccc2)cccc([N+](=O)[O-])c1 N1(C(C(C=C)C)=O)CC2(CCCC2CC(N2CCn3nccc3C2)=O)C1 C1(C(=O)NC(c2nncs2)C)CN(C(c2ccn(C(F)F)n2)=O)CC12CC2 Cc1cc(Br)ccc1CC(=O)Nc1ccc(Br)c(O)c1 C1(OC)CC(F)CN(c2nnc(-c3ccc(Br)s3)n2CCC(=O)N(C)C)C1 n1(C(C)C)cc(C(O)CN(C(=O)C(=O)NC2CC2)C2CC2)cn1 c1(OC)ccc(Cl)cc1C(=O)NC1CC(NC(=O)CCCCCN(C)C)C1 C1(O)(CNC(CNC(CC)=O)=O)CCCN(C(=O)CCOC2COC2)CC1 N1(C(CCCC#C)=O)CC(C)CN(C(=O)Cc2nccs2)CC1C Cc1cc(C)n(CC(N2CC3CCC3(CNC(C3CCOC3)=O)C2)=O)c(=O)n1 C(=O)(C1CCCc2c[nH]nc21)NC(CNC(c1n(C)c(O)nc1)=O)C1CC1 S(=O)(=O)(c1ccc(C#N)c(NCC2CCSC2C)c1)N1CCCC(C=C)C1 CC(CN=c1nc2scnc2c(NCC(C)(F)F)[nH]1)C(C)(F)F N1(C(CCC(=C)Cl)=O)CCN(C(c2ccc(C3CC3)nn2)=O)C(CF)C1 Cc1ccnc(C(=O)NC(C)(C)CNC(=O)CN(C)C(N)=O)c1F C(=O)(CCC1=NNC(=O)CC1)N(C)CC1(C)CCCCN1C(=O)OC(C)(C)C CC(C)(C)C(=O)C(=O)NC1CN(C(c2c(O)cccc2F)=O)CCC1C(F)(F)F Cn1ncc2ccc(C(c3ccccc3)NCCCOCc3ccccc3)cc12 c1(C(=O)NCCC(C(C)C)NC(c2c(C)ocn2)=O)cnc2[nH]cnc2c1 C1(O)(CCNC(C2N(C)C(=O)CC2)=O)CCN(C(=O)CC2CCCNC2=O)CC1 Nc1ccc(CNC(C2(c3ccc(F)cc3F)CCC2)=O)cc1Cl C1(CNC(C2ON=C(CC)C2)=O)CN(C(C2CC3CCC2C3)=O)CCC1(F)F C1(NC(=O)C=C2CCC2)CCCN(C(c2ccncc2)=O)CC1F C1(CN(C)CCN2CC(F)(F)C2)CCCN1C(C1CCC(O)C1)=O C1(C(N2CCC(C)(CCNC(CCC(=C)Br)=O)C2)=O)C(C2CC2)C1(F)F C1(OCC)CCC1NC(C)C(C)=C(C)C Cc1sc(N)c(C(N2CC(CCO)(NC(=O)C=Cc3cccc(O)c3)C2)=O)c1C c1(C(=O)NCC2(F)CC(NC(C(CC#C)C)=O)C2)ccc([N+](=O)[O-])cc1 N1(C(CN(C(C(N2CCNC2=O)C)=O)C)=O)CCC(C(N2CCCC2)=O)C1 c1(C(=O)OCc2cc(O)cc(Cl)c2Cl)ccc2c(=O)cc[nH]c2c1 c1(C(N2CCC(=O)NC2=O)Cc2ccc(C)cc2)cccc(S(C)(=O)=O)c1 C1(CN(C(=O)C(CO)c2ccccc2)C)CCCN(C(C2CCS(=O)(=O)C2)=O)C1 C(=O)(CCCC(F)F)N1CC(NC(C2(C)C=CCC2)=O)C(n2cccn2)C1 C1(CC(=O)NCC(CC)(C)OC)Cc2ccccc2CN1C(c1cc(C)co1)=O N1(C(C(C)NC(C)=O)=O)CC=CC1C(N1CC(CN=[N+]=[N-])C1)=O C(=O)(C1=NNC(=O)CC1)N(C(CNC(C1CCC(=O)N1)=O)C1CC1)C c1(OC)ccc(C(=O)NCC(C2CC2)N(C(=O)C(C)n2ccnn2)C)c(O)c1 c1(NCC2CN(C(C(CC)OC)=O)C(C)C2)nc(Cl)nc(CC)c1C#N C(=O)(CCC(=O)C(C)(C)C)N1CC(O)(CNC)C1.c1(COC)ccsc1C=O C12(C(N3C4C(CNC(c5c(C(C)C)ccs5)=O)C(C4)C3)=O)CCCC1CC(=O)C2 CC(CCCNC(=O)CC1(O)CCCC1)NC(C1(c2ccno2)CCC1)=O CCCC(CCCO)C(=O)NCCOC1CN(C(C2CCCCC2(C)C)=O)C1 C1(c2n(C)nnn2)(NC23CCC(N4CCCC4)(CC2)C3)CC2CCOC12 CCCS(=O)(=O)C(C)C(=O)NCC1CC2(CC2)CN1C(=O)C(C)OCCN(C)C C12(CC(=O)NC(CC=C3CC3)=O)CCC1CN(C(c1nonc1N)=O)C2 CC1(C)CC(C(=O)NCC2(C)CCCN(C(=O)C=Cc3ccc[nH]3)C2)CCO1 N1(C(CCOCCN(C(c2c(CC)cco2)=O)C)=O)CCS(=O)C(C)C1 CC#Cc1cncc(-c2cscc2C(=O)NC2(C#N)CCOCC2)c1 C#CC1CN(C(=O)CC2C=CCCC2)CCN1C(c1cc2ccccn2n1)=O n1(CCCC)cc(C(=O)NCC2CC2NC(=O)CC2(NC(C)=O)CC2)nn1 c1(C(N2C(C(C)NC(=O)Cn3cccn3)CCCC2)=O)c[nH]nc1S(N)(=O)=O N1(C(CCCC)=O)CCC2(CC1)CC(NC(=O)C=C1CCCC1)CO2 c1(C(N(CCCCNC(c2ccncc2)=O)C)=O)cccc2c1CCC2 C1(CC)(CC)CN(c2nnc(Cc3ccccn3)n2CCOC)CCS1=O c1(C(N2C3CN(C(CC4CCN(C)CC4)=O)C(C3)C2)=O)nccc2ccccc12 c1(C(=O)NC2CCC(C)(CNC(c3c(C)c[nH]n3)=O)C2)cc(C)c(C)c(Cl)c1 c1(CC(=O)N(CCCNC(=O)CC2C=CCCC2)C2CC2)ccc2nn[nH]c2c1 N1(Cc2c(C(=O)OCC)cccc2)CCC(NC(C2CC(=O)N2)=O)CC1C c1(C(=O)NC2(CNC(C3(C)CC3(Cl)Cl)=O)CC2)nn(C(C)(C)C)cc1Cl N1(C(C(CC)NC(N)=O)=O)CC2(CCN2C(C2CCCC2C(F)(F)F)=O)C1 Cn1cc(Cl)c(CC(=O)NCCCCNC(c2ccc(C3CC3)s2)=O)n1 Cn1ccc2cc(-c3nn[nH]n3)ccc12.C12=NC(C)=CC(=NCC3CCCCC13)N2 C1(COC)(CNC(C2CC2CF)=O)CCN(C(C2CC3C(C2)C3(F)F)=O)CC1 n1(CC)cc(C(=O)NC(C)(C)CC(C)(C)C=CC(=O)Nc2coc(SC)c2)nn1 c1(OC)ccc(F)cc1NCC1(O)CCN(S(=O)(=O)C2CCC2C(=O)O)CC1 C(=O)(CCCC(N)=O)NCC(C1CCCN(C(C2CC3CCC2CC3)=O)C1)(C)O c1(C(=O)NC2CC(NC(c3cc(Cl)c(Br)[nH]3)=O)C2)cccc2c1CCOC2 CC(C)(Cn1cc(C(C2CCCC2)O)nn1)CC(F)F c1(C(N(CCN(C(=O)CC(C)F)CC)CC)=O)ccc(O)c(C(C)C)c1 CCC(C)(CO)C(=O)NCC(C(C)(C)C)NC(c1cc(O)cc(O)n1)=O CC1(Br)CC1C(=O)N(CCCN(C)C)CCNC(=O)Cc1cccs1 C(=O)(CCCC(F)F)N(C)CC1CCN(C(=O)Cc2cnccn2)C1 C(=O)(CC1OCCc2sccc21)NC1(CCCCNC(c2c(C)cccc2)=O)CC1 c1(CC(N2CC(C(=O)NC3CN(C)CC3O)OCC2)=O)ccc(S(C)(=O)=O)cc1 c1(C(N2CCCC2C2CCN(C(C3CCS(=O)(=O)N3)=O)C2)=O)cnc(C)nc1N.CO C1(C(=O)NCC(CC)NC(C2CN3CCC2CC3)=O)CC1C1CCCC1 c1(NC(C)CNC(c2ccc3c(c2)CCCS3)=O)ncc2ncn(C)c2n1 C1(NC(C2CC(N(C)C(c3n[nH]cc3C3CC3)=O)C2)=O)CC2CCC(C1)C2O C1(C)(CCNC(CC2C(C)(C)CC2)=O)CCN(C(c2c[nH]nc2Cl)=O)C1 C(CS(=O)(=O)CC(=O)N(CCC(N1CCC(CC(C)(C)C)C1)=O)C)OC c1(C(=O)NC2CC(C)(NC(C=C(CC)CC)=O)C2)ccc2snnc2c1 C1(C)(CC)C=C(C(=O)N2CCCC(NC(C3CCCO3)=O)C2C)C1 CCCCCCCC(O)C(=O)NCCCCCNC(c1nncn1C)=O C1(c2onc(-c3cc(C)c(Br)cc3)n2)CCN(C(=O)OC(C)(C)C)C2COCC12 C(CCC(=O)N1CC(O)(CN(C)C(C2CCC(C(N)=O)C2)=O)C1)OCCOC C1(F)(C(=O)Nc2c(OC)cccc2)CCCN(C(c2cc(C(N)=O)no2)=O)C1 C(N=c1[nH]c(-c2ccccc2)nc(=NCC=C(Cl)Cl)[nH]1)N1S(=O)(=O)CCC1 N1(C(CN2CC(C)(OC)C2)=O)CC(CCNC(C2CS(=O)(=O)C2)=O)OC(C)C1 c1(C(=O)NCC2(OC)CCN(C(C3CNC(=O)N3C)=O)C2)cc(C)c(C)c(F)c1 c1(NC(=O)NCCN(CCCC)C)ccc2c(OC)nccn12 C1(NC(CCSCC(C)C)=O)CC2(C1)CC2NC(=O)CC(C)c1ccco1 c1(OC)ccc2c(n1)NC(C(=O)NC1CCCCN(C(C3CC=CCC3)=O)C1)C2 C1(C(=O)NC(c2nc(C)[nH]n2)C)CCN(C(c2ccc(CC#N)cc2)=O)C12CC2 C1(CC(=O)NCC(COC)NC(c2n[nH]cc2Cl)=O)CCC(OC)CC1 N1(C(c2c(C)noc2)=O)CCC(C2CC2)(CNC(=O)C=Cc2cnccn2)C1 n1(NC(CCOC)(C)c2nnnn2C(C)C)cc(C)ccc1=O CC1CCC(NC(C2CN3CCC2CC3)=O)CN1C(c1ccc(CO)nc1)=O C1(C)(NC(CC2N(C(C(CC)COC)=O)C3CCC2C3)=O)CC(C)(C)OC1=O C1(CNC(CSCCCC)=O)(NC(c2ccn(C(C)(C)C)c2)=O)CCCCCC1 c1(N2CC(S(=O)C3CCN(CC(F)F)CC3)CC2)nccc2c(Cl)cncc12 Cc1cc(C(=O)NC2CCCC(C(=O)NCCOc3ccc(Cl)cn3)C2)cn1C c1(C(=O)NC(C(=O)N(CCC(=O)OCC)C)Cn2ccnn2)ccccc1O c1(C(=O)NC2CC3CC(OCC)C3C2)c(C(F)(F)F)cc(F)cc1F C1(C)(OC)CCCN(C(C(=O)Nc2c(C)cccc2C)C(C)C)C1 Cc1ccc(CNC(=O)COC2CCN(C(C3CCC(C(N)=O)C3)=O)C2)c(F)c1 n1(CCC(=O)NC(CNC(C2N(C)CCC2)=O)C2CCC2)ccc2ccccc12 c1(C(N(CC(O)CN(c2cc(O)nc(C3CC3)n2)C)C)=O)cnc2ncccn12 N1(C(c2scc(CNC(COC(C)=O)=O)c2)=O)CCC2(CCOCC2)C1 C1(NC(=O)OCC)CCCN(C(=O)Nc2cccc(C3(C)CCO3)c2)C1 C12(C(N3CC(CCNC(CC4CCC(C)CC4)=O)C3)=O)CCC(C(F)F)(CC1)C2 c1(C(=O)OCC)cc(NC(=O)NCC2(COC)CC=CC2)cc(SC)c1 N1(C(c2coc(C(F)F)n2)=O)CCC(c2ncco2)CC1 C1(COC)(CNC(C2CC(SC)C2)=O)CCN(C(=O)Cc2ncsc2Cl)C1 CC1(C)CCN(C(C2CC2c2ccccc2Cl)=O)CC1NC(C1CCC1)=O C(CCOC)(C(=O)N(C(CO)C1(O)CC1)C1CC1)NC(C(N1CCCCC1)C)=O C(C(CNC(c1ccc(CO)cn1)=O)S(C)(=O)=O)NC(CCCC=C)=O c1(NC(C)=O)nc(C(=O)NCC(C2CC2)N(C(=O)CCn2cnc(C)c2)C)cs1 N1(C(C(C)NC(=O)OC)=O)CCCC(F)(C(=O)NC2(CO)CC3(CCC3)C2)C1 N1(CCOC)CC(C(N2CCC(c3scnc3C)CC2)=O)CC1=O c1(NCc2cc(C)cc(C(F)(F)F)c2)cccc2c(OC(F)F)nccc12 C(=O)(C(C(C)C)N(C)C(=N)NC(C)=O)NCC1CCC(CNC(CCCC)=O)C1 N1(C(CN(C(C)=O)C)=O)CCCC(C(C)NC(c2csc(C3CC3)n2)=O)C1 C(=O)(CCCCCC(C)(C)C)NCCC(C)NC(c1nc2ncc(C)cn2n1)=O c1(OCC)ccc(C(=O)NC(C)(CNC(=O)CC2CCC(=O)N2)C(C)C)cn1 c1(C(=O)NC(C)CCN(C(=O)C(F)=C2CCC2)C)cc(F)c(F)c(F)c1F C(C)(CCC(=O)NC1CCC(F)(CNC(=O)CCc2ccc[nH]2)C1)SC Cc1nccc(C(N2CCOCC2CN(C)C(c2cn(C)nn2)=O)=O)c1O CC(C)CCC(O)C(=O)NCc1nocc1C(=O)NC1CC1CN(C)C C1(C(=O)NC2C(C(N)=O)CCCC2)CC2(CCN(C(C34CCC(C3)OC4C)=O)C2)C1 c1(OCCC(=O)N(CC(C)NC(C2CC2(C)C)=O)C)cc(F)ccc1F c1(NCC(C)NC(C2CN(c3cc(C)[nH]n3)C(=O)C2)=O)cnc2n1CCCC2C c1(CNC(C(C)(C)O)=O)cc(C(=O)Nc2cncc(Br)c2)ccn1 C12CC3CC(CC13)NC(=O)C(=O)N2.C(C1CCC1)=CC(=O)N.C(COCC)OC C1(N(C(=O)NCC(C2CC2)OC)CC2CC2)CCN(c2nccs2)CC1 Cc1cccc([N+](=O)[O-])c1C(=O)NC1COCCC1NCc1cccc(F)c1F C1(CC)CN(C(C)C)CCN1C(=O)NCCc1cn[nH]c1 CC(C)CC(C)CC(=O)N1CC=CC(NC(c2cc(O)nc(N(C)C)n2)=O)C1 C1(C(=O)OC)CCN(c2nnc(-c3ccc(CO)o3)n2Cc2ccccc2)CC1 C(C)(CCCNC(C1CCC(OC2CC2)C1)=O)NC(CC1CC(OC)C1)=O C1(C2=NOC3CC23)C(=O)N1C.Cc1cc(CNC2(C)CCC2)sn1 c1(C(=O)NC2(C(=O)NC3CCC(O)C(O)C3)CCSC2)ccn2ccnc2c1 C1(CNC(c2ccc(CCC)s2)=O)CCCCC1NC(c1cnc(C)nc1)=O C1(C(=O)NCCCN(CCCNC(C2N(CC)CC2)=O)C)CC1[N+](=O)[O-] c1(OCC)ccc(-c2noc(C3CC(F)C(=O)N3)n2)cc1 CC1CCCC(C2=NOC(C(=O)Nc3ccc(Cl)nc3)C2)C1 C=CC(CC)C(=O)N(c1cccc(C(F)(F)F)c1)CCO N1(C(CCOC)=O)CCC(CNC(=O)CN2CCC(C(F)(F)F)CC2)C12CC2 c1(C(=O)OCC2CCC(NC(C)=O)CC2)nn(C)c2ccccc12 c1(C(OCOC2CC(C(=O)OC)C2)=O)cnn(Cc2nn[nH]n2)c1 c1(CC(=O)NC(CNC(C(F)OC)=O)C)coc2cc(C(C)(C)C)ccc12 CC1CCCC1(C)NC(c1c(CNC(c2cc(Cl)cn2C)=O)cnn1C)=O N1(C(C2(CC)CCCO2)=O)CCC2(CC=CCO2)C1.c1(CNC=O)cnnn1C C1(NC(CC2C(C)CCO2)=O)CCC(C)N(C(c2cc(F)ccc2O)=O)C1 CCCC(CC)CCC(=O)N1CCC=C(C(=O)N2CC(C)(CSC)C2)C1 n1(CCC)ccnc1C(C)NC(c1ccc(CC)o1)c1nnnn1CCC C1(CC(=O)NCCCO)CCCCC12NC(=O)NC2=O N1(C(c2c(CC)nco2)C(=O)NC2CCOCC2)CC(C)(C)OCC1C(F)(F)F c1(C(N2CCC(CN(C(C(n3c(C)ncc3)C)=O)C)C2)=O)cc(F)c(N)cc1F C1(NCc2c(F)cc(C3CCC3)cc2)CS(=O)(=O)C12CCCC2 c1(C(C)C)ccc(C(=O)NCC2CC(F)CN2C(=O)CCCCC2CC2)nc1 CCC(C)(F)C(=O)NCCn1cc(C(=O)NC2CC(=O)N(C3CC3)C2)cn1 C1(C(=O)NCC(CC=C)NC(=O)Cc2ccc(C)nc2)Cc2ccc(F)cc2C1 C1(CC(=O)NCCCN(C(=O)COC2CCOC2)C)CCCCC(=O)N1 N#CC12CN(C(=O)Nc3ccc(O)cc3)CC1CS(=O)(=O)C2 C1(NC(CC2(OC)CCC2)=O)CCCCC12CCCN(C(c1cnoc1)=O)C2 N1(C(C2CCN2C(=O)C(c2ccccc2)F)=O)Cc2ccc([N+](=O)[O-])cc2C1 C=CCC(F)(F)C(=O)NC1C=CC(CNC(=O)C(C)(O)C(C)C)C1 N1(C(C(C)C)=O)CCCC1C(N1CC(C)(NC(c2cc(-c3cccs3)[nH]n2)=O)C1)=O Cc1cscc1C(=O)NCC1CCN1C(=O)CC1CC=CC1 Cn1nc(COC)c2c1CCN(c1ncnc(Cl)c1C(F)F)C2 Cc1ccc(C(N2CC(C(=O)NCC3(C#N)CCC3)C(F)C2)=O)c(F)c1 C1(C(N2C(CN=[N+]=[N-])CCC2)=O)N(C(C2(N3CCCC3)CC2)=O)CC12CCCC2 Cc1cc(CC(=O)N(C(C(=O)N(C2CCCC2C)C)C2CC2)C)no1 c1(C(C(N2CCC(NC(C3(OC)CCC3)=O)C2)=O)O)ccccc1Cl c1(-c2cccc(C(=O)OCC)n2)cc2n[nH]cc2cc1C n1(CC)ccc(CC(=O)NC2C(C(=O)NCC(C)(O)C3CCC3)C2(C)C)n1 CC(CC(=O)OCC(C(F)F)n1cccn1)n1cccn1 C1(C(=O)NCCn2c(C)cnn2)CCN(C(=O)CC2CCOC2=O)CC1 Cc1cncc(CCC(=O)NC(C)C(CO)NC(=O)C(O)Cn2cncn2)c1 N1(C(C2CCCN(CC)C2)=O)CCC2(NC(=O)Cc3sc(O)nc3O)CCCC12 C=CCCCCCCCCCNc1ccc(N2CCN(C)CC2)c(Cl)c1 C1(O)(CC(=O)Nc2ccn(C(F)(F)F)n2)CCN(CC(N2CCCCC2)=O)CC1 C1(C(N2CCC(NC(C)(C)C)CC2)C(=O)NCCC(=O)OC)CCC2(CC1)CC2 C1(C(C)C)NC(=O)N(C2(N(C)C(=O)NCCc3nc[nH]n3)CCCCC2)C1=O CCCC(CC)C(=O)NCCC1(C(=O)N(CCC(C)(C)C)CC)CC1 N1(C(C(C(CC)CC)C)=O)CCCC(C2CCN(C(C3C4COCC34)=O)C2)C1 C(=O)(C(CC)C(=O)NCC1CC1NC(=O)CN(C)CC)OCC CP(C)(=O)C(O)C(=O)NCC1(C)CCC(NC(=O)C=C2CCSCC2)CC1 C12(CNC(C(C3(O)CCC3)NC(C=CC)=O)=O)CC(C)(CCO1)C2 C1(C(N2CC(O)(CNC(c3ccc(C(=O)OC)o3)=O)C2)=O)CN2CCN1C(C)C2 CCC(CC)(CN=c1ccnc(NCc2nc(C(C)C)n[nH]2)[nH]1)OC c1(CNC(c2ncccc2F)CC)cc(F)cc(I)c1 C1(C(=O)NCC2(NC(COc3ccc(C)cc3C)=O)CC2)CCn2nnnc2C1 C1(NC(c2c(C)nc(CO)s2)=O)CN(C(C2CCCSC2)=O)CCC1C CC1=CC(C)=NS(=O)(=O)N1CC(N1CC(F)(F)CC1CNC(C1OCCO1)=O)=O C12(CCC(C)(N3CCCCC3)CC1)C(=O)N2.Cn1c(C2CCC2)noc1=O C1(C(=O)Nn2ccc(CNC(C3(N(C)C)CC3)=O)n2)CN(C(N)=O)CCN1C S(=O)(=O)(c1cccnc1N1CCCC(C)(C)C1)NCC(C(=O)NC)C N1(C(c2nc(=NC)[nH]c(C)c2)=O)CCC2(CCCN(C(C34CC3C4)=O)C2)C1 Cc1ccc(F)cc1-c1noc(C2CC2)n1.NC(=NCC1CCCC(C)C1)NC1CC1 c1(C(=O)Nc2cncc(-c3ccc(-c4ccccc4)s3)c2)cnc2ccccn12 C1(C(N2CCOCC23CC3)C(=O)NCCC2(C)CC2)CC2CCC1CC2 O=C(C1=CCN(C(=O)C=Cc2ccc[nH]2)CC1)NC(CO)CCO CC(CC(=O)N(CCC(=O)NC1CCCCC1(F)F)CCCO)C(F)F C1(C(=O)NCCCOCC)CCN(C(=O)CN2CCC(C)C2)C12CC2 c1(Nc2c(-c3c(OC)ccc(OC)c3Br)nccc2)nc2c(C)cccc2s1 N1(C(C)C(=O)NC(CO)C(=O)NC(C)(C)C2CC2Nc2ccccc2)CCCCCC1 N1(C(C)C(=O)NC2CC(CNC(=O)C=Cc3ccncc3)C2)CCP(C)(=O)CC1 CC(C(=O)NCC(C)(C)CN(C(=O)C(F)(F)C(O)c1ccccc1)C)S(N)(=O)=O C=C(C)C1CN(C(C2(C)C=CCN2C(c2ccc([N+](=O)[O-])[nH]2)=O)=O)CCO1 Cc1nn(CC(=O)NCC(C)(C)C(=O)NCCCCCF)c(=O)o1 C1(N(C(C2(COC)CN(C(C3CCSC3)=O)C2)=O)C)CCCCC1(C)C C1(NC(c2c(SC)n(C)nc2)=O)CN(C(c2sccc2C(C)=O)=O)CCC1CO CC1=C(C(=O)N2CC(CC(=O)NCC(Cl)C(C)(F)F)CC2(C)C)CCCO1 C1(NC(C(C)SCCCC)=O)CC2CN(C(=O)Cc3cc(C)ccc3C)CC2C1 N=c1ccc(C(N2CCC(OC3CCCCC3)C2)=O)c(Cl)[nH]1 c1(C(=O)NCCCCC(C)NC(CC2C(OC)COCC2)=O)cc(C)cc(F)c1 N1(C(CC(CC)CC)=O)CC(C)CN(C(c2conc2C2CCCC2)=O)C(C)C1 c1(OC)nc(Cl)ccc1C(=O)N(C(C)CCNC(=O)CC(=O)N(C)C)C C(C(C)(C)C(=O)N1CC(O)CC1CC(=O)NCC1CCCCO1)OC(C)C C1(C(C)C)N(C(c2cscn2)=O)CC12CCN(C(=O)CCC1CCC(C)O1)CC2 c1(C(N2CCC(CN(C(c3cc(OC)n[nH]3)=O)C)C2)=O)cncc(F)c1Cl N1(C(C(C)CO)=O)CC2CCC1CN2C(=O)C(c1cnn(-c2ccccc2)c1)=O CCCC(C#N)C(=O)NCCN(C)C(c1cc(C)ccc1NS(C)(=O)=O)=O C(=O)(CC(C)C(F)(F)F)N1CCC(CNC(c2cccc(OC)c2)=O)C1 C1(NC(C(CC=CC)C)=O)CC2CC1N(C(c1ccc(F)cc1C(F)(F)F)=O)C2 C1(C(=O)OC)CCC(C(N2CCC2Cn2cc(C3CCOC3)nn2)=O)CC1 Cc1cc(CNC(=O)C(C2CCC2)NC(c2cccnc2C)=O)cc(C)n1 C(CC)(C(=O)N(CCC(C)(C)NC(C1CC1(Cl)Cl)=O)C)=CCCC C(CC(C)(C)C(=O)N1CCCC(CC(N)=O)C1)NC(C(CCC)OC)=O C1(C(=O)NC2(CCNC(c3cc(CC)no3)=O)CCC2)CNC(=O)CC1C N1(C(c2cnc[nH]2)=O)CCCC(N(CCF)C(C23CC(C)C2C3)=O)C1 C1(C(N2CCC(NC(c3ccc(C(N)=O)o3)=O)C2)=O)CN2CCCC2CO1 O=C1CNc2ncc(C(N3CC(CNC(C4CC=CCC4)=O)C(O)C3)=O)cc2N1 C(=O)(CC1OCc2ncccc21)NCC1CC(C)(C)CN1C(=O)CCCF N1(C(c2cc(C)c(O)nn2)=O)CCC(C)(C)C(C(N2CC3CC2(C(F)F)C3)=O)C1 CC(N)(CS(C)(=O)=O)C(=O)NCCc1nc2cc(F)ccc2o1 c1(OC)ccc(C(N2CCC(C)C2CNC(C2CC3(CC3)C2)=O)=O)cn1 C1(C(=O)NCCC2CCCN(C(C3CN(C)C(=O)N3)=O)C2)(CC)CCCCO1 c1(OC)ccc(C)c(NC(=O)CC2CC(C)N(C(=O)C3=CC(C)(C)C3)C2)c1 C1(NC(CC2C(C)C2)=O)CC2CCC(C1)N2C(=O)Cc1cnc(C(F)(F)F)s1 N12CC3(CCC(C3)NCCOCCC1=O)C2.c1(CO)csc([N+](=O)[O-])c1 CC(C)CC(C)C(=O)NC1(c2cn(CCNC(=O)CC(C)(C)C)nn2)CCOCC1 c1(C(=O)NC2CC(NC(c3c(CC)cccc3CC)=O)C2)cc(S(N)(=O)=O)c[nH]1 CC1CN(C(=O)C(=O)NCCC(N)=O)C(C)CN1C(c1ccc(Cl)c(N)c1)=O N(C(=NCCc1ccc(F)cc1)NCCS(=O)(=O)N1CCCC1)C1C(C)C1 C(=O)(CC(CN(C)C)C(F)F)NC1(CCC)CCN(C(C(C=C)O)=O)CC1 C1(N=[N+]=[N-])(C(=O)NC(C)(C)CNC(=O)CCCC2CCCC2)CCOCC1 N1(C(C2CN(C(C3CC(F)(CF)C3)=O)CC2F)=O)CC(O)(C2CCC2)C1 C(C(N=[N+]=[N-])C(=O)OCc1ccoc1C(=O)NCC1COCCOC1)OCC c1(C(N2CCC(CNC(CCCOCC)=O)C2(C)C)=O)ccc2cc[nH]c2n1 c1(CC)nocc1C(=O)NC1CC1COC.C12C=CCN1C2=O c1(CC(=O)NCCC(C)NC(Cc2nnc(C)s2)=O)csc2ccccc12 C(CC(C)C(=O)NC1CC(CNC(C2(C)CCOC2C)=O)C1)=CC N1(C(Cc2cn(C)nc2Cl)=O)CCOC(C)(CNC(c2cn[nH]c2)=O)C1 c1(CCCNC(c2n(C(C(=O)OC)C)nnn2)CCCC2CC2)cccc(Br)c1 Cc1cc(Cl)cc(NC(=O)CCC2CCCN2C(C2CCCCC2(F)F)=O)c1Cl CCC(F)(F)CC(=O)NCC1(F)CCC(NC(c2cncc(Br)c2)=O)C1 N1(C(c2c[nH]c(=NC)s2)=O)CC2(CCN(C(C3CCCN3C(=O)C3CC3)=O)C2)C1 C1(C(N2C(CCOC)CN(C(=O)CCC(C)(C)O)CC2)=O)CCCCC12CCC2 Cc1ncc(C(=O)NCCC2CC(NC(C3(n4cnnn4)CC3)=O)C2)n1C CCC(C)(CCC(C)C)C(=O)N1CCCN(C(=O)CCCN=[N+]=[N-])C(C(C)C)C1 C1(C(N(CCC)CCNC(C2CC3(CC3)C2)=O)=O)(COC)CCCCO1 C(CCC(O)C(=O)NCc1cn(C)nn1)NC(C=CC)=O C1(NC(c2c(NC(C)=O)c[nH]c2C)=O)CC2CC(C1)N(C(C)CN(C)C)C2 Cc1c(C(=O)NC(C)CNC(c2scnc2C(C)(C)C)=O)ccn1C1CC1 c1(NC(C(CC(C)C)O)=O)cccc(Cl)c1C#N.C12C3CN(CC13)C2=O Cc1nc(O)nc(O)c1CCC(N1CC(NC(=O)C=CBr)C(C)C1)=O c1(C(N2CC(NC(C(C)CCO)=O)CC2(C)C)=O)ccnc2ccc(F)cc12 N1(C(CCCC(=O)OC)=O)C(CNC(=O)Cn2cnccc2=O)CC2COCC12 CCCCC(C)CCC(=O)NC(C(=O)N(C(C)CC(=O)OC)C)c1ccoc1 C1(C(=O)NC(C2CN(c3nc4ccccc4s3)C2)C)CCc2ncncc2C1 c1(C(=O)Nc2ccc(C)c(OCC(F)(F)F)c2)cc(S(=O)(=O)N2CCC2)c[nH]1 c1(OCC)oc(C)nc1C(N1CCC(CF)(NC(C23COCC2C3)=O)C1)=O CON1CCC(C(=O)NC(C2CC(CCCc3cn(C4CCC4)nn3)C2)=O)CC1 C(=O)(CC(CC)C(C)(C)C)N1CCCC(N(C(CCC#CC)=O)C)CC1 CCCCCC(O)C(=O)N1CCCC(C)(NC(C2CCC(C3CC3)CC2)=O)C1 c1(OC)cnc(C(=O)NC2(CO)CN(C(=O)C=CCO)C2)c(F)c1 N1(C(C2C(C(C)C)(CC)C2)=O)C2CCCC1CN(C(=O)CCN(C)C(C)=O)C2 N1(C(CCC=CC)=O)CCC(COC)(NC(c2ccncc2N)=O)CC1 N1(C(C(CCC)C)=O)CC2(CCC(CNC(=O)CS(=O)(=O)NCC)O2)C1 c1(OC)nc2ccc(C(N3CC(C)CN(C(=O)CC4CSC4)C(C)C3)=O)cc2[nH]1 C(CCN=C(NCc1cnn(CC(F)(F)F)c1)NCC1CCOC1)(C(F)(F)F)OC c1(CC)ccccc1C(=O)NC(C(=O)NC1(C)CC(N(C)C)C1)C(C)C Cc1cc(NC(=O)CCOC2COC2)ccc1NC(=O)C(F)(F)C(F)F c1(C(N2CCN(C(=O)CC3CC=CC3)C(CF)C2)=O)cc([N+](=O)[O-])n[nH]1 c1(NC(CN2CCC(c3ccc(C)cc3)C2)=O)ccc2ncc(C=NO)n2c1 Cc1ccc(NC(N2CC(C)OCC2C)=O)cc1N1CCCS1(=O)=O N1(C(C2CCN(C(=O)CNc3ccccc3)CC2)=O)CCC2(CCCCO2)C1 C1(CC(=O)NC(CNC(CS(=O)(=O)NCC)=O)C2CC2)CC2(CCC2)CO1 c1(C(C)C)cc(-c2ccccc2)sc1NC(C1CC(O)CN1C(=O)C(C)NC=O)=O n1(CC(N2CC3C(CNC(C4(C)CCC4)=O)(C3)C2)=O)cnc([N+](=O)[O-])c1 c1(CC(=O)NCC(C)N(C(c2cn(C3CC3)nn2)=O)CC)cccc(Cl)c1 N1(C(C2(CC#C)CCCCO2)=O)CCCOC(CNC(c2ccoc2)=O)C1 C1(C(N(OC)CC2CC3CC3C2)=O)CCCN(C(c2nocc2C)=O)CC1 c1(C(N2CC(NC(c3ccncn3)=O)CC23CCC3)=O)cc2c(cn1)OCCC2 Cn1nc(CN(CCC(=O)NC(=O)COC2CCCC2)CCCO)oc1=O CCC(C(=O)NCC1CCC(F)(CNC(=O)CCn2ccc(C)n2)C1)C(C)C C(=O)(CCCC(=O)NC(C(=O)NCCc1scnc1C)C1(C)CC1)OCC N1(C(C(C)NC(C)=O)=O)CCCCC1CN(C)C(c1cocn1)=O CC1CN2CCN1C(C(=O)NC1CC3CCC1C(NC(c1cscn1)=O)C3)C2 C1(NC(c2ncn(C(C)C)n2)=O)CN(C(=O)CC#N)CC1C C(=O)(C(C)CC(=O)OCC)NC(CC)CNC(c1cc(C(F)(F)F)ns1)=O C1(C(=O)NC(CCC)CNC(C2(CC)CC2)=O)NC(=O)CC1C(F)(F)F N1(OC(c2c(Br)ccc(SC)c2)=O)CCC12CCS(=O)(=O)C2 C12(CNC(C)=O)CC(C1)C(NC(C1(NC(=O)C3CC3)CC1)=O)CO2 Nc1cc(C(=O)NCC(Cl)NC(=O)CCC2CCCO2)c2ccccc2c1 Cn1cc([N+](=O)[O-])c(CC(N2CC3CCC2C(NC(=O)COc2ccsn2)C3)=O)n1 C1(C(=O)NCC2(COC)CN(C(C3CC(F)(CF)C3)=O)C2)CCNC(=O)C1 C1(NC(=O)CC(C2CC2)C2CC2)CCN(C(c2cc3sccc3[nH]2)=O)CC1F C1(c2n(C)nnn2)(NCCCc2ccccc2OC(F)F)CCCC1OC(F)(F)F Cc1cc(C(=O)NCC2CC2CNC(C2(C)CCCC2(F)F)=O)c(C)cc1Cl n1(CC)cc([N+](=O)[O-])c(C(=O)NCC2CCC(CNC(c3cocn3)=O)CC2)n1 C1(NC(CCC)=O)C2CCCN(C(=O)CCC3CCCCO3)C2C1(C)C C(C)(c1ccco1)=CC(=O)N(C(C)C(=O)NCC1CCOC1(C)C)CCC Cc1nc(N2CC(NC(c3cc(Cl)nc(Cl)c3)=O)C(C)(C)C2)cc(O)n1 N1(C(c2cn(C)c(Br)c2)=O)CCC(NC(=O)CN2CCCC2)C12CC2 CCC(C#N)(CC)C(=O)N1CCC(N(C(=O)CC2C=NN(C)C2=O)C)C1 C1(CN(C(c2ccn(CC)n2)=O)C)CCCCN1C(=O)COc1ccc(F)cc1 N1(C(c2c(C(=O)OC)c(C)cs2)=O)CCCN(Cc2cn(CCC3CC3)nn2)CC1 N1(C(CC2CCC(C)CC2)=O)CC2CCCC(CNC(c3cscc3F)=O)C2C1 N1(C(C)C)C(=O)CCC1C(=O)NC1CC1CNC(c1ccc(C(N)=O)nc1)=O Cc1ccncc1C1CCN(C(=O)NCC2(N(C)C)COC2)CC1 C12CC3CCC1(C3)NN(c1cc(C)on1)C(=O)c1cn2nn1.C(=O)(COC(F)F)OC.C CC(C)C(O)C(C)C(=O)NC1CC2(C1)CN(C(c1ccccc1SCCO)=O)C2 C1(NC(CC2OCCN(C(CCc3ccn(C)n3)=O)C2)=O)CCC2(CCC2)CC1 c1(NCCNC(CN(CCOC)CC)=O)ncnc(OC)n1 c1(CC(=O)NCC=CCNC(Cn2ncc(C#C)c2)=O)ccc2ccn(C)c2c1 C(=O)(C1=CCC(F)(F)CC1)NCC(C1CCN(C(c2c(C)nc(C)s2)=O)CC1)F c1(C(=O)NC2CN(C(C3CCC(CC)CC3)=O)C(C)C2)ccc(N(C)C)c(F)c1 Cc1cc(CCC(N2CC3COCC2C3)=O)cc(C)n1 c1(C(=O)NC(C)CNC(=O)CP(C)(C)=O)cc2c(o1)CCCC2 CC#CCCCC(=O)N1CCC1c1cn(C2CCC(=O)N(C3CC3)C2)nn1 c1(C(N(CC(C)C(=O)N(CCC(F)(F)F)C)C)=O)cccnc1S N1(C(c2c(O)ncc(CC)c2)=O)CC(C)CN(C(=O)CCCOC(C)(C)C)C(C)C1 CC1(CC(=O)NCC2CC(NC(c3ccnn3CCF)=O)C2)CCCO1 C(c1cnccn1)=CC(=O)N(C1CCN(C(C2CC(C#N)C2)=O)CC1)CCC Cc1cnc(CC(=O)NC(CNC(=O)Cc2cnc(C)o2)C2CC2)[nH]1 C1(CSC)CCN(C(=NCCc2c(C)nn(C)c2C)NCCc2cccs2)C1 C1(CC(C)NC(=O)Cc2ccno2)CC2CCC(C1)N2C(c1ccc(O)cn1)=O C=CC(CC)CC(=O)NC(C(=O)NCc1noc(C(N)=O)n1)C1CC1 N1(C(C(CC)C)=O)CC2(C(=O)NC3CN(CC(F)F)C3)CC1CO2 CC1CCC(NC(=O)CSCc2ccccc2)CN1C(c1ccccc1CO)=O C1(NC(C=C(C)C)=O)CCN(C(=O)CCC(=O)c2cccc(N)c2)CC1F c1(C(=O)NC2CC(F)(CNC(c3cnco3)=O)C2)csc2ncnc(O)c12 N1(C(CSCC)=O)CCC(C)N(C(=O)CCc2nnc(S)n2C)CC1 Cc1cc(C(=O)NC2CC23CC(NC(=O)C=Cc2cncc(O)c2)C3)cc(O)n1 C1(NC(=O)CSC(F)F)CCN(C(=O)CCCCO)CCC1c1ccccc1 C=CC(C)(O)CC(=O)N1CC(NC(=O)Cc2cnsc2)C(n2ccnn2)C1 c1(C(N(CCCNC(=O)C(C)(C)CF)CC)=O)cc2c(Br)cccc2cn1 N1(C(C(c2ccn(C)n2)C)=O)CC(NC(=O)CN2CCC(O)CC2)C2CCCC12 N1(C(CNC(=O)OC)=O)CCCCC12CN(C(C1CCN(C)C(C)C1)=O)C2 C1(C(=O)NCC=CCOC)CC(C)(C)CCN1C(c1occ2c1CCC2)=O C1(NC(C=CC(C)(C)SC)=O)CC=CCC1C(=O)NCC1(CO)CC1(C)C c1(C(=O)NC2CC(NC(C(c3ccc(F)cc3)OC)=O)C2)c(F)cccc1I N1(C(C(=O)NCCOCCOC)=O)CC(NC(C23COCC(C2)C3)=O)CC1(C)C c1(CC(N2CCC(O)(CN(C(C(C=C)O)=O)C)CC2)=O)ccc2sccc2c1 c1(C(=O)NCC2(OC)CN(C(=O)CC3CCC(=O)N3)C2)cc2c(O)cccc2[nH]1 C12CCCC(C1)C2.N1(C(c2c(CNC(=O)C3CC3)occ2)=O)C2CCC1CC2 c1(CN2CCN(C(CNC)=O)C(C)C2)ccc(F)c(-c2noc(C(C)C)n2)c1Cl Cc1c(F)cc(CN2CCC(NC(c3cccc(C)c3O)=O)C2)cc1F Cc1ccc(C(=O)NOC(CC(C)C)C(=O)NCC2CCCS2)nc1O C(=O)(C(CC(C)C)ONC(C1CC(=O)C1)=O)N(CC=C)C1CC1 Cn1cnc2c(NC3CCCC3C3CC3)[nH]c(=NCC34CCCN3CCC4)nc12 C(=O)(C1c2ccccc2CN1C(c1ccco1)=O)NC(C1CCCCC1)C#N c1(CSC)nc(N(C)CCOCC(=O)Nc2ccccc2C)cc(C)n1 C12(CNC(C(C)SCC)=O)CC(COC)(CN1C(c1ccc(C)cc1Cl)=O)C2 C1(C(=O)NCC2N(C(c3c(C)cc[nH]c3=N)=O)CC2)C2C3CC4C1C1C2CC3C41 c1(C(N2CC3C(CC(=O)NCC4(CF)CCC4)(CC3)C2)=O)ccc2[nH]ccc2c1 C(=O)(C(C)(COC)OC)N(CCC)CCN(C(=O)C(C)Cc1cccnc1)CC c1(CC(=O)NC2CCC23CCN3C(c2cnon2)=O)ccc(Br)c(F)c1 N(C(=NCCC(C)=O)NC1CCC(C(N)=O)C1)C1CCN(C(=O)OCC)CC1 C1(C(=O)NC(C=C)C)(CCNC(=O)Cc2nonc2C)CCCC1 C(=O)(C(Cc1cnc[nH]1)NC(=O)C(O)CSC)NC(c1ccccn1)COC C1(NC(C2CCC(OC)CC2)=O)CC2CN(C(=O)CC(C)(C)COC)CC12 C#CC1CN(C(C2CN(C(=O)COCCC=C)CC2CCC)=O)CCO1 N1(C(c2ccc(OC)nn2)C(=O)NCCOC)CCN(CCC#N)C(=O)C1 C(C1c2ccccc2CCN1C(c1nnn(C(C)(C)C)n1)=O)NC(C(CCC)O)=O c1(C(=O)NC(C)CCCCNC(c2cncnc2)=O)ncc(Cl)cc1Cl C(CN(CC(=O)N(C)CCN1CCOCC1)N1CCC(O)(CCO)CC1)OC C1(C(=O)NCCN2CCN(C(Cc3c(C)nn(C)c3)=O)CC2)CCCCC(=O)C1 C=CCC(F)(F)C(=O)NC(CN(C)C(c1cn(CC)nc1C1CC1)=O)CC C1(NC(CC2(OC)CC2)=O)CN(C(=O)Cc2cncs2)CC1C C(=O)(C(C)(C)C(F)(F)CC)NC1(CC=C)CCN(Cc2noc3c2CCCC3)C1 c1(C(=O)NC(C)=O)ccc(CNC(=O)CC2CC(F)C2)cc1.C12CCCN1C2=O c1(C(=O)O)[nH]c2ccccc2c1I.c1(C2NCCSC2)cc(F)ccc1F c1(CC(C)NS(=O)(=O)C2CCN(C(=O)OC(C)(C)C)C2)cc(F)cc(C#N)c1 N1(C(C23C(CN(C(C4C(C)C5CCC4C5)=O)C2)C3)=O)CC(C)(C)C12CCC2 c1(C2CCN(C(C3CCN(C(CCC)=O)C3)=O)C2)ccc(Cl)c(Cl)c1 C12(CC)CN(C(C3CCCC(C)C3)=O)C(CNC(c3ccn(C(F)F)n3)=O)(C1)C2 C12(NC(N(CCOC)CC)=O)CC1CN(Cc1ccc(N3CCC(C)CC3)cc1)C2 N1(C(CCOCCCOC)=O)CC(O)C(O)C1C(=O)NCC(O)CCSC c1(C(=O)NC(CC)CN(C)C(C2(CO)CCCO2)=O)nnc(S)n1C c1(C(N2CCC(N(C(C3C(CC)C3)=O)C)C3(C2)CC3)=O)nc2ncc(Br)cc2[nH]1 c1(CCCC)nc(C(=O)NCC(C)N(C(=O)CCOC2CCOC2)C)cs1 Cc1ccc(F)c(C(=O)NCC2(CNC(c3c(F)cccc3Cl)=O)CC2)c1 c1(C(N2C(CNC(c3c(CC)noc3C)=O)CC(F)C2)=O)ccc(O)c(C)c1C Cc1cc(C(N2CC=C(C(=O)NCCCCCO)C2)=O)nnc1C C1(NC(C2CC(C)OCC2)=O)CC2CC1CN(C(c1ccsc1C(F)(F)F)=O)C2 CCC(O)C(F)(F)C(=O)NCc1cc(C(N2CCCC(C(C)(C)C)C2)=O)n(C)n1 c1(C(=O)OCc2nc(Br)cs2)ccc(O)nc1 CCN=c1[nH]cc(C(=O)NCC2CN(C(=O)C(O)P(C)(C)=O)C(C)(C)C2)s1 c1(C(N2CC(CNC(C(C)SC)=O)C2)=O)cnc(COC(C)C)s1 C(C(CNC(=O)C(Cl)=CCl)C(F)(F)F)NC(=O)CN1CCS(=O)CC1 c1(CC(=O)OC)nc(NCCCCCNC(=O)CCc2cccnc2)c(C)s1 C1(NC(COCCOCC#C)=O)CCCC(CNC(=O)CCSC)C1 C=CCC(CC)C(=O)N1CCCC1C(C)NC(c1ncc(C)cn1)=O C1(NC(C(C)CO)=O)CCCCC12CCN(C(c1nn(C)c(Cl)c1Cl)=O)CC2 N1(C(=O)Nc2nnc(-c3ccc(F)cc3)s2)CC2CC(C1)C2(F)F C=CC(CCC)CC(=O)N1CCC(CN(C)C(c2cc(C3CC3)ncn2)=O)C1 Cn1nc(Br)nc1C(N1CCC(c2ccc(Cl)cc2)C1)C(=O)NC1COC1 c1(C(N2CCC(OCC(F)F)CC2)C(=O)NC(CC)C)c(C)nn(C)c1Cl c1(C(=O)NCC2C(NC(C(C)NC(C)=O)=O)CCC2)cccc2c1OCCCO2 c1(C(=O)NC2(CN(C)C(c3n[nH]c(C)n3)=O)CC2)coc(-c2ccsc2)c1 Cn1nc(C(N2CC3CN(C(=O)Cn4nnc(=O)[nH]4)CCC23)=O)c2c1CCSC2 Cc1cccc(C(N2CCC(CO)(NC(=O)CC3CC(C)(C)CO3)C2)=O)c1O N1(C(C(CCCC)O)=O)CCC2(CC1)CC2NC(=O)C(C1CCOCC1)F C1(C)(C(=O)NCCC(C)NC(C2CCC(C)O2)=O)CCS(=O)(=O)CC1 Cc1cc(C(N2CCC2C(N2CCN(c3ccccn3)C(C)C2)=O)=O)nc(C)c1 CC1CC(C)(C(N2CC(CNC(c3cnc(Cl)c(C(F)F)c3)=O)C2)=O)CCO1 c1(C(CC)C)cc(N2CCOC(c3ccc(C(=O)O)cc3)C2)ncn1 Cc1cc(C)c(C(=O)NCC(C)(C(C)C)NC(c2cc(C#N)c(C)s2)=O)c(O)c1 Cc1cccc(C(=O)NC(C)C(=O)NC23CC(C2)N(C(=O)CC2(O)CCC2)C3)c1 N1(C(C2N(CC)CCC2)=O)CCC2(CC1)CC2NC(c1nnn(C)c1C1CC1)=O CCC(C)CCC(=O)N(C1CCN(C(=O)CCOC2CCCCC2)C1)C N1(C(CC(CNC(c2c(C)ncnc2C)=O)C2CCC2)=O)CC(C)(C)C(O)C1C C1(N(C)C(C2CCN(C(c3cscc3Cl)=O)C2)=O)CCOCC1(C)C c1(CN2CCC(O)(C(=O)Nc3cnn(CC)c3C)C2)c(Br)cc(F)cc1Br c1(CCOCC)nncn1C(=O)N.c1(OC(CCOC(C)(C)C)=O)ccccc1 C(=O)(C(C(C)C)N(C)C)NCC(C)(C1CC1)NC(C(c1ccccc1)SC)=O c1(OC)ccc(Cl)cc1-n1nc(C(C)C2CC2)nc1C1COC(=O)O1 C(CC)(C(=O)NC1(C(=O)NC(C)(C)CCN(C)C)CC1(C)C)OCC C1(C)(C(=O)NC(C2CCN(C(C3C(C)C3C)=O)CC2)C)CCS(=O)(=O)CC1 C1(CCC(=O)NCC2CC2CNC(c2c(Cl)cn(C)n2)=O)CCC(=O)NC1=O C(=O)(C1CCc2c(Cl)cccc21)NC1CC(NC(=O)Cc2cn[nH]c2)C1 Cc1nn(C(F)F)c(C)c1CC(=O)NC(C)CN(C(=O)CCc1cnn[nH]1)C(C)C O=C1OC2CON(C(=O)c3cc(-n4cccn4)ccn3)CC2O1 c1(C(=O)NCC2CC2NC(C2C3CN(CC(F)(F)F)CC23)=O)cc(F)ccc1O CC(C)CC(C(=O)N1CCN(C)C(CNC(c2cc(C(N)=O)c[nH]2)=O)C1)C(C)C S(=O)(=O)(c1ccccc1-c1ccc(Br)cc1)NC(c1ccc(Cl)cc1)CC c1(C(C(=O)N(C2CCC(O)C2)C)C2CC2)ccc(Cl)cc1 C1(CN(C)C(C2CC23CC3)=O)CCN(C(c2csc(Br)c2)=O)C1 C1(CNC(c2cc(C)ns2)=O)CC2CCC1N2C(C1(C)CC12CCC2)=O CC(CC(=O)NCC(CO)NC(=O)C=C1CCCCC1)c1cccnc1 c1(C(=O)NCCCCCCn2cc(CCc3nn[nH]n3)nn2)cccc(CO)c1 C1(NC(=O)COCCn2cnnn2)CC2(NC(c3ccccn3)=O)COC1C2 C(C)(C)(CCC(=O)N1CCCC(CO)(CSC)C1)NC(c1c(CC)oc(C)c1)=O c1(C(C)(C)C)ocnc1C(N1CC(CO)(NC(c2csc(C(F)(F)F)c2)=O)C1)=O C1(C(=O)NC(C)CCN(C(=O)C(C)c2ccco2)C)CC(F)(CF)C1 C12(CCCC1)CN2.C1(C(N(C2(C(N)=O)CCC2)C2CC2)=O)CCCCO1 c1(CC)ccc(C(N2CC(C(C)NC(c3cc(Cl)c(Cl)n3C)=O)C2)=O)c(O)c1 N#Cc1ccc(=NCC(=O)N2CC=CC2CNC(=O)C=CC2CCC2)[nH]c1 CCCC(O)CC(=O)N1CC2CC(CNC(=O)CCCn3nc(C)cc3C)C2C1 n1(CC)nc(C)c(C(=O)NCC2(NC(=O)C(C)NC(C)=O)CCCCC2)c1C C(=O)(C1=CC2CCCC12)NCC(C(C)(C)C)NC(=O)C1=CCCOC1 c1(C(=O)NCCOCCNC(CCC=C=C)=O)ccc(CCC)c(N)c1 C1(CC)CN(C(c2ccccc2Cl)=O)CCC1NC(=O)CSc1cccc(C)c1 n1(CC)nnc(C)c1C(=O)NCC(C)NC(c1cnoc1-c1ccccc1)=O C1(CCC)CN(C(=O)C(C)CC(N)=O)CCN1C(=O)CCc1ccc[nH]1 C(=O)(C(F)(F)C(F)(F)F)NC(CCN(C(C(C)(C)NC(=O)NCC)=O)C)C1CC1 c1(C(=O)NCCC2(NC(C3C(C)CN(C)C3)=O)CC2)csc2cc(Cl)cnc12 C(=O)(CC(C(C)C)c1ccon1)N(C1CC1)C.c1(OC(CC)=O)ccccc1 C1(COC)CN(C(=O)COCCF)CCN1C(c1cnnc(O)c1)=O CCC(CCC(=O)NC(C)(CNC(c1cc(C)cc(C)n1)=O)C1CCC1)OC Cn1cc(CNCC2CCn3nnnc3C2)c2ccc(Cl)cc12 C1(c2sc(SC)c(C)n2)(NS(=O)(=O)C(C)CSC)CCN(C(=O)OC(C)(C)C)CC1 S(=O)(=O)(c1ccc(C#N)c(NCc2cnc(C)s2)c1)N1CCC(CC)C(C)C1 CCC(C)(C)C(=O)C(=O)NCC(CC(F)(F)F)NC(c1cc[nH]c2nccc1-2)=O C1(C(CNC(=O)CCCc2nccs2)F)CCN(C(=O)CCOC2COC2)CC1 C=CCC(C(=O)NCC=CCNC(c1occc(=O)c1OC)=O)C(C)C Cc1ccc2c(=NCc3cnns3)[nH]c(N3CC(=O)NC4(CC4)C3)nc2c1 C1(C(=O)NCCNC(C2(COC)CC(=C)C2)=O)CCCCN1CC(F)F C(=O)(CCS(=O)(=O)NC)NC(CC=C)CNC(C1(n2cnnn2)CCCCC1)=O c1(C(C(=O)NCCN(C)C)N(C)CCOCC2CC2)ccc2ccc(Cl)cc2n1 N1(C(C(CC2CC2)OC)=O)CCC2CCCC12C(N1CCC(C(N)=O)CC1)=O CC(C)CC(=O)NCC(=O)NCCC1CN(C(=O)CC2CC=CC2)C1 C1(NC(CSCCC(C)C)=O)CC(O)CN(C(c2ccnc(N(C)C)c2)=O)C1 S(=O)(=O)(c1ccc(NCCc2cn3c(C)cccc3n2)c(Cl)c1)N(C1CC1)CC Cc1cc(OCCNC(=O)CC2CCCN(C(=O)C(N)=O)C2)cc(O)c1 c1(C(N2CCOCC(NC(c3ncncc3F)=O)C2)=O)cc(Cl)cc([N+](=O)[O-])c1 C1(CNC(C2(C(C)C)CC2)=O)CCN(C(c2nn[nH]c2Cl)=O)C12CC2 c1(NC(c2nnnn2CCC2CC2)(CC)C2CC2)cccc2c1OC(C)(C)C2 CC(C)C(O)C(=O)NCC1(C)CC(NC(=O)CSc2cn[nH]c2)C1 Cc1cc(C)c(C(N2CCCC2CN(C)C(c2ncoc2CC(C)C)=O)=O)[nH]1 Cc1c[nH]c(CC(N)=O)c1C(=O)NC1CCN(C(C2COC(C)C2)=O)CC1 O=C(C(O)C(F)(F)F)NC1CN(C(c2nncs2)=O)C1 n1(CC(C)C)c(N2CCC(C(C)(C)NC(=O)OC(C)(C)C)CC2)nnc1C1CCC1.O c1(C(N2CC(CCNC(CC(C)CN(C)C)=O)C(C)C2)=O)ccc2ccoc2c1 Cc1noc2cc(C(N3CC(NC(c4cc(Cl)no4)=O)C(C)C3)=O)ccc12 C1(NC(C2CCC(CC)O2)=O)CN(C(=O)C(c2ccc(F)cc2)C)CCC1C C1(CNC(C(C)NC(=O)NC)=O)CCN(C(c2cnn(CCO)c2)=O)C(C)C1 C(=O)(C(O)C(C)(C)C)N(CCOC(C1(C(=O)OCC)CC1)=O)C CCCC(CC(=O)NCc1ncccc1O)NC(=O)C(O)CC N1(CC)CCN(CC(=O)N(CC(=O)O)C(C2(c3ccccc3)CCCO2)C)CC1 c1(C(=O)NCCCC2N(C(c3c(C)nn[nH]3)=O)CCC2)ccc2nc(O)cn2c1 C(=O)(C1CCOc2ccccc21)N1CC=CC(NC(=O)CC2COCCO2)C1 c1(C(=O)NCC2(O)CCN(C(c3c(CCC)onc3C)=O)C2)coc2c1COC2 N1(C(c2ncc(CC)nc2)=O)Cc2nccn2CC(NC(=O)CC2C=CCC2)C1 N1(CCN(C)C(c2nccc3ncccc23)=O)CC(=O)C2C3CCC(C3)C12 N1(C(C(CC)N(C)C)=O)CCC(CNC(c2ccc(-c3ccco3)[nH]2)=O)C12CC2 c1(OC)ccc(F)cc1C(=O)NC1C2CN(C(C3CCC(C)(C)O3)=O)CC12 c1(C(=O)NC2C(C)N(C(=O)COC3(C)CCCC3)CC2)cc2n(n1)CCCC2O N1(C(C(=Cc2cnc[nH]2)C)=O)CCN(C(c2nc(C)ccc2F)=O)CC1C1CC1 N1(C(C(CC)=CC)=O)CCC2(CC1)CC(NC(=O)Cc1cncn1C)CO2 N1(C(C(Cc2cscn2)OC(C)(C)C)=O)CC2(C(=O)ON3CCC(Br)C3)CC1C2 c1(C(=O)NCCOCCCN(C(=O)C=Cc2nccs2)C)ncc2ccccn12 C=CC(CC)CC(=O)C(N1CCCCC1)=O.C1(C(=O)OC)CN(C=O)CC1O N1(CC(=C)C)CCC2(CC1)CN(C(C1CN3CCCN1CC3)=O)C2 n1(CC#C)c(C(=O)N(CCCN(C(=O)C(O)C2CCC2)C)C)cc2ccccc12 C(=O)(C(C)S(N)(=O)=O)N(C)CC1CCN(C(C=C(CC)CC)=O)C1 CC(C)CC(C(=O)N1C2CCC(C2)C1CNC(C1CC1C)=O)n1ccnc1 C1(C)(NC(C2C(OC)CCCC2)=O)CCCN(c2nccc(C(N)=O)n2)C1 c1(N2CC3(OCC(C)C3)C2)nccc(=NC2CCOc3ccccc32)[nH]1 N1(C(C(C)=CC2CC2)=O)CC(C2CCN(C(c3cnc4scc(C)n34)=O)CC2)C1 C(=O)(C1Cc2ccc(Cl)cc21)NC(CNC(c1ccc(OC)nn1)=O)(C)C1CC1 c1(C(=O)NC(c2ccc(CC)cc2)CNC(=O)CCS(C)=O)cccn(C)c1=O N1(c2cc(NCc3nnc(C(C)C)s3)ncn2)CC(C)OCC1C N1(C(C(C)N(C(C(C)NC(=O)NC)=O)C)=O)CC(C)CC(O)C1 CCCCC(F)C(=O)NCc1cc(C(=O)NCC2CCCC2O)n(C)n1 CC(C(=O)NC(CNC(=O)CC1CC2(CCO1)CC2)C1CCC1)C(C)(C)C c1(OC)cccc(SCC(N2CC(N(C(=O)CSC(F)F)C)C(O)C2)=O)c1 N1(C(COC)=O)CCC2C1CCN2C(=O)CCSC1CCCC1 C1(CNC(=O)Cc2sccc2-c2ccccc2)(NC(C2CCC2(F)F)=O)CCOC1 c1(OC)ccc(F)c(C(N2CC(CNC(C3C(C)C3(F)F)=O)CC2(C)C)=O)c1 CCC1=NOC(CC(N2CC=CC2Cn2cc(CC(F)C(C)(C)O)nn2)=O)C1 C(=O)(C1=CNC2=NCCCN12)N1CC(N(C(c2c(CCC)nsc2N)=O)C)C1 C1(CNC(CNC(CCC)=O)=O)C(C)CCCN1C(c1cn(C2CCC2)cn1)=O c1(C(N(CCCCC)C)=O)occc1CNC(c1ccncc1)=O N1(C(C(COC)NC(C(CC)COC)=O)=O)CCn2c(cnc2C)C1 C1(C(=O)OC)CN(C(c2ccnc(OC(F)F)c2)=O)c2ccc(F)cc2O1 c1(N(C(=O)NOC2CC(C(=O)O)C2)C)cnccc1C(F)(F)F CCCCCC(O)C(=O)N1CC2(C(N3CCC(SC)C3)=O)CCC1CC2 C1(CNC(c2scc(C)c2C)=O)CCCCN(C(=O)CC2COCCO2)C1 N1(C(c2cc[n+]([O-])cc2)=O)CCC2(CC1)CN(C(C1CC3C=CC1O3)=O)C2 C1(C)(C(=O)NCC2(C)CCC2)CCCN(C(=O)CCCCN=[N+]=[N-])C1 C1(NC(C(C)OCC)=O)CC(F)CN(C(c2cc(Cl)n(C)n2)=O)C1 C=C1CCN(C(=O)CCOCCN(C(=O)C(CC)n2cnc[n+]2[O-])C)C1 c1(-c2cccc(CS(C)=O)c2)cnc2c(C(=O)NCc3cc(Br)no3)c[nH]c2c1 c1(C(=O)NCCC2CN(C(C3CSC3)=O)CC(C)O2)cccc2nccnc12 c1(CNC(=O)C(=O)NC2CC3CCCCC23)cn2cc(F)ccc2n1 CCCC(C(=O)N1CCC(CNC(=O)CC2CCC3(CCC3)O2)CC1)S(N)(=O)=O N1(C(c2nc(C(C)=O)sc2)=O)CC(NC(=O)C(F)(F)c2cccnc2)CC1C Cc1[nH]c2ncccc2c1C(=O)N(CCNC(=O)Cc1cc(CO)on1)C(C)C C1(CNC(c2ccc(F)cn2)=O)CC12CCN(C(=O)C(O)Cn1cncn1)CC2 c1(C(N(C)CCNC(c2cc(F)c(Br)cc2F)=O)=O)cc2c(=O)[nH]ccn2c1 Cc1nc(C(=O)NCC2(O)CN(C(C3CC4OC3C3CC43)=O)C2)c2ccnc-2[nH]1 C1(NC(c2nc(C)oc2)=O)CC2CCC(C1)N2C(=O)CCc1ncccn1 N(C(=NCCC1CCCCC1)NCCc1cccc[n+]1[O-])CC(=O)NC CC1C(C(=O)NC(C)(C)CCn2ccnc2)CCN1C(C1CCC(C)(C)C1)=O C(=O)(CC(C)(C)CNC(c1ccn(C)n1)=O)NC(COC)CCO CC(C)(C#N)C(=O)NCCC(O)CNC(=O)C1=C(Cl)CC1 Cc1cc(NC(=O)CC2COCCN2C(=O)C(O)C(C)C)cnc1Cl C=CC(C)(CCOC)C(=O)NCC1(C)CC(NC(c2csnc2OC)=O)C1 N1(c2cc(CC)ncn2)CCOCC(NC(c2c(C(F)(F)F)coc2C)=O)C1 c1(C(=O)NC2CC3CN(C(CCC(=O)OC)=O)CC3C2)cnc2snc(C)c2c1 c1(C(=O)NCC2=CCN(C(C3C(C)(C)C3(F)F)=O)CC2)ccc2c(c1)C(=O)NC2 C1(O)(C(CNC(C2(CC(=O)OC)CC2)=O)C)CCN(C(=O)C=NOC)C1 c1(NC(COC)=O)nncn1NC(=O)C1CN(C(=O)C(c2cccnc2)OC)C1 C1(NC(C(C(=C)Cl)(C)C)=O)CC1C1CCN(C(C2CC3(C2)CC(F)C3)=O)CC1 c1(C(N2CC(NC(c3n(C(C)C)ncn3)=O)C(O)C2)=O)c(O)cccc1Cl C=C(C)CC(C(=O)N1CC(c2nc(=O)o[nH]2)C1)NC(=O)C(C(C)C)SCC N1(C(c2scc(C)c2)=O)CC(F)CC1CC(=O)NCCN1CCOCC1 c1(CC)oc(C)cc1C(=O)N(CCCCCCNC(C1(C(=O)N(C)C)CC1)=O)C C(C(CC(=O)NOCCCCF)C1CCC1)NC(C1CC(C)(F)C1)=O N1(C(C(CC)N(C)C)=O)CCC2(NC(C3CCN(C(C)C)CC3)=O)CCCC12 C1(COC)(CNC(=O)CC2CN(C(=O)C(C)c3cc[nH]n3)CCO2)CCC(=O)N1 C1(NC(=O)NC(CCc2c(C)c[nH]c2C)=O)CN(CCNC(C)(C)C)CCC1C CC1(C)CN(C(C2CCc3nc[nH]c3C2)=O)CCC1NC(C1(CF)COC1)=O N1(C(C(C)(C)C2CCOC2)=O)CC2(C1)SCCC2NC(=O)COCc1nc[nH]n1 CCC(CCOC)C(=O)NCC1CN(C(c2ccnn2COC)=O)CCN1C N1(C(CCC)=O)CC(CNC(c2cnc(N3CCCC3)s2)=O)C2CC12 c1(OCC(N2CCN(C(C(=O)NCC)=O)C(CO)C2)=O)c(C)cc(Cl)cc1C C(=O)(C(O)(C(F)(F)F)C1CC1)NCCOCCCNC(c1c(C)cco1)=O N1(C(C(C(C(C)C)O)C)=O)CCN(C(c2cnc[nH]c2=N)=O)C2CCCC2(C)C1 C1(=CC(=O)N(CC(C)O)CCNC(=O)COC2(C)CCC2)CN2CCC1CC2 N1(C(C(C(=C)Cl)(C)C)=O)CC2CCCC2(NC(=O)CCC)C1 Cc1cc(C(=O)NCCC2CCN(c3ncccc3C#N)CC2)n2ncnc2n1 CCCC(C#N)C(=O)N1CCN(C(=O)C(CO)OC)CC1c1cnn(C)c1 c1(C(N2C(CC)CN(C(=O)CC3CC(F)C3)CC2)=O)cc2c(s1)CCCNC2=O N1(C(CCSCC)=O)CCN(C(=O)C(C(C)C)NC=O)CC1c1ccnn1C Fc1cccc2c1CCN(Cc1cc(-c3ccccc3)nc3ccccc13)C2 C(=O)(C(C)(CO)CO)Nc1c(C(=O)Nc2ncn(C)c2C(F)F)scc1 C1(NC(C2(OC)CC2C)=O)C2CC3C1C3C2C(=O)NCC(=O)OC(C)C c1(C(N2C3CN(C(=O)Cc4ccsc4Br)C(C3)C2)=O)n[nH]c2c1CCCC2 C(Cn1cncn1)(CCC(=O)O)NC(c1cnn[nH]1)=O C1(C(=O)NC2(CCNC(C(C)(C)F)=O)CCC2)CC(=O)CC(=O)C1 c1(N2CCC(NC(c3cc(C)[nH]n3)=O)C2)cc(C(C)(C)C)ncn1 C1(C(=O)NCC(C(C)C)NC(C2C(c3ccccc3)C2C)=O)CC(C)(C)CN1C C(=O)(CCCCC(C)C)NCC1(C(C)NC(c2ncc(OCC)nc2)=O)CC1 Cc1cccc(C(N2CC(N(C)C)C(CNC(C3(O)CC3)=O)C2)=O)c1Cl c1(C(=O)NCC2CN(C(COCC)=O)CC2C)ccc(C#N)cc1 c1(C(N2CC(NC(c3cccs3)=O)CC23CCC3)=O)ccc2ncccc2c1 c1(C(=O)NCC(C)(CO)NC(C(C)OCC#C)=O)ccc(C(=O)OCC)cn1 N1(C(c2cc(C)c(O)nn2)=O)C2CCCC1CN(C(c1ccc(C(F)F)s1)=O)C2 c1(C(N2CCC(O)(CCNC(C=CC)=O)C2)=O)cn(C(C)C)c(C)cc1=O C1(COC)CN(C(=O)Cc2ccc(C)o2)CCN1C(c1occc1F)=O C1(N(C)CC)CCN(C(C2C=CCN2C(=O)CC2C=CCCC2)=O)C1 c1(NC2C3CN(C(C(C)OC)=O)CC2CC3)nc2ccc(C(F)(F)F)cn2n1 C1(C=C)(C(=O)NC(C(=O)NC(CC#C)C(=O)OC)CCOC)CCOCC1 N1(C(C(CC)C)=O)CC2CCCN(C(=O)CCc3ccsc3Cl)C2C1 C(C)(CCCCNC(C1CC1CF)=O)NC(COCC(C)C)=O c1(C(=O)NC(C(=O)NC(CCCCC)C)C(C)(C)C)c[nH]c2ccccc12 N1(C(CC(C)F)=O)CCC(C)(C)C1CC(N1CCC(CC(F)F)C1)=O N1(C(Cc2nc(CC)sc2)=O)CC(NC(c2ccc(Cl)cn2)=O)C(C)(C)C1 c1(C(N2CCC(NC(CN(CC)CC)=O)(CF)C2)=O)c2c(nn1C)CCCC2 N1(C(CCc2c(C)nccc2)=O)CCN(C(=O)C(C2CCOCC2)C)CC1CO c1(C(N2C(CCNC(C(CC(C)C)O)=O)CCCC2)=O)cccc2oc(O)nc12 C1(CC(=O)NCCOCC)C2CN(C(=O)CCC(C)=O)CC12.C12CC(C1)O2 CCC(O)CC(=O)N=c1ccc2cc(S(C)(=O)=O)ccc2[nH]1 CC(C)(CCCNC(=O)Cn1cc(C2CC2)nn1)C(=O)NCC1CNC(=O)CO1 N1(C(CN(C)C(N)=O)=O)CCC(C2CC2)C1CNC(C1CC(S(C)(=O)=O)C1)=O N1(C(c2nc(C)oc2)=O)CCC(NC(=O)CC2CC2C(F)(F)F)C(C)C1 c1(C(N(CCC)CCNC(=O)C(O)c2cnc[nH]2)=O)cc2sc([N+](=O)[O-])cc2[nH]1 c1(C(=O)NC2CCN(C(C(C(CC)O)C)=O)C2C)ccc2nc(C)nc(O)c2c1 c1(C(=O)NC2(C)CN(C(CN(CCCCCC)C)=O)C2)cnc(C(C)C)n1C C(=O)(C1=NOC2(CCC2)C1)NC1CN(C(C2(C)N(C)CC(O)C2)=O)CC1(F)F C(=O)(C(C(C)C)c1cccnc1)NCC(C1CC1)NC(c1n(CC)ccc1)=O c1(C(=O)NCC2OCCN(C(Cc3c(C)noc3)=O)C2)cnc2[nH]nc(O)c2c1 c1(C(=O)OC)cc(OC)c(S(=O)(=O)N2CCCC(C3CCCC3)C2)c2ccccc12 c1(-n2ncc(C(=O)NC(CNC(CCSC)=O)C3CCC3)c2)ccccc1Cl C1(C)(CNC(CCn2ncc(C)c2)=O)CN(C(C2(O)CC2(C)C)=O)CCO1 c1(C(=O)NCC2(O)CCN(C(c3cc(OC)n[nH]3)=O)C2)ccc(Br)c(C)n1 N1(C(CC2(CSC)CC2)=O)CC2(CC(C(=O)NCC(O)C(F)F)CO2)C1 c1(OC)ccc(C(N2CC3CC(C2)N3C(C2CCNC(=O)C2)=O)=O)c(Br)c1 C(C(C)(C)CC(=O)NCCc1ncc(-c2ccccc2)s1)N(C)C N1CCC2(C1)N(C)C2.C1CCCOCC1.CS(=O)(=O)CCc1ncc(-c2nccs2)s1 C1(O)(CNC(c2[nH]cc(C)c2C)=O)CCCN(C(c2cc(Cl)cnc2O)=O)C1 N1(C(c2cccc(C#C)c2)=O)CCC2CN(C(=O)C=Cc3cn(C)cn3)CC2C1 N1(C(C=CC(C)C)=O)CCC2(COC(CNC(c3cccn3C)=O)C2)C1 N1(C(c2ccc(N)c(Cl)n2)=O)CC2(C1)CN(C(=O)CC13CCCC1C3)CC2CO c1(C(N2CCCC(O)(C(C)NC(=O)CC(C)F)C2)=O)cncc2cc(Cl)ccc12 N1(C(CC2CC(=C)C2)=O)CCC(NC(=O)C(F)Cc2ccccc2)C1(C)C c1(C(N(CC(=O)NC(c2cc(C)on2)CC)C)=O)ccc(C#N)cc1 N1(C(=O)NCCc2cc(CC)no2)CCCC(c2nncn2C2CC2)C1 C1(CNC(C(C)SCC)=O)CC(O)(CNC(c2scnc2C(C)C)=O)C1 C1(C(=O)NC2(C(N3CC(F)(COC)C3)=O)CCSC2)(N(C)C)CCCSC1 C1(CC)(NC(=O)CSc2ccccn2)CN(C(c2cn(C(C)C)nn2)=O)C1 Cc1n[nH]c(C)c1CC(=O)NCC1C=CCN1C(c1cc(C2CCC2)[nH]n1)=O CCCC(CC(=O)N1CCCC(C2CCCN2C(c2cc[nH]n2)=O)CC1)C1CC1 c1(SCCN(S(Cc2c(C)ocn2)(=O)=O)CCO)ccccc1[N+](=O)[O-] c1(C(=O)NC2(CNC(=O)CC3CCC4CC34)CCC2)cccn2c(O)nnc12 C1(NC(=O)NC2C3CC4C2C4(C(=O)O)C3)CCC2(CC2)CCC1 C1(F)(CNC(CC2CC(=O)NC2)=O)COCCN(C(C2C3(CC3)C23CC3)=O)C1 N(S(=O)(=O)N(C)C(c1csc(CO)n1)C)CCOC(C)=O.c1(O)ccccc1 c1(C(=O)NCC(c2c(CC)cccc2)NC(=O)C(CO)SC)ccc(Cl)nc1N c1(OC)cc(C(N2CCCC2C(N2CCC(C)(OC)C2)=O)=O)c([N+](=O)[O-])cc1F CC1COCC(C(N2CCOCC2C(=O)NCCc2ccccc2)=O)O1 c1(C(C(N2CC(COC)(CNC(=O)CCSC)C2)=O)N(C)C)ccccc1Cl Cc1cc(Cl)ccc1NC(=O)CC1CCCCC1NC(=O)CCN1CCCCC1 c1(C(=O)NC2CC(CC)C2)coc(CNC(c2ocnc2C)=O)c1 c1(C(N(CC(C)NC(=O)C(OC)OC)CC)=O)cnc(O)n1CC N12CC(NC(=O)OC(C)(C)C)CC(C1)NC2=O.C=CC1(C(=O)OC)CCC1 c1(C(N2CC=C(CNC(C3CCC4(CC4)C3)=O)CC2)=O)cnn2c1CCCC2 N1(C(CCNC(COC)=O)=O)CC(NC(C23CCCC(C2)OC3)=O)CC(O)C1 C1(C(=O)OC)(CNC(CC(c2ccccc2)OC)=O)CN(C(c2cc(Cl)no2)=O)C1 C=CCC(C)(C)CC(=O)NC1CCN(C(C23CSCC2C3)=O)C1CC N1(C(c2nc(C)sc2C)=O)CC2CCC(C1)C(NC(C1(C(F)F)CCCC1)=O)C2 C1(NC(CSC)=O)COC2(CCN(Cc3scnc3C)CC2)C1 CCC(CC(=O)N1CCCCC1C1(NC(=O)Cc2oc(C)nc2C)CC1)C1CC1 C1(NC(COCCNC(C(COC)(C)O)=O)=O)CCCCNC1=O N1(C(C2C(CCOC)C2)=O)CCC(C)(CNC(=O)CC2CCCS2(=O)=O)CC1 C(CC(CC)(CC)NC(C=CC(=O)OCC)=O)NC(=O)C(F)Oc1cnn(C)c1 C1(CC(=O)NC(C(C)NC(CCCOC(C)C)=O)CO)C=NN(C)C1=O CN1CCC(C)(C(N2CCC(F)(F)C(CNC(C3CC(N4CCC4)C3)=O)C2)=O)C1=O C1(S(C)(=O)=O)(CNC(NC2C(C)C2)=NCCc2cccs2)CCCC1 Cc1coc(C(N2CCCC2CNC(=O)CCc2ccc(=N)[nH]c2)=O)c1F N1(C(C(CC)(F)F)=O)CC(C2CCN(C(C3(CO)CCCCO3)=O)CC2)C1 c1(C(N2CCC(N(C(c3ccc(F)o3)=O)CC)C2)=O)ccn(CCO)c(=O)c1 c1(CC(=O)NC(C)CNC(=O)C=CCO)csc(-c2ccccc2)n1 C(=O)(CCCCSC)NCC(=C)CCNC(c1nonc1C(=O)NC)=O N(C(=NCCNC(CC)C)N1CCCC(NC(=O)OC)C1)Cc1ccc(F)cc1 CC1CCCCC1OCC(=O)NC(C)(C)CCCNC(=O)CC1CCC(F)(F)C1 CC1CN(C(c2nncs2)=O)CC(C)CN1C(c1cc2ncccc2[nH]1)=O N1(C(c2cc(-c3ccc(C)s3)on2)=O)CCc2nc(=N)[nH]cc2C1 C1(OC)CC(C(=O)N(C)CCNC(C2CCC(C(C)C)NC2=O)=O)CC1OC C1(N(CC(=O)OCC)C(=O)COCCCC(C)C)(NC(C)=O)CCCCC1 CC1(C)CC(CNC(=O)NCCc2ccccc2F)CC1O c1(C(c2nnnn2C2CCCC2)NCCCCCC)cc(F)ccc1F.CCOC c1(C(=O)NC2(CNC(C(CC)C#N)=O)CCOCC2)cccc2c1CCCC2 c1(OC)cccc(C(=O)N(CCC(=O)NC2(C(N)=O)CCOC2)C)c1 N1(C(COCCC(C)C)=O)CCN(C(=O)C=Cc2ccccc2C#N)CC(O)C1 C(=O)(CS(=O)(=O)CC(=O)OCC)N1C2CCC(CNC(C(C=C=C)C)=O)(CC2)C1 c1(C(N2CC(CNC(C(CC=C)C)=O)OCC2)=O)ccc(-n2ccnc2)c(F)c1 C1(F)(CNC(C2(C3CC3)CCC2)=O)CCN(C(=O)CCCF)CC1 c1(N(C)CC2CC2(C)C)ncccc1S(=O)(=O)NC1(C)CC(C)(C)C1 C1(C(=O)Nc2cc(C(F)(F)F)n[nH]2)C=CCN1C(c1cc(C(N(C)C)=O)c[nH]1)=O Cc1ccc(S(=O)(=O)NCC)cc1.C(=O)(C(C)(C)CC(C)C)NCC=CCNC(CO)=O Cc1ncc(C(N2CCCCC(CNC(C3(CC(F)F)CCC3)=O)C2)=O)c(=N)[nH]1 CCC(CO)N(C(=O)C=C(C)CNC(=O)CC1CC(NC(C)C)C1)C C1(n2cc(C(CC3CC3)NC(=O)O)nn2)CCCN(C(=O)C(n2ccc(=N)[nH]2)C)C1 C1(NC(C2(COCC)CCCC2)=O)CN(C(=O)C=C(C)C(C)(C)C)C2(CCC2)C1 N1(C(CNC(=O)NC)=O)CCCC(O)(CNC(C2(CF)COC2)=O)C1 N1(C(C2C(C)(C)C2)=O)CC2(NC(=O)CS(=O)(=O)CC3CCCO3)CCC1CC2 C1(N=c2[nH]nc(O)s2)(C(C)(C)C)CCN(C(=O)CN2CC3CC3C2)CC1 c1(C(=O)NC2C(C(=O)NC(C)(CO)C(F)F)CC=CC2)cccc2ccoc12 C1(NC(C2(C)C(CC)CCN2C(=O)CC(Cl)Cl)=O)CCCCN(C)C1=O Cc1csc2ncnc(N3CC4(CCN(C(=O)CCC(N)=O)C4)C3)c12 CC1(C)CCC(CC(=O)NC2CCN(C(C3CCNC(=O)C3)=O)CC2)C1 CC(C)(C)C1=NOC(C)(C(N2CC(n3cc(C4(CCO)CC4)nn3)C(O)C2)=O)C1 C1(CC=C)(NC(=O)CCC#CC)CCN(C(=O)CSC2CCOC2=O)C1 C1(NC(=O)CC2CC3(CC3)C2)C2CCN(C(c3c[nH]nc3C3CCC3)=O)CC12 c1(C(N2C(C)CCC(NC(C3CC4(CSC4)C3)=O)C2)=O)cnc2cccnc2c1 C1(CC)CCC(C(=O)NCC2CC2NC(=O)CCC(=O)Nc2nnc(C)s2)CC1 c1(C(=O)NCC(N(C(=O)C(C)OCC)C(C)(C)CC)C2CC2)cncc(CC)c1 C(c1ccccc1)=CC(=O)NC1CC(C(N2CCCC(CCCO)C2)=O)C1 Cc1c(C(N2CCCC(CC(C(=O)O)NCCOC(N)=O)C2)=O)cccc1N C1(CC(=O)NCC2N(C(c3cc(C(C)(F)F)on3)=O)CCC2)CCC=CCC1 C1(C(=O)NCCCNC(c2ncc(C(F)F)s2)=O)CC2CCCCN2C1 c1(OC)sccc1C(=O)NC(CNC(c1coc(C(F)(F)F)n1)=O)CO N1(C(C)(C)C)CCC(NCC(O)CCCNC(c2csc(C#N)c2)=O)C(C)(C)C1 c1(OC)ccc(CCC(=O)NC2COCC2NC(C2CN(S(C)(=O)=O)C2)=O)cc1 c1(C(N2CCC(NC(c3cncc(CC)c3)=O)C2)=O)ccc(F)c(Br)c1 C(=O)(CCCC(=O)N(CCCCCNC(c1ncc(Cl)s1)=O)C)NC(C)C c1(C(=O)NCCN(C)C(C2CC2Cl)=O)cccc(-c2cccc(Cl)c2)c1 C#CCC(CC#C)C(=O)N1CCCC(CCNC(=O)C(C)Oc2cccnc2)C1 C(=O)(C(F)C1CCC1)NCCC1(C(=O)NC2(CN(C)C)CC2)CC1 CS(=O)(=O)c1cc(C(N2CC3CC2(CNC(=O)COC2CCCOC2)C3)=O)co1 c1(C(=O)NCC2N(C(C(CC(C)C)OC)=O)CCC2)cn2c(n1)COCC2 c1(C(=O)NC2CCN(C(c3cnccn3)=O)C2)cc(Br)cc(F)c1F c1(C(N2C(CNC(CCCNC(C)=O)=O)CCCC2)=O)cc2nc[nH]c2cc1N C1(NC(C2CN(C)C(=O)C2)=O)CC2CN(C(=O)CC3C=CS(=O)(=O)C3)CC12 C1(CNC(C(CC=C)C)=O)CN(C(c2cc(OC)cnc2F)=O)C(C)(C)C1 CC1(O)CCCCC1C1(N)CC1.c1(C(C2(c3ccoc3)CC2)=O)nnnn1CC(F)F C(=O)(C1=CCCCC1)N(CC(CNC(c1c(C)nc(CC)o1)=O)O)C c1(OC)ccc(CC2(CNC(=O)CC3(O)CCNCC3)CCNC2)cc1 CC1(C)CCc2nc(C(N3CCCC(O)(CNC(=O)CC(F)F)C3)=O)ccc2C1 C(=O)(C1=CCC(F)(F)CC1)NCC=CCNC(C(CO)NC(C)=O)=O c1(C(=O)NCC(C2CCCC2)NC(=O)CCc2ccco2)cccn(O)c1=O C(C)(CNC(=O)CC1CCCN1C(C)=O)(C(C)C)NC(c1cnc(CC)s1)=O C1(N(CCOC)CC23CCC2C3)CCN(C(c2cc(OC)ncn2)=O)CC1 C(=O)(C(O)CC1CCCC1)NCC(CN(C(CCC)=O)C)O N1(C(C2CCC3(CCC3)C2)=O)CC2CCN(C(=O)C(F)C(F)(F)F)CC12 c1(CNC(COC2CCC(C)CC2)=O)cccnc1CNC(c1csnn1)=O CC1(C)CC(NC(=O)C(C)(F)C(C)(C)F)CN(C(c2ccccc2)=O)C1 c1(C(=O)NC2CN(C(C(C)C3CCCC3)=O)CC(F)C2)cnc2[nH]cnc2c1 N1(C(Cc2c(C)scc2)=O)CC(NC(C2(C3CCCCO3)CC2)=O)CC12CCC2 C1(C(=O)NC(C)(C)C)CCC(O)CN1C.N12CC3C(C3C1)C(=O)NCC(C)NC(=O)C2 Cn1[nH]c(C2CC(NCc3ccnn3C(F)F)CC(C(F)(F)F)C2)nc1=O C(C)(CCCN=c1[nH]c(=NCC2CSC2)[nH]c2c1CCC2)c1cccc(OC)c1 C1(C(=O)NCc2ncc(C)nc2)CN(Cc2ccc(O)cc2)CCC1O c1(OC)cccc(CSC)c1C(N1CC(n2cc(-c3ccc(C#N)s3)nn2)C1)=O C1(NC(CC2N(C(C)C)CCC2)=O)CN(C(=O)C(F)(F)c2ccccc2)CC1F C1(CNC(C(CC=C)NC(C)=O)=O)CC2CCC1N(C(c1cc(Cl)no1)=O)C2 Cn1oc(-c2ccccc2)cc1=O.N12CCC(C1)n1cc(nn1)C=CC2=O C(=O)(C1CCCc2scnc21)N1CC(CCNC(C2(S(N)(=O)=O)CC2)=O)(OC)C1 c1(C(=O)NC(C)CNC(C2CCCCN2C)=O)ccc(F)cc1OC(F)F N1(C(C2C(CCC)C2)=O)CC2CCC2(CNC(c2cnc(S)n2C2CC2)=O)C1 N1(C(C(C)NC(=O)C(C)(C)C)=O)CC2CCC(Nc3nccc(C#N)n3)C2C1 C(=O)(C1COc2ccc(Cl)cc21)NCCC1CCCN(C(CSC)=O)C1 c1(C(=O)NC2(c3cn(-c4ccc(C)c(F)c4)nn3)CC2)c[nH]c2cc(C#N)ccc12 CCCCC(C)(F)C(=O)N1CCOCC(CNC(=O)CCNC(=O)OC)C1 C1(C#N)(C(=O)NCC2(C)N(C(CCC3CC(OC)C3)=O)CCC2)CCC(=O)CC1 c1(C(=O)NCC2(F)CCN(C(Cc3cc(C)on3)=O)C2)ccc(I)c(Cl)c1 N1(c2snc(C)c2C#N)CCC2(CC1)CN(C(c1cncs1)=O)CC(C)O2 C12(CNC(c3cn(CCO)nn3)=O)CCC(CC1)N(C(=O)CCOC1CC1)C2 CCCCCC(F)C(=O)NCC1CCCCN(C(c2oc(CC)nc2C)=O)C1 C(C(C)(CNC(c1cncc(CNC(=O)CCCn2cccn2)c1)=O)CO)OC Cc1nc(=NCC2C(C)CCCN2C(=O)Cc2nn(C)cc2Cl)[nH]cc1Br C(=O)(CCCC(N)=O)NC(C1CCC(OCc2ccccc2)C1)C.CCC1C(=O)N1 N1(C(CCOCC#C)=O)CC(C(=O)NCc2n[nH]cc2COC)C2(CCC2)C1 N1(C(c2c(N)ccc(C)c2F)=O)Cc2ccccc2C(NC(=O)CC2CN(C)C2)C1 C1(C(=O)NC(C=C)(CC)CC)CN(C(=O)C(F)CC(C)(C)C)CC1C1CC1 CC1=C(C)CC(C)(NC(c2occc2CNC(=O)C(C)(C)CO)=O)CC1 O=C1CCN(CC23CCC(CC2)OC3)C(=O)N1CCCCCCCOC(F)(F)F C1(CNC(c2c(CC)csc2)=O)CCC2(CCC2)C1NC(=O)C(Cl)=CCl Cc1ccc(C(N)=O)c(C(N2CC(Cn3cc(-c4cccc(Cl)c4)nn3)C2)=O)c1 c1(C(N(C2CCN(C(C3CN(N=O)C3)=O)C2)CC2CC2)=O)cc2n(n1)CCO2 C(=O)(CCCCCC#N)N1CCCC(C)(CNC(c2ccc(C(C)=O)cn2)=O)C1 c1(CN2CC3C(C(=O)NCc4cccc(OCC)n4)C3C2)cc(O)ccc1F C(CCC(C)(F)F)N(C(CCC1(C)CN(C(C(C)n2cccc2)=O)C1)=O)C CC1(C)CN(c2nc(Cl)ncc2C(F)(F)F)CCC1NC(=O)CCC1CCCO1 n1(CC(=O)NC(CN(C(c2cnns2)=O)CC)C)nccc1C N1(C(C2CCOC2)=O)CCN(C2CC2(F)F)CC1.c12cn(nn1)CCC2C(=O)O N1(C(C(C(C)C)O)=O)CCCC2(C1)CN(C(c1ccnn1-c1ccccc1)=O)C2 C(=O)(C1CCOc2c(F)cccc21)N1CC(CC(CC)NCc2cc(F)n[nH]2)C1 Oc1ccc2c(c1)C(Nc1ncc(C(c3ccccc3)(F)F)s1)CCC2 c1(C(=O)NCCCC(CCC)NC(C(CC=C)C)=O)noc2ccccc12 c1(NC2(C#N)CN(C(COC(C)(C)C)=O)C2)cc(F)c(F)c(F)c1F N1(C(CSCCC)=O)CC2CCN(C(c3cn(C(F)F)c(C)n3)=O)CC12 C1(CNC(=O)COCCF)COCCN(C(=O)Cc2cccnc2)C1 N1(C(CCCCCC)C(=O)NC2CC2)CCn2c(nc(C(F)(F)F)c2Br)C1 C(=O)(CC(C)(C)C(C)=O)NCC1N(C(C(C)OCCOCC)=O)CCCC1 C12(CC3C(C(=O)NCCCNC(C=C(CC)C)=O)CC3)CC3CC1C2C3 C1(NC(Cc2n(C)ccc2)=O)CC2CC(NC(C3CCC(=O)N3)=O)CC2C1 C(C(C)(C)CN(C(=O)C(CN)OC)C)OC.C12(OC)CN(C1)C(=O)C2 N1(C(c2c(C)onc2)=O)C2CCC1C(F)C(NC(=O)CCn1ncn(C)c1=O)C2 O=C(CCNC(=O)OCc1ccccc1)NNC(=O)NCCNC(C1CCCS1)=O C1(CNC(C=C=C(C)C)=O)CCN(C(=O)CC2(CO)CC2)CC1(F)F C1(C(=O)NCCCN2CCC(NC(=O)C(Cl)=CCl)C2)OCCOC12CCC2 CC1(C)CN(CCCO)CCN1C(c1ncc(Cl)cc1F)C(=O)NC1CC(F)(F)C1 C1(C(N2CCCCC(NC(c3ccc(CCC)s3)=O)C2)=O)CC2CCCC(C1)C2 CC1CC(NC(C2CC(O)C2)=O)CN(C(c2cc(CN(C)C)ccc2Cl)=O)C1 C(N=c1[nH]c(Cl)ncc1Br)C1(F)CCN(C(CSc2cccc(OC)c2)=O)CC1 C12(CC(=O)NCC3(O)CN(C(CNc4cn(C)nc4)=O)C3)CCCCC1C2(F)F C1(NC(C2(C)CCCCC2)=O)Cc2ccccc2C1NC(=O)CC1(C)CC1F N1(C(C2(OC(C)C)CC2)=O)CC=CC(C(N2CC(N(C)C(N)=O)C2)=O)C1 C(C(CC1CCCC1)C(=O)NC(C)C)NC(C(=O)NCC)=O.C1CCS1 c1(OC)cccc(-n2nc(C3CC3C)nc2-c2cccc(SCC3CC3)n2)c1 N1(C(C(C)=C2CC2)=O)CCC(c2ccccc2)(NC(=O)C(O)CCc2ccccc2)C1 Cc1cc(C)n(CC(=O)NCC2CN(C(=O)C(C)(C)c3cscn3)CC2O)n1 c1(C(N(CCOC)CCNC(=O)CNc2cnn(C)c2)=O)cncc2c1CCC2 c1(C(N2C3C(NC(CC4(C=C)CC4)=O)C(C3)C2C)=O)cc(F)c(Cl)cc1F c1(C(=O)NC2CC(CCNC(C3(n4cncn4)CC3)=O)C2)cc(Cl)c[nH]1 c1(C(=O)NCc2c(CCNC(CC(COC)C)=O)ocn2)cc(C)c(Cl)cc1F c1(C(=O)NC2C(CNC(C(CCOC)C)=O)CC2)ccc2c(c1)C(=O)NC2 C1(C(N2CCC(C(=O)OC)C2)=O)CCC2CCC1N2C(=O)C=C(C)C NS(=O)(=O)CCCC(=O)NCC(CO)NC(=O)CSCc1ccncc1 CCC(C)CCC(=O)N1CC(NC(C2(n3cncn3)CC2)=O)C(CC)C1 C1(CCNC(C)=O)CCN(C(C2(C3(O)CCOC3)CC2)=O)CC1(F)F Cc1scc(C(=O)NCC(C(C)C)NC(c2ccc(CS(C)(=O)=O)o2)=O)c1C c1(NC(C2C3(CN(C(C(C)(C)C)=O)C3)C2)=O)cnc(Cl)cc1Br N1(C(c2c(C)coc2)=O)CCCC2C(NC(c3cccc(C)c3N)=O)C(C)(C)C12 N1(C(C2CCC(NC(c3c(C)cns3)=O)CC2)=O)CC2OCCN(C)C2C1 CCC(C)(CO)C(=O)NCC1(CNC(c2ccc[n+]([O-])c2)=O)CCCCC1 C1(NC(c2c(SC)csc2)=O)CCN(C(=O)CCN(S(C)(=O)=O)C)CC12CC2 C#CCC(C(=O)NCc1nc(CNC(=O)CSCC(F)(F)F)cs1)C1CC1 CC(CC(C)(C)C)C(=O)NCC1CCC(CNC(c2cc[nH]c(=N)c2N)=O)CC1 N1(C(CC(C)(C)SC)=O)CC2(CNC(c3cnc(C)[nH]3)=O)CC1CCO2 CCCC(CNC(=O)CCOC1CCC1)C(=O)NOC=Cc1cccnc1 C12(C(N(c3cccc(Br)c3)C(C)C)=O)CC1CN(C(c1nc(Br)cs1)=O)C2 N1(C(c2c(CNC(c3cc4ccsc4[nH]3)=O)ocn2)=O)CCSC2COCC12 C(=O)(C#CC1CCOC1)N(C(C)C)CCNC(C1(CCc2ccccc2)CC1)=O c1(C(=O)NCC2C(NC(C=CCC)=O)CCC2)cc2c(nc1N)CCC2 c1(C(N2CC(C(C)NC(C(CC)C(=O)OC)=O)C2)=O)ccc(Cl)c2ncccc12 c1(C(N2CCC(CCC(=O)NCCc3ccn(CC)n3)C2)=O)cnncc1NC c1(OCc2cn(CCC(=O)NCC(CNC(CC)=O)F)nn2)cccnc1F c1(C(=O)Nc2c(C(=O)NCc3c(CC)cccc3)n[nH]c2)cc(Cl)nc(Cl)c1Cl C#Cc1cccc(OCC(=O)NC2CC3CC2N(C(c2cccnc2C)=O)C3)c1 C1(CC(=O)N(C2CN(C(C3(O)CCOCC3)=O)CC23CC3)C)CCC(C)(O)CC1 c1(OC)cccc2c1OCC(C(=O)NCCN(C(=O)C(O)CC(C)C)C(C)C)C2 C1(C(=O)NCC(CNC(C2C(CCC)CCC2)=O)(C)C)(COC)CC2(CCC2)C1 N1(C(c2scc(C)c2C)=O)CCC(CNC(c2ccn(C(C)(C)C)c2)=O)C(C)C1 N1(CC(=O)NCC(C)NC(=O)CSc2cccc(O)c2)CCS(=O)(=O)CC1 N1(C(C(C)C2CC2)=O)CC2CCC1C(CNC(c1coc(S(C)(=O)=O)c1)=O)C2 CC1(C)CC(CC(N2CCC3C(NC(=O)CCN4CCCCC4)C23)=O)CCO1 N1(C(c2c(SCC)cccc2)=O)CC2CC(C1)CN(C(=O)C(CO)C(F)(F)F)C2 N1(C(c2ccncc2O)=O)CCC2CCN(C(c3c[nH]cc3Br)=O)CC2C1 C(CCCC(CO)NC(C1CC2CC2C1)=O)NC(CCc1c(C)nn(C)c1)=O c1(CC)c(C(=O)NCC2(O)CCN(C(c3ocnc3C)=O)C2)cnn1C(C)(C)C c1(C(=O)NC(C)CCCNC(=O)Cc2cncs2)ccc2nc(CO)[nH]c2c1 N1(C(C(CC)C(C)C)=O)CCCC2(CCN(C(c3ccncc3C)=O)C2)C1 c1(C(N2CC(C(C)NC(c3nnc(S)n3C)=O)C2)=O)c(F)ccc2[nH]ccc12 N1(C(Cc2cc(C)no2)=O)CC(C)(C(=O)NC(CO)CCO)CC1(C)C C12(CC(=O)N(C3CCCC3SC)CC)CCC1CN(C(c1c(C)nsc1N)=O)C2 C(=O)(C1=C2CCCN=C2NN1)NCC(CO)NC(C(n1ccc(C)n1)(C)C)=O CC1(C)C(C)(NC(=O)C(=O)NCC23CCC2C3)C1(C)C C1(OCC)(CNC(=O)CC2CCC(O)C2)CN(C(c2coc(Cl)c2)=O)C1 c1(NC(C(CNC(c2[nH]cc(C(C)=O)c2)=O)O)=O)cc(CO)cc(C)c1 N1(C(CN(CCC)C)=O)CC(C)(C)CC1CC(N1CCC1C1CCC1)=O C1(CNC(CCN(CCCCC)C)=O)CN(C)CCN1C(=O)CNC(=O)OC Cc1ccc(F)c(CN2CC=CC2C(=O)Nc2ccc(Cl)c(O)c2)c1 CCCCCCC(C)(C)C(=O)N(CC(CC)NC(=O)C(F)CC1CCC1)C CC1(CC(=O)NCC2CCOC2C(N2CCC(C(F)F)C2)=O)CCOC1 N12CC(C3CC3)(C1)OCCNC2=O.N(CC)(CC)CC n1(CCC(=O)NC2CC(C(=O)NC(c3ccncc3Cl)C)C2)ccccc1=O C(C(C)(O)CNC(=O)CC1(C2CC2)CC1)NC(CN(C1CC1)CC)=O CC1CC(C(N2CCOCC2CN(C(=O)C=CC(N)=O)C)=O)CCO1 C12(C(N(C)Cc3c(CNC(C(C)OCC)=O)cccc3)=O)CCCN1CCC2 c1(C(=O)NCC2C(NC(c3c(CC)noc3)=O)COC2)cn2nc(OC)ccc2n1 C1(CNC(CSCC#C)=O)CN(C(C23CC(N(C)C)(C2)C3)=O)CCC1(C)C c1(NC(C(C)(Cn2ccnc2)C(=O)O)=O)cccc2ncnc(O)c12 CC1(C)CCC(C(=O)NO)(NC(c2ccc(C(N3CCCC3)=O)o2)=O)C1 c1(C(N2CCC(C(C)NC(=O)Cc3nc[nH]n3)C2)=O)cnn(C(C)(C)C)c1N Nc1c(C(N2CCN(CCF)CC2c2ccccn2)=O)cccc1I C1(C(=O)NC(CC=C)CC(F)F)CCN(C(c2cccc(O)c2F)=O)C12CCC2 c1(C(=O)NC(C2CCN(C(=O)C(C)(C)CN(C)C)CC2)C)ncc2[nH]ncc2n1 C1(C(=O)NC2CCC(C)N(C(c3cccc[n+]3[O-])=O)C2)CCCC2(CCC2)O1 Cc1scc(C(=O)NCC(CO)NC(=O)CCC2CCC(=O)NC2)c1Br S(=O)(=O)(c1ccc(N2CCC(O)CC2)c(F)c1)NC(C=C)C1CC1.C(COC)OC Cc1ccc(CCC(=O)NC(C)(CNC(C2CCC2(C)C)=O)CO)s1 C1(C(N2CCCC(CCC(N3C4(C)CC4CC3)=O)C2)=O)CC2(CCCO2)C1 C1(NC(Cc2c(C)ccs2)=O)CCN(Cc2cc(-c3cnn(C)c3)no2)CC1O C(C(C)(C)CN(C(=O)CC(C)O)CC)NC(CC1(CC)CCC1)=O C1(NC(c2nc(CCC)sc2)=O)CCN(c2nc(Cl)ncc2C)CCC1CO c1(C(=O)NC2CCN(C(=O)CCc3cccnc3)CC2F)cnn2ccccc12 c1(OC)ccccc1C(N)CC(=O)NCC1CC1c1ccc(F)cc1 C1(C(N2C(C=C)CC2)=O)N(C(=O)C=Cc2cocn2)CC12CCCC2 C1(CCNC(c2nc(OC)c(F)cn2)=O)CN(C(=O)CNC=O)CCS1(=O)=O Cc1c(C(F)(F)F)nc[nH]c1=NCC1CC2(C1)C(F)(F)C21CC1 C1(C(=O)NC2C(NC(c3c(OC)nccc3)=O)CC2)CCCN1S(=N)(=O)N(C)C C1(n2cc(CCNC(c3nccs3)=O)nn2)CCCN(C(=O)CSC2CC2)C1 C1(C(N(C)C)=O)CC(F)(F)CN1C(c1cccc(N(C)C)c1)=O c1(C(=O)NC2C(N(C(=O)CCCF)C)CCCC2)cc(F)c(Cl)cc1Cl C(=O)(C1=C(Cl)CCCC1)NCC1(F)CCC(CNC(C(=O)N(C)C)=O)CC1 C1(C)(C(N2CCCC(CC(=O)NC(CC)C(=O)NC)C2)=O)CCC2CC2C1 N1(C(C(CCC)C)=O)CCC(C(C)(C)C)CC1CNC(c1cnc(C(C)(C)C)[nH]1)=O C12(CNC(CCCC#C)=O)CC(CO1)N(C(C1(C)CC=CC1)=O)C2 C(N=c1cc(C#N)nc(C2CC2)[nH]1)C1(NC(CC2CCCC(C)C2)=O)COC1 Cc1c(C=CC(=O)NC2CC(NC(C3(F)CC3)=O)C2)cnn1C Cc1ccc(C2CC2C(=O)NCCCC2(NC(c3nc(O)sc3C)=O)CC2)c(C)c1 N1(C(C(C)C2CCCC2)=O)CC(C(=O)NC2COCCC2(F)F)C(F)(F)C1 C1(C(=O)NCCCCCC)C2C(CN1Cc1cc(C)ccc1Br)C2(C)C N1(C(c2n(CC#C)cnn2)=O)CCN(C)C(CNC(c2ccc(C)c(F)c2)=O)C1 C(=O)(C(O)P(C)(C)=O)NC1(COC)CCN(C(c2csc(-c3nc[nH]n3)n2)=O)C1 Cc1cncc(C(=O)NC(Cn2ccnn2)C(=O)NC2CC(CCO)C2)c1 CC(C)CCC(=O)NC1C=CC(CC(=O)NOCCCC(C)C)C1 CC(C)(C#N)C(=O)NC1CCN(C(c2cnc(-c3ncccn3)s2)=O)C1 CC(CCC(=O)NC(Cc1cc[nH]n1)C(=O)NCCc1ncc[nH]1)N(C)C Cc1c(C(=O)NCC2CCN(C(=O)CCCCC(F)(F)F)C2)oc2c1C(=O)CCC2 C#Cc1ccc(Cl)c(C(=O)NCC2(F)CCN(C(C3CCCOC3)=O)C2)c1 CC1N(C(C2CC(F)CCN2C(=O)C(O)C2CCC2)=O)CC(C)OC1(C)C N1(C(c2c(C)onc2)=O)CCC(CNC(=O)Cc2ccc(Cl)c(Cl)c2)C(C)C1 C(=O)(CCCOC)C1CC1.c1(CSCC)ccccc1.C1(C)=CC2(CC2)N(C)C1=O C1(S(C)(=O)=O)(C(=O)NC2CCC(C)N(C(=O)C3=NNC(=O)CC3)C2)CCCCC1 c1(C(=O)NC2CCN(C(c3nnc(C)s3)=O)CC2C)c(F)ccc(F)c1F N1(C(Cc2cc(C)on2)=O)CC2CC(C(=O)NCc3ccc(O)cc3C)C(C2)C1 C#Cc1ccc(C(N2CC(CCC(=O)N)C2)=O)nc1.C1(N(C)C)CCSC(C)C1 C1(C(=O)NC2(CC(C3CC3)NC(C3(O)CCC3)=O)CCCC2)CC2(C1)CC21CC1 C1(CC)CN(C(c2cc(C)sn2)=O)CCN1C(C1CCC1(F)F)=O C1(C(N2CCC(CN(C(C(C)NC(C)=O)=O)C)C2)=O)CCc2cnn(C)c2C1 c1(C(N2CC(CCCNC(C(C)N(C)C)=O)OCC2)=O)c(O)cccc1F S(=O)(=O)(c1cccc(C(=O)NCCCCCCNC(c2coc(C)c2)=O)c1)NC C#CCCCCC(=O)NCC(C1CCCN1C(C1(C)CCC(=O)N1)=O)(C)C N1(C(c2n(C)c(S)nc2)=O)CCC2C(C1)NC(=O)CN2C(=O)CC1CCCC(=O)N1 C1(c2n(C(C)C)nnn2)(NCCn2cncn2)CCC2C3CCC(C3)C12 N1(C(C(C(C)C)(C)O)=O)CC(NC(=O)COC2CC(F)(F)C2)CC12CCCC2 C(=O)(C(C)(O)C(C)C)N(CCNC(=O)C(=O)Nc1ccccc1SC)CC CC1(C)C(CNC(c2cc(Cl)sc2Cl)=O)CCN1C(=O)C=Cc1nccs1 CON(CCC(=O)N1CC=CC(O)C1)C(=O)C1CC1CNC N1(C(c2nnc(C(c3ccccc3)=O)s2)C)CC(c2ccccc2)N=CC1C c1(C(=O)NCc2cc(-n3ccnc3)ccn2)ccc(CO)cc1 C(=O)(C(C)C1=CCCC1)NC(CC)CNC(c1ccn(C)c1C)=O C(=O)(C1=C(F)CN(C(C2CC2=C)=O)CC1)N(CCC=C)C Cc1ccc2ncc(C(=O)NCC(C)CN(C)C(C3CC3C3CC3)=O)n2c1 C(=O)(C(CC(F)F)N(C(=O)C(C)c1cccs1)C)N(C(C)CCO)C N1(C(C(c2ccccc2)OC)=O)CC(CNC(C2CNC(=O)N2C)=O)CC(C)C1 c1(C(=O)NCC2N(S(C(C)C)(=O)=O)CCCC2)c(Br)ccnc1Cl N1(C(C2N(CC)CCC2)=O)CCCC2CN(C(C3CCC(C)CC3)=O)CC12 C1(NC(C(COC)C)=O)CCCCC12CCN(C(C1CSCCS1)=O)CC2 C1(NC(C(CCOCC)NC(c2cccc(F)c2)=O)=O)CN2CCC1(F)CC2 N1(Cc2c([N+](=O)[O-])ccc(C)c2)CC2(CCN(C(C)C)CC2)CNC1=O C1(C(=O)NCC(C)NC(=O)CSCC(c2ccccc2O)=O)CC12CC(C)(C)C2 C(S(=O)(=O)c1ccc(Cl)c(Cl)c1)OCCOc1c(-c2c(C#N)cccc2)cccn1 C1(C(=O)NCCNC(=O)COC(C)CC)(SC)CCOCC1.C1(NC(C)=O)CC1 C1(C#N)(SC)CN(C(=O)CN2CCC(Oc3ccccc3Cl)C2)C1 CC1(CNC(c2ccco2)=O)CCN(C(C2CCCN2S(C)(=O)=O)=O)CC1 CCCCC(C)CCC(=O)N1CCCCC1CN(C(=O)CCCCCN)CC N12CC3C(C3C1)NC(=O)NC(F)(F)C2=O.c1(OC)ccc(C2CCOC2)cc1 N1(C(C(C)OCC(F)(F)F)=O)CCC(C)C(CNC(c2cc(C#N)n(C)n2)=O)C1 C1(CC(N2CC(=C(CNC(c3nnn(C)n3)=O)F)C2)=O)CC2COCC12 N1(C(C=C(C)COCC(=O)Nc2ccc(=O)oc2)=O)CCOC(C)C1 C(=O)(CCCC(N)=O)NCC(CNC(C1N(CCCC)CCOC1)=O)C C12(NC(c3cn(C)nn3)=O)CCC1CN(C(=O)C(O)Cc1cccc(Cl)c1)C2 C(F)(C(=O)NCC(C)NC(=O)Cc1cn[nH]c1)OC c1(Cc2c(OCC(=O)O)cccc2)ccc(Br)cc1CN1CCC(C(F)(F)F)C1 C1(C)(NC(c2nc(OC)oc2)=O)CCCCC1NC(C12CCCC1C2(F)F)=O N1(C(c2c[nH]c(=N)s2)=O)CC2OCC(NC(C3CCCCO3)=O)C2C1 O=C1CC(C(=O)NC2(CCNC(=O)CCCc3ccccn3)CCCC2)CCN1 C1(C(N(C)CC2CN(C(C3CC(=O)CO3)=O)CCO2)=O)CCc2ccnn2C1 C1(CC)CN(C(C2CCCC2CNC(=O)Cc2ccc3c(c2)CC3)=O)CC1(C)C C1(C(N2CC(F)(C(=O)NC(C(O)CO)C3CC3)C2)=O)CCNC1=O N1(C(CC)=O)CCCC(C(=O)NCc2ccc(OC(C)CC)nc2)C1 C1(C(N2CC(C)(CC=C)C2)=O)CC2CN(C(c3ccncc3OC)=O)CC2C1 CC(CBr)N=c1cccc(S(=O)(=O)N2CCC(CCCC(N)=O)CC2)[nH]1 C#Cc1ccc(C(N2CCCC(C)(C)C2CNC(=O)C(O)CCCC)=O)cc1F Cc1cc(C)n(CCC(N2CCC(C(C)C(N3CCC(C(F)F)C3)=O)CC2)=O)n1 c1cnc(Cl)c(C)c1.C1C(CC2CCCC2)C(=O)N1.C1CC(=O)N1.CC(=O)OCC c1(SC)ccc(Cl)c(C(N2CCC(N(C(=O)Cc3nncn3C)CCO)C2)=O)c1 c1(NC(CCCc2onc(CCC)n2)=O)ccc([N+](=O)[O-])cc1C CCCCC(C(=O)NC)NC(=O)C(C1(O)CCC1)NC(=O)CC1OCCCO1 N1(C(C2C(C(=O)OC)C2(C)C)=O)CC2CC2(NC(=O)Cc2sccc2Cl)C1 c1(C(=O)NCC(CC=C)NC(=O)C=Cc2sccc2C)cc(Cl)c2c(c1)OCO2 C(C(CC(C)C)C(=O)OCc1occc1C(=O)OC)c1c(OCC)c(F)ccc1 CC1=C(C(=O)NC2CCOC(C(=O)N(C)Cc3noc(C)n3)C2)SCCO1 c1(C(=O)NCC=CCNC(c2nn(C)c3c2CCC3)=O)ccc2c(c1)CCC2(F)F CCCC(C)C(=O)NC1CN(C(c2cnn(C(C)C)c2C)=O)CC1CCO N1(CCCc2c(C)ncs2)CC(NC(=O)COC(F)F)C2(CCOCC2)C1 c1(C(N(C2CCN(C(C3CC(=O)N(C(C)(C)C)C3)=O)C2)C)=O)cn2ncccc2n1 N1(C(c2c(C)c(Br)ccn2)=O)CCC(N=c2[nH]c(-c3cnn(C)c3)no2)C1 C1(NC(Cc2c(C)noc2C)=O)CN(C(c2ccns2)=O)CCC1C C1(N(C(CCCC(C)C)=O)C)CCC2CN(C(=O)CSCCC(F)(F)F)CC12 c1(Sc2ccccc2CC(=O)N(C(C(C)C)CO)C(C)C)cccc(F)c1 c1(C(N2CC3(C(C(=O)NCCOCCCCl)C3)C2)=O)cc(C(F)(F)F)ccc1Br N1(C(C2(C(C)C)CC2)=O)CCCC(C(=O)N(C2CCC(O)CC2)C)CC1 C(C(CNC(c1sc(C)nc1OC)=O)C(C)C)OC c1(C(=O)NCC2CC3(CC3)CN2C(c2nncs2)=O)cnc2occc2c1 c1(N2CCCC(C(N3CCC(OCC)CC3)=O)C2)cc2c(OC)[nH]c(=N)nc2s1 C(=O)(C(F)CC(C)(C)NC(=O)C(C)CC(F)(F)F)NCC(C)O C1(CC)(CO)CCOCC1.n1(CC2CCCO2)cc(C2CC2)cn1 N1(C(c2ccc(OC)nc2)=O)C2CCCC1CC(NC(=O)C=C1CCSCC1)C2 C1(CC)CN(C)C(=O)CN1C(=O)NCCN1C(C)CCC1C CCS(=O)CC(=O)NCC(C)N(C(c1cccc(-c2csc(C)n2)c1)=O)C1CC1 C1(C)(C(=O)NCCN(C)CC)CC12CCN(c1nccc(N)c1C)CC2 Cn1ncc(C(=O)NC2CCCC2(C)C)c1F N1(C(CCCN(C(C)=O)C)=O)CCC(C)C(CNC(=O)CNc2cnn(C)c2)C1 C(CCCCC(=O)NCC1CCO1)N(C)C(c1coc(C(N)=O)c1)=O c1(CC)c(C(=O)N(CCCCNC(=O)C(C(C)C)c2cnn(C)c2)C)csc1C C1(NC(C(CC)SC)=O)CC2(C1)CC2NC(c1cncc(C)n1)=O c1(OC)ccc(C)cc1C(=O)NCC1CC(NC(=O)C=C2CN3CCC2CC3)C1 c1(OC)ccc(C(=O)NCC2C3CC2N(C(=O)CCc2cscn2)C3)nn1 CN1CCOc2cc(CN3C4CCC3CC(C(=O)NCC3CNCCO3)C4)ccc21 C1(CNC(C(C)C2CCCC2)=O)CCN(C(c2nnn(C)c2N)=O)C(C)C1 Cc1[nH]c(C)c(C(=O)NCC2CCC2NC(c2nc(Br)c[nH]2)=O)c1C Cc1cc(C)n2nc(CC(N3CCC(CNC(C4(F)CC4)=O)C(C)C3)=O)nc2n1 N1(C(C(CC)C)=O)CCC2(CC1)CC2NC(c1cc(F)ccc1C)=O C=C(Br)CCC(=O)NC(C1CCN(C(=O)C(C)n2ccnc2)CC1)(C)C C1(NC(C(CCOC)NC(=O)CCC2OCCO2)=O)CCc2nncn2C1 N1(C(CS(=O)(=O)NC)=O)CCC(C2CC2)(CNC(=O)Cc2cc(C3CC3)no2)C1 C1(C(=O)NCC(c2ccccc2)O)COCCN(C(c2c[nH]cc2C2CC2)=O)C1 c1(-c2cn(C3C(C(=O)Nc4nc(C)nn4C)C3)nn2)c[nH]c2cccc(F)c12 N1(C(CCN(CCC)C)=O)CCCC(CCOCCOCCOCCO)C1 C1(C(C)C)(C(=O)NCC2CC3CC3C2)CCCN1C(=O)CC1(n2cccn2)CC1 c1(CC(N2CC(CCNC(C=CCC)=O)C(C)C2)=O)cc2cc(Cl)ccc2[nH]1 CC1(C)OCCC1C(=O)NCC1CC(NC(=O)CNC(=O)C2CC2)CC1O N1(C(=O)Nc2ccc(-n3cc(CCCCCO)nn3)o2)CC2CC3CC2C1C3 N1(C(c2cn(CCCC)nn2)=O)CC(NC(=O)C(C)SC)C2CC2C1 Cc1noc(C)c1CN(S(=O)(=O)CCCc1ccccc1)C Nc1nn2ccccc2c1C(N1CC2CCCC2(C(F)F)C1)=O Cc1ccc2occ(C(N3CCC4CCN(C(=O)C=CCF)C4C3)=O)c2c1 c1(OC)ccc(F)c(CN2CC3CN(C(c4cc(F)ccc4F)=O)CC23)c1F c1(C(N2CCC(F)(CNC(C(C)(C)OCC)=O)C2)=O)c(OC)ccc2c1CCC2 C1(C(=O)NC)(CC)CCN(C(c2ccc(OC)nn2)=O)C1 N1(C(C)=O)CCCC1C(N1CCCC1C(C)(C)NC(=O)C=C(C)C(C)C)=O c1(C(=O)NCCC(C)NC(CCc2cnc(C)o2)=O)cnc(Br)c(N)n1 Cc1ccc(CCC(=O)N(CC(O)CNC(C2(C(N)=O)CC2)=O)C)o1 N1(C(C2N(C)CC2)=O)CC2CC(C1)CN(C(C1(C)CCCO1)=O)C2 c1(OC)cccc2[nH]c(=NCc3sccc3C)[nH]c(=NC(C)CN(C)C(C)C)c12 C=CC1(C(=O)NCCCCCO)CCNC1 C1(OC)CC(CNC(=O)C(c2ncccc2C)(F)F)N(C(C2(CCF)CC2)=O)C1 c1(C(=O)NCC(C)N(C(=O)Cc2ccn(C3CC3)n2)C)ccc(F)c2c1CCC2 C1(CC(=O)NCCCCNC(=O)CCSc2ccc(F)cc2)CCC2(CCC2)O1 C1(C(=O)NC2CC(CNC(C3CCOC3)=O)C2)(OC)CCCCC1 C#Cc1ccc(C(=O)NC2C3CC(NC(=O)C(C)(CC)OC)CC23)cc1C Cc1ccc(Cl)c(O)c1C(N1CC2CC(CNC(C3(C)C=CCC3)=O)C2C1)=O C1(C(=O)NCC2(OC)CCN(C(=O)C(C)(C)N(C)C)CC2)CCn2nnnc2C1 c1(C(N2CCC(OCCNC(=O)CC3CC4(CC4)C3)C2)=O)ncc[nH]c1=O c1(CCN(C(CC2(C#N)CCC2)C(=O)NCC(F)F)C)cccc(F)c1 c1(CC)cnc(C)c(NC(=O)CCOCCN(C(=O)C(C)(COC)OC)C)c1 C1(CC(N2C(C(C)(C)NC(C3(C=C)CCC3)=O)CCC2)=O)CC(C)(C)OC1(C)C Cc1cc(OC(=O)C(C)C(=O)O)ccc1-n1cccc1C(C)C CC(C)(C)C(C)(C)C(=O)N1CCCC(CNC(C2CN(S(N)(=O)=O)C2)=O)C1 N1(C(c2cc(C)cc(F)c2)=O)CC(NC(C2C(C)C2C)=O)CC12CCCC2 C1(C(N(C(CNC(Cc2nc(CC)sc2)=O)C)C)=O)CC(C)(C)CCO1 CCCC(CCc1ccccc1)C(=O)Nc1ccc(I)c(C(=O)OC)c1 S(=O)(=O)(c1c[nH]ccc1=NCC1CCCOC1)N(C(c1ccc(Cl)cc1)C)C C1(CN(CCC)C)CCN(C(c2nc(-c3cnn(C)c3)cs2)C(=O)NC)C1 C1(CC(=O)NC2CCN(C(=O)CC3(C)CC3(F)Cl)CC2)(CN(C)C)CCOCC1 Cc1oc(C2CCOCC2)nc1C(N1CC(CNC(C2COC2)=O)CC1C)=O N1(C(C2(OC)CCCC2)=O)CCC(C)C(CNC(C2(F)CCCC2)=O)C1 C1(CC(C)C)CCCN(C(=O)C(CCO)NC(=O)CC(Cl)Cl)C1 c1(OC)cc(OC)c(C(N2CCN(C(=O)Cc3ccsc3)C(C(C)C)C2)=O)cn1 c1(OC)ccc(CC(N2CC3(NC(c4ccc(CO)o4)=O)CCC2C3)=O)c(C)c1 C=CC(CCC)CC(=O)N1CCC(C)(NC(=O)CC2C=CCC2)CC1 C(=O)(CCC(=O)N1CCC(CC(=O)NCC(COC)OC)C1)OC C1(C(N(CC(CC)NC(=O)C#CC(C)(C)O)C)=O)CCc2cncn2C1 c1(CN(CC=C)C)ccc(C(=O)N(CC(C)NC(C2(C)C=CCC2)=O)CC)cc1 C(CC(=O)Nn1ccnn1)(C(C)(C)C)NC(c1c(OC)cncn1)=O c1(C(N2CCC(c3ccccc3)C2)=O)cc(-c2ccnc(O)c2)c2[nH]ccc2c1 c1(-c2nc(C)sc2)cccc(CNC(=O)C(=O)NCCC(O)C(=O)O)c1 C(CCC(O)C(=O)NCC1(CO)CCOC1)NC(C1(OC)CCCCC1)=O N1(C(c2c(C)ccc(C)n2)=O)CCN(C(=O)Cn2cnnn2)C(C)C1C N1(C(C(O)NC(=O)OCC)=O)CC2CN(C(c3ccnnc3SC)=O)C2C1 c1(CCC(N2CCC(OCn3cc(CC4CCCC4)nn3)C2)=O)ccccc1Br CC1CCC=C1C(=O)N1CC(C(=O)NCc2ccc(C(F)(F)F)cc2)C2(CC2)C1 Cc1cc(C(N2CCC(C)N(C(c3nnsc3N)=O)CC2)=O)c(C)c(C)c1 N1(CCC(=O)NCC(CNC(c2c(CC)nccn2)=O)(C)O)CCP(C)(=O)CC1 c1(CC)cc(C(N2CC3CC(NC(c4ncoc4C4CC4)=O)C2C3)=O)cc(O)n1 N1(C(C23CC(OC)C2C3)=O)CCC(CNC(=O)Cc2csc(C)c2)CC1C C1(C2CCN(C(C3CCCO3)=O)C2)CCCCN1C(C1(N2CCOCC2)CC1)=O c1(CCNC(C=CC(C)NC(=O)C=CC(C)(C)C)=O)noc(=O)n1C c1(CC(=O)NC2C(NC(CC(=O)OC)=O)CCOC2)c(F)c(F)c(F)c(F)c1F c1(CCn2cc(C3N(C(=O)CC4CC4)CCCC3)nn2)ccc2c(c1)OCCCO2 C(=O)(CCCC(=O)NCC)N1CC(CNC(COCC(=C)C)=O)C(C)C1 c1(C(N2CC(C)C(CNC(=O)C(O)C(C)(C)C)C2)=O)cc(F)c(CO)c(F)c1 c1(C(=O)NCC(CNC(C2(OC)CCCOC2)=O)O)cc2ccccc2nc1O Cc1nc(NCc2ccc3nonc3c2)cc(=NC(C)c2ccc(F)cc2F)[nH]1 N#Cc1c[nH]c2ncnc(N3CC4CCN(C(c5ncc(Br)cc5Cl)=O)C4C3)c12 C(=O)(C(CC(C)C)C(N)=O)N1CCC(NC(C2C(OCC)C2)=O)(CC)CC1 C1(NC(=O)Cc2ccn(CC(F)F)n2)(CO)CCN(C(=O)CC2CSC2)C1 N1(C(c2ccc(CC)o2)=O)CC(NC(C2CCCN(C)C2)=O)CCC1C N1(C(c2c(CC)cccc2)=O)CC(C)(C)CC1CNC(C1CCCO1)=O C(=O)(CC(C)(C)C(=O)NCCC(C)NC(c1ccc(F)c(C(F)F)c1)=O)OC C12(NC(C3C(CN)CCCC3)=O)CCCC1NCC2 C=CCC(CNC(=O)C(C)NC(C1CC(C)=NO1)=O)CC(C)C c1(SCc2onc(-c3c(COC)n(C)nc3)n2)ccc(Cl)c(-n2nnnc2C)c1 Cc1ccc2nsnc2c1C(=O)NC1CCN(C(c2cnn(C)c2F)=O)CC1F c1(C(=O)NCC(C2(O)CCN(C(c3c(CC)scc3)=O)C2)C)cc([N+](=O)[O-])c[nH]1 c1(CC(=O)NCC(CN(C(CN2CC(C)(OC)C2)=O)C)O)ccnc(Br)c1 n1(C(CC)C)nnnc1C(c1cnc(Br)s1)NC(C1(C(C)C)CC1)=O C(C(C)C(=O)NCc1ccc(C(N2CC(CC(C)(C)C)C2)=O)s1)OCC c1(C(=O)NC2(CNC(c3cc(Cl)c[nH]3)=O)CC3CCC2C3)ccnc2ncnn12 n1(CCC)cc(C(c2nnnn2C2CC(F)(F)C2)NCC(C)(C)OC)nn1 C1(CNC(C2(CC#C)CC=CCC2)=O)(CO)CCN(C(c2cc[nH]c2)=O)CC1 Cn1cnc(C(=O)NCCN2CCCN(C(=O)CC3=CCCC3)CC2)cc1=O c1(CC(N2CC(NC(C3N(C)CCCC3)=O)CC2(C)C)=O)c[nH]c2cccnc12 Cc1occ(C(F)(F)F)c1C(=O)NC1CCC(NC(=O)C=Cc2cnc[nH]2)C1 CC1=CC(C(=O)NC)SC1.C(C)(C(CO)N)NC(=O)C=CSCc1ccco1 C(C1=CCCCC1)NC(C1CSCN1C(=O)Cc1cnsc1)=O c1(C(=O)NC2COC(C)(C)O2)cccnc1C(=O)NCCCCOCC N1(c2cc(C)c(C#N)cn2)CCCC2(CCCCC2NC(=O)C=CS(C)(=O)=O)C1 C(C(CCC)CCC)NC(CC1(C=C)CN(C(c2cc(OC)no2)=O)C1)=O C=CCCCC(C(=O)N(C)CCC1CCOCC1)NC(=O)C(c1cccn1C)=O CC(C)CCCC(C)CNC(=O)CC1C2CCC(C2)N1C(=O)C(C)C(C)(C)C c1(C(=O)NC2(C)CCN(C(c3ncsc3C3CC3)=O)C2)cc2ccccc2[nH]1 C(=O)(C(F)CCCC)NCC(CCCC)NC(=O)Cc1csc(S)n1 C(=O)(CCC(CC)CCC)NC(CC#CC)C(=O)N(CC(O)COC)C c1(COC(=O)CCCN2CCOC(NC(=O)NCC)C2)cncc2ccccc12 C#CCC(CC(F)F)C(=O)N1CCC(C)(C)C1C(N1CCN(C)C(C)C1)=O C(=O)(C(C)(C(C)C)OC)N(C1CCN(C(C=CCCC)=O)C1)CCC c1(OC(c2nnc(Br)n2C)C(=O)NC(C=C)(C)C)ccccc1CC C(=O)(C(CC(C)C)N(C)C(C1CCOCC1)=O)N1CCC(OCC)CC1 c1(CC)ccc(C(=O)NC2(CNC(=O)CCC=CCC=C)CCC2)cc1Br c1(C(=O)NCC(N(C)C(c2cnc(C(C)(F)F)s2)=O)C2CC2)cccn(O)c1=O C(=O)(CC1=CCOCC1)N1C(C(=O)NC(CCC)c2ccco2)CC1C C1(C(C)NC(COC(C)=O)=O)CN(C(c2ccc(-c3ncc[nH]3)nc2)=O)CCO1 CN=c1ccc(C(=O)NCCC2CCCN2C(=O)CNS(C)(=O)=O)c[nH]1 CN1CCC(C(=O)NCCC2(O)CCCCC2)(NC(=O)CCC2CC2(F)F)C1 C1(C(=O)Nc2ccc(OC)cc2)CC2CCC(C1)N2C(=O)C(O)CCSC C(=O)(CCCCCC#N)NC1CC(COC(C(=O)OC)CCSC)C1 C1(CNC(c2cc(C)c(Cl)s2)=O)CCC(C)CN1C(c1cn2ccnc2s1)=O c1(C(N(CCN(C(c2[nH]cc(C)c2)=O)C)C(C)C)=O)cc(Cl)c(O)c(Cl)c1 C1(C(N2CCC(C(C)NC(=O)CCC3CCCOC3)CC2)=O)C2C3CCC(C3)C12 C(CC(C)(C)CC(=O)NCCC(O)CNC(c1cnn(C2CCC2)c1C)=O)OC c1(CC)sc(=N)[nH]c1C(N1CCC(CCNC(=O)C(C(C)C)NC=O)C1)=O c1(NCC(=O)N(C2CCN(C(C3C(C)(C)C3(F)F)=O)CC2)CC)ccc(F)nc1 N1(C(c2scnc2Cl)=O)CCOC2(CCN(C(c3cnc4[nH]cncc3-4)=O)C2)C1 n1(CC)nccc1C=CC(N1CC(NC(c2cc(C)c[nH]2)=O)CC1C)=O C=Cc1cc(C(=O)NCC(C)CNC(c2cccc(F)c2C)=O)cc(F)c1 N1(C(c2c[nH]c(=NC)s2)=O)CCC(C)(NC(=O)Cn2nc(C(F)(F)F)cc2C)C1 CCCCC(C)(F)C(=O)N1CCN(C(C2CC2(Cl)Cl)=O)C(C)C1 C1(CCOC)(NC(=O)CCCn2cncn2)CCN(C(=O)CC2C(=O)NN=C2C)C1 C1(NC(c2cncc(CC)c2)=O)CC(O)CN(C(=O)C=Cc2cncs2)C1 CCC(C)(C)CC(=O)N1CC(CNC(C2CCC(C3CC3)C2)=O)C(F)(F)C1 c1(CC(=O)NCc2nc(CNC(CC)CC(=O)OCC)sc2)ccc(Cl)c(C)c1 c1(C(=O)NCCNC(COc2cc(C)c(Cl)cc2)=O)ccc2c(c1)C(=O)NCC2 c1(CN2CC(C)N(C(C3CCCS3)=O)CC2)ccc(O)c([N+](=O)[O-])c1 Cc1cc(C(N2CCN(C(=O)Cc3cc(C4CC4)no3)C(CO)C2)=O)ccc1F c1(CC)ncc(C(=O)N(CC(CC)NC(C2CC3CC3C2)=O)C)c(O)n1 NS(=O)(=O)CCCC(=O)NC1COCCN(C(C2CC2(F)Cl)=O)C1 c1(OC)cc(-c2nc(Cc3ccc(C)c(C)c3)no2)cc(Br)c1 c1(CC(=O)NCC(N(C(=O)C(F)=CCCF)C)C2CC2)c(F)cc([N+](=O)[O-])cc1F C#Cc1ccc(C(N2CCN(C(=O)C(CC3CCCC3)C(C)C)C(C)C2)=O)nc1 N1(C(c2nc(CCCCC)sc2)=O)CCC2OCCN(C(=O)C#CC3CC3)C2C1 CC1CCN(C(=O)CNc2ncccn2)C(CNC(c2cc(F)cc(Cl)c2)=O)C1 C=CCCCC(N)C(=O)N1CCCC(O)(C(F)(F)F)CC1 N1(C(C(c2cscn2)N(C)C)=O)CCN(C(C2CCCCC2)=O)C2(CCC2)C1 C1(C)(C(=O)NCC(N2CCCCCC2)C)CCCN(C(=O)CSc2ccsc2)C1 C1(CC(=O)NCCNC(C=Cc2nnc(C(C)C)o2)=O)CCCC(C#N)C1 C1(NC(C(C)Oc2ccccc2)=O)CCCN(C(c2ncccc2Cl)=O)C1 C#CCC(C)C(=O)NCCCOCCN(C(c1ccnn1C1CCOCC1)=O)C1CC1 c1(C(N2CC(C)N(C(c3csnn3)=O)CC(C)C2)=O)cc(=O)c2ccccc2[nH]1 C(CCC(C)NC(=O)Cc1nocc1C)NC(C(c1cccnc1)OC)=O c1(C(N2CCCC(C3N(C(COCC)=O)CCC3)C2)=O)cc2cc(Cl)ccc2[nH]1 c1(C(C(=O)N(CCCNC(C2COC(=O)N2)=O)CC)(F)F)ncccc1F N1(C(C2C(CC)OCC2)=O)CCC2CN(C(c3cnccn3)=O)CC12 C1(CNCC(N2CCCS2(=O)=O)C)CCCN(C(=O)OC(C)(C)C)CC1 CC(O)(CNC(=O)COCCF)NC(C1(CF)CC1)=O c1(OCC(C)C)cc(C(=O)N(CCNC(c2ccc[nH]2)C)CC)ccn1 c1(N2CC(C(=O)Nc3cc(C)ns3)C(C)(C)C2)ncnc2sc3ccccc3c12 c1(C(N2CCC(N(C(CN(S(CC)(=O)=O)C)=O)C)C2)=O)cnc(C(C)C)nc1 C(=O)(C(O)CNC(C1CC(C)(F)C1)=O)NC(c1cncs1)C c1(C(=O)OCc2ccc(OCC=C)cc2)ccc2c(c1)nc(Cl)n2C C1(C(N(c2cncnc2)C)=O)CCC(n2cc(-c3cncn3C)nn2)C1 CCC(CCOC)C(=O)N1CC2CC2C1C(N1CCC(CF)CC1)=O c1(C(C(=O)NCCOC)N(CCCO)C(C)C)nccc(Cl)c1Cl C12(C(=O)NCC3N(C(c4cnn(C)c4Cl)=O)CC3)CC1COC2(C)C C(=O)(C(C)CC(C)(F)F)NC1CCN(C(C2C(C(C)C)CCO2)=O)C12CC2 c1(N(CC(CCC)C)C)nc2ccc(=NCC3(C)CCCCC3(F)F)[nH]c2s1 Cc1ccnc(C)c1C(=O)NCC(C)CNC(=O)CCn1ncn(C)c1=O C(=O)(C#CC1CCCOC1)NC(C(C)NC(=O)C(C)(F)F)CCc1ccccc1 c1(CNC(C2C3CCCC2CC3)=O)ccc2c(c1)CN(C(c1ccnnc1)=O)C2 c1(N(C)C)nc(C(N2CC3(NC(=O)CCC4CC4(F)F)CCC2C3)=O)cc(O)n1 C1(NC(Cc2c(C)n[nH]c2C)=O)CC(C)CN(C(c2ccc(CO)nc2)=O)C1 CC(CCCCNC(=O)COC(F)F)NC(=O)CCC(=O)C1CC1 CC1CC(CNC(C2OCCC2(C)C)=O)CN(C(C2CCCC(CF)C2)=O)C1 C(O)(CN=c1ccc2c([nH]1)CCC2)C1CCN(C(c2ccc(F)cc2)=O)CC1 CCC(C)(C)CCC(=O)NC1(CC)CCN(C(=O)C(C)(C)CN(C)C)CC1 C1(CNC(CSc2c(C)n[nH]c2C)=O)CC(F)(F)CN1C(c1ccccc1Cl)=O N1(C(c2c(C)snn2)=O)CCC(C)(C)C(C(=O)NCC(Cl)C(C)(F)F)C1 C1(C(=O)NC(CN(C(C(F)=CC)=O)C)Cc2ccccc2)CCCN1CC(C)C Cc1cnn(C)c1C(=O)NC(C)(CNC(=O)CC1CC1(Cl)Cl)C(C)C N1(C(CCC2CC(NC(C(C)CC3CC3)=O)C2)=O)CCCC(N2CCC2)C1 C(C(C)(C(=O)NCC1(F)CC(CNC(c2cc(N)ccn2)=O)C1)OC)OC Cc1nn(C)c(C=CC(N2CC(NC(=O)CC(C)C)C(O)C2)=O)c1NC(C)C c1(CC)noc(C(=O)N(CC(O)CN(C(=O)CCCOC(C)=O)C)C)n1 C1(CC)CN(C(C2COC3(CCC3)C2)=O)CCN1C(=O)CSC(C)(C)C C=CCC(C)(C)CC(=O)NCCCC(CCC)NC(=O)CC(C)CN(C)C CC(CC(C)(C)C)C(=O)NCCC1CCN(C(=O)C(F)(F)CN(C)C)C1 c1(C(N2CC(CNC(CCCOCC=C)=O)C(O)C2)=O)coc2ccc(F)cc12 C1(NC(C2CC3CCC2CC3)=O)CC2CC1CN(C(c1c[nH]nc1C(F)F)=O)C2 c1(SC)nc(N2CC3CC2(CNC(=O)Cc2cnc(C)nc2O)C3)c(C)c(Cl)n1 N1(C(C(C)OCCC=C)=O)CCC(N(CCC)C(c2cc(CCCO)on2)=O)C1 CC1CN(C(=O)CC(F)F)CC1CCNC(=O)C(C)NC(=O)OC(C)(C)C c1(CC(=O)NCC2(C)CN(C3CC3)C2=O)cc2ccc(F)cc2s1 C(=O)(C#CC(C)(C)CNC(=O)C1=CCCC1)N1C(CC)C(O)CC1 c1(C(CNC(C(C)OC(c2cc(C(F)(F)F)n[nH]2)=O)=O)F)ccccc1 Cc1ccc(NC(=O)C(N2CCC(CCNC(C3(CF)CCC3)=O)C2)=O)cc1C C1(NC(C(n2cc(Cl)cn2)C)=O)C2CC1N(C(=O)CCc1cnc[nH]1)C2 C(CC(=O)NC1(c2ncc[nH]2)CC1)(C(F)(F)F)NC(c1nc(COC)oc1)=O c1(C(N2C(CNC(c3nnn(C)c3C(F)F)=O)C=CC2)=O)cc2cnn(C)c2s1 C(=O)(C(CCc1ccccc1OC)N1CCCC1C(=O)NCC1CC1)OC c1(CC=C)cccc(CN2CC(C(C)NC(c3cnc(C)s3)=O)C2)c1.C(C)C N1(C(C(c2ccccn2)C)=O)CCOCC(CNC(c2cncc(F)c2Cl)=O)C1 Cc1cc(C(=O)NC2CCC(C(=O)NCC3CC(=C4CC4)C3)CC2)ncn1 C(C)(CNC(C1(C)CCC(=O)N1)=O)(CC(C)C)NC(c1c(C)cnnc1)=O C1(C)(C(=O)NCc2ccc(CC)cc2)CN(C(C2C3CC(=O)CC23)=O)C(C)(C)C1 Cc1cc(NCC2CN(C(c3cnc(O)c(C)c3)=O)CCN2C)nc(C)n1 Cc1nn(CC(=O)NCC2CC(F)(CNC(C34CCCCC3C4)=O)C2)c(=O)n1C C(C(N=[N+]=[N-])C(=O)NC(C(N1CCC(F)(C#N)C1)=O)C1CC1)OCC N1(C(C=CCC)=O)CCC2(CCCCN(C(=O)Cc3csc(C)n3)C2)C1 C(=O)(N=c1[nH]ncn1C)C1C(O)CCN(Cc2cc(OCC)c(OC)cc2)C1 c1(-c2cnc(NCCN(CC(C)C)C)nc2)ccccc1C#N c1(NC(=O)Nc2cccc(F)c2Cl)cccc2c1CCO2.C1CCCCC(=O)N1 C12(CNC(C3(C(c4ccc(Cl)cc4)O)CCNCC3)=O)CNCC1COC2 N1(C(CC=CC(C)(C)C)=O)CCC2(CCC2NC(C2CCNC(=O)C2)=O)CC1 c1(OCC)cc(Br)ccc1C(N1CC(F)CC1C(N1CC(O)C(O)C1O)=O)=O Cc1cc(C(N2CCCC2CCCNC(=O)C(C(C)C)NC(N)=O)=O)c(C)s1 c1cccc(S(=O)(=O)N(CP(C)(C)=O)C(C)=O)c1.N1CCOCC1 C12(CNC(C(C3CCCCC3)N(C)C)=O)CC1CN(C(C1CCCOC1)=O)C2 CCCCCC(O)CC(=O)N(CCNC(=O)CC(CC)C(F)F)C(C)C c1(C(=O)NC(CN(C(c2nc(O)c(C)s2)=O)CC)C)ccc(F)c(F)c1C CC(C)C(CN(C)C)C(=O)NC1CCN(C(=O)C(C)(C)N=[N+]=[N-])CC1O C1(C(=O)NCCC2(C(N(CC(O)CO)CC)=O)CC2)CCCCS1 Cc1cc(F)cc(Cl)c1NC(C1CC12CN(C(c1ncccc1F)=O)C2)=O C12(NC(C3C(COC)(CC)C3)=O)CC1CN(C(=O)CCNc1cnccn1)C2 C1(OC)CN(C(c2cnccc2C)=O)CC1C(=O)N(C)Cc1csnc1C N1(C(C(=O)N(C)CC2CCCSC2)=O)CCOc2ccc(Cl)cc2C1 Cc1nnc2c(C(=O)NCC3(F)CC(CNC(=O)Cc4cnoc4)C3)cccn12 Cc1ccc(CN(C=O)Cc2ccc(O)c(Cl)c2)cc1C(F)(F)F N1(CCC(=O)N(CCC)CCNC(=O)C(C)n2ccnc2)CCP(C)(=O)CC1 C#Cc1ccc(C(=O)NC2(C)CC(NC(=O)CCC34CCC(CC3)C4)C2)o1 N1(C(CCSCCC)=O)CC2(C1)OC1(CO)CC2(NC(c2cc(C)c(C)o2)=O)C1 S(=O)(=O)(c1ccc(C(=O)NC2CC(CNC(c3ccc[nH]3)=O)C2)cn1)NC c1(C(C)C)cc(CCNC(=O)NC2CC2c2cnn(C)n2)on1 N1(C(c2c[nH]c(=N)s2)=O)C2CCC1CC(O)(CNC(=O)CCCS(N)(=O)=O)C2 C(=O)(C(C)(C)CS(C)(=O)=O)NCCCC(C)(C)NC(=O)C=Cc1cnc[nH]1 c1(C(=O)NCC2(OC)CN(C(C3CN4CCN3CC4C)=O)C2)c(F)cc(F)cc1Cl c1(C(C(=O)N(C(C)CNC(=O)C(F)(F)CSC)CC)O)ccc(C(F)(F)F)cc1 Cc1c(Br)cc(Cl)c(C(N2CC3CC2CN3Cc2c(O)cccc2Cl)=O)c1Cl C1(CNC(C(C)SC)=O)CCC(CNC(C2CC(C)C2)=O)CC1 C1(C(=O)NC2COCCC2NC(C23CCC(CC2)C3)=O)CC2CCCC(C1)C2 C1(C(C)NC(c2c(COC)scc2)=O)CCCCN1C(C1C(C(F)F)C1(C)C)=O N1(C(c2c(CC)nc[nH]2)=O)CCCN(C(=O)CCOCCOC)CCC1 c1(NC)cnccc1C(=O)NCC(C)CNC(C1OCCOC1C)=O N1(C(CCCC(C)=O)=O)CCCC2CN(C(C3CCc4nnnn4CC3)=O)CC12 Cc1cc(C(N2CC(O)CC2(C)C(=O)NC2CCC3(C(C)C)CC23)=O)nc(O)n1 N1(CCNC(=O)Nc2c(-c3cn(C)nc3)ccc(Cl)c2)C(=O)NC2(CC2)C1=O c1(CNC(c2nnnn2CCSC)C2CN(C(=O)NC)C2)csc(C(F)(F)F)c1 N1(Cc2ccc(C(=O)OC)cc2C)CCC(N=c2nc(Cl)c3c([nH]2)COC3)C1 CCS(=O)(=O)CC(=O)N1CCCC1(C(=O)NC1CC2(CC2)C1)C(C)C N1(C(CN(C(C(CCC)F)=O)CC(C)C)=O)CCC(C)C1(C)C C1(C(N(C)CCN(C)C2CC2)=O)CC(=O)CN1C(c1ncc[nH]1)=O N1(C(C(C)(Cl)CCl)=O)CC2(CC(C(=O)NCC3CC3(F)Cl)CO2)C1 N(C(=NCCF)NC1CCN(C2CC2)CC1)Cc1cccc(C(C)O)c1 Cc1cc(C(=O)NC2CC(CO)N(C(=O)Cn3nc(C)c(C)c3C)C2)nc(O)c1 C1(C(N(CCC#N)CC)=O)CCN(S(=O)(=O)C(C)C)CCC1C N1(C(c2c(OC)nn(C)c2)=O)CC2CCCC2(NC(c2nc(=O)n(C)[nH]2)=O)C1 Cc1cc(C(N2CCCN(C(=O)C(C)NC(N)=O)CC2CO)=O)c(O)nc1C CC1(C)CN(C(c2cnn(C(C)(C)C)c2)=O)CCN1C(c1c(F)cccc1F)=O N1(C(C(C)OCCOC)=O)CCC(NC(C23CCC(CO)(CC2)C3)=O)C(CO)C1 c1(N(C(=O)Cc2cnoc2)CC2(NC(C3(C)CCC3)=O)CC2)ccc2c(c1)OCO2 c1(OC)cc(C(C)NC2CCCC(C)C2)c(F)cc1OC(C)C C1(CCC)CCCCN1C(=O)CN(C(c1cc(C)cs1)=O)CC1CC1 CC1CCCN(Cc2nc(-c3cc(-c4ccco4)cc(Cl)c3)on2)CC1 N1(C(=O)NCC2(c3ccccc3Br)CCCCC2)CCC2C(CCCN2C2CC2)C1 C1(CC(=O)NCC2(O)CN(C(c3cc(CCC)on3)=O)C2)(CC=C)CCCCC1 c1(CC)cccc(C(=O)NC2CCC(N(C(=O)C(C)(C(C)C)OC)C)CC2)c1N C(=O)(C1=Cc2ccccc2OC1)N1CC(N(C(=O)C#CC2CC2)C)C(C)(C)C1 C1(NC(C2(C#C)CCC2)=O)CCN(C(c2cccnc2S)=O)CC1CC c1(C(=O)NC(CNC(C=Cc2nnn(C)n2)=O)(C)C2CC2)cc(C(F)F)cc(Cl)n1 c1(OCCC(N2CC3C(NC(CSC(C)C)=O)(C3)C2)=O)cc(F)cc(Cl)c1 N1(C(C(C)=CC=C)=O)CCOC(C(=O)NCC(C)(C)C(C)O)C1 N1(C(c2c(COC)cco2)=O)CC2(C1)CN(C(=O)C(C)(C(C)C)NC(C)=O)CC2CO C1(C2CC2)(CNC(C2CCCC2O)=O)CCN(C(c2cn(CCCF)nn2)=O)C1 c1(C(N(CCCNC(C(C)(C)O)=O)CCO)=O)nccn2c(Br)cnc12 N1(C(CSCCC(C)C)=O)CC(F)(F)CC1CCNC(c1nocc1C(C)C)=O c1(C(=O)NCCN(C(CC(C=C)c2ccccc2)=O)CC)c[nH]c(=N)nc1C C(=O)(C1=C(C)CCC1)N1C(C2(NC(C3(C#C)CC3)=O)CC2)CCCC1 CCC(O)C(C)C(=O)NC1CC(F)(CNC(c2cnn3ccsc23)=O)C1 c1(C(N2CCC=C(CNC(C(COC)OC)=O)C2)=O)ccc(OC)c2cnccc12 c1(C(=O)NC(CNC(c2ccc(COC)s2)=O)C)cn2c(n1)CCC2 C1(NC(CCCC)=O)CCN(C(C2CCOC2C)=O)CC1 N(C1CN(C(=O)C=Cc2cccs2)CCc2ccccc21)C(C1C(C)C1C)=O N=c1[nH][nH]c2cc(OCCNC(N3CCC34CCCOCC4)=O)ccc12 Cn1nccc1C(C(=O)NCC1(CCO)CC1)Nc1ccccc1 c1(C(=O)NC(c2cccc(N)c2)C(C)C)cc(F)ccc1Cl C1(NC(c2c(C)cco2)=O)C2CN(C(=O)CC3CCCC3C)CC12 C(=O)(C(O)CC(N)=O)NCC1CC(NC(CCN(C)C(=O)OC(C)(C)C)=O)C1 N1(C(c2ccc(C(OC)OC)o2)=O)CCC(NC(=O)C(O)CC(N)=O)C(C)C1 Cc1nc(C)c(C(=O)NCCC2(C(=O)NC3CCCC3C)CC2)s1 CC(C)CC(F)(F)C(=O)NCCN(CC(C)O)C(C1CCSC1)=O C1(C(N(C(C)C)CCNC(=O)CCC(N)=O)=O)CCC2CC1CO2 C1(C(=O)NC(CC)Cn2cncn2)(CNC(=O)CCOCCOC)CCCCC1 N1(C(C2(COCC)CC2)=O)CCC(C2CCCO2)CC1.N12CCC1C(=O)N2 c1(NCC(CC)CCO)ncnc(NCC(C(C)CC)OC)c1C C1(C=O)OC(N(C2CC(C#N)C2)CC#C)=CC(Br)=C1OC(F)(F)F c1(-c2cnc(SC)nc2)cncc2sc(C(=O)Nc3ncc(F)cc3Cl)cc12 N1(C(C(=O)NCCN(C)C)=O)CC2CCCC(C1)N2Cc1csnn1 c1(C(C(=O)NCC(CO)NC(C2N(CCC)CCC2)=O)(C)C)ccc(C#N)cc1 N1(C(CCN(CC#C)C(C2CN(CCC)C2)=O)=O)CCC(N(C)CC)CC1 c1(CC(=O)NCC=CCNC(C2CNC(=O)N2)=O)nccc(OC(F)F)n1 Cc1cccc(O)c1C(=O)NCC(C)(F)CNC(C12CC(CO)(C1)C2)=O C(=O)(C#CC1CCOC1)NC1CN(C(C(C)CSc2ccccc2)=O)CC(F)C1 C(=O)(C(C)C(C)S(C)(=O)=O)NCCCCNC(C=Cc1ccc(OC)c(F)c1)=O C1(CC(=O)N(CC(C)C)CCCO)C(COC)CC1(F)F C12(CC(N3CC(CCC)OCC3)=O)CCC1CN(C(C1(CO)CCCC1)=O)C2 N1(C(C(C)(C)c2ccno2)=O)CCCN(C(=O)C(c2cccnc2)O)CC1 C(=O)(C(O)CC(F)F)NC(CCCC)CNC(=O)C=Cc1cc(C)no1 Cc1cccc(C(=O)NCC(C)(C)CNC(c2cnc(O)c(Cl)c2)=O)c1Cl N1(C(C=Cc2n(C)ncc2)=O)CCC(C=CCOCC(N2CCCC(C)(C)C2)=O)CC1 C1(C(=O)NC2(C)CCN(C(CC(C)n3cccc3)=O)C2)CC2C=CC1CC2 N1(NC(c2cccc([N+](=O)[O-])c2)(CC)C)CCS(=O)(=O)C(C)(C)C1.C c1(CC(=O)NC2CC(NC(=O)CC34CCC(CC3)C4)C2)cc(O)nnc1O c1(OC)ccc(-c2cn(C3CN(C(=O)Cc4ccc(C)cc4Br)C3)nn2)cc1F C(=O)(CC(O)C(=O)N1CC1)NCCC(C)(C)NC(C1CCN1C1CCCC1)=O c1(C(N2CCN(C(CSCCC#N)=O)C3C2C3)=O)ccc2nc(O)oc2c1 c1(C(=O)NCC(C)(CO)NC(C2CCC(N(C)C)C2)=O)cc(Cl)c(Br)[nH]1 CC(CC(=O)N(CCCNC(=O)C(C)CC1CC1)C1CC1)n1cc(Br)cn1 C1(NC(CCCN(C)C2CC2)=O)(CF)CCN(C(=O)C(CO)NC(N)=O)C1 C(=O)(C(CNC(c1cnsn1)C1CC1)CC1CCCC1)NCC#CCC C1(C)(NC(CC2CN(C)C2)=O)CN(C(=O)CSC(=N)N)C1 CC(C)CC(O)C(=O)N1CCOC(C)(CNC(C2CN(C)CCO2)=O)C1 C(=O)(CS(=O)(=O)c1ccccc1)NC1C(C#N)CN(C(=O)CCc2cccs2)C1 c1(C(N(C2CCN(Cc3occc3Br)C2)CCC)=O)cncn1C c1(C(=O)NCCOCCCNc2nccn2C2CC2)cnc(Cl)cn1 Cc1ccc(C(=O)NCC(C)(C)CCNC(=O)CC2CCC(C)C2)c(C)c1 c1(C(=O)NCC2CCC(NC(C3C(OCC)C3)=O)C2)cccc2oncc12 N1(c2ccc(CN3C(Cc4c(C)con4)CCC3)cc2)C(=O)c2ccccc2C1=O c1(CSCC(O)Cc2ccccc2)ccc(OC(F)F)c(F)c1 C1(CC(=O)N(CC(C)CNC(=O)CC2(C)CC2)C)CC2CCC(C1)N2C CC1(CNC(=O)Cn2ccccc2=O)CCCN(C(C2(Cl)CCCCC2)=O)C1 CCC(CC1CCCC1)C(=O)N1CC=CC1CNC(C1CS(=O)(=O)C1)=O C1(CC(=O)NCCC(C)NC(c2ccccn2)=O)CC2(CCOCC2)CO1 c1(CC)cc(C(N2CC(CN=c3[nH]nco3)C(C(F)F)C2)=O)ccc1C C1(C(=O)NC(CC)CNC(=O)CCn2ccc(O)nc2=O)CCCC2(CCC2)O1 N1(C(C2N(C(c3nn(C)c(O)c3)=O)C3C(O)CC2C3)=O)CC(=O)N2CCCC2C1 c1(C(C2CCOC2)CNC(c2csc(N(C)C)n2)C)ccccc1 Cc1cccc(C(=O)NCC2CCC(C(=O)NCCC3CCC(C)(C)C3)O2)c1O c1(C(=O)NC2(CCOC)CCN(C(c3nc(Cl)c(Cl)s3)=O)C2)cc(C)nc(C)c1 C1(C(=O)Nc2cccnc2)CCCCN1CCNC(=O)CC1(CO)CCC1 C1(CN(C(c2c(SC)cnn2C)=O)CC)CCN(C(C2CC2C)=O)CC1 N1(C(C(C(COC)C)C)=O)CC2CCCC(C1)N2C(C1(Cl)CCCCC1)=O c1(C(C)C)n[nH]cc1C(=O)NCC1CCCC1NC(=O)CC(=O)Nc1nccs1 c1(C(=O)NC2CN(C(CCSCCC)=O)CC3C2C3)[nH]c2ccc(C)cc2c1Cl c1(CC)nc(-c2cccc(-c3ccc(C)nn3)c2)n(CCc2ccncc2)n1 CCC(CC)(C(N)=O)NC(=O)C(c1ccoc1)NC(c1csnc1C)=O c1(OC)cc(OC)c(NC2CC(N)CN2C(c2cc3ccccn3n2)=O)cc1F C1(C(=O)NCCC(=C)CNC(=O)C=C2CCOCC2)CCCC(F)C1 C1(NC(C(CC)(F)F)=O)CCCC(NC(c2ccc(Cl)cc2NC(C)=O)=O)CC1 Cc1cnc(CNC23CC2CN(C(=O)CNC(=O)Cc2ccc(O)cc2)C3)nc1 C1(COC)CN(C(=O)Cc2cccc(Cl)c2)CCN1C(=O)Cc1cnns1 CCCCC(CC)CC(=O)N1CC(NC(=O)Cc2n[nH]c(=NC)s2)CC1(C)C N1(C(c2c(C)nns2)=O)C(CNC(=O)C=Cc2ncco2)CC2CCCCC12 Cc1c(C(N2CCCC2CC(F)(F)F)=O)cn2[nH]cnc(=O)c12 c1(CC)ncccc1NC(C1CC(F)CN1C(=O)CCc1ccc(C)nc1)=O C(CC(C)(C)NC(C1CNC(=O)C1)=O)=CC(=O)N(CCN(C)C)CC C12(OCC)CCCC1(NC(=O)NCC1(C)COC(C)CO1)CCO2 C(=O)(C(C(F)(F)F)C(F)(F)F)N1CC1.c1(CC(=O)NCCO)c[nH]nc1O N1(C(C2(SC)CC2)=O)CC2(CCN(C(=O)Cc3cccc4nsnc34)C2)C1 Cc1nn(C)c(F)c1C(=O)NCc1ccc(C(C)NC(=O)C(C)C(C)(C)C)cc1 C1(C(=O)NC2C(NC(C(COC)(C)C)=O)CCOC2)CCn2c(C)cnc2C1 Cc1cc(C(N2CCCC(CC(=O)Nc3cc(C)ccc3O)C2)=O)nc(Cl)c1 c1(SCC)ccc(CC(=O)NCCC(O)CNC(C2(O)CC(F)(F)C2)=O)cc1 N1(C(C(C(C(C)C)O)(C)C)=O)CCC2(CC1)CN(C(C1(C)CC(C)C1)=O)CCO2 c1(OC)ccc2nc(N(C3C4Cc5ccccc5C34)C(=O)C(C)C)sc2c1 C(=O)(CCCCC(=O)NC12CC(NC(=O)CCCSC(C)(C)C)(C1)C2)NC c1(C(N(C2C(C)CN(C(c3ncc[nH]3)=O)CC2)C)=O)ccc2nc(O)n(C)c2c1 C#Cc1ccc(C(=O)N(CCNC(C2CCC2)=O)CCOC)c(F)c1 CCCCCC=CCC(=O)NCc1ocnc1C(=O)N(C)OCC(F)(F)F CC1(C)CCCC(C(=O)NC2C3CC(NC(=O)CSc4cn[nH]c4)CC23)C1 c1(OC)ccc(C(N2CCC(C)(NC(=O)CC3CCC(=O)NC3)C2)=O)c(F)c1F Cc1ncc(C(N2CC3CC(NC(C4CN(C(C)C)C4)=O)C2C3)=O)cc1N n1(CC)nnnc1C(c1nc(C)no1)NCCCC(=O)NC1CCOC1 Cc1cc(CN(CC(C)NC(C2CC3(CCC3)C2)=O)C)cc(F)c1 C1(CC(=O)NC2CCCN(C(C3(NC(C)C)CC3)=O)C2)CCCC(C)(C)C1 C(CC(C)(C)CC(=O)NC(COC)(C)C(C)C)NC(=O)CCCC1CC1 N1(C(CC2(C=C)CN(C(=O)C#CC3(C)COC3)C2)=O)CCC(F)(F)C(F)C1 C1(C(=O)NC(CN(C(CSC(C)C)=O)C)(CO)CO)CSc2ccccc2O1 C(CCCCC(=O)NC1CC(C)N(C(c2cc(N(C)C)ccn2)=O)C1)OC C1(C(=O)NC(CNC(C2CC2c2ccccc2)=O)C2CC2)CCCN1C(=O)C1CC1 Cn1nnc2c1C(C(=O)NCC1CCCN(C(=O)C(F)(F)C3CC3)CC1)CCC2 C=CCCC(C(=O)NCC(CC)OC)NC(C1CCN1C)=O N1(C(C(C)OC2CCCCCC2)=O)CCC(NC(c2cnccn2)=O)C(O)C1 N1(C(CN2C(C)CCC2)=O)CCOC(C(N2CC(C(C)(C)C)C2)=O)CC1 C(=O)(C(C)(C)CO)NC(C)C(CO)NC(=O)Cc1cccc(C(F)(F)F)n1 N(C1COCc2ccccc21)C(N(C)C(c1ccccc1)C1CC1)=O N1(C(c2c(CC)con2)=O)CCC2(CCOCC2)C(NC(=O)Cc2cnc[nH]2)C1 CC1(C)CN(C(C2CN(C3COC3)C2)=O)CCC1NC(C1(n2nccn2)CC1)=O c1(OC)cc(F)c2c(C(N3CCC3CNC(c3ccc([N+](=O)[O-])o3)=O)=O)cnn2c1 C(=O)(CCCC(F)(F)F)N1CC(C)(CNC(c2cc(C)c(F)nc2)=O)C1 CN1N=C(CC(=O)N2CC3CCCC(NC(c4cccc(=O)o4)=O)(C3)C2)CC1=O N1(C(c2c(NCC)scn2)=O)CCC(C(F)(F)F)C(NC(=O)CS(N)(=O)=O)C1 c1(OC)cccc(C(N2CCCCC2CN(C)C(c2ncc(Cl)s2)=O)=O)n1 c1(CC)cc(C(=O)NCC2(NC(=O)CC3CC4(CC4)C3)CCOC2)cs1 c1(C(=O)NC2CC(C)CN(C(c3cnn(C4CC4)c3)=O)C2)ccc2n[nH]cc2n1 C1(C#N)(C(N2C(CC)C(NC(c3ccn(C)c3)=O)CC2)=O)CCOCC1 C(=O)(C(O)C(CCC)NC(=O)CCCC)N1CC(C#C)OCC1.C1(=O)CCCN1 C12(CO)CN(C1)C(=O)N2.C1(COC)(COC)CC(C(=O)OC)C1 c1(C(=O)NCCC(Cn2cc(CN(C)C)nn2)F)coc2c1CCCC2 C1(NC(C(C)SCCCC)=O)CC(C)(CNC(=O)C=CC(C2CCCC2)=O)C1 N1(C(C2CC(SC)C2)=O)CCCC(CC(N2CCCC3(C2)N=N3)=O)CC1 c1(C(N(CCN(C(c2[nH]c(C3CC3)nc2C)=O)CC)CC)=O)cccn2nnnc12 c1(C(=O)NC(CNC(c2c(C)[nH]nc2Cl)=O)C2CCC2)cnc(O)c([N+](=O)[O-])c1 C1(C(=O)NCCN(C(=O)CC2(O)CCCCC2)C)CCN(S(N)(=O)=O)CC1 c1(C(N(CC=C)C2CC2)=O)ccn(CCNC(=O)C(CO)N(C)C)c1 C1(C(c2ccc(-c3ccncc3)s2)=O)CCCC1N(C(C1CC=CCC1)=O)CCO CCN=c1[nH]c(C(=O)N(C2CCN(C(c3csc(Cl)n3)=O)CC2C)C)cs1 N1(C(Cc2c(C)scc2)=O)CCC(C)(CCNC(C2(C)CC(F)(F)C2)=O)C1 C1(NC(c2c(C(N)=O)csc2)=O)CCN(C(c2coc(C3CCC3)n2)=O)CC1F C1(CC(=O)N(C)CCO)Cc2ccccc2CN1C(c1ccc2ccn(C)c2c1)=O C#Cc1cccc(C(=O)NC(CO)C(C)NC(C2(CC(F)F)CCC2)=O)c1F C(=O)(CCCC(=O)NCC(C)CNC(c1oc(CC)nc1C)=O)NCC c1(C(=O)NC2(C)CC(NC(C3CCCN3S(C)(=O)=O)=O)C2)cnn2c1CCCC2 N1(C(Cn2c(C)ccn2)=O)CCC(NC(C2CCN(C)S2(=O)=O)=O)CC(O)C1 C1(CNC(c2ccnc(S)c2)=O)CCN(C(=O)C(O)C2CCCC2)CC1O Cc1ccccc1C(=O)NCc1cccc(Cc2nnnn2C2CCC2)n1 N1(C(C2C(CC)C2)=O)CC(NC(c2cncc(C)n2)=O)CC2(CCC2)C1 c1(CNC(C(C2(O)CN(C(c3c(C)cn(C)c3)=O)C2)F)=O)cccc(F)c1C C(=O)(C1=CCCCCC1)NCCC1CC(CC(C(=O)C(CC2CCC2)N)=O)C1 Cn1cc(C(=O)NCC(=O)NC23CCCCC2C3)ccc1=O C1(NC(C=CCC(C)(C)NC(Cc2n(C)nnc2)=O)=O)CCCC2(CC1)CC2 C1(C(=O)NC(CC(=O)N(C2CCN(CC)CC2)C)C2CC2)CC(=O)OC1(C)C C(c1c(C)noc1C)=CC(=O)NC1CC(C(C)NC(C2(COC)C=CCC2)=O)C1 CC1(C)C(N)CCN1C(=O)CCC(=O)N(C)C.C(c1cc[nH]n1)=CC(=O)C(CN)=O C1(NC(C2(O)CCC2)=O)CCN(C(=O)C2=CCCCC2)CC1F N1(C(C(CC2CN(C(C3(C)CC=CC3)=O)C2)F)=O)CCCC(F)CC1 C(CC(C(=O)N(C(C)CC(=O)OC)C)NC(=O)C(C)N(C)C)SC c1(N(C)C)ccc(CNC(C2C3CC3CN2C(C2CC2(Cl)Cl)=O)=O)cn1 N1(C(Cc2cc(C)no2)=O)CC2CC1CN2C(c1sccc1-n1ccnn1)=O C1(C2N(C(C3COC4(CCC4)CO3)=O)CCC2)CNc2ccccc2O1 Cc1cccc(C)c1OCC(=O)NCC1(O)CC(NC(=O)C(C)C2CCC2)C1 c1(CN2CC3(OCC(NC(c4c[nH]c(Br)c4)=O)C3)C2)cccc2ccccc12 C(=O)(C(F)(F)C(C)(C)O)NC(C)CCCC(=O)NCc1cnn(C(C)C)c1 N1CC2CC1CN2c1cc(NCC)nc(C(C)C)n1.c1(CCC)ncccc1C c1(NCC(C)C(O)C2CCCC2)c[nH]nc1-c1ccccc1 CC1(F)CCN(C(C2CCN2C(=O)Cc2ccon2)=O)C1 c1(CC(=O)NCCN(C(=O)CC2(N3CCCC3)CC2)CCC)cc(C)ccc1F CC(C)C(O)CC(=O)N1CCCCC1CN(C(=O)CCOCc1ccncc1)C C=CC(C)(O)CC(=O)N1CCC(OCCNC(=O)C(C)(C)C2CCCO2)CC1 CC1CC(NC(c2nc(Cl)ccc2Cl)=O)CCN1c1nccnc1F C1(C(N2CC(OC)C(NC(c3cc(C)nn3C)=O)C2)=O)Cc2cc(Cl)ccc2O1 N1(C(CSC)=O)CCC2(NC(=O)C(c3ccc(F)c(F)c3)(C)C)CCCCC12 CCCS(=O)(=O)C(C)C(=O)NCC1CCN(C(C2CCC(O)CN2C)=O)CC1 C1(n2ncc(N(C)C)n2)CCN(C(=O)C(N2CCCC(F)C2)=O)CC1 c1(C(=O)NCCC2CCCN(CCn3cccn3)C2)ccc(F)c(Cl)c1 O=C(CC(F)(F)C(F)(F)F)N1CC(O)(CCNC(C2(C3CC3)CCC2)=O)C1 c1(CC)ccc(C(=O)NCC(O)CN(C(=O)Cn2nc(C)oc2=O)C)nc1 N1(C(CN(CCC)C)=O)C2CCC(C(=O)NC3(CN(C)C)CCC3)C1CC2 CC(CCN=c1cc(Cl)nc[nH]1)NC(c1ccn2c(O)nnc2c1)=O C1(C)(NC(c2noc(CC)c2C)=O)CCCN(C(=O)CCCC#N)C1 Cc1nc(CO)nc2ccccc12.n1(C)cc(CC(C(=O)OC)NC(=O)C(C)O)nn1 C(=O)(CCCS(C)(=O)=O)NC(C1CCN(C(C2(C(F)F)CCC2)=O)C1)C Cc1cccc2c1CCOC2C(=O)NC1(CF)CCN(C(=O)CSC)C1 c1(NCCC2N(C)CCC2)nccc(=NCc2ccnc(C#N)c2)[nH]1 C1(CC(=O)NC(c2nc(C)[nH]n2)(C)C)C2CCCC2N1C(c1ccc(C)nc1)=O N1(C(C(CCC)NC(N)=O)=O)CCC(C(=O)N(CCCCCO)C)C12CC2 N1(C(COC(C)=O)=O)CCC=CC1C(N1CC2CC1CS2)=O c1(N2CCCC(CSC)C2)nc(=N)[nH]c(=NCCc2c[nH]nc2O)[nH]1 C1(c2nc(COCC)[nH]n2)CCCN(C(=O)NC2(O)CCNCC2)C1 C1(CNC(c2c(C)c[nH]n2)=O)CN(C(C2CCCCO2)=O)C(C)(C)C1 c1(OC)ccc(C2(C(=O)NCCCCCCN(C(=O)C(C)OC)C)CCC2)cc1 Cc1ccc(F)c(C(N2C3CCC(C3)C2CNC(=O)C(C)OCC2CC2)=O)c1F C1(CN(C(C2(NC(C(CO)NC(=O)OC)=O)CCC2)=O)C)CCC(C)CC1 c1(OC)cc(NC(C2CCC(C)N2Cc2ccc(F)nc2C)=O)c(Br)cc1Br c1(C(N(C2CCN(C(=O)CCC3CCC(=O)NC3)C2)C)=O)ccc(C#N)n1C C1(CC(=O)NC(CNC(C2(C(=O)OC)CC2)=O)C2CC2)CSCCS1 c1(C(=O)NCc2ccccc2CNC2CC2C(=O)NC2NC(=O)O2)ccc2n[nH]cc2c1 c1(CC)ccc(N)c(C(=O)N(CC(C)(C)CNC(c2cc(F)ccc2F)=O)C)c1 C1(C(N(CC(=O)NCC)CC)=O)C=CCCN1C(C1CC2(CC2)CO1)=O c1(CCC(=O)NC2CN(C(C3C(OC)CCCC3)=O)C2)c(C)nc(SC)nc1O C12(CNC(CCOC(C)C)=O)CCCC1CCN2C(c1ccnn1C(C)C)=O C1(F)(C(=O)NC2CC(C)(NC(CCSc3nc(C)[nH]n3)=O)C2)CCCN(C)C1 c1(OCC(=O)NCC(C)CNC(=O)CCC2CCOC2)ccc(C)c(C)c1 c1ccc2nc[nH]c2n1.c1(C(N2CCC2)=O)cc(F)ccc1OC(F)F C(C)(C(C)NC(C1(N(C(=O)CCn2cncn2)C)CC1)=O)(C1CC1)OC C1(C(N2CCCC(NC(Cc3ncc(C)s3)=O)C2)=O)Cc2c(F)cccc2O1 c1(C(=O)NC2C(CC)N(CC(N3CCOCC3)=O)CC2)cnn2ccccc12 c1(NC(C(c2cn(CC(=O)OC(C)(C)C)nc2)=O)=O)cc(F)c(Cl)cc1C C1(COCC(=O)NCCN(C(C)C)C(C2(CO)CCCC2)=O)CCCCO1 C12CCCN(C1)C(=O)CNC(=O)N(CC)CCn1nccc1C(=O)NC2.NC CC1CC(CC(=O)N(CC(N2C(C)CCC2C)=O)CCO)CC(C)(C)C1 N#Cc1c[nH]c(C(N2CC=CC2CNC(=O)C(c2ccccc2F)F)=O)c1 C1(NC(C=Cc2ncn(C)c2)=O)CC2CC1N(C(C1(C)CC1(F)F)=O)C2 c1(C(=O)NC2CN(C(=O)CCCCBr)CC(F)C2)n[nH]c2cccnc12 CCC(CC)C(=O)NC1CCC(NC(=O)CC(C)NC(C2CCCC2)=O)CC1 c1(OC)nscc1C(=O)NC1(C(=O)NCc2cc(CSC)no2)CCCC1 C(C(C)(C)C(=O)NCC1(F)CCN(C(C2CC(=O)N(C)C2)=O)C1)OCC C1(CC#C)(C(=O)NC(C2CCOCC2)CO)CCN(C(=O)C(COC)OC)C1 C(=O)(CC(C)C(=O)N1CC(F)CC1CNC(=O)C(C(C)C)C1CCC1)OCC c1(C(N(C(C)CNC(c2cccc(C(N)=O)c2F)=O)C)=O)cc2ccccc2o1 C1(CNC(C(Cc2c(C)nc[nH]2)O)=O)CC12CCN(C(=O)Cn1cnnc1)CC2 CC1(C)CC(C(N2CCCCC2CCO)=O)CC(C)(C)S1 c1(COCC)nc(N2CCC(C)(NC(=O)Cc3ccon3)C2)cc(C)n1 N1(C(Cc2c(C)cco2)=O)CC(C)CN(C(c2n[nH]c(=N)[nH]2)=O)C(C)C1 N1(C(CS(=O)(=O)NC)=O)CCC(CNC(c2ccc(S(C)=O)cc2)=O)C(F)(F)C1 c1(CCC(=O)NCCCN(C)C(=O)NC2(c3cc[nH]n3)CC2)cccc(Br)c1Cl C12(CC(=O)NC3(CNn4cccn4)CC(c4ccccc4)C3)CC(CN1)C2 C(C(COC)CC(=O)NC1COCC1C(N1CCC1C1CCCC1)=O)OC N1(C(c2cncs2)=O)CC2CCN(Cc3cc(Cl)ccc3O)CC2C1 C1(C(N2CC(NC(COC3CCC(=O)NC3=O)=O)C2)=O)CC2(CCC2)CCO1 N1(C(C(CC)n2cccn2)=O)CCC(C2(NC(c3ccc(CO)nc3)=O)CC2)C1 Cc1nc(NC(c2ncccc2F)C)cc(NC2CC(C(C)(C)C)C2)n1 c1(CNC(C(=O)NC(c2ccnn2C)CC)=O)cccc2c1OCCCO2 C(N=c1[nH]cnc2c1COC2)C1N(C(C2CCCC(C)C2)=O)CCC1 c1(C(N2CC3(CNC(C45CSCC4C5)=O)CC2CO3)=O)ccc(F)cc1F C1(C(=O)NCc2cc(Oc3cccc(C)c3)ncc2)CCN(C2CC2)CC1C N1(C(CC)=O)CCC(CNC(=O)C(C)OCC)(OC)C1 c1(CCC)ccccc1C(=O)NCC1CCCN(C(=O)C(c2cnn(C)c2)O)C1 CCCCCC(O)CC(=O)NCC1=NOC2CN(C(C3CC4CC4C3)=O)CC12 C1(C(N2C(CN(C(c3ccon3)=O)CC)CCC2)=O)CCc2c[nH]nc2C1 N1(C(C(C=C)OC)=O)CCC(C2CC2)C1C(=O)NC(COCC)C(C)C CC1(COC(=O)CCc2ccccc2F)COCC(C)(C)O1 n1(CC)ccnc1C=CC(=O)NC(C1CCCC1)CNC(c1ncoc1C)=O c1(C(=O)NC(C2CCC(F)(F)CC2)CC)cn2c(n1)CCC2 C(CCC(CO)NC(=O)CC1CCCC1C(=O)O)NC(C(=Cc1cccs1)C)=O CC1(CNC(C2CC(=C3CC3)C2)=O)NC(=O)NC1=O.C12CCOC1CCNC2=O CC1(CNC(C2C3CCN2CC3)=O)COCCN(C(c2ccc(O)cn2)=O)C1 N1(C(c2cc(OCC)n[nH]2)=O)CCCCC1C1CCCN1Cc1csnn1 N1(C(C(COCC)(C)C)=O)CCN(C(=O)CCC=CBr)C(CF)C1 Cn1cnnc1C1CCN(Cc2cnon2)C1 c1(NCCN(CCS(CCCC)=O)C(=O)OC(C)(C)C)cc(Cl)ccc1C c1(NC(CC)C(C)C)ccc(S(=O)(=O)NCCCSC)cc1Cl.OCC C=CCCCCC(=O)NC1(CC=C)CCCN(C(=O)CC2CCS(=O)(=O)CC2)C1 CCC(C)C(CC(=O)N(C)CC1CCCN(C)C1)NC(=O)C(C)(C)n1cccn1 C(C(C)CC(F)(F)F)NC(CN(C(c1c(C(C)C)nco1)=O)C(C)C)=O c1(C(=O)NC(C2(CNC(c3ccc[nH]3)=O)CC2)C)ccc(F)c(Cl)c1F N1(C(C(=O)NCC)=O)CCCC1(C)C(=O)NC1CC2CC2C1 c1(C(N(CC(N2CC(CC)OC(C)(C)C2)=O)CC=C)=O)ccccc1[N+](=O)[O-] c1(OCC=C)ccccc1C(c1nnnn1CC)NCc1ncc(C)o1 N1(C(CNC(CCC(C)C)=O)=O)CCCCC(NC(C2CCCS(=O)(=O)C2)=O)C1 C1(NC(CCNC(=O)NC)=O)CCN(C(=O)C(C)c2ccco2)CC1CO Cc1c(NCCCCC(C)C)ncnc1N(C)CC1CCC1 C1(C(N(C2CN(C(c3ncnc4sccc34)=O)C2)C)=O)CCC2(CCOCC2)C1 c1(CC)nc(C)c(C(N2CCC(O)(CCNC(=O)CN3CCCOC3=O)C2)=O)s1 C=CC1CN(C(C23CC2CCN3C(c2cnn(C)c2N)=O)=O)CC1O C=CCC(C(=O)N1CCC(C=CC(N2CCC(C3(C)CC3)C2)=O)CC1)C(C)C c1(CC(N2CCN(Cc3ccc(Br)nc3)CC2)=O)ccc(O)nc1 N1(C(c2ccc(F)c(N)c2F)=O)CCC2(CCCN2C(=O)C=C2CCOCC2)C1 N1(C(c2cc(C(=O)OC)sc2)=O)CCC(F)C(NC(=O)C(C(C)O)N(C)C)C1 n1(CC=CC)nc(C)c(C(=O)NOCc2cn(CC3(Cl)CC34CCC4)nn2)c1C n1(CC)nc(C(=O)NC2(C)CC(NC(=O)Cc3ccnn3C)C2)c2c1CCOC2 c1(C(N2CC(F)(CN(C3CC(=O)N(C4CC4)C3)C)C2)=O)ccc(N)cc1Cl N1(C(C(C)OCCN(C)C)=O)CC(F)(F)CC1CNC(C1CCCCN1N=O)=O c1(OC)ccc2[nH]c(=NCc3cc(Cl)nc(Cl)c3)nc(N3CCCC(C)C3)c2c1 N1(C(c2c(C)cc(=N)[nH]c2)=O)CCCC2(CCCN2C(=O)C2=CCCC2(C)C)C1 C1(CNC(CN(CC)CC)=O)CN(C(=O)CC2CCC(C)(C)O2)CCCO1 Cc1cccc2c1CN(C(=O)NC1(C)CC(NCc3ccnn3C)C1(C)C)C2 c1(NC(C2CCC(C)NC2)=O)ccc2nc(-c3cccnc3)oc2c1 N1(c2cc(C)ncn2)CC(C(=O)NCC2C3(CCC3)C23CCC3)CCC1(C)C c1(C(=O)NCC2N(C(CSCCC)=O)CCCC2C)cc2cccnc2nc1C C1(C(N2CCC(N3CCC3)CC2)=O)CCCC1C1CC1.C123COC(C1)(C2)C(=O)N3 c1(C(=O)NC(CNC(c2c(NCC)scn2)=O)C2CC2)ccc(C2CCC2)nc1 N1(C(CC2C(C)(C)OCC2)=O)CCC(F)(C(=O)NCCN2CCCC2)CC1 c1(CC(N2CC(C)C(CS(N)(=O)=O)C2)=O)cc(F)c(F)cc1[N+](=O)[O-] C1(NC(C)=O)CCCCC1C(N1CCC(CCNC(=O)CCC2CCCO2)CC1)=O N1(CCC(=O)NCCN(C(C2C(CC)C2)=O)CC2CC2)CCNC(=O)C1 N1(C(c2ccc(NC)cn2)=O)C2CCC1CC(CNC(=O)C(=O)CC(C)C)C2 c1(C(=O)NCC23CCC2CN(C(c2ccc(=O)oc2)=O)C3)nccn2nccc12 C(=O)(C(C)(O)CC)NCCC(=C)CNC(c1cccn1-c1cc(Cl)ccn1)=O Cc1cccc(C)c1OCC(O)CNc1ncnc(C(C)(C)C)n1.C(CCSC)NC N1(CC)CC(NC(=O)CC(C)(C)NC(C2OCCC2(C)C)=O)C(C)C1 C(=O)(C(CNC(=O)CCC(=O)N(C)C)C(C)C)NCC(=O)OC c1(C(C(=O)NCC(C)NC(C2(C)CC(=C)C2)=O)C)cccc(C(F)(F)F)c1 CONC(=O)C(C)(C)CCN(C)C(c1cc(O)ncn1)=O C(CCCCC(=O)NC(C)(CNC(c1ncn2c1CCC2)=O)CO)OCC N1(C(c2cccc(OC(C)C)n2)=O)CC(NC(=O)C(F)CC2CC2)CCC(O)C1 N1(C(C2C=C(C)CS2)=O)CCC(CC(C)NC(=O)C(C)Cc2cnc[nH]2)CC1 N#Cc1cc(NC(=O)CC2CN(C(c3cc(O)c(O)c(Cl)c3)=O)C2)ccc1Br C(=O)(C(C)(O)CCN(C)C)N1C2(C(=O)NCC3CCN(CCC)C3)CC(C1)C2 c1(CN2CCCC(CC(=O)NC(c3ccc(F)c(Br)c3)C)C2)cc(F)c(O)cc1F C1(CC)(NC(=O)CCC(C)(C)OC)CCCN(C(C2CSC2)=O)C1 C(=O)(CCC(C)(C)N(C)C)NCC(C)(CNC(=O)C(C)C(C)(C)C)OC C1(C(C(=O)NC(CC2CN(C(CC3(SC)CC3)=O)C2)C)C)CCCCC1 C1(NC(c2[nH]cc(C(C)=O)c2)=O)CS(=O)(=O)CC1NC(c1coc(CO)c1)=O c1(C(C)(C)CCN2CCC(CO)(NC(=O)C(N)=O)C2)cccc(C(F)(F)F)c1 C1(C(N(C)CC2COCCN2C(C2(C)C=CCC2)=O)=O)CCCC(F)(F)C1 N1(C(CSCC)=O)CCCC(C)(C)C1C(=O)Nc1ccc(N(C)C)nc1 c1(CNC(C)C)ccc(S(C)=O)cc1.C1(CC)CN(C(=O)C(=O)N)C1 C(CC1=CCN(C(=O)C(C)(CO)NC(=O)C2CC2)CC1)NC(c1c(C)ncn1O)=O N1(C(C2(NC(C3ON=C(CC)C3)=O)CCOCC2)=O)CCC(C2(C)CC2)C1 c1(OCC)cccc(C(CNC(=O)CC(=O)Nc2ccc(F)cc2)OC(C)=O)c1 CCCC(C(=O)NC(c1cnccc1C)c1ccccc1Cl)OC C#Cc1nc(C(=O)N(C(CNC(C2CSCCS2)=O)C2CC2)C)cs1 C1(C)(N(C)Cc2ccccc2)CCN(C(c2cccc(I)c2)C(=O)NCC(F)F)C1 Cc1c(CC(=O)NCc2cc(C(=O)NCC3CCCC(O)C3)cs2)ncn1C N1(C(CNS(N(C)C)(=O)=O)=O)CC(N(C(=O)C=Cc2cnccn2)C)C2(CC2)C1 C1(CNC(C(C)Cn2cccn2)=O)CCCCCN1C(C1CC2(CSC2)C1)=O N1(C(CCCCNC(C)=O)=O)CCC2(NC(C3CC3C(C)O)=O)CCCC12 N1(C(C(c2ccc(F)c(F)c2)C)=O)CCCCC(NC(=O)Cc2cnn(C)c2)C1 Cc1cc(C(N2CCC(F)C(NC(=O)Cc3cn(C)nn3)C2)=O)nc(O)n1 C1(C(=O)NCC(C2CCN(C(C(CC)OC)=O)CC2)(C)C)CCCCC(F)(F)C1 c1(C(=O)NCC(N(C)C(c2cccc(CO)n2)=O)C2CC2)cc2n(n1)CC(F)C2 N1(C(C2(S(C)(=O)=O)CCC2)=O)CCC2CCCC12CNC(c1cc[n+]([O-])cc1)=O C(=O)(CCCC(=O)N1CCC(C)C(CNC(C23CCC(C2)OC3)=O)C1)NC(C)C N1(C(C2CC(F)CN2C(C2CCC(CO)CC2)=O)=O)CC2C(C1)C2(F)F Cc1coc(C=CC(N2CC3CC3(NC(=O)CCCCN(C)C)C2)=O)n1 c1(C(=O)NC2C(C)CN(C(C3(C)CCOCC3)=O)C2)cccc2c1CC(=O)N2 CCCC(CNC(C1CCCSC1C)=O)C(=O)NCCc1c(C)noc1C C1(NC(COCCC#C)=O)CC(O)CN(C(c2cccc(Cl)c2)=O)C1 C(=O)(NNC(=O)CCc1ccccn1)N(CC(=O)Nc1ccc(F)cc1)C1CC1 C1(CNC(c2c(C)onc2)=O)CC(F)(F)CN1C(=O)CSCc1cccnc1 C#CCC(CC#C)C(=O)NCC1(C(N)=O)CN(C(=O)C(COC)N(C)C)C1 CC(O)(CNC(=O)C(C1(O)CCCC1)F)CNC(C1CCCC1)=O c1(C(=O)NC2C3CN(C(CCOCC)=O)C(C3)CC2)csc2c(C)cccc12 C1(O)(CN(C(=O)COC2CC2(F)F)C)CCN(C(=O)CC2CCCSC2)CC1 c1(C(=O)NCc2ccnc3[nH]ccc23)nc2c(s1)CC(C(F)(F)F)CC2 c1(C(=O)NC(C2CCOC2)CNC(C(=CC2CCCC2)C)=O)ccnc(C)c1C CCC(F)(F)C(C)(C)C(=O)NCC1C=CC(NC(c2ccc(=N)[nH]c2)=O)C1 CN1CC2(CC2)CC1C(=O)NC1CCC(C(=O)NCCCC2(C)CC2)CC1 N1(C(c2cc(C)ns2)=O)CCC2(CC1)CN(C(=O)Cc1ncsc1Cl)C2C(C)C C(=O)(Nn1cnnc1C)C1N(C(C(C(C)(C)C)OC)=O)C2C(C1)C2 N(C1COc2cc(Br)ccc21)c1nccc(N2CCC(C)OC(C)C2)n1 C12(C(=O)NCC34COC(C3)C(O)C4)COCC1CN(CC1CCN(C)C1=O)C2 c1(C(=O)NC2CC(CC(=O)Nc3cc(CC)c(C)cc3)C2)cccc2nccn12 N12CC(OCC1(C)C)CC2=O.c1(CC)cnn(CC(C)CC)c1 C1(CNC(c2c(C)cnnc2O)=O)CCCC2(CN(C(c3ccsc3C)=O)C2)O1 c1(NC(=O)CC2CCN(C(c3cccc(O)c3F)=O)CC2)cnccc1[N+](=O)[O-] N1(C(C(c2scc(C)n2)C)=O)CCOC(C(C)NC(c2nccn2C)=O)C1 O=C(CCCC(=O)N1CCCC(O)(CNC(C2CC(C3CC3)=NO2)=O)C1)C1CC1 C1(N2CC(C#N)CC(C)C2)CC2CN(C(=O)OC(C)(C)C)CC2C1 CON(CCC(=O)Nc1ccc(C2CC2)nc1)C(=O)C1(C(C)(C)O)CC1 N1(C(C(C)(C)c2cnsc2)=O)CCOC(CCNC(=O)C=Cc2cc[nH]n2)C1 C(c1c(C)coc1C)=CC(N1CCC(C(CNC(C(CC)=CC)=O)C)CC1)=O C1(CC)CCN(C(=O)Cc2cccnc2)C(C(=O)Nc2cncnc2O)C1 C1(CC(=O)OC)CCCCN1C(=O)C(C)(C)NC(=O)CC1CCCC1(F)F c1(-c2cccc(NC(N)=O)n2)csc(=NC2CCC(=O)NC2)n1C1C2(CC2)C12CC2 C1(CC)CN(C(C2CCOC2CNC(c2ccc(O)nn2)=O)=O)CC1O c1(C(=O)NCC(N2CCN(C(C(C)(C)CF)=O)CC2)=O)cc2c(cc1Cl)NCC2 CCCCCCC(C)C(=O)NCc1ccc(CNC(c2csc(CO)n2)=O)cc1 N1(C(c2c(COC)cc[nH]2)=O)CCC(C)C(N(C(=O)CCCOC2CC2)C)C1 N1(C(CC(C(=O)OC)C)=O)CC2(C1)SCCC2NC(=O)Cc1ccn(C(F)F)n1 C#CCC(C(=O)NCc1occc1C)NC(c1ccc(C)cc1)=O CC(CC(=O)NC1CCOCC1NC(=O)C(C)(C)CC#N)C(C)(C)C C1(NC(C2(C)CCC(C)C2)=O)CN(CCCOc2ccc(Cl)cc2)CCC1C N1(C(C2C(C)C2)=O)CCCN(C(C2CCN(C)C2c2ccc(Cl)cc2)=O)CC1 c1(C(=O)NC2C(CC)CN(C(C3CC=CC3)=O)CC2)cccc2cnccc12 N1(Cc2ccc(C)o2)CCCC(c2nc(C(C)O)nn2CCN2CCCCC2)C1 N1(C(c2c(CC)ncs2)=O)CCCCC(CNC(=O)Cn2cc(C(F)F)cn2)C1 N1(C(CN2CCc3n(cc(C)n3)C2)=O)CCc2cc(Br)cc(F)c21 CCC(C)CCC(O)CC(=O)NCC1CCCCN(C(=O)C(C)(C)C(C)C)C1 C(=O)(C1=C(C)OCCS1)N1C(CC)C(C(=O)NCC2C(C)(C)C2(C)C)CC1 C1(N(C(c2c(C)cccn2)=O)C)CCCCN(C(=O)CNC(c2cscn2)=O)C1 c1(NC(C2N(C(c3ccc(C)nc3Cl)=O)CC(F)C2)=O)ccc2ccoc2c1 c1(C(N(C)CC2C3CCN(C(=O)OC(C)(C)C)CC23)=O)cncc2ccsc12 C1(CC)C(C(NCS(=O)(=O)CC2CC2)=O)CCCN1C(c1scc(C)c1C)=O C(C(C)(C)C)=CC(=O)N(CCCOCCN(C)C(C1CC(CCO)C1)=O)C O=C1NCCC1C(=O)NCC(O)C(=O)NCc1nc[nH]n1 C1(C2(O)CCOCC2)(C(=O)NC2C(NC(c3cc(C(C)C)on3)=O)COC2)CC1 C(CCCCC(=O)NC(C)(C)C(C)NC(C1CC(C)(C)C1)=O)OC Cc1cc(C(=O)N(CCNC(=O)CC2CCCC(C)O2)C2CC2)cc2c1CCC2 N1(C(c2c(C)oc(C)c2C)=O)CCC2CCN(C(=O)CC(C)C(C)C)C2C1 c1(C(=O)NCCCCC(C)NC(CN(CCC)C)=O)ncn2c1CCCC2 N1(C(c2c(OC)ccnc2)=O)CCCC(CNC(C2(CC(C)C)CCC2)=O)CC1 CC(C)CS(=O)(=O)CCC(=O)N1CCCC1(C)CNC(=O)C(CO)NC(=O)C(C)C N1(C(CCCN(C(C)=O)C)=O)CC2OCCN(C(=O)C(C)CC3CCCC3)C2C1 N1(C(Cc2n(C)ccn2)=O)CC2CC1CCC2NC(=O)COCC1CCCC1 CC(CCC(C)(C)C)C(=O)NCC1CNCCC1C c1(NC2(CNC(c3n[nH]cc3Br)=O)CCOCC2)ncc2c(n1)CCOC2 C1(C(=O)NC2CCCCC2n2cc(CCCC3CC3)nn2)CC2(CCOCC2)C1 c1(CCC(=O)NC2CCC(NC(C(=O)NC)=O)C2)ccc(NS(=O)(=O)CC)cc1 C(CC(CC)C(=O)NC(C)CC1CN(C(=O)C(CC)(CO)OC)C1)=CC c1(CNC(CC2(C)C(C)C2)=O)cccc(CNC(C2CC23CCC3)=O)c1 Cn1ncc2c(C(=O)NC3C4CN(C(C5OCCO5)=O)CC34)ccnc12 C1(CC(=O)NC(C)C(C)(C)CO)CN(C(c2ccn(CCF)n2)=O)CCC1C c1(C(=O)NC(c2cncc(OC)c2)COC)cc2cccn2c(O)n1 CC1=C(C)CC(C(=O)NC2CN(C(c3ccccc3C3(C)CC3)=O)CC2F)CC1 Cc1c(C(=O)NCC2CCN2C(=O)C(C)CC2CC2)cncc1Br C1(C(N2CC(O)(C(C)C)C2)=O)CC=CC(NC(C2COCCOC2)=O)C1 CC1CCN(C(c2cnc(C3CCC3)o2)=O)C(C)C1NC(=O)Cn1cnnn1 C(=O)(C(C)CC(F)(F)F)N1C(C(=O)NCc2nc(CC)sc2)CC(F)C1 Cc1cnc(C(=O)NC2CCC(CNC(=O)C(F)(F)c3nccn3C)C2)nc1 C1(NCCSCC(N2CCOCC2C2CCCOC2)=O)CCc2nnnn2CC1 C1(NCC(N2CC3COCC3C2)=O)CCc2ccccc2C1 c1(C(C(=O)NC(C)C(C)NC(c2cnc(C(N)=O)s2)=O)=O)cc(F)cc(Cl)c1 c1(NS(NC(C)=O)(=O)=O)cc(S(=O)(=O)N2CCC(Sc3ccc(C)n3C)C2)c[nH]1 C1(C(N(CC(CCC)O)C)=O)CCN(C(=O)CC2CC(CC)=NO2)C1C C#CC1CC2CCC1N(C(C1C3CCN(C(=O)C=Cc4ccn(C)c4)CC13)=O)C2 C12(C(=O)NC(CC=C)CNC(c3cccnc3S)=O)CC3CC(C(=O)N1)C2C3 C1(OC)CC(COC)N(C)C1.C12CCCC1C(=O)N2 C12(NC(=O)NC(c3nnc4ccccn34)C)CCCC1CC(F)(F)CC2 CCCCC(CO)NC(C1(C(C)NC(C2C(C)(C)C2(C)C)=O)CC1)=O c1(CC(=O)NC(CNC(C(C2CCCC2)OC)=O)(C)C2CCC2)cccc(F)c1 Cn1ccn2ncc(C(=O)NC3CCN(C(=O)CNC=O)C(c4ccccc4)C3)c12 CN1CCOc2ncc(NC(=O)C(=O)NCc3ccnn3C(F)(F)F)cc21 N1(C(c2c(C)cc[nH]2)=O)CC2CCC(N=c3[nH]c4cc(Cl)cc(Cl)c4o3)C2C1 c1(NC(C2C(OC)C2)=O)nccn2ccnc12.C12CN(CCC1C(F)(F)F)C2=O N1(C(c2c(CC)n[nH]c2)=O)CC(O)CC1(C)C(=O)NOCC(=O)N(C)C c1(CNC(c2cc(OC)n[nH]2)=O)ccc(C(=O)NCCC2CCCN2C)nc1 c1(C(=O)NCC(CNC(c2c(CC)onc2C)=O)F)ccc(O)c(F)c1F C1(CNC(C2C(=C)CC2)=O)CC2CCC1N2C(=O)C1=C(C)OCC1 N1(C(C(C)(C)SC)=O)C2CCC1C(C)C(NC(c1cc(C)oc1C)=O)C2 C(=O)(CC(F)(F)C(F)F)N1CCCC(C)(C(=O)Nc2ccc(C(=O)NC)nc2)C1 C(CCN(C)C(c1cccc(Cl)n1)=O)(C(C)C)NC(CC1(OC)CC1)=O C1(CCNC(C2CC(SC)C2)=O)CC(F)(F)CN1C(C1CC2(C1)CC(C)C2)=O c1(CN2CC(C)(CC(N3CCCC(F)(F)C3)=O)C2)cc2ccccc2[nH]1 CC(CCCCNC(C1CCCCN1C)=O)NC(=O)CC1CN(CC(F)(F)F)C1 c1(OC)cncc(C(=O)NC(CNC(=O)C(F)C(C)(C)O)C2CC2)c1C c1(OCC=C)ccc(CC(N2CCC(NC(C3CCCO3)=O)C2CC)=O)cc1 c1(N2CCC(OC(C)(C)C)CC2)nc2c(c(=NCC3C(C)(C)C3(F)F)[nH]1)COC2 c1(C(=O)NCC(O)CNC(c2coc(CC3CC3)n2)=O)csc([N+](=O)[O-])c1 c1(CNC(N2C(c3cn(CC)nc3)CSCC2)=O)ccc(S(C)=O)cc1 C(=O)(CCC1CCc2ccccc21)N1CCCCC(NC(c2onc(C)n2)=O)C1 C1(NC(c2nc(C)nn2C)=O)CN(C(=O)C=C2CC2)CCC1C C1(CC=C)(NC(C2CCCN2C=O)=O)CCCN(C(c2cc(COC)[nH]n2)=O)C1 c1(C(=O)NC2CC(C)N(C(c3ccc(C(F)F)cn3)=O)C2)cc2ccsc2n1C C(CC(C)C(=O)NC1CCC1NC(=O)CCOCC1CC1)=CCC C1(NC(c2c(OC)cccc2)=O)CN(CC(O)CC(F)(F)F)CCC1O C1(NC(C2OCCO2)=O)CCN(C(=O)COc2ccc(F)cc2)CC1F c1(C(N2CCN(C(C3N(C(C)(C)C)CC3)=O)CC2)=O)ncsc1S(N)(=O)=O c1(C(=O)NC(CC(=O)NCCC(C)N2CCCC2)C(F)F)cc[nH]c2nccc1-2 N1(C(C2C(CCOC)C2)=O)CCC(C(=O)Nc2ccnc(SC)c2)C(C)C1 O=C(C(CO)c1ccccc1)NCC1(NC(=O)C(C2CCC2)C2CCC2)CCC1 C1(CN(C(CC2(C=C)CCC2)=O)C)CN(C(C2CSCCS2)=O)CCO1 C#CC1COCCN1C(=O)C(CC(C)C)N(C(=O)CCOC(C)=O)C CC(C)(CC#N)C(=O)Nc1cccc(NC(=O)C(C)(C)CF)c1 n1(CCCC)nc(-c2ccc(C(F)(F)F)cc2)nc1C1CCCN(C(N)=O)C1 N1(C(C2C(C)COC2)=O)CCN(C(C2C3CC4C(C3)C24)=O)CC(C)(C)C1 C1(OC)(CO)CCN(C(C2CCC3CC23)=O)CC1.C(=O)(C1CC1)O c1(NC(=O)NC(C(=O)OCC)C2(C)CC2)ccc(OC(F)F)c(Cl)c1 C(=O)(C(CC(C)C)Nc1ccccc1C#N)N1CC=CC(C(=O)OC)C1 Cn1cc2c(n1)CC(C(N1CCC(F)(CNC(c3ccnc(O)c3)=O)C1)=O)CC2 c1(CC)ccc2c(c1)C(CC(=O)NCCNC(c1ccsc1S(N)(=O)=O)=O)C(=O)N2 c1(C(C)C)cnc(O)c(C(N2CCC(C(C)NC(=O)CCCCC3CC3)C2)=O)c1 c1(N(C)CCOCCNC(c2nnnn2C)=O)cc2occc2n1C c1(C(C)NCC(c2c(C)cccc2)O)ccc(F)cc1Cl C(N=c1[nH]c(N(C)Cc2ccc(C(C)(C)C)s2)nc2ccsc12)C1CCN(C)CC1 c1(C(=O)OC)cnc(NC(=O)OCC)c(Br)c1.C12C3CC4C(C3)C14C2 c1(C(=O)OC)nsc(N(CCCCNC(=O)Cn2cc(CO)nn2)C)n1 c1(C(=O)NCCC2CCCN(C(CC(=C=C)C)=O)C2)cc(OC)cc2c1OCC2 C(CCC(=O)N1CCC(N(C)Cc2c[nH]c(=N)s2)C1)NC(CCC)=O C(CCC(C)(C)C)(OC(F)F)NC(C(C)SC(F)(F)F)=O C1(NC(C(C)CCO)c2nnnn2CC2CC2)CC2(COCCO2)C1 C12(C(=O)NC(C3CC=CCC3)C(=O)NCCCOCC(C)C)CC1CNC2=O N1(C(C(C)CC2CCC2)=O)C2CCC1CC(F)(CNC(C13CCC(C1)OC3)=O)C2 C(=O)(CCCCC=C)N1CC(C#C)(C(N(CCCc2cnn(C)c2)CC)=O)C1 n1(CCNC(CN2CC3C(OCC)C3C2)=O)cc([N+](=O)[O-])cn1 C1(CC(=O)NC2COCC2CNC(C2(C)CC(F)C2)=O)(OC)CCOCC1 N1(C(C23CCC(OC)C2C3)=O)CCC(NC(=O)CN(C2CCCC2)C)C12CC2 N(C(=NCCCCl)N1CCC(C)(OC)C1)Cc1c(OCCOC)ccc(OC)c1 c1(-c2nc(NC(N3CCc4cccc(Br)c4C3)=O)on2)cc(Cl)cc2ccncc12 CCC(C)(CNC(=O)CCOCCCOC)NC(c1cscc1Cl)=O C1(OC)CN(C(c2ccc(C(N)=O)o2)=O)CC1Cc1ccnc(N(C)C(C)=O)c1 C(=O)(C(C)C(=O)N1CC(O)(CNC(=O)CCCc2cccc(Br)c2)C1)OCC Cc1ccnn1CC(=O)N(CCCCCNC(c1cc(C2CCC2)no1)=O)C n1(Cc2cnc(NC(=O)NC3CCNCC3)s2)nc(CC(F)(F)F)o1 c1(C(=O)NCCN(C(=O)Cc2ccccc2C)CC)c(C)ncn(C)c1=O Nc1ccc(Cl)c(C(N2CCC(NC(=O)CCc3ccoc3)C(F)C2)=O)c1 CC1=NOC(C(=O)NCC2CC(C(=O)NCC3(C(C)(C)O)CC3)C2)C1 C1(NC(c2[nH]nnc2C2CC2)=O)CC(C(=O)N2CCOC(C3CC3)C2)=CC1O c1(CC(=O)NC2(C)CC(NC(C3CCCCCCC3)=O)C2)ccc2c(c1)COC2 C(C#CC(=O)NC(C)C(C)(C)OC)NC(C(C)OCC=C)=O c1(OC)sccc1C(=O)NCC12CC(NC(=O)CCn3ccnn3)(C1)C2 C(C(C)C)(C(O)C(=O)N1CCCN(C(=O)Cc2cc[nH]c2)C(C)C1)OC C1(CC(=O)NCCCOCCNC(CNC(=O)OC)=O)CCC2CC12 N1(C(C23CC(NC(c4scc(C#N)c4)=O)(C2)C3)=O)CC2(CCC(=O)NC2)C1 Cc1ccc([N+](=O)[O-])cc1C(N1CCC1c1cn(-c2ccncc2C)nn1)=O c1(C(=O)NCC2(F)CCCN(C(CSC)=O)CC2)n[nH]c2ccc(F)cc12 C=CC(CC)CC(=O)N1CC(CNC(c2cnc(NC(=O)NC)o2)=O)C(C)C1 N1(C(C(C)CSC(F)(F)F)=O)CCN(C(c2nncn2C2CC2)=O)CC1 CCCC(C(=O)NC1CCC(C(N2CCC(CO)(COC)C2)=O)C1)OCC n1(CNC(C2(C)C(NCC)CCC2)=O)cc(Cl)c(CC(C)(C)C)n1 CCCC(CC(C)C)C(=O)N1CC(O)CC1CC(=O)NC1CCC([N+](=O)[O-])CC1 CC1C(N(C(=O)CCOCCNC(=O)C=C2CCC2)C)CCN1C N1(C(C2CC(C#N)C2)=O)CC2CC1CN(C(c1coc(-c3ccccc3)n1)=O)C2 c1(CCCC)ccc(C(=O)N(C(C)C)C(c2cccc(F)c2)=O)cc1N N1(C(c2c(C)nc(C)s2)=O)CCC2C1CCN2C(c1ccc(F)c(Br)c1)=O N1(C(CC(CN(C)C)O)=O)CCOCC(CNC(c2cn(CC3CC3)cn2)=O)C1 c1(C(=O)NC2C(C(C)C)N(C(c3ccsc3)=O)CC2)nn(C)c(C(F)(F)F)c1Cl N1(CC(=O)N(CC(C)NC(c2ccc(CN(C)C)[nH]2)=O)CC)CCC(C)(O)C1 Cc1cc(C)n(CCC(=O)NCC2COC(C(C)C)C2)n1.C12(CC1)C(C)NC2=O Cc1ccc(C(N2CCOC(CN(C)C(C3CCCC(C)(C)C3)=O)C2)=O)nc1C C1(N(C(=O)CN2CC(CO)C2)C)CCN(C(c2cc(C(F)F)[nH]n2)=O)C1 c1(C(C)CNC(N2CC(N3CC(C)CS3(=O)=O)C2)=O)cccc(S(N)(=O)=O)c1 N1(C(CCCCC)=O)C(CNC(C2(CN(C)C)CCCCC2)=O)CC2COCC12 C1(C(N2CCC(NC(CCCc3nc(C)sc3)=O)C2)=O)CC2C=CCC(C1)C2 N1(C(C(C2OCCC(C)C2)c2cccc(Br)c2)=O)CC2C(C1)C2(F)F N1(C(CCCSC)=O)CC2CN(C(c3ccoc3C)=O)CCC12 C(CCCCC(=O)N1CCC(C)(CC(=O)OCC)C1)OCC=CC C(C1CCc2ccccc21)N(C(=NCc1ccc(SC)cc1)NCC(C)(C)C)C N1(C(C2(COC)CN(C(C3CCC4(CCC4)C3)=O)C2)=O)CCn2nccc21 Nc1ccc(C(N2CCC3C(NC(C4C=CCC4)=O)C23)=O)cc1F C1(NC(C2N(C(CC)=O)CCCC2)=O)CC2CC1N(C(c1cc(C)cnn1)=O)C2 N1(C(CCN2CCC(C)CC2)=O)CC2C(C1)N2S(=O)(=O)CCCCl c1(C(C)C)cc(C(=O)NC2CC(N(C)C(C3CC4(CCC4)C3)=O)C2)n(C)n1 Cc1ccc(-c2cn(C3(C(=O)Nc4cccc(I)n4)CC3)nn2)c(CO)c1 C1(C2(Cl)CC2)(CNC(C(C)NC(=O)NC)=O)CCN(C(C2CC2COC)=O)C1 C1(C(=O)NCC2(CCNC(c3c[nH]c(=N)s3)=O)CC2)CCC(CO)CC1 C1(NC(c2ccnc(C)n2)=O)CC(F)CN(C(=O)CCN2CCCCC2C)C1 C1(c2n(C)c(C3(C)CCS(=O)(=O)CC3C(F)(F)F)nn2)CCN(S(N)(=O)=O)C1 C#Cc1ccc(C(N2CC3CC3(C(=O)Nc3c(C)cccc3F)C2)=O)cc1 c1(C(N2CCC(CNC(C3C(=C)CC3)=O)(CO)CC2)=O)ccc(N)cc1[N+](=O)[O-] NC1CC2(C1)CC1(CC(F)(F)C1)C2NCc1cnc2n1CCC2 C1(C(=O)NCCCC(=O)OCC)CCCCCN1C(=O)CC1CC(C)=NO1 C1(N(C2CCCCC2)C(=O)C(=O)N(C2CC2)C2CC2)CCCOC1 c1(CN(C(=O)C(N2CCOC(Cc3cccc(F)c3)C2)=O)C)cccc(F)c1F C1(C(=O)NC(C#C)C2CC2)CC2(CC2)CN1C(=O)C(C)NC(C)=O c1(C(=O)NCCC(=O)NCC(=O)NCC=CCNc2ccccc2)cccnc1 c1(OC)cc(CN2CC3CCN(C(=O)Cc4ccsc4)C3C2)cc(CN(C)C)c1O C(=O)(N=c1ccn(CC(C)C)[nH]1)C1CCN(Cc2cncc(C#C)c2)C1C CCC(O)C(=O)N(C(=O)CN)CCCCOCCOc1ccccc1.C(COC)N.C(C)(C)O C(CC1=CCCCC1)N(C(CN(C1CCC1)C(C1C(C(N)=O)C1)=O)=O)C1CC1 c1(NC2C(C(F)(F)F)CCN(C(C3(C)CCCC3)=O)C2)c(F)cccc1[N+](=O)[O-] C1(C(N(C(CC)C)C)=O)CN(C(c2cn(CC)cn2)=O)CCC1(C)C Cc1nc(C)n(CC(=O)N(C2CCCC2)CCNC(=O)C=Cc2ccoc2)n1 c1(OCC)ccc(Cl)cc1C(=O)N(C1CN(C(c2cc(OC)no2)=O)CC1O)C c1(CC(=O)NC(CN(C(=O)C(CC)OC)CC)C)cc[nH]c(=N)c1 CC1OC2CCC1(C(=O)NC1CC1NC(C1C(C)C1C)=O)C2 C(=O)(C(C)(C)S(C)(=O)=O)Nc1ccc(NC(c2c(OC)ccc(CO)c2)=O)cc1C O=S(=O)(c1ccc(N2CC3CC3C2)cc1Cl)NCc1cccc(Cl)c1 N1(C(CS(CC)=O)=O)CC(CNC(c2cn(C3CCCC3)nc2C)=O)C2(CC2)C1 CC1(C(=O)Nc2cc(F)ncc2F)CCCN(C(c2c(Br)cccc2Br)=O)C1 c1(C(=O)NCCN(C(=O)CCC=C(C)C)CCOC)nnc2ccccn12 C(=O)(CC(COC)NC(C1CC2(CCC2)C1)=O)NCC(NOC)=O c1(CCC)nc(C)c(C(=O)NC(C2CCCC2)CNC(c2c[nH]c(Br)c2)=O)o1 N1(C(c2cnc(C)nc2C)=O)CCC(NC(C2(C)CC2)=O)CC(C)(C)C1 C1(NC(CCc2c(C)n[nH]c2C)=O)C2CC1CN(C(c1ccc(=O)n(C)c1)=O)C2 N(C(=NCc1ccc(CS(C)(=O)=O)cc1)NCC1(CF)CCC1)C(C=C)C C1(C2(O)CN(C(=O)CN3CCCNC3=O)C2)(CNC(C(C(C)C)C)=O)CC1 C1(CCC)CN(C(c2c(C)cccc2O)=O)CCN1C(=O)C(C1CCCC1)OC Cc1cc(CC(=O)NCC2CCCN2C(=O)CC2CCCCN2C)cc(C)c1 Cc1nn(C)c(C)c1C1OCCC1NC(C1CC2(C1)CC(CNC(=O)CO)C2)=O C(c1cnccn1)=CC(=O)NCC(CNC(C(F)=CC)=O)(C)O Cc1cc(=NC2CN(C(=O)CN3CCS(=O)(=O)CC3)CC3(CCC3)C2)[nH]cc1C#N CC1CCCN(CCc2nc(CCC(N)=O)n(-c3ccc(F)cc3)n2)C1 C1(C(=O)OCc2ccc(C(=O)OCC)s2)CCCC2(CCOC2)O1 c1(C(C(=O)N(C(C)CNC(=O)Cc2nc[nH]n2)CC)C)cnn(C)c1 N1(C(C2CC=C(C)CC2)=O)CCN(C(=O)CC(O)C2CCCC2)C(C)C1 N1(C(C2N(CC)CCC2)=O)CCCC(F)(C(=O)NCCCC2C=NNC2=O)C1 CN1CCN(c2ccnc(NCCNC(=O)C(F)(F)F)n2)C2CC12 c1(N(C(C)CCC2CCCC2)C(N2CC=CC2)=O)ccccc1 c1(C(=O)NC(CCNC(c2n(C=C)nnc2)=O)(C)C)cc(Cl)c(Cl)n1C C1(NC(C2CCCN2CCCC2CC2)=O)C2CN(C(c3cccnc3)=O)CC12 C1(O)(C2CCN(C(=O)OCC)CC2)CCN(N2CC(O)C(F)C2)C1 C(C)(C(C)(C)NC(c1cnc(Br)s1)=O)NC(CCOC(C)=O)=O O=C(N=c1ccc(N2CCCCC2)n[nH]1)Nc1ccc(F)c(F)c1Cl N1(C(CC(C(C)C)C)=O)CC2CCC1CC2NC(c1cc(Cl)n[nH]1)=O N1(C(C(C2CCCC2)OC)=O)CCCC(CN(C)C(C2CCC(=O)NC2)=O)C1 CN(C1CCc2ccccc21)N1CCOC(c2ccc(Br)cc2)C1 c1(CCC)cc(C(=O)NCC2CCN2C(=O)CSC2CCOC2=O)n(C)n1 N1(C(C2ON=C(CC)C2)=O)CCCC2CN(C(C3CC(=O)C3(C)C)=O)CCC12 C(=O)(C(C)(C)C(N)=O)NCC(CC(=O)N(C(C)COC)CC=C)C1CCC1 C1(N(C(C2C(=C)CC2)=O)C)CCC(NC(c2ccncc2N)=O)CC1 c1(C(N(C2CCN(C(CC3(C(=C)F)CCC3)=O)C2)C)=O)nc[nH]c2ncnc1-2 N1(C(CCC(=O)NCC)=O)CCC(NC(=O)CN2C(=O)CCC2=O)CCC1 c1(OC)ccc(C(=O)NCCCN(CCO)C(C2OCCOC2C)=O)nc1Cl CC12CN(C(c3cnc(O)s3)=O)CC1CN(CC(c1ncccc1N(C)C)=O)C2 C(=O)(CCCCC(C)CC)N1CC(O)(CNC(COCCSC)=O)C1 N1(CCOC)CC(C(N2CCCC(CC(=O)Nc3csnc3C)C2)=O)CC1=O c1(C(N2CCCC(CC(=O)NC3(CO)CCC3)C2)=O)cccn2nccc12 c1(N2CCOCC(C(=O)NC(C)(C)C)C2)ccccc1S(C)=O.C1(=O)OCCN1 CC1(C(=O)NCc2csc(C(=O)NC3(C(N)=O)CCCC3)c2)CC=CC1 c1(CC(=O)NC(CCCCNC(CC(=C)C)=O)C)cc(OC)ccc1F CC(C)CC(CNC(=O)COCCF)C(=O)NCC(C)(F)C(C)C C1(C(N(CC(C)(O)C2CCC2)C)=O)CCCN(C(C2(C#N)CCCC2)=O)CC1 CCC(C(=O)N1CC(C2C(=O)N2)C1)C(C)(C)CC.C(C1=NOC2COCC12)OC C1(CC(=O)NC2CC(C)(NC(c3cc(C(C)C4CC4)n[nH]3)=O)C2)CCCCN1C c1(C(N2CC3(OCC(NC(c4ccc[nH]4)=O)C3)C2)=O)n[nH]c2cc(Br)ccc12 Cc1cc(C#N)cc(NC(C2CCCO2)C)n1 CC1(NC(=O)COCC2CC2)CCCN(C(=O)C(F)(F)c2cccnc2)C1 C(=O)(CC(C)(C)N(C)C)N(C1CCN(C(C2CCC=CO2)=O)C1)CCC C(=O)(C1=CCCC1)NC(C(=O)NCCCC(=C)Cl)(C)C1CCC1 N1(C(CCS(=O)(=O)NC)=O)CCC(C)(C)C(NC(c2c(C)ncnc2C)=O)C1 C(CO)(C(C)(C)C)NC(C1C(NC(C(CC)OC)=O)COC1)=O O=C1CCC(CC(N2CC3CC2(C(=O)NCC2CCCO2)C3)=O)CC1 c1(C(=O)NC2CCN(C(C3(CC)CC3)=O)CC2O)ccc(Br)c(C)c1C C(C(O)C(=O)N=c1ccn(CC(N)=O)[nH]1)NC(C1(NC(C)C)CC1)=O C1(C)(C(N(C(C(=O)OC(C)C)C)C)=O)C2CC3CC(C2)CC1C3 Cc1cccc(CN2CCN(C(c3cccc(Br)c3Cl)=O)C3CC23)c1F CC1(NC(C2CC2c2ccccc2)=O)CC(NC(c2ccsc2C(F)F)=O)C1 Cc1cc(N(C)CC2CCOC(C)C2)ncc1S(=O)(=O)N(C1CC(F)(F)C1)C CCC(CC)C(F)C(=O)NCCOCCCN(C)C(C1CCN(C(C)=O)C1)=O CCC(C)CC(C(=O)Nc1ccsc1)c1ccccc1 C1(NC(COCC=C)=O)CCC2(CCCN(C(c3cocc3Br)=O)C2)C1 N1(CCN=C(NC(CC)C)NCc2cn3c(n2)SCC3)C(=O)C2CC=CCC2C1=O C#CCCC(N)C(=O)N1CC(O)(CCC(C)(C)C)C1 Cc1ccc2cccnc2c1C(=O)NCCCCCCNC(=O)C(C#N)C1CC1 C(=O)(C1CCc2ccc(OC)cc21)NCCCN(C(C1C(=C)C1)=O)C Cc1ccnc(F)c1-c1csc(CNC(c2cc(O)ccc2F)=O)c1 C1(C(N(CC)CC2CC2)=O)N(C(C2CCC(O)CC2)=O)CC12CCCC2 c1(C(=O)NCC(CNC(CC(C)C)=O)CO)ccc(N2CC(F)CC2=O)cc1 C1(C(=O)NC(CCOC)CNC(C2(C)CC2C)=O)CC2(CCCC2)C1 C(CC(C)C)(C(=O)NC1CCN(c2ccc(-c3ccccc3)o2)C1)OC C1(CCC)CN(C(=O)C=CC=C(Cl)Cl)CCN1C(=O)CC1CCCC(C)(C)C1 c1(C(=O)NCCCCC2CN(C(C3CCC(SCC)O3)=O)C2)ccc(OC)nn1 CC1C(NC(c2cc(C3CC3)nn2C)=O)CCN1C(c1ccc(C2CC2)cn1)=O C1(NC(c2cc(OC)cc(Cl)c2)=O)CC2(CCN(C(C3CCC3(C)C)=O)C2)C1 C1(N(C(C2C(CC)C2)=O)C)CN(C(c2cccc(C3CC3)c2Cl)=O)CC1(C)C CC(C)CCC(C(=O)NC1CCN(C)C1(C)C)NC(=O)C(C)OC(C)(C)C c1(C(N2CC(NC(c3ccc(Cl)c4occc34)=O)C2)=O)ccc2ccnn2c1 N1(c2c(OC)cncn2)CCN(C(c2cn(C3CCOCC3)nn2)=O)CC(O)C1 Cc1ccc(Br)c(F)c1C(=O)NC1(C)CCOC1C1CC1 C#Cc1ccc(C(=O)N(C(CNC(C2(CC(F)(F)F)CC2)=O)CC)CC)c(F)c1 N1(C(c2cnc(C3CC3C)s2)C(=O)NCCCC(=O)OC)CCNC(=O)C1(C)C C1(C(N2CSCC2C(=O)NCC(C)C(F)F)=O)(OC)CCC(C)C1 c1(N2CCCC(CCNC(c3c(C)c(I)ccc3)=O)C2)ncnc2cc(I)sc12 c1(N(C)CCN(C)C)cc(Br)ccc1S(=O)(=O)NC1CC1c1ccc(C#N)nc1 c1(OC)cnc(F)c(C(=O)NCC2(OC)CN(C(C3CCCN(C(C)C)C3)=O)C2)c1 c1(C(N(C2CCN(C(=O)CCNC(=O)NC)CC2)CCC)=O)cccc(C)c1Cl c1(OC)ncc(CN2CCCC(C(=O)Nc3ncc(C(F)(F)F)cn3)C2)cc1C N1(C(CC2(N(C)C)CCC2)=O)CCCC(O)(CNC(=O)CC23CCCC2C3)CC1 N(C(=NCc1ccccc1)N1CCC(C(=O)Nc2cc(C)ccn2)C1)C(C=C)C c1(C(N(CCNC(c2cc(C(CC)CC)no2)=O)C)=O)ccc2[nH]c(=N)[nH]c2c1 CCCC(CCC)C(=O)N1CCC(N(C)C(C2CCCC23CC3)=O)C1 c1(C(=O)OC)cc(C(=O)NCC(CNC(C2COC(=O)N2)=O)OC)n(C)n1 CC12COCC1CN(C(C1N(C(=O)C3=NNC(=O)C3)CC13CCCC3)=O)C2 c1(CC(=O)NCC(C)NC(C2CNC(=O)CC2C)=O)ccc2c(n1)CCC2=O CC(C)C(O)CC(=O)NC(Cc1ccoc1)C(=O)NC1CC(CF)C1 Cc1cc(C(N2CC3CC3(NC(=O)CCc3ccsc3)C2)=O)c(C(F)(F)F)o1 c1(C(N(C)CC2CN(C(C34CCCN3CCC4)=O)C2)=O)cc([N+](=O)[O-])ccc1F N1(C(c2c(C)c(C(F)(F)F)n[nH]2)=O)CCC(C)N(C(c2cc(Cl)cnc2O)=O)CC1 C(=O)(C(CC(=O)N1C2CCCC1COC2)SC)OC C(C(O)C(=O)N1CCCC1C(C)(C)CNC(c1cc(Br)n[nH]1)=O)N(C)C c12cc(F)c(c(F)c1)CC(=O)N1CCC(C1)N(C)C2=O.C1(OC)COCCN1C Cc1ccc(-c2ncc(NC3CC4CCC3N4C)s2)cc1C C#Cc1ccc(C(N2CCC2CNC(c2cnn(CC3CCCC3)c2)=O)=O)cn1 C(=O)(C1=CS(=O)(=O)CCC1)N(C(CNC(C1CCC2CC2CC1)=O)C1CC1)C N1(C(CNC(CC)=O)=O)CC(NC(=O)C(CC(C)C)NC(N)=O)CC12CCC2 N1(C(C2C=CCC(C(C)=O)C2)=O)CCC(C)(n2cc(C3CCCC3O)nn2)CC1 Cc1ccc(F)cc1CNC(=O)CSCCNC(=O)CC1CCCCC1O N1(C(C=CCN(C(C(C)SC)=O)C)=O)CC(F)(F)C1 c1(CCNC(c2n(C)nnn2)CC#N)ccccc1[N+](=O)[O-] CCC(C)(C(c1nnnn1C1CCCCC1)NCCCc1cccs1)OC c1(-n2c(C3(NCCCN4CCCC4)CC(OCC)C3)nnn2)cccc(Cl)c1 C1(CNC(COCCSC)=O)C=CCN1C(=O)Cn1cc(C2CC2)cn1 N1(C(=O)CNc2nccs2)C2CCC1CC(NC(C1(O)CCOC1)=O)C2 c1(CNC(C(C)C2(NC(=O)COCC3CCC3)CC2)=O)csc(CC2CC2)n1 N1(C(CC2(OC)CC2)=O)CCCC(C)C1C.C12CC(C1)C(=O)N2 N1(C(c2cc(CCOC)no2)=O)CCOCC1C(C)(C)C(=O)O c1(NC(=O)C(c2cccnc2)NC(C2C(C)C2C2CC2)=O)nccc2[nH]ccc12 C1(C(=O)N(CC(O)CO)C(C)C)(CC)C=CCN1C(=O)Cn1nnc(C)n1 c1(C(=O)OC)cccc(Cn2cc(CC3CCN(C(=O)CCC(F)F)C3)nn2)c1 c1(CN(CC(=O)Nc2cc(C(=O)NC)nc(O)c2)C)cc(F)c(F)c(F)c1 C(=O)(C#CC1CCCC1)N(C1CCC(NC(c2c(OC)c(Cl)sc2)=O)CC1)C c1(SC)cccnc1NC(=O)C(COC(C)C)NC(=O)CSCC(N)=O n1(CC(=O)NC(C)(CNC(c2nccnc2O)=O)C2CC2)cnc([N+](=O)[O-])n1 C(c1ccc(F)cc1F)=CC(=O)NC(C1CC(NC(=O)CCN2CCCC2)C1)C c1(C(=O)OCC)cn(CCC(=O)N2CC(Cc3nnc(OC)s3)C2)nn1 CC1(CNC(=O)Cc2ccc(F)cn2)CCCC1NC(C1(O)CCOC1)=O C(=O)(C(C)CCCC)NC(CC(=O)NC(C=C)CO)COC c1(CNC(c2n(CCOCC)nnn2)c2ccnn2C(C)CC)c(F)cccc1Cl c1(C(C(=O)NCCN(C)C(C23CCCC2C3(F)F)=O)(C)C)ccc(F)c(Cl)c1F C(CCS(C)=O)(C(=O)NC1CCC(NC(c2ocnc2C2CC2)=O)CC1)N(C)C C1(CNC(CC(=C)C)=O)CC(C(C)C)CCN1C(c1cnccc1OC)=O Cc1ccc(F)cc1C(N1CCCCC(NC(=O)C(C)(O)Cc2ccccc2)C1)=O N1(C(CC=CC)=O)CCCCC1C1(NC(c2cc(C)co2)=O)CC1 c1(C(N)=O)ccc(C=CC(N2CC(NC(C3(CF)CC3(F)F)=O)C(F)C2)=O)o1 C1(CNC(c2c(F)ncc(C)c2)=O)CC2(CCC2)CN1C(C1CCC(=O)N1C)=O N1(C(Cc2c(C)[nH]c3ccccc32)=O)CCCC(C2CN(C(C3CC34CC4)=O)C2)C1 c1(C(N2C(CC3N(C(C(CSC)O)=O)CCC3)COCC2)=O)cncn(C)c1=O C1(N(C(=O)Cc2ncc(C)s2)CC)CCN(C(C2CC2F)=O)CC1 C1(C)(NC(CCC(=O)NCCC)=O)CCN(C(C2(C)CC(O)CN2)=O)CC1 Nc1c(C(=O)Nc2ccc(N3CCCC3=O)c(F)c2)cc(Cl)nc1Br CC1=C(C(=O)NCC2CCOC2C(=O)NCC2CC2c2ccoc2)CC1 c1(C(=O)NCC2CCCC(NC(CCOC)=O)C2)c[nH]c2ccc(C)cc2c1=O N1(C(CC(=O)NCC#C)=O)CCN(C(C2(c3ccc(F)cc3)CC2)=O)CC(O)C1 N1(C(C2CC(C)(CC)C2)=O)CCC(NC(c2ccc(CCOC)cc2)=O)C1(C)C c1(C(=O)NCCOCCN(C)C(c2cc([N+](=O)[O-])nn2C)=O)cc(F)c(F)cc1Cl CCC(O)C(F)(F)C(=O)NC1CC(NC(=O)CN2CC(C)(C)C2)C(O)C1 C1(C)(CNC(c2nc(C(C)C)sc2)=O)CC(F)(F)CN1C(c1coc(Cl)n1)=O CN=C(NC1CSC1(C)C)N1CCCC(Oc2ccc(Cl)cc2)C1 c1(CCCC(=O)NCC(CC=C)NC(C2(COC)C=CCC2)=O)ccccc1Cl C(=O)(CC(C)(C)O)NCC=CCC1N(C(c2c(CCC)[nH]cc2)=O)CCC1 c1(CNC(CC(C)(C)N(C(C2(NC(C)=O)CCC2)=O)C)=O)c(O)cccc1F c1(CCC(=O)NC(C2CN(C(C3(C#N)CC3)=O)CCO2)C)cc(F)ccc1F C1(NC(c2c(C)nc(COC)s2)=O)CC(F)CN(C(c2cc(C)ncc2C)=O)C1 C=CCC(CNC(c1[nH]ccc1C1CC1)=O)C(=O)N1CCC(CO)C1 C12(C(=O)NCC3C(NC(c4ccc(-c5cccc(Cl)c5)s4)=O)C3)CC1CNC2=O CN(CCCC(=O)NC(C)(C)CNC(c1ccc(F)cc1OC(F)F)=O)N=O c1(C(C)C)cc(C(=O)NCC2CCCCN2C(=O)Cc2cncs2)ccc1F C1(NC(=O)CC2(O)CCCCC2)CCCN(C(=O)CCc2ccsc2)CC1F C1(NC(c2ccc(C)s2)=O)CCCCCC1C(N1CCC1CN=[N+]=[N-])=O CCC(CC(=O)NCC1(CCCO)CC1)N(C(=O)C(C)=CCO)C c1(C(N2CC(C(=O)O)C(C(=O)OC)C2C)=O)cc(C)c(Br)c(Cl)c1 C1(NC(COCCNC(CC(C)n2ccnc2)=O)=O)CN(C)C(=O)C12CC2 C(=O)(C1Cc2ccccc21)N1CCN(C(c2cc(CSCC)on2)=O)CC1CC N1(C(C2CC(C#C)(O)C2)=O)CC2CC1CCN2C(C1CCCOCC1)=O C1(NC(C(C(CC)O)C)=O)CCN(c2nc(C(F)F)nc(=N)[nH]2)CCC1CO Cc1ccnn1CC(=O)NC(CNC(=O)C(C)Cc1ccccc1)C1CC1 C(=O)(C(F)CC(C)(C)NC(C1CN(c2cccnc2)C1)=O)N(C1CCCSC1)C CCCCC(C(=O)NC(CCN(C(=O)CC12CCCC1C2)C)C(C)C)NC(N)=O c1(CC)cccc2c(C(=O)NC3CCCCC3NC(C3CCCCS3)=O)c[nH]c12 N1(C(c2c(NC)scn2)=O)CCC2(CCCN2C(=O)C(C)CC(=O)N(C)C)C1 c1(C(N2C(CCNC(C3COCCN3C)=O)CC(OC)C2)=O)cc(N)ccc1Cl c1(CC)cc(C(=O)NCCOCCCNC(=O)Cc2ncc(Cl)s2)ccc1F c1(C(=O)NC23C(CN(C(CC4CC(=O)NCC4)=O)C2)C3)nncc2ccccc12 c1(C(N(CCCCN(C)C(C2(C)CCCS2)=O)C)=O)ccncc1C1CC1 C1(CC)CN(C(c2cccc(C3CC3(F)F)c2)=O)CCN1C(c1ccc(C)o1)=O C(=O)(CCCC(=O)N(C)C)N.N12CCOC(C1)CN(C)C(=O)C1(CCC1)C2=O.CN C1(C(=O)NC(C2CCCO2)(C)C)C=CC(NC(c2ccc(C(F)F)o2)=O)C1 CC(CC(C)(C)CO)NC(=O)CC1N(C(c2cnn(C)n2)=O)CC1(C)C C#CCC(CC(F)F)C(=O)N1CC(NC(=O)Cc2sc(O)nc2O)C2CC2C1 O=C(C1=CS(=O)(=O)c2ccccc21)N1CC2CCN(C(c3ccsn3)=O)C2C1 C(=O)(C(C(C)(F)F)c1ccccc1)N(CCN(C(=O)C=CCO)CCOC)C1CC1 C1(C(N(CCCOCCNC(=O)CSc2nc[nH]n2)C)=O)CC12CC(O)C2 c1(OC)cccc(OCc2nc(-c3cccc(Cl)n3)nn2CCCO)c1 N1(C(=O)CC2CC=CCC2)CC2CCCC2(Nc2ncncc2Cl)C1 N1(C(c2cccc(C)n2)=O)CC(=O)NC2CN(C(c3ccccc3Cl)=O)CCC12 c1(OC)cc(C)c(Cl)cc1C(N1CC2C(C1)N2C(c1cc(F)c(C)c(F)c1)=O)=O N=c1[nH]cc2c(c1C(N1CCC3(CCC3)C(CNC(=O)C3=CCSC3)C1)=O)CCC2 N1(C(Cc2nnc(C)s2)=O)CC2(C)CN(C(C3CC3C)=O)CC2(C)C1 C(=O)(C(C)(C)CC(C)C)NCCCN(C(CCCNC(=O)NCC#C)=O)CCOC Cc1onc(Cl)c1C(=O)NC1CN(C(C2SCCS2)=O)CC1CC1CC1 CC(C(=O)N(C)CCOCCCNC(C1CCN1C(C)(C)C)=O)C1CCC1 C1(NC(C=CC)=O)CN(C(c2cnn(-c3nccs3)c2)=O)C2(CCOC2)C1 c1(CC(=O)NCC2(C)CCN(C(=O)CN3CC=CC3)C2)cccc2ccccc12 c1(CCC(=O)NCC(C(C)(C)C)NC(C(COCC)C)=O)cc(F)cc(F)c1 C123CCC(CC1)(C2)NC3=O.CN1CCCCC1C(=O)NCC1OCCC1C(=O)O C1(NC(CCn2ncc(C)c2)=O)C2CCCN(c3ncnc(O)c3Br)C2C1(C)C N1(C(c2nc(C)oc2C)=O)CC2CCC1CN2C(=O)C(C(C)(C)C)n1ccnn1 c1(CCC(=O)NC2(CC=C)CN(C(C3(C)CCCN3C)=O)C2)ccc(F)cc1C c1(C2CC(=O)NC2)cccc(C(=O)NCC2CCCN2C(=O)CC2CC2)c1 c1(C(N2CCC3CN(C(C4CCSC4)=O)C3C2)=O)cc2nccc(Cl)c2s1 c1(NC(CC#C)COC)cnc(Cl)c(C2CC2)c1 C(C(C)C(C)C(=O)NC1(CCC(=O)NCc2ncoc2C2CC2)CCC1)OC C(=O)(C1=COCCO1)NCC12C(CN(C(C(c3n(C)ccc3)=O)=O)C1)C2 CCC(CC)(CCNC(c1nccc(N)c1Cl)=O)NC(=O)CCc1cncnc1 C(C)(C(O)C(=O)NCCCN(C)C(C1(OC(C)C)CCOCC1)=O)OC N1(C(C23CN(C(C4CC(C#C)(O)C4)=O)C(C2)C3)=O)CC2(C1)CC1(CCC1)C2 C#CC(C(C)OC)NC(C1(C)CC(NC(c2cc(O)cs2)=O)C1)=O N1(C(C=Cc2ccc(SC)s2)=O)CCCN(C(c2ccc(C#N)s2)=O)CC1 c1(C2(CNC(c3c(CC(C)(C)O)cco3)=O)CC2)ccccc1Br c1(C(=O)NCC(CNC(=O)CCc2cn[nH]c2)OC)cnc(S)n1C1CC1 CC(F)(F)C(F)C(=O)NC1CC(NC(c2cc(Br)cnc2O)=O)C1 c1(C(=O)NC2(C)CC(NC(C(CCC)O)=O)C2)c[nH]c2cc(OC)ccc12 N1(C(C2C(C)(C)CCO2)=O)CC2(C1)CN(C(c1ccc(-c3ccncc3)s1)=O)C2 N1(C(c2nc(COC)sc2)=O)CCCC(NC(C2CCCCS2)=O)CCC1 c1(OC)ccc(C(=O)N(C2CCN(C(=O)CCc3ccc(=N)[nH]c3)CC2)C)nn1 N1(C(CS(=O)(=O)NC)=O)CCCC12CCN(C(=O)Cc1ccc(O)cc1C)CC2 C1(C(N(C)CC2N(C(C(CCC)O)=O)CC(F)C2)=O)CC(c2ccncc2)=NO1 c1(CN2C(C(=O)NC3CN4CCC3CC4)CC3CC32)c[nH]c2cccc(Cl)c12 C(CCC(C)(C)C(=O)OC(C)(C)C)OC.C1(CO)CCCCNC(=O)N1.C(=O)O c1(CNC(c2n(CCCC)nnn2)c2cnc(CCOC)s2)ccc(Cl)c(Cl)c1 N1(C(c2scc(C)c2)=O)CC(O)CC1CC(=O)NCC(C)C C=CCC(CC(=O)NCc1cnc(CC)nc1)NC(=O)CCc1ccncc1 C12OCCC1CNC2=O.C1(CC)OCCC1NC(=O)C(C)(C)OC(C)(C)C C1(C(=O)Nc2cnccc2Cl)CC12CCN(C(=O)Cn1cccn1)CC2 c1(CC(=O)NC(C2N(C(CC(=O)OC)=O)CCCC2)C)nsc2ccccc12 c1(CNCCC2(C)CC2(Cl)Cl)ccc([N+](=O)[O-])s1 C(C)(CCCC(=O)NC(CC)(CC)C(C)C)NC(C1C(=C)C1)=O C1(COCC(=O)NCCN(C(=O)CSc2nc[nH]n2)C)CC2CC1C2 C(=O)(C1CCc2c(Cl)cccc21)NC1CCN(C(C2CC(C)(F)C2)=O)C1 c1(C(c2nnnn2C)Nc2c(C)nn(C)c2C)ccc2oc3ccccc3c2c1 c1(NCCOc2cccc(C#N)c2)nccc(=NCC2CCCC2N(C)C)[nH]1 c1(C(=O)NC2C(C(=O)Nc3nccc(C(C)C)c3)CCC2)c(F)cncc1Br Cc1cncc(C=CC(=O)NCC(C)CNC(c2cnccc2C(F)F)=O)c1 c1(CC)cnoc1C(=O)NC(C)CCCNC(=O)C=Cc1ccsc1 C1(C(C2CC2)=O)(CN(S(=O)(=O)CC2CC3(C2)CC3F)CC)CCCCC1 C1(CNC(C(F)=C(C)C)=O)CN(C(C23CC2COC3(C)C)=O)CC12CC2 C1(O)(C)CCOCC1.C1(C(=O)N)CCOCC1NC(C1CC1C(F)F)=O C1(NC(C2C(=C)C2)=O)CCCN(C(=O)CC(C)(O)c2ccccc2)C1 Cc1cc(C(F)F)oc1C(=O)NC(C)CCNC(=O)CC1COCCN1C N1(C(C2N(CCC)CCC2)=O)CC2CCCC2(NC(c2ccc(CF)cc2)=O)C1 N1(C(C(C(C)C)C)=O)CC(NC(c2cc3sccc3cn2)=O)CCC(O)C1 C(=O)(C(C)C(F)(F)F)NC(C)CCCNC(C1(C(F)F)CC1)=O C12(NC(CS(=O)(=O)NC)=O)CCC(CN(C(C34CCCC3C4(F)F)=O)C1)C2 O=C(C1CSc2ccccc21)NCCCCNC(c1nccc2ccsc12)=O C1(OC)(CNC(C2CN(C(=O)Cc3c(C)cnn3C)C2)=O)CC(C)(CO)C1 C1(C(N2CC(OCCNC(C(C)n3cnnn3)=O)C2)=O)CC=CCC1C(N)=O c1(C(=O)NC(CNC(C(C(C)C)(C)C)=O)C(C)(C)C)nc2ncc(Br)cc2[nH]1 C1(OC)CN(C(=O)Cc2nocc2C)CC1NC(c1sc(CC2CC2)nc1C)=O S(=O)(=O)(c1ccc(Br)cn1)Nc1ncc(C(=O)OCC)s1.c12cc(Cl)ccc1S2 c1(C(N2CC(O)(C(C)NC(C=Cc3n(CC)ncc3)=O)C2)=O)cccc(C)c1Cl c1(C(=O)NC(C)(C)CCNC(C2(C)CC2(F)Cl)=O)cc(N)cnc1Cl c1(-c2ocnc2C(=O)NCC=CCOCC)cccc2ccccc12.C(=O)(C(C)O)N CCCCCCCCS(=O)(=O)N1CC2CN(C(c3cc(Br)cc(I)c3)=O)CC12 O=C1CCN(C(C2CCN(CC(F)(F)F)CC2)=O)CCC2CCCN12 CC1CCOCC1C(=O)NCc1cccc(NC(=O)Cn2cccnc2=O)c1 C1(n2cccn2)(C(=O)NCCCSCCNC(c2ccccc2)=O)CCCC1 C1(C(N2CCC(NC(CSCC#C)=O)C(CO)C2)=O)CC(=O)C12CCCC2 N1(C(C(c2ccc(OC)c(Cl)c2)(F)F)=O)CCNC(=O)c2cc(Cl)ccc21 CC1C(C)N(C(=O)Cc2cncnc2)CCN1C(c1cnn(C)c1N)=O CC(C(C)C(=O)NC1C=CCN(C(c2ccc(F)cn2)=O)C1)S(C)(=O)=O C1(CNC(C23CC(C(=O)Nc4cccc(F)n4)(C2)C3)=O)CCC2CC2C1 N1(C(C2(C)CCC(=O)N2)=O)CC2CCC(C1)N2Cc1ccn(-c2ccccc2)n1 N1(c2cc(NCC3(CCC)CC3)ncn2)CCC(Cc2ccccc2)C(C)C1 c1(C(=O)NC(C(C)C)C(C)NC(C2C3CCC2CC3)=O)ccc2ccoc2c1 Cn1ccc(C(=O)N(C2CC2)CC2CCCN2C(=O)C=CC(F)(F)F)cc1=O c1(CC(=O)NCC2N(C(CC=C)=O)CC(OC)C2)cc(OC)c2c(c1)CCO2 N1(C(c2cc(Br)cs2)=O)CCOCC1Cc1cn(Cc2ncccn2)nn1 C1(NC(CCCOCC)=O)CN(C(C2(SC)CC2)=O)CC1C c1(C(=O)NC(C(C)C)CCNC(=O)CCS(C)(=O)=O)cc2c(cc1N)OCCO2 CC(O)C(C(N)=O)N(CC(C)O)C(=O)COC(C)(C)C c1(C(=O)NC2C(NC(C3C(C(N)=O)C3)=O)CCC2)cccc(C(F)(F)F)c1 C(N=c1nc(N2CCc3nc[nH]c(=N)c3C2)c2[nH]ccc2[nH]1)C1(SCC)CC1 CCC(C)CC(C)C(=O)N1CC2CC1(C(N1CCC(CC3CC3)CC1)=O)C2 N1(C(c2c(CC)ccs2)=O)C2CCC1CN(CCN1CCCCC1=O)CC2 CCCC(O)C(CO)NC(=O)C(C)N(C(=O)C(C1CCCCC1)C)C1CC1 N1(C(C2CSCCN2C(c2cnccn2)=O)=O)C2CCC1COC2 c1(C(N2C3CN(C(CC(C(C)C)C)=O)C(C3)C2)=O)ccc2cncn2c1 C1(CCCNC(C=C(COC)C)=O)CCCCN1C(C1CCCCC1O)=O Cc1ccnnc1C(=O)NCCC1CN(C(=O)Cc2nonc2C)CC1C N1(C(C2(C)C(CC)CCC2)=O)CC(C(=O)NCC2(C)CCCN(C)C2)C2(CCC2)C1 S(=O)(=O)(c1cnn2ccc(N(CC(F)F)C)nc12)N(CC)CC1CCSCC1 C(CSC)(C(=O)NCCC1CN(C(=O)C(c2ccccn2)O)C1)OC C(=O)(C1=C(F)CN(C(C2CNC(=O)C2)=O)CC1)NC1C(C#N)CCCC1 N1(C(CN(C(C)=O)C)=O)CCC(C)(CNC(c2ccc(C(F)(F)F)nc2)=O)CC1 C1(C(=O)NCC2CC(NC(c3cc(C)c(F)nc3)=O)C2)CCc2nn[nH]c2C1 C(CC(C)C(=O)N(C)CCNC(c1ccc(-c2cnn(C)c2)o1)=O)=CCC C1(C(=O)NC(CO)CCO)CN(C(=O)C=Cc2cc[nH]c2)CC1F c1(C(=O)NC2(C)CC(NC(c3csc(C(F)(F)F)c3)=O)C2)cc2n(n1)CCCC2 C12(C)CCCN(C1)C2=O.Cc1nccn1CCCC(=O)NCCS(C)(=O)=O c1(C(C)=O)ccccc1C(=O)NC1CCCC1NC(=O)C(C)(C)c1ccnn1C n1(CC)nc(C)c([N+](=O)[O-])c1NCC(C)NC(c1cc(C(F)F)n(C)n1)=O c1(OC)cc(N(C2CC3CNC2C3)C)c(Br)cn1.c12cccc(OC)c1OC2=O C(CC(O)C(=O)N1CC(C2CCCN2C)C1)NC(C(C)c1ccco1)=O CC1CC(C(=O)NCC(O)C(F)F)CN(C(=O)CNC(=O)NC2CC2)C1 N1(C(c2cnc(CC)[nH]2)=O)CCC2C(CCN2C(=O)CC=Cc2ccccc2)C1 CC1(C)COCCC1C(N1CCC(NC(C2CC3(C2)CC32CC2)=O)CC1)=O c1(C(N2CC(CN(C(=O)CCSc3n[nH]c(=N)s3)C)C2)=O)n[nH]c2c1COCC2 CCC(CC)(CC)C(=O)N1CCC(CF)(NC(c2ccc3nc[nH]c3n2)=O)C1 N1(C(CNC(CC)=O)=O)CCN(C(=O)C(c2cnccc2C)(C)C)C(CCO)C1 C1(O)(CN(C(C2(N(C(C(C)n3cccc3)=O)C3CC3)CCC2)=O)C)CCOC1 N1(Cc2n[nH]c(C)c2Br)CC(C)NC(=O)C12CC2.N12CCC(CC1)C2=O C(C(C)C(F)C(=O)NOCCC(C)C)NC(c1c(CC)nns1)=O C1(C(=O)Nc2ccc(-c3c(C)ncs3)cc2)CCc2nncn2C1 CC1CN(C(=O)C(F)C2CCCC2)CC1CNC(=O)CCCOc1ccccc1 C1(NC(C=CC(C)C)=O)CCN(C(=O)CCC2CCC(=O)N2)C12CC2 C1(NC(Cc2cc(C)c(F)cc2)=O)CC2CC(NC(=O)CC3(C)CC3)CC2C1 Cc1cccnc1CC(=O)NCCCNC(=O)C(C)n1cccn1 c1(OC)cccc(C(C)C(N2CCCC2CN(C(=O)C(C)OCC2CC2)C)=O)c1 c1(OC(C)=O)ccc(C(=O)NCC2(NC(=O)CN3CCSCC3)CC2)cc1 C1(OC)CS(=O)(=O)CC1NC(c1cnn(CCCl)c1)Cc1ccccc1 c1(OC)ccnc(C(=O)NC2(C)CCN(C(C3CCCS(=O)(=O)C3)=O)C2)c1C c1(NC(C(=O)N(CC(C)CNC(c2cscn2)=O)C)=O)ccccc1 C12CN(CC1C(c1ccccc1)CC)C(=O)CN1CC2C1.C(=O)(CNC(N)=O)NC N1(C(c2cn(CC(=O)NC)nn2)=O)CCCCC(NC(c2cnc(C3CC3)s2)=O)C1 C1(C)(C(N(CC(C)NC(C2(C3CCCO3)CCOCC2)=O)C)=O)CCCCO1 CC1CC=CCC1C(N1CCC(N(C(=O)CCNC(=O)C(C)(C)C)CCO)C1)=O N1(CC(=O)N(CC(C)N(C)C(c2ccc[nH]2)=O)C)CSCC1=O N1(C(C(CC=C)C)=O)CCC2(CC1)CC(NC(=O)CCNC(=O)COC)CCO2 C#CCC(CC(=O)NCc1nc(CC)cs1)NC(=O)CN(C)CCOC CC(C(=O)NCc1cn(CCN2CCCCCC2)nc1)C(F)(F)C(F)F C1(N(C)CC2CC2(C)C)CCC(c2cccc(OC(F)F)c2)CC1 C1(C)(CC)CC(C(=O)NCCCCCCNC(=O)C(C)CN(C)C)CCO1 N1(C(C(CC(C)C)O)=O)C2CCCC1CC(NC(c1cnn(C3CCC3)n1)=O)C2 C1(OC2CCN(C(C(C(C)SC)NC(=O)C(C)(C)NCC#N)=O)C2)CCN(C)CC1 c1(NC(C(=O)NCC2C(Sc3ccccc3)C2)=O)cc(C(=O)O)n2ccsc12 N1(C(C(C2CC2)SC)=O)CC2CC2(CNC(c2nc(C(F)(F)F)cn2C)=O)C1 c1(C(C)(C)C)nccc(=NCC2CN(C(C3COCCOC3)=O)CC23COC3)[nH]1 c1(C(C2CCN(C(=O)NC3CC(C)S(=O)(=O)CC3)C2)=O)ccc2c(c1)nnn2C C12CC(C(OC)C1)N2.C12(C(=O)OC)CC(C(=O)NC(c3ccsc3)COC)(C1)C2 c1(C(C)NCCC2CCN(C)C2=O)cccc2ccccc12 N1(C(c2cnn(C(C)C)c2C2CC2)=O)CCC(CNC(C2CC2(C)Br)=O)C(C)C1 N1(C(CC2CC(=C)C2)=O)CCCC(O)(CN(C(c2snnc2C)=O)C2CC2)CC1 C#Cc1ccccc1CCN1CC(CC(=C)Cl)C1 c1(C2CCN(C(c3n[nH]c(C)c3C)C)CC2)nc(O)c2cc(Cl)ccc2n1 CC(CN=c1nc(-c2ccccc2)[nH]c(=NC2CC2C(C)(C)C)[nH]1)C(C)(F)F N1(C(C(=Cc2ccco2)C)=O)CCC2(CCCC2NC(=O)CCC(C)(C)C)C1 C(=O)(CCCCCC(C)O)NC1CC2N(C(c3n(CC)nc(C)c3)=O)C(CC2)C1 N1(C(=O)OC(C)(C)C)CCC(Nc2cccc(O)c2[N+](=O)[O-])CS1(=O)=O [N-]=[N+]=NC1(C(N2CC3CC2CC3O)=O)CCN(C(=O)Cc2ccoc2)C1 c1(N2CCC(NC(C3(O)CCOCC3)C)C2)ncc2ncn(C)c2n1 Cc1nnc(C(C)NC(Cc2ccccc2)CC(C)C)nc1C C1(CNC(COCCSC)=O)CN(C(=O)Cc2ccnn2C)CC1(C)C NS(=O)(=O)CC(=O)NCC1CCCN(C(c2cn[nH]c2)=O)C1 c1(CC)ccc(C(=O)NC(C)(CNC(=O)C(c2ccc(C)s2)C)CC)cc1 CCCC(C(=O)NCC(C)(CC(C)C)NC(c1sc(C)nc1C)=O)C(C)C Cc1sc2ccccc2c1C(=O)NCC(C)N(C)C(c1cnc2cncn2c1)=O CCC(C)CCC(=O)N1CC(NC(=O)COc2c(C)cccc2Cl)C(C2CC2)C1 c1(CC)cc(C(=O)NC2CC3CC(NC(C4CC(SC)C4)=O)CC23)c(C)nn1 C(c1cn[nH]c1)=C(C)C(=O)N1CCC1C(=O)NC(C)COC(F)(F)F C(=O)(CC(C)(C)C(F)(F)F)Nc1c(CN(CC=C)C)cccc1 C1(NC(C(F)OC)=O)CCCN(C(=O)CC2CCN(CC(=O)OC(C)C)CC2)C1 N1(C(CCCOCCC)=O)CC(NC(C2OCC3CCCC23)=O)C2(CC2)C1 c1(C(N)=O)ccc(F)nc1NC(C1CN(C(=O)CCN2C(=O)C=CC2=O)CCO1)=O c1(OC)c[nH]c(Cn2cc(C(C)NC(=O)CC3(O)CCCN(C)C3)nn2)cc1=O C1(CNC(c2cc[n+]([O-])cc2)=O)(NC(C2CCCSS2)=O)CCCCC1 C1(NC(COC(CC)C)=O)CN(C(c2n[nH]c(C)c2C(F)(F)F)=O)CCC1(C)C C1(C(=O)NC23CC(CNC(C(CSC)C)=O)(C2)C3)CC2(CCO1)CC2 c1(C(=O)NC(CCC(C)C)CO)cc2c(s1)CCN(Cc1ccc(Br)c(Cl)c1Cl)C2 C1(O)(CC#C)CC(C(=O)NCC(C2CC2)NC(c2ccnn2CCC)=O)C1 C1(C(=O)NCC2CN(C(C(C)(C)F)=O)C2)C2Cc3cc(Cl)ccc3C12 C(=O)(C(C)CC=CCc1ccccc1)N(CCOCCN(C(C1C(C=C)C1)=O)C)C C(C(CNC(c1nc(=N)cc[nH]1)=O)C(F)(F)F)NC(C1N(CC)CCC1)=O C1(C(CNC(C=C(C)Cl)=O)F)CCN(C(c2cc(C(F)(F)F)on2)=O)CC1 C1(C#N)(C(=O)NC23CC(NC(C=C(CC)CC)=O)(C2)C3)C(C#N)C1(C)C C1(CC(=O)NCC(CNC(C(c2c(OC)cccc2)O)=O)C)CC(=O)NC(=O)C1 C(=O)(CCCC(=O)N1C(C(=O)NCCOc2ncccn2)CCC1C)OCC c1(OCC)ccc(C(=O)NC2CCN(C(=O)C=C(CC)CC)C2C)cn1 c1(C(=O)NCCC2(O)CN(C(c3cc(N)c(Cl)cc3)=O)C2)cc(F)c(O)c(F)c1 S(=O)(=O)(c1ccc(Cl)cn1)N1CC(CC(N2CCOC3(CC3)C2)=O)OCC1 CC1(C)CC(NC(=O)CCCCO)CN1C(=O)CSCC1CCCO1 Cc1nc(C)n(C2CCCN(C(=O)Nc3cc(N4CCCC4)ncn3)C2)n1 C=C(C)C1OCCC1C(N1CCC(C(N2CCCC2(C)COC)=O)(CC)CC1)=O CCC(CC(=O)N1CCC(C)CC1C(=O)NCC1CC2(CC2)C1)C(F)F N1(C(c2n(CC=C)ccc2)=O)CCCC(CC(=O)NC2CCCC2C)C1 C1(C(=O)NCCC2(OC)CN(C(=O)C(C)(O)C(C)C)C2)CCc2ccccc2O1 c12ncnc3sc(cc13)c(=O)[nH]2.n1(CC)cc(CN2CCCC2CO)cn1 c1(OC)cc(CC(N2CC3C(C(=O)NC4(C(C)C)CCC4)C3C2)=O)ccc1O c1(C(CNC(CCC=C)=O)NC(=O)Cc2nnc(C)s2)ccccc1OC C1(OC)CN(C(c2ccc(C)[nH]2)=O)CCC1NC(c1ccc(-n2ccnc2)cc1)=O c1(OCC(=O)NCC2CCCN(C(=O)CCn3cccn3)C2)cccc(Cl)c1 CC1(C)CCC(CNC(c2ccc(F)o2)=O)N(C(c2c[nH]nc2C(F)F)=O)C1 C(N=c1[nH]nc(C(C)(C)C)s1)C1CC(C)N(C(c2cnoc2)=O)C1 C12(NC(c3c(C)ccc(C)n3)=O)CC3CCC(C1C2)N3C(c1ccnc(C)c1)=O C1(C(C)C)CC2CCC(C1)N2C(=O)NCC(CO)N(C)C c1(C(N(C2CN(C(C3CCC(C)(C)OC3)=O)C2)C)=O)cncc2ccc(F)cc12 N1(C(C(CCC)NC(N)=O)=O)C2CCC1CC(NC(C1OCC1(C)C)=O)C2 c1(OC)ccc(C#N)c(NC(C2CC2C(=O)Nc2ccccc2F)=O)c1 CC1(CNC(=O)C(F)(F)CO)CN(C(c2ccc(C(N)=O)cc2)=O)CCO1 c1(SCCCOC)cccc(C(=O)Nc2cccc(-c3nc(C)cs3)c2)c1 C(=O)(C1CCCn2nccc21)NC1(CF)CCN(C(C(CC)COC)=O)C1 C1(C(=O)NCCC2CC(NC(C(CCC)C)=O)C2)CSc2ccccc2O1 CC(C)(C)C1=NOC(C(N2CC(CNC(c3ccsc3)=O)C3(CCC3)C2)=O)C1 c1(C(=O)NCC2(CC3CC3)CC2)cc(C(=O)Nc2nncn2C2CC2)on1 N1(C(c2cc(I)cn2C)C(=O)Nc2c(OC)cccc2)CCn2c(nc(C)c2C)C1 CCCC(CCCNC(=O)C(Oc1ccc[n+]([O-])c1)OC)NC(C1CN(C)C1)=O C=C=C(C)CC(=O)NC1CCCN(C(C2CCCN2C2CCCC2)=O)C1 C12(C(=O)NC(C(=O)NCC(CC)C)CC)CCN(CC1)CC2 c1(C(=O)NCC(CO)NC(C2CC2c2cccnc2)=O)nn(C2CC2)cc1Cl CN1CCC2(CCN2C(=O)CC(C(F)F)NC(=O)Cc2cnnn2C)C1 C1(CNC(c2c(C)snn2)=O)CC2(CCN(C(c3cccc(CO)c3)=O)CC2)C1 C1(C(=O)NC2CC(CCNC(c3cccc(CCC)c3)=O)C2)CC(=O)C12CCC2 CC1CN(C(c2csc(CNC(=O)CC3CCCC4CC34)c2)=O)C(C)C1C c1(C(N2C(CN(C(=O)Cc3nc[nH]n3)C)CCCC2)=O)cc2n(n1)C(C)CCC2 C(=O)(C(C(F)(F)F)=CC(C#N)C(=O)OC)N(C)CCNC(=O)CCSC1CC1 C(=O)(C1=NN2CCCN=C2N1)NC(C(C)C)C(C)NC(=O)CCC1CCOC1 c1(C(N2CCCC(CC(=O)NC(c3cnc[nH]3)C)C2)=O)cc(Cl)ccc1Cl c1(C(C(=O)N(c2cc(C)ccn2)CC)Sc2cccnc2)cccc(C)c1 CCCCCCCCOCC(=O)NCC1COCCN1C(=O)CC1(C)CCCO1 c1(C(N2CCN(CC(C)(C)NC(C=COCC)=O)CC2)=O)cc(Cl)c(F)c(Cl)c1 C1(O)(C(=O)NCCN(CCCN(C)C)C(=O)CC2COCCO2)CCCCC1 c1(C(=O)NC2(C)CC(NC(C(CO)OC)=O)C2)cc(NC(C)=O)ccc1Cl c1(C(N2CC3C(C(=O)NCC(C)(C)CO)C3C2)=O)cncc2ccccc12 CC1CC(C(=O)NCC(C)(F)CNC(c2cc(C3CCC3)[nH]n2)=O)CC(=O)N1 c1(C(N2C(C(=O)NCc3nc(C)sc3)CC(O)C2)=O)ccc2c(c1)OCCO2 C1(O)(C(C)NC(CC=CC=C)=O)CCN(C(=O)CCC(C)C)CC1 C#CCC(C)(CNC(=O)COC1CCN(C(c2cnco2)=O)C1)CO CC1CN(C(C2CCCN2C)=O)CCCN1C(=O)CCCNC(N)=O c1(OC)c(C(=O)NCCC(C)(C)NC(=O)Cc2cccc(F)c2Cl)ccnc1Cl Cc1cnc2c(C(=O)NC3CC(CNC(C4(C)CC4)=O)C(O)C3)cnn2c1 c1(OC)ccc2c(c1)C(C(=O)NC1CC3(CN(C(C)=O)C3)OC1)C(C)N2 CN1C(=O)CSC1=CC(=O)N1CCCOC(CNC(=O)CC2CC=CCN2C)C1 S(=O)(=O)(c1ccc(Nc2cccn2C)c(Br)c1)NN(CCOCCC=C)C C(C)(C1OCCc2ccccc21)c1nnc(-c2occ(C)c2C)n1C CCN(OC)C(=O)CNC(=O)CC1CC(C)(C)CN1C(c1n[nH]c(C)c1O)=O c1(CCC(N2CCC(F)(CNC(C(CCC)(C)O)=O)C2)=O)ccc2ncsc2c1 C#CCC(CC#C)C(=O)NC1(C)CC(NC(=O)CN(S(C)(=O)=O)C)C1 Cc1ccc2c(c1)CN(C(C1CCCC1NCc1cnn3cccnc13)=O)CC2 C1(NC(c2c(CC)cno2)=O)CCC(CNC(=O)C(C)OCCC(C)C)CC1 C1(CNC(CCc2nc(C)c(C)o2)=O)CN(C(=O)CC2(C#N)CC2)CCC1(C)C N1(C(CCC(C)O)=O)CCC2(CCCCN(C(C3(CO)CCC3)=O)C2)C1 Cc1nc2n(n1)CC(C(=O)N(CCNC(c1coc(C#N)c1)=O)C(C)C)CC2 c1(C(=O)OCC(=O)N(CC#C)CC=C)cn2cc(Cl)ccc2n1 C1(NC(=O)CC2CCCCC23CC3)CCN(c2nccnc2F)CCC1CO c1(CCCNC(C)(C)CNC(=O)NCCC2CC(F)C2)ccccc1F N1(C(c2c[nH]c(=NC)o2)=O)CCN(C(=O)CC2CC3CCC2O3)C(C)C1 C1(C(N2CC(CCC)C2)=O)CCC(C)(C)N(C(C2CC2Cl)=O)C1 CCC(C)CC(C(=O)NCC(C(C)C)C(C)C)NC(=O)CC1CCCC(=O)C1 c1(C(=O)NCC(C2CC2)NC(CC2CCC(C)O2)=O)cccc(C2(C#N)CC2)c1 C1(NC(=O)CC2CCOC2)CN(C(c2cocn2)=O)C2(CCCCC2)C1 C(CCCCNC(=O)Cc1cncs1)N(C(=O)CCN1CCOCC1)C(C)C c1(CC(=O)NCC(CC)NC(C2CC=CCC2)=O)c(F)ccc(Cl)c1F c1(N)cc(C)ccc1[N+](=O)[O-].C12CCN(CC1)CCN2C(C12CC(C)(CO1)C2)=O.CO C1(C(=O)NCCCC(CO)NC(CC(C)(C)O)=O)CCC(=C(F)F)CC1 C(=O)(C1CCc2nccn21)NC(C1CCN(C(c2c(CC)noc2)=O)C1)C c1(COC)ccc(C(=O)NCCN(C(c2ccc(CO)[nH]2)=O)C(C)C)c(OC)c1 C(=O)(C1=CC2CC=CCC12)N(C1CCCCCC1)CC C1(NC(C2C(NC(c3ccc4ccoc4c3)=O)CC2)=O)CCC2(CCC2)CC1 C1(C(N(C(C(C)C)CO)C)=O)CC(F)CCN1C(c1cc(O)n(C)n1)=O c1(C(N(C2CN(C(CC(CC)C)=O)C2)C)=O)[nH]nc2ncc(Br)cc12 S(=O)(=O)(c1ccc(C#N)c(NCC2CCCO2)c1)N1CCCC(CC)(CC)C1 Cc1nc2n(n1)CCN(C(=O)CCNC(c1cc(Cl)n(C)n1)=O)C2 n1(C(CC)C)ncc(C(=O)NC(C)CCNC(c2cccc(F)n2)=O)c1C C(=O)(CC(C)CC(C)C)N(CCC)CCNC(=O)CCc1nc(CC)[nH]n1 c1(C(=O)NCC2CN(C(C(C)N(C)C)=O)CC2(F)F)cccc2nc[nH]c12 C1(CN(C)C(C2CCC(c3ccccc3)O2)=O)C=NN(C)C1=O Cc1ccc(CN=c2ccnc(N(C)CC3COC(=O)O3)[nH]2)cc1C#N C1(C(=O)NC(C)CCNC(=O)CCCc2cnccn2)CCCCN1S(C)(=O)=O N1(C(CCCN(C)C)=O)CCC2(CCCN2C(=O)CC2CC(O)C2(C)C)CC1 c1(COC(c2cccc(SCCC)c2)=O)cc(S(N)(=O)=O)ccc1Cl N1(C(CNC(=O)OCC)=O)CCC2(CCCC2N2CCC(C)(N(C)C)CC2)CC1 c1(C(N2CC(NC(C(C)(C)OC)=O)C(N3CCOCC3)C2)=O)ccnc(C)c1C C1(COC)(CNC(=O)CN2OC(C)CC2=O)CCN(C(=O)C(COC)N(C)C)C1 c1(C(N2CCC(CN3CCCCCC3)CC2)=O)cc2c(s1)CCC2=O N1CCCC2(C1)CC=C(C(CC)CS(=O)(=O)O)C1C2(O)COC1.C=O N1(C(CC(=O)NCC2CC2)=O)CCC2(CO)CN(C(=O)CC3CSC3)CC2C1 CCCCC(O)C(=O)N1CCC(NC(=O)C=CCN2CCC2)C(C(C)C)C1 c1(C(C)NC(c2cn(-c3cccc(Cl)c3)cn2)=O)ncccc1Br N1(C(c2ncn(C(C)C)n2)=O)CC(CNC(=O)Cc2cnoc2)OC2(CCC2)C1 C1(N(C(CSCCC)=O)C)CC2CC1N(C(C1CCCC(C)(C)C1)=O)C2 c1(CC(=O)NCC2(NC(CCC(=O)c3ccc(C)s3)=O)CC2)c[nH]c2ccccc12 C1(CCNC(c2cc(C)n(C)c2)=O)CC(F)(F)CN1C(=O)C(C)C1CCC1 Cc1nn(CC(=O)N(C2CCC(NC(=O)CS(C)(=O)=O)C2)C)cc1[N+](=O)[O-] c1(NCC(c2ccc(F)cc2)NC(CS(CC)(=O)=O)=O)snc(Cl)c1C#N C1(CNC(C2(NC(CCCOC(C)=O)=O)CC(F)(F)C2)=O)CCCCC(=O)N1 C(N=c1[nH]c(=NC)[nH]c(=NCc2cccc3c2NC(=O)CO3)[nH]1)C1N(CC)CCC1 N1(C(C(C)SCC)=O)CCOC2CN(C(c3csc(C(=O)OCC)n3)=O)CC12 N1(C(c2ccc(C)o2)=O)CCN(C(=O)C2=C(Cl)CCOC2)C(C)CC1C c1(N2CCC(NC(C(CCCC)O)=O)C(F)C2)ncnc2c(Br)nn(C)c12 C#Cc1ccc(C(=O)NC(C)C(C)C(=O)NC(C)(CC(C)C)C(N)=O)c(C)c1 C1(CC)(NC(=O)CC2CC(CF)C2)CCN(C(C2CC2(F)Cl)=O)CC1 C1(C(=O)NCCC(=O)OC)CC(O)CN1C(C1CCCN1C=O)=O C(=O)(C1=NOC2(CCC2)C1)NC(c1ccccc1)C(=O)N(C1CCN(C2CC2)C1)C CCCC(O)CC(=O)NC(CNC(c1cc(C2CC2)nn1CC)=O)CCOC C1(C(=O)NC(C)C(C)NC(c2csc(C3CC3)n2)=O)OCCOC1(C)C c1(C(N2CCC(C)(NC(CCCC#C)=O)C2)=O)nn(CC)c(=O)c2ccccc12 c1(OC)cc(F)c(S(=O)(=O)N(CC(C)(C)O)C)cc1Br N1(C(c2n(CC)nc(C)c2)=O)CCC2(C=C(C(=O)NCCSCCO)C2)C1 C1(CNC(c2ccn(C3CC3)n2)=O)COCCN1C(c1cncs1)=O Cc1cc(C(=O)NCC2CCCN2C(=O)COCc2ccnn2C)ccc1F C1(C(CNC(C(C)N(CC)CC)=O)(C)C)CCN(C(C2CCC(=O)N2C)=O)CC1 N1(C(C2(SC)CC2)=O)CCC(CCNC(=O)CSc2nnnn2C(C)(C)C)C1 Cc1nc(C(=O)NC2CCN(C(=O)CCC3(C)CC3)C2C(C)C)cn1C N1(C(C(Cn2cccn2)NC(CCSC)=O)=O)CCc2n[nH]cc2C1 N1(C(Cc2cc(C)c(Br)cn2)=O)CC2(CNC(=O)N2C)C1 c1(OC)cc(C(N2CC(COC)CC2CNC(=O)C(C)(C)C2CCC2)=O)ncn1 C(C)(C)(CCCNC(=O)Cc1cncc(O)c1)NC(CCOCCOC)=O Cc1cc(C(N2CC=CC(C(N3CC(CO)CC3CO)=O)C2)=O)c(C)cn1 c1(OCC(=O)NCC(C)CNC(=O)C(C)N2CCC2)cccnc1 c1(OC)noc(C2CC2)c1C(=O)N(CC(C)CNC(c1ccnc(S)c1)=O)C C=C1CC(C(=O)NC(C(O)CO)C2CC2)(CNC(C2CC=CCC2)=O)C1 N1(C(C(CCC)CC)=O)CCC(NC(c2ccn3nccc3n2)=O)C(C)(C)C1 C1(CNC(COCc2cc(C)on2)=O)CN(C(=O)CC#N)C2CCN1C2 CCCCC(CNC(=O)C=Cc1cnc[nH]1)NC(c1cc(Cl)c(Br)[nH]1)=O Cc1c(C(=O)NC2(CO)CCN(C(=O)C(C)O)CC2)oc(=O)c2ccccc12 Cc1cc(C(N2CC(NC(c3c(C)noc3C(F)(F)F)=O)C(C)C2)=O)cc(Cl)n1 c1(C(N2CC(C(=O)OC)C2)=O)n[nH]cc1CNC(=O)CC1CC1(C)C C1(NC(c2c(C)c[nH]n2)=O)CCN(C(c2ccnc(C3CC3)n2)=O)CC1(C)C C12(C(=O)NCC3N(C(Cc4nnc(C)o4)=O)CC=C3)CCC(O)(CC1)CC2 CC(CS(C)=O)C(=O)NCCCCCCN(C)C(c1cnc(O)c(Cl)c1)=O C1(c2ccccc2)(C(N2C(C)CSC2)=O)CC2(COC2)C1 N1(C(C2C(C(C)=O)C2(C)C)=O)CCN(C(C2CCCC3CC23)=O)CC1C c1(OC)cccc(C)c1-c1ccc(CNC(C2CCN(CC(F)(F)F)C2=O)=O)nc1 C(=O)(C(F)(F)CCn1cccn1)NCC1(C(C)NC(C2(C)CC=CCC2)=O)CCC1 C1(C(N2CCCC2CNC(=O)CC2CCC(=O)C2C)=O)(CC)CC(F)(F)C1 N1(C(CSC)=O)CC2(C1)C(NC(=O)CC1CCS(=O)(=O)C1)CCS2(=O)=O N1(C=O)CCC2COCC2C1.CC(C)C(C(=O)NC(N1CCCC(N)C1)=O)C1CC1 C1(NC(CCCC)=O)CC(NC(=O)C(C)Cc2c(C)noc2C)C(O)C1 C=CC(C(=O)NC(c1cccnc1)C(=O)NCCN(CC)CC1CCCC1)OC N1(C(C(C)(C)N2CCCCC2)=O)CCCC(O)(CNC(=O)COC(=O)CO)C1 O=C(CCN=c1[nH]ccs1)NC1(CCNC(C2CCO2)=O)CCC(F)(F)CC1 C1(O)(C(C)NC(CSCC=C)=O)CCN(C(c2cncc(OC)n2)=O)C1 C1(NC(C(COCC)C)=O)CCC(NC(=O)Cc2ccc(C(F)(F)F)nc2)CC1 N1(C(C2(C3CC3)CN(C(C3(COCC)CC3)=O)C2)=O)CCC2OCCC2C1 C1(C(=O)NC2CCN(C(c3n(OC)cnc3C)=O)C2)CCC2(CC1)CNC(=O)C2 N1(CC(=O)Nc2onc(-c3ccc(=NC)[nH]c3)n2)C(=O)C(=O)N(C)C1=O C12(C(N(C(C)CCNC(=O)CCCCc3ccccc3O)C)=O)CCC(F)(CC1)C2 N1(C(C2(OC)CCN(C(=O)C(C)n3cccc3)C2)=O)CCC(O)C(CO)C1 C(C(C1CCCC1)NC(=O)C1=CCSC1)(C(C)C)NC(C(=Cc1cnc[nH]1)C)=O C1(CCC)CN(C(c2cncc(F)c2)=O)CCN1C(c1ccnc(CO)c1)=O C1(CC)C(NC(=O)CCSc2cccc(N(C)C)c2)CCCN1C(=O)C(C)SC N1(C(CCCn2cc(C3C(C)(C)C3)nn2)=O)CCC(F)(C(=O)NC=O)CC1 CN1CC(O)CC1C(=O)NC1CC(NC(c2ncc(Cl)s2)=O)C1 C1(CC)CCCC1N=c1nc2sccc2c(NCc2nc(C(C)(C)C)cs2)[nH]1 C1(CN(C)C(C2CCC(=O)O2)=O)CCN(C(c2ccnn2CC2CCC2)=O)CC1 c1(C(=O)NCC(C)(C)OCC(=O)NCCC2CCOCC2)cccc2cncn12 C(c1cccs1)=C(C)C(=O)NCCC1CC(NC(C2CC(C(F)(F)F)CO2)=O)C1 C1(CNC(=O)Cc2cc(-c3ccccc3)on2)COCCN(c2cc(O)ncn2)C1 Cc1cc(=NCC2(CCN(C)C)CCC2)[nH]c(=NCc2cnn[nH]2)[nH]1 c1(CC)nn(C)c(C(N2CC(C)N(C(C)C(=O)NCCC3CC3)C(C)C2)=O)c1Cl c1(OCC(=O)N(C)CC2(NC(CC3CC(OC)C3)=O)CC2)ccccc1Br N1(C(C(C)OCCC#C)=O)CCC(C2CC2)(NC(=O)COc2cccc(F)c2)C1 CCCCCC(O)C(=O)NC(C1(CNC(c2cn(C)c(=O)c(C)n2)=O)CC1)C c1(OC)ccc(C(=O)NC(C2CN(C(=O)C=Cc3cn(C)nn3)CCO2)C)nc1 N1(c2ncc(OCC)cn2)CCN(Cc2cnc(Br)s2)C(C)C1 C(=O)(C1CCC(=O)c2cccn21)NC(C1CCN(C(C2CCC(=O)N2)=O)CC1)C N12CCCC(COC)(C1)C2=O.C1(CCC)(NC(C2CC2COC)=O)CCNC1=O c1(C(=O)NCC23CC2CN(C(c2ncc(F)cn2)=O)C3)ccnc2nccn12 C=CCC(C)(C)CC(=O)NC1CC(O)C1CC(N1CCNC(=O)C1CC)=O C(=O)(C(C)Cc1ccco1)NC(CC)CNC(=O)CNC(=O)NC1CC1 c1(CNC(C(=O)Nc2n(C)nc(-c3ccccc3)c2)=O)ccc(F)cc1O c1(C(=O)NCCN(C(C(C2CCOCC2)OC)=O)C(C)C)oc(C2CC2)nc1C C12(NC(c3n(C)cc(C(F)(F)F)n3)=O)CCCC1N(C(c1ccsn1)=O)CC2 Cc1ncccc1CCC(=O)NCCC(C)(C)CNC(=O)Cc1ccc(Cl)cn1 C(=O)(C(C(C)C)C(C)C)N1CCC(OCCNC(C=Cc2c(C)cccc2)=O)C1 c1(CC)ccc(OC(C)C(N2CC3CC2C3NC(=O)CCCCN(C)C)=O)cc1 CC(C)CC(C(=O)N1CCCOC(CNC(C2CSC2)=O)C1)C(N)=O c1(C(=O)NC(CC2CN(C(C=CC)=O)C2)C)cc(F)c(CO)c(F)c1 c1(C(=O)NCCC2(NC(=O)C(Cl)=CCl)CC2)c(Cl)ccc2ccncc12 C1(C)(C(=O)NC2(CC=C)CC2)CC(O)CN1C(C1CC(C)(C)CN1C)=O Cc1ccc(CC(=O)OC2CC(F)(F)C2C)c(F)c1F CC1CC(NC(=O)CNC(=O)C2CC2)CN(C(c2occ3c2CCC3)=O)C1 C1(C(=O)NCC(=O)NCc2nccn3nccc23)C2Cc3ccccc3C12 CON(CCC(=O)Nc1cc(C)cc(F)c1)C(=O)C(C)NC=O c1(C(N2CC(NC(=O)C=Cc3cccs3)C2)=O)cccc2c(O)ncnc12 N1(C(c2nc(C)oc2)=O)CCCN(C(C23CC(CCO2)C3)=O)C(C)C1 c1(OC(C(=O)NCC(CC)NC(=O)C=C(C)C)CC)ccc(Cl)c(C)c1 N1(C(c2c(C)ccnc2C)=O)CCC2C(CCCN2C(c2cn(C)cc2C)=O)C1 N1(C(c2c(C)ccc(F)c2)=O)CCc2cc(CN(S(=O)(=O)CCCl)C)ccc2C1 N1(C=O)CCC(C2CCCN(C(C3(C4CC=CC4)CCC3)=O)CCC2)CC1 C1(CNC(CC(CN(C)C)O)=O)CC(C(C)(C)C)CN(C(C2(C)CC2)=O)C1 CC1CCC(CC(=O)NC2CC(NC(c3ccccc3NC(N)=O)=O)C2)CC1C N1(C(C23CC(C)C2C3)=O)CC2C(NC(=O)CC3C(C)(C)C3(C)C)C2C1 C1(CNC(CNC=O)=O)(NC(=O)CCc2nnc(C3CCCC3)o2)CCOC1 CC1CC(=O)NCC1C(=O)N(CCCOCCN(C(=O)C(C)(F)F)C)C C(=O)(C1(C)CC(=O)N(C)c2ccccc21)NCCCCCNC(C(C(C)C)C)=O c1(C(N2CC(C)(CCC(=O)NC(C3CCN(C)C3)CC)C2)=O)cccc(=O)n1O N1(C(C(C(C)(C)C)O)=O)CC(C(N2CC(O)CC2CO)=O)CC12CCC2 C1(C(=O)NC(C)CN(C(=O)CCCc2cccs2)C)CC(C(=O)OC(C)(C)C)=NO1 C=CC1CN(C(=O)COCc2scnc2C)CC1NC(c1ccnc(C)c1)=O c1(OC(C)C)ccc(C(=O)NC2CN(C(C3C=CCC3)=O)C(C)(C)C2)c(Cl)c1 N=c1[nH]c(C(N2CC=CC(NC(C3CCCC(F)(F)C3)=O)C2)=O)nc(=N)[nH]1 n1(CCC(N2CC(OCCNC(CNC(N)=O)=O)C2)=O)cc(Cl)cn1 C1(NC(C(C)c2cccs2)=O)CCSC12CN(C(=O)CC1CC3CC3C1)C2 N1(C(C(COCC)(C)C)=O)CC2(CCCCN2C(=O)C(C)=C(C)CC)C1 C(=O)(C(C(C)(C)C)N1CCOC1=O)Nc1nc(CC(=O)OCC)c(C)s1 N1(C(C(C)c2ccsc2)=O)CCC(C(=O)NCCC2(O)CCOC2)C1 C(=O)(N=c1[nH][nH]cc1I)N1CCN(C)C(c2cc(Cl)cc(Cl)c2)C1 CC(C)C(C(=O)NCc1ccn(CC(F)F)n1)N(C)C Cc1nc(NC(C2CCN(C(=O)CCC3CCC3)C2)C)c2ccsc2n1 Cn1cc(C(=O)NC2CCC(CCNC(C3(N4CCCC4)CC3)=O)C2)cn1 C1(C(=O)NC2CCC(CO)CC2)CC(O)CCN1C(=O)C1=C(Cl)CCC1 C1(NC(c2c(CC)nc(C)o2)=O)CCC2CCN(C(c3cccc(O)n3)=O)C1C2 C=CCC(C)(C)C(=O)N1CC2(C(=O)NCCc3ccccn3)CC1CO2 c1(CCC)ccccc1C(=O)OCC1CCN(C(=O)OC)C1 CC(=O)CCCCC(=O)N1CCCC1C=CC(=O)N(C)CCC1CC1 C1(C(C(=O)NC(C(=O)N(CC(C)(C)O)CCC)c2ccco2)O)CCCCC1 C(C)(C)(CC(C)N=c1ccnc(NC2C(C3CCCCCC3)C2)[nH]1)OC N#Cc1c[nH]c2ncnc(N3C4CN(Cc5ccc(-c6ccncc6)o5)CC34)c12 C1(CNC(c2csc3nnsc23)=O)(NC(C2CC2(F)F)=O)CCC(F)(F)CC1 c1(OC)cc(C(N2CCCCC(NC(C3(CF)CCC3)=O)C2)=O)cc(F)c1 c1(C(=O)NCC(=CC(=O)N(CC)CC2(O)CCC2)C)cc(C)ccc1O c1(C(=O)NC2CCCN(C(C(CC)O)=O)CC2)cc2cc(C)ccc2s1 c1(C(N2CCC(C(C)NC(c3scc(OCC)c3)=O)C2)=O)cc(CC)cc(C)c1 C(=O)(CCCCN=[N+]=[N-])NC(C)(CNC(c1csc(-c2nc[nH]n2)n1)=O)CO CC(CNC(=O)CN(C(=O)CCc1ccoc1)CC1CC1)CC1CCC1 N1(C(C2CN(C)C(=O)CC2)=O)CCCC2(CCN(C(=O)CCc3cnc[nH]3)C2)C1 Cc1ccc2occ(CC(c3nnc(N(C)C(C4CC4)C4CC4)n3C3CC3)O)c2c1.C C#CCCC(O)C(=O)N1CCC(NC(=O)CCCN=[N+]=[N-])C1c1ccccc1 c1(C(=O)NCC2(C)CCN(C(c3nc(C)[nH]n3)=O)C2)csc(N=S(C)(C)=O)n1 Cc1c(O)ccc(C(=O)NC2CC(C)(NC(=O)Cc3csc4cncn34)C2)c1C c1(C(=O)NC2CCCC(C(=O)NC(CC=C)CC)C2)nnc(O)nc1O N1(C(CC(C)CF)=O)CC2(CCN(C(c3ccnn3CCN(C)C)=O)CC2)C1 C(=O)(C(CCC)C(=O)OC)NC1CC(CNC(c2c(CC)cno2)=O)C1(C)C C(CC(C)C(=O)NCC1(NC(=O)CSc2nnnn2CCSC)CCC1)OC N1(C(CN=S(C)(C)=O)=O)CCC(C2CC2)C1CNC(=O)C1=CCCS1 C(=O)(C(CC1CCCCC1)NC(=O)CCc1cn(C2CCCC2)nn1)OC C12(C(=O)NCC(CC)NC(=O)C(C)c3cc[nH]n3)CCCCC(OC)(C1)C2 C12(C(N3CC(C#N)(F)C3)=O)CC(CN(C(=O)CCC3CCCO3)C1)C2 CCC(CC)(CN=c1[nH]c(C(C)C)nc(C)c1Br)NC(c1ccccc1SC)=O N1(c2nccc(C)n2)CCOC2(CCN(C(=O)CCC3CC3(C)C)CC2)C1 C(=O)(CC1=CCCCC1)NCC(c1ccc(OC)cc1)NC(c1cc(C)no1)=O CC1(NC(=O)CN2C(=O)CNC2=O)CCC(NC(C2(Cl)CC23CCC3)=O)CC1 N1(C(c2ccc(CC)[nH]2)=O)CCC(C(=O)N(C)C(c2ccccc2F)C)C(C)C1 c1(C(=O)NC(CCNC(c2c(C)n(C)cc2)=O)C)cnc2ccccc2c1 C1(O)(COC)CCCN(C(=O)C(C2(C)CC2)NC(=O)C(C2(O)CCCC2)F)C1 CC1CCN(C(c2ncnn2C)=O)CCN1C(=O)CCOCc1ccccc1 N1(c2nccc(OC)n2)CCN(C(c2cc(C(C)(C)C)[nH]c2C)=O)CC1C C(C(=O)N1CC2C(C(=O)NCC3CCCCC3)C2C1)(C(C)C)SC Cc1c(C(=O)Nc2cccc3ncsc23)ccc(Br)c1F.N12CCCC1C2=O C1(C(C)C(=O)N(C)CCOCCN(C(=O)COC2CC2)C)CCCOCC1 C#CC1(C(N2CCCC2CNC(=O)C(C(C)C)NS(N)(=O)=O)=O)CCCC1 Cc1cncc(C)c1C(=O)NCC1CCN(C(=O)CCCc2cccnc2)CC1 c1(-c2[nH]nc(C(=O)NNC(=O)c3cn[nH]c3)n2)ccc2cncn2c1 C1(CN(C)C(c2cccnn2)=O)CCCC(NC(c2cc(C3CC3)nn2C)=O)C1 c1(OC)cccc(C(=O)NOCc2cn(CC3CC4CCC3C4)nn2)c1 c1(OC)cc(F)cc(CN2CCCN(C(=O)C3CC3)CC2)c1N C(=O)(CS(=O)(=O)C1CC1)NCCN(CC)Cc1csnc1Cl C1(C(N2CCC(NC(CS(CC)(=O)=O)=O)C2(C)C)=O)CCCN(S(N)(=O)=O)C1 CC(C)(C)CC(=O)NNC(=O)NC1CCCCC1(C)C c1(C(=O)NCc2ccsc2C(N2CC(F)(F)C2C2CC2)=O)cc(F)ccc1Br c1(NC(=O)NC2CCC(CS(C)(=O)=O)CC2)ccc(Br)cc1-n1ccnn1 Nc1cc(C(N2CC=C(CNC(=O)CC(F)(F)F)CC2)=O)ncc1F CC1CN(C)C(=O)CN1N1CCC2(CC1)CN(Cc1cn(C)nc1Br)CCO2 CC(C)CCC(C(=O)NC1CN2CCCC1C2)NC(=O)CSC(F)(F)F c1(C(=O)NC2(CNC(=O)C=CCO)C(C)CCCC2)cccc2cccnc12 CC(CC(C)(C)C)C(=O)NCC(C1CC1)N(C)C(c1cnc(O)s1)=O C=CC1(C(=O)NCCN(C(=O)COc2cc(F)cc(F)c2)CC)CCCCC1 c1(OC)cnn(C)c1CNCc1c[nH]nc1-c1ccc(O)cc1 C1(CN(C(=O)C=Cc2ccn(C)c2)C)CN(C(=O)C(O)CC(N)=O)CC12CC2 c1(OC)cc(C(=O)N(CCC(C)(C)NC(c2c[nH]c(C(N)=O)c2)=O)C)sn1 c1(C(=O)NC(CNC(C=Cc2cn(C)nn2)=O)(C)CO)cc2ccncc2[nH]1 c1(OC)ccccc1CCC(=O)NCCCCCNC(c1onc(C)c1C)=O c1(C(=O)NC(CCCCNC(COCCCOC)=O)C)ccnc(Cl)c1Cl C1(C(=O)NC(C(C)(C)C)CNC(C2(C#N)CC3(CC3)C2)=O)CCc2cncn2C1 N1(C(C#CCNC(CC(CC)C)=O)=O)CCOC(C)CC1 N1(C(C2CN(CCC)C(=O)C2)=O)CCCC(C)(CNC(c2nnc(C)s2)=O)C1 N1(C(C2CCC(=C)CC2)=O)CCCCC1C1CCCN1C(=O)C=Cc1ccsc1 Cc1cc(CCC(=O)NC(C)CCCNC(C2(C)CCCC2C(C)C)=O)nn1C C(=O)(CCC(F)(F)F)NC(CN(C(C1(OC)CC(COC)C1)=O)C)(C)C c1(CN2C(C(=O)NCc3ccc(NC(C)=O)cc3)CC(F)C2)cc(Cl)cnc1Cl C1(C(=O)N(C)CC2(O)CCOC2)(CC)CCCN1C(=O)CC1CC(C)(C)CO1 c1(CC2C(=O)N2)ccccc1Br.C(C(F)(F)CO)NC(c1sccc1CO)=O C1(NC(CCNC(C)=O)=O)C=CCN(C(C23CC(OC(C)(C)C)(C2)C3)=O)C1 C(F)(C(=O)NCCC(C)NC(=O)CCSCC(F)(F)F)=CC CS(=O)C1(CNC(=O)COC2CCN(C(c3cscc3Cl)=O)C2)CC1 c1(C(N(C(C)CNC(C2(C)CC(C)(C)C2)=O)C)=O)ncn2c1CCC2 CON1CCC(C(=O)NCCC2CCCN(C(=O)Cn3cccc3)CC2)CC1 n1(CC(=O)NC2CN(C(CSC(C)(C)C)=O)CC2O)ncn2nccc2c1=O N1(CC(N2CCC(C)(NC(CC(=C)Br)=O)C2)=O)Cc2ccccc2OC1=O CCC(CC)C(C)C(=O)NC(C1CN(C(=O)Cc2ccccc2C(C)C)C1)C C(CCCCC(=O)NCc1ncon1)n1cc(CCC2C(C)C2)nn1 CC1CN(C(c2cc(Cl)c(Br)cn2)C(=O)NCCC2CC2)Cc2c[nH]nc21 C(c1cncnc1O)=CC(=O)NC(CNC(c1c(C)scn1)=O)(C)CO Cc1nccn1CCC(=O)NCC1CCC(NC(=O)C(C)CO)C1 N1(C(C2CC(C)(C)C2)=O)CCC2CN(C(C3(C)CCCC(F)(F)C3)=O)CC2CC1 C1(C)(NC(C)=O)CCN(C(=O)C(C)N(C(C23CCC(C2)OC3)=O)C2CC2)C1 C(=O)(C(C(C)Nc1ccc(CCC(=O)NC2CCOC2)cc1)C(C)C)OC c1(CC)cc(CNC(C2CC2)NC2CCC(C(C)O)C2)ccc1C C1(CC(=O)NCCC2(CNC(C(C)NC(=O)OC)=O)CCC2)COCCO1 C(=O)(C1=CNC2=NCCCC2=C1)NCC1C(C)CN(C(=O)CSc2cn[nH]c2)C1 C1(CNC(C2(NC(c3cc(C)on3)=O)CC(O)C2)=O)CCCCCC1 Cc1c(C(N2CC3(NC(c4cc(C(C)(C)C)no4)=O)CC2C3)=O)ccn1C c1(-c2c(C(=O)NC3CC(O)(CC(=O)OCC)C3(C)C)occ2)ccc(F)c(F)c1 c1(CC(N2CCC(CNC(C3CCC(OC)CC3)=O)C2)=O)ccc(F)c(Cl)c1F C1(C(NOCCCCCNC(C2CCCS2)=O)=O)(CC)CC2(CC2)C1 c1(C(=O)NC2CN(C(c3cc(CCC)on3)=O)C2)c(F)ccc(Cl)c1N N1(C(Cc2n(C(C)C)ccn2)=O)CCC(NC(=O)COc2ccon2)C1C1CC1 C(=O)(N1OC2CCC1CC2)C1(F)CCN(C(c2ccnc(O)c2)=O)C1 c1(C(=O)NCC2CN(C(CCSC)=O)CC2(C)C)cc(F)c2ccccc2c1 C(=O)(C#CC1(C)COC1)NC(C(=O)NCC(C(CC)CC)C)CO N1(C(C=CCCC)=O)Cc2ccccc2C(NC(=O)Cn2nnc(=O)[nH]2)C1 CC(CC(=O)NCC1CCN(C(=O)Cn2cnnn2)C1)P(C)(C)=O c1(CC)cc(C(=O)NC2CCC2CNC(c2cnn(C)c2)=O)ns1 C1(C(N2CC(C)(NC(c3cc[nH]c3C3CCCC3)=O)C2)=O)CCCC(F)(F)C1 C1(NC(c2cccnc2-n2ccnc2)=O)CN(C(=O)C=Cc2ccsc2)C2CC12 C(=O)(C1CCc2nccn21)N1CC2CN(C(c3cc(OC)c(F)cc3)=O)CC2C1 c1(C(N2C(c3cccc(C)c3)C(C)C2)C(=O)NC(C)(C)C)ccc(F)c(F)c1Br N1(Cc2ccc(OC)c(O)c2)CC2(CCCC2NCc2nnc(C(C)(C)C)s2)C1 C1(C(=O)NC2CC(C=C)C2)CN(C(C2CCN(C)C2=O)=O)CC1(C)C CC1CCC(CC(N2CC(C(C)NC(C34CCCN(CC3)C4)=O)C2)=O)CC1C N1(C(C2C(C(=O)OCC)C2)=O)CC2CC(C1)N(C(c1cnc(C3CCC3)s1)=O)C2 Cc1cccc(C(O)C(=O)NCC2CN(C(C3NC(=O)C4CC34)=O)C2)c1F C1(CC)(NC(c2ccc(C(F)(F)C(F)(F)F)nc2)=O)CCN(C(=O)C(C)O)CC1 C(N=c1nc(NC2CCNC2)c2c([nH]1)c(C)nn2C)c1cnn(CCC)c1C N1(C(c2c(CC)cno2)=O)CC(NC(=O)CC2(c3ccc(F)cc3)CC2)C(C)C1 c1(CC)cc2c(cc1NC(=O)C(=O)NC1(CC(F)F)CC1)OC(C)C2 c1(C(N2CCC(NC(C3CCCN(CC)C3)=O)C2C)=O)cc(C)c(C#N)cn1 CCCC(C(=O)N(C(C)CN(C)C(C1(COC)CCC1)=O)C)NC(N)=O c1(OC(C)C)ccc(S(=O)(=O)N2CCC(NC(C(CN(C)C)C)=O)CC2)cn1 C1(NC(=O)OC)CCN(C(=O)C(C)N(C)C(C2CC23CC3(F)F)=O)CC1 N1(C(C=CCCC)=O)CCC(C2CCN(C(c3ccnc4[nH]nnc34)=O)C2)C1 c1(C(=O)NCC2N(C(CC(=C)C)=O)CC=C2)cc(-c2ccccc2)oc1C CC1CCCCC1NC(C1CN(Cc2csc(Br)n2)C1)=O Cc1cccc(C(C(=O)NC(=O)NC2CCNC2=O)N(C)CC2CCCCC2)c1 c1(C(=O)NCCC(C)NC(=O)C(C)(C(F)F)c2ccccc2)cccc(Cl)c1N C1(CCC(=O)NC2CC(CO)CO2)CCCCN(C(c2cn(CCO)nn2)=O)C1 C(C(C)C(F)C(=O)NCC(C)(C)O)NC(C(C(C)C)SCC)=O Cn1cc(C2CC2C(=O)N(CCCNC(=O)C=CC2CC2)C2CC2)cn1 N1(C(CCSCCCC)=O)CCOC(C(C)NC(C2CCC2C)=O)C1 CC1(C)C(C(N2CCC(O)C2)=O)CCN1C(=O)C(=O)NC1CC1 C1(CCNC(c2cccc(SCC)c2)=O)CCN(C(=O)C2=COCC2)CC1(F)F C=CCCC(C)NC(c1sccc1CNC(C1CCCN1C(C)=O)=O)=O C(CC(C(C)C)NC(c1cc(N2CCCCC2)ccn1)=O)N(C(COC)=O)C N1(C(c2cn(CC)nc2)=O)CC(C)N(C(C23CCC(CC2)C3(C)C)=O)C(C)C1 CCCCC(C(=O)NC)NC(C1CN(C(C2(OC)CCCC2)=O)CC12CC2)=O N1(C(C23CC(C(C)C)(C2)C3)=O)CCC(C)N(C(c2csc(C(C)C)n2)=O)CC1 N1(C(c2ccnn2CC2CC2)=O)CCC2C(CCCN2C(c2ccns2)=O)C1 N1(C(c2c(C)nsc2N)=O)CCOCC(C(=O)N(C(C)CN(C)C)C)C1 CC(C)CC(CNC(c1cccc(I)c1)=O)NC(c1ccon1)=O Cc1cc2ccc(C(=O)NCC(C)(C)CCNC(C3(F)CC3)=O)cn2c1 C1(CCOCC(=O)NC2(C)CCC2)CCC2(CC1)CC2.C12(CC1)N(C)C2=O C=CCCN=C(NCC1(C(O)C(C)C)CC1)NCc1cccc(C(F)(F)F)c1 C1(O)(C(C)NC(c2cnc(C(F)F)s2)=O)CCN(C(=O)CCCC2CCC2)CC1 c1(OCC(=O)NCC(=O)NCCCC(C)C)cccc2c1OC(C)(C)C2 c1(OCC(=O)N(C2CCN(C(c3cc[nH]c3)=O)CC2)C)cccc(OC(F)F)c1 N1(C(=O)NC(c2ccccc2)CC#C)C2CCCC1CC(F)(F)C2 c1(C(C)C)csc(S(=O)(=O)N2CCC(c3cc(O)n(C)n3)CC2)c1 C(=O)(NN1CC(NC(=O)OC(C)(C)C)CC1=O)N(C(CC(=O)N)C1CC1)C.C1CC1 N1(C(C2CCC3C(C2)C3(F)F)=O)C(C(=O)NCC2CC(O)C2)CC2CCCCC12 Cc1nc2c(Nc3ccc(C(=O)Nc4cc(I)ccc4C#N)nc3)ncnc2[nH]1 C1(C(=O)NCC(CCCC)NC(C2C(=C)CC2)=O)C2Cc3ccccc3C12 CC(C)CCCC(=O)NC(c1ccccc1)C(C)NC(C1(C)CCC2CC2C1)=O N1(C(C2C(C=C)C2)=O)CCC(N(C(=O)CC(c2ccc(F)cc2)C)CCO)CC1 c1(CC(C)C)cc(C(=O)NCC2CC2NC(=O)C(C(C)C)NC(N)=O)n(C)n1 C1(C(=O)NC(C)(CNC(c2ccsc2C(F)(F)F)=O)C2CC2)CC2OC1C1CC21 Cc1nnc2n1CC(C(=O)NCCNC(C1(Nc3ncccn3)CC1)=O)CC2 c1(CCC)cc(C(=O)N(C(C)CNC(C2(CC)CC2(F)F)=O)CCOC)ccn1 c1(SCC(C)C)cccc(C(=O)NCCC(O)CNC(C2(O)CCSC2)=O)c1 c1(C(N2CCN(C(c3nc(CC)oc3)=O)CC2)=O)cc2c(s1)CCC(C)(C)C2 c1(CC(C)NC(=O)NCC(C2CC(F)(F)C2)OC)c[nH]c2cc(F)ccc12 c1(OC)ccc(OC(c2sc(-c3ccccn3)nc2C)=O)cc1[N+](=O)[O-] C1(C(=O)NCc2c(C(=O)NC(C(C)(C)O)(C)C)nco2)CN2CCN1CC2 C1(CC(=O)N(CC=C)CC2CC2)COCCN(C(=O)CCCCCC)C1 N1(c2ccc(S(N)(=O)=O)c(N3CCCC3)n2)C(=O)C2CCC(F)CN2C1=O C12CCC13CCN(CC3)C(=O)COC2.c1(SC)cccc(NC(=O)C2CC2)n1 N1(C(c2ccccn2)=O)CC2CC1CN2Cc1ccc(SC(F)(F)F)cc1 C(CC(C(=O)N1CCCC(C(=O)NC2C(C#N)C2(C)C)C1)N(C)C)N(C)C C(C(C)C(F)C(=O)NCCc1nc(C)no1)NC(C(CO)OC)=O C#CC1CC2CCC1N(C(C1CC(NC(c3c(C)cccc3O)=O)CCO1)=O)C2 c1(C(=O)NC2(CO)CN(C(Cn3ncc(CC)c3)=O)C2)cccc(C(C)(C)C)c1 C1(C)(CC)CC(NC2CCCCC2OC)CCO1 c1(C(=O)NC(CC=C)CNC(=O)C(C)C2CCCC2)ccc(Cl)c(C)c1 C1(OC(=O)N(C2CCOC2)C2CCC2)CCN(c2ccccc2)CC1 N1(C(CCN(CCC)C)=O)CC(NC(c2sc(F)cc2C)=O)CCC1C C(C)(CO)(C(=O)NCC1CCCN(C(C2CC(Cl)(Cl)C2)=O)C1)NC(C)=O CC(C)CC(C)CC(=O)NC1CC2(C1)CC2C(=O)N(C)CCc1ccc(Cl)s1 CC(C)CCC(O)C(=O)NC(C)(CNC(=O)Cc1ccc(Cl)cc1Cl)C(C)C Cc1cc(C(=O)NC(C)(C)CCC(=O)N2CCOC(C)(C(N)=O)C2)cc(C)n1 C1(CCOC)(NC(CC(COC)C)=O)CCN(C(C2(C)CCCOC2)=O)CC1 Cc1cc(CO)oc1C(N1CCCCC1CCNC(=O)C(C)Cc1ccco1)=O c1(CC)nc2c(C(=O)NCC3CN(C(=O)CCC[N+](=O)[O-])CC3C)ccnc2[nH]1 n1(Cc2cn(CCC(=O)NC(c3cc(Cl)nc(Cl)c3)C)nn2)ccc2ccccc12 C(=O)(C1=NNC(=O)CC1)NCC1(F)CC(NC(c2cn(CC)nc2C(C)C)=O)C1 c1(OC)ccc(CC(N2CCN(C(=O)C=CC3CCCC3)CC2CF)=O)cc1O C1(NC(CN(CC)CC)=O)CCCC1NC(=O)C[SH](c1nccn1C)C1CCCC1 c1(CCC)cc(C(=O)NC2CCC(CNC(=O)CC3(SC)CC3)CC2)n(C)n1 c1(C(N(CCC(=O)Nc2cnc(CC)nc2)CC#C)=O)cc(C)ccc1CC N1(C(Cn2cc(C(C)=O)nn2)=O)CCCC(C(C)NC(c2nnc(S)n2C)=O)C1 n1(CC(N2CC3C(NC(C(C)C(C)(F)F)=O)(C3)C2)=O)ccc2nc(O)nc(O)c12 c1(OCC)nscc1C(=O)NCCN(C(C1C(C)CC1C)=O)Cc1ccccc1 Cn1ccnc1CC(=O)NC(Cn1cncn1)C(=O)NC1CCOC1 N1(C(C(C)c2cc[nH]n2)=O)CC(C)(C(N2CCC(CN(C)C)C2)=O)C1 C1(C)CCCN(C(=O)NC)C1.c1(NC(=O)NCC(=O)NCC(CO)N)ccccc1 CCCC(C)CC(=O)N1CC(F)CC1C(=O)NCC1(C)CC1 C1C(C(F)(F)F)N1.c1(CN(CC(=C)C)CC)ccccc1 N1(C(C)C(=O)N(C)Cc2ccc(-c3cc[nH]n3)cc2)C(=O)c2ccccc2C1=O c1(CC)nc(=NC(CNC(C2(C3CCCC3)CCC2)=O)CC)s[nH]1 N1(C(C(C)(C)CC2CC2)=O)CC2CN(C(C3CC4CCC(C3)O4)=O)CC2C1 C=CCCC(F)(F)C(=O)NCC1(CCNC(C2CN3CCCN2CC3)=O)CC1 C(=O)(C(C)(C)CNC(C1CN(C(C2(C)CCCO2)=O)CC1CC)=O)NCC C1(C(N2C(CNC(COCc3ncc(C)o3)=O)CCC2)=O)COCCC1(F)F c1(C(N2C(C(=O)NCCCC=C)CSCC2)=O)cccn2cncc12 N1(C(CC(=O)OCC)=O)CCCC2(CCCCN2C(=O)C(c2ccc(C)o2)C)C1 CCC(C)(C)C(C(=O)NCC(=O)OC)OC.c12cccc(c1)OCC(=O)N2 C(CCCOC)(C(=O)NCCN(C)CCOC)NC(CC=CCCC)=O C1(CC(=O)NCc2c(C(N3CC(CCOC)C3)=O)c[nH]n2)CCCC12CC2 c1(SC)ccc([N+](=O)[O-])cc1C(=O)NC1CN(C(C2CCCN2C=O)=O)CC1C c1(CC(=O)NCCC2CN(C(C3C(=C)CC3)=O)C2)ccc(-c2ccnn2C)cc1 C1(CNC(C(C)c2ccco2)=O)CCN(C(=O)C=Cc2cccnc2)C12CCC2 N1(C(CC)=O)CCN(C(C2(CO)CCN(C(=O)C(C)C3(O)CCC3)C2)=O)CC1 c1(C(=O)NCC(=O)N(CC(CC)NC(=O)Cc2cccs2)C)c[nH]nc1O c1(COC)csc(C(N2CC(CC(C)NC(=O)Cn3cc(C4CC4)cn3)C2)=O)c1 C1(C(=O)NCC=C)N(C(=O)CC2OCCO2)CC12CCCC2 N1(C(CN2CC(C)(C)C2)=O)CCCCC12CC(NC(=O)C(O)CC1CCCCC1)C2 CC(C)C(C)(O)C(=O)NC1CCN(CCOCc2ccccc2)C1 Cc1cc(C(=O)NC2CCC2C(=O)N(C)C)ccc1C(F)F.c1(C)cn(CC)nn1 N1(C(c2ccc(OC)s2)=O)Cc2ccccc2C(NC(c2ccc(SC)s2)=O)C1 c1(N2CC=C(C)CC2)nc(C)nc(-c2ccccc2)c1C CC(C)CCCCC(=O)NCC(O)CCNC(c1c(C2CCC2)cnn1C)=O C#CC(C)(C)C(=O)NCC(O)CN(C)C(c1cnncc1C(F)(F)F)=O Cn1cc(C(N2CCC(CC(=O)NCc3cccc(O)c3)CC2)=O)cc1C#N C(=O)(C1c2c[nH]nc2CN1C(c1sccc1Cl)=O)NC(CC(=O)OC)(C)C c1(CC(=O)NCCN(C(=O)C(N)=O)CCC)csc(C(C)C)n1 Cc1csc(C=CC(=O)NCC2(C)CCC(NC(c3[nH]ccc3C)=O)C2)n1 c1(C(N2CCC3C(C2)CN3C(=O)CC2=CCCCC2)=O)cnc2c(c1)CCCC2 N1(C(CC(C)(C)OC)=O)CCC2(CCCN2C(c2cc(C)c(Cl)cc2F)=O)C1 c1(C(=O)OC(C(C(=O)OC)O)C(C)C)nc2ncccc2cc1C N1(C(=O)NCC(CC)CC(F)F)CCc2cncnc2CC1 N1(C(c2c(C)nc(O)cc2)=O)CCCC2(NC(=O)COCC(F)F)CCCC12 C12(CNC(C(C)OCC(F)(F)F)=O)CC(CO1)N(C(=O)CCOCC1CC1)C2 N1(C(C=NOC)=O)CC2ON=C(CNC(c3cc(NC)ccc3Cl)=O)C2C1 c1(-c2ccc(OC)cc2)nc(C2CN3CCN2CC3)n(C2CCc3ccccc32)n1 c1(CCC(=O)NC(CC)CNC(=O)C=Cc2cscn2)ccc(Cl)nc1 N1(C(C(C)OCC=C)=O)CCC(CNC(=O)CCN2CCC2)(COC)C1 N1(C(C(N2CCN(CC(=O)NC)CC2)C)=O)CC2CC1CN2C(c1nocc1Cl)=O C(=O)(C(=O)C(C)(C)CC)NC1(C(=O)NCC2CC(=C)C2)CC(CO)C1 C1(CCCNC(=O)CO)CCCCN1C(c1cc(-c2ccco2)on1)=O C(=O)(C(F)(F)C(F)F)NCCCCCNC(c1c(C)nn(C2CCOC2)c1)=O N1(C(CC(=C)C)=O)CC(O)CC1CNC(C1(Cc2cnn[nH]2)CCCC1)=O c1(C(N(C)CCn2ccnc2)=O)cnc2n[nH]c(-c3cnn(C(C)(C)C)c3)c2c1 N1(C(=O)COC2CC=CC2)CCC2CCN(OC(C3C(C(=O)OC)C=C3)=O)C2C1 CC1CCCN(N(C)CCOCF)C(OC(C)(C)C)C1 C1(C2(O)CCC2)(CC(=O)N(C2CCCC2)CCCNC(=O)C=Cc2cc[nH]c2)CC1 c1(C(N(CC2CCCN(C(C(CC)OC)=O)C2)CC)=O)c(OC)cccc1Cl c1(C(N2CCC(C(C)CNC(=O)C3CC3)CC2)=O)ccc(S(=O)(=O)C2CC2)cc1 C(c1ccncn1)=CC(=O)NCCCN(C(C)C)C(C1CCCN(C(N)=O)C1)=O C(CC(C)(C)CC(=O)N1CCC2(CC(NC(C3CC4CCC3C4)=O)C2)C1)OC N1(N(C(c2sncc2Br)C(=O)NCC)CC(C)C#N)CCOCC1 N1(C(C2C(C(=O)OC)CC2)=O)CCCCC(NC(c2cnc3n2CCC3)=O)C1 c1(CC(C(=O)NC(C2N(C(CC)=O)CCC2)C)O)ccc(Cl)cc1 C(CCC(C)C(=O)OCc1cn(C2CCCNCC2)nn1)OC c1(C(=O)NC2CN(C(=O)C3=CCCC3)CC23CC3)cc(=O)c2ccc(Cl)cc2o1 N1(C(C(CC)(O)c2cccc(Cl)c2)=O)CCC(NC(=O)CCc2ccon2)C(F)C1 C1(C)(OCC(=O)NC(C(=O)N(CC(C)C#N)C)C2(O)CCC2)CCCC1 N1(C(C(CC)=CCCC)=O)C2CCC1CC(CNC(c1cc(N)cnc1C)=O)C2 N1(C(C(CCC)(C)O)=O)CC2CCC(C1)N2C(=O)Cc1cc(F)ccc1Br N#CC1(C(=O)NCCOCCNC(c2cnsc2)=O)CCOC1 Cc1cccc(NC(C(C)N(CCC(F)(F)F)C(C2CCN(C)CC2)CC)=O)c1 N1(C(C(CCSC)O)=O)CCC(C)(C)C(CNC(c2cn(C)cn2)=O)C1 C(=O)(CC(=O)N(C(C)(C(=O)N(C)CC1CCOC1)C1CC1)C)N(C)C C1(NC(C2(CC)CCN(C(=O)C(COC)N(C)C)C2)=O)CCN(C)CC1(C)C C(c1cncnc1O)=CC(=O)NCC1(O)CN(C(C2CC2F)=O)C1 c1(C(N2CCC(O)C2CN(C)C)C(=O)NCC=C)ccc([Si](C)(C)C)s1 CCC(C)C(C)C(=O)NCc1coc(C(=O)NCC23CCC(CC2)CC3)c1 C12(C(=O)NCC(CC)NC(c3cnoc3-c3ccc(C)o3)=O)CC(C#N)(C1)C2 c1(C(=O)NC(CNC(CCSCC)=O)C(C)C(C)C)cc(S(N)(=O)=O)n(C)c1 c1(NC(C2CC(CNC(C(CC3CC3)OC)=O)C2)=O)cc(C)cc(C)c1 c1(NC(c2nccn2-c2cccc(F)c2)=O)ccnc2cc(Br)ccc12 C1(C(=O)NCCOC2CN(C(C3(CCF)CCC3)=O)C2)CC12CCCCC2 C1(C(N2CCCC(OCC)C2)=O)CN(C(=O)C(=O)C2CC2)CCC1O c1(C(=O)NCC(C)NC(c2cn(C)c(=O)n2C)=O)ccc(F)c(F)c1 CN1CC2CC1CN2C(=O)CC(CC1CC1)NC(=O)C(C)(C)CC#N C(=O)(C(F)(F)C(C)O)NCc1c(CCNC(c2nc(CS(C)(=O)=O)sc2)=O)ocn1 N1(C(CC2OCC(C)(C)OC2)=O)CCC2C(CCCN2C(c2cnc[nH]2)=O)C1 c1(C(N(CCNC(C2(C)CNC(=O)C2)=O)CC)=O)ccc(F)c(S(C)(=O)=O)c1 Cc1ccc(Br)c(C(N2CC(O)(CNC(C3CC3CN(C)C)=O)C2)=O)c1F N1(C(CC2CCN(C(c3c(C)ccs3)=O)C2)=O)CCN(C)CC1C1CCC1 CC1(C)OCCCC1NC(=O)NCC1(O)CCCC1 Cc1ccc(C(=O)NC(C)CNC(=O)CC2CCC(=O)NC2)cc1C#N C1(C(N2CCC(CNC(CC(C)C3CC3)=O)C2)=O)COCCN1C(c1ccco1)=O Cc1cc(Cl)ccc1CC(=O)NC1CC12CC(NC(c1occc1C)=O)C2 c1(CC)cc(C(N2CC(CNC(c3ccc(Cl)nc3N)=O)C3CC23)=O)ccc1F N1(C(c2ccsc2)=O)CCC(=CCNC(C23CC(C2)C(C(F)(F)F)O3)=O)CC1 N1(C(Cc2c(C)n(C)nc2)=O)CCC(NC(C2(C3CCCO3)CC2)=O)C(F)C1 Cn1nnc2cc(C(=O)NCC3CC3NC(=O)Cn3nc(Cl)ccc3=O)cnc12 c1(OC)cc(C(=O)NC2CCOCC2NC(C2(C)C(C)(C)C2(C)C)=O)ccc1F C1(C(=O)NCCN(C)C(C2COC(C)(C)CO2)=O)CCC(=O)N(CC(F)(F)F)C1 CC(=O)CC(C)(C)C(=O)N1CCCC(C(C)C(=O)NC(C)C(C)(C)C#N)C1 N1(C(c2cnn(C)c2F)=O)CCC2C1CCCN2C(c1cc(C(C)(C)C)on1)=O C1(NC(C(=O)NC2CCN(CC(C)(C)CO)CC2)=O)CCCC1C1CC1 C1(C(=O)NC(C(=O)NC)CC2CC2)N(C(=O)CCc2cc(C)[nH]n2)CCC1(C)C Cc1c(C(=O)NC(CO)CCCCNC(C2C(C)C2C)=O)cccc1[N+](=O)[O-] c1(CNC(C(=O)NC2CC(OC)C23CCC3)=O)cn(C)c(=O)nc1O C1(C(=O)C(C2(N(C)C)CCCC2)=O)CCC12CCCO2.c12ccc(cc1)CNC2=O CC1CCC(CC(=O)N(CCCCCNC(c2nc(Cl)cs2)=O)C)C1 CC(C)CC(C(=O)NC(C(=O)NCC1CC2(CCC2)C1)C1(O)CCC1)C(N)=O C(=O)(C(O)CC(N)=O)NCc1ccc(OCC(COCC)O)cc1 Cc1cc(C(N)=O)cc(C(N2CCC(CNC(=O)CC3(C)CCCO3)CC2)=O)c1 N1(C(C2CCC(C)O2)=O)CC2(COC(CNC(=O)C(O)(C3CC3)C3CC3)C2)C1 c1(C(C(=O)NCC(CC=C)NC(C23COCC(C2)C3)=O)C)ccc(Cl)cc1 c1(C(N(CCOC)CCNC(c2nnc(C)s2)=O)=O)cn2c(C)cccc2n1 C1(CNC(CCOC)=O)CCCC2CN(C(C3CC4CCC3C4OC)=O)CC12 C(C)(C(C)C(=O)N(CCO)OC)NC(c1ccnc(OC)n1)=O c1(CNC(C(CC)C)C)cc(F)c(N2CCOCC2)c(F)c1 CN1C(=O)c2ccccc2C1C(=O)NCC=CCNC(C1(O)CC2CCC1C2)=O N1(C(C(COC)O)=O)CC(C2CCN(C(c3cnc(C)c(N)c3)=O)CC2)C1 Cn1cc2c(C(N3CCCCC34CN(C(C3CCCOC3)=O)C4)=O)cccc2n1 C1(CC)CCCCC1OCC(N1CC(O)CC1CNC(=O)CSC(F)F)=O CCCC(C#N)C(=O)NCC(C1CC1)NC(c1ccnc(S)c1)=O C(=O)(C(C(C)(C)C)N1CCCC1=O)NCCNC(C(CC)c1ccccc1)=O Cc1cc(C(=O)NC(C)CNC(C2(C(F)F)CCCO2)=O)nc(O)n1 c1(C(N(C)CC2CC(=C)C2)=O)c[nH]nc1CNC(=O)CC1CC=CCC1 c1(OCC(=O)NC(C2CCCCC2)CNC(C2C(C)C2)=O)ccccc1 CCCC(C(=O)NCC1CCCCCN1C(c1cnc(C)cc1C)=O)S(N)(=O)=O c1(C(=O)NCC)cc(C)nnc1C(=O)OCC1CC1 c1(C(N(C2CCN(C(C=C(C)C3CC3)=O)C2)C)=O)cc2ccc(Br)nc2[nH]1 C1(CC)CN(C(=O)C(=Cc2cccs2)C)CCC1NC(C1CC2(CCC2)C1)=O C1(NC(C2CCCN(CC)C2)=O)CN(c2cc(Cl)nc(SC)n2)C2CCCCC12 C1(CNC(c2n(CCC)ncc2)=O)(COC)CCCN1C(C1CC(O)C1)=O c1(CCC)ccc(C(=O)N(C2CCN(C(C3CC(CCO)C3)=O)C2)C)cc1 CCCCCC(F)C(=O)N1CC(CNC(c2ccc(O)nc2C)=O)CCC1C C1(NC(c2ccc(C#C)o2)=O)CC2CCC1N2C(C1SCCCS1)=O c1(C(=O)NC(C)CCNC(=O)CC=CC(C)(C)C)ccccc1-n1ccnn1 C1(C(N2CCC(C(C)NC(=O)Cc3cnccn3)C2)=O)CCCC(F)C1 C(=O)(C(C(C)C)N1CCCCC1)N1CC(C(C)NC(C(C)=C2CCC2)=O)C1 c1(C(=O)NC(C)CCN(C(=O)C(CO)NC(N)=O)C)cc(C(N)=O)cc(F)c1 c1(C(=O)NCC2N(C(c3c(F)cccc3Cl)C)CC2)n[nH]c2c1CCCC2 c1(N2C(C(=O)Nc3cc(Cl)c(Cl)cc3Br)CC(=C)C2)ncnc2n[nH]cc12 c1(NC(c2ccc(Oc3cccc(OC)c3)cc2)=O)nc2ccc(Cl)cc2s1 C(C(CCN=C(NCCc1ccccc1)N1CCC(C)(OC)C1)OC)OC C(=O)(C(CC(=C)C)NC(=O)C(CC)N(C)C)N1CCC(C=C)C1 CCC(C#N)C(=O)NCCC1CN(C(c2csc(C3CC3)n2)=O)CCO1 c1(CNC2CCC(C(N3CCn4ccnc4C3)=O)C2)ccc2c(Cl)n[nH]c2c1 N1(C(c2[nH]nc(OC)c2Cl)=O)CCCC(C2(NC(c3nnc(C)s3)=O)CC2)C1 O(P(=O)(CCC1CCCN(C(c2ccc(C3CC3)c(C)c2)=O)C1)OCC)CC CC12CN(C(c3ccccc3Br)=O)CC1CN(C(c1ccsn1)=O)C2 C1(NC(=O)Nc2ccccc2OC2CC2)CCN(c2cc(C)c(I)cn2)CC1O N1(C(=O)O)CC2(CCC1CO)CC2.C(CCCCCN1CC(=C(F)C#N)C1)C(C)(C)C c1(C(c2c(C)cccc2)NCCc2ccccc2)cc([N+](=O)[O-])ccc1Cl C(CNC(=O)CNC=O)(CCOC)NC(CC1(OC)CCC1)=O C(CC)(CCCC(=O)NCC1(C)CCN(C)CC1)NC(c1c(CC)n(C)nc1)=O C#Cc1ccc(C(=O)NC(CCC)CCCNC(C2CS(=O)(=O)C2)=O)nc1 Cc1c(NC2(c3nnnn3C3CCCC3)CCC(C)(CO)CC2)cccc1C#N C(=O)(C(O)CC(F)(F)F)N1CCCC(CC)C1C(=O)NC(c1ncc[nH]1)C C1(C(=O)NCCOC2CCN(C(CCC=C=C)=O)C2)CCC(C)C(C)C1 C1(Cl)(C(=O)NCC(c2ccccc2)N(C(CN(CCC)C)=O)C)CC1(C)C Cc1c(C(=O)NC(C)C(C(C)C)NC(=O)Cc2ccsn2)ccn1CCO CC(C(=O)N1CCCOC(CNC(C2(C)CC2Br)=O)C1)C(C)(F)F c1(C(C2=CCCCN2C(C)=O)=O)ccc2nncn2c1 N1(C(C(F)=CC)=O)CCC2C(CCCN2C(c2n[nH]cc2Br)=O)C1 c1(CC(=O)NC2C(NC(C(CCCCC)O)=O)C2)cccc2cc(OC)ccc12 N1CC(C)OC(C)C1.c1(OC)ccccc1C(CF)NC(=O)CSCC(=O)OC Cc1cc(=NCc2ccccc2S(=O)(=O)N(C)C)nc(S)[nH]1.C1(N)CCCC(OC)C1 N1(C(C(CSCC)NC(c2nnc(O)nc2O)=O)=O)CC2(CCC(O)CC2)C1 C1(NC(CCCC(CC)C)=O)CCN(C(c2cnc(=N)[nH]c2)=O)CC(C)(C)C1 C1(NC(C(C(C)C)NS(C)(=O)=O)=O)CCC2(CC1)CN(C(c1cnnn1C)=O)C2 CC(C)CCCC(=O)N1CC2(NC(c3nn(C)nc3C(=O)OC)=O)CC1C2 N1(C(CC(CC)CC)=O)C2CC=C(C(=O)NOCC3CCC3)C1CC2 C1(CN(C)C(C2CCS(=O)(=O)N2)=O)CCCN(C(=O)CN2CC(F)(F)C2)C1 C1(CNC(C(C)N(C2CC2)CC2CC2)=O)COCCN1C(=O)C=CCN1CCCCC1 C1(C(=O)NC(c2ccncc2-c2ccc(OC(F)(F)F)cc2)C)C2CC1N(CO)C2 c1(C(N2CC(CC(=O)OC(C)C)(OCC)C2)=O)ccc(OC(C)=O)cc1F C=CC(CC(=O)NCC#CCNC(C1CCN1Cc1ccsc1)=O)c1ccccc1 N1(C(CCC=C)=O)CCCC(C2(NC(c3n[nH]c(C)c3C(F)(F)F)=O)CC2)C1 S(=O)(=O)(c1ccc(NCCC2CCC2)c(F)c1)NC(C)COCC1CC1 C1(C)(C(N2CC3(N(C(CC4(OC)CCOCC4)=O)CC3)C2)=O)CC(C(C)C)=NO1 C(c1ccccc1Cl)=CC(=O)N(CCCNC(c1cc(F)ncc1Br)=O)C c1(C(=O)NCC(CC)N(C(C2CC(C#N)C2)=O)CC)ccccc1C1(C)CCO1 C1(NC2(C)CC(C(=O)Nc3nc(Cl)c(C#N)s3)C2)CC2CCCCN2C1 C1(OCC)CCCN(c2cncc(C(=O)N(C)C(c3cc(C)on3)C)n2)C1 Cc1nc(C#N)cc(=NCC23CCC(NC(=O)CCc4cc[nH]n4)(CO2)C3)[nH]1 C(CCC(C)(C)C(=O)N1CC=CC(C(N2CCCC(CCO)C2)=O)C1)OC c1(C(=O)NCC(CC=C)NC(=O)Cc2cccnc2F)cc(O)n(CC)n1 C12(NC(c3cnn(C(C)C)c3Cl)=O)CCCN(C(C3CCCC(=O)C3)=O)CC1C2 c1(-c2ccc(CNC(C3CC(C(N4CCOC5CC45)=O)C3)=O)o2)cccc(Cl)c1 N1(C(c2cc(OCC)ncc2)=O)CC2CCN(Cc3ccc(N(C)C)s3)C2C1 N1(C(C(C)c2ccco2)=O)CCCN(C(c2cccc(C(F)F)c2F)=O)C(C)C1 CCCC(C)(C)CC(=O)N1CCCN(C(=O)C(=O)NCCC(N)=O)CC1CO c1(COC)c(C(=O)NCC2CNCC(F)C2)sc2ccccc12 C1(CC(=O)N(C2CCCC2)CCC)CN(C(C2CC(O)C2)=O)CCC1C C12(C(=O)NCc3cnc(C)o3)C(NC(=O)CCC3CC3(F)F)C3CC1C2C3 CCC(CC(=O)NCC(O)CCNC(c1cnn(CCO)c1)=O)C(C)(C)C C1(C(=O)NC(c2cn(C)nn2)C(N2CCOCC2)=O)CCCCC1F N1(C(c2cncc(C(F)(F)F)c2)=O)CCC2(CCCC2)C1 N1(C(CCOCCOC)=O)CC2C3CCC(C(NC(c4cscc4Cl)=O)C3)C2C1 C=CCC(C)(C)C(=O)N(C)CP(C)(C)=O.N1CCCC1CC=O c1(C(=O)NC(c2ccc(C(F)F)cc2)C)ccc2sc(C3CC3)nc2c1 C(CCC)(C(O)C(=O)N1CCCC1CN=[N+]=[N-])NC(C(C=C)O)=O Cc1nc2nccc(C(=O)NCC(C)(O)CNC(C3(C)CCNC(=O)C3)=O)n2n1 c1(C(N(CC(C)(C)C)CCC#C)=O)ccc2occ(C)c2c1 N1(C(Cc2c(C)cccc2)=O)CCN(C(c2cc(CO)[nH]n2)=O)C(C)C1C N1(C(C(C)C)=O)CCC2CCC(NC(c3ccc(Cl)c(Cl)c3)=O)C1C2 C1(NC(c2c(C)n(C)nn2)=O)CCN(C(c2ccnnc2)=O)CC1F N1(C(C2C(C)OCC2)=O)CC(C2CCN(C(=O)Cc3c(Br)cnn3C)CC2)C1 c1(C(=O)NC2(CF)CCN(C(C(CN(C)C)(C)C)=O)C2)cc(F)cc(F)c1 C1(OC(C)(C)C)CC2(C1)CN(C(=O)CC1NC(=O)NC1=O)C2.C12CC(C1)C(=O)N2 C1(NC(C(CCCCC)O)=O)CN(C(C2CC3C=CCC(C2)C3)=O)CC2(CCC2)C1 CC1(C(N2CC(NC(=O)CCc3ccc(Cl)cc3)C(O)C2)=O)COCC1(F)F Cc1c(O)ccc(C(N2CCN(C(C34CC(C)(CO3)C4)=O)CC2)=O)c1C C1(F)(C(=O)NCc2cccc(CC)c2)CCCN(C(C2(CC)CCCCC2)=O)C1 C(CCCC(C)NC(=O)CCc1cc[nH]n1)NC(C1(OC)CCSC1)=O c1(C(N2CCC(NC(CC(CCC)C)=O)(CO)CC2)=O)cn(C)c2ccccc12 C1(CNC(C(C)(C)OCC)=O)CN(C(c2cc(C(N)=O)no2)=O)CCN1C C(=O)(C(C)(C)C#N)NC(C1CCCN(C(=O)CSc2ccccc2F)C1)C C1(CNC(c2c(C)nc[nH]2)=O)(CO)CCN(C(=O)CC2OCCC2(C)C)C1 c1(C(N2CC3C(NC(c4cscn4)=O)(C3)C2)=O)cnc(O)c([N+](=O)[O-])c1 N1(C(COC2(C)CCC2)=O)CC2CC(C(=O)NC(CO)CC(F)(F)F)(C2)C1 N1(C(CC2C(CC)C2)=O)CCN(C(=O)COCCCCCCCC)CC12CCC2 CCCCCC(O)C(=O)NCC1CCCN1C(c1oc(C2CCC2)nc1C)=O C1(NC(C2CC(NC(CCCC=C)=O)C(O)C2)=O)CCCC(O)CC1 c1(NC(CCNC(C(C)SCC)=O)=O)cccc(F)n1 c1(C(N(C)CC2N(C(C(C)OCCC=C)=O)CC(F)C2)=O)cccc(N)c1Br N1(C(c2c(C)ocn2)=O)CC2C(CN(C(=O)Cc3ccsn3)C)C2C1 N1(C(COC(CC)C)=O)CC2(CC(CNC(C3CC4(C3)CC43CC3)=O)C2)C1 C(c1cccc(O)c1)=CC(=O)NCC1CCCN(C(C2C(C)=CCC=C2)=O)C1 C1(O)(C(C)NC(=O)C(N2CCCC2)C2CC2)CN(C(=O)C=C2CCC(C)C2)C1 N1(C(CC(C)F)=O)C2CCC(C2)C1C(=O)NCCCN1CCC1 CC(C)(C(=O)N1CC=C(C(=O)Nc2cccc(NC=O)c2)C1)C(N)=O N1(C(CCCOCC)=O)CCN(C(=O)C(C)N2CC(C)C2)CC1c1cccnc1 C1(n2cc(N(C(C)C3CC3)C(C3CC4CCC3C4)=O)nn2)CCC(N(C)C)CC1 Cc1ccc(OCCC(=O)N(C)CC2CCN(C(=O)C=CC3CC3)CC2)cc1C c1(C(=O)NC2CC(NC(CC3(C)CC3(Cl)Cl)=O)C2)ccc(O)c(CO)c1 c1(C(N2CCCN(C(C(C(=O)OCC)F)=O)CC2)=O)cc2ccc(C)cn2n1 N(C(=NCCF)N1CCCC2(CCC2)C1)CCN(C(=O)NCc1ccccc1)CC c1(C(N2CC(C(C)NC(c3cc(=O)cc[nH]3)=O)OCC2)=O)nn(C)c(Cl)c1Cl CC1(C(=O)NCC(CO)NC(c2csc(C(F)F)c2)=O)CC(C2CC2)=NO1 C(=O)(C1c2ccccc2OCC1(C)C)N1C(CNC(c2ncc(C)c(Cl)c2)=O)CC1 N1(C(c2ccc(OCC(C)C)cc2)=O)CCN(C(=O)C(O)C(F)F)CC(C)(C)C1 C1(NC(CCn2ncc(C)c2)=O)C2CC1CN(C(=O)Cc1csc3nccn13)C2 CC1CCCC(C(=O)NCC2CCN2C(=O)Cc2ccnc(C(F)(F)F)c2)C1 C1(NC(c2c(CC)c[nH]n2)=O)CCCC(N(C)C(C2CC(O)C2)=O)C1 c1(C(C(=O)N(CC(C)NC(=O)C(C)(C)C2CCOCC2)C)C)cccc(C#N)c1 c1(C(N2CC(CNC(Cc3c(C)non3)=O)N(C)CC2)=O)n[nH]c2c1CCSC2 N1(Cc2ccc(S(CC)(=O)=O)s2)CCC2(CC1)CC(C(N1CCOC(=O)C1)=O)C2 N1(CC(=O)N(C)Cc2ccc(Br)cc2)CCC2(CC1)CC2N CN1CCN(CCC(=O)N(CCCNC(C2CCC(O)C2)=O)C)CC1 CS(=O)(=O)c1cccc(-c2cnc(CC(=O)NCc3ccc(Cl)c(Cl)c3)nc2)c1 C1(OC)C(NC(c2[nH]ccc2CNC(c2ccoc2Cl)=O)=O)CC1O CON1CCC(C(=O)NCCN(CC(C)O)C(=O)CC2CC(C)(C)CO2)CC1 C1(C2CC2)(NC(C(CC(C)C)NC(C2CC3CCCC3C2)=O)=O)CCCCC1 CC1N(C(=O)C(Cn2cccn2)NC(=O)CN2CCNC2=O)CCCC1(C)C c1(CNC(C(=O)N(C2CCCC2)CC(C)NCC)=O)c(C)nc2sccn12 c1(N2CC(CC)C(O)C2)cc(Br)ccc1S(=O)(=O)N1CCN(C)C(C)(C)C1 N1(C(CCCCCOCC)=O)CCC2(CNC(c3ncccc3Cl)=O)CCCC12 c12cccnc1N(Cc1ccn(-c3ccccc3)n1)C2=O.C1(C(C)O)CC(NC=O)C1 CCCC(CC)C(=O)NC(CCSC)C(=O)NCCN1CCCC1 c1(C(=O)NC2CCCN(C(C=CC=CC)=O)CC2)ccccc1S(C)(=O)=O C1(CCNC(c2ccccn2)=O)CSCCN1C(=O)CNC(=O)C(F)(F)F c1(CCC)ccc(N)c(C(=O)NC2CCCC2NC(=O)C=CC2CCOCC2)c1 C1(CNC(c2nc(C)oc2)=O)CC2COCC2N1C(=O)CNC(=O)C(F)(F)F C1(CC#C)(C(N2CCC(C(C)NC(=O)C(F)C3CCOC3)C2)=O)CCOCC1 C1(NC(c2ncc(Br)s2)c2nnnn2C2CCCC2)CCn2nccc2C1 N1(C(C2N(C(C(=O)NC3CC3)=O)C3(CC2)CC3)=O)CC2COCC2(CO)C1 c1(OC)nccc(C(=O)NC2CC(CC(=O)NCC(C)O)C2)n1 c1(C(N(CCNC(C2C(C(C)C)CCO2)=O)C)=O)cnc(Br)c(N)c1 CC1=CCC(C)(C(N2CC3C(CNC(c4cnn(C5CC5)c4)=O)C3C2)=O)CC1 C1(NC(c2cc(-c3ccc(F)cc3)[nH]n2)=O)CC2CC1N(C(=O)CCF)C2 N1(C(COCCN(C)C)=O)CC(O)CC1(C)C(=O)Nc1nccn1COC1CC1 N1(C(CC2CC(N(C)C)C2)=O)CCC(NC(c2cnc(S)[nH]2)=O)C(F)(F)CC1 CCCCC(C)(F)C(=O)Nc1cc(N2CCCC(C)(C(=O)OCC)C2)nc(C)n1 CCC(=O)CCC(=O)N1CCOCCC1C(=O)NCC(c1ccccn1)O N1(C(CCc2onc(C)n2)=O)CCCCC(C2CN(C(=O)CC3CC(F)(F)C3)C2)C1 C#Cc1cccc(NC(C2(NC(c3cnn(C(F)F)c3)=O)CC(CO)C2)=O)c1 c1(C(N2CCC(NC(C3(C)CC3)=O)C2C2CC2)=O)cnnc2ccccc12 N1(C(CCC(=C)C)=O)CCCN(C(=O)CC(C)OC)C(C)C1 N1(C(c2cc(C)c(Cl)s2)=O)C2CC=C(C(=O)N3CCC(F)(CF)C3)C1CC2 C(c1cncc(OC)c1)=CC(N1C(C(N(CCOC)CCO)=O)CSCC1)=O c1(C(=O)NCCOCCN(C(C=C2CCC(C)CC2)=O)C)cnc2c(c1)CCC2 N1(C(COCCN(C)C)=O)C2CCC1CC(NC(c1ccnc(OC(F)F)c1)=O)C2 c1(C(c2nnnn2C(C)(C)C)NC(c2ccc(F)cc2)COC)cnn(C)c1Cl C1(CC)C(C)CC2CN(CCc3[nH]cnc3C)CCN12 Cc1c(C(=O)NCCC2CN(C(=O)C3=CCCC3C)CCO2)cncc1N C1(C(C(=O)NC(C)CC2CC(O)C2)C)CCN(C(C2CCC(F)CC2)=O)CC1 C1(NC(C(CN(C(C2(C=C)CCC2)=O)C)C)=O)C2CCCCC12 c1(OC)ccsc1C(=O)N(C1CC1)Cc1cccnc1.C1(C)C=CC(=O)N1 C1(C)(C(=O)NCC2(C)CCN(C(C(C(C)C)N(C)C)=O)C2)CC(C(C)C)=NO1 C#Cc1cccc(NC(=O)CNC(=O)C(CC)Nc2ccc(Cl)nc2)c1 N1(C(CC(C)Oc2ccccc2)=O)CCCCC1CNC(c1cncs1)=O C1(C(N2CCC(C(C)NC(=O)COc3ccc(F)cc3)CC2)=O)CC2C=CC1CC2 CCCCCC(O)CC(=O)NC1CCCC(NC(=O)CCCc2nncn2C)C1 c1(OC)ncnc(OC)c1C(=O)NCC(C)(C)CNC(=O)C=Cc1cn(C)nn1 c1(C(N2CCC(CC)(CNC(c3n[nH]cc3Cl)=O)C2)=O)ccc2occc2c1 c1(CCNC(c2n(CCOC)nnn2)C2(C3CC3)CC2)nc(C)sc1C c1(CCc2ccccc2)ccc(I)cc1.n1(CC(N)=O)nnc(C)n1 C(=O)(C1CCCc2nncn21)NC1(CO)CCCN(C(CSCCCC)=O)C1 Cc1nc(C(=O)NCC2(NC(=O)CSc3nccn3C)CCC2)c2ccnc-2[nH]1 c1(NC(C(Cc2cn[nH]c2)NC(C=CC=CC)=O)=O)ccccc1Cl N1(C(c2c(C)nc(O)nc2C)=O)CC2CCC(C1)N(C(=O)Cc1cscn1)C2 c1(C(=O)NCCCN(C(C2COC3(CCC3)C2)=O)CC)sc2cccnc2c1Cl C(CC(C(C)(C)C)NC(c1ncnc(O)c1Cl)=O)N(C(C(CC)(C)O)=O)C N1(C(C(CC)Nc2ccccc2)=O)CC2CC2(NC(=O)NCc2[nH]nnc2C)C1 c1(C(=O)NCC2CC3(C2)CN(C(=O)Cc2ccoc2)C3)ccn2cnnc2c1 N1(C(C2(OC)CCC2)=O)CCC(O)(CCNC(C2CC2C(C)C)=O)C1 C(C(C)C(C)C(=O)NC1(CCNC(C2CCCN(C)C2)=O)CC1)OC N1(C(Cc2c(C)nccc2)=O)CCC(C)C(NC(=O)CCC2CCCCC2)C1 C1(C(N(CC(C)(C)NC(c2c[nH]nc2C2CC2)=O)C)=O)CCCCC(F)(F)C1 C1(CC(=O)N(C)CC2N(C(COCC(=O)NC)=O)CCC2)CCOC1(C)C N1(C(COC)=O)CCCC(C)(C(=O)Nc2cnncc2Br)C1 N1(C(c2cccc(SCC)c2)=O)CCOCC(F)(CNC(C2(C3CC3)CC2)=O)C1 C(CNC(=O)CP(C)(C)=O)(CC(F)(F)F)NC(Cc1nnc(C)o1)=O CCCCC(C)(F)C(=O)NC1CC2CC(C1)N(C(=O)Cn1cnc([N+](=O)[O-])n1)C2 N1(C(c2c(CCC)onc2C)=O)CC2(CC(NC(=O)C(CC)N(CC)CC)C2)C1 C1(C(=O)NCC2(O)CCC(C)C2)(NC(C2CCCS2)=O)CCc2cc(Br)ccc2C1 C(C)(CNC(C1CC(C(F)(F)F)(OC)C1)=O)(C(C)C)NC(C=C(COC)C)=O C1(C)(N(C(C(C)NCC)=O)CC)CCC(C(F)(F)F)CC1 CC1=C(C(=O)N2CCN(C(C3(n4cccn4)CCOCC3)=O)CC2)CCO1 c1(OC)cc(C)cnc1NC(=O)C(F)(F)C1CCCC1N c1(OC)cc(C(=O)NC2CC(CC(=O)N(CC(N)=O)C)C2)ncn1 c1(OC)ccc(C(=O)NC2CCC(NC(=O)COCC3(F)CC3)C2)nn1 N1(C(c2ccc(-c3n(C)ncn3)cc2)=O)CCCC(NC(=O)CC(F)(F)F)C(F)C1 c1(-c2nc(C(=O)Nc3cccc(CC)c3)sn2)cnn2c1CCC2 C(CCCCC(=O)N1CC(COC)CC1CNC(c1cccc(Cl)c1)=O)=CC C1(C(=O)NC(C(=O)NCC(C)C(C)(C)C)(C)C)CC2(CCC2O)C1 c1(C(=O)NC2CCN(C(c3c(C)n(C)cc3)=O)C2C)nc(Cl)c(Cl)c(N)c1Cl c12cccc(n1)NC2=O.CCC(CO)N(C)C(C1CCC1)=O CC1CCCn2c(C(N3CCN(C(C4CCC(C)(C)C4)=O)CC3C)=O)cnc21 C1(C(N2C(C)(C)C(CNC(=O)CC3CCCC3)CC2)=O)COC2(CCC2)CO1 c1(C(N(C2CC(NC(C3CCC(C)O3)=O)C2)C)=O)[nH]c(=N)sc1C(F)(F)F C(c1ccco1)=C(C)C(N1CCC(NC(c2cnnn2C)=O)C1)=O c1(C2CC(NCc3n(CC(F)(F)F)ccn3)C2)ccc2c(c1)OCO2 Cc1nc(CO)sc1C(=O)NC1CCOCC1NC(C1CC(O)C1)=O CC1CN(C(c2cc(Cl)no2)=O)CC1CCNC(=O)C(C1CCCCC1)=O c1(C(N2CC(C(C)NC(c3ncccc3F)=O)OCC2)=O)cc([N+](=O)[O-])nn1C N1(C(c2ccc(C)n2C)=O)CC2OCC(NC(=O)C=Cc3cnn(C)c3)C2C1 N1(C(C(CCSC)O)=O)CCC(O)(CN(C(=O)C(C)CC(C)C)C)CC1 C(=O)(CCS(N)(=O)=O)NC(C(C)C)CCNC(c1cc(C(F)F)no1)=O c1(CN(C(C(=O)NCC2CCCC(C)O2)=O)C)ccc2[nH]ccc2c1 CCCCCC(O)CC(=O)NC(C)C(CO)NC(C1CCOC(CC)C1)=O N1(C(C(C)CC2CC2)=O)CC2(CNC(C3CCCC(C)CC3)=O)CC(F)(C1)C2 C12CCc3cc(ccc3C1=O)N2.c1(C(c2nnnn2C)SC)cnc(Cl)s1 c1(C(N(CCNC(c2cnccc2C(F)F)=O)CC)=O)ccc([N+](=O)[O-])n1C c1(OC)ccc2c(C(=O)NC3CCN(C(=O)C#CC4CC4)CC3F)csc2c1 c1(CN2C3CC(NC(C(C)(C)OC)=O)CC2CC3)ccc2ccn(C)c2c1 N1(C(C(CC)OC)=O)CCC(NC(C2CC=CCC2)=O)C1C c1(OC)cc(C(=O)NC(CCN(C(=O)C(O)C2CCCC2)C)C(C)C)cc(C)n1 C(CS(=O)(=O)c1ccc(C)cc1)NC(c1cc(F)ccc1F)CC=C c1(OC)cc(C(N2CCC3CCN(C(=O)C4CC4)CC23)=O)cc2c1OCC2 C(=O)(C1=CC2C=CC(C1)C2)N(C)C(c1cnc2cc[nH]c2c1)=O.C12(CC1)CN2 c1(C(=O)NCCCN(C(CN(CC(=O)NC(C)C)C)=O)C)nc2ncccn2n1 CN1C(=O)Cc2ccc(C(=O)NCC3(C)CCN(C(C4CCC(=O)N4)=O)C3)cc21 N1(Cc2ccc(COC(C)=O)o2)CC(NC(c2c[nH]cc2C#N)=O)C(C#N)C1 c1(C(N(CC(C)O)CCNC(c2ccn(C)c2)=O)=O)ccc(Cl)c(Cl)c1N c1(CN2CCCC(CNC(CNC(C(CC)CC)=O)=O)C2)cc(Br)ccc1OC C(=O)(C1CCc2scnc21)N(CCCCCCNC(CCSCC(C)C)=O)C N1(C(=O)NCc2ccc3c(c2)OCCO3)CCCC2CC3(CCC3)C12 c1(C(N(C)CC2N(C(CCCC)=O)CCOC2)=O)cnc2c(C)cnn2c1 c1(C(=O)NCCCN(C)C(c2cccc(N)c2F)=O)cc2cc(F)ccc2s1 c1(-c2[nH]cc(C(=O)NCCN(C(=O)C(C)CN(C)C)C(C)C)n2)ccc(Cl)cc1 C(Cc1ccco1)(C(=O)NCC(F)CO)NC(CSCC(N)=O)=O Cc1coc(C(C)(C)C)c1C(=O)NC(C)C(CO)NC(=O)Cc1cccs1 Cc1ccc(C(N2CC(NC(=O)C(C)(CO)CO)C(F)C2)=O)cc1F c1(CC)n[nH]c(=NCC2CCN(C(=O)CSCc3cccc(Cl)c3)C2)o1 C=CC(CCC)CC(=O)Nc1c(F)cc(COC)c(F)c1 Cc1n[nH]cc1NC(c1nc(CNC(=O)Cc2ccoc2)cs1)=O C12(CCOC)CCN(C1)C(=O)C(F)(F)CNC(=O)C1C(C1)C(=O)N2.C(COC)OC Cc1c(C(=O)NCC(O)CCNC(C2SCCCS2)=O)noc1-c1ccccc1 N1(C(CCN(C(=O)CC2CCCO2)C(C)C)=O)CC(F)CC(F)C1 N1(C(=O)NCC2(OC)CCCC2)CCCC2(CCCCN2)C1 C(=O)(C(C)(CSC)NC(c1n[nH]c(C)c1Cl)=O)NC(CC)CN1CCCC1 N1(C(C(COCC=C)C(F)(F)F)=O)CC(N=c2nc[nH]s2)CC(C)(C)C1 CC(CCN(C)C)CCNC(=O)C(C)OCOC.C1=CN=CNC1c1c[nH]nn1 CC(C)(C)CC(C(=O)NOCC1CC2C=CC1C2)NC(C1(O)CC1)=O c1(NCC2CC(NC(CC3C(OC)CC3)=O)C2)nc(C)ns1 CCC(CC)CCCN(C)C(C1CC(C)N1C(=O)C=Cc1cc(C)no1)=O c1(C(C)NC(N2CCCC(CCN=[N+]=[N-])C2)=O)nc(Cl)c(Cl)s1 C1(C(N2CC(C)(CC)C2)=O)CC2CC1CN(C(C1(CO)CC1)=O)C2 C1(C(=O)NCCOCCN(C(C2(COC)CC2)=O)C)CC2(CC2)C1 C12(CNC(c3cc(C(F)(F)F)n[nH]3)=O)CC(CN1C(=O)COC1CCCOC1)C2 C(N=c1nc2ncn(C)c2c(NC2CCCC(C)CC2)[nH]1)c1c(OC)cccc1 N(C(=NCCCNS(C)(=O)=O)NCC1CC2CCC1CC2)CC1CN(C(C)C)C1 C(=O)(CC(C)CC(C)C)NC1C(NC(CC(C)c2ccco2)=O)CN(C(N)=O)C1 C1(N(CCC(=O)N(CC(N)=O)C)C)CCCCN(C(C(C)(C)C)=O)C1 C=C1CC(C)(C(=O)N(C(c2ccccc2)C(C)O)C)C1 Cc1cccc2c(C(=O)NC3CCCC(NC(C4CC4C)=O)C3)cccc12 N1(C(C=CC=CCC)=O)CCC(CNC(c2cn3ccnc3s2)=O)C12CC2 c1(C(N2C3CN(C(c4ccn(C)c4)=O)C(CC3)C2)=O)cc2cc(Br)cnc2[nH]1 c1(C(C(=O)NC)N(C)Cc2cnn(C)c2)ccc(N2CCCC2)cc1OC.C(N)=O CC(C)(C(=O)NCC1CCCN1C(=O)CC1CC=CCC1)N1CCOCC1 N1(C(CCC2CCN(C)CC2)=O)CC(NC(C2CSCN2C)=O)C(C2CC2)C1 c1(CC(=O)N(CCNC(=O)CCn2nc(C)nc2C)CC)ccc2occc2c1 C1(C)(C(C)NC(C2CCCO2)=O)CN(C(=O)CSc2nncn2C)C1 N1(C(CC2N(C(C(SC)SC)=O)CCOC2)=O)C2C=CCC1CCC2 C1(NC(C2(C(F)(F)F)CCC2)=O)CCCC(NC(C2(C(F)F)CCCO2)=O)C1 c1(N2CCCC(COCCOC)C2)ncccc1S(=O)(=O)NN1CCC(CO)C1 C1(CNC(C=CC(C)C)=O)CN(C(c2cc([N+](=O)[O-])c[nH]2)=O)CCC1C c1(CC)ccc2occ(C(N3CC(CNC(=O)C(C)CC)C(F)(F)C3)=O)c2c1 CC1(C)CN(C(c2ccn(C(F)(F)F)n2)=O)CCC1NC(=O)Cc1ccno1 C12(C(=O)NCCC3(O)CN(C(C4CC45CCC5)=O)C3)CCCCC1NC(=O)CC2 c1(NC(C2N(C(C3CCC(=O)NC3)=O)CC=C2)=O)nc2cccc(Cl)c2s1 c1(SC)ccc(C(N2CCC3(CO)CCCC23)=O)cc1C#N c1(OC)ccc(C)c(C(=O)NC2CCOC(CNC(=O)C(C)(C)Br)C2)n1 CC(C)C(O)CC(=O)N1CC(CNC(=O)C(C(C)C)NC(N)=O)CC(C)C1 c1(SC)ccc2[nH]c(=NCCCN(C(=O)CC3CCCCC3C)C)sc2c1 CCC(O)C(C)(C)C(=O)NOC(CC(C)C)C(=O)N1CCCC(CF)C1 C1(CNC(COCCC)=O)CC(F)CN1C(=O)Cn1nnnc1-c1ccccc1 C1(CC)CN(C(=O)C(C)c2ccco2)CCC1NC(C1CCCO1)=O c1(NC(=O)CC(Cl)Cl)cccc(CO)c1F CCCCCC(C(=O)N(C1CCCN(C(=O)C(C#N)CC)C1)CC)C(C)C N1(C(C(C)n2ccnc2)=O)CCC(C)(NC(c2cnn(CC3CC3)c2)=O)CC1 C1(NC(c2c(C(C)C)onc2)=O)CCN(C(C2CC2c2ccn(C)n2)=O)CC1F O=C1NC(=O)c2ccccc2N(C(CC2CCOC2)C(=O)NCCC2CC2)C1 C(=O)(C1=C(Cl)CCC1)NC1(CF)CCN(C(COCCCCC)=O)C1 CC1(C)COCCC1CNC(c1ccc(I)s1)c1nnnn1CCCF C1(NC(C2(C)CCC2)=O)CC1C1CCCN(C(C2(c3ccc(F)cn3)CC2)=O)C1 Cc1ccc(C(N2CCCC2NC(N)=O)C(=O)NCCOc2ccc(F)cc2)nc1 C(=O)(C(CN(C)C)C(C)C)NCCC(=C)CNC(c1nc(Cl)ccc1N)=O C1(NC(=O)C2CC2)CCCCN(C(=O)CCC(=O)Cc2ccc([N+](=O)[O-])cc2)CC1 N(C(=NCCc1cn(C2COC2)nn1)NCC1CC1)C1C(OC)COC1 c1(C(N(CCNC(=O)CSC2CCCCO2)CC)=O)ccc(Cl)c(Cl)c1C C1(C(=O)NC(CSCC)C(=O)NCCCc2cccnc2)CCC(=O)N(C)C1 C(C)(C(C(C)C)NC(c1cncc(C(=O)N(C)C)c1)=O)NC(c1c(C)nns1)=O C1(CCNC(CNC(N)=O)=O)CCCN1C(c1cnc[nH]1)=O C1(C2CCCCO2)(C(=O)NC2C(NC(=O)Cc3ccccc3F)C2)CCOCC1 C1(C(=O)NC)CCN(C(=O)C(C(C)(C)C)NC(=O)C(C(CC)CC)OC)O1 CC1CC(CNC(C2CCN(CC(F)F)CC2)=O)CN1C(=O)C=CC1CCC1 c1(C(N2CCN(C(c3c(Cl)ncc(C)c3)=O)C(C)C2)=O)ccn2ccnc2c1 C1(C(=O)OC(C)(C)C)COC2CN(C(c3cc(CNC(C)=O)on3)=O)CC2O1 C1(CC)CN(C(C23CC(CO)(CN2C(c2cn(CCO)nn2)=O)C3)=O)CCCO1 N1(C(c2c(OC)nccc2)=O)CC(CNC(=O)Cc2ncc(Cl)s2)CC1(C)C N1(C(CNC(=O)OC)=O)CCCCC(C(N2CC(NC(C)=O)C2(C)C)=O)C1 c1(C(=O)NCCN(C(C2(CC)CCCO2)=O)C)cnn(C)c1C(C)(F)F c1(C(N(CCNC(C(C)OCCC=C)=O)C)=O)c(C)nn2c1CCCC2C C1(CC)CC2CCC1N2C(=O)CC1N(C(C2(CO)CCCCC2)=O)CCC1(C)C Cc1cc(C2(NC(=O)C(CC3CC3)NC(C3CC(F)CS3)=O)CC2)no1 N1(C(CN(C2CCCC2)C)=O)CC(CNC(=O)CCc2ccsc2)C2(CC2)C1 CC1CCC(NC(=O)Cc2cccc(Cl)c2)CN1C(=O)CN1CCCS1(=O)=O N1(C(C2(CCOC)CC2)=O)CCCC(CO)(NC(c2ccnn2C2CC2)=O)C1 N12CCN(CC1C1CCC1)C(=O)COCCC2=O.C(CC(C)C)NC(COC)=O O=C1CCC2CN(C(=O)NC(c3cccc(OC(F)F)c3)C(F)(F)F)CC2N1 C1(NC(c2cccc(CO)c2)=O)CN(Cc2cnc(Cl)nc2Cl)CC1(F)F N(C1CCc2cc(Cl)ccc21)C(=O)NC(c1ccc(O)cc1)CC N(S(=O)(=O)N1CC(C(N2CC(O)C(O)C2)=O)CC1C)C(C)C N1(C(c2c(C)nc(C)[nH]2)=O)CCC(C2CN(C(=O)C(O)C3CC3)C2)CC1 CC(C)(CCS(C)(=O)=O)C(=O)N1CC(CNC(=O)COCCCF)C2(CC2)C1 C1(CCC(=O)N(CCNC(c2ccc(C3CC3)cc2)=O)C2CC2)NC(=O)NC1=O O=C(C#CC1CC(F)(F)C1)NCC1CCCC1NC(C12CCC(F)(CC1)C2)=O C1(c2cn(CCCOC)nn2)CC2CCC(C1)N2C(C1CCCCN1C)=O N1(C(c2cc(C)nn2-c2coc3ccc(Br)cc23)=O)CCOC2(CCSC2)C1 C1(C(N(C)Cc2c(C)cccc2)=O)CCCN(C(C2CC3(C2)CC3(F)F)=O)CC1 C(=O)(C(F)CCC(C)C)NCC1CCCN(C(c2cncc(C#C)c2)=O)C1 N1(C(c2[nH]ccc2CC)=O)CCCCC1C(=O)NC(CC)CN1CCCC1 C1(C(=O)NCC2C(CNC(c3cc(C(C)(C)C)on3)=O)C2)C2(CC2)C12CC2 C(=O)(C(C(C)C)c1ccncc1)NCC1CCC(NC(c2c(SC)csc2)=O)C1 N1(C(C(C)SC)=O)CC(NC(=O)C(F)(F)C(F)(F)OC(F)(F)F)CCC(O)C1 Cc1cc(F)cc(C(=O)NC2(CF)CCN(C(C34CCCN(CC3)C4)=O)C2)c1N Cc1cc(F)c(C(=O)NCC2(CCNC(C3C4CS(=O)(=O)CC34)=O)CC2)cc1F CCCCS(=O)(=O)NCC(=O)NCCCN(C(C1CC1C(F)(F)F)=O)C(C)C C1(C(=O)NCC23C(CN(C(c4c(C(C)C)ncs4)=O)C2)C3)CC2(C1)CC(F)C2 N1(C(CCC=CC)=O)CCN(C(=O)C(COc2ccccc2)OC)CCC1C C=C=CCCC(=O)NCCn1cc(C(=O)NCc2nc(C)cs2)cn1 c1(C(N2CC(F)(CNC(c3ccc(CO)o3)=O)C2)=O)ncnc(O)c1Cl N1(C(c2c(C)n(C)cn2)=O)CC2CC(C1)N(C(=O)Cn1ncccc1=O)C2 CC1CC(C(=O)N(CC(=O)NC(C2(CC(C)(C)C)CCC2)=O)C2CC2)CN1C Cc1cnc2c(C(=O)NC3CCCC34CCN(C(C3(F)CC3)=O)C4)cnn2c1 C12(NC(c3cccc(C)c3F)=O)CCN(C(c3nn(C)cc3N)=O)CCC1C2 N1(C(C(CCC)C)=O)C2CCCC1CC(NC(c1nnn3c1CSCC3)=O)C2 Cc1cc(C2CC2)ncc1C(N1CCOCC1CNC(c1ncn(C)n1)=O)=O CCC(CC)(CN=c1[nH]cnc2cc(Br)ccc12)NC(C1CC=CCO1)=O C1(NC(CCCCN(C)C)=O)CCN(C(c2c(N)cnn2C)=O)CC(C)(C)C1 c1(SC)cccc(C(=O)N(CC(C)N(C(=O)C(O)CN2CCOCC2)C)C)c1 Cc1cc(N2CCC3(CC=CCO3)CC2)nc(=NC(C)Cc2ccc(Cl)s2)[nH]1 C(=O)(C1Cc2ccccc21)N1C(C)CCC(CNC(C2CCCC2CF)=O)C1 C1(C(=O)NC2CC3CC(NC(CCC)=O)CC3C2)CC2CCC1CC2(F)F c1(N(N2CCCC2)C(=O)NCc2ccc(Sc3ccccc3)cc2)ccc(Cl)cc1 c1(C(=O)NCC2CN(C(C(C)SCCCC)=O)CC2C)cncc(C)c1C c1(C(=O)NC2(CNC(CCCc3scc(C)n3)=O)CC2)ccc2c(n1)OCCO2 C1(C(=O)NCC#CCNC(c2cc(SC)c(C)o2)=O)CC2CCCC(C1)C2(F)F CCC(O)C(C)(C)C(=O)NC1CC(NC(=O)C(Cl)=CCl)C1 C(=O)(C(F)C(C)(C)O)NCc1ccc(CN(C(=O)CCC2CCN(C)C2)C)cc1 Cc1cc(F)ccc1N(C(C1CN(C)CCO1)C(=O)NC1CCCC(C)C1)C NS(=O)(=O)c1cc(C)cc(NC2CC3CCC4C2C34)c1[N+](=O)[O-] C12(CC)CCC(C(=O)NCC(C3CCOC3)NC(c3cnns3)=O)(CC1)CO2 C1(CC=C)(NC(c2ccn(CC(C)C)n2)=O)CCCN(C(C2CC(F)(F)C2)=O)C1 C1(COC)CN(C(c2cnc(C3CC3)s2)=O)CCN1C(=O)C(O)C1CCCC1 N1(C(C2(NC(=O)C=Cc3cc[nH]n3)C(C)(C)C2)=O)CCCC(CO)(CO)C1 C12(NC(c3cc(CC)c(F)cc3)=O)CCCC1N(C(=O)C1=C(Cl)CCOC1)CC2 CC1(C)CCCC1C(=O)NCC1(C(N)=O)CN(C(c2n[nH]cc2Cl)=O)C1 N1(C(c2cc(C)sn2)=O)CCCC(C2CN(C(c3ccc(CCO)cc3)=O)C2)C1 c1(C(=O)NCC(C#C)OC)[nH]ccc1CNC(=O)C(C)C N1(C(Cc2c(C)non2)=O)CCC(O)(CNC(=O)COCc2cccnc2)CC1 c1(CNC(C(OC)OC)=O)cc(C(=O)N(C2CCOC2)C2CC2)co1 c1(C(=O)NC2C(N(C(CN(CCC)C)=O)C)CCCC2)nn(C)c2c1CSCC2 CC(C(=O)NCC1CN(C(=O)C=Cc2ccncn2)C1)C(C)S(C)(=O)=O c1(OC)cc(Cl)ccc1C(N1CC(NC(c2cnn3c2CCC3)=O)CC1C)=O N1(C(c2snc(C)c2N)=O)CCCCC2(C1)CN(C(C1CC(F)(CO)C1)=O)C2 c1(N(C)C)ccc(C(N2CC(NC(c3c[nH]nc3C(F)F)=O)C(CO)C2)=O)nc1 c1(C(=O)NCC(CCNC(CC(CC)C)=O)O)cccc(C)c1N N1(C(c2cccc(C(C)C#N)c2)=O)CCC12CCN(C(c1cc[nH]n1)=O)CC2 C1(N=[N+]=[N-])(C(=O)NC2CC3CC(OC)C3C2)CCN(C(=O)C(C)(CO)OC)C1 C1(C)(CC(=O)OCC)CCN(C(c2ccc[nH]2)=O)CC1.C1CC(=O)N1 c1(CC(=O)NC(CNC(C2CC(O)(CC#C)C2)=O)CO)ccccc1SC N1(C(CC(CN(C)C)O)=O)CCC(C)(C)C(CNC(=O)CCSCC(N)=O)C1 N1(C(C2CCS(=O)(=O)C2)=O)CCC2(CCC2)C(CNC(C2(CF)CC2)=O)C1 C(=O)(C(C)(C)CCC#N)N(C(Cn1cc(C2C(C)C2)nn1)(C)C)C1CC1 C1(NC(c2cc(CNC(COC(C)=O)=O)no2)=O)CCOC2CC12 Cc1cnc(C(=O)NCCCCN(C)C(C2(C(C)C)CNC(=O)C2)=O)c(F)c1 Cc1ccncc1CNC(C1CC(NC(=O)CCCCC2CC2)C1(C)C)=O C1(NC(CC(C)C)=O)CCN(C(=O)C(C(C)C)c2ccn(C)n2)CC1 CC1(C)CN(C(C2CC(F)(F)C2)=O)CC2(CN(c3ccnc(S(C)(=O)=O)n3)C2)O1 n1(CC)nccc1C(=O)N(CCCc1cn(CCCO)nn1)C1CC1 Cc1[nH]nc2c(C(=O)N(CCC(C)NC(c3nnc(O)nc3O)=O)C)cccc12 Cc1ncsc1C=CC(=O)NCC1CN(C(c2cccc(C3CC3)c2)=O)CC1O CCC(CC)CCCC(=O)N1CCC1CNC(=O)Cn1cnnn1 C1(=CC(=O)NC2C(CC)CN(C(=O)CCC3CC3(F)F)C2)CCC(C)(C)CC1 C1(C(=O)NCc2cccc(C#C)c2)CCC(C)(C)N(C(=O)C=CCCC(C)C)C1 c1(C(=O)NC(CCCNC(c2c(OC)nccc2)=O)(C)C)ncc(F)cc1N c12ccnc(c1)C(=O)NC2.O=C(CC(C1CCC1)C1CC1)N(C1CCCC1O)C.OCC C1(C(=O)NC2C(C(=O)NCC3OCCN(CC)C3)CC2)CC(C)(C)CCO1 c1(C(N2C(C(=O)NOCCOCCF)(CC)CCC2)=O)cc(O)nc(O)n1 Cc1nc[nH]c(=NCCC2CCN(C(C3CC4(CSC4)C3)=O)C2)c1Br c1(C(N2CCCC(CNC(C(CCC)NC(N)=O)=O)C2)=O)ncc2ccccn12 c1(C(=O)NC2CC(C)N(CC(=O)Nc3ccc(Cl)[nH]3)CC2)cncc2ccccc12 N1(C(CC(=O)NCC)=O)CCC(CNC(C2(Cl)CC2(C)C)=O)C(C)C1 c1(CNC(c2cc3ccccn3c2)=O)nc2c(s1)CN(C(C1(O)CCC1)=O)CC2 c1(C(=O)NCC2C(NC(C(C)NC(C)=O)=O)CC2)ccc(O)c(Cl)n1 C(C1=NOC2CN(C(=O)CCCS(N)(=O)=O)CC12)NC(c1noc(CC)c1C)=O C1(C(=O)NCC2C(C)CN(C(=O)CC3(O)CCOCC3)C2)CC2(CCCC2)CO1 C1(C(N(CC#C)Cc2ccco2)=O)CCC(CC)N1C(C1CCCC(=O)O1)=O N1(C(Cc2c(C)scc2)=O)CCN(C(=O)C(C#N)C(C)C)C2(CCC2)C1 c1(C(=O)NCCC(C)N(C(CCC(C)OCC)=O)C)cc(C#N)c(O)nc1N c1(OC)ccc(Cl)c(F)c1C(N1CC(CNC(=O)CC(C)OC(C)=O)C(O)C1)=O n1(CC(N2CC(CNC(C(CC)SC)=O)C2)=O)ccc2cc(Br)ccc12 C#Cc1cnc(C(=O)NCCN(C(=O)C(C(C)C)C(C)C)CC)c(C)c1 N1(C(C=C2CCC(C)C2)=O)CCCCC2(CCN(C(=O)C(c3ccccn3)C)C2)C1 C1(NC(CCSCC)=O)CN(C(=O)Cc2cnns2)C(C)(COC)C1 C(=O)(C1=NOC(C2(O)COC2)C1)N(C(CNC(c1cc(C)ncc1)=O)C1CC1)C N1(C(c2nc(CC)oc2)=O)CC2CC1C2CNC(=O)CC1(O)CCC1 Cc1cc(C)c(C(N2CC(CCCCNC(c3ccoc3C)=O)C2)=O)s1 CC1(C)C(Nc2cc(-c3cccs3)ncn2)C(C)(C)C1C(N1CC2CC1CS2)=O c1(CCNC(C(C2(C)CC2)NC(C2C(CC)OCC2)=O)=O)cnn(C)c1C C1(C)(CC)CC(C(=O)NC(C)C=Cc2ccc(OC(F)(F)F)cc2)CCO1 N1(C(C2C(C)CCC2)=O)CCCN(C(=O)C(c2cccc(C(F)(F)F)c2)O)CC1 c1(C(N(CC(CC)NC(c2cc(Cl)c[nH]2)=O)C)=O)csc(Br)n1 CCC(O)C(C)(C)C(=O)N(CC(O)CN(C(=O)CCc1ccnn1C)C)C Cc1cc(C(N2CC(NC(=O)C(F)C(F)(F)F)C(C)C2)=O)c(F)cc1F C1(C(=O)NCC2(NC(=O)Cc3nc([N+](=O)[O-])n[nH]3)CCC2)CCN2CCOCC12 C(=O)(C(F)(F)C(F)(F)F)N(C1CN(C(c2cccc(CC=C)c2)=O)C1)C1CC1 c1(C(N2C3C(N(C(CSCC(C)C)=O)C)CC(C3)C2)=O)ccc2oc(=N)[nH]c2c1 c1(NCCc2c(O)nccc2)nc(N2CCC=C(F)C2)nc2ccc(Cl)cc12 c1(CC)onc(C)c1C(=O)NC(C)CC(C)NC(C1(CC)CC(C)(C)C1)=O C1(C(=O)NCC2CCN(C(c3c(C)nc(C)o3)=O)CC2)CNC(=O)CC12CCC2 C(C(C(C)(C)C)NC(=O)C(C)(C)c1ccc(CO)s1)NC(c1c(OC)nsc1)=O C1(C(=O)NCC(CC)(CC)NC(C2C(CC)C2)=O)CCc2c(n[nH]c2C)C1 C1(CC)CCN(C(=O)C2=NOCC2)C(C(=O)N(CC(C)C(=O)OC)CC)C1 C=CCCCCCC(=O)N1CC(CNC(=O)CCCn2nc(C)nc2C)CC1C N1(C(C2(C#N)CC3(CC3)C2)=O)Cc2nccn2CC(NC(C2CC23CCC3)=O)C1 C(=O)(C(C)(F)C(=O)NC1CCN(C(=O)COC(c2ccccc2)=O)C1)OCC C(C)(CO)(C(=O)N1CCCC(SCCN(C(=O)CSC)C)C1)C(=O)C(F)(F)F.CO n1(C(C)C)nc(Br)cc1CNc1ccnn1Cc1cccc(O)c1 Cc1ccc(NC(C2CC3CN(C(C4CC45CCC5)=O)CC3C2)=O)c(C)c1O c1(C(=O)NC2C=CCN(C(Cc3ccc(C)s3)=O)C2)ccc2ccnc(O)c2n1 C(C(C)(C)NC(=O)C(F)C1CCC1)CCNC(COCCOC)=O C1(CC(N)=O)(NC(C(C)OCC=C)=O)CCN(C(C2CCCC(C)(C)C2)=O)CC1 Cc1cc2[nH]c(C(=O)OCCCCCC3CC3)cc2o1 Cc1cccc(C)c1NC(=O)CNC(C1CCC1CF)=O.C1(C=O)CCN(C)C1C c1(NC(CN2CC(n3ncc(C)c3)C2)=O)cccc(Br)c1-n1cnnn1 c1(N(Cc2[nH]nc(-c3c(C)c[nH]n3)n2)CC2CC2)cccc2ccncc12 c1(C(=O)NCC2C(NC(c3cncs3)=O)C2)c[nH]c2ccc(Cl)cc2c1=O Cc1cc(NC(C2CN(Cc3ccccc3C(=O)O)CCO2)=O)cc(F)c1 N1(C(=O)CCc2ccc[nH]2)CCC(n2cc(COCC3(O)CCCC3)nn2)C1 C1(C#CC(=O)NCC(C)CN(C(=O)CC2(C)CCCC2)C)(CC)COC1 N1(C(c2n(CC)c(O)nc2)=O)CCCC2(CCC2NC(c2cc(=O)cc[nH]2)=O)C1 N1(C(CCCC(=O)NCC)=O)CCC2(CC1)CC(NC(C1(C)CC(F)(F)C1)=O)C2 C1(CC(=O)NC2CC23CCN(C(c2cnsn2)=O)CC3)CCCCCC1(F)F Cc1ccc(CC(=O)NC(CC(=O)NC(C2CCC2)C)C2CC2)cn1 C#CCC(C(=O)NCC(C)(O)C(F)F)NC(=O)CC(COC)N(C)C C(=O)(CCCC(=O)NC(C)C(C)NC(=O)C(C)(C)C1CCOC1)NCCC C1(C(N2CCC(C)(CCC)C2)=O)CCCCN(C(c2snnc2C2CC2)=O)C1 Cc1cc(C#N)ccc1-c1nc(C(=O)NC(c2cnc[nH]2)C)c(C)s1 N1(C(C(=O)C2CCCC2)=O)CC2CC(C(N3CCOC4(CCC4)C3)=O)CC2C1 c1(C(N2CC=CC23CCCC3)=O)c[nH]c2cc(Cl)ccc12 Cc1c(F)ccc(N)c1C(=O)NCC(C)CNC(=O)CN(CC(C)(C)C)C c1(C(=O)NCC2N(C(C=CCOC)=O)CC2)csc(-c2nc[nH]n2)n1 C(C1CCOCC1)=CC(=O)NC(C(=O)N(CCCO)CC)CC1CC1 C1(NC(c2cc(C)cc(O)n2)=O)CC2CC1CN(C(c1cc3occc3s1)=O)C2 Cc1cc(=NC2CC(CN3CCCC(C)(CO)C3)C2)[nH]c(N2CCCCC2)n1 CCCC(CCCO)C(=O)NC1CCN(C(=O)C(C(C)C)c2cnn(C)c2)C1 c1(C(N(C(CNC(CCCC=C)=O)C2CC2)C)=O)noc2c1CC(C)CC2 CC1(C(=O)NCC2CC2CNC(c2cncnc2)=O)CC(F)C1 N1(C(C2CC(=C)C2)=O)CCCCC(C(=O)N(C2CC2)Cc2scnc2C)C1 c1(OCC(=O)OCC2C(C)(C)C(O)C2)ccc(Cl)c(Cl)c1 Cc1cc(C)c(N2CCC(N3CCC(OC(C)C)CC3)CC2)c(C)c1 N1(C(c2cc(C)on2)=O)CCC(C(=O)NCC(=O)NC(C)(C)C)C12CC2 c1(SC)ccc(C=CC(=O)NC(C)CCNC(=O)Cc2ccc(C#N)cc2)cc1 c1(CC)[nH]nc(C(=O)NC2C3CCN(C(C4CCCC(C)C4)=O)C23)c1Br c1(C(C)C)nc(C(=O)NCC(O)C(=O)N2CCCC2C(O)CO)co1 c1(Cc2cn(C3(C(=O)NCc4ccsc4)CC3)nn2)ccc(O)cc1 N1(C(CC(C)OC)=O)CCOC2(CCN(c3ncc(C#N)cc3Br)CC2)C1 c1(CCC)cc(C(C)C)ccc1C1CC1.C12CCCN(C1)C(=O)NC2 C1(C(=O)NC2(C)CCN(C(C(CC)(C)C)=O)CC2)CCCCC1C1CC1 C1(C2N(C(CC3N(C(C(=O)Nc4ccccc4)=O)CC3)=O)CC2)CCCCC1 c1(C(C(=O)N(CCC)CCNC(C2C(=C)C2)=O)C)ccc(OC(F)F)cc1 C(CC(C)CC)(C(=O)N1CCN(CC2CC2)CC1)NC(c1cc(OC)ncc1)=O c1(C(C)(F)F)cccc(C(=O)NCC(CO)NC(=O)CCCc2cnccn2)n1 O=C(CC(C(F)F)C1CC1)NC1CC(CCNC(C2(c3ccccc3)CC2)=O)C1 C#CCC(CC(=O)NCCOC)NC(C1CCCC(=O)CC1)=O C(=O)(N1OC2C=CC1CC2)C1N(C(C(C(C)C)(C)C)=O)CC(=O)C1 Cn1c(C(=O)NS(=O)(=O)CC23CCCC2C3)cnc1C(F)(F)F CC(c1ccccc1F)=CC(=O)N(C(CNC(=O)CCC1CCCO1)C1CC1)C CS(=O)(=O)C1(C(N2CC3CCCC3(NC(C3CCC(=O)C3)=O)C2)=O)CCSCC1 CC(=O)C(C)(C)CC(=O)NC(C)C(N1CCCC1(CO)CC1CC1)=O C12(CNC(CCc3cncc(C)c3)=O)CC(NC(=O)CC3(C)CC3)(C1)C(C)(C)O2 CC1(C)CN(C(c2ccc(CCO)cc2)=O)CC1CNC(=O)COC1CC1 C(=O)(C(CC)C(=O)N1CC(F)(CNC(c2nccc(C)c2F)=O)C1)OCC CCCCCCCCC(=O)NCC(C(C)C)NC(=O)CC(c1cccc(C)c1)C N1(C(c2c(C)ncc(Cl)c2)=O)CC2CCCC2(NC(=O)C=C2CCC(C)C2)C1 CC1COCCC1CNC(C12CC(C1)C(C)N2)=O CCCC(C(N)=O)NC(=O)C(CCC1CC1)NC(=O)CN(C)C(C)=O NS(=O)(=O)c1cccc2c1CCN(N1CCCC1C1CCCCC1O)C2 N1(C(C=CCOC)=O)CCCCC(NC(=O)C(C)CC2CCCC2)C1 c1(NC(CC)=O)cncc(C(=O)NCC2CC2NC(=O)Cn2cnnn2)c1 n1(C(C)C)cc(CC(=O)N(CC(C)N(C(C2(CCN(C)C)CC2)=O)CCO)C)cn1 N1(Cc2nc(CC)on2)CC(NC(c2conc2C(F)(F)F)=O)CCC1C C(C(=O)NCCOCCC=C)(C1CCC1)NC(C(=O)OC)C1CCCC1 N1(C(C(C)C2CCC2)=O)CCCC(CO)(NC(=O)C=CC(F)(F)F)C1 c1(C(N2CC3C(CNC(CCOC)=O)(C3)C2)=O)cc(F)ccc1I c1(C(=O)NC(C2CCN(C(Cn3ccc(C)n3)=O)C2)C)cc2c(F)cccc2[nH]1 c1(C(N2CC=C(CNC(c3c(C)scc3)=O)CC2)=O)n[nH]c2c1CSCC2 c1(NC2CC(CNC(C3CCN(C)C3)=O)C2)cc(C(=O)OC)nc(Br)c1 c1(CN(CCC#C)C(CSCC2CC2)=O)ccncc1.C1(CCC)CCC1 N1(C(c2c(C)ccnn2)=O)CCC2CCCC12CNC(=O)CC1CCSCC1 N1(C(C2(OC)CCC2)=O)CCCC(F)(C(=O)N(C)Cc2ccc(C)cc2)C1 CCC(CC(=O)N1CC2(CC(NC(=O)C(F)(F)CC)C2)C1)C(C)C CC(CCNC(=O)CCC1(NC(=O)CC2CCCC2)CCC1)C(F)F c1(C(N2C(CNC(C(CC=C)NC(C)=O)=O)C=CC2)=O)nc(OC)ccc1C CCC(CC(=O)NC1CC(CO)N(C(=O)CC2(C)OCCO2)C1)C(C)C CCCCC(C)C(=O)N1CCN(C(=O)CCOc2ccc(C(C)C)cc2)C2CC12 C(N=c1[nH]c2cc(F)c(F)cc2[nH]1)c1n(C(c2cccc(C#N)c2)C)ccn1 C1(C(C)C)CCN(C(c2cnc[nH]2)=O)C(CNC(C2CC2c2cc[nH]n2)=O)C1 N1(C(c2c(CC)nc(C)s2)=O)CCN(C)C(CNC(=O)C(C)(C)C2CC2)C1 C(C(=O)NC1(CO)CCN(C(=O)Cn2cc(C3CC3)nn2)C1)(C(C)C)SCC C12(CNC(=NCc3ccc(OC)cc3)NC3CCSC3)CCC(C1)C(C)(C)O2 C#CC1(O)CN(C(C2CSCN2C(c2sccc2CO)=O)=O)C1 C1(C(=O)NCC2N(C(c3c(-c4ccc(C)o4)onc3)=O)CC2)CC2(C1)CC(C)C2 N1(C(CN(CCOC)C)=O)CCCC1C1CCCCN1C(c1sccc1Cl)=O C12(CC(F)(F)C1)C(=O)NCCN2.c1(NS(C)(=O)=O)nc(C(C)(C)C)cs1 C#CCCC(O)C(=O)N1CCC(CNC(c2ccncc2Br)=O)(OC)C1 C#CC1(C(N2CC(O)(c3cn(CCC(=O)OCC)nn3)C2)=O)CCCC1 c1(CCC(N2CC(F)(N(C(C=CC=CC)=O)CC3CCCC3)C2)=O)cccc(O)c1 n1(CC)nc(C)c(C(=O)NCCOC(C)(C)CNC(=O)CC(CC)C(=O)OC)c1C N1(C(c2n(CCOC)ncc2)=O)CC(C)(C)OCC1CNC(=O)C1=C(C)CC1 c1(C(N(C)CC2(CNC(CSCC#C)=O)CC2)=O)cnn2c1OCCC2 C(=O)(C1=CS(=O)(=O)c2ccccc21)NCC1(O)CN(C(C2C(C=C)C2)=O)C1 C(=O)(C(F)(F)C1CC1)NC(CNC(CCN(CCCCC)C)=O)C N1(C(CCSCC)=O)CCN(C(C2CCCOC2C)=O)C(C2CCCC2)C1 C1(NC(C#CC(C)C)=O)CCC(C)(NC(C2CC2c2ccccn2)=O)CC1 C1(CC)CC(C(=O)NCC2(F)CN(C(C3CCCCCC3)=O)C2)CC(=O)N1 c1(NC(C2(C(C)NC(=O)CC3CC4CCC3O4)CC2)=O)ccc(F)c(F)c1 Cc1ccn(C)c1CC(=O)NC1CC(CC(=O)NC(C)(C)CN(C)C)CCO1 S(=O)(=O)(c1cccc(=NCc2ccco2)[nH]1)NCc1scc(C(N)=O)n1 C=CC1(CC(N2CCC(C(C3CC3)OC)CC2)=O)CN(C(=O)C=CC)C1 Cc1ccc2c(CC(N3CCC(NC(c4cnsc4)=O)CC3)=O)ccc(O)c2n1 C1(CNC(C(F)=CC)=O)CCCCCN1C(c1ccc(OCF)cc1)=O C(C)(N=c1nc2scnc2c(N(C)Cc2ccc(Cl)c(Cl)c2)[nH]1)n1ncc(C)c1 N1(C(c2ccc(C(N)=O)[nH]2)=O)CC2(C=C(C(=O)N3CCCCCCCC3)CO2)C1 N1(C(C(C)SC(C)C)=O)CCC2CC2(C(N2CC(OCC(C)C)C2)=O)CC1 C(=O)(CCCC(C)(C)C)NC1(CNC(n2ccc(=O)n(C)c2=O)=O)CC(OC)C1 C(=O)(CCCC(N)=O)NCCOC1CN(C(C(CC)C)=O)C1 C(=O)(CS(=O)(=O)C1CCCC1)NC1CCC(CNC(C(C)C(C)(F)F)=O)C1 CCC(CC)CCC(=O)N1CCC(C2CCCN2C(=O)CC2(OC)CCCC2)C1 C12(NC(c3ccc(=O)oc3)=O)CCCC1N(c1nc(Cl)ncc1F)CC2 C1(CNC(C2ON=C(C(C)C)C2)=O)(NC(=O)C=CCO)CC2CCC1CC2 N1(C(C2C(=C)C2)=O)CCc2sccc2C1CNC(c1c(C)nc(CC)nc1C)=O C(=O)(CCCC(F)(F)CO)N1CCC(CCNC(c2c(C)cc(C)s2)=O)C1 c1(CNC(C2(OC)CCN(C(C)=O)C2)=O)cc2cncc(Br)c2o1 C(=O)(C1CCc2ccccc21)N1CC2CC(NC(c3c(Cl)ncc(C)c3)=O)C2C1 C(c1ccc(Br)o1)=CC(N1C(c2cc(C)no2)CCC1)=O C(=O)(CCCn1ccnn1)NCC(CNC(=O)CCC1OCCO1)OC CCCCC(O)C(=O)N1CCOC(CCNC(=O)C(=O)Nc2ccc(Cl)cc2)C1 C1(NC(c2cn(C)c(=O)n2C)=O)CCCCC12CCN(c1cncc(Cl)n1)CC2 N1(C(c2n(CC=C)ccc2)=O)CCOCC1CCNC(=O)C(C)CNS(C)(=O)=O CC(C(=O)N(CCCOCCN(C)C)CCO)N(C1(CC2CCC2)CC1)C S(=O)(=O)(c1nc(N(C2CCCCC2)N(C2CCC2)C)ccc1Br)NC(C=C)COC C1(C2(O)CCC2)(C(=O)NCC(N2CC3CC3(CO)C2)=O)CC1 c1(NCCN2CCN(C(=O)NCC3(C)CN(S(C)(=O)=O)C3)CC2)cc(Cl)ccc1I CCCCC(O)C(C)C(=O)N(CCNC(C1CCCC1F)=O)CC N1(C(CCCSC)=O)CCC(CNC(C2CCCN2C)=O)C(F)(F)CC1 C1(C(=O)NCCOC(C)C)CC(O)CN1C(=O)Cc1cn(C)nn1 N1(C(C2(NC(C(c3n(C)ncc3)=O)=O)CCSC2)=O)CC(S(C)(=N)=O)C1 CC1CC(C(=O)NCC(=C2CN(C(=O)CCN3CCCCC3)C2)F)CC(C)C1 CCCC(C#N)C(=O)N1CC(O)CC1C(=O)NCC(=O)N(C)CC N1(C(C(C(C)O)N(C)C)=O)CCCCCC1C(=O)NCCn1cccn1 c1(C(C)C)ccc(C(=O)COC(=O)C(c2cnn(C)c2)C)cc1 C1(C(N2CCN(CCNC(c3n(C=C)ncc3)=O)CC2)=O)CC2C(C1)C2(F)F N1(C(C2(CC)CC(F)(F)C2)=O)CCCC(CNC(=O)C(F)=CC2CC2)(OC)C1 c1(C(=O)NCC2N(C(c3c(CCC)ocn3)=O)CC2)cc(CC)c(=O)n(C)c1 C1(CC=C)(C(=O)NCCc2csnn2)CCN(C(=O)CC(C)F)C1 C(CN=C(NCC1CC1)NC1CCC1(C)C)c1cc(C)sc1C S(=O)(=O)(c1cc2sc(=NC(C)c3nccn3CC)[nH]c2cc1Cl)NC(CC)C(C)C N1(C(c2c(C)occ2)=O)CCC(C2CC(NC(=O)Cc3cc(F)ccc3F)C2)C1 c1(CC(=O)NCCC(C=C)(C)C)nc(C)c(C)n1-c1ccccc1 c1(NC(C2CCN(C(CCCC#CC)=O)C2CC)=O)ccc(C)c(C#N)c1 CC(C(=O)NCCN(C(=O)CNC(=O)C1CC1)C)NC(C1CCCC1)=O N1(C(CCc2c(C)nccc2)=O)CCC2CN(C(c3cc(C#N)c[nH]3)=O)CC12 C(C(C)C(C)C(=O)NCCCCC(C)NC(=O)C=CC1CCCCCC1)OC CCCCC(C(=O)NC1CCN(C)CC1C)NC(=O)CCCCC1CC1 Cc1cccc(C)c1C(=O)NC(C1CCN(C(c2csc(C)c2C)=O)C1)C c1(C(=O)NCc2c(C(=O)OC)cn[nH]2)cc(S(N)(=O)=O)ccc1Cl CC1=C(C)CN(c2ncnc(NCc3cnn(CC(C)C)c3C)c2C)CC1 C1(NC(CCOC)=O)CCCN(C(C2(NC(C)C)CCCCC2)=O)CC1 c1(C(=O)NC2CC(NC(CCC(C)SC)=O)C2)cc([N+](=O)[O-])ccc1SCCO c1(C(N(CC(C)(C)NC(c2nc(C(=O)OCC)sc2)=O)C)=O)cc2c(s1)CCC2 C1(C(N2CCC(OCC#C)C2)=O)(CC)CCCN1C(=O)COc1ccccc1 C(c1ccccc1)=CCC(=O)N(CC(C(=O)NC(c1cccs1)C)C)C Cc1cccc(NC(c2cc(C)n(CC3CC3)c2C)=O)c1Cl CCC(CNC(=O)C(C)C(C)NC(=O)Cc1nonc1C)CC(C)C c1(C(N2C(C(=O)NCCC)CC(F)C2)=O)ccc(OC)c(O)c1O C(CCC=O)(C(C)C)NC(c1cc(-c2ccccc2)nn1C)=O.C=C1CC(C)C1 C(=O)(C(F)CC(C)(C)NC(c1cnc(OC)nc1)=O)N(C(C#C)C)C c1(OC)cccnc1C(F)(F)C(=O)N(C(F)CO)CC(C)C c1(C(C)NC(c2n(CC(=C)C)nnn2)c2occc2CC)ccc2c(c1)CCC2 C(C(=O)NNC(=O)OC1CN(C(c2cnc(OCC(C)(C)C)s2)=O)C1)C(C(C)C)C c1(C(=O)NC2CCCCN(C(COCCOCC#C)=O)C2)cc(C)c(Cl)cc1F N1(C(Cc2ncn(C)c2)=O)CC2CCN(C(=O)COCCF)C2C1 C#CCCC(C(=O)Nc1cnn(CC#C)c1)NC(=O)CCC(C)CN(C)C C1(C2(C=C)CCC2)(C(N2CC(NC(C(CN(C)C)(C)C)=O)C(O)CC2)=O)CCC1 c1(OCC(CC2(N(CCCN)C)CC2)O)cccc(NC(C(CC)C)=O)c1 C1(C(=O)NC(CNC(C(C)SCCCC)=O)(CC)CC)CCC2(CCC2)C1 c1(C(=O)Nc2scc(C(=O)OCc3ccc(F)cc3F)n2)cc(Cl)cc2cc[nH]c12 N1(CCOC)CCN(C(=NCCc2nccs2)NCc2cnc3n2CCC3)CC1 n1(CC(=O)NCCC2CCC(NCC3C(C(=O)OCC)CC3)C2)cc(C#N)cn1 C1(CC(N2CC(NC(CNC(CC)=O)=O)(CC)C2)=O)CCCCN1C N1(C(Cc2c(C)nsc2)=O)CC2CN(C(=O)Cc3coc4ccccc34)CC2C1 C(CCC(CCC)NC(=O)C(N1CCCCC1)=O)OCCCCCCC N1(C(C2N(C(CCN(C)C)=O)CCC2)=O)CCN2C(=O)CCC2C1 C=CC(C)(O)CC(=O)N(CCC(C(C)C)NC(=O)C=Cc1ccco1)C C1(NC(C2C(=C)CC2)=O)(CNC(=O)CCOCC2CCC2)CCC(C)(C)CC1 Cc1cc(C(=O)NC2(C)CC(NC(c3coc(C(F)F)c3)=O)C2)n2ncnc2n1 C1(NC(=O)OC)CCN(C(=O)CC(C2CC2)NC(=O)CCc2ccncn2)C1 c1(OC)ccccc1CNC(=O)NC1CCC(c2ccccc2)C1 C12CCCCC1NC1(c3ccccc3Cl)CN(C1)C(=O)N2.n1(C(C)C)cncn1 CC(C)(C)C(C(=O)N1CCCC(NC(=O)C=Cc2cccnc2)CC1)C1CCC1 C1(NC(C(C)NC(c2ccco2)=O)=O)CCC(NC(C2CN(C)C2)=O)C1 c1(CN2CCC(NC(N(c3cccnc3)C)=O)C2)cccc2cccnc12 C#Cc1ccc(C(=O)NCC2(C(F)F)CCN(C(C3(CCF)CC3)=O)C2)nc1 C1(CNC(=O)C2=CCCSC2)CC2CCC(C1)N2C(C1CC2CCC1C2)=O c1(N(CCOCC=C)C)nc2ccsc2c(=NCc2cn3c(n2)SCC3)[nH]1 C(=O)(C(C)(O)C(F)(F)F)NC1CN(C(c2c(OCCC)cccc2)=O)CC1SC c1(C(C)(C)C)cnn2c(C(N3CCC=C(CCn4cc(CO)nn4)C3)=O)ccnc12 Cc1cc(N(C)C)ccc1C(=O)NCCC1(NC(=O)COC2CCOC2)CC1.C(N)=O C1(CC)C=CCN(C(=O)CC(C)(C)NC(=O)C(O)C(C)C)C1 N1(C(c2c(C)ncc(Cl)c2)=O)CCC2CC1CN(C(=O)Cc1ccccc1F)C2 C1(C(N2CC(NC(CC=C=C)=O)C(F)CC2)=O)CCN(S(N)(=O)=O)CC1 CC1=CCC(N(c2ccccc2)C(=O)CC2CCN2C(=O)C#CC2CC2)CC1 N1(C(C2C(C(=O)OC)CC=CC2)=O)CCCc2c(F)cc(F)cc21 Cc1ccc(-c2nc(C)c(C(=O)NC3(C)CN(C(C4C(C)C4C)=O)C3)s2)c(C)c1 N1(Cc2c(COC)cccc2)C(=O)NC(c2cnccn2)C1=O N1(C(=O)NC2C(C#C)OCC2)CCCC(O)(C(F)F)C1 C12(C(=O)NCC(C)NC(c3c(OC)noc3C)=O)CC3CC(F)(C1)CC(F)(C3)C2 C(=O)(C1=NN(C2CC2)C(=O)CC1)NC(CNC(c1nc(C)sc1C)=O)C1CC1 N1(C(NC)=O)CCC(CCCO)CC1.c1(CC(C(=O)CCCC)=O)nccn1C c1(C(N2CC(C3C(=O)NCCS3)C2)=O)ncnn1C(C)C.CCOCC C1(C(=O)NCC=C(Cl)Cl)CCCCCCN1C(C1CCC2CC1CO2)=O CCCCC(F)C(=O)NC(Cc1cn[nH]c1)C(=O)N1CC(c2n[nH]c(C)n2)C1 C1(SC)CN(C(=O)Cc2cc(C)cs2)CC1n1cc(C2CCN(C)C2)nn1 Cc1coc(C2CC2)c1C(N1CC(NC(C2NC(=O)OC2C)=O)C(C)C1)=O CCC(F)(F)CC(=O)NC(C)(CNC(=O)CC1CCC(C)CC1)C1CC1 C1(c2n(CCCCC)c(N3CCSC(C(C)C)C3)nn2)C(C)(C)CCCC1(C)C C1(C(=O)NCc2cccc(C)c2)CC2(CCN1C(=O)C(O)CC1CCCC1)CC2 C1(C)(C(N(CCOCCCNC(C2CC(SC)C2)=O)C)=O)C=CCC1 c1(NC(C2CCCN(C(C(=O)OCC#C)C)C2)=O)csc2cncn12 C1(C(N2CCCC(C(F)(F)F)C2)=O)N(C(C2CCCC23CCC3)=O)CC12CCCC2 n1(CC(=O)N(C2CCN(C(c3cc(F)c[nH]3)=O)C2)CCC)cc2ncccc2n1 CCC(C)CCCC(=O)N(CCNC(C1OCC2CCCC1C2)=O)CC c1(OC)ccc(C(=O)C(=O)NC2CCN(C(c3cnc(C4CC4)[nH]3)=O)C2)cc1 C(CCCCCC(=O)NCC1CCC1(F)F)NC(CCCC)=O CC(C)C(C)C(C)CC(=O)N1CCN(C(=O)CC(C)(C)C)CC1c1ccccn1 CCCCC(C(=O)NC(CC(=O)NCCCCC1CC1C)C(C)(C)C)C(C)C C1(NC(C(COCC)C)=O)CC2CC(NC(c3ccc(CF)cc3)=O)C2C1 C(=O)(CCCn1nnnc1C(C1CC1CO)NCc1cnc(C)s1)OC C(=O)(C1CCCc2nc[nH]c21)NC1CCC(C)N(C(c2cnc(C(C)O)s2)=O)C1 C1(C(=O)NCC2CN(C(C#CC3(C)CC3)=O)CC2O)Cc2cccc(F)c2O1 c1(CCCNC(C2(C)CN(C(C3CC3C3CC3)=O)C2)=O)cccc(F)c1 N=C(N)NC(=N)N1CCN(c2ncccc2C(F)(F)F)CC1 c1(C(=O)NCC(CNC(C(CN(C)C)(C)C)=O)F)c(N)c(F)cc(F)c1F c1(C(N2C(CNC(C(C)O)=O)C=CC2)=O)ccc2ccccc2c1F N1(C(C(=CC2CCCC2)C)=O)CC2CC2(CNC(c2nc(C)oc2C)=O)C1 N1(N(C(c2ccc(O)c(O)c2)CNC(C)C)C)CCC2(N)CC2C1.Cc1[nH]nc(O)c1CC C1(OC)CN(C(=O)C=C(C)C)CC1NC(c1ccnc(OCCO)c1)=O c1(OCC=C)ccc(C(=O)NCCC(C)NC(=O)OC(C)(C)C)cc1 c1(C(=O)NC(CC)(C)CNC(=O)CCN(CCO)CCO)cc(Cl)n(C)n1 Cc1ccc(CC(CCBr)NC(c2c(C)nn(C)c2-n2ccnc2C)=O)cc1Br C1(C(=O)NCCNC(C(CC(C)C)C)=O)Cc2ccccc2C(C)(C)C1 N1(C(C2(COC)CC(=C)C2)=O)CCCCC1CNC(=O)CC1CC(F)(F)C1 C12(CNC(c3onc(C)c3C)=O)CCC1CN(C(c1c[nH]nc1C1CC1)=O)C2 c1(COC)cccc(C(=O)NCC#CCNC(c2ccncc2Cl)=O)c1C c1(OC)cccc(O)c1CN1CCC(C(=O)NC2CC(=O)N(C3CCCCC3)C2)C1 c1(N2CC=CC(NC(C(C(C)O)(F)F)=O)C2)ncnc2c1CCC2 c1(C(N(C)CCNC(=O)CCc2ccc(F)nc2)=O)cccc2c(C#N)c[nH]c12 c1(C(=O)NCC(CO)NC(C2N(CC)CCC2)=O)cnn(C)c1N C(C(C)CN=c1[nH]nc(C(C)(C)C)s1)NC(COC(CC)C)=O C=CCCCCCC(=O)N1CC(=O)NCC1C(=O)NCCC(C)C(C)C N1(CC(=O)N(C2CCCC2)CCCNC(c2cocc2C(N)=O)=O)CCSCC1 c1(C(N2CCC(NC(C=C(C)C)=O)C(C(C)C)C2)=O)ccc2nn[nH]c2n1 N1(C(C(C)C2CC2)=O)CCCCC(NC(=O)CN2CCCC2=O)C1 c1(C(=O)NCC23C(CN(C(CSC)=O)C2)C3)c(C)ccc(Br)c1C C(C(=O)OCC1C=CCCCC1)(C(C)C)Sc1cn(CC)nc1 CC(C)CCC(=O)NCCOCCOCCN(C)C(C1(S(C)(=O)=O)CC1)=O C12(CNC(CSc3nc(C)[nH]n3)=O)CN(C(=O)CSC(C)(C)C)CC1CCO2 C1(NC(Cc2c(C)n(C)nc2)=O)CCN(C(=O)CC2CC(F)C2)CCC1CO C1(C(N2C3CN(C(CSc4cccc(C)c4)=O)C(C3)C2)=O)CN2CCN1CC2C C(=O)(CS(=O)(=O)CCO)N(CCCNC(=O)CC1CCC1OC)CC N1(Cc2c(C)nc[nH]2)CCC(F)(F)C(CNC(c2ccccc2Cl)=O)C1 Cc1ccc(F)c(C(N2CCCOC(CNC(=O)C(C)n3cccc3)C2)=O)c1 N1(C(C2N(C(c3c(C#C)cn(C)n3)=O)CC(=O)NC2)=O)CCOC2(CCC2)C1 c1(C(N2CCCC(N(C(=O)CC3(COC)CC3)CC)C2)=O)c[nH]c2ncccc12 N1(C(c2onc(C)n2)=O)CCC2(CC1)CC2C(N1CCC2(CCOC2)C1)=O c1(CN2CC(NC(=O)Cc3ccccc3N3CCCCC3)C2)cccc(O)c1O c1(C(=O)NCC2C(NC(C(CC3CC3)OC)=O)CCC2)cccc2c1C(=O)NC2 c1(OC)cc(C(N2CC(CC(=O)N(C)Cc3ccns3)CC2C)=O)nn1C O(NC(=O)C=Cc1cc[nH]n1)CC1CC1.C12CN(C1)C2=O C1(C(N2C(CNC(C3CC(O)CN3CC(C)C)=O)CC3CC23)=O)(OC)CCCCC1 N1(C(C2CCC(C(=O)NCc3c(C)n(C)nc3)C2)=O)CCOc2ccccc2C1 N1(C(COc2ccc(C)cc2F)=O)CC2CN(C(c3nccc(C)n3)=O)CC2C1 C1(C(N(C(CO)C2CC2)C)=O)N(C(C2(O)CCCCC2)=O)CCCC1(C)C C(=O)(C1COCc2ccccc21)NCCC1(CNC(c2cc(C)oc2C)=O)CC1 c1(N2CC3C(CCN(C(c4ccnn(C)c4=O)=O)C4CC4)C3C2)cccc(F)c1C#N n1(CCCCNC(=O)CC2CSC2)cc(CCCCCN2CCOCC2)nn1 C1(NC(C=CC(C)C)=O)CCN(C(=O)CC(O)CN(C)C)CC(C)(C)C1 C(C)(C)(CC(=O)NCC1(F)CN(C(C2CC2c2cccc(Cl)c2)=O)C1)N(C)C CC1(NC(c2ncccc2Cl)=O)CCN(C(C2(C)CC=CCC2)=O)CC1 CCCC(CC)CCC(=O)NC1(C(=O)NCc2cnn(C)c2)CCCC1 C12(CNC(C3C(=C)CC3)=O)CCCC1N(C(c1nncs1)=O)CCC2 C1(C(=O)NCCNC(C(c2cccc(Cl)c2)(C)C)=O)COCCN1C1CCCC1 CN1C(=O)OCC1C(=O)NC1C2CN(C(C3CC(Cl)(Cl)C3)=O)CC12 C1(C)(CN(C(CC(c2cn(CCC)nn2)OC)=O)CC)CCCS1(=O)=O C1(NC(c2c(C)nc(CO)s2)=O)CCN(C(c2c(C)nc(C)n2O)=O)C1(C)C c1(CC(=O)N(C2CCN(C(Cn3ncc(C)c3)=O)CC2)CCO)ccc(C)c(Cl)c1 c1(-c2cn(CCC(=O)NC3CC4C(NC(N)=O)C4C3)nn2)ncn2c1CCCC2 c1(C(=O)NCC(C)(C)NC(C(C)SC)=O)cc(C)c2ncccc2c1C c1(C(=O)NC2C(CNC(CC3ON=C(C)C3)=O)CC2)cc(S(=O)(=O)NC(C)C)c[nH]1 c1(C(C)NC(c2ccc(C(=O)O)o2)C)cccc(F)n1 N1(C(c2cc3[nH]cc(-c4cn(C)nc4)c3cc2)=O)CCC(C2CCOCC2)C1 c1(C(CNC(CC2(C=C)CC2)=O)NC(=O)C(C2CCC2)C2CC2)ccccc1F C1(NC(c2c(CC)cccc2)=O)CCN(C(=O)CC2(C)CC2(Cl)Cl)CC1F N1(C(CN(CC)CC)=O)CCC2CN(C(=O)Cc3ccnn3C(F)F)CCC12 C(C)(C(CCC=O)N=c1ccnc2[nH][nH]cc1-2)c1cccc(OC)c1 CCC(C)(CC(=O)N1CCC(C(C)(C)NC(c2cc(C)no2)=O)CC1)C(=O)OC N1(C(CCCc2[nH]c(=N)sc2)=O)CCCC(CNC(C2CC3(CC3)CO2)=O)CC1 N1(C(CC2C(NC(c3c(CC)cc[nH]3)=O)CCCC2)=O)C2CCCC1CC2 c1(C(=O)NC2CC(N(C(CCC=CC(C)C)=O)C)C2)cc(Cl)c(Br)[nH]1 C(=O)(C(O)CC1CC1)N(CCN(C(=O)CC(n1cccc1)C1CC1)CC)CC C1(CNC(CN(C(=O)C2=CCCC2)C)=O)CCCC(F)C1 C1(C(=O)NCCCNC(C2(c3cc[nH]n3)CC2)=O)CC12CCOC2 N1(C(C(=O)NCC=C)COC)CCCC(C(C)C)(COC)C1 C(C(C(C)(C)C)NC(=O)NCc1ccccc1)NC(=O)NC(C=CC)C1CC1 C1(C(=O)NCC2(CNC(C3(C)CC3(F)F)=O)CC2)CCCC(=O)O1 C1(CC(=O)N(C2CCC(NC(c3sccc3C3CC3)=O)CC2)C)CCCCCO1 CC1CC(NC(c2cnn(CC(F)(F)F)c2)=O)CN(C(C2CCCC2)=O)C1 c1(C(=O)NC2C(NC(C(c3c(C)noc3C)C)=O)COCC2)cccc(Cl)c1F N1(C(Cc2c(C)nsc2)=O)CCC(CCCNC(c2nc(Cl)c(Cl)s2)=O)CC1 N1(C(c2c(C)ccn2C)=O)CCc2c(CNC(=O)CC3(C)CC3F)cccc2C1 N1(C(Cc2ccc(OC)cc2C)=O)CCCC12CCN(C(C1(C)CC(C)C1)=O)C2 C1(NC(c2cc(C)no2)=O)CCC(C)(CNC(c2cnc(=N)[nH]c2)=O)CC1 C1(C(=O)O)(CC)CN(C(=O)C(F)=CC(C)(C)C)C1 c1(C(=O)NCC#CCNC(CCN(CCCCOCC)C)=O)n[nH]cc1[N+](=O)[O-] c1(OC)ccc(C(F)(F)C(=O)NC2CN(C(=O)C=CCN(C)C)CC2C)cc1 c1(OCC)cc(C(=O)NC(C)(CNC(=O)C(C2CCCC2)OC)CC)[nH]n1 c1(CCC)n[nH]cc1C(=O)NCc1cc(C(=O)N(CCCO)CC(C)O)cs1 n1(CCNCc2c(C)nco2)c(C)nc2ccccc12.C1C(=O)O1 c1(CC)nn(C)c(C(N2CCC(NC(c3cc(CC)c[nH]3)=O)C(F)C2)=O)c1Cl C1(C2(N(C(=O)C)C)CC2)CCCN1C(C1(C(=O)O)CC1)=O.c1ccsc1 c1(CC(=O)N(C(c2cccc(Cl)c2Cl)C(=O)OC)C)ccc(C(F)(F)F)c(F)c1 c1(OC(=O)C2=CCCCC2)cccc2c(Cl)nccc12 Cc1nnc2n1CC(C(N1CCCC(N(C)C(c3csc4nccn34)=O)C1)=O)C2 C1(C(=O)NCCC(CNC(=O)C2=CC(C)(C)C2)OC)CC2CCCCC2O1 c12occc1C1=CCN(CC1)CC(=O)N2.C(=O)(N=c1scc(C(=O)O)cc1C)OC c1(C(N2CCC(C(=O)NCCN3CCOC3=O)C2)=O)cc(F)cc(F)c1O c1(C(N2CC(OCCNC(CNC(C)=O)=O)C2)=O)c(C)csc1Cl c1(C(N2CCC(CCNC(c3nnn(C)c3N)=O)C2)=O)ccc2c(c1)CCC=C2 c1(C(C)C)cc(C(=O)NC(C(C)NC(c2cccc(Cl)c2)=O)C(C)C)ccc1F c1(C(=O)NCC2C(NC(C34CC(C)(C3)C4)=O)CC2)cc(C(F)F)ccc1O Cc1cc(=O)n(C)nc1C(=O)NCCCC1CCN(C(C2CCC2(C)C)=O)CC1 c1(CN2CCC(NC(c3cnco3)C)C2C)cccc([N+](=O)[O-])c1 C1(NC(=O)CCc2cscn2)CN(C(=O)CC2CS(=O)(=O)C2)CCC12CCC2 c1(C(=O)NCC(C)N(C(=O)CC2CC2c2cnc[nH]2)C)ccccc1CC#N CC1CCCCC1(C)C(N1CC2(C1)CN(C(c1cc(O)ccc1Cl)=O)C2)=O N1(C(c2n[nH]c(CC)c2Br)=O)CC2CC(NC(=O)C(C)(C)N3CCCC3)C1C2 c1(C(=O)NCC2N(C(CCCC#C)=O)C3C(C2)C3)ccc(C)cc1C(C)=O c1(OC)cc(F)ccc1CC1CCCN(C(c2cnccc2N(C)C)=O)CC1 C1(NC(C(C)Oc2c(OC)cccc2)=O)CCN(C(=O)CC2CC2)CCC1CO N12CCOC(C1)C2=O.c1(C(C(=O)NCCC2CC(SC)C2)N(C)C)cncn1C N1(C(COCCCC)=O)CCCCCC(NC(C2CC3(C2)CC(O)C3)=O)C1 C1(C(=O)OC)CCCC(C(N2CC3(NC(=O)CCCC4CCC4)CC2C3)=O)C1 Cc1nccc(Br)c1NC(C1CCN(c2ccccc2)CC1C)=O C1(C=O)C2CC3C(C2)C13.C(=O)(C(F)C=CC=C)N(CCC)CCNC(C)=O C=CCC(C)(C(F)F)NC(=O)C(C)CC=CCC.C1=CC(=O)NC(C)(C)C1 c1(C(=O)NCC(CC)NC(C2NC(=O)C3CC23)=O)c(F)ccc2c1OCC2 C(=O)(C(O)CC(F)F)NCC12CC(NC(CC3C(OC)COCC3)=O)(C1)C2 c1(SCC)ccccc1C(=O)NCC(C(C)C)NC(=O)CCCC1CC1 Cc1nnc(C(=O)NCC2CC(F)(CNC(=O)CCCc3sccc3C)C2)s1 c1(OC)ccc(CC(=O)N(CC(=O)NC(c2cscn2)CO)C(C)C)nc1 Cc1ccc(Br)c(F)c1C(=O)OCC(=O)N(CC(N)=O)C CC1N(C(C2(CNC(=O)C3=CCCC3C)CCCCC2)=O)CCCC12CCC2 c12cnn3cc(cnc13)NC2=O.N1(S(C(C)C)(=O)=O)CCOC(C(F)(F)F)C1 O=C(Cc1cccnc1)NNC(=O)c1ccc(CNSc2ccc(Cl)cc2)o1 c1(COC(=O)Cc2cccc(F)c2Br)cc2c(o1)CCCC2 C1(C(=O)NC2CC(C)(C)N(C(C3(CC4CC4)CC3)=O)C2)CNC(=O)CC1(C)C CCC1(C)CNC(=O)CN(C)N(Cc2ccccc2)C1=O.C1(NC(C)=O)CCCC1 c1(C(N(C2CCN(C(C3CCCN3C)=O)C2)C)=O)c[nH]c2cc(Br)ccc12 C(=O)(CC1=CCCC1)NC1CC(C(N(OC)C)=O)C1(C)C c1(C(=O)NC2CC(CNC(c3cc(C)nnc3)=O)C2)cc2occc2[nH]1 c1(CSCC(=O)NCCN(C(=O)CC2CCCO2)CCC)ccc(Cl)cc1 CC1=C(C(=O)N2CC(C)(OCC(N3CCn4ccnc43)=O)C2)CCCO1 c1(C(=O)NCC(=C)CCNC(=O)COC(C)CC)ccncc1C(F)(F)F c1(C(N2CC(CNC(c3nc(OC)oc3)=O)C(C)C2)=O)cc2cnn(C)c2s1 CCCC(C)(C)CC(=O)N1CC(NC(c2cc(C#N)cs2)=O)C(C)C1 c12cn(nn1)CCCN(C)C(=O)C1(CC1)CCO2.C(=O)(C1CC1)N.COC c1(C(=O)NC(C(C)NC(c2c(CCC)occ2)=O)C)onc(Br)c1C c1(SC)ccccc1NC(=O)C(CCN(C)C)NC(=O)CCc1ccn(C)n1 Cc1nc(C)c(CC(=O)NCC2(NC(c3c[nH]nc3Cl)=O)CCOC2)s1 CN1CCCCC1CCCC(N1CCCCC1CNC(=O)CNS(C)(=O)=O)=O C(CCN=c1[nH]cc2ccnc-2[nH]1)N1CCN(C(c2cccc3sncc23)=O)CC1 C(=O)(C(C)(C)CCCF)N1CCN(C2N(C(CSCCCC)=O)CCC2)CC1 N1(C(C(CC#C)CC#C)=O)CCCC12CCN(C(C1OCC3CCCC13)=O)CC2 Cc1c(Cl)ncc(F)c1CNC(c1cncc(-n2ccnc2)n1)=O c1(N(CCCC)C(=O)Cn2cc(Cl)cn2)[nH]c(C)cc1C.N1CCC(=CC)CC1 C(=O)(C(O)(C(F)(F)F)NC(=O)CC(C)C)NCC1(OC)CCOC1 C1(N(C(C=NOC)=O)C)CCCC2CN(C(=O)CSC(C)C)CC12 c1(C(N2CCC(CN(C(=O)C=C3CC3)C)C2)=O)csc2ccccc12 C(=O)(C(C(C)C)C(C)C)NC1(C(=O)NC(C(=O)NC)C)CC1 C1(C(=O)NCCCNC(CN(C)C(=O)OC(C)(C)C)=O)C2CCC12 C1(C(=O)NCC(C2CCN(C(C3CNC(=O)N3)=O)CC2)C)CCCN1C=O C1(C(=O)NC(C(CC)(C)C)c2ccccc2)CCCN(CCn2cc(Cl)cn2)CC1 N#Cc1cnc(NC(C2CC23CN(C(C2CCCCO2)=O)C3)=O)c(Cl)c1 C(=O)(C(C(=O)NCC1CCCN1C(=O)CCCc1ccc(C)s1)C(C)C)OCC c1(C(=O)NC2CC(C)(NC(C(CCSC)O)=O)C2)c[nH]c2nccc(Cl)c12 N1(C(C2C(NC(CC(=O)OCC)=O)CCCC2)=O)CC2(COC(C)C2)C1 C=C1CCN(C(c2cnnc(O)c2)=O)C(C(=O)NC2CN(C(N)=O)C2)C1 C1(=O)C(Cn2cncn2)N1.C12(O)CN(C1)C(=O)C2.C1(C(N)=O)CC1(F)F c1(NCc2[nH]nc(OCC)n2)cc(I)c(Br)c(F)c1F c1(C(N2CC(C)C(C)CC2)C(=O)NC2(C)CC2)cccc2c1OCCO2 Cc1cc(=O)n(C)cc1C(N1CCC(NC(=O)C2=CS(=O)CCC2)C(C)(C)C1)=O Cc1cc(=NC(=O)C(=O)NCC2(O)CC(NC(=O)C(CC(C)C)C(N)=O)C2)[nH]o1 c1(N2CCC(O)(C(=O)NCCS(=O)(=O)NC)C2)nccc2nc[nH]c12 c1(C(N2CCC(C)(CNC(=O)CCOC(F)F)C2)=O)ccc2cc(F)ccc2n1 C(C)(CO)(C(=O)NCCCC(C)(C)NC(c1ccc(N(C)C)nc1)=O)NC(C)=O C1(CC(C)OC)CC2CCC(C1)N2C(=O)CC1(CSC)CC1.C1CC(=O)N1 Cc1cc(O)cc(O)c1CN(C)CC1CCCCO1.C12CN(C1)C2=O C1(C(=O)NCC(C2CC2)NC(CCC(=O)NCC)=O)(COC)CCC(F)(F)C1 C(=O)(C1=CCCCC1)N1CCC(C(C2CC2)NC(CC(=O)N(C)C)=O)CC1 CCC(C)(C)C(c1nnnn1C1COC1)Nc1ccc(C(F)(F)F)cc1.C1CO1 CCCS(=O)(=O)C(C)C(=O)NC1CCCN(C(C2CCC(F)(F)C2)=O)C1 C1(CC(=O)NCC(C)N(C)C(C2CC23CC(O)C3)=O)CCCOCC1 C(=O)(C1=CCC(C)CC1)NC(CCCNC(C1(CC#C)CCOC1)=O)(C)C N1(C(c2ccc(CC)nc2)=O)CCCC(NC(=O)CCC2CCCO2)C1CC N1(Cc2ccc(NC(C)=O)s2)CCCC(C(=O)Nc2ccncn2)C1 c1(C(N(C(C)C)CCN(C)C(C2(C)CCCOC2)=O)=O)ncnc2c1CCCC2 CC1CC(C(=O)N2CCN(C(c3cnn(CCO)c3)=O)CC2CC2CC2)=NO1 Cc1coc(C(=O)NC(c2ccccc2F)c2cc(C)n[nH]2)c1C.C1CC1 CC(CC(C)NC(c1c[nH]nc1I)=O)NC(=O)C(=O)N(C)C c1(C(=O)NC2CC(NC(CC3C=NN(C)C3=O)=O)C(O)C2)cccc(Cl)c1O C(=O)(C#CC(C)(C)CNC(=O)C=CCOC)N1C(CC)(CC)CC1 c1(C(=O)NC(C(=O)NC(CCSC)CO)C(C)(C)C)c[nH]c2cnccc12 N1(C(C2CCCC(C(N)=O)C2)=O)CCOC(C)(CNC(c2cncn2C2CC2)=O)C1 C1(C(N(CCC(C)C)C)=O)CN(C(=O)CCCCNC(N)=O)CCC1(C)C c1(OC)cc(C)ccc1C(C)Nc1nccc(N(C)Cc2nccs2)n1 CCC(C(=O)N(CCCNC(c1cc[nH]n1)=O)C)C(F)(F)F c1(C(C2CCCCC2)n2c(N(CC(=O)OC(C)=O)C)nnn2)cc2ncccc2o1 C1(C)(C(N(CCN(C)C)C)=O)CCN(C(=O)C=Cc2cn(C)nn2)CC1 C1(NC(NCc2n(CCC)cnc2)=NCCSC)CCCCC12CCC2 C12(NC(C(C(=O)OCC)OC)=O)CCCC(NC(=O)CCCOC)(C1)C2 C(=O)(C1=CC2C=CC(C1)C2)N(CCOCCC(N1CC(C#C)(F)C1)=O)C C1(C)(CC)CC(NC(=O)CCCn2cncn2)CN1C(=O)C=Cc1ccncn1 c1(C(=O)NCc2nc(CNC(C(OC)OC)=O)sc2)ccc(C)nc1 c1(C(N2CC(C#N)(C(N3CC4CCC(CC4)C3)=O)C2)=O)cccc2cc(F)ccc12 c1(C(N(CCCNC(CC(C)CN(C)C)=O)C2CC2)=O)cc(Cl)c(F)c(Cl)c1 N1(C(COCC#C)=O)CC(C)CC1C(=O)NCC1CC2CCC2C1 C1(NC(C2CCCOC2C(=O)O)=O)CNCC(F)(F)C1 N1(C(C)(C)CO)CCN(C(=O)C(C2(O)CCC2)NC(c2cccnc2)=O)CC1 c1(C(=O)NC2CC(CCC(=O)N(CC(F)(F)CC)C)C2)ccc2occc2c1 c1(CC(N2CCC(NC(C3C(=C)CC3)=O)C23CCC3)=O)c[nH]c2c(F)cccc12 c1(CNC(C(C2CCN(C(c3cc(C)sn3)=O)C2)F)=O)ccc(F)cc1C N1(C(C(C)NC(C)=O)=O)CCCC(O)(CCNC(C2(N(C)C)CCOCC2)=O)C1 N1(C(CSCCCC)=O)CC2(CCN(C(c3ncc(F)cn3)=O)CC2)CC1C CCCC(CC(=O)Nc1ccccc1C)NC(=O)CC1(COC)CC1 N1(Cc2n(CC)nc(C(F)F)c2)CCC(=O)N(Cc2cccc3[nH]ncc23)C1=O c1(SCC(=O)NC(Cn2cc(C(CC)O)nn2)C)cc(C)ccc1C O=C(C1CCSc2ccccc21)NCC1CN(C(C23CCC(CC2)C3)=O)CCO1 c1(N(C)C)cnccc1C(=O)NC1CC(F)(CNC(=O)CCc2nccn2C)C1 n1(CCC=C)nc(-c2cccc(N(C)C(C)=O)c2)nc1C1CC1F C1(C(=O)NC2CCN(C(CCC(C)N(C)C)=O)CC2)CCN(C)S1(=O)=O CC(C)C(O)CC(=O)N(C)CC1CCN(C(C2(C)CCCC2O)=O)CC1 c1(C(N2C(C(C)NC(C3(CCC=C)CC3)=O)CCC2)=O)nc2ccccc2s1 CN1C(=O)c2ccccc2C1CCSCC1CCc2nccn21 C1(Cn2cc(C(CC)(C)O)nn2)C(C2CC2)CCN1C(=O)CCn1cccc1 NS(=O)(=O)c1cc(C(=O)NC2C=CC(C(N3CCCC(F)C3)=O)C2)c(O)cc1Cl c1(C(=O)NCC2CC(C)N(C(=O)CCC#N)C2)cccc2nccn12 N1(C(COc2c(C)cccc2)=O)CCC(CNC(C2C(C)C2C)=O)C12CCC2 C1(NC(c2nc(CCC)oc2)=O)COCCN(C(C2(C(=O)C3CC3)CC2)=O)C1 c1(CCC)[nH]ccc1C(=O)N(CC(CC)NC(=O)CC1CCN(C(C)C)C1)C c1(C(N2CC(NC(c3cnn[nH]3)=O)CC3(C2)CC3)=O)ccc2c(c1)CCC=C2 N=c1nc2cc(C(=O)NC3(CNC(=O)CNc4ccccn4)CC3)ccn2[nH]1 C(N=c1cc(C)nc(-c2ccc(Br)cc2)[nH]1)c1c(CC)n[nH]c1 Cn1c(=O)sc2cc(S(=O)(=O)NCC(O)CN3CCOCC3)ccc12 N1(C(c2cc(OC)c(O)nc2)=O)CC(C2CCN(C(C3(C)CC=CC3)=O)CC2)C1 C1(C(C)CO)CC2CCC(C1)N2C(=O)CCCSC1CCC(C(C)=O)CC1 N1(C(CCOCCC)=O)CC(NC(C2CCC=CCC2)=O)C(c2ccnn2C)C1 C(c1nc(C)c(C)[nH]1)=CC(=O)NCC1(NC(c2c[nH]c(=NC)s2)=O)CC1 C1(NC(C2OCCC(NC(c3cccc(CC)n3)=O)C2)=O)CCn2nnnc2C1 c1(C(=O)NCC(CO)NC(CCCc2n(C)cnn2)=O)cc(Cl)c(Cl)[nH]1 C12(NC(CS(=O)(=O)NCC)=O)COCCC1CN(C(c1cc(C)nc(O)c1)=O)C2 CC(CC(=O)N1CC(NC(c2occc2C2CC2)=O)C1)C(F)F C(=O)(C1=CCCCC1)N1CC(CCC2(C)CC(F)(F)C2)(CNC(C=C(C)OC)=O)C1 C=CC(O)C(=O)NCC1CC(NC(=O)C=CCOC)C1 c1(NCC(N2CC(CNC(CC)=O)C3(C2)CC3)=O)ccc(SC)c([N+](=O)[O-])c1 C(=O)(C1=CC2C=CC1C2)N1CCC(C(C)CNC(=O)CC2(C)CC2(F)Cl)CC1 CCCCC(C(=O)NC1CNC(=O)C12CC2)NC(C1CCCCNC1=O)=O C(=O)(C1=NNC(=O)CC1)NCC1CC(NC(Cn2c(=N)nc[nH]2)=O)C(O)C1 c1(C(=O)NC(C)C(CCc2ccccc2)NC(=O)C2=NOCC2)cc2cccnn2n1 CCCCCCC(CC)(CC)C(=O)OCC1CCNC(=O)CC1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CN(C(CCN=C)=O)CC1S(C)(=O)=O C1(NC(C(CC)N(CC)CC)=O)CN(C(=O)Cc2nonc2C)CC1C Cc1cc(F)c(CNC(c2ncoc2-c2ccccc2)=O)c(Br)c1 c1(CC(N2CCC(CNC(c3c(C)csc3)=O)CC2)=O)nc([N+](=O)[O-])n[nH]1 c1(CC(=O)NCC2CC3(CCCCC3)C2)ccc2c(c1)OCCO2 N1(C(C#CC(C)C)=O)CCC2(CCCCC2NC(c2cc[nH]n2)=O)C1 N1(C(C(C2CCCCC2)C)=O)CCCC1(C)C(=O)N(C)CC1CC(F)(F)C1 c1(C(N2C(C)CC(CNC(CCCOCC)=O)C2)=O)nc(C)ccc1OC C(CN(C)C1CC1)(CC(C)C)NC(C=CCNC(CC=C(C)C)=O)=O N1(C(c2cc(C(C)C)cc(Cl)c2)=O)CC2CC1CCC2NC(c1cocn1)=O c1(N(C(=O)OC)CCOC)sc(C)c(C)c1NC(=O)C(=O)NC1CCCSC1 C12(C(=O)OCC)CCCC1CN(C(c1n[nH]c(C)c1Cl)=O)C2.C1(=O)NCCN1 n1(CC)cnc(C(=O)NC(C(=O)N(CCC(=O)NC(C)C)C)C2CC2)c1 CC1CN(C(=O)CCC2CC2(F)F)CCC1Nc1ncnc(O)c1Br N1(C(Cc2nc(C(C)(C)C)sc2)=O)CC(NC(=O)C(Cl)=CCl)C2(CCC2)C1 c1(C(=O)NC(C(=O)N(C(CC)C)CCC)C)nc(C)c(=O)[nH]c1OC c1(C(=O)NC2C(NC(C=Cc3occ(C)n3)=O)CCC2)cc2c(nn1)CCCC2 N1(C(CC(C)OC)=O)CCC(C)(CNC(C2(Cc3ccccc3Cl)CC2)=O)C1 C1(CNC(C=CCCC)=O)CC2(CC2)CN1C(C1C2CC3C(C2=O)C13)=O N1(C(C2C(C)SCCC2)=O)CC2(CC(CC(=O)NCC3CCC(=O)NC3)C2)C1 N1(C(C2(Cl)C(C(C)=O)C2)=O)CC(C=C)(CC(=O)NC2CC(n3ccnc3)C2)C1 Cc1ccccc1CC(C)NC(C1CC=CCC1)=O.N12CCN(CC1)C(=O)C2 N1(C(CCN(CC#C)C(c2c[nH]c(=N)o2)=O)=O)CC(CC2CC2)C1(C)C c1(C(=O)NCCC(C)NC(C=C(COC)C)=O)cc(F)cc([N+](=O)[O-])c1 C1(C(=O)NCC(Cn2cc(-c3cccc(N)c3)nn2)OC)CC2(CC(=O)C2)C1 c1(C(C(=O)NCCCF)N(CC(=O)NC)C)csc(C2CCC2)n1.OCC c1(C(N2CCC3(NC(=O)CCCn4ccnn4)C(C2)C3)=O)cc2ccccc2[nH]1 C(=O)(C(F)C(C)C)N(C(CNC(c1ccn(CCCC)n1)=O)C)CC C1(NC(c2c(CNC(CCCN(C)C)=O)cco2)=O)CC2(COCCO2)C1 C(=O)(C1=NOCC1)NC(C(C)NC(=O)CCc1ccccc1)(C)C c1(C(=O)NC(CCN(C(C(C(C)C)n2cc(C)nc2)=O)C)C)cc(C)nc(C)c1 C=CCCCC(C(=O)N1CCC(OCCO)C1)NC(c1cncc(F)c1)=O c1(NC(=O)NCC(=O)OCC2CCCC2)cccc(Br)c1Cl Cc1cc(COC(C)C(=O)NC2CCCC2NC(=O)C(C)C)no1 N1(C(c2cc(C)cc(F)c2)=O)CCCC(NC(c2ccn(C)c(=O)c2)=O)C(F)C1 N1(C(c2cc(C)cc(C)n2)=O)C(C)CC2CN(C(=O)C(F)(F)CC3CC3)CC12 C12(NC(=O)COc3cccc(F)c3)COCCC1CN(C(c1nsnc1O)=O)C2 C=C=CCCC(=O)N(C)CC1CCCN(C(=O)C(C)(C)c2cncs2)C1 N1(C(c2ccc(O)nn2)=O)CC2CC(C1)CN(C(=O)CCN1CCOC1=O)C2 C1(C)(CC)C=C(C(=O)NCC2(C)CCCN2C(=O)Cc2c(Cl)cnn2C)C1 Cc1nnc2n1CCC(C(N1CC(CNC(=O)CCc3cccnc3)C1)=O)C2 C1(NC(=O)CC2C=CCCC2)CCC(O)CN(C(c2csc(C3CC3)n2)=O)C1 C12(C(N3CCC(C)C(NC(=O)C=CC4CCCO4)C3)=O)CCC(CC1)C2(C)C c1(CC(=O)NCCN(C(C(C)=C2CC2)=O)CC(C)O)ccc(C)c([N+](=O)[O-])c1 C1(NC(CCOCC#C)=O)C(C)CN(C(=O)COc2cccnc2)CC1C C=C(C)C1OCCCC1C(=O)NCCC(C)N(C(=O)CC12CCC(CC1)CC2)C C1(NC(c2c(OC)cnc(C)c2)=O)CCCC12CN(C(c1cc(=O)cco1)=O)C2 N1(C(COCC)=O)CCC2(CCCN(C(=O)C(c3cnc(O)nc3O)(F)F)C2)C1 Cc1ccc(F)c2oc(C(=O)NCC3CC(C)(C)CCO3)cc12 C(=O)(C(C)(C)CN1CCOCC1)NCCC(C)NC(CC1(COC)CCCC1)=O S(=O)(=O)(c1cccc(N2CCSC3CCCC23)n1)NCCc1n(C)c(O)nn1 C(=O)(C(CCSCC)OCC)OCC.c1(C)cc(C)n(CO)n1 CN1CCCC12CCCN(C(=O)C(=O)NC1C3CCC1(C)C3(C)C)C2 c1(CC)nn(C)c(CC)c1C(=O)NC1CCCC1NC(=O)CC1CCN(C)C1 CP(C)(=O)c1ccc(C(N2CCN(C(=O)C=CCO)C(c3ncc[nH]3)C2)=O)o1 N1(C(CCN(C(CC)CC)C)=O)CCCC(C(=O)NC)(NC(=O)CNC=O)C1 Cc1nc(NCC2CC(C)(C)CCO2)cc(NC2CC2C2CCCC2)n1 C(C(=O)N1CCCc2nncn21)C1OCCN(C(C(C)Cc2ccco2)=O)C1 N1(C(CSCC)=O)CCN(C(=O)C(Cc2ccccc2)N(C)C)C2CCC12 N1(C(c2cc(C)c(C)s2)C(=O)NCSc2ccccc2)CCOCC1C1CCCO1 c1(C(N2CCCC(NS(CCC)(=O)=O)C2)=O)cc2c(nc1O)CCC(C)(C)C2 C(=O)(C1=COc2ccccc2O1)NC1CC(C)(NC(C(CCC)O)=O)C1 N1(C(=O)NC2(COC(C)C)CC3CCC2O3)CCn2c(nc(C(F)(F)F)c2Br)C1 N1(C(c2c(C)ccc(F)c2)=O)CCC(NC(C2(F)CCOC2)=O)CC(C)(C)C1 C(=O)(C1=NOC(C)C1)NC(C(=O)NC1(CCC)CCC1)CC1CCC1 N1(C(C(C)(C)C2CC2)=O)CCC2(CC(NC(=O)C(c3ccc(Cl)s3)=O)C2)C1 CC1(CNC(C2CNC(=O)C2)=O)CCCN1C(c1ccsc1-n1cnnn1)=O Cc1cccc(C(=O)NCCN2CCN(C(=O)CC3CCC(C(N)=O)O3)CC2)c1O N1(C(C(C=C=C)C)=O)CC(=O)NC2CN(C(c3c[nH]nc3C3CCC3)=O)CCC12 C1(CCNC(CCCNC(=O)OC)=O)(NC(c2csc(F)c2)=O)CCOCC1 N1(C(CCCN=[N+]=[N-])=O)CC(CO)C2(C1)CN(C(c1nc(=O)cc(N)[nH]1)=O)C2 C1(S(N)(=O)=O)(C(=O)NC(C(c2ccccc2)NC(C2CC(SC)C2)=O)C)CC1 C1(C)(C(=O)NCC(COC)NC(C23CCCN2CCC3)=O)CCCCCC1 c1(N(C)Cc2ccc(-c3noc(C(F)(F)Cl)n3)cc2)n[nH]c2ccc(C#N)cc12 CC1(C)COC(CC(=O)NC2CCN(C(=O)Cc3cccnc3)C2C2CC2)C1 c1(C(N2C(CNC(C3(n4cncn4)CC3)=O)CC(OC)C2)=O)ccc(C#N)cc1C C1(CNC(=O)C=CC2CCOC2)CCCCC1NC(=O)Cn1cc(C2CC2)cn1 c1(CC(=O)NC2(COC)CN(C(=O)C(C3CCC3)OCC)C2)cc(C)n(C)n1 c1(COCC)cncc(C(N2CC(O)(C(F)C(=O)Nc3[nH]c(C)nc3C)C2)=O)c1 N1(C(CN(CCC)C)=O)CCC(NC(=O)C(C)(C)C2CCCO2)C(CC)C1 C1(NC(CC(=O)OC)=O)CCc2nc(C(=O)NCC3CC4C=CC3O4)ncc2C1 C=CCC(CC(C)C)C(=O)NCC(C)(C)CC(=O)NC(c1ccnn1CC)C CCC(C)C(C(=O)N1CCC(O)C(NC(c2cnns2)=O)C1)NC(=O)OC N1(C(c2c(C)n(C)nn2)=O)CC(NC(=O)CCSCC(C)C)C2(CCC2)C1 c1(OCC)ncccc1C=CC(=O)NCC(Cl)=CCl CCC(F)(F)C(C)(C)C(=O)NC1CCC1CNC(c1[nH]cc2c1CCS2(=O)=O)=O Cn1ncc(C(=O)NCCC2CCCN2C(c2cn(-c3ncccn3)cn2)=O)n1 C1(NC(c2c(C)cco2)=O)C2CCC1CN(CC(F)(F)Cl)C2 C1(C(=O)NC2(CCCC(=O)N(C3(CCO)CCC3)C)CCC2)CCCN(C)C1 c1(C(N2CCCC(NC(C3(N(C)C)CC3)=O)CCC2)=O)nc2cc(F)ccc2s1 c1(C(=O)NC(CNC(C(C)n2ccnn2)=O)C(C)(C)C)ccc(F)c(F)c1O C1(CC(N2C3C(NC(c4c(C)nc(C)[nH]4)=O)CC(C3)C2)=O)CCC2(CCC2)CO1 O=S(=O)(c1ccc(NCC(O)CF)cc1Cl)NCCSc1ccc(F)cc1F c1(C(=O)NCCCN(C(C(COC)(C)O)=O)C)csc2nnsc12 N1(C(C(CC#C)(C)NC(C2C(C#N)C2(C)C)=O)=O)CCC2(CCSC2)C1 c1(-c2ccc(CNC(C(=O)NC34CC(CC)(OC3)C4)=O)cc2)c(C)cccc1C Cc1cc(C)c(C(N2CCC(O)(CCNC(c3coc(Cl)n3)=O)CC2)=O)cn1 CC1CN2CCCCC2CN1C(=O)CCc1cc(Br)ccc1F C1(NC(CC2(N(C)C(C3CC3F)=O)CC2)=O)CCc2c[nH]nc2C1 CCP(=O)(CC)c1ccccc1C(N1CCC2CCN(C(=O)C3=CCC3)C2C1)=O C1(NC(C2(C)CC2C(F)(F)F)=O)CNC(=O)C12CC2 N#CC1CN(C(C2C3CC4C(C3NC(C3CC(=C5CCC5)C3)=O)C24)=O)CCO1 C(=O)(CCS(N)(=O)=O)N1CC(CNC(C(c2ccc(C)cc2)C(C)C)=O)C(O)C1 c1(C(=O)NC2CCC23CN(C(c2nn[nH]c2Cl)=O)C3)ccc2cc[nH]c2c1 CCCC(NC(=O)N(CCC)CC1CC1)CC1CC1 CCC(CCOC)C(=O)NCCC1CN(C(c2c(C(F)(F)F)nn(C)c2C)=O)C1 c1(SCC(=O)NC(CNC(C(c2ccc(OC)cc2)O)=O)C)cc(C)ccc1C C=C=CCCC(=O)NC1CCC1NC(=O)C=CC(C)C C1(N(C)C)CCN(C(=O)CCC2CC(NC(=O)CCOC3CCCC3)C2)CC1 N1(C(C(C=C=C)C)=O)CC2CC1CC2NC(c1conc1-c1ccccc1)=O C(=O)(C1=CC2CCC=CCCC12)NCC1N(C)CCN(C(C2CNC(=O)N2)=O)C1 c1(C(=O)NCC2(CO)CN(C(C(CC)OC3CCCCC3)=O)C2)cncc(N)n1 c1(C(N2CCC(CNC(C34CCCCC3C4)=O)C2)=O)cnc2sccn12 C(=O)(CCCC(CC)CC)N1CC(C(C(N2CCC(CCCC)C2)=O)O)C1 C1(NS(C)(=O)=O)CC(CO)N(CC=O)C1.n1(CC(=O)OC)ncn(C)c1=O C1(OC)CCCC1C(N1CCC(C(F)C(=O)NC2(CO)CC2(C)C)C1)=O c1(C(=O)NC2(CNC(CC3C(C)CCO3)=O)CCC2)cc(F)cc2c1NCCC2 C(C(C(C)(F)F)c1ccccc1)OC(C1(CC#C)CCC1)=O c1(C(=O)NCCCCNC(C(C)NC(=O)C(C)(C)C)=O)cnn(C)c1S(N)(=O)=O c1(C(N2CCC(NC(C3C(C)C3C)=O)(CF)C2)=O)cncn(C)c1=O c1(CC)ccc(-c2cn(CC3CC(NC(=O)COC4CCCCO4)C3)nn2)cn1 Brc1ccc2c(c1)C(NC1CCNCCCC1)CCO2 N1(Cc2n(C)ccc2)CC(C(N2C(C(=O)O)CC3CC23)=O)C(F)(F)C1 C(=O)(C1=NOC(CNC(=O)C=C(C)c2ccco2)C1)N(C1CCCC1)CC N1(Cc2c(CC)onc2C)CC2CC1CN2C(c1coc(C)n1)=O C(=O)(C1CCCc2nccn21)NCC1(C)CCCN(C(c2cnnc(Cl)c2)=O)C1 C1(CC(N2CCCC2C2CCCN(C(C3(CF)CCC3)=O)C2)=O)C=CS(=O)(=O)C1 Cc1ccc(C(N2CCCN(C(c3csc(C)c3N)=O)CC2)=O)cc1Cl CC(C)(C)CC(F)C(=O)N1CCC(C)(CNC(=O)C=CCN2CCC2)C1 CC1CC(C(N2CC(C(N)=O)C2)=O)N1C(c1ccoc1)=O S(=O)(=O)(c1[nH]c(=NC2CCC2O)ccc1Br)N1CCC(N2CCC(C)CC2)CC1 C#Cc1cc(C(=O)NC2C3CN(C(=O)CC4(C#C)CCC4)CC23)cc(F)c1 C(=O)(C(CNC(C1CC=C(C)CC1)=O)C(C)(C)C)NCCS(CC)(=O)=O C1(CC(=O)N(CCCCCNC(c2cc(CCOC)on2)=O)C)CCC2CC2C1 CC1(C)CN(C(C2(Cl)CC2)=O)CC1CNC(C1CCCCN1C1CCCC1)=O CC(CC(=O)NCC(C)CNC(C1CCCS1)=O)N(C)C C1(N(C)C)CCC(C(=O)N=CCC(N2CC(F)(CO)C2)=O)C1 c1(CC(=O)NC(C2CCCCC2)CNC(c2cnc(SC)s2)=O)cnn(C)c1C C12(C(N3C4(C(N(C)CCc5nccs5)=O)CC4CC3)=O)CCC(CC1)CC2 n1(CC(=O)NCC2CN(C(C(C)C)=O)C(C)(C)C2)nc2n(c1=O)CCCCC2 c1(OCC(C)N)ccc(O)c(C(=O)NC2(C3CCC3)CC2)c1 N(C(=NCCF)N1CCC(c2ccco2)C1)CC(C)(C)C.C(C(F)(F)F)N CC(CN=C(NC(C1CC1)C1CC1)NCC1CNC(=O)O1)Oc1ccc(C)cc1 c1(OC)ccc(C(=O)NCC(COC)C(=O)NC2CC2)c(F)c1 N1(C(CNC(CC)=O)=O)CC(C)(OCC(=O)NC(c2cnn(C)c2)C)C1 C=C(C)C(CC(=O)NCC1CCC(C(=O)Nc2ccc(CO)cc2)CC1)OCC N1(C(CCCCOC)=O)CCCC(C)(CNC(c2c(OC)cccc2F)=O)C1 N1(C(C(=O)NC(c2ccccc2)C)C2CCOC2)CCOC(C(C)(C)C)C1 c1(C(N(C2CN(C(=O)CC3CCCO3)C2)C)=O)cc(S(N)(=O)=O)oc1Cl N1(C(CCOCC(C)C)=O)CCC(CO)C(NC(c2nn(C(F)F)cc2Cl)=O)C1 C1(NC(=O)NC)CCCC(C2CC(C(=O)NCC3CC3)C2)C1.C1(=O)CN1 C1(C(C)C)COCCN1C(C1CCN(C)C1)=O.c12cn(nn1)CCCOC2=O N1(C(C(CC(C)C)ONC(c2c(OC)cncc2)=O)=O)C2CCC1CC(=O)NC2 CC(C)CCC(O)C(=O)N1CCCC(C(=O)NC2CC2)C1 c1(C(=O)NCCC2CCCN(C(C(C(C)C)(C)O)=O)C2)ccc(P(C)(C)=O)nc1 C(=O)(C(C)C(O)C(C)C)N1CC(CCNC(c2sc(C)c(Br)c2)=O)C1 c1(C(=O)NC2CN(C(C(C)OC)=O)C2)cnc(-c2ccccc2)o1 N1(C(COCCCC)=O)CC2(CCN2C(c2ccnn2CCF)=O)C1 c1(C(N2CC(C(=O)Nc3ncc(I)cc3I)CC(F)C2)=O)cccc2nscc12 O=C(CCCCC1CC1)N1CCC(N2CCN(C(C3CC3(F)F)=O)CC2)C1 N1(C(C(CC)n2cncn2)=O)CCC(C)N(C(=O)N(c2ccc(F)cc2)CC)CC1 C1(C(=O)NCC(=O)NC(C)(C)C)(CF)CCN(C(c2cnn(CCO)c2)=O)C1 N1(C(c2nccc(C)n2)=O)CCN(C)CC1CNC(=O)CCc1cc(C)on1 CC1CN(C(c2cc(O)ccc2Br)=O)CCN1C(c1n[nH]cc1I)=O c1(CCC)csc(C(C(=O)NC2CCOC2)N(C)Cc2ncnn2C)c1 Cc1c(C(N2CC3(CC3)CC2C(N2CCN(C3CC3)CC2)=O)=O)cc(F)cc1Cl N1(C(c2c(C)noc2)=O)CC2CCC1CN2C(=O)C(C)CO C1(OC)CC2(C1)CN(C(=O)C(CNC(c1ccc(O)nn1)=O)CC1CC1)C2 c1(CC2C(=O)N2)ccc(OCC=C)cc1.C(C)(C)(C)OC(N(CC=C)C)=O N1(C(c2cnc(SC)s2)=O)CCOCC1CN(C(=O)Cc1ccn(C)n1)C Cc1cccc(N)c1C(=O)NCC1CCN(C(C2(n3cccn3)CCC2)=O)C1 C1(NC(c2ccn(C)c(=O)c2O)=O)COC2(CCCN(C(=O)C(C)(C)C#N)C2)C1 C1(N(C(C(c2ccccc2)SC)=O)C)CC2CCC(C1)N2C(=O)C1=CCCO1 CCC(C#N)C(=O)N1CC(N(C)C(c2nn(C)cc2C)=O)C1 Cc1cc(F)c2cc(C(=O)NC3(CO)CCN(C(=O)CN4CCC4C)C3)[nH]c2c1 N1(C(c2c(COCC)con2)=O)CCCN(CCc2noc(C3CC3)n2)CC1 c1(C(N(CCNC(c2c(C)csc2)=O)C2CC2)=O)cc(N)ccc1Br N1(C(c2c(C)cc(Br)cc2I)=O)CCc2c(C#N)cccc2C1 Cc1nnccc1C(N1CCCCC1CCNC(=O)CC1CN(C)C1)=O n1(CCC2(C)CC2)nnnc1C(C1(CC(F)(F)F)CCC1)N.C1(C)CC1 c1(N(C(c2c(CC)scn2)=O)C)cc(C2CC2)ncn1.C12CCCN1C2 c1(C(=O)NC2CC(CNC(C3CCC(C(N)=O)O3)=O)C2)ccc2cnnn2c1 C1(C(=O)NC)CCCCC1CNC(CN1CCC(CNC(=O)C2CC2)CC1)=O N1(CCOC)CCN(C(=O)C(=O)N(c2nc(C)cs2)C(C)C)CC1 c1(NC(C2(C(C)C)CCN(C(COC(CC)(C)C)=O)C2)=O)cn2ccccc2n1 C1(C(N2CCC(C)(CNC(c3c(CC)[nH]c(=N)s3)=O)C2)=O)CN2CCN1C(C)C2 c1(CC(=O)NCC(C)(CO)NC(CN(CCC)C)=O)cccc(Cl)c1NCC C(=O)(CC(C)(O)COC)N1CCCC(C(N(CCOCC)CC)=O)C1 CCCC(C#N)C(=O)N1CCCC(CCNCCCn2cccnc2=O)CC1 C1(CNC(C(CC)N(C)C)=O)CC2(CCC2)CN1C(c1cc[nH]c2nccc1-2)=O C1(NC(c2c(C)n[nH]c2)=O)CC12CCN(C(=O)CCOC(C)C)C2 C1(C(N2CCC(C(C)C(=O)N(C3CC3)CC3CC3)CC2)=O)CCC=CCCC1 Cc1ccc(OC(C)C(=O)NCC2CC(F)(F)CN2C(=O)CC(C)(C)O)c(C)c1 C1(c2ccc(CC)o2)CN(CCCc2ccc(OCC(=O)O)cc2)CCO1 C=C(C)CCCC(=O)N1CCC=CC1C(=O)NCC=CCl N1(C(C(C)n2cccc2)=O)CCOC(C(C)NC(=O)CC2CCC3CC23)C1 CC1C(NC(c2cccn2C2CC2)=O)CCCN1C(c1cscc1Cl)=O C(c1ccc(Cl)c(Cl)c1)=CC(=O)NCC=C1CCN(C(C(C)(C)C)=O)CC1 Cc1cnn(C)c1C(=O)NC1C=CC(C(=O)N(CC(C)(CO)CO)C)C1 Cc1c(C(=O)N(CC(C)C)CCc2nn[nH]n2)oc2c(F)cccc12 C1(F)(C(=O)NC(c2c(Br)ccc(C)c2)C)CC2CCC(C1)N2C(=O)OC(C)(C)C C(=O)(C(O)CCS(C)=O)NC12CN(C(Cc3cccc(C)c3)=O)CC(C1)C2 C1(C(=O)NC2C(C#C)N(C(=O)OC(C)(C)C)CC2)CCn2ncnc2C1 c1(CC(=O)NCC(C2CCN(C(C3C(=C)CC3)=O)CC2)(C)C)cc(O)cc(Br)c1 C(=O)(C1COc2ccc(Br)cc21)NC1(C)CCN(C(c2ccn(C)n2)=O)C1 C(C1CCCN1C)=CC(N1CC(C(C)NC(C(c2cccc(F)c2)C)=O)C1)=O c1(C(=O)NCC(C2CC2)NC(c2cnc(OC)s2)=O)cccc(Cl)c1C C=CC(C)CC(=O)NC(CCSCC)C(=O)NC1CC(C)(C)C1 c1(N2C3CN(C(c4cc(C)cc(Cl)n4)=O)C(CC3)C2)nccc(C)c1[N+](=O)[O-] C1(NC(c2cnn(CCNC(=O)Cn3ccnn3)c2)=O)CCOCC1F C(C(C(=O)N1CCCC(C)(CNC(c2sncc2C)=O)C1)C(C)(C)C)OCC=C c1(NC(C(C2CCCOC2)N)=O)cccc2c1CNS(=O)(=O)CC2 C#Cc1ccc(C(N2CCC3CC23C(=O)NCC2(C)CCCCO2)=O)nc1 n1(CC)cc([N+](=O)[O-])c(C(N2CC(NC(=O)C(C)=CC3CC3)CC3(CC3)C2)=O)n1 c1(C(N2CC(C)(C)C(NC(C3CCC(=O)O3)=O)C2)=O)csc(S(N)(=O)=O)c1 C(=O)(CCCC(F)(F)F)NC(C1(CNC(C2CCC=CCCC2)=O)CC1)C Cc1ccsc1C=CC(=O)NCC(CO)NC(=O)CC1CCC1(C)C C1CC(C)N(CC)CC1C.c1(CCC)ccc(Cl)cc1C C1(C2CCCN(C(c3coc(O)n3)=O)C2)(NC(CC(C=C)CC)=O)CC1 c1(CCC)ccccc1C(=O)N(C1CN(C(=O)COc2ccccc2CC)C1)C c1(OC)cc(C(N2CCC(NC(=O)C(O)CC3CC3)C(CO)C2)=O)ccc1Br N1(C(CNC(c2c(C)occ2)=O)=O)CCN(C(=O)CC2(C)CCCC2)C2(CC2)C1 CCCCCCC(C)C(=O)N1CCC(CC(=O)N(S(=O)(=O)CC)CC(C)C)C1 C(=O)(CCCC(C)(C)CC)NCC(CNC(c1n(CC#C)cnn1)=O)F Cc1cn(C)nc1C(=O)NCCC1CN(C(C2(C(C)C)CCC2)=O)CC1C CC1(C)CC(C(=O)NCCCc2cccs2)CN1C(C1(C)CCCS1)=O C1(CC)C(C(=O)NC(C)Cc2nc[nH]n2)CCCN1C(c1coc(C)n1)=O CCCCCC(C)CC(=O)N1C2CCC1CN(C(=O)Cn1nnc(=N)[nH]1)C2 c1(C(=O)NC(CC(C)NC(c2cncc(C)c2)=O)C)cc(N)nc(Cl)c1 CCC(CC(F)(F)F)C(=O)NCC(C)(CC(C)C)NC(C1CC1C(F)F)=O C=C1c2ccccc2C(=O)N1C(C)C(=O)OCC1OCCC12CCC2 Cc1c[nH]nc1CNC1CC(OC(C)C)C1n1cccn1 c1(C(C)Nc2c(C)ccc(OC)c2)oc2ccccc2c1C C1(NC(CCc2n(C)ccn2)=O)CCOC12CCN(C(=O)Cn1nnc(=O)[nH]1)CC2 C12(CC(=O)NCc3nc(CC)on3)CCC1CN(C(C1(C)C(C)(C)C1(C)C)=O)C2 c1(-c2cn(CCN(C(=O)CC3CCC(C(F)(F)F)O3)C)nn2)cccc(C#N)c1 C(=O)(C(COC(C)(C)C)NC(C)=O)NC(COC)CNC(C1(C)CC1C)=O c1(C(N2CC(CCCCNC(C3CCNC3=O)=O)C2)=O)c[nH]c(=O)c2ccnn12 C1(CCOC)CN(C(=O)CC2(OC)CCC2)CCN1C(=O)CCC1CCCO1 c1(C(N2CC3C(NC(CCC4CCC(=O)N4)=O)(C3)C2)=O)cc2nc(Cl)ccc2s1 N1(C(COC(C)=O)=O)CCC(OCc2cn(Cc3cnn[nH]3)nn2)C1C(C)(C)C C1(NC(C(C(C)OC)O)=O)CC2(C1)CN(C(c1oc(C(C)C)nc1C)=O)C2 Cc1cc(C(=O)NC2CCN(C(C3CCCCO3)=O)C2)co1 FC1(F)CCCCC(Sc2c(-c3ccccc3)cnn2CC(F)(F)F)C1 c1(C(=O)NC2CC(N(C(C3C(=C)C3)=O)C)C2)cc(S(N)(=O)=O)sc1Cl Cc1cc2ccc(C(=O)NC3CCCC(n4cc(CN(C)C)nn4)C3)cc2o1 C1(CC(=O)NCC(=O)NCCNC(c2cncc(C(N)=O)c2)=O)CCCC2CC12 C1(CNC(C2C(C)C2)=O)CCCCN(C(=O)C(C)(C)COC2CCCC2)C1 n1(CC)nnc(C(=O)NCC2CCN(C3CC3)C2)c1C.C12(CC1(C)C)C(=O)N2 C(=O)(CCCC(C)NC(c1ccc(NC=O)cc1)=O)NC(C)C(C)(C)CN(C)C c1(C(=O)NCCN(C(C(=O)NCCC)=O)CC)c[nH]c2c(C)c(C)ccc2c1=O N1(C(c2c(=N)[nH]cnc2)=O)CCC2(NC(c3ccc4nsnc4c3)=O)CCCC12 C1(NC(c2n(Cc3sccc3)nnn2)C2CCCC2)CC2CCCC2C1 CCC(C#N)C(=O)N(C1CCCCCC1)Cc1ccco1 Cc1ccc(C(C)(CNC(=O)NC2CC(O)C2)CO)cc1 C1(NC(C(C)C(C)O)=O)COC2(C1)CN(C(c1ccc(O)c(F)c1F)=O)C2 c1(CC(=O)NCC2C(NC(CCC(=C)C)=O)CC2)ccc2nc(O)[nH]c2c1 c1(C(N(c2ccc(Cl)cc2Cl)CC(=O)NC)=O)cc(F)c(C)c(F)c1 N1(C(c2nc(C)nc(O)c2)=O)CCC2(CC1)OCCC2NC(C1CCC1(C)C)=O C1(c2nnnn2CCC(C)(C)C(=O)OC)(NC2CC2)CCCC(C2CC2)CC1 C1(CNC(C2=C(C)N(C)CC2)=O)CCNC2CCCC12 CC1CCC(CC(=O)NCc2cc(C(=O)NC(c3nccs3)C3CC3)cs2)O1 C1(NC(Cn2nc(C)c(Cl)c2)=O)CC2CCC1N2C(c1snnc1C)=O N1(C(c2c(CCNC(=O)C=CC(=O)NC3CC3)ocn2)=O)CCCCC1CO c1(CCC(=O)NC)ccc(F)cc1C(=O)OC.C12=C(C)C(=O)N(CC1)CC2 N1(C(C2(C#C)CCN(C(C3CCC(F)CC3)=O)C2)=O)CC2(CNC(=O)OC2)C1 C1(NC(c2scc(C)n2)=O)CC2CC1N(C(c1cccc(-n3cccn3)c1)=O)C2 C1(CC)C(C(=O)NCC2(CCO)CC2)CCN1C(c1c[nH]c(C#N)c1)=O C(C(C(=O)NCC(CC1CC1)OC)C(C)(C)C)NC(c1nc(COC)oc1)=O C1(NC(CN(C(=O)C(C)n2cncn2)CCOC)=O)CC(CN(C)C)C1 c1(C(=O)NC2CC2NC(=O)CN2CCOCC2=O)cnc(C2CC2)nc1 CC(CC(=O)NC1CCC12CN(C(C1=CC=CC=C(C(F)F)O1)=O)C2)C(F)(F)F CC1CCN(C(c2cnc(N)cn2)=O)CC1CC(=O)NCCOc1cncc(Cl)c1 N1(Cc2cc(OC)ncc2)CC(NC(C2(C)CCOCC2)=O)CCC1C N1(C(C2C(CCOC)C2)=O)CCC(F)(CNC(=O)C(F)CC2CCCCC2)CC1 Cc1n[nH]c2cnc(C(=O)NCC3COCCN(C(C4(Cl)CC4)=O)C3)cc12 C1(NC(C(=O)NCCc2nc(C(F)(F)F)cs2)=O)COc2cc(F)ccc2O1 c1(C(=O)NC2CCN(C(CCCCOC)=O)CC2F)cc(C)c(C)nc1C C1(CN(C(=O)CC2CC2C)CC)CCN(C(c2cc(C3(C)CC3)on2)=O)CC1 C1(C(=O)Nc2c(C)cccc2)CN(C(=O)C=CC2CC2)CC12CC2 c1(C(=O)NC2(CNC(C(C)n3cnnn3)=O)CCOC2)cc(Cl)ccc1N C1(CCNC(CCC)=O)CN(C(c2cnc(C)cc2C)=O)CCS1(=O)=O Cc1nc(NCC2CC(C)N(C(=O)CC3CCCC(=O)N3)C2)c2ccsc2n1 c1(C(N2CCCC(N(C(=O)Cc3cncs3)CC)C2)=O)nccc(Cl)c1C C(=O)(CC(CC)C(C)(C)C)N1CCC(NC(C(=Cc2ccc(F)cc2)C)=O)CC1C c1(N2CCC(C)(NC(C(CCOC)C)=O)C2)nc2c(cc1C#N)CCC2CO C12(CC)CCCN(C1)C(C(=O)NC)c1nc(n[nH]1)CC2.N1(CCCCSC)CC2CCC1C2 c1(C(N2CCC(F)(CNC(Cc3cc(C)sn3)=O)C2)=O)c(F)cc(F)c(F)c1F c1(C(=O)NCC2(CNC(Cn3c(C)ccn3)=O)CC2)ccc(CCF)cc1 Brc1ccc2nnc(=NCCCc3cccs3)[nH]c2c1 C(C)(CCCNC(c1cc(-c2ccc(Cl)s2)[nH]n1)=O)NC(CCC)=O c1(C(=O)OC(CC(N2C(C)CC2C(=O)N(C)C)=O)=O)ccccc1Cl c1(C(=O)NCCC2CCN(C(C(C)(C)OC)=O)C2)c(Cl)cccc1Cl c1(C(=O)NCC(C2CCOC2)NC(c2cnc(CC)s2)=O)ccc(F)cc1C C1(NC(COCC#C)=O)CC2CCC(C1)N2C(=O)C(C)Cc1cccnc1 C1(NC(C=CC(C)(C)NC(=O)C2=CCCC2)=O)CCOCC1O c1(C(N2CCN(C(C(C(C)C)C)=O)C(c3cn[nH]c3)C2)=O)cc(N)c(Cl)c(O)c1 Cc1cc(C(N2CC(NC(c3nc(Cl)sc3C)=O)C(O)C2)=O)n2ncnc2n1 C1(NC(c2noc3c2COCC3)=O)CN(C(C2CCSC2)=O)C2(CCCCC2)C1 C(=O)(C(C(C)=Cc1ccccc1)N1CCCCC1c1ccc(F)cc1)NCCC c1(C(=O)NC(C2CCCC2)CNC(C(CSC)OC)=O)cc(Cl)ccc1C Cc1cc(Cl)cc(Cl)c1OCC(N1CC2CC(NC(=O)C=C(Cl)Cl)CC2C1)=O c1(C(=O)NC(C(=O)NC(CC#CC)C)COC)cnn(C)c1C(=O)OC C1(N(C(C(C2CCCOC2)OC)=O)CC2CC2)CCN(C(=O)C(C)(C)CF)CC1 c1(NCCC(=O)N(C)C)ccc(S(=O)(=O)NCC2CCN(CC(F)F)C2)c(Cl)c1 C1(C(N2CC=CC2Cn2cc(C(C)C)nn2)=O)(COC)C=CCC1 N1(C(c2cccc(-c3c[nH]n(C)c3=N)c2)=O)CC(C(=O)O)C2(CCOCC2)C1 C#CCC(C)(C)C(=O)N1CCC(C)C(CNC(C2(CC(C)C)COC2)=O)C1 CC1C(NC(c2sc(N3CCCC3)nc2Cl)=O)CCCN1C(=O)CN1CCCC1 CC1=C(C(=O)N2CCC(F)C(NC(=O)C(C)OC3CCCCC3)C2)CCCO1 c1(C(N(CCNC(C(C)(C2CCC2)OC)=O)C)=O)nccc2occc12 N1(C(C2(SC)CCSCC2)=O)CCC(NC(=O)C=Cc2ncc(C)[nH]2)C(CO)C1 C1(NC(c2nccc3ccccc23)=O)CCC2(CC1)CN(C(=O)C=CCO)CCO2 c1(C(=O)NCC2N(C(C3C(C)C3)=O)CC(F)(F)C2)cn(C)cc(Br)c1=O C1(NC(c2n(C=C)nnc2)=O)CN(C(c2scnc2Cl)=O)CC1C1CC1 N12C3CC4C5CC(C4C3O)C5c3c(n(CCCC)ccsc1n3)C=C2 N1(C(CC(C)OC)=O)CCN(C(=O)CCCCNC(c2ccccc2)=O)CC1CF CS(=O)(=O)C1CCCN(C(c2ccccc2-c2ccnc(N3CCCC3)c2)=O)C1 C1(NC(C(CC)(C)OC)=O)CCC2(CC1)CC(NC(=O)C=Cc1scnc1C)C2 c1(C(=O)NCC(C(C)C)(C)NC(=O)Cc2nncn2C(C)C)cccc2ncoc12 N1(C(C2(OC)CCOCC2)=O)CCC2(NC(=O)CCC(C)CN(C)C)CCCC12 CC1(C(=O)NCCC(Cc2ccccc2)NC(=O)C=C2CCC2)CCC(=O)NC1 c1(C(=O)NCC(C)N(C(c2ccc(CO)cn2)=O)CC)cc(OC)cc(C)c1 N1(Cc2cc(C)n(C)n2)CC2CN(C(=O)C(=O)Nc3ccco3)CC12 N1(C(CC)C)CCCC(C2CCCN(c3ccnc(C(C)(C)NC(=O)OC)n3)C2)C1 c1(C(=O)NC2(CCNC(C3(CC)CC3(F)F)=O)CCCC2)ccc2sccc2c1 n1(C(C(=O)NCC2(NC(CC3(OC)CC3)=O)CC2)C)cnc(C#N)n1 C1(C2CN(C(=O)CCc3cn(C)nn3)C2)(NC(CC2N(C)CCC2)=O)CC1 c1(CCC(=O)NCC2(F)CC(NC(c3cc(C)n(C)n3)=O)C2)ccc(Cl)c(F)c1 C(=O)(NNc1oc(C(C)C)nc1C#N)N1C(CC)CCC(C)C1 c1(C(=O)NCC(CC2CC2)C(=O)NC2(C(=O)OCC)CC2)ncc(F)cc1F c1(CCC(=O)N(C2CC(C(=O)OC(C)(C)C)C2)C)ccc(CO)cc1 N1(C(C(P(C)(C)=O)O)=O)CCC2(CCC2)C(CNC(=O)CC2(O)CCCC2)C1 C123CCCC1N(CCC2)C(=O)N3.c1(CN(C2CCS(=O)(=O)C2)C)ccccc1F N1(C(C2C(C(C)C)CCO2)=O)CCC(c2ncc(C(F)(F)F)[nH]2)(C(=O)O)C1 C#CCC(CC(=O)N1CC(C)(C)CC1CO)NC(CC(C)C#C)=O C(CCCCCNC(C1CC12CC(O)C2)=O)NC(c1cc(-c2cccs2)[nH]n1)=O CC1CSCCN1N1CC(C(c2ccccc2)C)C1 CCCCS(=O)(=O)NC(C)C(=O)NC(C)CNC(c1cn(C(F)(F)CO)nn1)=O c1(CC)ccc(N)c(C2CC2C(=O)NCC2(C(=O)NCCCN(C)C)CCC2)c1 CC(N=[N+]=[N-])C(=O)NC1CCCC(CC(=O)NC2CCC(CN(C)C)CC2)C1 C1(CC(N)=O)(NC(=O)C(C)SC(C)C)CCN(C(c2cnc(C(C)=O)s2)=O)CC1 O=CC1N(CCO)CCN(C(=O)COCCN(C)CCO)C1 CN1C(=O)CCC1CC(=O)NCCNC(C1CN(C(c2ccoc2C2CC2)=O)C1)=O C(=O)(C1=CCS(=O)(=O)C1)N1CCCC(NC(C=Cc2ncn(C)c2)=O)CC1 c1(C(N2C(C)CC(NC(C3(c4ccc(F)cn4)CC3)=O)C2)=O)ccc(N)c(F)c1 N1(C(CN2CCN(CC)CC2)=O)CC(C)N(C(=O)CNC(=O)NC2CC2)CC1C C(=O)(CC(C)CC(C)C)NCCC1(CNC(c2cccc(CC)n2)=O)CC1 CC1(C)C(CNC(=O)CCSC(F)(F)F)CCN1C(=O)CSCC(N)=O CC1(NC(c2cccn(C#N)c2=O)=O)CCCN(C(=O)CCn2ccnn2)C1 C(CC(C)C)(C(=O)NC(CNC(=O)C=CC(C)(C)C)CC(C)C)NC(C)=O N1(C(C2ON=C(CC)C2)=O)CCCN(C(=O)CC2(OCC)CCOCC2)C(C)C1 N1(C(C=CCNC(N)=O)=O)CC(N=[N+]=[N-])C1.C1CC(=O)N1 c1(SCC(=O)NCC(CNC(C(C)(C)SC)=O)F)cccc(C)c1 Cc1ccc(Cl)c(C(=O)NC23CC(CNC(=O)C4=COCCC4)(C2)C3)c1 C(=O)(C1CCCc2ccccc21)N(CCC(C)NC(c1cc(C(C)C)on1)=O)C Cc1ccc(NC(=O)C(C2CC2)N(C)C(c2cccc(Cl)c2)=O)c(C)c1O CC1(C)C(CC(N2CC(N3CCN(C(C4CCCS4)=O)CC3)C2)=O)C1(C)C N12CCC(C3(CCC3)C1)C2=O.c1(OC)nc(N2CCN(C(=O)CO)CC2)ncc1F c1(CC)ccccc1CNC(C1CC(C)CN1C(=O)C(C)(C)C#N)=O C1(CC=C)(NC(c2ccc(C)c(C)n2)=O)CCCN(C(=O)C(N)=O)C1 N1(C(C(=C(C)C2CC2)F)=O)CCOC2CCN(C(C3CCOC(=O)CC3)=O)CC12 c1(CN(C(c2ccccc2F)C(=O)NC(C)C)C(C)C)ccccc1Cl c1(C(=O)NCC(C2CCC2)NC(C(CCCC)C)=O)cncc2c1CCC2 Cn1ncc(C(=O)NCCNC(C2CSCCN2C(=O)CCCC#N)=O)c1C(F)F c1(NCC(CCC)C)cc(C)[nH]c(=NCCN(C)C(C)C)n1 C1(C(N(C2CCN(C(=O)CC3CCC(C)CC3)C2)CC)=O)CC(=O)NC(=O)N1 N1(C(COC(CC)C)=O)CCC(C(=O)NCC#CCOC)C12CC2 c1(COC)ccc(C(=O)NCC(=O)N(C)Cc2nnc(C)o2)o1 N1(C(CS(=O)(=O)N(C)C)=O)CC(NC(=O)CCNS(C)(=O)=O)CC1(C1CC1)CO c12cccc(c1)NC2.c1(N(c2ccccc2)CC)ccc(C(=O)N(C)OC)nc1 CCC(F)(F)C(=O)NCCCN(C(=O)CC(n1nc(C)cc1C)C)C N1(C(c2cccc(CC)c2)=O)CC(F)(F)CC1C(=O)Nc1cnccc1Br CCCC(CCCNC(C1CCC(=O)N1CC)=O)NC(=O)CCNC(=O)COC C=CC(C)(C)CCNC(=O)C(C(C)C)n1cc(-c2ccncc2C)nn1 Cn1ncc2c1CCNC2C(=O)NCc1nnc(-c2ccco2)o1 CC1(C(N2CC(NC(=O)Cn3cncn3)C(O)C2)=O)CCCCCC1 C(CO)(C(=O)NCc1cc(C(=O)NC2(CCF)CCC2)cs1)NC(C)=O C(=O)(C(F)CC(C)(C)C)NCC(C)N(C(=O)C(C)=CC(C)(C)C)CC c1(OC)ccc(C#CC=O)cc1.c1(C2(C3CCCC3)CC2)cccnc1 C1(C(=O)NCC2CCC(=O)N2)CN(C(=O)CCc2cn[nH]c2)CC12CCC2 c1(Cc2cc(C(N3CC(CC#N)C3)=O)on2)ccccc1Br C(=O)(C1=COc2ccccc2O1)N1CCC(CNC(Cc2c(Cl)cn(C)n2)=O)C1 N1(C(C(COCC)C)=O)CCCCCC1CNC(=O)CCC1(C)CCC1 c1(C(=O)NCC(CN(C(C(C)OCCOCC)=O)C)C)c(N)cccc1[N+](=O)[O-] C1(CC)CC2CN1C(=O)N2.c1(CNC(=O)OC(C)(C)C)ccc(-n2cccn2)o1 n1(C(C)(C)C)nnc(C(=O)NC2(Cn3cccn3)CN(C(c3coc(Br)n3)=O)C2)n1 C(=O)(C1CCCc2scnc21)N1CC(NC(c2cc(N)cc(C)c2F)=O)C(C)C1 C(=O)(CS(=O)(=O)c1ccccc1F)N1C(CNC(C2CCCC(F)C2)=O)CCC1 Cc1oc(C#N)cc1C(N1CCC(CNC(C2CCCN2C2CC2)=O)C12CC2)=O c1(-c2cc(OC3CN(C(C(C=C)O)=O)C3)oc2)ccc(Cl)cc1.C12CSCN1C2=O C1(NC(C2CC=C(C)CC2)=O)CN(C(c2cc(Cl)c(Cl)s2)=O)CC(F)(F)C1 C(=O)(CCCN(C(=O)CNC(c1csc(CC)c1)=O)C)OCC C(=O)(C(C(C)(C)C)NC(C1CC=CCC1C)=O)N1CC(CC(=O)OC)C1 Cc1nc2c(CC(=O)OC3CCCCCCC3)cccc2o1 CC1CN=C2NC(C(=O)NCC3(O)CN(C(C4CC5CCC4O5)=O)C3)=NN2C1 n1(CCC(=O)NC2C(NC(C(C)OCC#C)=O)CC2)ccc(O)nc1=O C1(C(N(C)CCC2OCCO2)=O)(NC(C2CC(F)C2)=O)CC(F)C1 C1(CNC(CC(CC)n2cccn2)=O)CC2CCC(C1)N2C(C1CC(SC)C1)=O c1[nH]nc2ncnc(O)c12.C12(C(=O)NCC(C)CNC(=O)CC#N)CCN(CC1)CC2 C1(NC(CSCC#C)=O)CC(C2CCN(C(c3cc(C)c(F)cc3N)=O)C2)C1 N1(C(C(c2ccc(N)cn2)C)=O)CC2(C)CN(C(C3CC(O)C3)=O)CC2(C)C1 C1(NC(c2ccnc(-n3cccn3)c2)=O)CN(CC2(C3CCCOC3)CC2)CC1O N1(C(c2scc(OC)c2)=O)CC2(CCC(CNC(C3CCC(=O)NC3)=O)O2)C1 C1(=C(CNC(CN(C)C(N)=O)=O)F)CN(C(C2(c3ccno3)CC2)=O)C1 c1(C(N2CCC(C(C)NC(c3cn(C)cn3)=O)C2)=O)ccc(Cl)c(C#N)n1 C(=O)(C1Cc2ccc(Cl)cc21)N(C(c1cn(-c2nccc(C)n2)nn1)C)C CC1CC2(CCO1)CC2C(=O)NCC1C2CN(C(=O)CCCc3csc(=N)[nH]3)CC12 c1(CC(=O)NCC(CNC(CC=CCC)=O)F)ccc2nonc2c1 C(C(=O)NCC(C1CC1)NC(c1ccnn1CC(F)(F)F)=O)(C(F)(F)F)OC(C)=O c1(C(=O)NC2CN(c3nc(C)cc(OC)n3)CC(F)C2)c(F)cc(C#N)cc1F c1(C(N2C(C)CC(NC(c3c(OCC)ccs3)=O)C2)=O)cc(C)cc(Cl)n1 C1(C(N2C(C(=O)NCC(CCC)OCC)C3CC3C2)=O)CC2(CCC2O)C1 Cn1ccc(-n2cnc(C(=O)NC3CCC3NC(=O)CNc3cccnc3)c2)n1 Cc1cc(C)n2ccc(C(=O)NCC(C(C)(C)C)NC(=O)CCP(C)(C)=O)c2n1 C1(NC2C=CCCC2)COC2CC1C2 c1(-c2cn(C(C)C(=O)NCC3(c4ccccn4)CC3)nn2)ccc(F)cc1 C1(CC)CCN(C(=O)C(F)OC(F)(F)F)C1CNC(=O)Cn1cc(C(F)(F)F)cn1 N1(C(CC(CC)OC)=O)CC(C2CN(C(=O)C(CC)CCOC)C2)C1 CC1CN(c2cc(N3CCC(CC4CC4)C3)nc(C(F)F)n2)CCN1C1CC1 C1(CN(CCOC)Cc2nc(-c3ccccn3)no2)Cc2ccccc2O1 N1(C(c2cnc(S)nc2)=O)CCCCC2(CCN(C(C3CCCOC3)=O)C2)C1 N#Cc1c[nH]cnc1=NC1CCCN(C(C2(c3cccnc3)CCC2)=O)C1 Cc1nc2ncnn2cc1C(=O)NC1CC(O)CN(C(=O)CC2CC=CCC2)C1 C(=O)(CCCC(=O)NC1CCCN(C(c2n[nH]cc2C(F)(F)F)=O)C1C)NCC c1(NC(C)=O)cc(C(=O)NC2CC(NC(C)=O)C2)ccc1F.C12CCCN1C2=O C(=O)(N=c1cc2n([nH]1)CCCC2)C1C(CC)N(C(c2cnn(CC)c2)=O)CCC1 c1(CNC(C2CN(C)C(=O)N2)=O)n[nH]c2c1CN(C(=O)CC1OCCCO1)CC2 n1(C(C)C)ncc(C(=O)NCC2(NC(=O)CCCC3CCC3)CCOC2)n1 C1(CNC(C(CC)F)=O)CN(C(c2[nH]cnc2C)=O)CC(C)(C)O1 c1(SC)nc(C)cc(=NC(C)c2ccc(CC(c3cc(F)cc(F)c3)=O)cc2)[nH]1 N1(C(c2cc3ccccn3n2)=O)CC2CCN(Cc3ccc(I)c(F)c3F)C2C1 N1(C(=O)CCC2CC2)CCC(O)(C2CCN(C(c3ccc(C4CC4)nn3)=O)CC2)C1 C1(NC(C(C)OCCCC)=O)CCCCN(C(c2nc(C)c(N)cc2C)=O)CC1 N1(C(CC2CCC(NC(C(C)(C)N3CCCCC3)=O)C2)=O)CCC=C(F)C1 C123CC(C1)(OC2C)CNC3=O.C1(NC(CCNS(C)(=O)=O)=O)CCN(C)CC1 C12(CCCCCC1)C(=O)N2.c1(CNC(c2cc(O)cs2)=O)cnn(C2CC2)c1 C12(NC(C(C)C)=O)CC(CNC(c3cnn4c3CCCC4)=O)(C1)OC2(C)C C=CCC(C)(C)CC(=O)NCC(C)(C)OCC(=O)NCC1(O)CCOCC1 C(=O)(CC(O)C(Cl)(Cl)Cl)N1CCC(NC(c2cc(C(C)C)c(N)cc2)=O)C1 CN1CCN(C(c2sccc2F)=O)C(CNC(c2cc3occc3s2)=O)C1 O=C(N=c1cc(CCO)[nH][nH]1)C1CC(F)CN1C(c1cc(O)cc(Cl)c1)=O N1(C(c2ccc(NCCOC)cc2C)C(=O)NC)CCN(CC(F)F)CC1C C(c1cc(C)cc(C)c1)=CC(=O)NCC1(C(C)NC(C(COC)(C)O)=O)CC1 CCC(CCC(=O)N1CC(OCC(C)C)C1)OC(=O)CCCCCF C1(C)(C(=O)NCCC2CC(NC(CC(=O)NCC)=O)C2)CCCC1O CCC(O)(CC(=O)NC1C2CN(C(=O)C=C(C)C3CC3)CC12)c1ccccc1 c1(C(=O)NCC(CNC(c2cccc(OC)c2F)=O)(C)O)coc2c(C)cccc12 N1(C(Cc2ncc(CC)[nH]2)=O)CCC(C2CC2)C1CNC(c1cc(Cl)ns1)=O N1(C(c2c(SCC)cncc2)=O)CCC2(CCC2NC(C2CCCO2)=O)CC1 N#CC1(C(=O)NCC2(C(F)F)CCN(C(C3(n4cncn4)CC3)=O)C2)CC=CC1 N1(C(=O)OC)CCCC(N(C(CNC(=O)C=C2CCC2)=O)C)C1 C#Cc1ccc(Cl)c(C(=O)NC2(CCNC(=O)C=Cc3sccc3C)CCC2)c1 c1(C(N2CCC(CCNC(CNS(CC)(=O)=O)=O)C2)=O)cccc(SC)n1 Cc1oc(C(=O)NC(C)CCNC(C2CCCCC2O)=O)cc1-c1ccccc1 Cc1cccc2c1OC(C(=O)NC1CC3(NC(=O)C4=CCCCO4)COC1C3)C2 C1(OC)CC(CNC(C2(CO)CCCO2)=O)N(C(=O)CC2CC3(CC3)C2)C1 c1(C(=O)NCCN(C(c2c(OCC)c[nH]n2)=O)C)cccc2c1C(=O)CCCC2 C1(N(C2CN(C(=O)CC(C3CCCCCC3)N)C2)C)CN(C)CCO1 c1(C(=O)NC(CN(C(=O)C(O)C(F)F)CC)C)cc(O)ccc1OC c1(CNc2nccc(-c3ccc(OC)cc3F)c2)ccccc1[N+](=O)[O-] N1(C(c2nc(C)sc2)=O)CCN(C(C2=CC(Cl)(C(C)C)C=C2)=O)CC1C c1(C(=O)NC2CC(C)N(C(c3ccns3)=O)C2)c(F)cccc1Cl C1(C(=O)NCCC(C)(C)SC)CCN(C(c2c[n+]([O-])c(C)cn2)=O)CCO1 c1(C(=O)NCCN(C(CC(OCC)OCC)=O)C)cn2cc(C)nc2s1 C1(CC)C(NC(=O)C(O)CC(F)F)CCCN1C(c1cnn(C2COC2)c1)=O C(=O)(CCCCCN=[N+]=[N-])NCCOCCCN(C(C(C(C)C)(C)O)=O)C NC1CC(C(=O)Nc2cccc(OCCO)n2)C12CC(F)(F)C2 N1(C(C(C(CC)C)=O)=O)CCC(C(=O)Nc2cc(O)c(F)cc2F)=C(F)C1 C(C)(N(C)N1CCC(C)C1)c1c(C)n(C)nc1 CC1CCN(C(c2cc(F)cnc2O)=O)CCN1c1nc(C(C)(C)C)nc(=N)[nH]1 C(=O)(C(C)(C)C(=O)NCC1CCC(NC(c2ccnc(C)n2)=O)C1)NC S(=O)(=O)(c1cccc(C(F)F)c1)NCC1N(C(C2C(C)CC(=O)N2)=O)CCOC1 CN1CCn2ncc(C=O)c2C1=O.C1(F)(CNC(=O)C(=O)O)CCOC1C C1(C(=O)NCC(CC)C)N(C(c2ccc(O)c(C)c2)=O)CCC1(C)C N1(C(c2c(CNC(C(C)O)=O)cco2)=O)CC2(C1)CN(C)CCO2 Cc1c(C(=O)NC(C2CCCCN2C(=O)CCc2cn[nH]c2)C)nnn1C N1(C(COc2c(OC)cccc2)=O)CC(NC(c2cnnn2C)=O)CC1(C)C CC(C)(CO)C(CO)NC(=O)C1=CCN(C(=O)C=CC(=O)NC2CC2)C1 C1(C(N2CCC(CN(C(CCSC)=O)C)CC2)=O)Cc2ccccc2S1 C=CCCCCCCCC(=O)NC1CS(=O)(=O)CC1NC(C1CCCCC1)=O C(=O)(CC(C)(C)Cc1cn(-c2ccc(Br)c(C)c2)nn1)N(CC(CC)C)C N1(C(CC2C(NC(c3snc(C)c3N)=O)CC2O)=O)CCC(F)C(O)C1 Cc1ncc(C(=O)NCCOC2CCN(C(=O)CC(C)N3CCCC3=O)C2)s1 Cc1cc(C#N)nc(=NCCN(C(C2CCS(=O)(=O)N2)=O)CC2CCCC2)[nH]1 N1(C(C2(CC)CCCCC2C)=O)CCN(C=O)CC12CC2.n1(C(C2CC2)C)nccn1 C1(C(F)F)(OC)CCN(C(=O)CCc2nnc(C)n2C)CC1 C1(C(=O)NC2C(C(=O)OC)CC2)N(C(=O)CCc2ccccn2)CCCC1(C)C c1(C(N(C2CN(C(=O)C(C)(C)c3ncco3)CC2F)C)=O)cc(Cl)cnc1O C1(C(=O)NC(C(C)C)C(=O)NCC2(CN(C)C)CC2)C2CCC(C2)C1C C1(CNC(CC=C=C)=O)C(C2CC2)CCN1C(c1cnc(C)[nH]c1=N)=O c1(N2CCCC(OCC)C2)ccc(Br)c(S(=O)(=O)NCc2cc(C)ccn2)n1 n1(CC(=O)NC2(COC)CCN(C(c3c[nH]nc3C)=O)C2)cc(P(C)(C)=O)cn1 C1(C(N)=O)(NC(COCCC#C)=O)CCCN(C(=O)CC(C)C(=O)OC)C1 c1(C(N(CC)Cc2cccs2)=O)cc(-c2ccccc2SC)cc2[nH]ncc12 Nc1ccccc1CCNC(=O)NCCc1coc(-c2ccccc2)n1 C(=O)(CCCC(=O)NC)N(CCC)CCC.C12CCCN(CC1)C2=O c1(NC(CC)(CNC(=O)CNS(C)(=O)=O)CC)cnc2ncnn2c1C C1(C(N2CCC(CCOC)C2)=O)CCN(C(C2CCCCC2)=O)CCO1 c1(C(=O)NCCCN(C)C(c2cncnc2)=O)cnn(C)c1Br c1(CS(=O)(=O)NC(C(C)(c2ccccc2)N(C)C)=O)ccc(Cl)cc1 C(=O)(C1=NOCC1)NC(C(=O)N(C)Cc1cnsc1)CC1CCCCC1 N1(C(c2ccc(C)cc2)=O)CC(NC(c2c[nH]nc2F)=O)C(N=[N+]=[N-])C1 c1(CC)cccc2[nH]c(C(N3CCC(CNC(=O)C(C)SC)C34CCC4)=O)cc12 C(N=c1[nH]c(-c2cc3sccc3[nH]2)cs1)c1c(C)noc1C Cc1ccccc1C(C)NC(c1ccc(C2CCCO2)cc1)=O C1(C(=O)NCC2(CC(=O)OC)CCCC2)CN(C(C23CCC(C2)C3)=O)CCO1 C12(C(=O)NC(CCC)c3ccco3)CCCC1N(C(C1CCCSC1C)=O)CC2 C1(C(=O)Nc2cccc(NC(C(c3n(C)cnc3)O)=O)c2)CCCC(C)(C)CC1 N1(C(C(C(C)C)C)=O)CC2(C1)SCCC2CNC(c1ccc(OC(F)F)cc1)=O c1(OCC(=O)NC(C2CN(C(C3OCCO3)=O)CCO2)C)cc(Cl)cc(Cl)c1 c1(C(=O)NC(CNC(C(N2C(CC)CCC2)=O)=O)C2CC2)cc(C2CC2)nc(O)c1 C1(C(=O)NC(c2cnn(C)c2)C(=O)N(CCCC)C)CC(C)(C)C1 C(=O)(CC=C(Cl)Cl)NC(C(=O)NC(COC(C)C)C)C1CCC1 C(C(F)(C(=O)NC1(C2CCCO2)CC1)C(C)C)NC(C(C)(C)OC(C)=O)=O N1(C(=O)C(c2cccc(Cl)c2)O)CCC2(CC1)CC2C(N1CCCCCC1)=O CC(CC(F)(F)F)C(=O)NC(c1nc(C(=O)N(C2CCC(C)(C)C2)C)co1)C N1(C(CCC2C(=O)NC(=O)N2)=O)CC2(CC(C=O)C2)C1.O=CC=C1CCC1 C1(NC(c2cnc(CC3CC3)[nH]2)=O)CN(C(C2CC2CF)=O)CC1C1CC1 N1(C(C=CC(C)=O)=O)CCC2(CCN(C(=O)C(C)(C)S(=O)(=O)C3CC3)C2)C1 N1(C(c2n(CC)ccn2)=O)CCN(C(C2(C(=O)N(C)C)CC2)=O)CC1C(C)(C)C N1(C(c2ccnc(C(N3C(CC(N)=O)CCCC3)=O)c2)=O)CC2(CC(O)C2)C1 c1(C(=O)NCCCCCN(C(C(C)NC(C)=O)=O)C)cc(Br)cnc1C c1(C(=O)NC2CC(NC(c3nn(C)c(O)c3)=O)C2)cc2cccn2c(O)n1 C(=O)(CC(C)(C)C(F)F)N1CC(O)(C(C)NC(=O)C=Cc2ccc(Cl)s2)C1 c1(C(=O)NC(c2cn(C3CCCNC3=O)nn2)COC)cc2ccccc2s1 c1(NC(=O)C(C)(C)C(N)=O)c(C)cc(-c2cn(CC(F)(F)CO)nn2)cc1C C1(NC(CCc2nnc(C)n2C)=O)CC12CCN(C(C1CNC(=O)N1C)=O)CC2 CC1CCCn2c(C(=O)NCCC3CCCCN3C(=O)CCN(C)C)cnc21 C(=O)(C#CC(=O)NC1CCC(NC(=O)CC2COC3CC2C3)CC1)N(C)C c12cc3c(s1)CCC(C3)CN2.C(=O)(CCCONC(=O)OC(C)(C)C)NC C1(CNC(C2(F)CCN(C(C3CCCSC3)=O)C2)=O)CC2CCCC2C1 S(=O)(=O)(c1cc(C(F)(F)F)cc(Br)c1)NC(CCCC)(C)C(N)=O N1(C(CCCC(N)=O)=O)CC2CCCC2(NC(c2coc(CC3CC3)n2)=O)C1 C1(CC)CN(C(=O)CCc2cc(C)no2)CCC1NC(=O)Cc1n[nH]c(=N)s1 c1(OC)cc(CN=C(NC(C)C)NC(c2cccs2)C)c(F)cc1Cl C1(NC(C=CC(C)C)=O)CCCCC1CNC(=O)CCCN1CCCC1 C(=O)(C1CCCn2cc(C)nc21)NCC1C(NC(Cc2cn(CC)nc2)=O)CC1 c1(C(=O)NC2(C)CN(C(C3(CC=C)CC3)=O)C2)cc(C(F)(F)F)ccc1N N1(CCC)CCCCC1C(N1CC(CNC(=O)COCCCOC)C(O)C1)=O CC1(C)CC(C)(C(=O)NC(C)(C)CNC(=O)CCNC(C2CCCC2)=O)C1 C(C)(CC(=O)NCC(C)(C)CNC(=O)C(F)(F)c1cnnn1C)OC Cn1[nH]c(CNCC(CO)NC(=O)CC2CNC2)nc1=O c1(C(=O)NC2CCCN(C(c3c(C)noc3)=O)C2)n[nH]c2c1CCSC2 C#CC1CCCN(C(=O)C(F)CC2CN(C(C3CN(C4CCC4)C3)=O)C2)CC1 c1(C(=O)NC2CN(C(C(C)N(C)C)=O)CC2N=[N+]=[N-])c(Cl)nc2ccccn12 N1(C(c2n(C)c(S)nn2)=O)CC(=O)N2CCCC2C1.C1C(=O)N1 N1(Cc2c(OC)cc(C)cc2C)CC2(CCCC2)c2c(F)cccc21 C1(C(=O)NC2CN(C(CCc3ccc(CC)cc3)=O)CC2C)CC(C)(C)CN1C c1(CC(=O)NC(CC=C)CNC(C2CC(O)CN2C)=O)cc(C)ccc1O Cc1cc(C)c(CC(=O)N(C2CC(NC(=O)CC3CC4CC4C3)C2)C)c(C)c1 c1(N2C(CCNC(C3(C#C)CC3)=O)CCC2)cc(C(=O)OC)nc(Cl)n1 CC1(C(N2CCC(O)C(CNC(=O)C(O)C(C)(C)C)C2)=O)CCCCCC1 CC1CCCN(C(c2n[nH]c(=N)s2)=O)C1CNC(C1CCNC(=O)C1)=O C(C)(C(CO)NC(C1CCS1(=O)=O)=O)NC(C(C)NC(C)=O)=O c1(OCCOCC)cncc(C(N2CCC(COC)C2)C(=O)NCCC#N)c1 c1(CC)nc(=N)[nH]cc1C(N1CCCC1C1CC1NC(=O)CCOCCOC)=O C(=O)C(C)(C)N(C)CCN(C)CCSC(F)(F)F.C(COC)OC Cc1ccc(O)cc1NC(=O)CCN(C(=O)C(C)C(C)(C)C)CCCO CCC(CNC(C1(N(C)C)CCCC1)=O)(CC)C(=O)NC1CC(C)OC1=O N1(C(=O)NC2C(C)CN(C)CC2)C(C(=O)O)C2CC(O)C1C2 c1(C(=O)NCC(CNC(C(CC=C)OC)=O)(C)F)cccc(O)c1F C1(C(N2C(CCNC(c3nc(CC)sc3N)=O)CCC2)=O)CCCCC12CCC2 c1(C(C(=O)NCCC)N(CC(C)CC)CC)ccc(Cl)cc1Br c1(NC)cccc(C(=O)N(C)CC2CCCN2C(c2csnc2C)=O)n1 C12(C(=O)NCC(CC)NC(c3ccc(C)s3)=O)CCCCC1C2(F)F c1(C(=O)NCC2OCCN(C(c3cnc(CC)[nH]3)=O)C2)ccc(F)c2[nH]ccc12 n1(COC)nncc1C(C(=O)NCCC#N)N(CC(C)C)C(c1ccccc1)C C1(NC(C=C(COC)C)=O)CCC12CN(C(c1nc(O)sc1C)=O)C2 c1(C(=O)NC2C(C(N(CC#C)CC=C)=O)CCC2)cc(Cl)cnc1OC Cc1ncncc1C(N1CC=CC1(C)C(=O)NCC(C)(C)CC1CC1)=O C12(C(=O)NCCC(C)NC(c3cncn3C)=O)CC(CC(F)F)(C1)C2 C1(C(C(=O)N2CC(CCO)C2)NC(C2CCC2(F)F)=O)CCCCC1 C(CN=c1nc2sccc2c(NCc2ncc[nH]2)[nH]1)(C1CC(F)(F)C1)OC c1(C(=O)Nc2cc(C(F)F)ccc2CO)cc2ccccc2o1 CCCC(CC)C(=O)N1CCN(C(=O)Cc2cnsc2)C(c2cn[nH]c2)C1 C1(NC(CC(=C)C)=O)CC(C2CCN(C(c3cc(O)ccc3F)=O)C2)C1 C1(C(=O)NC2CCC2)CC2(CC(NC(C=CC(=O)OC(C)(C)C)=O)C2)C1 C(=O)(CS(=O)(=O)C(C)C)NC1CCN(C(c2c(CC)n(C)cc2)=O)CC1F CC(C)C(O)C(F)(F)C(=O)N(C)CC1(O)CN(C(=O)CN(C)C(C)C)C1 C1(NC(C(CC#C)(C)C)=O)CN(C(=O)CC(C)(C)COC)CC1N=[N+]=[N-] CN1CCN(C(C)(C)CNC(C2CCN(C(c3ccccn3)=O)CC2)=O)CC1 N1(C(C(c2cnccn2)C)=O)CCC=CC1C(=O)N(C)CC1CCCN(C)C1 N1(C(C2CC(=C)C2)=O)CCCC(CCC(C)C)(NC(c2cc(C#N)cn2C)=O)C1 C1(N(C(Cc2c(C)cc(C)s2)=O)C)CCN(C(C23CC(C2)C(C)O3)=O)CC12CC2 C1(C(=O)NCc2c(OC)cccc2)CN(C(=O)CCC2(C)CC2)C(C)(C)C1 C1(NC(Cc2nc(CC)on2)=O)CC1C1CCCN(C(c2cc3sccc3s2)=O)C1 C1(CNC(c2scc(C)c2)=O)CCCCN(C(c2ccnc(Cl)c2O)=O)C1 C(=O)(CCCNC(=O)CSCCN)OC(C)CCc1ccccc1 C1(CC(N2CCC(N(C(c3csc(C(C)OC)n3)=O)CC)C2)=O)CCC(=O)N1C C(C(C)N=c1[nH]c2cc(Cl)cc(Cl)c2o1)(C1CCCCC1)NC(CCC(=C)C)=O C12(COC)CC(CNC(c3ccccc3C3CC3)=O)(CN1C(c1ccsc1)=O)C2 c1(CNC(N(C2CC3COCC23)C)=O)ccccc1OC1CCCC1 C1(C#N)(C(=O)NCCC2(CNC(C(C)OCCC(C)C)=O)CC2)CC2CC2C1 c1(OC)ccc(C(N2CC(NC(c3ncccn3)=O)CCC2C)=O)cc1Cl C(=O)(C1=CS(=O)CCC1)N(C1CCCN(C(=O)CCC2CCC2)C1)CC C1(CNC(C=C(C)C(F)F)=O)CC2CCC1N2C(c1cc(C(F)F)[nH]n1)=O Cc1nc2ncc(C(=O)NCC3CC3NC(c3cc4c(s3)CCOC4)=O)cc2o1 C1(NC(C(CC)N(C)C)=O)CN(C(=O)Cn2ccc(=O)cc2C)CC12CCCC2 C1(O)(CC)CCC(NC(C2(CO)CCN(C(c3cnn(CCO)c3)=O)C2)=O)CC1 CC1CNCC(CNC(c2cc(C3CC3)n(-c3ccccc3)n2)=O)O1 c1(OCCC(=O)NCC2CN(C(C(CC#C)C)=O)CC2C)ccc(F)cc1F N1(C(c2c(C)onc2-c2ccccn2)=O)CC(NC(=O)C=CCO)C2(CCC2)C1 C(C(C(C)(C)C)NC(C1CCC(C)CC1)=O)NC(C1=CC1CC(=O)OC)=O C1(NC(c2cccc(-n3cc(C4(C)CCCOC4)nn3)c2)=O)CC1C1CCOCC1 N1(C(C2(CC)CCN(C(=O)C=CCOC)C2)=O)CCCC(C)(C)C1C CCCC(C)(CC)C(=O)NC12CCCN(C(=O)CCNC(c3ccco3)=O)CC1C2 CC(C)C(C)(O)C(=O)N1CCCC(CCNC(C2(c3ccno3)CC2)=O)C1 C(=O)(CC(F)(F)C(F)(F)F)NC1CCN(C(C(COC)COC)=O)CC1(C)C Cc1ncc([N+](=O)[O-])n1CC(N1CCC(NC(=O)COC(C)C)C1)=O C(=O)(C1=CCOCC1)N(CC)CC1CCCCN1C(=O)CCCc1cc[nH]n1 n1(CCCN(C)C)nc(-c2cccc(Cl)c2)nc1-c1cnc(N(C)C)o1 c12nc(OC)cc(n1)O2.c1(COC)ccc(C(C)NCCc2ccnn2C)o1 C1(N(C(c2cnc(C(C)(C)C)s2)C(=O)NCCCF)CCC)CCCCCC1 c1(OCC)ccc(C(F)(F)F)cc1OC.N1(CC=O)CCC1(C)C(=O)OCC Cc1nn(C)c(-n2cccn2)c1C(=O)NCc1n[nH]c(C2CC2)c1Cl N1(C(CCOC(C)C)=O)CCC2C(C1)CN2C(=O)CCCC(F)F C(=O)(C(C)(C)CCNC(c1ccnc(O)c1)=O)NCC=CC(C)(C)C C(=O)(C(F)C(F)(F)F)NC1C2(CC(NC(=O)CCCCc3ccccc3)C2)C1 c1(OCC)ncnc(OCC)c1C(N1CCC(NC(C2(F)CCCOC2)=O)C1)=O