SMILES N1(C(CCNC(c2cc(C)cc(F)c2)=O)=O)CCC(C)N(C(=O)C=CC2CC2)CC1 c1(C(=O)NC(C2(CNC(C(CC)C)=O)CC2)C)ccc2c(c1)C=CS2(=O)=O c1(N2CCC(COC)(CO)C2)ncnc(NCc2ccccc2CC2CC2)c1C C1(OC)CN(C(=O)CN2CCC(C)CC2)CC1NC(C1CCCN(C(C)C)C1)=O Cc1nn(C)nc1C(=O)NC1COCC1CNC(=O)CC(C)c1ccccc1 C1(O)(C(C(=O)NC(c2cnsc2)C)NC(CCCOCC)=O)CCCCC1 c1(CNC(C2CCCC(C)(C)CC2)=O)ccc2cc(Cl)ccc2n1 C(=O)(C(C(C)O)NC(N)=O)NCC(n1cc(C(C(C)C)NC(N)=O)nn1)C c1(NC(CC)CC#N)ccc(S(=O)(=O)NCC2(CCOC)CC2)c(Br)c1 c1(CC)cc(C(=O)NC2CCCC(CNC(C3CCCC(=O)O3)=O)C2)nn1C Cc1cc(C(=O)NC(c2nocc2C(=O)NCC2COC(C)(C)C2)C)ncc1F Cn1cnnc1CC(=O)NC(C(=O)NCC1CC1C(N)=O)C1(C)CC1 N1(C(c2c(OCC)ccc(C)c2)=O)CC(NC(=O)Cc2cncs2)CC(F)(F)C1 c1(C(N2CCCCC(Nc3c(C#N)c(Cl)ncn3)C2)=O)cc2cccc(F)c2o1 Cc1cc(-c2cn(CSC3CCN3C(=O)C(C)CSC(F)(F)F)nn2)cc(C)c1 C1(C(N(C2(C(=O)OC)CC2)CC)=O)CC(C)N1C(=O)CCC1CC1 CCC(CN=c1[nH]c(N(C)Cc2cc(F)cc(Cl)c2)nc2c1CCCC2)OC c1(OC)cc(Cl)ccc1C(C)NC(C1(C)CCCN1NCCF)=O C1(O)(C(=O)NC2CN(C(c3c(OC)c(C)cs3)=O)CC2O)CCC(C)(C)CC1 c1(C(=O)NC2CCN(C(c3c(NC)cccc3)=O)CC2C)nnc2n1CCOC2 N1(C(C(C=C)O)=O)CCn2ncc(CN(C)C(c3nccc(C)n3)=O)c2C1 C(=O)(CC(O)C(C)C)NC(C1(CNC(c2cn(CCOC)nn2)=O)CC1)C c1(CC)ncc(C(=O)NC(C)(C)CNC(C2CC2CF)=O)s1 c1(C(N(C2CCN(C(c3c(CC)c(C)sc3)=O)CC2)C)=O)cc2occc2s1 C1(NC(c2cn(CCC(C)C)nn2)=O)CN(C(=O)C=Cc2ccoc2)CC12CC2 c1(NC(C)(C)C(=O)NC2C(OC)COC2)cncc(OC2(CCCCO)CC2)c1 c1(C(=O)NCCCC2CCN(C(C(OC)OC)=O)CC2)cn2ncccc2n1 Cc1csc2c(CC(=O)Oc3nnc(Br)s3)cccc12 N1(C(C(C=CCCC)O)=O)CCC(NC(c2cc(C(F)F)ccn2)=O)C(F)C1 N1(C(CC(C(F)(F)F)OC)=O)CCC2(C=C(C(=O)N=c3ccn(C(C)C)[nH]3)C2)C1 O=C(CCCSCc1ccccc1)NCCC(C)NC(=O)C(c1cccnc1)O CC1(C)CC(NC(c2ccc(C(F)F)s2)=O)CN(C(c2cc(N)cc(F)c2)=O)C1 N1(C(C2(CC)CCC(O)CC2)=O)CC2CCCCC2(NC(C2CCCC2O)=O)C1 c1(OC)ncc(F)c(Nc2ccc(C(=O)Nc3cc(F)c(C)cn3)nc2)n1 C1(C(N2CCCC(CNC(c3ccsc3Br)=O)C2)=O)CCCC1C1CC1 N1(C(CN2CC(CC)C2)=O)CCCN(C(=O)C(C)(F)CC)CC1 CCC(C)(COC)C(=O)NCC1CCC1NC(c1cc2n(n1)CCC2)=O c1(NC(CCOC)=O)cnc2ccnn2c1.C1(=O)C(F)CC2CN1C2 C1(N(C(c2cn(CC(F)(F)F)nn2)=O)CC)CCCN(C(C2CCC2)=O)C1 CS(=O)(=O)c1cncc(C(=O)NC2CCCN(C(C34CCC3C4)=O)C2)c1 N1(C(COC(CC)C)=O)CCC2CCN(C(c3c(O)cc(F)cc3F)=O)CC2C1 N1(CCN(C)C(C2(c3cccs3)CC2)=O)CCC(c2ccon2)C1 c1(OC)cc([N+](=O)[O-])ccc1C(=O)NCC1CN(C(=O)CC(C)c2ccccc2)C1 C1(CNC(CC(=O)NCC)=O)CN(C(=O)Cc2cc(C)nn2C)CCC12CCC2 C1(C(N2CC3C(CNC(Cc4cnc(C)[nH]4)=O)(C3)C2)=O)CC2(C1)CC(C)C2 c1(C(=O)NC23C(CN(C(Cc4c(C)ccnc4)=O)C2)C3)ccc2nnnn2c1 N1(C(C(C)NC(C)=O)=O)CCC(NC(=O)Cc2scnc2-c2ccccc2)C(F)C1 Nc1cc(C(=O)NCC2(NC(=O)CC3(O)CCC3)CC2)cc(F)c1 C1(CC(=O)NC(C2(O)CN(C(c3cc(N4CCC4)ccn3)=O)C2)C)CC(=O)NC1=O N1(C(CNS(NC)(=O)=O)=O)CC(CNC(=O)Cc2nonc2C)N2CCC1C2 c1(OC)ccc(Cl)c(C(N2CC(N(C)C(c3ncoc3C)=O)C3(CC3)C2)=O)n1 c1(OC(F)F)cc(CCNC(c2ccnc(OC)c2)=O)cc(F)c1OC.CO CC1(C)C(NC2CCC23CCCC3)CC1O N1(C(C2(SC)CC(=O)C2)=O)CC2(CC(CC(=O)NCC(C)C3CC3)C2)C1 C(C(CC(=O)N1CC(CN2CCC(=O)CC2)C1)NC(c1ccoc1)=O)OC CC1=NOC(C(N2CCCC2C(C)(C)CNC(C2(N3CCOCC3)CC2)=O)=O)C1 C1(C(=O)NCC2(F)CCN(C(CP(C)(C)=O)=O)C2)CC1C1(C)COC1 N1(CC(=O)Nc2cccc(NC(Cc3cccc(C)c3)=O)c2)CCNC(=O)CC1 S(=O)(=O)(c1cnc2ccoc2c1)N1C(C)CC(c2ccc(F)cc2)C1 C1(C(N2CC(OCC)C2)=O)CCN(C(c2[nH]nnc2CC)=O)CC1(C)C N1(C(CC)=O)CCCC(C(N2CCC3C(NC(c4ncn(C(C)C)n4)=O)C23)=O)C1 c1(C(N2C(CN(C(C(COCC)C)=O)C)CCC2)=O)cnn(C2CCC2)c1C CC1CC(NC(C2(C)CCN(C)C2=O)=O)CCN1c1nc(C(C)(C)C)nc(=N)[nH]1 C(=O)(C(CCCCN)CC(F)(F)F)Nc1cn(-c2nnc(C(=O)OCC)o2)nc1 C(C(N=[N+]=[N-])C(=O)NCC(C)NC(=O)C(C)CC(F)F)OCC N1(C(c2cnc(CC)s2)=O)CC(CNC(c2cc(Cl)n(C)n2)=O)C(C(F)(F)F)C1 C1(NC(C(C)(N(C(c2nc(OCC)oc2)=O)C)C2CC2)=O)CC2COCC2C1 c1(N(C(C2CCCN(C(C(C)SCC)=O)C2)=O)CC)c(OC)cc(Cl)cc1F C(CCN=C(NCc1ccc(SC)o1)N1CCC(C(N)=O)(CO)C1)OC Cc1ccc(N2CCCC2C(=O)OCCCO)cc1.N1(CC(C)C)CCCC1 N1(C(c2cc(OC)nc(F)c2)=O)CC2CC(C1)C(CO)C2NC(=O)C(C)(F)F C(=O)(C(C#N)C(C)(C)C)NC(C)(C)CCNC(=O)Cc1cncc(O)c1 N1(C(c2c(C)c[nH]c2)=O)CC(C)N(C(c2cc(Br)c(Cl)cc2C)=O)CC1C C(C1=CCN(C(C2CC(C3CC3)=NO2)=O)CC1)NC(c1ccc(=O)oc1)=O c1(C(N(C2CCN(C(=O)CC3CC34CC4)C2)C)=O)ccnn1CC1CCC1 CC1CCN(C(C2CC2OC(C)(C)C)=O)CCO1.c12csc(c1)CNC2=O C1(C2CCN(C(=O)C(C)(C)C(C)O)CC2)(NC(C(CCC)N(C)C)=O)CC1 N1(C(CC(CCC)c2ccccc2)=O)CC2CCN(C(c3ncncc3Cl)=O)CC12 C1(C(=O)NCc2occ(C(N3CCC(OC)(CO)C3)=O)n2)CC2COCC2C1 N1(S(=O)(=O)CCCl)CCN(Cc2cc(Cl)cc(Cl)c2F)C2(CC2)C1 N#CC1CN(Cc2ccc(Br)[nH]2)CC1NC(c1cncc(-c2ccccc2)c1)=O C1(OCC(=O)NC2CC(N(C(=O)Cn3cnc(=N)[nH]3)C)C2)CC(CO)C12CCC2 C#Cc1cc(C(=O)NCC(C)(O)CNC(=O)C=CCC)cc(N)c1 C(=O)(CC(C)(C)C(=O)NCC1(CNC(=O)C(C)O)CCOCC1)OC c1(CC(C(=O)NCC(N(C(COCCCC)=O)C)C2CC2)O)ccc(Cl)cc1 C12(OC)CCCN(C1)C2=O.c1(NC(C2CCOC2=O)=O)ncccc1C1CC1 C1(C(=O)NCCC2N(C(C3C(C)CCOC3)=O)CCC2)CC(=O)NC(=O)C1 C1(NC(C2C(C(C)NC(C(CC)CN(C)C)=O)C2)=O)CC2(CCCCO2)C1 CCC(C)CCCC(=O)N(C)CC1CCCCN1C(c1cccc(C#N)c1)=O Cc1ccc2c(CNC3CCCN(c4ncnc5cnccc45)C3)cn(C)c2c1 C=Cc1cc(C(=O)N(C)CCN(C(c2cc(CN(C)C)on2)=O)C(C)C)cc(F)c1 CC1CCCC(C(N2CCCC2CCNC(C23CCC(CC2)C3)=O)=O)C1 C1(CNC(c2c(N)nccn2)=O)CCCCN(C(C2(C(F)F)CCCO2)=O)C1 c1(C(N2C(CNC(CC(C)OC)=O)C(C)(C)CC2)=O)cccc2c1C(=O)CC2 c1(C(=O)NC(CC2CN(C(c3ccc(C(C)C)o3)=O)C2)C)cc(O)nc(O)n1 CC(O)C(=O)NNC(=O)NCc1cccc(F)c1I C1(NC(C2N(C(C=NOC)=O)CCOCC2)=O)CCOCC12CCC2 N1(C(C(C(C)CC)N(C(CC=CC)=O)C)=O)C2CCC1CC1(CC1)C2 c1(ON)ccc(F)c(N)c1C(=O)NC(c1ccc(-n2cncn2)c(F)c1)C C1(CC(=O)NC(CNC(CSCCOC)=O)C(C)C)CCCCCO1 C1(NC(Cc2nc(C)[nH]n2)=O)C2COCC1CN(C(c1cnncc1C)=O)C2 C=CC1CN(C(=O)NC(C(=O)OC)C2CC2)CCO1 CC1(CNC(C2CC(NC(c3ccc(O)cn3)=O)CCO2)=O)CC=CCC1 CC(C)=C=C1C(=O)NC1CCCCC1C(CCCCC)CC(F)C(=O)N1 C1(C(=O)N(C)C)CCC(NC(C2CC(n3cc(CN(C)C)nn3)CC=C2)=O)CC1 CCC(CC)(CO)C(=O)NC1CC(NC(=O)Cn2cc(Br)nn2)C1 CC(C)(C)C(C(=O)Nc1ccc(C(N2CCCC2)=O)cc1)c1ccc(Cl)cc1 C1(NC(C(C)OCC=C)=O)CC(C)(C(=O)NCC=CC(C)(C)C)C1 N1(C(Cc2cc(C)sc2C)=O)CCN(C(=O)CNC(c2cccs2)=O)C2CCC12 C(=O)(C(C)CCCCCC)N1CC(NC(CCCC=C)=O)C2(C1)CCC2 c1(C(=O)NC(C2CCCN2C(C2(Sc3ccno3)CC2)=O)C)csc(C2CC2)n1 C1(C(N(C(CCCC)C)C)=O)CN(C(=O)Cc2c(C)cnn2C)CCN1C c1(OC)c(Cl)cc(C(=O)NC23CCCC2CN(C(c2cnc(S)[nH]2)=O)C3)nc1Cl Cn1cnc(C(N2CC(O)(C(C)(C)CNC(C3(CF)CC3)=O)C2)=O)c1 CCCC(CCCNC(C1CCC1C)=O)NC(c1c[nH]nc1-c1ccn(C)n1)=O N1(C(C)=O)CCCC1(C)C(=O)NCC1(O)CCN(C(=O)CCCC2CC2)C1 C#Cc1c[nH]nc1C(=O)NCC1CC(F)CN1C(c1ccoc1Cl)=O c1(C(=O)NCC(CC=C)NC(c2ncn(C(C)C)n2)=O)ccc(C2CC2)cc1C c1(C(=O)OC)ccc(NCC2CCCN(C(=O)C(=O)OC(C)=O)C2)cc1Cl N1(C(C(C)N(C(c2cnnc(C)c2C)=O)C)=O)C2CCC1CC(C)C2 c1(NC(C2(C)CCC3(CC2)CC3)=O)nc2c(F)cc(Cl)cc2s1 C(CC(CC)C(=O)NCC(O)CC(=O)N(CCC(N)=O)C1CC1)=CC C(=O)(CCCC(C)(C)C)N1CC(C(=O)NCCCC(=C)Cl)C(C)C1 n1(CC)cc(C(=O)NC23CC2CN(C(C2CC(F)(F)C2)=O)C3)c(C)n1 N1(C(=O)OCC)CCCC(C(=O)NC23CC(NC(=O)CC4CCOC4=O)(C2)C3)C1 C1(N(C(c2cc(CCO)on2)=O)CC)CCCN(C(=O)Cn2ncc(Cl)c2C)C1 c1(C(=O)NCC2C(C)CCN(C(=O)C(C)(C)CO)C2)ccc(S(N)(=O)=O)nc1 C(=O)(C(C)(C)C(N)=O)NCC(C)OC(=O)NC(C1C2CN(C(C)(C)C)CC12)=O CCCC(CCCNC(=O)Cc1cc(C)[nH]n1)NC(C1(CO)CCCCC1)=O CC1(C)CCN(C(c2csc(Cl)n2)=O)C1C(=O)NC1C(=O)OCC1CO CCC(CC)C(c1nnnn1Cc1ccco1)NC1CC1C(C)(C)C CC1CCC(NC(=O)CC2(O)CCCOC2)CN1C(c1cc(N)ccn1)=O CN1C(C)(CNCCCCc2ccc3c(c2)OCO3)CCS1(=O)=O C1(CNC(CC(C)(C)NC(=O)CCNC(=O)CO)=O)CC2(CCCO2)C1 c1(CN2c3ccoc3C2=O)cc(F)c(Cl)c(Cl)c1.N1(CC)CCN(C2COC2)CC1 C1(n2cc(CCC(=O)NCC(CC#N)N)nn2)CCC(C(=O)O)CC1 c1(NC(C2CCC(C)CN2C(C2CN(C(N)=O)C2)=O)=O)cncc2ccccc12 CC1CN(C(c2c[nH]c(=S)cn2)=O)CCN1C(=O)C(O)Cc1ccccc1Cl c1(C(N(CCNC(CC2C(OC)COCC2)=O)C(C)C)=O)ccc(S(N)(=O)=O)o1 c1(CC)nc(C)oc1C(=O)NCCOCC(=O)N(CC(O)CO)C C1(C(=O)NC(CCSC)C(=O)NC2CC(C#N)C2)CCc2c[nH]nc2C1 c1(C(N2CC(CC(C)NC(=O)C(F)=C3CCC3)C2)=O)cc2ccccc2s1 c1(C(N2CC3N(C(C4C(=C)CC4)=O)C(CC3)C2)=O)ccc(C2=NOC(=O)C2)cc1 c1(C(=O)NC(C)CN(C)C(C2CCCO2)C2CC2)cc(C(F)(F)F)ccc1F C12(C(=O)NC3CCN(C(CC4CCC(=O)C4)=O)CC3F)CC3CC(C1)CC(F)(C3)C2 C(CCCC(=O)N(C1CCC1)C)N(C(C=C(C)C(C)C)=O)C1CC1 N1(Cc2ccc(OCCCC)cc2)CC2CN(C(c3ccc(C)s3)=O)CC12 C(C(=O)N1CC(NC(C2(C)CC=CCO2)=O)C(C)C1)(C(C)C)NC(C)=O c1(CSC2CCC(C)OC2)cc(F)ccc1N(C)C c1(C(N2CC3OCC(NC(CC4C(C)(C)C4)=O)C3C2)=O)cncc2ccccc12 C(CC(N)=O)(C(=O)N1CCC(C)(C)CC1)NC(c1c(OC)noc1C)=O C(=O)(CCCCO)NC(CC(C)NC(C(C)OCCCC)=O)C C1(N(C2CCOCC2)CCCC)C2CC(n3cc(-c4ccncc4)nn3)C1C2 c1(OC)ncc(NC(C23CC2CN(C(c2cncc(C#N)c2)=O)C3)=O)cc1C C=CCCCC(=O)N1CCCC1CCNC(C1(OC)CC(C)C1)=O Cc1ccc(Br)cc1NC(N1CC(NC(c2ccc(Cl)cc2C)=O)C(F)(F)C1)=O N1(C(C2(F)CCN(C(CCNC(COC)=O)=O)C2)=O)CC(C#N)C2(CCC2)C1 C(=O)(C#CC1(C)COC1)NC1(C)CCN(C(C2CC(CCC)OCC2)=O)CC1 C1(CNC(c2ncc(C(F)F)cn2)=O)CC2(CCC2)CN1C(=O)Cn1cnnc1 c1(C(=O)OC)[nH]c2ccccc2c1C(C(=O)CC1CC1C)=O.C1(C=O)CCCC1.C1CN1 N1(C(C2(C)CC(C)C2)=O)CCC2(CCN(C(=O)CC3(C)CCS(=O)(=O)N3)C2)C1 C(=O)(C#CC1CC(F)(F)C1)NC(CNC(C(CCCC)(C)F)=O)(C)CO C1(CCC)(NC(=O)CCc2cc(C)[nH]n2)CCCN(C(=O)CS(=O)(=O)CC)C1 c1(C(N(C(c2ccccc2)COCC)C)=O)cc(F)c(O)c(Cl)c1 C1(C(=O)NC(CC=C)C2CC2)CC(C)(C)CN1C(c1ccnc(O)c1F)=O c1(CC(=O)N(CC(C)(C)CNC(c2cnn(C)c2)=O)CCC)ccc(CO)cc1 C1(NC(C2CSC2)=O)COC2(CCCN(C(=O)COc3cncc(Cl)n3)C2)C1 CCCC(C)(O)C(=O)NC1CC(C)(NC(C2CCC2(C)C)=O)C1 c1(C(N2CCC(C)C(NC(=O)CN3CCN(C)CC3)C2)=O)cccc2ccoc12 CCCCC(CNC(c1ccc(SC)cc1)=O)NC(c1n[nH]cc1C1CCC1)=O C1(N(C(=O)C=C(C)C(F)F)CC)C2CN(C(=O)CCN(C3CCOCC3)C)CC12 CC(C)CC(O)C(C)C(=O)N1CCC(N=[N+]=[N-])(C(=O)NC2CC(N3CC(O)C3)C2)C1 N1(C(C)C)CCCC1C(=O)NC1CCC1CNC(=O)Cn1cnnc1 c1(C(N2CCOCC(NC(C(CC)(C)C)=O)C2)=O)cc2c(F)cc(F)cc2[nH]1 c1(O)ccccc1F.C(=O)(CC(C)C1CC1)N(CC(=O)OC(CSC)C)CC N=c1[nH]cnc2c(C(N3CCCC(NC(=O)C(F)=C4CCC4)CCC3)=O)cnn12 c1(C(C(=O)OC)Sc2cnn(C3CCS(=O)(=O)C3)c2C)cc(Br)cc(Br)c1 Cc1c(C(=O)NC(C)(CNC(C2CC(C(F)F)C2)=O)CO)ccn1C c1(C(=O)NCC2(C)CCCN2C(C2CCSCC2)=O)ncc2ccccc2c1O N1(C(CN(C)Cc2n(C)ccn2)=O)CCC(CO)(NC(C2CCSC2)=O)C1 C(=O)(CCN=C(NCC(=O)N(C1CCCC1O)C)NC(c1cnn(C)c1)C)NC C#Cc1ccc(NC(C2CCC(CNCc3coc(C)n3)CC2)=O)cc1 c1(CN(C(c2cn(C)nn2)C(=O)NCCCC)CC)ccccc1Br CC(C)(CC(=O)NCC1CCC1NC(c1cc(F)ccc1F)=O)CC(F)(F)F C(CC(C)C)(C(=O)N1CCC(C(N)=O)CC1)ONC(c1c(CC)n[nH]c1)=O N1(C(CCC=C=C)=O)CC(NC(=O)C(CCC)C(C)C)CC(C)(C)C1 CC(C)(C#CC(=O)NCc1nc(C(C)(C)C)ns1)CNC(=O)OC(C)(C)C C1(NC(c2cccc(OCC#C)c2)c2nnnn2C2CC2)CCN(C)C(C)C1 c1(NC(=O)NCCC=C)c(-c2cccc(Cl)c2)noc1-c1ccccc1 N1(C(c2n(CCC)ncc2)=O)CCCC(NC(c2cncc(C(C)(C)C)c2)=O)C1 C1(C(=O)NCC(=O)OCC)CC(C)CCN1C(c1cc(F)n(C)n1)=O C12(CNC(C3N(CC)CCCC3)=O)CCC(CC1)CN2C(=O)C(C#N)C(C)C CC1(C)CCC(C(=O)NC2CC3C(C(N4CCC(F)(CF)C4)=O)C3C2)C1 C#CCCN=C(NCC1(Cl)CCOCC1)N1CC(C(=O)OCC)S(=O)(=O)C(C)C1 C1(CC)CC(C(N2CC3CC2(C(=O)NCC(C)CC2CC2)C3)=O)CCO1 C1(CNC(C2C(CC)CCC2)=O)CC(O)CN1C(=O)CCCc1ccsc1 C1(C(N2CC(CN(C)C(C3CCCS3)=O)OCC2)=O)CC(C)(C)CCO1 CC(C)(CNC(C1(C)CC2CCC1O2)=O)CC(=O)NCc1cnn[nH]1 C12(C(N(C(C=C)C3CC3)C)=O)CC(C)(C1)OC21CCC1 CC1=C(CNC(C2CC(NC(=O)Cc3ccoc3)C(O)C2)=O)COCC1 C1(NC(C2CC3CC3C2)=O)CCCCN(C(c2cc(Br)cnc2O)=O)C1 C1(OCCNC(C(CC)OC)=O)CCCN(C(C2(C(C)(C)C)CCCCC2)=O)C1 N1(C(c2c(C)nc(C3CC3)[nH]2)=O)CCN(C(=O)Cc2occc2C)C(CO)C1 CC1(C)COC(C(=O)NCC(C2CC2)NC(=O)CCN2CCOC2=O)C1 CC1(C)CCN(C(C2CCC3(CCC3)C2)=O)CC1CC(=O)NOCCCO c1(OC)cc2c(cc1C(=O)NCC(C)NC(C1CC1C#N)=O)OCO2 S(=O)(=O)(c1ccc(N2CC3CC2C3)cc1Br)NCC1(c2cccs2)C(C)C1 N1(CC(=O)NC2CC(Cc3ccccc3)=NO2)CC2C(C1)C2(F)F.N12CCC1C2=O C1(C(=O)NCC(CNC(CC2(OC)CCCCC2)=O)O)CNC(=O)C(C)(C)C1 C(=O)(C(C(C)CC)NC(c1cccc(=O)o1)=O)NC(C#C)C(C)(C)C CCC(C#N)C(=O)NCCC(C)NC(=O)CC(C)(C)OC N1(C(C(=O)NCCn2ccc(C#N)n2)=O)CC2COCC(C2)C1 C1(C(=O)NC(c2c(C)nns2)C)CC(C)(C)CCN1C(=O)CC12CCCC1C2 N1(C(=O)C=CSc2nc[nH]n2)CCN(C(c2cnsc2)=O)C(CC(F)(F)F)C1 CCC(C)CC(C(=O)N(C)CC1CCCCCC1)NC(=O)CC1CCCSC1 C1(NC(C2(CSC)CC2)=O)CCOCC1C(=O)NCCc1ncn(C)n1 N1(C(CCCCSC)=O)CCCC2(CCCN2C(c2ccsc2S(N)(=O)=O)=O)C1 N1(C(c2cc(CCC)n(C)n2)=O)CCC2CN(C(C3(CF)CCC3)=O)CCC2C1 c1(C(=O)NCCC(C(=O)OCC)(C)C)cc(F)c(F)cc1OC C1(CC(=O)NC23CCCC2C3)(NC(c2cc(F)ccc2F)=O)CCCCCC1 C(=O)(C1CCc2c[nH]nc21)NCC1CC(CN2C(C)CCCC(C)C2)C1 c1(OCC(=O)OC)ccccc1CNC(C1(CNC2CC3C=CC2C3)CC1)=O c12cc(F)c(c(F)c1)[nH]c2=O.C1(C(C)O)CCCN(Cc2ccn(C)n2)CC1 n1(CC)cnc(C(=O)N(CCc2nccs2)CC2CC2)c1 c1(C(N2CC(C(C(=O)NC(c3ccco3)CO)OC)C2)=O)cncc(F)c1C C(=O)(C1CCCc2ncnn21)NC1C(NC(=O)Cc2csc(-c3ccoc3)n2)C1 C=CC(O)C(=O)N(C)CC1(NC(=O)CN(c2cnccn2)C)CC1 c1(OC(CC)C(=O)NCC2CC(NC(=O)CCc3nccs3)C2)ccccc1F CC1CN(C(=O)C(F)=CC2CC2)CCN1C(c1ccc(-n2nccc2C)cc1)=O C12(C(=O)NCCCN(C(=O)CC3OCCO3)C(C)C)CC3CC(C1)CC(O)(C3)C2 C(C(C)(C(=O)NCC(C)(Cn1cccn1)NC(C1CCCN(C)C1)=O)OC)OC c1(OC)ccccc1-n1ncc(-c2nc(CC(C)OC)nn2C2CCC2)c1C CN1C(=O)CSC1=CC(=O)N1CCC(NC(c2ccnc3cccnc23)=O)C1 C1(CN(C(C2(CCCC)CC2)=O)C)COCCN1C(c1ccoc1COC)=O C1(F)(CNC(C=C(C)C(F)F)=O)CCN(C(C2CC2(F)Cl)=O)CC1 Cc1cncnc1C(=O)NCC1CC(O)(CNC(c2ccccc2C2CC2)=O)C1 CC12CN(C(C3OC4CCC3CC4)=O)CC1C1C=CC2C1 C12CCN(CC1)N(C1CN(C(C3N(CCC)CCC3)=O)C1)C2=O.C(C)(=O)NC C=CC(CCC)CC(=O)N1CCC2(CNC(=O)CC3C=CCC3)CCCC12 N1(C(C(C2CC2)OC)=O)CC2(NC(=O)Cc3csc(Br)c3)CCC1CC2 C1(CN(C(=O)CCSc2ccc(C)cc2)CC)CCCN(C(=O)CS(C)(=O)=O)C1 N1(C(C2(CCCC)CC2)=O)CCN(C)CC1C(N1CCC(CF)C1)=O C1(CC#C)(C(=O)NC(c2nnc(C)o2)C)CCN(C(=O)C=Cc2ccoc2)C1 C1(CC(N2C(CNC(C3CC3C3CC3)=O)CCC(C)C2)=O)CCCC2(CCC2)O1 c1(C(N2CC(C)(C)C(NC(c3ccc(O)cc3)=O)C2)=O)ccc(P(C)(C)=O)cn1 C1(C)(CNC(c2c(C)cno2)=O)CCCN(C(C2(n3cncn3)CC2)=O)C1 C12(CC)CN(C(c3[nH]nnc3C)=O)C(CNC(C3CC3C)=O)(C1)C2 c1(CNC(C2CN(C)C2)=O)ncccc1C(=O)NCC=CBr C(C(=O)NCC(C)(O)CNC(c1ncnn1C(C)C)=O)(C(C)C)OCC CC(C)CC(C(=O)NCCCC1C=NNC1=O)NC(c1cccc(F)c1O)=O C1(NC(C2(F)CC2)=O)CCCN(C(=O)CCOC2CC2)C1 CC1CCn2cc(C(=O)NC3CCN(C(C4(C#N)CCOC4)=O)CC3F)nc2C1 CN1C(=O)CCC1(C)CNC(C1(CO)CCN(C(C2CCCC2C2CC2)=O)C1)=O c1(CN(C)C(=O)NC2CCCN(c3ccccn3)C2)cccc(C(F)(F)F)c1 C(=O)(CCCS(C)(=O)=O)NC1C(CNC(C(C)CSc2ccccc2)=O)CC1 CCC(CC)CC(F)C(=O)NC1CC(CCNC(c2cc(C)oc2CC)=O)C1 c1(NC(=O)NC2CC(C(F)CO)C2)nc(Cl)nc2c1CCOC2 C1(O)(CN(CC=C)C(=O)NCC(=C)Br)CCOCC1 C12(NC(C(CC#C)C3CC3)=O)CCCC1N(C(=O)CC1(O)CC1)CC2 C=CCC(C(=O)N1CC(C(N)=O)(N(C)C)C1)NC(=O)Cc1cn[nH]c1 C(=O)(C1=CCC(C)(C)CC1)N1C(CNC(c2c(C)nsc2C)=O)COCC1 N(C1CCCOc2ccc(Br)cc21)C(=O)NCC1CN(C)CC1C(F)(F)F C1(CC(=O)NC2C3CCN(C(c4ccnnc4)=O)C23)CCS(=O)(=O)CC1 C1(NC(CCCC(N)=O)=O)CC2CC(C1)N(C(=O)OC(C)(C)C)C2 C1(C(=O)NC(C(=O)NC(C(CCC)O)CO)CCOCCO)CCC2(CCC2)O1 C1(CC(=O)NCC(CC)NC(c2cc(O)ccc2N)=O)CCCC(C)(C)O1 c1(C(C)C)ccc(C(N2CC(O)(CNC(c3ccc(-c4ccco4)s3)=O)C2)=O)o1 CN1CCN(C(C2(C)C=CCC2)=O)C(CNC(c2cn3c(n2)SCC3)=O)C1 c1(C(=O)NC2C(C)CN(C(=O)C(C)(C)CC3CC3)C2)c[nH]c2ccc(F)cc12 c1(OCCOC)cc2c(cc1CNC1(C(F)(F)F)CCSCC1)OC(C)C2.C(CO)S c1(OC)ccc(Br)cc1S(=O)(=NC(=O)CNS(C)(=O)=O)C(O)C1CC1(C)C c1(C(N2CCC(NC(COCCCCC)=O)C2CC)=O)ccc2ccsc2c1 C1(C(=O)NCC(CC(C)C)NC(c2cc(O)cnc2Cl)=O)(OC)CCC(C)CC1 C(CN=C(NC(c1cn(C)cn1)CCNC(C)(C)C)NC1CC1C)NC(C(C)C)=O c1(OCC)cc2ccccc2cc1C(=O)NC1CC2(CCC2)CN1C(C)=O c1(C(=O)NC2CC3CN(c4ncnc(=N)[nH]4)CC32)ccc([N+](=O)[O-])c(Cl)c1 C(=O)(CCCCCNC(C)=O)N1CC(CC=C)(OC)C1.C12(CCC1)C(=O)NC2 c1(C(=O)NCCCCN(C)C(c2cnc(O)n2C)=O)ccc(Cl)c(C(F)(F)F)c1 N1(C(COCCCCCC)=O)CCN(C)CC1CNC(=O)CCSCC(C)(C)C N1(C(C2COCC(C)O2)=O)CCCC(C)(C(N2CCC(CC3CCCC3)C2)=O)C1 CCC(C#N)(CC)C(=O)N1CCC(N(CCO)C(C2CC23CCSCC3)=O)C1 C1(C(=O)NC2(CNC(c3nc(OCC)oc3)=O)CCCC2)OC2CCC1C2 C(=O)(C(CC(=O)OC)N)C(=O)CC(C)CNC(C)=O.C(C1CO1)OCC c1(C(N2CC(NC(CCC(=O)OC)=O)C(F)C2)=O)cccc(S(=O)(=O)C(C)C)c1 c1(CN2C(C)C(NC(=O)C=CC3CCCCC3)CCC2)cccc2occc12 C12(CNC(CS(=O)(=O)N(OCC)CC)=O)CC(CC)(CN1C(=O)C(C)(C)O)C2 C1(CC(=O)N(C(C)CNC(=O)CCn2cccn2)C)CCC1C(F)(F)F C(C(F)(C(=O)N1CC2CCC2(C)C1)C(C)C)NC(c1c(C)cc(CC)o1)=O C=C(C)C(C)(C)C(=O)NCCCN(C(c1ccc(OCCOC)nn1)=O)C1CC1 N1(CCSCC)CCN(c2ccccn2)CC1.Cc1nc(C(C(C)C)NC(=O)O)no1 C(C(C(C)(C)C)NC(=O)C(C)(F)c1ccon1)NC(c1c(OC)nsc1)=O C1(C(N(c2ccc(C)s2)CCOC)=O)CCCN(C(=O)CCC(C)C)C1 C1(NC(c2c(COC)ccs2)=O)CC2CCC1N(C(=O)CCS(C)=O)C2 C1(NC(c2c(C(C)C)cco2)=O)C2CCC1N(C(=O)Cc1cnc[nH]1)C2 C1(OCC(=O)NC(C)(C)CCNC(=O)Cc2nc[nH]n2)CCCCCC1 N1(C(c2c(C)ccnn2)=O)CC(F)(F)CC1CNC(=O)CCC(C)C Cc1[nH]nc(Br)c1CNC(=O)C(n1cc(CN2CCNC(=O)C2)nn1)C N1(C(Cn2ncc(C)c2)=O)CCC(C2(NC(c3sc(Cl)cc3Br)=O)CC2)C1 C12CCN(C(=NCCSC(F)F)NC1)C2.C(F)(F)(C(F)(F)F)C1(OCC)CCC1 O=C(CCCCCNC(C1CC1F)=O)NOCC1CCSCC1 c1(C(=O)NC(C(CO)NC(c2c(F)ccc(OC)c2)=O)C)cc2c(s1)CCCC2 C1(OCC)CCCC1NC(c1c[nH]nc1CCNC(=O)CCc1ccncc1)=O c1(OCC)n[nH]c(NC(=O)NCCNC(C2CCC(O)CC2)=O)c1Br C1(C(=O)NC(C)CC2CN(C(=O)CCCC(F)F)C2)CCCc2ccccc2C1 C1(CNC(c2cc(C)nc(C)c2)=O)CCC2CN(C(=O)C#CC3(C)COC3)CC12 c1(C(=O)NC(CNC(=O)C=Cc2ccccc2Cl)CO)c[nH]c2cccnc12 C1(CC(=O)N(CC(C)CNC(=O)CS)C)CCCN1CS.C(C(N)=O)S(C)(=O)=O N#Cc1c(NC2CC23CC(NC(c2cnccc2C(F)(F)F)=O)C3)ncnc1Cl C(=O)(CC(C)(O)C(F)(F)F)N(C)CC1(NC(c2cc(SC)c(N)cc2)=O)CC1 C(=O)(C(C(C)(C)C)C1CCC1)N1CC(N(C(c2cnc(CC(C)C)s2)=O)C)C1 c1(C(N2CC(OCC)C(CNC(c3cc(Cl)no3)=O)C2)=O)c(Cl)ccc(C)c1O N1(C(C(C(CC)C)NC(c2nnccc2C)=O)=O)CCCC(N=[N+]=[N-])C1 N1(Cc2cn(CC)nc2)CC=CC2COCC12 c1(CC)cc(C(=O)NC(C)C(C)NC(c2ncccc2-n2cccn2)=O)sc1C c1(C(N2CCCC(NC(c3sc(C)c(Br)c3)=O)C2)=O)cccc2nncn12 CCC(CCCC(=O)N1CC2CC2(C(=O)OC)C1)NC(C1OCCC1(C)C)=O c1(C(=O)OC)cccc(NC(N2CC(C)CC2c2cccc(F)c2)=O)c1Br N1(CC)CCCC(C(=O)NCC2CCCC2NC(C23COC(COC)(C2)C3)=O)C1 N1(C(c2cnc(Cl)s2)=O)CC2CCCC2(C(=O)NCC2=NOCC2)C1 C1(C(N2CCN(C(C(CCCCC)O)=O)C(C)CC2)=O)CC2(CCOCC2)CO1 c1(COC)cc(=NCCC2CCC(NC(c3csnc3C)=O)C2)[nH]cn1 CC(CC(F)(F)F)C(=O)NCCCOCCNC(=O)C(O)C1CCC1 N1(c2cc(C)ncn2)CCC2CCC(NC(c3cc(Cl)on3)=O)C1C2 C(=O)(CCCC(F)(F)F)NCC(C)(Cn1cccn1)NC(c1occ(C)c1C)=O N1(C(c2cc(CCC)[nH]n2)=O)CC2(COC(CNC(=O)C(C(C)C)OC)C2)C1 Cc1cc(Cl)c(C(=O)NC2COCC2NC(c2ccnc(C(F)F)c2)=O)cc1N C(CN(C)C)(C(=O)N(C)CCn1cncn1)NC(C(C)c1ccco1)=O CC(N=[N+]=[N-])C(=O)NC1CCCCC1C(N1CC(N2CC(O)C2)C1)=O n1(C(C)(C)C)cc(C(=O)NCC(C2CC2)NC(=O)C=CC2CCCC2)c(Br)n1 C(=O)(C1CCCc2nc[nH]c21)N1CC2(CC(CNC(C(C)OCCCC)=O)C2)C1 C(=O)(CS(=O)(=O)CC(=O)NC1CCCCC1N=[N+]=[N-])OC(C)(C)C C=CCC(CC(=O)C1C2CCC(C2)NCC1)NC(c1ccc(CC)[nH]1)=O C1(NC(Cn2ncn(C)c2=O)=O)CC2CC(C1)N(C(C1C=CC=CC=C1)=O)C2 O=C(C#CC1CCCC1)Nc1ccc(CO)nc1.N12CCC(C1)OCC2=O NS(=O)(=O)N1CCC(C(=O)NCC=CCNC(c2coc(C(F)(F)F)n2)=O)CC1 C(=O)(C(C)n1cncn1)NCCCN(C(C1(CC)CC1)=O)C CC1CN(C(=O)C(=O)NCCOc2cccnc2)CCC1C c1(NC(C2C(NCc3ccc(OC)c(O)c3)C2)=O)ccc(CCO)c([N+](=O)[O-])c1 N1(C(c2ncc(C)cn2)=O)CC(O)(C2CCN(C(=O)C(C)CF)CC2)C1 Cc1ccc(C(C)(C)C(N2CCC(C)(NC(=O)CC3CCC(=O)N3C)C2)=O)cc1 c1(C2(O)C(C(=O)C3CC3)C2)ccc(F)cc1.C12(CCC1)C(=O)NC1(CC1)CS2 C1(NC(C)=O)CCN(C(=O)C(Cc2ccoc2)NC(=O)CN2CCNC(=O)C2)CC1 CCC(CC(C)C)C(=O)N1CCC(CCNC(c2ncncc2F)=O)C1 N1(C(CCc2ccc(OC)cc2)=O)CCN(C(=O)CN(C2CCCCC2)C)C2CC12 C(=O)(C1=NN2CCCN=C2N1)NC(C)CN(C)C(C1CCC(C2CC2)C1)=O c1(SC)ccc(C#N)c(Cl)c1.C=C1CC2N(C1)C(=O)c1c(cccn1)NC2=O Cc1cc2cc(NC(C3CCN(C(c4ccncc4Br)=O)CC3O)=O)ccc2[nH]1 C(C(CO)(CO)NC(=O)Cc1nocc1C)N(C(C(COC)NC(C)=O)=O)C C(CO)(C(=O)NCC(F)C1CCC1)NC(CN(C(C(C)C)=O)C)=O N1(C(c2c(C)nn[nH]2)=O)CC2(CCCC2NC(C2CC(=O)N(CC3CC3)C2)=O)C1 C1(CC)CCC(NC(=O)CC(C)N(C(=O)C(C)N2CC(C)C2)C)CC1 C1(CNC(C(CC)n2cccn2)=O)CN(C(=O)CC2CCC(=O)O2)CCC1(C)C c1(C(CNC(C2CC2NC(c2nocc2Br)=O)=O)N)ccc(OC)cc1.CC n1(CC)cc([N+](=O)[O-])c(C(=O)NCC2CN(C(=O)COC(C)=O)CCN2C)n1 C(=O)(CC(C)(C)COC)N1CCC(CCNC(C2CN(CC)C(=O)C2)=O)C1 c1(C(N2CCN(CCNC(c3c(C)nco3)=O)CC2)=O)c(C)cc(Br)cc1F c1(C(N(C(CNC(C(CCC)C#N)=O)C2CC2)C)=O)ccc(O)c2c1CCCC2 S(=O)(=O)(c1cccnc1NC(c1ccc(C)s1)C)N(C(c1cc(C)on1)C)C C1(NC(CCNC(COC)=O)=O)CCCN(C(c2cc(C(F)F)n(C)n2)=O)C1C C1(O)(C(=O)NC2CCN(C(=O)OC)CC2)CCN(C(C2CC23CC3)=O)CC1 c1(C(=O)NCCCCN(C)C(c2cncs2)=O)c(O)nnc2c1CCCC2 C12(N)C3C4C1C1C2C3C41CO.C1(C=O)C2CC1CN(C(C1CCOCC1)=O)C2 C1(C(=O)NCCN(C(CCc2cc(C)no2)=O)C(C)C)CCC2C1C2(F)F C1(N(C)C(C2(F)CCC2)=O)CC2CC1N(C(=O)CC1C=CCC1)C2 c1(-c2cn(CCC3CN(C(C4C(C)CC=CC4)=O)C3)nn2)ccc2ncsc2c1 N1(C(CC2OCCN(C(c3cncc(OC)c3)=O)C2)=O)CC(C)CCC12CC2 c1(NC(C)CCNC(C2CCCC(=O)N2)=O)nc2c(cc1C#N)CCC2 c1(C2(C(N(CCNC(CCc3cnc(C)s3)=O)C3CC3)=O)CC2)cccnc1Cl c1(OC)cccc(CCC(N2CCCC(NC(=O)C(C)(C)C(N)=O)C2C)=O)c1F c1(CNC(C2(C)CCCN2C(c2cc(C#N)c[nH]2)=O)=O)ccc(F)c(Cl)c1 C(=O)(C(C)(CSC)NC(c1cnc(=N)[nH]c1)=O)NCCN(C)CC C(CCC(=O)NCC1CNC(=O)CO1)(C(C)C)NC(C1C(C(=C)C)OCC1)=O c1(C(=O)NCCOCCOC)oc(C(C2CC2)Cc2ccc[nH]2)cc1C c1(OCC)cc2c(cc1NC(=O)NCc1nc(C3CC3)n[nH]1)OC(C)C2 C1(C(=O)NCC(C(C)C)NC(C2(C)CC=CC2)=O)CCOC(C(F)(F)F)C1 c1(OC)ccc(OC)c(C(=O)NNC(=O)C2CCN2CC2CCCO2)c1 N1(C(c2c(C)c[nH]n2)=O)CC(C)(C)OCC1CNC(=O)Cc1ccn(C(C)C)n1 NCS(=O)(=O)c1ccc(C(=O)NC2CCCC(NC(c3nncs3)=O)CC2)cc1 C1(C(=O)NCC(CCC)OC)CCN(C(=O)NCc2ccco2)C1(C)C c1(Nc2ncc(CN(C3CCCNC3)CC)cn2)cccc([N+](=O)[O-])c1[N+](=O)[O-] CC1(C)CC(C(=O)NCC2CC3CC3N2C(=O)CN(C2CCCC2)C)CNC1=O Cc1[nH]c2c(CN(CC(O)CN3CCC(N(C)C)CC3)C)cccc2c1C N1(C(c2c(CCC)occ2)=O)CCC2C(C1)CN2C(c1ccn2ncccc12)=O C1(C(=O)NCC(C)CC(=O)OC(C)(C)C)(C(=O)O)CCC(C(F)F)CC1 CN1CCCC(Nc2ccccc2)C1.C1(C(C)(C)C)COCC(C2CC2)N1 C1(CC(=O)NCCOCC(=O)NC2CC(N(C)C)C2)COCCO1 Cc1cccc2cc(C(=O)NC3CC3NC(=O)C=Cc3ccc(Cl)s3)cnc12 N1(C(c2c(C)c[nH]n2)=O)CCOC2CN(C(C3(C)CC=CCC3)=O)CC12 N1(C(C=CC=CC)=O)CC(NC(c2cccc(SC)c2)=O)CC1CO c1(C(=O)NC2CCN(C(CCN(C(C)C)C)=O)CC2CO)cc(Cl)c(N)cc1F Cc1sc(N)c(C(=O)NC2CCCC(NC(c3cccc(=O)o3)=O)CC2)c1C C(C(=O)NCCCN(C)C(c1cn(CCF)nn1)=O)(C(C)(C)C)SC N1(C(C2C(C)(C)C(F)(F)C2)=O)CC2(C=C(C(=O)NOCCF)CO2)C1 Cc1nc(NCc2ccsc2Cl)cc(N(C)Cc2ccc(C)s2)n1 C1(C(=O)NCC(CN(C)C)O)CC=CCN1C(=O)C=C(C1CC1)C1CC1 C(=O)(C1=CC2(CCOC2)C1)N1CCC(CNC(CC(C)(F)F)=O)C12CC2 Cc1cc(C)nc(-c2cn(C(C)C(=O)NC(c3cccc(C#N)c3)C)nn2)n1 c1(CC(=O)N(CC(N2CCC(OCCO)C2)=O)CCOC)ccccc1C C1(C(=O)NCCCNC(CSCC(=O)NC(C23COCC2C3)=O)=O)CCCCC1 N1(C(C(CC)OCC)=O)CCC(F)(CNC(C2(c3cccs3)CCCCC2)=O)C1 Cn1nnc2cc(C(=O)NC3CCC(C)(CNC(c4cccnn4)=O)C3)cnc12 CC1(C)CN(C(C2C=CCC2)=O)CC(CNC(=O)COc2ccccn2)O1 c1(OC)cc(C(=O)NCCCF)ccc1OCC(F)(F)F.c12nnnn1C2.C1CC1 C(=O)(CCC(=O)C1=CCOCC1)NC1C(CNC(CS(CCC)(=O)=O)=O)CCC1 CCC(CC)C(C)C(=O)NC(C)C=CC(=O)NCC1CCC(F)C1 c1(C(N2CCC(C)(NC(c3c(CC)nn(C)c3)=O)C2)=O)nn(C)c(C)c1Br C(C(C)(C)CNC(C1(F)CCOC1)=O)N(C(=O)C(F)C1CCCC1)CC C1(N(C(=O)CC2CC3CC3C2)CC#C)CCN(C(=O)CCCOC(C)(C)C)CC1 Cc1cccc(C(F)(F)C(N2CC3CC2C3NC(C2CCC(F)C2)=O)=O)c1 C12CC(C)CN(C1)C(=O)N2.C(=O)(CS(=O)(=O)N1CCSCC1)OC c1(C(N(C2CCS(=O)(=O)C2)CC)=O)ccccc1C(N)=O C(CCC)(C(=O)NC(C)(C)CNC(CC1(C(=O)NCC)CC1)=O)=CCC.C1CO1 C1(CNC(c2occ(C)c2)=O)CCN(C(c2c(C)nsc2N)=O)CC1CO c1(CC)conc1C(=O)NCCCN(C)C(C)C.c12cc(cs1)C(=O)NC2 c1(C(=O)NCCCCCCNC(c2cncc(C)c2)=O)ccc(C)c2c1CCC2 C1(NC(C(C)=C(CC)C)=O)CCCC12CN(C(=O)C(c1c(F)cccc1F)C)C2 c1(C(=O)NC(CNC(C(C)SCCCC)=O)C(C)(C)C)cnc2cc(C)nn2c1 c1(SCC(N2C(C)(CNC(C3CCC(=O)C3)=O)CCC2)=O)ccc(C#N)cc1 c1(C(=O)NCC(C(C)C)(C)NC(=O)C(N2CCN(C)CC2)C)ccc(Cl)cc1Cl c1(C(=O)NCC2C3CN(c4nccc(SC)n4)CC32)nccc2ccn(C)c12 c1(N(CCCC(C)(C)C)c2n(CCCCCC)nnn2)ccnc(OC(F)F)c1Cl N1(CC#C)CCC(C(=O)NC(C2CCCC2)CNC(c2nc(Cl)c(Cl)s2)=O)CC1 c1(C(N2CC3CN(c4c(C)cncn4)C3C2)=O)cc2cn[nH]c2cn1 c1(OC)n[nH]c(C(N2CCCC2c2ncon2)=O)c1Cl N1(C(=O)NC(C)C2CC2)CC(CO)C(C2CCOCC2)C1 c1(CC(=O)NC(C2CC(F)(F)C2)CC#C)ccc(Br)c(Cl)c1 N1(C(=O)O)CC(CC(c2csc(-c3ccccc3)c2)=O)OCC12CC2 c1(C(N2CC(NC(C(COC)C)=O)CC(C)(C)C2)=O)ccc2c(O)ncnc2c1 CC(C)C(CC(=O)N1CCN(C)C(CO)C1)NC(c1cc(F)ccc1F)=O N1(C(C)=O)CCC(N=c2nc3c(ncn3C)c(NCCCCCO)[nH]2)C1 Cc1cnc(NC(CO)CCO)c(S(=O)(=O)N2CCC(CCCO)C2)c1 N1(C(C(COC(C)=O)N)=O)CCOCC(CN(C)C)C1 N1(C(=O)Nc2ccccc2C(F)(F)F)CCC(C(N2CCNCC2)=O)CC1 c1(C(=O)OCC2OCCCO2)cccc(N2CCC2)c1 C1(C)(CC)CCCN1Cc1cccc(-c2nnn(C)n2)c1 c1(C(C)NC(c2cnc(-c3ccccc3)s2)=O)cccc(OCC2CCCOC2)c1 C(C(COC)C(=O)NC(Cc1cc[nH]n1)C(=O)N1CCCC1C1CC1)OC C#CC(CNC(C1(F)CCN(C(c2cnnc(C)c2)=O)CC1)=O)CC(C)(C)C n1(CC(=O)NC2(CN(C(=O)COC3CCCC3)C)CCC2)ncccc1=O c1(NC(C2CC23CCN(Cc2cn(C)nc2)C3)=O)c2c(nn1C)CCC2 c1(C(=O)NCC2C(C)CN(C(C3COC(C)(C)C3)=O)C2)ccc(O)c(C(C)C)c1 c1(C(=O)NCC=CC(=O)NCCC(CCC)C2CC2)cc2cc[nH]c2cn1 C(CNC(C1C(C)CCN1C(c1cccc(C)n1)=O)=O)(CC(C)C)OC C1(N(C(Cc2c(C)cccc2)=O)C(c2ccncc2)C)CCC2(CC1)CNC2 C(=O)(N=c1ccc(C2CCOCC2)n[nH]1)N(C(c1ccncc1Cl)C)C1CC1 C1(C(N(CCCNC(COC(CC)(C)C)=O)C)=O)CCN(C2CC2)C1 c1(N2CC(C)(O)C2)ccc(NC(=N)NC2(S(C)(=O)=O)CC2)cc1 N1(C(CCCNC(=O)C2CC2)=O)CCN(C(C2C3C4CCC(C4)C23)=O)C(CO)C1 c1(SCC(=O)NCC(C(C)C)NC(C2CN(C(N)=O)C2)=O)c(F)cccc1Cl C1(CC(=O)NCCC(C)NC(C(C)(C)OCCC)=O)CCC2(CC1)CC2 c1(OCC(CN(CCOC)CCN(C)C)O)cccc(Cl)c1 C(=O)(C1=CC2(CCOC2)C1)NCC(CCCC)NC(C1(C2CCCO2)CCC1)=O c1(NC)nc(C(N2C3CCC2CN(C(c2ccc(Cl)o2)=O)C3)=O)ccc1[N+](=O)[O-] c1(OC)cc(C(N2CC(NC(=O)C=CC(C)(C)C)C(O)C2)=O)c(O)c(Cl)c1 c1(Cc2onc(-c3c(OCC)cc(Cl)cc3)n2)c(Br)sc2ccccc12 N1(c2nc(C)nc(N3CC4CCC(C3)O4)c2)C2CCC1CC(CC)C2 C1(C(=O)NCc2cccs2)COCCC12CN(S(=O)(=O)c1cccc(Cl)c1)C2 c1(CC(=O)N(C2CCNCC2)CC#C)sccc1Br C1(C)(c2c(C(=O)OC(c3cncc(F)c3)CC)cccc2)NC(=O)NC1=O N1(C(c2ccc(C(C)=O)cc2)=O)CCN(C)C(CNC(=O)C(C)c2ncco2)C1 N1(C(=O)CC2COC(=O)C2)CC(C)(C(O)C(=O)NCCN(CCCO)C)C1 N1(C(C(C(C)C)OC)=O)CCC2(C)CN(C(=O)CC3(C)OCCO3)CC12 c1(OC)ccc2oc(C(N3CC(NC(C4C(C)C4C)=O)CC(F)C3)=O)cc2c1 CC1CN(C(=O)CC(CNC(C2CCC(C)(C)OC2)=O)C2CCC2)CC(=O)N1 Cc1cn2c(n1)C(C(=O)N(CCCCNC(=O)CC1(O)CCCOC1)C)CCC2 c1(N2CC3CC(NC(c4cc(CCC)[nH]n4)=O)C3C2)cc(C)c(C#N)cn1 N1(C(C(C)=CC)=O)CCN(C(C2CCC(=O)N(CC(F)(F)F)C2)=O)C(CCC)C1 c1(C(=O)NCC2N(C(C(COCC)(C)C)=O)CCOC2)cc2cccnc2[nH]1 c1(C(=O)NC2CN(C(Cc3cnc(C)s3)=O)CC(C)C2)cnc2ncccc2c1 c1(C(=O)NCC(C)(O)Cn2cccn2)nc2nc(O)c3ccccc3n2n1 c1(C(N2CC(C(=O)OC)C23CCOCC3)=O)nc2ccccc2nc1O N1(C(CCCC=C)=O)CCN(C(C2COCCO2)=O)C(Cc2ccc(F)cc2)C1 C1(C(=O)NC(CCNC(CCc2cc(C)n(C)n2)=O)C)CCc2c(nnn2C)C1 CCCCS(=O)(=O)CC(=O)NC12CCCC(NC(c3ccns3)=O)(C1)C2 C1(F)(N(C(=O)NC(C)CCC2CCCO2)CC2CC2)CCCC1 Cc1nc(C)c(CNC(=O)CC2COCCN2C(c2cnn(-c3nccs3)c2)=O)[nH]1 c1(N2C(CCNC(C3ON=C(CCC)C3)=O)CCCC2)ncc(C#N)cc1F c1(OC)ccc(NC(C2CC(O)CN2Cc2ccnc(Cl)c2Br)=O)cc1[N+](=O)[O-] CCC(O)C(C)(C)C(=O)NCC1C=CC(NC(=O)CC2C=CCCC2)C1 C12(NC(=O)Cn3ncnn3)CC3CC(C1)CC(NC(c1csnn1)=O)(C3)C2 C1(C(=O)NCc2c(C)nn(C)c2)CCN(C(C2CCCC(C#N)C2)=O)CC1(C)C C1(NC(CC)=O)CN(C(c2ccc(-c3sccc3C)s2)=O)C2(CCCOC2)C1 C1(CC(=O)NCC(CSC)OC)CC(O)CN1C(=O)C=Cc1ccsc1 Cc1cc(NC(C2CCCN(Cc3n[nH]c(C)c3C)C2)=O)n(-c2ccccc2)n1 C1(C(=O)NCCCN(C(C2(C=C)CCC2)=O)C)CNC(=O)CC1C N1(C(C(COC)NC(C)=O)=O)C2CC1CN(C(c1cc(O)nn1C)=O)C2 CCC(F)(F)CC(=O)N1CCC(C)(NC(=O)C(c2cc(F)cc(F)c2)(F)F)C1 Cc1cnc(C(=O)NCCCCCCNC(C2(CC(F)F)CC2)=O)c(O)c1 C(c1ccc(F)cc1)=CC(=O)NC(CN(C(C(C=C)O)=O)C)(C)C c1(CC)oc(C)cc1C(=O)NCC(C)(F)CNC(c1nc(O)c(C)s1)=O Cc1nc(C(N2CCSCC2CCNC(=O)C(N2CCCCC2)C)=O)c(C)s1 c1(C(N2CCN(CC3CN(C(c4nc(Cl)oc4Cl)=O)C3)CC2)=O)ccc(O)nn1 c1(C(=O)NCCC2CCCN(C(C=Cc3cn(C)nn3)=O)C2)ccc(Cl)cc1Cl C1(CNC(Cc2cn(CC)nc2)=O)CN(C(=O)CC2COCC2O)CC(C)(C)C1 C1(NC(=O)CSCc2cscn2)CCCCN(C(=O)CCc2cnc[nH]2)C1 N1(C(c2c(C)ccnc2)=O)CC2(C1)CN(C(C1(C)CC1Br)=O)CC2CO N1(C(C2CCN(C(C)=O)C2)=O)CC2(C(N3CCSCC(C)C3)=O)CC1CO2 C1(C(=O)OC)CCN(C(=NCC=CBr)NCc2nnc(CO)s2)C1 Cc1ncnc(Cl)c1NC(=O)CC1CCCN(Cc2cccc(Br)n2)C1 c1(NC(C2C(NCc3ncc(C)cc3F)C2)=O)n[nH]c2c(Cl)cccc12 c1(C(=O)NC(c2ccncc2)CC)cccnc1CNC(c1coc(C)c1)=O C1(O)(CN(C)CCNC(c2ncc[nH]2)=O)CCCN(C(=O)CNC(=O)C2CC2)C1 c1(C(N(CC(C)NC(c2c(C)cns2)=O)C)=O)nccnc1N C(c1ccoc1)=CC(=O)NCCN(CCC)C(C1CC1OCC)=O Cc1oc(C(F)(F)F)nc1C(=O)NCC1CC1NC(=O)CC1C=NN(C)C1=O N1(C(c2cccc(C(C)C)c2O)=O)CCC2(CCN(S(=O)(=O)CCCCl)C2)C1 C1(C(N2CC3CN(C(CCCCc4ccccn4)=O)CC23)=O)CN2CCC1CC2 c1(N2CC(N(CC(=O)NC)C)C2)ncnc2ccc(OC)nc12 Cc1cc(C(=O)NC2CCC(C)(CNC(=O)CC3C=CCCC3)CC2)ccc1Cl Cc1cnc(C(=O)N(C)CCN(C)C(c2csc(-c3ccccc3)n2)=O)cc1Cl C(=O)(CC(C)C(F)F)N1CCC(CONCC(=O)OC)CC1 c1(C(=O)O)cc(S(=O)(=O)Nc2cc(Cl)c(CO)cc2N)cc(Cl)c1F CCCC(CC)C(=O)N1CC(O)CC1CNC(c1sc(Cl)cc1Cl)=O C1(NC(c2ccccc2)=O)CCN(C(C(CF)C(F)(F)F)=O)CC1 C(=O)(CCCCC(N)=O)NC(CC)CN(C(=O)C=CC(c1ccccc1)=O)C C12(C(=O)NC(CN(C(CCOCC)=O)C)Cc3ccccc3)CC(F)C1C2 CCCCCC(O)C(=O)NCCC1(NC(=O)CC2CCCO2)CCC1 c1(OC)ccc(CCC(C(=O)NCC(C)C)N2CCOC(CC(N)=O)C2)cc1 c1(C(=O)NCC2C(CNC(C(C)S(N)(=O)=O)=O)C2)cnc2c(c1)CCCO2 n1(CC(=O)N(C2C(C)CCN(C(CCOC)=O)C2)C)ccc(=O)n(C)c1=O C(CCC(=O)NNC(=O)C(C)(C)CCCCNC(=O)C#CC1CCC1)OCCOC N1(C(C(C)c2cccs2)=O)CCCCC1CCNC(=O)CNC(=O)CN(C)C N12CCC(CC1)OCC2=O.C(=O)(C(C)(CO)N(C)C)NCN(C(CNC(C)=O)=O)C CC1CCCN(C(=O)CC2CC2C2CC2)C1CNC(=O)C1=C(Cl)CCC1 c1(C(=O)NCCC(C)F)conc1CNC(c1ccco1)=O Cc1ccc([N+](=O)[O-])c(C(N2CC(NC(C3(O)CC3(C)C)=O)C(O)C2)=O)c1 c1(C(=O)NC(CN(C(c2nc(C(C)C)sc2)=O)C)C)cc2ccccn2n1 C1(NC(c2c(C)cc(CC)o2)=O)CC2CC(NC(c3ccc(F)s3)=O)CC12 C(=O)(C(C)C(C)S(C)(=O)=O)NC(C1(O)CCN(C(c2ncc(Cl)s2)=O)CC1)C c1(C(=O)OCC)sc2nc(COC)nc(N3CCC(C)C(C)(C(=O)O)C3)c2c1C C=CC(O)C(C)(C)C(=O)N1CCOC(CC(=O)NCc2cc(F)ccc2Cl)C1 C1(C(=O)NCC(C2CC2)SC)CC2(CC2)CN1C(=O)CC(=O)N(C)C N1(C(C(CCC=C)NC(=O)COC(C)(C)CC)=O)CCC2(CCCC2)CC1 C1(N(C(=O)CC2(C)CC2)C)CN(C(c2ccccc2OCC(F)(F)F)=O)CC1F C1(OC)CN(C(=O)CNC(c2ccccn2)=O)CC1NC(=O)CC1(O)CCOC1 c1(OC)nc(C(=O)NCC2(F)CC(NC(=O)CN3C(=O)CCC3=O)C2)ncc1F c1(N(CC(CC)C)C)[nH]c(=NCC(C(C)(C)C)OCCO)nc2scnc12 Cn1nc(C(=O)NCCCC2CN(C(c3ccc[nH]3)=O)CCO2)cc1C(N)=O C1(C)(C(=O)NC)CC(OC)CN1C.N12CCOC(C1)C2=O.C1(CCC)CCCC1OC N1(C(CCOCC#C)=O)CC(C(=O)NCC2CCCC2(C)C)C(C)C1 c1(OC)cc(C(=O)NCCC2CCC(NC(=O)Cc3cccs3)C2)cc(Cl)c1O N1(C(c2cccc(CC)c2C)=O)CC(NC(=O)C=Cc2nccs2)CC(F)(F)C1 n1(CC)cnc2[nH]c(=NCc3csc(Cl)c3)[nH]c(=NC(C)C(C)C)c12 CC1CCCC(CC(N2CCC(C)(NC(C3(CC4CC4)CCCC3)=O)C2)=O)C1 C12(CCNC(C=CC=CCC)=O)CCC1CN(C(c1cccnc1NC)=O)C2 Cc1[nH]cc(C(=O)NCCCc2ccc3n[nH]cc3c2)c(=O)c1Br c1(C(=O)NC(C2CCCN(C(c3cc[nH]n3)=O)C2)C)cccc2c1COCCN2 CC1CN(C(=O)CN(C)C2CC2)CC(C)N(C(c2ccc3c(c2)CC(=O)N3)=O)C1 C1(NCn2cc(C(N3CCN(CC)CC3)=O)nn2)(CO)COCCN1C N1(C(=O)NCCS(CC)=O)CC(n2ccnn2)C(O)C1 C1(CC=C)CCCN(C(=O)C(C)(C2CC2)N(C(=O)CN(C)CCC)C)C1 N1(C(C=CCCC(C)C)=O)CCC2(CCCN(C(=O)COCC3CCC3)C2)C1 n1(CC(N2C(CNC(=O)C(=O)NC3CC3)CC(OC)C2)=O)ccc(=O)n(C)c1=O c1(OC)cc(CC(=O)NCC(O)CCNC(C2OCCO2)=O)cc(Cl)c1 c1(C(N2CCn3c(C)cnc3C2)=O)ccnc2cc(Cl)ccc12 Cc1cc(C(=O)NC(C)(C)CN(C(=O)CC(C)c2ccccc2)C)nn1C N1(C(c2ccc3cnsc3c2)=O)CCC(C2CN(C(C3COC3)=O)C2)CC1 Nc1cc(F)c(F)cc1C(N1C2CCC(C2)C1CNC(=O)COC(F)(F)F)=O N1(C(CCSCC(N)=O)=O)CCC2CCN(C(c3nnc(O)nc3O)=O)C2C1 C(=O)(CN1C(=O)CCc2ccccc21)NCC(CNC(CC1(OC)COC1)=O)F C#Cc1ccc(CNC(=O)CC(=O)NCc2cccc(OC)c2OC)cn1 c1(CC)ccoc1C(=O)N(CC(N1CC(Cl)(Cl)C1)=O)C(C)C C1(OC)CC2CC(C(=O)N(C3CC(NC(C4(C)CCN(C)C4)=O)C3)C)CC12 Cc1ccc(C(=O)NCC2CN(C(=O)C(F)C3CCC3)CC23CC3)c(N)c1 N1(C(C=C(C)C(F)F)=O)CCC(NC(C2CC3CC2C2CC32)=O)CC(O)C1 C(CCC(C(=O)NCCN=[N+]=[N-])NC(c1cc(F)ccc1O)=O)OC C(C1=CCCCC1)NC(=O)C(C1CCN(C(C2CCN(C3CC3)C2)=O)C1)F C#CC1(O)CCCN(CC2CN(C(=O)COCCOCCO)C(C)(C)C2)C1 N1(C(C(CC=C)C)=O)CCN(C(=O)C=Cc2cccs2)C2CCC12 c1(-n2cc(C(CC)(C)O)nn2)cccc(CNC(c2ccc(Cl)s2)=O)c1 C(CN=c1[nH]cnc2ccc(O)cc12)(N(C(C(c1ccccc1)OC)=O)C)C1CC1 c1(C(=O)NCCNS(CC)(=O)=O)n[nH]c(C)c1[N+](=O)[O-].c12cn(nn1)CC(C)S2 C(=O)(C(O)C(C)(C)C)N(CCOCCN(C(=O)C(c1ccccc1)O)C)C C1(CNC(c2ccn(CCN(C)C)n2)=O)C2CN(CC(O)CC3CCCO3)CC12 C1(NC(c2cc(C)n(C)c2)=O)CCN(C(=O)CCc2cnn(C)n2)CC1CO N1(C(c2cnc(C(C)C)[nH]2)=O)CC(NC(c2cnncc2C(F)(F)F)=O)C(O)C1 Cn1cnc(NCCC2CCC(NC(C3CC3C3CCCCC3)=O)C2)c(Br)c1=O C1(C(=O)NCC2(CN=c3[nH]nc(CCOC)s3)CCCC2)CCCC2(CCC2)C1 CC1(C)CNC(=O)c2cc(NC(=O)C(c3cccc(Br)c3)O)ccc2O1 C1(CNC(c2nc(Cl)c(Cl)s2)=O)CC12CCN(C(c1cnsn1)=O)CC2 c1(OCC)c(C(=O)N(CC(C)Nc2cnc(C#N)cn2)C)nc(O)nc1O C1(NC(Cc2cc(C)no2)=O)CCCC1(C)CNC(=O)C(c1ccccc1Cl)C c1(CNC(C(C2CCC2)NC(COCC)=O)=O)ccc(CO)o1 C(=O)(C1=CCC(NC(c2csc(=N)[nH]2)=O)C1)NCC(CC(=O)NC)C N1(C(C2(CC)CCCC2O)=O)CC2CN(C(C3CCC=CCCC3)=O)CC(C1)O2 C1(OC)CN(C(C2(C)CCCS2)=O)CCC1NC(=O)CCC1CCCCC1 N1(C(COc2cccc(C)c2)=O)CCCCC(NC(C2CCN2S(C)(=O)=O)=O)C1 N1(C(C2CC(C)(O)C2)=O)CC2CC(C1)N(C(=O)CCC1CC1CC1CC1)C2 CC1CN2CCN1CC2C(=O)N(CCCNC(C12CCC(CC1)OC2)=O)C1CC1 N1(C(c2cc3sccc3[nH]2)=O)CC2CCN(C(c3cnc(Cl)s3)=O)CC2C1 c1(OCC(Cc2cn(CC(CCC(=O)OC(CC)C)F)nn2)O)ccccc1C C1(C(=O)NCC(C)(Cn2cccn2)NC(CN(CC(C)(C)C)C)=O)CCS(=O)(=O)N1 c1(OCCC)cccnc1C(=O)NCCNC(=O)C(C)NC(=O)C(C)(C)C C#Cc1cccc(NCC(=O)NC2CC3CC2N(C(C2CCCN2CC)=O)C3)c1 C(=O)(CC(O)(C(F)(F)F)c1ncco1)NCC=CCNC(c1c(C)cncc1)=O C(=O)(C1COc2ccccc21)N1CC2C(CNC(c3n(C)nnc3)=O)C2C1 N1(C(C2CCC(=C)CC2)=O)CC=C(CC(=O)NC2CSC2)CC1 c1(-c2nnc(NC(N3CCC(CO)(CO)C3)=O)o2)ccc(F)cc1Cl CC(C)CC(C)(C)C(=O)NCCn1cnc(C(N2CCOCCC2C2CC2)=O)c1 c1(CN(CC)CC)ccc(C(C)(F)F)cc1.C12CC(c3nnnn3C(C)CC)(C1)N2 N1(C(C2C(CC)OCC2)=O)CC2=C(C1)CN(C(c1cccc(F)c1F)=O)C2 C(=O)(C1=COc2ccccc2O1)NCCC(C)(C)NC(=O)C=CC(=O)NC1CC1 c1(C(=O)NC2CC(CNC(C(CSC)(C)C)=O)OCC2)cnc2n1CCCCC2 O=C1NCCOC2CN(C(=O)CN3CCc4ccccc4C3=O)CC12 Cc1ccc(C(=O)NC2CC(O)CN(C(=O)CCc3ccc(O)cc3)C2)cc1C c1(NC(c2cscn2)CC)cc(Cl)cc(Br)c1I C1(N(CC(C)C)C(c2cc(C)oc2)=O)CCN(C(=O)CC2CCC=CCC2)CC1 c1(OCC)nc(Cl)ccc1C(N1CCCC(F)(C(=O)NCC23CCCC2C3)C1)=O c1(CNC(CC2N(C(C3(SC)CCC3)=O)CC2)=O)ncccc1O N1(C(C(n2cc(Cl)cn2)C)=O)CCC(C2CCCCN2CCn2cc[n+](C)c2)CC1 Cc1csc2cc(C(=O)NC3CC3CNC(=O)C(N)=O)[nH]c12 C(=O)(C(CCC(N)=O)NC(=O)CCCN(C(C)C)C(C)C)N1C(CC)CC(C)C1 c1(NC(C(=O)Nc2cccc(-c3ccncc3)c2)=O)ccc2c(c1)CCNCC2 N1(C(CC2ON=C(C)C2)=O)CCN(C(C2(CN(C)C)CC2)=O)CC1 N1(C(COCCC=C)=O)CC2CN(C(c3cnc(OC)c(Cl)c3)=O)CC2(C)C1 C(=O)(CC(C)C(C)(C)NC(c1sc(C)cc1C)=O)NC1CC(C#C)C1 C=CC1(O)CC(C(=O)NC(C(=O)NCCc2cccs2)C(C)OC)C1 Cc1ccc(C(=O)NCC2(NC(C3CCCC(=O)N3)=O)CCCCC2)nn1 c1(C(=O)NCCCN(C(=O)C(C)C2CCC2)CC)cc2ccncc2s1 N1(C(c2cc(C)c(C)s2)C(=O)NCCOC)CCCc2ccc(C)cc21 Cc1ncc(CC(=O)NC2CC(CCNC(c3coc(C4CCC4)n3)=O)C2)o1 C1(C(N2CC(N(CC=C)C)C2)=O)CCCN1C(=O)CNC(=O)C1CC1 Cc1noc(C2CC2)c1C(=O)NCC1(C)CCCN1C(=O)CC1(C)CCCCC1 c1(N2CC(c3sc(C)c(CC(=O)N(C)C)n3)C2)sccc1S(=O)(=O)N(C)C N1(C(N2CC3C(N(CCO)CC)C3C2)=O)CCC(C(C)CO)CC1 N(C(=NCc1ccc(N2CC=CC2)cc1)N1CCC(F)C1)C(CC)C C1(C(=O)NCC2(C)CCCN2C(c2cnc3sccn23)=O)NC(=O)C2CCC12 N1(C(C(c2cnccn2)C)=O)CC=CC1CNC(c1n[nH]cc1C1CC1)=O c1(C(N2CCC(N(C(C3CC4CC4CC3C)=O)CC)C2)=O)ccnc2ccsc12 CC1CCCn2cc(C(N3CC(O)(CNC(=O)C(c4ccccc4)O)C3)=O)nc21 C1(C2(NC(N3C(c4nc(OC)c(C)s4)CCC3)=O)CC2)CCC2(CC1)CC2(F)F CC(C)(CS(C)(=O)=O)C(=O)NC1COCCN(C(C2CCCS2)=O)C1 C1(NC(c2c(OC)ccs2)=O)CCCCN(C(c2cc3ccccc3[nH]2)=O)CC1 CC1CCC(C(N2CCN(C(=O)CCF)CC2)=O)CN1C(=O)Cc1ccnn1C Cc1ccc(-n2nnnc2N2CCC(CC(=O)NC(C)COC(C)C)C2)cc1 Cc1noc2cc(C(N3CC4CC(NC(=O)CC(C)(F)F)CC4C3)=O)ccc12 C1(C)CN(C(=O)COc2cccc(O)c2)CC1(F)F.NC(=O)N(CCN)CC1CC1 c1(C(=O)NC2C(C)N(Cc3ccccc3)CCC2)cnc2cnccc2c1 c1(C(=O)NC23CCCC(NC(C4CC45CC5)=O)(C2)C3)cccc(O)c1[N+](=O)[O-] N1(C(C(C)C2CCCC2)C(=O)NCCC#N)CC(C)C(C2CCC2)C1 N1(C(CCOCC(C)C)=O)CCC(CF)(NC(C2CCC(=O)NC2)=O)C1 c1(C(N(C)CC2(NC(C=C(CC)C)=O)CC2)=O)nccc(Cl)c1C N1(CCNC(=O)NCc2cc(Br)ccn2)CC2C3C=CC(CC3)C2C1 C(=O)(CCCCC(F)F)NCC1(C)CCCN1C(c1n[nH]c2c1CC1CC21)=O C(=O)(C1=COCCO1)N1C(CNC(c2ccc(CN3CCOCC3)o2)=O)C=CC1 C(c1ccc(=N)[nH]c1C)=CC(N1C(CNC(CCOCCOC)=O)CC1)=O C(=O)(C1=CNC2=NCCCC2=C1)N(C1CCCCCC1)CCNC(C(CC)C)=O C1(C(N(C(C)CC(N)=O)C)=O)CC2CCC(C1)N2C(C1CC1C1CC1)=O C(=O)(C1=CCCCC1)N1C(C(C)NC(c2csc(O)n2)=O)CCCC1 N1(C(N2CCCC2CO)=O)CCC(C(=O)NC2CC(n3cncn3)C2)CC1(C)C c1(CNC(C(=O)NC(C2CC(C)C2)C)=O)cccc(C(F)F)n1 C(CN=c1[nH]c(N2CCC(P(C)(C)=O)C2)nc2c1CCCC2)Sc1c(C)nc[nH]1 C1(N(CCNC(C(CC)CCOC)=O)C2CC2)CCCCN(C)C1=O C1(C)(CNC(CC2(C)CCOC2)=O)CCCN(C(=O)Cc2ncc(Cl)s2)C1 N1(C(=O)CC2(O)CCOC2)CCCCC(NC(C2(C3CC3)CC=CC2)=O)C1 CC1(C)C2CCC1(C(=O)NC1CCC(NC(C34CC5CC3C4C5O)=O)CC1)C2 CC1=C(F)CN(c2nccc(C3CC4CCCC4C3)n2)CC1 C1(CCCC)CN(C(=O)CC(C)(C)OC)CCN1C(c1ccnc(SC)c1)=O C1(N(C(C(F)OC)=O)CCO)CCN(C(c2cc(C3CCC3)[nH]n2)=O)C1 Cn1cnc(CCNC(C(CCCO)c2ccccc2)=O)c1 C1(NC(Cc2c(C)ccs2)=O)CCN(C(C2CC3CCC2CC3)=O)CC(C)(C)C1 Cn1cccc1C(=O)C(=O)NC1CC(CNC(c2ccnn2C2CC2(F)F)=O)C1 CON(CCO)C(=O)c1coc(CNC(c2c(O)cccc2F)=O)c1 C(=O)(CC(C)C(=O)NCC1CC1CC(=O)Nc1cnn(C(C)C)c1)OC N1(C(C(C)NC(COC)=O)=O)CC2(CCC2)CC1C(=O)NC1CC2CCC(C1)N2C c1(CN(C)C(c2ccc(C(N)=O)o2)=O)cccc(C(=O)NC2CCCCCC2)n1 CC(C)(C)CN=C(NCC1(O)CCOC1)NCC(C)(O)c1ccsc1 c1(C(N2C(C)C(NC(=O)CCC3CCC3)CCC2)=O)ccnc2ccnn12 C(=O)(C(C)(C(C)C)OC)N(CC(C(=O)NC1CC(CC)OCC1)(C)C)C CCC(C)(C)CCCC(=O)N1C(CC(=O)NC(C(C)C)C(C)C)C2CCCC12 C1(C(N2CCCC(OC)C2)=O)CC2(CCN1C(=O)C(CC1CCC1)OC)CC2 Nc1cc(F)c(CC(=O)NC(CNC(=O)CCC2CC2CC2CC2)CO)cc1F c1(C(=O)NCCCC(CCC)NC(=O)C=C2CCCC2)cncc2ncccc12 C1(N(C(C(C2CC(F)(F)C2)OCC)=O)C)CCCN(C(=O)Cc2cccnc2)C1 c1(C(N(C2CCN(C(=O)CN3C(=O)CNC3=O)CC2)CC)=O)ncc(F)cc1F C1(C(c2n(CCC)nnn2)NC2CC(OC)C2)CCC(S(C)(=O)=O)CC1 C(CCOCCO)(C(=O)NCc1occc1C)NC(CC1CC(=C)C1)=O C1(NC(CC(C=C)CC)=O)CN(C(c2cc(CC)[nH]n2)=O)CCC12CCC2 C1(CNC(C(C2CCC2)OC)=O)CN(C(c2cnc(O)o2)=O)CC1n1ccnn1 CCC(O)C(C)C(=O)NCC1CCC(CN(C)C(c2snnc2C)=O)CC1 C=CCC(CNC(c1sccc1F)=O)NC(=O)C(F)(F)C1(O)CCC1 Cc1cc(Cl)cc(NC(C2CC23CCN(C(c2cncc(Cl)c2Cl)=O)C3)=O)c1I N1(C(C2CN(C(CC(C)OC)=O)CC2F)=O)CCC(C)CC(C)C1 CC1(C)CC(NC(=O)Cc2cn[nH]c2)CN(c2ncc(Cl)cn2)C1 c1(C(=O)NCC23CC2CN(C(=O)Cn2cccc2)C3)cncc2nc(O)[nH]c12 n1(CC(=O)OC)nccc1C(N1CCC(N(C)C(C2CCCC2OC)=O)C1)=O C(=O)(C1=CC2CCCCCC12)N1CC2CCC(NC(=O)CCCCF)CC2C1 C(=O)(C(C)(O)C(C)C)NCCNC(Cc1cn(CC)nn1)=O.C12CCCN(C1)C2=O c1(C(N(C(CCNC(Cc2cn(CC)nc2)=O)C)C)=O)ccncc1CC c1(NC(C(C)OC(=O)C(Cc2ccccc2)N(C)C)=O)cccc(Cl)c1 C(=O)(C1=C(Cl)CCC1)NCCCC(=O)N(CCC1N(C(=O)OC(C)C)CCC1)C N1(C(C(CC)n2cncn2)=O)CCN(C(c2cccc(SO)c2)=O)C(CO)C1 c1(C(N(CCCN(C(C(CCCC#C)C)=O)C)C)=O)ccc2ncc(Br)n2c1 c1(C(=O)NC(C(N2CCC23CC(O)C3)=O)C2CCC2)cnc2n1CCC2 Cc1ccc(OCC(=O)NCC2(C)CN(C(=O)CCS(C)=O)CC2C)cc1C c1(C2c3n(nnn3)CCN2)cccc(C(=O)OC)c1F.C1(C)(OCC=C)CCC1 N1(C(C2CN(CC(C)C)C2)=O)CCCC(CN(C(=O)CCN)C)C1.S(C)(=O)(=O)C1CC1 C(=O)(C1=C(C#N)CCC1)N1CCN(CCCNC(C(C)C2(O)CCC2)=O)CC1 CC(c1ccccc1F)=CC(=O)NC(C)(C)C(C)NC(c1c[nH]nc1F)=O c1(C(N2CC(NC(=O)CN3CSCC3=O)C(F)C2)=O)oc2ccccc2c1Cl C12(NC(c3c(CC)c[nH]c3)=O)CCCC1N(C(=O)COCC1CCCOC1)CC2 c1(C(=O)NC2(CNC(C(C)CC3CCC3)=O)CCC2)c[nH]c2cccc(C#N)c12 C1(C(=O)NCC(C)(F)F)CC12CCN(C(=O)C=Cc1cc[nH]c1)C2 c1(C(N(CC(C)N(C(C(CCC)OC)=O)C)C)=O)cccc(C2=CCOCC2)c1 Cc1cn2nc(C(=O)NCC(O)CNC(c3c(C)cccc3O)=O)cc2c(=O)[nH]1 C1(C(=O)NCC(CCC)(C)C)CC(C)(C)CCN1C(c1ccc(F)cc1F)=O c1(C(N2CCC(N(C(c3ccc(O)nc3Cl)=O)CC)C2)=O)ccnc2ncnn12 Cn1ncnc1CCC(=O)N1CCC1CNC(c1cn(C)nn1)=O.C1(N)CCCCC1 C1(C)(CNC(CC2(SC)CC2)=O)CCCN1C(C1CC1c1ccc(C)o1)=O CCC(C)(CC)C(=O)NCC1CC1CC(=O)Nc1cnc(Cl)nc1C c1(SCCC(=O)NC2(CNC(CC)=O)CCOC2)ccc(F)c(F)c1 N(C(=NCCc1ccn(CC)n1)N1CCC(c2ccccc2Br)C1)C(CC)C c1(C(=O)NCCC2COCCN2C(C2CCCCO2)=O)c[nH]nc1[N+](=O)[O-] c1(Nc2cn(CC)nc2C)cc(F)c(C(=O)O)cc1C C=CCCCCC(=O)N1CC(C(=O)NCCC(C)c2cn[nH]c2)CCC1C CCCCCCn1nnnc1C(CC1CCCS1)NC1(n2ccnn2)CC1 Cc1nc(C(=O)NCC(C)(CO)NC(c2cscc2Cl)=O)nn1-c1ccccc1 c1(OC)ncnc(C(=O)NCCC(C(C)C)NC(c2cc(=N)[nH]c(Cl)n2)=O)c1F C(N=c1[nH]cnc2cc(F)ccc12)C1(NC(c2c(C)nn(C)c2)=O)CCC1 N1(C(COCCC)=O)CCCCC1C(C)NC(c1occc1CC)=O N1(C(c2c(C)cccn2)=O)C2CCC1CC(CC(N1CC(F)C(F)C1)=O)C2 c1(CC)cn2c(C(=O)NCC(O)CNC(=O)C(C)NC(N)=O)cccc2n1 N1(C(c2c(C)nc(C(C)C)o2)=O)CCN(C)CC1CNC(C1CC12CC2)=O C#Cc1ccc(F)cc1CNC(=O)NC1CCCC1SC(C)(C)C N1(C(C2N(CCC)CCC2)=O)CCCC(CN2CCN(C(=O)COC(C)=O)CC2)C1 c1(CCC)cc(C(N2CC3CC2C3NC(=O)C(C2CCOCC2)C)=O)c(C)o1 N1(C(C(C)NC(C)=O)=O)CCCCC1CCN(C)C(C1(N2CCCC2)CC1)=O c1(C(N2CC(OC)C(NC(=O)Cc3cnn(C)c3C)C2)=O)ccc(C#N)nc1O C1(CC(=O)NCC2CC2Cl)(NC(=O)CC2CSC2)CCCCC1 Cc1cc(C(N2CCCC2(C)C(N2CCn3ncnc3C2)=O)=O)cc(C)c1O CCC(CC)(CO)C(=O)N1CCCOC(CNC(c2cn(C)nc2C)=O)C1 C1(C(=O)NC(c2cc(-c3ccco3)[nH]n2)C)CC12CCN(C1CCOC1)CC2 CC(C)(C)C(CNC(=O)CCc1ccc(N)cn1)NC(c1sccc1C(F)F)=O c1(NC(C2C(C(=O)NC(C)CO)C2)=O)onc2ccccc12 N1(C(c2scc(C(N)=O)c2)=O)CCN(C(C2CC2CF)=O)C(c2ccccn2)C1 c1(NC(C2(C)C(C)C2)=O)cccc2c1CCN(CC(=O)NCCc1cc[nH]n1)C2 N1(C(C(C)S(N)(=O)=O)=O)CC(NC(C2CC3(C2)CC(F)C3)=O)CC(C)(C)C1 C1(NC(=O)COCC2CC2)CC2CN(C(c3ncc(Br)cc3O)=O)CC12 C(=O)(C(C)(CC)C(=O)N1CC2CN(C(=O)CCN3CCC(F)C3)CC2C1)OCC c1(C(=O)NCC2CC(CC)CN2C(c2cnsn2)=O)cnc(OC)cc1F C1(C(=O)NCC(CC=C)NC(c2coc(C(F)(F)F)c2)=O)CCC2(CCC2)C1 C1(C(N2C(CC)CC(CC)CC2)=O)CCC2(CC2)N1C(c1cc[nH]c1)=O n1(CC)nnnc1C(C1CC1C1CC1)NCCNC(=O)C(C)C C12(CC(=O)N(CC(C)NC(=O)C(C)CC3CCCC3)CC)CCC(CC1)OC2 C12(C(N3CC(COC)(CNC(c4nnsc4C)=O)C3)=O)CCCN(CCC1)C2 C1(C(N(C)CC2CN(C(c3c(O)cc(C)nn3)=O)C2)=O)CCc2nnc(O)n2C1 C(C(F)(F)C(=O)N1CC(NC(c2cc(=O)cc[nH]2)=O)C(CC2CC2)C1)OC CCC(CC)C(F)C(=O)N1CCCC(F)(C(=O)NCC(n2cccn2)C)C1 C1(C2CC2)(CNC(C=C(COC)C)=O)CCN(C(=O)C=CI)C1 C1(C(=O)NC(COC)C2CC2)CCCC1NC(c1ccsc1)=O C(=O)(CC(C)(O)C(F)(F)F)N(C(=O)CC1CCn2cncc2C1)C N1(C(C(C)OCC=C)=O)CC(=O)NC(=O)C1 N1(C(C=NOC)=O)CCC(C)N(C(=O)CCOc2ccc(Cl)cc2F)CC1 Cc1cc(C(=O)NC2CCC(C)N(C(c3cc(C#N)c[nH]3)=O)C2)cnc1C C1(NC(c2c[nH]nc2[N+](=O)[O-])=O)CCC2CN(c3cnc(F)cn3)CC2C1 N1(C(c2n(C)nc(C(F)F)c2)=O)CC(NC(c2ccc(F)s2)=O)C2(CC2)C1 C(=O)(N=c1ccc(SC)n[nH]1)NC1(C(C=CC(=O)OC)=O)CCC(C)C1 CCCCC(C)(CO)NC(=O)CCCCCNC(=O)CCc1cc(C)nc(C)c1 C1(C(=O)Nc2ccc(CC(=O)OC)cc2)CC2(CCOCC2)CO1 c1(OC)ccc(CC(=O)NCC2(NC(C3(O)CCC3)=O)CC2)cc1 CCN=c1ccc(C(N2CCCCC(CNC(=O)C(=O)NCC3CC3)C2)=O)c[nH]1 N(C(=NC(C)C1CCC1)NC1CCC1)C(C#C)Cc1ccccc1 Cc1nn(CC2CCC2)cc1CNc1ccc(C2(C)CCO2)cc1 c1(C(=O)NC2(CNC(CCC)=O)CCCC2)cnncc1C C(N=c1[nH]c(=NCCCN(CCCC(F)(F)F)C)[nH]c2c1CSC2)c1c(C)coc1 c1(C(N2C(CNC(=O)COC3C=CCCC3)CCCC2)=O)ccc(Br)c(O)n1 N1(C(C(=O)N(C)CC2(OC)CCCCCC2)=O)CCC(C)CC(C)C1 n1(-c2ncc(C(=O)NCC(=O)N(C3CCC3)CC#C)s2)c(C)ccc1C C(=O)(C1=C(Cl)CCC1)NCCNC(=O)CCC(=O)c1ccccc1OC(F)(F)F C1(CC(C)C)CN(C(C(=O)NCCCF)C2CC2(Br)Br)CCO1 Cc1nccnc1C(=O)NC(C)CCN(C(=O)Cc1cncs1)C C(C(C)(C)CNC(=O)CSC)N.CC(C(=O)C(C)=O)=CC1CC1 C(=O)(CCCC(C)(C)C#N)NC(C(=O)NCCC(CC)(CC)OC)C1CCOC1 CC1(C(=O)NCCNC(=O)C2CC2)CC12CCN(C(N)=O)CC2 c1(CCC)c(NC(N2CCC(C)(CN(C)C)C2)=O)cnn1-c1ccc(Cl)cc1 N1(C(CCC(C)SC)=O)CC(NC(c2ccnc(C(F)(F)F)n2)=O)C2(CC2)C1 c1(OC)cc(C(N2CCN(C(=O)C3=CCCOC3)CC2)=O)c(OC)cc1Br C1(C#N)(C(N2CCCCC(c3n(C(C)C)cnn3)C2)=O)CC2CCC1CC2 N#Cc1c(I)c[nH]c1C(=O)NC1(c2ccc(Br)cc2)CCCOC1 N1(C(C2(NC(C3=CCCC3C)=O)CCCC2C)=O)CCN2CCCC2C1 C1(CCC)CN(C(C2CNC(=O)C2)=O)CCN1C(c1cc(Cl)cnn1)=O CCCC(CC1CCCC1)C(=O)NCC(C)(C)OCCNC(=O)Cc1ccsc1 c1(SC)cccc(NC(=O)Cc2ccc(C3CCNCC3)cc2)c1 Cc1ccoc1CC(=O)NC(C)CCN(C)C(C1COC(c2ccccc2)C1)=O c1(C(N2C(C)(CNC(c3c(COC)noc3)=O)CCC2)=O)cc(O)cc(O)c1 C=CC(CC(=O)NCC(C)NC(c1sc(F)cc1Br)=O)c1ccccc1 C1(CC(=O)NC2N(C(C(CN(C)C)N(C)C)=O)CC=CC2)CC(C)(C)OC1=O Cc1csc(=O)n1CC(=O)NCCCN1CCN(C(=O)CCc2cnc[nH]2)CC1 c1(O)cccc(Br)c1.CC1C(=O)OC2CC(C2)N1.c1(CCN)nccs1 N1(C(CC2N(CC)CCC2)=O)CCC(NC(=O)Cc2ccc(C)s2)C1C C(=O)(C(C)C(C)c1ccccc1Cl)NCCCN(C(c1c(CC)noc1)=O)C c1(COC)nc(=NCC2(CCNC(c3cnsc3C)=O)CC2)s[nH]1 C1(CNC(CCC)=O)C=CCN1C(=O)CCCc1ccc(C)o1 N1(C(CC(C)NC(=O)OC(C)(C)C)=O)CCC(N(C)C(c2cnc(Cl)s2)=O)CC1 c1(N(c2ccc(NC(=O)C(C3CCOCC3)N)cc2)C)ccc(I)c(Cl)c1 C(C)(C)(CCCNC(=O)COCC(F)F)NC(C1N(CC(C)C)CC1)=O CC(C)CCC(F)C(=O)N(CCC(=O)C(C)C#N)C.N C12(CCOC1)C(=O)N(CC)C2.C1(CO)CCC1CC1CCCC1 c1(OC)ccc2c(C(=O)NC(C)CCNC(C3(C(N)=O)CC3)=O)cc(O)nc2c1 C1(C2CCN(C(=O)C(C)C(C)(C)C)CC2)(NC(C2C(C)C3CCC2C3)=O)CC1 C1(C(N(CCN(C(=O)CN2CC3CC3C2)CC)CC)=O)CCCCCC1(F)F C1(C)(C(N2CC(C(C)NC(c3c(COC)cco3)=O)C2)=O)CCC(=O)N(C)C1 C(=O)(CCS(=O)(=O)Cc1ccncc1)OCCCC1(C(C)(C)C)CC1 C1(C(C)NC(=O)CCCC#N)COC(C)(C)CN1C(c1cnc(C(C)(C)C)nc1)=O CC(C)C(N=[N+]=[N-])C(=O)NC(C(N1CC2(CCCN2C)C1)=O)C1CCC1 c1(-c2cc(OCC)cc(OC)c2)n[nH]c2c1CN(C(=O)C(C)O)CC2 CCCCCC(C)(CC)C(=O)N1C2CCC1CC(NC(=O)C#CC1CC1)C2 c1(C(=O)NC(C)CN(C)C(C2CC2C2CC2)=O)cc2ccccc2n1C C1(F)(CNC(c2c(C)c[nH]n2)=O)CCC(CNC(=O)C(c2cccn2C)=O)CC1 c1(C(=O)NCC2CN(C(C(C=C)O)=O)C(C)CC2)nn2cccnc2c1Br C1(CC)(CNC(C2CCC(C)N2C(c2occc2C)=O)=O)CCCCO1 c1(C(=O)NCCN(CCC)C(c2ccn(C)c2)=O)ncoc1-c1cnn(C)c1 C(CCN(C)C)(C(=O)NOC1CCC1)NC(C(c1cc(C2CC2)on1)C)=O c1(OC)ccc2cc(C(N3CCC(C)(NC(c4ncoc4C)=O)C3)=O)n(C)c2c1 N1(C(CSc2nc(C)cc(C)n2)=O)CCC2CCN(C(=O)Cc3cnc[nH]3)C2C1 C=CC1OCCC1C(=O)NCC(C1(O)CN(C(=O)CC(C)C2CCCC2)C1)(C)C C1(=O)C(C)NC(=O)N(C)CCCN1CC.C(C)(C)(C)OC.C1(=O)CO1 N1(C(Cc2nnn(C)n2)=O)CCCCC1CC(C)(C)CNC(=O)C1=C(Cl)CC1 C1(c2cn(CCN(C)C)nn2)CCN(C(c2ccc(F)c(F)c2)=O)C1(C)C c1(CN2CCC(O)(C(=O)Nc3cccnc3Cl)C2)ccc(Cl)c(I)c1 C1(C(=O)NCC2CN(C(c3cccc(CCO)c3)=O)CC2O)COC2(CCC2)C1 Cc1nn(C2CCCN(C(=O)C(C)Cc3cnn(C)c3)C2)c(C)c1Cl.c12cn-1nn2 C12(C(N(CC(CN(C(c3ccc(CC)[nH]3)=O)C)O)C)=O)CCC(C1)OC2 c1(C(N2C(CCC)CN(C(C3CCS3(=O)=O)=O)CC2)=O)nccc2ncccc12 CC1C(NC(=O)N(c2ccccc2)CCCC(C)O)CCCN1C(=O)OC(C)(C)C C#CCC(CC#C)C(=O)N1CC(CNC(=O)CC(C)C(F)(F)F)C(COC)C1 Cc1cccc(N)c1C(=O)NCC#CCNC(=O)C(C(C)C)c1ccccc1 Cc1ccc(NC(C2CCN(C(c3c[nH]ccc3=O)=O)C2C(C)C)=O)c(O)n1 N1(C(c2n(CC)ccc2)=O)CC2(CC(NC(=O)C(N3CCCC(C)C3)=O)CO2)C1 Cc1[nH]c2ccccc2c1C(=O)NC1CCCC1C(=O)NCCC1CCOC1 c1(-c2n(-c3c(OC)cccc3)nc(C3CC3(C)C)n2)cc(Cl)nnc1O N1(C(COC(CC)(C)C)=O)CCCC1C1CCN(C(=O)CNC(=O)CN(C)C)C1 C(=O)(C(F)C(F)(F)F)N(C)CC1CCCN(C(=O)Cc2ccn(C(F)F)n2)C1 C(=O)(C=CS(F)(F)(F)(F)F)N(CC(CN(C(CNS(CC)(=O)=O)=O)C)O)C c1(C(CNC(c2cc(C)[nH]n2)=O)NC(=O)C(F)(F)c2ccccn2)ccc(F)cc1 C1(CC=C)(NC(=O)Cc2cncc(C(F)(F)F)c2)CCN(C(=O)C(N)=O)CC1 C12CCCN1C(=O)C21CC1.c1(CNC(=O)Cn2cncn2)cccnn1 CCCCCC(=O)N1CCCC(N(C)C(C2CC2(F)F)=O)C1 C1(CNC(Cn2ccc(C)n2)=O)CN(C)CCN1C(c1ccc(C(C)C)cn1)=O c1(C(N(C2CC(CNC(=O)CSC(F)(F)F)C2)C)=O)cccn2ccnc12 C1(C(=O)NC(CNC(c2c(CC)n(C)nn2)=O)C2CC2)C2CCCCCC12 N1(C(C(COC)OC)=O)CC(C(N2CC=CC2)=O)CCC(O)C1 C1(C(N2C(CCNC(=O)C(F)C3CC3)COCC2)=O)CC2CCC1CC2 c1(CC)ccc(CCNC(c2cc(C)[nH]n2)c2nnnn2C(C)(C)C)cc1 NS(=O)(=O)c1ccc(C(=O)NCCNC(CCCCO)c2ccccc2)[nH]1 C1(NC(=O)CCc2cnco2)CCN(C(=O)C(O)C2CC2)C(c2ccccc2)C1 C1(C(=O)NCCOCC#C)CCC2CCC1N2C(c1cnn(CCC)c1)=O C12(C(N(CCCNC(=O)Cc3cc[nH]n3)CCO)=O)CCC(F)(CC1)CC2 N1(C(c2cn(C)nc2)=O)CCC(NC(c2ccc(C#N)o2)=O)C(C(N)=O)C1 Cc1cc(C(N2CC(N3CCN(C(=O)Cn4cnnc4O)CC3)C2)=O)c(O)nn1 CC(CC(=O)N(CC(C)CNC(C1CC(C)(C)C1)=O)C)c1ccco1 N1(C(c2c(CC)nc[nH]2)=O)CCC2CN(C(=O)C(O)CC[S+](C)C)CC2C1 C1(C(N2CCCC2CCNC(C2(C)CC(F)(F)C2)=O)=O)(OC)CCCC(C)C1 CN1CCN(CC(=O)NC2(C)CC(NC(=O)Cc3nc(C4CC4)no3)C2)CC1 c1(NC(CC)(CNC(=O)C(C)CF)CC)ccc(C#N)c(C)n1 c1(C(N2C(C(=O)Nc3cc(C(N)=O)cc(F)c3)CC2)=O)c[nH]c2ccc(F)cc12 C1(NC(CC2N(C)C(=O)CC2)=O)CCCCCCC1NC(C1(C)CC1(C)C)=O CS(C)(=O)=NCC(=O)NC1CCN(C(=O)Cc2cccnc2Br)C12CC2 Cc1ccc(CCC(N2CCN(C(=O)CC3NC(=O)NC3=O)C3CC23)=O)cc1Cl C(CCCC(C)NC(=O)C(CN(C)C)Cc1cccc(F)c1)NC(CCC#C)=O C(=O)(CC(C)CC(C)(C)C)NC1CN(C(c2cnc(C)n2C)=O)CC1O CC1CC(NC(=O)C(=O)Cc2ccccc2)CCN1C(=O)Cc1cocn1 CCC(CC)C(=O)NC(CC)CC(=O)NCC1CCC(OC)C1 CCCCCCCCCC(O)C(=O)NCCCCC(CO)NC(=O)C(O)C1CC1 c1(-c2nc(-c3nc(C(C(C)C)(C)C)sc3)on2)ccccc1Cl C(=O)(CCCSC)NC(C)(C)CN.C1(N(C(C=C(COC)C)=O)C)CCCC1 C(CCCNC(=O)CCC1CCCOC1)(c1ccccc1)NC(C=C(C)Cl)=O CCCC(C(=O)N1CC(N(C(=O)CN(C)C)CC)C1)S(N)(=O)=O c1(CN2CC3CN(C(c4ccc(CC)cc4)=O)C3C2)c(C)cc(F)cc1C C1(C(N2C(C(C)C)CCC2)=O)CCN(C(=O)COC2CC=CC2)O1 C1(CC)(NC(=O)C(C)CC(F)F)CCN(C(c2ccncc2)=O)CC1 c1(C(=O)NCC2(NC(CSC)=O)CC2)sc(C)nc1C1CCCO1 c1(N(CC=C)C)ccc(Br)c(S(=O)(=O)NCCc2c(F)cncc2F)n1 c1(CC(=O)NC2(CF)CC2)ccccn1.CC C1(CNC(C2(OC)CCCCC2)=O)CC2CCC(C1)N2C(=O)C(C)C1CC1 N1(C(Cc2c(OC)c(F)ccc2)=O)CC2CCCC(C1)N2C(=O)C(=O)NC1CC1 Cc1cccc2[nH]c(C(N3CCC4CCC(C3)N4C(=O)CNC(N)=O)=O)cc12 C1(C)(c2cn(C(CC)C)nn2)CCCN(C(c2cccn2C)=O)C1 C(CN=c1nc(C#N)cc(C)[nH]1)C1N(C(Cc2cnc(C)s2)=O)CCCC1 C12(NC(c3ccn(CC(C)C)n3)=O)CCCC1CN(C(C1(CF)CC1)=O)C2 C(=O)(C(C)(C)CC(C)C)NCC1N(C(c2cnc(CC)[nH]2)=O)CC1 C1(C(=O)N(C2CC23CCOC3)CCOCC(F)(F)F)COCCN1C1CCCC1 Cc1cc(Br)c(Cl)cc1Nc1ncccc1C(F)(F)F.C12CC1C(=O)N2 C1(C)(NC(C(C)CCN(C)C)=O)CCCN(C(=O)CC2CCC(C)C(C)C2)C1 C1(CNC(c2c(C)snn2)=O)CC2CCCCC2N1C(=O)Cn1cccnc1=O N1(C(CCCOC)=O)CC(NC(c2[nH]nc(C(F)(F)F)c2C(F)(F)F)=O)C(C)C1 c1(C(=O)NC23CN(C(CCNC(=O)NC)=O)C(C2)C3)c(C)[nH]c2ccccc12 Cc1ccc(OCCNC(C2CCN(C(C3COC(=O)C3)=O)CC2)=O)c(C)c1 c1(OCC)ccc(C(=O)NCC2CN(C(=O)C(CO)N(C)C)CC2O)c(OC)c1 C(=O)(C#CC1CCCCO1)NCCCN(C(c1c(Br)ccc(C)n1)=O)C(C)C Cc1cccc2oc(N3CCC(C)C3CNC(c3cnc4ccccn34)=O)nc12 c1(C(C)C(=O)NCC2(F)CN(C(C3CCCOC3)=O)C2)nc(F)ccc1Cl N1(C(C(C(CC)O)C)=O)CCc2cc(CNC(c3ccc(F)cc3)=O)ccc2C1 N1(C(C(C)SCCCC)=O)C2CCC1CC(C(=O)Nc1ccc(Cl)cc1O)C2 c1(C(=O)NC2(CCNC(C(C)OC3CCOC3)=O)CCC2)ccc(N)cc1Cl C(=O)(C(CNC(c1ccn2nccc2c1)=O)CC(C)C)NCCN(C(=O)OC)C C1(CNC(C2CCC(=O)NC2)=O)CC2(CCN(C(c3cc(Cl)cnn3)=O)C2)CO1 CN1CC(C)(C)CC1NC(N1CCCC1c1c(F)cccc1Cl)=O Cc1cc(C(N2CCCCC(NC(c3ccc(F)nc3F)=O)C2)=O)nc(C)c1 C(=O)(C1=NOCC1)N(CC(CC)NC(=O)Cc1cccc(OC(F)F)n1)CC N1(C(CC2C(C)=NN(C)C2=O)=O)CCC2CCN(C(c3nnsc3C)=O)C2C1 CN1N=CC(CC(=O)NCC2CN(C(C3CCS(=O)(=O)C3)=O)C2)C1=O CCC(C#N)C(=O)N(C)CC1CCCN1C(C1(c2ccno2)CCC1)=O c1(C(=O)NCCN(C(CC(C)n2ccnc2)=O)C)ccc(C(=O)OC(C)C)c(F)c1 c1(C(=O)OC2(COC)CC(COC)C2)ccc(C)c(Br)c1 C1(C(=O)NCC2(C(=O)NCCSC(F)F)CCCO2)CC2(CC2)CO1 C(=O)(C1=CCc2ccccc21)N1C(CNC(c2cc(COC)on2)=O)CC1 c1(CC(C)NC(=O)C2=CCCC2)c[nH]c2ccccc12.N12CC3(C1)SCCC3C2 Cc1nn(CC(F)F)cc1-c1nc(-c2occc2C)nn1CCN(C)C c1(C(=O)NCC2C(NC(C3CN(CC)C(=O)C3)=O)CCCC2)cncc(Cl)c1C N1(C(C(COC)(C)O)=O)CCN(C)C(CNC(=O)Cn2nc(C)cc2C(F)F)C1 c1(OC)cc(C(=O)NCC2(NC(c3cccc(F)c3Cl)=O)CC2)cnc1Cl C#CC1CC2(CC2)CN1C(=O)NCC(C(C)(C)C)c1ccccc1 N1(C(CN(CC)CC)=O)CCC2CCCC12C(=O)NCCC1CCC(C)(C)O1 C1(=O)CCCCCCC(=O)NC(CO)C(C)NC(=O)C(C)(OC)C1CCOC N1(C(C2CC(O)CN2S(=O)(=O)CCc2ccccc2)=O)CC2(CC2)CC1CN C(=O)(CC1=CCCCC1)NCC(=O)N(CCNC(C=CCOCCOC)=O)C1CC1 CN1CC2CC1CN(C(=O)CCC1CCCCN1C(=O)COc1ccsc1)C2 C1(NC(C2CCCC(C)CC2)=O)CC2CCC1N(C(=O)C=Cc1cccnc1)C2 C1(C(=O)NCc2cc(C(=O)NCC(C#C)C(C)C)ncc2)CCC(=O)NC1C C1(CNC(CC(C)CCN(C)C)=O)CC2(CCN(C(c3cc(F)n[nH]3)=O)CC2)C1 c1(C(C)C)ncc(Br)c(=NC(CNC(C2CCC(=O)N2C(C)C)=O)C(C)C(C)C)[nH]1 C1(C)(C(=O)NCC(CC(C)C)NC(COCCCOC)=O)CCC(C)=C(C)C1 c1(CC(C(=O)NCCNC(CCNC(=O)NC)=O)O)ccc(F)cc1F c1(C(N2CC(CO)C(C)(C)C2)C(=O)NCCCCCC)nccc2ccc(Cl)cc12 N1(C(C2(CC#C)CCCO2)=O)CC(C(N2CC(F)(CF)C2)=O)CCC1(C)C C(C1CCCC1)=CC(=O)NCCC(=O)NCCCOc1cccnc1 N1(C(C(CSC)O)=O)CC(NC(=O)CCc2csc(C)n2)C(C2CC2)C1 CCC(C)(C(=O)NCc1ccoc1C(=O)NCCC1CC(C)=NO1)OC N#Cc1cnn2cc(Cc3nc(-c4ccco4)nn3C3CCCS(=O)(=O)C3)cnc12 C(=O)(CCCCC(C)C)N1CC(NC(C(CC)=CCCC)=O)CC1(C)C C(C(O)C(C)(C)C)N(C(C1C(NC(c2scc(COC)c2)=O)CCC1)=O)C c1(C(N2CC3CCN(C(C(C)C4CC4)=O)CC32)=O)cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 CCC(C)(C)C(O)C(=O)NCCC(=O)NC(CN(C)C)CO C#Cc1ccnc(C(=O)N(C(C)C(=O)NCC2=NOC(C)C2)C)c1 c1(C(=O)NCCOCCN(C(Cc2c(OC)ccs2)=O)C)[nH]c(C)nc1C c1(C(=O)NC(CCC)CCCNC(=O)CC(CC)C2CC2)cn2cccnc2n1 Cc1noc(C)c1SC1(C(=O)NC(C)C(C)NC(=O)CCc2ccccc2)CC1 C1(C2CCC2)(C(=O)NC2C(CNC(=O)Cc3cccc(Cl)c3)C2)CC1(F)F C1(NC(c2cc(C)cc(F)c2N)=O)CCCC2CN(C(=O)C3=CC(C)(C)C3)CC12 C#CCC(CC(=O)NCC(c1cnn(C)c1)C)NC(=O)CC1(C)CCOCC1 C(=O)(C1CCc2nccn21)N(C)CC1CCCN1N1CCCCC1.C(=O)C(N)=O C(=O)(C(CC(C)C)OC)NC(C(C(C)C)NC(COCC=C)=O)C c1(CC)cc(NC(CN2CCC(N(c3ccccc3)C)C2)=O)nc(C)n1 N1(C(CSCC#C)=O)CCCCC1C1CCCN1C(c1ccnn1CCF)=O C1(NC(=O)COc2cccc(F)c2F)CCCC2(CC1)OCCO2 C1(O)(C(C(=O)NCC(c2ccccc2)C)F)CN(C(=O)CCCC2CCC2)C1 C1(C)(CNC(c2c(OCC)ccs2)=O)CCC(NC(=O)CCCCOC)C1 c1(Nc2c(C)ccc(C)n2)ccc(S(=O)(=O)C2CC2)cc1 c1(OC)c(Br)ccc(F)c1C(c1nnnn1CC(F)F)NC(C1CC1)C1CC1 C(C(CC(C)C)C(=O)NC1CN(C)C(C)(C)C1)NC(c1cn(CCC)nn1)=O C(=O)(C(C)CC(F)(F)F)NC1C(SC)CN(C(C2C=CCS2)=O)C1 c1(C(N(C2CCN(C(C34CCC3C4)=O)C2)C)=O)cccc(C#N)c1 c1(CNC(c2nc(C)ccc2Br)c2n(C(CC)C)nnn2)cc(C#N)ccc1O C(=O)(CCC(F)F)NCCCC(=O)N(C(CN)C(C(=O)CCF)CC)C N(C(=NCCCF)NCC(C1CCCCO1)c1ccco1)C1N(C)S(=O)(=O)CC1 C1(F)(CNC(c2c(C)onc2)=O)CC2CCC(C1)N2C(=O)Cc1ccsn1 CC1CN(C(c2cccc(C#N)c2)=O)CCC1Nc1ncc(Cl)cn1 N1(C(CC(=O)NCC)=O)CC(NC(=O)COC2CCOC2)C(c2cnn(C)c2)C1 c1(NC)cc(Cl)ccc1C(=O)NCC1CC(NC(C2CCCC2(F)F)=O)C1 c1(C(N2C(C)CCC(NC(C3CC34CCOCC4)=O)C2)=O)cccc2c1OCCN2 c1(OC)ccc(C(N2C3CCC2(CNC(c2c[nH]c(=N)s2)=O)CC3)=O)cc1F C1(NC(c2n(C)nc(CNC(=O)CCCCCF)c2)=O)CC2(C1)CC(C#N)C2 N1(C(c2c(C(C)C)scn2)=O)CCN(C(c2cc(CN(C)C)no2)=O)CC1CF CCCCC(C(=O)N1CC(C(N2CC(C)CC2COC)=O)CC12CCC2)C(C)C C(CC1CC1)(CC(=O)N1CC2C(CC#C)C2C1)NC(CSCC#C)=O N1(C(C2C(C)CCC2)=O)CCC(CF)(NC(=O)C(C)OCC(F)(F)F)C1 CCC(CCC(=O)N(C(C)CN(C)C(c1ccc(C2CC2)s1)=O)C)OC C(=O)(C1=CC2CCCC12)NCC1(O)CCN(C(C(C(C)(C)C)NC(N)=O)=O)CC1 C1(CN(C(C2(C)CC(C)C2)=O)C)CCCN(C(C2CN(C)C(=O)N2)=O)C1 C12(CNC(C3C(C#N)C3)=O)CCC(NC(=O)CSc3cccc(Cl)c3)(CC1)CO2 CC1=C(C(=O)NC(c2ccc(F)cc2)C(=O)OCc2ccc(F)cc2Br)CCO1 Nc1cc(C(N2CCC3(NC(c4cn(C5CC5)nn4)=O)CC3C2)=O)ncc1Cl N1(C(c2nocc2Cl)=O)CC2CCCC2(C(=O)NCC2=NOC3CCCC23)C1 c1(N(C(CNC(Cc2c(CC)cccc2)=O)C)CCOC)ncc2ncnc-2[nH]1 CC1CN(C(c2cnnn2C)=O)CC1NC(C1(C)C=CCC1)=O N1(C(C(=O)OCC)=O)CC2CC2(C(=O)NC2CCC(C(=O)O)CC2)C1 C1(C(=O)NCC(CNC(=O)CC2CCSCC2)O)CCCC(CC2CC2)C1 C1(C(=O)NCC2CC(F)(CNC(Cc3n[nH]c(=N)s3)=O)C2)CCCN1C=O CC1COCC(CC(=O)NCc2ccc(C(=O)NC(c3nnnn3C)C)s2)O1 N1(C(c2c(C)cnnc2)=O)CC2CCCC(C1)N2C(C12CCC(C)(CC1)CC2)=O c1(OCC)cncc(C(=O)NCC2(F)CN(C(c3cnc(OC)s3)=O)C2)c1 c1(C(=O)NCCC2(O)CCN(C(=O)CCC3CC3(F)F)C2)cc(Cl)cnc1O c1(C(N2CCC(N(C(=O)C3=NOCC3)CCC)CC2)=O)cn2c(n1)CCC(C)C2 C1(N(C(N=S(CC#C)(C)=O)=O)C)CCOC2(CCC2)C1 C(C(C(=O)NC1(CCF)CC1)C(C)(C)C)NC(CCCC#C)=O CC(C)CC(C)(CNC(C1CCC(N(C)C)C1)=O)NC(=O)CCC(C)(C)F C#CC1CCCC(NC(=O)CC(CNC(=O)CCC(C)(C)OC)C2CCC2)C1 Cc1cnn(C)c1CC(N1CC(N(C(=O)CN2CC(C)C2)C)C(O)C1)=O C(=O)(C1c2c[nH]nc2CN1C(C1CCCN1C=O)=O)NCc1cc(OC)ncn1 N1(C(c2nc(OC)oc2)=O)CCC(NC(=O)C=Cc2ccccc2Cl)C(C)(C)C1 c1(CC)cc(F)ccc1C(=O)NC1CCCN(C(=O)COc2cnn(C)c2)C1C C1(C(=O)NCC2(CNC(c3c(C)cc(Br)o3)=O)CCC2)CCC2CCC(=O)N12 O=C1NCC2(CCN(C(C3C4CN(Cc5c[nH]ccc5=N)CC34)=O)CC2)N1 Cn1ccc(C(N2C3CCC2C(CNC(C2CCCC2O)=O)C3)=O)cc1=O Cc1ccn(CC(=O)NCC2CC2C(=O)NC(=O)CSCCC(F)(F)F)n1 C1(CNC(c2c(C(C)NC(c3c(C)n[nH]c3)=O)noc2)=O)CC(C)(C)CO1 C1(O)(N(C)C)CCN(C(=O)C(C2CCCCC2)NC(C2(C(N)=O)CC2)=O)C1 Cc1n[nH]c(=NC(C)CC2CCN(C(c3cnn(C)c3C)=O)CC2)o1 C(=O)(CCC(=O)c1ccc(F)cc1)NC(CNC(C(C)n1cnnn1)=O)C1CC1 C1(C(=O)NC(CC)CN(C)C(c2cn(C(C)C)nn2)=O)Cc2cccnc2C1 C1(C(=O)Nc2cc(COC)on2)N(C(=O)CC2(O)CN(C(C)=O)C2)CC1(C)C c1(C(=O)NCC(C)(CC)NC(CC(C=C)(C)C)=O)c(Cl)cc(Cl)c(Cl)c1F N1(C(C2CCN(C(=O)OC)CC2)=O)CCN(C)C(CNC(C2CCCSS2)=O)C1 n1(CC(=O)OC)cc(SCC(=O)NCCN2CCCC2=O)c2ccccc12 c1(NC(C2(C(=O)OC)CC2C)=O)ncc(Br)cc1OC(C)C C1(C)(NC(C2(CC#C)CCCO2)=O)CCN(C(=O)C#CC2CC2)CC1 N1(C(Cc2c(S(C)=O)cccc2)=O)CCC(C2CCCN(c3nnns3)C2)CC1 CC1(C)C2CCC1(C(N1CCN(C(c3cc4scnc4[nH]3)=O)CC(O)C1)=O)CC2 c1(OC)c[nH]c(C(=O)NCCCCCCC(c2cncn2C)C(=O)NC)cc1=O Cc1cccc(C(=O)NCCC(C)CCNC(=O)C(F)n2ccnc2)c1C C1(c2ccccc2F)(CNC(=O)NC(C)C)CCCCC1 C1(NC(C(C)Oc2cccnc2)=O)CC(N=c2nn[nH]n2-c2ccccc2)C1 C1(NC(C(CC)SC)=O)CCN(C(=O)C(C2CCC2)C2CCC2)CCC1C(N)=O C1(O)(CNC(C2(OC)CC2)=O)CCCN(C(=O)CCCc2nncn2C)C1 C12(CNC(c3ncc[nH]3)=O)CC(CN1Cc1cccc(CO)c1)C2 c1(CC(N2C(C)CC(NC(C3CCCC3CF)=O)CC2)=O)ccc2[nH]ccc2c1 CN1CC(C)(NC(=O)CCn2cc(C(C3CC3)NC(=O)OC(C)(C)C)nn2)CCC1=O N1(C(C(C(C)C)O)=O)CCOC2(CCCCC2NC(C2CNC(=O)C2)=O)C1 C1(NC(c2c(C(C)C)ncnc2)=O)CC2CN(C(C3(C#N)CCC3)=O)CC2C1 c1(C(=O)NCC(C)NC(c2cnc(CC(C)C)[nH]2)=O)ccc(Br)c(O)n1 C1(C(=O)OCC)(C(N2CCN(CCC(=O)O)CC2)=O)CC2CCC1CC2 CC(C)P(=O)(CC(=O)NCC1(O)CCN(C(C2C=CCCC2)=O)C1)C(C)C CCCC(C(=O)N(C)Cc1ccc[nH]1)NC(c1cc(C(=O)OC)ccn1)=O c1(OC)cc(N)ccc1C(N1CC(NC(C2CN3CCN2CC3)=O)C(C)C1)=O CCC(CC)(CCNC(C1CCC(C)(O)CC1)=O)NC(=O)C(COC)CC c1(C(=O)NC(CNC(c2c[nH]c(C)c(Cl)c2=O)=O)C)cccn2c(O)nnc12 C1(CC)CN(C(c2ncoc2CNC(=O)Cc2c(C)noc2C)=O)CCN1C C1(NC(=O)OC(C)(C)C)CCCCC1CNC(C1CN(C(=O)C(N)=O)CCO1)=O N1(C(C2(OC)CCN(C(=O)Cc3ccnn3C)C2)=O)CC2COCC2(C)C1 C(=O)(C(CCCC)C(C)C)NCC(C(=O)NCCOCC=C)CC1CC1 N1(C(C2(N(C(=O)C=C3CCCCC3)C)CC2)=O)CCOC2(CCC2)CC1 C(=O)(C(C)(C)CF)N(C)CC1C(NC(C(CC)OC)=O)CCC1 c1(C(N2CCC(NC(=O)CCC(F)F)CC2C2CC2)=O)ccc(Cl)c(F)c1F CCC(CN=c1ccc(S(=O)(=O)NC2CCC3(CCC3)O2)c[nH]1)N1CCCC1=O Cc1cccc2[nH]c(=NC3CC(CCNC(=O)CC(C)(O)C(F)(F)F)C3)oc12 N1(C(C=CC(C)NC(Cn2nnc(C)n2)=O)=O)CCC(OC)C1(C)C C1(C(=O)NCC2N(C(CC3C(C)CCC3)=O)CCC2)CC2C=CC1C21CC1 CC1CSCCCN1C(C1CC(C)N1C(C1CCCC1)=O)=O C1(C(=O)NCCn2cc(C(N3CC(OCC)C3)=O)nn2)OCCC1(C)C N1(C(c2c(CCC)nns2)=O)CCC(F)(F)C(CNC(c2sc(F)cc2C)=O)C1 C1(OCC(=O)NCC#CC)CCN(C(C2CC2C(C)C)=O)C1 N1(C(=O)Nc2cc(C)[nH]c2C)CCCc2cccc(OC(F)F)c21 N1(C(COC)=O)CCOC(C)C1Cn1cc(C(=O)NC2CC(NC(C)=O)C2)nn1 CC(C)CC(C)CC(=O)N1CCC(F)C(NC(=O)C(C)(C)c2cscn2)C1 c1(C(N2CC(CC)C(C(=O)NC(c3ccncc3)C)C2)=O)cccc(C)c1O N1(Cc2cc(CC)[nH]n2)N=C(C(=O)NC2CC(C(=O)OCC)C2)CCC1=O N1(C(C2(CC)CC(C)(C)C2)=O)CC(CNC(=O)C(C2CC(F)(F)C2)O)CC(C)C1 C1(C(N2CC(CC(C)NC(C(CC=C)(C)C)=O)C2)=O)CN(C)C(=O)CCO1 CC1C(NC(C2CCCS2(=O)=O)=O)C(C)CCN1C(=O)CC1CN2CCN1CC2 CCCC(O)(CCC)CC(=O)NC(C)(CNC(c1n[nH]cc1Cl)=O)C1CCC1 c1(SCC#C)ccccc1C(=O)N(CC(C)NC(c1ccc(SCC)cc1)=O)C c1(C(=O)NCC2CN(C(C(=O)NCC)=O)CC23CC3)ccc2nnn(O)c2c1 C1(C(=O)NC2CCC(CNC(=O)CCc3ccon3)C2)(CC)CCNC1=O c1(C(N2CC(C(C)NC(COCCC)=O)C2)=O)cn(C)nc1-c1ncccn1 c1(C(=O)NC(C)C2CC2)cnc(C=O)nc1.c1(C(=O)NC)cn(C2CC2)cn1 N1(C(C2(C=C)CCN(C(=O)CCOC3CCC3)C2)=O)CC(C)OCCC1C N1(C(c2nc(C)sc2)=O)CC2CC(C1)C2C(=O)CC1CCCC1C c1(CC)ccc(NC(C2(N(C)C(=O)OC(C)(C)C)CC2)=O)c(Br)n1 C1(NC(c2cc(C)nn2C)=O)CCN(C(C2C3COCC23)=O)C(C)C1 C(=O)(C(C(C)NC(c1ncccc1Cl)=O)C(C)C)Nc1c(OC)cc(F)cc1 C12(CNC(c3ncn(C)c3)=O)CC1CN(C(=O)CCCC1CCOCC1)C2 C1(CC(=O)Oc2n(CC)nc(-c3ccccc3)c2)CN2CCC1CC2 C(=O)(CCCC(C)(C)C)N1CC1.CC1CCCc2n[nH]cc21 c1(CC)oncc1C(=O)NC1CCC(CNC(=O)C(N2CCOC2=O)C2CC2)C1 C=C(C)c1cccc(NC(=O)C(CNC(=O)C(C(C)(C)C)OC)CC(C)C)c1 c1(CC)nc(N2CC3C(CNC(=O)CC(C)(O)COC)C3C2)c(F)c(Cl)n1 CC1(C)CCC1C(=O)NC1CC(CNC(c2ccn(CCSC)n2)=O)C1 N1(C(C(CC)SC)=O)C(C)C2CC1C2NC(=O)CNC(C1CCCC1)=O C1(NC(c2ncc(C)cn2)=O)CC2CCC(C1)N2C(=O)CCS(C)(=O)=O C1(CNC(C2CC(O)CCN2Cc2cccc(C(F)(F)F)c2)=O)=CN=C(O)C(N)C1 c1(CC)cccc(C(N2CCOC(C(C)NC(=O)CSCC(C)C)C2)=O)n1 N1(CC(=O)NC(C)CCc2ccccc2)CCC(C(N)=O)(CO)C1.C(N)=O C1(OCC)CN(C(=O)C(F)=CC2CC2)CC1NC(=O)CCOC1CCC1 c1(C(C)(C)C)scnc1C(=O)N(CCNC(C1CCCN1C1CC1)=O)C1CC1 C1(C(=O)NCCCNC(CC=C)=O)CC2(C1)CC(F)C2 C1(OC)CC(NC(c2cncnc2)=O)CN(C(=O)Cn2ncc(Br)n2)C1 C1(CCN(C(CC(=C)C)=O)C)CCN(C(=O)C(C)Cc2ccc(C)cc2)CC1 C(=O)(CCN=C(NCCF)N1CCN(C2CCN(Cc3nccs3)CC2)CC1)NC CCCCC#CC(C)(C)NC(C1CC(C)N1C(C1CCC(=O)N(C)C1)=O)=O Cc1cc(=NC(=O)C(=O)N2CC(CC(C)NC(C3CC(=O)C3)=O)C2)[nH]o1 C(CC(C(=O)NC1CONC1=O)NC(C1CCCN1C(=O)C(C)(C)C)=O)SC C1(C(N2CC(C#N)(CCF)C2)=O)CCCC(NC(=O)CN2CCCC2)CC1 N1(C(c2cc(C)[nH]c2C)=O)CCCC(CO)(NC(C2CCSC(C)C2)=O)C1 c1(CNC(C2(NC(C)=O)CC2)=O)occc1C(=O)N(C)CCF c1(OC)ccc(F)c(CC(=O)NCC2CCN(C(=O)COC(C)=O)CC2)c1 c1(CC(N2CC(F)(CNC(C(C(C)C)C3CCC3)=O)C2)=O)c(F)cccc1F C(=O)(C(C1=CCSC1)N1CC(C)CCC1(C)C)NCCCOC N1(C(CCc2cc(C)on2)=O)CCCC(C2CN(C(=O)C(C)c3cc[nH]n3)C2)C1 c1(OCC(=O)N(CC(CC)NC(=O)Cc2cncc(F)c2)C)cncc(Br)c1 C1(C(N2CC(C(N)=O)(CNC(CCC)=O)C2)=O)CCN(C)C(C)C1 C1(C(N2CCC(NC(CN(C(C)C)C)=O)C2)=O)CC(c2ccccc2)=NO1 C1(C(=O)NCC(C#C)CC)C(C)CCN1C(=O)C=Cc1cocn1 N1(C(c2cccc(Cl)c2C)C(=O)NC)c2c(Br)cccc2CC1C N1(C(C2(CSC)CC(=O)C2)=O)C2CCC(C2)C1C(=O)Nc1ccc(Cl)cc1O Cc1cn2c(n1)CC(C(=O)NCCC(C)NC(c1nnn3c1CSCC3)=O)CC2 N1(CC)CC(C(N2CCCCC2CCCNC(c2cnoc2C)=O)=O)NC1=O c1(OC)ccccc1CCOC(=O)CC1CCCC(C)C1 C1(C(=O)NCCc2ccccc2Cl)CN(Cc2ccc(Br)cn2)CCC1O c1(C(N)=O)ccc(F)c(NC(C2CCC(NCc3cccc(I)c3O)CC2)=O)c1 CC1CC=C(C(=O)NC2CCCCC2NC(=O)COc2ccc(Cl)nc2)CC1 N1(C(Cc2cn(C)nc2)=O)CCCCCC(C(=O)Nc2ccccc2[N+](=O)[O-])C1 c1(NC(C2C(NC(c3ccc(OC)cn3)=O)C2)=O)ccc(Br)c(F)c1F O=C(N=c1[nH][nH]c2c1CCCC2)C1CCN(Cc2cc(Br)ccn2)CC1 N1(C(c2cnc(C3CC3)nc2)C(=O)NC2(C)CC2)CCSC2CCCCC12 CCCC(C)(CCC)C(=O)NC1C2CC3C1C3C2C(=O)NC(COC)C(C)C C(c1ccc2c(c1)COCC2)=CC(=O)NC(C1CC(NC(COCC)=O)C1)C N1(C(C2N(C(c3cc(C)c(C)nn3)=O)CC(O)C2)=O)CC2(CCC1CO)CC2 C(=O)(C1=CCCCCC1)NC(CC(=C)C)C(=O)N(C)CC1CCCC2CC12 N1(C(C2(C)CCCS2(=O)=O)=O)Cc2ccccc2C(CNC(C2(F)CCC2)=O)C1 c1(CC(=O)NC2(CC=C)CN(C(=O)CC(C)(C)COC)C2)ccc2[nH]ccc2c1 c1(C(=O)NC)cc(NC(=O)CN(C(=O)CNC(C)=O)CC)cc(OC)c1 CC(C)CC(O)C(=O)N1CCOCC1CNC(=O)CCN1CCCCCC1 c1(C(=O)NCC2C(NC(C3C(CC)N(C)CC3)=O)C2)c(F)cc(Cl)cc1F c1(C(N2CC3C(NC(c4cnc(C5CC5)o4)=O)(CC3)C2)=O)cc(Cl)cc(F)c1F C1(CC(=O)NCCc2cncs2)COCCN1C(c1scnc1Cl)=O C1(N(C(C(C)OC)=O)C)CC2(C1)CC2NC(c1cccc(Cl)c1)=O S(=O)(=O)(c1ccc(NC2CCCC3CC23)cc1Br)N1C(CC#N)CC(F)C1 c1(CNC(C)=O)ccc(CO)cc1.N12CCCC(C1)c1cn(nn1)C(C)C2=O N1(C(C2CC(N(C)C)C2)NC(=O)CCC2CCCCO2)CCOCC1CC(F)F Cc1cc(Cl)c(Cl)cc1CN(C1CN(C(c2c(C)cccc2C)=O)C1)C Cc1ccc(S(=O)(=O)C(C)C(=O)N2CCC2CNC(=O)C#CC2CCCOC2)cc1 C1(COC)CN(C(C2CC2c2cnc[nH]2)=O)CCN1C(C1CCCCCCC1)=O c1(C(=O)NCC2CC(C)N(C(c3cnc4sccn34)=O)C2)c[nH]c(=N)nc1O C1(NC(C2C(CC)CCCN2)=O)CCC2(CCNCC2)C1 c1(CC)noc(C(=O)N(CCCN(C)C(C2CC2C(N)=O)=O)C)c1C Cc1cc(C)c(C(=O)NC(C2CC2C(=O)NCc2nn[nH]c2C2CC2)C)s1 CCCCCC(CC)C(=O)N(CCCNC(C12CC1COC21CCC1)=O)C1CC1 C(=O)(C#CC1(C)CC1)NC(C(c1ccccc1)NC(COCCSC)=O)C CCC(CN(C)C)CC(=O)NCC(C)CNC(c1nc(OC)ccc1C)=O C(CC(C)C(=O)NC(C)CCNC(c1cn(C2CCC2)nn1)=O)=CCC CC(C)CC(C(=O)NC1CCC1NC(c1coc2c(F)cccc12)=O)C(N)=O C(=O)(C(C)CS(C)(=O)=O)NC(C1N(C(c2cncc(C(C)C)c2)=O)CCC1)C N1(C(C(CC)C#N)=O)CCC(C2(NC(c3cc(C4(C)CC4)ccc3F)=O)CC2)C1 N1(C(CSCC=C)=O)CCC2(CCN(C(=O)COCc3ccc(C#N)cc3)C2)C1 N1(c2nnc(CC)o2)C(CNC(c2coc(C)n2)=O)CC2COCC12 c1(C(COC(=O)CC(c2ccon2)C2CCCC2)=O)ccccc1Cl c1(C(=O)NC2(CC=C)CCN(C(c3cc(C)c(Cl)s3)=O)C2)cccc(F)c1F c1(CC)noc(C)c1C(=O)NCC1(F)CC(CNC(C2CC2(C)Br)=O)C1 N1(C(c2c(C)nc[nH]2)=O)CC(N(C)C(c2ccnc(C3CC3)c2)=O)C2(CC2)C1 Cc1nc2ccccc2n1CC(=O)NC1CN(C(c2cn[nH]c2)=O)CC1N=[N+]=[N-] CC1(C)CC(C(O)CNC(=O)COC2CCN(C(c3cccnc3)=O)C2)C1 C(C)(C(=O)N1CC(c2ncccn2)C1)(C1CCC1)NC(COCCSC)=O c1(C(N2CCOC(CN(C)C)C2)C(=O)NC(CC)(C)C)cc(F)cc2c1CCC2 c1(OCC)ncc(F)c(N2CC(NC(c3cc(C#N)c[nH]3)=O)CC(F)C2)n1 c1(OC)ncnc(OC)c1C(N1CC(CCNC(C2CCCCC2(C)C)=O)C1)=O CC1(C(=O)NCc2cc(-c3ccco3)on2)CC(N)C1 c1(C(=O)NCCN(C(c2cc(C)on2)=O)CC2CC2)cc(F)cc(Cl)c1N c1(C(C)(C)C)cc(C(=O)NC2CC(O)(CNC(=O)C=Cc3cccs3)C2)on1 C=Cc1ccc(C(=O)NC2(CNC(C3CCN(C4CC4)CC3)=O)CC(OC)C2)cc1 c1(CC(=O)N(CCNC(C2C(OC)CC2)=O)C)cccc(C)c1Br c1(NC(C2CC3CC3N2C(c2cc3sccc3s2)=O)=O)ccc(F)cc1O c1(NCC(N2CC3CC3C2)=O)cc(=O)n2c(n1)CCCC2.N12CCC1C2=O c1(C(=O)NCCS(CC)=O)cnc2c(C)cccn12 C#CCCCCCCC(=O)NCC1N(C(C2CCC(C(N)=O)C2O)=O)CCC1(C)C n1(CC(=O)NC2CCC(NC(=O)CNC(=O)CC3CCCCC3)C2)nnc(=O)[nH]1 C1(c2n(CC(=C)C)nnn2)(Nc2nccn2CC)CCN(C)CC1C CC1CC(NC(c2occ3c2CCC3)=O)CN(C(=O)Cc2cnns2)C1 O=C(N=c1ccn(CCn2cc(CCC3CCCN3C)nn2)[nH]1)C1CCOC1 C1(NC(CC(COC)C)=O)COC2CN(C(=O)C=C3CCCCC3)CC12 C1(F)(CNC(C2C(CC(C)C)C2)=O)CCC(Cn2cc(-c3ccn(C)n3)nn2)C1 C1(C(C)(C)C)CCCCN1C(=O)CCNC(c1c[nH]c(C#N)c1)=O C1(C(N2C(COC)(CNC(c3coc(Cl)n3)=O)CCC2)=O)CC2C(C1)C2(C)C C1(COC)CCC(NC(=O)CC2CCCN2C(=O)CC2CC(SC)C2)CC1 c1(CC=C)cccc(NC(=O)NCCc2ccc(F)cc2)c1 C12CCCCC1N(C)C2=O.Cc1nc[nH]c1C(=O)NCC1CCN(S(C)(=O)=O)C1 O=C(NNc1cc(F)c(Br)c(F)c1)NCc1ncco1 C1(C(N2CCC(C(N)=O)C2)=O)CC2CCCCC2N1C(c1cccnc1)=O c1(CN=c2scc(-c3ccncc3)[nH]2)cccn2c(O)nnc12 C1(NC(c2cccc(SCC#C)c2)=O)(CO)CCCN(C(=O)C(C)NC(C)=O)C1 N1(C(c2n(CC)nnc2)=O)CCC2CCN(C(=O)C=Cc3nccs3)C2C1 C1(C2CN(C(C3CC(C)N(C)C3)=O)C2)(NC(c2c(C)nc(C3CCC3)o2)=O)CC1 CCCCC(=O)OC1CC(CCCNC2(C3CCCCO3)CC2)C1 C1(NC(c2ncc(C)cn2)=O)CCN(C(C2(NC(N)=O)CC2)=O)CC1CO C1(C(=O)NCCc2n(C)ncc2)COCCC1NC(C1CCC(O)C1)=O C12(CNC(C3CCC4(CC4)C3)=O)CC1CN(C(C1(CF)CC1)=O)C2 c1(Cc2nnc(-c3ccccc3)s2)ccc(Cl)cc1.CN(C)CCS c1(C(=O)NCCN(C(C2CCC(C(C)C)NC2=O)=O)C)cn2cc(Cl)cnc2n1 C(=O)(C1=C(Cl)CCOC1)NCC(C1CCCCC1)NC(c1c(C)cc(O)nc1)=O C1(CNC(=O)C(N2CCC(C3CC3)C2)=O)CCC2(CCCCCC2)O1 N1(C(c2n(CC)ncc2)=O)CCCC(C)C1CNC(=O)C(C)(C)c1ccno1 Cc1cc2c(cc1C)C(C(=O)NCCCCC(C)NC(C1CCCSS1)=O)CO2 C1(C(=O)OCC)CCC1(C)C(=O)N(CCCN(C(=O)C(C)CC)C)C C1(C(=O)NC2(C)CN(C(c3cncc(OC)c3)=O)C2)C2Cc3ccc(Cl)cc3C12 C(=O)(C(C)CN(C)C(C1CCCN1C(=O)CCCC1CCCO1)=O)OC N1(C(C=C(CC)CC)=O)CCN(C(=O)CCc2cncs2)CC(O)C1 CCCN(C1CC1)N1CCOC(C(C)NC(=O)C(C)(C)OCC(C)C)C1 CC(C)CCCC(C)C(=O)Nc1cccc2c1OCC2.C1(=O)CCN1C1CCC1 c1(C(N2CCC(CC)CC2C(N2CCC=C(Cl)C2)=O)=O)cccc2ccccc12 c1(-c2cc(C(=O)NC3CN(C(C(CSCC)O)=O)C3)no2)ccc(OC)cc1 N1(C(CS(CC)=O)=O)CCCC(C)C1CNC(c1cn(C)ccc1=O)=O N1(C(c2cccc(C(C)C)n2)=O)CCCC12CCN(C(c1cncs1)=O)CC2 N1(C(C(C(C)(C)C)NC(C)=O)=O)CC2CC(C1)N(C(=O)CCC1OCCO1)C2 Cc1cc(N2CCN(C(=O)CCN3CCCCC3)CC2)cnc1O N1(C(c2ncn(CC)c2)=O)CCCOC(CNC(C2(C)CC2Br)=O)C1 N1(C(c2c(C)c(N)ccc2)=O)CCCC(C2(NC(=O)C(C(C)O)N(C)C)CC2)C1 C(c1ccccn1)=C(C)C(=O)NCC1CC(NC(=O)CN2CSCCSC2)C1 C1(OCC)COCCC1CC(=O)NCC(C)N(C)C(c1ccoc1Br)=O c1(C(N2CCN(C(C3CCC(C)O3)=O)CC2C)=O)nnc(O)c2ccccc12 c1(COC)ncc(C(=O)Nc2cccc(CNC(=O)CSCCC(C)C)c2)cn1 C(CN=c1ccc(C(F)(F)F)c[nH]1)COCCNC(CN(CCC)C)=O C1(NC(c2c(OC)csc2)=O)CCC2(CCN(C(=O)C3=NOC4(CCC4)C3)C2)C1 C1(CNC(C2N(CCC)CCCC2)=O)CCCC12CCN(C(=O)CSCC)CC2 c1(N(C(C2N(CCC)CCC2)=O)C)cccc(OC)c1Br CC1(C)CC(F)(F)CN1C(=O)C(Cc1csnn1)NC(=O)OCC.C(C)(C)(C)O c1(C(N(CC(C)NC(C=C(CC)C)=O)C)=O)ccnc(CC(C)C)n1 c1(CC)cccc(F)c1C(N1CCOCC1CCNC(=O)C=Cc1ncc[nH]1)=O N1(C(C2(C)CCN(C)C2)=O)CCCC(NC(=O)CCN2CCCC2)CC1 N1(C(c2ccncc2O)=O)CC2(C(=O)NCC3(CO)CC=CC3)CC1CO2 C(=O)(C(C)(C)CS(C)(=O)=O)NCC(C)N(C)C(c1csc(C(F)(F)F)n1)=O C1(C(=O)NCC2(NC(c3c(C(C)=O)c(C)[nH]n3)=O)CCCC2)CCCCN(C)C1 c1(C(N2C(CNC(c3c(SC)ccs3)=O)CC(C)(C)C2)=O)cc2ccncc2[nH]1 Cc1cc(Br)cnc1C(=O)NCCC1CCN(C(C23CC(OC)C2C3)=O)C1 C(C)(C(=O)NC1CCCCN(C(=O)CCc2cncn2C)C1)(C(C)C)OC CC(C)(C)C1=NOC(C(=O)NCCNC(=O)C(c2ccccc2F)(C)F)C1 Cc1cccnc1C=CC(N1CCC(NC(=O)CCc2cn(C)cn2)CC1C)=O N1(Cc2nn(CC)nc2Br)CCn2ncc(C(F)F)c2C1 N1(C(c2cc(OC)cc(F)c2)=O)CCC(C2CC(NC(c3csc(C)n3)=O)C2)C1 CC(C)C(C(=O)NC1(C)CN(C(=O)C(C)(C)O)C1)NS(C)(=O)=O N1(C(C2C(C)N(C)CC2)=O)CCOC2CN(C(=O)CCn3cnccc3=O)CC12 C(CCCCC(=O)NC1CCN(C(c2cnc(OC)c(Cl)c2)=O)CC1C)OCC C(=O)(C1=CC2(CCOC2)C1)N1C(C)CC(NC(C2CC(=O)CO2)=O)CC1 C1(C)(CC)C=C(C(=O)NC(C(=O)N(C)CC)C2CCC2)C1 CC1(C#CC(=O)NCC2CN(C(=O)CCOc3cc(Cl)cc(Cl)c3)CCO2)CC1 C1(C2N(N3CC(C(C=O)OC)C3)CC2)CCCCC1.C(C)(C)(C)OC=O C1(CC(=O)NCC2(CNC(c3csnn3)=O)CC=CC2)CC=CCC1 C(=O)(C(CC)C(=O)N(CC(C)(C)CNC(=O)CC1CCC1C1CC1)CC)OCC N1(C(C)=O)CCCC(C)C1CNC(=O)CCc1ncc[nH]1 c1(OC)ccc(CCC(=O)N(C(C)CNC(=O)CC2CCCCO2)C)cc1OC C1(C(=O)NC2C=CC(COCC(=O)NC3CCOC3)C2)CC2OC1C1CC21 N12CC3CC1CN3C(=O)Cc1cccc(c1)C2=O.c1(CC)nccnc1OC C1(C)(C(N2CCCC(CN(C(C(C(=O)NC)(C)C)=O)C)C2)=O)CCC(C)C1(C)C N1(C(COCCCCC)=O)CCN(C(C2(CC)CC2)=O)C2(CC2)C1 Cc1ccc(S(=O)(=O)N2CCN(CCN3CCN(C)CC3)C(C)C2)c(C#N)c1 C1(C(=O)NC2CC3CN(C(CN(C(COC)=O)C)=O)C2C3)CCS(=O)(=O)C(C)C1 N1(C(C)C)CCCC(CC(=O)NC(C)(C)CNC(C2CCCCN2C(C)C)=O)C1 Cc1cccc2nc(N3CCCC(C(C)NC(c4cnc(C(C)O)s4)=O)C3)sc12 Cc1cccnc1-n1cc(-c2ncccc2C)nn1 C1(C(N(CCC)CC)=O)CCN(C(c2cn(Cc3nnc(CC)o3)nn2)=O)CC1 N1(C(C(C)OCC=C)=O)CCC2(CCN(C(=O)CCCNC(C)=O)CC2)C(C)C1 N1(C(CCC2CCC(C)O2)=O)CC2CCC(C1)N2C(c1ccc(F)cn1)=O c1(C(N(CC(CN(C(C(CC)F)=O)C)O)C)=O)cc(OC)ccc1[N+](=O)[O-] c1(C(=O)NCC(CN(C(CSCCOC)=O)C)C)cccc(-c2nc[nH]n2)c1 c1(C(=O)NCCOC(CC2ON=C(C)C2)=O)cc(OC(C)C)c2ccccc2n1 c1(OCC)cccnc1C(=O)NCC1C2CN(C(=O)CC3CCC(F)(F)C3)CC12 C1(CC(=O)NC2CCCC2)CCCN(C(C)C)C1.CCC1CCN1 N1(CC(=O)NC(CCCCNC(c2c[nH]cc(C)c2=O)=O)C)CCc2sccc2C1 C1(C(=O)NCC(COC)(C)CO)CCOCCN1C(=O)Cn1ncnn1 c1(SCCC(=O)N(CC(CC)NC(=O)CN2CCC(C)CC2)C)ccccc1O C(c1ccncc1)=CC(=O)NCC1(F)CC(NC(C23CC(C(C)(C)C)(C2)C3)=O)C1 c1(C(=O)NCC2N(C(C(CC=C)C)=O)CCOC2)c[nH]c2cccc(F)c12 C1(C)(CNC(c2c(CC)con2)=O)CCCN(C(c2nn(C)cc2C(C)=O)=O)C1 C1(NC(CC2CCC(=O)NC2)=O)CCS(=O)(=O)C12CN(C(=O)CCC[N+](=O)[O-])C2 c1(N2CC(C)OCC2)nc(N2CCC3(CCCC3)CC2)nc2c1CSC2 c1(C(CC(=O)O)NCCc2ncc(CC)s2)ccc(Br)c(C)c1 C12(CNC(CC=C=C)=O)COCCN1C(=O)CN(C(c1nc(C)ncc1Cl)=O)C2 N1(C(C2(C)CC=CCC2)=O)CCCC(C(=O)N(C2CC2)C2CC2)CC1 N(C1Cc2ccccc21)C(=O)CCn1cc(-c2cc(F)ccc2Cl)nn1 C1(NC(c2csc(Br)c2)=O)CCN(Cc2cc(Br)c[nH]2)CC1F C(=O)(C1CCCc2nc(C)[nH]c21)N1CCC(NC(c2cc(C)c(F)cn2)=O)C1 O=C(CCC1=CCCCC1)NCCNC(c1ccsc1)=O C1(C(=O)NC(C2CN(C(c3cnc(SC)s3)=O)C2)C)COC2COCC12 c1(N(C(C(C=C=C)C)=O)C2CCN(C(C)=O)C2)cc(F)cc2[nH]c(COC)nc12 c1(CC(COC(COC(Cc2nnc(C)o2)=O)=O)=O)ccc(C)c(C)c1 C1(C(=O)NCC2N(C(c3ccc(C)nc3C)=O)CCOC2)CC2CSCC(C1)C2 c1(C2(C(=O)OC)CC2)ccc(-c2ccnc(NCc3ccc(F)cn3)c2)cc1 N1(C(c2nc(C)oc2C)=O)CCCC(C)(CNC(C2(c3cc[nH]n3)CC2)=O)C1 N1(C(N2CC3CC3C2)=O)CCC(N=c2[nH]c(C(F)(F)F)nc3c2CCC3)C(F)C1 c1(OC)ccc(C(O)C(N2CC(F)(CNC(c3cn(CC)nc3C)=O)C2)=O)cc1 C(C(C)C(C)C(=O)N1CCCC(NC(=O)COc2cccc(C)c2C)C1C)OC c1(OC)ccc(C(=O)NCC2C3CCC(C3)C2C)c(C)c1 C12(CNC(CN(C)CC)=O)CC1CN(C(c1ccnc(C(F)F)c1)=O)C2 N1(C(CCOC(CC(C)C)C)=O)CC(NC(=O)C=Cc2nccs2)C2(CCC2)C1 N1(C(c2c(CC)occ2)=O)CCN(C(=O)C(C)(COC)COC)CC1C CC1CCCN(C(=O)C=Cc2cnn(C)c2)C1CNC(=O)CCCCC1CC1 C(=O)(C(O)CCC(C)C)NC(C(=O)NC(CC=C)CO)CN=[N+]=[N-] C(C(C)(C(=O)NCC1CC(O)CN1C(=O)CC(C)C1CCCC1)OC)OC c1(N2CCC(C=C)CC2)[nH]c(=NCc2c[nH]nc2C2CCCCC2)nc2scnc12 n1(CC(N2CC(CC)N(C(=O)Cc3cc[nH]c3)CC2)=O)ccc2c(C)cccc12 c1(NC(N(CC(O)C2CC2)C)=O)ccc(N2CCOCC2)nc1C C(=O)(CCCCCCCC1CC1)NCCNCCCNC(Cc1ccn(CC)n1)=O C1(C2CCN(C(=O)Cn3ccnn3)C2)(NC(C(C)C(C)(F)F)=O)CC1 C1(C(=O)NCC2N(C(CCCn3c(C)cc(C)n3)=O)CC2)CCCC1S(C)(=O)=O c1(CC)nn(C)c(CC)c1C(=O)N(C)CC1CCCN1C(=O)CN(C)CC C1(CNC(C(C)NC(=O)NC)=O)COCCN1C(c1ccc(C)cn1)=O C1(CNC(c2c(C3C(C)C3)noc2)=O)CN(C(=O)CC(C)(F)F)CC12CC2 C(=O)(C(C)CC(F)F)C(CCN(C(C)C)C(C1(C)CC2(CC2)C1)=O)=O.OC c1(C(N(CCNC(C(C)OCCC=C)=O)C2CC2)=O)ccnc2c1ncn2C CCCCCCCC(=O)N1CCOC(CNC(=O)CC2CC(F)(F)C2(F)F)C1 CCC(CC(=O)NC1(C)CCN(C(=O)Cn2nc(C(C)(C)C)cc2N)C1)C(C)(C)C N1(Cc2ccc(C(=O)O)[nH]2)CC2CCN(S(=O)(=O)c3nccs3)CC2C1 c1(C(=O)NCC2CCN(C(c3ccc(C(N)=O)s3)=O)C2)ccc(O)c(CO)c1 Cc1ccc(OCC(N2CCN(C(=O)CC3(C)CC3)C3CC23)=O)c(Br)c1 C1(C(=O)O)C(N)CCCN1C(c1ccc(N2CCOCC2)o1)=O CC1CN(C(c2cc(F)c[nH]2)=O)CCCN1C(c1c[nH]c(Br)c1)=O Cc1n[nH]c(C)c1CC(N1CC(C(C)NC(=O)CCCc2cccnc2)C1)=O c1(C2(NC(=O)NC(C(C)(C)C)Cl)CC2)ccc(OCC(F)(F)F)cc1 c1(C(C)NC(=O)NC2CC(CO)C3CC23)nccc(Cl)c1O C(=O)(CS(=O)(=O)C(C)(C)C)NCC1(F)CCN(C(C2(NC(C)C)CC2)=O)C1 C1(CC(=O)N(C2(C)CCN(C(=O)CCc3cnc[nH]3)C2)C2CC2)CN2CCC1CC2 Cc1c(C2OCCC2NC(=O)NCC2CCNC2=O)cnn1C CCC(CN(C)C)CC(=O)N(CC(C)C(=O)NCCCC(N)=O)C CCCC(C(F)(F)F)NC(C1CCC(C2CC2)N1C(c1sccc1OC(C)=O)=O)=O Cc1n[nH]c(C)c1C(C)CC(=O)N(CC(C)O)CCNC(C1(CC(F)(F)F)CC1)=O Cc1ccc(C(=O)N(C2CN(C(=O)CCCC(C)(F)F)C2)C)c(N)c1C C123CC4CC1C2C4CNC3=O.c1(SC)cccc(Cn2cc(C3CCCO3)nn2)c1 Cc1ccc(CC(N2CCN(C)CC2CNC(=O)C(=O)NC2CC2)=O)c(F)c1F C(=O)(C(C)C(C)(F)F)N1C(CCOC)C=CC1.c12ccc(cc1)-c1cn(nn1)C2 N1(C(C=C(C)C)=O)CC2CCC(C1)N(C(c1cncc(F)c1C(F)(F)F)=O)C2 C#CCCCCCCC(=O)N1CCC(C(C)C(N2CCOC(C#C)C2)=O)C1 C1(C(=O)NCCCN2C(C)CCCC2)CN(C(=O)Cc2cnsc2)C(C)(C)C1 C1(CCC(N2CCC2C=O)=O)CCCN(CC)C1.C(CCCN(C)C)N(CC)CC CC1(C)CC(CC(=O)NCC2CC2CN(C(c2cccn2C)=O)C2CC2)CO1 c1(C(N2C(CC)CN(C(=O)CN3CC4CC4C3)CC2)=O)ncnc2c(C)csc12 CC12CC(C(N3CCN(C(C4CC5CCC(C4)S5)=O)CC3)=O)(C1)C1(CCC1)O2 c1(C(N(C2CCCN(C(CC(CC)SC)=O)CC2)CC)=O)cn2c(n1)CCCC2 N1(C(CN(S(C)(=O)=O)C)=O)CC2CC(NC(c3sncc3Br)=O)CC2C1 C(=O)(CCC(=O)NC1CC1CNC(C1CCN1C)=O)NCC c1(C(=O)NC2(CNC(C(N3CC(C)C3)C)=O)CCC2)ccc(Br)c(F)c1 c1(C(N2C(C)CC(NC(c3ncc(C)cn3)=O)C2)=O)cc(N)cc(N)c1 C=CCC(CN(c1ccccc1)C(=O)CCOC)NC(=O)C=C(Cl)Cl c1(CNC(C(C)OC(C)=O)=O)ccc(C(N2CCC2(C)C(C)C)=O)s1 c1(OCC(=O)NC(CC(=O)OC)C)cnc(SC)nc1O N1(C(c2cncc(Br)c2)C(=O)NCCCSC)CCn2[nH]c(=N)nc2C1 C1(C)(CC)C=C(C(=O)NC2COCC2NC(c2ccc(F)cc2)=O)C1 C1(C(=O)NCC(CC=C)NC(=O)CCCC2CC2)CCN(c2ccccc2)CC1 C(CCC(C)C(=O)NC1CCCC(NC(=O)CCCNS(C)(=O)=O)C1)OC CCC(COC(c1cnn(-c2ccc(C)cc2C)n1)=O)CC(F)F c1(C(=O)NC(CCCNC(C(CC)n2ccnc2)=O)C)ncnc(OC)c1F C1(C(=O)NCC(CC)NC(=O)CN2CC3CC3C2)CCCN(C(C)=O)C1 Cc1cc(C(=O)NCC2CC3CC3N2C(=O)CC2(OC(C)C)CC2)n(C)n1 C1(C(=O)NCCC#CCO)(CNC(c2cc(CCO)on2)=O)CC2(CC2)C1 Cc1cc(C(=O)NC2CS(=O)(=O)CC2NC(c2sccc2C(F)F)=O)cc(O)n1 C1(OC)CC(C)(C)C(C)(C)C1.C(=O)(CC(=O)NCCC1CN1)OCCCOC Cc1csc(COC)n1.C1(=O)C(CNC(c2c[nH][nH]c2=N)=O)N1 c1(C(=O)N(CCO)C2CC2)cscn1.O=C(CN)N c1(C(N(CC(C)NC(c2cc(CSCC)on2)=O)C)=O)n[nH]c2c1COCC2 CP(C)(=O)c1cnc(C(=O)Nc2cc(Br)cc3c2OCCC3)cn1 C(C(C)(C)CC(=O)NCCCCCCNC(=O)Cn1cnc(C(F)(F)F)c1)OC N1(C(C(CCC)C)=O)CC2(CC(C(=O)NC(C)CCC(F)(F)F)CO2)C1 N1(C(c2c(OC)cc(C)cc2)=O)CC2CCCC(CNC(=O)C(C)OC)(C2)C1 N1(C(C(=O)NCc2ccc(OC)cc2)C(C)C2CC(F)(F)C2)Cc2ncsc2C1 C1(NC(C2(C)CS(=O)(=O)C2)=O)CCC2(CCCN(C(c3cc(Cl)c[nH]3)=O)C2)C1 C#Cc1cncc(NC(=O)C(CC(F)F)NC(c2cn(C)ccc2=O)=O)c1 c1(C(=O)NCCNC(=O)Cn2cnc3c2CCCC3)cccn2c(O)nnc12 CC(C)C(C(=O)NCCC(C)NC(=O)CCc1cccc(O)n1)c1cnn(C)c1 c1(C(=O)NC(C(C)NC(c2cnc(CC)[nH]2)=O)C(C)C)ncc(C)cc1C C1(NC(c2ccon2)=O)CCN(C(C2CCCC23CC3)=O)C12CCC2 C(=O)(CC(O)CC(C)(C)C)N(CC(=O)NC(c1cc(C)on1)C)CCOC C1(N(C)C(=O)N(C2(C(F)(F)F)CC(O)C2)CCO)CCC2CC2C1 C1(CNC(c2scc(OC)c2)=O)CCCCN(C(=O)Cc2cc(C)cc(F)c2)C1 c1(CNCC2CCN(C(CC(CC)SC)=O)C2)ccc(CC)cc1F c1(C(N2CC(NC(C#CC(C)C)=O)C(F)C2)=O)cc2c(Cl)ccc(Cl)c2[nH]1 C1(C(=O)NCC=O)COCC(=O)N1C1CC1.C(=O)(C=C(C)C)N(CCOC)C C(=O)(C1Cc2ccccc21)N1C(C#C)CC1.C1(=O)CC(C)N1CC C(=O)(CCC(F)(F)F)NC(CC1CCCN(C(c2c(C(C)C)ncnc2)=O)C1)C C1(NC(CC(C)(C)c2cccs2)=O)COC2CN(C(c3cnc(=N)[nH]c3)=O)CC12 N1(C(C2CCC(=O)N2)=O)CCC(N2CCC3CCOC3C2)C2(CC2)C1 c1(C(N(C)CC2(NC(C(C3CC3)OC)=O)CC2)=O)ccc(Cl)cc1 Cc1nc2ncc(C(=O)NC(C3CCOC3)CNC(=O)C#CC3CC3)cc2o1 c1(C(N2CCC(NC(C3C(C)C3C)=O)CC(F)C2)=O)ccc2[nH]nc(Cl)c2c1 N(C(=NCCSC)N(CC)Cc1cscn1)C(CC)C C12(C(=O)NCC(CCNC(=O)C3CC3)O)CCC(CO)(CC1)CC2 c1(NC(C2N(C(CC)C)CC2)=O)ccc(F)c(F)c1 C1(CC(=O)NCC(C)(C2CCC2)NC(c2occc2CN(C)C)=O)CCOCC1 c1(OC)ncc(NCc2ccc(CN3CCC4(C(C(=O)OC)C4)C3)o2)cc1CO S(=O)(=O)(c1c[nH]ccc1=NCCCCNS(C)(=O)=O)N1CC(C)S(=O)(=O)C(C)C1 C1(CN(C(C2(CCC)CCC2)=O)C)CCCN1C(=O)CNC(=O)CN(C)C c1(CC(=O)NC2C(CNC(CC)=O)C2)sc(C)nc1C.C1C(=O)N1 C1(CNC(CCCOCC)=O)(OCCNC(C2CCC(O)C2)=O)CCOCC1 CN=c1[nH]nc(CC(=O)NC2CC2NC(c2ccc(SC)cc2)=O)s1 C1(O)(CC)CCCN(C(=O)CC2(CNC(C3CCCN(C)C3)=O)CC2)C1 C(=O)(C#CC1CCCCO1)N1CCC(O)(CNC(c2c(Cl)cnc(C)n2)=O)C1 N1(C(=O)CC2COCCO2)CCC2OCCN(C(c3ccc(CO)o3)=O)C2C1 N1(C(CCC2(C#N)CCC2)=O)CC2CCC2(C(=O)NC2CC(CO)C2)C1 c1(C(=O)NC2CN(C(Cc3cccc(C)c3)=O)CC(C)C2)ncccc1N=[N+]=[N-] C1(CC(=O)N(C(c2ncccn2)C)C2CC2)CN(C(=O)CC(C)(C)O)CC1C CC1CCN(C(C2CCCN(C(c3cc(=O)cc[nH]3)=O)CC2)=O)CC1(F)F c1(C(N2CCC(C)(NC(c3cc(F)c[nH]3)=O)C2)=O)ccc(O)c2c1CCCC2 c1(C(N(C2CCCN(C(CC)=O)C2)C)=O)cccn2c(O)nnc12 C1(C(N2CC(NC(COCCCC#C)=O)CC2(C)C)=O)CCS(=O)(=O)C(C)C1 C12(CC(F)(F)C1)CNC(=O)N2.N1(OC)CCCC1(C)C1CCC1 Cc1nc(C(F)(F)F)sc1C(N1CCC(C2(CO)CC2)C1)=O c1(C(N2CCC(NC(C3CC3CF)=O)CC2)=O)ccn2ccccc12 c1(C(N(C2CCN(C(c3cc(CCC)n(C)n3)=O)C2)C)=O)[nH]cc2c1CCCC2 c1(CC)cc2c(NCC3CN(C(C4(O)CCSCC4)=O)C3)nc(C)nc2s1 Cc1ccc(F)cc1OC(=O)CCC1CCCCN1S(=O)(=O)CC1CC1 CCCCCCCCCN1CCC(O)(C(N2CCCC(F)(F)CC2)=O)CC1 N1(C(C(=O)N(C)C)=O)CCC(CNC(=O)CC2CCOC2)C1(C)C S(=O)(=O)(CC(=O)NC(C)(CNC(C1(COC)CCC(=O)N1)=O)C1CCC1)NC C1(NC(CN(c2ccccc2)C)=O)CCOC2(CCS(=O)(=O)CC2)C1 Cc1nc(O)nc(S)c1CN1CCCC1Cn1ccnc1 C1(C(=O)NCCCCC2N(C(C3CCC(C)C3)=O)CCC2)CC2C=CC1C21CC1 n1(COC)ncc(C)c1C(C(=O)NCC1CCOC1)NC(c1cccc(C)c1)(C)C C(=O)(C1=C(Cl)CCC(C)C1)N1CCC(N(C(C2(COC)CC2)=O)CC)(COC)C1 CCCCC(C)C(=O)NCC(CNC(c1ccc(Br)cc1Cl)=O)CO C12(C(=O)NCC(CNC(C(C(C)C)n3cnnn3)=O)C)CC(C)(C1)OC21CCC1 CC1(C)COCC1CC(=O)NC1CC1CNC(=O)C(c1ccc(Br)cc1)O c1(C(N(C2CC(CNC(=O)C(c3cnn(C)c3)O)C2)C)=O)cc(O)ccc1F C1(C(N)=O)CC(C(=O)NC(C2CCOC2)CNC(=O)C(=O)NC2CC2)C1 Cc1cc(F)ccc1S(=O)(=O)NC(C1OCCOC12CCC2)=O c1(C(=O)NCC(C)NC(C=C(C)c2ccsc2)=O)cc2c(ccn2C)[nH]1 N1(C(CSCC=C)=O)CC2CC2(CNC(C2CC(C(F)F)C2)=O)C1 N1(C(c2c(OCC)ccs2)=O)CC2CCC2(NC(C2CCCO2)=O)C1 C(=O)(C(CO)C(F)(F)F)N1CC2C(CNC(c3cncnc3C3CC3)=O)C2C1 C1(C(=O)NCC(CC)NC(COCCSC)=O)CCOC(C)C1.OC C1(NC)CCN(C(C=CC(=O)NC2(CF)CCC2)=O)C1.c12n[nH]cc1NC2=O c1(C(C)NC(C2CN(C(C=NOC)=O)C2)=O)cccc(Cl)c1 CCCCC(C)(F)C(=O)N1CC(CCNC(C2CC23CCCC3)=O)(OC)C1 Nc1cc2c(cc1C(=O)NCCCCCNC(=O)CCc1cncnc1)OCO2 N1(C(CC2N(C(C3C(C)CC3)=O)C3C2CCC3)=O)CCOC2COCC12 C(=O)(C(C)(C)C(=O)N1CCCC(CCNC(=O)CC2CC3(CCC3)C2)C1)OCC c1(C(=O)NCC(C)C)cccc(C(F)(F)F)c1.C1C(C)(C)C2CN(C2)C1=O N1(C(C(=O)NCc2nc(NC(C)=O)sc2)=O)CCOC(c2cccc(O)c2)C1 N1(C(C(C)(C)OC(C)C)=O)CCCC(CCC(=O)NCC(C)CC2CCC2)C1 C1(NC(CCCNC(=O)C=CC2CCOC2)=O)CCn2ncnc2C1 C1(C(C)C)CNC(=O)C2CC2CC(=O)N1.C1(CC)CC(CC(=O)OC)C1 Cc1nc(CC(=O)N(CCC(C)NC(C2CCCO2)=O)C)c(Cl)s1 c1(C(=O)NCC(CCC)NC(c2c(C)n[nH]c2C)=O)cc2ccnc(Cl)c2[nH]1 c1(C(=O)NCCC(C(=O)N(CCO)CCO)OC)c[nH]c2nccc-2c1C C1(C(=O)NCC2CCN(C(C3C=CCCC3)=O)CC2)CN2CCCN1CC2 S(=O)(=O)(c1ccc(C(N2CCOC(CNC(c3nncs3)=O)C2)=O)cn1)N(C)C CC1CCN(C(c2cnsn2)=O)CC1NC(=O)Cn1nncc1N CCCCCCC(=O)NCCCCn1ccc(=O)cc1.N1(C=O)CC([N+](=O)[O-])C1 C12(C(=O)NCC3(C)CCN(C(C(CCCOC)C)=O)C3)CCC(CF)(CC1)CC2 c1(C(N2C(CCC)CCC2)C(=O)NCCOC)ccc2c(OC)cc(OC)cc2n1 C(C(C(=O)NCC(C)NC(=O)CN(C)Cc1ccccc1)OC(C)(C)C)SC C1(CNC(CC2(C)CC2)=O)CC2(CO1)CN(C(C1C(F)(F)C13CCC3)=O)C2 C(=O)(CC1=CCCC1)NC1CCC(NC(C(CC)(O)c2cccc(Cl)c2)=O)CC1 C(=O)(C#CC1(C)COC1)N1CCC(C)(NC(c2cc(C)ns2)=O)C1 C1(C(N2CC(C(c3ccccc3)C)C2)=O)Cc2cc(F)ccc2O1 c1(CN2CCCC(C(C)NC(c3ccc(F)c(Br)c3)=O)C2)cc(F)c(O)c(F)c1 N1(C(C=C(CCN(C)C)Cl)=O)CC(CO)(NC(=O)Cc2cncnc2)C1 c1(C(=O)NC(C2(C(N(C3CC(OC)C3)C)=O)CC2)C)cccnc1 C(c1sc(Cl)nc1Cl)=CC(=O)NCC1C2CN(C(CN(C(=O)OC)C)=O)CC21 C1(CNC(C(CC)N2CCCC2=O)=O)CCCCN1C(=O)CCOCCOC c1(OCCOC)cc(O)ccc1NC(=O)C(c1ncccc1C)O C(=O)(C1=Cc2ccccc2C1)NC1C=CC(NC(C(C)Oc2ccncc2)=O)C1 C(CCCC(=O)NCC12CCCC1C2)N(C(C1(CC)CC1)=O)C Cc1c(C(=O)N(CC(O)CNC(C2CCCN2C)=O)CCO)cnn1CC(C)C C1(CNC(C(OC)OC)=O)COCCN1C(=O)Cn1cc(-c2ccccc2)cn1 C12(NC(C3C(C)C3C)=O)CCC1CN(C(c1cc(-c3c[nH]nn3)ccc1F)=O)C2 C(=O)(C1=C(F)CN(C(=O)Nc2ccccn2)CC1)NCCNC(=O)CC1CCC1 C(=O)C(CC=C(Cl)Cl)c1ccccc1.CCC(C)CC(=O)O C(C)(CC(=O)N1CCC(CC(=O)NCc2ncc(CO)o2)C1)OC C1(C(N2C(CN(C(c3c(C)occ3)=O)C3CC3)CCC2)=O)CCC12CCC2 C(CCCC(=O)NCC1(F)CC(C(=O)Nc2cnccc2Br)C1)OCCC=C C12(CNC(c3cc(CSC)no3)=O)CC1CN(C(=O)CCOC1COC1)C2 c1(C(CC)O)nnc(C2CCCC2)n1CCC(c1ccccc1)C1CC1 n1(CC)nnnc1C(CCOC(C)=O)(C(C)(C)C)NCCc1noc(C(C)C)n1 CCCC(CNC(=O)C=CC1CCCC1)C(=O)N(c1ccccc1)C.C1CO1 C(=O)(CCn1cccn1)NCC1(CN(C(=O)C=CCF)C2CC2)CC1 c1(NC(C2CC(NCc3nc(C)c(Br)cc3)C2)=O)cccnc1[N+](=O)[O-] C1(NC(C2C(C=C)C2)=O)CN(C(c2cc(F)ccc2C(F)(F)F)=O)C2(CCC2)C1 N1(C(C(CC2CC2)NC(=O)OC(C)(C)C)=O)CC2CC2(C(=O)Nc2cnc[nH]2)C1 Cc1nn(C)cc1C(N1CC(CC(N2CC(CC3CC3)C2)=O)CC1C)=O c1(CC)ncncc1C(=O)NCC12CC1CN(C(=O)C(=Cc1cccnc1)C)C2 C(=O)(CCCC(N)=O)NC1(C)CCN(C(Cc2c(C)cco2)=O)C1 C(=O)(C(C(=O)NCC(CC)NC(=O)C(F)Cc1ccccc1)OC)OCC CC1(CNC(c2ccoc2CC(N)=O)=O)CCCN(C(C2CNC(=O)C2)=O)C1 CCCCCC(CC)C(=O)N1CCCC(C)(C)C1C(=O)NC(CO)CC(F)(F)F c1(C(N(CCC)CCNC(C2CCCC2(F)F)=O)=O)ccc2cc(O)ccc2n1 N1(C(C2(C(C)C)CCN(C(=O)CCOC3COC3)C2)=O)CCC(F)C(O)C1 C1(CC=C)(NC(=O)C=Cc2cc[nH]n2)CCCN(C(C2CCC3CC2CO3)=O)C1 N1(C(C2CCCO2)=O)CCCC2CN(Cc3nnc(-c4ccccc4F)s3)CCC12 C=CC1CN(C(=O)Cc2cn(C)nn2)CC1NC(=O)CN1CCCCC1=O N1(C(c2c(C)nc(C)o2)=O)CCCC(C)(CNC(=O)C(c2ccccc2)F)C1 C1(N(C(=O)CN2CCOCC2)C)CN(C(c2cc(C(C)(C)C)nn2C)=O)CC1F CCCCC(O)C(=O)N1CC(NC(c2cncc(C(C)(F)F)c2)=O)CC1(C)C c1(OC(C)C)ccccc1CC(=O)NCCN(C)C(C1C(C)(C)C1(C)C)=O CCC(C)C(C(=O)N1CC(OC(F)F)C1)NC(=O)Cc1cnsc1 c1(C(=O)NCC2CCC3CC23)ncccc1N(C(=O)CC(C1CC1)C1CC1)C1CC1 c1(COC)cnc(OC)c(C(=O)NC2CC(NC(=O)Cc3ccc(F)nc3)C2)c1 c1(CC2CCN(C(C=COCC)=O)C2)ccc(O)c(O)c1O CC(C)(C(=O)Oc1ccc(Nc2ccccc2)cc1)C(=O)NC1(C)CC(=O)NC1=O C12(C(=O)NCC3CC(NC(C4(CO)CCOC4)=O)C3)CC(C(F)(F)F)(C1)C2 N1(C(c2c(C)ocn2)=O)CC=CC1(C)C(N1CCC1(C)CC1CC1)=O c1(C(N(C2CCN(C(c3cc(C(N)=O)[nH]n3)=O)CC2)CC)=O)cc(Cl)c(Cl)[nH]1 CC(c1ccccc1Cl)=CC(=O)NC(CNC(c1c[nH]ccc1=N)=O)C(C)C C1(NC(c2c(SC)ccs2)=O)CCC2CC1CN2C(=O)CC1(O)CCCOC1 C=CCC(CC=C)C(=O)NC1CCN(C(c2c[nH]c(=N)nc2CC)=O)C12CCC2 C(N=c1nc2ncn(C)c2c(NCc2cccnc2Cl)[nH]1)c1cccc(C)c1F C1(COC)(CNC(C2CC23CC(O)C3)=O)CCCN1C(=O)C(C)(C)O c1(C(N2C(CCCOC)CCC2)=O)ccc(C(F)F)cc1 C(=O)(CC(C)C(=O)N1CC(CN(C)C(c2nc(-c3ccco3)sc2C)=O)C1)OC c1(C(=O)NCC2CC(NC(c3occc3C3CC3)=O)C2)ccc2[nH]nc(O)c2c1 C1(NC(CC(CC)C2CC2)=O)CN(C(c2nnn3c2CSCC3)=O)CC(C)(C)C1 CC1CN(C(c2sccc2Cl)=O)CCC1NC(=O)Cc1cnn(C(F)F)c1 N1(C(C=C(CCC)CCC)=O)CCN(C(c2[nH]ccc2C2CC2)=O)CC12CC2 C1(C)(C(N(CCC(N)=O)CC)=O)C=CCN1C(=O)C(C)OC CCCCC(C)CCC(=O)NCC1C=CC(NC(c2ccoc2Br)=O)C1 c1(OCCN(C)C)cccc(F)c1.C12COCC1C(=O)NC2 c1(OC)nccc2c(C(=O)NCCCCNC(c3cc(C#N)n(C)n3)=O)c[nH]c12 N1(C(Cc2c(C)ocn2)=O)CCC2(CC1)CN(C(=O)C1=NOC(C)C1)CC(C)O2 c1(-c2cc(NC(N3CC(C)N(C)CC3)=O)on2)ccc2c(c1)OCCO2 N12CCC(C1)N(C)C(=O)NC(C)CC2=O.C1CCCO1.C(C)(C)(C)OC(C)=O Cn1nnc2cc(C(N3CCCC3(C)CNC(=O)CC3CC4CC4C3)=O)ccc12 c1(C(C)C)ccc(C(=O)NCCCC2CCCN2C(c2ccc(Cl)s2)=O)c(O)c1 N1(C(C(COCC)F)=O)CC(CO)CC1Cn1cc(C(O)C2CC2)nn1 c1(C(N(CC(=O)NCC(COC)C)C2CC2)=O)conc1C1CCC1 c1(CNC(CC2OCCN(C(C(C)(C)CCl)=O)C2)=O)ccc2ncnn2c1 CC1(NC(C2CC2C(=O)NCCC2CC2)=O)CN(C(N)=O)C1 C#Cc1nc(C(=O)NCC(C)(C)CN(C)C(c2cc(C(N)=O)no2)=O)cs1 CCC(CC(=O)N1CCN(C(c2cc(C)nc(O)n2)=O)C(CF)C1)C(F)F CC(C)CC(CNC(=O)CN1CC(=O)NC1=O)NC(c1cnn(C)c1Cl)=O CC(C(=O)N)C(=O)NNc1nc(Cl)c(C#N)n1C.n1(C)cncn1 c1(C(=O)NCC(CCCC)NC(c2ccoc2CCC)=O)[nH]cc2c1CCC2 C(=O)(C(C)(CCC)CCC)N1CCC(NC(CCC#CC)=O)C(C)C1 N1(C(Cc2c(C)nsc2)=O)CC2CCCN(C(C3CC4C=CCC(C3)C4)=O)C2C1 CC1(C)C2CCC1(CC(=O)NC1C3CN(C(C4(C#N)CCC4)=O)CC13)CC2 C1(CNCC2CC(C(F)(F)F)OC2)CC12CCCCC2 C(c1cnn(C)c1)=C(C(=O)NC1CCC(CNC(c2c(CCC)[nH]cc2)=O)C1)C c1(CCC(=O)NCCOCCC(=O)N(CC(C)C#N)CC)nc(C)cs1 C(CC1=CCN(C(c2ccnn(C)c2=O)=O)CC1)NC(C1C(C)CSCC1)=O C1(N(C(CCn2cc(CC=C(C)C(F)F)nn2)=O)CC2CC2)CC2(C1)CC(C)C2 c1(CN2CCCC(C(=O)Nc3c(C)cc(Br)cc3F)C2)cccc2c1cnn2C C1(C(=O)NCC2CC(O)(CNC(c3cc(C)[nH]c3C)=O)C2)CCCCC1(C)C C1(COC)CN(C(c2ccccn2)=O)CCC1NC(c1ccc(SC)o1)=O C=C(F)CN=C(NC1CCC(C(N2CCOCC2)=O)CC1)NC1CN(CCOC)C1 NS(=O)(=O)c1c[nH]c(C(=O)NC2CC(C(=O)O)C2)c1 c1(C(=O)NCCCNC(C2CC(C)(F)C2)=O)cccc(N=S(C)(C)=O)c1 c1(OC)ccc(C(=O)NC2CCCC(N(C(=O)CC3CCSCC3)C)C2)c(C)c1 C(C(C)(C)CC(=O)N1CCC2(CC2C(=O)NC2(CF)CC2)C1)N(C)C C(=O)(C1CCc2c[nH]nc21)NC(CNC(C(=Cc1ccccc1)CC)=O)C C1(NCC=CCNC(CN2CCC(OC)C2)=O)CCC(F)(F)CC1 N1(C(c2c(NC)cccc2F)=O)CCC2(C(=O)NC(C)C(=O)OC)CCCC12 CC1CC(NC(C23CC(c4nc[nH]n4)(C2)C3)=O)CN1C(=O)Cc1cnc[nH]1 C(CCC(O)C(=O)N1CC2C(C1)C2(C)C)NC(c1nc(OCC)oc1)=O N1(C(Cc2n(C)nnc2)=O)CC2CCC2(NC(=O)CNS(C)(=O)=O)C1 CC(C(=O)N(CC(=O)N(C1CC(Nc2ccoc2)C1)C)C)c1cccs1 c1(C(=O)NCC2CN(C(CCCCN(C(C)=O)C)=O)C(C)C2)cc2cc[nH]c2cn1 c1(N(C2CC3CNC2C3)C(C(C)NC(C)=O)=O)cccc(N2CCOCC2)c1 N1(C(c2n(C)ccc2)=O)CCC2C(C(=O)NC3CCCN(O)C3=O)C2C1 C(=O)(C1=CC2CCC1C2)NC1CN(C(CC2CCC(=O)N2)=O)C(CO)C1 c1(C(=O)NC2C(NC(c3cn(C)c(=O)cn3)=O)CCC2)c[nH]c2ccccc12 c1(C(=O)NC2C(C)N(C(C3CCNC(=O)C3)=O)CC2)cc2c(ccn2C)s1 C(CCC(O)C(=O)NCC(C)(C)CC(F)F)NC(C(C)=NOCC#N)=O c1(C(=O)OCCC2CC(C)CC(C)C2)c(F)cc(F)cc1Br Nc1cc(F)c(C(N2CC(C3(NC(c4ccc(F)c(F)c4)=O)CC3)C2)=O)cc1F N1(C(Cc2c(C)n(C)cn2)=O)CCCC(C)C1CCNC(=O)CCN1CCCC1 c1(C(N2CC(NC(CC(CC)CC)=O)C(O)C2)=O)c(F)cc(C)cc1Br c1(CC)cc(C(N2CCC(COC)(NC(=O)CC(C)(C)N(C)C)C2)=O)cc(O)n1 C1(CC=C)CCCCN1C(C1C(C)CN1C(=O)C=CCC)=O C1(C(=O)NC(C)CC(=O)NCCC(=O)NCCO)CC2C=CC1C2 c1(OCC(=O)NCCCCNC(C2N(C)CC2)=O)ccccc1C#N Cc1c(F)ccc(C(N2CC(C3(NC(=O)CCC4CC4(C)C)CC3)C2)=O)c1C C1(CC=C)(NC(c2cnn(CC)c2C)=O)CCN(C(=O)C(C)S(C)(=O)=O)CC1 CCC(CC)C(C(=O)N1CC(C(=O)NOC(C)(C)CO)C2(CCC2)C1)OC C(=O)(CCCCCCSC)N(CC(CC)NC(c1cccc(C2CC2)c1)=O)C CCC(O)CC(=O)NC1CCC1NC(c1ccc(-c2ccc(C)cc2)cc1)=O CCC(COc1ccc(OC(=O)C(C)S(N)(=O)=O)cc1)(CC)CC C1(CNC(COC(C)=O)=O)CN(C(C2CC2CN(C)C)=O)CCN1C C1(NC(C2CC=C(C)CC2)=O)CCN(C(=O)Cc2ccn(C)n2)CC1F C=CCC(CC(=O)NCC(C1CCCC1)C)NC(=O)CS(C)(=O)=O N1(C(C(CC(C)C)(C)O)=O)CCCC(C2(NC(c3nn(C)cc3Cl)=O)CC2)C1 c1(C(C)C)c(C(=O)NC23CC2CN(c2cc(F)ncn2)C3)cnn1CCO c1(CCCO)nc(CC2CCCC2(F)F)n(-c2ccccc2)n1 C(C(C)(CC(C)C)NC(c1ccc(C)cc1C)=O)NC(CC=C)=O CC1CCC(C(C)Nc2ccc(C3(O)COC3)cc2)CC1 C1(F)(C(N(CC(C)NC(=O)C(c2ccc(Cl)cc2)(C)O)C)=O)C(C)(C)C1(C)C C(CCC)(C(=O)NC(C1CCN(C(c2ccc(C(C)C)cn2)=O)CC1)C)=CCC N1(C(C(CC)C(C)O)=O)CCCC(C2CCN(C(C3COCCN3)=O)CC2)C1 c1(C(=O)NC2CCN(C(C(CCC)OCC)=O)C(C)C2)cccc2cccnc12 Cc1nc(C(=O)N(CCC#N)C(C2CCCC2(C)C)=O)nn1-c1nc[nH]n1 C1(C(=O)NC23CC(C2)C3)(CC)CCCN(C(=O)CC2CCCOC2)C1 C(CN=C(NCC(CC1CC1)OC)NC(C)(C)COC)c1c(OC)cccc1 C(=O)(CCCCCc1cccc(O)c1)NCC1C(NC(C=C(C)C2CC2)=O)C1 c1(C(=O)NC(CC)(C)CNC(c2nsnc2O)=O)cc2c(cc1C)OCO2 C(C)(C)(CC(F)C(=O)NC1CN(C)CC1(C)C)NC(c1c(NC)nccc1)=O C(=O)(CC(F)(F)C(F)F)N(CCCNC(=O)CCC(F)(F)F)CC c1(OC)cccc(C(=O)N(CC(C)C(=O)N(C)C(c2nc(C)no2)C)C)c1 C(=O)(C1=COCCC1)NC(C)=O.C1(=O)CCC(C)NCCN1C c1(CCC(=O)NCC2CN(C(CSC)=O)C3C2C3)c(C)nc(O)nc1O C1(C(=O)NCC(CN(C)C(N)=O)O)CCCN(C(=O)CCOc2ccsc2)C1 c1(CC(=O)NC2C(NC(CC3ON=C(CC)C3)=O)C2)ccnc2ccccc12 CCC(CC(=O)N1CCC(C(=O)NCC(F)C(C)(C)O)(CC)C1)CC(C)C c1(C(C)=O)cccc(Cl)c1.c12nc(cs1)C(C(=O)NC1CC1)N(C)C2 N1(C(C2(C#C)CN(C(=O)C(O)CCSC)C2)=O)CCC(CO)C(O)C1 Cc1sc(Cl)nc1C(=O)NC(CNC(c1cc(C2(C)CC2)on1)=O)C(C)C c1(CCC)ccc(O)c(C(=O)NCC2CCCN(C(=O)C(=O)NCCC(N)=O)C2)c1 c1(OC)cc(-c2cn(C(C)C(=O)N3CCC(SC)C3)nn2)ccc1O c1(C(=O)NC2(CC(=O)Nc3ccc(Cl)nc3Cl)CCC2)ccc(F)c(Br)c1 C1(NC(c2c(C)oc(Cl)n2)=O)CCN(C(=O)CCC(C)(C)C)C(C2CC2)C1 C(=O)(CCC(F)(F)C(F)(F)F)NCC1N(C(=O)C(O)CC2CC2)CCN(C)C1 N1(C(c2nnc(C)s2)=O)C2CCC1CC(CNC(c1ncc[nH]1)=O)C2 C1(C(=O)NCCN(C(=O)CO)C)CCCN(C(c2ncccc2CO)=O)C1 C=CCCC(C(=O)NC1CCOC1)NC(=O)CC1(C)CC1 N1(C(CSC(C)C)=O)CC(C)CN(C(c2ccc(F)cc2Cl)=O)C(C)C1 C1(C(=O)NCC(C2CC2)NC(CC2CCC(=O)N2)=O)CN2CCC1CC2 C(=O)(CCCCC(C)C)NC(CC=C)CNC(=O)Cc1nc(C2CC2)cs1 C1(CC=C)(NC(c2cnc[nH]2)=O)CCCN(C(c2cnc(C(F)F)cn2)=O)C1 CC(C)CC(C)(C)NC(=O)NC(C)CC1CCCCO1 Cc1ccncc1CC(=O)NC1CCC(Nc2ncccn2)CC1 C1(NC(C(C2CCN(C(=O)C3=CCCOCC3)CC2)C)=O)CC2(CCCO2)C1 c1(C(=O)NCC2CC(F)(CNC(C3(C)C=CCC3)=O)C2)cccc2nc(O)oc12 C12CC(CO)N(C1)C(=O)CO2.c1(CNC(C=C(C)C(C)C)=O)ccncc1 C1(O)(CCNC(CSCC#C)=O)CCCN(C(c2nocc2C(C)C)=O)C1 c12cccc(c1)C(=O)N2.CC(C)(COCCNC(=O)COCCO)CS(C)(=O)=O C1(C(=O)NCC(O)CNC(=O)C(C)SCC)(NC(=O)OC)CCCC1.C(C)(C)(C)O Cc1cc(C)c(C(N2CCC3CC23C(=O)NCc2nccn2C(C)C)=O)cn1 c1(C(=O)NCC2(COC)CCCN2C(=O)CNS(N)(=O)=O)ccc(F)c(O)c1 C12(C(=O)NC(CNC(=O)C(F)CC3CCCC3)C3CC3)CCC(CC1F)C2 C1(C#CC(=O)N2CCCC(CCNC(C3(C)CCCOC3)=O)C2)(CC)CC1 c1(C(N2CCCN(C(c3c(CC)occ3)=O)C(C)C2)=O)ccc2nc(O)oc2c1 c1(CNC(N(CC)Cc2cccnn2)=O)c(F)c(F)c(N)c(F)c1F N1(C(=O)NC(C)C=CCCc2ccccc2)CC2(CCCO2)C1 N1(CC)CCCC(C(N2CC(C(=O)NC(C)CCO)(SC)C2)=O)C1 Cc1ccc2c(C(=O)N(CCCCN(c3cncc(Cl)n3)C)C)cnn2c1C c1(C(=O)NCC(C2CC2)NC(=O)CC2(O)CCC2)ccn2c1CSCC2 c1(C(N(CC(=O)NC(c2cn(CC)nc2)C)C2CC2)=O)ccncc1Cl C(CC(C(=O)N1CC([N+](=O)[O-])C1)NC(=O)CC1(N(C)C)CC1)SC n1(CC)nc(C)c(C(N2CCOC(C)C2c2nnc(C)o2)=O)c1C(F)(F)F C1(C#N)(C(N(C2CN(C(c3cnc(C4CC4)o3)=O)C2)C)=O)CCOCC1 N(C(=NCCC1(C(=O)N(C)C)CCOCC1)NCC1CCCO1)C1C(C)C1 C1(C(=O)OC)CC(C)N1C(c1cnn(CCNC(C2CS(=O)C2)=O)c1)=O C(=O)(CCCCCn1cc(-c2cccnc2N)nn1)C(=O)C(c1ccccc1)F N1(C(C(N2CCCC(OCC(=O)NC)C2)=O)=O)CC2(CCOCC2)CC1C C12CN(CCO1)C(C)c1nc(co1)C(=O)NCC2.C(=O)(C1=CCCC1)N(C)C c1(N)cc(I)ccc1Cl.C1(C(=O)NCCOC)COCCN1Cc1ccccc1 C(=O)(C(F)CC(C)(C)NC(c1cn(C)c(C)n1)=O)NC(CC=C)CC C(CC(C(=O)NCCn1cnnn1)NC(c1n[nH]c(C)c1Cl)=O)=CC c1(CN2C(C)(C(=O)Nc3ncc(Br)nc3I)CC2)c(F)cc([N+](=O)[O-])cc1F c1(C(=O)NC2CCC(NC(C(C)CC(N)=O)=O)C2)ccc2nc(C3CC3)cn2c1 c1(C2C(C)CCO2)c(Oc2cccc(Cl)c2)ccc2ccccc12 c1(C(N(C)CCNc2nccc(C3CC3)n2)=O)ccc(CO)c(F)c1 c1(CC)c(C(N2CCCC2C(C)(C)C(=O)NCC(C)O)=O)nnn1C CCCC(C(=O)N1CCOCC1)NC(C1CN(C2CCC2)C1)=O C1(C(N(CCCCNC(C(c2ccc(C)s2)C)=O)C)=O)CCc2n[nH]cc2C1C Cc1cccc(C(=O)Nc2ccsc2C(N2CCOCC2CC(C)C)=O)c1C Cc1ccc(Br)cc1C(N1CCCC(C(N)=O)C1)C(=O)NCC1CC1 C(=O)(C#CC(C)(C)O)NC(C(C)NC(c1cn(C(C)C)nc1)=O)C(C)C c1(C(N2CC(OC)(CNC(C3CCCC3C)=O)C2)=O)coc2c1CCCC2 N1(C(c2cnc(=N)[nH]c2)=O)CCC2(CC1)CCN(C(c1cccnc1Cl)=O)C2 c1(-c2nc(-c3cccc(Cl)c3)oc2)ccc(F)c(F)c1.c12ccc(s1)NC2 CCC(CC)C(C)C(=O)NCC(C1CCCC1)NC(c1cc2c([nH]1)CCCC2)=O N1(C(c2cccc(CCC)c2)=O)CCN(C(=O)C(F)CC2CCCC2)CC(O)C1 C(=O)(C(COCC)NC(=O)CCn1ccnc1)N(C1CCN(CC)C1)C(C)C.O.C c1(C(=O)NCCN(C(CC(COC)C)=O)CC2CC2)cc(Br)ccc1OC c1(CC)ccc(C(=O)NCC2CC(O)CN2C(=O)CCCOCC=C(C)C)cc1 N1(C(c2ccc(C#N)cc2)C(=O)NC2CCC2)CC(=O)N2CCCCC2C1 c1(C(=O)NC(C(C)NC(Cc2cc(OC)nn2C)=O)CO)ccc(CO)c(F)c1 CC1CN(C(C2CC(C(C)(C)C)C2)=O)CC1(C)CNC(c1ccsc1)=O n1(CCC)c(N2CCN(CCN3CC(O)CC3=O)CC2)nnc1-c1cc(Br)cn1C N1(C(C(C(=O)OC)CC)=O)CCC2(CC1)CN(C(c1ccoc1OC)=O)C2 C(=O)(CCC(C)(C)[N+](=O)[O-])N(C1CCN(C(c2c(OC)c(Cl)ccc2)=O)C1)C C(=O)(C(C(C)(C)CC)OC)N1CC(O)(CNC(c2n(CC(=O)OC)ncc2)=O)C1 CN1C(=O)CC(C(=O)Nc2ccccc2NC(=O)CSC(F)F)C1c1ccccc1 CC1(C)CN(C(=O)CC2(O)CCOCC2)CCC1C(=O)NCCCOC(=N)O N1(C(Cc2ncc(C)s2)=O)CC2(CCC2C(=O)Nc2cccc(N3CCCC3)c2)C1 c1(C(N2CC(CNC(CCC(C)SC)=O)C(C)C2)=O)ccc(CN(C)C)c(F)c1 C#CCCCC(C)C(=O)NC(CCC1CCC1)C(=O)NCC(C#N)CC c1(C(=O)NCC(CCNC(C(C)=C2CCC2)=O)O)c(Br)ncn1C CC(CC(=O)NC1C=CCCC1)C(C)(C)NC(C12CSCC1C2)=O Cc1cc(C(N2CC(CNC(C3(O)CCCCC3)=O)C3CC23)=O)c(C)n1C Cn1ccc2cc(C(N3CCCC3CNCC3COC4(CO)CC3C4)=O)ccc12 c1(C(N2C(Cn3cc(C(C(C)C)O)nn3)CC2)=O)nn(C)cc1N N1(C(C2CCCCN(C(C(N3CCCC3=O)C)=O)C2)=O)CC2(CC(CO)CO2)C1 Cc1ccc2c(N3CCC(F)(F)C3)nc(=NCC3CCC4(CCC4)O3)[nH]c2c1 C1(NC(c2ccc(CC)s2)=O)CN(C(c2cc3ccoc3s2)=O)CC(F)(F)C1 c1(OC)cc(C(=O)NCCc2cn(CC3CC(F)(F)C3)nn2)cnc1OC C1(NC(C(C)NC(CCCC)=O)=O)CN(C(=O)CSC2CCCCC2)CCC1O C1(CC)C(C(=O)NC2(CO)CC(O)C2)CCCN1C(=O)C(C)CSC c1(OC)ccc(C(=O)NCC2CCCN2C(=O)C(c2ccccc2)OC)cc1N C1(N(C(CSCCC(C)C)=O)C)CCN(C(c2ccoc2)=O)CC1C C(=O)(C(C)(O)C(F)(F)F)N1CC2C(CNC(c3ccc(C(C)C)nc3)=O)(C2)C1 CC(C)CCCCC(=O)NC1(C(=O)NC2CCC3CCC23)CSC1 C1(C)(CC(N2C(C(=O)NC(c3ccn(C)n3)CC)CC2)=O)CC2(CCC2)C1 N1(C(c2cncc(SC)c2)=O)CCC2(CCC2NC(=O)Cn2nnc(C)n2)CC1 c1(NCC2N(Cc3cc(O)c(O)c(O)c3)CCOC2)ncnc2[nH]ccc12 C#Cc1cc(F)c(C(=O)NCCCOCCN(C(=O)C(N)=O)C)c(F)c1 C1(=O)C(C(C)C)N(CC)CC(C)N1.C1(C)(NC(=O)NC)CCCC1 N1(C(C23CC(COC)(OC2)C3)=O)CCCN(C(c2cnns2)=O)C(C)C1 C(=O)(C(CCSC)N(N1CC(O)(NC(=O)Cc2nc(Br)cs2)C1)C(C)=O)OCC c1(C(N2CCC(CNC(c3c(COC)ncs3)=O)C2)=O)cc([N+](=O)[O-])ccc1C c1(C(=O)NCC(CNC(C2(C)CC=C(C)CC2)=O)O)coc2c1C(O)CCC2 C12(C(=O)NC(CC)CNC(C3CCCN3C(=O)NC)=O)CCCC1CCC2 C1(CNC(c2c(-c3c(C)cccc3)cccn2)=O)C(C)CCCN1C(=O)C=CCF N1(C(c2c(NC)c(F)ccc2)=O)CCC2CCCN(C(=O)C3=CCCCO3)C2C1 C1(C2CCC2)(C(N2CC(O)(CNC(C(c3ccccc3)OC)=O)C2)=O)CC1(F)F c1(OC)ccc(Cl)c(CC(=O)NCC(C2CCC2)NC(C2CC2F)=O)c1 Cc1cccc(COCCOCC(=O)N)c1.C1CC(=O)NCC(C)S1.C(CO)O C(=O)(C1=NOC(C)C1C)N1C(CC)C(NC(c2ccnn2C(C)C)=O)CC1 c1(NC(C2CN(C(c3ccc(C)cc3F)=O)CC(F)C2)=O)cnc(Cl)c(Br)c1C C1(C(C)C(=O)NCC2(O)CCN(C(=O)CC3CSCCS3)C2)CCC(C)(C)CC1 C#CC(C)(C)C(=O)NC(C)CNC(=O)CCc1cccc(SC)c1 c1(NCC2(OC(C)C)CCOC2)cc(=NCCc2nc[nH]n2)[nH]c(C(F)(F)F)n1 C#CCC(O)C(=O)NC1CC1CNC(=O)Cc1csc(-c2ccc(Cl)cc2)n1 CCC1=C(C(=O)NC2CCC(C(=O)NCC3CC(C)=NO3)C2)CCCO1 c1(C(=O)NCC(C2CCOC2)NC(c2cc(OC)n[nH]2)=O)c(OC)ccc(F)c1N C#Cc1cc(NC(=O)C(=O)NCc2ccc(O)nn2)cc(F)c1 Nc1ccc(Cl)nc1C(=O)NCCCCCCNC(C1CC(CC2CC2)C1)=O C1(C(=O)NCC2(F)CCN(C(CCSC)=O)C2)CCC(NC(=O)OC(C)(C)C)CC1 N1(C(C2(C)CC(=C)C2)=O)CCC=C(C(=O)N2CCCC(OC)CC2)C1 c1(C(=O)NCC(CN(C)C(C2CCOC2C2CC2)=O)O)ccc(S(N)(=O)=O)c(F)c1 C1(C(N(C(CNC(=O)CCCCO)C2CC2)C)=O)CC(=O)NC1(C)C N1(C(C)=O)CCC(CC(=O)NC2CCN(C(=O)Cc3ccoc3)C2CC)CC1 C1(C(N2CCC(C(=O)NCC(C)C)C2)=O)Cc2n[nH]cc2C(N)C1 C1(C[Si](C)(C)C)CCC(N=c2nc(-c3cc(Cl)cc(Cl)c3)[nH]o2)C1 CC1CN(C(=O)C(F)C(C)(C)O)CCCN1C(c1cc(Cl)n(C)n1)=O CCCC(C)CC(=O)NCC(C1CCCCC1)CNC(C12CC(C1)C(C)O2)=O N1(C(C(C2CC2)OCC)=O)CC2(CCC2NC(c2ccc(OC)s2)=O)C1 c1(OC)cncc(C(N2CC=CC2CNC(=O)CCOCC(F)(F)F)=O)c1 S(=O)(=O)(c1cccc2c1OCCCO2)NC(c1ccc(=NC)[nH]c1)=O C(C)(C(F)(F)C(F)(F)F)=CC(=O)NC1C(C(=O)NCC(COC)CO)C1 Cn1cc(C(=O)NC(CNC(C2(S(C)(=O)=O)CCC2)=O)CO)n(C)c1=O C(=O)(CC(CC)CC(C)C)NC(CC)CNC(C1C=CCN1C(=O)OC)=O c1(C(N(C)C)=O)n[nH]c2cccc(-c3ccc(C4(C)OCCO4)cc3)c12 N1(C(C2(C)CC2)=O)CCN(C(C23CCCC(C2)OC3)=O)C(Cc2ccccc2)C1 CC1=NOC2(C1)CC(C(N1CCC(NC(=O)Cc3cncc(C)c3)C1(C)C)=O)C2 c1(C(=O)NCC(CC)NC(=O)C(F)(F)C2(O)CCC2)ccc(COC)s1 C1(NC(CCOC)=O)CCCC1NC(=O)COCC1CCC1 Cc1cc(C)c(CC(=O)NCC(C2CCCN2C(=O)COC(F)(F)F)(C)C)c(O)n1 c1(C(=O)NC2C(NC(CCc3cc(C)on3)=O)COC2)cnc2[nH]nc(O)c2c1 CCC(CN(C)C)C(=O)NC1CC(C(C)(C)O)C1.C12CCCC1CC(=O)N2 CC(C)(CO)CC(O)CC(C)C(F)(F)F.N1CCCC1 Cc1cc(CCC(=O)N(C2CCCN(C(=O)C(N3CCSCC3)C)C2)C)n(C)n1 Cc1ncc(C(=O)NC2CC(C(N3CCC(CC(N)=O)C3)=O)C2)cn1 N1(C(c2c(CC)nc(C)cc2)=O)CCN(C(=O)C(CN(C)C)N(C)C)CC(C)(C)C1 CC(C)C(C(=O)NCC1CCC1NC(=O)CSS(C)(=O)=O)NS(N)(=O)=O N1(C(c2ccc(CC)cc2)=O)CC(C)N(C(=O)CCCCC(C)C)CC1C N1(C(C=CCCC)=O)CCN(C(=O)CCN(CCC2C(=O)N2CC)CC)CC1.OC.CC c1(CC(N2CC(CN(C)C(C3CN(C)CCO3)=O)C2)=O)cc(F)ccc1Br CC1(CNC(=O)CCN2CCOCC2)CCN(C(c2cnc(C3CC3)s2)=O)C1 c1(C(=O)OCC)cccc(NC(=O)NCC(C)NC(C2CC=CCC2)=O)c1 C1(NC(C=Cc2n(CC)ccn2)=O)CN(C(C2CCCCC2(C)C)=O)CCC1O N1(C(C(F)=CC)=O)CC(NC(c2ccc(-c3ccco3)o2)=O)CC1C C(N=c1nc(N2CCC(C(N)=O)C2)c2c([nH]1)CCC2)C1(C(C)(C)C)CCCC1 C(CC(=O)NCC1(C)CCN(C(c2ccc(CO)cc2)=O)C1)(C(C)C)OCC C1(CC)CN(C(=O)CCc2nc(C(C)(C)C)no2)CCN1C(=O)C1=COCCO1 N1(C(CCc2cc(C)on2)=O)CCC(C)(CNC(=O)Cc2ccc(Br)cn2)C1 n1(CCC)ncc(C(=O)NCC2CN(C(c3cc(F)cs3)=O)C2)c1C C(=O)(C1=NN(C)C(=O)CC1)N1C(CC)C(NC(c2cncn(C)c2=O)=O)CCC1 c1(C(N(CCCNC(c2[nH]cc(C(=O)OC)c2)=O)C)=O)cnnc2ccccc12 c1(C(=O)OC)ccc(Nc2ncnn2C)c(CNC2CCCN(OC)C2)c1 N1(C(c2c(N)cnc(Cl)c2)=O)CC2CCCN(C(c3cnn[nH]3)=O)C2C1 C1(CC(=O)NCC2=C(C)CC2)N(C(C2CCN(C)C2C)=O)CCC1(C)C C1(C(N2CCC(C(C)C(=O)NC3CCCC3CCO)CC2)=O)CCS(=O)CC1 N1(C(=O)NC(C2C(c3ccc(C#N)c(Cl)c3)C2)C)CCN2CCCC2C1 CC(Cc1ccccc1)C(=O)NCC(F)CNC(C1CN(S(C)(=O)=O)C1)=O c1(C(=O)NC(C2CCN(C(c3c(C)ccc(O)c3)=O)C2)C)c[nH]c2cccnc12 CC(F)(F)C(C)(C)CN(C(=O)C(=O)NC1CC1)CC1CCC(=O)N1C1CC1 CCCC(CCC)=CC(=O)N(CCNC(=O)Cn1nccn1)CC CC1(C)CCCN(S(=O)(=O)N2CCC(F)(F)CC2CN2CC3(CCC3)OCC2CO)C1 CC1CCC(CNC(c2nccnc2C(F)(F)F)=O)N(C(c2csc(=N)[nH]2)=O)C1 C1(c2n(CCCSC)nnn2)(Oc2ccccc2)CCOC1C.C1(N)CC2CC2C1 O=C(C)C(S(=O)(=O)N1CC(c2ccc(F)c(F)c2)C1)c1cccc(F)c1 CON(CCC(=O)Nc1cc(OC)ccn1)C(=O)C1=C(C)CCCC1 C(=O)(C(CC1CCOCC1)NC(=O)CC1CC1CC)N(CC=C)CC1CCCC1 C(=O)(CC(C(F)(F)F)NC(c1csc(O)n1)=O)NCC(COC)OC N1(C(C(CCC)C#N)=O)CCCC2C1CCN2C(=O)CC=Cc1ccccc1F C1(CCC)CN(C(C2CC(F)(F)CS2)=O)CCN1C(=O)CCC12CCC(CC1)C2 C1(NC(CSCCCC)=O)CCC12CN(C(c1ccco1)=O)C2 c1(OCC)ccc2c(c1)C(O)CC2.C12(C)CC(N(C)C)C1NC(=O)C(=O)N2 c1(NC(C(CCC#C)NC(=O)Cc2nc(=N)[nH][nH]2)=O)cccc2c1CCO2 N1(CC2CCC(F)C2)C2CCCC1CC(O)C2 c1(COC)cnc2ccccc2c1Br.C1(OC)CCN2CC12 Cc1cc2sc(NC(=O)NCC=Cc3ccc(F)cc3F)nc2cc1F N1(C(c2c(C(C)C)nns2)=O)CC2CCC1CN2C(c1cnc2ncccn12)=O C1(C(=O)NC(CC#C)CC#C)CCN(C(=O)C(CC(=C)C)OC)C12CCC2 N1(C(CCC2N(C(c3cnc(COC)s3)=O)CCC2)=O)CCC(CO)C(C)(C)C1 N1(C(c2cccc(CC=C)c2)=O)CCC12CN(C(C1CCN(C)S1(=O)=O)=O)C2 C#CC1CCN(C(=O)C(F)C2CC(NC(C3(N(C)C)CC3)=O)C2)C1 C(=O)(C(CCOC1(C)CC1)N1CCC1(C)c1ccccc1)NC C(=O)(CC(C)C(C)C(C)C)N1CCC(CNC(c2c(CC)scc2)=O)C(C)C1 c1(C(=O)NCC(C)N(C(C(C2CCC2)OC)=O)C)c(C)cncc1F C1(CNC(c2ccncc2)=O)CC(F)(CNC(C23CCC2CC3)=O)C1 c1(OC)ccc(C)c(NC2(CC(=O)NCc3cc(C(C)(C)C)no3)CCC2)c1 C(=O)(C1=CNC2=NCCCN12)N1CC(CN(C(=O)C=CC(C)(C)C)C)OCC1 c1(C(=O)NC2C3(CC(C(=O)OC)C3)CC2)cc(Br)c2c(c1)[nH]c(=N)n2C c1(CN(CCN(C)C)C(c2cccnc2N2CCCC2)=O)cccc(C(=O)O)c1 C1(O)(CCNC(C=CC(C)C)=O)CCN(C(C2CCN(CC(C)C)C2)=O)C1 C1(OC)CC(NC(=O)CCc2cc(C)on2)CN(C(C2CC(C)(O)C2)=O)C1 C1(C(N(C(C)C)CCN(C(=O)CN(C)CCO)C)=O)CCOC1C(F)(F)F C(C(C(C)(C)C)NC(=O)CC(C)O)NC(C1N(CC)CCC1)=O C1(C(=O)NCC(C)=CC(=O)NCC2CCC(=O)O2)CC12CCCC2 Cc1ccc2cc(C(=O)NC(C)(C)CN(C(=O)C=Cc3cn(C)nn3)C)[nH]c2c1 n1(CC(N2CC(CNC(c3cc(C)on3)=O)C(O)C2)=O)ccc(=O)n(C)c1=O c1(C(N2C(CNC(C(CC3CC3)NC(C)=O)=O)CC2)=O)ccc2c(c1)CCC(=O)N2 c1(CN(C(c2n(C(CC)C)ncc2)=O)CCOCc2ccoc2)ccc(Cl)nc1 C1(c2n(C)nnn2)(NC(C2CC2)C2CC2)CC2(CCCOC2)C1 CCCCC(CC)C(=O)NCc1occc1C(=O)NCC(CC)n1cccn1 c1(CC(N2CC3C(CNC(c4c(C)ncnc4)=O)C3C2)=O)cccc2c1OCO2 N1(C(c2ccc(C(C)(C)C)[nH]2)=O)CCN(C(=O)C2=C(Cl)CCOC2)CC(O)C1 C(=O)(C1CCCn2c(Br)cnc21)NC(C)CN(C)C(c1cc(F)ccc1O)=O N#CC1CN(c2ncc(I)cn2)CCN1c1ncncc1F C=C1c2ccccc2C(=O)N1CC(N1CCC(C)S(=O)(=O)CC1)=O N1(C(C=CCN(C)C)=O)CCN(C2CCN(C(c3csnn3)=O)C2)CC1 CCCCCCC(C)C(=O)N1CC(CNC(c2cc(C)on2)=O)C(C)C1 C(=O)(C(F)C(C)(F)F)NCC1(COC)CCCN1C(c1cccc(C(C)C)n1)=O O=C(CC(C1=CCCCCCC1)N(C1CC1)Cc1ccsc1)OCC(F)F c1(CN2CC(C)N(C(c3cc(CO)ccc3O)=O)CC2)ccc(Br)c([N+](=O)[O-])c1 C1(NC(C2CC=CC(O)C2)=O)CCC(=O)NC1C.C12(O)CN(C1)C(=O)C2(C)C C1(OC)CC2(C1)CC(C(=O)NC1CN(CC3CC34CC(O)C4)CCC1C)C2 c1(C(=O)NCc2ncccc2C(N2CCCC(O)C2)=O)cnc2c(Cl)cccn12 C1(NC(CN)=O)CCN(C(=O)CCOc2ccc(CC(=O)C(C)=O)cc2)CC1F.OC C1(COC)(NC(c2ccc(OC)s2)=O)CCCN(C(=O)C(C)SC)C1 C1(NC(c2cc(OCC)c(OC(F)F)cc2)=O)CC(C)(C)NC(C)(C)C1 c1(C(=O)NCC2COCCO2)cccc(N2CC=CC2)c1 N1(C(C(c2c(C)noc2C)C)=O)CCC(NC(c2ccn(C)n2)=O)C(C)(C)C1 N1(C(c2nc(CCCC)sc2)=O)CC(CNC(=O)C(C)(C)OC(C)C)CC1C C1(OC)CC(C)CN(C(c2cc(C3CC3)oc2C)C(=O)NC(C)(C)C)C1.C(=O)OC C1(CN(C)C(C2(CO)CC2)=O)CCCCN1C(=O)CCc1cccnc1Cl C1(C(C)C)CN(C(c2cc(Br)n(C)n2)=O)CCN1C(C1CCCCO1)=O n1(CC)nc(C(=O)NCC2CC(C)N(C(=O)Cc3ncoc3C)C2)cc1C Cc1ccc2cc(CN3CCNC(=O)C3)sc2c1.c12cc(F)ccc1CC(=O)N2 c1(C(=O)NCC2CC(F)(CNC(C(C3CC3)OCC)=O)C2)cn(C)nc1O C(CC)(C(=O)NC(C)CNC1(OC(C)=O)CCC1)=CCCC C1(CC=C)(C(=O)N(C)Cc2cc(C)ccn2)CCCN1C(=O)C(F)F C1(C(N(CCNC(=O)CSc2cccc(Cl)c2)CC)=O)CCCCC12CCC2 N1(C(C2(CC)CCCCO2)=O)C2CCC1CC(O)(CNC(=O)C(O)c1cnc[nH]1)C2 c1(C(=O)NCC2(OCc3ccccc3)CN(C(COC)=O)C2)ccc(C)nc1O CC1=NOC(C(=O)NCCOCCCN(C)C(c2ccncc2Cl)=O)C1C N1(C(c2ncc(C)[n+]([O-])c2)=O)CC2(CCOCC2)C1c1cn(CC(C)(C)C)nn1 c1(C(N(CC2CC2)CC2CC(O)C2)=O)cnccn1.O=C1CO1 c1(C(=O)O)cc(N(C(CCc2c[nH]c(=N)s2)=O)c2cccs2)cc(F)c1 N1(C(c2scc(C)c2)=O)CC2CCCC(NC(c3cnoc3)=O)C2C1 N1(C(CCC)=O)CCC2(CCC(NC(C3CCC(O)CN3C)=O)CC2)C1 C1(C(=O)NCCC2(C)N=N2)CCN(C(c2cc(Cl)n[nH]2)=O)CC1O CC1(C2(C(=O)NCCc3cc(C(=O)O)no3)CC2)CC1 C1(C(=O)NCCC(C)NC(=O)C(C)(C)C2CCCO2)CCC(N(C)C)CC1 n1(CCC(=O)NCC(CN(C(Cc2cc(C)n(C)n2)=O)C)O)ccc(O)nc1=O c1(C(c2ncccn2)NC(C2C(C)(C(F)F)C2)=O)cccc2ccoc12 c1(C(N2C(CNC(C3C(C)C3C)=O)C(O)C(O)C2)=O)cc(=O)c2ccccc2[nH]1 C1(NC(c2cc(C(C)C)on2)=O)CC(O)CN(C(C2OCCCC2(C)C)=O)C1 c1(CC)nc(CNC(=O)C(c2ccnn2C)NC(=O)CCc2cc(C)on2)co1 C1(C(N2CC(O)(CCNC(c3nocc3Cl)=O)C2)=O)CCC2(CC1)CC(O)C2 C=CCC(C)(C)CC(=O)NC1COCC1NC(C1CCCN(C(=O)NC)C1)=O Cc1nn(C)c(C)c1C(=O)NCCc1cc(CN)ccc1C(F)(F)F N1(C(C)=O)CCCC(OC(=O)C(C)(C)n2ccc(C3CC3)n2)C1.C1(=O)C(C)CN1 N1(C(C(C)O)=O)CC(C)N(C(=O)C=C2CCC2)CC1C C(C(=O)N1CC(C)(O)CO1)C1N(C(CC2C=NN(C)C2=O)=O)CCN(C)C1 C1(N(C(CNC(C=CCCC)=O)=O)C(C2CCC2)C2CCC2)CC(C#N)C1 C(=O)(CCC(=O)N(C)C)NC(C)CNC(=O)C(C)C1CCCC1 N1(C(C(CC#C)NC(c2cccc(CO)c2)=O)=O)CCCC(C)(C#N)C1 Cc1ncnc2c1CC(C(=O)NCCC(C(C)C)NC(c1cnn(C)c1)=O)CC2 N1(C(c2cc(C)sn2)=O)CCCC(C2CCCN(C(=O)CC3OCCC3(C)C)C2)C1 C1(C(=O)NC2C=CC(C(=O)NCC(C)O)C2)C(C)(C)C1(C)C S(=O)(=O)(c1cccc2cnc(C)cc12)N(CCOC)CCF C(CCCC(=O)N(CC(C)(C)CNC(C1COCC1C(N)=O)=O)C)(OC)OC c1(C(N2CCCC(NC(C=C3CCC(C)C3)=O)CC2)=O)c2c(nn1C)CCCC2 c1(OCC(=O)N(CCCCCC)CCNC(C2CCCO2)=O)cnc(SCC)nc1 CCCC(C)(O)C(=O)NCCCCCCNC(c1cc(C)n(-c2ccccc2)n1)=O N1(C(CN2C(C)CCCC2)=O)CC2ON=C(CNC(=O)CSc3cn[nH]c3)C2C1 CCCCC(O)C(=O)NC1(C)CC(NC(C2(C)CCOCC2)=O)C1 n1(CC(=O)NCCC(C)NC(c2nc(C3CC3)cs2)=O)nc(O)ccc1=O C(CCS(C)(=O)=O)(C1CC1)NC(C(=O)NC(C1CC2C=CC1C2)C)=O Cc1nc(C)c(C(=O)N(C2CCN(C(=O)CCc3nc[nH]n3)CC2)C)c(C)n1 N12CC(C(F)C1)NCc1cc([nH]c1)C2=O.c1(C=O)c(C)ncn1C.CO c1(C(C)=O)ccc(C)nc1N1CCCC(CCNC(C2CCCOC2)=O)C1 c1(C(=O)NC2CCC(C)N(C(=O)CP(C)(C)=O)C2)ccc(Cl)c(S(C)(=O)=O)c1 C(=O)(C1COc2ccc(Cl)cc21)N1C(CNC(COC)=O)C(C)CCC1 c1(C(=O)NC2CC(N(C(CCc3cc(C)[nH]n3)=O)C)C2)nccc2occc12 C12(C(N3CC(CNC(c4cnc(CC)s4)=O)OCCC3)=O)CCCCN1CCC2 CC(C(=O)NCC1=CCCN(C(C2(F)CCOC2)=O)C1)S(N)(=O)=O C(C(=O)NNC(=O)COc1ccc(C(N)=O)cc1Cl)c1cc(C)oc1C C1(CC(=O)NCCCN(CCCCNC(=O)CNC(=O)NC)C)CCC(C)CO1 Cc1cc(CNC(c2ccc(C(F)F)o2)=O)ccn1.C12CC(C)N1C2=O N1(C(CCCCCC)=O)CC2=C(C1)CN(C(C1CC3CCC1C3)=O)C2 c1(C(N2CC(COC)N(C(C3CC3(C)C)=O)CC2)=O)ccccc1P(C)(C)=O C(=O)(C(C)(F)C(=O)N(CC(C)NC(=O)CN1CCCC1)C)OCC N1(C(C(N2CCOCC2)C)=O)CCCC1CC(=O)NCC1(CC2CCC2)CC1 C12(C(N3CC(C)C(CC(=O)NCC4CNC(=O)C4)C3)=O)CCCC1OCC2 C#CCCCC(C)(c1nnnn1-c1ccc(Br)cc1)NCc1ccoc1C Cc1ccccc1CNC(N1CCCC(NC(=O)CC(C)(C)C2CC2)C1)=O C(=O)(C(F)(F)CCNC1CCCCC1)NC(C)CCN(C(=O)CC12CC(C1)C2)C N1(C(CCN(C)C(N)=O)=O)CC(CNC(=O)C=CCO)(NC(=O)C(C)(C)C)C1 N1(C(c2cn(CC)nn2)=O)CCC2CN(C(=O)C(F)(F)C(O)C3CC3)CC2CC1 C1(NC(C2CC(n3cc(CCC(C)O)nn3)C2)=O)CCCCC1C1CC1 C12(CCC(=O)N(C3(C#C)CC3)C)CCC1CN(C(=O)C(C)=C1CCCC1)C2 C1(C(=O)NCC(C(C)C)F)CN(C(C2(N(C)C)CC2)=O)CC1CC1CCCO1 c1(CCC(N2CC=C(CNC(C(CSC)C)=O)CC2)=O)cccc(S(N)(=O)=O)c1 c1(CC(=O)NCC(C(C)C)NC(C2(CO)CC2)=O)cccnc1Cl C1(C(N2C(CN(C(C(CC)OC)=O)C)CC(F)C2)=O)COc2ccc(F)cc2C1 c1(C(=O)NC(CN(C(C(CC)n2ccnc2)=O)C)C)cc(C)c(F)o1 C1(C(=O)NCCC(C)(C)NC(=O)CC2CC=CCC2)CC12CCCC2 c1(CNCc2c(C)nns2)cccc(N2CCOC2=O)c1 c1(S)cccc(S(C)(=O)=O)c1.C1C(F)C(=O)N2CC(C2)CN1.N(C1CC1)(CC)C c1(C(=O)NCC2CC3CC3N2C(=O)CC2CC=CC2)[nH]nc2ncnc(O)c12 C(=O)(C1=CCCC1c1ccccc1)N(C)CCNC(=O)COCCF c1(CC(=O)NCCCCC2CC2)cnc2cccnn12.C1(OC)CC2N(C1)C2=O C1(CC(=O)NC(CNC(c2c[nH]nc2-c2ccncc2)=O)C2CC2)CCOCC1 c1(OCC(=O)N(C(C)CNC(c2ccc(C(C)O)cc2)=O)C)cc(F)cc(F)c1 C(=O)(C(C(C)O)NC(C1CCOC1C)=O)N(CCC#C)CCOC C1(F)(CNC(c2ccc(C)s2)=O)CCN(C(c2cccc(OC(C)C)c2)=O)CC1 c1(C(N(CCOC)CCNC(C23CC(C)C2C3)=O)=O)cccc(C(C)C)n1 c1(C(=O)NCC(CCNC(=O)CC2CCC2)O)ccn2nccc2c1 N1(C(C(CC)COC)=O)Cc2ccccc2C(NC(=O)Cc2ccc(O)cc2)C1 C12(C(=O)NCC3(COC)CCN(C(=O)C(C)CC#N)C3)CC(C)(CCO1)C2 Cc1cc(N)cnc1C(N1CCC(F)C(NC(=O)C(C)CC(C)C)C1)=O C(CCCC(=O)NC1CC(CNC(=O)C=Cc2cccs2)C1)NC(N)=O C(=O)(CC1=CCCC1)NCC(C)NC(c1cnn(-c2cccc(Cl)c2)c1)=O c1(C(N(C)CC2N(C(C3(CC(C)C)CCCC3)=O)CCC2)=O)cccnc1O c1(C(=O)OC)ccc(C(F)(F)F)c(C(=O)NC2(c3ccon3)CCCC2)c1Cl c1(C(N(C2CCCC(NC(c3ccnnc3O)=O)C2)C)=O)nccn2ccnc12 N1(C(C2=CC(C)(CC)C2)=O)CCC2CCN(C(c3sc(C)cc3Cl)=O)CC12 c1(OC)ccc(OC)c(C(=O)NC(CCNC(C2CC(F)(CO)C2)=O)C(C)C)c1N c1(N2CCC(C)(NC(C3CCCC(=O)N3)=O)C2)ncc(C#N)cc1F CCCCCCC(C)(C)C(=O)N1CC(O)(CCNC(=O)C=CC=C(Cl)Cl)C1 c1(C(N(CCCn2cc(C)nn2)C(C)C)=O)oc(Br)nc1C.C(CCOC)OC c1(C(=O)NC2(CNC(COC)=O)CCC2)cc2c([nH]1)CCOC2 C1(C(N2CC(=C(CNC(c3c(C)ncs3)=O)F)C2)=O)C2CCCCC12 N1(C(C)=O)C(C)CS(=O)(=O)CC1C.c1(NC(=O)OC)c(SC(F)(F)F)cccc1F CC1CCC(C(=O)N2CC(n3cc(CN(C4CC4)CC4CC4)nn3)CO2)CC1C n1(CCC)nc(C)cc1C(=O)NCC1CC1C(=O)NCC1CN(C)CC1O c1(C(=O)NC(CC(C)C)CNC(=O)C(C)(O)C(F)(F)F)ccc2cc[nH]c2c1F C1(NC(c2cc(C(F)(F)F)cs2)(c2nnnn2C2CC(F)(F)C2)C)CCCC12CC2 C1(CNC(COCC(=O)OC)=O)CC(C)(C)CN1C(c1nnn(C(C)(C)C)n1)=O C1(C(C)NC(=O)Cc2ccnn2C)CCN(C(C2CC2C2CCCO2)=O)CC1 N1(C(c2c(C)nn[nH]2)=O)CCCOC(CNC(C2(C)CC2(F)F)=O)C1 CC12CCC(C(=O)OCCNC(=O)NOCC=CCl)(CC1)CO2 C1(C(=O)Nc2cccc(C)n2)C2CCC1N(C(c1ncccc1C)C)C2 N1(C(CCC(C)OC)=O)CC2CC2CC(NC(C2(C)CC2(F)F)=O)CC1 C(=O)(CCC(C)(C)O)NC(C1CCCC(OCC(=O)OC)C1)C.C(CF)N.OC N1(C(C2=C(C)OCC2)=O)CCC(NC(c2cc(Br)c[nH]2)=O)CC(C)(C)C1 C=C(C)C(O)CC(=O)NCC1CCC1NC(c1cc(-c2csc(C)n2)c[nH]1)=O N1(C(C=C(COC)C)=O)CC2CC1C2C(=O)N(C)C.C12CN(C1)CCN2 C(=O)(C1=CCC(F)(F)CC1)NC1(CNC(C(C(C)OCC)O)=O)CCOCC1 C1(C(=O)NCCOc2ccc(NC(C(C)OCF)=O)cc2)CCc2c[nH]nc2C1 c1(C(C)C)cc(=NC2CC3CCC(C2)N3C(C2CC3(C2)CC3F)=O)[nH]c(Cl)n1 c1(C(N(C2CCCN(C(=O)C=CCF)C2)CC)=O)ccc2sncc2c1 c1(C(=O)NCCC2(C)CCN(C(CCCC#C)=O)C2)nnc(O)nc1O Cc1ccc(Cl)c(O)c1C(=O)NCC1CCCC(CNC(=O)C2=CC(C)(C)C2)C1 c1(-c2c(C(N3CCC4(CC=CC4)C3)=O)cccn2)ccc2cnccc2n1 CC1(C)CCC(F)(F)CC1C(=O)NCC=CCNC(c1cccc(N)n1)=O CON1CC(C(N2CCCC2C(=O)NC2CCCOC2)=O)CC1=O CC1(C)CN(C(=O)CCCn2cccc2)CC(CNC(C2(F)CC2)=O)O1 N1(C(Cc2ccc(C)cc2)=O)CCN(C(=O)C(C)n2ccnc2)C2CC12 N1(C(CC(=C)Br)=O)CCC(NC(=O)Cc2ncc(CC)[nH]2)C(CC)C1 Cn1cc(C(=O)NCCCCCNC(=O)C(C)(C)n2cccn2)c(C(C)(F)F)n1 C1(C(N2CC(C3OCCN(C(C#CC(=O)N(C)C)=O)C3)C2)=O)CCn2cnnc2C1 c1(C(=O)NCCC(C)NC(C2CCC(C)CC2)=O)cc(=O)c2ccncc2o1 C(C(F)(F)CCC(=O)N1CCC(CN=c2ncc(O)c[nH]2)C1)c1cccc(OC)c1 N1(C(Cc2n(C)c(S)nn2)=O)CC2CCN(C(C3(F)CCC3)=O)CC2C1 Cc1cc(=NC(=O)CSCC=Cc2cccc(C#N)c2)[nH]n1-c1cccnc1Cl c1(C(=O)NC2(CCC)CC2)ccoc1CNC(=O)C(C)(C)OC(C)=O C(=O)(C(C)C(C)(C)C)NCC(CNC(=O)C=Cc1ncc[nH]1)OC N1(C(=O)COCC2CNCCN2)CCCC(C(F)(F)F)(C2CC2)C1 C(=O)(C(F)(F)CCc1ccccc1)NCCN(C(C1(C)CCC(C)C1)=O)CC C1(C(N2CC(OC)C(NC(C3CC4CCC3O4)=O)C2)=O)CC2(C1)CS(=O)(=O)C2 N1(C(C2(C#C)CC2)=O)CCC2CCN(C(=O)Cc3cccc([N+](=O)[O-])c3C)C2C1 C1(C(=O)NCC(C)(C2CC2)NC(c2c(CC)occ2)=O)CCN(C)C1C N1(C2CN(c3c(OC)cnc(SC)n3)CC(F)C2)C2CCC1CN(C)C(=O)C2 C1(COC)(CNC(=O)C(N)=O)CN(C(=O)CCOC(C)CC(C)C)C1 c1(C(=O)NCC(C2CC2)NC(CCSC)=O)cc(C#N)c(F)cc1F CCC(C(=O)NCCOC1CCN(C(=O)Cn2ncnn2)C1)N(C)C C1(NC(C(Cc2c(OC)cccc2)(C)C)=O)C2CCC1N(C(=O)CCSC)C2 C1(NC(C2C(NC(C(C(C)C)=O)=O)CCC2)=O)CCCC2(CC1)CC2 CN1C2CCC1CC(=CC(=O)NC13CC1CN(C(c1ccc[nH]1)=O)C3)C2 c12ccc(cc1)CNC(=O)CN1CCC(C1=O)NC2.c1(CC)nc(CC)no1 CC1CC(C(N2CCC2(C)CCO)=O)CCN1C(c1csc(F)c1)=O C1(CNC(c2occ(C(N)=O)c2)=O)CCCCN(c2ccc(C#N)nc2)C1 N1(C(C(C)OCCC=C)=O)CCC2(CC1)CCN(c1nc(C)nc(C)c1F)C2 C1(C(N(C2CCOC2)C)=O)C2CN(C(C3(C(F)(F)F)CCC3)=O)CC12 N1(C(CCCOCC=C)=O)CCC(NC(C2(S(C)(=O)=O)CC(O)C2)=O)C12CCC2 C1(NC(C2CC(=C)C2)=O)C(C)CCC1C.C12(CC1(C)C)C(=O)N2 c1(C(N2CC(N3C(=O)CC(NC(CC=C=C)=O)C3)C2)=O)ncc([N+](=O)[O-])cc1C C1(C(=O)NCc2n(CC)cnn2)CCN(C(c2sccc2Cl)=O)C1C C(=O)(CCCN=[N+]=[N-])N1C(CC(=O)NC(C=C)C2CCC2)CC1 CC(C)CCC(=O)NCCCC(C)NC(c1ccc(C2CCCCC2)s1)=O CC(O)C(C)C(=O)NC1C2CC1N(C(=O)CCc1nc(-c3cnc[nH]3)no1)C2 C1(CC=C)(C(N2CC(N=[N+]=[N-])C2)=O)CCN(C(c2cc[nH]c2C)=O)C1 N1(C(C(CC)OC)=O)CCN(CC2CC(F)(CNC(C3(C)COC3)=O)C2)CC1 C12(NC(c3scc(C(N)=O)c3)=O)CCCC1CN(C(C13CCC(CC1=O)C3)=O)C2 C(=O)(C#CC(C)(C)CNC(C1(CCN(C)C)CC1)=O)NC(C)Cc1nc[nH]n1 C1(CC(=O)N(C(C)C(=O)NC23CC(C2)C3)C)CCOC1=O CC(C)C(O)CC(=O)N1CC(O)(C(C)NC(=O)CSc2nccn2C(C)(C)C)C1 C(=O)(C1CSc2ccccc21)N1CCC(NC(c2scc(C)c2)=O)CC1 N1(C(c2c(OC)nccc2)=O)CCC(C2CC2)C1CNC(c1ccccc1C)=O CC1CC2CCN(C(=O)C(=O)NC3CC4CCC4C3)CC12 c1(C(=O)NC2C(NC(c3c(OC)cc(O)nc3)=O)CC2)cc2cccn2cn1 C1(C)(C(N2CCC(CNC(C(CC#C)O)=O)CC2)=O)CC(C(C)(C)C)=NO1 N1(C(C)=O)CCC2(CC1)CN(S(=O)(=O)CCCOC(C)=O)CC(C)O2 c1(C(=O)NCCCCNC(C2(C(=O)NC3CC3)CC2)=O)coc(-c2cccs2)n1 c1(C(N2CCC(CCNC(c3n(CC)ccc3)=O)C2)=O)cc(C2CC2)ccc1F c1cc(C(C=COC(C)(C)C)=O)cc2c1OCO2.OC(F)F N1(C(c2nn(CC)c(C3CC3)c2)=O)CC2(CC2)CC1CNC(=O)CCC(F)F C1(NC(C2C(OC)CN(C(COCCCC#C)=O)C2)=O)COCCN(C)C1 C1(NC(C2CCCN2CC(F)F)=O)CN(C(=O)COC2CCOCC2)CC12CC2 CC(C)C(C)CC(=O)N1CCCC1CCC1CCN(C(C2CC2(F)F)=O)CC1 N(C1CCOc2cc(F)cc(F)c21)C(N(c1c(C)cccc1)CCC#N)=O CC(C(=O)N1CC(O)(CNC(c2cc(Cc3ccccc3)c[nH]2)=O)C1)C(C)O c1(OC)cc(OC)nc(NC2CC2C(=O)Nc2c(C)ccnc2F)n1 N1(C(CCC=C)=O)CCC(CNC(c2cc(C(N)=O)c[nH]2)=O)C12CC2 N1(C(COC2CC(C#N)C2)=O)CC(=O)NCC1C(=O)NC1CC(n2ccnn2)C1 c1(NC(C2N(c3ncc(C)c(C)n3)CCCC2)=O)cc(Br)c([N+](=O)[O-])cn1 C1(CC)CC(c2nnnn2C2CC(F)(F)C2)(NC2CSC2)CCO1 C1(NC(C)=O)CC2(C1)CN(C(c1cccc(C(F)F)c1F)=O)C2 N1(C(c2ccc(F)s2)=O)CCC2CN(C(=O)C(F)=CC3CC3)C2C1 c1(C(C(=O)N(C2CN(C(C(CC)SC)=O)C2)C)O)ccc(Br)cc1 CC(C)C1=NOC(C(N2CC(O)CC2CC(=O)Nc2cnc(Cl)nc2)=O)C1 N1(C(C(C=C)O)=O)CC(NC(c2cnccc2C(F)(F)F)=O)CC2(CCC2)C1 N1(C(=O)CC2CCCN(C(c3cnn4cc[nH]c34)=O)C2)CCCC(C2CCC2)C1 C1(C(N2C(C)COC(C)(C)C2)=O)CCN(C(=O)CC(O)CC(C)(C)C)CC1(C)C C(=O)(C1=CC2CC=CCC12)NCC1CC(NC(c2cc(C)c(Cl)c(N)c2)=O)C1 C1(NC(c2[nH]nc(OC)c2Cl)=O)CC2CC1CN2C(=O)CC(C)(C)C C1(NC(c2cc3nnn(C)c3s2)=O)CCN(C(c2ncc[nH]2)=O)CC12CCC2 Cc1cc([N+](=O)[O-])cnc1NCCC1CCCN(C(=O)C(C)CF)C1 c1(C(=O)NCC(C2CCCC2)NC(C(C)(C)N(C)C)=O)cccc2c1CCN2 Cn1cc(C(F)(F)F)cc(NC(=O)CC(=O)NCCCc2ccccc2)c1=O C=CCCCCC(=O)N1CCOC(CNC2CC(C(=O)Nc3ccccc3)C2)C1 CC(C)(CC(F)(F)F)C(=O)NCCOC1CCN(C(=O)CN2C(=O)CCC2=O)C1 CC(CC(=O)NC1COCCC1NC(=O)C1=CCCSC1)C(F)(F)F c1(C(=O)NC2CCC(C(=O)NCc3occ(C)n3)CC2)ccn2nccc2c1 C(=O)(CC(C)(C)C(F)(F)F)NC(CN(C(=O)C(c1cccc(F)c1)(C)O)CC)C CC1=C(C(=O)NCC2CC3CN(C(=O)CCC4OCCO4)CC23)CCC1 c1(C(=O)NC(CNC(C(CCC)OC)=O)C2CC2)cc2n(n1)CCNC2=O C1(C)(C(N2C(CN(C(=O)CC3CN(C(C)=O)C3)CC)CCC2)=O)CCCNC1=O Cn1c(C(=O)NCCOCCCNC(c2cnn3c2OCC3)=O)ccc1C#N c1(C2C(C(N(CCCNC(C(CC)(C)O)=O)C)=O)C2)c(Cl)cccc1Cl C(CC(C)C)(C(=O)NCC(CC(C)C)NC(c1coc(C2CCC2)n1)=O)OC C1(O)(CNC(C2(CCOC)CCC2)=O)CCCN(C(=O)CCn2ccc(C)n2)C1 c1(C(=O)NC(C(C)NC(c2ccn(C(C)C)c2)=O)CO)cc2ccncc2[nH]1 Cc1nn(C)c2nc(C(N3CCC(F)(CNC(=O)C4=CCC4)C3)=O)ccc12 N1(C(C(C)C2CCCC2)=O)CC2(C(=O)NCCCC(C)(F)F)CC1CO2 N1(C(CC)=O)CCN(C(c2ccc(CC)nc2)=O)CC(O)C1 C(C(C)(COC)C(=O)NC1C=CCN(C(=O)C(O)Cc2[nH]cnc2C)C1)OC C1(C(C(=O)NCC2CC(NC(C3(CCOC)CCC3)=O)C2)C)CCC(=O)N1 C(C1CCc2cc(F)ccc21)NC(=O)C1CC1c1ccc(C(F)(F)F)cc1 C1(CCNC(CN(C)C)=O)CN(C(=O)C(CO)NC(N)=O)CCO1 N1(C(C=CC(C)C)=O)CC(CNC(c2cn(CC(F)F)cn2)=O)CC1(C)C N1(C(C(C=C=C)C)=O)CCN(C(c2cc(Br)sn2)=O)C(C(F)F)C1 FC(F)(F)C1=CCN(c2ccnc(N3CCOC(C4CCCCC4)C3)n2)CC1 N1(C(C(C2CCC2)OC)=O)CC=CC1(C)C(=O)NC1(C2CCCCO2)CC1 C(c1ccncc1)=CC(=O)NCC(CNC(c1nnc(C(C)(C)C)s1)=O)OC C1(CCNC(COCCCC#C)=O)CCN(C(c2ccnn2C(F)F)=O)C(C)C1 N1(C(CC2C(C)C2)=O)CCC(CNC(=O)C(C)Cc2ccccc2F)C1(C)C N1(C(C(CC2CC2)NC(C2(CC(C)=O)CC2)=O)=O)CC2CC1CS2=O C12(CNC(COCC(=C)C)=O)CCCC1N(C(=O)CSCCCC(C)C)CCC2 N1(CC)CCC([N+](=O)[O-])CC1.c12cc(c(C)nn1)C(=O)N1CCCCC1c1n[nH]cc1-2 N1(C(c2c(N)nccn2)=O)CCCC(NC(c2nn[nH]c2C(F)(F)F)=O)C(F)C1 C1(N(C)C)CCN(CC(N2CCCC2CNC(C2(C)CCCC2)=O)=O)CC1 C#Cc1ccnc(C(=O)NC(CNC(c2cc(=O)n(C)cn2)=O)CO)c1 c1(CN2CCC(C(=O)NCc3cn(CC)nc3)C2)ccc(F)cn1 N1(C(C2(n3cncn3)CC2)=O)CCC2CN(C(=O)Cn3ncnn3)CC2C1 CCC(C)(F)C(=O)N1CCC(NC(=O)C(O)Cc2[nH]cnc2C)CC1 CCC(CC)(C(=O)NC1CC(C)N(C(c2cccc(N)c2)=O)C1)OC N1(C(N(c2cccc(NC(=O)C(=O)O)c2)CCOC)=O)CCC12CCCOC2 Cc1ncc(N)cc1C(=O)NC(C)CC(C)NC(c1ccncc1N(C)C)=O C1(OC2CCN(C(C)=O)C2)CCN(C)CC1.C(=O)(C(F)=C1CCCC1)N1C(C)C1 N1(C(CC(CC)C(C)C)=O)CCC(C(=O)NC2CC3CCC2C(O)C3O)=C(F)C1 C1(NC(c2nc(C)[nH]n2)=O)CCN(C(c2cnn(C(C)(C)C)c2Cl)=O)CC1(C)C C1(C(N(C(C)CNC(=O)C(C)OCCN(C)C)C)=O)CCCCC1 C1(NC(CC(CCC)(C)C)=O)CCn2c(-c3cn(CC(N)=O)nn3)nnc2C1 C#Cc1ccnc(C(N2CC(NC(c3ccc(F)cc3)(C)CC)CC2C)=O)c1 c1(C(N(CC(C)(C)O)C)=O)cnc(C(=O)NCCCCO)cc1 N1(Cc2scc(C)n2)CCOC(C)(CC(C)C)C1.C(=O)(C(C)(C)C(F)F)N C1(NC(C(c2ccn(C)c2)C)=O)CCOCC1C(=O)NCC(C)(C)CO CN=c1c(C(=O)NC(C)C(C)NC(=O)Cn2cncc2C)c[nH]c2ccccc12 C1(C(=O)NCC(CCC)OCC)C(C)OCCN1C(=O)CSC(F)(F)F N1(C(C(C)SC)=O)CCC2C(NC(=O)CCOC3CC3)CC12 c1(C(COC)N(C)C)ccc(CCC(=O)NC(=O)C(C)(C)C2CCCCO2)cc1 c1(-c2c(Cl)occ2)nc(-c2ccco2)nn1-c1ccnc(F)c1 C(c1ccc(C)s1)=CC(=O)NCC(c1cnn(C)c1)NC(C1CCN(CC)C1)=O C1(C(=O)NC(C)CC(=O)NC(C)Cc2ncn(C)n2)(OC)CCOCC1 c1(CC(=O)NC(=O)C=CC(C)(C)SC)cccc(C)c1C.CCC1(C)CCN1 N1(C(C(CC)OC)=O)CC2(CCCCN(C(C3(OC)CCCC3)=O)C2)C1 N1(C(c2cncc(C)c2)=O)CCC2(CCN(c3cc(C)ncn3)C2)C1 CC(C)C(C(=O)N1CC(C(=O)Nc2ccc(C(F)F)nc2)C(C)C1)C1CCC1 C1(N(C(CC(C)c2cccnc2)=O)C(c2ncccc2Cl)C)C2CCC1CNC2 C1(C(=O)OCC(C)OCC)CCc2nc(-c3cccc(C)c3)sc2C1 c1(C(=O)NC(C(CC)CC)C)cc(C(=O)O)c(OC)c(OC)c1 N1(C(COCCCOC)=O)CCC(NC(c2ccccc2-n2cccn2)=O)C(C)C1 C(=O)(C1=NNC(=O)C1)N1CCC2C(Sc3ccccc3)C21.CC1CCN2C1C2 C#CCCCC(=O)N(C1CCN(C(=O)C=C2CCCO2)CC1)CCOC Cc1n[nH]c(C)c1CC(=O)NC1CN(C(=O)CCCCc2ccccc2)CC1CO c1(-n2cc(C(=O)NCC(O)CC3CCCCC3)nn2)cccc(Br)c1 c1(CNc2c(C(=O)Nc3c(Cl)cc(C)cc3Cl)scc2)cccc2cnccc12 C1(NC(c2n(C)nc(CC)c2Cl)=O)CC2CCC1N(C(=O)CC(C)C(C)C)C2 S(=O)(=O)(c1cc(Br)c(Br)s1)Nc1ccc(C(=O)NS(=O)(=O)c2ccccc2Br)nc1 c1(C(=O)NCC(C)(C2CC2)NC(C(C)OCC#C)=O)cccc([N+](=O)[O-])c1 N1(C(C(C)OCCOCC)=O)CCCN(C(=O)C=CC(C)(C)C)CC1C CCCCC(CC(=O)Nc1cn(C)nc1C)NC(C12CCCN1CCC2)=O C(=O)(CCCCCNC(=O)Cc1n[nH]c(C)n1)N1C(CC)(CC)CC1 CC1C(C)NCCN1C(=O)Nc1nc2c([nH]1)CCC2 C(=O)(CS(=O)(=O)C(C)C)N1CC(NC(c2cc(CC)[nH]n2)=O)C(n2cccn2)C1 C1(CNC(C2(COC)CCCN2C(=O)CC(C)(C)C)=O)CC2CCC(C1)C2 N1(C(c2ccc(-c3cccs3)[nH]2)=O)CCCCC2(CCN(C(=O)C(Cl)=CCl)C2)C1 C(=O)(C(F)CCC(C)C)N1CCC(C)(c2cn(CCC(C(=O)OCC)(F)F)nn2)C1 c1(NC)cccc(C(N2CC=CC(NC(=O)C=C3CCC(C)CC3)C2)=O)n1 c1(N2CCC(C)C(NC(c3c(C)oc(CO)c3)=O)C2C)ncc2ncn(C)c2n1 c1(C(N2CC(NC(C(C)SC(F)(F)F)=O)C2)=O)ccc(C2CCC23CCC3)cc1 Cc1nnc2n1CCCC2C(=O)N1CC(C)CN(C(=O)C(C)C2CC2)CC1C C1(NC(CC=CC(C)(C)C)=O)CCCC(C(=O)NCC(O)C2(Cl)CC2)C1 c1(C(=O)NCC2(F)CCC(NC(C(C)=C3CC3)=O)C2)cc(=NS(C)(=O)=O)cc[nH]1 c1(C(=O)NCC(C)(C2CC2)NC(CCCn2ncc(C)c2)=O)cncc(C)n1 C1(C2CCOCC2)(C(=O)NC(CNC(c2c(Cl)ccc(C)c2)=O)C)CC1(F)F C1(C(=O)NCCSCC=C)CCC(O)CN1C(c1ccn(C)c1C1CCC1)=O N(C1CCCc2ccc(Br)cc21)C(C(C)(C)CC#N)c1n(CC=C)nnn1 N12CCC(c3ccc(Br)cc3)(C1)C2.CC(C)(C)C(N)C1CCC1 c1(C(N2CC3C(CNC(CC(=O)OC)=O)(C3)C2)=O)cc(F)cc([N+](=O)[O-])c1 c1(OC)ccc2c(n1)CC(NC(=O)NCC(c1cnccn1)C)CC2 CCC(C)C(O)C(=O)N1CCCC(C)(NC(=O)Cc2nc(=O)o[nH]2)C1 c1(C(CC2CC2)CNC(N2CCCC2CC2CC2)=O)ccc(Br)cn1 C1(NC(c2c(OCC)n[nH]c2)=O)CN(C(=O)CC(C)C(=O)OC)C(CC)(CC)C1 CC1CN(C(=O)C(Cc2cc[nH]n2)NC(=O)C(C)(C)C2CCOC2)C(C)C1C N1(C(C2(SC)CC2)=O)CCC2CN(C(=O)CC3CNC(=O)O3)CCC2C1 C1(OC)CCC(C)(c2nc(-c3ccc(F)cc3)nn2C2CCCSC2)CC1 C(CC(=O)N(C1CCC(NC(=O)CCCN(C)C)C1)C)(C(F)(F)F)OC N1(C(CC(COC)C)=O)CC2(CNC(c3ncsc3C)=O)CC1CO2 C1(C(=O)NC2CCN(C(c3ccn(CC)n3)=O)C2C(C)C)CS(=O)(=O)CC12CC2 C1(CC)CC(C(=O)N2CCN(CC3CC(F)(F)C3)CC2C)=NO1 C1(CNC(C=C(COC)C)=O)CC(C)CCN1C(=O)C(C)n1cncn1 c1(C(N2CC(CCC)C(NC(c3nc(O)sc3C)=O)C2)=O)cc(C)ncc1C N1(C(c2nccc(OCC)n2)=O)CC(C)CN(C(=O)C(C)SC(F)(F)F)C(C)C1 c1(C(=O)NCC(C(C)C)NC(=O)CC2CCN(C)CC2)cc(C#N)c(N)cc1O N=c1[nH]c(=NCC2CCCC23CC3)[nH]c(=NCCc2cn[nH]c2)[nH]1 Cc1cc(N)c(C(N2CCCCC2CCNC(C2(C)CCCO2)=O)=O)cc1C c1(CC(=O)NC(C)C=CC(N2CCC(C(N)=O)C2(C)C)=O)cnc(O)nc1O CC1(C)CN(C(C2CC3(C2)CC(F)C3)=O)CC(CNC(=O)CC2CC2(Cl)Cl)O1 C1(NC2CCCN(C(c3c(C)nn[nH]3)=O)C2)CCCCC1(C)C.C12CCCN1C2=O C1(CCNC(c2c(C)coc2)=O)CN(C(=O)Cn2cc(Br)cn2)CCO1 C1(C)(CNC(C(CCOC)(C)C)=O)COCCN(C(=O)C=Cc2ccncn2)C1 N1(C(c2c(C)[nH]nc2C(F)F)=O)CCOCC(C(=O)NCCN2CCOCC2)C1 N1(C(C2CC(C(=O)OC)C2)=O)CCC(C2(NC(C3CCCCCCC3C)=O)CC2)C1 c1(C(=O)OC(C)(C)C)ccc(C(=O)NCC2CC2CNC(c2cnc(S)[nH]2)=O)o1 C1(C(=O)NC2CC(NC(Cc3cc(=N)[nH]cc3)=O)C23CCC3)CC2CCC(C1)C2O C(=O)(C1=CN(C)S(=O)(=O)N=C1C)N1CCC(CNC(C(C)OCC#C)=O)C1(C)C C1(CC(=O)NC(C(=O)NC(C=C)(C)CC)CSCC)CCCC12CC2 C=CC(CC)CC(=O)NCCC1(O)CCN(C(c2cnc(OC)c(C)c2)=O)C1 N1(C(C(=O)NCc2scc(C)c2)=O)C(C=O)c2ccccc2-c2ccccc21 C1(C2CCN(C(=O)CNC(=O)NC3CC3)C2)(NC(=O)CC2COC(=O)C2)CC1 C1(CCC)CCC(C(=O)NCC2CC(NC(c3cccc[n+]3[O-])=O)C2)CC1 C=CCC(C)(C(=O)N1CC(C)(C)CC1CNC(c1ccncn1)=O)N(C)C C1(=CC(=O)NCCC2COCCN2C(c2ncccc2F)=O)CN2CCC1CC2 c1(NC(=O)CCCOc2cccnc2)ccc2scnc2c1.C12CC1C(=O)N2 C1(CC(C)C)C(=O)NC(C)C(=O)NO1.C1CC2CCC1O2.CCO c1(COC)cccc(C)c1NNC(=O)NCc1cc(C2CCC2)n[nH]1 C(=O)(CCCCC(C)C)N1C(CCCNC(CCSCCC)=O)CCC1 C1(CNC(C(C=CC)O)=O)CC2(CO1)CN(C(C1CSC1)=O)C2 N1(C(C(=O)NCC2(OC)CCC(F)(F)CC2)=O)CCC2(CC1)CCC(F)(F)CO2 C(=O)(CCCS(N)(=O)=O)NC1CCN(C(C(c2ccc(C)nc2)(F)F)=O)CC1C N1(Cc2nnc(C)s2)CCC(C)(NC(=O)CC2CC=CC2)C1 Cc1cc(C(=O)CNC(=O)C(C)(C)C2(O)CCOC2)cnc1Br N1(C(CNC(c2c(OC)cccc2)=O)=O)CC(C(=O)O)C2(CCNCC2)C1 Cc1ccc2[nH]c(C(N3CCN(C(=O)C(O)C4CC4)CC3)=O)c(Cl)c2c1 Cc1cc(=O)oc2ccc(OCC(=O)NCC(O)CCNC(=O)CN(C)C)cc12 c1(C2C(CC)C2)csc(NC(=O)N(c2cnn(C)c2)C2CC2)n1 Cc1cc(=NCc2nc3c(s2)CCC3)[nH]c(N2CC3CC2CS3=O)n1 C1(C(=O)NCCCC2(NC(CCc3c(C)ncs3)=O)CC2)CC1C1CCCC1 c1(C(=O)NC2C(NC(=O)CCc3ccon3)CC2)ccccc1OC(F)F c1(C(=O)NCCC(O)C(=O)N2CCCC2C2(C(=O)O)CC2)ccn2nccc2c1 N1(C(C(C2CCCC2)OC)=O)CCCC1C(=O)N(C1CCN(CC2CC2)C1)C c1(OC)c(CN2CCCCC2c2ccc(C(=O)NS(C)(=O)=O)cc2)cccc1F N1(C(CN(CC)CC)=O)CC(NC(c2cccc(-c3nccs3)c2)=O)CCC1C N1(C(c2n(C)[nH]c(=N)c2)=O)CCC(NC(=O)CCSc2ccc(F)cc2)C(O)C1 Cc1c(C(N2CC3CC3(NC(=O)C(C)CN(C)C)C2)=O)c[nH]c2nccc1-2 c1(C(=O)NC(C2CCN(C(C3(OC)CCSC3)=O)C2)(C)C)ccccc1Cl C1(NC(C=CCC(C)(C)NC(=O)Nc2cccc(Cl)c2)=O)CC1C1CCCC1 C1(N(C(CC(OCC)OCC)=O)C)CCCN(C(=O)C(C)(C)C)CC1 c1(C(=O)NC(C2CC(C(=O)OC)C2)=O)cnn(C(C)C)c1C.C12(O)CN(C1)C2 C1(OC)CN(C(c2ccns2)=O)CCC1NC(=O)CN1CC2CC2C1 S(=O)(=O)(c1cc(F)c(F)c(F)c1)N1CCN(C(c2c(N)c(F)c(Br)cc2)=O)CC1 n1(C(C)C(=O)N(CCCN(C(=O)CC2(CO)CC2)C)C)nnc(-c2ccccc2)n1 C1(C(=O)NCC2CCCN2C(c2cc[nH]n2)=O)(COC)CCOCC1 c1(C(C)C)cccc(OCC(=O)NC2CN(C(c3c[nH]ccc3=O)=O)C2)c1 c1(OC)cc(N2CCC(C)(NC(C3CCC(CC)CC3)=O)C2)nc(C(F)(F)F)n1 C1(C(N2C(CC(C)C)CC2)=O)N(C(C2CCC(=O)CC2)=O)CC12CCCC2 C1(C(=O)NC(c2ccc(F)cc2)CNC(CCCOC(C)=O)=O)CCCC1(C)C N1(C(COC(C)=O)=O)CC(C(=O)NCc2cncnc2C)C2(CCC2)C1 CCCCC(CCC)NC(=O)CC(C)(C)NC(C1CC(F)C(=O)N1)=O C12(NC(C(CC)SC)=O)CCCCC1N(c1ncc(I)cn1)CC2 N12CCC3CC(C1)CN(C3)C(=O)C(O)C2=O.N1(CC(=O)C2CCC2)CCOCC1 c1(CC(=O)NCC2CC(NC(C3(CC)CCC3)=O)C2)c(C(C)C)cccc1Br.OCC C(C(C)(C)C(=O)N(C1CC(C(=O)Nc2cnc(SC)nc2)C1)C)SC N12CCC(C1(C)C)N(c1ccc(F)cc1)C2=O.c1(-c2c(C)coc2)nc(C)c(C)s1 CC1(C)CC(CNC(c2cncnc2)=O)CN1C(=O)CCC12CCC(CC1)C2 C12(C(=O)OCc3cnn4c3CCC4)CCCCN1CCC2 Cc1cc(C(N2CCCC(O)(CN(C(=O)CN3CC=CC3)C)C2)=O)c(C)cn1 c1(C(=O)NCCC2(OC)CN(C(C3(C)CCCS3)=O)C2)cnn(C)c1C(F)F c1(C(=O)NCC2N(C(CC3(C)CCCO3)=O)CCC2)ccc(Br)cc1F C1(N(C)C(c2cnc(O)n2C)=O)CCCCCC1NC(=O)C(c1cnn(C)c1)O C1(CNC(C(C=CC)O)=O)CN(C(=O)Cn2cc(C#N)cn2)CCC1C Cc1c(CC(=O)NC2CC(CC(=O)NC34CCC(CC3)C4)C2(C)C)ncn1C C12(NC(=O)Cn3cc(C(F)(F)F)cn3)CC1CN(C(c1ccc(CO)cc1)=O)C2 Cc1cnc(C#N)nc1N1CCC(NC(C2CC3CCC3C2)=O)C(C)C1 c1(C(=O)NC2CCCN(C(=O)C(F)OC(F)(F)F)C2)ccc2ccccc2c1F C1(C(=O)NC(CCNC(CCOCCOC)=O)C(C)(C)C)CC1C1CCOCC1 Cc1nc2sccn2c1C(=O)N(C(C)CNC(C1(Oc2cnn(C)c2)CC1)=O)C c1(-c2c(OCC(=O)OC)cccc2)cc(S(=O)(=O)NCCC(N)=O)ccc1OC C1(NC(C(c2cccc(C)c2)O)=O)CCC(C)(CNC(=O)C=CCO)CC1 N1(C(C2C(C)OCCC2)=O)CCC(NC(c2ccc(C(F)F)c(F)c2)=O)CC1C N1(C(C(=O)NCC(=C)C)C2CC(C(=O)OC(C)(C)C)C2)CCCC1C1CCC1 C1(NC(=O)CCC2CC2)CCCCCC1n1cc(-c2cscn2)nn1 c1(OC)c[nH]c(C(=O)NCCC(Cc2ccccc2)NC(C2(Cl)CC2)=O)cc1=O C1(C(=O)NC(C(C(C)C)NC(C2CSC2)=O)C)CC2(C1)CC1(CC1)C2 C(=O)(C1=NOC2(CCC2)C1)NC1(CC=C)CN(C(=O)CC2CCCN(C)C2)C1 c1(C(=O)Nc2nsc3ncccc23)cc([N+](=O)[O-])c(O)cc1F.CC12CN(C1)C2 C1(NC(c2c(OC)nccc2)=O)CCN(C(=O)C(=Cc2cccs2)C)CC1F c1(C(N2C(CCNC(C(CC#C)C)=O)CSCC2)=O)ccc(OC)c(C)c1 Cc1onc(C(N2CCC23CN(C(C2CCC(=O)N2C)=O)C3)=O)c1[N+](=O)[O-] C1(C(C)NC(CCCOCC)=O)CN(C(c2ccc(C(=O)N(C)C)[nH]2)=O)CCO1 CC(C(=O)N1CCN(C(c2ccon2)=O)CC1CC(C)(C)C)C1=CCCC1 N1(C(C2(N(C(c3c(C)nco3)=O)C3CC3)CCC2)=O)CC(C)(C)OCC1C N1(C(CNC(C2C(C)(C)C2)=O)C(F)F)CCN(C(=O)C=C2CCCC2)CC1 N1(C(COCCOCC)=O)C2CCC1CC(O)(CNC(c1cc(C)ccn1)=O)C2 c1(CC)cn2c(n1)CCC(C(=O)NCC1C=CCN1C(c1cnsc1)=O)C2 N1(C(c2c(N)cc(Cl)nc2)=O)CC2CCC(C1)N2C(=O)CSCc1ccccc1 c1(C(=O)NC2CC3CCC(C2)N3C(C2CSC2)=O)cc2c(F)c(F)cc(F)c2[nH]1 c1(C(=O)NCC2OCC(CNC(CC=CC(C)(C)C)=O)C2)ccc2ncnn2c1 c1(C(N2CC(C(=O)NC(c3ccco3)C)C2)=O)cnc(N)cn1 c1(C(N2CCC(NC(C(C(C)C)C)=O)CC2)=O)cc(Cl)cc2c1CCC2 C1(CC)CCN(C(=O)CCOCC(C)(C)C)C1C(=O)NCc1cnn(CC)c1C c1(C(N2CCC(C(C)(O)CNC(=O)CO)CC2)=O)ccccc1[N+](=O)[O-] c1(CSC2C(C)C2C)cccc(NC(=O)C(c2ccccc2)=O)c1.C(CCO)OC C1(C(=O)NC(C(NOCc2ccc(C)cc2)=O)C)CCC(C)(O)CC1 N1(CC)CCCN(C(=O)CC(C)c2ccco2)CC1.C1(=O)CCCCN1 c1(NC2C=CC(C(=O)NC)C2)nc(N2CCCOC(C)C2)c2ccccc2n1 C1(C(=O)NC(C=C)(C)CC)CCN(C(=O)Cc2cccs2)C12CCC2 C1(NC(c2c(C)nccn2)=O)CN(C(=O)Cn2nnnc2C(C)C)C2(CCC2)C1 C1(NC(CC(CC)(C)C)=O)CCCC12CCN(C(=O)CN(C)CCOC)C2 c1(SC)cccc(C(=O)NC2CCC(NC(=O)C(C)(C)C(N)=O)C2)c1[N+](=O)[O-] c1(C(=O)O)ccc(CNCc2c(I)ccnc2Cl)cc1Br C1(CC(=O)NC2C(C)COCC2)N(C(=O)CCCn2ccnc2)CCC1(C)C N1(C(CC(C=C)CC)=O)CCc2c(cnn(C)c2=O)C1 CC1(C)CN(C(c2c(F)cc(Cl)cc2Cl)=O)CCC1NC(c1cc(O)cc(Cl)c1)=O N#Cc1cc(C(=O)C(=O)NCCn2cc(C3CC3)nn2)ccc1F CS(C)(=O)=NCC(=O)N1CCCC(CNC(c2cn(C3CCOC3)nn2)=O)CC1 CC1(C)CC(NC(c2cc[nH]n2)=O)CN1C(c1cc(C2CC2)nnc1O)=O c1(COC)ccccc1C(=O)NCC1CN(C(C2CC2(C)C(C)C)=O)CCO1 c1(-c2nnc(C)o2)ccccc1C(N1CCN(Cc2cccc(Br)c2)CC1)=O N1(C(CCC(C)C)=O)C2CC1CN(C(=O)CCNC(c1ccccc1)=O)C2 N1(C(C(CCC)OC)=O)CCN(C(=O)COc2ccon2)CC(O)C1 N1(C(C(C(C)C)n2cnnc2)=O)CCC(C)N(C(C2CN(C3CCC3)C2)=O)CC1 CCCCC(C)C(=O)NCCCN(C(=O)CC(C)(C)OC)CCO c1(CC)nc(CNC(=O)NCCC2CC2)oc1C N1(C(C=CC(C)(C)NCCN2CCCCC2)=O)CCCC(C)(C)C1C(N)=O C(=O)(C(C)SC(F)(F)F)N(C(CNC(C)=O)C1CC1)C1CC1 N1(C(CC2(C)CCOCC2)=O)CCC2(CC1)CC2CNC(=O)C(F)(F)C(F)(F)F c1(C(=O)NCC2(CNC(CCN(C)CC)=O)CCCC2)cccc(C(C)C)c1N O=C(C1CCCc2n[nH]cc21)NC1CN(C(=O)CCC(F)F)C2(CCC2)C1 S(=O)(=O)(c1ccc(NC(C2CCOC2)C)cc1Cl)N1CCC(CC)(CC)C1 CC1(NC(=O)CC2(O)CCCCC2)CCN(C(C2(O)CC2(C)C)=O)CC1 N1(C(c2c(F)cc(OC)c(N)c2)=O)CCc2[nH]nc(CNC(=O)C(C)(C)F)c2C1 C1(CNC(C=CCOC)=O)CC2(CCOCC2)CN1C(c1cc(O)nc(C)n1)=O C(=O)(C(CC(C)C)ONC(C1CC(=O)NC1(C)C)=O)NC(CCC)C(N)=O c1(CC)nnc(C)cc1C(=O)NC(c1ccccc1)CNC(C1CC(C)(O)C1)=O c1(SC)ccc(O)c(C(=O)N(C)CC2CN(C(C3CCCC3O)=O)CC23CC3)c1 C1(CNC(CC=C=C)=O)CN(C(=O)C(O)CCC)CCC12CCC2 CCC(N)CCC(=O)Nc1cccc(Oc2cccnc2)c1 Cc1cc(C)c(C(=O)NCC(C)CNC(c2cn(C(C)(C)C)nc2C)=O)[nH]1 C(=O)(C(C)CC(F)(F)F)N1CCC(C#C)(C(=O)Nc2ccccc2OC)C1 C1(O)(CNC(CCC(C)SC)=O)CCN(C(c2cn(C)c(C)n2)=O)CC1 C1(CC#C)CN(C(=O)NCCNS(=O)(=O)CC2OCCCO2)CCO1 C(=O)(C1=NN(CCO)C(=O)CC1)NCC1(O)CCN(C(c2c(C(C)=O)ccs2)=O)C1 C12(NC(c3ccnc(CO)c3)=O)CCCC1CN(C(c1ccc(F)c(F)c1)=O)C2 C1(NC(C(COC)NC(C(CCC)NC(C)=O)=O)=O)CCCCC1(C)C CN1CCCC(C(C)(C)C(N2CCC(F)(CNC(C3CC(O)C3)=O)C2)=O)C1 c1(OC)ccc(C)nc1C(=O)NC1(CO)CN(C(c2cc(C(F)F)[nH]n2)=O)C1 N1(C(CNC(=O)OC)=O)CCC(C)N(C(=O)CCc2cncc(Br)c2)CC1 Cc1nc2sccn2c1C(N1CCC(CNC(=O)C(O)C(C)(C)C)C12CCC2)=O C1(NC(c2cc[nH]c2)=O)CCCC2CN(C(C3(n4cnnn4)CC3)=O)CC12 C1(NC(c2nc(-c3cccnc3)cs2)=O)CCNCC1CO N1(C(CC(CNC(C2CC(OC)C2)=O)OC)=O)CC2CC(O)CC1C2.C1CC1 c1(CNc2c(OOC)cc(OCC(N)=O)cc2)ccc2oc(C)nc2c1 CC(CC(=O)NCC1CCC(NC(=O)CCc2nc[nH]n2)CC1)C(F)(F)F N1(C(COC(CC)CC)=O)CCC2(CO)CN(C(=O)C3=CCCOC3)CC12 c1(C(C2CCCC(C)(C)C2)NC(=NC)NCCCOC)ccc(F)c(F)c1 c1(C(=O)NCCC2CN(C(C#CC(C)C)=O)CC2C)noc2c1COCC2 C1(C#N)(C(=O)NCC(CNC(CC(C)OC)=O)OC)CC(=O)C1 C1(NC(C2(c3cc(C)on3)CC(C)(C)C2)=O)CN(C(=O)C(C)C)CC2(CC2)C1 C(=O)(C1=CC2CCCC12)NCC1(CNC(c2[nH]c(=NC)sc2)=O)CC1 Cc1ccc(C(=O)NC2(CO)CN(C(c3cc(C(N)=O)ccc3C)=O)C2)nc1C CCCC(C(O)C(=O)NCC(C)(C)CO)NC(C1(C)CCOCC1)=O N1(C(CCN(c2ccc(F)cc2)C(C(C)(C)C)=O)=O)CCCC(NC(N)=O)CC1 C(C(C)(C)CC(=O)O)NC(c1cnn(C(CC)C)c1-c1ccccc1)=O C12(NC(c3ccnnc3O)=O)CCCC1N(C(=O)C=CSc1nc[nH]n1)CCC2 C(=O)(C1=CS(=O)(=O)CCC1)N1C2CC(NC(=O)C=CCN3CCCC3)CC1CC2 CC1(C)CN(C(=O)C(Cc2ccsc2)NC(=O)CN2CCCC2=O)CCC1CO N1(C(C(C2CC2)OC)=O)CCC2(CCCC2NC(=O)CC2CCCC3CC23)CC1 C1(CNC(CSCC=C)=O)N(C(C2CCC(=O)N2CCC)=O)CCC1(C)C C1(C(=O)NC2CCN(C(C=CC(C)(C)SC)=O)CC2)Cc2nccn2C1 CC(CNC(C1CN(CC(F)(F)F)C1)=O)CN(C(=O)CCc1cn[nH]c1)C CN1C(=O)C(=O)N(CC(=O)NCc2cccc(N3CCNCC3)n2)C1=O C1(c2ccccc2)(COC)NC(=O)N(CC(=O)NC(c2cc(F)cc(Br)c2)C)C1=O N1(C(c2cnc(CC)o2)=O)C(C(=O)NC2CCNC2=O)CCC1C c1(C(=O)NCC2C(NC(C(C)CC3CCC3)=O)C2)ccnc(F)c1F C(CCCCCNC(C1CCCC1NC(=O)CCc1cnn(C)c1)=O)N(C)C c1(NC(C2C(C(=O)NCC(C)F)CCCCC2)=O)cccc2cccnc12 C1(CNC(CC(C)OC)=O)CC2(CO1)CN(C(=O)C(C)(F)c1ccccc1)C2 Nc1nc2c(cc1C(N1CC3CCC(C1)N3C(C1CCCCO1)=O)=O)CCCC2 N1(C(C2(C(N(C)C)=O)CC2)=O)CCC2CCCN(C(c3c[nH]c(=O)cn3)=O)C2C1 N1(C(COCCCCC)=O)CCC(N(CCC)C(C2(C)CCOC2C)=O)CC1 c1(C(=O)NC2CCN(C(C3CC(OC)C3)=O)C(C)C2)c[nH]c2cc(F)ccc12 Cc1ccc(O)c(C(=O)N(C)CCO)c1.C1(C[Si](C)(C)C)C(=O)N2CCN1CC2 C1(CN(C)C(C2CCCN2C(=O)Cc2cncs2)=O)CCCC2CC12 C(C(C)(C)C(C)(C)O)C(N(CCCNC(C1CC12CC2)=O)C(C)C)=O N1(C(C2(C)CCCN(C(CC(CC)(F)F)=O)C2)=O)CCOCC(C2CCC2)C1 C(C(C)(C)CNC(=O)CC1CC1(Cl)Cl)N(C(=O)Cn1ccc(C(F)F)n1)C NS(=O)(=O)c1c[nH]c(C(=O)NCC2CCCC(NC(C3(C(N)=O)CC3)=O)C2)c1 c1(N(CCN(C(c2cc(SC)ncn2)=O)C)C)nc2c(cc1C#N)CCC2 N1(C(c2cc(OC)nn2C)=O)CC(C2(NC(=O)Cn3cc(C(C)O)nn3)CC2)C1 c1(CC)c(C(=O)N(C2CN(C(=O)CC3CCCC3(F)F)C2)CCO)ccn1C CC1(C#CC(=O)N2CC3CCCC3(C(N3CCC(CN=[N+]=[N-])C3)=O)C2)COC1 C(CCCNC(C1CC(CCC)C1)=O)NC(CSCCCC)=O c1(OC)cc(OC)c(NC=O)c(OC)c1.C1(=O)C(C2CC2)NC2C(C2)N1 N#CC1(O)CC(C(=O)NC2CCN(C(c3csc(Br)c3)=O)C2)C1 C1(CC(=O)C(C2CC(N)C2)=O)CC2(CC2)C1.CC(C)CN(CC(C)C=O)C CCCCC(CNC(C1CC1C#N)=O)NC(c1ccoc1CC(N)=O)=O Cc1c(C(=O)NCC(C)CN(C(=O)CC(C)C(F)F)C)cc(C(C)C)n1C c1(NC(=O)CC2CN(Cc3ccc(Cl)nc3Cl)CCO2)cc([N+](=O)[O-])ccc1I N1(C(C2(C(N)=O)CC2)=O)CC(N(C(=O)COCC2CCC2)CCO)C1 Cc1onc(Br)c1C(=O)N(CCC(C)NC(C1CC1F)=O)C N1(Cc2c(-c3cn(CCC)nn3)cnn2C)CCCNC(=O)C1CC1CCCO1 N1(C(C)C)CC2CC1CN2C(=O)CN(C(=O)Cc1ccco1)C(=O)C1CC1 C(C(=O)NC(CC1CCC1)CO)(N(C(=O)C=CCO)C)C1CC1 N#Cc1ccc(C(=O)NCC(CNC(C23CCC(CC2)OC3)=O)C(C)C)c(O)c1 C(=O)(C#CC1CCCCO1)NCC1C(NC(c2ncc(C)cc2F)=O)CC1 C(=O)(C(O)C(F)F)N(CCN(C(c1cccc(Br)c1)=O)CC)CC CC(C)(O)C#CC(=O)NC(CNC(=O)C(C)(C)CC1CCCC1)CO N1(C(c2cncc(C)c2)=O)CCCC(C)C1CNC(c1cn(C)nc1Br)=O C1(CC)(NC(=O)Cn2ncnn2)CCN(C(C2CC2c2ccc(C)cc2)=O)CC1 C1(N(C(CC2(NC3CCCC3)CC2)=O)CCO)CC=C(C(=O)N(C)C)C1 CC(C)C(C(=O)NOCC(F)(F)F)NC(=O)CCCCC1CC1 N1(C(C=NOC)=O)CCC2(CC1)CN(C(c1conc1C1CC1C)=O)CCO2 CC1(C)CN(C(=O)C2=NOCC2)CCC1C(N1CC(O)(C(F)(F)F)C1)=O C1(NCC(C(=O)N(C)C)c2ccccc2)CCCNS1(=O)=O N#Cc1cc(Br)ccc1C(=O)NC1CCN(C(c2cnn[nH]2)=O)C(C2CC2)C1 C(=O)(CC(C)(C)CC(=O)N1CCC2C(NC(c3nnc(S)n3C)=O)CC12)OCC N1(C(CNC(N)=O)=O)CCC2CCN(C(=O)Cn3c(-c4cccs4)nnc3S)C2C1 n1(CC(=O)NCCN(CC=C)C)ncc(C#N)c1N C(N=c1[nH]c2c(c(=NC(C)C3CCOCC3)[nH]1)COCC2)C1CN(C(C)C)C1 c1(CCC)nc(C)c(C(=O)NC2CC(CCNC(n3nnc(=O)[nH]3)=O)C2)o1 N1(C(C(C)Cn2cccn2)=O)C2CCC1CN(C(=O)COCCCF)C2 C#CC(C)(C)C(=O)NCC(C1CC1)NC(=O)C(C1CCOCC1)F C1(NC(c2cscc2Cl)=O)CCN(C(c2cncc(Cl)n2)=O)CC1F CC(C)(C)C(C(=O)N1CCC(F)(CO)C1)NC(c1ccncc1O)=O C(=O)(C(C)(F)C(C)(C)F)N1CCN(C(c2c(C)oc(CO)c2)=O)CC1C1CCC1 C1(N(C)C)CCCN(C(=O)C(CC2CC2)NC(c2nnn(C)c2N)=O)C1 c1(C(=O)NC(CCOC)CNC(C2CC2c2cccnc2)=O)ccncc1F O=C(O)C(CNC(C1CCCOC1c1cnn(-c2ccccc2)c1)=O)CCO CC1CN(C(C2CC2C(=O)NC2CCN(S(C)(=O)=O)C2)=O)C1(C)C n1(CCN(CC(C2CCS(=O)(=O)CC2)(C)C)C)c(=O)oc2ccccc12 C1(CCNC(c2cc(OC)ncc2)=O)CN(C(=O)C(C#N)=CC(C)C)CCS1(=O)=O C1(C(=O)NC(C)CCN(C)C(c2cncc(N)c2)=O)CCS(=O)(=O)C1(C)C c1(C(N(CC(C)NC(=O)C(C)(c2ccccc2)N(C)C)C)=O)cncn1C C(C)(CCCCNC(c1cn(C)nc1C(C)C)=O)NC(COCC=C)=O CC1C(NC(=O)C(C)(C)CC(F)F)C2CCCCC12 N1(C(C2C(CCOC)C2)=O)CC(CCNC(=O)CC2CN(C)C2)C(C)C1 C1(CN=C(NC2C(C)C2)N(C)Cc2ccco2)C(F)(F)C12CCOCC2 O=C(CNC(=O)C(F)(F)F)N1Cc2ccccc2C(=O)N1 CC(C)C(C#N)C(=O)NC1C=CC(CC(=O)NCCC2CC(CF)C2)C1 C(=O)(C(C)C(C)COC)NCc1c(C(N(CCCC=C)CC)=O)cccn1 CCC(C)C(C)C(=O)Nc1cccc(C)c1C.n12cc(nn1)CN1CC2C1 C1(N)CC2CC(C1)N(C(=O)C=CC=C(Cl)Cl)C2.CCCCCC=CCC=O c1(C(C(=O)NC2CCC(CNC(C)=O)C2)O)ccc(F)c(F)c1.c1(C)cccc(N)n1 CCC(CCC(C)C)NCC(O)COc1ccccc1Br Cc1ccc(OCC(=O)NCC23COC(CNC(c4cnc[nH]4)=O)(C2)C3)cc1 O=C(C1CCCc2nnnn21)NC1CCOCC1NC(C1(C2CC2)CC1)=O C1(=O)C(C(C)(C)C)N1.c1(C(N2C(C)(C(=O)OC)CC2)=O)cc(OC(F)F)cc(F)c1 C(CC(C)C(=O)N1CCCC1(C)CCC(=O)NCC1(C)CCCC1)=CC CN1CCC=C(CNC(C2C=CCCN2C(=O)C(O)C(F)(F)F)=O)C1 c1(CNC(c2cccnc2)=O)ccc2c(c1)CCCC2NC(=O)C1CC1 c1(C(N(C2CCN(C(c3cccc(CO)n3)=O)C2)C)=O)ccc(C#N)c(Cl)c1 C1(C)(C(=O)NCC(N(C(c2cnc(OC)nc2)=O)C)C2CC2)CCCNC1=O C(C(C(C)C)NC(=O)C(F)(F)c1ccccc1)NC(CSCC#C)=O C1(CC(C)C)COCCN1C(=O)C(=O)NC1(CO)CC1(C)C C1(N(C(c2c(C)cco2)=O)C)CCCCC1N(C)C(C1(c2ccno2)CC1)=O c1(C(=O)NCc2cccc(NC(=O)C(O)Cc3cnc[nH]3)c2)ncc(F)cc1F CC1(C)CC(C(=O)Nc2cnc(Cl)c(F)c2)CN(C(c2cc[nH]c2)=O)C1 C1(CNC(=O)CSC(F)F)CC2(CC2)CN1C(c1c[nH]c(=O)cn1)=O CCC(CNC(c1ccsn1)=O)(CC)NC(C1CCN(C2CCC2)CC1)=O C1(F)(CC)CCN(C(=O)C(C)(C)CN(C(=O)CCc2nncn2C)C)C1 CCC(CC)(CO)C(=O)NCC(F)CNC(=O)CC1(C)CC1(Cl)Cl N1(C(C2C(COCC)C2)=O)CCC(NC(c2cscc2CC)=O)C12CC2 C1(CCONC(CN(C(CNC(=O)OC)=O)C)=O)CCOC(C)C1 C=CCC(C(=O)N1CCCCC(CC(=O)N(CC#CC)C)C1)C(C)C C(=O)(C#CC(C)(C)C)N(C)CC1CCN(C(c2cncc(NC)n2)=O)C1 Cc1cc(=NCc2cnc3n2CCC3)[nH]c(NC2C=CCCCC2)n1 C(C)(C)(C(C)CC(=O)N1CCC(C)(C#N)C1)NC(c1ccc(COC)o1)=O n1(C(C)C2CC2)cc(C2CNCC2OC(F)F)nn1 C1(OC)CC(CNC(=O)C(C(C)C)c2ccc(Cl)cc2)N(C(=O)Cc2ccsc2)C1 c1(NC(CCCCn2cc(C(COC)(C)O)nn2)=O)ccc(S(C)(=O)=O)c(C)c1 c1(C(=O)NCC(CC(C)C)NC(c2cccc(O)n2)=O)coc2c1C(=O)NCC2 N1(C(C(C)Oc2ccccc2C(F)(F)F)=O)CC(O)C(O)C1 C1(C(=O)NCC2CCN(C)C2)C2CC1N(C(=O)CC1(O)CCC1)C2 C(=O)(C1=Cc2ccccc2C1O)N1CCC(NC(C2=CCC(C)CC2)=O)C1C N1(C(=O)C(F)n2ccnc2)CCOCC(CNC(C2CC(OC3CC3)C2)=O)C1 CCC(CO)C(=O)NCCCCC(C)NC(c1scnc1C)=O C1(NC(C=C(C)C(F)F)=O)C(C)(C)CN(C(=O)C=CC2CCCN2C)CC1(C)C C1(CCOC)CN(C(c2sc(=N)[nH]c2C)=O)CCN1C(c1ccns1)=O C(CC)(CC)(CCNC(CCOCC#C)=O)NC(=O)CC(N1CCN(C)CC1)C N1(C(c2ccc(F)cc2)=O)CCC2(C1)CN(C(=O)CC1COc3ccccc31)C2 N1(C(C2C(=C)C2)=O)CCCC(C2(NC(C3CC(O)C3)=O)CC2)C1 N1(C(c2nocc2C)C(=O)NCCCCCC)CCc2c(Cl)cccc21 N1(C(C2(C)C(C(=O)OC)C2)=O)CCC2(CC1)CC(NC(=O)CCCC(F)(F)F)C2 C1(=O)C(C(C)CC)OC2(CCCC2)C(=O)NCCN1CCOC.CCNC CCC(CC)CC(=O)NCC=CC(N1CC=CCC1C1CC1)=O N1(C(=O)Cc2c[nH]ccc2=O)CC2CCC1CN2CCC(c1ccccc1)O N1(C(c2c(SC)n(C)nc2)=O)CCOC2CN(C(=O)C(C)=C3CC3)CC12 C1(NC)CCN(C(c2cccc(OCCO)c2)C(=O)Nc2cccc(Br)c2)CC1 C(=O)(CC(C=C)CCC)NC(CC=C)CNC(c1cc(C(C)C)oc1C(C)C)=O c1(CN=C(NCCOC)NC2CC2)cc(OC)c(O)cc1C O=C(C1=CC2(CCN(C(=O)CCc3cncs3)C2)C1)N1CCC(Cn2ccnn2)C1 CN1CCc2cc(C(=O)NCC3CC3CNC(c3cc(O)nn3C)=O)ccc2C1 C1(CNC(C2CCN(c3ccncc3)C2)=O)CC(O)(CNC(C2CC=CC2)=O)C1 C(=O)(CC(CC1CCCC1)C(F)F)N1CC(C)N(C(=O)CCCC(N)=O)CC1 C(=O)(C#CC1CCOC1)NCC(c1ccc(C)cc1)NC(C1CC(O)C1)=O C1(C(=O)NC2CN(C3CN(C(CCC#C)=O)C3)C(=O)C2)CC12CC(F)(F)C2.C1(C)CC1 N1(C(C(C)SCC)=O)CCC(O)(C2CCN(C(c3nc(OC)c(C)s3)=O)CC2)C1 C12(C(N3CC(CCNC(C4CC(C)(C)C4)=O)C3)=O)CCC(=O)N1CCS2 c1(CN2CC3(CN(C(c4csc(-c5ccccc5)c4)=O)C3)C2)ncc(Cl)cc1Cl C1(CNC(C=CC)=O)CC(NC(c2c(N)c(C(F)(F)F)nn2CC)=O)C12CCC2 C1(OC)CN2CCCC2(C(=O)NCC(C)(C)NC(=O)CC=C(Cl)Cl)C1 c1(CC(=O)NC(CCN(C(C=CCCC)=O)CC)C)noc2ccc(OC)cc12 c1(SC)ccc(O)c(C(=O)N(CCNC(C2CCSC(C)C2)=O)C2CC2)c1 C(c1c(Cl)cccc1Cl)=CC(=O)NC1C(F)CCN(C(CCOCCOC)=O)C1 c1(OC)cc(C(N2CCC2CNC(=O)CC23COC(C)(C2)C3)=O)ccn1 C(N=c1[nH]c(N2CCOC(CCO)C2)nc2cc[nH]c12)C1CC(CC)OC1 C(=O)(C(C)C(CC)CC)N1CCN(C(CNC(CCCC(=C)C)=O)=O)CC1 c1(OCC)ccc(Br)c(CN2CCC(C(=O)Nc3cc(OC)cc(C)c3)C2)c1F N1(C(NOC(C)(C)C)=O)CCCC(CNC(C2(C)C(SC3CC3)CC2)=O)C1 N1(C(C(CC)OC)=O)C2CCC1C(NC(c1cccc(N(C(C)C)CC)c1)=O)C2 c1(CN(C)C(c2csc(C(F)F)c2)=O)ccc(CNC(C2CCCCC2)=O)cc1 N1(C(c2c(CC)nc(C)s2)=O)CCP(=O)(OCC)CC1 C(=O)(C1c2c[nH]nc2CN1C(c1cnc(=N)[nH]c1)=O)NCC(C(=O)NC)(C)C c1(COC)nc(NCc2cccc(Br)n2)cc(N(C)CCn2ccnc2)n1 C1(NC(C=CC=CC)=O)CCSC12CN(C(=O)CC13CCC(CO)(CC1)CO3)C2 C(CN=c1[nH]n(C)cc1[N+](=O)[O-])(C(C)(C)C)NC(CC1CCC(C)(C)CO1)=O c1(C(=O)NCCOC2CCN(C(c3c(C)coc3C)=O)C2)cc2n(n1)CC(F)C2 n1(CC(=O)NCCN(C(=O)C(CC)NC(C)=O)CC)cc(CC2CC2)nn1 c1(C(=O)NCCC(C)NC(=O)CC(=O)c2cnn(C)c2)ccc(O)cn1 N1(C(c2cc(C(C)C)no2)=O)CCSCC1CCNC(=O)Cc1cnc[nH]1 CN1CC(NC(C2(NC(c3cc(=N)[nH][nH]3)=O)CC2(C)C)=O)C(=O)N1 C1(CC)(NC(=O)C(F)(F)c2nccs2)CN(C(=O)C(c2cncnc2)C)C1 C1(CNC(CCc2onc(C(C)(C)C)n2)=O)CCCCN1C(c1csc(O)n1)=O Cc1cc(C(=O)NC2CCCC(NC(=O)Cc3ccc(F)c(F)c3)C2)cc(C)c1 C(=O)(C(CO)C(C)(C)C)NC12CC(NC(C=CCCC(C)C)=O)(C1)C2 c1(CN2C(C(=O)NCC3CCCOCC3)CCC2C2CC2)cc2cccnc2[nH]1 Cc1cc(Cl)cc(C(=O)NC2CC(CNC(=O)C(N3CCN(C)CC3)C)C2)c1O CC(=O)CCCC(=O)NC1CC(F)CN(C(=O)CCN2CCN(C)CC2)C1 N1(C(c2ncn(C)n2)=O)CCC(O)(CC(N2CCC(F)(C(N)=O)C2)=O)CC1 CCC(CC)C(C)C(=O)N(C)CCN(CCCCCC(=O)Nc1cccc(C)c1)C N1(C(C2N(C(C3CCN(OC)CC3)=O)CC=C2)=O)CC2CCCC2C12CC2 N1(C(C(C)=C(CC)C)=O)C(C(N2CC(C(=O)OCC)C2)=O)CC1C C1(CNC(c2ccc(C)cn2)=O)CCC(C)CN1C(c1nscc1Br)=O N1(C(C(C)n2ccnc2)=O)CC(NC(c2nn[nH]c2Cl)=O)CC2(CCOCC2)C1 c1(C(=O)NCC(C2CCOC2)NC(c2nc(C(C)=O)sc2)=O)nnn2c1CCC2 CCC(CC(=O)N(C)CCN(C)C(C1CCSC1)=O)NC(=O)CNC(N)=O c1(NCC2(NC(C3(COC)CC3)=O)CC2)nccc(OC)n1 N1(C(C(C)S(C)(=O)=O)=O)CC2CCN(C(=O)C(C)(Cl)Cl)CC(C2)C1 C1(NC(C=C(C)C(F)F)=O)CCCC1CNC(c1ncoc1-c1ccco1)=O N1(C(CCSCC)=O)CCC(C)(C)C(C(=O)NC(c2ccco2)CO)C1 N1(C(=O)NC(c2cc(Cl)ccc2Cl)C)CCNCC2(C)CCCC12 C1(CC)CCCCN1C(=O)C(CNC(=O)CCCN(C)C(C)C)CC1CCCC1 C1(CCNC(C(=Cc2ccncc2)C)=O)CCN(C(=O)CN(C)C(C)C)C(C)C1 CCCCCC(O)C(=O)N1CC2C(CC(=O)NC3CCCC4(C3)N=N4)C2C1 CC(CCNC(=O)C(C)N1CCC1)N(C(=O)CSCc1ccco1)C C1(C)(CCOC)CN(CC(C2CCC(F)(F)CC2)C)CCO1 c1(C(=O)NCC(CNC(C(C)n2cccn2)=O)O)cc2c(o1)CCCNC2=O c1(N(c2ccc(C(CC)(C)C)cc2F)C(c2ccccc2)=O)ccc(Br)cc1Cl n12cc(nn1)C2=O.c1(C(=O)OCCCO)cnn(CCNC2CC2)c1.C1(C)CCC1 c1(C(=O)NCCN(C(C(CC)F)=O)CCOCCO)oc(C)nc1C Cc1cc(N)ccc1C(=O)NCC(C)(C)CN(C)C(C1CCN1C)=O c1(C(N2C(CNC(C(CC)NC(N)=O)=O)C(C)CC2)=O)cncc(N)c1C C12(NC(=O)NCC3C(C(C)(F)F)C3)CCCCC1C2(F)F C(=O)(C(C)C(O)CC)N(C(c1ccccc1)CNC(CCC(C)OC)=O)C C(=O)(C(C)CC(C)(C)C)NCCC(C)(C)NC(CSc1ccc(C)cc1)=O N1(C(c2cn(C3CN(C4C(C)OCC4)C3)nn2)c2ccccc2)CCS(=O)CC1 CC(N=c1ccnc(N2CCC3(CCCO3)CC2)[nH]1)c1cccc(F)c1 Cc1nc(C2CCCN(C(C3C4CN(C(=O)CC5CC5)CC34)=O)C2)oc1N(C)C CC(CC(=O)OC(C)(C)C)NC(=O)CC1CSCN1C(=O)C(C)(C)F C1(CCNC(c2c(CC)nn[nH]2)=O)CCCN(C(C2CC(C#N)(OC)C2)=O)C1 N1(C(c2ccn(C)n2)=O)CCC(CNC(=O)C(F)CC2CCC2)CC1 C1(C(N2C(CNCCC(CC)(C)C)CCC2)=O)CNC(=O)CN1C(C)=O CC1CC(NC(c2cccc(Cl)n2)=O)CN1C(c1cc(O)n[nH]1)=O C1(C(C)C)(C(=O)NC2CCCC2C(=O)N(C)Cc2ccco2)CCCC1 N1(C(C23CCCC2C3)=O)CC2CN(c3nnc(O)s3)CC2C1 N1(C(C)C)CCN(C(=O)NCC(C2CCOCC2)F)CC1C C1(CCC(=O)NCCNC(C2CN(C(c3cc[nH]n3)=O)C2)=O)CCCCC1 N1(C(C2(C)CCCO2)=O)CC2(CCCCN(C(c3cc4n(n3)CC(F)C4)=O)C2)C1 C(=O)(C(=O)N=c1nc(-c2ccccc2F)[nH]o1)N(CC(C)O)CC(C)O C1(CCN(C(=O)CC2(C)CCC2)C)CCCCN1C(c1ncoc1C1CCC1)=O C1(c2nc(CNC(COC)=O)[nH]n2)CCCN(C(C2CCCCN2C(N)=O)=O)C1 n1(CC(C)C(=O)N2CC(CC(C)NC(=O)CC(F)F)C2)ccc2ccccc12 S(=O)(=O)(c1cccc2nsnc12)NCC1N(C(c2cscn2)=O)CC2C(C)(C)C21 c1(C(=O)NC(=O)CCn2cc(C)nn2)cc(P(C)(C)=O)cs1.CC(=O)NC c1(CC(=O)NCC(CNC(C2CCN(CC)CC2)=O)O)nsc2ccccc12 N1(C(CC(C)C)=O)CCC2(CC1)CC2C(=O)N(CCC(O)C(F)(F)F)C(C)C c1(CN=C(NC(C#C)C)NC2CCCC2C(N)=O)cc(Cl)ccc1N(C)C N(C(=NCCOC)NC(c1cnn(C)c1)C)C(c1nc(CC)sc1)C c1(NC(C(=O)NCCc2c(C)ccnc2)=O)ccn2c(C(F)(F)F)nnc2c1 CCC1CCC(=O)N(C(C)C)CCN(C)C(=O)C1.C(=O)(NC)OC N1(C(COCC(C)C)=O)CCCCC(N(C)C(C2CN(C(C)C)C2)=O)C1 C1(NC(c2cnc(C3CCCC3)s2)=O)CCCCN(CCCC2CCOC2)C1 N1(C(c2ccc(Cl)c(F)c2)=O)CC(C2CCCCN(C=O)C2)C1.C(CCN)OC CN1CCCC1(C)C(=O)NC1CC(CNC(c2ncoc2C2CCCO2)=O)C1 C1(CNC(C2CC3CCC2O3)=O)CC12CCN(C(c1cc(F)ccc1F)=O)CC2 C=Cn1nncc1C(=O)NCc1cc(Br)n[nH]1.c12cn(nn1)C1CN(C1)C2=O c1(C(N2CC3C(CN(C(c4c(C)cccn4)=O)C)C3C2)=O)ccc2nncn2c1 Cc1nc(C)c(CC(=O)NC2C=CCN(C(=O)CC3(O)CCOC3)C2)s1 CC1(C)CN(C(=O)C(=O)NCC2CC(=O)N2)CC(C)(C)O1 S(=O)(=O)(c1ccc(NC2CCC(S(C)(=O)=O)C2)c(Cl)c1)NCC(C)C C1(NC(=O)CSc2ccsc2)CC2C(NC(=O)CCc3cccs3)C2C1 c1(C(=O)NC(C(C(C)C)NC(c2cc(C)nc(C)c2)=O)C)cccc2sccc12 c1(CN2CCC(=O)N(Cc3ccccc3)CC2)cc2cc3c(cc2[nH]1)OCCO3 C(=O)(CC1C(=O)Nc2c(F)cccc21)N(CCCN1CCCC1)C c1(C(=O)NC(CNC(c2c(C)coc2)=O)CO)ccc(-c2nnc(O)o2)cc1 C1(C(N(c2c(OCC(CCC)O)c[nH]n2)c2ccncn2)=O)CC2CCC(C1)N2 C12(CNC(CCCCCCC)=O)CCCCC1N(C(c1cc[nH]c1)=O)CCC2 Cc1csc2c(CC(N3CCCC3C(=O)N(C)C(C)C)=O)cccc12 N1(C(COCCCCC)=O)CCC2CN(C(c3cc(C#N)ccc3F)=O)C(C)C12 c1(C(=O)NCCCNC(C2(C(C3CCC3(F)F)=O)CC2)=O)ccc(CCO)cc1 C(=O)(CCCCCF)NC(C1CCN(C(c2ccc(CC)cc2)=O)C1)C Cc1ccnn1CC(N1CC(CNC(=O)C(F)C2CCC2)C1)=O C1(CNC(C(c2ccc(Cl)s2)C)=O)COCC1NC(C1(c2ccccc2)CC1)=O Cc1cc(C(=O)NC2CCN(C(=O)CCn3cccn3)C(C)C2)ncc1Br C1(NC(C2(CCOC)CCC2)=O)CCOC(NC(=O)COCCCOC2CC2)C1 CC1CN(C(=O)CN(C)C2CC2)CCN(C(c2cc(CO)on2)=O)C1 N1(C(c2c(OC)nsc2)=O)CCC(NC(c2nc(C(F)(F)F)cs2)=O)C(F)C1 N1(C(CCCCC)=O)CCCOC(CNC(c2n[nH]cc2Br)=O)C1 N1(c2nc(C)nc3c2cc[nH]3)CCC2(CN(C(C3CCCC3O)=O)CC(C)O2)C1 C(CN=C(NCC1(C)OCCO1)NCC1CCC(C2CC2)O1)SC1CCCC1 C(=O)(C1Cc2ccc(F)cc21)NC(CC1N(C(CNC(=O)NC)=O)CCC1)C1CC1 C1(NC(C(CC)N(C)C)=O)CN(C(c2c(Cl)cccc2Cl)=O)CC2(CCC2)C1 c1(CC(=O)NC2(C3CCCN3C(c3cnc(Br)s3)=O)CC2)nc2ncccn2n1 c1(CN(C)C(=O)Nc2c(C)c(F)ncc2)cc2n(c1)CCCC2 c1(C(=O)NCC(CC)(C)NC(c2n[nH]cc2[N+](=O)[O-])=O)ccc(C)c(Cl)c1F N1(C(C(C2(O)CN(C(C(CC)(F)F)=O)C2)F)=O)CC(=O)NC(=O)C1 c1(NC(CCSC)=O)ccc([N+](=O)[O-])c(C(N)=O)c1.N12CC3C(C3C1)C2=O CC1(C(=O)NC(CNC(C2CCCN2N=O)=O)C2CCC2)CS(=O)(=O)C1 C1(C(C(=O)NC(C2CCC2)C)C)CCCN(C(=O)C2CC2)C1 c1(CN2CC(NC(C3Cc4ccccc4C3)=O)C(F)C2)c[nH]c2ncc(Br)cc12 CC1CCC(CNC(=O)C(C)(C)C(F)F)CN1C(c1coc(C#N)c1)=O C1(NC(CCC2(C)CC2(F)F)=O)CCN(C(c2ccncc2N)=O)C1C1CC1 C(=O)(C(C)CCC(C)(C)C)N1C(CNC(C=CCOC)=O)(COC)CCC1 C12(NC(C3N(CC)CC3)=O)CC(CNC(=O)C=Cc3cnc[nH]3)(C1)OC2C C1(CC=C)(C(=O)NC2CCC2C(=O)OC)CN(C(=O)CCCNC(C)=O)C1 Cc1cccc(C)c1C(=O)NC1CC2(C1)CC2NC(=O)CC1(C)CC(F)(F)C1 C(=O)(C1=CC(O)CCC1)NC1(CNC(C=Cc2ccc(OC)cc2)=O)CC1 c1(OC)ccc(N(C(=O)COCCS(C)(=O)=O)CC)c(Br)c1F c1(NC(C(CC)C)CN(C)C)cc(C)nc(NCC2CCCOC2(C)C)n1 C1(NC(C2CCC(C(C)C)CC2)=O)CCN(C(=O)CC2COC(C)(C)C2)CC1O C1(C(C(=O)NC(COC)CNC(c2ncccn2)=O)OC)CCC(F)(F)CC1 CC1(C)OCc2c1n[nH]c2C(=O)NC1CCCC1NC(c1cnc(S)nc1)=O N1(C(CC(=O)OC)=O)CCC(C(=O)Nc2cncc(N(C)C)c2)C1(C)C C1(NC(C(CC)n2cncn2)=O)CCCCC1CC(=O)N(C1CCOC1)C C#Cc1ccnc(C(=O)NCCN(C(=O)CCc2nncs2)CC(C)O)c1 N1(C(c2c(C)nc(C(C)C)s2)=O)CCOCC(NC(=O)C(C)(O)C(C)C)C1 C1(F)(CNC(=O)Cc2cnns2)CCC(CNC(=O)CN2C(=O)CCC2=O)C1 c1(C(=O)NCC2N(C(C3C(C)OC3(C)C)=O)CCC2)c(F)ccc(F)c1Cl C1(CC)CN(C(=O)C=Cc2nccs2)CCC1NC(C1CC(C)(C(C)(C)C)C1)=O CC1(C)CC=C(C(=O)NCC23CCC2CN(C(c2ocnc2C2CC2)=O)C3)CC1 C(CCCCNC(C12CCC1CC2)=O)NC(=O)CCn1ccnn1 CC(C)(O)CC(=O)NC(C)(C(N1CC2CCC1C2)=O)C1CC1 C1(F)(CC)CCCN(C(=O)NCCOCCn2nc(C)cc2C)C1 N1(C(C(c2cccc(C)c2)C)=O)CC2(CNC(c3c[nH]nc3C)=O)CC(F)(C1)C2 C1(OC)CC(NC(=O)CCNC(C)=O)CN(C(=O)CC2CC(C)C2)C1 N1(C(c2c(C)cc(Cl)cc2)=O)CCC(C2CCOCC2)C1 C(=O)(C1=NN(CCO)C(=O)CC1)NCC(C1CCOC1)NC(C(C)(C)C(N)=O)=O C(=O)(C(C)(F)C(C)(C)F)N(C1CN(C(c2c(F)ccnc2F)=O)CC1(C)C)C C(=O)(C(C)(C)O)N(CCC(=O)NCC(CC1CC1)OC)CCCO Cc1ccc(C2(C(=O)N(C3CN(C(c4ncccc4N)=O)C3)C)CC2)c(F)c1 CCC(C)(Cc1cc(C)nc(OC)n1)C(=O)N(C1(O)CCCOC1)C1CCOC1 CCCC(C)(CC)C(=O)N1CC(C)C(C)(C(=O)N(CC(=O)OC)C)C1 N1(C(c2cc(CC)on2)=O)CC(F)(F)CC1CNC(C1CC12CCC2)=O c1(NC(C)=O)ccc(NC(=O)NCC2(C)CC=CCO2)c(C(=O)N(C)C(C)C)c1 CN1CC=CCC1CC(=O)NCCN(C(C1(CO)CC1(F)F)=O)C1CC1 c1(C(N2CCC(CNC(C(COC)OC)=O)CC2C)=O)ccc2ccccc2c1 C=CCC(CC=C)N1CCC(NC(c2cccc(Br)c2)=O)C1 CCCC(C)(O)CC(=O)N(C)CC1CN(C(=O)CC2(CO)CCCCC2)CCO1 C(=O)(CCCC(C)(C)C#N)N1CCC(C)N(C(c2cn(C)nc2Br)=O)CC1 C1(CCC(=O)N(CCCN(C(CSCCCC)=O)C)C)CCCCCC1 N(C(=NCC12CC(CO1)C2)N(C)Cc1ccnn1C)C(C)C Cc1nnc(CC(N2CC(CC(C)NC(=O)CCCC3CCCO3)C2)=O)o1 c1(C(C)C)ccc(C(=O)NCC2CC2CNC(C2CC(n3cnnc3)C2)=O)s1 N1(C(C(C=C)OC)=O)C2CCC(C2)C1CC(=O)NC1CCOC(C)(C)C1 C(CC(C)C(=O)NC(C1CCN(C(=O)CCc2cccnc2F)C1)(C)C)OC c1(CC(=O)NC2CC3(C2)CN(C(C2CCC4(CCC4)C2)=O)C3)cnc2n1CCOC2 Cc1cc(O)c(C(=O)NC2CCCC2CNC(=O)CN2C(=O)CNC2=O)nn1 C(=O)(N=c1ncn(C(F)F)[nH]1)N(C(c1ccccc1F)CC)C c12ccc(cc1)Cn1cc-2nn1.C(C)(C(=O)N(CCN(C)C)C(C)C)OCC C1(NC(CC(CC)(C)C)=O)CN(C(c2cc(C(F)F)ncn2)=O)CC12CCC2 C1(C(=O)N(C)CCNC(=O)Cc2ccc(NC(C)=O)cc2)(COC)CCC(=O)N1 C=CCC(C(=O)NCC(CCC)NC(c1[nH]c(=N)sc1CCC)=O)C(C)C c1(C(=O)NCC2N(C(C=C3CCN(C)CC3)=O)CC=C2)csc2nccn12 c1(CCC)nc(C)c(C(N2CCCC2C2(NC(c3cnn(C)n3)=O)CC2)=O)o1 c1(C(=O)NCC2(C)N(C(C3C(C)OC(=O)N3)=O)CCC2)ccc(N)c(Br)n1 C1(COC2(C)CCOCC2)CN(C(c2ccccc2)C(N)=O)CCCO1 C(N=c1nc2sccc2c(NCC23CCC(CC2)O3)[nH]1)c1ccc(=O)[nH]c1 C1(C(C)C)C(=O)N1.c1(OC)cc(C(=O)NC(CC2CCC2)CO)on1 c1(C(=O)NC2C(CNC(c3occ(C)c3)=O)COC2)cnn(C(C)(C)C)c1C C1(NC(C2N(C)C(=O)CCC2)=O)CCC2CCN(C(C3(n4ccnn4)CC3)=O)C12 C1(N2CCC(NC(c3cccc(OC(C)=O)c3)=O)C2)CCCNCCC1 N1(C(c2nc3ccccc3s2)C(=O)NCCCC)CCC2(CCCOC2)C1 CC1(C)CC(C(=O)NC2C=CCN(C(c3nccnc3C(F)(F)F)=O)C2)CC1 c1(C(N2C3CN(C(CC(C)=C(C)C)=O)C(C3)C2)=O)cc2ccc(N(C)C)cc2[nH]1 c1(C(=O)OC)ccc(NC(=O)C(O)Cc2ccc(Br)cc2)c(OC)c1 N1(C(=O)NCCC2C(C)C(=O)CC2)CCCC2(C1)OCCCO2 C(=O)(C(F)CC(C)(C)C)NCc1cc(C(N2CCCC(C=C)C2)=O)sc1 Cc1cc2n(n1)CCN(C(=O)Cc1ccc(-c3ccccc3)cn1)C2 c1(C(=O)OC)c(C)cnc2ccccc12.C1(C)C(=O)N1.C1(=O)CC2(CC2)CCN1 N1(C(c2c(OC)cnc(Cl)c2)=O)CCC(NC(=O)C(C2CC2)OC)C12CCC2 c1(OC)nccc(C(=O)NCCCCN(C)C(c2sccc2CC#N)=O)c1F Nc1ccc(C(=O)NC(C2CCOC2)CNC(C2CCCC2)=O)c(F)c1F C1(C(=O)NCC(CCO)OC)CCCN(C(C23CSCC2C3)=O)CC1 c1(NCC(=O)NC(CC)(C)CNC(C2CCN(C)C2)=O)ccc(Cl)cn1 C(C1(C)CCOCC1)=CC(=O)NC(C1CN(c2ccncn2)C1)C c1(C2C3OCC(NC(CC(C(C)C)O)=O)(C3)C2)c2ccccc2nn1C.C1C(=O)O1 CN(C)NC(=O)CCC(=O)NCC=CCNC(=O)CC1CCC(O)C1 CCCCC(CNC(c1c[nH]nc1CC)=O)NC(c1cc(C2(Cl)CC2)n(C)n1)=O C(=O)(C1CCCc2ccccc21)N1C(C)CCC(NC(c2c(CC)cco2)=O)C1 C1(CC)(NC(=O)C=CC(C)(C)C)CCN(C(=O)CCS(N)(=O)=O)CC1 c1(C(C)C)nc(CCN(C)C)n(-c2cccnc2OC(F)(F)F)n1 C1(NC(COCC=C)=O)CCN(C(=O)CN2CCOCC2=O)C(C2CC2)C1 c1(N(C)CC2CCCCN2C(=O)C#CC2CCCO2)ncc(C#N)cc1F N1(C(C2(COC)CC2(F)F)=O)CCC(F)(CNC(c2cccnc2C)=O)CC1 C1(NC(C(N(C(c2c(C)cns2)=O)C)C2CC2)=O)CCCCC1(F)F Cc1cc(C(C)C(N2CCCC(N(C)Cc3cnnn3C)C2)=O)cc(C)c1 Cc1c(NC(=O)OC(C)(C)C)cnn1CCCSc1cc(=N)[nH][nH]1 N1(C(OC(Cc2c(C)cccn2)=O)=O)CCN(C2CCOCC2)C(=O)C1 Cc1cc(C(=O)NCC(Cc2ccccc2)NC(c2cccs2)=O)cn1C(C)C C1(C)(CC(=O)N(CC(C)NC(COCCC#C)=O)C)CCS(=O)(=O)N1 Cc1cc(O)ccc1CC(N1CC2CC2(NC(=O)CCNC(=O)C2CC2)C1)=O C1(C(=O)NC2(CO)CC2)CC2(CC2)CN1C(=O)CC1CCCOC1 N1(C(Cc2ncc(C)[nH]2)=O)CC(CNC(c2ccc(Cl)cn2)=O)C(C)(C)C1 CCCCCCCCCCCC(=O)N1CC2CC1CN2C(C1CCOC(=O)N1)=O N1(C(C(C)CNC=O)=O)CCCCCC(NC(=O)COCCC2CCCC2)C1 C1(CC(=O)OC)CCCN(C(N2CCC3(CC2)CC3)=O)CC1 c12ncccc1C(=O)N2.C1(N(CCCC)C)CCN(C(=O)CSc2cccs2)C1 c1(C(=O)NC2CCN(C(C(CC)COC)=O)CC2)ccc(C(F)(F)F)cc1OC CCC1=C(C(=O)NCC2CCN2C(=O)CC(C)OC)CCCO1 C(=O)(CCCCC(C)(C)C)NC1CN(C(CC2N(CC)C(=O)CC2)=O)CC1O N12CCC(CC1)OCC1C(C1)C2=O.n1(CC(=O)N(CCOC)C)nccn1 C1(CNC(CC)=O)CN(C(c2ccncc2-n2cccn2)=O)CC1(F)F C1(F)(C(=O)NC2CCN(C3CCNC3=O)CC2)CCC(CO)CC1 N#Cc1ccc(C(=O)NCC=CCNC(c2ncsc2-c2ccccc2)=O)o1 N1(C(=O)CC2CN3CCC2CC3)CCC2(C1)CN(C(C1CCCCO1)=O)C2 C1(C2CCN(C(=O)C(C)(C)SC)CC2)(C(N(CC(CCC)O)C)=O)CCOCC1 C12(NC(Cc3c(C)noc3Cl)=O)CCCC1N(C(=O)CCC1CCC1)CCC2 c1(C(=O)NC2CCCC(CNC(C(C)=C(C)C)=O)C2)c(F)ccc(F)c1O c1(C(N(C(CC)C(=O)NOC2CC2)C)=O)cc(C)c(C)cc1C C(=O)(C1Cc2ccccc21)N1CC(CNC(C(C(CC)C)O)=O)C(O)C1 Cc1ccc(CNC(=O)NCCCC(=O)NC2CCN(CCCCO)C2)cc1 C1(CNC(c2cc(CC)[nH]n2)=O)CN(C(c2cc3ccsc3s2)=O)CC(C)(C)O1 c1(C(=O)OC)c[nH]c(C#N)c1C.C1(C)CCN(C(=O)CN(C)C)C1(C)C C(=O)(CS(=O)(=O)C1CC1)N1CC2C(CNC(c3ccc(C(C)C)s3)=O)(C2)C1 N1(C(c2cnc[nH]2)=O)CCC2CN(C(c3c(OC(F)F)cccc3Cl)=O)C2C1 CCC(CCC(=O)Nc1cnc(C)c(Cl)c1)NC(C1CC(Cl)(Cl)C1)=O C1(CC=C)(NC(=O)CCSCC(N)=O)CCN(C(=O)CN(C)C)CC1 C1(C)(COCC)CC(NC(=O)CCC=C(C)C)CN1C(=O)Cc1ccsc1 c1(C(N2CC(CSC)OCC2)C(=O)NCC2CC2)ccc2ccc(F)c(F)c2n1 N12CCCC(C1)C2=O.O=C1CCC(CCC(=O)NC2CC(N3CCC3)C2)C1 Cc1cnn2ccc(C(N3CCCC3C(C)NC(C34CC(C)C3C4)=O)=O)nc12 c1(C(N2CCCC3CN(C(C4CCC5CC45)=O)CC23)=O)[nH]nc2ncnc(O)c12 c1(N(CC#CC)C)nc(=NCC2CCC(F)C2)nc(N2CCOCC2)[nH]1 CC1COC2(CCC2)CN1C(C1C2CC3C(C2NC(C2(C#N)CC(=O)C2)=O)C13)=O C(=O)(C(C)C(CC)CC)N1CC(C=C)(CC(=O)N(C)Cc2cnn(CC)c2)C1 C(C(N=[N+]=[N-])C(=O)N(C)CC1CN(C(c2cc(C)cnc2C)=O)C1)OCC C(CNC(c1cccnn1)=O)(C(=O)N1CC(n2ccnc2)C1)N(C)C c1(-c2nn(C(COC)COC)c(CCC(F)(F)Cl)n2)cc(F)c(N)c(F)c1 CC1CCC(C(F)(F)F)CN1c1nnc(-c2ccc(Cl)cc2)n1CCC#CCO C1(C(=O)NC2CCC(NC(C3CC3c3cccs3)=O)C2)(CO)CC(F)(F)C1 N1(C(COc2c(Br)ccc(C)c2)=O)CCC2(CC1)CC(C(=O)N=c1[nH][nH]cc1Br)C2 C(CCOCCO)(C(=O)NCc1ccns1)NC(C(CC(C)C)O)=O c1(C(N2CC(CNC(CCC=C=C)=O)C3(C2)CCC3)=O)nc2nc(C)ccn2n1 c1(CCCC)ccc(C(N2C(CNC(c3n[nH]c(C)n3)=O)CC3CC23)=O)cn1 Cc1cccnc1C=CC(=O)NC1(CNC(c2ccnn2C)=O)CCCCC1C N12C3CCC1CC(C3)C(=O)C(=O)CN(C)CC2=O.N1(CC)CC(C2CC2)C1C1CC1 C#Cc1cc(C(=O)NCC(C)N(C(=O)C(C)(O)COC)C)ccc1C C1(C(=O)NCc2nc(CNC(c3n(C)cnc3)=O)sc2)CCC2(C1)CC2(F)F N1(C(c2n[nH]c(=N)[nH]2)=O)C2CCC1CN(C(C1COCC1C(N)=O)=O)C2 C12(NC(C(=O)NCCOCCOC)=O)CCCN(C(=O)CCC(C)(C)C)CC1C2 c1(NCC(CSC)OC)ccc(S(=O)(=O)NCc2cncs2)c(Cl)c1 Cn1c(C(N2CCCCC2CNC(C2CC23CC(O)C3)=O)=O)cnc1O c1(C(=O)NC2C(O)CCN(C(C(COC)OC)=O)C2)ccc(OC)c(OC)c1C C(CCCC(C)NC(=O)Cn1ccsc1=N)NC(C=C(C)Cl)=O c1(CCC(=O)NC(C)CNC(=O)CCOCC2CCCO2)cccc(F)c1Cl C1(C(N(CC(C)NC(c2c(CC=C)cccc2)=O)CC)=O)CC2(CCCC2)CO1 c1(OCC=C)ccc(Cl)c(C(N2CCCC(O)(CNC(c3ccc[nH]3)=O)C2)=O)n1 C1(C2CC2)(CNC(c2cccc(OCC#C)c2)=O)CCN(c2nc(C)ns2)C1 N=c1ccc(C(=O)NC2C=CC(CNC(c3cn(CC(F)(F)F)nn3)=O)C2)n[nH]1 c1(NC(C2CS(=O)(=O)CC2n2cccn2)=O)nc2cccc([N+](=O)[O-])c2s1 c1(C(C)NC(C(=O)NCCCC)CC)ccc(OC)cc1 c1(C(=O)NCCNC(C(C=C)(C)C)=O)cc(C)cc2c1NCCC2 Cc1cccc(N)c1C(=O)NC1CC(O)CN(C(=O)CC2CSCCS2)C1 C1(C(=O)NCC2C(C(F)(F)F)CCN(C(CSC)=O)C2)CCc2nn[nH]c2C1 Cc1cc(C)c(CNC(=O)CSCCNC(=O)CCC2CCC2C)s1 c1(NC(C2N(C(c3c(C)n(C)nc3)=O)CCSC2)=O)ccc(Cl)c(F)c1Cl N1(C(C(C=CCCC)O)=O)CC2CC(C1)CN(C(c1ccnc(Cl)c1OC)=O)C2 c1(C(CC)NC(c2nc(Cl)cs2)c2nnnn2C2CCOC2)ccc(OC)c(Cl)c1 CC(C(=O)NCCCOCCO)C(C)NC(c1nccnc1O)=O c1(CC(=O)NCC2CN(C(C=CCOC)=O)C3C2C3)c(C)nn(C)c1Cl C1(C(N2CCCC(C)CC2)=O)CCC(C)(C)N(C(=O)CCc2cnoc2)C1 c1(CNC2CC(C(N3C(C(=O)OC(C)(C)C)CC(F)C3)=O)C2)cc(I)ccc1F c1(CCC(=O)N(CCOC)CC2(CO)CC(Oc3ccccc3)C2)ccnn1C C(=O)(C(F)(F)C(F)(F)OC(F)(F)F)NC(CC=C)CNC(c1cc(Cl)c[nH]1)=O Cn1c(=O)oc2c(C(N3CCCC(CCCCSC(F)(F)F)C3)=O)cccc12 CCCCCC(C(=O)NCC1CCN(C(=O)CC2CCOCC2)C1(C)C)C(C)C c1(CC(=O)N(C(C)C(=O)N(CC)CCC(C)CCO)CCC)ccon1 Cn1cc(C=CC(=O)NCC(C2CCCC2)NC(c2cc(N(C)C)ccn2)=O)cn1 N1(C(c2cc(OC)ncc2)=O)CCC(C)N(C(=O)C(C)SC)CC1 C1(C2NC(=O)N2)(N(CC(O)CO)C(C)=O)CCN(C(=O)C(F)(F)c2csc(C)c2)C1 C1(NC(CCCC#CC)=O)CCOC12CCN(C(=O)CC1NC(=O)NC1=O)CC2 Cc1ccc(C(=O)NC2CC(CNC(=O)CC3CC(F)(F)C3(F)F)C2)cc1Cl C1(N(C(c2c(C)snc2)=O)C)CC2CC1N(C(c1cccn1C)=O)C2 N1(C(COc2ccc(C#N)cc2)=O)CCN(C(C2CCSCC2)=O)CC(O)C1 CCC(C)C(C)C(=O)N1CC(=C(F)CNC(c2ccc(SC)s2)=O)C1 Cn1c(C(=O)NC(C)(CNC(=O)C(C)(C)C#N)C2CCC2)ccc1[N+](=O)[O-] N1(C(C2CC(C)C2)=O)CCC2CN(C(c3cccc4c3OCC4)=O)CC12 N1(C(C(c2c(C)scc2)C2CC2)=O)CC(c2ccccc2)C1(C)C CSC1=C(C(=O)NCC2(O)CCCN(C(=O)C(c3cnn(C)c3)=O)C2)CCCC1 c1(C(=O)NC2CCCN(C(C3(NC(C)=O)CCCC3)=O)C2)n[nH]c2c1CCC2 c1(CN2CCC(C)C(N(C)C=O)C2)c2c(nn1C)CCC2 c1(C(=O)NC(CCNC(Cc2cccc(C)c2Cl)=O)C)n[nH]c2c1CC(C)(C)C2 C1(CC)C(NC(=O)C(C)O)CCCN1C(=O)CC1(COC)CC1 c1(C(=O)NCC(CC(=O)NC2CCN(C(N)=O)C2)OC)ccc(C#N)c(C)n1 C1(NC(c2ccc(NC(=O)Nc3c(OC)cccc3)cn2)=O)CCCCC1(F)F CN1CC(C(N2CCOC(CC(=O)NC34CC3COC4(C)C)C2)=O)CCC1=O CC1CC(NC(=O)Cc2ccc(F)c(F)c2)CN(C(c2cc([N+](=O)[O-])n[nH]2)=O)C1 CCC(CCCC(=O)NC1CCCC1(C)O)NC(c1ncccc1F)=O N1(CC)CC2(CCN(C(c3cnc(Cl)cc3C(F)(F)F)=O)CC2)C1 C1(NC(c2ccc(Cl)cn2)=O)CCN(C(c2csc(-c3ncc[nH]3)n2)=O)C12CC2 CC1OCCC1(F)F.C12CCN(C(=O)OC(C)(C)C)C1NC2 c1(C(N2CC3(C2)CN(C(c2ccc(O)nn2)=O)C3)=O)c(Cl)cc(Cl)cc1Cl c1(C(=O)NC(CNC(C=C(CC)C)=O)CO)cc2cc(C)ccc2[nH]1 C(=O)(CC(C)C(=O)NCCCCNC(c1cnccc1Cl)=O)OCC C1(O)(CNC(c2cc(=O)cco2)=O)CCCN(C(C2CC(O)C2)=O)C1 C(=O)(CC(C(F)(F)F)NC(=O)CC1CCC1)N1CCC(CSC)C1 N1(C(COCCCCCC)=O)CC(NC(=O)C(F)(F)Cc2ccccc2)C2CC12 CC1(F)CN(C(=O)CN2CCOCC2)CCN(C(C2(C(F)(F)F)CCCC2)=O)C1 C1(C2(NC(C3CCN(C(=O)c4ccon4)O3)=O)CC2)(OC)CCC1 N1(C(c2c(C)occ2)=O)CCC(C)(C)C(C(=O)NC(C)(C)CCF)C1 N1(C(CC(CC)NC(CCCC#C)=O)=O)C2CCC1COC2 CC1=CCCN(C(C2(F)CN(C(=O)CC3CCCC(C)O3)C2)=O)C1 c1(OC)ccccc1CC(C)(C)C(=O)NCC(CNC(=O)CCC1(C)CC1)CO c1(CNC2(c3n(C(C(=O)OC)C)nnn3)CC(C)C2)c(Cl)c(C)nn1C Cn1ncc(C(=O)NC(CC2CCC2)C(=O)NC(c2ccccc2)CF)n1 C(=O)(CCS(=O)(=O)CC(C)C)N1CC(NC(c2ccnc(C)c2Cl)=O)C1 C(=O)(C(C)SC)N(CCNC(C1(SCC)CC1)=O)CCOCCO N1(C(c2c(OC)scc2)=O)CCN(C(=O)C(C)OCC(F)(F)F)CCC1C C1(OC)NC(CNC2CC(c3ccc(F)cc3)C2)CCC1Br C(CN(C(=O)C(c1ccccc1Cl)O)C)(CO)(CO)NC(CC1CC(=C)C1)=O c1(CCC)ccc(C(N2CC(C(=O)NCc3ccccc3F)C(O)C2)=O)cc1 C1(C)(C(=O)NCC(CC)NC(=O)CCN2C(=O)CCC2=O)C=CCCC1 CC1CC(C)C1CNC(=O)COc1ccccc1.c12cn(nn1)CC(=O)N2 N1(C(C2CC(CCC)OCC2)=O)CC=C(CCNC(c2cn(C)cc2C)=O)CC1 C1(C(=O)NCC(COCC)O)CN(C(=O)CCCC2CCCO2)C(C)(C)C1 C1(C(N2CC(OC(=O)NC)C2)=O)CCN(C(c2cc(C)[nH]n2)=O)C1C C1(CNC(C2=NOC(C)C2)=O)C(C2CC2)CCN1c1nnc(C(N)=O)s1 C=C1Cn2c(C(N3CC4CCC4(CNC(c4ncn(CC)n4)=O)C3)=O)nnc2S1 c1(CC(=O)NC(CC)(CNC(C2CC3C=CC2C3)=O)CC)ccc(F)c(OC)c1 C1(NC(c2cc(C)ns2)=O)CC(C)CN(C(c2ncoc2C(C)(C)C)=O)C1 Cc1cc(C(N2CCCC(F)(CNC(C3CCN(C)C3=O)=O)C2)=O)cc(C)c1F c1(OCC=C)ccccc1C(N1CCC(C(=O)NC(C)CCC(=C)C)CC1)=O c1(C(N(CC(CC)NC(c2ccsn2)=O)CC)=O)cccnc1SC(F)F c1(C(C(=O)OC)C)cccc(C(=O)NC(C2CCCO2)Cc2ccccc2)c1 CC(C)C(C#N)C(=O)NCC(C)N(C)C(c1ccc(C(F)(F)C(F)F)cn1)=O N1(C(c2c(OC(F)F)cc(C)s2)=O)CCN(C(C2CC(C)C2)=O)CC(O)C1 c1(C(=O)NC2C(C)(C)N(C(=O)Cc3ccsn3)CC2)noc2c1COCC2 CC(C)CCCC(=O)NCC1CN(C(=O)C2=CCCCO2)CC1O C(=O)(C1CCC(=O)c2cccn21)N1CCN(C(C(C(C)C)NC=O)=O)CC1C C1CN=C(N2CCOC(Cc3cccs3)C2)NCC1.N1(CCC)CCCCC1C Cc1nocc1CN(C(=O)C(C1(O)CCC1)NC(=O)C(C1CC1)N(C)C)C Cc1c(C(=O)NC2CCN(C(=O)C(C)C(C)C)C2)cc([N+](=O)[O-])cc1Br C=Cc1cnn(C)c1C(=O)NCC(C)NC(c1ccc(-c2ccccc2F)[nH]1)=O N1(C(C2CCC(C(=O)O)C2)=O)CCC(CCCCOC(C2CCCC3CC23)=O)CC1 C12(C(=O)NCC3(CC(=O)NC(c4nc(C)on4)C)CC3)CCC(CC1F)C2 C1(NC(C(CCCC)C)=O)CCC2(CC1)CN(C(c1cccnc1OCC)=O)C2 C1(NC(c2ccc(C)s2)=O)CCN(C(C2CCC2c2nnc(S)n2C)=O)CC1(C)C C1(C(=O)NCCS(=O)(=O)NC)N(C(=O)CCCC#N)CC12CCCC2 c1(C(N2C(CN(C(C(n3cc(Cl)cn3)C)=O)C)CCC2)=O)nnn(C)c1N C1(NC(C(C)SC(C)C)=O)(CNC(=O)CCC2CCCCO2)CCOCC1 N1(C(c2cnc(-c3cnccc3)s2)c2nnnn2C2CC2)CCCN(CCO)CC1 C(=O)(C1=CS(=O)(=O)CCC1)N(CC(C)N(C(=O)Cc1cn2c(n1)CCCC2)C)C CCC(C)(COC)C(=O)NCC(CO)NC(=O)CN(C)CC1CCCCC1 c1(C(N2CCC(CCNC(C=CC(N)=O)=O)C2)=O)cnc(O)c(Cl)c1 CC1CN(C(C2CN(C(c3cc(CO)oc3C)=O)CC2(C)C)=O)CC1(C)CO N1(c2cc(C)nc(CO)n2)CCC2(COC(CNC(=O)C=C3CCCCC3)C2)C1 C1(C(C)CN(C)Cc2c(C)nn(C(F)(F)F)c2C)CCn2ccnc2C1 Cc1cnc2n1CCC(C(=O)NC1(CON)CCN(C)C1)C2 Cc1ccc(O)c(C(=O)NCCCCCCNC(c2cc(C)[nH]n2)=O)c1 c1(COC)nn(C)cc1C(=O)NCC1C=CCN1C(=O)C(O)COC N1(C(c2on(C)c(=O)c2)=O)CC2(CCN(C(C3(c4ccccc4)CC(O)C3)=O)C2)C1 c1(C(N(CC(C)(C)NC(C23CCCC2C3)=O)C)=O)n[nH]c2c1CCC2 Cc1cc(C(=O)NC(C)(CNC(=O)CC2CCCC23CC3)C(C)C)[nH]c1C CCC(C)(C)C(=O)C(=O)N1C(C(=O)O)CCC1C1CCC1 C(C(O)C(=O)NCC(C)NC(=O)CSC1CC1)=CCCC N1(C(N(C)C2CC2)=O)CCN(c2ccc(C(F)(F)F)nn2)C(CO)C1 c1(CC(=O)NCCOC)ccccc1SC.C1(C(=O)N)CCC1C(=O)OC.C1C(=O)N1 C(Cn1ccnn1)(C(=O)NOCCF)NC(C1CCNC1=O)=O c1(C(=O)NC(C)C)ccc(C(=O)NC(C)(CNC(C2COC2)=O)C(C)C)cc1 c1(CNC(CC(c2ccc(C)cc2)C)=O)cccc(O)c1C C1(CC=C)(C(N2CC(CCNC(=O)CNC(=O)C(F)(F)F)C2)=O)CC=CC1 CCCC(C(=O)NCC)N(C)CC.C1(C=O)(N(CCCN(C)C)CC(C)C)CCC1 C1(C(=O)NC23CC(C(=O)NCCN(C)CCO)(C2)C3)CCC(C2CC2)C1 c1(C(=O)NCC(=O)NC(C2CCCC2)CCCOC2CCC2)cccnc1 N1(C(c2cc(CC)[nH]n2)=O)CCC(C)(NC(=O)C(C)COC(C)=O)C1 C1(CNC(c2cccc(C(C)C)n2)=O)CN(C(=O)C(O)CC(N)=O)C2(CCC2)C1 c1(C(c2nnnn2CC2CCCO2)NCCCn2c(C)ncc2)cccc(C(C)C)c1 N1(C(C2C(C=C)C2)=O)CC(NC(c2ccccc2SC)=O)C(c2cncn2C)C1 C1(C(=O)NCCCc2n(C)ncn2)CN(C(=O)Cc2ccc(Br)s2)CCC1F c1(OCC=C)ccc(Cl)c(C(=O)NCC2CCN2C(c2cc(CCC)[nH]n2)=O)n1 C(=O)(C(C)(C(F)F)c1ccccc1)OC(C)CC(C1CC1)NC(=O)OC(C)(C)C c1(C(=O)NCC2C(C)(C)N(C(=O)Cn3ccnn3)CC2)ccc(N)c(F)c1F Cc1[nH]c2ncccc2c1C(=O)NCC1CN(C(=O)C(C)CS(C)=O)CCCO1 c1(N2CCC(N3CC(C)(C)C3)CC2)nc2c(c(=NCC(Cl)Cl)[nH]1)CCCCCC2 N1(C(C2N(C(C)C)C(=O)CC2)=O)CCCC(O)(CCNC(c2ccnnc2)=O)C1 C#CCCCC(C)C(=O)NCC1C(C(=O)N(CCC(C)(C)O)C)C1(C)C C12(CNC(c3cc(CCC)n(C)n3)=O)CC(CO1)N(C(=O)Cc1n[nH]c(=NC)s1)C2 c1(CNC(CSCC=C)=O)nc(CNC(=O)CNC2CC2)cs1 CCC(CC)C(=O)NCCCC(=O)NC1(C(=O)NC(C)(C)CC(N)=O)CCC1 N1(N2C(c3ccc(F)cc3)COCC2)CCc2cc(-c3ccccc3)[nH]c2C1 N1(C(CC2CCC(=O)O2)=O)CCCC(NC(=O)CSCc2cccnc2)C1 c1(C(=O)NCCC(C)N(C(=O)CSc2n[nH]c(O)n2)C)cc2cccc(F)c2o1 C1(CC(=O)NC2C(NC(c3c(COC)noc3)=O)CCC2)CCOCC1OC C1(NC(C2(COC)C=CCC2)=O)COCCN(C(C2(N(C)C)CCCCC2)=O)C1 N1(C(C2(CSC)CC2)=O)CCC(C)(C)C(C(=O)NC2CCCC2F)C1 N1(C(C(C=CCCC)O)=O)CCC(C)(C)C(CNC(=O)Cc2ccsc2)C1 N1(c2nc(C)cc(OC)n2)CC2(CCOCC2)CC1CNC(C1CCCOC1)=O CC1(NC(=O)CCC2CC=CCC2)CCCN(C(C2CC2c2ccccc2)=O)C1 c1(C(C)C)cccc(OCC(N2CC3C(CNC(=O)Cc4cnc[nH]4)C3C2)=O)c1 C1(CCC)(NC(=O)CCCC2OCCO2)CCN(C(c2cnc(C)nc2)=O)CC1 n1(CC(=O)OCC)cc(C(=O)NCC(O)CN(C(=O)C(C)n2cncn2)C)nn1 N1(C(=O)OC)CCCC(N(S(C)(=O)=O)C(C2CC2(F)F)=O)C1 N1(C(C2(C)CCCC2)=O)CCCC(C2CCN(C(=O)C(F)OC(F)(F)F)CC2)C1 C(=O)(C1=NOC2(CCC2)C1)NC(C)CCNC(C1(C)CCC(C(C)(C)C)OC1)=O C(CCCC(=O)NCC(C)=CC1CC1)N(C(c1n(C(C)C)cnc1)=O)C Cc1c(CC(c2nnnn2C2CCCCC2)NCCCCO)cccc1C(F)(F)F C(CC(F)F)(C(=O)N1CCCOCC1)NC(c1cc(CO)cc(F)c1)=O c1(C(N2CC(C)(CC(=O)NCCN3CCCC3)C2)=O)nnc2ccc(Cl)nn12 C#CCC(O)C(=O)NC1CCN(C(c2ccn(C3CC3)n2)=O)C1C CC1(C(N2CCC(CNC(c3cc(F)ccc3Cl)=O)C2)=O)CCC(F)(F)C1 CC1CCC(CNC(=O)C2=CCCOC2)CN1C(=O)Cc1cncnc1 C1(NC(C2C(CNC(c3ccc(C)nc3)=O)CCC2)=O)CC=C(C(C)C)CC1 C12(NC(C3CC(=C)C3)=O)COC(C1)C(NC(=O)CCC(C)N1CCOCC1)C2 C(=O)(C(C(C)(C)C)NC(=O)CC(F)(F)CC)N1CC(CC)(CC)C1 N1CC2(CCN(c3cc(O)nc(=O)n3C)CC2)CC1C.n1(C(C)C)ncc(C)n1 CC(C(=O)N=S1(=O)CCC2(CCCN2)C1)c1cccs1 Cc1ccc2scc(C(N3CCN(C(=O)CC4CCC5CC45)C(C)C3)=O)c2c1 C1(CNC(CSc2n(CCC)c3c(n2)cccc3)=O)Cc2cc(C)cc(Br)c2O1 c1(C(N2C(C3(NC(C4CCOCC4)=O)CC3)CCC2)=O)cc2ccccc2[nH]1 c1(N(C(C(=O)NCCCSC)C(C)C2CCCOC2)C)cc(C)c(Cl)c(C)c1 N1(C(C(CC#C)C)=O)CCN(C(c2cnc(N)c(Cl)c2)=O)CC1CCC O=S(=O)(c1cccnc1NCc1ccc(C2CC2)cc1Cl)N1CCSC(F)(F)C1 c1(C(=O)NCC2(C)N(C(C(F)=C(C)C)=O)CCC2)ccnc2[nH]c(C)nc12 C(=O)(C=CS(C)=O)NCCNC(C1CN(C(C2C(C)OCC2)=O)C1)=O c1(C(=O)NC23C(NC(COCC=C)=O)CC(CC2)C3)c(C)ccc(F)c1N Cc1cccc(C(=O)NCC2CC2NC(c2cc(F)ccc2OC(C)C)=O)c1O N1(C(C=CCOC)=O)CCC(C(=O)NCC(O)CN(C)C)C1.C(C=C)=C C(=O)(C1=C(C)CC(C)(C)CC1)NC1C(CO)CCN(C(C2C(=C)C2)=O)C1 c1(CC)ccc(CCCC(=O)NCC(O)CNC(c2coc(OC)n2)=O)cc1 c1(CNc2nccc(-c3cn(C)nc3)c2)cc(S(C)(=O)=O)ccc1O C1(NC(C=CC=CC)=O)CCN(C(C2CC2C(=O)OCC)=O)CC1F CC1OCCC1C(=O)C(=O)N(CCNC(=O)CC1CCCC1O)C1CC1 C12COCCN1C2.C(C)(CC(=O)N1CC(CO)(NC(=O)CC2CCC2C)C1)OC C(C(C(=O)NC1CCN(C)CC1C)C(C)C)NC(C1(COC)CCC1)=O c1(CC(=O)NC2CC(CCNC(c3cc(OC)no3)=O)C2)cc(F)ccc1F C(C)(CC1CCCCC1)(C(=O)NC(C)CCN(C(=O)Cn1nncc1C)C)OC c1(OC)ccc(F)c(C(=O)NC2(CO)CN(C(C3(OC)CCOC3)=O)C2)n1 c1(C(=O)NCC(CNC(c2cn(CCOC)nc2)=O)O)ccc2c(c1)CNC2=O CC(C)C(O)CC(=O)NC1CCCN(C(c2coc(C(F)F)c2)=O)CC1 c1(C(=O)NC2CC(NC(C3(C)CCC(C)C3)=O)C2)n[nH]c2cccnc12 c1(OC(C)(C)C)cccc(C(c2nn[nH]n2)NC(C2C(C)(C)C2(F)F)=O)c1 CCC(C(=O)NCCN(C)C(C1CC(C)(F)C1)=O)OC1CCCC1 n1(CC(=O)NC2C(OC)CN(C(c3cnc[nH]c3=N)=O)C2)cnc2c1CCCC2 c1(C(N2CC(NC(C(C)SCCCC)=O)(CO)C2)=O)c(C)cccc1F C=Cc1ccc(CC2(OC)CN(C(C3CC(C(C)(C)C)C3)=O)C2)cc1 CN1CCC(C)(C(=O)NC2(C)CCCN(C(c3nscc3N)=O)C2)C1=O N1(C(C(C)CC2CC2)=O)CC(C(=O)NC(C)(C)CC2CCCC2)C(F)C1 CC(CC(=O)NCC(C)NC(c1cnn(-c2ccccc2F)c1)=O)C(F)F C1(COC)(NC(C2CC2c2cc[nH]n2)=O)CCN(C(=O)Cn2nc(C)cc2C)C1 C(=O)(CCC(C)C)NCC1(COC(CNC(CCN(CCCC)C)=O)(C)C)CC1 C(=O)(CCCC(C)CC)NC(CC#C)CC(=O)NCCCN1CCOC1=O N1(C(CCC#C)=O)CCC2(CC2)CC1C(=O)N(C(CF)CF)C N1(C(c2nc(C)[nH]n2)=O)CCOCC12COCCN(C(=O)C(C)(C)C1CCC1)C2 Cc1ccc(C(N2CCC(C)C2CNC(=O)Cc2cc(Cl)ccc2F)=O)cc1Cl C(=O)(C(C)N=c1cc[nH]cc1)NC1CCN(C(C(C)CF)=O)C1(C)C C1(COC)(NC(=O)Cc2ccsc2)CCN(C(c2cn(C3CC3)cn2)=O)C1 C#Cc1cccc(C(=O)NCC(C2(O)CN(C(=O)C=C3CCC3)C2)(C)C)c1C c1(C(=O)Nc2cccc(CNC(c3cc(C)oc3C)=O)c2)[nH]c(=N)ccc1C CC1(CNC(c2ccccc2C(N)=O)=O)CCCN1C(=O)COC1CC(F)(F)C1 c1(N(C(=O)CCCc2ccc(Br)s2)C(c2cccs2)C)nc(Cl)ncc1Br CC1(C)CCN(C(C2CC3CCC2CC3)=O)C1CNC(c1ccc(N)c(Cl)c1)=O CC(C)(C(=O)NCC(O)C(=O)N1CCCC1CN=[N+]=[N-])C1CC1 c1(CNC(CC2(C)CCN2C(=O)COc2ccsc2)=O)n[nH]c2c1CCC2 C1(NC(CCCC2(NC(C(C)C(C)(C)C)=O)CCC2)=O)CCCCN(C)C1=O N1(C(C(C)(C)c2ncco2)=O)CCN(C(c2cccc(=O)o2)=O)CC12CCC2 Cc1nc(C(=O)NC2CCC2NC(=O)COC2(C)CCCC2)c(C(F)(F)F)[nH]1 CC(C(C)(C)NC(c1cnn(-c2ccccn2)c1)=O)NC(=O)C(C)N(C)C C1(C2CCCCC2)(NC(C2CC(C(=O)N3CC4CC4(CO)C3)=NO2)=O)CC1 N1(C(c2ccno2)=O)CC2COCC(C1)N2C(c1cc2cnccc2[nH]1)=O C(=O)(CC(C)(C)C=C)N(C1CCN(C(c2ccc(F)c(CC)c2)=O)CC1)CC#C C1(CC(=O)NC2CC(NC(C=Cc3n(C)cnc3)=O)C2)CCC2(CC1)COC2 C#Cc1ccc(C(N2CCC(NC(=O)Cc3c(C)n[nH]c3C)C(O)C2)=O)cc1Cl c1(-c2c(C(=O)NCCc3cc(OC)cc(F)c3)nccc2)ccccc1[N+](=O)[O-] C1(C(N(CC(O)C2CCC2)C)=O)CCC2CCC1N2C(c1ncn(C)n1)=O O=C1NC(=O)C2(CCCCCC(c3ccc(Cl)cc3)CC2)CCN1 N1(Cc2cc(OC)c(Br)cc2)CCC2(CC1)CC2C(=O)NCC1(C)OCCO1 C1(NC(=O)CSCC(N2CCCC2)=O)COCC1NC(c1ncc[nH]1)=O Cc1cc(-c2cn(C3CCN(C(c4c(C)ccn4C)=O)CC3)nn2)ccc1F c1(C(=O)NC(CC)CNC(=O)CC(C)(C)OC)cc(F)cc2cccnc12 C1(COC)CN(C(c2nnn(C(C)C)c2C)=O)CCC1NC(=O)CSC(F)F Cc1cccnc1C(F)(F)C(=O)N(c1ncc(C(F)(F)F)cn1)C1CCCNC1 C(=O)(C(C)(C)CC(C)(C)C)NC(CC)CN(C)C(C1COC2(CO)CC1C2)=O C1(C(=O)NC(C(C(=O)OC)C)C)CCN(C(=O)C=C(C)C(C)(C)C)C(C)(C)C1 C=CCC(C(=O)NCC1CCC(C(=O)NC(c2cn[nH]c2)C)C1)C(C)C n1(CC)cnc2c1C1=NC(=NCC3COCCN1C3)N2.c1(SC)ccccc1Br c1(C(C)NC(C2(C)CCN2CC2CC(F)C2)=O)cccc(C(F)(F)F)c1F CC1C(=O)OCCCC(=O)N(C)C2C3CN(C1=O)CC32.C(C)(C)(C)SC(C)(C)C C(=O)(CC(C)(C)C(F)F)N1CCCC(CNC(C2OCC(C)(C)C2)=O)C1 N1(C(=O)NCCc2ccc(Cl)cc2C(F)F)CCCC1C1CCCO1 c1(C(C)=O)cc(NCCCNC(C2CCC(=O)N2)=O)ncn1 c1(CC(=O)NC(CCCNC(CC=C)=O)C)coc2cc(Cl)ccc12 c1(C(N(CCN(C(c2c[nH]nc2C)=O)CC)CC)=O)ccnn1C(C)(C)C c1(C(=O)OCCc2ccccn2)ccc(NC(c2ccon2)=O)cc1 c1(N2CCC(NC(C(n3ncc(C)c3)C)=O)C2)cc(O)nc(C)n1 c1(C(=O)NCCCN(C(C2C(C=C)OCC2)=O)C(C)C)cnc(O)c2cncn12 Cc1cccc(CN(C(c2cnc(C(C)(C)O)s2)=O)Cc2ccccn2)c1 c1(-c2[nH]nc(C(CC)CC)n2)nn(C)c2ccccc12 C(=O)(C(CC)CCCC)NC(CCC)CNC(c1ccc(C)nc1O)=O N1(C(C2CCN(C(C)=O)C2)=O)CC(NC(=O)CN2CCC(C)(C)C2)CC(F)C1 N1(C(c2n(C)c(C(N)=O)cc2)=O)CC2CCC(C1)C(NC(=O)C(F)C(F)(F)F)C2 c1(C(=O)NC(CC)(C)CN2CCN(C)CC2)cc(OC)c(C)cc1F CC1CN(C(c2c[nH]c(Br)c2)=O)CC2(CCN(Cc3cc(Cl)ccc3Cl)C2)O1 N1(C(c2cc(OC)n[nH]2)=O)C(C)C2CC1C2NC(=O)C(c1ccnn1C)C C=Cc1ccc(C(N2CC(NC(=O)CCC3C(=O)ON=C3C)C(C)(C)C2)=O)cc1 C1(=CC(N2CC3C(CNC(=O)CN4C(=O)CCC4=O)(C3)C2)=O)CN2CCC1CC2 C(=O)(C#CC(C)(C)CNC(=O)C(C)CC(C)C)NCCC(=O)NCC c1(NC(C2(C)C(C(=O)OC)C2)=O)cc(O)c(Br)s1.c1(C(=O)C2CC2)ccc(Br)cn1 N12CC3CC(C1C3)N(C)C(=O)CC1CC(C1)C2=O.c1(CC(=O)OC)nocc1CN C1(N(C)C)CN(C(C2C=CCCC2)=O)CCC1CNC(=O)CC1CC=CCC1 Cc1ncn2ccc(C(N3CCC(O)(C(C)NC(=O)CCCC4CC4)C3)=O)cc12 N1(C(CC(=O)OCC)=O)CCCCC1C1CN(C(=O)C(C)(C)COCC)C1 c1(C(N2CC=CC(NC(CCCC#C)=O)C2)=O)ccn2c(C)cnc2c1 C1(C(N(CC(C)(C)CNC(c2ccnc(CO)c2)=O)C)=O)OCC2CCCC12 C1(OC(C)C)CCCN(C(=O)CCCCN(C)C(c2c[nH]nc2C(C)C)=O)C1 N1(C(c2ccc(C#C)o2)=O)CCN(C)C(CNC(=O)C=CC(F)(F)F)C1 C1(C(N(CC(CN(C)C(c2n[nH]cc2[N+](=O)[O-])=O)O)C)=O)CCCCC(F)(F)C1 C1(CNC(CCCCC)=O)COCCN(C(=O)C(C)Cc2c(C)nn(C)c2C)C1 N1(C(C(CCC)O)=O)CCC(C2CC2)C1CNC(c1cccc2nsnc12)=O CCCC(CNC(c1cccc(O)c1F)=O)C(=O)N1CC(C)CC1CC C(C(C(=O)NCc1cnc(F)c(C)c1)C(C)(C)C)NC(C(CCCC)O)=O C(CCCCC(=O)NCC(C)C1CCC1)NC(Cc1c(C)noc1C)=O C#CCCCC(C)C(=O)N1CC2=C(C1)CN(C(=O)C(C)(C)CF)C2 C(c1ccccc1C)=CC(=O)NCC1(CNC(C2C=C(C)CS2)=O)CCCCC1 C12(N(C(=O)C#CC3CCOC3)CCCCNC(C(C)(F)F)=O)CCCN(CCC1)C2 C(=O)(C1=NOC(C)C1C)NCc1occ(C(N2C(C(C)=O)C=CC2)=O)c1 C(=O)(C(=O)C(C)(C)C)N1CC2C(C(N(C)CCC3CCCO3)=O)(C2)C1 C(=O)(C(C)CC(F)(F)F)NC(CNC(c1c(C)n(C(C)(C)C)nc1)=O)C1CC1 N1(C(CC2(OC)CCOCC2)=O)CCC(O)(C(C)NC(C2CCCC2O)=O)CC1 c1(C(N(CCOCCN(C(C(CC)OC)=O)C)C)=O)ncc(OC)cc1F.C1CC1 c1(C(=O)NC2CN(C(c3ccnnc3)=O)CC3(CC3)C2)cnc2ncccc2c1 O=C(C(C1=NOCC1)N1CCCC1C1CCCOC1)NCCc1ccc(Cl)cc1 C(=O)(N1CCC(C(=O)NC(C)(CC)CO)O1)c1nc(CCC)oc1 C(=O)(C(CNC(c1nc(C)oc1C)=O)CC(C)C)NC(c1nc[nH]n1)CC CCC(C)(C(=O)N1CCN(C(=O)CC#N)C(c2ccc(F)c(F)c2)C1)C(N)=O CC(C)C(C)(CNC(=O)CCc1nccn1C)NC(C1(C(C)C)CNC(=O)C1)=O c1(CC(=O)NCC2C(C(N(C3(C#C)CC3)C)=O)OCC2)cccnc1O c1(C(=O)NCC(C2COCCN2C(=O)CC(F)(F)F)(C)C)ccnnc1O CCCCCCCCC(=O)NC1C2CC1N(C(c1cc3c(nc1O)CCC3)=O)C2 CCC(C)C(O)C(C)C(=O)NC(CC(F)F)C(N1CCC2(CCCC2)C1)=O C1(C(N2CCC(CN(C(=O)C(C)(C)n3cnnn3)C)C2)=O)CCCC(C)(C)CC1 C=CCCCCN(C(=O)C(Cc1cc[nH]n1)NC(=O)C(COC)N(C)C)C N1(C(Cc2n(C)ccn2)=O)CCC2(CCCN2C(=O)CC2SC(=N)NC2=O)C1 c1(C(N(C(C(=O)NCc2nnc(O)n2C)C2CC2)C)=O)ccnnc1O c1(C2(NC(C(n3ccnc3C3OCCC3C=C)C)=O)CCCC2)ccccc1Br C12(CNC(C3(CC)CC3(F)F)=O)CC1CN(C(C1(C(F)F)CCCCC1)=O)C2 C1(NC(c2cnc(CN(C)C)[nH]2)=O)CCC(CNC(=O)CC2CC=CCC2)CC1 c1(NC(CC2(NCc3n(C)ncc3)CCC2)=O)sc2c(c1C#N)CCC2 C1(CNC(c2cc(CCC)on2)=O)CCN(C(C2CC(C)C2)=O)CC1(F)F c1(C(N(CC(CNC(c2nccc(C)n2)=O)C)C)=O)cc(N)c(C)cc1C N(C1CCCn2ccnc21)C(CCC(CC)NC(=O)Cc1cnns1)=O n1(CCOC)cc(C(=O)NCCC2CCCN2C(C2CC(CF)C2)=O)nn1 N1(C(C2(OC)CC(C)C2)=O)CCC(F)(F)C(CNC(c2nc(Cl)sc2Cl)=O)C1 N1(C(c2c(C)c[nH]n2)=O)CC(C)CCC1CNC(c1ccc(F)c(CO)c1)=O N1(C(C2C(=C)CC2)=O)CC2CCC1CN2C(C1(C#N)CCOC1)=O n1(CC(=O)N(C(CCNC(C2N(CCC)CCC2)=O)C)C)cc(C#N)cn1 C(=O)(C(CC1CCC1)NC(=O)C(C)(C)NC(C1CNC(=O)O1)=O)OC Nc1ccc2nc(-c3ccc(CN(C4CCCCC4)CCCO)o3)sc2c1 CC1(C)CC(NC(C2CSC2)=O)CCN(c2nnc(C#N)s2)C1 C(c1c(C)coc1C)=CC(N1CCC(N(C(=O)C(C)C2CCC2)CC)C1)=O Cc1cc(CNC(C2(C3CC3)CN(C(c3cc(O)nc(O)n3)=O)C2)=O)cc(F)c1 c1(C(=O)NC(n2cccc2)CNC(=O)CC2CCCC2)cc2sccc2[nH]1 C1(N(C(C(CCC)N(C)C)=O)CC)CCCN(C(=O)Cc2cnn(CC)c2)CC1 C1(NC(c2nc(CC)oc2C)=O)CC2CC1CN(C(c1cc([N+](=O)[O-])c[nH]1)=O)C2 CN(C(=NCCc1ccccc1)NCCN1CCCC1=O)CC1CC1(Cl)Cl N1(C(C(N2CCN(C)CC2)C)=O)CC2CCN(C(c3cccc(=O)o3)=O)CC2C1 CCCCC(C)CCC(=O)NCCCOCCCNC(=O)CCc1ccccc1 N1(CC2CC(C)OCC2)C(=O)CN(Cc2ccccc2C(C)(C)C)C1=O C1(C(=O)NC2CCCC(OC)C2)CCOCCN1C(c1ccc(Cl)o1)=O c1(NCc2nc(CN(CCOC)C)on2)cnn(CC(C)=O)c1-c1ccccc1 c1(OC)ccc(NC(CCCNC(C)(C)C#N)=O)cc1 C1(C(C)C)(C(=O)NC(C23CCC(CO2)C3)C)CCCN1C(c1cncc(O)c1)=O CCCC(CNC(=O)Cc1ccsc1C)C(=O)NCC(C)OCCO C(=O)(C(CCC1CCC1)NC(C1(CSC)CC1)=O)NC(C1(OC)CCC1)C c1(C(=O)NC(C2CN(C(C3(CCCC)CC3)=O)C2)C)cccc2c1C(=O)CC2 N1(C(C(CC)C)=O)CCCOC(CCNC(c2cnc(CO)nc2C)=O)C1 C1(CCNC(c2ccc(CO)o2)=O)CC(F)(F)CN1C(C1C=CCCC1)=O N1(C(C(CN(C)C)O)=O)CC(C(=O)NCC(F)(F)CO)CC1CO C1(C(=O)NC2(CNC3CCCO3)CCC2)OCCCC1c1ccccc1 c1(OC)cc(C(=O)NCC(C)N(C(=O)CCN2CCC(O)CC2)C)cc(N)c1O C1(C(N2C(C3(NC(c4cc(C)on4)=O)CC3)CCC2)=O)CCc2n[nH]cc2C1C C1(NC(=O)NCC2CNC(=O)C2)CC2C=CCC(C1)C2 C1(NC(c2coc(C3CC3)n2)=O)CCCN(C(C23CC(C(F)F)(CO2)C3)=O)C1 Cc1ccncc1C(N1CC(OCCC(=O)NCC2CC=CCC2)C1)=O C(CN=c1ccn2ncc(I)c2[nH]1)NC(C1(C(C)C)N=N1)=O c1(C(C)NC(C2CC(C)(NC(=O)CC3CSCCO3)C2)=O)ccc(O)nc1 c1(C(N2CCC(c3ncco3)CC2)C(=O)NC2CCOC2)nnc2n1CCC2 Cc1cc(O)c(Cl)cc1C(=O)NC1CCC(NC(=O)CSCCC(C)C)C1 Cc1ccnc(NC(C)(CCCO)c2nnnn2CC2CC2c2ccccc2)n1 C1(CC(=O)NC(COC)(C)C)CCCCN1C(c1cn(C2CC2)nn1)=O c1(C(N2CCC(CNC(CN(C(COC)=O)C)=O)C2)=O)c(C)oc2ccccc12 Cc1[nH]nc2c1CCC(C(=O)NCC1CCN(C(C3(C)COC(=O)N3)=O)CC1)C2 C1(NCCNC(CN(C)CC)=O)CC(C)N(CC(F)(F)F)C1 C1(CCC)CN(C(C2CC2F)=O)CCN1C(c1cc(C2CCCC2)nn1C)=O C1(NC(=O)CCNC(C2CCC2)=O)CCCC(C(=O)NCc2n(C)ccn2)CC1 C1(O)(CNC(C2C(C(=O)OC)C2)=O)CCCN(C(C2(OC)CCC2)=O)C1 CC1CC(c2nccn2C)CN1C(=O)NC1C2CC1(c1cccc(Cl)c1)CO2 CC1CN(C(C2CCC2)=O)CC(CCNC(c2cnn(-c3cccnc3)c2)=O)O1 C1(C(C)NC(=O)Cc2ccns2)CCN(C(=O)CCC2CCC2)C1 N1(CCC2CCC(=O)NC2)CCN(C(c2ccc(C(F)(F)F)cc2)=O)C(=O)C1 Cc1cc(CCC(=O)NCC(C)CNC(C2CCC2(C)C)=O)on1 C1(NC(C(C)n2ccnc2)=O)CC2CCC1N2C(=O)Cc1ccc(Cl)cc1F C1(CCNC(C=C(C)C(C)(C)C)=O)CN(C(=O)C(N2CCSCC2)C)CCO1 c1(C(N2CC(CC(=O)NC(CC)CO)C2)=O)cc(C(F)(F)F)cc(F)c1 c1(C(=O)NCC2CCC(NC(C3(C#C)CCC3)=O)C2)c(C)c(C)c(C)c(C)c1C C(=O)(C(CC(C)(C)C)C1CCCC1)N(C1CN(C(=O)OC(C)(C)C)C1)C c1(CC)nnc(C)cc1C(=O)NCC1CCC(CN(C(=O)C=C2CC2)C)CC1 C(CCCCCNC(=O)C(C1CCCCC1)O)N(C(COCCC=C)=O)C c1(C(C(N)=O)N(C(=O)C(N2CCOCC2)C2CC2)C)ncccc1Cl C1(CCNC(C)C)CN(C(=O)OC(C2CC2c2ccnn2C)=O)CCS1(=O)=O N1(C(c2cnn(C)c2C(F)(F)F)=O)CC(NC(c2nnc(S)n2C)=O)CC1(C)C N1(C(C(COC(C)=O)C)=O)CCOC(C(=O)NCC2CC(F)(F)C2)C1 c1(C(C(=O)NCCCCCC)N(C2CCCOC2)CC)cccc(Cl)c1Cl N1(C(C(=O)NCCc2c(C)ocn2)=O)CCCC(OC(F)(F)F)C1 c1(C(=O)NCC2CCN(C(CCOC(C)=O)=O)CC2)cccc(F)c1C1CC1 n1(CC(=O)NCC(CC(C)C)NC(=O)C(O)c2cnc[nH]2)cnc([N+](=O)[O-])c1 N1(C(COCCC)=O)CCN(C(=O)Cc2cccc(Br)c2C)CC1CO N1(C(CC2C(C)CCN(C(Cc3ccn(CC)n3)=O)C2)=O)CC2(COC(C)C2)C1 C(C(C)(O)CC(=O)N1CCCC(CCNC(C2CC3(C2)CC3(F)F)=O)C1)OC C(=O)(C#CC1CCC1)NCC1CC(CNC(C2CC(C)(C(=O)O)C2)=O)C1 Cc1ccoc1C(N1CCCC1CNC(=O)CN(C(=O)CC1CCCCC1)CC)=O N1(C(CCOCCOC)=O)CCC2(CC2)CC1C(=O)NCCCc1cncn1C Cc1cc(F)c(Cl)cc1C(=O)NC1(C)CCC(NC(=O)C(F)CC2CCC2)CC1 C1(C(=O)NCC(C)(C2CCC2)NC(c2nn(CC)c(C)c2)=O)COC(C)(C)CO1 CC1COCC(CC(N2CCSCC2C(N2CCC(N3CCCC3)C2)=O)=O)O1 C(=O)(CCC(=O)c1ccc(Br)cc1)NC(CNC(=O)C(F)=CCCF)CO C(C(=O)NC(C)Cc1ccsc1)(C1=CCSC1(C)C)N(CC)CC1CC(F)(F)C1 n1(CCOCC)ncc(I)c1NC(=O)Nc1cccc(OC)c1 C1(CC(=O)NCC2CCN(C(c3c(C)nc[nH]3)=O)C2(C)C)CCCCCC1(F)F C(=O)(C(C)C(O)C(C)C)NCC1(NC(c2cc(CC)ncc2)=O)CCCCC1 C(=O)(CCN=c1ccc(C)c[nH]1)N1CC(OC)C(NC(=O)CCC=C(C)C)C1 c1(C(=O)NCC(C)CN(C(=O)C(O)C2CCC2)C)cccc(C(C)(C)C)n1 c1(C(C(=O)N(CCC)CCNC(=O)CN(C2CCCC2)C)F)ccccc1F C1(CNC(C2(SC)CCC2)=O)CC2(CC2)CN1C(C1CCCC(CF)C1)=O c1(C(=O)NCC23CC(NC(C4CCCN(C)C4)=O)(C2)C3)c([N+](=O)[O-])cnn1C C1(C(=O)NCC2(O)CCC2)CC2CC2N1CC1(c2ccccc2)CCCC1 c1(C(=O)N(CC2(CC(=O)NC(CC)(C)C)CC2)C(C)C)cncc(N(C)C)n1 CCC(CN(C)C)C(=O)NC(Cc1cnn(C)c1O)C(=O)N(C1CCOCC1)C c1(C(N2C(C)(C(=O)Nc3ccnc(Cl)c3)CCC2)=O)cnn2cccc(F)c12 CN1CC2CN(Cc3cn(-c4ccnc(F)c4)nn3)CCN2C1=O N1(C(c2cnn(CC(C)C)c2)C(=O)NCC)CCOCC(CC2CC=CCC2)C1 C1(C)(CCC)CCCN1C(=O)CCc1ccccc1C c1(-c2c(C)ccc(CO)c2)cc(C(N2CC(C)(OC(C)C)C2)=O)c2cc[nH]c2c1 c1(C(N2CC(O)(C(C)NC(c3ccc(C)nn3)=O)C2)=O)ccc2c(c1)NC(=O)C2 N=c1ccc(C(N2CC3(NC(c4cnc(C5CC5)nc4)=O)CC2C3)=O)c(Cl)[nH]1 C1(N(C(CC(C)NC(CC(=O)NCC)=O)=O)C)CC(C)OC(C)C1 C1(CC)CN(C(=O)CC2(C(F)(F)F)CC2)CCC1NC(C1(OC)CCCSC1)=O C1(NC(c2c(OC)c[nH]c2C)=O)CC2CCC(C1)N2C(=O)OCc1ccccn1 C1(C)(NC(CN(C2CCCS2)C)=O)CC(NC(C2(C3CCCO3)CCC2)=O)C1 CCN=c1[nH]c(C(N2CCOC(CCNC(=O)COC3CC(F)(F)C3)C2)=O)cs1 N1(C(C(C2CCC2)OC)=O)CC23CCCC2(C1)CN(C(=O)CCP(C)(C)=O)C3 c1(CN2CC(NC(C(CCC)N(C)C)=O)C(C)C2)ccnc(F)c1Cl c1(NC(C2C(NC(C(C#C)(C)C)=O)C2)=O)cc(C#N)ccc1Cl C1(C(=O)NC2C(CNC(=O)C=Cc3cncc(F)c3)CC2)CCn2nncc2C1 CC(CCCC(=O)Nc1cncc(F)c1)NC(c1ncc(F)cn1)=O c1(C(N2CCC(NC(C3(COC)CC3)=O)C2)=O)cccc(F)c1C c1(CC(C)C(N2C(C(=O)NCc3cccc(Cl)n3)CC3CC23)=O)ccc(O)cc1 c1(NC(C)C)nccc(=NC(=O)C2(C)CCCN2S(=O)(=O)c2cnc(Cl)c(Cl)c2)[nH]1 N1(C(C23N(C(CC(=O)OCC)=O)CCC2CCC3)=O)CCC2C(=O)NCC2C1 C1(CC(=O)N(C(C)C)CCO)CCN(C(=O)CC2CC3(CC3)CO2)CC1 c1(C(=O)NC(CC)CN(C(=O)Cc2csc(C)n2)C)nc(C(C)C)oc1C C1(NC(C2CCC(=O)O2)=O)C(CNC(C2(CC3CC3)CCC2)=O)CCC12CCC2 c1(C(=O)NCC(C2CCCOC2)OC)ccc2c(c1)NC(=O)C2 C1(CNC(c2c(CC)non2)=O)CC2(CC2)CN1C(c1cn(C2CC2)nn1)=O c1(C(CNC(N(CC#CC)C)=O)C(=O)OC)ccc([N+](=O)[O-])cc1 Cc1nccc(F)c1C(C1CC1)NC(=O)Nc1ncccc1C(F)(F)F N1(C(CCCCOCCC=C)=O)CCCCCC1CNC(C1C2CCCC12)=O.C(C)(=O)O Cc1oc(=O)oc1C(=O)Nc1ccccc1C(=O)OC(C)C CC1SCCCC1C(=O)NCC1CC(C(=O)NOCC2(C)CCC2)C1 c1(C(=O)NCC2COCCN(C(c3cc[nH]n3)=O)C2)c(Cl)ccc(Cl)c1O C1(CNC(C(C)=CC=C)=O)OCCC1C(=O)NC(c1ccns1)C N1(C(C(C)Sc2cccc(C)c2)=O)CCN(C(c2sc(C)nc2C)=O)C2CC12 c1(C(N2CCN(C(C3CCCC(=O)O3)=O)CC2)=O)ccc2ccccc2c1 N1(C(CN2CCC(C)C2(C)C)=O)CC(C)(C)OC2(CCOCC2)C1 c1(C(=O)NCCCNC(C2CC2c2ccsc2)C2CC2)csc(Cl)c1 C1(C(=O)NCc2cc(C)[nH]n2)CC(C)CN(C(c2occ3c2CCC3)=O)C1 CN1CC2CN(C(C34CCC(CC3)N(C(=O)CC3C=CCC3)C4)=O)CC2C1 N1(C(c2ncc(OC)cc2F)=O)CC(CNC(=O)CNC=O)C2(CCC2)C1 N1(C(C2(OC)CCSCC2)=O)C2CCCC1CC(NC(c1csnc1OC)=O)C2 S1(=O)(=O)c2ccc(c(F)c2)N1.C12(C(N(CCCOC=C)C)=O)CCSCC1C2 N1(C(C(CC2CCC2)OC)=O)CC2CC1(C(=O)NCC(C)C(F)F)C2 N(C1c2ccccc2CC1NC(=O)C(F)(F)CO)C(c1ccc(OC)cn1)=O N1(C(C(CC2CC2)NC(C2CC(O)(CC#C)C2)=O)=O)CC(CN(C)C)C2(CC2)C1 C(=O)(NN1CCCCC1=O)c1c(OC(=O)NC2CCCS2)cccc1 C1(C)(CNC(C2C(=C)C2)=O)CCCN(C(c2cscc2F)=O)C1 c1(CNc2c(C)noc2C2CCC(F)(F)CC2)nnc2c(=O)[nH]ccn12 N1(C(CCc2c[nH]c(=N)[nH]2)=O)CCC2C(C1)CN2C(C1CCS1(=O)=O)=O c1(C(=O)NC2CCN(C(c3cncc(C)n3)=O)CC2CO)cc(C)c(N)cc1Cl C=C(C)CCCC(=O)N1CC(NC(C2CCCN2N=O)=O)CCC1C N1(C(C2C=CCN(C(CC3ON=C(C)C3)=O)C2)=O)CC2CC(O)C2C1 c1(C(=O)Nc2c(CNC(C3(COC)CC3)=O)cccn2)cnn2c1OCC2 c1(-c2c(C(=O)NC(C)C(C)C)ncc(SC)c2)ccc2[nH]c(C(F)(F)F)nc2c1 CC(CN(C)C)CCC(=O)NC1(CO)CCCN(C(=O)CN2CCOC2=O)C1 c1(OC)cnc2c(c1)c(C(C)C)nn2C.c12ccoc1S(=O)(=O)N2.c1ccccc1 C1(OC)CC2CC1CN(C(=O)C(CNC(c1cnc(OC)s1)=O)C(C)C)C2 c1(C(c2n(CCCOC)nnn2)NCCCC2CCCCO2)cn(C)nc1I C(CC(=O)NC1(Cn2cc(CC3CCOC3)nn2)CCC1)(OCC)OCC C1(C(=O)NC2CCC(C)N(C(=O)Cc3ccco3)C2)CCn2ccnc2C1 Cc1ccc2cc(C(=O)NC(C3(O)CN(C(c4cc(=O)cc[nH]4)=O)C3)C)[nH]c2c1 C(=O)(CC(=O)N(C)C1CC1)N(CC(CC)NC(=O)CC(C)C1CCCCC1)CC C(=O)(C1CCc2cccc(F)c21)NC(C1CCN(C(CC(C)OC)=O)CC1)C C1(C(N2C(C=C)CC2)=O)CC(O)CN1C(c1c[nH]c(C#N)c1)=O c1(C(=O)NCC2C(NC(COCCC=C)=O)COC2)cc(N)ccc1F C1(C(=O)NC2C(SC)CN(C(c3coc(SC)c3)=O)C2)COc2ccccc2C1 c1(C(N2C(C)(CNC(c3c(C)ncnc3C)=O)CCC2)=O)nc[nH]c2nccc1-2 C(=O)(C1CCc2ccccc21)NC(CNC(C(C1CC1)OCC)=O)CC(C)C C(C(=O)N1CC(OCC)C1)(C(C)C)OCC.C1(=O)CCN(C)C(=O)NCCN1 N1(C(C(C)NC(CC)(C)C)=O)CCCN(C(=O)CS(=O)(=O)C(C)C)CCC1 N1(C(C(CC)OC2CCCCC2)=O)CC(C)(C)CC1CNC(=O)CCOC(C)=O C1(C(C)(C)NC(CSCC#C)=O)CCN(C(C2CCCCO2)=O)CC1 C1(C(N2CC(N(CC=C)C)C2)=O)CN(C(=O)CC(C)COC)CC1F C1(C(C)NC(C2C(CC)C2)=O)CCCN(C(C2CC2c2cccnc2)=O)C1 N=C1NC2=NCCc3c(cnn3-c3ccccc3)CCCN=C(N2)N1.C1CC1 c1(CNC2C(CNC(c3cc(CC)on3)=O)CCC2)ccc(NS(C)(=O)=O)nc1 c1(C(=O)NCCC(O)CNC(c2cnn(C(F)F)c2)=O)cnoc1CC1CCC1 N1(C(c2cc(C(C)=O)oc2)=O)CCN(C(=O)C=Cc2cncc(F)c2)CC1C c1(C(=O)NCC(=C)CCNC(C2CC2C(C)(C)C)=O)ccc(-c2cc[nH]n2)cc1 N1(C(c2cc(OC)ncc2)=O)CC(C(N2CC(C(F)(F)F)N=N2)=O)CC2OCCC12 C1(NC(=O)Nc2c(F)cc(C)c(F)c2)CCOC2(CCSCC2)C1 N1(C(CC(=O)NCC)=O)CCC2(CC1)COCC(CNC(C1CCOC1)=O)O2 c1(CC)ccc([N+](=O)[O-])cc1NC(N1CC2NC(=O)OC2C1)=O c1(C(C)C(=O)NCC2(NC(c3ccc(F)cc3)=O)CCOC2)nc(F)ccc1Cl O(CP(C)(C)=O)CC(=O)NCC(C1CCCC1)NC(CN(C1CCCCC1)C)=O c1(C(N(CCNC(c2scc(C(C)=O)c2)=O)C)=O)n[nH]c2c1CCCC2 c1(CC(CO)NC(C2C(NC(c3c(C)scc3)=O)CCC2)=O)ccc(O)cc1 C(=O)(C1=C(Cl)CCC1)NC(C1(O)CN(C(=O)C(N2CCC(C(F)(F)F)CC2)=O)C1)C N1(C(CCc2onc(CCC)n2)=O)CCC(NC(c2snnc2C)=O)C(F)C1 c1(C(=O)NC2(CNC(C34CC(OC)C3C4)=O)CC2)nc(C)n2ccccc12 C(=O)(C(C(C)(C)C)N(C)C)NCC1OCCN(C(CCc2nc(C)c(C)[nH]2)=O)C1 C1(C(=O)NCC(=CC(N2C(CC)COCC2)=O)C)CC(C)(C)CN1C c1(C(=O)NCC(CNC(CC(C=C)CC)=O)O)cc(Cl)c(C)cc1Br C1(N(C(c2cn(CC)nc2C2CC2)=O)C)CCCN(C(c2ccc(F)s2)=O)CC1 c1(OC)cc(C(N2CC3CC3(C(=O)Nc3cn(C)nn3)C2)=O)c([N+](=O)[O-])cc1O C12(C(=O)NCC(C(C)C)(C)NC(c3cc(C(F)F)ccn3)=O)CC1COC2(C)C c1(NC(C2(CC#C)CCN(C(C3C(C)(C)C3(C)C)=O)C2)=O)nn(C)cc1C#C C(C)(CC(=O)N(C)CC1CCCN1C(c1ccc(C(N)=O)o1)=O)OC N1(C(C2CCN(CCC#C)CC2)=O)CCN(C(c2snnc2C)=O)CC(CO)C1 N1(CC)CCOC(C(=O)NC2CC(CNC(c3c(C)cnn3C)=O)C2)C1 N1(C(CC2(C=C)CCC2)=O)CCC(C)(NC(=O)C(c2ccccn2)C)C1 c1(CC(=O)NC23CC(NC(C=C4CCC(C)C4)=O)(C2)C3)ccc(F)cc1Br C(=O)(C1=CC2CCC(C1)N2)N1CC(N(C)C(C2CC(n3ccnc3)C2)=O)C1 c1(C(=O)NCC(=C)CCNC(=O)COc2cc(C)on2)cc(O)cc(Cl)c1 N1(C(C2N(C)C(=O)OC2)=O)CCS(=O)(=O)C(CCNC(c2ccccc2)=O)C1 CC(C)C(C(=O)CN1CCOCC1)NC(c1csc(Br)n1)=O C1(COC)CN(C(=O)CN2CCCCC2=O)CCN1C(c1cc(CN)sn1)=O C(CC(C)C(=O)NCC1CC1NC(c1cnc(C2CC2)o1)=O)=CCC Cc1ccc(C(C)CC(=O)NCC2(C)CCN(C(=O)C(F)(F)C3CC3)C2)cc1 C1(CC)CCCCN1C(c1cn(-c2ccc(C)nc2)nn1)C c1(CC)cc(C(=O)NC(CNC(c2cnncc2O)=O)CC(C)C)sc1C c1(C(N(CCN(CC#CC)C)C)=O)cc2cc(C)ccc2s1 c1(NC(C2(C)CCN2C(C2(O)CCOCC2)=O)=O)cc(Cl)cc2[nH]ncc12 N1(C(C2(CC=C)CCN(Cc3nc4cccnc4[nH]3)C2)=O)CCCC(C)(C)CC1 c1(C(CC(=O)NCC(O)CNC(=O)CC2CCSCC2)C2CC2)ccc(O)cc1 C(=O)(CC(C)(C)C#N)N1C(C(=O)Nc2c(CC)n[nH]c2)CC1 C(=O)(C1=CC2(CN(C(c3csc(Cl)c3)=O)C2)OC1)N1CC(C)(C(F)(F)F)C1 C=CCC(F)(F)C(=O)NCCC(CNC(=O)C=Cc1cn[nH]c1)OC O=C(CCN=c1[nH]c(=NCCCF)[nH]c2c1CCC2)C1CCCC1 N1(C(C(C(C)O)C)=O)CCC(CO)(NC(=O)CC2OC(C)(C)OC2=O)CC1 Cc1nc(F)ccc1CNC(=O)CC1CCCC1NC(C1CC(O)C1)=O C1(CC(=O)NCCCCN(C(=O)CSc2ccc(Cl)cc2)C)CCC(C)(C)CO1 c1(-c2ccc(SC)cc2)nc(C)cc(=NC2CN(C(=O)C(F)C(C)(C)O)C2)[nH]1.CS N1(C(c2c(SCC)nccn2)=O)CCC2C1CCCN2C(=O)CCC(C)(F)F N1(C(c2c(C)nn(C)c2C(F)F)=O)CC(NC(c2cccn2C)=O)C(C2CC2)C1 CC(C)(F)CCC(=O)NC1(CC(N2CC(O)(c3cc[nH]n3)C2)=O)CCC1 N(C1CCOc2ccc(Br)cc21)S(=O)(=O)c1cccc(N2CC(F)C(F)C2)n1 n1(CC)cc(C(=O)NC(C)CCCCNC(c2cnoc2)=O)c(C)n1 C1(C(=O)NC2C(NC(C3CCC(F)(F)C3)=O)CC2)C2CCC1(c1cscn1)C2 C1(NC(CCC(C)(F)F)=O)CN(C(=O)CC2CCCCC23CC3)C2(CCCC2)C1 C1(CCCCNC(c2ccc(CC)o2)=O)CCCN(C(=O)CCN2CCC2)C1 N1(C(CC2(COC)CC2)=O)CC(C(N2CCC(C(F)(F)F)C2)=O)CC12CCC2 c1(NC(N2CCCC(CNC(c3cccc(F)n3)=O)C2)=O)cccc2c1OCC2 Cc1cc(C(=O)N(C2CCC(NC(c3ccnnc3C)=O)CC2)C)nc(C)c1 C(=O)(CC(F)(F)C(F)F)NCCC(C)N(C)C(C1C(F)(F)C12CC2)=O C1(NC(=O)NC(CC(C)C)C)CC2(C1)CN(C(=O)CN1CCCC1)C2 N1(C(C(C)C#N)=O)CCC(NC(C2CCC(c3ccccc3)C2)=O)C(C)(C)C1 C(=O)(C1=CCC2(COC2)OC1)NCC1CCCC(NC(C(C)(C)S(C)(=O)=O)=O)C1 N1(NC(C)(C)CNC(C2CC3CCC3C2)=O)CCN(C(=O)CC2CC2)CC1 N1(C(c2cc(C)c(Cl)cc2)=O)CC2OCCN(C(=O)CC3CCCN(C)C3)C2C1 C1(NC(CCOCC)=O)(CNC(C2CCCCC2n2cccn2)=O)CCOCC1 CC(CN(C)C)CCC(=O)NC1CCCC1CC(=O)NC1C(C)C1(C)C C(=O)(CCCOc1cccnc1)NC(C)CCC1CN(C(c2cncn2C)=O)C1 c1(OCCCCOC)nnn(C2CCS(=O)(=O)C2)c1NC(=O)C=Cc1ccsc1 c1(NCC2C(O)CCC(C)(C)C2)[nH]c(=NCc2nc[nH]c2Br)nc2sccc12 C1(CNC(CC(CC)OC)=O)CN(C(=O)C=CSC)CCC1(F)F c1(OC)cc(C(=O)NC(C)(C)C(C)NC(=O)CCc2cnc[nH]2)sc1Br CP(C)(=O)c1cccc(C(N2CCCC(NC(=O)Cn3cnnc3)CC2)=O)c1 C(CCC(c1ccccc1)N1CCCC1)NC(C1CC(CC2CCCO2)C1)=O C(C(=O)NC1CC1)(C1CCSC1)N(C)CC1(C)CC1 C=CCC(C)(C)C(=O)NCC1CN(C(=O)C(F)(F)CO)CC1O C1(C(C)C(=O)NCCF)CCCN(C(=O)C(C)(C)N(C)C)C1 C(=O)(CCCC(=O)NCCC)NCCCC1OCCN(C(C(COCC)C)=O)C1 Cc1cc(C(=O)NCC2CN(C(c3cc[nH]c3)=O)CC2C)c2cccc(C)c2n1 C1(C(C)(C)C)CCc2nc(NC(=O)Cc3cc(Cl)c(Br)c(Cl)c3)sc2C1 CC1(C)CN(C(=O)CCC2CCC2)CC1NC(=O)C1=NNC(=O)C1 c1(N(C)Cc2c(C)occ2)cc(Br)ccc1S(=O)(=O)N1CCCC(C2CCC2)C1 N1(CC(N2CC(O)(CNC(c3ccc(Br)o3)=O)C2)=O)Cc2ccccc2C1=O CCCCS(=O)(=O)NC(=O)C(CCC)OCC(N1CCOC(CN)C1)=O C1(CNC(c2n(CC)ncn2)=O)CCC(C)N(C(c2cnsc2C)=O)C1 C1(N(C(C=CC)=O)C)CCCCN(C(C2CC=C(C)CC2)=O)C1 C1(CC)C(NC(=O)C=Cc2ncc[nH]2)CCN1C(C1CCS(=O)CC1)=O Cc1nc(=NC2CN(C(C3CC4(CCCC4)C3)=O)CC2C)s[nH]1 N1(C(C(CCC)C#N)=O)CCC2(CC1)CC2C(=O)NCc1nc(COC)no1 N1(C(CC2CC(C)(C)C2)=O)CC(F)(F)CC1CNC(C1CC1C(F)F)=O N1(C(c2c(C)cccn2)=O)CC2(C1)CN(c1ncc(Br)cn1)C2 C1(C(=O)NCC(CC(C)C)NC(C23CCC(C2)OC3C)=O)CCC2(CC1)CC2 Cc1ccc(C(F)(F)F)cc1CN1CCC(Br)CC1.N12CCC(C1)CC2=O C1(C(=O)NC(c2ccc(C)cc2)CC)CCCN(C(c2ccc(N)cn2)=O)CC1 C1(Cc2cn(C3C=CCC(C(=O)NC(CC=C)CC)C3)nn2)CCC(C)(C)CC1 C1(C2CN(C(C34CCCN3CCC4)=O)C2)(NC(C(CC)N2CCCC2=O)=O)CC1 C1(NC(C2N(C)CCN(CC)C2)=O)CCCC2(CC1)CC2 Cc1ccc2nc(C(N3CCC3CNC(c3ccnn3C3CC3)=O)=O)cn2c1 N1(C(C2(C#N)CC(C)C2)=O)CCC(NC(=O)CC2(C)CCCC2)C(C)(C)C1 C1(C(=O)NC(C(C2CCN(C(C34CC(CC)(C3)C4)=O)C2)C)=O)CC(=O)N(CC)C1 C1(NC(=O)Cc2cc(Cl)cc(Cl)c2)CN(C(=O)CNC2(CN)CC2)CC1C1CC1 C(=O)(CC(C(F)F)N(C)C)NCCCCNC(c1c(SCC)cccc1)=O c1(NS(C)(=O)=O)ccc(C(=O)NC2CCSCC2)cc1.C1(CN)CC1C=O c1(C(=O)NC(C(C)C)(C)CNC(C2CCCCN2C)=O)cnn2c(=O)cc[nH]c12 C(N=c1[nH]nc(CO)s1)C1C(NC(C2(C)CNC(=O)C2)=O)CCCC1 N1(C(=O)C2=CCCCC2)CCC(C2CCCN(C(C3COCCO3)=O)C2)CC1 Cc1ncnc2c1CC(C(=O)NC1(CCNC(=O)C(CO)N(C)C)CC1)CC2 C1(C(=O)NC(C2CC2C(N2CCC=C(C)C2)=O)C)CCCCC(=O)N1 C(=O)(N=c1ccn(CC(F)(F)F)[nH]1)N1CCC(C(C)C)C1 N1(CCC)CCC(CC)(NC(c2nn[nH]n2)=O)CC1 C1(O)(CNC(CCCc2scc(C)n2)=O)CCN(C(=O)CSC(F)(F)F)CC1 c1(CC(=O)NCC(=O)NC2(C(=O)NC)CCOC2)ccc(OCC)nc1 S(=O)(=O)(C1CCOC2(CCOCC2)C1)N1CCC(C)C(F)(F)C1 C1(CC)(CC)CCN(C(C2CCCN(C(c3cc(C)c(C)[nH]3)=O)C2)=O)CC1 c1(OC)ccc2cc(C(N3CC(CNC(=O)C(Cl)=CCl)CC(C)C3)=O)n(C)c2c1 C=CCCC(C(=O)OC)NC(c1cc(OC)c(-c2ccnc(O)c2)cn1)=O c1(SC(C(=O)N(C2CCN(C(CCNC(C)=O)=O)C2)C)C)ccc(C#N)cc1 N1(C(c2cc(C)[nH]c2)=O)CC2(CC2)CC1C(=O)NCCc1ccon1 CC1CC(C(=O)NC(C)(C)C)N(C(=O)OCC2CN(c3ccccc3)CCO2)C1 Cc1ccc2nc(-c3nc(CC4CCOCC4)nn3Cc3ccccn3)cn2c1 CC1CCC2(CCC2)CN1C(=O)NC1CCN(c2ccc(Br)cc2)C1 c1(OCC)ncc(C(C)NC(=O)NCCCC2CCCCC2)cc1C C1(C(=O)NC2CCN(c3ncccn3)C2)CC2(C1)CC(F)C2 Cc1cnn(C(C)C(=O)NC2CCC(CNC(C3CC(F)C3)=O)C2)c1 CCC(C)C(CC(=O)NCCC(C(C)C)OC)NC(=O)C(O)CC(N)=O n1(CCC(=O)OC(CC(C)C)(C)C)ccc2ccc(F)cc12 C1(CNC(=O)Nc2c(C)snc2)CN(C(=O)C(=O)Nc2ccccc2)CCN1C c1(OC)nccc(=NC(=O)C2CCN2C(c2cc(C)ccc2F)=O)[nH]1 N1(C(c2c(N)cc(Cl)cc2)=O)CCOC2CN(C(c3cnc(N(C)C)o3)=O)CC12 c1(CNC(N2C(C(C)Nc3csc(C(F)(F)F)c3)CCC2)=O)cccc(F)c1F Cc1nc(CC(C)C)c(C(=O)NC(C)C(CO)NC(=O)CSC(F)(F)F)s1 N1(C(C2C(C)=CCS2)=O)CC2CCN(C(c3c(C#N)cnn3C)=O)CC12 n1(CC)ccnc1C(=O)NCCCCCN(C(=O)CC1CC1(Cl)Cl)C c1(C(=O)NCc2ccn(CC)n2)c[nH]c2cc(C3=CCCCC3)cnc12 c1(CC(=O)NCC2CCN(C(c3ccc(CCC)[nH]3)=O)C2)ccc(F)c(Cl)c1F C(CC1=CCN(C(=O)CC2CCCC(C)C2)CC1)NC(c1c(COC)ccs1)=O C(=O)(CC(=O)NCC(CNC(=O)CC1CCCOC1)CO)OCC c1(OC)cccc(C(C)=CC(N2CCN(C(c3ccc(C)s3)=O)C(C)C2C)=O)c1 CN1CCC12CN(C(=O)CCC(C)(C)NC(c1cc(O)cc(=O)o1)=O)C2 N1(C(C2CCN2C(C2(N(C)C)CCCC2)=O)=O)CCNC(c2ccc(Br)cc2)C1 N1(C(C2CCC(C)(C)OC2)=O)CCCC12CCCN(C(=O)C=CC=C(Cl)Cl)C2 c1(C(N2C(C(N3CCN(S(C)(=O)=O)CC3)=O)CC(=C)C2)=O)ccc(Cl)c(OC)c1 N1(C(C(C)OCC)=O)CCC(NC(c2cnc(F)c(Cl)c2)=O)C(CC)C1 c1(OCC)ncc(C(=O)NC2CCOC2C(N2CCCC2c2nc[nH]n2)=O)s1 N1(C(CC=CC(=O)N(C)C)=O)C(CNC(C2CC2(C)C)=O)CC2CCCC12 CC1CN(C(=O)C#N)CCN1C(C1(c2cc(Br)ccc2O)CC1)=O C(=O)(C1CCCn2cncc21)NCC1CC(NC(Cn2ncc(C)c2)=O)C(O)C1 c1(OC)ccnc(C(=O)NC(C)C(C)NC(=O)C(C)P(C)(C)=O)c1OC N1(C(c2c(CCC)onc2C)=O)CCN(C(=O)C(C)CF)C(c2cn[nH]c2)C1 N1(C(C2(OC)CCOCC2)=O)CCC(CC(=O)O)C(NC(c2[nH]cnc2C)=O)C1 N1(C(C2CCN(C(CNC(C(C)(C)C)=O)=O)C23CC3)=O)CCOCC2(CC2)C1 C1(NC(C=Cc2n(CC)ccn2)=O)CN(C(c2cc(C)cc(C)c2)=O)CCC1F C(C(CNC(C1C2COCC12)=O)C(F)(F)F)NC(=O)CCCSc1ncccn1 c1(C(=O)NC(C)CN(C)C(C2CCC(=O)N2)=O)cncc([N+](=O)[O-])c1 c1(C(C)=O)ccc(CC(=O)NC(C(C)(C2CC2)NC(C2CC(C)=NO2)=O)C2CC2)s1 c1(N2CCC(OCCNC(=O)NC34CCC3C4)CC2)cccc2c1OCCO2 c1(C(N(CCNC(c2cccc(CC)n2)=O)C)=O)ccc2c(c1)COCO2 Cc1ccc(Br)c(F)c1CNC1CCC(=O)NC1=O c1(C(=O)NCc2nc(CNC(CCNC(C)=O)=O)sc2)cnn(CCC#N)c1C Cc1ccc(C)c(CCCC(N2CC(NC(=O)CC3C=CCCC3)C(O)C2)=O)c1 c1(C(=O)NCC(C2CC2)NC(C2(OCC)CCOC2)=O)cnc(=NCCF)[nH]c1 C(C(=O)N(C)OCC)NC(C(C1CCN(C(c2nc(OCC)oc2)=O)C1)(C)C)=O N1(C(C=NOC)=O)CC2CC(NC(C3(C4CCOCC4)CC3)=O)CC2C1 C=CC(C(=O)NC1CCCC1NC(=O)COC1CCCC1)c1ccccc1 C1(C(=O)NCCCOCC)C(CC)CCN1C(=O)C=CCOCCN(C)C N1(C(CCOCC#C)=O)C(C(=O)NCC2CCCSC2)CC2CCCC12 c1(C(=O)NCC(C)N(C(CNC(C(CC)C)=O)=O)C)c(C)cncc1C c1(CC(=O)NCCCN(C(=O)C(N2CCOCC2)C)C)csc(S)n1 C1(C)(CNC(C(CC2CCCC2)NC(CCC)=O)=O)CC(C)(C)C1 Cc1ccc(C(=O)NC2CC(C(N3CC(OCC(N)=O)C3)=O)C23CCC3)nc1O CC(C)C1=CCC(C(=O)N(CC(=O)NCC2(C)CCCO2)CCO)CC1 c1(CC)oc(C)cc1C(=O)NCC(CC)NC(=O)CSc1nncn1C Cc1cn2ccc(C(=O)NCC3(CNC(c4c(C5CC5)cnn4C)=O)CC3)cc2n1 c1(C(=O)NC(C)CNC(c2c[nH]nc2-c2ccoc2)=O)ccc(Cl)cc1O C(=O)(CCCC(=O)N(C)C)NC1(CF)CN(C(c2c[nH]c(=NC)o2)=O)C1 C(CCCN=[N+]=[N-])NC(C(C1CC1)NC(C(C)n1cccc1)=O)=O O=C(C(F)C(F)(F)F)NC1(CO)CCN(C(=O)CN2CC3CC3C2)C1 C#CCC(C)(C(=O)N1CCCC1CNC(C)=O)NC(=O)CC1CCOC1(C)C c1(C(=O)NC(CC=C)CNC(C2CN(C(C)=O)C2)=O)ccc2cc(Cl)ccc2c1 C(=O)(C(C(C)C)NC(=O)CC(C)C)NCC(=O)NC1C(OC)C(O)C1 c1(C(=O)NCC(C)(CO)NC(C2C(C)N(C)CC2)=O)cc(C(F)(F)F)ncc1N N1(C(C(c2cccc(Cl)c2)C)=O)CCC(NC(c2n[nH]cc2C(C)C)=O)C1C c1(CC(=O)NCC(O)CCNC(c2ccc(C(F)F)nc2)=O)cncnc1O N1(C(CNC(=O)OCC)=O)CCC(F)(CNC(=O)CC2CCCOC2)C1.C1(C)CC1 c1(OC)ncnc(OC)c1NC1CCN(C(=O)CN2C(=O)CCC2=O)C(C)C1 c1(C(=O)NCCCCCNC(C(C)Cn2cccn2)=O)cnc2c(ccn2C)c1 c1(C(=O)NCC(CC(C)C)NC(C2(C)CC=CCC2)=O)c(F)ccnc1Cl C(=O)(C#CC(C)(C)CNC(C1CCC(C2CC2)C1)=O)N1CC(C)OCC1 N1(C(CSCC)=O)C2CCCC1CN(C(=O)COC1(C)CCC1)C2 CC(=O)CCC(=O)NC(Cc1cn[nH]c1)C(=O)NC(c1cnsc1)C C1(CNC(C2(OC)CCN(C(C3CC3(C)C)=O)C2)=O)OC(=O)NC1(C)C c1(OC)cccc(C2CC(O)CN2C(=O)C(C)n2ccnc2)c1 N1(C(c2[nH]cc(C(C)(C)C)c2)=O)CCC(C2CCCN(C(=O)C3CC3)C2)C1 N1(C(c2ccc(CC)o2)=O)CCC(NC(c2cnn(C(C)(C)C)c2Cl)=O)C1C C1(CN(C(=O)CSCCC#N)C)CCCN1C(=O)CCc1ccncc1 c1(OC)ccc(Cl)c(C(=O)NC(CNC(=O)CCNC2CCCCC2)C2CC2)n1 C(CC1CCCCC1)(C(=O)NC(C)(CNC(=O)CNc1cnn(C)c1)CO)OC Cc1cc(C(=O)NCC2CN(C(=O)C(c3ccn(C)n3)C)CC2(F)F)cc(F)c1 S(=O)(=O)(c1cnn(C)c1)NCC(=O)NCC1(F)CCC(NC(C(C)N(C)C)=O)C1 N1(C(c2nn(CC)nc2C)=O)CCC(C)C(CNC(c2cc(F)cnc2Cl)=O)C1 C#CC1(C(=O)NC2CN(C)CC23CC3)CCN(C(=O)CN2CC(C)(C)C2)CC1 C(C(C(=O)N(CC(O)COC)C)NC(=O)Cn1cc(C(C)=O)nn1)OC C=Cc1ccc(-c2cncc(C(=O)NCCC(N)C(C)(C)C)c2)cc1 C1(C(N(CC(C)O)CCNC(=O)C=C2CCN(C)C2)=O)CCc2ccnn2C1 N1(Cc2cnc(COC)s2)CCN(C(=O)CCC(C)C)C2CC12 c1(CC(=O)NC2C(CNC(c3cc(OC)no3)=O)CCC2)cnn2c1OCCC2 c1(CC(=O)NCC(CC)NC(=O)CC2CC3CC3C2)cnn2ccccc12 C1(NC(CCc2onc(C)n2)=O)CC2CN(C(c3nc(Cl)oc3C)=O)CC12 C=C(CNC(=O)CN(CC)CC)CCNC(=O)Cc1n[nH]c(C)n1 C(C1=Cc2cc(Cl)ccc2OC1)=CC(N1CCCC(NC(CC=CC)=O)C1)=O C1(C(=O)NC2C(CNC(c3c(CC)n[nH]c3)=O)CCCC2)CCC(=O)NC1=O C1(CNC(CCN2CCC(C)CC2)=O)CCN(C(=O)CCS(N)(=O)=O)C1(C)C c1(CC(=O)NC2C3CCN(C(C(N4CCCC(O)C4)C)=O)C32)ccnc(Cl)c1F N1(C(C(N)CCc2cnc[nH]2)=O)CCCC(c2ccncc2)CC1 N1(CCC)CCC(C(=O)NC2CN(C(=O)CN(C)C(C)C)C3CC23)CC1 c1(CC)oc2ccccc2c1C(N1CCOC2(C1)CN(C(=O)C(C)(F)CC)C2)=O N1(C(c2ccc(CO)o2)=O)CCCCC(C2CN(C(c3ccncc3Cl)=O)C2)C1 CCCC(C(=O)OC)C(=O)N(CC(O)CNC(=O)COC(C)C)C N1(C(CC2CN(C(C)=O)C2)=O)CCC2(CC2C(=O)NC2CCCCCC2O)C1 CCC(C)C(O)CC(=O)NCCC(C)(C)NC(c1cn2ccsc2n1)=O c1(CCNC(CNC(=O)CNC(=O)Cc2ccsn2)=O)cccnc1O Cc1ocnc1CNC(=O)C(c1ccnn1C)NC(=O)COC1CC=CC1 c1(CC(=O)NCC(CC)NC(c2nocc2Cl)=O)csc(C2CCOCC2)n1 C1(N(C(=O)CC2CC2)CC)CCCN(C(c2ccc(C3(C#N)CC3)cc2)=O)C1 Cc1cc(F)cnc1C(N1CCCC1CN(C)C(c1cnc(C)n1C(F)F)=O)=O c1(NC(C(=O)OCCNC(C)=O)C)cc(C)nn1CC(F)(F)F CC1CN(C(=O)C=CC(C)(C)C)CCN1C(C1CCCN1C(N)=O)=O C(C)(CCNC(C1(OC)CC1)=O)N(C(C=C(CC)C)=O)C N1(C(C(C)S(N)(=O)=O)=O)CCC2C1CCCN2C(c1nccc2n[nH]cc12)=O C1(CNC(c2cc(OCC)ns2)=O)N(C(C2CCS2(=O)=O)=O)CCCC1(C)C C(=O)(C1CCc2c[nH]nc21)N(C)CC1(O)CCN(C(C2CC(OC)C2)=O)C1 CC1CC2CN(C(=O)C(C)O)CC2N1C(=O)Cn1cnnn1 O=C1CSCN1CCN1CCC(CC(=O)NCC(c2cccs2)O)C1 Cc1cc(Cl)ncc1S(=O)(=O)N1CCC2CN(C(=O)CN3CC4CC4C3)CC2C1 CCC(C)(C(=O)N1CCC([N+]C)C1)NCc1nccc(OC(F)F)n1 CCCCS(=O)(=O)CC(=O)N(C)CC1(O)CCN(C(c2ccccc2CO)=O)C1 CC1(C)CN(Cc2ccccc2Cl)CC1NCC1C2CCOCC12 CC(C(=O)NC1CCN(C(=O)Cc2nc(C3CC3)nn2C)C1C1CC1)C(C)(C)C Cc1ccc(C(N2CC(CC(=O)NC3CC(C)OC3=O)C3(CC3)C2)=O)c(O)c1 Cc1nc(C(N2CCCCC(NC(C3(CF)CCC3)=O)C2)=O)ccc1Br N1(C(C(COC)C)=O)CC(NC(=O)CSc2ccccn2)C(CC(N)=O)C1 c1(NC(N2CCC(CCO)CC2)=O)cnc2sccn12.c12cn(nn1)CC(=O)N2 c1(C(N(CC)CC)=O)ccc(C(=O)NCCC(c2ccccc2)O)cc1 N1(C(c2cccc(N)c2)=O)CCC(C)N(C(c2c[nH]ccc2=O)=O)CC1.CCN c1(NC)cnncc1C(=O)NCC1CCC1C.c1(CCN(C=O)C)cc[nH]n1 c1(C2(C(=O)NC(C)CNC(=O)CCn3cncn3)CC2)cn[nH]c1 c1(OC)c[nH]nc1C(=O)NC1CCC(NC(c2ccc(C)o2)=O)C1 c1(C(=O)NC2CN(C(C(COC)C)=O)CC(O)C2)nn(C)c(=O)c2ccccc12 C(=O)(C(C=C)CC)NC(COCC)C(=O)N1CC(CC)C1 C1(C(N2C(CNC(c3cccc4ccoc34)=O)CCC2)=O)CCc2ccnn2C1 c1(C(N2CCCCC(NC(CCSC)=O)CC2)=O)cnc2nccnc2c1 C1(CC(=O)NCC(C2CCC2)NC(C2CC(N(C)C)C2)=O)CCCCN1C c1(C(=O)NCCOCCCNC(c2c(CC)noc2)=O)[nH]cc2c1CCCC2 N1(C(c2c(OC)cncc2)=O)CCCC2(CCC(NC(=O)COC(C)=O)C2)C1 CCC(CC(=O)NC(C)C(C)n1cncn1)NC(=O)COCCCOC C1(C(=O)NCC(C)CNC(=O)CCc2ccsc2)C2CCN(C)CC12 c1(OCC(N2C(CNC(C(C)OC)=O)C3CC3C2)=O)cccc(F)c1F c1(C(C)O)ccccc1-n1ccc(-c2cnc(-c3cccs3)nc2)n1 N1(C(c2c(C)ccn2C)=O)CCC=C(C(=O)NCc2cnn(C(C)C)c2)C1 c1(C(=O)NC(C2CCCCC2)C)cccc(CNC(=O)C(O)c2ccsc2)n1 C1(C(=O)NC(C)CNC(=O)CCc2cnco2)CCC(=O)N1 CC1(C)CC(NC(C2(C)CCC(=O)N2)=O)CN1C(C12CC(C(C)(C)C)(C1)C2)=O C1(C(=O)NCCC(C)(C)NC(=O)C(CO)NC(N)=O)CCCCC1(F)F N1(C(c2c(CC)c[nH]c2)=O)CC(C)(C)C(NC(=O)C(C)CC2CCC2)C(C)(C)C1 C(=O)(C(CNC(=O)CCSC)Cc1ccoc1)NC(C#C)CC1CCCC1 N1(C(CCC=C(C)C)=O)CCCC(C)(C)C1CNC(c1cnc2c(c1)COC2)=O C1(CC(=O)NCCOC(CNC(c2n(C)nnc2)=O)(C)C)CCC(C)(C)O1 CN=S(=O)(c1ccc(C(=O)Nc2ccnc(-c3nn[nH]n3)c2)cc1)N(C)C Cc1cccc(F)c1C(=O)NC1CN(C(=O)Cc2ccc(F)cc2)CC1C(F)F c1(C(=O)NCC(CNC(C2CC(F)(F)C2)=O)C(F)(F)F)cccc2c1COC2 c1(C(=O)NCC2(NC(C3C(C)CCCC3)=O)CCC2)n[nH]c2c1CC1CC21 O=S(=O)(c1cnc(NCc2sncc2Br)c(Cl)c1)N1CCCC2(C1)OCCO2 CC1CCN(C(C2(C)CCN(C(c3ccc(CO)cc3F)=O)C2)=O)CC1(F)F Cc1ccc(C(N2CCC(C)(NC(c3cc4sc(C)cc4[nH]3)=O)C2)=O)c(F)c1F c1(C(=O)NCC2C(CNC(CCCN(C)C)=O)C2)cncc(N)n1 C1(CNC(C(CC#C)C2CC2)=O)CCN(C(=O)CCCCC)CCC1CO C(=O)(CCCCCCNC(C1(O)CCOCC1)=O)NC(C(CC)C)C(=O)NC n1(CC)nc(-c2ccc(Cl)cc2)nc1C(C)CN1CC(COc2ccccc2)C1 c1(NC(CC)(CC)CO)cc(Br)c2nccnc2c1Br N1(CC(=O)N(C(C)CNC(C)C(=O)N(C)C)CC)C(=O)CCCC1=O N1(C(C=C(CC)CC)=O)CCCCC1CCC(=O)N(C)CC1CCOC1C CCC(C)C(C(=O)N1CCCC1CNC(C1OCCC1CC)=O)OC N1(CC(C2CCCCO2)(C)O)CCCC(OC2CN(CC(=O)NC3CC3)C2)C1 c1(C(=O)NCCC(C)N(C(C(CC)OC)=O)C)cc2cc(F)cc(F)c2[nH]1 N1(C(c2cccc(C)n2)=O)C2CCC1CC(NC(C13CCC1C3)=O)C2 c1(C(N2C(CN(C)C(c3nnsc3N)=O)CCC2)=O)ccc(O)nn1 C1(NC(c2cccnn2)=O)CCCC12CN(C(c1cc3nc[nH]c3cn1)=O)C2 C1(C(C)C)CCCC(NC(c2ccc(CNC(=O)CC(C)(F)F)s2)=O)C1 C1(C(=O)NCC2CC(OC)CN2C(c2cncc(Br)n2)=O)CCC(N=[N+]=[N-])C1 C(c1nc2ccccc2[nH]1)=CC(N1C(CNC(C(C(C)C)(C)O)=O)CC(F)C1)=O C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CNC(CC(C)O)=O)CC(F)(F)F Cc1cn2c(C(=O)NC3CN(C(=O)C(C)CC(N)=O)C4CC34)cnc2s1 c1(C(=O)NCCC2CN(C(C(CCC)C)=O)C2)ccnc2cc[nH]c12 C1(C(NOCCOCC)=O)CN(C(=O)C(C)(C)CF)CC(C)O1 c1(C(=O)NC2C(NC(CCCC)=O)CCC2)ccc(C(C)C)cn1 c1(OC)cccc2ccc(C(=O)NCC(C)NC(c3cc(=O)n(C)cn3)=O)nc12 CC1CN(C(=O)CCc2nncs2)CC1(C)CNC(=O)C(c1cccn1C)=O C12(CN(C(=O)COC3CCOC3C)C1)C(=O)N2.c1(C2C(N)C2)ccncc1.CC C1(C(=O)NC23C(CN(C(c4ccc(C#C)cn4)=O)C2)C3)CC2(CCOCC2)CO1 N1(C(c2cccc(OCC(C)C)n2)=O)CCC2(C1)OC(=O)NC2(C)C O=S(=O)(c1cc(Cl)c(I)s1)Nc1cc(F)c(F)cc1Br C(CC(C)(C)NC(=O)Cc1cn[nH]c1)=CC(=O)N(C)CCc1cccs1 C1(C(=O)NC(C)CCO)CCCN(C(c2cc(Cl)c(Cl)s2)=O)C1 Cc1cc(CNC(=O)C(CCF)NC(c2ccc(CO)nc2)=O)cnc1F C1(C(N2C(C(=O)NC3CC(C)(CC)C3)C3CC3C2)=O)CC2OC1C1CC21 c1(C(=O)NCCC2(NC(c3cnn(C(F)F)c3)=O)CC2)ccc2c(c1)CCO2 N1(C(C2CC(CNC(c3nn(C)c(O)c3)=O)OC2)=O)CC2(CC(CC(F)(F)F)C2)C1 C(=O)(C(C)CC(C)(C)C)N1C(CN(C(=O)CC(C)(C)C(F)F)CC)CCC1 CCCC(O)CC(=O)NCCCCN(C(c1scnc1C1CC1)=O)CC N1(CC)CCCC(Cc2cnc(NC(=O)C(=O)NC)s2)C1.c12ccccc1c2=O N1(C(CC2(C)CN(C(c3coc(Cl)n3)=O)C2)=O)CCC(O)C(C)(CO)C1 Cn1cc(C#N)cc1C(N1CCC(O)(CNC(=O)CCC2CC2(F)F)C1)=O c1(C(N2C(C(=O)Nc3cnc(COC)nc3)CC3CC32)=O)cc2cn[nH]c2cn1 C(=O)(C(CC(C)C)N(C)C(c1sc(C)cc1C)=O)NC(C#C)C(C)OC N1(C(C(CCNC(=O)COC2CCCOC2)O)=O)CC(O)(C2CCC2)C1 c1(C(C)NC(CC(C)n2cccc2)=O)ccc(CNC(=O)COC2CC2)cc1 CC(C(=O)N1CC(CNC(c2sc(F)cc2Cl)=O)C2(CC2)C1)C(F)(F)C(F)F c1(C(=O)NC2(C)CCN(C(C(C)NC(CC)(C)C)=O)C2)cc2c(Cl)nccc2o1 C1(C(NOC(C(C)C)CN2CCCCC2)=O)(CF)CCN(C(=O)CP(C)(C)=O)C1 C1(n2c(C(CC)O)nc(CC(C)CC)n2)CC2(C1)CC1(CCCC1)C2 CC1(C)CCN(C(c2cccc(F)c2F)=O)C1CNC(C1CC=CCO1)=O c1(C(N2CC(NC(c3coc(Cl)n3)=O)C(O)C2)=O)cnc2ccccn2c1=O c1(CC)ccccc1CN(C)CC1CCCN1C(c1ncnnc1OC)=O C(C1=CCN(C(=O)CCCSC)CC1)NC(CCc1onc(C(C)OC)n1)=O O=C(CCCCC(F)(F)F)N1CC2(C1)CN(C(C1CC3(CCCCO3)C1)=O)CCO2 C(=O)(CCCCC(=O)NCC1CC1NC(=O)COCCc1cccs1)OC c1(OCCC(=O)NC2C(NC(C(CC)N3CCCC3=O)=O)CC2)cccc(C#N)c1 CON(CCC(=O)NC1C=C(C)CCC1)C(=O)Cc1nc(C)cs1 N1(C(C=COCC)=O)CCC2C(CCN2C(C2C(c3ccccc3)C2(F)F)=O)C1 C(=O)(CS(=O)(=O)C1CC1)NC(C)CN(C)C(C1CCCCN1S(C)(=O)=O)=O C1(N(C)C(=O)NC2CCCC23CC3)CCN(CCc2ccccc2)CC1 N1(C(c2ccccn2)=O)CCN(CC2CN(C(c3scnc3Cl)=O)C2)CC1 Cc1cnc(N2CCOC(C(C)NC(c3cc(Cl)ns3)=O)C2)nc1 c1(OC)ccc(C(=O)NCCC(C)CCNC(=O)Cc2cc(CC)no2)c(F)c1 C(C(C)(C)CNC(c1ccoc1Cl)=O)N(C(C1C(CC)C1)=O)CC Cc1nc(Cl)ccc1CC(=O)NCC1CCCCC1NC(=O)C(C)n1cccn1 N1(C(C2(OCC)CC2)=O)CC2CCC1C(NC(=O)C(C)CN(C(=O)C(C)C)C)C2 C1(CC(=O)N(C2CCCC2)CCCNC(CC(C)(C)C2CC2)=O)CCC(=O)NC1 C1(CC)CN(C(C2CC(=O)N(c3cc(OC)ccc3Cl)C2)=O)CC(=O)N1 C(=O)(CCC(CC)CC)N1CCC2(C(N(CCCC)CCCC)C2)C1 N1(C(C(C)(C)C2CC2)=O)CCC(O)(C2(NC(C3C(Cl)(Cl)C34CC4)=O)CC2)CC1 C1(CC(=O)NCC(CO)OC)CCCN(C(c2ccc(C#N)o2)=O)C1 N1(C(CNC(C)=O)=O)CCCC(O)(CN(C(=O)C=Cc2cccn2C)C)C1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCc1cccc(CNC(CCCCOC)=O)c1 c1(C(=O)NCC2(NC(=O)CNC(=O)C(F)(F)F)CCC2)cc(F)c2cn[nH]c2c1 C(=O)(CCCCCF)NCCn1ccc(C(=O)NCC(COC)C(C)C)c1 c1(C(CC)C)ccccc1C(=O)NCCN(c1cccc(N)n1)C(=O)COC c1(C(N(C)CCNC(=O)CCOCCO)=O)ccc2nc(O)[nH]c2n1.C1CO1 c1(OC)cccc(C(F)(F)C(=O)NC(CNC(=O)C=CC(=O)N(C)C)C2CC2)c1 N1(CC(=O)OC)CCC(=O)N(CCc2c(OCCC)cccc2)C1=O C1(CC(=O)N(C)CC)CC(C)(C)CN1C(=O)Cn1nccc1C c1(C(N(C)CC2(CNC(c3nocc3Cl)=O)CC2)=O)c[nH]c(=S)cn1 N1(C(C(C)(C(C)C)NC(C)=O)=O)C2CCC1CN(C(=O)C1=C(Cl)CCC1)CC2 c1(OC)cc(C(N2CC(NC(=O)C(c3ccc(F)cc3)C)C(CO)C2)=O)ccn1 N1(C(CC)=O)CCC(C)(C)C1.C(=O)(N(C(CSC(C)C)=O)C)C1CC1 C1CC(C(=O)NOCC)Oc2ccc(cc2)N1.CCCCCn1ccnc1 c1(C(=O)NC2(CC=C)CN(C(CC(=O)NCC#C)=O)C2)cccc(S(C)(=O)=O)c1 C(=O)(C(=O)N=S(C)(C)=O)N1CC(CNC(CCCCOC)=O)C(C)(C)C1 N1(C(C2C(=C)C2)=O)CC(C(=O)NC2CNC(=O)C23CC3)CC(C)(C)C1 c1(C(N2CCC(C(CNC(CCC(=C)Cl)=O)O)CC2)=O)ccc(C#N)cc1 CC1(C)CN(C(C2CC3CCC(C2)O3)=O)C(CNC(c2cnns2)=O)CO1 c1(CC(N2CCC(NC(c3ccc(C(C)C)nc3)=O)CC2)=O)ccc(Cl)c(F)c1 Cc1nc2ccc(Br)cc2cc1C(N1CC(O)(CNC(C2(CCF)CC2)=O)C1)=O c1(CC(=O)NCC(=O)N(C(c2ccccc2)CC)C)ccc(C)cn1 N1(C(C2(COC)CCCC2)=O)CCN(C)C(CNC(C2CC2(C)C(F)F)=O)C1 c1(-c2cccc(NC(Cc3cc(C)on3)=O)n2)cc(C(=O)N(C)C)ccc1F c1(C(N(CCC(C)NC(c2ccc(C3CC3)o2)=O)C)=O)snnc1C(C)(C)C C(C1C(=O)N1)OC.C1(C(=O)OC)CC(C(F)F)(NC(=O)CC(C2CC2)C2CC2)C1 C1(C(=O)NCCOCCOCCNC(c2cn(C)nc2)=O)CCS(=O)(=O)N1 c1(OC)c(Cl)ccc(C(N2CC(NC(=O)CC3(C)CC3(Cl)Cl)CC2C)=O)c1F C1(C(=O)NCCN(C(C(C)(C)OCC)=O)CC2CC2)CN2CCN1CC2 c1(C2(C)N=N2)ccccc1.C1(C(=O)O)(C)CC(NC(=O)OC(C)(C)C)C1 C12(C(N3CCN(C4CN(C(=O)COCCO)C4)CC3)=O)CC1CCC2(F)F C=CC(C)(C)CC(=O)N1CCC(COC)(NC(=O)C(C(C)C)n2ccnc2)C1 C1(C(N(C(C)CO)CC)=O)CSCN1C(=O)C.c1(CCC(=O)N)cccn1C C1(C(N(c2ccccc2)CC(OC)OC)=O)CC12CCN(C(c1ccsc1Br)=O)CC2 c1(C(N2CCCC(CC#N)C2)C(=O)NC(C(=O)OC)C)cc(F)c(OC)cc1Cl N1(C(C=CC)=O)CCCC(C(=O)NC(CO)C(C)CC)C1CC CC(C(C)C(=O)NC(c1ccccn1)(C)C)NC(=O)CCCC1CCCC1 c1(C(=O)NCC2N(C(C(COC)COC)=O)CC2)ccnc(S(N)(=O)=O)c1 Cc1cc(Br)cc2cc(C(=O)NCC(O)CN3CCC3)[nH]c12 C1(OC)CCCCN(CC(=O)NC(C)CNC(c2ccc3nn[nH]c3n2)=O)C1=O c1(C(N2CC(c3ccccc3)(C(=O)OC)OCC2)=O)nc2cc(F)cc(F)c2[nH]1 C1(CC(=O)NC2CC(n3cc(C(CC)(C)O)nn3)C2)(CO)CCCCC1 C(C)(C)(CC(=O)NC1(CF)CCN(C(C2CC2OC(C)(C)C)=O)C1)OC N1(C(C2C(CNC(c3c(C)cccc3C)=O)CC2)=O)CCCC2CCCC12 CC1=C(C)CC(C)(C(=O)NC(C)CCCNC(C2(C)CCC(C)C2)=O)CC1 c1(-c2ccc(C)o2)cccc2[nH]c(C(=O)Nc3cccc(Cl)c3)cc12 C1(C)(C(N(CCCCCC)C)=O)CCN(c2ccnc(NC)n2)C1 CCC(CC)CCC(=O)N1CCN(CC(=O)NCC(C)OO)CC1 c1(OC)cc(O)ncc1C(=O)N(CCCCN(C(=O)C(C)SC)C)C N1(C(c2c(C)noc2)=O)CCN(C(c2nc(C(F)(F)F)ccc2F)=O)CC1C C(=O)(CCCc1ccccn1)N(CC)CC1CCCN1C(=O)Cc1ccco1 CCC(C)C(CC)(c1nnnn1CCC1CC1)NC1CCCCC1=O.C1(N)CC1 C1(C(N2C(C3CCN(c4c(C)cncn4)CC3)CCCC2)=O)CN2CCCN1CC2 CC(C)CCC(O)C(=O)NC1CCCC1NC(c1cc(F)cc(F)c1F)=O C1(CNC(C2CCC(=O)N2)=O)CCN(CCN2CCCC2)CC1O N1(C(CC(C=C)C)=O)CC2CCC1C(C(=O)NC(C)Cc1cnc(C)s1)C2 N1(C(C=CC(=O)OCCCC)=O)CC(C)(C(=O)NCC2(C)CC(O)C2)CC1(C)C CCS(=O)CC(=O)N(C(c1ccccc1CC)CNC(=O)C(C)OC(C)(C)C)C CC(C)CCC(O)C(=O)NCCC1CCN(C(=O)CCCn2cnc(C#N)n2)C1 N1(C(c2cc(C)nc(Cl)c2N)=O)CC(C2CCCN(C(C3(CF)CC3)=O)C2)C1 n1(CC)c(C)cc(C(N2CCCC2(C)CNC(c2csc(C)c2OC)=O)=O)c1C FC1(F)CCCC1CCC(C1CC12CCCC2)c1nnnn1C1CC1.c1(O)ccncc1 C1(CNC(c2cccnc2Cl)=O)CCN(c2ncc(I)cn2)CC1(F)F C1(C2CN(C(=O)Nc3cn[nH]c3)C2)CCCCC1=O C(=O)(C1CCCc2sc(C(=O)OC)cc21)NCC1CC(F)(CNC(C(C)=CC)=O)C1 N1(C(CC=C)=O)CCN(C(=O)NC2CCC(C(=O)OC)C2)CC1 C1(NC(c2c(C#N)scc2)=O)CCCC12CN(C(=O)CC1CCC3(CC1)CC3)C2 c1(NC(N(C)CC2(C#N)CCOCC2)=O)ccc2nn(C)cc2c1 N1(C(C2ON=C(C(C)C)C2)=O)CCC2(CCC2NC(C2CCC(C)=C(C)C2)=O)CC1 C1(CNC(c2cccc(C(=O)NC)n2)=O)CN(C(=O)C(F)CC2CC2)CCCO1 c1(NC(C2(OC)CCSC2)=O)ccc(NC(=O)C(C)CC(C)C)cc1C C1(C(=O)NC(c2nnc(O)o2)C)C(CNC(C2CC=CCO2)=O)C1(C)C C12(C(=O)NCCC3(OC)CN(C(C4CCCN4C)=O)C3)CC1COC2(C)C C1(NC(C2C3C4CCC(C4)C23)=O)CCC2(CC1)CC2NC(=O)C=CCn1cncn1 C1(NC(c2c(C)snn2)=O)CC(C)N(C(c2ncsc2Br)=O)C1 c1(C(N2CC(C(=O)Nc3cnnc(Cl)c3Br)OCC2)=O)ccc([N+](=O)[O-])cc1 c1(C(=O)NC2C(OC)CN(C(=O)C(C3CCOCC3)C)C2)cc(S(N)(=O)=O)co1 C1(NC(CCC(C)O)=O)CCSC12CN(C(c1cccc[n+]1[O-])=O)C2 c1(CN2CCN(C(c3cc(C)ns3)=O)CC2)cncc(C#N)c1 Cc1ccc(C(O)C(=O)NCC2CCCN2C(=O)CCC=CC(C)C)cc1 Cn1cnc2ccc(CN3CCOCC3CC(F)F)cc12 C1(C(NOCC(=O)OCC)=O)C=CCN1C(=O)CC(C)F Cc1cccc2c(C(N3CCCC(F)(CNC(=O)C(F)C(C)C)C3)=O)n[nH]c12 CCC(C)C(C(=O)NC1CCCC1CN(C)C)NC(=O)CCOC c1(C(=O)NC(C2(O)CN(C(c3c(COC)nn[nH]3)=O)C2)C)cnc2cccnn12 C1(NC(=O)Cc2ccns2)CCCCC12CCN(C(=O)Cc1cnoc1)CC2 C1(C(=O)NC(C)(CNc2cnc(C#N)cn2)C2CCC2)CCc2nnc(O)n2C1 N1CC2CCN(C(=O)Cc3ccc(Cl)s3)C2C1.O=C1CCCN1CCO CCC(CC)(CC)C(=O)NCC(CC(C)C)C(=O)N(C(C)CC1CC1)C N(C(=NCCc1c(F)cccc1F)NCC(F)F)C1C(F)(F)COC1 C1(C(=O)NCC2CN(C(C3C(C)(Br)C3)=O)C2)Cc2cc(F)ccc2C(=O)O1 c1(COC)cc(C(=O)NC2CCCC2NC(=O)C=Cc2cc[nH]c2)n(C)c1 C1(CC)C(CC)CCC1N(C)OCC(O)CCF c1(C(N(C)CC2(CNC(C(C)CF)=O)CC2)=O)noc2c1COCC2 C1(n2cccn2)(CNC(C(CSC)O)=O)CCN(C(C2CC2C(F)F)=O)CC1 N1(C(=O)OC(C)(C)C)CCOC(C)(CCNC(=O)CCS(C)(=O)=O)C1 c1(C(=O)NC2CCN(C(c3c(SC)cccc3F)=O)C2)ccn2cc(C)nc2c1 n1(C(C)C)cc([N+](=O)[O-])c(=NCC2CCCN(C(C3CC=CCC3)=O)C2)[nH]1 C(C(CC(C)C)C(=O)NC)NC(C(CNC(CCOCC#C)=O)OC)=O N1(C(C(C)(C)N2CCCCC2)=O)CCC(C(N)=O)(NC(=O)CSCC(=O)NC)CC1 C1(CC#C)(NC(=O)CCC(C)NC(c2ccn(CC)n2)=O)CCOCC1 N1(C(CN(C(C(C)SCC)=O)C2CCC2)=O)CC(CO)C(C)(C)C1 N1(C(Cc2ccc(C)cc2)=O)CC(=CCC(C)(C)NC(=O)CC2CC2)OC(C)C1 c1(C(=O)NC(CNC(CCOC)=O)(C)CC(C)C)sc2cccc(F)c2c1Cl c1(CN(CCC(=O)OC(C)(C)C)CCCC2CC(F)C2)cccc2occc12 N1(C(CC(=O)OCC)=O)CCC2(CCC(C(=O)NCc3ccnc(Cl)c3)C2)CC1 C12(C(=O)NCC(C=C)(C)C)CC(CO)(CN1C(=O)CCNC(=O)OC)C2 C1(C(=O)NC2CC3CC3C2)CC(O)CN1C(C1CN(C2CC2)C1)=O C(CC(C)CCNC(=O)Cc1ccccc1CC=C)NC(CC=CC=C)=O C1(CNC(c2ncn(CC)c2)=O)CN(C(c2cc(SC)ccc2C)=O)CCN1C CCC(C)(COC)C(=O)N1CCCCC(C(=O)NCC(C2CCC2)OC)C1 N1(C(c2cccc(Cl)c2Br)C(=O)NCCSC)CC(C)CCC12CC2 c1(COC)cc(C(=O)NCCN(C)C(C2CCCC2C(=O)OC)=O)c(F)cc1C C12(C(N3CCC(CNC(CC4C(C)C4(F)F)=O)CC3)=O)CCC(F)(CC1)CC2 CC1(CNC(C2CCCOC2)=O)CCN(C(=O)CCCCN2CCCC2)C1 C1(C(N(C)CC2(NC(CC3C(C)OCC3)=O)CC2)=O)CC2(C1)CC(O)C2 C=C(Cl)C(C)(C)C(=O)NCC1CCCCN(C(C2CCN(S(C)(=O)=O)C2)=O)C1 c1(CC(=O)N(CC(C)NC(C2(O)CC2C(F)(F)F)=O)C)nc(F)ccc1Cl C1(C(N2CCCC(NC(c3cnns3)=O)CC2)=O)CC(=O)C12CCCC2 c12cccnc1C(=O)N2.C1(C(CC)=O)CC(NC(c2ccc(Cl)o2)=O)C1(C)C C1(C)(C(=O)NC(C(=O)NC)O)CCCN1C(=O)CC(C1CC1)C1CC1 N1(C(c2c(C)occ2)=O)CCC2CCN(C(C3CCC(N=[N+]=[N-])CC3)=O)CC2C1 N1(C(C(N2CCCC(N(C)C)C2)=O)=O)CCc2cc(Br)cc(Cl)c2C1 N1(C(c2nc(C(C)=O)sc2)=O)CCC(CC)C1CN(C(c1ccco1)=O)C1CC1 Cc1ccc(C(=O)NC(C)CC(=O)N(C)C)cc1O.C1C(C)(C)OCC(=O)N1C N1(C(C=Cc2ccn(C)c2)=O)CC(C)(C)CCC1CNC(c1cnco1)=O c1(C(=O)OCC)c(NC(C2CC2NC(=O)Cc2ccc(F)cn2)=O)sc(C)c1C CCC(C)CCC(=O)NCc1ccc(CNC(C2(F)CC=CCC2)=O)cc1 CC1CN(C(=O)C(Cl)Cl)CC1(C)C(=O)N(C)CC1(CO)CC1 CC1(C(=O)NCCCNC(=O)CC2(CO)CC2)CC(F)(F)C1 C(C(C)C(C)C(=O)N(C)CC1CCN(C(C2CC(OC)C2)=O)CC1)OC N(C1CC2(CN(C(c3ccc(F)s3)=O)C2)n2ccnc21)C(c1ccc(C)nn1)=O c1(NC)c(C(=O)N(C)CCOCCNC(C2CC2C)=O)sc2nccnc12 N1(C(C(CC)(F)F)=O)CCN(C(c2cc(CCCO)on2)=O)C(CCO)C1 c1(OC)cccc(C(=O)NC(Cc2ccccc2)CCNC(=O)C2CC2)n1 C1(NC(c2cnc(OC)nc2)=O)CC2CC(NC(C3CC3C(F)F)=O)CC2C1 C1(CC(=O)NCC(CCC)OC)CCCCC1NC(=O)C(=O)NC1CC1 C1(NC(CCc2nc(C)c(C)[nH]2)=O)CC2CCC(C1)N2c1ncnc(=N)[nH]1 N1(C(c2ccc(SC)s2)=O)CCC(O)C(N(C(=O)CCc2ncc[nH]2)C)C1 c1(CCC(=O)NCC2(CNC(c3c(C)scc3)=O)CC2)ccc(Cl)cc1Cl N1(C(c2c(CC)csc2)=O)CC2(C(=O)NCC(c3nccs3)C)CCC1CC2 N1(C(C2(OC)CCCCC2)=O)CC2CC(NC(c3ncnn3C)=O)C2C1 Cc1ncc(NC(=O)C(C2CCCC2)NC(=O)CC2C=CCCC2)c(C)c1 N1(CC)CCOC(C(=O)NC(CNC(=O)CCOC2CCOCC2)C(C)(C)C)C1 N1(C(c2occ(OC)c(=O)c2)=O)CCCC2(CCC2NC(C2CCCC2C)=O)C1 C(=O)(C(CC(C)C)C(C)C)NCC1C2CN(C(c3c(C)scc3)=O)C1C2 N1(C(C(CC=CC)NC(=O)CCc2ccsc2)=O)CCC(C)C(O)CC1 C(=O)(C#CC1CCC1)N1CC(OCC(=O)N(C)CC2CCC(=O)N2)C1 C(=O)(C(Cc1ccsc1)NC(=O)C(N)C1(C)CC1)OC CCCCC(CNC(c1snc(Cl)c1Cl)=O)NC(c1ncc(NC)nc1)=O CC(CC1CC1)C(=O)NCC1CCN1C(c1occc1Cl)=O C(=O)(C(C)(F)C(C)(C)F)NCC(C(C)(C)C)NC(c1ccc(C#N)cn1)=O c1(C(N2CC(C(C)OC)C2)=O)cnn(CCNC(=O)C(C)C2CCCO2)c1 c1(OC)cccnc1CNC(C1(NCc2cccs2)CCC(C(CC)CC)C1)=O CN1CC(NC(=O)C(=O)Nc2ccn(-c3ccccc3)n2)CC12CCOCC2 C(=O)(CC(C)(O)COC)NCC(C)N(C(=O)Cn1nnc(-c2ccsc2)n1)CC N1(C(CSCc2cn(CC(C)(C)CO)nn2)=O)CCC(O)(C(F)(F)F)C1 Cc1c(C(N2CCCC(CNC(=O)CS(C)(=O)=O)CC2)=O)ccnc1Cl CCC(CC(=O)N1CC(CNC(c2ccc(-n3cnnn3)cn2)=O)C(O)C1)OC c1(C(=O)NC2(CC=C)CN(C(c3ccn(CCF)n3)=O)C2)nc2c(s1)COCC2 CC1CC(C)N(C(c2ccnn2CCF)=O)CCN1C(c1cc(O)nc(Cl)c1)=O C1(CC=C)(NC(c2cnc(C3CC3)nc2)=O)CCN(C(=O)C(C)n2cncn2)C1 c1(C(=O)NC2CCN(C(COC)=O)C2)cnc2c(c1)CCC(=O)N2 N1(C(C)=O)CSCC1NC(=O)OCC1(F)CC(C(C)(C)C)C1 N1(C(CC(CC)OC)=O)CCC(C2CC2)(CNC(C2CCCN2C(C)=O)=O)C1 C1(C(N(C2CC(SC)C2)C)=O)CCC(O)CN1C(=O)Cc1cccc(F)c1 c1(OC)cc2ccccc2cc1C(N1CC(CNC(=O)CC2CCC(=O)N2)C1)=O N1(C(Cc2c(C)ocn2)=O)CCC2(CCCN2C(C2CC=CCC2C)=O)C1 c1(NC(C2CC23CN(C(c2cc(Cl)c(Cl)s2)=O)C3)=O)nc(Cl)ccc1I N1(C(C(C=C=C)C)=O)CCCCCC(NC(c2cc(C)cc(C)c2C)=O)C1 Cc1cn2c(n1)C(C)CC(C(=O)N(CCCN(C(=O)CCC1CCCO1)C)C)C2 CC1(C)CC(CNC(=O)C=Cc2cnc[nH]2)CN1C(c1cccc(N)c1)=O c1(OC)cc(C(=O)NC2CN(C(=O)CCC3CC3(F)F)CC2OC)ccc1Cl C12(CCNC(CC3C(=O)NC(=O)N3)=O)CCC1CN(C(=O)C(=O)NC1CC1)C2 N1(C(C(C)C2CCCC2)=O)CC(C2(NC(=O)CCN3CCC3)CC2)C1 n1(CC(N2CC3C(CNC(c4cc5sccc5[nH]4)=O)(C3)C2)=O)ccc(O)nc1=O Cc1nccn2ncc(NC(=O)C(N3CC4CCCC4(N)C3)=O)c12.C1CO1 N1(C(C2N(C(C(CC)n3cncn3)=O)C3(CC2)CC3)=O)CC(O)C(O)C12CCC2 C1(C)(C(=O)NCC(C)(F)CNC(C2CC3CC3C2)=O)CCC2CC2C1 Cc1cc(C)n(CCC(=O)NCC2(C)CCC(NC(=O)CCOC3CCC3)C2)n1 c1(C(N2CCOC(CN=c3[nH]nco3)C2)=O)ccn2ccccc12 C1(CN(C(C(CC)OC)=O)C)CCCN(C(c2ccc(CSC(F)F)o2)=O)C1 c1(C(=O)NCC2C3CN(C(C4CC(=C)C4)=O)CC32)cc(F)c(C)cc1F N1(C(C(C(C)NC(c2cc(C(N)=O)co2)=O)C)=O)CC(O)(C2CCC2)C1 C(=O)(CC(=O)N1C(C(=O)NC(c2ccncc2)(C)C)CC1C)NCC c1(SCC(N2CC(NC3C(C(=O)OCCSCC)C3)C2)=O)ccccc1OC n1(CC#C)cccc1C(=O)N(C)CCNC(C12CC(C1)C2)=O N1(C(c2c(C(C)C)n[nH]c2)=O)CCC2(CCN(C(C3CCC(C)O3)=O)CC2)C1 c1(CC(N2CC(N(C(COCCOCC)=O)C)C2)=O)c[nH]nc1O c1(NC(C2(C)N(C(C3C(C(=O)OCC)C3)=O)CCC2)=O)cnc(Cl)nc1C c1(C(N(CCNC(=O)COc2ccsn2)CC)=O)cccc2nc(C)sc12 C=Cn1nccc1C(N1CC(NC(=O)C=CCOCC(F)(F)F)CC1CO)=O C1(NC(c2c(C)noc2)=O)CC(F)CN(C(=O)C(C)Oc2ccc(Cl)cc2Cl)C1 CC(CC(=O)NC1CCC(NC(=O)CN(C)C)C1)C1CCCC1 N1(C(C=C(CCC)C)=O)CCSCC1C(=O)NC(c1ccc(C)cc1)CO C1(CC(=O)NC(CC)(C)CNC(c2nncs2)=O)CC=CCN1C CC1CCC(NC(=O)COCCCF)CN1C(c1ccnc(-n2cccn2)c1)=O C1(C(N(C)CCn2cnnn2)=O)CCCCC1NC(C1CC(CCO)C1)=O C1(NC(C=CCN(CC)CC)=O)CC2CC(NC(C3(C)CC4CC4C3)=O)CC2C1 c1(C(N(CCN(C(C2SCCCS2)=O)CC)CC)=O)cnn2c1N(C)CC2 C(=O)(C(C)N(C(C1CN(C2COC2)C1)=O)C1CC1)N(CC)CC C1(O)(CNC(c2ccco2)=O)CCCN(C(C2(c3ccccc3)CC(O)C2)=O)C1 C1(C(N2CC(C(C)NC(c3ccc(SC)nc3)=O)C2)=O)NC(=O)N2CCCCC12 C=CCCCCCC(=O)NC1(CN(C)C(C2(C)CCC(F)(F)C2)=O)CC1 n1(CC(=O)NCCc2ccc(C)s2)cc(Nc2oc(C)nc2C)c2ccccc12 N1(C(C2C(COC)CCO2)=O)CC2CC1CN(C(c1cc3occc3n1C)=O)C2 C1(NC(CC2(C(=C)F)CCC2)=O)CC2(CCN(C(c3cccc(N)n3)=O)C2)C1 C(=O)(C#CC12CC3CC(CC(C3)C1)C2)N(CC=C)CC12CCC(CC1)C2 C1(NC(c2c(CC)c[nH]c2)=O)CN(C(c2cc(C(F)(F)F)n(C)n2)=O)C2CC12 CC1(C)NC(=O)CC1C(=O)NCC1(C(N)=O)CN(C(c2ccc(Cl)nc2O)=O)C1 c1(Cc2c(OC)cccc2)nc(C)ccc1C(=O)N(CC(C)C)C CCCCCCCCC(=O)N1CCCC(NC(c2ncc(C(F)F)cc2C)=O)C1 Cc1cn2nc(N3CC=C(CCNC(=O)Cc4cc(O)nc(O)n4)CC3)sc2n1 C1(NC(c2c(OC)ccs2)=O)CN(C(c2cc(O)nc(Cl)c2)=O)C2(CCOC2)C1 CCCC(CC)CCC(=O)NC1CCN(C(=O)CCSCC(N)=O)C1C CN1CC(CNC(=O)CC(C)(C)CNC(=O)CC(C2CC2)C2CC2)CC1(C)C C1(C(=O)NCC(=O)O)CC2(CCN(C(=O)Nc3ccc(C(=O)CF)cc3)C2)C1 c1(C(=O)NCC(CC)(CC)NC(=O)Cc2cncs2)nccc2n[nH]cc12 C(c1cn(C)cn1)=CC(=O)N(C)CCNC(C1(O)CCSC1)=O N1(C(C2CCC(C(=O)OC)C2)=O)CCC(C(C)(C)C)(CNC(=O)CC(F)(F)F)C1 C=C(Cl)CC(C(=O)N1CC(C)(CSC)C1)NC(=O)CCC(C)(C)F NS(=O)(=O)c1cc(C(N2CC(C3(NC(=O)Cc4cncnc4)CC3)C2)=O)c(Cl)o1 N1(C(CC(CC)CC)=O)CCS(=O)(=O)C(CCNC(=O)CC(C)C(F)(F)F)C1 CC(C(=O)NC1CC2(C1)CC(NC(C1OCCN(C)C1=O)=O)C2)C(C)(C)C c1(C(N(CC(C)(C)NC(Cc2ccc(C)c(Cl)c2)=O)C)=O)cc(Cl)cc(F)c1F Cc1cc(C(N2CCCC(C(=O)NC3(C)CCOCC3)CC2)=O)nnc1C C(CC(=O)N(CC(O)CN(C)C(c1sc(COC)nc1C)=O)C)(C(C)C)OCC C1(NC(CCc2ccc(OC)cc2)=O)CN(C(C2CC2)=O)CCC1CO.C1CC1 N1(C(c2ccc(OC)cc2F)=O)CCC2(CC1)CN(C(=O)CC1CC(F)(F)C1)C2 C1(CNC(C=CC(C)C)=O)CC(O)CN1C(=O)CCc1cc[nH]n1 c1(C(c2nnnn2Cc2nnn(C)n2)NCC2C(C)C2)csc(Cl)c1Cl C(CCCCCCCC1OCCO1)(c1nnnn1C1CC1)NC(C(C)N=[N+]=[N-])C CCC(C)C(O)C(=O)N1CCOC(CCNC(c2ccc(C#N)nc2)=O)C1 c1(NC(C2N(C(c3cn(CCC)nc3)=O)CCC2C)=O)ccc(O)c(=O)cc1 N(C1CCCc2ncccc21)C(=O)NCCC1CCCC1(F)F C1(O)(CNC(Cc2scc(C)c2)=O)CCN(C(C2CC(CN(C)C)C2)=O)C1 c1(C(=O)NC(COCc2cccs2)C(=O)O)ccc2c(c1)OC1(CCCCCC1)O2 C1(C(N2CCC(N(C(=O)C(F)=C3CCCC3)C)C2)=O)CCc2c(ncn2C)C1 S(=O)(=O)(c1ccc(C)cc1)N1CCCC(C(=O)Nc2c(CC)noc2C)C1 C1(N2CCCC(C)(O)CC2)CC2(CCN(C(=O)COC3CCOC3)CC2)C1 N(C1CC(C)(C)Oc2ccc(Cl)cc21)SCC(=O)N(CC(F)F)C Cc1cc(C(=O)N(C)CCNC(C2CC2C(F)(F)F)=O)cnc1C(F)(F)F c1(OCCCOC)ccc(Nc2nccc(N3CCC(C)(C(F)(F)F)C3)n2)cc1 CS(=O)c1ccc(CC(N2CC(CNC(c3cccc4ccnn34)=O)C2)=O)cc1 C(=O)(CCCC(C)(F)F)N1C(C)CC(NC(c2cccc(OC(F)F)c2)=O)CC1 N1(C(C(CC=C)(C)C)=O)CCOCC(C)(CNC(C2(F)CC2C)=O)C1 N1(C(C=C(CC)CC)=O)CC2CC(NC(=O)Cc3cc(F)ccc3Cl)CC1C2 c1(C(=O)NCC2CCN(C(c3ccco3)=O)CC2)cccc2c1CCO2 CCCC(C)(C)CC(=O)N1CCCC(CC)(NC(C2CC3(C2)CC(C)C3)=O)C1 c1(CC=O)ccc(Br)s1.CC(CCN(C(=O)Cc1cn[nH]c1)CC)N(C)C C(CCC(C)C(=O)NC1CCC(CNC(c2occc2C(C)C)=O)CC1)OC Cc1cc(C)c(CC(=O)NC2CCN(C(c3cn(C)c(O)n3)=O)CC2)s1 Cc1cn2cc(-c3sc(C(N4C(C(=O)NC5CC5)CC5CC54)=O)c(C)n3)sc2n1 C(C)(CN=c1[nH]c(C)cc(=NCc2nc(C)ccc2Br)[nH]1)OC N1(C(CC2(COC)CC2)=O)CCC2(CCCCN(C(C3CC3C3CC3)=O)C2)C1 C1(COC)CN(C(C2CCS2(=O)=O)=O)CCN1C(=O)CC1(C)CC1 N1(C(c2cscn2)=O)CCN(C(=O)Cc2ccc(O)c(F)c2)C2CC12 c1(C(N(CCCNC(Cc2scc(C)n2)=O)C(C)C)=O)ccc(O)cn1 C1(CNC(C(C)OC)=O)CC(F)CN1C(=O)C(C)Cc1cnc[nH]1 c1(C(C)C)ncc(CNC(=O)C(N2CCC(C)C2)=O)cn1 c1(C(N2CCC(N(C(C34CC(C3)C4)=O)CC)C2)=O)cc(OC)ncc1F CC(C(=O)NCC1(CNC(=O)CNC(=O)NC2CC2)CC1)C(C)(F)F C1(C(N(C)C)=O)CCN(C(=NCCCC2CCCO2)NCCCOCF)C1 N1(C(COCCCC)=O)CCOC(CNC(=O)Cc2ccc(OC)s2)C1 C(C)(C)(CCCC(=O)NCC1CCCC(OC)C1)NC(CCC=CC)=O c1(C(N2CC(CNc3nc(C)nc(Cl)c3)OCCC2)=O)cc2c([nH]1)CCCC2 CC1(C)CCOC1CCC(N1CCC(NC(=O)Cn2ccnn2)C1)=O N1(C(CC(CNC(CCSC(C)C)=O)(C)C)=O)CC2(CC(CO)CO2)C1 c1(-n2cc(OC3CN(C(=O)NCCCC(=C)Cl)C3)nn2)ccc(F)cc1 c1(C(=O)NCC2CCN(C(COCCCC)=O)CC2)cccc(C#CC2CC2)c1 Cc1cn2c(C(N3CC=CC3CNC(=O)COCC(C)C)=O)cnc2s1 C1(NC(c2ncccc2O)=O)CN(C(c2ccn(C(F)F)n2)=O)CC2(CC2)C1 N1(C(COC(CNC(CCC#C)=O)(C)C)=O)CC(CO)C(O)C1 C1(C(N(C)Cc2cnn(C)c2)=O)CCOCCN1C(C1CC2CCC1CC2)=O c1(C(=O)NC(C)C)ncc2c(n1)CCN(N1CCN(C(=O)OC(C)(C)C)CC1)C2 Cc1cc(F)ccc1S(=O)(=O)N1CCNC(C(=O)NCc2cncnc2)C1 CCCC(C(=O)Nc1ccsc1)NC(=O)C(Cl)Cl C1(NC(C2CCC(C)C2)=O)CCC2(CC1)CN(C(C1CCN1C)=O)C2 S(=O)(=O)(c1cccnc1NCC1CCC(F)(F)C1)N(C)Cc1ncc(C2CC2)o1 C1(C(N(C)Cc2nc[nH]n2)=O)C(C2CC2)CCN1C(c1cncc(CO)c1)=O C(c1c(Cl)nc2sccn12)=CC(=O)NCC(C1(O)CCN(C(=O)CCF)C1)C C(CC(C(=O)NC(C1CCC1)C)NC(=O)Cc1cnn(C)c1C)SC C(=O)(C(C)(C)CC(=O)N1CCN2CC1C2=O)OC.C1(OCCF)CC2(C1)CC2F C1(NC(C(C=C)OC)=O)CCN(C(=O)CNc2ccccc2)C1(C)C c1(CCC(=O)NCC(CCOC)NC(c2nc(C)nn2C)=O)ccccc1C C1(SCC)CCCN(C(=O)CC2CCN(C(=O)Cc3sccc3C)C2)C1 Cc1nn(C)c(C(=O)NCC2(NC(=O)C(C)(C)n3cnnn3)CC2)c1[N+](=O)[O-] C1(NC(CNC(C2C(C)C2)=O)=O)CC2CN(C(=O)C(F)(F)C3CC3)CC2C1 C1(N(C(=O)C(O)C(C)SC)CC)CCN(C(=O)Cc2ccccc2)CC1 N1(C(C(CC)COC)=O)CC2(CC2)CC1CNC(=O)Cc1ccccc1C(N)=O N1(C(CS(CC)=O)=O)CC2(C1)C(NC(c1nc(C)c(C)nc1O)=O)CCS2(=O)=O C(C)(C(=O)OC(C)(C)C)(C(=O)N1C(C)CN(C(=O)C(C)(F)F)CC1C)OC C1(NC(c2cc(COC)c(F)cc2)=O)CC2CN(c3nccnc3OC)CC2C1 Cc1cc(CC(=O)NC2CCC(N(C)C(c3cnc[nH]3)=O)C2)no1 C1(NC(CCC2(CCC#C)N=N2)=O)CC2CCCC(C1)N2C(C1(Cl)CC1(F)F)=O N1(C(CCC(CC)NC(c2nnsc2C)=O)=O)CCC(O)C(F)(F)C1 c1(C(=O)NC2CN(C(C(C=C=C)C)=O)CC(O)C2)cc2nccnc2cc1F N(C1CCCc2c1cnn2C(C)(C)C)CC(=O)N(C(C)CCO)C CC1CN(C(=O)CCOc2ccc(F)cc2)CC1NC(C12CCC(CC1)C2)=O C#Cc1cccc(C(N2CCN(C)C(CNC(C3CC(=O)N(C)C3)=O)C2)=O)c1 C(C(C(=O)N(C(C)CN(C)C)C)NC(=O)CC1CC=CCC1)OC C(CC(C(=O)N1CCC(C)(O)C1)NC(C1CC2(CC2)CO1)=O)N(C)C C=CC(F)(F)C(=O)NC1CC(CNC(c2cc(C)n(C)c2)=O)CC1O c1(C(=O)NCC2CC3(CN(C(CC(CC)OC)=O)C3)C2)n[nH]c2ccc(Cl)cc12 c1(C(N2C(C)C3CC2C3NC(=O)CCCNC(N)=O)=O)c(F)ccc(N)c1F CC1(C)C2CCC(C2)C1C(=O)NCCC1CCCN1C(=O)CCNC(=O)CO CN1CCCC(C)(C(N2CC(F)(CNC(C3CC4CCCC4C3)=O)C2)=O)C1 C1(NC(c2scc(CNC(C(C)=NOCC#N)=O)c2)=O)CNC(=O)CC1C c1(CNC(C(C=CC)O)=O)ccc2c(c1)CN(C(c1ccc(F)c(F)c1C)=O)C2 CCCC(C)(O)CC(=O)NC(CC(=O)N(C1(c2cc[nH]n2)CC1)C)C(C)OC C(=O)(C(COC)CC(C)C)NCC1(C(N2CCC(O)(CC)C2)=O)CCOC1 N1(C(c2cccc(OC(F)F)c2)C(=O)NC(CC)(C)C)CC2CCC(C1)C2(F)F c1(OCC)cc(C(c2nnnn2C2(C)CC2)NCCCC(=O)OC(C)(C)C)[nH]n1 C(CC1=CCN(C)CC1)NC(C(CCCNC(CC=CC)=O)O)=O N1(C(Cc2cc(C)on2)=O)CCC2(NC(=O)OC(C)(C)C)CCCCC12 C(CCN=[N+]=[N-])N(C(C(C1(O)CCC1)NC(=O)NC(CC)C)=O)C CCC(CC)CC(C(=O)NC)NCc1ccc(-c2cncnc2)cc1 N1(C(C(N2CCCCCC2)C)=O)CCCC1(C)CNC(c1ccoc1Cl)=O C1(C(=O)NCc2n(CCC)ccn2)CCC2CCC1N2C(=O)CC1CCCO1 c1(C(=O)OC)ccccc1S(=O)CC.c12nc(cs1)CNC(=O)C2 C1(C(=O)OC)C=CCN1C(=O)COC1CC(CNC(=O)Cc2conc2C)C1 C1(=CC(N2C3CN(C(CCCOC)=O)CC2CC3)=O)CCOc2ccccc21 c1(CN(C)CC2CNC(C)(C)C2)cccc(OCC(F)(F)F)n1 C1(C(=O)NCCC2CCSC2)CCCN(C(C2(Cl)CC2(F)F)=O)CC1 c1(C(=O)NCCN(C(c2c(C)[nH][nH]c2=N)=O)C)cc2cccc(F)c2o1 CC1(C)OCc2cc(NC(=O)Nc3cnn(-c4ccccc4F)c3N)ccc21 c1(C2(C(=O)NC3(CNC(c4c(C)nc[nH]4)=O)CCOC3)CCC2)ccccc1Cl C1(N(C(C(COC)NC(C)=O)=O)C)CN(C(C2CCC3(CC3)C2)=O)CC12CC2 O=C(C1CCSc2ccccc21)NC1CC(NC(C2CN3CCN2CC3)=O)C1 C(=O)(C(C)(COC)CC)NCCCN(C(c1c(CC)occ1)=O)C C(=O)(CC(C)CC(=O)N1CC2(C1)CN(C(C1(C(=O)N(C)C)CC1)=O)C2)OC N1(C(C23N(C(c4c(=O)ccn(C)c4)=O)CCC2C3)=O)C2CCC1CC(CO)C2 c1(C(=O)NCCNC(c2cc(C(C)(C)C)n[nH]2)=O)cnn2c1CCCC2 C12(C(=O)NCC3N(C(c4n(C(C)C)nnc4)=O)CCOC3)CC1COC21CCC1 c1(C(N2C(C)CCC2C(N2CCC(C(=O)N(C)C)C2)=O)=O)ccnc2ncccc12 C1(C(C)C)C(NC(c2ccn(-c3ccccc3Cl)n2)=O)CCN1C(=O)C1=CCC1 Cc1ncccc1CC(=O)NC(C)(CNC(c1cnn(C2CCC2)c1C)=O)CO c1(C(=O)NC(C(C)C)CNC(C2CC3CCCCC23)=O)cc(F)cc(Cl)c1O C1(Cn2cc(C(C)C)nn2)OCC2CCC1C2.C12C(C1(C)C)C(=O)NC2 CCC(C(=O)NCC1CC(F)(CNC(=O)Cn2nnc(C3CC3)n2)C1)C(F)(F)F c1(C(N2C(CCNC(C3(N(C)C)CC3)=O)CCCC2)=O)c[nH]nc1[N+](=O)[O-] c1(OC)cccc(C(C(=O)NC2(C)CC(C)(C)C2)N(C)Cc2ccc(F)cc2)c1 c1(CC(=O)NC(C)CN(C)C(C2(C#N)CCC2)=O)nn(C)c2ccccc12 C12(C(=O)NC3C(NC(c4nc(COC)sc4)=O)CCCC3)CC3CC(CC1C3)C2 c1(C(N2C(C)C(C(F)(F)F)CC2)C(=O)NC2CCC2)cc(Cl)c(Cl)c(Cl)c1 C1(NC(c2n(C)ncc2)=O)CCN(C(=O)CC2CCCC(=O)N2)C1(C)C C1(Oc2cn(C)nc2)CC(CO)N(C(c2cccc(CO)c2)=O)C1.C1(C(=O)N)CCC1 C=CCC(CC(=O)NCCN=[N+]=[N-])NC(=O)CCCC1(COC)N=N1 c1(SCC(N2C(C(=O)OC)CC(n3cc(CSC)nn3)C2)=O)cc(F)cnc1Cl c1(CCC(=O)NC(CNC(CCC(=C)Br)=O)C(C)(C)C)ccc(O)c(Cl)c1 C1(C(=O)NCC2(NCc3nc[nH]n3)CCCC2)CC2(CC2)C(=O)O1.CC1C(=O)N1 C12(CC(=O)NC(c3nc[nH]n3)CNC(=O)C=Cc3cccnc3)CCC(CC1)C2 c1(C(=O)NCC(C)N(C)C(c2cn(C)nc2Cl)=O)cccc2c1CNC2=O N1(C(c2c(C)con2)=O)CCC2(CCCC2NC(C2(F)CCCCC2)=O)C1 O=S(=O)(c1ccnn1C1CC1(F)F)Nc1cnn(-c2ccccc2)n1 CC(O)C(C)C(=O)NCCOC1CCN(C(=O)CNC(=O)CCN(C)C)C1 C(=O)(C1=Cc2ccccc2C1)N(CCCNC(=O)C(O)C1CCCC1)C C12(CC3CCC1CC3)NC2.CCCCCCC(C(C)c1nnnn1CCC)OC c1(CC(=O)N(CC(C)NC(C2CCS2(=O)=O)=O)C)ccc(N2CCCC2=O)cc1 C1(CNC(C2CCN(C(C)=O)C2)=O)CC(O)CN1C(C1(N2CCOCC2)CC1)=O C(N=c1[nH]c(=NCCCc2nccs2)[nH]c2c1CSC2)c1nc(C(F)F)sc1 N1(C(CC=CC=C)=O)CC(NC(=O)CC2(C)CC(F)(F)C2)CC12CCOCC2 C1(NC(Cc2cc(C)sc2)=O)CC2(CCN(C(=O)C3CC3)C2)C1 c1(C(=O)Nc2c[nH]nc2CNC(c2ccccc2C2CC2)=O)cnc(Cl)c(F)c1 CCC(C)CC(=O)C(=O)N1CC2CC(C(=O)NOCC=C(C)C)C(C2)C1 CCCC(C(=O)NCC1(C)CCCN1C(=O)C=CC(CC)=CC)NC(N)=O C1(=CCNC(C(COC)O)=O)CCN(C(C2CCCCS2)=O)CC1 C(C1c2ccsc2CCN1C(C1CCCCC12OCCO2)=O)NC(C(=O)N(C)C)=O C1(CCn2cc(SC(c3cnc(C(=O)OC)n3C)=O)nn2)CC2CCCCN2C1 N1(C(=O)OC(C)(C)C)CC2CCC2(C(=O)NC(c2nn[nH]n2)C2CC2)C1 C1(C(C(=O)NC(COC)CNC(=O)C(C)=C2CCC2)C)CCOCC1 Cc1ccc2c(c1)CCC(C(=O)N(CC(C)C)Cc1cnsc1)O2 N1(C(c2cc(CCNC(CC=C=C)=O)on2)=O)CCC(C)(C#N)C1 c1(CN2CCCC(NC(c3c(C)nn(C)c3)=O)CC2)cc(F)cc([N+](=O)[O-])c1Br Cc1c(C(=O)N(C)CC2CCCN(C(=O)CCc3nccs3)C2)ccc(F)c1F C1(NC(C(CC#C)O)=O)CCCN(C(c2cnnn2CC)=O)C1CC C1(NC(c2cc(C)c(C(F)F)nc2)=O)CCCN(C(c2sccc2Cl)=O)CC1F c1(CN(C(CCN(C(=O)C(C)n2cnnn2)CC=C)=O)C)cc(C)cs1 CC1CCN(C(=O)C=CCN(C)C)CCN1C(C1CCCCC1)=O Cc1nn(C)c(C)c1C(N1CC(n2cc(C(CC(C)(C)C(C)(C)O)=O)nn2)C1)=O N1(C(C2C(CC)C2)=O)CC2(C1)CN(C(=O)C(O)c1ccsc1)CC(C)(C)O2 CC1CN(C(=O)CCCOc2ccccc2)CC1CNC(=O)C=CI N1(C(c2cccc(CSC)c2)=O)CCC(C)C(NC(=O)CSC)C1 N1(C(C2CC=CCN2C(c2cc(CO)[nH]n2)=O)=O)CCC(CO)C(O)C1 C(=O)(CC(O)(C(F)(F)F)c1ccccc1)Nc1ccc(OCC#N)nc1 Cc1ccc(F)c(SCC2(O)CCN(C)C2)c1.N12CCC(C1)Cn1nnnc12 C(=O)(C1=CC2C=CC1C2)N1CC(C(N(C(C)CC2CC2)C)=O)OCC1 Cn1ncc(C(=O)NCC2CCCN2C(C2CCCCO2)=O)c1C(F)F C12(C(=O)NCC(C)N(C(C(CC)(C)OC)=O)C)CC3CC(C1)CC(C)(C3)C2 c1(C(=O)NCCCCN(C(C(C)SCCCC)=O)C)nc(C)c(N)cc1C N1(CCOC)CC(C(=O)NC(C)(C)CN(C)C(c2csc(C)n2)=O)CC1=O C1(NC(=O)CCOC2CCC2)CC2(CCN(C(=O)CC3CCCCCO3)CC2)C1 N1(S(CCOCOC)(=O)=O)CC2CCC1CN2.C1(C=O)C2COCC12 CC(C)CC(C)C(=O)N(C1CCN(C(c2coc(C3CCCC3)n2)=O)C1)C c1(C(N(CC(C)N(C(c2cc(OC)c(F)cc2)=O)C)C)=O)[nH]nc([N+](=O)[O-])c1Cl c1(NC(CC(=O)OCC)=O)ccc2c(c1)CN(C(c1nc(Br)c(Br)cc1Br)=O)C2 c1(C(C(=O)NC(CC)CNC(=O)C=CC(=O)N(C)C)F)c(F)cccc1F C1(NC(c2c(CNC(=O)CN3CCOC3=O)ocn2)=O)CC2(CCC2)C1O C1(CC(=O)NCC(C)(C)C(N)=O)CCCN(C(=O)CCc2cn[nH]c2)CC1 c1(C(=O)NC(C(C)NC(C2(COCC)CC2)=O)C)cc(C)nc(Cl)c1N c1(C(=O)NCCNC(=O)Cc2ccc(F)cc2C(F)(F)F)cnc2n1CCCC2 CC(C)C(CO)C(=O)N1CCC(OCCNC(=O)CC2CCC(C)(O)CC2)CC1 CN1CCCc2ccc(NCc3nc4ccccc4n3C)cc2C1 Cc1cc(Cl)ccc1-n1cc(CCNC(=O)CNC2CCOC2C)nn1 N1(C(c2occ(C)c2)=O)CCCC(N(C(=O)C(N)=O)CC2CC2)C1 CC(C(=O)NC1(CNC(C2C(C)(C)C2(F)F)=O)CC1)S(=O)(=O)c1ccc(F)cc1 CC1(C)C(CNC(=O)CCSc2ccccc2)CCN1C(C1CCS1(=O)=O)=O N1(C(C2CCC(=C)CC2)=O)CCC2C(CCCN2C(C2CCC(O)CN2C)=O)C1 Cc1ccc(CC(=O)NCC2CCC(C)N2c2ncncc2F)cn1 CC1(C)CCCCC1CN1CCC(=CC(=O)NC(c2ccccc2)C#N)CC1 c1(C(=O)NC2C(OC)CN(C(C(CC)F)=O)C2)cc2n(n1)CCNC2=O O=C1NC2CCC1CC2C(=O)NC1CCN(C(=O)C2=COCC2)C1 C1(CC(=O)NCC2CCN(C(=O)C=CC(C)CC)C2)(CC)CCOCC1 C1(C)(C(=O)NCC(CCOC)NC(=O)C(CO)OC)CC2C=CC1C2 C1(C(N2C(C)(C)C(CNC(=O)C(O)C3CCCC3)CC2)=O)Cc2nccnc2C1 C1(C)(C(=O)NC2CC(CCNC(c3c(C)cn(C)n3)=O)C2)CCOC12CC2(F)F Cc1onc(C(N2CC(NC(=O)Cc3ncccc3C)C3CC23)=O)c1Br N1(C(C(C)(C2CC2)NC(CC(=O)OC)=O)=O)CC2CC(OC)C(C2)C1 C(=O)CC(C(F)(F)F)NC(C)(C)C.C(=O)(C(CC)CCC)C(=O)COCP(C)(C)=O C(=O)(CC(O)C(Cl)(Cl)Cl)N1CC(OC2CCN(C(C(C=C)O)=O)CC2)C1 c1(C(N2C3CN(Cc4ccc(C(C)(C)C)s4)C(C3)C2)=O)cc2cc(Br)ccc2[nH]1 N1(C(COCCCC)=O)CCC(NC(=O)CC2CC2C2CC2)C1C1CC1 C1(C(=O)NC(CCN(C(=O)C(C)(C)NC(C)(C)C)C)C(C)C)(OC)CCCCC1 C=CC(C)(C)CCNC(=O)C(C1CCCCC1)NC(=O)C(C)NC=O CCCC(C)(C)C(=O)N1CCN(C(c2cc(C)ccc2Br)=O)C(CO)C1 C1(CC(=O)NCC#CCC)CC(NC(c2nc(C)oc2C)=O)C1(C)C C1(NC(C(C)NS(CC)(=O)=O)=O)C2CCCN(C(c3ccsc3)=O)C2C1(C)C N1(C(c2[nH]c(=NCCC)sc2)=O)CC2CC(CNC(=O)COC(F)(F)F)CC2C1 N1(C(c2ccn(C(C)C)n2)C(=O)NCC2CCCO2)CC(C)CC1C c1(CNC(N(C(C)CC(N)=O)C)=O)ccccc1OC1CCC1 C(C(C)(CC)C(=O)Nc1cncc(Cl)c1)NC(C(F)=C(C)C)=O N1(C(=O)CN2CCCC2)CCOC2(C1)CN(Cc1cc(O)ccc1[N+](=O)[O-])C2 C1(CC)CCCCC1C(=O)Nc1ncc(CCNC(=O)CSc2ccccc2)s1 c1(C(=O)NC(C(=O)NCC(CC)SC)C2CCCO2)ncncc1OC N1(C(C(COCC)C)=O)CCC(NC(=O)CCC2CCC2)CC(O)C1 c1(CC)ccc(C(C)C(=O)N(C)CCNC(=O)Cn2ccnn2)cc1 CC(C)C(C(=O)N1CCC(N(C(=O)Cc2cnsc2)CC2CC2)C1)n1ccnc1 c1(C(N2C(CN(C(c3cc(C)no3)=O)C)CCC2)=O)c[nH]c2cccnc12 c1(-n2cc(C3(C)CN(C(C(CC=C)C)=O)C3)nn2)cc(Cl)cc(Cl)c1 c1(CNC(C2CN(Cc3c(Br)cccc3Br)CCO2)=O)ccc2ccccc2n1 C1(C(=O)NCC2CCCC(CNC(C3(C(N)=O)CC3)=O)C2)CC2(C1)CC21CC1 c1(OCC(=O)NCC2CCCN(C(c3c(C)coc3C)=O)C2)ccc(F)c(F)c1 C1(C(N2CCCC(N(C(=O)CCNC(N)=O)CC)C2)=O)CCn2cc(C)nc2C1 C(C(C(=O)NC(C)CC(C)C)NC(=O)C(c1cnn(C)c1)=O)OC C1(COC)(CNC(=O)COC2CCCCC2C)CCN(C(=O)CC(C)C2CC2)CC1 c1(C(N2CCN(C(CC3CC(C(=O)OC)C3)=O)C3C2C3)=O)cccc2nccn12 c1(-c2ccc(OC)cc2OC)nc2c(s1)CN(C(=O)COc1ccccc1)CC2.OC c1(OC)c(C(=O)NC(CNC(=O)CCCN(C)C)C(C)C(C)C)cccc1C C(=O)(C1CCOc2ccc(Cl)cc21)NC1CC(NC(c2n(C)ncc2C#N)=O)C1 Cc1cc(CC(=O)NCCOC2CCN(C(c3cc(C4(C)CC4)n[nH]3)=O)C2)sn1 N1(C(C2C(C(=O)OC)CC2)=O)CCC(CN(C(=O)Cc2ccn(C)n2)C)C1 C=CC(F)(F)C(=O)N1CCOC(CCNC(c2cn(CC)nc2C)=O)C1 N1(C(C2N(CC)CC2)=O)CCCN(C(=O)COCC(=O)Nc2cnccn2)C(C)C1 Cc1conc1CC(=O)NC1CC(CNC(=O)C(C)N(C2CCCC2)C)C1 C12CC3CN(CC3C1)C2=O.c1(CC2CC(C(C=[SH]C)=O)C2)n[nH]c2ccccc12 CC1(C)C(CNC(=O)CCC2CC(NC(=O)CN3CCC(F)CC3)C2)C1(F)F C1(O)(CNC(CN(C(CCSCCCC)=O)CC)=O)CCC(C)C1 C1(NC(C2(COC)CN(C(C(CC#C)O)=O)C2)=O)CC(F)(F)C1(C)C C1(NC(c2c(C)[nH]nc2Cl)=O)CCCCCC1NC(c1cc(O)cc(Br)c1)=O C1(NC(C2CCN(C)C2)=O)COCCN(CCCC2CCC2)C1 C1(C=O)C2CCC1CN(C(=O)C(c1ccccc1)O)C2.C=CC(CO)C1CCOC1 C1(CCC)CC(C(N2CCC(CNC(=O)CN(C3CC3)CC)CC2)=O)CCO1 Cn1[nH]c(=NC(=O)C23CC(CO2)N(C(C2CN(C4CC4)C2)=O)C3)cc1C(N)=O Cc1cc(CCCC(=O)NC(C)CCCSCCCC(=O)OC(C)(C)C)cs1 N1(C(=O)CC(F)(F)F)CCC2C(C1)CN2C(c1cnn(CC(F)(F)F)n1)=O C(=O)(C1CCc2ccc(OC)cc21)NCC1N(C(C=CC=CC)=O)CCC1 c1(C(=O)CN(C2(C(=O)OC)CSC2)C)cc(C(F)(F)F)ccc1C C1(N(C(c2n(CC)nc(C)c2)=O)C)CN(C(=O)CCOC2CC2)CC12CC2 O=C(C1Cc2ccc(Cl)cc21)NCC12CC1CN(C(=O)CCC(F)F)C2 c1(OC)cccc2ccc(C(=O)N(CC(C)NC(C3(F)CC=CCC3)=O)C)nc12 C1(C(=O)NCC2CCN(CC)C2)CCCCN1C(C1CCCN1C)=O N1(C(C(C)Cn2ccnc2)=O)CC2CCCC(NC(=O)C(C)C3CCOC3)C2C1 C#CCC(C(=O)N1CCCCC1CCC)NC(c1oc(C)nc1CC)=O C1(CC(C)O)CCCN1C(=O)CCCC1CC1OC(C)(C)C C1(CC)CN(C(=O)C(C2CN(C(=O)C(=O)C(C)(C)C)C2)OC)C(C)CO1 c1(CCCC)nc(C)c(C(N2CCC(NC(=O)CSC3CC3)C2)=O)c(O)n1 c1(OCC(C)C)cccc(C(=O)N(C(C)CNC(=O)C=C(Cl)Cl)C)c1 C(C(C)C)(C(O)C(=O)NCC1(NC(C2CCC(=O)O2)=O)CCOC1)OC C12(NC(c3cccc(C)n3)=O)CCC(CC1)N(C(c1cc(Cl)cc(Cl)c1N)=O)C2 C1(Nc2ncc(C(=O)OCC)s2)CN(C(=O)Cc2ccc(O)nc2)CC2(CC2)C1 C1(COC(CCn2c(C)ccc2C)=O)CC2(CCCC2)CO1 CCC(C)CCCCC(=O)N1CCC(C)N(C(=O)CC(C)(C)OC)CC1 N1(c2cccc(OC)c2)CCCN(C(=NCc2cnn(C)n2)NCC(C)C)CC1 C#CCC(C)(C(=O)N=c1cc(C)n(CCO)[nH]1)NC(=O)CCN(C)CCO c1(CC)ccoc1C(=O)NCCCC1CCN(C(C2(OC(C)C)CCOC2)=O)C1 C(=O)(CCCC(C)(C)C)NCC1C(C)CCCN1C(c1ccc(O)c(N)n1)=O N1(C(c2cncc(N)n2)=O)CCN(C(=O)CC2CCS(=O)(=O)C2)C2CCC12 C1(NC(C2CN(CC)C(=O)C2)=O)CC2CN(c3nc(C(C)(C)C)ns3)CC2C1 CC1C(NC(c2cccc(F)n2)=O)CCN1C(=O)CCCc1ccccc1Cl CCC(C)(CC)C(=O)NCC1(C(=O)Nc2ccc(C)cc2COC)CC1 CC1CC(CNC(c2cnc(N)c(Cl)c2)=O)CCN1C(=O)Cc1cncc(F)c1 C1(COC)(NC(=O)C(O)Cc2ccccc2)CCCN(C(=O)C#CC(C)(C)C)C1 C1(NC(CCSCC(N)=O)=O)CCOCC1NC(=O)C(O)C(F)F Cc1cc(NC(C2CCN(C(=O)C(C)CC(F)F)CC2O)=O)cc(F)c1 c1(C(=O)NC2(CC(=O)NCCn3c(CC)nnc3)CCC2)ccc(C#N)[nH]1 C(=O)(N1CC2COCC2O1)C1C(CNC(=O)CN2CC(=O)NC2=O)CC1 c1(-n2cc(C(N(C(C)(C)COC(F)(F)F)C)=O)nn2)c(C(=O)O)cccc1C c1(C(=O)NCCCCNC(c2cn(CCC=C)nn2)=O)[nH]c2c(c1C)CCCC2 N1(C(C(CC)SC)=O)CC2CCC(N(C)C(c3ccc(C)nc3C3CC3)=O)C2C1 C1(C(C(=O)NC(C2(C(N(CC(C)C)CC3CC3)=O)CC2)C)C)CCOCC1 N#Cc1ccc(C2(C(=O)NC3CC3NC(C3(C4CCC4)CC3)=O)CCC2)cc1 C(C)(CNC(=O)CCc1cnc[nH]1)(C(C)C)NC(c1c(CC)c[nH]n1)=O N1(C(c2c(CC)n(C)nc2)=O)CCC(O)(CNC(c2ccc(Cl)cc2Cl)=O)CC1 C1(COC)(NC(c2cc(C(F)(F)F)c[nH]2)=O)CN(C(c2coc(C(C)C)n2)=O)C1 N(C1COc2ccccc21)C(CC(C(F)(F)F)NC(CCCC(C)C)=O)=O c1(C2CN(C(C(C)NCC(=O)OC)=O)C2)cccc(F)c1.n1(CC=C)nnnc1C c1(C(C)Nc2nnc(C(C)(C)C)o2)cccc(Cl)c1 O=C1CCCC(C(=O)NC2CCN(C(=O)CCc3ccc(Cl)s3)C2)O1 CCC(C)(C)C(O)C(=O)NCC1CC(F)(CNC(=O)CCN2CCC(F)C2)C1 c1(NC(c2cc(C(CC)=O)on2)=O)c(C)ccnc1C c1(C(=O)NCC(C)(C(C)C)NC(c2c(C)scn2)=O)ccc([N+](=O)[O-])[nH]1 c1(C(N(CCCN(CC(=O)OC)C)CC#C)=O)nc(N(C)C)nc(=N)[nH]1 c1(N2CCC(CCC)C2)ccc(S(=O)(=O)N(C)CCn2nccn2)cn1 C(=O)(C(CC)C(=O)N1CC(C=O)(OC)C1)OCC.N1CC(CC(C)SC)C1 c1(C(=O)NC(C(C)C)C(C)NC(=O)Cc2ccon2)cncc2cc(Cl)ccc12 c1(CNC(C(C)NC(CN(CC)CC)=O)=O)cccc2ccncc12 C(=O)(C(Cn1cccn1)NC(C1CC(CO)CO1)=O)NCC(C)C#N CCCCCC(=O)NCC(=O)NCC=CCNC(=O)CC1CCCC1(F)F N1(C(C(C)OCC)=O)CCC(C(N2CC(C#N)C2)=O)C1CC N1(C(CSS(C)(=O)=O)=O)CCC2CN(C(C34C5C6CC3C3C4C5C63)=O)C2C1 N1(C(c2c(C)nc[nH]2)=O)CCN(C(=O)CSCC(N)=O)C(NC(=O)C(C)C)C1 N1(C(C2C(CC)CCC2)=O)CC2(C1)CN(C(=O)CCc1cccc(F)c1)C2 CC(C)CC(O)C(=O)NC(c1cnn(C)c1)C(N1CC2(CC(OC)C2)C1)=O C1(CC)CCN(C(=O)CCOC(C)C)C1C(N1CC(CF)C1)=O c1(C(=O)NCCCN(C(c2c(C)nc(C3CC3)o2)=O)C)coc2ccc(Cl)cc12 N1(C(COCCOC)=O)CC(NC(=O)CC2C=CCC2)C(c2cncn2C)C1 C1(NC(CS(N)(=O)=O)=O)COCCN(C(c2cccs2)=O)C1 c1(C(=O)NCC2C=CC(NC(c3c(C)nco3)=O)C2)ccc(F)c2[nH]ccc12 C1(CNC(c2[nH]nnc2C2CC2)=O)CC2C=CC1C2.C12(CCCC1)C(=O)N2 c1(NCc2ncc(C)nn2)cc(Cl)nnc1O CCN=C(NCc1ccc(F)cc1)NCc1ccoc1 CCC(CC(=O)OC(=O)CCc1cccnc1)NC(=O)C(O)CCNC(N)=O N1(CC)CC(C(=O)NCC2C(C)CCN2C(=O)Cc2n[nH]c(C)n2)CC1=O c1(SCc2ccc(N(C(=O)NCC)CC)cc2)cc(Br)c(F)cc1O C1(NC(C(C)N)=O)(CO)CCN(C(=O)C(CC(F)F)C2CCC2)CC1.n1(C)cnnn1 Cc1ccc(Br)c(NC(C2COCCN2C(=O)OC(C)(C)C)=O)c1F c1(NC(C(CC)NC(=O)CC2CSC2)=O)ccc(F)cc1F c1(C(N2CCNC(=O)C23CCC3)C(=O)NC(CC)C)ccc([N+](=O)[O-])c(Cl)c1 c1(C(=O)NC2(CF)CCN(C(C3C(=C)C3)=O)C2)cc(OC)c(O)c(N)c1 C1(C(N2CCC(NC(CCC#CC)=O)(COC)C2)=O)COc2ccc(O)cc2O1 N1(C(C2CCC(C)CC2)C(=O)NCCC2(C)CC2)CCC2OC(=O)OC2C1 c1(SCC(N2CC(C)C(NC(=O)COC3CC3)C2)=O)nc2ccccc2s1 c1(CC(=O)NCCN(C2CCCC2)C(C2C(CN(C)C)C2)=O)ccc(O)c(Cl)c1 C1(NC(c2cc(C)ncn2)=O)CC2CN(C(c3csc(C(F)F)c3)=O)CC12 C(C(=O)NCC(F)CNC(C1CC1C)=O)(C(C)C)(C(C)C)NC(=O)OC C1(O)(CNC(CCC(N)=O)=O)CCN(C(c2ccsc2)=O)CC1 C1(CC(=O)NC(CCNC(CC(=C=C)C)=O)C)Oc2ccccc2NC1=O Cc1ncc(C(N2CCOC(C3CN(C(=O)Cc4cnc(C)s4)C3)C2)=O)c(=N)[nH]1 [N-]=[N+]=NCCCCC(=O)NC1(C(=O)NC(CCO)C(F)F)CCCC1 c1(CC(C(=O)NC2CCN(C(COCC=C)=O)C2CC)C)c(C)nn(C)c1C C1(NC(C2(OC)CCOC2)=O)CCCN(C(=O)Cc2cccc(Br)c2)C1 c1(OCC(=O)NCCC2CN(C(C3C(C)(COC)C3)=O)C2)c(C)occc1=O C(=O)(C1=CCC(NC(C2(F)CCCC2)=O)C1)NCC(c1ccncc1)C C(CCC(=O)N(C(C)CNC(c1cnc(C2CC2)s1)=O)C)NC(=O)OCC C1(O)(CCNC(C2(C)CNC(=O)C2)=O)CCN(C(C2CCCCC2)=O)CC1 c1(Cn2cc(C3CCN(C(C(CN(C)C)O)=O)C3)nn2)ccc(N)cc1 C1(C(N(CC)CC2CCOC2)=O)CC(NC(=O)CCc2ncccn2)C(O)C1 N1(C(CCC(C)OCC)=O)CC(C2CN(C(=O)C(C)CN(C)C)C2)C1 Oc1cncc(N=c2scc(C)n2C2CCCCCC2CO)n1 c1(NC)cnc(C(N2CCC(CC(=O)N(CC#CCCO)CC3CC3)C2)=O)cn1 N1(CC)C2CCCC1CC(NC(C1N(C(=O)CN3CC=CC3)CCC1)=O)C2 C(=O)(CC(C)CC(=O)OC)NCCOCCOCCNC(c1cn(CCC)nn1)=O c1(C(=O)NC(C)C(C)NC(c2n[nH]cc2[N+](=O)[O-])=O)cccc2ncn(C)c12 c1(CNC(=O)CCSc2nc[nH]n2)c[nH]nc1Cl CCC(C)(C)C(O)C(=O)N1CC2(C1)CN(C(c1nnn(C)c1C)=O)C2 C1(C)(C)CC(F)C(=O)N1.C(C(O)C(C)C)NC(C=CC(C)(C)SC)=O C#CC1(O)CCN(C(=O)C(C)NC(=O)CCCCCOC)C1 C(=O)(C1=CCN(C(=O)CC2CC3CC3C2)CC1)NCC1(O)CCC(C)C1 N1(C(=O)C(O)c2ccsc2)CCC2CN(C(c3cnc4c[nH]nc4c3)=O)C2C1 C(=O)(CC1=CCOCC1)NCCCC(C(=O)N(CC)CC1CC1)O c1(C(=O)NC(C2CN(C(=O)C(CO)C(F)(F)F)CCO2)C)c(F)ccc(N)c1F C1(C(=O)NCCN(CCC)CC)CC(C)N1C(C1(C)CC1(C)C)=O C1(CNC(c2cccc(=O)o2)=O)C(C2CC2)CCN1c1cc(C(F)F)ncn1 c1(C(N2CC(CNC(C(C(=C)Cl)(C)C)=O)C(O)C2)=O)ccc2c(c1)CC(=O)NC2 C1(NC(=O)N(C(c2cccc(C)c2)C(C)C)Cc2ccnc(Cl)c2)CC1C1CCCC1 N1(C(C(F)OC)=O)CCCC2(CCCCC2NC(=O)Cc2nc(C3CC3)n[nH]2)C1 C1(CCC(=O)NCCC2CC(NC(CN(C)C3CC3)=O)C2)CCC(=O)N1 c1(CC)cc(=NCc2cccc(C(C)C)n2)nc(CNC(=O)C(CC)C(C)C)[nH]1 Cc1cc(OC(C)(C)C)cc(C)c1.c12ccc(s1)c(=O)n2C CCCCC(O)CC(=O)N1CCC(C)(C(=O)NCCN(C(C)C)CC)CC1 N1(C(CCC)=O)CCC2C(C1)NC(=O)CN2C(C1CCCN1C1CCCC1)=O c1(C(N(C)CC2N(C(c3c(C(CSC)=O)cco3)=O)CCC2)=O)cnncc1C c1(C(CNC(N(CCCC)CC)=O)O)nn[nH]n1 c1(C(C(=O)NCC(C)C)N(CC(CCC)C)C)ccc(F)c(C)c1 N1(CC(=O)NCC(CC)NC(CSCC#C)=O)CCCOC1=O c1(C(C(=O)NCC2CC2)N(CCOC)CCC2CCCC2)cnc(SC)c(Cl)c1 C1(C(=O)NC(C)CCCCNC(=O)C(=O)C(C)(C)C)CCS(=O)(=O)C(C)C1 C(=O)(CC(O)CC(C)(C)C)N(CCC(N1CC2N(CC)CC(C2)C1)=O)CCCO C1(CNC(C2CC(=C)C2)=O)CN(C(c2ccc(=O)n(C)c2)=O)CCC1C c1(OC)ccc(CCNC(=O)CN(C2CCC(C)CC2)C)c([SH]=CC(F)(F)F)c1 CC1CC(NC(c2cc(C#N)on2)=O)CCN1C(c1ccc(Br)o1)=O CC1(CO)CCC(N=c2[nH]c(=NCc3cnc4n3CCC4)[nH]c3c2SCC3)CC1 c1(C(N2C(CNC(C(C(CC)O)C)=O)C(C)CC2)=O)ccc(C#N)nc1O C(=O)(C(CC=C)NC(c1coc(C(C)C)n1)=O)NC(C1CCCCC1)C#C c1(C(N)=O)cc(N(C(=O)C)C2CC2)cc(O)c1.c1ccc(-c2ccccc2)cc1 C1(NC(CC2CC(=O)C2)=O)CCN(C(c2csc(Cl)n2)=O)CC12CCC2 C(CNC(=O)Cc1csnn1)(CC(F)(F)F)NC(C(N1CC(C)C1)C)=O C1(CC(=O)NCC2(C(=O)NC(CC)C3CC3)CCCC2)CCN(C)CC1 N1(CC)CCN(CC(=O)NCCCCCNC(c2ccc(C(F)(F)F)[nH]2)=O)CC1 C(CNC(C1CCCSC1)=O)(CC(F)(F)F)NC(C(C)Oc1ccccn1)=O C12(NC(C(C)OCCOC)=O)CC(NC(c3coc(C)c3)=O)(C1)C2 c1(C2CC(C(=O)NCC(C3CCC3)NC(C=CC(C)(C)SC)=O)C2)ccccc1 N1(C(CCC(C)(F)F)=O)CCC2CN(C(=O)CN3CC4CCC3C4)CC12 C1(NC(C2(COC)CC(F)(F)C2)=O)CN(C(c2cn(C)cc2C)=O)C2(CCC2)C1 N1(C(C(C(CC)C)N(C)C)=O)CCC2(C=C(C(=O)NCCCC(=O)NO)C2)C1 Cc1cc(CC(N2CCC(C(C)NC(C3CC(O)C3)=O)C2)=O)ccc1Cl C(=O)(C#CC1CCCCC1)NCC(CCOC)NC(c1cn(CC)nc1C1CC1)=O CC1CCOC(C(=O)NCc2csc(CNC(C3CCC(C)(C)O3)=O)c2)C1 c1(C(=O)NCC23OCCC(NC(c4c(CC)[nH]cc4)=O)(C2)C3)ccc(Cl)c(N)c1Cl CCCC(O)C(CO)NC(=O)CC1CC1CNC(=O)CCn1cnnn1 c1(CC)ccc(C(=O)N(CCNC(=O)CCc2nc(=N)[nH][nH]2)CC)cc1CC c1(C(N(CCNC(=O)CC2CCCCO2)CC)=O)cc(C)nc(O)n1 C(=O)(C1=CCCCC1C)NCC12C(CN(C(C3(CCC=C)CC3)=O)C1)C2 C(CCCC(=O)NC(CNC(C1CCCCC1O)=O)CO)OCC CCN=c1ccc(C(N2CC(NC(c3cc(C)c[nH]3)=O)CC3(CC3)C2)=O)c[nH]1 C(c1ccc(S(N)(=O)=O)cc1)=CC(N1C2C(CNC(=O)C=CCF)C(C2)C1)=O CN1CCC2CC(C(=O)NCc3nccn3C3CCCCC3)CCC12 Cc1cc(C(=O)CCC(=O)NCC2CC2CNC(c2ccnc(O)c2)=O)c(C)s1 c1(C(=O)NCC(C)(C)NC(C2C(Cl)(C(=O)OC)C2)=O)cc2n(n1)CCCO2 C(=O)(C1CCc2nccn21)N1CC2(CC(CCNC(C(C)CC3CCC3)=O)C2)C1 C1(C2CCN(C(=O)CC3CCC(=O)NC3=O)C2)(NC(c2c(C)coc2)=O)CC1 C12(C(N3CCC(NC(CSCC(C)=O)=O)C(F)C3)=O)CCOC1CCOC2 C1(C(=O)NCCc2cn(CC)nc2)CCN(C(=O)CC2CCCN2C2COC2)O1 N1(C(c2c(C)cn(C)c2)=O)CC2CC(C(=O)Nc3ccc(F)nc3)C(C2)C1 C(=O)(C1CCCc2c1ncn2C)NCCCC1N(C(CCOCC)=O)CCCC1 N1(C(c2cc(CNC(C3C(C(C)C)OCC3)=O)no2)=O)CC(CO)CC(C)(C)C1 c1(OC)c(C(N2CCC2CNC(c2ccnc3[nH]ncc23)=O)=O)cc(Cl)cc1Cl N1(CC(N2CCC(N(CC(c3ccc(C)cc3)=O)C)C2)=O)CCCCS1(=O)=O CS(=O)CCC(=O)NCC1CCC1NC(c1scnc1C(F)F)=O c1(C(N(CC#C)C2CC2)=O)ccn(CCNC(=O)Cc2ccc[nH]2)c1 CCCCC(O)C(=O)N1CCC(CC(=O)NCC(C)(CC)CC)C1(C)C C1(NC(CC2CC(OCC)C2)=O)C=CCCC1C(=O)N(C)CC1OCCC1(C)C C1(N(C(C(C2CN(C(C(C=C)C)=O)C2)OC)=O)C)CCOC(C)C1 c1(C(C(=O)NCCC2(NC(C3CC4CC4C3)=O)CC2)CO)ccc(Cl)cc1 CC(C)S(=O)(=O)CC(=O)N1CCCC1CCNC(c1cc(C(C)(C)C)no1)=O c1(CC(=O)NCCNC(C2(CC3(O)CCC(C(C)C)C3)CC2)=O)ccc(Cl)cc1 N1(C(c2ncn(C)c2)=O)CCC2(CCCN2C(c2c(F)ccc(F)c2Cl)=O)C1 Cn1cc(S(C)(=O)=O)c(C(=O)NCC(C2CC2)NC(=O)Cc2ccccc2Cl)n1 C1(C(=O)NCC2(CNC(C3(CCC)CCC3)=O)CC2)CC2C(C1)C2(C)C C(=O)(C#CC1CCC2(CC1)OCCO2)N1CC(C)(NC(C(C)CF)=O)C1 c1(N2CC(NC(C3(CC(C)C)CCC3)=O)CC(F)(F)C2)ncnc2c(Br)c[nH]c12 C(=O)(C1=C(C#N)CCC1)NC1C(C(N(c2c(C)ccc(C)c2)C)=O)CCC=C1 c1(NCC2CC3CCC3C2)ccc(S(=O)(=O)NC2(C(=O)OC)CCCC2)c(Br)c1 c1(CNC(C(=O)OCC)Cc2ncccn2)n[nH]c2c1CCOC2 Cc1ccccc1C=CC(N1CCC(NC(C2(C)CC=CCO2)=O)C1)=O C12(CNC(C3(Br)CC3)=O)CCC1CN(C(=O)C(O)Cc1cnc[nH]1)C2 c1(CC(=O)NCC(C2CCC2)NC(C2CCCC2)=O)cnco1 c1(N(C(C(=O)NCC)C(C)C2CCCCC2)CCC)ccc(F)c(F)c1 C1(C(=O)NCC2(OC)CCN(C(=O)CCc3cnco3)C2)CCCC(C)(C)CC1 c1(CC(=O)NC(CCCNC(c2ccc(C)cc2F)=O)C)cnc2n1CCOC2 c1(C(=O)NC2CCC(C)N(c3ncc(Cl)c(O)n3)C2)cc2cc(F)ccc2s1 CC1(CNC(C2CC(O)C2)=O)CCCN(C(=O)CC2CC3(CCO2)CC3)C1 C1(C(=O)NC(C(C)C)CCN(C)C(c2cnco2)=O)C2Cc3ccccc3C12 C1(CCC)CCN(C(C2(C)CC(Oc3csc(CC)n3)C2)=O)CC1 c1(NC(C2CSC2)C)ccc(S(=O)(=O)N2CCC(OC(F)(F)F)CC2)c(Cl)c1 c1(CC(=O)NCCN2CCC(CC3CCCC4CC34)C2)c(F)cccc1Cl c1(SC)nccc(N2CC3C(CNCc4cnon4)C3C2)n1 N1(C(c2[nH]cc(C(=O)OC)c2)=O)CCOCC12CCN(C(c1nccs1)=O)C2 N1(C(c2ccc(C(C)C)cc2)=O)CCCC(C)(C(N2CCCC2C#N)=O)C1 CC1CC(CO)CCN1C(C1COCCC1NC(C1C2(CC2)C12CC2)=O)=O N1(C(CC=CC=C)=O)CCC2(CCOCC2)C(CNC(=O)Cn2[nH]cnc2=N)C1 C1(C(=O)NCC2CC(NC(C3CCS3(=O)=O)=O)C2)(OC)CCC12CCC2 C(CC1=CCCCCC1)NC(CC1OCCCN(C(C2=C(C)OCC2)=O)C1)=O C1(CC(=O)N(CCNC(c2cc(C)co2)=O)CC)COC(C)(C)C1 c1(CCC(=O)NC2CC(F)(CNC(C(C3CCC(=O)N3)C)=O)C2)ccc(Cl)nc1 C1(C(=O)OC)CCCC1C(=O)N(CCCCNC(c1cnc(CC(C)C)[nH]1)=O)C c1(CC)c(C(=O)NCC2CC(COC)CN2C(=O)CC)nnn1CC.C(C)=O c1(NC(C2CC3(C2)CN(Cc2cnccc2C(F)(F)F)C3)=O)nccc(Cl)c1I N1(C(c2c(C)[nH]c(C#N)c2)=O)CC(C(=O)NC(C)C(C)C)CC12CCC2 C(N=c1[nH]nc(Cl)s1)SCCNC(=O)CSc1ccc(Cl)cc1 c1(C(=O)NCC(N(C)C)C2CC2)cncc(N2CCCC2)n1.C1(N(C)C)CCCN1C C1(NC(c2ccc(C)nc2C)=O)CCN(C(=O)Cc2cccnc2O)CC(O)C1 Cc1cc(Br)ccc1S(=O)(=O)NC12CC(C(=O)N=c3cc(Cl)cn[nH]3)(C1)C2 N(C(=NCc1ccc(C(F)(F)F)cn1)N1CCC(CN(C(N)=O)C(C)C)C1)C(C)C c12ccc3nc(ccc3c1)NC2.C(=O)(C(COC(F)(F)F)N(C)C)OC C1(C(=O)NC2(CC(=O)NCC(C(CC)C)OC)CCCCC2)CCC(=O)N(C)C1 c1(C(N2C(CCCNC(C3CC34CC4)=O)CCC2)=O)cc([N+](=O)[O-])cc(Cl)c1Cl Cn1c(S(=O)(=O)N2CCOC(c3ccc(C(F)(F)F)cc3)C2)cnc1Cl CN1CCN(c2nc(C3CCCC3)ns2)C(CNC(c2cc(F)cnc2O)=O)C1 N1(C(C#CC2(C)CC2)=O)CC(NC(=O)CCC2CC2(C)C)C2(CCOCC2)C1 c1(CC)c(C(=O)NC2C3CN(C(C4CCCCN4C)=O)CC23)cnc2ncnn12 C1(NC(CNC(CC)=O)=O)CC2CCC(C1)N2C(=O)Cc1occc1C c1(CC)nc(C)[nH]c1C(=O)NC1CCCC(NC(c2cc(C#N)on2)=O)C1 N(C1CN(C(c2coc(C(F)F)c2)=O)Cc2ccccc21)C(c1cc(C)c(C)[nH]1)=O C1(C(=O)NCC2(C)ON=C(C)C2)CN(C(=O)C(C(C)C)N(C)C)CCC1(C)C c1(C(=O)NCC(C)(C)C(=O)N2CCOCC2)ccc2ncoc2c1 S(=O)(=O)(c1ccc(C(N2CC(N(C(=O)COC3CC3)C)C2)=O)cc1)NC CC1CC(=O)NCC1C(N1CCN(C(C2(C)CC2)=O)C(CS(C)(=O)=O)C1)=O c1(C(N2CC(C(N)=O)C2)=O)cc(Cl)cc(Cl)c1.C12COCCN1S(=O)(=O)C2 C1(C(C)C)CN(C(=O)Cc2ncccn2)CCN1C(=O)CCN1CCCS1(=O)=O C1(C)(C(=O)NCC2(CNC(CSC)=O)CCCCC2)Cc2ccccc2NC1=O C(=O)(C1=CCCCCC1)NCCCC1N(C(C(C)(Cl)Cl)=O)CCCC1 N1(C(=O)CCCC(F)(F)F)CCN(C(c2cnn3cc[nH]c(=O)c23)=O)C2CCC12 C12CCC(CC1)C(=O)NC2.c1(C(=O)NC23CC(CC)(C2)C3)cnccc1Br C12(C(=O)NC3(C(=O)OC)CC3)C(=O)C3CC1C2C3.c12ccnc(c1)CNC2=O C1(NC(c2cc(C(C)=O)on2)=O)CCCCN(Cc2ccc(C)cc2Cl)C1 N1(C(COCCOC)=O)CCC2(CC1)CC2(CO)NC(=O)CN1CC(C)(C)C1 N1(c2ncc(CCC)cn2)CCCC2(CCCN(C(C3CC=C(C)CC3)=O)C2)C1 c1(CNC(C2(C=C)CCC2)=O)cnn2c1CN(C(c1cc(C)on1)=O)CC2 C(=O)(CCCCC(=O)OC)N(CC(CC=C)C(=O)NC1CC(=O)N(C)C1)C c1(CC(=O)NC(C(C)C)CNC(c2cnc3n2CCC3)=O)nnc2n1CCOC2 Cc1coc(C)c1C=CC(N1CC(CNC(=O)C(F)n2ccnc2)C(O)C1)=O CC(C)CC(C(=O)NCC1CC2(CC2)C1)N(C)C(C1SCCS1)=O C(=O)(CC(C)C(C)(C)NC(=O)C(O)c1ccsc1)NC(CC=C)CC(F)F N1(CC(=O)NCC(c2ccncc2)C)CCCC(CNC(=O)C(C)(C)CO)C1 c1(C(=O)NC2(C)CCCN(C(C3C(C)C3)=O)C2)nc(S(C)(=O)=O)n2ccccc12 C1(C(N(C(CNC(=O)CC2CCC(O)C2)C2CC2)C)=O)CCC(=O)N1C1CC1 C=C(C)CC(C(=O)N1CCCN(C(C)COC)CC1)NC(=O)OC(C)(C)C.C(COC)N c1(CN2CC(O)C(F)C2)c(F)ccc2[nH]ccc12.c12cccc(c1)CNC2=O C(=O)(C(CC(F)F)c1ccccc1)NC1CC(CNC(CSc2cc(C)on2)=O)C1 N1(C(C2(C#N)CCCO2)=O)CC2CC(C1)CN(C(=O)CCc1cc(Cl)cs1)C2 N12CCC(C13CC3)C(=O)N1CC(CCC2C(=O)OCC)C1.c1(SC)ccccc1 Cc1ccc2c(C(=O)NCC(C)(O)CNC(C3CCC(O)C3)=O)n[nH]c2c1 c1(C(N2CCC(C)(NC(c3ccncc3)=O)C2)=O)cnc(Cl)c(Br)c1 c1(C(N(C(C)CNC(C2CCC3CC23)=O)CC)=O)cn(CCCF)nn1 N1(C(CC2(NC(CC3(C(=O)OC)CCC3)=O)CC2)=O)CC2(CCC(O)CC2)C1 c1(-n2ncc(C(=O)NCC3N(C(COC4(C)CCCC4)=O)CC3)c2)ncc(Cl)cn1 Cn1cnn(C(=O)NCC2CC2CNC(=O)CN2CSCC2=O)c1=O C=CC(C)(O)CC(=O)NCC1(CN(C)C(c2nccc(Cl)c2C)=O)CC1 C1(CNC(c2c(C(N)=O)csc2)=O)CCC(F)(CNC(C2CCC(O)C2)=O)C1 C1(NC(C2(OC)CCN(C(c3c(OC)nn(C)c3)=O)C2)=O)CC2CCC(C1)C2O CC(C)=C=CC(=O)NC(C(=O)NC(c1n[nH]c(CO)n1)C)C1CCOC1 C1(C(=O)NCC2(O)CN(C(C3(C)COCCO3)=O)C2)CC12CCOCC2 C12CC3(C1)CC(C3)C(=O)N2.C1(CNC)CC12CC(OCC)C2.C=C1CCC1 N1(C(CC(C)(C(F)F)N(C)C)=O)CCC2(CCCCN(C(=O)Cc3csnn3)C2)C1 c1(C(N2CC(F)C(F)C2)=O)cn2c(n1)CCC2 c1(N2CCC(CC(=O)Nc3cc([N+](=O)[O-])c[nH]3)C2)cc(Cl)nc(Cl)n1 N1(C(c2c(NC)cccc2)=O)CCC(C(=O)NCC2CCCN2C2CC2)=C(F)C1 C(=O)(C1=CS(=O)CCC1)NC1C(NC(C(C)CN2CCCCC2)=O)C1 c1(OC)ccc(C(=O)NC23CC(CNc4cc(Br)cc(Cl)c4Cl)(C2)C3)c(Cl)c1Cl CCS(=O)(=O)c1ccc(CNc2cc(C)ccc2NC(=O)C(F)(F)F)s1 C1(NC(C(c2ccc(C)cc2)F)=O)CC(O)CN(C(=O)CCCN2CCCC2)C1 c1(NC(C(CCCN(C)C)CNC(=O)OC(C)(C)C)=O)c2c(nn1C)CCC2 N1(C(=O)COc2cccc(Cl)c2Cl)CCC2CCN(C(C3(O)CCOC3)=O)C2C1 c1(CC)nc(C)sc1C(=O)N(C)CCOCCN(C(=O)Cc1ccccc1F)C c1(C(=O)NC(C)(CNC(C2CCNC2=O)=O)C2CC2)nc(C2CC2)n2ccccc12 c1(C(N2CC(NC(C3CCCC(CF)C3)=O)(CO)C2)=O)ccccc1F c1(C(=O)O)ccc(Br)c(O)n1.N12CC(CC(F)C1)C2=O.C123CC(C1)(C2)CNC3=O C1(NC(c2nc(CC)oc2)=O)(CO)CCCN(C(C2(C)CCC(=O)NC2)=O)C1 O1P(=O)(OCC)CCC2CCCCN12.CCCCC(C)C c1(C(=O)NCC(N(C)C(C2CC(=O)NC2=O)=O)C2CC2)cc(Cl)cc(Cl)c1F CC1(C)CCN(C(=O)C2=C(Cl)CCC2)CC1NC(=O)CC1CC1(Cl)Cl c1(C(=O)OCC)ccc(NNC(=O)C(C)OCC(C)C)cc1 N1(C(C2CCCN(CCC)C2)=O)CCCC(O)(CN(C)C(c2cccs2)=O)C1 C1(NC(c2cn(C)c(O)n2)=O)CC2(CCN(C(C3(CC#N)COC3)=O)C2)C1 n1(CCC)nc(C)c(C(=O)NCC2CC(NC(=O)C3=CCCCO3)C2)c1C CC1CN(CC2CN3CCC2CC3)CCC1NC(C(c1ccc(Cl)o1)C)=O C(=O)(C(C)(CO)NC(c1cccc(F)c1)=O)NCC(C(C)C)N1CCOCC1 c1(C(=O)Nc2cc(Br)ncc2O)nc(C(F)(F)F)n2c1CCCC2 c1(NC(C2CCCN(C(c3c(C)[nH]nc3C(F)(F)F)=O)C2)=O)ccc(O)c(Cl)n1 C(=O)(C(CO)C(C)(C)C)N1CC(NC(C(C2CCC2)OCC)=O)C(O)C1 N1(C(c2cnc(CC)s2)=O)CCOC(C)(CNC(=O)CC2(N(C)C)COC2)C1 CC(CCNCc1ccsc1)C(F)(F)CN=c1cc(N(C)C)nc(C(C)C)[nH]1 CC1(C)CCCCCC1NC(=O)CC1C2CCCC2N1C(=O)Cc1ccon1 c1(C(N(C(CCC)C)CCCC)=O)[nH]cc(C)c1C.C12C=CCN1C(=O)CO2 CC1=C(C(=O)N2CCOC(CCNC(c3cncc(Cl)c3Cl)=O)C2)CCCO1 c1(SC)cc(C(N2CC3CC(NC(=O)CSCC(F)F)C2C3)=O)ccc1N C1(CNC(c2onc(C)n2)=O)CCC(NC(=O)C(C)CF)CC1 C(N=C(NC1CC1)N1CCC(Oc2ccc(Br)cc2)C1)c1c(CCC)occ1 Cc1ccc(O)cc1C(N1CCC(C)C1C(=O)NCC1CCC(=O)N1)=O C1(CNC(COC2CCC(C)CC2)=O)CC2(CC2)CN1C(=O)C(F)n1cccn1 C1(C(N(C)Cc2n(CC)cnc2)=O)CCCN(C(=O)Cc2nccn2CC)C1C c1(C(N2CCC(C(=O)Nc3cc(Br)cnc3O)C2)=O)cc(F)c(F)c(F)c1F C1(C(C2CC2)NCCN(C(CCC#CC)=O)CC(C)O)CCC(O)(C(F)(F)F)CC1 N1(C(COCc2ncc(C)o2)=O)CCC(C)C(NC(=O)Cc2ccsc2)C1 Cc1cccn2ncc(C(=O)NC(C)CCN(C(=O)C=C3CC3)C)c12 C(=O)(CC(CC(N)=O)CC(C)C)NCC1N(C(C(CC#C)CC#C)=O)CC=C1 n1(CC(=O)NCC(CN(C)C(c2ncc(F)cn2)=O)O)ccc(=O)c([N+](=O)[O-])c1 N1(C(C2C(=C)C2)=O)CCC(CNC(c2cscc2C2CC2)=O)CC1C C(CC(C)N=c1[nH]c(N(CCCc2cccc(OC)c2)C)nc2ccsc12)SC C1(NC(C(C)n2cnnn2)=O)CCCC2CN(C(=O)C(O)CC(C)(C)C)CC12 c1(NC(=O)NC(c2ccc(F)c(Br)c2)(C)C)cncc(P(C)(C)=O)c1 C1(CNC(c2c(Cl)cn(CCC)n2)=O)CN(C(C2(C3CC3)CC2)=O)CC12CCC2 c1(CC)cc(C(=O)OCc2ccc(Cc3ccc(Cl)cc3)cc2)cc(CC)c1 C1(CC(=O)NCCN(C(C2Cn3c(C)ncc3CC2)=O)C)COCC2(CCC2)O1 c1(C(N2CC3CCN(Cc4cocn4)C3C2)=O)cc(I)ccc1[N+](=O)[O-] c1(CCNC(C2(COC)CN(C(=O)C(F)=CC(C)(C)C)C2)=O)cccnc1O N1(C(C(CC=C)CC)=O)CC2(CCC(CNC(=O)C(C)(C)C(C)C)O2)C1 N1(C(CCC=C=C)=O)CCC2CN(C(=O)C(C)(C)COC)CC2C1 C1(NC(C2CC(SC)C2)=O)CCN(C(C2(C(N3CCCC3)=O)CCC2)=O)C1 c1(C(N2CC(C)C(CCNC(C3CC3CF)=O)C2)=O)csc2c1CCC(C)(C)C2 N1(C(Cc2ccc(C(C)=O)s2)=O)CCN(C(=O)CCc2ccn(C)c2)C2CC12 C1(C(=O)O)COCC1NC(=O)NC(Cc1cccnc1)CO c1(C(N2CC(NC(c3nccc(OC)c3F)=O)C(O)C2)=O)cnc2scc(C)n12 Cc1cc(=O)n(CC(N2CC3C(CNC(c4ccon4)=O)C3C2)=O)cn1 C(c1ccc2c(c1)NC(=O)CO2)=CC(=O)NCC(CC)NC(CSCCCC)=O c1(CC(=O)NC(CC)(C)CNC(c2ccsc2OC)=O)ccc2c(c1)CCCO2 CCCC(C(=O)NCC(F)(F)C(F)F)NC(c1cn(CC)nn1)=O c1(C(N(C2CC(NC(C3N(CC)CCC3)=O)C2)C)=O)ccc(CO)c(Cl)c1 N1(C(C2C(CC)OCC2)=O)CC2CCC1CN2C(c1cc2ncccc2o1)=O C1(C(=O)NCCCOCC(F)F)(CC)CCCN(C(=O)CP(C)(C)=O)C1 C1(C(=O)NCCN(C(=O)Cc2ccon2)CCOCCO)CCCCC12CCC2 C(=O)(C(CN(C)C)C(C)C)NC(C(=O)NC(CCC)CCO)(C)COC c1(C(=O)NCCCOCCCNC(C=CC=CC)=O)ccc(C)cc1 C1(C(N(CCCCNC(Cn2c(C)cc(C(F)F)n2)=O)C)=O)CC(C)(C)CN1C N1(CCC(C)C)CCCCC1C(=O)NCc1ncc(CN(C)C)s1 Cc1cccc2ncnc(N3CC(NC(=O)C(c4cncn4C)O)CC3C)c12 C(CC(=O)N1CCCc2ccnn21)(c1ccccc1C)NC(COCCOC)=O c1(C(=O)NCCCN(C(=O)CN2CCCNC2=O)CC)cnn(CCO)c1N c1(C(=O)OC)cc(Br)cc(F)c1NC(c1cc(S(=O)(=O)N(C)CCO)c[nH]1)=O C(=O)(CC(F)(F)C(F)(F)F)N1CCC(N(C(c2ccnc(C)n2)=O)C)C2(C1)CC2 C1(NC(Cc2c(C)nn(C)c2C)=O)CCC2CCN(C(c3ccc(F)s3)=O)C1C2 c1(C(C(=O)NC(C(=O)OC)C)N(C2CCN(C)CC2)C)cc2n(c1)CCCC2 N1(C(C(C)Oc2ccccc2)=O)C2CC1CN(Cc1cccc(C(F)(F)F)c1)C2 CC1(C)CN(C(=O)CCNC(C2CCC2)=O)C1.c1(O)ccc(Cl)cc1 N1(C(C2C(C)CCO2)=O)CCC(C2CC2)C1C(=O)NCCc1ccncc1 CC1CN(C(C2(C)CC2(F)Cl)=O)CC(C)N(C(c2n[nH]c(C3CC3)n2)=O)C1 c1(CCN(C(CNC(=O)OC)=O)C)ccc(C)cc1.C1C(O)CSCC(=O)N1 CC1c2cc(Br)cc(Br)c2CCN1CC(=O)NCC1CCc2ccccc21 N1(C(C(CSC)O)=O)CC(C2CN(C(=O)C(C(C)C)NC(C)=O)C2)C1 N1(C(C(Cc2ncn(C)c2)O)=O)CCC(O)(CNC(=O)C(F)(F)CO)C1 CC1Cc2cc(O)ccc2C(C)N1C(=O)NCc1nnc(S)n1C C1(C)(OC)CC(Nc2cc(N3CCC=C(C)C3)nc(C(C)C)n2)CC1(C)C CC1CCN(C(=O)CC2COCCO2)CC1CNC(c1ccc(OCF)cc1)=O n1(CCC)ncc(C(=O)NC2CN(C(=O)COc3ccc(O)cc3)CC2C)c1C N1(CCCC)CCOCC1C(=O)NCC(C)NC(=O)CCc1ccc(C)s1 c1(C(=O)NCC(CC)NC(=O)C(C)(O)CC)cn(C)nc1C(=O)Nc1ccccc1 N1(C(C23N(C(c4ccc(OCC)cc4)=O)CCC2C3)=O)C2CCCC1COC2 C1(CCNC(C23CC(CO)(C2)C3)=O)(OC)CN(C(=O)COC2CCC2)C1 c1(C(N2CCC(C)(CNC(C3CC34CCCC4)=O)C2)=O)cnn2c1OCCC2 N1(C(C=CCC)=O)CCC(CCNC(=O)CC2(C)CC(F)(F)C2)C(F)(F)C1 C(=O)(C(O)CC(C)(C)C)N1CCCCC(C(=O)Nc2ccc(CN(C)C)cc2)C1 C#Cc1ccc(CCNC(N2CCN(c3cncnc3)C(=O)C2)=O)cc1 C1(c2ccccc2)(NC(=O)Nc2cc(C(CC)CC)no2)CCCOC1 CC1CCC(NC(c2cn(CCNC(C3CC3(C)C(C)C)=O)nn2)=O)CC1 N1(C(CC(CC)C)=O)CCOC(C)(CNC(c2c(Cl)sc(Cl)c2C)=O)C1 c1(C(=O)NCC(C)NC(C2CC3CCC2O3)=O)cc(Cl)c(Br)[nH]1 c1(NC2(C(c3nnnn3C3CC3)OC)CCOC2)c(C(F)(F)F)cc(Cl)cc1Br S(=O)(=O)(CC(=O)NC(CC1CCC1)C(=O)NCCC1CCCN1C)NC C1(C)(C(C)NC(c2ccc(F)cc2)c2cccn2C)CCC(O)CC1 N1(Cc2cn(CC3(SCC)CCCO3)nn2)CCC(C(N2CSC(C)C2)=O)CC1 C1(CNC(=O)Cn2cnnc2)CC2CCCC2N1C(=O)CSC1CCS(=O)(=O)C1 c1(OC)ccc(C(=O)NCC2CC(C)N(C(c3ccccc3C)=O)C2)c(OC)c1 N1(C(C(CC)(C)C)=O)CCN(C(c2cnc(OC(C)C)s2)=O)CC1C c1(C(C)C)ccc2c(c1)C(NC(N1CC3CC(O)CC3C1)=O)CCC2 c1(-c2c(C)nc(C)s2)c(C)ccc(C)c1N.N12CCN(C(C)C1)C2c1ccccc1 C(=O)(CC(C)(C)C(=O)NCC1CC1CNC(c1cncc(Cl)n1)=O)OC C12(C(N3CC(NC(C(c4ccccc4Cl)(C)C)=O)C3)=O)CC(C#N)(C1)C2 c12cncc(c1)NC2=O.C(C(=O)NCCC1(CNC(=O)N)CC1)SCC=C c1(C(=O)NCC(CNC(c2cccc(C3(F)COC3)c2)=O)O)cc(F)ccc1O c1(C(N2CCCN(CCNC(C(C(C)(C)O)F)=O)CC2)=O)cncc2[nH]ccc12 c1(NCc2ncc(OC)nc2)nccc(=NCc2cccnc2Br)[nH]1 C1(CC)CCCC(C(=O)NCC=CCNC(c2nc(C)oc2OC)=O)C1.C(=O)OC Cc1nn(C)c(C)c1C(C)C(=O)N(CCN(C)CCn1cncn1)C(C)C c1(C(N(C2CC(NC(C3(C(F)F)CC(F)(F)C3)=O)C2)C)=O)cnc2n1CCC2 C1(CCOC)(NC(=O)CC2CC2C)CCN(C(C2CN(C(C)C)CCO2)=O)C1 CS(=O)(=O)c1ccsc1C(=O)NCCCCC(CO)NC(c1cnc(S)[nH]1)=O C(=O)(CCN(OC)C(=O)C1CCN(C(C2CC(C)(C)C2)=O)C1C)OCC CC1CN(C(C2(O)CCC2)=O)CC2(CCN(C(C3CCCOC3C)=O)C2)O1 C12CC(F)CN1C(=O)C1N(CCC1)C2=O.C(C)(C(=O)OCCOC)OCC=C C(=O)(C(O)C(CCC)NC(=O)CC1CC(C)C1)N(C1(C#C)CC1)C C=CC1(CNC(C2CC2CC(C)(C)C)=O)CN(C(=O)CSCC(N)=O)C1 C1(CNC(C(C)(C)C)=O)CN(C(C2CCCCCC2)=O)CCC1CC(N)=O N(C1CCc2cccnc21)C(C1CCN(C(C2C=CC=CC=C2)=O)C1)=O N1(C(=O)OC(C)(C)C)CCCC2(CNC(C3(Nc4ccccc4Cl)CC3)=O)CC12 Cc1c(C(N2C(C(=O)NCC3CNC(=O)CO3)CCC2C)=O)cccc1C#N C1(NC(=O)CC2CCCCC2)CCCC12CCN(C(c1cc(Br)cs1)=O)C2 c1(C(=O)NC2CC(C)(CNC(c3cc(C(C)(C)C)n[nH]3)=O)C2)csc([N+](=O)[O-])c1 Cc1ccc(CCC(=O)NC2CCC(NC(C3SCCCS3)=O)C2)cn1 N1(C(CNC(CC(C)C)=O)=O)CC(NC(C2CC=CC2)=O)CCC1C C1(N(C(C(C(C)O)N(C)C)=O)C)CCCCN(C(c2ccc(O)cc2)=O)C1 Cc1cc(C#N)cc(C(N2CC(N(C)C(C3CCCCCC3)=O)C(F)C2)=O)n1 CC12CCCCC1(C(N1CCC(CCC(=O)NCCN3CCC(CO)C3)C1)=O)C2 N1(C(CCOC(C)=O)=O)CCC(CNC(=O)Cc2c(C)n[nH]c2C)CC1 c1(OC)cc(C=CC(N2CCN(C(=O)C(Cl)=CCl)C(C)C2)=O)ccc1F N1(C(C2CCCC(OC)C2)=O)CCN(C(=O)CCn2cnnn2)CC1CO c1(NC)ccc(C(N2CCCC2CCNC(=O)C(O)C2CCCC2)=O)c(C)c1 C1(CC(=O)NC(CC(=O)N(C)Cc2cn(CC)nc2)C2CC2)CCC2(CC1)CC2 N1(C(CC2CC(=C)C2)=O)CCOC(C(C)NC(=O)CSc2nncn2C)C1 C1(C(=O)NCC2C(NC(c3cn(C)nc3C(F)F)=O)C2)CCC2(CCC2)O1 c1(C(c2nnnn2C2COC2)NC(C)CCCCO)cc(Br)cc2c1OCC2 C1(C(=O)NC(C)CN2CCN(C)CC2)CC12CCN(C(c1cnns1)=O)CC2 N1(C(C=CC)=O)CCC(C2(NC(c3cccn3C3CC3)=O)CC2)C1 Cc1cc(C(=O)NC(C)CC2CCN(C(=O)CC(C)(C)F)C2)ccc1N(C)C=O C1(CNC(C2C(C)COCC2)=O)CC2(C1)CC(N)CCO2 c1(C(=O)NC2CC(CNC(C(c3n(C)ncc3)O)=O)C2)cccc(CO)c1 N1(C(C2CN(C(C)C)C2)=O)CCCN(Cc2nnnn2C2CC2)CC1 CC1CCC(NC(c2cn(C3CC3)cn2)=O)CN1C(=O)CCC(C)(C)C C1(NC(CCNC(C)=O)=O)CCSC12CN(C(C1C(C)C1C)=O)C2.c1nncn1C C1(NC(c2cncc(CC)c2)=O)CCCN(C(=O)Cc2ccnn2C)CC1 c1(C(=O)NCC(O)CCNC(C2(F)CCC2)=O)cnc2ccc(F)cn12 N1(C(CN(C(C(C)OC(C)(C)C)=O)C)=O)CC(CO)C(C)(C)C1 N1(C(c2cc(CC)c(C)cc2)=O)CCC2(C1)CN(C(=O)CC1(O)CC1)CC(C)O2 N1(C(C(c2cc(C)oc2C)C)=O)C2CCC1C(CNC(c1cc(F)n(C)n1)=O)C2 C1(NC(C2(C(C)NC(=O)C(O)c3ccsc3)CC2)=O)CC12CCOCC2 CC(C)(C)C(CNC(c1ncc(F)cn1)=O)NC(=O)C(F)C1CC1 c1(C(=O)OC)cnn2c1S(=O)(=O)CC2.CC(=NOCC#N)c1cn[nH]c1 N1(C(COCC=C)=O)CC2(CCN(C(=O)Cc3csc(Cl)n3)CC2)C1 C(=O)(CC(C)CN(C)C)NCC(CC)NC(=O)CCc1ccc(C(C)C)cc1 C1(CNC(c2ccc(OCC#C)cc2)=O)CN(C(C2CCCN2C)=O)CC12CC2 c1(CCOCC(=O)NCCCCN(C(=O)C(O)CC2CCC2)C)ccccc1 C1(OC)CN(C(=O)CCCNC(=O)C(C)(C)C2CC2)CC12CC2 S(=O)(=O)(c1c[nH]ccc1=NCc1cc(C)ccn1)N1CCC(CS(CC)(=O)=O)CC1 c1(C(N2C(C(N3C(C(=O)NC)CC3)=O)C(O)CC2)=O)cnc(O)c(F)c1 C1(OC)(CNC(c2ccc(F)cc2)=O)CCN(C(=O)C(c2cncn2C)(F)F)C1 Cc1csc2ncc(C(N3CC4CCN(C(=O)CC5CCCO5)C4C3)=O)c(=O)n12 C1(NC(Cc2n(C)ccc2)=O)CC2CCC1(C(=O)NCCCC(C)(C)O)C2 N1(C(c2ccc(C)c(Cl)c2Cl)=O)CC2COCC(C1)C2NC(=O)C=CC(C)(C)C C(=O)(CC(C)CC(C)(C)C)N1CC(O)(C(C)NC(CC=CC)=O)C1 C=CCCC(C(=O)OC)NC(=O)C(C)(C)C1CCCN1C(C1CCC(F)(F)C1)=O c1(CC(=O)NC(C(CO)NC(CC(CC)C)=O)C)cccc(C#N)c1 C1(C(=O)NC(CC)CNC(c2cc(Cl)c(Cl)s2)=O)CCc2nncn2C1 Cc1cnc(CN2CC(C(N3CCCCC3)=O)CC(F)C2)c(F)c1 c1(C(N2C(C)CC(NC(c3cc(CCC)[nH]n3)=O)C2)=O)coc2c(C)cccc12 CN1CCN(C(C2(F)CCN(c3ccc(C(C)N)cn3)C2)=O)CC1 c1(C(=O)OCC)c(C)sc(C(=O)NCC2CCCN2C)c1Cl N1(C(C2CCC3CC3CC2)=O)CC2CCCC(C1)N2C(C1CCS(=O)(=O)N1)=O c1(CC)cc(C(N2CC=CC2CNC(C2CC(OC3CC3)C2)=O)=O)ns1 Cc1cc(OCC(=O)NC2(CNC(c3cc(Cl)cn3C)=O)CCCC2)cc(C)c1 c1(C(N2CC(CNC(C3CC(CC(C)(C)C)C3)=O)C2)=O)ccc(O)cc1O O=S(=O)(c1ccc(NCC2CCN(CCF)C2)c(Cl)c1)NCC(O)CCC1CC1 CC1CN(C(C2CCN(C)CC2)=O)CCC1N=c1[nH]c2c(F)cccc2o1 C1(CNC(c2c(OC)ccs2)=O)CN(C(C2C3(CC3)C23CC3)=O)CC2(CCC2)O1 C1(NC(Cc2cccc(C)c2)=O)CCC(C)(CNC(C23CC(C)(C2)C3)=O)CC1 N#Cc1cccc(C2CCCN2C(c2ccc(-c3ccc(F)cc3)nn2)=O)c1 Cc1sc(C(=O)NC2CC(NC(c3ccc[n+]([O-])c3)=O)CC2O)c(C)c1C c1(CC)ccc(C(C)C)cc1.C(C)(CC(=O)O)N(CC(=O)O)S(C)(=O)=O C1(CCNC(=O)C(C2CC2)C2CC2)CSCCN1C(c1ccc(CF)cc1)=O N1(CCCCNCCCC(C)OCCOCCOC)CCCC(C)C1 c1(-c2cn(CCO)nn2)ccc2nccnc2c1.O=C1OCCC1CCO C1(C(N2CCC(OCC(=O)Nc3c(CC)ncnc3)C2)=O)CC(C(C)C)=NO1.C1CC1 Cc1nc(C(N2CCN(C3CN(C(=O)C(F)F)C3)CC2)=O)c2ccccn12 Cn1c(C(N2CCCCC23CC3)C(=O)NCC2CCCO2)cnc1[N+](=O)[O-] C1(NC(C=C(CC)C)=O)(COC)CN(C(=O)CCCn2ccnc2)C1 CC1C(NC(c2cnc(Cl)c(C3CC3)c2)=O)CCCN1C(C1CC2(CSC2)C1)=O C1(CNC(C(CC)C)=O)C2CCCC1N(C(=O)C(C)CN(C)C)C2 S(=O)(=O)(CCC(=O)OCCn1cnc(Cl)c1)N(C)C c1(C(=O)NC(CNC(C(CC)OC)=O)C2CC2)cc2nc(Cl)ccc2o1 CC(C)C(C(=O)NCc1ocnc1CO)C(C)NC(=O)C=CC(=O)N(C)C CC1(C)CC(CNC(C2=NC=CSC=N2)=O)CN(C(c2nnn3c2CSCC3)=O)C1 C1(C(C)NC(c2ccn(C(F)F)n2)=O)CCCN(C(=O)C=C2CCCC2)C1 N1(C(C(C2(O)CCC2)NC(CC2ON=C(C)C2)=O)=O)CC(O)CC1C(N)=O c1(C(C)=O)ccc(C(=O)NC(C2CCCCC2)C(C)NC(c2cncs2)=O)cc1Cl C(=O)(CCCCCCNC(C1CCCN1CCC)=O)N1CCC(C#C)C1 c1(OC)ccccc1C(O)C(N1CC(O)(C(C)NC(=O)C#CC(=O)N(C)C)C1)=O c1(C(N(c2n(C)nc(O)c2)C2CC2)=O)n[nH]c2c1CCN(C(=O)CCCC(F)(F)F)C2 N1(C(C=CCC#N)=O)CC(C2CC2)C1.c1(C2(CC(=O)NC=CC)CC2)ccccc1 C(c1ccc(Br)cc1)=CCCNC(c1c(C)nccc1)=O c1(C(N2CCC(C)N(C(=O)C(=O)NCC(F)F)CC2)=O)cccc2c1C(C#N)C2 C(=O)(C(C)CN(C(=O)CCc1cnco1)C)NC(C#C)CC CC1CCC(NC(=O)CCCSC(C)(C)C)CN1C(c1cc(C(F)(F)F)ncn1)=O C1(CNC(COCCOC)=O)CCN(C(C2(C(N(C)CC)=O)CCC2)=O)CC1 C12(C(=O)NCc3nccc(C)n3)CC(CO)(CN1C(C1CC3COCC3C1)=O)C2 C1(CCOC)(NC(=O)C(=O)NC(C2OCCC2C(C)C)=O)CCCC1 c1(NC2CC(C)N(C(=O)NC3CN(c4ccccc4)C3=O)C2)cc2nncn2cn1 c1(-n2cc(C(C)NC(=O)C(N3CCC(C)C3C)=O)nn2)cccc(Cl)c1C C(=O)(CC(C)CN=C(NCc1cccc(C(F)(F)F)c1)NCc1ccon1)OC C1(CC#C)(C(=O)NC23CC2CN(C(=O)CCc2cnc[nH]2)C3)CCCCO1 C1(N(CCC#N)CCCc2ccccc2)CC2CNC1C2.c12cc(ncn1)N2 C1(CCNC(C2(N(C(C(C)n3cnnn3)=O)C3CC3)CCC2)=O)CC(=O)N(C)C1 C1(CNC(CC(C)C(F)F)=O)CN(C(=O)CCn2ccnc2)C2(CCOCC2)C1 Cc1nc(C(N2CC(NC(=O)CCN(C3CCCCC3)C)C3CC23)=O)c(C)s1 c1(OC)cncc(C(=O)NCc2cc(C(=O)N(C3CN(C(C)C)C3)C)n[nH]2)n1 Cc1cc(NCC(N)C(C)(C)C)c(C)n1C1CCC(C)CC1 C#Cc1ccc(C(N2CCCC2CS(C)(=O)=O)=O)o1 N1(C(c2cnc(SC)n2C)=O)CCC(NC(C2CC2C)=O)C(F)C1 C1(c2cn(C3CC(NC(C(C4CCCCCC4)OC)=O)C3)nn2)COC(C)(C)OC1 C(=O)(C(F)C(=O)N1CCN(CCNC(c2ccncc2Cl)=O)CC1)OCC Cn1cc(Cl)c(C(=O)NC2CCCCC2NC(=O)C(O)CC2CC2)n1 C1(NC(C2COCCC2(F)F)=O)C2CC1CN(C(c1ccc(Cl)cn1)=O)C2 CN=c1[nH]cc(C(=O)NCc2c[nH]nc2C(=O)NC(C)C(C)n2cccn2)s1 c1(N2C(C(N(C)CCOc3ccncc3)=O)CCC2)nc(Cl)nc2[nH]cnc12 c1(CN2CCC3(CCC(N)C3)C2)cccc2[nH]c3ccccc3c12 c1(C(=O)NC(C)C(C)(C)NC(=O)C2=CCCC2)cc2ccnn2cn1 c1(C(=O)NC2(C(=O)NCCOc3ccon3)CSC2)cnncc1O c1(OC)ccc(C(=O)NC2CC(C=O)C2)c([N+](=O)[O-])c1.N1(CCO)CCC(C)C1 Cc1cc(C(=O)NCC23CC2CN(C(=O)C#CC2CC2)C3)ccc1F C12(CCCN(C(=O)C(C)C(F)F)C1)C(=O)NC2.C(COC)=CC C1(C)(CNC(CC2CCCC(C)O2)=O)CC(F)(F)CN1C(c1cnn[nH]1)=O CCC(C)C(O)CC(=O)N1CCCC1C(=O)NCC(O)(CC)CC C1(F)(C(N2CCC(C(C)CNC(c3cnccc3Cl)=O)CC2)=O)CCCC=C1F Cc1ccc(S(=O)(=O)NC2CN(Cc3cn(CC(O)C(C)CO)nn3)CC2O)c(F)c1 C1(CNCCNC(CSCC#C)=O)CC(O)CCN1C(=O)CO.C(C)(=O)NC CCCC(CC)C(=O)NC1CCCCC1CNC(c1ccc(F)s1)=O N1(C(Cc2c(C)cco2)=O)CCC(c2ccccc2)(NC(C2CC23CC3)=O)CC1 C(CSC)(C(C)C)OCCc1ccccc1.C(=O)(COCC(=O)NC)N1CC1.CC c1(OC)cc(NC2CN(C(C3(OC(C)C)CCOCC3)=O)CC2(C)C)nc(C)n1 Cc1nc(Br)sc1C(=O)NC(C1(O)CN(C(=O)Cc2cnoc2)C1)C N1(C(C=CC(CC)C)=O)CC(CNC(c2cn(C)nc2OC)=O)C(O)C1 c1(CC(=O)NC2C(CNC(C3N(CCC)CCC3)=O)CC2)nc2ccccc2s1 Cc1cc(N2CCOCC(NC(C3CCCCN3C(N)=O)=O)C2)nc(S(C)(=O)=O)n1 C1(NC(C2C(C(C)C)OCC2)=O)CCN(C)C(=O)C1.c12cncc(c1)C(=O)NC2 c1(C(N2CCN(C(CC(CCC)C)=O)CC2CCO)=O)cc(F)c(C#N)c(F)c1 C1(NC(C(C)=CC2CC2)=O)COC2(C1)CN(C(C1CC(=O)N(C(C)C3CC3)C1)=O)C2 CC(C)CCC(F)C(=O)N(CCCNC(=O)C(C)C1(O)CCC1)CCO C12(NC(C(c3cccnc3)C)=O)CCCC1N(C(=O)C(C)Cn1ccnc1)CC2 N1(C(c2c(CC)ccs2)=O)C2CCC1CC(NC(=O)CC1C=CCC1)C2 Cc1cccc2cc(C(=O)NC3CC4CN(C(C5CC6CC6C5)=O)CC34)oc12 CC(C)CC(C)(C)C(=O)NC1CCCC1NC(c1ccccc1CO)=O C1(NC(CC(C)F)=O)CCC(NC(c2nccnc2N)=O)CC1 C(=O)(C(C)CO)N(C(C(=O)NCCOC(C)C)C1CC1)C CN1CCN(CCC(=O)Oc2ccc(N(CCCF)CCC#N)cn2)CC1 CCCC(CNC(=O)C(C)(C)O)C(=O)NC(C)(CO)CCCC C1(NC(C(CC=C)OC)=O)COC2(C1)CN(C(=O)CC1OCCO1)C2 c1(CNc2c(C(C)NC(C3CCN(C(C)=O)C3)=O)cco2)cc(C)ccc1F N1(C(C2CCC(C)O2)=O)CC2CC(C1)CN(C(=O)CN1CCCCC1)C2 CC1(C)CNC(=O)C1NC(=O)C(=O)NCCC1CCC(C)(C(=O)O)CC1 c1(OC)ccccc1C(CNC(=O)C(C)CO)NC(=O)CNc1scnc1C Cc1c(C(=O)NCC(C)N(C(=O)COCCOC)CCO)cnn1CCO C1(C(N2CCCC(C=C)C2)C(=O)NCC(=C)C)Cc2ccccc2C1 c1(NC(=O)C(N2CCC(CNc3ccco3)C2)=O)ccc(F)c(I)c1 C1(N(C)C(c2cnc[nH]2)=O)CCCN(C(=O)C(c2ccccc2)OC2CC2)C1 Cc1cc(Cl)c(Cl)cc1C(=O)NC1CN(C(=O)CC2=CCCCC2)C2(CCC2)C1 N(C1CCCc2occc21)C(C(c1ccco1)NC(C(=CC1CCCC1)C)=O)=O C1(C2CCCN(C(=O)CN(c3ccncc3)C)C2)(NC(CN(C)C(N)=O)=O)CC1 c1(C(N(C2CCCC(N(C(=O)CP(C)(C)=O)C)C2)C)=O)ccc([N+](=O)[O-])[nH]1 C1(NC(=O)CN2CC=CC2)CC=CCC1C(=O)NC1CCCNC1=O C=C1CCN(C(C2COCOC2)=O)C(C(N2CCC(OCCO)C2)=O)C1 N1(C(CCc2c(C)nc[nH]2)=O)CC2(CCOCC2)C1c1cnn(C)c1 c1(C(=O)NCC(CC=C)NC(=O)CCCc2nc(C)no2)cc2c(s1)CCC2 N1(C(c2c(C)cccc2N)=O)CC(C)(CNC(C23CCC2C3)=O)CC1(C)C c1(C(=O)NCCN(C(C(n2c(C)ccn2)C)=O)C(C)C)cnc(=NCCF)[nH]c1 C1(NC(c2nc(C)n(C)n2)=O)CCSC12CN(C(=O)CCC1NC(=O)NC1=O)C2 c1(C(=O)NCC(C2CC2)NC(C=C(C)c2cnn(C)c2)=O)ccc(S(C)(=O)=O)s1 C12CC=C(C(=O)NCCSCC(=O)N1)C2.N1(CC)CCCC(N(C)C)C1 C(=O)(C1=CS(=O)CCC1)NCC(Cc1ccccc1)NC(=O)CCn1cccn1 C1(C(=O)NC(C)CCO)COC2(CCN(c3ncc4[nH]ccc4n3)CC2)C1 C1(C(=O)NCC(CC2CC2)CO)(CNC(=O)Cn2ncnn2)CCCC1 N1(C(C(C=C)(F)F)=O)CCOC(C)(CNC(=O)Cc2cnc(C3CC3)[nH]2)C1 CCC(C)(C)CC(=O)N1CCOCC(C(N2CC(OC)C2)=O)C1 CCCC(CNC(c1cc(C)nn1C)=O)C(=O)NC1CC12CC(OC)C2 C1(CC=C)(CNC(=O)Cc2cnoc2)CCCN1C(=O)C(O)CCN(C)C Cc1nc(CC(=O)NCCC2(O)CCN(C(C3(C)COC(=O)C3)=O)C2)c(C)s1 c1(C(N2CC(CNC(C(C(C)C)OC)=O)CC2(C)C)=O)cc2nn[nH]c2cc1F CN1N=C(C(=O)N2CCC3CCN(C(c4ccc(=N)[nH]n4)=O)C3C2)CCC1=O c1(NC(CN2C(C)CC2C=O)=O)cnc2ccc(Br)cc2c1 C(CC(=O)N1CC(O)CCO1)N(C(C(c1ccccn1)C)=O)C c1(CCC(N2CC(C(N)=O)(CNC(=O)CN)C2)=O)cccc(Cl)c1Cl.CC(C)C c1(C(N2C(CC)C=CCC2)=O)ccc(S(=O)(=O)N2CCCC(C(C)C)C2)cc1 Cc1ncc(NC(=O)NC2C(C(=O)OC(C)(C)C)CC2(C)C)cc1F c1(OC)ncc(-c2scc(C)c2C)cc1C(=O)Nc1ccccc1C(N)=O C(CCC(C(=O)NCCc1cocn1)NC(c1cc(CO)on1)=O)OC C(=O)(C1=CCN(C(=O)Cn2c(C)ccc2C)CC1)N(C(CC)CC)C CC1CC2CC2CC1C(=O)NCC1CN(C(=O)Cc2ccc(CO)cc2)C1 c1(C(=O)NC(CNC(c2cccc(CC)c2F)=O)C2CC2)ccn2cccc2c1 N1(CCCc2c(OC)cccc2)C(=O)CN(CCc2nccnc2OC)C1=O C12(C(=O)NCc3c(C)noc3)C(NC(c3ncc(F)cc3C)=O)C3CC1C2C3 CCCC(F)(F)C(=O)N1CCC(C(=O)NCC2(C)CC(F)(F)C2)CC1 C12(CCCCC1C)C(=O)NC2.c1(OC(CC)C(=O)NC2(CO)CC2)ccccc1C c1(C(=O)NCC(C)NC(C=Cc2ccc(SC)s2)=O)ccc2nc(O)n(C)c2c1 c1(C(=O)NCC(C)N(C(=O)C(C)OCC(C)C)CC)cnsc1C C#Cc1cc(C(=O)NCC(CC(C)C)NC(=O)CS(=O)(=O)N(C)C)cc(F)c1 C(=O)(C(C)CC(=O)c1ccc(F)cc1)N(CC(CNC(C(C)OCC)=O)C)C C1(C(=O)NCCC(C)NC(c2[nH]cc(CC(C)C)c2)=O)CCN(C)C1C c1(C(C(=O)NCC(CC)NC(C2(CC)CCOCC2)=O)O)cc(F)c(F)cc1F CC(C(=O)N(C)CCN(C)C(C1CC(=O)CO1)=O)S(C)(=O)=O C(=O)(CCCCCCCC12CCCC1C2)NC1CN(C2CN(C(C)=O)C2)C(=O)C1 CC(C)C#CC(=O)N1CCCC1C1(O)CN(C(c2cccc(C)c2)=O)C1 C1(C(=O)NCCNC(C2(C(=O)OC)CC(O)C2)=O)CCn2ncnc2C1 c1(-n2cc(C(=O)NCC(N3CCCC3Cc3cccs3)=O)nn2)ccccc1F c1(C(C(=O)NCC(=C)C)(C)N(c2ccccc2)CC2CC2)cn2cccc(F)c2n1 c1(C(=O)NC2CC(NC(C3CCC(OC)C3)=O)C2)cc(C)nnc1O c1(SCC(=O)NCC2CCCC(NC(C(C)CF)=O)C2)nc2ccccc2n1C C1(C(C)NC(C2(c3ccccc3)CC2)=O)CN(C(=O)OC(C)(C)C)CCO1 N1(C(C(c2ccn(C)c2)C)=O)CCCC(C)(C)C1C(=O)NC1C(C)CCC1C Cc1nsc(N2CCC(C)C(NC(=O)CS(N)(=O)=O)C2)c1C#N C(=O)(C(C)(C)S(C)(=O)=O)NCCC1(CNC(c2c(C(N)=O)ccc(C)c2)=O)CC1 Cc1ccc(Cl)c(F)c1C(=O)NC1CC(C(=O)O)C2CC12 N1(C(C2CN(CC)C(=O)CC2)=O)CC2(CC(NC(C3CC4CC4C3)=O)CO2)C1 c1(C(=O)NC(C)CNC(=O)COCc2nc(C(C)C)no2)cc(CC)cn1C c1(C(=O)NCCC2CN(C(CN(C)C)=O)C2)ccc([N+](=O)[O-])c(S(N)(=O)=O)c1 c1(C(=O)NCC(CNC(C(C)OCCOC)=O)O)sc2ncccc2c1Cl Cc1nc(O)c2cc(C(=O)NCC3CC3NC(C3CC4CCC3O4)=O)ccc2n1 C(C(CC(F)(F)F)NC(C1CCC1(C)C)=O)NC(C1(CC#C)CCC1)=O N1(C(CN2CC(=O)NCC2)=O)CC2CCC1CC2NC(=O)C=Cc1ccoc1 c1(C(=O)NC(C)(C)CF)cc(CNC(=O)C=CCO)ccn1 CCCCCC(O)CC(=O)N(CC(=O)NC(c1ccc(C)nc1)C)C n1(CC(=O)NCC2(NC(C3CC=C(C)CC3)=O)CCC2)nc(C)c2c1CCCC2 CCCCC(CC)CC(=O)NCCOCCNC(c1cc(Cl)ns1)=O Cc1ccc(C(N2CCCC(C(=O)NC3CN(C)CCC3O)C2)=O)cc1O C(=O)(C(F)(CNC(=O)C(C)(C)C(C)O)C(C)C)NCC1(C=C)CCC1 c1(N2CCC(C(C)NC(C(CCCC)C(C)C)=O)C2)nc(Cl)nc2[nH]c(O)nc12 C(CCCCCC(=O)N(C)Cc1ccoc1C)NC(CC(C(=C)C)OCC)=O C1(C(=O)NCCC2CCN(C(C=CC(C)(C)SC)=O)C2)CCCCC1O c1(C(=O)NCC(CNC(c2n[nH]cc2C2C(C(C)(C)C)C2)=O)O)ccncc1NC C1(NC(c2c(C)nc(N(C)C)s2)=O)CN(C(=O)C(F)C2CCC2)C2(CCOCC2)C1 C1(NC(C(CC)=CCCC)=O)CC(C2CCN(C(c3cscn3)=O)C2)C1 CCCC(CC(=O)NCCC(=O)NC(=O)CO)NC(=O)C(C1CCC(=O)N1)(C)C CCCC(CCCNC(c1ccc(CN(C)C)cc1)=O)N=c1nc(C)[nH]s1 C(=O)(C1CCc2c[nH]nc21)NCCN(C(c1cc2sccc2s1)=O)CC N1(C(=O)NCc2ccncc2)CCC(F)(Cc2ccccc2)C1 CC(CN1CCOCC1)C(=O)N(CCCNC(=O)C(C)CN1CCOCC1)C1CC1 c1(C(=O)NC2C(OC)CN(C(C34CC(C)(CCO3)C4)=O)C2)cn2ccnc2cn1 c1(C(=O)NCCC2CCC(NC(c3c(C)ncs3)=O)C2)nc(O)c(C)s1 N1(C(c2c(C(=O)OC)csc2)=O)CCC(NC(=O)CSC)C2(CCC2)C1 C1(C#N)(C(=O)NCC(C)N(C(=O)CCOCCN(C)C)C)CCCOC1 C(=O)(C1CCc2nccn21)N(C(CCNC(CC(C)F)=O)C)C n1(C2CN(C(C3(F)CCNC3)=O)C2)cc(Cl)ccc1=O Cn1[nH]c(C(=O)NC2(CC(=O)NCC3CC(CN=[N+]=[N-])C3)CC2)nc1=O N1(C(c2c(C)nc(O)cc2)=O)CCC2(NC(=O)Cc3cccnc3)CCCC12 C1(C(N(C2CCN(C(CC3(C=C)CC3)=O)C2)C)=O)(NC(N)=O)CCCCC1 C1(C(=O)N(CCNC(C2(N(CCC(=O)N(C)C)C)CCCC2)=O)N(C)C(=O)CC)CCC2(CC2)C1.C CC1(C)C=C(C(=O)NCCCC2CCCN2C(=O)CNSc2csc(=N)[nH]2)C1 N1(C(C(N2CCCCC2C)C)=O)CCC(O)C(C(=O)NOc2ccccc2)C1 c1(CCC(=O)NC(c2ccc(Cl)cc2)C(=O)O)ccc2[nH]c3c(c2c1)CCCC3 c1(CCC(N2C(CN(C)C(C3CC34CCOC4)=O)CCC2)=O)ccc(C#N)cc1 C1(C)(C(N2C(C)CC2CO)=O)CCN(C(=O)C(F)C2CCCC2)CC1 C1(NC(c2c(C)onc2-c2ccccc2Cl)=O)CCN(C(=O)C(C)C)CC1F N1(C(C(F)=CCC)=O)Cc2ccccc2CC1CNC(=O)CC1CNC(=O)C1 C(=O)(C(C)S(N)(=O)=O)N(CC)CC1CCCN1C(c1coc(CO)c1)=O n1(CC(=O)N(CCCC)CC(=O)NC(c2ccccc2)CF)c(C)ccc1C c1(CC)ccc(C(=O)OC)cc1NC(=O)C(=O)NC1CCN(C)C1C C(=O)(C1=CCC(NCC(=O)NC(=O)CN(C)C(C)C)C1)NC(C(C)O)(C)C C=CC(C)CC(=O)NC(C1CCCCC1)CNC(c1cc(CCCO)on1)=O C1(CN(C(C2CC2F)=O)CC)CCCCN1C(=O)C(CSC)OC C(=O)(C1=CCCC1C)NCC(C)N(C)C(c1cn(C)nc1C1CCOCC1)=O CC(F)(F)CC(=O)NC1CCN(CCNC(c2ccc(CO)cn2)=O)CC1 S(=O)(=O)(c1cccc(S(=O)(=O)NC(C)(C)C)c1)NCC(=C)CC c1(C(=O)NC2CCN(C(C3(CC#C)CCOCC3)=O)C2)cc(C#N)cn1C N1(CCn2cc(COC)nn2)CCN(C(C2C(C)CCN2C)=O)CC1 c1(CNC(C2CC(OC)CN(C(CCOCC#C)=O)C2)=O)ccc2ncsc2c1 N1(C(CC2ON=C(CC)C2)=O)CC2(CNC(=O)N2C)C1.C(=O)C1=C(C)OCCC1 c1(NC(C2N(Cc3n(C)cnc3)CCNC2)=O)cc(F)ccc1[N+](=O)[O-] c1(C(=O)NC2CC(CC(=O)NCC3CCCCO3)C2)cc(F)c2cc[nH]c2c1 C1(NC(=O)NC(CN(C(=O)CC(C)n2cccn2)CC)C)C2CC(=O)CC12 N1(C(c2nc(CC)oc2)=O)CCCC(O)(CCNC(=O)CN2CCCC2CO)C1 N1(N2CCC(C3N(C(CCCCSC)=O)CCCC3)CC2)CCN(CCO)C(=O)C1 N1(C(C=CC)=O)CC2CCC1CC2NC(=O)CC(C)(C)O N1(C(c2nc(CCC)oc2)=O)CC(NC(=O)CC(C)n2ccnc2)CC2(CC2)C1 c1(C(=O)NCCCC(C)NC(C2CC3C=CC2C3)=O)cnn2cc(C#N)cnc12 N1(C(c2cn(C)nc2)=O)CC(CNC(c2cccc(OCC(F)F)n2)=O)C(O)C1 C1(C(N(CC(C)C#N)C)=O)CC2CC1CC2NC(=O)CCC(N)=O n1(CC(=O)N(CCCNC(c2ccc(C#C)nc2)=O)CC)cc(P(C)(C)=O)cn1 C=CC(CC)C(=O)NCC1CCN(C(C2CC(OC(C)(C)C)C2)=O)CC1 Cc1cccc2oc(C(=O)N(C)CC3CCCN(C(=O)C#CC4CC4)C3)cc12 c1(C(=O)NCCOCCN(C)C(C2CNC(=O)N2C)=O)ccc2c(c1)CCCS2 c1(C(=O)NCC(C)CNC(c2ccnn2CC(F)F)=O)cccc(Br)c1 N1(C(CC=CC=C)=O)CCCN(C(=O)CCOCC(F)(F)C(F)(F)F)CC1C N1(C(c2cc(O)ccc2O)=O)CCN(C(c2cc(Cl)ncc2Cl)=O)C2(CCC2)C1 N1(C(C2(CC=C)CCOC2)=O)CCCC2(CCCN2C(c2cnn(C)c2C)=O)C1 C(C)(CCC(=O)NCC1CCN(C(c2csnc2Br)=O)CC1)SC Cc1cccc(C(c2nc(-c3cncnc3)nn2-c2nccn2C(C)(C)C)=O)c1C Cc1ccc(C(=O)NC2CC(C)CN(C(c3ccnc(C)c3C)=O)C2)cc1Cl C1(C(N(C2CCN(C)C2)CC)=O)COC(CNC(=O)CCCOC(C)=O)C1 C#Cc1c[nH]nc1C(=O)N(Cc1cncc(C(=O)O)c1)CC C(=O)(CS(=O)(=O)C(C)C)N1CCC(CN2CCN(C(COCCC)=O)CC2)CC1 c1(C(=O)NC2COC3CN(C(CCOC(C)C)=O)CC32)cnc(O)c2cncn12 CC(C)C(C)CC(=O)N1CCCC1CNC(=O)C(O)CCN(C)C n1(CC)nc(C)c(C(=O)N(CC(C)NC(c2n[nH]c(Cl)c2Cl)=O)CC)c1C C(=O)(C(CC(F)(F)F)c1ccc(Cl)cc1)NCC(C)N(C)C(C1CCNC1=O)=O C(=O)(CC(F)(F)F)N(C(Cc1ccccc1Br)C(=O)NC1CC(CF)C1)C n1(CC)nc(C)c(C(N2CCN(C(=O)C(C)C(C)(C)C)CC2C2CC2)=O)c1C C(CCN=C(NCC1CCCN1C)N1CCC(F)C1)OCC c1(C(N(CC(CNC(C=C(C)C2CC2)=O)C)C)=O)cnc2c(F)cc(C)cc2c1 N1(C(C2CCN(C(C)=O)C2)=O)CC2CC2(CNC(c2csc(C)n2)=O)C1 C1(C(C=CC(C)(C)SC)=O)CCN(C(C)C(=O)N2CCCC2)C1 C1(CNC(c2n(CCC)nc(C)c2)=O)C(O)C(O)CN1C(C1CC2(C1)CC2F)=O C12(C(=O)NC(Cc3cnc[nH]3)CO)CC(NC(C3CCCSC3)=O)(C1)C2 c1(CC(=O)NCCN(C(=O)C2=NOCC2)CC)cc(C(F)(F)F)cc(Cl)n1 CCCCC(C)C(=O)N1CCCC1CN(C(=O)CCc1nc[nH]n1)C N1(CC(C)(C)OCCn2ncc(NC(=O)NN)c2)CCCCCC1.C(CC(=O)O)C c1(CNC(C(C2OCCO2)OC)=O)cnccc1C n1(C(c2ccccc2)C)cc(NC(=O)C(C2(CO)CCOCC2)N)c(C#N)n1 CCC(CNC(=O)C(C)CNC(=O)CSCC(N)=O)CC(C)C C(=O)(C1=NOC2(CCC2)C1)NCc1cc(CNC(C(F)OC)=O)no1 Cc1nc2nccc(N(C)CC3(O)CCCN(C(=O)C(O)c4ccsc4)C3)n2n1 c1(-c2cn(Cc3n(CC)ncn3)nn2)ccc2c(c1)OCO2.C1(SC)CCCC1SC C1(NC(c2ccnnc2)=O)CN(C(=O)Cc2ccc(Br)s2)CCC1CO C1(C(=O)O)(NC(c2cnc(-c3ncccn3)s2)=O)CCNCC1 c12cccnc1N2.c1(C(N(CC(CN(C)C)O)C)=O)ccc(N)cc1.C(N)=O C(c1ccc(F)cc1)=CC(N1CCC(N(C(CC=CCC)=O)CC)C1)=O N1(C(C2C(=C)C2)=O)CC2(CC(NC(c3cn(C4CCC4)nn3)=O)c3nccn32)C1 C(=O)(C(F)CC(CC)CC)NC(CC=C)C(=O)NCC1CN2CCC1CC2 c1(C(N2CC(C)N(C(=O)CCC3CCCCO3)CC2)=O)nncc2c1CCCC2 C(C(O)CC(=O)NCC(F)CO)NC(CCc1n(C)ccc1)=O N1(C(c2cc(C)c(F)c(C)c2)=O)CCN2C(=O)C(C)CC2C1 S(=O)(=O)(c1ccc(NCCNC(C)=O)c(Br)c1)NCCN1CCN(CCC)CC1 C(=O)(C1=CCC(NC(C2CC(C3CC3)C2)=O)C1)N(CC)CC1CCOCC1 c1(C(=O)NC(CC)CNC(=O)C(CO)NC(=O)C(F)(F)F)cc2sc(C)cc2s1 N1(C(C(C)CC2CCNCC2)=O)CCC(=O)N(C)c2ccccc21 N1(Cc2ccc(C)cc2F)CCC2(CC1)CCN2C(=O)OC(C)(C)C C(CC(=O)NNC(=O)c1c(C)nsc1Br)n1cc(CCSC)nn1 c1(CNC(C2COCCN(Cc3cc(O)ccc3Cl)C2)=O)ccc2c(c1)OCCO2 C(=O)(CS(=O)(=O)CC(=O)N1CCCCC1Cc1cn(C2CC(O)C2)nn1)OC N1(C(c2c(C)noc2)=O)CCC(C(N2CC(F)(C3CC3)C2)=O)C(O)C1 C(=O)(C1=CCCC1C)NCC1(COC)CCCN1C(c1ccn(CC(C)C)n1)=O c1(CC)cnn(C)c1C(=O)N(CC(CC)NC(=O)C(C)(C)CO)C C1(OC)CCN(C(=O)C(F)C2(c3nn[nH]n3)CCC2)CC1C(N)=O c1(C(C)CC(=O)NCCN(C2CC2)CC2COC2)ccccc1Br C1(NC(C(C)(C)OC)=O)CCC(NC(=O)C=CC(C)C)CN1C(=O)OC(C)(C)C N1(C(C2CC(=O)NC(=O)N2)=O)CCC2(CC2)CC1C(=O)NCCOCF.C1CO1 S(=O)(=O)(CC#Cc1ccccc1)NC(C1CC(C)OC1=O)=O C1(NC(C2CCC=CO2)=O)CCC2CN(C(c3ccc4cccnn34)=O)CC2C1 C1(C(NCP(C)(C)=O)=O)CC2CC2N1C(c1ccn(C(F)F)n1)=O N1(C(C2OCCC(C)C2)=O)CCC2(CCCN(C(C3C=CC=CC=C3)=O)C2)C1 CCN=C(NCCC(=O)NCCCC(C)(F)F)NCC(c1ccccc1)OC n1(CC(=O)N(C2CCC(NC(Cc3cc(C)nn3C)=O)C2)C)nc(O)ccc1=O Cc1ccc(C)c(NCC(N2CCN(C(=O)CSC(F)(F)F)CC2CCO)=O)c1 C1(C(N(CC(O)CNC(=O)CNC(C2CC2c2ccsc2)=O)C)=O)CCCCO1 CN1CC2CCN(C(=O)CC(C3CC3)NC(c3ccc(C#N)o3)=O)C2C1 c1(C(N2CC(NC(C3(C#N)CC4CC4C3)=O)C2)=O)cc2c([nH]1)CCCC2 CC(O)(CC(=O)NC1C2CCC1N(C(c1[nH]nnc1C1CC1)=O)C2)C(F)(F)F c1(COC)ccoc1C(=O)NC(C)C(C)NC(c1ncccn1)=O n1(CC)ncn(NC(=O)c2cc3n(n2)CCCC3)c1=O.C12CCN(C1)C(=O)C2 Cc1cc(C(=O)NCc2cc(C(N3CC4CC4C3)=O)co2)c(C)s1 C(=O)(C1=CCC(NC(c2cnc(OC)s2)=O)C1)N(C1CC1)CC N1(C(Cc2c(C)ocn2)=O)CCOCC1CNC(=O)CSc1cn[nH]c1 CCC(CC)(CC)C(c1ccccc1)N(S(=O)(=O)CC(C)OC)C C1(NC(CCCOC(C2CCCC2)C)=O)CCN(C(=O)CCC2CC2(C)C)C1C N1(C(C(C)SC(C)C)=O)CCC2(CC1)CC(C(=O)Nc1nccn1C)CCO2 N1(C(c2c(C)ncs2)=O)CCCC(NC(=O)CC2CC3CC3C2)C1C Cc1oc(Cl)nc1C(=O)N(C1CCN(C(C2CCOC2C)=O)CC1)C(C)(C)C Cc1cc(C#N)cnc1C(N1CCC(C)C(N(C(=O)C=CBr)C)C1)=O C1(OC)CC(C(=O)NCc2nc[nH]n2)N(C(C2CCC(=O)N2)=O)C1 C(C)(CNC(C1(C)CCN(C(C)=O)C1)=O)(C(C)C)NC(C=CC=CC)=O C12(C(=O)NCC3(OC)CCN(C(C4(C#N)CC=CCC4)=O)C3)CCC(CC1F)C2 C1(C(N(C)CCOC(F)F)=O)(NC(=O)Cc2cncnc2)CCCC1C C1(C(N2CCN(C3CCCN(C(C4(CF)CCC4)=O)C3)CC2)=O)C2CC3C(C2=O)C13 c1(C(C)=O)ccc2sc(C(N3CC(O)CC3c3ccc(F)cc3F)=O)c(C)c2c1 C1(CC(=O)NC2CCC(CNC(c3cnc(C)[nH]3)=O)C2)CCCCC1O c1(C(=O)NCC2C(CNC(c3c(OC)c[nH]n3)=O)C2)c(C)[nH]cc([N+](=O)[O-])c1=O C1(N(C)C)CCC(C(N2CC(=C(F)CNC(=O)Cc3nnc(O)s3)C2)=O)CC1 C(=O)(CC(=O)NCC(C1CC1)N(C(=O)Cc1cncn1C)C)OC N1(C(CC2CCCN(C)C2)=O)CC2CC(NC(c3cncnc3)=O)C(C2)C1 Cc1ncnc(C(=O)NCCC(C)N(C)C(C2CC(=O)NC2(C)C)=O)c1C C(CC(C)(C)C)N(C(C(C)N(C(C1CCCOC1)=O)C1CC1)=O)C1CC1 CC(C)CC(C(=O)N(C(C)CN(C)C)C)ONC(=O)C(C)(O)C1CCC1 C1(C(=O)NC(CNC(c2ccc(C=C)cc2)=O)CC)CCOCC12CCC2 C(=O)(N=c1ccn(C)[nH]1)Nc1c(CC(C(=O)Nc2cccc(C)c2)C)c[nH]n1 N1(C(C(CCSC)NC(C2CC(F)(F)C2)=O)=O)CCn2nc(C)cc2C1 N1(C(c2c(C)ncs2)=O)CCCC(C2CCN(C(C3CCCN3C3CC3)=O)CC2)C1 CC(C)C(C)C(CNc1cccs1)N=c1cc[nH]c(=NCCCc2nccc(O)n2)[nH]1 c1(C(=O)NC(CC2OCCO2)CO)cncc2c1CCCC2 c1(NC(C2C3CN(Cc4cc(C)nc(C)c4)CC32)=O)ncnc2cnn(C)c12 C1(N(C)C(c2cnn(-c3cccc(F)c3)c2)=O)CN(C(=O)C(N)=O)CC12CC2 N1(C(c2cc(C)cc(OC)c2O)=O)CCCC2C1CCCN2C(C)=O C(=O)(N=c1cc(OC)n(C)[nH]1)C1(OC)CCN(C(c2ccc(C(=O)NC)cc2)=O)C1 C(=O)(C1CCc2cc(Cl)ccc21)NC(C(C)NC(=O)Cn1nccn1)(C)C C1(CNC(C(CNC(c2cc(O)cc(=O)o2)=O)O)=O)CC2(CCO1)CC2 c1(C(N(CC(=O)NCCN2CCCC2=O)C)=O)cc2cccnn2c1 c1(NC(C(c2cccc(Cl)c2)CC)=O)ccc2c(c1)oc(=O)n2C C1(NC(CCCC#CC)=O)CN(C(c2cc(Cl)ccc2OC)=O)C2(CCC2)C1 Cc1ccc(NC(=O)NCC(N2CCCC(n3cc(NC(N)=O)nn3)C2)=O)cc1 C1(NC(CCCOC)=O)CC2(CCN(C(C3C4CCC(F)(F)C34)=O)CC2)C1 c1(C(=O)NC2CC(C(C(=O)NC(CC)C(C)(F)F)F)C2)c[nH]c2cnccc12 N1(CC2CC3(CCC3O)C2)CCC2CN(C(=O)CC3(C#N)CCCCC3)C2C1 C(=O)(C(CC)CCOC)N1C(C(CNC(C(CC)CC)=O)(C)C)CCC1 C1(C(=O)NC2C(C#C)CCC2)CC2CC1CC2NC(c1ccn(C(C)C)n1)=O C1(CNC(c2ccc(Cl)nc2)=O)COCCN(C(=O)C(=Cc2c[nH]cn2)F)C1 C=C1CCC(C(=O)NC2CCC(CC(=O)Nc3cnccc3Cl)CC2)CC1 C(=O)(C1CCOc2c(F)cccc21)N1CCCCC(NC(CNC(N)=O)=O)CC1 N1(C(CC2CCN(C)C2)=O)CC2CCCC(NC(=O)CC=C(Cl)Cl)C2C1 N1(C(C2N(C)CC(C)(C)C2)=O)CCC2(CC(NC(=O)CCS(N)(=O)=O)C2)C1 C1(CNC(c2n(C)cnc2)=O)CC(NC(=O)CCCC(F)F)C12CCC2 C1(CNC(C(CC)(C)CC)=O)CCN(C(=O)Cn2cnc(Br)c2)CC1(F)F C1(C(=O)NC2C(NC(c3ccn(C)c3)=O)COC2)CCOC1(C)C c1(OC)cc(C(=O)N(C2CCCN(C(=O)CN(S(C)(=O)=O)C)C2)C)nn1C C12(C(=O)NC3C4CC(NC(CC(C)SC)=O)CC43)CC1COC21CCC1 c1(C(N2C(CN=c3c(C#N)cn(C)[nH]3)CCCC2)=O)coc2c1C(=O)NCCC2 c1(COC)cc[nH]c1C(=O)NCC(n1cc(C(=O)NCC2CC3(CC3)C2)nn1)C C(=O)(C(O)CCCSC)NCC(CNC(c1ccc(C(C)=O)[nH]1)=O)OC N1(CC)OCC(NC(=O)CC(F)(F)C2CC2)C1=O.c1(C(=O)OC)cc(CCO)on1 N1(C(CCOCCOCC)=O)CCCCC1C1CCCN1C(c1cncnc1)=O CCS(=O)(=O)c1cccc(C(=O)NC2CC(n3cc(C4CCC4)nn3)C2)c1 C(CC(C(=O)NCCn1cnnc1)NC(=O)C(c1cnn(C)c1)=O)=CC CC1(C)CC1(C(N1CC=CCC1)=O)NC(=O)CC1CCOC1 c1(C(C(=O)NCC)N(CCOCC)CC)ccnc2ccnn12.c1(CO)ccccc1 N1(C(CN(C)CC)=O)CC2CCCC(C1)N2C(=O)C1=NOC(C(C)(C)C)C1 c1(CC(=O)NC(C)(C)CNC(C2CCNC2=O)=O)c[nH]c2ccccc12 C1(C2CCC2)(C(=O)NCC2(C)CCCN(C(C(C3CCC3)OC)=O)C2)CC1(F)F C1(CC)CC(C(N2CCC(OCCNC(=O)COC(C)CC)CC2)=O)CCO1 c1(CC)conc1C(=O)NCC(C)(C1CCC1)NC(=O)CCc1ncnn1C [N-]=[N+]=NC1CCN(C(=O)C(O)C2CN(C(=O)COCC3CC3)C2)CC1O c1(C2(C3OCC(C)C3)CC2)ccc(-c2nccs2)cc1 CCCCC(O)CC(=O)NCCCN(C(=O)CCCC1(C)N=N1)C1CCCC1 C1(CN(C(=O)CCc2nocc2CC)CC)CCN(C(=O)C(C)CC2CC2)CC1 N1(C(=O)CN(C)C)CCCC1C(=O)NCC12CC(NC(C3CC(=C4CC4)C3)=O)(C1)C2 C1(NC(C2=NOCC2)c2n(C(CC)(C)C)nnn2)CC(C2CC2)(C2CC2)C1 c1(OC)ccc(C(=O)NCCNC(C2CCN(C)C(=O)C2)=O)c(Cl)c1 c1(CC(=O)NC2CC(F)(CNC(c3cnc(S)[nH]3)=O)C2)c[nH]c2cc(F)ccc12 N1(C(C(CCC)C(C)C)=O)CC(C2CCCCN(C(C3CN(C)C(=O)N3)=O)C2)C1 C(CN=c1[nH]c(=NCC2CC=CC2)[nH]c2c1COCC2)(C1CCCOC1)OC C1(NC(c2cc(CNC(C(C)c3cc[nH]n3)=O)sc2)=O)CCCCC1F c1(CC(=O)NC(CCCCNC(c2cc(CC)n(C)n2)=O)C)c(Cl)cccc1Cl N1(C(=O)CC2C=CCC2)CC2CCN(C(c3c[nH]cc(F)c3=O)=O)C2C1 N1(C(=O)NC2CN(C3CCN(C)C(=O)C3)C2)CCOCC12COCCN(C)C2 CC(C)CC(C)C(=O)N1CCCC(C)(CNC(c2cc(CO)ccc2Cl)=O)C1 CCC(CC(=O)N1CCC2C(CO)C12)NC(=O)OC(C)(C)C C1(NC(C(CC)OCC2CC2)=O)C2CC3CN(C(=O)CNS(=O)(=O)CC)C1C3C2 C1(C(=O)NCC2CN(C(=O)C3=COCC3)CC2(F)F)(OC)CCCCCC1 c1(C(N(CC(C)NC(c2cc(CC(C)C)on2)=O)CC)=O)sccc1S(C)(=O)=O C1(C(N(CCN(C(c2c(C)nc(C3CCC3)s2)=O)C)C)=O)CCCCC1N=[N+]=[N-] Cc1cnc(NCC(C)N(C(=O)CC2C(C)(C)C2(C)C)C)nc1S(C)(=O)=O C(=O)(C(C)(C)C(C)O)N1CC(OC)C(NC(=O)Cc2ncccc2C)C1 c1(CCNC(C(c2cccs2)NC(CCOCC#C)=O)=O)ccncc1C C1(C(=O)NC2C(CNC(C(C)OC)=O)CCC2)CC(=O)N(c2ccccc2Cl)C1 CC1CNc2c(C(=O)N(C)CCNC(c3nc[nH]c3C(C)(C)C)=O)cnn2C1 N1(C(c2c(C)ncn2C)=O)CC2(CC(CNC(=O)C=CC(C)(C)C)C2)C1 n1(C(C)(C)C)cc(C(=O)NC2CCC2NC(c2ncc(-c3cccs3)s2)=O)cn1 N1(CCC)CCC(C(=O)NC23CC2CN(C(=O)C=CC(C)(C)SC)C3)CC1 N1(C(CC2(COC)CC2)=O)CCCC(CNC(C2C3CC4C(C3)C24)=O)C1 c1(C(=O)NCc2c(F)cc(C)c(F)c2)c(F)cncc1C1=CCN(C)CC1 C1(C(=O)NC2CC(CCNC(C3(C)N(C(C)=O)CCC3)=O)C2)CC(C)(C)CCO1 C=C=C(C)CC(=O)N1CCC(F)(CNC(=O)CCn2cncn2)C1 N1(C(C2(NC(=O)Cc3ccn(C)n3)C(C)C2)=O)CCCCC1CCCO Cc1cccnc1CCC(=O)NC1(C)CCN(C(C2CCCN2N=O)=O)C1 CCC(CCC(=O)N1CCN(C)C(C(=O)NC2CN(CC)CC2OC)C1)OC C1(C(=O)Nc2ccc(OC)nc2C)CN(C(C2SCC=C2C)=O)CCC1(C)C c1(C(N2CC(CC(=O)NC(C(=O)NC(C)C)C)OCC2)=O)ncc(F)cc1F C(=O)(CC1=CCCCC1)N1CCCCC(CCC(=O)NC2(C)C(C)CCCC2)C1 C1(C(N(CC(=O)NC)C)=O)C(C2CC2)CCN1C(c1cc(Cl)ns1)=O C1(C(=O)OC(c2nccs2)CC)(CNC(=O)OC(C)(C)C)CCc2ccccc2O1 c1(OC)c(C(c2nnnn2C(C)(C)C)NCC23CCC(CC2)OC3)ccnc1F c1(NCC(S(=O)(=O)NC)C)cccc(S(=O)(=O)NCCCCCC2CC2)n1 N1(C(C(Cc2ccccc2)NCc2ccc(C(=O)O)o2)=O)CCCC(COC)C1 C12CN(CC13CC3)C2OC(=O)C(C)(C)Cc1ccc(Cl)cc1.C(C)(C)(C)OC(C)=O C12(NC(COC)=O)CC(NC(=O)COCc3nc(C)no3)(C1)C2 N1(C(CCNC(N)=O)=O)CCC(CN2CCN(C(C3CC3C(N)=O)=O)CC2)CC1 C(=O)(C(O)CC(C)(C)C)NCCC1N(C(CCCCCN(C)C)=O)CC(F)(F)C1 Cc1cc(C(=O)NCCC2CN(C(c3cc(C)[nH]c3C)=O)C2)n(C)n1 CCC(C(=O)NCCOCCNC(=O)CCCc1cc[nH]n1)OC CCCC(CNC(=O)C=Cc1ccnn1C)C(=O)N(C(C)CN(C)C(C)=O)C N1(C(C2(C)C(C)C2)=O)CC(C2CC2)(C(=O)NCC2CC(C#N)C2)C1 C1(NC(CSC)=O)CCC2(CCCN2C(=O)C(C(C)C)c2ccc(Cl)cc2)CC1 CC(Cn1nnc2c1CCCC2)N=c1[nH]c(=NCCCS(C)=O)[nH]c2c1CSC2 C#Cc1cccc(CC(N2C3CN(CCS(C)(=O)=O)CC23)=O)c1 CCC(C(=O)N1CCCC(CN(C)C(C23CCC(C(=O)O)(C2)C3)=O)C1)C(C)C C1(CNC(=O)CCF)COCCN(C(=O)CC2CC3CC3C2)C1 N1(C(CC(C)c2ccco2)=O)CCC(C)C(N(C)C(c2ccc(F)cn2)=O)C1 C=CC(C)CCNC(c1occc1CNC(=O)Cc1cnn(C)c1)=O N1(C(CN2CC(C)(C)C2)=O)CC2(CCC(CNC(C3CC=CCO3)=O)O2)C1 c1(NC(c2ccc(Cl)c(C#N)c2)c2n(C(C)(C)C)nnn2)ccc2nncn2c1 N1(C(C2C(C3C(C)C3)C2)=O)C2CCC1(CNC(=O)C(F)(F)C(F)F)CC2 c1(C(N2CC(OCCNC(=O)C(O)CC3CC3)C2)=O)cc(F)ccc1Cl C1(NC(c2c(C)nns2)=O)CC(C(=O)NCCCC2CCC2)C1(C)C CN=c1ccc(C(N2CCCC2CNC(=O)C(=O)NOC)=O)c[nH]1 C12(NC(C3CCN(OC)CC3)=O)CCC(CNC(=O)C(F)(F)CC3CC3)(CC1)OC2 c1(OC(C(=O)NCC(CC)NC(=O)CSC)(F)F)cc(Cl)cc(Cl)c1 c1(C(=O)NCC(C2CCCC2)NC(C2N(CC)CC2)=O)ccc(S(=O)CC#N)cc1 C(=O)(C1=NNC(=O)CC1)NCC1(CNC(c2cccc(NC)n2)=O)CC12CCC2 c1(CCC(=O)NCC2(CNC(C(CC)C)=O)CC2(F)F)cccc(C(F)F)c1 CC(C)C(C(=O)N1CCCC(NC23CC(C(N4CCCC4)=O)(C2)C3)C1)C1CCC1 c1(COC(C=CCCC(C)C)=O)cc(C#N)c2c(c1)OCCO2 C=CC1CCCN(C(C2CC2C(=O)Nc2cnccc2NC(=O)OC(C)(C)C)=O)C1 N1(C2N(Cc3nc(C4C=CCCC4)sc3)CCC2)CC2(CCCC2)C1 n1(CCC=C)cc(CC2(O)CN(C(C3(CCS(N)(=O)=O)CCC3)=O)C2)nn1 N1(C(C2CCC(C)(CC)O2)=O)CC(C)N(C(=O)Cc2cnn(C)c2C)C(C)C1 n1(CC)nc(C(=O)Nc2ccc(CN3CCCC3)c(Br)c2)c2c1CCOC2 C(=O)(CC(C)(C)C#N)N(CCCNC(C(C)Sc1ncccn1)=O)C c12cc(Cl)ccc1[nH]c(=O)n2C.c1(CC)ccnc(OC)c1 C(=O)(CS(C)(=O)=O)NC(C(=O)N1CC(SC)C1)COC(=O)C(C)C C1(C(=O)NCC2CCN(C(C(COC)C)=O)C2(C)C)Cc2cccnc2C1 Cc1nc2cccc(C(=O)N(C(C)CCNC(c3cccnc3)=O)C)n2n1 CCCC(C)C(=O)NCCN(C(=O)CC1CCC(O)C1)CCOCCOC C1(C)(CCNC(c2n(C(C)C)cnc2)=O)CCN(C(=O)CCn2ccnc2)CC1 c1(CN(C(C2CCN(C(C3CCCS3)=O)C2)=O)Cc2ccc(Cl)s2)ccccc1 C1(C)(C)CC(=O)NCc2cn1nn2.C1(C)CCN1C1CC1.CC(C(=O)O)OC1CCCC1 C1(CCC)CCN(C(=O)CSC(C)(C)C)C1CC.C1(=O)CN1 C1(N(C(Cc2ncc(C)s2)=O)C)CN(C(c2ccnc(C(C)(C)C)c2)=O)CC1O C1(CC)CC(O)CN1C(=O)CN(C(=O)Cn1[nH]cnc1=N)C(C)C C(=O)(C1=CCN(C)C1)NCCC(C)NC(c1cnc(CC)o1)=O CC1=C(C(=O)N2CCCC(NC(c3ccc(CO)cc3)=O)C(F)C2)CCCO1 CC1CN(C(c2nncn2C2CC2)=O)CC1CNC(=O)C(F)=CC1CC1 Cc1nn(C2CC2)cc1C(N1CCC(CNC(C2(C(F)(F)F)CCCC2)=O)C1)=O N1(C(C(COC)NC(=O)CCN(C)C(C)=O)=O)CCC2C(=O)NCC2C1 N(C1CCCc2c[nH]nc21)C(C(CC(C)(C)NC(c1cc2n(n1)CCC2)=O)F)=O N12CCC(C(C(=O)OC)C1)C2=O.c1(CC)ccccc1-c1ccc(C)cc1 N1(CCCC)CCN(C(=O)CC2CCCN2Cc2nccc(C(F)(F)F)n2)CC1 C1(COCC(=O)N(C2CCN(C(c3cnn(C(C)(C)C)c3)=O)C2)C)CCCCO1 C=CCC(CC(C)C)C(=O)N1CCCC(CC)(NC(=O)C(O)CC2CC2)C1 n1(CC)nc(C)cc1C(=O)NCCC(C)N(C(=O)C(c1ccnn1C)O)C c1(OC)noc(C2CC2)c1C(N1CCC(NC(=O)CCn2ccnn2)CC1)=O c1(CC(N2C(CCNC(CCC3C(C)C3)=O)CCC2)=O)ccc2c(c1)CCCC2 c1(C(CNC(c2n[nH]cc2Br)=O)NC(CC=C=C)=O)ccccc1F N1(C(c2n(C)ccn2)=O)CCCC2(C1)CN(C(c1cc(Cl)ncc1F)=O)CCO2 C(=O)(C1CC=Cc2ccccc21)N(CC(O)CNC(C1(F)CCC(=O)CC1)=O)C c1(N)cccn2ccnc12.c1(C2(NC(=O)CC3(C(=O)NC=O)CC3)CC2)nccs1 c1(CC)oc(C(N2CC=CC(NC(=O)C=C(Br)Br)C2)=O)cc1C C1(CC(=O)NC(C2(C(=O)OC)CNC2)C)(CSC)CCCCC1 C1(NC(c2c(C)n[nH]c2)=O)(CNC(C2(CC3CCC3)CC2)=O)CC2CCC1C2 CC(CC(=O)NC1(CF)CCN(C(=O)CN2CCCC2=O)C1)C(F)(F)F c1(C(C)C)ccsc1C(=O)NCCCN(C(=O)CCc1ncco1)CCO C1(CCCNC(C2COC(C(F)(F)F)C2)=O)CN(C(c2sccc2Cl)=O)CCO1 c1(CC)ccc(F)c(F)c1.CC1(CO)CCCN1CCC(=O)OC CC(O)CC(C)N=c1ccnc(NCC23CCCN2CCC3)[nH]1 N1(C(C2C(O)CCN(C(c3cc(OC)c(Cl)nc3)=O)C2)=O)Cc2ccc(F)cc2C1 N1(C(C(C2CC2)OCC)=O)CCOC2(C1)CN(C(C1CC1CC1CC1)=O)C2 N1(C(c2c(CC)nc[nH]2)=O)CCCC(NC(C23CC(C2)C(C)(C)O3)=O)CC1 C12(CNC(Cc3cnc(C)[nH]3)=O)CCC(CC1)N(C(=O)Cc1cccnc1)C2 O=C(CC1NC(=O)c2ccccc21)NCC1(NC(C2CCC3C2C3(F)F)=O)CC1 C1(N(C(=O)CCNC(C2CC(C(F)F)C2)=O)C)CCN(C(=O)CC2CCCO2)CC1 C#CC1(NC(C2(C(=O)O)CC(c3cn(CCCCF)nn3)C2)=O)CCCCC1 CC1(C)CC(NC(=O)CCNS(C)(=O)=O)CN(C(=O)CCCc2nccs2)C1 Cc1cc(C(=O)N(CC(C)O)CCNC(=O)C(C)(F)F)cc([N+](=O)[O-])c1Cl c1(C(=O)NC(C(C)NC(C(CC)N2CCCC2=O)=O)(C)C)cc(OC)n(C)n1 CCN=c1[nH]c(C)c(C(=O)NCC2CC(F)(F)CN2C(=O)CC=C(Cl)Cl)s1 N1(C(c2c(N)csn2)=O)CCc2c(CNC(=O)CC3CCNC3=O)cccc2C1 c1(OC)ccc(-c2n[nH]cc2C(=O)N(CCC(C)NC(C2(F)CC2C)=O)C)cc1 Cc1ccc2c(cnn2C)c1-c1cn(C(C)C(=O)NCC2CC23CCOC3)nn1 CC1(C#N)CCC(C(=O)NCCCCNC(c2sccc2-n2cccc2)=O)CC1 CC(C)CC(=O)N(C(CC1CCNCC1)CO)CC(F)F C1(c2c(C)sc(Br)n2)NC(=S)N(CC2CC2)C2=C1C(=O)NC2c1ccccc1 Cc1cccnc1C=CC(N1CC(C(N)=O)C(n2cc(CC(C)O)nn2)C1)=O C(=O)(C(CNC(=O)CCC1CCCO1)C(C)C)N1CC=CC(OC)C1 c1(CC(=O)NC2C3CN(C(CC4CN(C)C4)=O)CC32)c[nH]c2cc(F)ccc12 c1(C(=O)NCC2N(C(C3C(C(N)=O)C3)=O)CCCCC2)cc2cccnc2o1 N1(C(c2c(C(C)(C)C)c[nH]n2)=O)CC=CC(NC(C2(O)CCOC2)=O)C1 c1(-c2ccc(OC)cc2)ccc2nnc(C(=O)Nc3cc(OC)ncc3Br)n2c1 c1(C(=O)NCC(C)(CNC(=O)CC(C)C2CCCC2)OC)cc(C(C)C)n(C)n1 C(CO)(CCCCNC(=O)C(F)=C1CCCC1)NC(=O)CCC1CCC(O)CC1 C(CC(C)C)(C(=O)N(CC(C)CO)C)N(C(C(C)=CCO)=O)C c1(OC)ccc(C)cc1CN(c1ccc(C)cc1)C(C)C CC(C)CC(O)C(=O)NCCC1(O)CCCN(C(=O)C(F)(F)COC(C)C)C1 C1(C(N2CCC(OCCNC(c3cc(C)c(C)s3)=O)C2)=O)CCCN2CCCC12 C(=O)(C(C)CC(N)=O)N(CC)CC1CCCN(C(c2csc(C#N)c2)=O)C1 C(=O)(CC(C(F)(F)F)NC(=O)C(C1CCCCC1)F)NC1(CC)CC(C)C1 c1(OC)cccc(F)c1CNC(=O)CC1CN(Cc2ncccc2OC)C1 c1(C(=O)NCC2CC(OC)CN2C(C2OCCC2C(C)C)=O)cc2occc2[nH]1 C1(CC(=O)NC(C)C)CN(C(=O)C(C)C2CCCC2)C(C)(C)C1 c1(C(CNC(c2ccncc2C)=O)NC(CCC)=O)ccccc1CC C(=O)(C#CC(C)(C)CNC(c1cnc(N)cn1)=O)NC(C(=O)OCC)CO CCCCCCC(C)C(=O)NC1CN(C(=O)C=Cc2cnc(C)s2)CC12CCC2 C1(C(N2CC3C(C2)C3(F)F)=O)CC2CCCCC2N1C(C1CC1F)=O C(=O)(CC(C)(C)CCC)NC(C1(O)CCN(C(C2(CC=C)CCOC2)=O)CC1)C CC(C(O)C(F)F)NC(=O)C(C)(C1CC1)N(C)C(C1CC(F)C1)=O N1(C(C(C)OCC)=O)CC(NC(=O)CP(C)(C)=O)C2(CCC2)C1 C1(C)(CC(=O)NCCC=CCCC)CCN1C(c1cnc(C)o1)=O C1(C(=O)NC(CNC(COc2ccc(OC)cc2)=O)C)CC2CC1CC2=O N1(C(C(C)NC(C(C)=CC2CC2)=O)=O)CCOCC(O)C1 C1(CC)CC(C(=O)NC(CN(C(=O)CN(S(C)(=O)=O)C)C)CC)C1 Cc1cc(CN=c2[nH]ccs2)cc(Br)c1.c1(CC=O)cccc(C(F)(F)F)c1 CC1(C)CC(NC(c2c(F)cccc2Cl)=O)CN(C(=O)C(C)(O)c2ccccc2)C1 Cc1cc(OC(F)F)c(-c2sc(CN)nc2C)c(-n2cc(CC(C)O)nn2)c1 N1(C(C2CCC3(CC2)CC3)C(=O)NC)Cc2cc(F)ccc2CC1C c1(N(C)C)nc(Cl)c(C(N2CCOCC2CNC(=O)CCc2cnc(O)[nH]2)=O)s1 C=CCC(C)(C)CC(=O)NCC(C)CN(C)C(C12COC(CO)(C1)C2)=O N12CCCC(C1)CN(CC1CC1)CCC2=O.c1(C(=O)Nc2cnco2)ccncc1 N1(C(=O)C=Cc2ccncc2)CCC(S(=O)(=O)CCO)C1 CC1CC(C(=O)NCC=CCNC(c2cc(-c3ccncc3)nn2C)=O)CCN1C C1(CNC(CSCC(C)C)=O)CCN(C(=O)C(F)(F)c2ccccn2)CC1(F)F c1(OC)ccccc1OCC(N1CCC(NC(c2scnc2Cl)=O)C1)=O C1(CC=C)(C(=O)NC(Cc2cc[nH]n2)C(=O)NC)CN(C(=O)C=CCOC)C1 CC1(C)C=C(C(=O)NC2CCN(C(=O)CCCCCc3cccs3)C23CC3)C1 C=CC1CCCN(C(=O)C(=O)NCC(CCOC)C2CCC2)C1 C12(C(=O)NCC(CC)NC(=O)CCC3CCC(=O)NC3)CCCN1CC(OC)C2 C1(CC)CN(C(c2cnc(Cl)c(C)c2)=O)CCN1C(=O)Cn1cccn1 C1(C(C)C)COCCN1CC12CC1CN(S(=O)(=O)Cc1ccccc1)C2 C1(CC)CCC(C(=O)N(C)CC2COCCN2C(C2CCOC2)=O)CC1 c1(C(N2C(C)(CNC(c3csc(O)n3)=O)CCC2)=O)cc2ccccc2s1 c1(CC(=O)NCC(C)N(C(c2c(COC)onc2)=O)C)cn2cc(F)ccc2n1 CCCCC(O)C(C)C(=O)NC1CC(C(N2CCC2(C)CC)=O)C1 c1(NC(C(=O)NC(C(C)NC(=O)CC(C)(C)C)C)=O)cnn2c1OCC2 C(c1c(Cl)cccc1Cl)=C(C)C(=O)N(CCCCNC(=O)Cc1cnccn1)C C1(C(=O)NC(C)CCNC(c2cccc3c2COC3)=O)CCc2ccccc2C1 c1(-n2cc(CN(C(c3cnccc3CN)=O)C)nn2)ccc(F)c(CO)c1.CO c1(CNc2ccc(CC(F)F)cn2)cccc2ncnn12 N1(C(CC(c2c(C)n[nH]c2C)C)=O)CC(NC(C2(C(C)C)CCC2)=O)C(C)(C)C1 N1(C(C2C(C(=O)OCC)CC2)=O)C(C(N2CCC(O)(C(C)C)C2)=O)CCC12CC2 c1(OCC(=O)NCC2N(C(c3nn(C)c(F)c3)=O)CC(F)C2)cccc(C#N)c1 c1(-n2cc(CN(C(c3c(C)nc(Br)s3)=O)C)nn2)cccc2ncccc12 c1(C(=O)NC2C(CNC(CC3C(C)C3)=O)C2)cn2c(n1)COCC2 N1(C(CNC(C2CC=C(C)CC2)=O)=O)CCOCC(Nc2ccc(C)c(O)c2)C1 C1(C)(C(=O)NC(C)CCCCNC(=O)CC2CC(=O)C2)CCN(C)C1=O c1(CNC(C2(CNC(C(C)OC)=O)CC2)=O)ncn(C(C)C)n1 c1(C(=O)NC2C3CC(CNC(CCC(C)C)=O)(C3)OC2)ccc2c(c1)CCO2 C1(NC(CC(=O)NCC#C)=O)CC2CCC1N(C(=O)CC(C)SC)C2 Cc1[nH]c2ccccc2c1C(=O)NC1CCC1CNC(C1CCCC1F)=O C12CN(CC3(CCC3)O1)C(=O)CNC(CCC)C(=O)NC2.C(=O)(COC)OCC c1(C(=O)NC2C(NC(C3CC(C)C3)=O)CCCC2)cc(C2CC2)nc2ccnn12 C1(C(N(C(C)COC)CC=C)=O)CCCC(NC(=O)Cc2cc[nH]n2)CC1 c1(OCc2n(C)cnn2)c(Cc2cn(-c3ncccn3)nn2)nn2c1CCC2 c1(C(=O)NCCN2CCCC(CC)C2)cc2ccc(F)cc2o1 C1(NC(C(C=C=C)C)=O)CN(C(c2cccnc2SC(F)F)=O)CC12CC2 c1(CC2C(C(=O)NCCCCNC(C3CCCCO3)=O)(CO)C2)ccc(F)cc1 C1(C(=O)NC2C(CNC(CSCCC)=O)CCC2)CCS(=O)CC1 C1(NC(=O)CC2CCC3CC3C2)CC2(C1)CN(C(=O)C=Cc1cncc(O)c1)C2 CN1CCC(NC(=O)CCC(C)(C)C#N)C12CCCN(C(=O)C1=COCCO1)C2 c1(C(N(CCOCCCNC(C(CC)(C)CO)=O)C)=O)n[nH]c2ccc(C)cc12 N1(C(C(C)CCO)=O)CCC2(CCCC2CNC(c2cccn(O)c2=O)=O)CC1 C(=O)(CC(C)P(C)(C)=O)NCCCC1N(C(c2cc(CSCC)on2)=O)CCC1 Cn1c(O)nc2c(C(=O)NC3CCC(P(C)(C)=O)C3)cccc12 Cc1nnc(NC2CCCCN(C(=O)CCCC3CCC3)C2)c(C#N)c1C C1(C(N2C(C(=O)Nc3cccc(COC)c3)CC2)=O)C2C3CCC(C3)C12 c1(SC)ccc(C(N2CCC(CCNC(C3CC3F)=O)C2)=O)o1 CCCCCCC(F)C(=O)NCC1(C)CCN(C(=O)C(c2ccc(F)cc2)O)C1 C(c1cccc(O)c1)=CC(=O)NC1CC2(C1)CN(C(C1CCCS(=O)(=O)C1)=O)C2 C1(CC(=O)NC(CCC)CO)CCCN(C(=O)C(N2CCOCC2)C)C1 O=C(CC1CC(=O)NC1)NNC(=O)N1CCC(CC2CCOC2)C1 O=C(CCC(F)(F)F)NCC1CCCCN1C(C1(C(F)(F)F)CCC1)=O Cc1cc(Br)cc(CN2CC(NC(c3cnc(O)nc3O)=O)C(F)C2)c1O C12CC(C13CCC3)n1c(C)c(cn1)NC(=O)C(=O)N2.N1(CC(C)OC)CCCC1 C1(C(=O)NC(CC=C)CNC(=O)Cc2n[nH]c(=NC)s2)CCN(C)C(=O)C1 C1(CNC(C(C(C)C)SCC)=O)CCCCCN1C(=O)C1=CCCOC1 c1(OCC)ccc(C(N2CC(NC(C3CN(C(=O)CC)C3)=O)C3CC23)=O)cn1 N1(C(CCC=CC)=O)CC2(C1)C(NC(=O)Cc1cccc(F)c1)CCS2(=O)=O N#CC1(C(N2CCC(c3nncn3C3CC3)CC2)=O)CCCC(N)C1 C1(CC=C)(NC(C2CC2(C)CC)=O)CCN(C(=O)CSc2nncn2C)C1 c1(OC)nn(C)cc1NC(N1CCCC(C(F)F)C1)=O C=CC1(C(N2CCC(NC(N)=O)C2)=O)CCN(C(C23CC2CNC3=O)=O)CC1 c1(CNC(c2c(F)ccc(F)c2Br)c2n(CC)nnn2)nnc2n1CCCCC2 c1(CC(=O)NCC2CCN(C(CC(C)C3CC3)=O)C2)ccc(-n2cnnc2)cc1 c1(C(C(=O)N(C2CCN(C(=O)CC3CCCCC3)C2)CCO)O)cc(F)cc(Cl)c1 c1(C(=O)NC(CC)(C)CCNC(=O)CCc2cncc(F)c2)cc(C)cc(Cl)c1 c1(C(=O)NC2CC(C)N(C(=O)CCc3ccn(C)c3)CC2)cnn2ncccc12 C1(CNCCNC(C(=O)OC2CCCN(C)C2)=O)CCC2(CCOCC2)CN1 Cc1ccc(C(=O)NCCNC(=O)CCC(=O)c2cccnc2)cc1C(=O)O C1(C(N2CCC(Nc3ncnc(O)c3Br)C2)=O)CC2(C1)CS(=O)(=O)C2 Cc1scc(C(N2CCC(CF)(NC(c3cccc(C(C)C)c3)=O)C2)=O)c1C C12(C(=O)NCCNC(CC(C)Oc3ccc(CO)cc3)=O)CCC(CC1F)C2 C(=O)(CCCC(C)(C)CC)N1CC(CC)N(C(=O)CCCCCC(C)O)CC1 N1(C(C(CCC)S(N)(=O)=O)=O)CC(=O)NC2CN(C(C3CC(F)(F)C3)=O)CCC12 Cc1ccc(CC(=O)NCC2CCN(C(=O)CSc3nncs3)CC2)cn1 C1(CC=C)CCN(C(=O)CC=CCNC(C2(CSC)CC2)=O)C1C Cc1ccc(C=CC(=O)NC2CCCC2NC(c2ncoc2C2CC2)=O)cc1C c1(C(=O)NC2CC(=C)C2)conc1CNC(C1CC1C1CCCO1)=O C1(C(=O)NC2(CF)CCN(C(C3CCC(C)(CC)O3)=O)C2)CC2(CCCC2)C1 c1(N(C(CC)=O)CC2CC(C=O)C2)ccc(S(=O)(=O)N(C)C)cc1.C1CN1.SCC N1(C(c2c(C)cncc2C)=O)CCC2CCC(C1)N2C(c1ccc(Cl)cc1F)=O CCCC(F)(F)C(=O)NCc1cc(C(=O)NCC(C)(O)CO)on1 c1(C(=O)NCC(CC)NC(c2[nH]c(C)nc2C)=O)nc(COC)sc1N c1(C(=O)NCCNC(c2ccc(C)s2)=O)ccc2c(c1)OCCO2 c1(C(N2CC(NC(C3CCCO3)=O)CC(C)(C)C2)=O)ccc2c(O)n[nH]c2c1 C1(CCNC(C(C)OCC(C)C)=O)CN(C(C2(N(C)C)CC2)=O)CCS1(=O)=O C=CCC(C)(C)CC(=O)NC1CCN(C(=O)CCCc2ccc(Cl)cc2)CC1F Cc1ccc(C(c2ccccc2)NC(=O)CC2CCCNC2)nc1C1CC1 c1(OC)ccc(CCS(N2CCC(COc3ccccc3)C2)(=O)=O)cc1O c1(C(N2C(CNC(c3c(C)cn(C)n3)=O)CC3(CC3)C2)=O)ccc2cccnn12 c1(NC(C2C(NC(c3cn(C)cc3C(F)(F)F)=O)C2)=O)cc(Cl)c(Cl)cc1I CCC(CC)(C(=O)NC1(NC(=O)CC2(CNC(C)=O)CC2)CCOC1)OC C1(NC(c2c(CC)n(C)nn2)=O)CN(C(c2ccc(C)cc2O)=O)C2(CCC2)C1 c1(C(=O)NCCN2CCCC(CO)C2)cc2ccccc2c(I)c1O Cc1cc(C(N2CCN(C(c3c(C)ncn3C)=O)CC2C)=O)c(O)c(C)c1 C(=O)(C1=CC2(CN(C(C3CCC(F)C3)=O)C2)OC1)NCCc1n(C)cnc1 C(=O)(CC(C)CC(C)C)NCCC1N(C(CCCc2nnc(C)n2C)=O)CCC1 C(C(CCC)C(=O)NCCCOCCOC)NC(c1n(C=C)nnc1)=O N1(Cc2cccc(OCC)c2)CC2OCCN(C(C3CCC(F)(F)C3)=O)C2C1 c1(C(=O)NC)ccc([N+](=O)[O-])cc1.c1(CNCCOCC(C)C)cccc(OC)c1 C1(NC(c2c(N)non2)=O)CC2CCC(C1)N2c1nnc(-c2ccccc2)o1 N1(C(=O)COc2ccccc2F)CCCN(C(C2CC2CF)=O)CC1 N1(C(C(CC#CC)C(C)C)=O)CCOCC1C1CCCO1 N1(C(C(N2CCOCC2)C)=O)CCC(CN(C(=O)COc2ccon2)C2CC2)C1 c1(C(N(C)CC2CN(C(C(c3ccccc3)OC)=O)C2)=O)cc(SC)nn1C CC1=C(C(=O)NC2CCN(C(=O)Cc3ccc(F)cn3)C(C)C2)CCS1(=O)=O CC1(C)CCCCC1C(N1CCN(C(=O)CCOCC(F)(F)F)CC1CCO)=O c1(C(C)NC(C2CCCC(C(=O)O)O2)=O)c(F)cccc1F C(=O)(C1CC(=O)Nc2cc(F)ccc21)NC1(C)CN(C(C2COC(=O)N2C)=O)C1 c1(C(=O)NCC(c2cnc[nH]2)C)cncc(CNC(C2C=CCCS2)=O)c1 c1(C(=O)NCCCCCNC(COC(CC)C)=O)cncc(C(C)=O)c1 O=C(CC(C(F)(F)F)NC(c1cc2ncccc2[nH]1)=O)N1CCC(n2cncn2)C1 c1(CCC(=O)NCC2(O)CCN(C(c3cc(F)cs3)=O)C2)ccccc1Cl C12(CNC(C3(OC)CCCC3)=O)CC(CN(C(=O)CC3CC(SC)C3)C1)C2 CC1(C)CCCC(C(=O)NCc2ccc(C(N3CC(F)(C#N)C3)=O)o2)C1 C1(NC(CCCNC(C)=O)=O)CN(C(c2scnc2Cl)=O)CC1C Cc1cc(CC(N2CCC(F)C(NC(c3cc(C(C)C)on3)=O)C2)=O)ccc1O C(=O)(C(O)C(C)(C)CC)NCC(N1CCN(C(C(CC=C)(F)F)=O)CC1)C(F)F N1(C(C(C)NC(=O)C2CC2)=O)CC(CC(=O)NCC2(F)CN(C)C2)C2(CC2)C1 c1(C(N2CCC(CNC(C3(C)CCCCC3)=O)C2)=O)cccc(C#N)c1 C1(CN(C(C(COC)O)=O)C)CN(C(=O)Cn2cnnc2O)CCO1 c1(C(N2CC(COC)(CNC(=O)C(CO)N(C)C)C2)=O)cc2n(n1)CCCO2 CC1(C(=O)NCC2(CNC(c3cc(Cl)cs3)=O)CC(F)(F)C2)COC(=O)C1 CCC(CC(=O)NC(CNC(=O)CSCC(N)=O)CO)c1ccccc1 C=CCC(CNC(c1cc(C(=O)OC)ccc1Cl)=O)C(=O)O Cc1sc(C(=O)NC2(C3CCCN3C(c3cc(O)n(C)n3)=O)CC2)nc1O Nc1ccc2nc(N3CC4CC(NC(C5CC5Cl)=O)CC4C3)sc2c1 CCCC(O)CCN=c1ccnc(N(C)Cc2ncc(-c3ccccc3)[nH]2)[nH]1 N1(C(C(CN(C(c2c(CC)cncc2)=O)C2CC2)C)=O)CCC2(CC1)CC2 Cc1cc(=O)n(C)nc1C(N1CC(Oc2ccc(Cl)c(F)c2)C1)=O C12(C(=O)NCC(CCOC)O)CC(C)(CN1C(C1CC13CCC3)=O)C2 C1(NC(C(c2scc(C)n2)C)=O)CN(C(C2CC3CCC2CC3)=O)CC12CCC2 c1(C(N2CCN(C(C(=C)Cc3ccccc3)=O)CC2)=O)cc(OC)cc(F)c1 O(NC(=O)C(Cc1ccco1)NC(c1[nH]ccc1CSC)=O)CC(CC)C C1(NC(C2C(NC(=O)C=CCO)CCCC2)=O)CCc2nn[nH]c2C1 CCCC(CNC(c1ccnc(C)n1)=O)C(=O)N(C)CC1(OCC)CCC1 Nc1cc(C(N2CCOC(CNC(C3Cc4nncn4C3)=O)C2)=O)cnc1Cl C(=O)(C1CCCc2sccc21)NC(C(C)NC(C(C)C)=O)CO C=C(C)CCC(=O)N1CCN(CC2CCCN(C(C3CC3C(F)(F)F)=O)C2)CC1 N1(C(C=C(CNC(C(COC)N(C)C)=O)C)=O)CC2(CCC(=O)O2)C1 CC(C)P(=O)(CC(=O)NCCC1CN(C(=O)CC2CCCC2(F)F)C1)C(C)C N1(C(=O)C=Cc2ccc(F)cc2)CCC2(C1)CN(C(=O)Cn1nnc(=O)[nH]1)C2 N1(C(C=C(C)C(C)(C)C)=O)CCC(CCCCNC(=O)Cc2cccc(F)c2)CC1 c1(NC(C2CCN(C(C(COC)OC)=O)C2(C)C)=O)cccc2cccnc12 C=CC1CN(C(=O)C2=C(Cl)CC2)CC1NC(c1ccnc(-n2ccnc2)c1)=O C1(C(=O)NCCn2cc(C(N(C3CC3(C)C)C)=O)nn2)CCCCCN1C C1(NC(C2CC23CCC3)=O)(CO)CCCN(C(c2cnn(C3CCC3)c2)=O)C1 C1(C(=O)OC)CN(C(=O)Nc2cc(C)ccc2Br)CCC1(F)F c1(CNC(C2(C(C)(C)C)CN(C(c3cnsn3)=O)C2)=O)ccc2c(c1)C(C)CO2 N1(C(C(CSC)C)=O)CCCC2(C1)CN(C(C1(C#N)CCCOC1)=O)C2 c1(NC(C2(C(=O)NCc3ccc(S(N)(=O)=O)o3)CC2)C)nc2c(F)cccc2o1 CC(C)C(C#N)C(=O)NCCC1CN(C(=O)CCCNC(=O)C2CC2)CC1C c1(OC)ccc(CF)cc1.C1(C)(C)C(=O)NCC2C(C2(F)F)Cn2cc1nn2 Cc1ncc(C(=O)N(CCCNC(c2ccc(=O)n(C)n2)=O)CCO)c(=N)[nH]1 N1(CCCCOCCNC(C)=O)CCN(C)CC1.C12CCCN1CC(=O)NC2 Cc1cccc(CCC(C(CCCNCCCN)=O)=O)c1.C1(O)(C=O)CCCC1 CCC(C)(C#N)C(=O)N1CC2CC2(NC(=O)C(C)(C)NS(C)(=O)=O)C1 c1(C(N2CC(O)(C(C)NC(C(C)C3CCCC3)=O)C2)=O)ccc([N+](=O)[O-])cn1 Cn1cncc1C(=O)NC1(CO)CN(C(C2CCNC2=O)=O)C1 c1(C(N(CC(C)C)CC(c2cccs2)O)=O)cc(-c2cscn2)n(C)n1 C12(NC(CCSC)=O)CN(C(=O)C3=COCCO3)CC1CS(=O)(=O)C2 CCCCCC(O)C(=O)NC1CC(NC(C2(C(C)C)CCC2)=O)C1 Cc1cn2ccnc(C(=O)NCCC(C)N(C(=O)C=CCN3CCCC3)C)c2n1 C(CC(=O)NCC1COCCOC12CCC2)(C(C)(C)C)NC(=O)OC(C)(C)C N1(C(C2N(CC)CC2)=O)Cc2ccccc2C1CNC(=O)CN1CCOCC1 c1(C(N2CC(C(C)NC(C(CCC)OCC)=O)OCC2)=O)cc(Cl)c(Cl)cc1N N1(C(c2c(C)cccn2)=O)CCC(NC(c2cccs2)=O)C(C(C)C)C1 C(=O)(CC(C(F)(F)F)NC(C1C=CC1C(=O)OC)=O)N1C(CC)C(=O)NCC1 C1(NC(c2c(F)ncc(OC)c2)=O)CCCC12CN(C(=O)CCCSC)C2 c1(C(N(C2CC3CCC(C2)N3)CC(C)OC)=O)cc2cccc(Cl)c2nc1Cl O=C(CCCCN1CCCC1)NCC1CCCCN1C(=O)C=Cc1ccncc1 C1(C(N2C(C3(C(=O)NC4CC(OCC)C4)CC3)CCC2)=O)C2CC3C(C2)C13 c1(OC)cc(NC(C2CCC3(CCC3)C2)=O)c(C)cc1C c1(C(C)(C)NC2CCCN2c2nccc(N3CCSCC3)n2)ccc(C#N)cc1 N1(C(C2C(C(C)(F)F)C2)=O)CCCC1CNC(C1CC(c2ccccc2)C1)=O CC1OCCCC1C(=O)NCC1C2CC1N(C(c1cnccn1)=O)C2 N1(C(C(CC)C)=O)CCOC(CNC(=O)CC2CC3(COC3)C2)C1 C12(C(C)NC(C3CN(C(C4CC(C)OC4)=O)C3)=O)CCC(O)(CC1)CC2 c1(C(NCCCCO)=O)coc(NC(=O)CCC2CCCC2)n1.CC N1(C(c2nc(C(C)NC(C(C)SCCOC)=O)oc2)=O)CCCC2(CC1)CC2 c1(CC(=O)NCCN(C(=O)C(C)C(F)(F)F)CC(C)O)cc(O)nc(O)n1 CCCCCCCCNCC(N1CC2(C1)CN(Cc1cc(OC)c(Br)s1)C2)=O c1(C(C(=O)NCCCOCC)N(CC(C)(C)N(C)C)C)cc(C)cc2c1CCC2 N1(C(C2(Cc3cc(C(F)(F)F)ccc3F)CC2)=O)Cc2ccncc2C1 c1(C(C(=O)OC)NC(C2CCC(C(=O)OC)CC2)=O)ccc(Cl)c(C(=O)OC)c1 C(=O)(CS(=O)(=O)C(C)C)N1CC=CC(NC(c2cc(OCC)n[nH]2)=O)C1 c1(CC(=O)NC2C3CC2CN(C(=O)CC2C=CCC2)C3)ccc2c[nH]nc2c1 CS(=O)CCC(O)C(=O)NCC1CN(C(=O)CC2(C(F)F)CC2)C1 c1(C(N(C)CC2OCCN(C(C(CCC)O)=O)C2)=O)nn(C)c(=O)cc1C CN1N=C(CC(=O)NC(C)(CNCC2(C)CCOCC2)c2nn[nH]n2)CC1=O C(=O)(C#CC1CCOCC1)N1CC(N(C(COCCCOC)=O)C)OCC1 C1(C(=O)NC(C=C)(C)CC)CCC(NC(C2(C)CCCCC2)=O)CC1 Cc1ccc2c(c1)C(C(=O)NC1CC3CC1CN(C(c1cnccn1)=O)C3)CC2 C1(CC)CN(C(c2csc(O)n2)=O)CCC1NC(=O)Cc1ccc(F)cc1C N1(C(C=C(C)C)=O)CCC(N(C(=O)Cc2ccccc2CC(N)=O)CCO)CC1 c1(C(n2nc(-c3cc(Cl)ccn3)nc2-c2cnc(O)n2C)C)c(F)cccc1F C1(OC)(CNC(C2(CC(=O)NCCC3CCCC3)CCC2)=O)CCCC1.N(C)C c1(C(N(C2CCC3(CC2)CSC3)C)=O)cc(C(=O)O)ccc1P(C)(C)=O C(=O)(C(C)S(=O)(=O)Cc1cn(-c2ccsc2C(F)(F)F)nn1)N(CCCC)CC c1(CNC(CCN(CC#C)C(C2CC(C)(O)C2)=O)=O)cc(CC)on1 CC1(C)CN(C(c2cnsn2)=O)C(CNC(c2ccc(F)c(C(F)F)c2)=O)CO1 c1(C(=O)NC2CC(C)(NC(=O)Cn3cnnc3O)C2)c(F)cc(Cl)cc1F C(=O)(C(C)(C)CC(F)(F)F)NCc1c(C)ncs1.C12(CC1)CCN2 C(=O)(C(CC(=C)C)NC(=O)CC1CCCN(C)C1)NC(C=C)C C1(CC)CCN(C(=O)C=CC(C)NC(c2ncoc2C2CC2)=O)CC1 c1(C(N2CC(OCCNC(C3(CC)COC3)=O)C2)=O)cncc(Cl)n1 N1(C(c2sc(C)c(O)n2)=O)CCCC1C1CCCN1C(=O)CCCSC(C)(C)C c1(C(N2CC(NC(c3c(C)nn[nH]3)=O)(CO)C2)=O)nn(C)c(=O)c2c1CCC2 C1(NC(C(C=C)O)=O)CCC(CC(=O)Nc2cnc(SC)nc2)CC1 C12(C(=O)NCC(=O)NCC(=O)NCCCc3ccccc3O)CCCCC1C2 c1(C(=O)NCC2CC2C(=O)NC(C2COC2)C)cccs1 C(=O)(C1Cc2ccc(Cl)cc21)N1CC2C(NC(=O)CC3CC3)(C2)C1 c1(NC(N(CCC)C)=O)cnn(CCOC)c1 C1(C)(CNC(C2(F)CC(C(=O)OCC)C2)=O)CN(C(=O)C(O)C(C)CC)CC1C Cn1ncc(C(=O)NC2CCC2NC(=O)C(O)C2CCC2)c1Br N1(C(C(COC)(C)C)=O)C2CCC1(CNC(C1CCC(F)CC1)=O)CC2 C1(CNC(CC2C(C(=O)OCC)C2)=O)CC(F)CN1C(c1ccsc1C)=O Cc1nnc(O)c(C(=O)N(C)CC2(NC(=O)C(C)SC(F)(F)F)CC2)c1C c1(C(=O)NCCCN2CCN(c3cc(OC)ncn3)CC2)cccc2nccn12 C1(C)(CNC(CC=CC=C)=O)CCCN(C(C2(C)COC(=O)N2)=O)C1 C1(CC=C)(CNC(=O)C(=O)Nc2ccnn2CC2CCOC2)CCOCC1 C1(C(C)NC2CCCC2)CCC(N)C1 CCC(C#N)C(=O)NC1CC(N(C(=O)C=Cc2cnccn2)C)C1 C1(N(CC(=O)NC)C)C2CN(C(C3(N)CCC3)=O)CC12 c1(C(=O)NCC(C)CNC(C2(O)CC2(C)C)=O)ccccc1N(C)C c1(C(=O)NC2(C)CC(NC(c3c(C)cn[nH]3)=O)C2)nc2n(c1Br)CCC2 C(=O)(C1CCCc2nc[nH]c21)NCC(CNC(=O)CC(c1cccc(F)c1)O)O N1(C(c2cccc(N(C)C)n2)=O)CC(NC(C2(CCF)CCC2)=O)C(C2CC2)C1 C1(C(=O)NCCC(=O)OC)CCC=CC1NC(=O)CC=O N1(C(C2C(N(C)C)CC2)=O)CCCN(C(C2CC3C=CC2CC3)=O)CC1 N1(C(C(CC2CC2)OC)=O)CCCCC(NC(c2ccc(CNC(C)=O)o2)=O)C1 C1(CN2CCN(C(=O)NCc3ncc(Cl)s3)CC2)CCOC12CCCCC2 CC1CCN(C(=O)CN(C)CC2CC2)C1NC(=O)CC1CN(C)C1 C(=O)(C1CCCc2sccc21)N1CC(C)(NC(c2onc(C)n2)=O)C1 CC1CC(c2ccccc2)CN(C(C2CCCN(Cc3nccn3C)C2)=O)C1 C(=O)(CC(O)CC(C)C)Nc1ccc(C(=O)NC(CCC)C(F)(F)F)cn1 Cc1cc(CC(=O)NCC=CC(=O)NC2CC(CO)C2(C)C)nn1C C(=O)(C(F)(CNC(C1C2(CC2)C12CC2)=O)C(C)C)N(C)Cc1ccn(CC)n1 C1(NC(c2cnn(C(C)C)c2F)=O)CC2CN(C(=O)C(C)n3ccnc3)CC2C1 c1(C(N2C(CN(C(=O)CN(C)S(N)(=O)=O)C)CCC2)=O)cc2c(ncn2C)s1 Cc1ccc(CCC(=O)NC2CCN(C(=O)C=C3CC3)CC2C)cc1C C1(CNC(C(CCCOC)C)=O)CC2(CCC2)CN1C(C1CCCN1C=O)=O c1(CNC(C2(CC=C)CCCC2)=O)csc(CNC(C2CC23CC3)=O)n1 c1(C(=O)NC2CC(NC(C(C)NC(c3ccc(F)cc3)=O)=O)C2)cn2ccnc2s1 C(=O)(N1OC2C=CC1CC2)c1sc2ccccc2c1Br.O=C1CN1 N1(C(CN(CC(C)(C)C)C)=O)CCC(C2CC2NC(=O)Cc2csc(S)n2)CC1 c1(CCN2CCCC(CNC(C3(C)CCOCC3)=O)C2)c[nH]c2ccccc12 c1(C(=O)NCCC(C)CCNC(=O)C=Cc2ccco2)cc2c(s1)CC(C)(C)C2 N1(C(c2ccc(C)s2)=O)CCC(C)(CCNC(C23CC(CF)(CO2)C3)=O)C1 Cc1oc(C(C)C)cc1C(N1CCC(CNC(=O)C(C)c2ccsc2)C1)=O C(=O)(CCC(=O)NC(C(C)NC(c1cc(OC)ncn1)=O)C(C)C)NCCC Cc1noc(NC(C2CN(C(c3cccc(=O)n3C)=O)C2)=O)c1C#N S(=O)(=O)(CCCS(=O)(=O)NC(C1CCC(C)CC1)=O)NC1CCCOC1 N1(C(c2c(C)ocn2)=O)CC2(CCC2)CC1CNC(c1ccc(CCO)cc1)=O N1(CC)CCC(C(N2CC=CC2(C)C(N2CCOC(CC)C2)=O)=O)CC1 CC1CC(=O)N1.c1(N(CCC(N)=O)C(=O)NC2(C)CC2)ccccc1 C(=O)(C1=C(C)Oc2ccccc2C1)N1C(CNC(C(CC)(C)C(N)=O)=O)CCC1 C(=O)(CC(CN(C)C)C(F)F)N(C1(CCOC)CC1)C.C1C(=O)N1 C(CC(CC)C(=O)N1CC=CCC1C(=O)NCCC1CCC(C)C1)=CC C(C(=O)Nc1ccsc1CNC(c1cccc(CO)c1)=O)(C(C)(C)C)N(C)C N1(C(=O)C2=C(Cl)CC2)CCCC(C2CN(C(=O)COCCO)C2)C1 c1(CC(=O)NCCN(C(c2cnc(C3CC3)[nH]2)=O)C2CC2)ccc(F)cc1 N1(CCC)C(=O)CCC1C(=O)N(C)CC1CCCCN1C(c1coc(CO)c1)=O C1(CC)CCN(C(c2ccn(CCF)n2)=O)C1C(=O)NCC=CCOC N1(C(COCCCC#C)=O)CCC2CCN(C(=O)CCCCCCCOC)CC2C1 C1(NC(C2(C)CCNC2=O)=O)C2CC3CN(C(c4cc5occc5s4)=O)C1C3C2 CC1CN(C(C2(C(F)F)CC3(CC3)C2)=O)CC(CCNC(C2CC(O)C2)=O)O1 c1(CCC)cc(C(N2CC(CNC(=O)CCc3nncn3C)CC2C)=O)n(C)n1 c1(C(=O)NCC(c2ccc(F)cc2)NC(CCOC)=O)cncc(C(F)(F)F)c1 C(CC(F)F)(C(=O)NC(C)CN1CCOCC1)NC(Cc1c(C)nccc1)=O C(C)(c1ccccc1C)=CC(=O)NC1CC2CC(NC(C=C(CCC)C)=O)C1C2 N1(C(COCC(=O)OC)=O)CCN(C2CCN(C(=O)CCCN(C)C)CC2)CC1 c1(C(N2CC(CNC(C(CC)(C)F)=O)OCC2)=O)ccc([N+](=O)[O-])cc1Cl C1(C(N2CCCC(CCNC(C(C)=C(C)C)=O)CC2)=O)CC2CSCC(C1)C2 C(CC1CC1)(C(=O)NCCC1COCC1O)N(C(=O)COC(F)F)C.C1CC1 C=CCN=C(NCCCC1(C)OCCO1)N1CCC2(OC)CCCCC2(OC)C1 c1(NC2CCC(CNC(=O)Nc3ncc(Br)cc3Cl)C2)c(Cl)cccc1[N+](=O)[O-] C1(CC(N2CCN(C(C)=O)CC2)=O)CC2(C1)CN(C(C1CCC1(F)F)=O)C2 N1(c2n(C)c(Cc3ccccn3)nn2)Cc2cnn(C)c2CC(C)(C)C1 C(CCCCCN=[N+]=[N-])NC(CC1OCCN(C(C(C)=NOCC#N)=O)C1)=O C1(O)(C(C)NC(=O)CCc2cn[nH]c2)CCN(C(=O)C(N2CCC(O)CC2)C)C1 CCC(O)C(C)(C)C(=O)N1CCC(CNC(c2sccc2F)=O)(OC)C1 c1(CC)ncc(Cl)c(C(=O)NCC2CN(C(C)C(=O)N(C)CC)CCN2C)n1 C(=O)(C1=NOC(c2ccccc2)C1)NCCC(COCC)NC(C)=O c1(CC(C)NC(C2CC3(C2)CC3F)=O)ccccc1Br C1(OC)CCN(C(C2C=CCCN2C(=O)CC2(O)CCC2)=O)C1(C)C O=C1Cc2cc(C(N3CC(NC(c4cscn4)=O)C(F)C3)=O)c(Cl)cc2N1 N1(C(c2c(C)ccs2)=O)CCCC(CNC(c2c(C)cnn2C(C)C)=O)CC1 CCC(CC(=O)NC1CC(CNC(c2sccc2-n2ccnn2)=O)C1)C1CC1 C12(C(=O)NCCN3CC(C)OCC3)CCCC1CCN2C(c1ncn(C)n1)=O CC1N(C(=O)C(O)C2CN(C(c3ccc(F)c(O)c3)=O)C2)CCCC1(C)C CC12CC(NC(=O)CC3CCC(=O)NC3)(C1)C1(CN(C(=O)Cn3cnc(=N)[nH]3)C1)O2 C(=O)(N=c1[nH][nH]c(C)c1C)c1nc(-c2c(OC)cccc2Br)sc1 N1(C(=O)NCc2cccc(NC(C)=O)c2)CCC(C)(Cc2ncc(C)s2)CC1 C(CCOCCO)(C(=O)NCCC1CC(F)(F)C1)NC(C1CCC(F)(F)C1)=O C1(NC(C=COCC)=O)CC2CCC1(CNC(c1cnc(C3CC3)o1)=O)C2 c1(NC2N(C(CCNC(CCOCC)=O)=O)CC(OC)C2)cccc(OC)c1C c1(C(=O)NCCN(C(C2(CC#C)CCCO2)=O)CCC)ccc2nc[nH]c2c1F c1(OC)cc(OC)ccn1.N1(Cc2ccc(OC(F)F)cc2)CCNCC1CC N1(C(CN(S(C)(=O)=O)C)=O)CCN(C(=O)CCN2C(=O)CCC2=O)C2CC12 Cc1cccc(C2(NCC(N3CCC(O)C3)=O)CCC2)c1 Cc1ncnc(C)c1CC(=O)NCCN(C(=O)COC1CC1)C1CC1 C1(C2CCCCN2)(C(N(CC(C)CO)C)=O)CCOCC1 CC1(C)CN(C(=O)OC(C)(C)C)CC(C(=O)NCCn2ccc(=O)nc2Cl)O1 N1(C(C2C(C(C)C)C2)=O)CCC2CN(C(=O)CSCc3cccnc3)CC12 CC(CCC(=O)NC1CC(NC(C2CN(C)C(=O)N2)=O)C(O)C1)N(C)C C1(CC(N2CC(C(N3CCN(C)CC3CCO)=O)C2)=O)Cc2ccccc2O1 CCCCC(C)C(=O)N1CC2(C1)CN(C(c1ccc(NS(=O)(=O)CC)cc1)=O)C2 C1(C(=O)NCC(COC)NC(C2CC(O)C(F)C2)=O)CCCC12CCC2 N1(C(=O)CC2CSC2)CCCC2(C1)CN(c1ccnc3ncnn13)CCO2 Cc1cc(OC2CC2)cc(CNC(Cc2nncn2C)C(=O)O)c1 C1(C(=O)O)(NC(C2(COC)CN(C(=O)C=CC3CC3)C2)=O)CCSCC1 C(=O)(CC(C)C(C)(C)NC(c1cc(OC(C)=O)ns1)=O)N1CCN(CCCC)CC1 N1(C(CC(=O)NCC#C)=O)CC2COCCC2(NC(c2ccc(F)cc2C)=O)C1 N1(C(c2c(F)ccc(C)c2)=O)CCC2(NC(c3cc4c(s3)CCC4)=O)CCCC12 Cc1cnn(CC(C)C)c1NC(C1CN(c2ccc(NC(N)=O)cn2)C1)=O c1(C(=O)NC2C(NC(C=C(C)C(F)F)=O)CC2)ncnc2c1CCC2 C1(NC(C2CCN(C(=O)OC(C)(C)C)CC2)CC)CN2CCN1C(C)C2 CCCCC(C)CC(=O)NC1C=CC(C(=O)NC(C)CCC)C1 Cc1cn2ccc(C(N3CC(CNC(=O)Cn4nnc(=O)[nH]4)C3)=O)cc2n1 n1(C2CN(Cc3cc(C)nn3C)C2)ccc(=NC(=O)c2ccc(C(C)C)cc2)[nH]1 C=CC(C)(CC)C(=O)N1CCC(CCCCNC(c2ccc(C)nc2O)=O)CC1 C=CCCCCC(c1nnnn1CCC(=O)OCC)Nc1cccc(F)c1 C(=O)(CCCCC(F)(F)F)NCCN(C(=O)C(C(C)C)SCC)CCOC.C(C)=O C12(C(N(CCCCO)CC)=O)CCN(C(c3nc(O)sc3C)=O)CCC1C2 c1(C(=O)NC(CC)CN(C(=O)CNS(=O)(=O)N(C)C)C)cccc(Cl)c1C c1(C(N2CCC(NC(Cc3cnc(C)s3)=O)CC2C)=O)cccc2c1CNC2=O c12ccc(cc1)OC(=O)C(c1ccoc1)NCC2.C(CCOC)OC C(C1=NOC2CCCC12)NC(C(C1CN(C(CCC=C)=O)C1)O)=O C1(CC(=O)N(CCNC(c2cccc(CSC)c2)=O)CC2CC2)OCCOC1(C)C C(=O)(C(C)(C)CCF)N1CC2C(C(=O)NCCC(C)N3CCC3)(C2)C1 c1(N(CCNC(CCSCC)=O)C(=O)NC)ccccc1Cl.C12CCN1C2 C1(C(=O)NC(c2nc(C(N3CCC3CC(C)(C)C)=O)co2)C)(CO)CC=CC1 c1(OC)ccccc1-n1cnc(C(=O)NCCNC(=O)CCCC2CC2CN)c1 CC(C)(C)C(CNC(c1ncn(C(C)(C)C)n1)=O)NC(C1CC2(C1)CC2F)=O N1(C(C(c2ccc(Cl)cc2)C)=O)CC2(C1)CN(C(=O)C(C)(C)S(C)(=O)=O)CCO2 C#CC1(C(=O)N(C(C)CO)C)CCN(C(C2CCCCO2)=O)C1 c1(C(N2CC(CCCCCCNC(C(C)(CO)OC)=O)C2)=O)cnc2ccnn2c1 N1(C(C=CCOC)=O)CCC(C)C1CNC(c1csc(-c2cc(Cl)c[nH]2)n1)=O CCCCCC(CC)C(=O)NC1CCC(CNC(=O)Cc2ncsc2Cl)C1 CC1CCCC2CCCN(C(=O)NC3CC34CCOC4)C12 c1(OC)cnc(Cl)[nH]c1=NC(=O)C1CC1NS(=O)(=O)C(Cl)(Cl)Cl c1(N2CCCC(C(C)NC(C(CC=C)(C)C)=O)C2)ncnc2[nH]ccc12 C12(C(=O)NCCSCC(=O)NC(COC)CC(C)C)CCCCC1CCCC2 CCC(C)CC(C)C(=O)N1CCC(CNC(=O)C(CC)OC)(COCC)C1 CCC(CCC(=O)N(C)Cc1ccc(O)cn1)NC(c1cnnn1C)=O CCCN(OC)C(=O)CC(CCC)NC(=O)C(N)CC(C)C C(=O)(C(C)(C)C(=O)N1CCC(NC(=O)C=C2CCN(C)C2)C(O)C1)OCC Cc1c(C(N2CC(=C(F)CNC(=O)C(F)C(F)(F)F)C2)=O)oc2ccc(F)cc12 C1(F)(C(N2CCN(C(C(C)SC(C)C)=O)C(CCO)C2)=O)CCC(F)(F)CC1 Cc1n[nH]cc1CNC(c1sccc1CNC(=O)C(=O)NCC1CC1)=O C1(NC(c2nc(COCC)sc2)=O)CCN(C(C2(CC)CCC2)=O)CC12CCC2 c1(C(N(C(CC)C(=O)N2CCCC2C(N)=O)C2CCCCC2)=O)ccnc(NC)n1 C(CC(C(=O)NCc1cncnc1C)NC(=O)Cc1ccon1)=CC C1(C(N(CC(O)CF)CC)=O)CC2CN(C(c3cccn4cncc34)=O)CC2C1 Cc1nc(C(N2CCCC2C2(C(=O)NCCNC(N)=O)CC2)=O)nn1C c1(C(=O)NC(C(C)NC(c2cc(C(C)(F)F)n[nH]2)=O)C)c[nH]cc(Cl)c1=O c1(CC)ncc(C(N2CCC(NC(c3csc(Cl)n3)=O)CC2C)=O)c(C)n1 CC1CN(C(=O)NCc2ccc(F)cc2O)CCN(C)C1 N1(C(C(C)(C)C2CCCO2)=O)CCSCC1C(=O)NCCc1ccco1 C(C(CO)(CO)NC(C1OCCC1(C)C)=O)N(C(C1(CC)CC1)=O)C c1(OC)ccc2c(c1)CCC2N=c1[nH]c(=NC)[nH]c(=NCc2cc(C)ns2)[nH]1 c1(C(=O)NC23CC(NC(C4C(C)(CC)C4)=O)(C2)C3)nc2sc(C)cn2c1C C1(C(=O)NCC2CC(C)(C)OC2)CN(C(=O)CCCn2ccnc2)CC12CCC2 CC(CC(N)=O)C(=O)N1C(C(=O)NCCN2CCCNC2=O)CC2CC12 C(C)(CCCCNC(c1cccc(SC(C)(C)CC)n1)=O)NC(C=CC=CC)=O N1(C(c2cc(CC)on2)=O)CC2CC(CNC(=O)CCc3ccnc(Cl)c3)CC1C2 C1(NC(Cn2ncc(C#C)c2)=O)CC2CCC1CC2NC(c1cc(C)c(C)[nH]1)=O C(CO)(CCCNC(C1C(CN=[N+]=[N-])C1(C)C)=O)NC(C=CCC)=O c1(C(C)C)cccc(F)c1C(=O)NCCC(C)NC(c1c(Cl)cnn1C)=O N#CC1CCC(CC(=O)NC2(CNC(c3cc(C4CC4)n[nH]3)=O)CC2)C1 N1(C(c2cc(SC)c(C)o2)=O)CC(C)C(NC(=O)CC2SC(=N)NC2=O)C(C)C1 N1(CC)CCN(CC(N2CCC(C(=O)NC3CCN(C(N)=O)CC3)C2)=O)CC1 c1(C(=O)NC(CC(C)NC(c2cnc(C(N)=O)s2)=O)C)ccc(-n2cnnn2)cc1 C(=O)(C1=CC2CCCC12)NCC1CCN(C(c2c[nH]c(=NC)s2)=O)CC1 C1(C(C)C)CN(C(=O)C2=NOC(C(C)(C)C)C2)CCN1C(=O)C=Cc1cnc[nH]1 C1(NC(c2c[nH]c(=O)cn2)=O)CC2CCC(C1F)N2C(C1CCC=CCCC1)=O N1(CC(=O)NC(CNC(C(CC)F)=O)(C)C2CC2)CCN(C)CC1 c1(C(N(C2CCN(C(C3CC3F)=O)C2)CCC)=O)cc2c(nn1)OCCS2 c1(OC(C)C)nc(N2CCC(O)C(C(=O)NC3CC3)C2)ncc1Br.C12CN(C1)C2 C=CCC(C)(C)CCN(C(=O)C(c1cccs1)NC(C)=O)C Cc1ccc(C(=O)OCC2CC=CCC2)nn1 C1(C(N2CCN(C(C)=O)C3C2C3)=O)CC2(CCCCC2)C1 Cn1c(C(=O)NC2CC(NC(C3(CO)CCCO3)=O)C2)cnc1S CC(O)C(C(=O)NC1CCC1)NC(C1CC1C(F)F)=O c1(C(=O)NC2(C(=O)NC3C(C)CCC3)CCCC2)cc(Cl)ccn1 C1(C(=O)Nc2ccc(Cl)s2)CSCCN1C(=O)NC1(c2cccnc2)CC1 c1(C(N(CCCNC(C2CC2c2ccccc2)=O)C)=O)c[nH]c2cccc(Cl)c12 C(=O)(C1=CNS(=O)(=O)N=C1C)N(CC(C)O)CCNC(C(C)OCC)=O C1(CCCN(C(C2C(C)(C)C2C#N)=O)CCCC(O)C(N)=O)CC(=O)CC(=O)C1 C1(NC(CCCc2n(C)cnn2)=O)CN(C(C2(c3ccnn3C)CC2)=O)CC1F Cc1ccc(C(=O)NC2CCN(C(c3cc(O)nc(Cl)n3)=O)CC2F)c(C)c1 c1(C(=O)NC(CC(C)C)(C)CNC(C2CC=CCO2)=O)ccc2cncn2c1 O=C(C1=Cc2ccccc2C1O)NC1C=CCN(C(c2csc(Cl)c2)=O)C1 N1(C(CN2CCC(OC)C2)=O)CC2(C(=O)NCCCCCCOC)CC1CO2 N1(C(CSCC(C)C)=O)CCCC(CN(C)C(c2cc(C(N)=O)cn2C)=O)C1 c1(C(=O)NCC(CN(C(=O)CC2CCC(C#N)C2)C)(C)C)cn(C)nc1Br Cc1cc(C(=O)NC2CC(O)CN(C(c3ccccc3C(C)C)=O)C2)cc(C)c1 N1(C(C2CN(C)C(=O)C2)=O)CC2(C=C(C(=O)N3CCCOCC3)CO2)C1 C1(c2ccc(NCC3(CC(N)=O)CC3)cc2)CCc2ccccc2C1 C1(CC(=O)NC(C)CC2CCC2)CCCCN(C(C2(C#N)CCCO2)=O)C1 c1(CC(=O)NC(C2CCN(C(c3ccc(C(N)=O)[nH]3)=O)C2)C)nnc2n1CCCC2 c1(N2CCC(C=C)(CCO)CC2)nc2ccsc2c(=NCC2(CC)CCCC2)[nH]1 c1(C(N2CCC(C)(NC(CS(=O)(=O)N(C)C)=O)C2)=O)ccc2c[nH]nc2n1 c1(NCC(N2CCOCC(CNC(C(CC)(C)O)=O)C2)=O)c(C)cc(C)cc1C c1(C(N2C(CCNC(C(C)(C)F)=O)CCC2)=O)cnc2cc[nH]c2c1 CCCC(O)CC(=O)NCC12CC(CNC(c3n[nH]c(C)c3Cl)=O)(CO1)C2 CCN=C(NCc1cccc(N(C)CS(C)(=O)=O)c1)N1CCC(O)C1 C(CCC(C)NC(Cc1ccc(C(C)(C)C)s1)=O)OCC c1(CC)cc(C(=O)N(CC)CC2CCN2C(=O)CC2CCCO2)ns1 C1(CNC(C(CC)(C)OC)=O)N(C(=O)CCCOC(C)C)CCCC1(C)C C=Cn1nncc1C(=O)NC(COC(C)C)C(=O)N(C)CC1COCCO1 N#CC1CCCC(C(N2CC(CC(F)C(=O)NCC(C)(C)NC=O)C2)=O)C1 CN1CCC(C(=O)NC2CC(N3CCC3)C2)CC1.N1(CC)CC(CO)CC1=O c1(N(C)Cc2nnnn2C2COC2)ccc2oc(Cl)cc2c1 Cc1ccc2c(c1)ncn2CC(=O)NCC(C)NC(=O)CC(O)C1=CCCCC1 Cc1cc(C(N2CCCC2(C)CNC(=O)CCC2CC3CCC2C3)=O)c(C)s1 N1(C(C(=Cc2cn[nH]c2)C)=O)CCOC(CNC(C2(C(C)(F)F)CC2)=O)C1 C(=O)(CS(=O)(=O)C1CC1)N1CCCCC(N(C(C(C2CCOCC2)C)=O)C)C1 C(CNC(=O)C=CC1CCC1)(CC(F)(F)F)NC(C(C1CC1)OC)=O c1(CCN(CC(=O)OC)CC(C)N)cc(Br)sc1Br C1(NC(c2c(COC)scc2)=O)CC2CCC(C1F)N2C(=O)Cc1cc(C)on1 c1(CC(=O)NCC(CN(C)C(C2C=CCS2)=O)O)cncnc1O N1(C(CCN(C(c2nc(C(C)C)oc2)=O)C)=O)CCC(C2CC2)C1 C1(C)(C(=O)NC2CCCN(C(c3c(C)cncc3)=O)C2)C(C)(C)C1(C)C c1(CC)nc(C)c(CC(=O)NC(C)CCCNC(=O)C(C)CO)c(C)n1 C1(CC(=O)NC(C2CCN(C(=O)NCC)CC2)C)CC(O)C12CCC2 O=Cc1cccc(-c2nc(-c3ccccc3)nn2CC2CCC2)c1Br C1(CC)OCCC1C(=O)NC(CO)C(=O)N(CC1(CO)CC1)CC CCCC(C(=O)OC)C(=O)NCC(C(C)C)NC(=O)C(C)Oc1cccc(Cl)c1 c1(C(=O)NC(C2(O)CCN(C(=O)C=Cc3cocn3)C2)C)nc(O)nc(O)c1F CCCCCCCCOCCN(C(C1(NC(=O)CNC(=O)C2CC2)CC1)=O)C C1(NC(c2c(C)nccc2)=O)CN(C(=O)CCc2ccncc2)C2CCCCC12 CC(C)CC(C(=O)NCCC1CC(NC(C2(CF)CC2(F)F)=O)C1)C(C)C c1(C2(Nc3nc(CO)cs3)CCN(C(C)C)C2)cc(Br)ccc1F C(=O)(CC(O)C(C)C)N1CCC(OCCNC(c2nc(C)c(C)s2)=O)CC1 N1(C(C2CC(C)=C(C)CC2)=O)CC2(CCCC2NC(=O)COCC2CCCC2)C1 N1(C(c2ccc3c(c2)CCC3)=O)CCC2(CC1)CCN2C(c1ccccc1F)=O CCC(O)C(C)(C)C(=O)N(CCCNC(c1cc(-c2cccnc2)on1)=O)C c1(C(=O)NC2C=CC(CC(N3CCC(OC)C3)=O)C2)nccc(C)c1N CCC1(CNC(=O)N(C(C)CN(C)C)CC)OCCc2ccccc21 C=CCC(C(=O)N1CC(C(O)C(N2CCCC(OCC)C2)=O)C1)OC N1(C(C(CC)(CC)OC)=O)CC(NC(=O)CCCCCOC)C(C2CC2)C1 Cc1cccc(CN2CCC2)c1.C1(CCC(=O)OC)CCCN1C.c1(S)ccccc1 N1(C(c2c(C)noc2)=O)CC2CC1CN(C(=O)C(C(C)C)n1ccnc1)C2 C(CCC(=O)N1CC(N(C(C2CCC(=C(C)C)C2)=O)CCO)C1)N(C(C)=O)C CC(C)(CCCNC(c1sccc1F)=O)NC(=O)COc1ccccc1C(N)=O c1(CC)nsc(CNC(=O)C(C)CN(C(=O)Cc2nc(=N)[nH][nH]2)C)n1 N#Cc1ccc(C(N2CCC2CC(=O)Nc2ccc(C3CC(=O)C3)cc2)=O)nc1 C(=O)(C1=NNC(=O)C1)NC(C(=O)NCC(CC(C)C)O)CCC1CC1 CCCCC(CN1CCCC1)N=c1nc2c(ncn2C)c(NCCCC2CC2)[nH]1 c1(C(=O)NCC(CNC(c2ccccc2F)=O)OC)cc(S(N)(=O)=O)oc1C C(=O)(C(C)(C)C(=O)NCC1CC(C)(C)CN1C(=O)C(CC(C)C)N(C)C)NC CN1C(=O)C2CN(C(=O)CCn3cc(C4CCCCCC4)nn3)CC2C1=O Cn1nnc2cc(C(=O)NC3CCC3NC(C3CC(C4CC4)=NO3)=O)sc12 C1(COC)(NC(c2cc(Cl)cnn2)=O)CCN(C(=O)CCCc2ccccn2)C1 C(=O)(C(=O)CCC(C)C)NC1C(CC)CN(C(=O)COC2CCOCC2)CC1 C1(CC)CN(C(c2cc(C)ccc2I)=O)CCN1C(c1cnc(Cl)s1)=O C1(NC(C(C)NC(=O)OC)=O)CC(C)(NC(=O)C(c2ccccc2)C)C1 c1(C(CNC(=O)C(O)C(F)F)NC(c2c(C)n[nH]c2)=O)ccc2ccccc2c1 C(CCN1C(C)C(CCCc2ccccc2)C(=O)C1)N(C(CC(=O)OC)=O)C c1(N(C)C)cc(Br)ccc1CN1CC2CC1CN2C(c1ccnn1C(C)(C)C)=O C#Cc1ccc(OC)c(C(=O)NC2COCC2NC(c2conc2C2CC2)=O)c1 C1(C(=O)NCCC(=O)NCC(CN(C)C(=O)Nc2cncnc2)O)CCOCC1 C1(NC(CN(C(=O)COC)CC)=O)CCC12CCOCC2 C#CCCCCC(=O)NC(c1cn(C)nn1)C(N1CCC(C)(O)C1)=O C1(C(F)(F)C(=O)NC2CC(NC(=O)Cc3cnsc3)C2)(OC)CCOCC1 C1(CC(=O)NCC2CSC2)C(NC(c2snnc2C2CC2)=O)CC1O C12(CNC(c3cnn(C)c3Cl)=O)CC(C1)C(NC(=O)C(O)c1ccsc1)CO2 CN=c1[nH]cc(C(=O)NC(CCOCC)C(=O)N2CCC(C3CCCO3)C2)o1 Cc1cc(C(=O)NCC(C)(CO)NC(C2CC(n3cccn3)C2)=O)ncc1F c1(C(C(N2CC(OCC)(CNC(c3cc(F)c[nH]3)=O)C2)=O)(F)F)cccc(C)n1 c1(C(N2CC(NC(C3(O)CCOCC3)=O)CC(O)C2)=O)cccc2ccccc12 C(=O)(C(C)CC(=O)OC)NCCCN(C(c1ccc(Cl)o1)=O)CC Cc1nc(S)sc1CC(=O)NC(C)(C)CNC(c1ncccc1Cl)=O N(C1CN(C(C2(F)CC2C)=O)CCc2ccccc21)C(c1cc(SC)nn1C)=O C1(OC(C)C)CC(C(=O)NCCOCCCNC(=O)COC(F)F)C1 N(C1CN(C(=O)CSC2CC2)Cc2ccccc21)C(C1(C(C)C)CCCCC1)=O c1(NC(=O)NC2CC(SCCCOC)C2)c(C)nn(-c2ccc(F)cc2Cl)c1C C(c1cnc(C)nc1O)=CC(=O)NC1CCN(C(c2cn(CC)nn2)=O)C12CC2 C(=O)(C(=O)N=S(C)(C)=O)NC1C(C)N(C(=O)CCC(C)(C)F)CC1 c1(OC)ncc(F)cc1C(=O)NC(C)(C)CNC(=O)C(C)c1ccon1 CN1OCCC1C(=O)NC1COCC1CNC(=O)C(C)(C)n1cncn1 c1(C(N(CCNC(=O)CCc2cccnc2Cl)CC)=O)c(C)cccc1C c1(C(C)C)ccc(C(=O)NCc2cc(C(N3CCCC3CO)=O)on2)s1 C1(N(C)C(c2coc(C(F)(F)F)c2)=O)CCCC(N(C)C(c2cnn[nH]2)=O)C1 c1(C(N2CCCN(C(C3(C)OCC(C)(C)OC3)=O)CC2)=O)cc2ccccc2o1 c1(C(N(C2C3CN(C(=O)C=CC=C(Cl)Cl)CC23)C)=O)cc2c[nH]cnc-2n1 N1(C(CC2(C)CCC2)=O)CCC(O)(CCNC(c2ccc(F)cc2)=O)C1 C1(NC(c2scc(OC)c2)=O)CCOCC1C(=O)NC1(CCO)CCCCC1 C(=O)(C1=CS(=O)CCC1)NC1CC(C)(NC(CN2CC(C)(OC)C2)=O)C1 CCCCC(=O)C(=O)N1CC(CC(=O)Nc2ccc[n+]([O-])c2)C(C)C1 CC1CC(C(F)(F)F)CN1C(=O)C#CCNC(c1cc(=N)[nH][nH]1)=O Cc1nn(C)cc1C(=O)N(C1CC2CNC1C2)CCc1nc(=N)[nH][nH]1 c1(CCC=C)ccc(C(=O)NCC(C)(O)CNC(C2CCCOC2)=O)cc1 C1(C(=O)NCc2ccc(OC)s2)C2CN(C(C3C4CCC3(C(=O)OC)C4)=O)CC12 CCC(C)(CO)C(=O)NCC1CCN(C(c2cc(O)ccc2C(C)C)=O)C1(C)C C(CCO)N(CCN(S(C)(=O)=O)C1CC1)NC1CC1.CC1CC1 c1(C(=O)NCC2(OC)CN(c3ncc(C#N)cc3C)C2)sc2nccn2c1C N1(C(C(CCOC)C)=O)CCC(C2(NC(=O)CSCC(C)C)CC2)C1 c1(C(=O)NC(C)CN(C)C(C2(Cl)CC2(F)F)=O)ccc2c(c1)CCCC2 c1(CNC(C(C2CCCOC2)OC)=O)cccn1C(c1ccncc1)C C(=O)(C(C#N)(CC)CC)N1CCN(C2CCN(C(C(C(=C)Cl)(C)C)=O)C2)CC1 Cn1nc(CNC(=O)NCC(C)(Cn2cccn2)SC(F)(F)F)cc1O CC1=C(C(=O)NC2C=CCC(C(=O)NCCC3CC4CCC3O4)C2)CCC1 C(CC(N)=O)(C(=O)NCCc1cc(C)n(C)n1)NC(CCC=C=C)=O c1(CC(=O)NCCC2(OC)CN(C(C3(C(C)(F)F)CC3)=O)C2)cccnc1F O(NC(=O)CCCC(C)(C)Nc1cnc(OCC)cn1)CC.N12CCC(C1)C2 C(CN=C(NCC(=O)NC(c1ccc(F)cc1Cl)C)NC1CC=CCC1)SC c1(C(N(CC(C)C)CC(=O)NCC(C)C(F)F)=O)ncccc1O c1(C(=O)NC2C(NC(C3CC(=C)C3)=O)CCOC2)cc(=N)[nH]c(Cl)n1 c1(C(=O)NC2CCCC2NC(c2ncc(Cl)s2)=O)cnc2[nH]cnc2c1 Cc1cc(C(N2CCC(c3ccon3)C2)C(=O)NC2(C)CC2)cs1 c1(CC)cc(C(=O)NCC(C)CN(C(=O)CC(C)OC)C)n[nH]1 c1(C(N(CCCNC(CC(CSC)O)=O)C2CC2)=O)ccc(C#N)c(C)n1 Cc1c(C(=O)NC(C)(CNC(=O)CSCC#N)C(C)C)cnn1CCC(C)C N1(C(C2C(CNC(C(C)n3ccnn3)=O)CC2)=O)CCN(C(C)(C)C)CC1 N1(C(CC=C(C)C)=O)C(C(=O)N(C)Cc2ncc(C)o2)CC2CCCC12 c1(C(=O)NC(C2CCCN(C(c3cc(F)n[nH]3)=O)C2)C)ccc2nsnc2c1 C(=O)(CS(=O)CCC(F)(F)F)NC(C(C)NC(C1(C(N)=O)CC1)=O)CO C1(NC(C=NOC)=O)CCC2(CCCN2C(c2cccn(C)c2=O)=O)CC1 N1(C(c2c(CC)c[nH]n2)=O)CCCC2(C1)CN(C(=O)CN1OC(C)(C)CC1=O)C2 C#Cc1cccc(NC(=O)C(C)NC(=O)CCC(C)SCC)c1 N1(C(C(c2n(C)ccc2)=O)=O)CCOC2(CCN(C(C3CC(F)(F)C3)=O)C2)C1 c1(C(=O)OC)cc(NC(=O)C(=O)Nc2ccc(SCC(C)C)cc2)c(C)cc1F c1(C(=O)NC(CN(C(CC(c2ccc(F)cc2)C)=O)C)C)ccc2ncnn2c1 c1(NC(=O)NCC(c2c(C)cncc2)C)cc(Br)cc(N)c1C Cc1ncc(C(=O)NC(C)C(=O)NC(C(O)CO)C2CC2)c(C)n1 c1(OC)cc(Cl)c(I)cc1N(C1CCNCCC1C)C(=O)CCN1CCOCC1 c1(C(=O)NC2(C(F)F)CC(NC(C(C)Cc3ccco3)=O)C2)ccsc1C#N CC1C(NC(c2ccc([N+](=O)[O-])s2)=O)C(C)CCN1C(=O)Cn1cccc1 CC1(C)COC(NC(=O)COC(=O)CCCn2cc(C3CC(F)(F)CNC3)nn2)C1 N1(CCNC(=O)C(N2CCCCC2n2cncn2)=O)CCN(C2CCOC2)CC1 C(=O)(CC(F)(F)C(C)C)N(C1C2CN(C(C=CC=CCC)=O)CC21)C C1(NC(C(CC)(F)F)=O)CCC2CC1CN2C(=O)C=Cc1ccccn1 CC1CN(C(c2cc(C(C)(F)F)n[nH]2)=O)CCCN1C(C1CCCN(C)C1)=O C(CC1=CCOCC1)NC(C1N(C(CC2N(CC)C(=O)CC2)=O)CC(C)C1)=O c1(N(C)CC2CC(=C)C2)nnc(CC2CC2)n1CCCCCC CC1(CNC(C2(C(F)(F)F)CC(=O)C2)=O)CCCN1C(c1cccc(CO)c1)=O C1(CC(=O)NC23CC(NC(C=C(C)C=O)=O)(C2)C3)C=CS(=O)(=O)C1.C1(SCC)CC1 c1(C(N(CC)CC)=O)ccc(C(=O)NCC2CCC2NC(C2CC2(C)C)=O)cc1 C1(C(N2C(CN(C(CSCC=C)=O)C)CCC2)=O)CCc2ncccc2C1 C(=O)(C(C)(C)C)NC1C(C(=O)OCC(N2C(CC)CC2)=O)CCC1 C1(CCNC(C2(C(CC)=O)CC2)=O)C(C)CCCN1C(c1coc(O)n1)=O c1(CCS(=O)(=O)CNC2(CO)C(C)(C)CC2)c(Cl)cccc1[N+](=O)[O-] c1cn(C2CCN(C(=O)C(C)(C)c3ccnn3C)C2)nn1.C(C)(C)NC(C)=O c1(C(=O)NC(CCCCNC(c2c(NC)cccc2)=O)C)cc2n(c1)CCC2 n1(CC(=O)OC)cc(CNC(c2coc(C)c2)=O)nn1.c12ccsc1CNC2=O c1(NCCC(C)(C)NC(C2N(C)CCOC2)=O)ncnc2c1COC2 N1(C(CC(C)CF)=O)CC(F)(F)CC1CNC(c1cc2n(c1)CCC2)=O c1(C(N(C)CC2(NC(=O)Cc3c[nH]ccc3=O)CC2)=O)cc2c(Br)cccc2[nH]1 N1(C(CNS(SC)(=O)=O)=O)CCCC2(C(=O)Nc3cccc4[nH]ncc34)CCCC12 CC(N=c1cc2n([nH]1)CCNC2=O)c1cnc[nH]1 C1(CNC(=O)C(c2ccccc2)=O)C=CCN(C(=O)CNc2ccc(O)cc2)C1 Cc1cc([N+](=O)[O-])ncc1C(=O)NCC1CN(C(c2ccc[nH]2)=O)C2CCN1C2 C1(C(N2CC(C)N(C(C34CCC(C3)C4)=O)CC2)=O)COc2ccc(Cl)cc2C1 C(C1=CCN(C(c2scnc2Cl)=O)CC1)NC(C1C(C)C1C)=O c1(C(=O)NC2CN(C(C(C=C=C)C)=O)C(CO)C2)c[nH]c(=N)nc1CC C12(NC(CCCc3ccc(C)cc3)=O)CCCCC1CN(C(c1cnc[nH]1)=O)C2 c1(C(=O)NC(C)CCCNC(=O)C(F)(F)C2CCOCC2)cnc2sccn12 N1(C(c2cc(C#C)cc(Br)c2)=O)CCC2CN(C(=O)CCC(F)F)CCC12 C1(NC(c2ccc(Cl)s2)=O)CC2CCC1N(C(c1ncc(F)cn1)=O)C2 C1(NC(c2n(C)ncc2Br)=O)CCCCCN(C(=O)CC2COC(=O)C2)C1 N1(C(C(c2cccc(O)c2)C)=O)CC2CCC(C1)N2C(C1CCC2(CCC2)C1)=O c1(NC(COCCOCCOCC#C)=O)c(O)cccc1Cl Cc1c(C(=O)NC2CC(C)(CNC(=O)CCCCN(C)C)C2)cccc1O C#CCCCCCC(=O)NC1(C)CCC(NC(=O)C(C)CO)CC1 C1(C)(C(=O)NC2CN(C(CC(C)CN(C)C)=O)C(C)(C)C2)CC2(CC(O)C2)C1 C1(N(C(c2cnc(C(C)C)[nH]2)=O)C)CCCC(NC(=O)C=CSc2nc[nH]n2)C1 CC(C)(C)C(O)C(=O)NC1CC(NC(c2cc(C(N)=O)cs2)=O)CC1O C(CC(CC)C(=O)N1CC(C(=O)NOCC(C)(C)C)CC(C)C1)=CC N1(C(C2C(O)CCN2C(C2CC2c2ccc(F)cc2)=O)=O)CC2CCCCC2C1 C12(NC(C(C(C)C)Oc3cccc(Cl)c3)=O)CCCC1CN(C(c1ncc[nH]1)=O)C2 c1(C(N(C(CC)C)Cc2ccccc2)=O)cc(Br)cc([N+](=O)[O-])c1C c1(NC(C2C=CCN(C(C=C(C)C(F)F)=O)C2)=O)c(O)cccc1Cl C1(C(=O)NC2CCC(N(C)C)C2)CC(C)N(C(=O)OC(C)(C)C)C(CCC)C1 C1(NC(C23N(C(CSCC)=O)CCC2C3)=O)CCCCC1C#N C(=O)(CCC(=O)N(C)C)NC(C1CN(C(C2CCC(=O)O2)=O)C1)C C(CCSC)(C(=O)NC(C)CCC)NC(CCC#C)=O c1(C23C(C(N(CC(=O)OC(C)(C)C)C(C)C)=O)(CCC2)C3)cccnc1Cl C1(CNC(c2c(CC)c[nH]n2)=O)C2CN(C(=O)CC3CCC(=O)CC3)CC12 S(=O)(=O)(c1cc(Cl)cc(Cl)c1)NC.n1(C(C)C)nccc(N)c1=O CC(C)S(=O)(=O)CC(=O)N1CC(NC(=O)CC2CCCCC2(F)F)C(C(F)F)C1 CCC(CC1CCCC1)C(=O)N(CC(C)CNC(c1nnn(C)c1C)=O)C N12CCCC(C1)C(=O)N(c1ccccc1)CC2=O.C(=O)(CC(F)F)C(CN)=O.CC(=O)OCC C1(CNC(CN(CCC#C)C)=O)CN(C(=O)C(O)CCSC)CC1F c1(NCCC(OCC)OCC)cc([N+](=O)[O-])cc(=O)n1C C(=O)(C(F)(F)CC(C)C)N1CC(OC)(CNC(c2ccc(CO)cc2)=O)C1 N1(C(c2c[nH]c(=NC)c(N)c2)=O)CCCC1C1CCCN1C(C1CCC=CCC1)=O C1(C(=O)NCCCC=C)CCC(O)CN1C(c1cnc(=N)[nH]c1)=O C1(C)(C(=O)NCc2ccc(C3C(C)C3)o2)CCCN1C(c1ccsc1C#N)=O CC1CC(NC(=O)C2=NNC(=O)C2)CN(C(c2cc(=N)[nH]c(=N)[nH]2)=O)C1 c1(NC(C2C(Nc3cc(C)ncn3)C2)=O)nc(C)c(C)cc1Br N1(S(CCOCC)(=O)=O)CC2CN(C(c3cnn4c3CCCC4)=O)CC2C1 N1(C(C2C(CCC)C2)=O)CC(N(C(=O)CCOCc2ccccc2)C)C(O)C1 C1(NC(CS(=O)(=O)NCC)=O)CC2(CCN(C(=O)C(CC)N(C)C)C2)C1 C(C(CC(=O)NC1CC(C(=O)Nc2ccc3oncc3c2)C1)C(F)(F)F)N(C)C c1(C(N)=O)ccc(C(=O)N(CCNC(C2CCCC2C2CC2)=O)C2CC2)o1 C=CCC(C(=O)N(C)CCOC(=O)C(C)NC(C)=O)NC(=O)OC(C)(C)C C1(NC(C=C(CCC)C)=O)CCC(NC(=O)Cc2sccc2C)CC1 N1(C(c2c(C)ncs2)=O)CCC2CCN(C(=O)Cn3nnc4c3CCCC4)C2C1 N1(C(c2cc(C(=O)OCC)no2)=O)CCC(C)N(C(c2cn(CC)cn2)=O)CC1 c1(CC(C)NCC(c2cccc(C)c2)OC)c(F)cccc1Cl C1(C(=O)NC2CC(CNC(C(CN(C)C)(C)C)=O)C2)CCC(N=[N+]=[N-])CC1 C1(C(C)(C)C)(C=O)CCCC1.c1(NC(C2SCC(NC(C)=O)C2)=O)cnccn1 Cc1nc(O)ccc1C(=O)NC1CCN(CCNC(=O)C(C)Cn2cco2)CC1 C1(CC(=O)NCC2C(OCC)CN(C(=O)C(C(C)C)OC)C2)OCCCC1(C)C C1(C(=O)NC(CN(C(c2cccs2)=O)CC)C)CCCN1S(C)(=O)=O c1(NC(C23C(CN(C(C4(Br)CC4)=O)C2)C3)=O)cc(Cl)ccc1[N+](=O)[O-] N1(C(C2C(C)(C)COC2)=O)CC2(C=C(C(=O)NCCC34CCCC3C4)CO2)C1 C(=O)(CCCC(=O)N1CCCC1)N1CC(O)(CNC(c2cscc2C(F)F)=O)C1 N1(CCCC)CC(NC(c2cnc(-c3cccc(CC4CC4)c3)nc2)=O)C(C)C1 c1(CC)cc(C(=O)NCC2(CC)CC2)ccn1.C12CC(F)(C1)CNC2=O N1(C(CN(C)C)=O)CCOC2CN(C(=O)C=Cc3ccco3)CC12 Cc1ccc2nc(NC(C3(C)CN(C(=O)C(c4ccc(Cl)cc4)C)C3)=O)sc2c1 C1(CNC(c2ccc(Cl)s2)=O)CCCN(c2ccnc(N3CCCC3)n2)C1 Cc1cc2nccnc2cc1C(=O)NC(C)CCNC(C1CC2(CCC2)C1)=O C=CC1(C(N2CC(OC)CC2CNC(C2COCCO2)=O)=O)CCCCC1 Cc1cnc(C2=NN=C(C)C2C2CCN(C(=O)CCS(N)(=O)=O)CC2)nc1S(C)(=O)=O CCCCC(O)CC(=O)N1CC2CC2(CNC(c2ncc([N+](=O)[O-])n2C)=O)C1 c1(OCC)ccnc(CN(CC(O)CNC(CNC(C2CC3(C2)CC3F)=O)=O)C)n1 NS(=O)(=O)c1ccc(C(N2CCOCC2C(=O)Nc2sncc2C#N)=O)c(Cl)c1 c1(CCC)cc(C(=O)NC(C)CC2CN(C(=O)CC3CC3C)C2)n[nH]1 N(C1CCCOc2ccc(F)cc21)C1(c2n(CCCC)nnn2)CCOCC1F C1(NC(c2sc(OC)c(Br)c2)=O)CN(C(c2cc[nH]n2)=O)CCC12CCC2 c1(C(N(C2CCN(c3cc(CC)cnn3)C2)CCC)=O)ccc2c(c1)OCO2 CC1CC(C)(NC(=O)C(c2ccco2)NC(C2CNC(=O)N2)=O)C1 c1(OCC=C)ccc(Cl)c(C(=O)NC(CNC(C2CC2C#N)=O)CC(C)C)n1 C12(CO)CCC(CC1)NC(=O)NC2.C(CCCCCc1ccccc1)OC C1(C(N2CCC(N(C(C3(C)CC4CC4C3)=O)CC)CC2)=O)CCCC1C1CC1 c1(C(C(=O)NCCCC)N(CCC)CCc2cccs2)scnc1Br c1(C(=O)NCC2N(C(C3C(C=C)CC3)=O)CC(O)C2)cc(Br)ccc1OC Cc1ccccc1CNC(c1nnnn1-c1cccc(Br)c1)CC1CCCCC1 N1(C(c2cc(C3CC3)on2)C(=O)NCC2CCOCC2)CCSC2CCC12 C(=O)(CCC(CF)CF)NC(C)C=CC(=O)NCCC1CCN(C)C1 C(=O)(CCCC(F)(F)F)NC(C1CCN(Cc2nc(Cl)ccc2Cl)CC1)C CC(CC(=O)N1CC(C)(OCC(N2CCC(C3CCCO3)C2)=O)C1)OCCO c1(CC2N(Cn3cc(C(CC)(O)CC)nn3)CCC2)cn2ccsc2n1 c1(CCN(CCC)Cc2cnc(-c3ccccn3)s2)cccnc1 c1(C(=O)NCC)oc2ccccc2c1O.C1(C)(CN)CCN(C(=O)C(C)CC)C1 C(=O)(C1=CC2C=CC1C2)N1CCC(C(C(N2CC(C3CC3)(OC)C2)=O)(C)C)CC1 C#CC1CN(C(c2sccc2Cl)=O)CCN1C(c1ccc(N(C)C2CC2)cc1)=O c1(C(N2CCC(C)C(NC(=O)CSc3nnnn3C)C2)=O)ccc2nccn2c1 c1(C(N2CCOCC2)N(C(C(=O)NCCC(C)SC)=O)C)cc2ccccc2o1 CC(C(CO)NC(=O)CCSC(F)(F)F)NC(=O)CCCOc1cccnc1 N1CC2(C1)CN(C(=O)CCC#N)CCO2.C1(CCC)NC(=O)N(Cc2ccccc2)C1=O C1(NC(C(C)NC(CC)=O)=O)CC12CC(NC(c1cnn(C3COC3)c1)=O)C2 c1(C(N2CCCC(CC=C)C2)C(=O)NCC2CCCO2)nc(C)ccc1Br N1(C(C2C(OC(C)(C)C)C2)=O)CC2(C1)CN(C(=O)C1=CCCOC1)C2 c1(C(N2CC(=C)C2)=O)oc(CNC(c2ccc(CC)s2)=O)cc1C N1(C(CC=CCC)=O)CCC(F)(CNC(C2(C(C)(C)OC)CC2)=O)C1 N1(C(CC2(C=C)CC2)=O)CCN(C(=O)CCn2cc(C)cn2)C(C(C)C)C1 c1(NC(c2nnc3ccccn23)C)nccc(=NC(C)c2c(Cl)cccc2Cl)[nH]1 N1(C(C(=O)NC2(CCO)CN(C(C3C(COC)C3)=O)C2)C)CCP(C)(=O)CC1 C1(C(=O)NC2(C)CN(C(c3ccn4nccc4n3)=O)C2)CCc2nn[nH]c2C1 C1(C)(NC(C(COCC)C)=O)CCN(C(C2CCCS2)=O)CC1 C1(NC(c2cncc(C)n2)=O)CC2CCC1N(C(c1sc(CO)nc1C)=O)C2 C1(NC(c2cc(COC)no2)=O)CN(C(=O)CC2CC3(CCC3)C2)C2CCCC12 C1(n2cc(C)nn2)CC2CCC(C1)N2C(C1C2C=CC(CC2)C1C(F)F)=O C1(CC(C)NC(CCOCCCC)=O)CCN(C(=O)C(C2(O)CCCC2)F)CC1 C1(C(=O)NCCN(C(CC2CCC(OC)CC2)=O)C)C2Cc3cc(Cl)ccc3C12 c1(C(=O)NCC(=O)NCC(=O)N(C(C)CO)C)ccc(C#N)o1 N1(C(Cn2cc(C(C)OCC)nn2)=O)CC2CN(S(C)(=O)=O)CC2C1 C(C1c2ccccc2CCN1C(C1(OC)CC1)=O)NC(C1CCC(CC)O1)=O c1(C(=O)NC2CC(C)CN(C(=O)C(F)CC3CCCC3)C2)ccc(N=[N+]=[N-])cc1 C1(O)(CC(N2CC3CC(O)C2C3)=O)CCN(Cc2cc(-c3cccs3)[nH]n2)CC1 Cc1nc(O)ccc1C(=O)NCC1CCN1C(C1(CO)CC1(F)F)=O C1(CC)CCN(C(=O)CN(C)C(C)=O)C1CNC(c1cc(CC)no1)=O C1(NC(=O)Cc2ccsc2)CN(C(=O)C=CC=CCO)CC1F NS(=O)(=O)c1cc(C(N2CCCC2C(=O)NCC(O)C(F)(F)F)=O)c(Cl)cc1F N1(C(C(C)C2CCCC2)=O)CC(CC(N2CCC(C(C)(C)C)CC2)=O)C2(CC2)C1 Cn1cc(C(N2CCN(C(=O)C(C)(F)F)C3CCC23)=O)c2cccc(Cl)c12 c1(C(=O)NCC(CNC(CC(CC)CN(C)C)=O)F)ccn2cncc2c1 C1(n2ncc(C(=O)NCC3CCOC(C)C3)c2)CCN(Cc2c(C)onc2)CC1 C(C(C(C)C)NC(=O)CC1CCN(C(=O)Cc2cc[nH]c2)C1)OC(C)=O N1(C(CC=CC=C)=O)CCOC2(C1)CN(C(=O)C1=C(C)OCC1)C2 C(=O)(C1Cc2ccccc21)NCC1C(C(NOC(C=C)C)=O)C1 CC(C)C(O)C(F)(F)C(=O)N1CCC(CO)C(NC(=O)COc2cccnc2)C1 C(=O)(C(C)CC(F)(F)F)NCC(C)(C)OCCNC(Cc1c(C)cc(F)cc1)=O C1(CNC(c2c(C)c(Br)sc2)=O)CCC(C)CN1C(=O)CCC1CC1 C1(CN(C(C2CC(=C)C2)=O)C)CCCC(NC(=O)CCCc2ccc(Cl)cc2)C1 N1(C(c2c(C)ncs2)=O)CC(F)(F)CC1CNC(=O)C(C)S(N)(=O)=O n1(CC(N2CC(NC(=O)CC3CCC(O)C3)C(O)C2)=O)cnc2c1CCCC2 CC(O)(C(=O)NC1COCC1C(=O)NC1CCN(S(C)(=O)=O)C1)C(F)(F)F c1(-c2c(N(C)C)ccc(C(F)(F)F)c2)nc2cc(C3=COCCC3)cnc2[nH]1 c1(SC(C)C(N2CCC(NC(C3CC34CC(F)(F)C4)=O)C2)=O)ccc(F)c(F)c1 C1(C)(NC(C(CCC)O)=O)CCCN(C(=O)CCCOc2ccc(C)cc2)C1 C(CNC(=O)C(C)(C)C)(CC(=O)NCCc1c(N)cnn1C)OC C1(=CCNC(CCC2CC(C)C2)=O)CCN(C(C2CCC(C)CO2)=O)CC1 Cc1nc(C)n(CC(=O)NCCC2CCCN(C(C3(C#N)CCCO3)=O)C2)n1 C12(NC(C3(C(F)F)CC(=C)C3)=O)CCN(C(c3cccc(OCCC)c3)=O)CC1C2 N1(C(c2c(C#C)cn(C)n2)=O)CC2=C(C1)CN(C(=O)CCc1cc(Cl)cc(Cl)c1)C2 c1(C(N(C2CCN(C(=O)Cc3sccc3C)CC2)CC#C)=O)ccc(C)cc1Cl c1(C(N2C(C(N3CCN(C(C(C)C)=O)CC3)=O)CC2C)=O)cccc2ccnn12 C12CC3(CCN(C3)C(=O)N1)C2.C(CC(=O)OC(C)(C)C)OC(=O)OCC Cc1ccc([N+](=O)[O-])cc1C(=O)NCC(CO)NC(=O)C(C)SC(F)(F)F C(=O)(CC(C)C(F)(F)C(F)(F)F)NCC(C)(CO)NC(C(C)=C1CCC1)=O c1(COC)nn(C)cc1C(=O)NC1CCC(NC(=O)CC2CCCC(C)C2)C1 N1(C(C2CN(C(C)C)C2)=O)CCCC(C)(CNC(=O)CCCN=[N+]=[N-])C1 c1(-c2cn(CC(C)NC(=O)CC3CCOC3=O)nn2)ccc2ncsc2c1 CC(CCCC(=O)NCCCC[Si](C)(C)C)N(C)C1CC1.C(C)(C)C c1(C(=O)NC(COC)CNC(=O)CC2C(C)C2(F)F)ccc(C)cc1 c1(OC)ccc(CCC(=O)NCCCN(C(c2occc2C)=O)C(C)C)c(F)c1 Cn1cnc2c(N3CCCC(C(N4CCc5ccccc54)=O)C3)nc(Cl)nc12 C1(C)(C(N(CCCNC(C(C)OCc2c(C)cccc2)=O)C)=O)CCC12CCC2 c1(CCC(N2C3C(NC(C=CC)=O)C(C3)C2)=O)cc(Br)ccc1C C(=O)(CCC(C)(C)F)N(c1ccc(N(C)C)cc1)CCNC(C1C(C)C1C)=O C1(NC(C(N2CCCC2C2CC2)c2ncc(C)cn2)=O)CCC(F)(F)CC1.C(=O)OC C1(OCC(C(=O)Oc2ncccc2F)N(CCCCO)C(C)C)CCC(F)(F)CC1 C=CC(CC)C(=O)NC1CC(CNC(C2(CCC)CCC2)=O)CC1O C1(=O)C(CCn2ccnn2)N1.CC1(CCN(C(=O)Cn2cnnn2)C2CC2)CCC1 Cc1cncnc1C(=O)NCCC1CC(C(=O)NCCCc2nncs2)C1 c1(C(N(CC(C)(C)CNC(=O)CC2CC(=O)C2)CC)=O)cc(C)n(CC2CC2)c1C C1(OCC(=O)Nc2onc(C)n2)CCN(Cc2cn(C3CCOCC3)nn2)CC1 CC(C(=O)N1CC(CCNC(C2(Cl)CC2)=O)C1)N(C)C Cc1c(C(=O)NC2CCCN(c3cc(C(F)(F)F)ncn3)C2C)cncc1Cl CC1=C(CNC(c2cccc(C)c2)C)SCCO1 C1(N(c2ncc(-c3ccccc3)s2)CC)CCC(F)(F)CC1.c1n[nH]c(C)c1Cl c1(C(N(C)Cc2scc(C)c2)=O)cc(CNC(=O)C(F)CC2CCOC2)nn1C c1(CC)cccc2c(C(=O)NC(C)CNC(c3cc(=O)n(C)o3)=O)c[nH]c12 N1(OC)CCCN(CC(N)=O)C(=O)C1.C1CCCC1C c1(C(=O)NCC2C(CNC(CC3CC(=O)C3)=O)C2)ccc2ncc(=O)[nH]c2c1 C1(CNC(C2(CCC)CCNC2=O)=O)CN(C)CCN1C(=O)Cc1nc[nH]n1 N1(C(C=CCCC)Cc2ccccc2)CCCC(NC(C2CNC(=O)C2)=O)C1 c1(C(=O)NC2C(OC)CN(C(C(CCC)O)=O)C2)c[nH]c2ccc(Br)cc2c1=N N1(C(c2c(O)nnc(C)c2C)=O)C2CCCC1CC(NC(=O)CC1CC=CC1)C2 CC1SCCC1N=c1nc(N2Cc3nccn3CC(CO)C2)c2c([nH]1)CCS2 c1(C(=O)NCC(CO)NC(C(CC)N(C)C)=O)cc(C(=O)OC)cc([N+](=O)[O-])c1 C(CC(CNC(c1coc(-c2ccsc2)c1)=O)NC(=O)C(C)SC)OC C1(NC(C2=C(C)CCC2)=O)CCOC2(CCN(C(c3cc(CO)[nH]n3)=O)CC2)C1 N1(Cc2c(C)nc(C)nc2C)CCS(=O)(=O)C(CCNC(c2cc(C)sn2)=O)C1 c1(CC(C(=O)NC(C(=O)OC)COC(C)C)C#N)ccc(C#N)cc1 C1(NC(=O)COC2CCC2)CCN(C(C2(C(F)F)CCCC2)=O)C1 CC1CCCC(OCC(=O)NC(C)(C)CCNC(=O)CN2CCC2)C1 c1(OC)cc2nc(NCC3CCCN(Cc4ccccc4)C3)[nH]c2cc1OC n1(CC)nc(Br)nc1CNCCCc1cnc(C)o1 c1(C(N2C(CN(C(C(C)(C(C)C)OC)=O)C)CCCC2)=O)ccc2occc2n1 c1(C(=O)NCCC2(NC(C(C=C)O)=O)CC2)c(F)ccc(OC(F)F)c1F c1(C2(Cc3cccnn3)CC2)cn(CCCC(=O)NC(C)C(=O)O)nn1 c1(C(N2CC(c3c(CNC(c4ccc(OC)s4)=O)nco3)C2)=O)cnnc(C)c1 C1(CN2CCC(OC(C34CCC(CO3)C4)C)C2)COCCN1C.C1(=O)CO1 C1(C(=O)NCCC(C)C2C(CCC=C)C2)CN(C(=O)CCC)CC1(C)C c1(CCCC(=O)NC(C(C)NC(C2(CSC)CCC2)=O)CO)ccc(Cl)cc1 N1(C(C(CC=C)NC(C)=O)=O)CC2C=CC1C(C(N1CC(C(=O)OC)C1)=O)C2 N1(C(c2c(CC(=O)OC)scc2)=O)CC2CCN(C(=O)CCC(C)SC)C2C1 CCC(CCOC)C(=O)NC(CCSC)C(N1CC2(CCN2C)C1)=O Cc1ccc(NC(=O)C(C)NCc2cn(CC(c3ccccc3)O)nn2)c(Cl)c1 C1(NC(c2c[nH]c(=N)s2)=O)CCN(C(c2cc3n(c2)CCC3)=O)CC1F C12(C(=O)NCC3N(C(C4CC(N(C)CC)C4)=O)CCC3O)CCCCN1CCC2 Cc1oc(C2CC2)nc1C(=O)NC1(CO)CN(C(C2(F)CCC2)=O)C1 N1(C(c2n(CC)ncc2Cl)=O)CC2CCCC(C1)N2C(=O)C(C#N)C(C)C C1(CCNC(C2CC(=O)OC2)=O)CN(C(C2(CO)CCOCC2)=O)CCO1 C1(NC(c2cn(CC)nc2C2CC2)=O)CCN(C(c2cccc(N)c2N)=O)CC1F CCC(CC(C)C)C(=O)N1CC(NC(C2CN(CC)C2)=O)C1 CCC(C)(CC)C(=O)N1CCOC(CNC(C2(C#N)CC3(CC3)C2)=O)C1 C(C(=O)N=c1ccn(C2COC2)[nH]1)Oc1c(C)cc(Cl)cc1 CC(C)C(=O)C(=O)NC1CC(C(=O)NCc2nccn2C)C1(C)C CC1CCC(=CC(=O)NCCOCCCN(C)C(c2cn(CCO)nn2)=O)C1 Cc1cc(CC(=O)NC2CC(CNC(=O)CCN3CCCC3)C(O)C2)ccc1O c1(SC)cc(O)ccc1NC(=O)CC1CCCN1C(=O)Cc1ccccc1O C(C)(C(C)C(=O)NCC(=O)OC(C)(C)C)NC(c1cc(OCC)no1)=O C1(NC(=O)C(c2ccccc2)F)CCCC(C(=O)NCC2N(C(C)C)CCC2)C1 CCCC(C)CNC(=O)CC1CCN1C(=O)C(O)C1CC1 C1(NC(N2CCN(C(c3cccnc3)=O)CC2)=O)CC2(CCC2)C1CC(=O)O Cc1nc(N2CCCC(CNC(c3ccno3)=O)CC2)c(C)c(Cl)n1 C=CCCCCCCCC(=O)NC1CN(C(=O)Cn2ncn(C)c2=O)C(C)(C)C1 N1(C(c2c(C)con2)=O)CCCC2(NC(c3c(F)ccc(O)c3F)=O)CC2C1 N1(C(C=CC(C)NC(=O)C2=C(Cl)CCOC2)=O)C2CCCC1CN(C)C2 c1(C(=O)NCC(C)(C2CC2)NC(=O)Cc2csc(S)n2)ccn2nccc2c1 c1(-c2nc(CCC(C)(C)C)nn2Cc2ccccc2)ccc(F)cc1C(F)(F)F C=CCN(OC)C(=O)C(F)CC(C)(C)NC(C1CCS(=O)CC1)=O CCC(C)(COC)CNC(=O)CC1(C)CCN(C(=O)CC2(C)CCOCC2)C1 C1(F)(C(=O)NCC(O)CC2CCCC2)CCCN(C(c2cc3n(n2)CCC3)=O)C1 N1(C(CC(C=C)CC)=O)CC(C)CN(C(c2cnn(CCC)c2)=O)CC1C Cc1ccc2oc(C(=O)NCCC3CN(C(c4ccnnc4O)=O)C3)cc2c1 CCCC(CNC(C1(C#N)CCC1)=O)C(=O)NC(C(C)C)C(C)C Cc1nn(CCO)nc1C(=O)NCCCOC1CC1(F)F.C(C)(C)(C)N c1(C(=O)NC(CCNC(c2nc(C)oc2)=O)C)cc(S(N)(=O)=O)co1 CC1C(NC(=O)C2=CCC2)CCN1C(c1cc(C2CC2)cs1)=O C12CC(=CC1O)C(=O)N2.CCCC(C)CC(=O)N1CCC(OCC)CC1 c1(C(N2CC(C)(CCC(N3C(C(N)=O)CC3)=O)C2)=O)cc2ccccc2[nH]1 N1(c2ncnc(C)c2Br)CCC2CCC(C1)N2C(=O)CC1CCOCC1(C)C C1(NC(C2CCOCC2)=O)COC2(C1)CN(C(=O)Cn1nccn1)C2 c1(NC(COc2ccc(CC)cc2)=O)ccc(NC(C2(CO)CNC2)=O)cc1F c1(CC)nnc2cc(N3CCC(NC(c4ccnc(C)n4)=O)CC3C)ncn12 C1(c2cn(C)nc2)CN(C(c2ccoc2)=O)CCN1C(c1cc(C(N)=O)co1)=O N1(C(C2CN(CC)C(=O)C2)=O)CCC(C2CC2)(NC(=O)CCOC(C)=O)C1 n1(CCOC)nc(C(N2CC(N(C(=O)Cc3nc[nH]n3)C)C(F)C2)=O)ccc1=O N1(CCSC2(C(C)(C)C)CC2)CCC2CC(O)CCC2C1 Cc1ccc(Cl)c(C(N2CCC(C(C)CNC(=O)Cc3ccnn3C)CC2)=O)c1 O=C(CCCCCn1cc(C2COCC2O)nn1)NNC(=O)CCCCC1CC1 C1(NC(C2C(C)CCCC2)=O)C2CC3C1C3C2C(=O)NC1CC1F C1(NC(c2cc(C(C)C)n[nH]2)=O)CC(NC(C2(CO)CC(F)(F)C2)=O)C12CCC2 CC(C(F)(F)C(F)(F)F)=CC(=O)NC1CCCC1N1CCN(C(C2CC2F)=O)CC1 C1(C(=O)NCC2(CCOC)CC2)CN(C(c2c[nH]nc2C)=O)CCO1 C(CN=c1[nH]nc(-c2ccco2)o1)NC.c1(NC(=O)N)ccnc(Cl)c1Cl Cc1ccc(NC(=O)CC2CC(F)CN2C(=O)C(=O)C(C)C)c(F)c1F N1(C(CC#N)=O)CCC2(CC1)CC(NCc1cccc3c1CCCC3)C2 CCCC(C)(C)CC(=O)N1CC(NC(c2c[nH]c(Br)c2)=O)CCC(O)C1 C1(C(=O)NCCN(CC(C)O)C(c2cccn3cnnc23)=O)OCC2CCCC12 CC1=C(C(=O)NC2CCC2NC(C2(N(C)C)CCCCC2)=O)CCC1 C=CCCCC(C(=O)NCC(C1CCCCC1)O)NC(C1CC(=O)N(C)C1)=O N1(C(c2cc(C)c(Cl)s2)=O)CCN(C(c2cnc(CCC3CC3)s2)=O)C(C(C)C)C1 C1(O)(C(=O)NC2CC2)CCN(C2CCN(CCF)C2=O)CC1.c12ccccc1N2 C(=O)(CCC=CBr)NCC(CN(C(Cc1ccn(CC)n1)=O)CC)(C)C c1(C(=O)NCC(CO)NC(CNC(C)=O)=O)cc2c(ccn2C)s1 C1(CC(N2CCCN(C(C(P(C)(C)=O)O)=O)CC2)=O)Oc2ccccc2NC1=O C1(C#N)(NC(c2c(OC)csc2)=O)CCN(C(c2cc(Cl)ccc2C)=O)C1 C=CC1(C2(C(=O)NCC3CCN(C(c4c(C)cnn4C)=O)C3)CCC2)CCC1 CCCC(CCC)=CC(=O)NC1CCCN(c2nnc(C(F)(F)F)s2)C1 c1(C(=O)NC2CCN(C(C(C)S(C)(=O)=O)=O)CC2F)nc2ccccc2[nH]1 c1(C(N2CC(C(C)NC(=O)CN3CSCCSC3)C2)=O)cccc2occc12 C1(C(=O)NCCC2CSCCN2C(=O)CCC(F)(F)F)CC2(C1)CC2(F)F N1(C(=O)Cn2cc(CC3CCCCO3)nn2)CCOC(c2ccc(Cl)cc2)C1 c1cc2c(CN3CCCCC3c3cc[nH]n3)[nH]nc2cn1 N1(C(c2cc(OC)no2)=O)CC2CCC2(CCNC(=O)Cc2ccno2)C1 C(CCCCCC(=O)NC(c1ccccn1)CO)NC(c1ccc(SC)o1)=O c1(OC)cccc(CCC(N2CCN(C(C3(C)CC4(CC4)C3)=O)CC2)=O)c1F C(=O)(C(C)(C)CCS(C)(=O)=O)N(CCCN(C(C(=C(C)C1CC1)F)=O)C)C c1(OC)ccc(C=CC(=O)N(C2CCN(C(C3CC(SC)C3)=O)C2)C)c(OC)c1 CN(CC(=O)c1cccnc1C1CC1)N1CCN(c2ccc(O)cc2)CC1 N(C(=NCCCF)NCCC1CCOC1)Cc1ccnc(OC)n1 C(=O)(C(F)(F)CCn1cccn1)NC(CNC(C(OC)OC)=O)Cc1ccccc1 C1(C(N2C(C)C(NC(=O)CCc3nc(O)n[nH]3)CCC2)=O)CCCCC12CCC2 n1(CCC(C)C)ncc(NC(=O)NC(C)CC(C)(C)O)c1Cl c1(C(=O)NCC(=O)NC2COCC2CNC(C2C=CCC2)=O)ccc(Br)s1 c1(CC(=O)NCC(CC)NC(c2ccc[n+]([O-])c2)=O)nccc2ccccc12 CC(=NOCC#N)C(=O)N1CC(CC(=O)NCCC2NC(=O)NC2=O)CC1C C1(N(C(=O)C(C)NC(C)=O)CC)(Cc2ccn(C3CC3)n2)CCN(C(C)C)CC1 C1(CNC(=O)CC2CCCCC2)CC2(CCN(C(c3csc([N+](=O)[O-])c3)=O)C2)CO1 C(=O)(C(C)(F)C(F)(F)F)NCC1(C)CCCN(C(c2c(C)nc(O)[nH]2)=O)C1 C12(C(=O)NCCN(C)C(C3C4(CC4)C34CC4)=O)CCC(CC1F)C2 N1(C(c2cc(Br)ccc2C)C(=O)NCCOC)CCC(F)(F)CC1C C#CCC(CC(=O)NC(C)CCCOC)NC(c1ccsc1Cl)=O C(=O)(C#CC1CCCO1)N1CC(O)CC(NC(c2cc(=O)cc[nH]2)=O)C1 Cc1nc(O)ccc1C(=O)OC(CSc1ccccc1Cl)C(C)C c1(C(=O)NCCCCCCNC(C(C)NS(CC)(=O)=O)=O)ccc(C)c(C)n1 C1(C)(C(=O)NCC(C)(C(C)C)NC(CCc2c(C)nccc2)=O)CCC(=O)NC1 C1(C(C)C)CCCC(C(=O)NC2(F)CCOC2)C1.n12cc(nn1)C(=O)N1CC2C1 C1(CN(C(c2nocc2Cl)=O)CC)CCCCN1C(=O)COC(C)C CC1(C)CCC(CC(=O)NCC2C3CN(C(C4(C#N)CCCOC4)=O)CC23)CC1 c1(CCC)n[nH]c(=NCCC2CCN(C(=O)Cc3cc(F)cc(Cl)c3)C2)s1 C1(NC(c2n(C)ncc2Cl)=O)CCN(C(c2ncc(Br)cn2)=O)C12CC2 C=CCC(C)C(=O)NCC1CC(O)CN1C(=O)CSCc1ccc(Cl)s1 C1(=O)C(C)C(C)NCCSC2(CC(=C)C2)CO1.C(C)(C)(C)OC(=O)NCC c1(C(C)(C)NCc2n(C)cc(Br)n2)cc(Cl)ccc1I c1(C(=O)NC(C(C)NC(Cc2cn(CC)nc2)=O)CO)cccc2sncc12 CC(C)(C)CC(O)CC(=O)NC1CC(C)(NC(=O)COCc2nccs2)C1 C12(NC(c3ccc(C)s3)=O)CCC(CN(C(c3csc(C)c3C)=O)C1)C2 CC1OC2(C)CC1(C(N1CCOC(CNC(C3C4CCCC34)=O)C1)=O)C2 C1(OC)CCCC(CC(=O)OCc2ccc(C(=O)OCC3CNC(=O)O3)cc2)C1 N1(C(C(CCC)NC(C)=O)=O)CC2CCN(C(=O)CCC(=O)NN(C)C)CC2C1 c1(C(=O)NC2C(NC(c3c(C)nsc3)=O)CC2)cccc(-c2nnco2)c1 C(C(C(=O)NC1CC1[N+](=O)[O-])N(C)C)N(C)C.C1(=O)CCOCCN1 C1(C(=O)NC2CN(C(C(=O)NCC)=O)C(C)(COC)C2)Cc2ccncc2C1 C12(C(=O)NCc3c(CC)nns3)CCCC1CN(C(=O)C(C)(C)C#N)C2 c1(OC)cc(Br)ccc1CC(=O)NC1C=CC(C(=O)Nc2ccc(Cl)cc2O)C1 C1(F)(CNC(C2CN(C(C)=O)C2)=O)COCCN(C(C2COC(=O)N2)=O)C1 c1(C(N(C2CN(C(C3CC3C(C)(C)C)=O)C2)C)=O)cncc(-c2ccccc2)n1 C12(C(N3CC(NC(C4CCCC45CC5)=O)C(O)C3)=O)CC(CO)(C1)OC21CCC1 C1(CNC(=O)CC2C=CCCC2)CC2CCC1N(C(c1ncnc(O)c1Cl)=O)C2 C1(C(N2CC(NC(=O)OCC)C2)=O)CC(=O)CN1C(=O)CC1CC2CCC1C2 c1(CCCC(N2CCC(C)(NC(C3CC3F)=O)C2)=O)ccc(C#N)cc1 Cc1coc(C(=O)NC2CC(CCNC(=O)C(=O)N(C)C)C2)c1 Cc1nn(C)c(C)c1CNC(C1(C)CCC(NC(=O)C(O)C2CCCC2)CC1)=O Cc1ccc(C=CC(=O)NC2CCC(N(C(=O)CC3CCC(=O)C3C)C)C2)o1 c1(C(=O)NC(C2CCN(C(C3CCCC3O)=O)CC2)C)snc2ccccc12 C(C1=NOC2CN(C(=O)CCN3CCCC3)CC12)NC(c1cc(C)nc(C)c1)=O c1(CC(=O)NCC2CCN2C(=O)C(c2ccc(Cl)cc2)O)c(F)ccc(F)c1F Cc1c(NC(c2c[nH]nc2CCNC(=O)C(C(C)O)N(C)C)=O)cnn1C c1(C2C(C(N3CCC(C(F)F)(NC(CC)=O)C3)=O)C2)c(F)cccc1Cl C1(C(=O)OC(CCC)CC)CCC(F)(C(=O)OC(C)(C)C)C1 C1(CC)CCN(C(=O)C(C2CCCO2)NC(C2COC(=O)N2C)=O)CCO1 C1(NC(CC2(CC)CCC2)=O)COC2(C1)CN(C(=O)CC(C)SC)C2 c1(NCC2N(C(=O)C=CBr)CCC2)ccnc2ncnn12 N1(C(CCOC(C)=O)=O)CCC(CCN(C(C2OCC2(C)C)=O)C2CC2)CC1 C1(NC(c2nncc(C)c2)=O)CCC2CN(C(c3n[nH]c(O)n3)=O)CC2C1 C1(C(=O)NCC2(CNC(c3ccc(C#C)o3)=O)CCOCC2)CC(=O)NC1(C)C N1(C(C=COCC)=O)CCC(C#N)(NC(c2ccc(I)c(Br)c2)=O)C1 N1(CC(=O)NC2CCC(NC(C3(CC)CC3)=O)C2)CCC(=O)NC1=O C(=O)(C1=C(C)CCCC1)N1CC(Br)=C(C)CC1 C1(CNC(CC(C)(C)OC)=O)CN(C(c2occc2Br)=O)C2(CCC2)C1 c1(C(N2CCC(N(C(C(C)CO)=O)C)CC2)=O)ccc2c(=O)n(C)cnc2c1 C1(C2(CCOCC)CC2)CCC(NC(=O)C(c2ccccc2)OC)C1 CCC(C)C(O)C(=O)NCC1C2CN(C(=O)CC(F)(F)CC)CC12 C1(C(=O)NCCCN(C(=O)Cc2ccoc2)C)CC(c2cccc(Cl)c2F)=NO1 C1(C)(CNC(COCC)=O)CC(F)(F)CN1C(C1CCc2n[nH]cc2C1)=O c1(C(=O)NC2(C)CCCN(C(CNC(CC)=O)=O)C2)ccc(S(=O)(=O)CC)cc1 c1(C(=O)NC)cccc(NC(C2(C)CCN(c3ncc(C(C)C)cn3)C2)=O)c1 C1(C(=O)NC2CCN(C3CC3)C2)(CNC(=O)CCOC2CC2)CC12CCC2 c1(CC(=O)NC2(CC=C)CCN(C(C3(F)CCOC3)=O)C2)cc2ccccc2cn1 Cc1cccn2cc(C(N3CCC(CCNC(=O)C4CC4)C3C3CC3)=O)nc12 C(=O)(CC(C)(C)C#N)N1CCC(C(C)(C)CNC(=O)CSCC(N)=O)CC1 Cc1cc(C(=O)N(C2CC2)CC2CCCN2C(c2ccc(C(C)C)o2)=O)nc(C)n1 c1(C(=O)NC2C=CCN(C(=O)CCc3ncco3)C2)occ2c1CCC2 c1(C(=O)NC(C)CCN(C(=O)C(C)(O)C(F)(F)F)C)cnc2ncccc2c1 c1(-c2c(C(=O)NC(C)CN(C)C(C3CSCCS3)=O)c[nH]n2)cc(F)cc(F)c1 Cc1c(-c2cnc(C3CCCN3C(=O)Nc3nccs3)[nH]2)cccc1F N1(C(C2N(CC)CC2)=O)CC(CC(=O)NCC2CCC(C)(C)O2)C(C)C1 CCC(C)C(O)C(=O)N1CCOCC1CC(N1CC2CSCC2C1)=O c1(C(N(C2C(C)CC2)C2CC2)=O)cnc(CNC(=O)CCc2cccnc2)nc1 c1(C(=O)NC2CCC(CNC(c3cc(Cl)c(Cl)[nH]3)=O)CC2)ccc2cccnn12 CS(=O)c1cccc(C(N2CC=C(CCNC(C3CC34CC(O)C4)=O)CC2)=O)c1 C1(CC)CCN(C(=O)CC(C)C2CCC2)C(C(=O)NC2CC(C(C)O)C2)C1 C1(CNC(c2ccn(CC)n2)=O)CN(C(=O)CSCC(C)C)CCC1C c1(CNC(CCCCC#C)=O)nnc2n1CCN(C(=O)CCC1CCC(O)CC1)C2 C1(C(N2CCC(N(C(=O)Cc3cnc[nH]3)CCC)C2)=O)CCCC1C(N)=O CCCN(OC)C(=O)c1c[nH]nc1CNC(=O)C1=CCCC1C N1(C(COC(CC)(C)C)=O)CCN(C(c2ccn(CCO)c(=O)c2)=O)CC1CO c1(C(=O)NCC2(C)CC(NC(=O)C3=NOCC3)C2)cn(C)c(=O)n(C)c1=O N1(C(CC(C)C(=O)c2ccc(Cl)cc2)=O)CC2CNCC2(C(C2CCC2)=O)C1 C#Cc1cn(C)nc1C(=O)N(C1CCCC(NC(c2cncs2)=O)C1)C CC(C)(C)C(O)CNC(c1ncc(Cl)s1)c1nnnn1CCOCC1CC1 C(=O)(CC(C)(O)C(F)(F)F)N1CC(N(C(=O)CCOc2ccccc2F)C)C1 N1(C(C(C)n2ccnn2)=O)CCOCC(NC(=O)C(O)CC(N)=O)C1 C1(NC(c2nnc(CC)s2)=O)CCCN(C(=O)CCc2cc(C)[nH]n2)CC1 C1(C(=O)NCC2N(C(c3cn(CCC)nc3C)=O)CC(F)C2)CCOCC1(C)C c1(CCC)nc(C)c(C(N2CC(F)CC2CNC(c2cnn(CC)c2C)=O)=O)s1 c1(OC)nocc1CCNC1CC1(C)CNS(C)(=O)=O C1(CNC(CCN(C(=O)CSc2cccnc2)CCOC)=O)CC(C#N)C1 C1(NC(CC(C)C2CCCC2)=O)CCCCN(C(=O)C(C)(C)N=[N+]=[N-])C1 N1(C(Cc2n[nH]c(=NC)s2)=O)C2CCCC1CN(C(c1coc(Br)c1)=O)C2 c1(C(=O)NC(CN(C(c2cc(C)on2)=O)C)(C)C)ccc2c(n1)CCC(C)(C)C2 c1(NC(C2CCCCN2C(=O)CN2CCCC2)=O)cncnc1O c1(CC)ncccc1C(=O)NC1CCCC1C(=O)NCC(F)Cl c1(NC(C(=O)NC(CC(O)COC2CCOCC2)CC)=O)cccc(CCN)c1 N1(C(c2ccc(CC)o2)=O)CCC(O)(C(C)CNC(c2ccsc2Cl)=O)C1 C1(C2CCN(C(=O)C(O)C3CC3)C2)(NC(c2ccc(C(=O)O)cc2Cl)=O)CC1 C=CCC(C(=O)N(C1CN(C)CC1O)C)NC(c1cc(Cl)n(C)n1)=O C=CCC(C(=O)N1CC(NC(c2ccc(OC)cc2C)=O)C1)C(C)(C)C c1(C(N(CCC#N)C)O)ccccc1.C1(CC(=O)NC)CN(CC)C1 N1(C(Cc2n(C)ccn2)=O)CCC2CN(C(=O)CC3CCCS3(=O)=O)CC2CC1 c1(C(N2C(CNC(C)=O)C=CC2)=O)cccc(N2C(=O)CCC2=O)c1 C1CCCCC(=O)N1.C1(NC(C(CCC)N(C)C)=O)CC2(CCCO2)CC1 Cc1nc(C2CCCOC2)sc1C(N1CCOCC1CN(C(=O)C=CCO)C)=O c1(C(N(C2(CC(N3CC4COCC4C3)=O)CC2)C)=O)c[nH]c2nccc-2c1 CC1(C(N2CCC(NC(=O)C(C3CCOCC3)F)C2)=O)CNC(=O)C1 c1(NCC(c2ccoc2)C)nccc(NC(CCO)c2nccs2)n1 C1(NC(c2n[nH]c(C)c2O)=O)C2CC1CN(C(c1cc(F)ccc1Br)=O)C2 C1(C(=O)N(C2CCN(C(c3c[nH]nc3C)=O)C2)C)(OC)CS(=O)(=O)C1 c1(Nc2c(C(N3C(C(=O)OC)COCC3)=O)cccc2)ncnc2c1ncn2C C1(CC)CN(C(=O)CNC(c2ccccn2)=O)CCN1C(=O)COC c1(OC)ccccc1C1(C(=O)NC2CCC(NC(=O)COC(F)(F)F)CC2)CCC1 Cc1cccc(C(=O)NC2CN(C(=O)C(c3cccc(Cl)c3)O)CC2O)c1Cl C(CN=c1[nH]c(=N)[nH]c(=NCC(C)NC2CC2)[nH]1)NC(=O)OC(C)(C)C Cn1cc(C(=O)NCCNC(C2CCCC3(C2)CC3(F)F)=O)c(=O)n(C)c1=O C1(C(=O)NC2(C)CCCN(C(=O)COCCO)C2)OCC2CCCC1C2 c1(C(N2CCC(C(N(C)Cc3cc(C)nn3C)=O)CC2)=O)cc(O)ccc1I CC1(C)CCCN(C(C(=O)NC(C2CC2)C2CC2)c2ccsc2)C1C(N)=O C1(C(=O)NCCNC(=O)Cn2cc3ccccc3n2)CN2CC3CC2(CO1)C3 CCC#CCN=c1nc(N2CCCC(C(=O)NC)C2)c2ccccc2[nH]1 Cc1cc(CNC2CC3(C2)CC(NCc2cccnc2)C3)cc(O)n1 N1(C(CN(C(CCOC)=O)C)=O)CCCC2CN(c3ccncn3)CCC12 Cn1cc(C(F)(F)F)nc1C(N1CCC(CNC(=O)C=Cc2ncco2)CC1)=O N1(C(C(C(C)C)NC(Cc2c(C)n[nH]c2C)=O)=O)CC2CCCCC2C1 S(=O)(=O)(c1ccc(F)cc1F)NCC(=O)NC1CCC1(F)F CN1CCc2cc(C(N3CC(NC(c4scnc4Cl)=O)CC(O)C3)=O)ccc2C1 N1(C(C(C(C)OC)OC)=O)CCCc2cnnc(O)c21 N1(C(CC(C)(C)O)=O)CCn2nc(CNC(c3snc(O)c3Cl)=O)cc2C1 CC1(C)CC1(C)C(=O)NCCC1(CNC(c2cc(Br)n[nH]2)=O)CC1 c1(CC)nc2n(n1)CC(C(=O)OCC1(c3ccccc3)CC1)CC2 N1(C(c2cc(C(C)C)nc(O)c2)=O)CCC(N(CC(O)C(F)(F)F)C)CC1(C)C C(C(=O)N1CCC(F)(c2cn(C(C)C(=O)NC)nn2)C1)(C(F)(F)F)OC(C)=O c1(C(N2C(CCCNC(c3c(COC)occ3)=O)CCC2)=O)nccc(Br)c1C Cc1nn(C)c(C)c1OC(C(=O)OCCC1CCC(C)(C)C1)C(C)(C)C c1(C2CN(C(C(n3cc(Cn4c(C)cc(C)n4)nn3)C)=O)C2)c(Cl)cccc1Cl Nc1nc(Cl)ccc1C(N1CC2CC1C2NC(c1ccc(Br)o1)=O)=O Cc1ccc(C(=O)NC2CCCCC2C(=O)N(C2CCC2)CCO)nc1O C1(CC2C(C(=O)NC3(CCOC)CCCC3)C2)CC(C)(C)CN1C(C)=O CC1CN(C(=O)CC2CCCC2NC(c2ccncn2)=O)CC(C)(C)O1 c1(C(=O)NC(C2(O)CN(C(C(C)c3cc[nH]n3)=O)C2)C)cn2c(n1)COCC2 N1(C(COCCC=C)=O)CCCC1CCCNC(C1CCC(F)C1)=O C1(NC(=O)Cn2cc(Cc3ccccc3)nn2)C2CNCC1(CO)C2 C1(C(=O)Nc2c(C)cccn2)CN(Cc2cc(Cl)c(F)c(Cl)c2)CCC1(F)F C(=O)(C1CCCc2sccc21)NC1CC(OC)CN(C(CCC(=O)OC)=O)C1 Cc1cc2c[nH]nc2cc1C(=O)NC(C)(CNC(c1cnn2ccsc12)=O)CO CCCC(O)CC(=O)N(C)CCOCCNC(=O)CC1OCCC1(C)C CC(C)C(F)C(=O)N1CCC(NC(=O)C(c2ccc(F)cn2)(F)F)C1C n1(CC)nc(C(=O)NC2CC(O)C2CC(=O)NC2(C)CCSC2)cc1O C1(NC(C=C(COC)C)=O)CCN(C(c2cnc[nH]2)=O)C(C2CC2)C1 C1(C(=O)NCC(C(C)C)(C)Nc2cc(Cl)nc(C3CC3)n2)CNC(=O)CC1C N1(CC(N2CCC(OCCNC(C3(C4CC4)CC3(F)F)=O)C2)=O)CCCNC1=O C1(NC(C2C(NC(Cn3c(C)nc(C)n3)=O)CCO2)=O)CC2(C1)CN(C)C2 C(=O)(CC(C)C(F)(F)F)NCCC1CC(OC)CN1C(c1cnc(C)s1)=O CC(CC(F)(F)F)C(=O)NC(C)CC(=O)O Cc1c(NC(=O)CC#N)c(C(=O)OCC23CCC(CC2)N3)nn1C Cc1nc(Cl)ccc1CC(N1CCC(CNC(=O)C=CC2C(C)C2(Cl)Cl)CC1)=O c1(CNC(c2[nH]nc(OC)c2Cl)=O)cc(C(=O)NCCC2CCCN2C)n(C)n1 N1(C(C(C)C2CCCC2)=O)CCCC(CNC(c2cnc(=N)[nH]c2)=O)C1 C1(NC(c2c(OC)n(C)nc2)=O)CCN(C(=O)CCCCSC)CC1C(N)=O N1(C(CC2(C)CC2(F)F)=O)CCCC(C(=O)NCCN2CCCC2)CC1 c1(NC2C(NC(CC(C)(C)N3CCCCC3)=O)CCC2)ccc(S(C)(=O)=O)cn1 C(=O)(C1=CC(O)C(NC(=O)COCCOCCO)C1)NCCS(CC)=O c1(C(C(=O)NCCN(C(C2(C)CCOC2)=O)CC)(C)C)ccc(Br)c(C)c1 C=CC1(CC(=O)NCC2CC(C)C2(C)C)CN(C(=O)C=CC2CCCCC2)C1 c1(OC)ccc([N+](=O)[O-])c(C(N2CCC(NC(c3cnns3)=O)C(CO)C2)=O)c1 C123CC1CN(C2)C3=O.Cc1cnn(C(C)C(=O)Nc2ccc(C)s2)c1 C(=O)(CC(C)CC(C)(C)C)NCCC(C)NC(c1ccc(C#C)cc1)=O C12(NC(C3(F)CCC(F)(F)C3)=O)CCN(CC1)C(=O)NC2.C(=O)(CC1CC1)OC CCCCCC(CC)C(=O)N1CCCC(NC(C2CN3CCC2CC3)=O)CC1CC C12(CNC(CC(CC)SC)=O)CCCCC1N(C(=O)CCc1ccon1)CCC2 C#CCCCC(C)(C)C(=O)N(C1CCC(N(C(=O)CCSCC)C)CC1)C C1(C(N2C(C)COCC2)=O)CCN(C(=O)C2CCC2C)O1 c1(CCC(=O)NC(c2ccc(OC(F)(F)F)cc2)C(C)C)nnc2n1CCNC2 c1(C(=O)NCC2(NC(C3CCCN3C3CCCC3)=O)CC2)ccncc1Br c1(NC(C2CN(Cc3cc(B(O)O)co3)C2)=O)nc2cc(Cl)ccc2s1 C=CC(C)(O)CC(=O)N1CC(CNC(=O)C(C)(C)C2CCCC2)C(O)C1 Cc1cc(-c2cn(CCC(=O)NCC3OC(=O)NC3(C)C)nn2)cc(C)n1 C12(CC)CCC(C(N3CCC(CNC(c4ccncc4F)=O)(OC)C3)=O)(CO1)C2 C#Cc1ccc(C(C(=O)NCCC)N(C)Cc2n[nH]cc2Br)cc1 C(=O)(C(F)(F)C(F)(F)F)NC1CCCC(CNC(c2ccc(OCC)cn2)=O)C1 N1(C(CN(CCC)CCOc2cccc(O)c2)=O)C2CCC(C(=O)NC)C1CC2 c1(OCCC)ccccc1CN1CC2C(C1)N2C(C1CCC(F)(F)C1)=O C1(C(=O)NCC(C)(C)n2ccnn2)CC2(CC2)CN1C(C1CC2(CC2)C1)=O C(=O)(CS(=O)(=O)C(C)C)N1C2(CNC(c3c(C)c(N)ccc3)=O)CCC2CC1 C1(CC(N2C(CCCCNC(CCOCCOC)=O)CCC2)=O)CCCCCC1 C1(C(=O)NC(CC)CNC(c2cc(C)c(C)o2)=O)CCCN(S(N)(=O)=O)C1 CC1(CCNC(c2ccns2)=O)CCN(C(C2CCC(=O)N2C2CC2)=O)CC1 N1(C(C(CC)F)=O)CCCCCC1CNC(c1c(Cl)cnn1CC)=O C1(NC(C)=O)COCCC1NC(c1ccc(-c2ccccn2)nc1)=O C1(NC(COCc2ccc(C)s2)=O)CCOCC1NC(=O)Cc1cncnc1O C1(CNC(CSC)=O)CCN(C(=O)C(COC(C)(C)C)OC(C)=O)C1 C#Cc1cccc(C(=O)NCCC(C)NC(C2CC3(C)CC2CO3)=O)c1 N1(C(C(F)OC)=O)CCN(C(c2csc(C(N)=O)n2)=O)C(CC2CC2)C1 Cc1cnc(Cl)cc1NC(C1(C)CCN(Cc2ccc(F)c(O)c2)CC1)=O CC(CC(C)(C)O)N1CCC(CNC(C2(c3ccc(F)cc3)CCCC2)=O)C1 C(CCCC(=O)N1CCC(O)C1C(C)(C)C)NC(C(C)SC(C)C)=O C=CCCCCN=c1nc2scnc2c(NCC2CCCN2CC(F)F)[nH]1 Cc1cc(C(=O)NC2(CNC(=O)CNC(=O)CC(F)(F)F)CC2)nc(O)n1 c1(C(=O)NC(C(C)NC(CCCOCC=C)=O)C(C)C)ccc2[nH]c(=N)oc2c1 N1(C(C2CCCC(C)CC2)=O)CCCN(C(c2ncnc(O)c2F)=O)CCC1 C(=O)(C1=CCCCCC1)N1C(C)CC(CCNC(=O)CC2(O)CCC2)CC1 N1(C(C2C(CNC(C(C(C)C)OC)=O)CCC2)=O)CCC2(CC1)CN(C)C2 C=CC(CCC)CC(=O)N1CCOC(CCNC(c2ccc3c(c2)COC3)=O)C1 c1(C(=O)NC2CC3CN(C(C(CC)C#N)=O)CC(C2)C3)cnc(O)c([N+](=O)[O-])c1 CC(F)CN=c1[nH]c(=NC(C)c2ccccc2CO)[nH]c2ccccc12 C1(OC)CN(C)CC1NC(c1occc1CNC(c1cc(Cl)cs1)=O)=O C=CC1CCN(C(=O)CC2CC3(C2)CN(C(=O)C(c2cc(C)no2)=CC)C3)CC1 CCC(CNC(=O)C(F)(F)c1ccsc1Cl)(CC)NC(=O)CCN(CCO)CC C1(C(=O)NCC2C(C=C)C2)CCC(n2cc(-c3ccccn3)nn2)CC1 C1(CNC(c2[nH]nc(C(=O)OCC)n2)C)CC12CCOc1ccccc12 C(C(=O)NCC1COCC1NC(c1c[nH]c(C#N)c1)=O)(C(C)C)OC c1(OCCC(=O)NCc2cc(CNC(CCSCC)=O)no2)cc(C)ccc1C C=CCC(CC(C)C)C(=O)NCC1(CO)CN(C(=O)C(N2CCCCC2=O)C)C1 CC(C)(C)C#CCCNC(=O)C(CNC(c1cc(F)c[nH]1)=O)CC1CC1 N1(C(CC2(C)CCCCC2)=O)C2CCC1CC(CNC(=O)C=CC1CCOC1)C2 c1(C(=O)NCC(N2CCN(C(C3CCCCS3)=O)CC2)C)cc(O)ccc1F C12(NC(CCCCN(C(C)C)C)=O)CCC(C1)N(C(c1cc(F)ccc1F)=O)C2 Cc1cccc2cc(C(=O)NCCn3cc(C4(C(C)C)CCCO4)nn3)[nH]c12 c1(C(=O)NC2CC(C)N(C(c3csc(=N)[nH]3)=O)C2)cccc([N+](=O)[O-])c1 c1(C(=O)NC(C)CO)c[nH]c2ccc(-c3cccc(NCCF)c3)cc12 n1(CCOC)nc(C)c([N+](=O)[O-])c1NC1CCC(NC(=O)Cn2ncc(Cl)c2C)C1 c1(C(=O)NC(CNC(CS(CC)(=O)=O)=O)CO)cc(F)c(C#N)c(F)c1 C1(n2cccn2)(C(=O)NC(C(=O)OC(C)C)C)CCN(C(=O)CCCCCF)CC1 C(=O)(C=C1SCC(=O)N1C)N1C(CCC)(NC(c2cccc(N)c2)=O)CCC1 CC(C(=O)N1CCCC(F)(C(=O)NCC(O)CCC2CC2)C1)C(F)(F)F c1(NC2C(CO)COCC2)c(CCc2ccccc2)cc(Cl)cc1Cl c1(C(=O)NC(CCC)C)coc2c1CN(C(C1CCC1NC)=O)C2 N1(C(c2c(C)cco2)=O)CCCC2CN(C(=O)CCn3cncn3)CCC12 c1(C(=O)Nc2cccc(CNC(CC(=C)C)=O)c2)cc2c(ncn2C)[nH]1 C1(C(N(C)CC2(CNC(C34CSCC3C4)=O)CC2)=O)CCCCO1 C(CC(F)(F)F)NC(c1cn(CC2CCCO2)nn1)=O c1(OC)cncc(C(=O)N(C(C)C(=O)NCc2csc(C)c2C)C2CC2)n1 c1(OC(C(=O)NCC2CC(NC(c3c(C)nsc3)=O)C2)C)cccc(Cl)c1 C1(NC(c2cc(C)nnc2O)=O)CCCCN(C(=O)CCCC(C)C)CC1 N1(C(=O)NCc2c(C(=O)OC)occ2)CC2(CCCCC2)CC1C C1(C(=O)NC2CC(C)(CNC(c3c[nH]c(Br)c3)=O)C2)Cc2ccccc2O1 C1(C(N(CC(CNC(CC(C)=CC)=O)(C)C)C)=O)CCOCC1(C)C c1(N(CCNC(c2cc(C)nn2C)=O)C2CC2)cc(C)nc(Cl)n1 c1(C(=O)NCC(C)(C)NC(CSCCC)=O)cc(O)cc(Cl)c1 CCCCC(CNC(c1occc1Cl)=O)NC(C1CCC(C)(C)C1)=O n1(C(CC)C)nc(C(=O)NCC2CCCN(C(=O)CCOCC(F)F)C2)cc1C C(=O)(C(C1=CCC2CC2C1)N1CCC1COc1ccccc1Cl)NC CCCC(CNC(=O)COCCCF)NC(c1cc(=N)[nH][nH]1)=O CCC(CC(=O)NC1CN(C(c2sc(C)c(C)c2C)=O)CC1O)C(F)F c1(C(N2CCC(O)(CCNC(C(n3ccc(C)n3)C)=O)C2)=O)ccc(N)c(N)n1 c1(OCC)sccc1C(=O)NCC1CCC(NC(C2(COC)CC2)=O)C1 C(C(C(=O)N1CC(C(C)NC(c2cn(CC(F)(F)F)nn2)=O)C1)N(C)C)OC N1(C(C2(COC)CC2)=O)CC2(CCC2)CC1CNC(=O)CC(C)SC C1(CNC(CC2C(C)OC(C)C2)=O)CCC2CN(C(=O)C(C)(C)CF)CC2O1 CC1(C)CN(C(C2(C)CC(F)(F)CN2C(=O)CC(O)Cl)=O)CCC1N1CCC1 C12(NC(c3cc(CC)ncc3)=O)CCCC1N(Cc1nc3c(o1)CCCC3)CC2 c1(C(C(N2CCC(O)(CN(C(=O)OC(C)(C)C)C3CC3)C2)=O)O)ccc(C#N)cc1 C1(N(C)C)CCC(C(=O)NCC2CCN2C(c2ccn(C)c2)=O)CC1 c1(C(=O)NCC(N2CCN(CCCC(C)(C)C)CC2)(C)C)scc2c1CCCC2 CC1(C)CC(NC(C2C=CCN(C(c3cscc3Cl)=O)C2)=O)C(C)(C)O1 C(=O)(C1CCCn2cncc21)NCC(CCCC)NC(=O)C(Cl)=CCl C1(C(=O)NCCCCC2CN(C(c3cc(C)no3)=O)C2)CCCCC12CCC2 N1(CC2(NC(C3CC3Cl)=O)CC2)CCN(C(=O)CCCC2CCOCC2)CC1 N1(C(c2cc(C(C)=O)[nH]n2)=O)CC2CC(C1)CN(C(C1CCC3CCC13)=O)C2 C1(NC(c2c(CNC(C(CN(C)C)(C)C)=O)occ2)=O)CCCC(F)(F)C1 C1(COC(COC(=O)C2=CCCC2)=O)CCC2(CCC2)C1NC(=O)OC Cc1cc(NC2CCOC(C3CC3)C2)c(S(N)(=O)=O)cc1[N+](=O)[O-] Cc1ccc(Cl)c(OCC(=O)NCC2(F)CC(NC(=O)C(=O)N(C)C)C2)c1 C12(CNC(C(C=CC)O)=O)CC1CN(C(c1cnn(C(C)(C)C)c1Cl)=O)C2 C1(CC(=O)N(C(C(=O)N(C)Cc2c(C)cco2)C)C2CC2)CC(C)(C)CO1 c1(NC(c2n(C(CC)C)nnn2)c2coc(C)n2)cccc(C#N)c1C c1(C(N(C2CCN(C(=O)CC3CC4CCC3O4)C2)CCC)=O)cc(=O)n(C)o1 C1(C#N)(CC(=O)N(C)CCOCCN(C)C(c2cccc(Cl)c2)=O)CCOCC1 CC1CC(C(=O)Nc2ccc(C(C)(C)C)cc2)N(C(=O)CC(F)(F)F)C1 Cn1ncc(CNC(=O)CCc2nncs2)c1C(=O)NC1CC(O)C1 C(=O)(CCC(C)(C)F)NC1C(CNC(c2nn(C)c(C3(Cl)CC3)c2)=O)CCC1 Cc1cc(Cl)ccc1-n1nc(CCC(C)C)nc1C1CCCN1CC(C)C c1(C(=O)NC2CCN(C(c3ccc(COC)o3)=O)C2)ccc2cnccc2n1 c1(C(N2CCC(OC)(CNC(c3ncccc3C)=O)C2)=O)ncc(C)cc1C CC(C)C(O)CC(=O)NCCCN(CCCNC(=O)CSc1cscn1)C N1(C(C)=O)CCc2cc(C(=O)NC3(c4nnnn4C)CCOCC3C)ccc2C1 c1(C(=O)NC(C(=O)OCCC)C)ccnc(CNC(=O)CN2CCCCC2)c1 N1CCCn2nncc2C1.Cc1nnc2n1CC(C(=O)N)C2 c1(N(c2nnn(C)n2)C(=O)C(=O)NCCC[Si](C)(C)C)ccc2c(n1)CCO2 Cc1cccc(CNC(=O)CC2(C)CN(C(c3c(C)n[nH]c3C)=O)C2)c1 C(C)(CNC(c1cc(C)n(C(C)C)c1)=O)(CC(C)C)NC(c1c(OC)ccs1)=O CCS(=O)CC(=O)NCCC1CC(NC(=O)CN2CCC(O)CC2)C1 CN1CNC(=O)C12CN(C(c1cccc([N+](=O)[O-])c1C(F)F)=O)C2 N1(C(c2[nH]cc(C(C)(C)C)c2)=O)CCC2CCC12CNC(c1ccc(O)nc1)=O C=CCCCC(=O)NC1(C)CN(C(C2(c3ccccc3)CC(F)C2)=O)C1 N1(C(c2nc(OCC)oc2)=O)CC=C(C(=O)NC2CCCCC23CC3)C1 N1(C(C=C(CC)C)=O)CCC(CF)(NC(c2ccc(C3CCOC3)s2)=O)C1 C1(F)(CNC(CCSCCC)=O)CCN(C(c2cc(C3CC3)n(C)n2)=O)C1 C(C)(C(O)C(C)C)NC(C(C1CCN(C(CCn2ncc(C)c2)=O)C1)C)=O C(=O)(C(C)(C)Cc1cccc(Cl)c1)N(C1CCN(C(C2CC3CCC23)=O)C1)CC c1(C(N(CCCCCC)CCNC(C2CCCS2)=O)=O)nccc2ncccc12 CC1CC(NC(c2cc(C#N)c[nH]2)=O)CN(C(C2(CF)CCC2)=O)C1 c1(OCC(=O)NC2C(NC(CC(CC)SC)=O)CC2)c(F)cccc1F N1(C(=O)OC(F)(F)Cl)CCC(O)C(C(=O)NC2CC3CCC2O3)C1.C1CO1 Cc1cc(C(N2CCCC(Nc3ncc(Cl)cn3)C2)C(=O)NC2CC2)cc(C)n1 Cc1ccc(F)cc1NC(=O)C(C)CNC(C1(C)CCCS1)=O c1(C(C)C)ccc(C(N2CC(F)(CNC(C3CCC3C)=O)C2)=O)c(F)c1 C1(C(=O)NCC(CN(C(=O)CC2(C(F)(F)F)CC2)C)(C)C)CCc2nccn2C1 c1(NC(=O)NC(C2CCS(=O)(=O)C2)=O)ccc(NC2COCCNC2=O)cc1Cl N1(C(CCOCCOCC)=O)CC(NC(=O)CC2CSCCS2)CC(C)C1 C1(C(=O)N(CC(N2CCC(n3ccnc3)C2)=O)C2CC2)CC2CCC1O2 C1(NC(C(CSC)OC)=O)CCCC(NC(c2cncc(C(F)F)c2)=O)C1 C1(C(N(CCCNC(C2CCC2(C)C)=O)C)=O)C(C)(C)C1(F)F C(=O)(C(C)CCC(C)(C)C)NCC1N(C(C=CC=CCCCCC)=O)CC1 N1(C(C(C2CC2)OCC)=O)CC2CC1CN2C(=O)C=Cc1cncs1 C1(CNC(c2ccc(OC)nn2)=O)CC2(CC2)CN1C(=O)C(C)(F)F c1(OC)ccc(F)c(C(=O)NC2CCC(N(C)C(c3nocc3C(C)C)=O)C2)n1 C(=O)(C(N)CC(C)(F)F)N(C)Cc1cccc([N+](=O)[O-])c1 c1(OC)ccc(O)cc1NC(C1CC(N(C)C(c2[nH]cc(C)c2C)=O)C1)=O c1(CNC(c2c(C)[nH]c(=NCc3nc(Br)cn3C)s2)=O)nccc2cccnc12 C(c1cccc(F)c1)=C(C(=O)NCCCCCCN(C(CC(C)C1CC1)=O)C)F N(C1CCCc2ccc(Cl)cc21)C1(c2nn[nH]n2)C(C)CN(C)C1 c1(C(N(C(C(=O)OCC)C)C)=O)csc(CNC(C2(C#N)CC2)=O)c1 C1(NC(C(COC)(F)F)=O)CC2CCC(C1)N2C(=O)CC1CCCCCC1(F)F C(C(CN=c1[nH]n(C(C)C)cc1[N+](=O)[O-])C(F)(F)F)NC(c1c(C)ocn1)=O C1(O)(C(C(=O)NCCCSC)F)CCCC1.N1(C=O)CCCCC1.C12(CC1)N(C)C2=O C1(C(=O)NCc2cncs2)CN(C(=O)CC2CCCC3CC23)CCO1 C1(O)(CNC(CCSc2n(C)ccn2)=O)CCN(C(C2C(C)(C)C2(F)F)=O)C1 N1(C(CC=C=C)=O)CCCCCC1C(=O)NC1CCC(N(C)C)C1 CC1CN(C(C2C3CN(CCN4C(=O)CCC4=O)CC23)=O)CCC1N(C)C C1(C)(NC(C2CC(CNC(c3cn(CCC)nc3)=O)C2)=O)CCC(=O)N(C)C1 c1(-c2cn(CC=C)nn2)nc(Cc2ccccc2C)nn1C1CCCCC1 N1(C(C(C#C)(C)C)=O)CCN(C(=O)Cc2cc[nH]n2)C2(CC2)C1 CC1CCC2(CCN(C(=O)CN(C(=O)CCc3ncccn3)C)C2)C1 C1(CNC(c2ccc(C)nc2O)=O)CN(C(c2cc(C)[nH]n2)=O)C2(CCC2)C1 C1(OCCC)CCC(NC(c2noc(C)n2)c2nnnn2C(C)(C)C)CC1 c1(C(=O)NC2C=CCN(C(C3(C)CC(=C)C3)=O)C2)ccc(C)c(Br)c1F c1(NC(c2nccc(CNC(Cc3ccc(C)nc3)=O)c2)=O)cnn(C)c1C#N C(=O)(C(CC(C)C)NC(c1ccc(F)c(C)c1)=O)N1CCC(SC)C1 c1(-c2onc(C(=O)NC(C)CN(C)C(C3SCCS3)=O)n2)ccc(Br)cc1 C1(NC(c2cc(C)ns2)=O)CC12CCN(C(c1ccc(C#N)n1C)=O)CC2 C=C1CCN(C(c2cnc(COC)o2)=O)C(C(=O)NCC(C)(O)C(F)(F)F)C1 N1(c2nnc(CCC(=O)NC3CC(N(C)C)C3)o2)CCN(C)CC1 c1(C(=O)NCC(C)N(C)C(c2nnc(S)n2C)=O)cc2cc(Cl)ccc2o1 C1(CC)OCCC1N=c1[nH]c(=NCC(=O)NC2CC2)c2ncccc2[nH]1 N1(C(CNC(c2ccccc2)=O)=O)CCCC(O)(CNC(C2CC2C2CC2)=O)CC1 C(=O)(C(CC)CC(C)C)NC(CCCC(=O)NCc1c(COC)noc1)C c1(C(=O)NCC2CC(NC(CC(CN(C)C)O)=O)CC2O)ccn2cc(C)nc2c1 c1(OC(C)C)ccc(CC(=O)NCC2(F)CC(NC(c3ccsn3)=O)C2)cc1 N1(C(C(CC)(C)C)=O)CC2CCC1C1CN(C(c3cnn[nH]3)=O)CC21 CC1(C)CC(CNC(C2(C3CC3)CCC2)=O)N(C(=O)C=CC2CC2)C1 c1(CNC(C(COCC)NC(CC=CC=C)=O)=O)ccc(O)cn1 c1(NC(C(=O)NCCC(=O)OC)=O)ccc(NC(c2cccc(I)c2)C#N)cc1 Cc1nncc(C(N2CC(O)(CC(N3CC(C(C)(C)O)C3)=O)C2)=O)c1C c1(C(=O)NC(C2(CNC(c3ccc[nH]3)=O)CC2)C)nccc2c(F)cccc12 c1(C(C)(C)C(=O)NCCC2CCN(C(=O)CS(=O)(=O)N(C)C)C2)ccc(F)c(F)c1 c1(C(=O)NC(C2CCN(C(c3c(CC)occ3C)=O)C2)C)cc(C)ccc1C C1(C(=O)NCCCCNC(C(P(C)(C)=O)O)=O)COc2ccc(F)cc2C1 Cc1cc(O)c(Cl)cc1C(=O)NCCCCCN(C)C(c1ccc(N)c(F)n1)=O N1(C(C2C(CCC)CCC2)=O)CCC(F)(CNC(c2ccc(C)[nH]2)=O)C1 C1(C(=O)NCCCN(C(c2nc3cnccc3s2)=O)CC)CCc2nn[nH]c2C1 CC1(C)CC(C(=O)NCc2nccs2)CN(C(C2COCC2(C)C)=O)C1 C1(C(F)(F)F)(C(=O)NC(C)CC(C)NC(C2(CC3CCC3)CC2)=O)CCOCC1 C(=O)(C(C)(C)C(F)(F)F)NCCCNC(CN1CCCC(C(=O)OCC)C1)=O C1(C(N(CC(O)C2CCC2)C)=O)CC=CCN1C(=O)C=CC(C)(C)SC c1(-c2ccc(CC)s2)csc(=NCC2C3CCOCC23)[nH]1 c1(CN(C(=O)CNc2nc3c(s2)CCC3)CC)cc2occc2n1C Cc1cc(C(=O)NC(C)CC(=O)NC2CSC2)nn1-c1ccccc1 C(=O)(CCCCCN=[N+]=[N-])NC(C(N1CC(NC(COC)=O)C1)=O)C N1(C(c2cnc(C)[nH]2)=O)CC(N(C)C(C2CCC(N(C)C)CC2)=O)C(O)C1 C1(C(F)(F)F)(CNC(C(COc2c(OCC)cccc2)C)=O)CC2CCC1C2 CCCCN=C(NCC1(C#N)CCC1)N1CCN(CC(F)(F)F)C(C)(C)C1 C12CC(=O)N(C1)CC(CC)(Sc1ccccn1)CC(=O)NCC(C)CNC2=O c1(OC)ccc(Br)cc1NC(c1ccc(C(=O)N(C)CCc2cc[nH]n2)cc1)=O N1(C(Cn2c(C)cnc2)=O)CCCC1(C)CNC(C1(C(C)C)COC1)=O c1(C(=O)NCC(C)NC(=O)C(F)(F)c2cscn2)cnn(C)c1N C(=O)(C1=CCCCCC1)NCC(CC)NC(c1cccc(C)c1[N+](=O)[O-])=O CCCC(F)C(=O)N1CC(CC(C)NC(c2cnccn2)=O)C1 C1(NC(c2ccc(C)n2C)=O)CCN(Cc2ncsc2C)CC1(C)C C1(OCCCC)CC(NC(=O)NCCSc2ccco2)C1(C)C C1(NC(c2ccc(C(F)F)cc2)=O)(CF)CCN(C(=O)C=C2CCOCC2)C1 C1(S(N)(=O)=O)(CNC(C2CCCN(C(Cc3c(C)occ3)=O)C2)=O)CCC1 c1(CC(=O)N(CCNC(C2CN(C(N(C)C)=O)C2)=O)C2CC2)nnc(O)s1 N1(C(C(C)OCCN(C)C)=O)CCCC(CNC(=O)CC2C=CCCC2)CC1 C#Cc1cnn(C)c1C(=O)NC1CC2C(NC(=O)C(C)SCCOC)C2C1 C1(C(N(C2CCN(C(C(C)OCCN(C)C)=O)CC2)C)=O)Cc2ccccc2S1 C1(CC)CN(C(c2c[nH]c(=NC)s2)=O)CCC1CNC(c1cnn[nH]1)=O N1(C(C2CN(C)C2)=O)CCC2(CC1)CC(NC(=O)CCCc1ccccn1)C2 Cc1cc(C(=O)NCC2CCC(NC(=O)CC(C)(C)O)C2)nn1C(C)(C)C Nc1cc(C(=O)NC2CCN(C(=O)C3=CCOC3)C2)c(Cl)c(F)c1F c1(SC)ccc(C)c(C(N2CC(CNC(C3(CO)CCOC3)=O)C(O)C2)=O)c1 N1(C(C2C(C(C)=O)COC2)=O)CCC(CC(=O)NCc2cnnn2C)CC1 C=CCCCC(C(=O)NCC1(C(C)(F)F)CC1)NC(C1(CC2CC2)CC1)=O C(=O)(C1=C(C2=C(CN(CC)C(S(=O)(=O)C(C)C)=O)N2C)CCCC1)OC C1(C(N2CCC(CSC)C2)=O)CC(CC)CCN1C(=O)CCc1cncn1C Cc1cc(C(N2CC3C(NC(C4(Cl)CC45CCOCC5)=O)C3C2)=O)c(O)c(C)n1 C=CC(O)C(=O)NC1CCC(NC(c2ccc(-c3cccnc3)s2)=O)C1 C(=O)(C1=Cc2cc(F)ccc2OC1)NC1CN(C(C2(C)C=CCC2)=O)CC2C1C2 C1(C(=O)NC2CCN(C(C3(CC=C)CCOCC3)=O)C2)CCCC2(CCC2)O1 c1(C(N2C(CNC(C=CC(CC)C)=O)COCC2)=O)nc(Cl)c(=O)[nH]c1N C1(C(=O)NC2C(C(=O)NCCC(CC)O)CCC2)OCC2CCCC12 Cc1nccc(C)c1NC(C1CN(C(C2CCOC2C2CC2)=O)CCO1)=O C=C(C)C1OCCC1C(=O)NCC(C)(C)OCCO.N1(C(CO)=O)CC2(CCCC2)C1 N1(C(C(CC)SC)=O)CCOCC1C1CCCN(C(c2cc(OC)ncn2)=O)C1 Cc1cc(C(=O)N(C2CC(C#N)C2)CC(=O)NCCN2CCCC2=O)c(C)s1 C12CN(CCO1)C2.C1(CCCC)CCCN1Cc1cn(Cc2csc(Br)n2)nn1 Cc1cc(F)c(NC(=O)NCC2CC2Cc2ccccc2)c(F)c1 Cc1nc2cc(C(N3CCCN(C(=O)CCC(C)(C)C)CC3C)=O)cc(O)c2o1 Cc1ncc(CC(=O)NCC(C)NC(C2CC3(CC3)C2)=O)s1 C1(C(N2C(C)(C(=O)NC)CC2)=O)CCCC(NC(=O)C=Cc2cc[nH]n2)C1 c1(CC(C)C)ccccc1COC(C1(C)CNC(=O)N1)=O N1(C(C(CCC)CC2CCCCC2)=O)CCC(C)N(C(=O)CCCC(F)F)CC1 CC1SCCCC1C(N1CC=CC1(C)C(=O)NC1CC(C)(C(N)=O)C1)=O c1(NCc2c(CC)nn(C)c2)[nH]c(=NCC2CC2C2CC2)nc2c1ncn2C C(=O)(C(C)(C)C(=O)NC(C1ON=C(C)C1)C1CC1)NC1(CC(F)(F)F)CCOCC1 C#CC1CCN(C(=O)C(c2ccnn2C)NC(c2scnc2Cl)=O)C1 C(=O)(C1(C)CCn2ccnc21)N(C1CCN(C(CC(COC)(C)C)=O)C1)C C(=O)(CS(=O)(=O)C1CC1)NCC1(C(C)NC(C)=O)CC1 C1(CC(=O)NC(C)CCCNC(=O)C(C)(C)n2cccn2)CC(C)(C)OC1=O C(CCC(C)NC(c1cnc(C(C)(C)CF)o1)=O)NC(COCC=C)=O C1(CNC(CC2(COC)CCC2)=O)CCCC(F)C1.c1(CC(=O)N)n[nH]c(C)n1 Cc1nn(C)c(C)c1CCC(N1CC2(CC2)CC1CNC(C12CC(C)(C1)C2)=O)=O c1(C(=O)NC(CNC(CCCCCCC)=O)CO)cc2cccc(OC)n2n1 C(=O)(CS(=O)(=O)CCO)N(C)CC1CCCN(C(=O)CC2CC3(CCC3)C2)C1 C(N=c1nc(C2CC2)c(F)c[nH]1)c1c(CNC(c2ccc(SC)o2)=O)nco1 Cc1ccc(C)c(C(N2CCN(C(=O)C=Cc3ccc(F)cc3F)CC2)=O)c1O c1(C(=O)NC(C(CO)NC(c2oc(CC)c(C)c2)=O)C)coc2c1COC2 c1(CCCNC(CCN(C(CCOCCOC)=O)C2CC2)=O)cccnc1 N1(C(c2nc(C)[nH]n2)=O)CCCN(C(c2nccc(Cl)c2C)=O)CCC1 C1(CC)CCCCN1C(=O)CC1COCCN1NC(c1cc(C)ccn1)=O C=C=CC(C)C(=O)NCCC1CCCN1C(=O)C(C1CC(F)(F)C1)OC CC1CCC(C(N2CC(CCNC(=O)C3=CCCCO3)C2)=O)C(=O)N1 N1(C(CNC(C)=O)=O)CCC(C(=O)NCC2CC2(F)F)(CO)C1 Cc1cc(C(F)(F)C(=O)NCC(C(C)C)NC(C2CCCN2N=O)=O)cnc1Cl C(=O)(CC(C)C(F)(F)F)N(C(CCNC(c1c(C(=O)OC)scc1)=O)C)C C(=O)(C1=NN(C)C(=O)CC1)N(C)CC1(CNC(=O)C=Cc2ccnn2C)CC1 CC(C)C(C)(CNC(=O)CSCc1ncc[nH]1)NC(=O)CC1CCCC1O C1(CCC(=O)OC)CCCN(CNC(c2ccc(-n3nc(C)cc3C)cc2)=O)C1 N1(C(CCC#C)=O)CCCC2CCN(C(c3cnc(CC)cn3)=O)CC12 C1(CNC(CSCC=C)=O)CC2CCC1N(C(c1nsc(C)c1N)=O)C2 c1(C(C)NC(=O)Nc2cn(CCC(C)(C)C)nn2)nnc2c(=O)n(C)ccn12 C1(CC(=O)NC2CCC(F)(CNC(c3c(C)ncn3O)=O)C2)(OC)CCOCC1 N1(C(C(CCCC=C)NC(=O)C(C)CC(F)(F)F)=O)CCCC(C2CCC2)C1 C1(C(=O)NCc2cn(C(CC=C)CC)nn2)CC2CC(C1)CS(=O)(=O)C2 N1(C(C2OCC(C)C2)=O)CCCC2CN(C(c3cnn[nH]3)=O)CC12 Cc1occc1C(=O)NCCN(C(=O)C(c1ccccc1)O)C1CCCC1.CCOC C12(NC(c3c(C)csc3)=O)CC1CN(C(=O)CN1CCC(C)C1)C2 c1(C(=O)NCCCC2N(C(Cn3c(C)nc(C)n3)=O)CCC2)cc(O)ncc1F Cc1ccsc1C(=O)NCC1CC(F)(CNC(C2CC2(c2ccccc2)C)=O)C1 N(C(=NCCCCl)N1CCN(C(c2ccco2)=O)CC1)CC(CC)C(C)C C(CN=C(NCCOC(C)(C)C)N1CCC2CCCOC2C1)N(C)OC(=O)C1CC1 C1(NC(c2cc(O)cs2)=O)CCCC(NC(c2cc(F)ccc2F)=O)CC1 CC1CCCN(C(=O)C(C2CC2)NC(=O)CS(C)(=O)=O)CC1 C1(NC(CC2CC(SC)C2)=O)C2CC(NC(c3ccc(Cl)cn3)=O)CC12 C(C1CCC(C)CC1)=C(C)C(N1CC(NC(c2c[nH]cc2C(C)C)=O)C(O)C1)=O C1(C(C)(O)CNC(=O)Cn2cncn2)(CCN(C)C)CCCC1.C1(=O)CC2(CC2)N1 C1(NC(C(CC(C)C)F)=O)CN(C(c2cocn2)=O)C2(CCCCC2)C1 Cc1ccc(CSCCC(=O)NCC2CCN2C(=O)Cn2nc(C)nc2C)cc1 C#CCCCCCC(=O)N1CC(O)CC1CNC(c1ccc2cnoc2c1)=O N1(c2ncc(C(=O)OCC)cn2)C2CCC1CC(NC(=O)Cn1cncn1)C2 c1(CNC(C2N(C(C(CC)n3cncn3)=O)CC2)=O)nnc(O)n1C CC1CC(NC(C2CCCCCC2)=O)CCN1C(c1cc(F)c[nH]1)=O Cn1cc([N+](=O)[O-])c(C(=O)NC(CNC(=O)C=CC2(C)CCOCC2)CO)n1 c1(-c2cn(C3CN(C(c4n(C(C)C)nc(Br)c4)=O)C3)nn2)cc(F)ccc1F C1(C(N(CCOCCNC(C(CC)OC)=O)C)=O)CC(=O)c2ccccc2C1 c1(C(NNC(=O)NC(c2sccc2Cl)C)=O)cccc2ccccc12 S(=O)(=O)(CCC(F)(F)F)N1CC(NC(C2CC3CCC2NC3)=O)C1 c1(OC)cccc(C(=O)OC)c1.c12csc(c1)C(C(=O)NC1(C)CC1)N(C)C2C C1(CNC(CCN(c2ccncc2)C)=O)CCCCN1C(C12CCOCC1C2)=O c1(-c2cc(C(NCOCCc3ccccc3)C)ncc2)ccc(F)c2[nH]ccc12 N1(C(C2CC2COC)=O)CC2CC(NC(C(C)Sc3ccccc3)=O)CC(C2)C1 c1(N2CCC(c3nccc(F)c3)C2)nc2ccccc2nc1NCC1CCSC1 C1(CCNC(C=CCC2(NC(C(C)(C)OCC)=O)CCC2)=O)OCCCC1(C)C c1(NC(c2nc(NC(c3ccc(OC)o3)=O)sc2)=O)cnnc(O)c1Cl C1(C(=O)NCCN(C(Cc2cn(CC)nc2)=O)C)CCCCC1(F)F c1(C(N2CC(F)(CNC(c3ncn(C)n3)=O)C2)=O)cc2ccccc2[nH]c1=N C1(C)(NC(C(CCC)=CCC)=O)CCN(C(=O)C(O)Cc2ccc(F)cc2)CC1 c1(C(=O)NCC(C2CC2)NC(C2COC2)=O)cc(Cl)c(Cl)s1 C1(N(C(=O)CC2CC3CCC2C3)CC)CCN(C(=O)CCn2ccnc2)CC1 Cc1occ(-c2ccccc2)c1C(N1CCC(NC(=O)CC2CC23CC3)C1)=O CC(C)(CNC(N1CCC(CCO)C1)=O)Cn1cc(CCCC#N)nn1 Cc1c(C(=O)N(C(C)CCNC(C2CCC2)=O)C)csc1Br N1(C(CC2(OC)CCC2)=O)CCC2CN(C(=O)Cc3cccn3C)CCC2C1 CC(CF)C(=O)NCCC1CN(C(=O)C(C)OC2CCOC2)C1 CC1CC(C(=O)N2CC(O)(C(F)C(=O)NC3CCCCC3(C)C)C2)=NO1 C(C(=O)Nn1nnc2c1CCCC2)(CC(C)C)NC(c1c(C)cncn1)=O CC(O)(CNC(=O)CCN(C(C1CC=CCC1)=O)CC1CC1)CCO C(=O)(CCC(C)CN(C)C)NCCC(CCNC(c1nn(CC)c(C)c1)=O)C C(=O)(C(C#N)C(C)(C)C)N1C(C)CC(CNC(CC2(CSC)CC2)=O)C1 C(=O)(C1=CCN(C(c2cc3ccccc3o2)=O)CC1)NC(C1CCC(O)CC1)C c1(C(=O)NCC2OCC(CNC(c3ccc[nH]3)=O)C2)oc2ccccc2c1Br CC1(C)CC(NC(=O)Cc2cncnc2)CN(C(=O)CNS(=O)(=O)C2CC2)C1 N1(C(c2n(COC)ncc2)=O)CCN(C(C2CCCCC2C(N)=O)=O)CC12CC2 c1(C(=O)NCC2(O)CN(C(CC(C)OC)=O)C2)cccc(OC(C)C)c1 N1(C(c2nc(C)[nH]n2)=O)CCCCC1CN(C)C(C1(c2ccncc2)CCC1)=O CC1OCC2(CCC(NC(N3CC(c4cccc(Cl)c4)C3)=O)O2)C1C N1(C(CC2(COC)CC2)=O)CCC(NC(=O)CC23COC(C)(C2)C3)C(C)(C)C1 C1(C)(C(N(C)CC2(O)CN(C(C(c3cccc(F)c3)C)=O)C2)=O)CCSCC1 N1(CCOC)CCC(NC(=O)C=CC(C)(C)NC(=O)C=CC2CCOC2)C1 N1(C(C(COC)OC)=O)CC2(CC(CC(=O)N(C3CC3(F)F)C(C)C)C2)C1 CCC(CC)C(=O)NCC(CO)NC(=O)C(Cc1ccccc1)CC N1(C(CSC)=O)CC(O)(CCNC(=O)CCOCC2CCCO2)C1 c1(-c2cccc(NC(C)C(=O)C3CC3)c2)ccc2c(c1)COC(C)(C)O2 N1(C(c2ccc(F)cc2)=O)CCC2CCCN(C(c3cc4[nH]ccc4s3)=O)C2C1 C1(C(=O)OCC23CC(C2)C(C(F)(F)F)N3)CCCCC1Cc1ccccc1 n1(CC)cccc1C(=O)NC1(C2CCCN2C(C2CC2[N+](=O)[O-])=O)CC1 N1(C(C2(SC)CC2)=O)CCC(N(C)C(C2(N(C)C)CC2)=O)CC1 C1(CC(N2CCC(C)CC2)=O)C2CCCC2N1C(c1cc(Cl)n(C)n1)=O C(CCCCNC(c1sccc1NS(C)(=O)=O)=O)N(C)C(c1cn[nH]c1)=O C1(OCC)CC(CNC(=O)C(C)NC(N)=O)N(C(c2[nH]c(O)nc2C)=O)C1 C12(NC(C3(CC=C)CC3)=O)COC(CNC=O)(C1)C2.c1ccc(-c2cscn2)cc1 C1(CC(=O)NCCC2(OC)CN(C(=O)C(F)=C(C)C)C2)CCCC(O)C1 N1(C(Cn2nnc(C)n2)=O)CCC(NC(C2(C(F)(F)F)CC(F)C2)=O)C(O)C1 C1(C(=O)NCCNC(c2c(CC)con2)=O)C2Cc3c(Br)cccc3C12 C1(NC(c2cn3ccsc3n2)=O)CC(O)(C2CCN(C(=O)C(F)(F)CO)CC2)C1 N1(C(C(CNC(C2(C#C)CC2)=O)(C)C)=O)CC(C)OC(C)(C)C1 c1(C(N2CCC(NC(C3CCSCC3)=O)CC2)=O)ccc2cnnc(O)c2c1 S1(=O)(=O)c2cc(Cl)ccc2N1.n1(C(C)C)ccc(NC(=O)N(C)C)n1 CC1(CNC(C2CCSC2)=O)CCN(C(=O)CCCC2CCC2)CC1 C(=O)(C(F)(CNC(=O)C(C)(C)C1CCC1)C(C)C)Nc1cncc(C#C)c1 Cc1cnc2cccc(C(N3CC(NC(=O)Cn4cncn4)CC34CCC4)=O)n12 c1(C(CCC(=O)N(C(C)CNC(C2(C)C=CCC2)=O)C)=O)ccc(F)c(F)c1F c1(C(N2C(CNC(C(CC#C)C)=O)COCC2)=O)cccc(C#CCO)c1 N1(C(C2C(C=C)C2)=O)CCN(C(c2c(C)ccnc2O)=O)CC1CCCC N1(CC(C)NC(C(C=C)O)=O)CCN(C(C2(C3CC3)CCC2)=O)CC1 N1(C(CN2CCN(CC)CC2)=O)CCC(C)(NC(c2ccc(C#N)s2)=O)CC1 c1(C(CNC(C2COCCN2C(=O)C2=C(Cl)CC2)=O)O)c(Cl)cccc1Cl N1(C(Cc2cc(COC)on2)=O)CC(NC(C2CC(C)=NO2)=O)C(C(F)(F)F)C1 n1(CCNC(C=C(CC)CC)=O)ccc(C(=O)N(CC)CC2COC(=O)N2)c1 CC1=C(C)CC(C(=O)NC2CC2CNC(C23CCC(CC2)CC3)=O)CC1 C1(C(=O)NC2CC(NC(c3cn(CCC)nc3C)=O)C2)CCN(C)C(C)C1 c1(C(=O)NCC(CN(C(C2CCC2)=O)CC)(C)C)c(C)ncn1C CN1CCN(C(c2ccc(C(N)=O)s2)=O)C(CNC(c2cnn(C)c2N)=O)C1 C(=O)(CC(C)CC(F)(F)F)N(C1CCCC1)CCNC(C(C)=CC)=O c1(C(c2nnnn2C2CC(F)(F)C2)NCCCSC)cc(F)c(N(C)C)cc1Cl c1(CNC2CC(NC(=O)NCCc3ccccc3Br)C2)cccc(I)c1F C(CC(C)(C)C)(C(=O)NCc1nc(CO)no1)NC(CN(CCOC)C)=O N1(CC(=O)NCCCC(C)NC(=O)CCSC(F)(F)F)CCCCS1(=O)=O C1(CNC(CCC)=O)CC(NC(=O)C=C(C)c2cccs2)CCO1 C1(C(=O)NCC(C)N(C(c2c[nH]nc2Br)=O)CC)CCC=CCCC1 Cc1ncnc(C(=O)NC2CC=C(C(=O)NC3(C)CC(C(=O)OC)C3)C2)c1C Cc1ccc(O)cc1CCCC(=O)NC1CCC(c2cn(C3CCC3)nn2)CC1 Cc1csc(C=CC(=O)NCC(C(C)C)NC(=O)COc2ccon2)n1 c1(C(=O)NCC(CC)NC(=O)CCNC(C2CCC2)=O)cc(Br)n[nH]1 Cc1cc(C)c(C(N2CC(O)(C(C)NC(C3(C)CCCC3)=O)C2)=O)c(Cl)n1 c1(C(=O)NCCCN(C(C(C)=C2CC2)=O)CC2CCCC2)c(Cl)cc(Cl)nc1N C(C(F)(F)CNC(=O)C(CC1CC1)OC)OC.C(=O)C(CO)OC c1(C(=O)OC)cc(C(C(=O)NC2CC2)N(C2CC(C#N)C2)Cc2cncs2)no1 c1(C(=O)NC23CC(CNC(c4ccc(Br)o4)=O)(C2)C3)cccc2nc[nH]c12 C1(NC(c2noc(CC)c2C)=O)CCCC12CN(C(=O)CC1COC(C)(C)C1)C2 CON(CCC(=O)N1CC(NC(C)=O)C(C2CC2)C1)C(=O)OC(C)(C)C C12CN(CC(C)(C)C1)C(=O)Cn1cc2nn1.C(COC1CCC1)(C1CCC1)OC C1(CCOC)CN(C(=O)CCC(=O)c2ccccn2)CCN1C(C1CC(F)C1)=O Cc1cc(F)cnc1C(=O)N(CCCCCCNC(=O)C(C)CC1CCCC1)C N1(C(c2ncc(C(C)C)s2)C(=O)NCCCF)CCCC2(CCCCC2O)C1 CC(C)CC(C(=O)NC(C)CNC(=O)Cc1coc(C(F)F)n1)N1CCCC1=O c1(CC)ccc(NC(=O)C(C)(C2CCC2)NC(=O)C(N2CCOC2=O)C)c(C)c1 c1(C(N2C(C3(NC(C4N(CC)CCC4)=O)CC3)CCC2)=O)cnn2ccccc12.OCC c1(C(N2CCN(C(COC(C)C)=O)C(C3CC3)C2)=O)cc2cn[nH]c2cn1 c1(C(=O)NC2CCN(C(CC(c3ccc(O)cc3)C)=O)C2)cn2c(n1)COCC2 N1(C(COCCC=C)=O)CCCC2(CCCN2C(C2OCCO2)=O)C1 c1(C(C)C)nnc(C=CC(=O)N(C)CCN(C(C2(F)CCCC2)=O)C(C)C)o1 C1(F)(CNC(=O)Cc2cnns2)CCC(CNC(=O)C(F)(F)c2ccncc2)C1 C1(NC(Cc2c(CC)cccc2)=O)CCC2CN(C(=O)CCNS(C)(=O)=O)CC2C1 N1(C(C2CN(CC)C(=O)C2)=O)CCC(C(=O)N2CCC(C)C(C)C2)=C(F)C1 c1(C(N(C)CC2CCCN(C(C(C)C#N)=O)C2)=O)cc2cccnc2cc1F C1(C(=O)NC(c2nccs2)CC)CCCN(C(C2CC3(CSC3)C2)=O)CC1 C1(NC(=O)OC(CNC(COCC)=O)C)CN(C(C)=O)CCC1C(F)(F)F CC(Cn1ccnc1)C(=O)NCCCNC(C1CC(F)C1)=O C1(CNC(C(CC)(C)O)=O)CCCCN(C(c2c(C)nc(C)nc2O)=O)CC1 c12ncccc1S(=O)(=O)N2.C1(CC)CCCCC1N(C)CC1CC1 c1(CC(=O)NCCC(C)(C)NC(C2C(C)C2)=O)c[nH]c2cc(Cl)ccc12 S(=O)(=O)(c1cc(C)ccc1NC(C)C(C)(C)O)NC(CCCC(=O)NCC)=O C1(C)(C(N2CCCC(N(C(C=CC(C)(C)C)=O)CCO)C2)=O)CCC(F)(F)C1 c1(C(N2CCC(c3cccc(NC(C)=O)c3)C2)C)ccc(C#N)cc1F CCCCC(C)C(=O)NC1(COC)CN(C(=O)CC2CCC(C)O2)C1 c1(NC(=O)COC(=O)CSc2cn[nH]c2)cccc(COC)c1 C(=O)(C(CC(N)=O)NC(C1CC12CCC2)=O)N1C(C)(CCO)CC1 C1(C(=O)NC(CCNC(C=C(CC)CC)=O)C)CCC(Nc2nccs2)CC1 C1(CC(C(=O)N)N(N2CCCC2)C)CC(C)(C)OC(C)(C)C1.c1(CC)cccs1 N1(C(c2ccc(N)c(F)n2)=O)CCC(C2CC(NC(=O)Cc3cn[nH]c3)C2)C1 N1(C(c2c(CC)c(F)ccc2)=O)CCC(C)(C)C(CNC(=O)CC23CC(C2)C3)C1 CC1=C(C(=O)N2CCC(NC(c3[nH]cnc3C)=O)C2C)C(=O)OC1(C)C c1(C(N2CCC(N(C(=O)C(F)=C(C)C)CC)CC2)=O)ccc2nc(C)ccc2c1 CCC(C(=O)N1CC2CC1CN2C(c1cnc2ccoc2c1)=O)C(F)(F)F C#Cc1ccc(OC)c(C(N2CCC(C)(CNC(c3cccs3)=O)C2)=O)c1 C1(NC(=O)C=CBr)COCCN(C(=O)CCc2cccc(F)c2Cl)C1 c1(C(=O)NC(CC)CN(C)C(c2cc(C)no2)=O)cncc(C(=O)OC)c1 c1(NC2CC(NC(C(c3c(C)noc3C)C)=O)C2)nccc(C#N)n1 c12ccc(cc1)NC(C(C)C)CCN(C)C(=O)C1CC21.C(=O)(C1=CCCO1)OC C(=O)(C(CC)C(F)(F)F)N1CC(C#C)(C(=O)NCCOC(C)=O)C1 C1(C(=O)NCC2(CNC(COCCCC)=O)CCCC2)C(C)(C)C1(F)F c1(C(N(CCCNC(C(CC)CN2CCCCC2)=O)C)=O)c(Cl)c(C)nn1C Cc1cc(C(C)C(=O)NC2CN(C(=O)C(C)CCO)C2)cc(C)c1 c1(C(C)C)cncc(C(=O)NCC2CC2CNC(C2(C(C)C)CC2)=O)n1 C(C)(CC(=O)NCCC1CCC(NC(=O)Cc2cccnc2)C1)OC C1(NC(COCCC#C)=O)CCOCC1NC(=O)C(c1cccnc1)O c1(C(N2C(CCNC(c3ccnn3CCF)=O)CCC2)=O)cn2ccsc2n1 CC1(C)CCCCC(C(N2CC(NC(c3ncccc3O)=O)C2)=O)C1 c1(C(=O)Oc2c(SCC)cccc2)c(Br)nn(C)c1C N1(CCN(C(CCC=C)=O)C)CCN(C(C2ON=C(C)C2C)=O)CC1 c1(C(N(CC(C)NC(CCC=C)=O)CC)=O)ccc2c(Br)cnn2c1 C(=O)(C(C(C)C)n1cnnn1)N(CCN(C(=O)C(C)(C)C)CC)CCSC C1(OC)CCCC1C(N1CCCC1CN(C(=O)C=Cc1ccsc1)C)=O N1(C(C=CCCC)=O)CCC2CC2(NC(c2cnn(C)c2C)=O)CC1 c1(C(=O)NC(CCOC)CNC(=O)CCCc2nccs2)cccnc1Cl c1(C(=O)NC2C(NC(c3n(C)c(S)nn3)=O)C2)cnc(O)c2cccnc12 C1(CC#C)(C(=O)NCC2CC2[N+](=O)[O-])CCN(C(c2sc(F)cc2C)=O)C1 CC1(CNC(=O)Cc2cscn2)CCCN(C(=O)CCC2NC(=O)NC2=O)C1 c1(C(=O)OC)cccc(S(=O)(=O)N2CCSC(C(N3CC(C)C3)=O)C2)c1 c1(C(=O)NCc2n(CC)cnc2)cc(=O)oc2ccc(O)cc12 Cc1c(C(N2CC3(CCN3C(C3C=CCC3)=O)C2)=O)sc2nnc(S)n12 C1(NC(Cn2ncc(C)c2)=O)C(C)CCN(C(c2cc(O)cc(N)c2Cl)=O)C1C c1(Sc2occ(C)n2)ccc(C)c(C(N2CCCCC2)C)c1 Cc1ccc(C(=O)NC(C(=O)N(C2CCOC2)CCO)C2CC2)o1 C=CCC(CC)N=c1nc(N(C)Cc2noc(C)n2)c2cnn(C)c2[nH]1 c1(SCCNC(c2n(CCC)nnn2)c2ccon2)ccccc1Br c1(C(=O)NCC2C(NC(CCCCNC(C)=O)=O)COC2)cc2sc(C)cc2s1 c1(CC(=O)NC(CCN(C(C2C(=C)C2)=O)C)C)sc(C2CC2)nc1C Cc1cc(=NC(=O)C2CCCC23CCN(C(=O)CCc2ccsc2)C3)[nH][nH]1 N1(C(CC2N(C)CCCC2)=O)CC(CNC(c2cc(C(F)F)no2)=O)CC1(C)C C1(NC(C2C=CCC2)=O)CC2(CCN1CC=CC(=O)OC(C)(C)C)CC2 N1(C(c2c(SC)cccc2)=O)CCCC(N(C)C(c2ccc([N+](=O)[O-])s2)=O)CC1 C1(NC(Cc2ncc(CC)[nH]2)=O)CN(C(c2cc(O)nc(O)n2)=O)CC(C)(C)C1 C12(CNC(C3CCCC3)=O)CC(CCO1)N(C(c1cccc(CF)c1)=O)C2 c1(NC(C(C)C)=O)cccc2c1C1CN(C(=O)COc3ccccc3Br)CC1O2 N1(C(C2CC(OC)(OC)C2)=O)CCC(NC(=O)C(c2ccc(C)cc2)C)C1(C)C C1(CNC(C(CCOC)C)=O)CC(NC(=O)C(=O)NC2CC2)C12CCC2 N1(C(c2cc(C(F)F)ccn2)C(=O)NC2CC2)CCC(C2CCCC2)C1 c1(N(C(=O)NC(C2(C)CSC2)=O)CCNC(=O)OC(C)(C)C)cnn(C(F)F)c1 CN1C(=O)CCCC1C(=O)NC1(CNC(C2(C3CCCO3)CC2)=O)CCCCC1 CCCC(C(=O)OC)C(=O)NC1CC1CNC(=O)CC1(COC)CC1 C1(C(COC)(C)C)(NC(=O)CC2(C)OCCO2)CCN(C(=O)C=C=C(C)C)C1 c1(C(N2C(CNC(C3(CF)CC3)=O)CC(OC)C2)=O)cc(Cl)c(Cl)c(Cl)c1 c1(C(=O)NC2CC3CC(NC(=O)CCc4csnn4)C2C3)ccc2nncn2c1 C(C(C)(CC)C(=O)NCCn1ccc(=O)cc1)NC(CCC(=O)NCC)=O N1(C(C2(C#C)CC2)=O)CCC(CO)(NC(=O)CCC(=O)c2ccc(C)cc2)C1 C(CCC(=O)NC(C)(CNC(C1CC1C(F)(F)F)=O)C1CCC1)N(CCC)CCC c1(C(=O)NCC2(F)CCCN(C(c3nc(=N)[nH]cc3)=O)C2)ccnc2cc[nH]c12 N1(C(c2nc(COC)oc2)=O)CC(C)CN(C(c2cc(Cl)no2)=O)CC1C C1(CC(=O)NCC(C)NC(=O)C(C)c2ccsn2)CC(F)(F)C1 c1(C(C(=O)NC2CC(C)(NC(C(CC)F)=O)C2)(F)F)ccccc1C C(=O)(C1=Cc2ccccc2OC1)N1CC(NC(=O)CC2CC(F)C2)C(C(F)(F)F)C1 C1(NC(C2(C(C)C)CCN(C(C3(COC)CC(=O)C3)=O)C2)=O)CC2CC1C(O)C2O N1(C(c2cccc(Cl)c2OC)C(=O)NCCCCCC)CC2OC(=O)N(C)C2C1 N1(C(c2cc(CCC)[nH]n2)=O)CC(NC(=O)CC2CC=CCC2)CC(C)C1 N1(C(c2nc(COC)oc2)=O)C2CCC1CN(C(=O)CCC=CBr)C2 C12(CNC(C(=O)NC(C)C)=O)CCC(CN1C(=O)C(C)C(C)(C)C)C2 C(=O)(C(C)(C)C(=O)N(C)CC1C2CN(C(=O)CC3COCCO3)CC12)OCC C=CC(C)(CCOC)C(=O)N1CC2(C1)CN(C(c1cn(C3CC3)cn1)=O)C2 C1(CCC)CCCN(C(C23CC2CN(C(=O)CC(C)SC)C3)=O)CC1 c1(CNC(C2C=CCCN2C(=O)CC2CC(=O)C2)=O)ccc(C2CC2)cc1 c1(C(=O)NCC2CCCN(C(c3c(C#C)c[nH]n3)=O)C2)cnc(C)cc1Cl Cc1ccc(CC(=O)NC2CCC2CNC(C2CCCSC2)=O)cc1 C1(F)(C(N(C2CCCO2)CC)=O)COCCN(C(=O)C=C(C)CN2CCOCC2)C1 C1(CNC(c2ccccc2CCCO)C)CC(C(=O)OC(C)(C)C)N(OC)C1 c1(C(N(CCC)CCNC(=O)Cc2nc(C)sc2C)=O)ccc(OC)c(C)c1 Cc1ccc(C(=O)NC(CCN(C)C)C(C)C)c(I)c1 C(CC(O)C(=O)NCc1ccccc1OC1(C(=O)NC)CC1)N(C)C.CC(F)F c1(C(C(=O)NC(CCNC(C2(CCC)CCC2)=O)C)C(C)C)c(F)cccc1F N1(C(C(CC)C)=O)CC(NC(c2ccc3nncn3c2)=O)CC(F)(F)C1 C(=O)(C(C)CC=CCC)N(CC(=O)NC(CC=C)CC)CC O=C(CCCCNC(=O)C1CC1)OCCCSc1ccccc1 CC(CCNC(C1Cc2ccccc2C1)=O)CC(F)(F)F CC1CCc2onc(C(N3CC(C(C)NC(=O)CCCC#CC#N)C3)=O)c2C1 Cc1nn(C)cc1C(=O)NC(CCN(C)C(C1CCC(C)CC1)=O)C(C)C c1(CCNC(C2(COC)CC2)=O)cc(C)n(-c2ccc(SC(N)=O)cc2)c1C Cc1cccc(CNC(C2CCC(CO)N2C(=O)Nc2ccc(F)cc2F)=O)c1O Cc1cc(C(N2CCCC(F)(C(=O)NC(c3ccncn3)C)C2)=O)ccc1O CC1(C)COCC(NC(=O)C(CNC(C2CCO2)=O)CC2CCCC2)C1 Cc1ccc(-n2cccn2)c(OC2CCC(Nc3nccc(N(C)C)n3)CC2)c1 C1(C2CN(C(=O)C=C(C)Cl)C2)(NC(C2CC(C(F)(F)F)(OC)C2)=O)CC1 N(C1CCCc2ccoc21)C(C1(C)N(C(C2C3CN(C)CC32)=O)CC=C1)=O c1(N(C)Cc2ccoc2)nc2c(c(=NCC3(C4CC4)CC3)[nH]1)CCCCC2 C=CCC(C)(O)C(=O)NC(c1cn(C)nn1)C(=O)NCCC(O)C(F)F c1(C(=O)NCC(CNC(CC2N(CC)CCOC2)=O)O)cc(F)ccc1F C1(C(N2C(CNC(c3coc(-c4ccccc4)n3)=O)CC2)=O)COCOC1 CCC(C(=O)N1CCN(C(c2ccn3c(Br)cnc3n2)=O)CC1)C(C)(C)CC C(CN1C(=O)Cc2ccccc21)NCc1cc2cccc(OC)c2o1 c1(C(=O)NCC(CNC(C(CN(C)C)NC(C)=O)=O)F)ccc(Cl)c(Cl)c1 CCC(CC)C(C(=O)N1CCCC1CCC(=O)Nc1cccc(Cl)c1)OC C12(C(N3CCC(NC(=O)CCOC4CC4)C(F)C3)=O)CC(CO)(C1)OC21COC1 Cc1c(C(N2CCC(CNC(=O)C(c3ccc(Cl)cc3)=O)CC2)=O)cccc1F Cc1cc(F)cnc1C(=O)N(C1CCN(C(C2CC(C)(F)C2)=O)CC1)C C1(C(N2C(C)(CNC(c3ccc(Cl)nc3)=O)CCC2)=O)CCOCC12CCC2 Cc1ccc(C)s1.C(=O)(C(C)S)NCC(N(C(=O)CNS(C)(=O)=O)C)C1CC1 c1(OC)oc2ccccc2c1COC(=O)NC1(CO)CCC1COC.C1(=O)CN1 Cc1nc(N2CCCCC2CNC(C2(C)CCCNC2=O)=O)ncc1Br N1(C(C2N(C(c3c(NC)cccc3)=O)CCCC2)=O)CCN2CCCCC2C1 c1(C(N2CCC(C(C)NC(C(C)=CC)=O)C2)=O)ccc(Br)cc1O c1(OC)cc(C)c(C(=O)NCCNC(=O)C2=NNC(=O)CC2)cc1OC CC(C)(CCCNC(C1CCN(C(=O)C=CCSC)C1)=O)NC(=O)OC(C)(C)C C1(O)(CCNC(C(CC=C)C)=O)CCN(C(c2cn(C(F)(F)F)cn2)=O)CC1 c1(C(N2CCCC(CN(C(=O)CC3CCCO3)C)C2)=O)ccc(C2CC2)nc1O c1(C(N2CCC(C)C2CNC(=O)Cn2cc(Cl)cn2)=O)cc(O)cc(F)c1 C1(CNC(C(CC)c2ccccc2)=O)CCC(C)(C)CN1CCC1(O)CCCC1 c1(C(N2CC3=C(CN(C(CCN(C(C)=O)C)=O)C3)C2)=O)ccc(F)c(C)c1C#N S(=O)(=O)(c1ccc(NC2C=CCC2)cc1Br)NCC1CC(C)(C)OC1(C)C CCC(CCC(=O)NC(C)(CC)CCO)NC(c1ccc(OC)nn1)=O c1(C(=O)NC(CC=C)CNC(=O)CCc2ncc(C)[nH]2)cc(C)c2[nH]cnc2c1 C12(C(=O)NC3(CC=C)CN(C(=O)C=CC(C)(C)C)C3)CC(C)(C1)OC2C N1(C(c2c(C)ccs2)=O)CC(C(N2CCSCC2C2CC2)=O)C2(CCC2)C1 O=C(C1=CC2CCCCC12)N(CCNC(=O)COCCF)Cc1ccccc1 c1(C(=O)NCC(O)CNC(C2CC(F)(F)C2)=O)cc(Cl)ccn1 Cc1cc(C(N2CC(NC(c3ccc(C)s3)=O)CC(C)C2)=O)n2ncnc2n1 N1(C(C2CN(C(=O)OC(C)(C)C)C2)=O)CCOC(c2ccccc2)C1 C1(CC)C(C(=O)N(C)CC2CCCCC2)CCN1C(C1COCC1C(N)=O)=O C1(C(=O)Nc2cccc(CC)c2)CCC(C)N(C(c2cc(F)ccc2F)=O)C1 C(=O)(C1=CCCCO1)N1CCC(CC(N)=O)(NC(c2c(C)nn[nH]2)=O)C1 c1(N(CC(C)NC(=O)CN2CC3CC3C2)C)ccnc(C2CCCC2)n1 Cc1cc(C(=O)N(C)CC2CCCN2C(c2cscn2)=O)ns1 CCCCC(C(=O)N(C)CCOCCNC(=O)Cc1cncn1C)C(C)C N1(C(C2(COC)C=CCC2)=O)CCN(C(=O)C=C2CCC2)C(CF)C1 c1(C(=O)NCCN(CC(C)O)C(c2cc(C(C)C)nn2C)=O)cnn2c1OCC2 C1(CC(C)NC(=O)CC2(O)CCC2)CN(C(=O)COC2CCC2)C1 CC(C)C(C)(O)C(=O)NCCn1cc(CNC(=O)C=Cc2cc[nH]c2)nn1 N1(C(CCC(C)OCC)=O)C2CCC1CC(NC(=O)C=CC1CCCC1)C2 N(C(=NCc1ccccc1F)NC1CC(NC(=O)COC)C1)C(CC)CC Cc1nccn1C(C)C(=O)NCC1(NC(C2(C3CCCO3)CCC2)=O)CCCC1 Cn1c(C(=O)NC2CC2CNC(C2CC=CCC2)=O)nnc1S c1(CCC(=O)NCC(C)CNC(C2(C#N)CC2)=O)c(F)cccc1F c1(N2CCOCC(CNC(=O)CCc3cncs3)C2)ncnc2[nH]ccc12 C(=O)(CCC(CF)CF)NC1C2CC(C(=O)NC(C)(C)CCF)C(C2)C1 C#CCCCCCCC(=O)NC1CCCN(C(=O)CC(C)(F)F)CC1 C(C(O)CC(=O)NC1CCC(=O)NC1)NC(C=C(CC)CC)=O c1(C(=O)NC(CC)CN(C(C2(O)CCSC2)=O)CC)cc(N)ccc1C C(N=c1[nH]c(=N)[nH]c(=NCC(F)(F)CC2CC2)[nH]1)C1N(C)CC(O)C1 c1(C(=O)NCC(CNC(C(C(C(C)C)O)(C)C)=O)O)nc2cncnc2nc1O CC(C)C(C)C(=O)NC1CCOC1C1CCN(C(C2(O)CC(F)(F)C2)=O)CC1 c1(OCC(=O)NCC2N(C(C(C)=C(C)C)=O)CCOC2)ccc(F)c(Br)c1 C12(CNC(C3CC34CCOCC4)=O)CCCC1CN(C(c1sccc1Cl)=O)C2 S(=O)(=O)(c1ccc(F)cc1)NC(=O)CCNC1CN(C(=O)C(F)(F)F)CCN1 N1(C(C(C)C2CCCO2)=O)CCOCC(NC(=O)COC2CCOCC2)C1 C1(CCNC(C2(C(C)C)CCC2)=O)(OC)CN(C(c2scnc2C)=O)C1 Cc1cc(=NC(=O)C(=O)N(C)C[Si](C)(C)C)[nH]n1CCC(C)(C)C N1(C(c2c(CC)ncnc2)=O)CC(C(=O)NCC(C)(C)C2CCC2)CCC1(C)C CCC(C)C(C(=O)NCC1(C(N2CC3C=CC3C2)=O)CCC1)N(C)C c1(C2C(C(=O)NC(C(C)NC(C(C)O)=O)CO)C2)ccc(N2CCCCC2)c(F)c1 c1(C(=O)NCC(CCNC(CSCCOC)=O)OC)cnn(C)c1C1CC1 N1(C(=O)NC)CCCC1CNC1(c2nnnn2CCCF)CC(OC)C1 N1(C(C(COC)C)=O)CCN(C(=O)C(C)=C(C)C)C(CCO)C1 C(=O)(C1=C(F)CN(C(=O)CSCc2ccccn2)CC1)NCC(C)C1CC1 Cc1ccc(NC(C2OCCC2CNC(c2ccccc2)=O)=O)cc1C Cc1ccc(C(=O)NCC2CCCC(NC(c3ncoc3C3CC3)=O)C2)nc1O N1(C(c2cc(CC)nn2C)=O)CC(NC(c2ncc(Cl)cc2F)=O)C2(CCC2)C1 c1(C(N2CCC(O)(CNC(C(C(C)C)SC)=O)C2)=O)cccc2cc[nH]c12 N#Cc1c(NC2CC(F)CN(C(=O)C3=NNC(=O)CC3)C2)cccc1Cl C1(OC)CN(C(=O)C(CC)Oc2nc(C)no2)CC1C(=O)NOCCCC1CC1 C(C(CCC)NC(c1nnc(C)s1)=O)NC(C(C)OCC=C)=O CCCCC(CC)C(=O)N1CC(NC(c2ccc(F)o2)=O)C1 C(CC(=O)N1CC2CCCC(C2)C1)(C(F)(F)F)NC(C1CC(N(C)C)C1)=O c1(OCC(=O)NC2CCN(C(c3cc(CC)no3)=O)C2)ccc(Cl)cc1Cl N1(C(C2CC(C)OC2)=O)CC2(CCN(Cc3cnon3)CC2)C1 C1(CN(C(N2CCCC(C)(c3cccc(F)c3)C2)=O)C2CC2)CCC2(CCC2)CO1 c1(C(N2C(C)(C(=O)Nc3ncc(F)cc3O)CC2)=O)cccc2nccnc12 C(=O)(C1=CS(=O)CCC1)NC1CCCN(C(c2n(CC)ccc2)=O)CC1 Cc1ccc(NC(C2CN(C(C3CCCC34CCC4)=O)CC2F)=O)c(O)n1 c1(NC(=O)CC2CN(Cc3ccc(C(F)F)cc3)C2)cc(C(F)(F)F)ncc1I c1(NS(=O)(=O)CCc2cn[nH]c2)cccc2c1OCCC2 C12CCN(C1)C2(C)C.N1(CCCN(C(=O)CCN(C)C(C)=O)C)CCOCC1 N1(C(C=CC=CC)=O)CCN(C(c2coc(-c3ccccc3)n2)=O)CCC1C N1(C(C(CCC)C)=O)CCN(C(C2CN3CCC2CC3)=O)C(COC)C1 C12(NC(c3c(F)ccc(O)c3F)=O)CC1COC21CCC1 C1(C(=O)NC(c2ccc(C)s2)C)CCn2cncc2C1 CCCCC(C)CCC(=O)NC1CC1C(=O)Nc1cccc2c1CCO2 CC1CN(C(=O)CC(C)(C)c2ccc(F)cc2)CC1NC(c1c[nH]c(=O)cn1)=O c1(OC)ccc(C(F)F)cc1C(=O)NCC12CC1CN(C(C1CNC(=O)N1)=O)C2 C1(NC(c2ccc(NC(N)=O)cc2)=O)COCCN(C(=O)CSC(F)(F)F)C1 N1(C(c2c(CC)nc[nH]2)=O)CCCC(N(C)C(C2(C)CCC(F)(F)C2)=O)CC1 CC(C)(C(=O)NCC1(CCNC(C2CC3(CCOC3)C2)=O)CC1)S(C)(=O)=O C#Cc1cccc(C(=O)NC2CCCCC2(C)CNC(C23CC(F)(C2)C3)=O)c1F C=C=C(C)CC(=O)N1CCC(N(C(C2(N3CC4CC4C3)CC2)=O)CC2CC2)CC1 Nc1cnc(C(N2CCC(O)(CCNC(c3cnncc3O)=O)CC2)=O)c(Cl)c1 C1(CC)CN(C(c2nc(O)sc2C)=O)CCN1C(c1cc(C2CC2)ccc1Cl)=O C(=O)(CN=c1ncnc2[nH][nH]c(Br)c1-2)Nc1ccc(OCC=C)cc1 C1(C(=O)NC(C(C)NC(c2[nH]nnc2C(F)F)=O)C)CC2(CCO1)CC2 c1(OCCC(C)C)ccc(CNC(=O)NC2CCCC(F)C2)cc1 Cc1cc(=NCC(C2CCCCC2)NC(=O)COCCCC(C)C)[nH]cn1 Cc1ccc(CCC(N2CC(NC(=O)Cc3ccccc3C)C(F)C2)=O)c(C)c1 CC1(C)CCC(CO)N(C(C2CN(C(=O)Cn3cnc(=N)[nH]3)CC2(F)F)=O)C1 C1(C(=O)NCC(CNC(=O)C(c2cccnc2)O)CO)CC12CCSCC2 CC1(C)OC2(CN(Cc3cncs3)C2)CO1 N1(C(CSCCCC)=O)CCN(C)C(CNC(=O)COC2CCOC2)C1 N1(C(C(C)SCCCC)=O)Cc2ccccc2C(NC(c2cnc(S)[nH]2)=O)C1 C1(C(N(C2(NC(CN(C(=O)OCC)C)=O)CC2)C)=O)CC2(CC(=O)N2)C1 C1(NC(C(COCC)n2cc(-c3cc(CC)no3)nn2)=O)CCN(CC)C(C)C1 C(=O)(C(O)CCCc1ccccc1)N(CC(C)(C)NC(C1N(CC)CC1)=O)C N1(C(CCc2ccn(C)n2)=O)CC2OCCN(C(C3CCCN3C=O)=O)C2C1 C=CC(CC(=O)N1CC(NC(c2csc(C#N)c2)=O)C(O)C1)c1ccccc1 c1(C(=O)NCC(CNC(c2cccc(OC)n2)=O)CO)cccn(C2CC2)c1=O C1(N(C(=O)C=CC2(C)CC2)C)CN(C(=O)C(c2cccc(C(F)(F)F)c2)O)CC1O C#CCCCC(C)C(=O)N1CCCC1C(=O)NC(c1ncc(C)o1)C c1(OC)ncc(Cl)cc1C(=O)NC1CC(CNC(=O)C(O)c2ccco2)CC1O c1(C2(C(N3C4C(NC(CCSC)=O)C(C4)C3)=O)CC2)ccc([N+](=O)[O-])c(C)c1 O=C(CC1=CCOCC1)N1CCCCC1C(N1CCCC(CCO)CC1)=O C1(NC(c2cc(SC)oc2C)=O)CCSC12CN(C(=O)C(c1ccccc1)F)C2 N1(C(CCCC)=O)CCN(C(=O)C(CC(C)C)Oc2ccccc2)C(C2CCC2)C1 C1(C(=O)NNC(=O)CC2SCCS2)CC(c2ccccn2)=NO1 N1(C(C2(COCC)CCC2)=O)CCCC(C(C)(O)CNC(c2ccoc2C)=O)C1 c1(CC(=O)NC(C)CCN(C(=O)C(C)O)C)ccc2cccnc2c1 C1(CN(C(C=CCCC)=O)CC)CCN(C(=O)Cc2cccn2C)C1 C(C(C(C)(C)C)NC(=O)CCc1ncccc1C)NC(C(=O)NCC)=O CCC(C(=O)N1CC2CCC2(NC(=O)CCc2nnc(O)nc2O)C1)C(C)C CC1OC2(C)CC1(C(N1CCC(CNC(c3ccnc(F)c3Cl)=O)C1(C)C)=O)C2 C1(NC(C(CC=C)OC)=O)CCN(C(c2ncn3c2CCC3)=O)C12CCC2 c1(C(=O)NCC2(F)CC(NC(CCC(=O)OC)=O)C2)ccnc(F)c1OC c1(OC)ccc(C(N2CCC(C)C2C(=O)N(C(C)CC(N)=O)C)=O)cc1O c1(C(N2CC3CN(S(CC)(=O)=O)CC3C2)=O)ccc(S(C)(=O)=O)cc1Br c1(CC)nc(O)c(C(=O)NCC(CC)(CC)NC(=O)C#CC2CCC2)cc1C N1(C(C(N2CCSCC2)C)=O)CCC(NC(c2cncc(Br)c2)=O)C(F)C1 C1(NC(C(C)SC(C)C)=O)CCN(C(=O)CCNC(=O)CO)CCC1(F)F C(C(O)CC(=O)N1CC(F)CC1CN(C)C(c1cc(CO)n(C)n1)=O)N(C)C C1(C(N2CC(CC(=O)NCCc3cscn3)OCC2)=O)CC2(CCO1)CC2 N1(Cc2cn(CC=C)nc2)CCN(C(c2cc(Cl)ccc2OC)=O)CC1CC C1(C(=O)NCCC(C)(C)OC)CCCC(NC(=O)C=Cc2cccc(C)c2)CC1 c1(CC)cc(C(N2CC(NC(c3cc(F)c[nH]3)=O)C(F)C2)=O)cc(C)c1 c1(C(=O)NCC(CNC(c2nc(CCCC)sc2)=O)O)ccnc2ccccc12 O=C(C(F)C(F)(F)F)NC1CCC(NC(c2ccc(C3CCOCC3)cc2)=O)C1 N1(C(Cc2c(C)con2)=O)CC(NC(c2ccccc2[N+](=O)[O-])=O)CC(C)(C)C1 c1(CCCC(=O)NCC2CC(F)(CNC(CC(=C)Br)=O)C2)nnc(C)n1C c1(OC)c(Cl)ccc(C(N2CCCN(C(=O)CC3C=CCC3)C(CO)C2)=O)c1F C1(NC(CCN(CC)CC)=O)CC2C(NC(c3cc(C)oc3C)=O)C2C1 c1(C(=O)NCCCCN(C(C(=O)NCC)=O)C)nnn(Cc2cc(C)no2)c1C c1(CC)cccc(C)c1C(=O)Nc1ccc(Cl)nc1NS(=O)(=O)C(F)(F)F C(=O)(CCCCCC(C)O)NC1CCC(CNC(c2cc(CC)nn2C)=O)CC1 C1(C(N(C(CCNC(C=C(CCN(C)C)Cl)=O)C)C)=O)CNC(=O)N1 C1(F)(C(=O)NCC2C(C)(C)C2(F)F)CCCN(C(=O)CCC2CCC(=O)NC2)C1 c1(C(=O)NCCC(C)c2cn[nH]c2)c[nH]nc1CCNC(c1ocnc1C1CC1)=O c1(C(N(CC(CC)NC(C2CC=CC2)=O)C)=O)ccc(-n2nc(C)cc2C)nc1 c1(NC(=O)COC2(CC#C)CC2)ccccc1NC(c1nnsc1SC)=O N1(C(=O)OC(C)(C)C)CCCC(C(=O)NCC#CCN(C(=O)C=CS(C)=O)CC)C1 CCC1=C(C(=O)NCC2(O)CC(NC(=O)C(C)(C)CC#N)C2)CCCO1 C1(C)(C(N2CCC(C)(CNC(C(CC)n3cncn3)=O)CC2)=O)CCC(=O)N(C)C1 C(=O)(C(CN(C)C)C(C)C)N1CCC(O)(CCNC(Cc2c(C)nsc2)=O)C1 c1(C(N2CCSCC2CC(N)=O)C(=O)NCCOC)c(Cl)ncn1C c1(C(=O)NC2CC3CN(C(C(C)OCC4CC4)=O)CC32)cccc2c1CNC2=O N1(C(CS(CC)(=O)=O)=O)CCC2CN(C(=O)COCCOCC)C(C)C12.OC CC#CC1CCN(C(=O)C(C)N(C(c2ccnnc2C)=O)C2CC2)C1 c1(C(=O)NC(CNC(c2cnn(CCC)c2Cl)=O)(C)CO)ncnc2c1CCC2 C1(C)(C(=O)NCCN(OC)C)CCN(C(=O)C=C(C)c2ccccc2)CC1 CC1OC2(C(N3CC4CC(NC(c5cnnc(O)c5)=O)C3C4)=O)CCC1CC2 C(c1nc2ccccc2o1)=CC(=O)NC1CCN(C(C=C(CC)C)=O)CC1CO c1(SCC(CC)CC)nnc(-c2ccc(OC)cc2)n1CCC#N N1(C(c2c(SC)scc2)=O)C2CCC1C(CNC(=O)C(O)CC(F)F)C2 Cc1ccc(CN(CCCNC(c2cccc(F)c2C)=O)C2CC2)cc1F n1(C(C)C)ncc(F)c1C(N1CC2CC2(CNC(C2CC=CCC2)=O)C1)=O c1(C(N2C(CNC(C3CCCO3)=O)CC(C)(C)C2)=O)cc(Br)c2c(c1)OCO2 C12(C(=O)NCC3N(C(CCC(C)(F)F)=O)CCCCC3)CCOC1CCOC2 N1(C(C(C(C)C)NC(COC)C)=O)CC2CCC(C1)N2Cc1ccc(C)cc1F N1(C(c2cnc(CC)s2)=O)CCC(C)(NC(c2n[nH]cc2CC2CCCC2)=O)C1 N1(C(CCC(C)SC)=O)CCN(C(c2ccc(C)cc2N)=O)CC1C1CC1 c1(C(N(CCC(C)NC(C(C=C)(C)CCOC)=O)C)=O)c(C)nn2c1CCCC2 c1(C(=O)NC2CC(CNC(CC(CC)C3CCC3)=O)C2)cccc2c1COC2 N1(C(C2N(CC)CC2)(C)C)CCC(C)(CC(=O)NCCn2ccnn2)C1 N1(C(c2c(C)nccn2)=O)CCCC12CCCN(C(=O)Cc1ccc(Cl)cc1)C2 C1(C(F)(F)F)(C(=O)OC)CCN(C(=O)NC(c2occc2C)C)CC1 CCC(C(=O)NCC1CC(NC(C2(C)CC(Cl)(Cl)C2)=O)C1)C(C)(C)CC C1(NC(CSSC)=O)CC(C)N(C(=O)COCC(F)F)C1 C1(C(N(CCNC(C2C(C=C)C2)=O)CC2CC2)=O)CC(F)C(=O)N1C C1(C(=O)NC23CC(C)(C2)C3)CCCN(C(=O)CC2CCCN(C(C)C)C2)C1 C12(NC(C3N(C(=O)OC(C)C)CCC3)=O)CC1CN(C(=O)CC(O)CN(C)C)C2 C1(F)(C(=O)NC2(CC)CCOCC2)CCCN(C(c2cc(C)c(C)o2)=O)C1 CC(C)CN=C(NCC(c1ccccc1)O)NC(c1ccn(C)c1)C C=Cn1nccc1C(=O)NCC1CC(NC(=O)C(C)N2CC(C)C2)C1 C1(O)(C(=O)NC(CCC)CNC(c2c[nH]nc2C2CC2)=O)CCC(C)(C)CC1 C1(C(N2CCC(CCC(=O)N(C)CCN3CCNC3=O)C2)=O)C(C)(C)C1(F)F C1(CNC(=O)CC2CCC2)CC(CNC(=O)CN2CCSCC2)CO1 C1(NC(CCc2cc(C)on2)=O)CCN(CC2CCC=CCC2)CCC1CO c1(CNC(C2CCCC(F)(F)C2)=O)cc(Cl)cc(Cl)c1.C12(CCCC1)C(=O)N2 c1(C(=O)NCC2CC(NC(=O)CCF)C(O)C2)cccc2c1COC2 C1(OCC)CCCN(C(=O)CC(C)NC(=O)CCCn2cncn2)C1 c1(C(N2C(CCNC(c3n(C)ncc3)=O)COCC2)=O)cnc2c[nH]nc2c1 CC1CCC(NC(C2CCC(=O)N2)=O)CN1C(C1CC(C)(C)CN1C)=O c1(C(=O)NC(C(CO)NC(c2c(C)occ2)=O)C)ccc(F)c(C)c1N C1(NC(CSc2cn(C)nc2)=O)CC2(C1)CC2C(=O)NC12CC(F)(C1)C2 N1(C(C(CC)=CC)=O)CC(NC(c2csc(SCC(F)(F)F)n2)=O)C(O)C1 CC(C)CC(CNC(C1(O)CC(C)(C)C1)=O)NC(c1csc(=NC)[nH]1)=O c1(Oc2c(C(=O)N=c3ccn(C4CC4)[nH]3)ccc(F)n2)ccc([N+](=O)[O-])cc1Br C1(C2CC2)(CNC(C(CCCC)N(C)C)=O)CCN(C(c2cc(C)c(C)o2)=O)C1 O=S(=O)(c1ccc(NC(C)C2CC2)nc1)NC1CC(n2ccnn2)C1 N1(C(CSc2ccc(C)cc2C)=O)CC23CCCCC2(C1)CN(C(=O)C(N)=O)C3 c1(C(C)C)ccc(C(N2CC(F)CC2C(=O)Nc2cc(C(F)F)cs2)=O)cc1 c1(N2CC(CCC)C(N(CC)CC)C2)cc(C#N)nc(C)n1 CC(CCCNC(c1cc(Cl)cs1)=O)NC(=O)CCc1nc(C(F)(F)F)n[nH]1 C1(NC(CC(CCC)CC)=O)CC2CCCC(C1)N2C(C1CCCCC1C)=O C(c1ccccc1C)=CC(=O)NCCNC(c1c(C)cn(C)c1)=O C1(N(C(=O)COCC(F)F)C)CCC(C)(NC(=O)C(F)Cc2ccccc2)CC1 N1(N(CCCC#C)CC2CCCO2)CCCC1CCCOCC CCCC(C)(CC)C(=O)N1CCN(C(=O)CCn2cnnn2)C(COC)C1 C=C1Cn2c(C(N3CCN(C(c4c(C)ccn4C)=O)CC3CC)=O)nnc2S1 c1(C(N2C(C)CCC(NC(c3nc(C)sc3)=O)C2)=O)ccc2ncccc2n1 C1(C(=O)NCC#CCNC(=O)CCCn2cncn2)CCCC2(CCOCC2)O1 c1(CC(=O)N(C(CCNC(C(CN(C)C)N(C)C)=O)C)C)ccc2c(c1)COC2 C12(C(N(C(C)CC(N)=O)C)=O)CC(CO)(CN1C(c1cc(C(N)=O)[nH]n1)=O)C2 C1(NC(c2cccc(CC)c2F)=O)CC2(CCN(C(c3cnsc3)=O)C2)C1 C1(CCNC(Cc2c(C)n[nH]c2C)=O)CN(C(=O)Cc2cnoc2)CC(C)O1 C1(C(N2C(CN(C(c3snc(C)c3N)=O)CC)CCC2)=O)C2CN(C)CC12 C12(CNC(Cc3ccc(OC)cc3)=O)CC(C1)C(NC(c1cnc[nH]1)=O)CO2 c1(C(=O)NC(C2CCN(C(C3NC(=O)CC3C)=O)CC2)C)ccc(Cl)nc1O C1(C(C)C)CN(C(c2nc(Cl)cs2)=O)CCCN1C(c1cc(C(N)=O)c[nH]1)=O C(=O)(CC(C)CNC(=O)CC(C)N(C)C(C1(CC)CC1)=O)OCC C1(CC=C)(NC(C2OCCC2C)=O)CCN(C(c2sccc2NS(C)(=O)=O)=O)C1 C1(C(=O)NCC2(F)CC(CNC(C3C(CCC)CCC3)=O)C2)CC(F)C(=O)N1 Cc1nnc2n1CCN(C(=O)C(CNC(=O)CN1CCCC1=O)CC(C)C)C2 c1(C(=O)NCC(CC)NC(c2ccnn2C)=O)coc2cc(C)c(C)cc12 CC1CCOC(C(=O)NC(CCCNC(C2(C#N)CC2)=O)c2ccccc2)C1 C1(N(C(CN(CCC)C)=O)CC2CC2)CCN(C(=O)COOC(F)F)C1 n1(CC)cc2ccc(C(N3CC(N(C)C(c4cnccc4OC)=O)C3)=O)cc2n1 c1(C(=O)NC2(C)CC(NC(CSCCOC)=O)C2)cc2c(F)c(F)ccc2[nH]1 C1(CC(=O)NCC(CCC)C)CN(C(c2cccc(CC#N)c2)=O)CC12CC2 CC(C)C(O)C(=O)NCC(C(C)(C)C)NC(C1(Oc2ccccc2F)CC1)=O Cc1cc(-n2ccc(C(=O)NCCC(C)(C)O)n2)ccc1Cl CC1(C)CCC=C1C(=O)N1CC2CC(CNC(=O)CCOCC(F)(F)F)C2C1 N1(C(C(C2CCOCC2)OC)=O)CCN(C(=O)CCCN=[N+]=[N-])C(C2CCC2)C1 C(=O)(C1CS(=O)(=O)c2ccccc21)N(CCNC(c1csc(C(F)(F)F)n1)=O)CC C12(CNC(COCCOCC#C)=O)CN(C(=O)C3=CCC3)CC1CS(=O)(=O)C2 c1(C(=O)NC(CC)CNC(=O)C(C)CC2CC2)noc2cc(F)ccc12 c1(C(N(C2CCN(C(C(CC)F)=O)C2)CC)=O)cccc(Cl)c1O N1(C(CSCC(C)C)=O)CC2CCCC(C1)N2C(=O)CCNc1ccccc1Cl CCCC(C(=O)NCCCC(=O)NCCc1noc(C)n1)OCC c1(NCC(=O)NC(c2ccc(F)cc2)C)cn2c(n1)CCCC2C(=O)O N1(C(c2cc(Br)c3c(c2)OCCO3)=O)CCc2c(Br)cncc2C1 N1(C(c2occ(C)c2)=O)CCN(C(=O)C(C2(O)CCCC2)F)CC1CC1CC1 C12(C(=O)NC3(C)CCOC3)C(NC(=O)COc3cccnc3)C3CC1C2C3 C(=O)(CC(C)(CC)C(=O)OC)NCCCC(C)NC(c1ccc(OC)cc1C)=O C#Cc1cccc(C(N2CC3CCC3(CO)C2)C(=O)NC2CCOCC2)c1 c1(CN2CC3N(C(c4cccc(O)n4)=O)C3C2)c[nH]c2ncc(Br)nc12 Cn1nc2c(c1C(=O)NC1CCCCC1NC(c1ccc(=N)[nH]n1)=O)CCC2 N1(C(C=COCC)=O)CC(F)(F)CC1C(=O)N(C)CC1CCN(C)C1 c1(CC(=O)NCC2(NC(C3CC3F)=O)CCC2)ccccc1Br c1(OC)cc(C(=O)NC2CN(C(C3CCCC3)=O)C2)cc(Br)c1OC(C)C c1(C(N(C2CCN(C(=O)Cc3ccns3)CC2)CC)=O)cnc(S(C)(=O)=O)s1 c1(C(C)=O)cc(C(N2CC(CC)(NC(=O)Cc3cnns3)C2)=O)co1 c1(C(=O)NC(CNC(C(C)NC(c2ccoc2)=O)=O)C2CC2)cc(Cl)cnn1 C1(COC)CC(CNC(C2(c3ccccc3C)CC2)=O)N(C(=O)Cn2cnnc2)C1 C(=O)(C1=CC2(CCOC2)C1)NC1CCC(CNC(C(=Cc2ccco2)C)=O)CC1 C1(C#CC(=O)N2CCC(C(C)(O)CNC(=O)Cc3cc(C)on3)CC2)(CC)CC1 C1(CC(=O)N(CC(=O)NCCC)CCC)CC(C)(C)CN1 C1(NC(c2cc(Cl)c(Cl)[nH]2)=O)CN(CCO)CCC1CO c1(C(N2CC(O)(CNC(Cc3scc(C)n3)=O)C2)=O)cc2c(F)ccc(F)c2[nH]1 C1(NC(CCOc2ccc(C)cc2)=O)CCN(C(c2ncc(F)cn2)=O)CC1C C1(CC)CCC(C(=O)N(CCCCCNC(=O)CCCc2csc(=N)[nH]2)C)O1 C(=O)(C1CCc2c[nH]nc21)OC(C)(C)C.C1=CC(=O)NC1(C)C.CC1CO1 C1(NC(=O)CC2CC=CCC2)CC(F)CN(C(c2cc(Cl)ccc2O)=O)C1 N1(C(C(CC2N(C(COC(C)=O)=O)CC2)F)=O)CC(O)CC(C)(C)C1 c1(NC(C2C3CCN(C(CN(C(COC)=O)C)=O)CC32)=O)cnc(C)c(C)c1 N1(CCNC(CCC2(C)CN(C(C=C(C)C)=O)C2)=O)CCCCC1=O c1(C(=O)NCCC2CN(C(c3[nH]nc(OC)c3Cl)=O)C2)n[nH]c(C)c1[N+](=O)[O-] Cc1cc(C(=O)Nc2cccc(NC(c3cc[nH]c3C3CCCC3)=O)c2)cn1C c1(OC)cc(CN(CCCn2cccc2)C)ncn1 CC1CCC(CNC(=O)C=C2CCC2)N(C(=O)CN(c2ccncc2)C)C1 c1(CNC(C(C(C)C)(O)c2ccccc2)=O)c2ccccc2nn1C CCCC(C(=O)OC)C(=O)N1CC(NC(c2cc(C(C)C)[nH]n2)=O)C(N=[N+]=[N-])C1 N1(C(C)C)CCCC1C(=O)N(CC(C)NC(=O)COCCOc1cn(C)nn1)C N1(C(C2CCCC(C)C2)=O)CC(NC(c2ccc(Br)nc2I)=O)C2(CC2)C1 CN1CCOC(C(=O)N(CCCNC(C2CNC(=O)N2)=O)CC2CCCC2)C1 c1(CNCc2ccc(OC)cc2)cc(Br)cc(Cl)c1F.N1(C(CO)=O)CCCC1C CC(C)C(CNC(=O)C(C)CC1CC1)C(=O)N(c1ccc(F)cc1)C N1(C(c2cc(NS(C)(=O)=O)on2)=O)CCC2CCN(C(=O)CNC=O)CC2C1 N1(C(CNC(CNC(C)=O)=O)=O)CCC(F)(CNC(c2cscc2Cl)=O)C1 C(c1ccc(C)cc1)=CCC(=O)NC(CN(C(=O)CCC(C)NC(C)=O)CC)C N1(C(C(C)SCCCC)=O)CCC(n2cc(-c3cnn(C4CCC4)c3)nn2)C1 C(CCC(C)C(=O)OCCn1ccc(O)nc1=O)OC CCC(C(=O)NCCCC(C)NC(C1(C(N)=O)CC1)=O)C(C)C O=C(CCCCc1ccccc1)N1CCC(NC(C2(O)CCCC2)=O)CC1 N1(C(c2c(C)nccc2)=O)CCC(C)C(NC(c2cc(C)ns2)=O)C1 C1(NC(CN(C)CC)=O)CC2CN(C(c3cc(C)nn3C)=O)CCN2C1=O c1(C(=O)NCCCCN(C(CS(=O)(=O)NC)=O)C)cc(F)ccc1C(F)F c1(C(=O)NCC(C2CCCC2)NC(=O)CCc2ncc[nH]2)cc(Cl)ccn1 c1(C(=O)NCCCCCNC(CCSC)=O)cnc(C(F)F)cc1C.C(=O)CO C1(N(C(C(OC)OC)=O)C)CCN(c2ccccc2C(F)(F)F)C1=O c1(NC(C2CC(=O)N2)=O)ccc2cnn(CCc3ccccc3)c2c1 N1(C(CC=C=C)=O)CC(NC(c2ccccc2NC(C)C)=O)CC2(CCC2)C1 C(=O)(C(O)CCC(C)C)NCC(CC(=O)N(CC)CC1CCOC1)C1CC1 c1(C(N2CCC(NC(C(C)n3cnnn3)=O)C2C)=O)cccc2c1CCCCC2 C(CCC)(C(=O)N1CCOC(CC(=O)N(C(C)COC)C)C1)=CCC C1(NC(C2(C=C)CCC2)=O)CCCCC1NC(=O)CCNC(c1ccoc1)=O C1(C)(C(N2CC(NC(CC(C)(C)OC)=O)C(F)C2)=O)COCC1(F)F N(C1CCc2cc(CNC(C3(C#N)CC(=O)C3)=O)ccc21)C(C1CCC(C)O1)=O C=CC1(C(=O)NCCC2(O)CN(C(c3ccc(CCC)[nH]3)=O)C2)CCC1 N1(C(C(C=CC)O)=O)C2CCC1CC(NC(c1ccc(OC)c(CC)c1)=O)C2 N1(C(c2c(C)ocn2)=O)CCCC2(CCCCN2C(C2CCCS2(=O)=O)=O)C1 c1(C(=O)NC2CN(C(c3[nH]cc(CC)c3)=O)CC2C(F)F)cccc2[nH]ccc12 C1(CC(=O)OC)C(=O)N(C)CCN1C(N1CC(OC(C)(C)C)C(C#N)C1)=O CCCCC(C)CCC(=O)N1CCC2C(C1)CN2C(c1cc(Cl)c(F)c(Cl)c1)=O N1(C(c2ncn(C)c2)=O)CCCC(Nc2cnncn2)C1 c1(C(=O)NC2CCC2c2nc[nH]n2)cc(Cl)ccc1Cl.C1C(F)CNC(=O)CO1 C1(C(=O)NCC23CC(NC(c4cn(CC)nc4C)=O)(C2)C3)CC2CCCCN2C1 C#CCC(CC(=O)NCC1CC2(CC2)C(=O)O1)NC(c1cc(Cl)c[nH]1)=O CCC(C)(C#N)C(=O)NC(CC(=O)NCC(C)(O)CSC)C(C)C N1(C(=O)CSCC2CCCO2)CCN(Cc2cn(-c3nccs3)nn2)CC1 c1(Nc2cc(N(C)CC3(C)CCCS3(=O)=O)ncn2)cc(Br)cnc1N c1(CC)[nH]nc(C(=O)NCCN(C(C2OCCO2)=O)CC2CC2)c1[N+](=O)[O-] c1(Nc2cn(C3CN(C(=O)NC(C(C(=O)OC)OC)=O)C3)nc2)cc(C)cc(F)c1 C1(COC)CC=C(c2ccc(C(=O)NCCC3CCCCO3)[nH]2)CC1 N1(C(CN2CC=C(C)CC2)=O)CCCC(CNC(c2ccn(C)c2)=O)CC1 C1(NC(C=CC=CC)=O)CCN(C(C2C(C=C(C)C)C2(C)C)=O)C12CCCC2 Cc1cc(=NCCCCC#N)[nH]c(=NCCOCCS(N)(=O)=O)[nH]1 c1(C(=O)NC2(CO)CN(C(COCc3cc(C)no3)=O)C2)cc(Cl)c(C)cn1 C1(C(=O)NC2CCN(C(C(C(C)O)(C)C)=O)CC2O)CS(=O)(=O)CC(=O)N1 C(=O)(C1=CCc2ccccc21)N1CC(N(C(C(CC(C)C)OC)=O)C)C(C)(C)C1 C(=O)(C(CO)C(F)(F)F)NC1(CC#C)CCC1.C12CCCC(CC1)NC2=O Nc1c(F)cc(C(=O)NC2CCC(CCNC(=O)CCCCC(F)F)C2)cc1F N1(C(CNCCC)=O)CC(NC(=O)C=CC(=O)OC(C)(C)C)C(C(F)(F)F)C1 C1(C)(C(N2CC3C(C(=O)N(C4CCCC4)CCOCC)C3C2)=O)CNCCC1(F)F Cc1cc(C(N2CCCC(O)(CCNC(=O)OC(C)(C)C)C2)=O)n2nc(C)cc2n1 N1(C(CN(C(C(CC)C)=O)C)=O)CCN(C(C2C(C)(C)C2(F)F)=O)CC1 CC1CC=C(C(=O)N2CCC2CNC(=O)Cn2ccc(Br)n2)CC1 C1(NC(CSCC(C)C)=O)CCN(C(=O)CCc2n[nH]c(=N)s2)CC1O C(CC1OCCc2ccccc21)N1C(=O)C(CCSC)N(C)C1=O C1(NC(Cn2c(=O)ccc(C)c2)=O)CC2CCC1N(C(=O)CCOC1CCC1)C2 c1(OC)ccc(CN2CCC(C(=O)Nc3cncnc3O)C(O)C2)c(F)c1OC C12(C(=O)NC(CNC(CN(C)C(=O)C3CC3)=O)C3CC3)CCC(CC1)CC2 Cc1cc(C(C)C(=O)NCCCCN(C)C(C2C3CCC(F)(F)C23)=O)cc(F)c1 c1(CC(=O)NC2CCN(C(C=CC)=O)CC2O)nnc(O)c2ccccc12 Cc1cc(CN2CC3CC3(C(=O)NCc3cccc(C4CC4)c3)C2)cc(C)c1Br C1(C(=O)NC2CN(C(c3c[nH]c(=NCC)s3)=O)CC2(C)C)CCCC2C1C2(F)F N1(C(C(CC)COC)=O)CCCC(C)(C)C1C(=O)NC12CC(C1)C2 C12(C(N(C)CCNC(C3CN(S(C)(=O)=O)C3)=O)=O)CC=CCN1CCC2 N1(C(c2ccc(OC)c(-c3cn(CC(=O)O)nn3)c2)=O)CCC2(CCC(O)C2)C1 CCCCC(O)C(C)C(=O)NCC1CN(C(c2ccc(C)cc2F)=O)CCCO1 C1(OCC)CC(N=c2nc(-c3ccccc3)nc(NC(c3ccn(C)n3)C)[nH]2)C1 C(=O)(C(CCCOC)NC(=O)Cc1cccnc1)NC1(C(=O)NC)CC1 c1(C(N(C2CCN(C(=O)CCC(C)(C)O)CC2)CC)=O)ccc2c(c1)OCCO2 Cc1ccnn1CC(N1CC(O)(CCNC(=O)CCSCc2ccccn2)C1)=O Cc1cc(C(N2CC3CC2C3C(=O)NCCc2ccccc2)=O)nc2nccn12 O=C(CCCCCn1cnnn1)NC1(C)CCCN(c2nnc(C(F)F)o2)C1 C1(NC(C2(CSC)CN(C(C3C(OCC)CC3)=O)C2)=O)CCCN(C)C1C c1(C(N2CCC(CNC(CCC(=O)OC)=O)C2)=O)sc(C#N)cc1Cl C(CCCCCC(C)C)NC(CC1N(C(CC(C)(C)NC(C)=O)=O)CCCC1)=O N1(C(Cn2ncc(C)c2)=O)CC2CCN(C(C3COCC3C(F)F)=O)CCC2C1 c1(C(N2CCC(NC(c3c(C)scc3)=O)CC2C)=O)cc([N+](=O)[O-])c(C)s1 c1(C(=O)NC2CC3(C2)CC3NC(=O)C(F)C2CC2)cc2c(nc1O)CCCCC2 C1(NC(Cn2nc(C)c(C)c2C)=O)CC12CCC(NC(c1cccnn1)=O)CC2 n1(CC(N2CC(C(C)NC(C3(CO)CC3)=O)C2)=O)nnc(-c2ccco2)n1 C=CC(C)(CCOC)C(=O)N(C(C)C(=O)NC(C)CCO)C1CCC1 C(=O)(CC(C)(C(F)F)N(C)C)N(C)CC1CCCN(C(=O)CC2=CCCCC2)C1 C1(C(=O)NCCC(C)NC(c2cnc(-c3cccnc3)s2)=O)CSCCS1 c1(NCC)ccccc1C(=O)NC(C1CCOC1)CNC(C1(C)CC=CCO1)=O N1(C(C(N2CC(C)C2)C)=O)CC(NC(C2CC(n3ccnn3)C2)=O)C2CCCC12 c1(-c2n(CCC#C)ccn2)ccc(OC2CCCCC2)c(F)c1 C(c1ccc(C)cc1)=C(C(=O)NC(CN(C(c1ccc(CC)nc1)=O)CC)C)C CCCC(C)(O)C(=O)NCCCCN(C)C(C1(C)CCN(C(C)=O)C1)=O c1(C2C(C(=O)NCC(C)NC(=O)Cc3c[nH]c(=N)[nH]3)C2)cccnc1O Cc1[nH]nc2c1CCC(C(=O)N(CCCCNC(C1CC3COCC3C1)=O)C)C2 C1(OC)CN(C(=O)C(F)(F)c2cnccn2)CCC1NC(C1CC(SC)C1)=O C(=O)(CC(C(C)(C)C)NC(=O)CC1(CSC)CC1)NC1(CCC)CC(C)(C)C1 CCN=c1[nH]cc(C(=O)NC2CC(CCNC(=O)CC3NC(=O)NC3=O)C2)s1 Cc1ncc(C(=O)NCC2CCN(C)C2)c(Cl)c1Br c1(C(N2CC3C(CNC(C(CCSC)NC(C)=O)=O)(C3)C2)=O)ccc(S(C)(=O)=O)[nH]1 C1(C)(C=O)CCN(C(c2ccno2)=O)C1.N1(C(C)CC2CC2)CCOCC1 N1(C(c2c(C)ncs2)=O)CC(NC(=O)C=CC2CCOC2)C(O)C1 c1(-c2cn(CCCCCCN(CC(=O)O)C)nn2)ccc(F)c(S(C)(=O)=O)c1 CC1CC(C(=O)NC2CC3(C2)CC(O)C3)CCN1C(=O)Cc1cn(C)cn1 N1(C(=O)Cn2cncn2)CCCC(CN(C(C23CC(CCF)(CO2)C3)=O)C2CC2)CC1 CC1(C(=O)NCC2(O)CC(NC(C3(N4CCCC4=O)CC3)=O)C2)CC=CCC1 c1(C(N2CC(CNC(c3cc(Cl)ccc3Cl)=O)C(O)C2)=O)ccn2ccccc12 c1(OC)ccc(CN2C(C(N3CCC(N4CCCC4)CC3)=O)CC3CC23)cc1F c1(C(=O)NCC(C2CC2)NC(C#CC2(C)CC2)=O)ncn2cc(Cl)ccc12 c1(-c2ccc(C(N3CC(C(=O)OC)N(C)CC3)=O)s2)nccn2cccc12 C1(c2c(OC)nsc2)NC(=S)N(c2cc(C)nn2C)C2=C1C(=O)OC2 c1(OC)ccc(F)c(C(N2CCCC(C(=O)NC(CO)C3CC3)C2C)=O)c1 N1(C(C2(C(C)C)CCN(C(C3CCN3C)=O)C2)=O)CC(=O)NC(=O)C1C C1(C(=O)NCC(C)CNC(c2cc[nH]c2)=O)CC(F)(F)CS1 CCC(C(=O)N1CCOCC1CNC(c1c[nH]nc1C(C)C)=O)C(C)C N1(C(c2ccn(CC)n2)=O)CC(C(N2CCC3C(C(=O)OC)C3C2)=O)C2(CC2)C1 c1(NCC(=O)NC)nccc(=NC(C)c2nc(O)n[nH]2)[nH]1 N1(C(C(=Cc2cnc[nH]2)C)=O)CCC2CN(C(=O)CCCN3CCCC3)C2C1 N1(C(c2c(Cl)cc(C)c(C)c2)=O)Cc2ccccc2CC1CNC(=O)CC(C)F Cc1c(O)ccc(C(=O)NCC2CCCC2NC(c2ccc(Cl)c(O)c2)=O)c1C C1(CNC(c2nc(C)sc2)=O)CC2CCC1N(C(=O)C1=CCOCC1)C2 N1(C(C(C(C)C)NC(c2ccc(Cl)cc2)=O)=O)CCC(O)CC(C)(C)C1 CP(C)(=O)CCNC(c1nnnn1C1CCOCC1)C1CC(n2ccnn2)C1 N1(C(CNC(CCCCC)=O)=O)CCCCC(NC(=O)C(=O)Nc2ncc[nH]2)C1 C(CC(=O)N1C2CCC1CC2)(C(F)F)NC(C1CCC(OC)CC1)=O C1(C(N(CC(=O)NCC(C)(CO)OC)CCOC)=O)CN(C)CCO1 C1(C(=O)NC2CCC(CN(C(C(CC)(F)F)=O)C)CC2)CCc2nccn2CC1 Cc1cc(C(=O)N(C)CCOCCCN(C(=O)C(F)n2cccn2)C)ccn1 c1(C(=O)NCC(C2CC2)NC(C2C=CCC2)=O)ccc(N2CCC2)cc1 C1(NC(C2CC(CCC)C2)=O)CCC(NC(C2CC3C=CC2O3)=O)CC1 C1(C(=O)NCCC(=O)NC)C2C(CN1C(c1c(F)ccc(Cl)c1F)=O)C2(C)C N1(C(CCC(C)C)=O)CC(C)N(C(c2cnc(Cl)c(C(F)(F)F)c2)=O)CC1C CN1CCC(C(=O)NC2CCC(C)(C)C2)(NC(=O)CS(C)(=O)=O)C1 C1(CCC)CN(C(C2(CCOC)CCC2)=O)CCN1C(=O)CSCCOC C1(NC(C2C3CN(C(C4C(C(C)C)CCO4)=O)CC32)=O)CCCCC1(C)C N1(C(C2(C)C=CCC2)=O)CCC(C(F)CNC(c2ncoc2C2CC2)=O)CC1 C(=O)(CCC(=O)NCc1cc(C(N2CCC(OCC(N)=O)C2)=O)n[nH]1)NC c1(OC)cc(Br)ccc1CN(CCC(O)c1cccs1)CCN(C)C N1(C(C(C=C)O)=O)CCCC2CN(c3ncccn3)CCC12 C1(NC(CN(CC)CC)=O)CC(OC)CN(C(=O)CC2CCC(=O)N2C)C1 c1(NC(C2C(NCc3c(C)n[nH]c3)C2)=O)ccc(I)c(C(N)=O)c1 C1(C(=O)NCCCOC2CC2)CC1C(N)=O.C1C(=O)N1CCC Cc1oc(C(C)C)nc1C(=O)NCC1CCCCN1C(c1cc(C2CC2)on1)=O c1(CNC(C=C(C)Cl)=O)cn(CCNC(C2CC(=C3CC3)C2)=O)nn1 c1(C(=O)NC2C(CNC(c3cn(C)nn3)=O)C2)ccnc(-n2cncn2)c1 C1(C(=O)NC2C(C(=O)NCCCCC#N)CCC2)CCNC(=O)C1 c1(C(N)=O)nc(NC2CCN(C(=O)NC3(c4ccsc4)CC3)CC2)ncc1Cl N1(C(c2cc(OC)c(Cl)cc2)=O)CCC2C(CCN2Cc2ncc[nH]2)C1 C1(C(=O)NCCCCCN2CCN(C(C=CC)=O)CC2)CCn2c(cnc2C)C1 CC1(C)Cc2cccc(C(=O)OCCOCC34CCCCN3CCC4)c2O1 N1(C(=O)OCC)CCC(C)(C(N2CCC(CSC)C2)=O)C1 c1(C(N2CC(NC(c3n(CCCC)ncc3)=O)C(C)C2)=O)cc(F)cc(C)c1N CCCCC(C(=O)OC)CC(C)NC(=O)C(C)(C)CNC(=O)CC1CC1CC C1(NC(c2c(C)scn2)=O)CCCC(NC(=O)Cn2cc(CO)nn2)C1 c1(SCC)ccc(F)cc1.C1(C)(C(=O)NCCCS)CC1C(=O)O.C1C(=O)N1CC CC1CCN(C(C23CC(C)(CO2)C3)=O)CC1NC(c1cccc(=S)n1O)=O C1(CNC(C(C)=CC)=O)CC2COCC2N1C(=O)C(O)Cc1ccccc1 N1(C(C(C)SC)=O)CCN(C(=O)C(c2cc(Cl)ccc2Cl)(C)C)CC1CO N(C1CN(C(=O)CCCC2CC2)Cc2ccccc21)C(CC1C(=O)NCCC1)=O c1(CC)cccnc1C(=O)NCCCC1CCCN1C(=O)CN1CCCC1=O Cc1cn2c(C(=O)NCC3(NC(C4CCC(=O)N4C)=O)CCCC3)c(C)nc2s1 CCS(=O)(=O)CC(=O)NCCCCCN(C(=O)C(C)CC1CCCO1)C c1(C2C(C3OCCN(C(=O)CCC4CCOCC4)C3)CN2)cccc2cncn12 CC1=NOC2(C1)CN(C(=O)C(=O)NC1(c3csc(N)n3)CC1)C2 c1(NC(C2CC(O)CN2Cc2nccs2)=O)nccc(Br)c1O CC1CN2CCN1C(C(=O)NCC1CCN(C(=O)CCCC(N)=O)C1)C2 N1(C(c2c(C#N)cn[nH]2)=O)CCC2(CCCC2NC(C23CC4CC2C3C4)=O)CC1 c1(C(=O)NC2CN(C(C3C(C(C)C)CCO3)=O)CC(C)C2)c(F)cc(F)cc1F C1(C(=O)NC2CCN(C(c3c(N(C)C)cccc3)=O)CC2)CCN2CCCC12 C1(C(=O)NCCCCN2CCCCC2)(CNC(c2cccnn2)=O)CC12CCC2 C1(C(N(CCN(C)C)CCO)=O)CC(NC(C2CC(F)C(=O)N2)=O)CCO1 N1(C(CC23CC(C)(OC2)C3)=O)CCN(C(C2CC3CC(=O)C2C3)=O)CC1C1CC1 CCCCCCC(F)C(=O)NCC1(NC(c2nccc3nn[nH]c23)=O)CCOC1 C1(OC)CC(NC(c2csc(-c3ccsc3)n2)=O)C12CCN(C(C)=O)CC2 c1(C(N2CC(NC(C(C)NC(=O)OC)=O)C(C)C2)=O)ccc2ccnc(O)c2n1 C1(NC(C(C)CC(F)F)=O)CN(C(c2nnc(O)nc2O)=O)C2(CCC2)C1 Cc1cc(C)c(C(=O)NCC2CCC(NC(=O)C#CC3(C)CC3)C2)c(S)n1 C#CC1CCC(C(=O)NC2COCCC2NC(c2[nH]nnc2C)=O)CC1 N1(C(C(C)N(C(c2ccn3cncc3c2)=O)C2CC2)=O)CCC2CCC(C2)C1 CC(C)(C)CCCNC(=O)C(C)(C)C1CCN(C(=O)C(F)C2CCCC2)C1 N1(C(C(=O)Nc2ncc[nH]2)=O)CC(CNC(c2ccccc2F)=O)N2CCC1C2 C1(C(=O)NCC#CCC)CCCCCCN1C(c1ncc2ccccn12)=O c1(CC2CCCN(C(=O)NC(C3COCCOC3)C)C2)ccc(Cl)cc1 c1(COC)nc(NC2CCCS2)cc(N2CCC(c3cc[nH]n3)CC2)n1 N1(C(C(N2CC(C)OCC2)=O)=O)CCCC2CCC(C)CC12 c1(NC(=O)COCCCn2cc(-c3cc(C)on3)nn2)cc2oc(Br)cc2[nH]1 c1(C(N(C)CC2CCN(C(c3cc(Cl)on3)=O)C2)=O)cc2ccc(F)cc2s1 c1(C(N2CCCCC(NC(CC(COC)(C)O)=O)C2)=O)ccc2c(c1)C(=O)OC2 C1(NC(CC(CCSC)O)=O)CCN(C(c2cnc(CC3CC3)s2)=O)CC1(C)C Cc1ncncc1C(=O)NC1CC2(C1)CC2NC(c1n[nH]c(C)c1F)=O N1(C(C(C)=C(C)C)=O)CCC(C)(CC(N2CCC(C)(F)C2)=O)C1 C1COC(C)(C)OC1.N1(C2C(=O)NC2)CC(N2CCCC2)C(C)(C)C1.CCOC c1(CCC(=O)NCC2CN(C(c3ccc(N(C)C)nc3)=O)C2)ccc(Cl)c(F)c1 CCC(C)(C)C(O)C(=O)N1CCC(C)C(NC(c2cc(C(C)C)oc2C)=O)C1C Cc1cn2cc(CC(=O)NCCC3CCCN3C(=O)CN3CCNC3=O)nc2s1 C(C(C)(C)C(=O)NC(C)CNC(c1cc(=N)[nH]n1C)=O)OC c1(CC(=O)NC(CNC(C=CC(C)C)=O)CO)ccc(S(=O)(=O)N(C)C)cc1 CC1(C)OCCOC1CC(=O)N(C)C.C(=O)(CCP(C)(C)=O)N1CC(C2CC2)C1 N1(C(c2[nH]cc(C)c2)=O)CCC(NC(=O)CCc2ncccc2C)C(CO)CC1 C1(C(C)NC(CCNS(CC)(=O)=O)=O)CCCN(C(c2[nH]c(C)nc2C)=O)CC1 C(=O)(CC(C)CC(C)C)N1CCC(NC(c2c(CC)ocn2)=O)C(CO)C1 C12(CNC(C(CC)C)=O)CCCC(CN1C(=O)CCOc1cccc(C)c1C)C2 c1(COC)ccc(CC(=O)NC2CN(C(=O)CCCc3cnn[nH]3)CC2O)cc1 C(=O)(C1CCCc2nccn21)NC(CC=C)CNC(c1ccc(C)nc1CC)=O c1(C(=O)NCCCC(c2ccccc2)NC(c2cnc(C)[nH]2)=O)ccc([N+](=O)[O-])o1 c1(C(=O)NC(COC)C)ncn2cc(-c3ccc(SC)cc3)sc12 Cc1ncc(Br)cc1NC(=O)C(O)C(F)F C(=O)(C(=O)N=[SH]1(C)CCCCC1)NCCn1cc(CN(S(C)(=O)=O)C)nn1 CCCCC(C)C(=O)N1CCC(C(=O)NCc2nnc(C)s2)(CO)C1 C(=O)(C(C)(O)CCC)N(CC(CNC(C(C)NS(CCCC)(=O)=O)=O)(C)C)C Cc1c[nH]c(C(=O)NC2(C)CN(C(c3ccn(C)n3)=O)C2)c1 c1(OCCNC(C2CCCN2C(=O)C=CCBr)=O)cccc(-c2cccnc2)c1 C1(COC)CCCCN1C(=O)C(=O)NC1CCCNC1=O c1(NC(=O)NC(c2c(C)cccc2)CC(C)C)ccc2c(c1)c(=O)ccn2C C1(N(C(C(CNC(=O)C=Cc2cscn2)OC)=O)C)CCCC1(C)O c1(C(CC)NC(=O)CN(C(c2cnns2)=O)CC)nccn1C CCS(=O)CC(=O)NC1CN(C(c2c[nH]nc2I)=O)CC1C C(N=c1[nH]c(N2CCC(OC)C2)nc2c1SCC2)c1cccc(CC)n1 C(C(C)(C(C)C)NC(=O)CC(C)(C)C)NC(C(C)n1cccn1)=O.c1(OC)ccccc1 C(=O)(C(C)(CSC)NC(C1OCCC1(C)C)=O)NC(CC)CCOCC C1(NC(c2c(C#C)c[nH]n2)=O)CC1C1CCN(C(=O)CCOCCCOC)CC1 Cn1nc(C(N2CCC(CCC(=O)N3CC(n4cccn4)C3)C2)=O)cc1O C(=O)(C#CC1(C)CCCO1)NCC(CC(=O)NCCn1c(C)cc(C)n1)C C1(c2ncco2)(OC(CSCC#C)=O)CC1C(=O)OCC c1(NC(=O)CC2CCN(Cc3cnn[nH]3)C2)ccc2c(n1)CCCC2 N1(C(CCCCOCCC=C)=O)CCC(C(=O)NCCCCCSC)C(O)C1 C1(NC(CSCCCC)=O)COCCN(C(=O)CCC2COC(C)(C)O2)C1 C(C)(C(C)(C)C(=O)NC(C)CSC)NC(c1c(COC)cc[nH]1)=O c1(N2CC(CC)S(=O)(=O)C(C)C2)nc(=NCC2CC3(CC3)C2)[nH]c2c1SCC2 C=CCC(CC(F)F)C(=O)NC1(CC)CN(C(c2c[nH]c(=N)o2)=O)C1 N1(C(C(CC)C)=O)CC(N(CC(=O)OC)C(=O)COCc2nc(C)no2)C(O)C1 C1(CC(=O)NCc2cc(OC)ns2)CC(C)(C)CN1C(c1nnn(C)c1N)=O C1(C2N(Cc3cn(CC(=O)OC)nc3)CCC2)CCC(C)CC1 CC1CN(C(c2cnns2)=O)CCCN1C(=O)CC(C)c1ccccc1 Cn1cc(Br)c(CS(N2CC(C(=O)O)C(C(F)(F)F)C2)(=O)=O)n1 CC1CCCC(O)(C(=O)NCC2CCN2C(c2ccc(C#N)n2C)=O)CC1 CN1CCn2cc(C(N3CCOC(CNC(=O)CCP(C)(C)=O)C3)=O)nc2C1=O N1(CC)C(=O)CCC1CC(=O)NCC(CO)NC(c1n[nH]cc1OC)=O c1(-n2c(C3C(=C)C3)nc(C3CCCO3)n2)cc2ccccc2n1CC c1(NCC2(CCC)CCC2)nc(N(CCC(C)C)C)c2ccsc2n1 N1(C(c2c(CC)n[nH]c2)=O)CCOC(C(=O)Nc2cnsc2)CC1 Cn1cc(C(=O)NCC(CNC(C2(n3ccnn3)CC2)=O)S(C)(=O)=O)n(C)c1=O C1(C(=O)NC2CCN(S(C)(=O)=O)C2)(CC)CCCN1C(=O)CCCN(C)C C1(C(=O)NC(C(C)(C)C)CNC(c2ccncc2)=O)CCc2nnc(O)cc2C1 n1(CC(=O)NC2CC(NC(C(CC)(C)O)=O)C2)c(C(N)=O)nc2ccccc12 CCCS(=O)(=O)C(C)C(=O)NCC(C)(CC)NC(=O)C1=C(C#N)CCC1 c1(C(N2CC(C)(CNC(CSCC=C)=O)OCC2)=O)cn2c(Cl)cccc2n1 N1(C(C(C)(C)C)=O)CCC(NC(=O)C(C)(C)Oc2ccc(F)cc2)CC1C1CC1 C1(CNC(CC2(C)CCCO2)=O)CC(O)CN1C(=O)CSc1ccc(O)cc1 Cc1cc(C(=O)NCC(C)NC(c2cc[nH]c2)=O)nc(C)n1 c1(C(=O)NCC(Cn2cc(CCCC)nn2)(C)C)cc2c(C)n[nH]c2cn1 C12(CNC(Cc3cc(C)no3)=O)CN(C(C3CCCCS3)=O)CC1CCO2 N1(C(C(C)(C)F)=O)CC(C(=O)NC2C(O)CC2O)C2(CC2)C1 Cc1cccc(C(C)NC(C2CCN(C(=O)COC3CCCC3)C2)=O)c1 Cn1c(C(N2CC3(CCC3CNC(C3(CO)CC3)=O)C2)=O)cnc1[N+](=O)[O-] C1(CNC(CCOC)=O)CCC2(CCC2)C1NC(c1cccc(O)c1C)=O CCCC(O)C(=O)NCCC(C(C)C)NC(=O)C(F)=C(C)C1CC1 C=CCC(C)(CC)C(=O)NCC(CO)NC(=O)CSC C1(C(=O)NC2(CC)CCCCC2)CCN(C(=O)C(C)OC(C)(C)C)CCO1 C(N=c1ccnc2[nH]n(C)cc1-2)c1nn(C)nc1Br C1(C(N2CCC(C3CCCCN3c3nnc(C4CC4)s3)CC2)=O)CC2CCC2C1 Cc1c(C(N2CCCC(O)(C(=O)O)C2)=O)cccc1Cl c1(C(=O)NC(C2CN(C(c3cnn(C(C)C)c3Cl)=O)C2)C)ncc2[nH]ncc2n1 C(C(C)(C)CC(=O)N1CCC(CNC(=O)C(O)Cc2cnc[nH]2)C1(C)C)N(C)C N1(C(CCNC(=O)CO)=O)CCCC12CCN(C(c1ccoc1Cl)=O)C2 C1(C(=O)NCC2CN(CC)C(=O)O2)CC2CCC(C1)N2C(=O)C(c1ccn(C)n1)C CC(CC(=O)NCC(C1CCC1)NC(c1nncn1C1CC1)=O)N1CCOCC1 NC(=O)CC(N=c1ccnc(NC2CC3CCCC3C2)[nH]1)c1ccccc1 CC1C(NC(=O)C=Cc2cccnc2)C(C)CCN1C(c1ccc(C(N)=O)[nH]1)=O CC(C)CC(CC(C)C)(c1nnnn1C1(C)CC1)NCc1cccc(Cl)c1F c1(OCC)cccc2[nH]cc(C(=O)N(C)C(c3ccccc3)C3CC3(F)F)c12 Cc1ccc2c(=NC(C)c3ccc(Br)cn3)[nH]c(=NCC(C)CO)[nH]c2c1 CC1CN(C)C(=O)CN1C(=O)CN(C1(CCN=[N+]=[N-])CC1)C(C)C N1(C(CCN(C(C2CC(C)(O)C2)=O)CC2CC2)=O)CC2(COC(=O)C2)C1 C=CC(C)CC(=O)NC1CCC(N2CCN(C(C3COC(=O)O3)=O)CC2)CC1 c1(-c2cccc(OC)c2)nc(=NCC2CCOC(C(C)C)C2)s[nH]1 C1(C(=O)OC)CC(N(C)C)C1.C1(=O)C(C)C(=O)CN1C1(OC)CC1 c1(OC)cccc(CN2CCCC(C(=O)NCC3CCO3)C2)c1C C1(COC)(NC(=O)CC(F)(F)F)CCCN(C(c2ccccc2C(C)(C)C)=O)C1 C(CC)(CCC(=O)N(CC(O)CF)C)NC(c1[nH]cc(C(C)=O)c1)=O C1(C(N2CC(F)(CNC(=O)C(CC3CCC3)OC)C2)=O)(CC)CC(=O)C1 N1(C(C2(C)CCNC2=O)=O)CC2(C1)CN(C(=O)C=Cc1cn[nH]c1)CCO2 c1(C(N2CCN(C(C3CCCSC3)=O)C3CC23)=O)ccc2c(O)nnc(O)c2c1 c1(NC(N2CCC(N3C(=O)CCC3=O)C2)=O)cc([N+](=O)[O-])n[nH]1 CC(C)CC(O)CC(=O)NCc1ccc(C(=O)NC2CC3CCC(C2)O3)c(F)c1 C1(NC(c2c(CNC(Cc3c(C)cccn3)=O)nnn2C)=O)CC2C=CC1CC2 C1(NC(C2CCCN(CCC)C2)=O)CC2(CCCN(C(c3cn[nH]c3)=O)C2)C1 Cc1cc(C(=O)NC(CNC(C2CCCC2O)=O)C(C)(C)C)nn1-c1ccccc1 CC1CCCn2c(C(C)(C)Cn3ncc(NC(=O)C(c4cccnc4N)O)c3)cnc21 n1(CCC(=O)N(CCNC(C2CCC(CC)C2)=O)C)c(C)cc(O)cc1=O c1(CNC(C(C2CCC2)OCC)=O)ccc(C(=O)N(CC(F)(F)Cl)C)o1 CC(C)(CC1CC1)C(=O)NCC1CCCCC1C(=O)NC1(C(O)CO)CC1 C1(C2CN(C(=O)CN3CSCCSC3)C2)(NC(c2c(C)cc(C)s2)=O)CC1 N1(C(CSCC)=O)CC(N(C(=O)CC(Cl)Cl)C)C(C)(C)C1 c1(C(N2CCCC(CNC(CC(COC)(C)O)=O)C2)=O)cnc2ncnn2c1C C12(NC(C3(NC(C)=O)CCCC3)=O)CC(C1)N(C(c1scc(C)c1C)=O)C2 c1(C(N2C3CN(C(c4c(OC)nsc4)=O)CC2C3)=O)ccc2cncn2c1 C1(CC(=O)NCCCC(C)NC(=O)C(F)(F)c2cccnc2)CC2(CCC2)C1 C(=O)(CC(C)C(=O)NCC(C)(F)CNC(C1CN(C)CCO1)=O)OC C1(CNC(=O)NC(CCNC(C2CC(C(=O)OC)C2)=O)=O)CCCOC1 N1(C(=O)Nc2ccc(C)[nH]2)C2CCC1C(C(=O)Nc1cccc(Cl)c1C)C2 C1(OC)CN2CCCC2(C=O)C1.C(=O)(CC(C)C(F)F)NCC(C(C)C)N C(c1ccc(Cl)cc1)=CC(=O)NCC1C2CN(C(C3C(C)(C)CCO3)=O)C1C2 c1(C(N(CCCCNC(C2C3CCC(=O)C23)=O)C)=O)n[nH]cc1[N+](=O)[O-] C#Cc1ccc(C(=O)NC(CNC(=O)C(C(C)C)SC)C2CCC2)c(C)c1 O=C(CC1CN(C(=O)NC(=O)C2CC2)CCO1)N=c1cc[nH]c(C(F)(F)F)c1 C1(CCNC(=O)Cn2nccn2)CCCCN1C(c1ncncc1Cl)=O C(CCCCC(=O)N1CCN(C)C(CNC(C2CCCC(C)(C)C2)=O)C1)OC C1(OC)CNC(=O)C1.C1(C)(C(=O)NOC2CCOCC2)C=CCC1 c1(CN2S(=O)(=O)CCC2)cc2cc(OC)ccc2nc1Cl.c12ccc(cc1)o2 c1(C(=O)NC(CNC(C2(CCOC)CCC2)=O)(C)CC)ccc(F)c(Cl)c1 C1(NC(=O)C=Cc2ncco2)C=CCN(C(C2CCC(=O)N2)=O)C1 c1(N(C(C)(O)C(=O)c2ccccc2)C(C(C)SC(=N)N)=O)ccc2ccccc2c1 c1(C(=O)OC)cc(C)nn1CC(=O)NC(C)CN(C)C(C1(F)CCCC1)=O c1(COC2CCCN(C(c3c(OCC)nn(C)c3)=O)C2)ccc(C(=O)O)c(F)c1 C1(C(=O)NC2CC3(C(NC(C4(C)C=CCC4)=O)C3)C2)CC(F)(F)CCC1(C)C c1(C(=O)NC2C(C)CN(C(=O)Cn3ncn(C)c3=O)C2)cnc2sccn2c1=O CC(C)(C(=O)Nc1ccc(-c2ccco2)[nH]1)c1cccs1.C12CC1CNC2=O C(=O)(CCN=c1cc(C)[nH]c(=NCC2CC3C(C2)C3(F)F)[nH]1)NCCC C1(C(=O)NC(CC#C)C(=O)NCC2CC3(CCC3)CO2)CC(C)(C)CCO1 C1(C(=O)NCCCN(C(=O)CSc2ccncc2)C)CC2(CCC2)CO1 C=CCC(C(=O)N1CCC(CC)C1C(N1CC(CO)CC1CO)=O)NC(C)=O C(=O)(CC(O)C(C)C)N1CCC(NC(C2(CC)CC2)=O)C1 N1(C(COCCOC)=O)CCC(NC(c2c(SC)cccc2F)=O)C1(C)C c1(C(N(CC(CNC(CC(C)(C)OC)=O)O)C)=O)cnc2cc(Br)ccn12 C(C(C)(C)CCNC(=O)C=C(C)C1CC1)NC(CCN(C(CCC)C)C)=O c1(-c2cn(CCN(C(C34COCC3C4(F)F)=O)CC)nn2)ccccc1[N+](=O)[O-] CC1(C)CCCC(C(CO)NCC2CC3CCC(C2)S3)C1 c1(C(=O)NC2C(CNC(C(C=C)(C)CC)=O)COC2)c[nH]c2c(Br)cccc12 c1(NC(C2C(NCc3cc(C)cc(F)c3)C2)=O)c([N+](=O)[O-])ncn1C C1(C(=O)NC(COC)CCl)CC12CN(C(=O)C=CC1CC1)C2 CC1C(C)N(C(=O)OCc2ccco2)CCN1C(=O)CN(C1CCC1)C C1(C)(CCNC(CCOC)=O)CCN(C(=O)C(C)Cc2ccc(N)cc2)C1 c1(CNCCCNC(c2coc(C3CCC3)n2)=O)cccc(C(F)F)c1 C1(NC(COCCCOC)=O)(CO)CCN(C(C2CCC3(CC3)C2)=O)C1 C1(OC)CC(NC(c2cscn2)=O)CN(C(=O)C(C)(O)c2ccccc2)C1 C1(OC)CC(CC(=O)NCCC(C)(C)NC(c2cnccc2Br)=O)C1(C)C C1(CC)CC(NC(=O)NC(C)C(C)(C)CN(C)C)CC(=O)N1 C1(NC(C(C)CN2CCCCC2)=O)CCN(CCC2CCCC2)C12CCC2 Cc1ncc(C(=O)NCCC2CCCN(C(c3sc(=N)[nH]c3C)=O)CC2)cc1N CC1(C)CCC=C(C(=O)NC2CN(C(C3CC34CC(F)(F)C4)=O)CCC2(C)C)C1 C12(NC(COCCCC)=O)CCC(CC1NC(=O)CCCCN(C)C)C2 C1(CC2C(C)(C)CO2)CCN(C(=O)C(=O)NCCc2ccccc2F)CC1 C1(C(=O)NCC(C2CCN(C(C3(C(F)F)CC(=C)C3)=O)CC2)C)CN2CCC1CC2 C(CC(C(=O)NC1(c2cc(Br)cs2)CC1)N1CCCC1)SC N1(C(CCC#CC)=O)CC2(CC(NC(c3cccc(OCC=C(C)Cl)c3)=O)C2)C1 C1(CC=C)(NC(C2CCN2CC)=O)CCCN(C(=O)CSC2CC2)C1 C1(C(=O)NCc2c(C(=O)NCCOCCC(C)C)[nH]cc2)CC2(CCO1)CC2 C=Cc1cncc(C(=O)NC2CN(C(=O)C(=CC3CCCC3)C)CCC2CO)c1 C(CC(C)(C)NC(c1cc(C2CC2)on1)=O)NC(C(C)N(C1CCCC1)C1CC1)=O C(CCCCCNC(C1CC(=O)N(c2nccs2)C1)=O)N(C(C1C(C)C1C)=O)C c1(C(=O)NC2CCN(C(c3ccc(CC)o3)=O)C2C)cc2scc(Cl)c2[nH]1 C1(C(N(C)CCc2nccs2)=O)CCCCN(C(=O)CCCF)C1 C12(C(=O)NC3C4CC(NC(c5c(C)n(C)cc5)=O)CC43)CC3CC(CC1C3)C2 C#Cc1cc(C(N2CCC(NC(=O)C(C)(C)OCC=C)C2)=O)cc(Br)c1 Cc1cc2c(cc1Br)N(C(C(=O)NCC1CC1(Cl)Cl)C1CC1Cl)CCO2 c1(C(N2CCC3CN(S(=O)(=O)c4ccc(Cl)s4)CC23)=O)cccc2ccnn12 c1(C(=O)NC(CN(C(CCC)=O)C)CC)ccn2ccnc2c1 CC1CC2(CC(C(=O)NCCCCC(=O)N3CCOCC3)C2)C1 C(C)(C)(C(C)CC(=O)NCc1cn(C(C)C)nn1)NC(CCC(C)=O)=O CC(C)CCC(O)C(=O)N1CCCC(CC(=O)NC2C(O)CC2O)C1 c1(OC)ncc(C(N2CCCC2C(=O)Nc2cncc(F)c2C)=O)cc1Cl N1(C(C(CC)N(C)C)=O)CCC(CNC(c2ccccc2OCCF)=O)(OC)C1 CC1(C)CN(Cc2cc(C(=O)O)cs2)C(C)(C)C1O N1(C(C2C(C)(C)CC2)=O)CCn2c(CNC(C3(C)C=CCCC3)=O)nnc2C1 c1(OCCC)ccc(C(N2CCSCC2C)C(=O)NCC(C)C)c(OC)c1 c1(C(N(CC(O)CNC(=O)COCC(F)F)C)=O)cnc2ncccn12 C1(CNC(c2ccc(C)n2C)=O)CN2CCCCC2CN1C(=O)COCC(F)F N1(C(c2nn(CC)c(C)c2)=O)CCC12CN(C(c1cc(CC(C)C)c[nH]1)=O)C2 C1(CCCC)CN(C(C2CC2C(=O)OC)=O)CCN1C(=O)CP(C)(C)=O c1(OCC)oc(C)nc1C(N1CC(CNC(=O)C=CC2(C)COC2)C(O)C1)=O C1(NC(C2N(C(C(CC3CCC3)OC)=O)CCC=C2)=O)CN(C)C2(CCC2)C1 c1(CC(CNC(=O)C(=O)NCC2CC3C=CC2C3)CO)ccccc1F c1(COC(c2c(=O)ccn(C)c2)=O)cc(F)c(Br)c(F)c1 C#CCCC(C(=O)NC1CC12CC2)NC(C1CN(C)C1)=O c1(CCC(N2CCN(Cc3ccc(Br)cc3F)C3CC23)=O)ccc(Cl)c(Cl)c1 c1(OC)cccc(-c2nc(COC(C3CC3c3cccc(C)c3)=O)cs2)c1 c1(CC)cscc1C(=O)NC1(CNC(c2cnsc2C)=O)CCOC1 CC(C)CCC(F)C(=O)N1CC(NC(C2CCC(CO)CC2)=O)CC(C)C1 C(C)(CNC(c1c[nH]nc1-c1ccoc1)=O)(C(C)C)NC(Cc1c(C)nc[nH]1)=O C(CC(=O)NCCC(Cc1ccccc1)NC(C1CCOC1)=O)(C(N)=O)NC(C)=O c1(NC(C2N(C(C(CC)C)=O)CCC2C)=O)cccc(C(F)F)c1OC(C)=O O=C1CC(C(=O)NOC2CCC(CCO)C2)CN1CCO.C(=O)CSC(F)F O=C(NOCC(=O)NCC(N1CCCCC1)=O)C(F)(F)CCn1ccnn1 C=CC1(CC(=O)NC2CC(NC(=O)C(C)c3cccs3)C2)CCOCC1 Cc1ccccc1CC(=O)N(C(C)C(=O)N(C)C(C)C)C Cc1ccc(CCNC(=O)C(=O)NC2C=CCCC2c2ccccc2)cn1 C1(C(N2CCCC(NC(CC3COCC(C)O3)=O)CC2)=O)CC2CC1C(O)C2O C(c1ccccc1OC)=CC(N1CC(NC(C(c2ccc(CC)s2)=O)=O)C1)=O Cc1c(O)c(=O)ccn1CC(=O)NCC(C1CCCC1)NC(=O)C(C)n1ccnc1 C1(CNC(CCCC)CO)CC2C(C1)C2(F)F.C1(=O)C(C)CC(=O)NC2CCCN12 c1(C(N2CCN(C(=O)CCc3ccccn3)C(CO)C2)=O)ccn2c1CSCC2 c1(NC2CCN(C(Cn3ccc(C)n3)=O)C(C)C2)ncnc2c1nnn2C(C)C c1(C(N(CCCN(C(C(C2CC(F)(F)C2)OCC)=O)C)C)=O)cccc(C#N)n1 CCCCCC(C)(C)C(=O)NCC(C)NC(=O)CCc1cccnc1F Cc1ccnc(Cl)c1C(=O)Nc1ccsc1C(=O)NCc1ccc(Br)cc1Br C1(N(C(=O)CSC2(CC3CC3)CC2)C)CCN(C(C2CCC2C)=O)CC1 c1(C(N(C)CC2CCCN2C(=O)CCF)=O)cc2cccc(Br)c2[nH]1 CCC(CC(=O)N1CC(NC(c2nnsc2C(F)F)=O)C(C)C1)c1ccccc1 N1(C(C2C(C)CCC2)=O)CCN(C(C2CC3(C2)CC3(F)F)=O)C2(CCC2)C1 Cc1ccc(NCC(N2CC(CNC(c3c[nH]cc3C3CC3)=O)C(C)C2)=O)cc1 c1(N2CCC(NC(C(CCC)OC)=O)C(F)C2)ncc([N+](=O)[O-])cc1C N1(C(N(c2cc(OCC)ncn2)CCCC)=O)CC(C2CC2)C1C1CC1 C(C(N)=O)C(=O)O.n1(C(C)C)ccc(C=O)c1.N12CCC(C1)CC2=O c1(CN2CC=CC2)cccc(C)c1.CCC1(C)CN(C)C(=O)N1 C1(NC(C2(CC#C)CCC2)=O)CCCCN(C(C2C3CNC(=O)C23)=O)C1 C1(NC(CC23CC(C)(OC2)C3)=O)CCC2CCN(C(c3c[nH]cc3Br)=O)C1C2 S(=O)(=O)(c1ccc(C)cc1C)NC(C(CC)NC1CCCCC12CCNCC2)=O c1(CCC(=O)NCC2C3CC2N(C(=O)C=Cc2ccoc2)C3)ccc(F)cc1F N1(C(C(n2cnc(C#N)n2)CC)=O)CC(NC(c2cnc(OC)nc2)=O)CC1(C)C c1(C(=O)NC2C(NC(C)=O)C2)cc(Br)c2nccn2c1 c1(N(C(C)=O)C)ccccc1C(N1CCC(CNC(=O)Cc2ccsc2C)C1)=O C(=O)(C1=Cc2ccccc2C1O)N1CCC(NC(CCC(=C)Cl)=O)(CC)CC1 c1(C(=O)NC2CC(C)(NC(CC3C(C)CCO3)=O)C2)ccccc1O N1(C(c2ccc(C(C)=O)nn2)=O)CCC(NC(c2cnc(C)nc2)=O)C(F)C1 C1(N(C)C)CC(CC(=O)NC(C2CCCC2)CNC(C2CC2F)=O)C1 c1(N2CCCC(CCC)CC2)nc2c(c(=NC(C)C3CC3)[nH]1)SCC2 C1(O)(C(C)NC(=O)CNC(N)=O)CN(C(=O)Cc2noc(-c3ccccc3)n2)C1 c1(C(=O)NCC(CNC(c2cccc(SCC)c2)=O)C)ccc(CC)cc1N c1(C(=O)NCCCCC(C)NC(C2C(C=C)OCC2)=O)ccc2c(c1)CCOC2 c1(C(N2C(CCNC(C(C)C3(O)CCC3)=O)CCC2)=O)coc2c1CS(=O)(=O)C2 n1(CCC(C)C)cc(Br)c(=NC(=O)c2cnn(C)c2)[nH]1 N1(C(C(C)n2cncn2)=O)CCCC(CCOc2ccccc2Br)C1 C1(NC(c2nc(OCC)oc2)=O)CC2CCC1N2C(C1CCCC1(F)F)=O N1(C(C(CNC(C(CC)C#N)=O)N(C)C)=O)CC2(CCC(=O)N2)C1 C(C)(CCCCCO)NC(C1(C)CN(C(c2nc(C)oc2C)=O)C1)=O C=CCCCC(C(=O)Nc1ccc(CC)c(F)c1)NC(=O)Cc1cncs1 C1(NC(Cc2cc(C(C)(C)C)on2)=O)CC(CO)N(C(=O)CC2C=CCC2)C1 c1(CN(C(C2C(CC)OCC2)=O)C)cccc(CNC(c2cccs2)=O)c1 c1(CSC)nn(-c2ccccc2)c(Cl)c1-c1ccccc1.C(CC(=O)N)S C=C(C)CC(C(=O)NCC1(C)CCCCC1)NC(C1CCC(=O)C1)=O c1(C(=O)NC(CC2CN(C(C3C(CCOC)C3)=O)C2)C)cccc(Cl)c1NC N1(C(Cc2ccn(CC)n2)=O)C2CCCC1CN(C(c1cc(C)cc(F)c1)=O)C2 Clc1cnc(SCCn2cc(-c3ccccc3)nn2)c(Br)n1 N1(CC(CNC(c2ccc(OC)cc2)(C)C)O)CCN(C)CC1 c1(C(C)=O)cc(-c2csc(C(C)CC)c2)cc(Cl)n1 C1(NC(C2(C)CC=CC2)=O)CCCCN(C(=O)CN2CCCC2=O)CC1 C(=O)(CCC(=O)N(C)C)NC(C1CCCN(C(=O)C(C2CC(F)(F)C2)O)C1)C CCC(CNC(C1CCNC(=O)C1)=O)(CC)NC(=O)CCc1ccc(NC)nc1 N1(C(CN(C)C(N)=O)=O)CCC(C2CC2)(NC(=O)C(C2CCOCC2)F)C1 c1(C(N(CC(C)CNC(=O)CCc2nc(C(F)(F)F)n[nH]2)C)=O)cnn(C)c1N CCC(CC)C(C(=O)N1CC(NC(=O)CP(C)(C)=O)CC(C)(C)C1)OC C=CC1CCCC(NC(=O)C(C)(CNC(c2cc(OC)no2)=O)CC)C1 C1(NC(=O)CNC(C2CCCCC2)=O)(CNC(=O)CC(F)F)CC(F)(F)C1 c1(CCNC(=O)C(=O)N(c2ccccc2F)c2cnn(C3CC3)c2)ccccc1Br CCS(=O)(=O)CCn1c(N(CC(C)C)C)nnc1C(c1nccs1)S.C1CC1 C(CCC(C)CC(=O)NC(C1CCN(C(c2ncsc2C)=O)C1)(C)C)=C(C)C Cc1cc(C(=O)NCC2N(C(=O)CS(N)(=O)=O)CCCC2(C)C)c(N)c(Cl)n1 c1(OC)cc(C(=O)NC2CCSC23CN(C(C2CC2(C)Br)=O)C3)cc(N)c1O C1(NC(C2CC(OC)C2)=O)CCN(C(=O)CCSC2CCCC2)C(C)C1 C#Cc1ccc(C(=O)NCC2(O)CCCN(C(=O)C(F)CCCCC)C2)cc1C C12(NC(CC)=O)CC(C)(C1)OC21CN(C(c2ccc3nc(=N)[nH]n3c2)=O)C1 n1(CC(N2C3(CNC(CC(=C)C)=O)CCC(CC3)C2)=O)ncn2cccc2c1=O O=C1CCc2cccc(C(N3CCOC(C(N4CCC5(C4)CC5(F)F)=O)C3)=O)c21 C1(N(C(CC(=C)C)=O)Cc2nccn2C)CCCN(C(=O)Cc2ccccc2C)C1 C(C(C)(C)C(=O)N1CCC(C2CCCCN2C(=O)C(O)C(C)C)CC1)OC c1(C(=O)NC2COCC2CNC(C2CC23CCCC3)=O)sc2ncccc2c1Cl N1(C(CCc2cc(C)[nH]n2)=O)CCCC(NC(c2csc(Cl)c2Cl)=O)CC1 C1(NC(=O)OC(C)(C)C)CN(N2CC3CCCCCC3C2)CC(C)(C)O1 CC(C)C(O)C(=O)NCC1CC(NC(C2CCCCN2CC(F)F)=O)C1 c1(C(N(C(CN(C(c2c(CC)nco2)=O)C)C)C)=O)cc2nc(C)[nH]c2cc1F N1(C(C(=O)N(C2CCCNC2)CCC)=O)CCC(C(C)(C)C)CC1 c1(-c2ncc(-c3n(CC(c4cccnc4)CC)ccn3)s2)cc(Br)cc(C)c1F C1(COC)CCN(C(=NCCc2ccc(F)cc2)NCc2nonc2C)C1 C(=O)(C(CN=[N+]=[N-])NC(c1snnc1C)=O)NCc1cnc(CC)[nH]1 c1(CNC(C(Cn2cccn2)NC(C(C)=CC)=O)=O)cnc(C(=O)OC)cn1 c1(N(C)C)ccc(-c2nc(Cc3ccn(C)c3)n(CCF)n2)nc1 N1(C(Cc2ccn(CC)n2)=O)CC2CN(C(C3(CC4CC4)CC3)=O)CC2(C)C1 C1(OCC)CC2CN(c3cc(NCCCN4CCC4)nc(C)n3)CC12 C(CCC(=O)O)(C(=O)N1CC2CCC2C1)NC(=O)OC(C)(C)C n1(CC)cc2ccc(NC(=O)NC3(C4CCC4)CC3(F)F)cc2n1 O=S(=O)(c1ccc(NCC2C3COCC23)c(Cl)c1)NCC1CCC1(F)F c1(C(=O)NC(CC)CNC(c2cnccn2)=O)ccc2c(C)cc(Cl)nc2c1 C1(COC)CN(C(C2OCCC2CNC(c2nonc2C)=O)=O)CCO1 C1(NC(C(C)(O)C2CCC2)=O)CC(C(=O)NCCCCCCCC2CC2)=CC1O C1(C(N2CC(O)(CCC)C2)=O)CNC(=O)CN1C(=O)COCC(F)F C1(C(N(CC(C)NC(CC2(C=C)CCOCC2)=O)CC)=O)CCCCC(C)(C)C1 n1(CC)ncc(C(N2CCC(CC(=O)N(C3CC3)Cc3nc[nH]n3)C2)=O)n1 c1(NCCN(C)C(N)=O)cnc(CC2CCN(c3nc(C(F)(F)F)ns3)C2)o1 c1(C(c2n(CC)nnn2)NC(c2coc(C)n2)C2CCC2)ccc(F)cc1 Cc1ccc(Cl)c(C(N2CCCN(CC3CC3)CC2)C(=O)NC2CCOC2)c1 CCC(F)(F)C(C)(C)C(=O)NC1CCCC(NC(=O)CCn2cnnn2)CC1 C(=O)(NNC(=O)C(C)(C)CCCCNC(C1CCC1)=O)c1c(C)ocn1.CC1CC1C Cc1ncnc(C(N2CCN(C(c3cnn4c3CCC4)=O)C(CCO)C2)=O)c1C c1(NC(C2CN(C(c3cccs3)=O)CCO2)=O)ccc(I)c(Br)c1 C(=O)(C1CCCc2scnc21)NCC1N(C(C2=CCCC2(C)C)=O)CCC1C1CC1 C(C1=CCCN(C)C1)NC(C1CCCN(C(c2c(C)occ2C(F)(F)F)=O)C1)=O Cc1ccc(F)c2oc(C(=O)NCC3(NC(c4ccnc(S)c4)=O)CCC3)cc12 c1(C(=O)NCCn2cc(C(N3CC=CC3)=O)nn2)ccc(O)cc1 C=CC(C)C(C)C(=O)NC1CC(NC(C2CC(F)(C(=O)OC)C2)=O)C1 c1(NC(CCCN(C(=O)OC)C)=O)cc(C)cnc1O.C(CCC=O)C1CCC1 C12(NC(CC(=O)NCC#C)=O)CCCC1CN(C(=O)C(C)(F)F)C2 c1(NCc2c(C(C)(C)C)noc2)[nH]c(=NCc2n[nH]c(=N)o2)nc2scnc12 C#CCCN=C(NCC1(CC2CCC2)CC1)N1CC(C)CC(C)C1 N1(C(C(c2ccnn2C)NC(C2=NOC(C)C2)=O)=O)CC2CCC(C1)C(=O)O2 c1(CC)cccc(C(=O)NC(C2CCN(C(c3[nH]ccc3C)=O)C2)C)c1 C1(C(=O)NC2CC(NC(Cc3cn(C(C)C)nn3)=O)C2)CC2(CC(=O)C2)C1 c1(C(C(=O)NCC(C)NC(c2cc3c(s2)CCC3)=O)=O)ccc2c(c1)CCOC2 N(C)(C(=NCC1CC1)NCC(c1cc(F)cc(Cl)c1)O)Cc1cccc(OC)c1 c1(C(=O)OC)cnccc1CNC(=O)CCC1(C)CCCN1C(=O)C#CC(C)C Cc1cc(=N)[nH]cc1C(=O)NCC(C)(C1CCC1)NC(c1cccs1)=O c1(C(=O)NCCN(C2CC2)Cc2n(C)ncc2)cc2ccoc2c(O)n1 N1(C(CCC(=O)N(CCC)CCC)=O)CC(=O)NC2CCCCC12 CCC(CO)CN=c1cc(NCC23CCOC2CN(C(C)=O)C3)nc(C(C)C)[nH]1 C1(C(N2CC3(CC(=C)C3)C2)=O)C(C2CC2)CCN1C(c1cc(C)cc(F)c1)=O Cc1cc(S(N)(=O)=O)ccc1NC(=O)NCC(C1CCCCC1)OCCCO c1(C(N(CCNC(C(CCC)OC)=O)CC2CC2)=O)cncc2ccc(F)cc12 Cc1cc(Br)cc(C(N2CC(F)(CNC(C3OCCN(C)C3=O)=O)C2)=O)c1F C1(C(=O)NCCC#CCC)C(CC)CCN1C(=O)C=NOC C1(C(=O)NCC2(COC)CC2)CCC(F)(F)CC1.C1(=O)C(CC2CCOCC2)N1 c1(C(N(CCC(C)NC(c2cnccc2Cl)=O)C)=O)cnc(O)c2ccsc12 C(CN=C(NCC1(F)CCCCC1)NC1CC1)=C(C)C1CC1 N1(C(C(C)NC(C=C)=O)=O)CC(C2CCN(C(=O)CSCCN(C)C)CC2)C1 CC(C)CCCCC(=O)N1CCCC(CNC(C2(C)CC(C)C2)=O)CC1 CCC(O)C(C)C(=O)NCC1C2CC1N(C(c1cc(F)ccc1C(F)(F)F)=O)C2 C1(N=[N+]=[N-])(C(N(CC(=O)NC)CCC)=O)CCN(C(=O)CCCC2CCCC2)C1 C12(NC(C3CC4(C3)CC(F)C4)=O)CCCC1N(C(c1cccnc1N)=O)CC2 c1(C(CNC(=O)CCCC2CC2)N(C)C(C2(F)CCC2)=O)ccc(Br)cc1 Cc1cncc(CC(=O)NC(C)(CNC(C2CC2(F)F)=O)CO)c1 N1(CCC(C(C)C)N)CCC(O)(C2CCC2)CC1 C1(C2CC2)(C(=O)NCCc2n(C)ccn2)CCN(C(c2ccco2)=O)C1 N1(C(C(C)N(C)C)=O)CC2CC(NC(c3occ4c3CCCC4)=O)C(C2)C1 C12(NC(=O)CCn3cnccc3=O)CCCC1N(C(C1CSC1)=O)CC2 c1(OC)ccc(F)c(CNC(=O)CNC(c2ccsc2)=O)c1.C12CC1C(=O)NC2 CC(C)C(O)CC(=O)NC1CN(C(=O)C(O)CF)CC1O N1(C(CCC=CCC=C)=O)CCCCC2(C1)CN(C(c1cnccn1)=O)C2 c1(C(=O)NCC(CC(C)C)NC(c2ncoc2C2CC2)=O)ccnc2cc[nH]c12 C=C(C)CC(C)C(=O)NCC(C)(CO)NC(=O)CC1(O)CCOCC1 c1(C(=O)NC2(CNC(C3C4CC4C4CC34)=O)CC2)cn2ncccc2n1 C1(C(C)NC(=O)C(C2CC=CCC2)N(C(c2cccs2)=O)C2CC2)CCCC1O c1(OC)cc(C(=O)OCc2ncc(Cl)s2)cc2c1OCO2 N=c1cc(C(N2CCC(CO)(NC(=O)C3=COCC3)CC2)=O)c(Br)c[nH]1 C(=O)(C(C)(C)CC(F)F)N1CC(CC(=O)NC(C(C)C)CCO)OCC1 CC1CC(NC(=O)CN2CCCCCC2=O)CCN1c1nccnc1F C1(CCN)CCC(NCC2CCCCC2c2ccccc2)CC1 Cc1[nH]nc2cc(C(N3CC(NC(C4CCS(=O)CC4)=O)CC3CO)=O)ccc12 C1(NC(C2(CCNC(=O)CCn3cccc3)CC2)=O)CC(C2CCCC2)C1 C1(NC(c2c(C(C)C)cccc2)=O)CCC(S(C)(=O)=O)CC1 c1(N(CCCC)C)ccc(C(=O)NCC(O)CNC(C2CC2C(F)(F)F)=O)cc1 N1(C(C(C)c2ccsc2)=O)CCC2C1CCCN2C(c1cc(Cl)c(F)cc1Cl)=O c1(C(=O)NC2C3(CC(NC(COCC=C)=O)C3)C2)ccc(N)cc1C Cn1cccc1CC(=O)NC1(C)CC1C(=O)O CCCC(C)(O)CC(=O)NCCn1cnc(CNC(=O)CC(C)(C)C#N)c1 C1(C(=O)NCCC2(OC)CCC2)CN(C(=O)Cc2cnc(C)s2)CC12CCC2 CC1CN(C(c2c(F)cccc2Cl)=O)CCCN1C(C1CCCC1(F)F)=O CCCCCC(C)(C)C(=O)N1CCC(N(C(=O)CCCN(C)C)C)C1 c1(NC(C(C2CCOCC2)NC(C)=O)=O)cccc(CNC(=O)C(C)C2CC2)c1 C1(CNC(C2(CC)CC2)=O)CC(C)(C)CCC1NC(c1c(C)nc(C)n1O)=O C12(C(=O)NC(C3CCCN(C(=O)CN(C)C4CC4)C3)C)CCC(CC1)CC2 C(C(=O)NOCCC1CC1)(C)(O)NC(CCCCOC)=O N1(C(C(CCC)NC(=O)CC2CC2C2CC2)=O)CC(C)OCC1C N=c1[nH]cncc1C(N1CC2C(CNC(c3coc(CC4CC4)n3)=O)C2C1)=O C12(CNC(c3c(C(N)=O)csc3)=O)CCC1CCN2C(c1ccnnc1)=O C(=O)(C(C)(CC)C(=O)NCCC1(O)CN(C(c2ncc(F)cn2)=O)C1)OCC c1(C(=O)NC(CC#C)C(=O)NC2(C)CS(=O)(=O)C2)ccc(F)c(C)c1 CC1(C)CCCCC1NC(N1CCC(=CC(N2CCOCC2)=O)CC1)=O c1(CC(=O)NC(C)CCNC(=O)C(C)N2CC2)ccccc1Cl n1(CCC)nc(C(=O)NCCNC(=O)C=Cc2nccs2)cc1C C1(CNC(C2CC(OC)C2)=O)CCC2(CN(C(c3ncccc3Cl)=O)C2)O1 c1(C(N2Cc3c(C(=O)NCC4CCC4)ncn3CC2)=O)cc(F)cc2cc[nH]c12 N1(C(c2cccc(OC)n2)=O)CCN(C(C2(C)CCCCC2C)=O)CC(C)(C)C1 C(=O)(CCCCCS(N)(=O)=O)NCC(CN(C(=O)CCn1cnnn1)C)O Cc1cccc2c1OC(C(=O)NCC(C)(O)CNC(=O)CNC1CCCCC1)C2 c1(C(CC)C)ccccc1OCC(N1CC(NC(=O)CCc2cccs2)C(C)C1)=O Cc1nc(O)ccc1C(N1CCCC(CCNC(c2cc(=O)cc[nH]2)=O)CC1)=O c1(CC(=O)NC2(CO)CCN(C(c3cc(OC)n[nH]3)=O)C2)cccc(Cl)c1F CC1CC(C(=O)N(CCCNC(c2snc(Cl)c2C#N)=O)C)Cc2nn[nH]c21 N1(C(CCN(C)CC)=O)CCC(C)(CNC(c2ccc(C)cc2SC)=O)CC1 N1(C(CC(=C=C)C)=O)CC(NC(=O)C=Cc2nc(C)cs2)CC2(CC2)C1 Cc1c(Cl)ccnc1C(=O)NCC1(CNC(=O)CC2CCN(C)C2)CCCC1 C(=O)(CCC[N+](=O)[O-])N(CC(C)CNC(c1ccn(C)c1)=O)C C1(CN(c2ncccn2)CC)CCCCN1C(C1(CC(C)C)CCNC1=O)=O C1(N=c2[nH]c(=NCC3(C)CS(=O)(=O)C3)[nH]c3ccc(F)cc23)(CN(C)C)CCCC1 N1(C(c2cncc(C)n2)=O)CCC2CN(C(C3CCC34CCC4)=O)C2C1 C1(S(N)(=O)=O)(C(=O)NC(C(C)(C)NC(C(C)SC(F)(F)F)=O)C)CCC1 Cn1cnc(C=C(F)C(=O)NCC(CC(=O)O)NC(=O)CC2CC2)c1 c1(C(=O)NCC2CCCN2C(=O)CCc2cccc(CO)c2)ccc([N+](=O)[O-])o1 C12(NC(C(CCC)NC(N)=O)=O)CC3CCC(C1C2)N3C(=O)CNC(=O)C1CC1 N1(C(C2C(C=C)CC2)=O)CCC(OCCCNC(=O)CSC)CC1 c1(N(C)C)cncc(=NC(=O)C(=O)NCC2CCC(=O)N2)[nH]1 c1(C(C)C)ncc(C(=O)NC2CCC(C(=O)CCN3CCCCC3C)C2)cn1 c1(C(=O)NCC(C)NC(=O)C(F)(F)C(C)(C)O)cnn2c1OCC(C)(C)C2 S(=O)(=O)(c1ccc(NCCOCCC)nc1)NC1CC(C)SCC1 C1(C(C)NC(=O)CC2CC(C(F)F)C2)CN(C(c2nccnc2N)=O)CCO1 C(=O)(C(C)C(O)CC(C)C)NCC1CCCN(CC(=O)NCC)C1 C(CC(CNC(=O)C(C)C#N)NC(c1ccc(C2CC2)s1)=O)OC.c1(S)ccccn1 C1(CC)CCN(C(=O)OC(C)(C)C)C1C(=O)NCC1CCSC1 CCCC(C)C(=O)NCC(CO)NC(=O)C(C1CCCCC1)F C=C1CC2CC1CN2C(c1ccc(C(C)(C)C)o1)C(=O)NCCCF C(C)(C)(CCCC(=O)NCC(CC)(CC)CO)NC(C(CC)OC)=O Cc1cccc2sc(N3C4CCC3CN(C(c3cnc5c(cnn5C)c3)=O)C4)nc12 c1(CC(=O)N(CC(C)(C)NC(=O)CC2CCCC(C)(C)C2)C)cc(F)c(F)cc1F Cc1c(C(=O)N(CCCc2ccccc2)C(C)C2CC2)cnn1-c1cccnc1 N1(C(C=CC(C)=O)=O)CCCC(C2CCN(C(=O)C(C)OC3CCCC3)C2)C1 Cc1nn(C)c2c(NCC3(C)CCOC3)nc(N3CCC(C(F)F)C3)nc12 N1(C(c2ccc(C)c(O)n2)=O)CC2CCCC(C1)N2C(=O)C(C)(C)N=[N+]=[N-] n1(CC(=O)NCCC2CC(NC(c3c(C)noc3)=O)C2)ccc(=O)c([N+](=O)[O-])c1 Cc1cc(C(=O)NCc2ccsc2C(=O)NC2CCOC2(C)C)ccc1C#N C(=O)(CC(CC)c1ccccc1)N1CCC(N(C(C=CC)=O)CC)C1 c1(CC)ncncc1C(N1CC(CC(=O)NCC2(O)CCOC2)CC1C)=O C1(CCC)CCN(C(=O)CC(C)(C)NC(c2cc(C(N)=O)[nH]n2)=O)CC1 c1(CCC(N2CC(N(C(=O)CCCc3nc(C4CC4)no3)C)C2)=O)cncc(F)c1 c1(C(N(CC(=O)NCc2c(CC)con2)C2CCC2)=O)cccc(OC)c1F c1(C(C(=O)NCC(C)(CO)NC(C(C)SCCCC)=O)(C)C)ccc(Cl)cc1F C1(CCC)(NC(c2ccc(O)c(N)n2)=O)CCN(C(c2[nH]ccc2C)=O)CC1 Cc1ncc(C)c(=NCCC2CCN(C(c3cnn(CC(F)(F)F)c3)=O)C2)[nH]1 C1(CCNC(Cc2nnc(C)o2)=O)CCCN(C(c2cccc(Cl)c2)=O)C1 c1(C(=O)NCc2ncn(C)c(=O)c2)ccccc1S(=O)(=O)NC(C1CCCC1)=O c1(Cc2cc(C)[nH]n2)nc(-c2cncs2)nn1C1CCSCC1 Cc1cc(O)cc(O)c1CNC1CCC(C(N2C3COCC2CC(F)C3)=O)C1 c1(CCC(=O)NCC(CN(C)C(c2coc(O)n2)=O)O)ccc(Br)cc1 C(=O)(C(C)(CCC)CCC)N1CC2C(C(=O)OCC(C(=O)C(F)(F)F)=O)(C2)C1 C1(C(=O)NCC2(NC(CCOCCC)=O)CCC2)CC(O)C(F)C1 C1(C(N2C(C3CCN(C(CCOC(C)=O)=O)CC3)CCC2)=O)Cc2cccnc2C1 N1(C(C2(CC)COC2)=O)CC2CN(C(C3CC4CCCCCC34)=O)CC2C1 C(=O)(C(F)(F)C(C)(C)O)N1CC2N(c3cc(-c4ccc(CC)cc4)nc(Cl)n3)C2C1 C1(C(=O)NCCCCCC)CCOC12CCN(C(=O)Cc1ncc(C)s1)CC2 C1(NC(Cc2c(C)ccnc2)=O)CCCC(NC(c2cc(Cl)ns2)=O)CC1 C1(c2cn(C(C)CNC(=O)CN3CCC(C)CC3)nn2)(OC)CCSCC1 c1(C(=O)NC2(c3ccccc3)CCN(C(C)=O)C2)ccc2c(c1)B(O)OC2 C1(C(N2CC(NC(c3cc(C)on3)=O)C(O)C2)=O)(NC(C)=O)CCCCC1 C=CCC(C)(C)CC(=O)N1CCCCC(NC(c2cncc3c2CCC3)=O)C1 N1(C(c2c(C)coc2)=O)CCC(c2ccccc2)(NC(=O)CCOCC(C)C)C1 c1(C2(C(=O)NC3CCC(n4cc(C(C)O)nn4)C3)CC2)ncccc1C c1(C(=O)OCC)c[nH]c(=NCC2CCCN2C(=O)Cn2ccnn2)s1 C(C(C)(C)C(=O)N(CC(O)CNC(=O)C(c1ccccc1)=O)C)OC(C)C N1(C(C2N(C(C(CC)NC)=O)CC(C)CC2)=O)CC(OC)C2(CCC2)C1 Cc1ccc(CC(N2CC(F)(C(=O)N(C)CC3CC3C)C2)=O)s1 N1(C(Cc2c(C)cnn2C)=O)CCN(C(=O)CC2COCCOC2)C(C)C1C CC(C(=O)N1CCC(n2cc(-c3cccs3)nn2)C1)S(N)(=O)=O CC(C)(C(=O)N1CCC(O)(CNC(c2ccc(N)cc2Cl)=O)C1)C1=CCSCC1 c1(C(=O)NC2CC(C)N(C(C3CC=CCO3)=O)CC2)cn2cccnc2n1 c1(OC)ccc(C)c(F)c1-c1ccc(C(=O)NCC2CC3C=CC2C3)nn1 N1(C(C2CCC(C)O2)=O)CCCC12CCN(C(c1cc(C3(C)CC3)on1)=O)C2 c1(CCC(=O)NCC(O)CNC(=O)C(=O)Nc2ncc[nH]2)ccncn1 c1(OC)c(C(=O)NC2COCCN(C(=O)C(C)c3cccs3)C2)c(C)nn1C CCC(C)(C)C(=O)OC.c12ccc(cc1)-n1cc(nn1)C(C1CCC1)NC2 C(=O)(C(CCF)NC(=O)CCCn1cncn1)N(CC(=O)NC(C)C)C C1(NC(c2cccc(NC(C)=O)n2)=O)CCN(C(=O)Cn2ncnn2)CC12CC2 c1(NC(=O)CC2CN(C(c3ccc4c(c3)OCC4)=O)C2)n[nH]c2cccc(F)c12 C(C(C)(CC(C)C)NC(=O)C#CC1CC1)NC(c1c(CC)nco1)=O c1(C(N(CCC)C)=O)cccc(C(=O)NC(=O)CCNCc2nn(C)cc2Br)c1 C(=O)(C1=NOC(C)(C)C1)NC1C(CNC(c2cc(C)nc(O)n2)=O)CCCC1 CC1CN(C(=O)C(C2CCOCC2)=O)CC1CC(=O)NC(C1CCN(C)C1)C C1(C(=O)NCC(C)(C2CCC2)NC(c2cnc(N)cn2)=O)CCC(=O)NC1 CC(C)CCN=C(NCCn1cccc1)NCc1cc(S(C)(=O)=O)co1 c1(C(=O)NC2C(C)N(C(=O)CCC3CCC(=O)N3)CC2)ccccc1P(C)(C)=O CCCCC(CNC(C1(C#N)CC1C)=O)NC(c1ccc(CC)nc1)=O c1(C(N2CCN(C(C(CC)C(C)C)=O)CC2C2CCC2)=O)c(C)nc(C)nc1C Cc1cc(C)c(O)c(S(=O)(=O)NC23CCC(C2)N(C(c2ccco2)=O)C3)c1 C12(C(N3CCC(N(CC(=O)NCc4cc(OC)ns4)C)C3)=O)CC3CC1C2C3 C#CCC(C)C(=O)NC1CCC1CNC(c1cncs1)=O c1(NC(C2N(C(Cn3c(C)nc(C)n3)=O)CCSC2)=O)c(C)cc(Br)cc1Cl N#Cc1ccc(S(=O)(=O)NCC=Cc2cncs2)cc1F C1(CNC(C(C)=C(C)C)=O)CN(C(c2nc(C3CC3)cs2)=O)CC1(F)F C(=O)(C(C)(C)C(=O)N1CC2(C1)CN(C(c1ccc(CO)c(F)c1)=O)C2)NC C1(CNC(c2nc(C(=O)OC)sc2)=O)CN(C(c2cc(CO)[nH]n2)=O)CC12CC2 CCC(C)(C)C(C(=O)N1C2CCC1CN(C(c1c(C)cc(C)oc1=O)=O)C2)OC c1(C(=O)NC(C(C)C)C(=O)NCc2nccn2C(C)C)cc2n(n1)CCC2 C1(CNc2cn(CC3C(OC)CCC3)nn2)CCCCCN1C N1(C(c2cnc(S(C)(=O)=O)s2)=O)CCCC12CCN(C(=O)Cc1cscn1)CC2 Cc1cccc(C(N2CCCCCC2CNC(c2ccnn2C)=O)=O)c1N C(=O)(CCCC(F)(F)F)NCC12C(CN(C(c3c(OC)ncc(Cl)c3)=O)C1)C2 N1(C(c2cc(C)cc(O)c2)=O)CCC2CCN(C(=O)CC3=CCOCC3)CC12 N1(C(c2ccc(OC)s2)=O)CCC(C(C)NC(c2cc(C3CC3)ns2)=O)CC1 c1(OCC)ccc(C(=O)NC(C)CCNC(c2cc(C3CCCC3)no2)=O)cc1 c1(CC)nn(C)c(CC(=O)NCC2(NC(=O)C(O)COC)CC2)c1Br C1(NC(C(C)(C)F)=O)CCN(Cc2ccc(C#N)cn2)CC1F c1(C(N2CCCC(C)(NC(C(C=CC)O)=O)C2)=O)cnc2cc(Cl)c(O)nc2c1 C(CC(=O)NC1CCN(C(c2cocn2)=O)CC1O)(C(N)=O)NC(C)=O N#Cc1cccc(C2CCN(C(=O)Oc3ccc(CNC)cc3)C2)n1.C1(N)CC1 C(CCCCCC(=O)N1CCc2sccc2C1)NC(C1(CC)CCCC1)=O N1(C(C2C(C)N(C)CC2)=O)CC2CN(C(=O)Cc3ccccc3Cl)CC2(C)C1 c1(C(N2CC(C)(C)C2C(=O)OC)C(=O)NCC=C)nc(C)n(C)n1 C#CCC(C(=O)Nc1cnc(SC)nc1)NC(C1CC1C#N)=O CCCC(CC)C(=O)NC1CCCCC1C(=O)NCc1c(C)cnn1C N1(C(Cn2c(C)ccn2)=O)CCN(C(=O)CC(C)F)C(CCO)C1 C1(CCNC(c2occ(C(F)(F)F)n2)=O)(NC(CC=C)=O)CCCC1 c1(OC)cc[n+]([O-])c(C(=O)NCC2CC(CNC(c3cc(Cl)c(C)cn3)=O)C2)c1 c1(C(=O)NC2C3CN(C(Cc4scc(CC)n4)=O)CC32)cnn2c1CCCC2C C1(CNC(c2cc(CC)n(C)n2)=O)CCC2CN(C(=O)C(O)CSC)CC12 C#Cc1cnn(C)c1C(=O)NCC(C1CCCCN1C(=O)C(COC)N(C)C)(C)C c1(CC(=O)N(C)CC2CCN(C(CC3C(COC)C3)=O)CC2)ccc(F)c(Cl)c1 c1(C(N2CC(OCCNC(C3(CO)CCO3)=O)C2)=O)ccc(C2CC2)o1 c1(OCC)c(C)cc(C(=O)NC2CC(NCc3ccccc3F)C2)cc1C C1(CC)CC(C(N2CC(O)(CNC(=O)COc3cncc(Cl)n3)C2)=O)C12CCC2 CCCC(C#N)C(=O)NCCN1CCC(NC(=O)CC2CC3C=CC2C3)CC1 CC1(C)CCCC1CCNC(=O)C=CCNC(=O)COCCCN(C)C N1(C(CN(CCCC(C)C)C2CCC2)=O)CCC(n2cc(CC(C)O)nn2)CC1 CC(C)CCC(C(=O)NCC(C)CC1CC1)NC(C12CCC(C1)C2(C)C)=O c1(C(N(C2CCCC2)CCCNC(COC(CC)(C)C)=O)=O)cc(Cl)c(Cl)n1C C=CC(C(F)(F)F)NC(=O)C(C1CCCN(C(=O)C(C)CC2CC2)C1)C C(=O)(CCS(=O)(=O)C1CCCC1)NCC1CC(OC)CN1C(C1CCCN1C)=O c1(C(=O)NCCC(C)N(c2ncnc(C(C)(C)C)n2)C)ccc(O)nc1 C(C(C(C)C(C)C)NC(c1cn(CC(F)(F)F)nn1)=O)NC(CCOC(C)C)=O C1(O)(C(C)NCC2CC3CCC2C3)CCN(C(=O)C(C)Oc2ccccc2)C1 C1(C(=O)NCC(C2CCC2)OCC)CCN(C(=O)C2CNC(=O)O2)O1 C(CCN=c1cc[nH]c(=NCCCCc2ncc[nH]2)[nH]1)c1cccc(C)n1 C1(NC(c2c(C)onc2)=O)CCN(C(=O)CC2CCC2)CC1c1ccccc1 C1(Nc2cc(CC)ncn2)(CNC(=O)CSC(=N)N)CC2CCC1CC2 C(=O)(C(C)(C)C1=CCSCC1)NC1CCN(C(CCC(CCC)CC)=O)CC1O N1(C(C2(F)CCCN(C)C2)=O)CC2CC1CCN2C(c1ncccc1Cl)=O C1(C)(COC)COCCN1C(C1CC(CCNn2cccn2)C1)=O N1(C(c2ccc(C)n2C)=O)CC2CCCC2(NC(=O)CC(C)CF)C1 c1(C(=O)NCC2(CC(N3CC(SC)(CO)C3)=O)CC2)cnc2ccncc2c1 C(=O)(C1c2c[nH]nc2CN1C(=O)C1=C(Cl)CCCC1)NC1CC(C)(C)C1 CC1(C)OCCOC1CC(N1CCCC1CCNC(C1CC12CCCCC2)=O)=O C1(C(N(C2CCCN(C(C(CC)CC)=O)C2)CCO)=O)CC(=O)NC(C)C1 c1(C(=O)NCCNC(C)=O)cc(CCNC(c2ccc[nH]2)=O)on1 c1(CN(C)C(=O)NCCS(=O)Cc2ccccc2)cccc(C(C)(C)C)c1 c1(C(N2CCC(n3cccc3)C2)=O)csc(-c2ccoc2)n1 C(CCC(C(=O)NC1COC1)N(CCOCc1ccccc1)C)OCC c1cc2c(nn1)CCC2.C(C(=O)N(CCOC1CCC1)C1CC1)N(C(=O)COC)C N1(C(C(C)NC(c2ccoc2)=O)=O)CC2CC2(CNC(=O)CC(C2CC2)C2CC2)C1 Nc1ccc(Cl)cc1C(=O)NC1COCC1CNC(C1CC1c1cncs1)=O C1(C(=O)NCCC(C)(C)NC(c2c(CCC)n(C)nn2)=O)C2CCC(F)(F)C12 c1(C(=O)NC2C(CC)N(C(=O)C(C)=C3CCCC3)CC2)[nH]c2ccccc2c1F c1(C(c2nnnn2Cc2ccccc2)NC(CC(=O)NC(C)C)C)nccn1C C(=O)(C(CCc1ccncc1)NC(=O)C(C#N)C=Cc1ccccc1)OCC C1(NC(C2CCN(CCO)C(=O)C2)=O)CC2(C1)CN(C(c1n[nH]cc1Br)=O)C2 Cn1nc2cc(Br)ccc2c1CN1CCCC(NS(=O)(=O)c2cccc(F)c2)C1 c1(NC(=O)NC(Cc2ccoc2)CO)csc2c1CCCC2 Cc1ccc2c(c1C)OCC2NC(c1cc(Br)c2c(c1)OCO2)=O Cc1cc(CCC(=O)NCCC2(NC(=O)C(C)CF)CCC2)cc(C)c1 C(=O)(CC(C(C)CC)NC(c1coc(C)c1)=O)NC(CCC=C)(C)C c1(C(F)(F)F)nocc1C(c1ccccc1)NCc1nnnn1C1COC1 c1(C(N2CCC(NC(CC(C)F)=O)C2)=O)ccc(N(CCO)CCCN)cc1.N(C)C C=CC(C)(C)C(=O)NCCCCC1CCCN(C(=O)CN2C(=O)CNC2=O)C1 O=C(C1COc2ccccc21)N1CCC(C2(NC(C3CC4(CSC4)C3)=O)CC2)C1 c1(C(=O)NCC(CC)N(C)C(C2CCCN2CC)=O)ccnc(S(N)(=O)=O)c1 c1(N(C(C=C)C)C)nnc(-c2ccco2)n1Cc1cc[nH]n1 CC1CC(N(C(=O)CCOCCN(C)C(C2(N(C)C)CCOCC2)=O)C)CCO1 C1(CCC)CN(C(=O)CN(CCO)C(N)=O)CCN1C(=O)COC(C)CC C1(CNC(c2cn(C(C)C)nn2)=O)CN(C(c2n[nH]cc2Cl)=O)CC12CCC2 n1(CC(=O)NC(C(C)C)CCN(C(=O)CC#N)C)cc2ccccc2n1 N1(C(C(C)NS(CC)(=O)=O)=O)CC2CC(CNC(C3OCCCO3)=O)C2C1 c1(C(=O)NCC2CN(C(C3CCC(C)(CC)O3)=O)C2)cc(N)c(C)c(N)c1 N1(C(C(C=C=C)C)=O)CCC(CNC(c2scc3c2CCCC3)=O)C(F)(F)CC1 C(=O)(C1=C(Cl)CCOC1)NC1(c2c(N)cc(F)cc2)CC1.N12CC3CC(C1C3)C2=O C1(CNC(c2cnc3ncccn23)=O)CCN(C(=O)C(O)C(F)(F)F)CC1(F)F CCN=C(NCCCc1ccccc1)NC1CCC(C(N2CCCC2)=O)C1 c1(CNC(c2ccc(C(=O)NC)nc2)=O)cc(O)cc([N+](=O)[O-])c1 C1(C(=O)NCCCNC(=O)OC)C(C)OCCN1C(C1CCC(C)C1)=O N1(C(CC=CCC)=O)CCN(C(=O)Cc2cc(OC)cc(C(F)(F)F)c2)C2CC12 Cc1ccc(CC(N2CCC(CCNC(=O)C(n3ccc(C)n3)C)CC2)=O)cc1 Clc1ccc(C2(Cc3nc(-c4cccc(Br)c4)no3)CCCCC2)cc1Cl c1(CC(=O)NC(c2cn(Cc3cccs3)nn2)CCC)cccc([N+](=O)[O-])c1 CCC(CC(=O)NCCC(F)Cn1cc(CCc2nc(=N)[nH][nH]2)nn1)C(F)F CC(N=c1cc[nH]cc1S(=O)(=O)NC1(C)CCCC(C)(C)C1)C12CCCC1C2 N1(Cc2ncn(C)c(=O)c2)CCC(NC(=O)CCC2NC(=O)NC2=O)C(C)(C)C1 C(=O)(C1=CCCCCC1)NCC1C(CC)CN(C(=O)CC2COCCN2C)CC1 Cc1ccccc1C(N1CC2C(CN(C)C(c3coc(C4CCC4)n3)=O)C2C1)=O C1(CC(=O)NC(C2CCCO2)CC)CCCC1NC(=O)C(C)n1ccnn1 C1(C(N2CCCC(C)C2)=O)N(C(=O)OCc2ccccc2)CCC1(C)C C(CC1CCC1)(C(=O)NOCCCC1CC1)NC(c1cccc(CC)n1)=O C(C(=O)NC1C=CC(C(N2CC(OC(F)F)C2)=O)C1)(C(C)C)SC C(=O)(C1CCCc2nnn(C)c21)NC1CN(C(c2c(CC)n[nH]c2)=O)CC(F)C1 C1(C(=O)NCCOCCCN(C(CSCCOC)=O)C)Cc2c(C)cccc2O1 Cc1c(Cl)ccnc1C(=O)NCC1(CN(C(=O)C(C2CCCCC2)F)C)CC1 N1(C(c2scc(C)c2C)=O)CCN(C(C2CC2F)=O)CC12CCC2 C(=O)(C1=Cc2ccccc2C1O)NCCN(C)C(c1cccc2nc(O)oc12)=O C=CC1(C(=O)NCCC(O)C(F)(F)F)CCN(C(=O)C(CCC)NC(C)=O)CC1 N1(C(NNC(=O)CCN(C(C(C(C)C)SCC)=O)C)=O)CCC2(C1)CN(C(C)=O)C2 Cc1nc(C(C)C)ncc1C(=O)NCC(O)CN(C(=O)C(Cl)=CCl)C c1(SCC)cccc(CC(=O)NCC2(NC(=O)CN3CCOC3=O)CCCCC2)c1 N1(C(C=C(C)C(F)F)=O)CC2C(CN(C(=O)CC(C)N(C)C)C)C2C1 C1(C(=O)NCC(C)(CO)NC(C=C(CCC)C)=O)CCN(C)S1(=O)=O C(CCCCF)NC(CCN(C(=O)Cn1cc(CO)nn1)C)=O N1(C(C(CCC)CCC)=O)CC2CCCCC2(NC(C2COC(=O)N2C)=O)C1 C1(NC(C(CO)N(C)C)=O)CN(C(c2cnc(C(N)=O)s2)=O)CCC1CO Cc1n[nH]c(=NC2CCCC3CN(C(c4c[nH]cc(Cl)c4=O)=O)CC23)o1 C1(CNC(C(C)OCCCC)=O)CCN(C(c2ccnnc2)=O)C12CC2 CCN=C(NCCc1ccco1)NCC1(C(F)(F)F)CCC1 CC1OC2(C(N3CCOC(CN(C)C(c4cccc(CO)c4)=O)C3)=O)CCC1C2 c1(C(N2CCCC(N(C(=O)COC(F)(F)F)CC)C2)=O)cn2ccn(C)c(=O)c2n1 N1(C(=O)N(C(C)C)Cc2cccc(N(C)CC)c2)C2C=CCC1CCC2 c1(C(N2CCC(C)C(NC(C3CCS(=O)(=O)C3)=O)C2)=O)c(N)nn2ccccc12 CN=c1ccc(C(N2CCCC2C(C)(C)C(N2CCSCC2C)=O)=O)c[nH]1 C1(NC(C2(C)CC3C=CC2C3)=O)CN(C(=O)Cc2ccsc2Cl)C2(CCCC2)C1 c1(NC)cncc(C(=O)NCc2cc(C(N3CCC(N(C)C)C3)=O)n(C)n2)c1 C1(O)(CNC(C=CC=CCCCCC)=O)CCN(C(=O)CC2CNC(=O)C2)C1 C1(NC(Cc2ccc(C)nc2)=O)CC2CN(C(=O)CC3CC4CCC3C4)CC12 C1(CN(C)C)CCN(C(=O)C=CC2CCCN2C(c2n[nH]c(=N)[nH]2)=O)CC1 N1(C(c2ccc(C)s2)=O)CCC(C2CC2)C1CNC(c1cc2cc(C)sc2[nH]1)=O C1(C(=O)OC(C)(C)C)(COC)CCS(=O)(=O)CC1.C12C3CN(CC13)C(=O)OC2 C(=O)(CS(=O)(=O)C1CC1)N1CCN(C(=O)C(F)C2CC2)CC1C1CC1 N1(C(C2NC(=O)OCC2)=O)CCC(C(F)(F)F)C(N)C1 C1(Cc2c(CC)non2)CCN(N2CC(CC=O)C2)CC1.C1(C=O)CCCN1CC C=C1CC(C)(C(=O)N(C)CC2CCCN2C(=O)C(C)N(C)C2CC2)C1 C1(O)(C(N2CC(C(=O)OCC)C(C3CC3)C2)=O)CC2(CCC(N)CC2)C1 c1(CN(C(C2(CC)CN(C(c3ccsc3C)=O)C2)=O)C)cccc(C)c1 c1(C(=O)NC(C)CN(C)C(C2CC2c2nccs2)=O)cnccc1N(C)C(C)C Cc1ccc(C)c(C(N2CCN(C(c3cn(CCBr)nn3)=O)C3CC23)=O)n1 N1(C(C=CC)=O)CCC(c2ccccc2)(NC(=O)C(CC)OCC)C1 C1(C(C#C)C)CCN(C(=O)C(C)(CO)NC(c2cnccn2)=O)CC1 c1(C(=O)NC(C2CN(C(CCOC(C)C)=O)C2)C)c(F)ccnc1Cl Cc1nn(C)c(C)c1C(=O)NC1CCCCC1C(N1CCCC(C(F)(F)F)C1)=O C(=O)(C(F)CCC(C)C)NC1CC(C(=O)NCc2ncc(CC)s2)OCC1 O=C1CC(C(=O)N2CC3(C2)CN(C(C2CC4CCC4C2)=O)C3)c2cccnc2N1 Cc1nc(N2CCC(NC(c3sccc3C(F)F)=O)C2)ccc1C#N Cc1ccc2c(CCC(N3CC(F)(CNC(C4CC4(C)CF)=O)C3)=O)c[nH]c2c1 CC(O)C(C)C(=O)N1CC(NC(=O)CN(c2ncccn2)C)C(C)C1 CC#CCC(C(=O)NC1CN(CC)CC1C)NC(C1CC2CC(=O)C1O2)=O C1(C(C)C)CC(CNC(=O)C(C)n2ccnc2)CN(C(C2(F)CCOCC2)=O)C1 C(=O)(CCC1=CCCCC1)NC(C(=O)NC1CC(C=C)C1)C1CCC1 C1(NC(C(CO)N(C)C)=O)COC2CN(C(=O)CC3CCSC3)CC12 C1(CNC(C2(SCC)CC2)=O)CCCCCN1C(=O)CCc1cn(C)cn1 N1(CC(COCC(C)C)O)CCC(C)(NC(c2cnc(Cl)c(Cl)c2)=O)CC1 C1(C(N(C2CC2)NC(C(=O)NC(C)C)=O)=O)CS(=O)(=O)CC12CC2.C1(C)(N)CC1 CC(N=c1[nH]c2cc(Cl)ccc2s1)C1CCCCN1C(=O)CC1CCC1 Cc1ccc(C(N2CC(NC(c3c[nH]c(=N)o3)=O)C3(CC3)C2)=O)c(C)c1 CC1=C(C(=O)NCC2CC3(CC(NC(c4cc[nH]c(=N)c4)=O)C3)C2)CCC1 CCC(F)(F)CC(=O)N1CC(O)(CN(C)C(C2CCCN2C(C)=O)=O)C1 CC1CCC(C(=O)C(C#N)C(=O)c2cccs2)C=CCC1 Cc1cnccc1-c1cn(CC2CCCC2NC(C2(n3cccn3)CC2)=O)nn1 N1(C(CC=CC)=O)CCN(C(c2ccnc(C3CCC3)c2)=O)C(C(F)F)C1 C1(O)(CNC(CSCCC)=O)CC(C)(C)C1.C12(C)CC(C1)NC2=O c1(C(=O)NC(CN(C(c2c(C)n(C)nc2C(F)F)=O)C)C)ccc2nn[nH]c2n1 c1(CC)ncc(C(N2CC(NC(C3(C4CCC4)CC3)=O)CC(C)C2)=O)c(O)n1 c1(C(N2C(C(N3CCOC(C(F)(F)F)C3)=O)CCCC2)=O)cc(O)c(Br)c(O)c1 CC1CN(C(c2ccncc2-c2ccccc2)=O)CC1NC(c1snc(Cl)c1Cl)=O Cc1nc(C=CC(N2CCCC2CNC(c2ccncc2)=O)=O)cs1 C(=O)(CC(C(F)F)n1ccnc1)N(CCCN(C(c1nn(CC)c(C)c1)=O)C)C c1(C(=O)NC(CCCCNC(CC2CC(=C)C2)=O)C)ccn2ncccc12 c1(NC(=O)CC2CN(Cc3ccc(Br)cc3O)C2)cc2cccc(Br)c2nc1Cl C1(C(C)(F)F)(C(=O)NC2(C)CN(C(C(C)NC(N)=O)=O)C2)CCOCC1 C=C(C)CCCC(=O)NCCOCCN(C(=O)C(C)(C1CCOCC1)OC)C Cc1cc2nccnc2cc1C(=O)NCCn1cnc(-c2ccccc2)n1 c1(C(=O)NCC2CCN(C(C3(C(=O)OC)C=CCC3)=O)C2)cccc2ncsc12 C(=O)(C(F)(F)CC(C)C)N1CC2C(NC(C(c3c(CC)cccc3)(F)F)=O)(C2)C1 N1(C(C2(C)CC=C(C)CC2)=O)CCC2(CC1)CCN(C(C1CC1C#N)=O)CC2 N1(C(c2sc(C)c(N)c2)=O)CCc2cc(C(=O)NCC3(O)CCNC3)ccc21 c1(C(=O)OC)n[nH]c(C(C)C)c1[N+](=O)[O-].C12OC3(C)CC1(C3)CNC2=O C(CCC(C(=O)NCCc1[nH]cnc1C)NC(c1ccsc1OC)=O)OC C1(NC(C(C)OC)=O)CCN(C(C2CCCC(F)(F)C2)=O)CC1F C1(NC(C2CCCC2)=O)COc2ccccc2O1.C1C(=O)NCC2CC2N1C c1(OC)ccc(C(=O)NC2CCC(CNC(=O)CCn3ccnc3)CC2)nc1Cl c1(CC)noc(C(=O)NC2CCC(CNC(=O)C=CC=C(C)C)C2)n1 C(=O)(CC1NC(=O)c2ccccc21)N1CCC(NC(CNS(NC)(=O)=O)=O)CC1 C1(NCn2ncc(P(C)(C)=O)c2)=CC=C2N=CC=C=C2N1.c12ccccc1S2 Nc1ccc(C(=O)NCC2CCCC(NC(=O)Cc3cn[nH]c3)C2)cc1O N1(C(c2ccc(OCC)cc2)=O)CC2CC(NC(=O)Cn3cccc3)C(C2)C1 c1(C(N2C(C(C)NC(=O)CC3CCC34CCC4)CCC2)=O)cnn2ncccc12 CC1C(=O)OCC1C(N1CCCC(Cc2cn(Cc3ccc(F)cc3)nn2)C1)=O N1(CC)CCC(NC(c2ncoc2CNC(=O)C(C)(O)C2CCC2)=O)C1 N1(C(C2CN(C(=O)C=CC(F)(F)F)CC2F)=O)CC(F)(F)CC1CO CCC(C)C(O)C(=O)NC1CCC(CC(N2CCCC(C(C)(C)O)C2)=O)CC1 CCC(C)(C)CC(=O)NCC(C)(F)CNC(=O)C=Cc1cncs1 CCC(C)C(C(=O)NC1CC(CCC(=O)NC2CCC(C(C)O)CC2)C1)N(C)C c1(OC)cc(C(=O)NCC2CCCC2NC(=O)C2=NOCC2)n(C)n1 C1(C(N2CCCC2CO)=O)CN(C(c2cnccc2-c2ccccc2)=O)CCO1 C(C)(C(C)(C)C(=O)N1CCCC(OC)C1C)NC(c1n(CC)nnc1)=O c1(C(N(C(CNC(C(C)(C2CC2)NC(C)=O)=O)C)C)=O)cc(Cl)nnc1O N1(C(c2ncc(C)[n+]([O-])c2)=O)CCC(C(N2CC(O)(c3cnn[nH]3)C2)=O)C12CCC2 C1N(C(C(n2cc(C(c3c(N)cccc3F)C3CC3)nn2)C)=O)CCCC12CCC2 Cn1nc(C(=O)NCCC2CCCN2C(=O)CC2(C)CC2(F)F)cc1C(F)(F)F c1(C(N2CCCC(N(C)C(c3ccsc3Cl)=O)C2)=O)ccc(Cl)c(F)c1O c1(C(N2CCC(CNC(c3ccc(O)nn3)=O)C2)=O)ccc[n+]([O-])c1 C1(C(N(C)Cc2onc(C)n2)=O)CN(C(c2[nH]ccc(=O)c2C)=O)CC1C1CC1 C(CO)(CCCNC(=O)CCCN(C)C)NC(C(c1ccn(C)n1)C)=O C=CC(C)(C)CC(=O)N1CCC(NC(C2(c3ccno3)CCOCC2)=O)CC1C N#Cc1ccc(C(=O)NC2CCCCC2NCC2CCOCC2)nc1 C(=O)(CC(C)(C)CC(=O)OC)NC(CC)CNC(C1CC2CCC1O2)=O c1(C(N2CCC(CCNC(C(C)NC(=O)C3CC3)=O)C2)=O)cccc(C(C)C)c1N Cc1nc2cccc(C(=O)N(CC(C)NC(=O)C=Cc3cncnc3O)C)c2s1 n1(CC(C)OC)cc(CC(O)C2CC2)nn1.C12(CN3C(=O)C3CO)CCC(C1)C2 C1(C(N2CC(=C(CNC(c3cc(C4CCC4)no3)=O)F)C2)=O)C(F)(F)C12CC2 C1(OCCC)CCCN(C(C2CN(C(=O)C(C(C)C)N(C)C)CC2C)=O)C1 Cc1c(C=CC(N2CC(NC(=O)COC3CC3)C(CC(C)(C)C)C2)=O)cnn1C C1(C(=O)NCCCNC(C(C)N2CCCC2)=O)CCN(C(=O)CS(C)(=O)=O)C1(C)C c1(C(=O)NCC2C3CN(c4c(C#N)cncc4)CC32)cc2c(nc1O)CCOC2 CCC(C)CCC(=O)N1CC(OC)CC1CNC(=O)CC1(C#N)CC1 N1(C(c2cnc(O)nc2)=O)CCc2ccc(-c3ccc4c(O)n[nH]c4c3)cc2C1 C#CC1CC2(CC2)CN1C(C1(CN(C(=O)CCCOC)C)CC1)=O C(CCF)(C(=O)NCCCNC(=O)OC)NC(C(CC)=CCCC)=O N1(C(CCc2cccc(NC)c2)=O)CC2(C1)CN(S(=O)(=O)c1cccs1)C2 C1(C2CC2)(CNC(C(C=C)C)=O)CCN(C(c2cc(CC)nnc2C)=O)C1 C(=O)(C(C(C)C)C(C)C)NCC1C(NC(CCCCN(C(C)=O)C)=O)CCC1 CC(C(=O)N1CCC(CNC(=O)C(F)CC2CCOC2)CC1C1CC1)P(C)(C)=O C1(NC(CC(C=C)C)=O)CN(C(C2CCC(=O)N2C)=O)C2CCCCC12 C1(C(=O)NCCC2(O)CN(C(=O)C3=CCCCC3)C2)CC2CCCC2C1 N1(C(c2cnc(OC)nc2C)=O)CC(NC(=O)Cc2cncs2)C(C2CC2)C1 c1(CC)cc(C(N2CCN(C(C3CC4CC4C3)=O)C(C3CC3)C2)=O)cc(O)n1 c1(C(=O)NCCNC(c2sc(Br)cc2F)=O)cc2c(cn1)COCC2 C1(NC(C2(C(C)C)COC2)=O)CCCN(C(C2C=NN(C)C2=O)=O)CC1 C1(C(N2C(CN(C(CNC(CC)=O)=O)C)CCC2)=O)CCCN1N=O c1(CCC)noc2ncc(C(N3CCN(C(C)=O)C(CF)C3)=O)cc12 C1(C(N2CCC3(CCC3)C2)=O)CCN(C(=O)C2CC2c2ccccn2)O1 C1(C(N2CCC(N(C)CC)C2)=O)CC(NC(C2CCCC2F)=O)C(O)C1 c1(OC)cccc(C(N2CC3CC2C3C(=O)Nc2cnc(Cl)nc2)=O)c1OC c1(C(N(CCC(C)NC(c2cn(CCC)nc2)=O)C)=O)sc2ccsc2c1C CC(C)(CN=c1[nH]nc(C#N)s1)NC(c1csc(Cl)c1)=O N1(C(C2(C)CC(F)C2)=O)CCCCC(C(N2CCC(OCC(N)=O)C2)=O)C1 N(C(=NCC(O)c1ccn(C)c1)N1CCC(O)(OC)C1)C(CC)CC C(=O)(CC(C)(O)C(F)(F)F)N1CC(C)(CNC(c2c(CC)ocn2)=O)OCC1 C1(NC(C(N2C(CC(C)(C)C)CCC2)=O)=O)CCC(c2ccccc2)CC1 C1(CNC(C(C)OCCOC)=O)CCC(C(C)C)CC1.c1(OCC(=O)N)cn(C)nn1 C1(C(=O)OCC)CC(O)CN(C(C2(NC(=O)Cn3nccn3)CC2C)=O)C1 c1(OC(C)(C)C)ccnc(CNCC23CC(CCO2)C3)c1 c1(C(=O)Nc2ccc(C3CC3)nc2)ccc2c(c1)CNCCN2 C1(CC)CCCCC1C(=O)N(C)CC=CC(=O)NC1CCN(C2CC2)C1=O C(=O)(CCC(F)(F)C(F)F)N1CCCC(O)(CNC(CC(CCC)O)=O)CC1 C(CC(C)C(=O)NC(CNC(C1(c2ccn(C)n2)CC1)=O)CC)=CC N1(C(C2C(C=C)C2)=O)CC(O)(C2CCN(C(c3c(F)cc(O)cc3F)=O)CC2)C1 c1(CCN(C(=O)CCOCCCOC(C)=O)CCC)ncccc1O C1(C(N2CCN(CCNC(c3c(CC)cno3)=O)CC2)=O)CC2COCC(C1)C2 CC1CCN(C(C2(CCF)CCOCC2)=O)C1CNC(=O)Cc1ccsc1Cl c1(OC)ccc(S(=O)(=O)N2CCC3(CC2)CC3(C)C(=O)O)c([N+](=O)[O-])c1.N1CCC1 C=CC(C)CC(=O)N1CC(N(C)C)C(CNC(C2(C(C)(F)F)CC2)=O)C1 N1(C(=O)CC2CCCCO2)CC2CCC1CN2C(c1ccnn1C1CCC1)=O CC(C(=O)NC1CC(O)CN(C(=O)Cc2n[nH]cc2Br)C1)S(N)(=O)=O c1(OC)ccc(Cl)cc1Cn1cc(C(c2ccccc2F)Cc2cccnc2)nn1 S(=O)(=O)(c1ccccc1C#N)NC(c1nc(Br)cs1)C C1(C(=O)OC)CCN(C(C2CCC(CNC(=O)C(O)CN(C)C)C2)=O)C1C N#Cc1cnn2cc(C(=O)NC3CCCN(C(c4ccccn4)=O)C3)cnc12 C1(C)(CC)CCC(NC(c2cc(CNC(C3CCCOC3)=O)ccn2)=O)CC1 c1(C(=O)NC2CN(C(C34OC(C)(C)C(C3)C4)=O)CC(F)C2)cnn2ncccc12 N1(C(C(CC)O)=O)CCOC2(C1)CN(S(=O)(=O)c1sccc1OC(F)(F)F)C2 CC(C)CC(CNC(c1ccn(CCNC(C23CC(F)(C2)C3)=O)c1)=O)CO C(=O)(CCCCC(C)=O)N1CC(C)(C(NOC)=O)C1.O1NC1=O C1(NC(CC(C=C)CC)=O)CN(C(=O)CCSC)CCC12CCOCC2 CC(O)(CC(=O)NCc1cccc(CNC(=O)C(c2ccccc2)O)c1)C1CC1 c1(NC(C)CN2CCCCC2)ccnc2ccc(C(=O)NC(C)(C)C)cc12 c1(C(N2CC=CC(NC(C(c3n(C)ncc3)(F)F)=O)C2)=O)c(O)cc(O)cc1O C=CCC(CNC(=O)CC1(C)CCN1C(=O)CC1CCCN1CC)CC(C)C CC(C)C(F)(CNC(C1C=CCS1)=O)C(=O)N1CC(C)(O)C1 C1(CNC(COC(C)C)=O)C2CN(C(=O)C(c3ccc(F)cc3)F)CC12 c1(C(=O)NCC2(NC(c3ccc(OC)nn3)=O)CCOC2)cc(F)c(F)c(F)c1 CC1(C)CN(C(=O)CC2CCOC2)CC(CNC(=O)C(F)=CC2CC2)O1 c1(OCCC(=O)N(C)CC2CCCN(C(C(CC#C)C)=O)C2)ccc(F)cc1Cl C(=O)(C1OCCc2ccccc21)N1CCCCC(NC(c2ccco2)=O)C1 C1(O)(CCNC(C=CCN(C)CC)=O)CCCN(C(=O)C(C)C2(O)CCC2)C1 C1(NC(CCC(=O)NC)=O)CCC(C)N(C(c2ccc(NC=O)cc2)=O)C1 C=CCCCCCCC(=O)NCc1ccnc(C(=O)N(CCCCO)C2CC2)c1 CC1(C)CC(CC(=O)NC2CCCN(C(=O)CCOC3COC3)C2)CCO1 C(C(C)(C)C(=O)NCC1(CNC(=O)C(C2CCOCC2)C)CC12CCC2)N(C)C CCC(C)CCC(=O)N(CCCN(C)C(C1(n2cc(C#N)cn2)CC1)=O)C N1(C(CC(=O)OC)=O)CCC(c2nc(NC(=O)C=C(C)Cl)cs2)CC1 N1(C(C(C)=C(CC)C)=O)CCC2(CCCC2C(N2CCC(C)(C)C2)=O)C1 C1(NC(c2c(OCC)ccs2)=O)CC2CC(C1)N(C(=O)CC1C(C)(C)C1(C)C)C2 C1(Cc2cn(CC(=O)NCCCS(C)=O)nn2)CCC(C)(C)CC1 c1(C(N(C2CCCCC2NC(=O)Cn2cc(Br)cn2)C)=O)cnn(C)c1F N1(C(CC)=O)CCCC1C(=O)NC1CC(N(C(=O)C(C)C2CCOC2)C)C1 N1(CC(C)C)C(=S)NC(c2ccc3nc(O)oc3c2)C2=C1CC(C)(C)NC2=O C(=O)(C(C(C)NC(C1CC2C=CC1O2)=O)C(C)C)NCc1c(C)nn[nH]1 C1(C)(Cn2cc(-c3c(CC)cccc3)nn2)Cc2ccccc2N1 C(=O)(CS(=O)(=O)C1CC1)N1CC(CNC(c2ccc(C)nc2N)=O)CC1(C)C C1(C)(CNC(c2cc(OC)ncc2)=O)CCCN(C(C2CC=CCC2)=O)C1 N1(Cc2cccc(-c3ccnc(C)c3O)c2)CCOC2COCC2C1 N1(C(c2ccc(C)n2C)=O)CCC(NC(=O)CC2CCOC2)C(F)(F)CC1 N1(C(C(C)(C)OC)=O)CC2CCCC(CNc3nccc(C)n3)C2C1 N1(C(C2(C)CCSCC2)=O)CCCC(CO)(NC(=O)C=Cc2ccncc2)C1 C(=O)(CCCCCSC)NCC(CNC(C(C)(C)OCC)=O)(C)OC CC(C)CC(C(=O)N1CC(n2cc(-c3nn(C)cc3Br)nn2)C1)C1CCCN1 C1(NC(COC(CC)C)=O)CCCCN(CC(=O)Nc2ccccc2)C1 N1(C(C2C(C(C)(C)O)C2)=O)CC(O)(CCNC(c2csc(-c3cnc[nH]3)n2)=O)C1 Cc1c(C(N2CC(NC(c3ccc(CC(C)C)s3)=O)C(O)C2)=O)ccn1C1CC1 Cc1nn(C)c(C)c1CCNC(=O)C(N1CCN(C(=O)OC(C)(C)C)CC1)(F)F N1(C(c2n(C(C)C)ncc2)=O)C2CCC1CN(C(C1CCO1)=O)CC2 C(=O)(C(CCC)NC(=O)C(COC)COC)NC(C#C)CC C12(C(=O)NCCCC(=O)OC)CCC(NC(c3cc(I)ccc3Br)=O)(CC1)CC2 Cc1cc(=NC(=O)C(=O)NC(CO)CC(c2ccccc2)C2CC2)[nH]n1C(C)(C)C C(C(C)(C(=O)N1CC2C(CC(=O)NCC3CC(N(C)C)C3)C2C1)OC)OC c1(C(N(CCCNC(C2C3CCC(=O)C23)=O)CC)=O)cccc2c1CCCC2=O Cc1cccc2c1CCC2NC(=O)Cc1ccc(OC(F)F)cc1Cl c1(C(C)C)c[nH]nc1C(=O)N(C(CCN1CCCC1)C)C.c1(C(=O)N)ccncn1 N1(C(c2cc(C3(C)CC3)on2)=O)CCC(NC(=O)C(C)(CO)N(C)C)C(O)C1 C12CCN(CC1)CC1CC(C1)C(=O)N(C)C1CCN(C1)C2=O.c1(CO)ccccc1 c12sccc1CNC2=O.C1(C(=O)NC)(NC(=O)CNC(=O)C2CC2)CC1 C1(C)(CC(=O)NC(C(C)C)CNC(C2CCOC2)=O)CC(F)(F)C1 Cc1cc(NCc2ncoc2C(F)F)nc(N(CC(C)(C)CO)C)n1 C(CCC(=O)NC1CCCC1CNC(c1cc(C(C)=O)c[nH]1)=O)=CC c1(C(=O)NC(CN(C(=O)CSc2ncccn2)C)(C)C)cccc([N+](=O)[O-])c1Cl C1(CNC(=O)C(F)n2ccnc2)C2CC1N(C(c1cccc(C(F)(F)F)c1)=O)C2 c1(NC2CCN(C(=O)CCN3CCOC3=O)C2)c(C)cncc1[N+](=O)[O-] c1(C(=O)NC2CCN(C(C3=NOC(C)C3)=O)C(C)C2)cc(Cl)cc(Cl)c1Cl c1(C(CC)C)nccc(N2CC(C)(NC(=O)Cc3ccnn3C)C2)n1 c1(N2CCCC(CCNC(c3cn4ccnc4s3)=O)CC2)nc2ccccc2s1 Cc1cc(-c2nc(C3CCCO3)nn2-c2ccc(C)c(Cl)c2)n2nc(C)cc2n1 c1(C(N2CCC(N(C(=O)Cc3cc(C)ns3)CCC)C2)=O)ccn2c1CSCC2 N1(C(CC(CCC)C)=O)CCC2(NC(=O)C(C)C)CCCC12 C1(C)(C(=O)NC(C2CCN(C(c3ccc(CC)s3)=O)C2)C)CCCOC1 N1(C(c2cc(Cl)cc(C)c2N)=O)CCN(C(c2nccs2)=O)CC(C)(C)C1 C1(C(=O)OCC)CCCN1C(=O)COCc1cn(C(c2ccccn2)C)nn1 c1(C(=O)NC(C(C)NC(CNC(CC)=O)=O)C)cnc(C)cc1C Nc1cccc(-c2cn(CCNc3cccc(CN4CCCC4)c3)nn2)c1 CCCCCCCCCC(=O)N1CCCC(N(C(=O)C(=O)C(C)(C)C)C2CC2)C1 C1(NC(c2cnc(Cl)s2)=O)CC2CC1N(C(c1ccc(-c3ccco3)s1)=O)C2 C1(CC)CCC(C(=O)NCC(CNC(=O)C(C)(C)c2cc[nH]n2)OC)CC1 C1(CC)CN(C(C2(C)CCCN(C(c3cnnn3CC)=O)C2)=O)CCCO1 c1(C(=O)NC(CNC(C(c2cccs2)SC)=O)CO)nc(Cl)cc(N)c1Cl O=C(C1=NOC2(CCN(C(c3cc(F)cc(Cl)c3)=O)C2)C1)Nc1cccs1 N#Cc1cc(S(=O)(=O)NC2CCn3cncc3C2)ccc1N1CC2CCCC2C1 Cc1[nH]c(=N)nc(O)c1CCC(N1CC(CNC(C23CC(F)(C2)C3)=O)C2CC12)=O C1(CNC(CC=CC)=O)CCN(C(c2ccc(C(C)C)nc2)=O)CC1O c1(CN(C(CNc2cccc(C(=O)NC)c2)=O)C)ccc(C)cc1OCC(C)C c1(C(=O)NC2C(C=C)CN(C(C3(C)CCCCO3)=O)C2)nccn2cc(C)nc12 C1(C(=O)NC(CCC)C2CCCC2)CCN(C(=O)C(C)CC#N)C(C)(C)C1 CCCC(CC)C(=O)N1CC(NC(C2(CC3CC3)CC2)=O)C1 C#CCC(C)(C(=O)NCc1ccc(O)nc1)NC(=O)C(C(C)C)N1CCCC1 c1(N2CC(C(=O)NC)C(CC3CC3)C2)ncnc(N(CC)CC)c1N c1(C(N2CC3C(CNC(=O)C(C4(O)CCCCC4)F)C3C2)=O)cccc(F)c1F c1(C(N2C(CNC(C(C(C)C)O)=O)C=CC2)=O)cncc2cc(Cl)ccc12 c1(CNCCC)cc(C)nn1C.C1CCCN1C(=O)COCC1CCCOC1 c1(CC)cccc(N(C2CCC2)CCOC)c1 C1(NC(C(Cc2ccccc2)OC)=O)CC(NC(c2snnc2C2CC2)=O)C(O)C1 N1(C(C(n2c(C)ccn2)C)=O)CCOC(CN(C)C(C2(F)CC=CCC2)=O)C1 C1(CNC(=O)NCC2CCC(C)(C)O2)CCCC(F)(F)C(=O)N1 c1(C(=O)NC(c2c(O)cc(C)c(Cl)c2)C)cc(F)c(F)c(Br)c1F c1(-c2cn(CC3N(C(C(C4CCOCC4)OC)=O)CC3)nn2)cncc(C)n1 c1(C(=O)NCCOCCCNC(C(C)c2cccs2)=O)ccc2c(n1)OCCO2 c1(OC2CC(=O)N2)ccc(CSc2ccc(OCCCO)cc2)cc1 N1(C(C2(CC)CC2)=O)CCCC(CN(C)C(C2CC(=O)N(c3cnn(C)c3)C2)=O)C1 c1(CC2(CC(=O)NCCl)COC2)ccc(CC(=O)N2CCC2)[nH]1.C1(O)CCOCC1 N1(C(C(CO)OC)=O)C2CCC(C(=O)NCC(C)(C)C(F)F)C1CC2 C1(CC(=O)NCCN(C)C(C2CC(O)(c3ccccc3)C2)=O)COCC(C)O1 N1(C(C(CC#C)O)=O)CCCN(C(c2coc3c2CCCC3)=O)CC1C C(=O)(C(CC(C)C)NC(=O)C=Cc1ccco1)NC(c1ccc(C)cc1)C CC1(CNC(=O)C=CBr)CN(C(c2ncc(F)cc2N)=O)CCO1 Cc1cc(=NC(CCO)C2CC2)[nH]c(C)n1 CCC(C)C(=O)N(C)CC1CCCN1C(=O)CSc1nnnn1C c1(N2CC(CC=C)(NC(C3CCCCC3O)=O)C2)nc2c(cc1C#N)CCC2 CC1(C)CN(N2CCC2C(O)CO)CC1C1CC1 C=C(C)C1CN(C(C2CC3(CCN(C(c4nnn(CC)c4C)=O)C3)C2)=O)CCO1 C1(C)(C(N2CC(COC)C2)=O)CN(C(C2(SC)CCC2)=O)C1 N1(C(C(C)NCC#C)=O)CC2(CC2)CC1CC(N1CCCC(C(C)C#C)C1)=O Cc1ccc(C)c(NC(C2(NC(c3cc(C)c(C)[nH]3)=O)CC(CO)C2)=O)c1 C(=O)(NNc1cc(C)nc(F)c1)N1CCC2(CCC(C(=O)OC)C2)C1 C1(N(C)C)CCN(C(=O)C(C2CC2)NC(=O)CCCc2cnn[nH]2)C1 N1(C(C(=C(C)C2CC2)F)=O)CCCCC1CCNC(C1CC(C)CCO1)=O C12(CNC(c3ccc(Cl)cc3)=O)CCC(CC1)N2C(=O)C(=O)NCC1CC1 C=C(C)CCC(=O)NCCC1CCCN(C(=O)C(O)C(C)C)C1 C1(C(=O)NC2CC(CCNC(C(CN(C)C)N(C)C)=O)C2)CCc2nn[nH]c2C1 N1(C(C(C2CC(F)(F)C2)OC)=O)CCCN(C(c2c(C)noc2C(F)F)=O)CC1C Cc1cn(CC(N2CCC2(C)C(N2CCOC3CC23)=O)=O)c(=O)nc1O Cc1nc(C(=O)N(C2C3CN(C(c4cc(C)c(Br)s4)=O)CC23)C)c(C)o1 C(=O)(CS(=O)c1ccc(Cl)cc1)N1CC(CNC(C(CC)CC)=O)C(O)C1 CN1C(=O)Cc2cc(S(=O)(=O)N3CCCC3NC(c3cncs3)=O)ccc21 CCC(C)(C)CCCC(=O)NC(CO)C(=O)NC1CC2C=CC1C2 c1(C(N2CC(C(F)(F)F)CC(C(N(C)C)=O)C2)=O)cccc2c1CNC2=O c1(NC)nc(C)ccc1C(=O)NC(C)CN(C(=O)CC1CCCN(C(C)C)C1)C C1(C(N(C(CC(=O)OC)C)C)=O)CCN(C(C23CCC(C2)C3)=O)C12CC2 c1(C(N(CCCNC(COCP(C)(C)=O)=O)CCO)=O)cncc2[nH]ccc12 N1(C(=O)CCOC2CC(=O)N(C3CC3)C2)CC2CCCC2(C(=O)NC2CC2)C1 c1(C(N(C)CC2CN(C(C3CCCN3C)=O)CC2O)=O)[nH]nc2c1COC2(C)C C1(C(=O)Nc2cc(C)nn2C(C)C)C2CC(CC2F)N1C(=O)C(Cl)Cl C1(C(=O)NCCCC2(NC(c3cn(C)nc3)=O)CC2)CCC(C)(C)OC1 N1(C(c2c(CC)ncs2)=O)CC2N(C(=O)Cc3ccoc3)CCC2(C)C1 Cc1cccc(C(N2CCC(NC(=O)CC3CC(C(F)F)C3)C(O)C2)=O)c1Cl c1(SCC(N2CCCC(NCC3CC4CC4C3)C2)=O)ccc(F)cc1 C(CC)(CC)(CCNC(c1coc(SC)c1)=O)NC(C(C=C)(C)O)=O N1(CC(=O)N(C(C)C(C)C)CC)CCC2(COCC(CO)O2)C1 Cc1cc2c(C(=O)NC(C)C(C(C)C)NC(=O)C=CC(F)(F)F)cccc2[nH]1 c1(C(N(C2CCN(C(c3csc(C(=O)OC)n3)=O)C2)CC#C)=O)coc(C2CC2)n1 N1(C(CN(C)Cc2cc(C(F)(F)F)cs2)=O)Cc2ccccc2S1(=O)=O N1(C(CCSCCCC)=O)C2CCCC1CC(NC(C1CCC3CC3C1)=O)C2 S(=O)(=O)(c1c(CC)cccc1C)NC(C(CC=C)(C)C)=O c1(C(=O)NC2C3CN(C(C4(C(C)C)COC4)=O)C(C3)C2)ccc2c[nH]nc2c1 C(=O)(CCCC(=O)OC(C)(C)C)N1CC(CNC(CC(C)N(C)C)=O)C1 c1(CC2(N3CC(NC(C(c4cccs4)NC(=O)NC)=O)C3)CC2)ccccn1 C1(O)(C(=O)NCCN(CCOC)C(c2cc(C)co2)=O)CCOC1 c1(OC)cc(Br)cc(CC(N2CCC3(CCC3NC(=O)NC3CC3)C2)=O)c1OC c1(OCCN(CC(C)NC(C(=Cc2cccs2)C)=O)C)ccccc1F c1(C(N(C2CCN(C(C3CCC3)=O)CC2)CCC)=O)nnn2c1CCCC2 c1(C(=O)NCC2CCCN(C(c3nc(F)ccc3Br)=O)C2)cc(Cl)cc(Cl)c1O C1(OC(C)(C)C)CC12CC(C)C2.S(=O)(=O)(CC1CCC1NC(=O)CN)CNC(C)C N1(C(c2c(C)ncc(Br)c2)=O)CCCN(C(=O)C(C)C#N)C(C)C1 CC(F)(F)CCC(=O)N1CCSCC1CCNC(=O)CCCc1ccncc1 c1(OC)ccc(Cl)cc1CN1CCCOC(CNC(c2ccc(Cl)nc2O)=O)C1 C1(NC(C2CCS2(=O)=O)=O)CCCC12CN(c1cc(Cl)nc(C(F)(F)F)n1)C2 c1(C(=O)OC)cc([N+](=O)[O-])cc(C(=O)NCC(O)C(F)F)c1C Cc1cc([N+](=O)[O-])cnc1NCCC1CSCCN1C(c1cncn(C)c1=O)=O C1(NC(=O)CSC2CC=CC2)CCCC(NC(c2nc(-c3ccoc3)no2)=O)C1 CCCC(CC)C(=O)NCC(C)(CC(C)C)NC(c1ccc(C2CC2)c(F)c1)=O c1(C(=O)NC(CC=C)CNC(c2sccc2CC)=O)ccnc(-n2cccn2)c1 c1(C(C(=O)NCC(CN(C(C=CC)=O)C)O)C)ccc(C(C)C)cc1 c1(C(=O)NCCOCCCNC(C(c2ccccc2)OCC)=O)ncncc1Cl c1(OC)cc(NC(=O)NCCOc2c(Cl)cccc2Cl)ccc1Br N1(C(COCC)=O)CCOCC1NC(c1cnn(C2CC2)c1C)C C1(C(=O)NC(c2ncc(C)o2)C)CCC2(CC2)N1C(c1cncc(O)c1)=O C(c1c(F)cccc1F)=CC(=O)NCCCCCCN(C(=O)CC1CCOC1)C N1(C(C2CN(C)CC(C)O2)=O)C2CC=C(C(=O)N3CCCC(CF)C3)C1CC2 CC1CON(C(=O)c2cc(-c3cccc(C(F)(F)F)c3)cs2)C1 C1(CNC(=O)C(C)N(C(=O)C(C)(C)OC(C)=O)CC)(CC)CCCO1 Cc1ccc(C(C)(C)C(=O)NCC2(NC(C3CCC4CCC34)=O)CC2)cc1 C12(C(=O)NCCOCC(=O)NC)CCC(NC(=O)C(C)S(N)(=O)=O)(CC1)C2 Cn1c(C(=O)NC(CNC(C2CCCC(O)C2)=O)CO)cc2sccc12 c1(C(=O)NCC(CO)NC(C(=O)NCCOC)=O)cnc(O)n1C N1(C(C=CC=CC)=O)CC2(CNC(c3oc(CC)nc3C)=O)CCC1C2 N1(C(C(C)c2ccco2)=O)CCCC12CCN(C(=O)COCc1ccncc1)C2 CC(N=c1[nH]c2ccc(O)cc2s1)c1ccc(N2CCCC(C)C2)cc1 C#CCC(CC(=O)Nc1cc(CO)cc(F)c1)NC(c1ncoc1CC)=O C(=O)(CCCC(C)(C)C)NC1CCN(C(c2ccc(CC)c(C)c2)=O)C(C)C1 C(=O)(C(CNC(=O)Cc1cc(C)on1)CC1CCCC1)NCC(CC)C c1(C(N(CCNC(=O)CC2CCCC2(F)F)CC)=O)cc(C)nnc1O C(CC(=O)N1CCC(CO)(OC)C1)(C(C)(C)C)NC(CCCCOC)=O C=CCC(C(=O)NOC(CC(C)C)C(=O)NCc1ncccc1F)OC c1(C(=O)NC2(COC)CN(C(C34CCCC3C4(F)F)=O)C2)ccc(C)c(Cl)c1 Nc1cc(Cl)nc(C(N2CCS(=O)(=O)C(CCNC(C3CC3F)=O)C2)=O)c1Cl CCCCC(O)C(=O)NC1CN(C(c2cccc(C3CC3)n2)=O)CC1C CC(CCNC(=O)CC1CCCOC1)CCNC(c1cc(=O)n(C)o1)=O c1(C(N2C(C)(C(=O)NCc3cnccn3)CCC2)=O)ccc2c(Br)cccc2n1 c1(Cn2cc(N3C(=O)CCC3)nn2)c(F)ccnc1F Cc1nn(C)c(C)c1CC(=O)NCC1(C)CN(C(=O)CC2COCC2O)CC1C Cc1nc(C)c(C(N2CC(N(C(=O)CCNC(=O)OC(C)(C)C)CCO)C2)=O)[nH]1 C(=O)(N=c1[nH]nc(-c2ccc(C)o2)s1)N(CC1CC(=C)C1)C(C)C N1(C(COCC(=O)NC)=O)CCC(O)(C(C)NC(c2sc(C)cc2Cl)=O)CC1 c1(C(N2C(CNC(CCC(=O)N(C)C)=O)CC2)=O)cc2c(F)cc(F)cc2[nH]1 C1(CNC(CN(C)C(c2cccs2)=O)=O)CCC(NC(=O)CC2(C)OCCO2)C1 c1(C(N2CCC(NC(C(C#C)(C)C)=O)C(C)(C)C2)=O)cccc([N+](=O)[O-])c1NC N1(C(C2CCN(OC)CC2)=O)CCN(C(c2sc(N(C)C)nc2C)=O)CC(C)C1 C1(CN(CC)CC)CCCN(C(=O)C=Cc2sccc2C)C1 CCCC(C)(O)CC(=O)N1CCC(C(=O)NC2CN(C(=O)C3CC3)C2)C(O)C1 Cc1cccc([N+](=O)[O-])c1OCC(=O)N(C(C)CNC(=O)CC1CC2(CC2)C1)C c1(OC)nc(N2CC3CCC(C2)N3c2ccnc(Br)n2)ncc1F C1(CCC(=O)NCC(c2ccccc2)NC(=O)CC2CCOC2)CCCC(=O)N1 c12cc(ccn1)N(CC)C2.C(CCCCNC(c1ccc(C)o1)=O)NC(C#CC)=O c1(C(=O)NC2CCC2NC(=O)C(O)Cc2ccc(F)cc2)cccc2ncccc12 c1(C(N2CC(COC)N(C(=O)C(C)N3CCC3)CC2)=O)c(C)cc(C)nc1S C(CC(C)(C)N=c1[nH]nc(C)o1)NC(C1C(C(=O)OC)C1)=O C1(C)(CNC(C(CC)n2cncn2)=O)CCN(C(=O)CC2CC(N(C)C)C2)C1 CN1CC(C(=O)NCC2CCCC(NC(c3cc(F)c[nH]3)=O)C2)CCC1=O C1(CN(C(c2c(C(C)C)c[nH]n2)=O)C)CCCN(C(=O)C(C)(C)CC2CC2)C1 C(=O)(CCCCCNC(=O)CC12CCCC1C2)NCC(C)(C)N(C)C C#Cc1ccc(C(=O)NCC2CC(F)(CNC(=O)CCc3ccon3)C2)cc1 c1(CC(=O)NCC(C)NC(CC2C(C)CCC2)=O)cccc(F)c1F C1(NC(c2n(CC=C)ccn2)=O)COC2(CCN(C(=O)CCNC(=O)NC)C2)C1 c1(C(N2CCN(C(c3cnn(C)c3Cl)=O)C3C2C3)=O)cc(Cl)c2ccccc2n1 c1(C(=O)NC(CNC(C2(C(F)(F)F)CC(C)(C)C2)=O)(C)C)cc(NC)ccc1O C1(C(CNC(c2c(C)ocn2)=O)F)CCN(C(c2c[nH]ccc2=O)=O)CC1 Cc1cc(CNC(c2c[nH]nc2C(=O)OC(C)(C)C)C)c2c(c1)CCC2 N1(C(C)C)CC(C(N2CCC(NC(c3cnnn3C)=O)CC2)=O)CCC1=O Cc1nsc(C)c1C(=O)NCC1CCN1C(=O)CC1CSCCS1 C1(C(=O)NC(CC)CC(=O)NC2CC3CCC2O3)CCC2(CC2)CO1 C=CCC(F)(F)C(=O)N1CC=CC(C(=O)NC(CC)C(=O)OCC)C1 N1(C(c2ccc(C(=O)OC)cc2)=O)CCCOC(CNC(=O)Cc2cnoc2)C1 c1(CNC(C2(N(C)C)CCN(C(c3csc(C)c3C)=O)C2)=O)nnc2n1CCC2 C(=O)(C(F)C(C)(F)F)NCCN(C(C)C)C(C1CC12CCSCC2)=O N1(C(CCCCSC)=O)CCC2(CC1)CCN(C(c1cn3cc(C)sc3n1)=O)C2 [N-]=[N+]=NCCCC(=O)N1CCCC1CCC(N1CC(O)CC(O)C1)=O c1(C(C(=O)NC)NC(=O)CC2CNCC2O)ccccc1Cl C1(C(=O)NCC(C2CCC2)NC(c2cncc(C)n2)=O)CCC(F)(F)CC1 N1(C(Cc2ccc(C)cc2)=O)CC2CC1CN2C(C1CCC(OC(F)F)CC1)=O C1(C(=O)Nc2c(OCC)scc2)CCN(C(=O)CC2(C)CCCO2)CC1C C1(CC(=O)NC2C(NC(C=NOC)=O)COC2)CC(C)(C)CCO1 Cc1cc(C(=O)NCC2(NC(C3CC(C)CC(C)C3)=O)CCCC2)cc(C)c1Cl C(CCCN=c1[nH]c2ccc(C(N(CC)Cc3cc(C)on3)=O)cc2s1)OC c1(CC)ccc(C(=O)NCCCCCCNC(C2CCNC2=O)=O)cc1Br Cc1cc(C)c(OCC(=O)NC(C)CN(C)C(C2(C)CCNC2=O)=O)c(C)c1 C1(COC)CC(CNC(C2(N(C)C)CC2)=O)N(C(=O)C(N2CCOCC2=O)C)C1 Cc1csnc1C(=O)NCC(F)CNC(c1ccn(-c2ccccc2)n1)=O C1(C(=O)NCC(C)(C)OC)CC=CCN1C(=O)C(C(C)C)NC=O C1(NC(Cn2ncc(C#C)c2)=O)CN(C(C2(OC)CCC2)=O)C2(CCCOC2)C1 C(C(C)C)(C(O)C(=O)NC1CCCCC1CNC(c1cc(Cl)cnc1O)=O)OC c1(SC)ncc(N)c(C(=O)NCCC(C)(C)NC(=O)C(C)(C)O)n1.CC#N c1(C(N2CCC(OC)(CNC(c3cncnc3C)=O)C2)=O)cnc(Cl)c(Cl)c1 N1(C(C2N(C(c3[nH]cc(C)c3C)=O)CC(=O)C2)=O)CC2CC1CS2=O C1(F)(CNC(C)=O)CCN(C(=O)C(c2cccc(C#N)c2)C)CC1 c1(C(N(CCNC(CCC2CC(OC)C2)=O)C)=O)cc(C)nc2c1c(C)nn2C O=C(C1CCCc2nccn21)NC1CC12CCN(C(=O)CCOCC(F)F)CC2 c1(C(=O)NC(C)CCCCNC(=O)CC(F)F)ccc(Cl)c(Cl)c1N c12ccc(C(CN(C)C)NC(CCC)=O)cc1O2.C(=O)(C(O)C(C)C)N c1(C(=O)NC2(CNC(c3c(C)n(C)nn3)=O)CC2)cnc2cc(F)ccc2c1 N(C1CCc2ccc([N+](=O)[O-])cc21)C(C(n1c(CC)ncc1)C)=O C(C1=NOC2COCC12)NC(C)=O.CCCCC(O)C(=O)NCC(N1CC(C)(O)C1)=O C1(NC(C2N(C(C(C3CC(F)(F)C3)OCC)=O)CC=C2)=O)CCCCC12CCC2 c1(CC)ccc(F)cc1C(=O)NC1CN(C(=O)C(O)CC(N)=O)CC1C(F)F C(=O)(C1=COCC1)N.C12(CCCC1)C(=O)N(CC)CCN(CC)C2=O.C(C)(C)(C)OCC c1(C(=O)NCC2CCN(C(C(c3ccc(F)cc3)CC)=O)C2)cccc(N)c1C C1(C(=O)NCC(C)N(C)C(c2cc[nH]n2)=O)CN2CCCC1C2 N1(C(C2C(=C)CC2)=O)CC2CC2(CNC(c2cncc(C(F)F)c2)=O)C1 c1(OC)ccc(C(N2CCC2(CO)CO)C(=O)NCc2cc(Br)ccc2F)c(F)c1 Cc1cc2ccc(C(=O)NC(CNC(=O)CCC3CCCOC3)C(C)C)cn2c1 c1(CC)oc(C(=O)NC2CC(CCNC(=O)C(c3ccccc3)C)C2)cc1C c1(C(=O)NC2CCN(Cc3ncc(Br)s3)C2)cc(O)ncn1 C(CCCCC(=O)N(C(c1n[nH]c(CC)c1C)=O)C)NCC(F)Cl c1(N(C)C)cc(C(N2CCC(C)(NC(c3nccnc3N)=O)C2)=O)cc(Cl)n1 C(C(COC)C(=O)NC1(CNC(C2CCCCN2C(C)C)=O)CCOC1)OC c1(OC)cccc2ccc(C(=O)NCCC(C)O)nc12.C12CC1C(=O)N2 C1(C(=O)N(C(=O)Cc2nc(C(C)C)cs2)C2CC2)CCC(CNC(CC)=O)C1 C(CCC(=O)NC(C)CNC(C1CC(F)(F)C1)=O)NC(=O)OCC N1(C(C(C)NS(C)(=O)=O)=O)CCC(C2(C(=O)NCC(N)=O)CCOCC2)CC1 N(C(=NCCC(C)=O)NC(c1cccc(Cl)c1F)C)C1CC(CC)C1 C1(NC(C(C)n2cnnn2)=O)CCC(O)CN(C(=O)C=CC(F)(F)F)C1 N1(C(c2cc(C)nc(O)n2)=O)CC2CC1CCC2NC(c1n[nH]cc1Br)=O CC(C)C(C(=O)NCC(C)O)N(C)C(=O)C1CC1 c1(C(N2CC(O)(CNC(c3c(C(N)=O)nccn3)=O)C2)=O)cnc2ccccn12 N1(C(C(C)OC2CCOC2)=O)CCC(NC(=O)C2=CC(C)(C)C2)C2(CCC2)C1 C(=O)(CN(CSc1ccc(Br)cc1)N(C)Cc1ccco1)OC N1(C(C(n2ncc(C)c2)C)=O)CC2CC(O)C1C2NC(c1cccc(Cl)c1O)=O c1(CC(=O)NC(CC=C)CNC(=O)C(n2cc(Cl)cn2)C)n[nH]c2ccccc12 N1(C(C2(C)CCCN(C(C3CCCCO3)=O)C2)=O)Cc2ccc(F)cc2C1 c1(C(=O)NC2C(CNC(c3c(OC)scc3)=O)CCC2)ccccc1C(C)=O c1(C(N(C2C3CCC3CN2C(=O)OC(C)(C)C)C)=O)cc(Br)c2occc2c1 c1(C(N2CCC(CC(C)NC(C=COCC)=O)CC2)=O)cc(N)c(Cl)cn1 n1(C(C)C(=O)N(C2CCOCC2)C)cnc2ccccc12 N1(C(C(CC(C)C)OC)=O)C2CCC1CC(CNC(c1cc(C(F)F)no1)=O)C2 C(=O)(C(CCOC)N(C(=O)COCC(F)F)C)NCC(CC)O CC1CN(C(C2CC(F)(F)C2)=O)CCN1C(=O)C=CSc1ccccc1 N1(C(Cc2c(C)occ2)=O)CCC(NC(=O)C=C2CCOCC2)C1(C)C CC(C)C1=NOC(C)(C(N2CCCC(NC(c3ccc(C#N)s3)=O)C2)=O)C1 c1(OCC(=O)N(c2c(OC)ccc(F)c2)C)ccc2c(c1)CCC2 C1(CCNC(C2(F)CCCC2)=O)CCN(C(C2CCCCC2O)=O)CC1 C1(CCCNC(C2OCCCO2)=O)(CNC(C2C(C)C2C)=O)CCCC1 CC(C)CC(C)(O)C(=O)NCC(C(=O)N(C)Cc1cn(C)cn1)C(C)(C)C C1(C(N(C(CCNC(c2cnn(CCOC)c2C)=O)C)C)=O)CCC(C)(C)CO1 CC(C(=O)N1CCCC1C(C)(C)NC(c1cncc(O)c1)=O)P(C)(C)=O C1(NC(c2ccc(C)cc2O)=O)CC2CC1CN(C(=O)C=Cc1c[nH]nc1C)C2 CCC(CC)(CO)C(=O)N1CCC(CCNC(=O)CCN2CCC(C)CC2)C1 C12(CC(N3C(CNC(c4coc(SC)c4)=O)CC(O)C3)=O)CCC(CC1)CC2 C(c1cccc2ccccc12)=CC(=O)NC1CN(C(c2c(C)occ2)=O)C2C1C2 c1(CCN(CCCN(C)C)CC#N)ccc(Cl)nc1.n1(CC(=O)O)cncn1 N1(C(C(CCC)OC)=O)CCCC(NC(=O)CSc2cnn(C)c2)C1C C1(NC(CCCn2c(C)ncc2)=O)CCC2CN(C(=O)C=CCF)CCC2C1 S(=O)(=O)(CCC(=O)NC(CNC(=O)CN1CC=CC1)C1CC1)NC Cn1nnc(Br)c1C(N1CCC(OC)C1)C(=O)NCCCF.c1cccc(F)c1 Cc1nnc2n1CCC(C(=O)N(CCCNC(c1cc[nH]n1)=O)C1CC1)C2 n1(CC(=C)C)c(N(CC(=O)OCCC)C(C)C)nnc1-c1csnn1 c1(C(=O)NC(CNC(C(CC)=CCCC)=O)CO)ccnc(Br)c1N C1(C(=O)NC(C)Cc2nn[nH]n2)CCC(C2CC2)N1C(c1c[nH]c(=O)cn1)=O CCC(C(=O)N1CC(O)(C2CCCN2C(=O)CSCc2ccncc2)C1)SC c1(OC)cc(C#N)ccc1-c1noc(-c2cc3scnc3[nH]2)n1 C(CC(=O)N(CCn1cncn1)CC)(C(C)(C)C)NC(C=CC=CCC)=O C(C)(C)(CC(=O)NCC1CCCN1C(=O)CC1(N2CCCC2)CC1)OC N1(C(c2n(CCC)nc(C)c2)=O)CCC2(CCC(NC(=O)C(C)(C)OC)CC2)C1 N1(C(CC2(OC)CCC2)=O)CCN(C(c2nn(C)cc2N)=O)C(C)C1 CC(C)C(CCNC(=O)C(c1cscn1)N(C)C)NC(=O)CN1CC=CC1 C=Cc1ccc(NC(C2CCN(C(c3cc(CCC)[nH]n3)=O)C2C(C)C)=O)cc1 C(C(C)(C)C(=O)NCC1CCCN1C(c1cnn(C(F)F)c1)=O)OCC CCCCC(CNC(=O)CCc1cccnc1C)NC(C1(C)CSC1)=O CC(CC(=O)NC1COCCC1(F)F)C(C)(C)NC(c1cccc2cncn12)=O c1(-n2ccc(C(=O)NC(C)C(CO)NC(=O)CO)n2)ccc(F)c(F)c1 C1(O)(CC(=O)N(C(CNC(c2cncc(C)n2)=O)C)C)CCCN(C)C1 c1(C(N2CCC(N(C(C3(CC)CCC3)=O)C)C2)=O)cc(F)cc2c1NCCC2 C1(C#CC(=O)N2CCC(N(C(=O)CC(C)(F)F)CC)CC2)(CC)CC1 c1(Cc2ccn(C)n2)cccc(NC(=O)Nc2cc(-c3ccccc3Cl)[nH]n2)c1 Cc1ccc(C=CC(N2CCN(C)CC2CNC(=O)Cn2cc(Cl)cn2)=O)cn1 c1(COC)ccc(C(=O)NOCCn2nnc(C(C(=O)O)C(N)=O)n2)cn1 c1(C(N(CCNC(C(CC)COC)=O)C(C)C)=O)ccc(Cl)c(C)c1Cl C(=O)(C(=O)N=c1ccn(-c2ccc(Cl)cc2Cl)[nH]1)Nc1c(=N)[nH]cnc1 C(CN=c1ncc(C(F)F)c[nH]1)C1CCN(C(C(C)SC)=O)C1 c1(Nc2c(CCSC)cccc2)[nH]c(=NC2CCCCCCC2)nc2scnc12 c1(OC)cc(C(N2C3CN(C(c4ccc(OCF)cc4)=O)CC23)=O)cnc1F N1(C(C2CC(=C)CN2C)=O)CCC(OC)C(C)(C)C1.c1(CN)cccc(OC)c1C c1(C(=O)NC(CNC(C2CCCN2C2CC2)=O)CO)cc(F)cc2ccncc12 C(C)(C)(C(C)CC(=O)NCCC(CO)C(C)C)NC(C(C)=CC1CC1)=O n1(CC(=O)NC(C)CCCNC(c2ccon2)=O)cc(C#N)c(O)nc1=O C(CC1=CCN(C(C2CC23CCCCC3)=O)CC1)NC(c1cccc(CO)c1)=O C1(OC)CC2CC(NC(=O)C(C3(O)CCC3)NC(c3cscn3)=O)CC12 C1(CN(C(C(F)=CCC)=O)C)CCCCN1C(=O)CC1CCC(=O)N1C c1(C(=O)NCC(C)(C)CCNC(=O)Cc2c[nH]nc2O)c[nH]c2cnccc12 C1(NC(C2CC(C)(C)N(C(C3C4CC5C(C4=O)C35)=O)C2)=O)CCCCC12CCC2 c1(C(N2C(CO)CC(NC(C(C3CCC3)OCC)=O)C2)=O)noc2c1CCCC2 C1(NC(C(C2CC(NC(C(C)OCOC)=O)C2)F)=O)CCc2n[nH]cc2C1 C1(C(N(C2CN(C(C(CC)OC)=O)C2)C)=O)CCCCN1C(=O)N(C)C C1(C(=O)NC(C(N)=O)CO)(NC(c2ncncc2Cl)=O)CC(F)(F)C1 CCCCS(=O)(=O)CC(=O)N1CC2CC1CN2C(c1[nH]nc([N+](=O)[O-])c1Cl)=O Cc1ccccc1-c1nc(C(=O)N(CC(C)NC(=O)COC(F)(F)F)C)cs1 c1(CCC(=O)NCC(CO)NC(COC(CC)CC)=O)nc(C)c(C)[nH]1 N1(CC)CCN(C(c2ccccc2OC)C(=O)Nc2cccc(Cl)c2)C(C)C1=O c1(C(=O)NC2(C)CN(C(c3c(COC)cco3)=O)C2)ncn2c1COCC2 C1(C2CCOCC2)(C(=O)NC2CN(C(Cc3c(C)nc[nH]3)=O)C2)CC1(F)F C(=O)(C1=NOC(C)C1)N1CCC(N(CC#C)C(c2n[nH]c(C)c2C(=O)O)=O)CC1 C1(C#N)(C(=O)NC(C2CCN(C(=O)C=CC3CCCC3)CC2)C)CC=CC1 c1(CC(=O)NC(CC=C)CNC(=O)C(C)O)cc(OC)ccc1OC Cn1nc(Br)c(CNC(=O)Nc2cncc(SC3CCOC3)c2)c1Br c1(C(=O)NCC(CC(=O)NC(CCOC)(C)C)OC)c(C)nc2ncnn2c1C CC1CCC(C)(NC(=O)CC2(NC(=O)CCCC#N)CC(OC)CC2)C1 C1(C)(C(=O)OC)CN(CC(=O)Nc2cn(C)c(C(F)F)n2)CCO1 c1(CC)ncc(C(=O)NC23CC(C(N4CCC4C)=O)(C2)C3)cn1 N1(C(C2C(C(=O)OC(C)(C)C)C=C2)=O)CCCC12CCN(C(=O)CCC(N)=O)C2 N1(C(C(CC=C)OC)=O)CCC2(CC1)CC2N(C(=O)C=C1CCC(C)C1)C1CCC1 CC(C)C(F)C(=O)NCCC1CC(NC(c2csc(Br)c2Cl)=O)C1 N12CCN(CC1)C(=O)C2.N(S(=O)(=O)N(C)C)C1CCN(CC)C1 C1(CC(=O)N(C)CCN(C(=O)CN2CCCCC2C)CC)(CC=C)CCCCC1 c1(C(N2CCC(N(C(C3C(C)C3C)=O)CC)C2)=O)cc(F)c(C)cc1Cl N1(C(c2ccc(OC)s2)=O)CC(NC(=O)CCc2ccc(C)nc2)CCC1C C1(C(=O)NCC2(NC(CC3(C)CC3)=O)CCC2)CC(=O)CO1 c1(C(N2C(CNC(C=COCC)=O)C=CC2)=O)nc(-c2ccccc2)cc(O)n1 c1(C(=O)NC2CN(C(Cc3c(C)con3)=O)CC2C)csc2ccc(Cl)cc12 C1(C#CC(=O)NC2CC(O)(CNC(=O)C3=CCCCC3)C2)(CC)CC1 N1(C(c2cc(C)n(C)c2)=O)CC2CCC(C1)N2C(=O)CSC1CCS(=O)(=O)C1 c1(C(N2CCN(Cc3ccccc3)C(C3CC3)C2)=O)cc(Cl)c(F)cc1F N1(C(C=Cc2c(C)cccc2)=O)CCC2CN(C(c3cc4c(s3)COCC4)=O)C2C1 c1(NC(=O)NC2CCCC(N3CCCS3(=O)=O)C2)ccc(N2C(=O)OCC2)cc1 N1(C(c2nc(COCC)sc2)=O)CC(C)CN(C(=O)C2=CCOCC2)CC1C C(=O)(CCCCN1C(=O)CCC1=O)NCCN(C(=O)CCCc1cnn[nH]1)CC C=C1CC(C(=O)N(CCOC)CCSC)(CNC(C2CNC(=O)C2)=O)C1 C1(C(=O)NCC2(C(=O)O)CCN(C(COCCC)=O)C2)CC2CCC(C1)O2 Cc1cnc(C(N2CC(CO)(NC(c3ccc[n+]([O-])c3)=O)C2)=O)c(Br)c1 c1(Cc2n3c(nn2)NC(=O)CN(C)CC3)ccc(C)c(C)c1.CCCOC n1(CC)ccc2cc(C(=O)N(C3CCN(CCO)CC3)CCCO)ccc12 C(=O)(CS(=O)c1ccc(Cl)cc1)N1CCC(NC(c2ccc[nH]2)=O)C12CC2 Cc1cccc(-c2c[nH]cc2C(=O)NCC2CCC(NC(C3(C#N)CC3)=O)C2)c1 C12(C(=O)NCCCCCNC(C(C)O)=O)CC3(F)CC(F)(C1)CC(F)(C2)C3 c1(SC)cscc1C(=O)N(CC(C)NC(=O)CCc1cnc(C2CCC2)s1)C CC1(C)OCCOC1CC(N1CC2CC1CN2C(=O)CC(C1CC1)C1CC1)=O C1(NC(C(C)=C2CCCC2)=O)C=CCN(C(C2CC(=O)N(C(C)(C)C)C2)=O)C1 c1(C(N(C2CCN(C(C3(COC(C)=O)CC3(F)F)=O)CC2)CC)=O)c[nH]ccc1=N c1(C(N(C(C)CNC(C2(F)CC2)=O)CC)=O)ccc(Cl)cc1Cl C(C(C)CC(=O)NNC(=O)C(C)(C)CCCCSC)NC(C(C(=O)OC)(C)C)=O c1(C(=O)NCC2C(NC(=O)CCCC3CC3)CCC2)ccc2n[nH]cc2c1Cl c1(OC)ccccc1NC(C(=O)N(CC(C1CCN(C)C1=O)(C)C)CC(F)(F)F)=O C1(CC(=O)Nc2cccc(NC(C(C)NC(C)=O)=O)c2)CN2CCN1CC2 N1(C(C(C2CCN(C(CC(CCC)C)=O)CC2)C)=O)CCCCCCC1C C(C)(C(CC(=O)N=c1cc(C)n(C2CC2)[nH]1)NC(=O)C1=CCCC1C)OC C1(C(=O)NC2(CC)CCCC2)(CC)CCCCO1.C1=CCNC1=O C1(NC(COCCCCCC)=O)CC(CCC#N)N(C(=O)CCC2CC2(C)C)C1 c1(OCC)ccccc1CCC(=O)NCC1CC(NC(C2CC(F)C2)=O)CC1O Cc1c(CN2CCCC(N(c3nccc(N4CCCC4)n3)CCO)C2)nnn1C N1(C(COc2ccn(C)n2)=O)CCC(NC(C2CS(=O)(=O)C2)=O)CC(O)C1 C1(C(=O)OC)CCOC1C(=O)NC12CC(NC(=O)CSc3ccccn3)(C1)C2 c1(NC(CC)COC(C)C)cc(N(C)Cc2ccc(=N)[nH]c2)ncn1 CC1CCCCC1C(=O)NCC(CNC(c1cc(C(N)=O)no1)=O)CO CC1CCN(C(=O)C(=O)N(C)C)CCN1C(c1cnccc1C(F)(F)F)=O c1(C(N(C2CCN(C(C=CCCC)=O)C2)CCC)=O)ccc(=O)n(O)c1 N1(C(CCC#C)=O)CCC2(CC2NC(=O)CN(C)C(C)C)C1 N1(C(Cc2n(C)ncc2Cl)=O)CC2=C(C1)CN(C(c1ncc3ccccn13)=O)C2 C1(CC#C)(C(=O)NC(C2CN(C(=O)C(C)(C)N3CCCC3)C2)C)CCCO1 C1(CC)CN(C(C2(NC(c3cc(C(C)=O)c[nH]3)=O)CCC(C)(C)C2)=O)CCCO1 c1(OC)c(Cl)cc(C(=O)NC2CCCN(C(=O)CN3CC=CC3)C2)nc1Cl C1(NC(C(C)OCC)=O)(COC)CN(C(=O)CSC2CC2)C1 c1(CC(=O)NCCNC(C2(C)CC=CCC2)=O)ccc([N+](=O)[O-])cc1Cl C1(CNC(c2scc(C)c2)=O)CC2CCC1N2C(c1cc(C(N)=O)ccc1C)=O c1(C(=O)NCC2CN(C(CC=C=C)=O)C2)cccc(NC2CCC2)n1 C#CCCCC(C(=O)NC(C)(C)CC)N1CCC(OCCN(C)C)C1 c1(CN(C(c2ccc(Br)cc2)CC)CC)ccc2c(c1)CCCN2C N1(C(c2cc(CCC)on2)=O)CCOC(CNC(=O)CCCCN2CCCC2)C1 Cc1nc(NC2CCCc3n[nH]cc32)c(Cl)cc1C#N.C1(=O)C(C)N1 N(C1CCc2cccnc21)C(C(CC(C)(C)C)NC(=O)CC1CC(F)C1)=O C1(NC(=O)CN2C(=O)CCC2=O)CCCCN(C(c2cocn2)=O)C1 c1(SCC(=O)NC(CCNC(C2(CC=C)CCCC2)=O)C)cccc(OC)c1 C1(O)(CN(C(=O)CCOc2cccnc2)C)CCCN(C(=O)CC2OCCO2)C1 N1(C(c2cc(C)sc2C)=O)CC(C2CC2)(C(=O)NC(c2ccsc2)C)C1 C(=O)(CC(F)(F)C(F)(F)F)NCC1N(C)CCN(C(C(COC)C)=O)C1 CC1(CC(=O)NCCC2CCCCC2)CCN(C(C2CCCO2)=O)CC1 C(=O)(C(CCSC)OC)N1CCC(NCC=C)C1.C1(C(=O)NC)(OC)CCOC1 C1(N(C(C2CC2(C)C)=O)CC)CCN(C(=O)Cn2ccnc2C)CC1 c1(C(=O)NCC2C(NC(CCOCCOC)=O)CC2)c[nH]c2ccc(F)cc12 C=CC(CC)CC(=O)N1CCCC(CC(N2CC(OC(=O)NC)C2)=O)CC1 C1(C(=O)OC)C=CCN1C(=O)CC1CCCN1C(=O)COC(C)C C1(NC(COCCC#C)=O)CC2CC(C1)N(C(=O)C=CC(c1ccccc1)=O)C2 c1(C(=O)NC2CN(C(C(=O)NC(C)C)=O)CC2O)cc2scc(Cl)c2[nH]1 c1(CC(=O)NCC(CO)NC(c2c(C(C)C)con2)=O)ccc(F)c(Cl)c1F C1(NC(=O)C=Cc2cscn2)C2CCC(C2)C1C(=O)NCC1CCCC1 c1(Cn2c(CC)nnc2N2CC=C(Br)CC2)cc(Sc2ccccc2)cc(F)c1 C1(NC(C2(OC)CCSCC2)=O)CCN(C(=O)CC2CC3CC3C2)CC1(C)C CC(C)(C(=O)N1CC2CC1C2CNC(=O)C(F)(F)CC1CCCO1)C(F)F CN(C1CCc2c(F)cccc21)C(C1CCCC1c1nc(S)n[nH]1)=O C1(CNC(CNC(CC)=O)=O)CC(C)(C)CCC1NC(=O)CSCCOC C=C(C)CC(C(=O)NC1COCC1C(=O)NC1CCC1(C)C)OC CC(C)C(F)(CNC(C1C2CC(=O)CC12)=O)C(=O)NC(c1cccnc1O)C c1(C(N2CC(C)(C)C(NC(C3CCOC3)=O)C2)=O)cc2cc(Br)cn2cn1 C1(NC(C(C)SC)=O)CN(C(c2c(C)nc(C)n2O)=O)CC2(CCC2)C1 C1(C(=O)NC(CCCCC(C)N(C(c2cc[nH]c2)=O)C2CC2)=O)CCCN(C(C)C)C1 C(=O)(C1=CCSC1)N1C(C)(CC(N2CC(C(C)OC)C2)=O)CC1 N1(C(C(C)Sc2c(F)cccc2F)=O)CCc2cc(O)ccc2C1 C1(O)(CCNC(c2cc(C)on2)=O)CCCN(C(c2cncc(O)c2)=O)C1 CCC(CCOC)N.C(=O)(C(O)C1CN(C(c2cnsc2)=O)C1)C(CC)CO C1(C(=O)OC)CCC(n2nnnc2Cc2scc(CN(C)Cc3ccon3)n2)C1 C1(C(=O)NCC(Cl)=CCl)CCC(C)(NC(C(C)n2ccnc2)=O)CC1 CCCC(CCC)CC(=O)N(C1CCC(NC(=O)CCN2CCCS2(=O)=O)C1)C c1(OC)c(C(=O)NCC(C2CCCC2)NC(C2CCC2(F)F)=O)cccc1Cl N1(C(c2cnn(C(C)C)n2)=O)CC(NC(c2cn(CCO)nn2)=O)CC(F)C1 C1(C(N(C2(C(=O)NCCS(C)(=N)=O)CC2)C)=O)CCCC1C1CC1 N#Cc1ccc(F)c(NC(C2CCCC2NC(=O)CCc2ncc[nH]2)=O)c1 N1(C(C(CNC(CCN(C)CC)=O)(C)OC)=O)CCCN(C)CC1C c1(C(=O)NC2CN(C(CC3C(C)(C)C(O)C3)=O)C2)nncc2c1CCCC2 C1(CNC(C(c2cccs2)SC)=O)CCCN(C(=O)C=Cc2ccsc2)C1 C(=O)(CCCC(O)NC(=O)COC1CCOC1)NCC C(=O)(CCC(C)(C)C#N)N1CC(N(C)C(C2C(=O)NCC2(C)C)=O)C1 C(C(C)CC(=O)NCC12CC(NC(=O)CNC(=O)CCSC)(C1)C2)OC c1(C(N2CC(C)N(C(c3cc(O)cc(F)c3F)=O)CC2)=O)cc(C#N)ccc1F c1(CCCC)ccc(C(=O)N(C(CNC(C2CNC(=O)C2)=O)C2CC2)C)cc1 c1(C(=O)NCc2c(C(=O)NCc3ccc(C)cn3)nco2)ccc(C)c(C#N)c1 C(=O)(C1CCCn2c(C)cnc21)NC1(CNC(c2nn(CC)c(O)c2)=O)CCC1 CC12CN(C(=O)C(=O)NCCCN3CCOC3=O)C(NC(=O)C3CC3)(C1)C2 c1(C(=O)NC(C)CC(=O)NCCC2CCCC2)cc([N+](=O)[O-])c[nH]1 N1(C(C(C)(C)NC(=O)NCC)=O)CCC(C)N(C(=O)CC2CCC(C)(C)C2)CC1 N1(C(C(CC)=CC)=O)CCCCC1CCC(C)(C)NC(=O)Cn1ccc(C2CC2)n1 Cc1ccc(C2(C(=O)NCCCC(C)NC(=O)CCc3ccco3)CC2)c(C)c1 N1(C(CSC)=O)CCCC(C2CCN(C(c3cncc(Cl)c3C)=O)C2)C1 C1(N(C(C2C(C=C)C2)=O)C)CN(C(=O)CCC2CC(F)(F)C2)CCC1O C(=O)(C(C)(C)C(C)(F)F)NCC(COC)NC(=O)COCC1CCC1 C1(NC(c2cc(C)c(Br)o2)=O)C2CC1CN(C(C1CCSCC1)=O)C2 c1(NC(C2(CCNC(C3CN(C)C(=O)N3)=O)CC2)=O)cccc2cnccc12 Cc1ccccc1CC(C)C(=O)NCC(C1CCC1)NC(C1(C(=O)N(C)C)CC1)=O C1(NC(C(C(C)C)NC(C)=O)=O)CCN(C(c2cc(C)cc(C)c2)=O)C(C)C1 C1(NC(c2nc(COC)sc2)=O)CC2CN(C(=O)C(F)C3CCOC3)CC12 CCCC(C(=O)N1CCC(O)(CC)C1)NC(=O)CC1CNC(=O)O1 C(=O)(CCCCCCNCc1ccccc1)N1CCN(C)CC1Cc1ccccc1 Cc1ncc(CNC(=O)C(C)CN(C(=O)C(=C2CCCCC2)F)C)o1 c1(OC)cc(NCC2CCCC2NC(C2CCCC2(F)F)=O)ncn1 N1(C(CC2CCCC(NC(C=CC(CC)C)=O)C2)=O)CCCC2(CCC2)C1 C1(C(=O)NCC(c2ccccc2F)NC(=O)CCC2CC2)CCCCCC1 C1(NC(c2ccc(OC)s2)=O)CC(NC(=O)C=CSC)C12CCC2 Nc1cc(F)cc(C(=O)NC2CCCC2c2ccc(Cl)cc2)c1F C12(NC(C3(N(C(c4nncs4)=O)Cc4ccccc4)CC3)=O)CC(F)(C1)C2 c1(C(N2CC(CCC)N(C(c3cnn(C)n3)=O)CC2)=O)ccc2snnc2c1 CCC(C)CCCCC(=O)NCC1CCC2(CN(C(c3nc(O)c(C)s3)=O)C2)O1 C=CC1CCN(C(=O)CC2CC(F)CN2C(=O)C(COCC)OC)C1 C=CCCCCC(=O)NCC(CC)NC(=O)C(C)Oc1ccccc1C(F)(F)F C1(C(N2CC(NC(C(C)OC3CCCC3)=O)C(O)C2)=O)CSc2ccccc2O1 C1(NC(C2(COCC)CCC2)=O)CN(C(=O)CC(F)(F)C(F)F)CC(C)(C)C1 C1(C(N(C2CN(C(c3cccc(OCC(F)(F)F)c3)=O)C2)C)=O)CCC(C)(C)C1 CC(C)CC(C(=O)N(C(C)C(=O)NOC1CCCCC1)C1CC1)C(N)=O n1(C(C)C)ncc(Br)c1-c1nc(-c2ccc(Cl)nc2)nn1C1CCCOC1 C#Cc1ccc(Br)c(C(=O)NCC(C2CC2)NC(C2CCN(C)S2(=O)=O)=O)c1 C1(CC=C)(NC(=O)CCS(C)=O)CCCN(C(C2CC2(c2ccccc2)C)=O)C1 C(=O)(N=c1cc[nH]c2ccc(I)cc12)C1N(Cc2c(Br)ccc(C)c2)CCC1 N1(C(CC(C)C(F)F)=O)CC(CNC(c2cn3c(n2)CCC3)=O)CC12CCC2 N1(C(C(C)=CC)=O)CC2CCOCC2(NC(=O)CCCc2cc[nH]n2)C1 CCCC(C)(O)CNC(C1(CNC(=O)Cc2coc(C)n2)CC1)=O c1(C(=O)NCC2CC(OC)CN2C(c2sc(C)nc2C)=O)ncc(C#N)cc1Cl c1(C(=O)NCC2CN(C(C3C(Cl)(Cl)C34CC4)=O)CCO2)ccc2nc[nH]c2n1 N1(C(CC2CC(C)(C)C2)=O)CCCC(C)(CNC(C2CC23CCCC3)=O)C1 C(C)(C)(CCNC(c1cncs1)=O)NC(C1C(C(C)C)(CC)C1)=O c1(C(=O)NC2CC(CCNC(C3(COC)CC=CCC3)=O)C2)c(N)sc(C)c1C NC(=O)CCCCC(=O)NCC1CCC(CNC(C2CC3C=CC2C3)=O)CC1 N1(C(C2C(CCC)C2)=O)CCC2C(C(=O)NC(C)(C)CC3CCOC3)C2C1 S(=O)(=O)(c1c[nH]ccc1=NCCC1(C)CC1)NC1C(c2cn(C)nc2)C1 Cc1cnc(C(C)OC(c2ccc(C)o2)=O)o1 c1(CNC23C(CN(C(=O)COc4ccccc4)C2)C3)cnc2n1CCC2 C(=O)(C#CC1CCOC1)Nc1c(C)cc(NC(C2C3CC4C(C3=O)C24)=O)cc1 C1(C)(NC(CC2CC(O)(CNC(CC(C)C3CCCO3)=O)C2)=O)CCSCC1 CN1CCCC12CCN(C(=O)C1=C(F)CN(C(=O)CCn3cccc3)CC1)C2 C(=O)(C1=NOC(C)(C)C1)NCCN(CC(C)O)C(C1CC2C=CC1CC2)=O n1(CC(=O)NC2C(NC(C3(C)CCC3)=O)CCC2)cc([N+](=O)[O-])cn1 N1(C(c2cn(C)c(O)n2)=O)CCC(NC(C2CC2Cl)=O)C12CCCC2 c1(C(=O)NCC(CNC(CC(=C)C)=O)OC)ccc2cnoc2c1 C(=O)(CCCCC(C)CC)NC1C2(CN(C(C(C=CCCC)O)=O)C2)SCC1 CC(C)CCCCCN=c1[nH]c(=NCCn2cc(Br)cn2)[nH]c2ccccc12 C=C(F)C1(CC(=O)NCC2CCC(NC(=O)C(F)=CCC)CC2)CCC1 CC(c1cnn(C)c1)=CC(=O)NCC1CC2(CC2)CN1C(C1CCC(C2CC2)C1)=O N1(C(C(CCC)C)=O)CCCC2(C1)C(NC(c1nc(Cl)oc1C)=O)CCN2C C1(NC(CN(C(=O)CC=CC(C)(C)C)CCC)=O)CCCN(CCC)C1 C1(NC(C2CCC(C)CC2)=O)COC2(C1)CN(C(=O)CCCc1ccccn1)C2 C(CNC(=O)C=CC(F)(F)F)(C(C)(C)C)NC(C1N(C(C)C)CCC1)=O c1(C(N2CC(NC(C3CC(CC)C3)=O)CC2(C)C)=O)cncc2cccnc12 CC(C)(C)CC(O)C(=O)NCC1(F)CC(NC(=O)CC2CCCC2(F)F)C1 C(=O)(C(CCSC)OC)NCCCCNC(c1c(OC)nsc1)=O C1(CNC(CCSC)=O)CN(C(c2cc(C)sc2C)=O)C2CCN1C2 Nc1ccc(C(N2CC(NC(=O)C=C3CCC3)C3(CC3)C2)=O)c(Br)c1F c1(C(N2C3(CNC(c4cncs4)=O)CC(C2)C3)=O)cnn2c1OCC(F)C2 CCC(C)(C)CCCC(=O)NCC(CC1CCNCC1)CO N1(C(CCNC(c2ccc(F)cc2)=O)=O)CC2CC(O)CC(C2)C1 C(CCC(C)CC(=O)NCCC1CSCCN1C(=O)Cc1csc(=N)[nH]1)=C(C)C C(=O)(CCC(CF)CF)N1CCCCC(C(N(C)Cc2cncs2)=O)C1 c1(CC(N2CCC(O)C(C(N)=O)C2)C(=O)NCCCC)ccc2ccccc2c1 C1(NC(C2(COC)C=CCN2C(=O)CCCCN(C)C)=O)CCC(=O)NC1=O C(N(C)N1CCN(C(C)(C)C)C2=NCC12)c1cc(C)cc(C)c1 C1(CC(C)C)C(=O)N1.C(C(C)(C)C)[SH](C(CC1CC1)CC1CC1)C CCCC(C(O)C(=O)NCC1CCCCN1CC)NC(=O)CC(C)F C=CCC(C)(C)C(=O)NC(C1CCCN(C(c2conc2C)=O)C1)C c1(COC)ccc(C(=O)OCC2(C(C)(C)C)CCCO2)cc1OC(C)=O c1(C(N2CC(CC(C)NC(c3c(C)nsc3)=O)C2)=O)csc2cc(Cl)cnc12 C1(N(c2cnn(C)c2)CC)CCCN(C(=O)C(N)=O)CC1 c1(C(=O)NCC2(O)CN(C(=O)Cc3ccc(F)c(F)c3)C2)n[nH]c2c1COCC2 C1(C(=O)OC)CC2(CCCC2)CN1C(c1cc(Cl)cc([N+](=O)[O-])c1N)=O C12(CNC(c3ccc[nH]3)=O)CC(C1)C(NC(C1CCCC(F)(F)C1)=O)CO2 CCC(N=c1cc(C)c(C#N)c(C)[nH]1)C1CCN(c2nncs2)CC1 CN1CCC(=CC(=O)NCCC(O)CNC(c2ccccc2C2CC2(F)F)=O)CC1 c1(C(=O)NCC2N(C(C3CC(=O)NC3)=O)CC(F)C2)ccc2sncc2c1 N1(C(COc2ccn(C)n2)=O)CC(NC(c2scnc2C(C)(C)C)=O)CC(O)C1 c1(NC2NCCN(C(CCc3nc(=N)[nH][nH]3)=O)C2)ccc(F)cc1[N+](=O)[O-] c1(NC2(C3CN(C(C(CC#C)C)=O)C3)CC2)c(C)cccc1[N+](=O)[O-] CC1S(=O)(=O)CCC1C(N1CCC(CO)(CNC(c2cnc[nH]2)=O)CC1)=O CCC(C(=O)N(CCNC(c1c[nH]c(=N)o1)=O)CC1CCCC1)OC C1(CNC(C=C(C)C(C)C)=O)CC(C(=O)NCc2cnc(C)o2)=NO1 C(CC(C)C)(C(=O)NC(C)C(=O)NCC(C)(C)C(N)=O)OC C1(C(N2C(CNC(c3ccc(C4CCCO4)o3)=O)CC2)=O)Cc2ccccc2O1 c1(N2CCCC(NC(c3cscc3Cl)=O)CC2)ncnc2cccc(F)c12 N#Cc1ccc(CC(=O)NCC2CCN(C(=O)C3=CCCC3)CC2)c(F)c1 c1(N(CCCNC(C=C(C)C2CC2)=O)C2CC2)cc(C)nc(C(C)CC)n1 CC(=O)n1cc(CN2CCSC(C(=O)Nc3ncccc3Cl)C2)c2cccnc12 n1(CCC)cc(C(N2CC(CNC(=O)COCC3CCCO3)(OC)C2)=O)nn1 N1(C(CN2CCC(OC)C2)=O)CCOC(C)(CNC(c2ncc(C)cc2F)=O)C1 Cc1ccnc(C(=O)NC2CCC(NC(=O)C(C)(C)NC(c3ccccc3)=O)C2)c1 c1(NC(C(=O)NC(C(=O)NCC)C)=O)cncc(Cl)c1C CC1(C)C(CNC(C2CC3CCC3C2)=O)CCN1C(c1cc(O)cc(F)c1)=O C(=O)(C(C)(C)CC(=O)N1CCOCC1CC(=O)NCCCCCCO)OC C1(C(N(CC(=O)NCC2C(C)(C)C2(F)F)CCC)=O)C2(CC2)C12CC2 Cc1ncnc(O)c1C(=O)NCC1CC(C)(C)CN1C(c1ccoc1)=O C1(C(=O)NCC2N(C(c3cc(C(C)(C)C)no3)=O)CC2)CC(=O)N(CC2CC2)C1 N1(C(C(C)=O)=O)CC(NC(=O)C(C)Cc2ccco2)C(C)C1 C1(N(C(C(c2ccc(Cl)s2)=O)=O)Cc2ccc(F)cc2)CCc2ccccc2C1 O=C(C1=C(Cl)CCCC1)NC1CCN(CCNC(=O)NC2CCCC2)CC1 CCC(CC)CC(=O)NCC(c1ccccc1F)NC(=O)C(C)CS(C)=O C(=O)(CC(F)(F)CC)N1C(CCNC(C=CC(CC)=CC)=O)CSCC1 N1(C(C2CN(C(N(C)C)=O)C2)=O)CC2CC1CC2NC(c1ncc[nH]c1=O)=O CC(CCC(=O)NC(C(N1CC(CO)(CF)C1)=O)c1ccco1)N(C)C CC(CS(C)=O)C(=O)N(C)CCNC(C1(CCF)CCOCC1)=O Cc1c[nH]cc([N+](=O)[O-])c1=NC(CNC(c1cc2cccnc2s1)=O)CC(N)=O N1(C(CCCOCCOC)=O)CC=C(C(C)(C)C(=O)N2CC(OC)CC2CO)C1 CC12CCC(n3cc(CC4(c5ncco5)CCC4)nn3)(CO1)C2 C(CN=c1cc(Cl)c(O)n[nH]1)(C1CCCC1)NC(C1CCC(C(F)(F)F)CC1)=O N1(C(C2CCN(C(C)=O)C2)=O)CC2CC(C1)C2NC(=O)C(C(C)C)n1cnnn1 c1(C(=O)NCC(C(C)C)NC(=O)C(C)C(C)(F)F)ccc([N+](=O)[O-])c(Cl)c1 c1(C(=O)NCC2N(C(CCC=C(C)C)=O)CCC2)cc(C(F)(F)F)cc(N)c1C N1(C(CC(C)(C)OC)=O)CCC(NC(=O)C(N2CCC(C)C2)=O)C(F)(F)CC1 N1(C(CC2C(C)C2(F)F)=O)C2CCC1CC(CNC(c1nnc(S)n1C)=O)C2 C1(C(=O)NCC2N(C(C(C(CC)C)OC)=O)CC(OC)C2)CN2CCN1C(C)C2 C1(C(CCC)NC(=O)C(O)Cc2[nH]cnc2C)CCN(C(=O)COC(C)=O)CC1 C1(NC(C(CO)OC)=O)CCCC1(C)CNC(=O)Cn1nc(C)cc1C(F)F c1(-c2nnc(CNC(=O)NC(c3nc[nH]n3)C)s2)ccccc1F n1(C(C)C)cc(CNC(=O)CC2CC(NC(=O)C(=O)C3CCCC3)C2)cn1 C1(NC(CN(C(COC)=O)C)=O)C(C)(C)CN(C(c2cnoc2C)=O)CC1(C)C C1(C(=O)Nc2ncn(Cc3ccccc3)n2)CC(CNC(=O)CC(F)(F)F)CCO1 N1(C(C=Cc2ccc(C)s2)=O)CC2CCN(C(C3CC3c3ccn(C)n3)=O)CC12 N1(C(C(CC2CN(C(CC(C)c3ccco3)=O)C2)F)=O)CCN(CC(N)=O)CC1 C1(F)(C(=O)NCCC2CC(NC(c3cnc(CN(C)C)[nH]3)=O)C2)CCCOC1 N1(C(CC2CC(=C)C2)=O)CC(C)CN(C(c2ccc(C)nc2OC)=O)CC1C CCCCC(C)C(=O)N1CC(C(=O)NCC(C)COCC)C2(CC2)C1 N1(C(C2CCNCC2OC(c2onc(C(=O)NC)n2)=O)=O)CCC(CO)CC1 CC1CN(C(=O)C(O)CC2CCOCC2)CCCN1C(=O)CCn1cccc1 Cn1cc(C(=O)NCC2CCN(Cc3cccc(F)c3Br)CC2)c(O)nc1=O C(=O)(C(CCC(C)C)NC(c1cc(C)[nH]n1)=O)NCc1cccc(CC)c1 C1(O)(CCNC(=O)COc2ccccc2)CCCN(C(c2cccc(=O)o2)=O)C1 N1(C(C2(Cc3ccccc3)CC2)=O)CCCC(CF)C1.C12(CCCC1)C(=O)NC2 C1(C)(CNC(C(COC)(C)C)=O)COCCN(C(c2cnc3[nH]nnc3c2)=O)C1 C1(CNC(C=CSC)=O)CCCC2(CN(C(c3n[nH]c4c(C)cccc34)=O)C2)O1 N1(C(c2nc(C)c(F)cc2)=O)CCC2(CC1)CC2(C)C(N1CCOC(C(N)=O)C1)=O C1(NC(c2c(CC)cns2)=O)C(CNC(=O)C=CSC)CCC12CCC2 CC1(CNC(c2cccc(C3CC3)c2)=O)CCCN1C(=O)Cc1nc[nH]n1 c1(NC(C2N(C(c3c(CC)ncs3)=O)CCC2O)=O)ccc(Br)cc1I c1(C(N(CCCN(C(COC(C)C)=O)C)C)=O)cc([N+](=O)[O-])ccc1OC(F)F N1(C(CCCCC)=O)CCCCC(NC(c2c(O)cccc2Cl)=O)C1 c1(C(=O)NC(C2CC(C)(C)C2)C(=O)OC)cc(-c2cccc(F)c2)n(C)n1 CCC(C)(CC)C(=O)N1CCOC(CCNC(C2(C#N)CC3(CC3)C2)=O)C1 N1(C(c2c(SC)scc2)=O)CCCC2(NC(C3(n4ccnn4)CC3)=O)CC2C1 C1(C)(OC)C=CCN1C(c1ccc(Cn2ccnc2)cn1)=O c1(CNC(=O)C=CC2CC2)ccc2c(c1)CCC2NC(=O)C1CCc2c[nH]nc21 c1(OC)ccccc1-c1ncsc1CC(=O)NCc1nc(C(F)(F)F)nn1C C(CCCCCNC(C1(CO)CCCO1)=O)NC(C1(C(F)(F)F)CCCCC1)=O N1(C(CCC(C)OC)=O)CCC(C)(C)C(C(=O)N(C(C)CCO)C)C1 c1(C(=O)NC(CN(C(c2ccc(C#N)[nH]2)=O)CC)C)ncnc(O)c1F c1(CC(=O)OC)cccc(CC(N2CC=CC(NC(=O)C3=COCC3)C2)=O)c1 C1(CC(=O)NCC2C(C)CN(C(C3(O)CCOC3)=O)C2)CCC2(CC1)CC2 N1(C(C(CCC)C)=O)CCC(C(=O)NC2CC2CCOC)C12CCC2 [N-]=[N+]=NCCCCCCC(=O)NC1CCN(CC2CC3C=CC2O3)C1 CC(C)C(F)C(=O)N1CCOCC1CC(=O)NCCCC(C)(F)F Cc1cc(Br)cc2c1CCN(C(c1ccc(-c3cncc(F)c3)nn1)=O)C2 C1(OC)(CO)CC2(CN(C(=O)NC(C)(C)C)C2)C1.N12CCCC(C)(C1)OC2=O Cc1ncn(C)c(=O)c1C(=O)NCCC(C)CCNC(c1cc(O)nn1C)=O N1(C(c2c(C)scn2)=O)CCC(O)(CCNC(=O)CCC2CCCN(C)C2)C1 C1(CN(C(COCC(=C)C)=O)C)CCCN(C(=O)COC2CCN(C)CC2)C1 N1(C(CC(=O)OC)=O)CC2CCN(C(C3CCC(=O)N3C)=O)CC2C1 c1(-n2ncc(C(=O)NCCC3CN(C(C=CSC)=O)C3)c2)cccc(F)c1 C1(CNC(CCC(=O)NCCC)=O)CCC(C)N(C(c2c[nH]nc2C)=O)C1 n1(CC(=O)N(C2CCN(C(=O)Cc3c[nH]nc3C)C2)CCC)cc(F)ccc1=O N1(c2nccc(N(C)Cc3cc(C(F)(F)F)ccc3O)n2)CCN(C)C(C2CC2)C1 C1(N(C(=O)CS(N)(=O)=O)C)CCCN(C(C2(COc3ccccc3)CC2)=O)CC1 c1(OC)ncnc(OC)c1C(=O)NCC1CN(C(C2CCCN(C)C2)=O)C1 CC#CCCCC(=O)NCCC1CCCN(C(=O)C=Cc2cncnc2O)C1 c1(C(N2C(CCNC(=O)CCc3cccc(F)c3)CCC2)=O)ccnc(CO)c1 C12(C(N(C3CCN(C(CN(CCC)C)=O)C3)C(C)C)=O)CC3CC1(CO)CC3C2 C1(NC(c2cnn(C)c2-n2cccc2)=O)CC2(C1)CN(C(C1CCC(O)C1)=O)C2 C1(O)(CC(=O)N(CC(CC)NC(=O)C=CCN(CC)CC)C)CCCN(C)C1 CCCCC(C(=O)NC1CCCC(O)C1)NC(=O)C(C)OCC1CC1 C1(C(=O)NCC(C2CCC2)NC(C=Cc2cn(C)nc2)=O)CN(S(N)(=O)=O)C1 C1(Cn2cc(C(C)(C)OC(=N)O)nn2)C2CN(C(c3ccco3)=O)CC12 C(=O)(CC(C)(C)CC)NCC1C(C(=O)Nc2ccc(C(C)=O)nc2)CCO1 N1(C(c2n(CCC)ccc2)=O)CC(CNC(=O)C(=Cc2cnn(C)c2)C)C(C)C1 CCCC(C)(C)C(=O)NCC1CN(C(C2C3(CCC3)C2C(F)(F)F)=O)CC1C C1(C(=O)NC2CCC2CNC(=O)C(F)(F)c2ccsc2)CCCC1CF CCCC(F)C(=O)N(CC(C)C(=O)N(C)CCN(C)C)C C(C)(CNC(C1CCOC1C(C)C)=O)(CC(C)C)NC(c1c(CC)csc1)=O C(CCNC(c1cccc(=O)o1)=O)(C(=O)NCC1COCC1O)OC c1(C(=O)NCC(CNC(c2ccc(CC)s2)=O)C)cc(C)nc2c1CCCC2 C=CCCC(C)(C)C(=O)NCc1nc(C(=O)NC(C)CCN2CCCC2)co1 C(=O)(C(F)C(=O)NCC1CCCCN1C(c1c[nH]nc1C1CCCO1)=O)OCC C(CN(C)C)(CCO)NC(CN(C(CN(C(=O)CCN(C)CCO)C)=O)C)=O c1(C(N2CCN(C(CN3CC(C)(C)C3)=O)C3C2CC3)=O)nn2cccnc2c1Cl c1(C(C(=O)N(C(CNC(C2CC23CC3)=O)C2CC2)C)C)ccc(Cl)c(Cl)c1 c1(N2CCCC(CNC(c3cc(F)cc(F)c3)=O)CC2)ncnc2c1COC2 N(C1CCCn2ccnc21)C(C(CC=C)CNC(=O)C(C(C)C)NC(C)=O)=O N1(CC(c2ccccc2)NC(C2CCN(C(=O)C3CC3)CC2)=O)CCCS1(=O)=O c1(C(=O)NCCC(CC)OC)ccc(N2CCOCC2)c(C(F)(F)F)c1 CC(C(=O)NC(Cn1cncn1)C(=O)N(CC(C)(C)C#N)C)S(C)(=O)=O Cc1c(C(=O)NCC(C2CC2)NC(=O)CCC2CC2(F)F)ccc(Br)c1F C(C(=O)N1CC(CN(C(=O)CCCn2cncn2)C)C1)(C(C)C)SC c1(CCNC(C(CSCC)NC(c2cnccn2)=O)=O)ccc(F)cc1 CCCCC(C(=O)NCCNC(=O)Cn1nc(-c2cccs2)oc1=O)C(C)C c1(C(=O)NC(C)CCNC(=O)C(c2cncc(F)c2)C)ccc(S(N)(=O)=O)cc1 c1(C(=O)NC(c2c(OC)ccc(Br)c2)C)ccc2c(c1)COC2=O c12ccc(o1)C=CC(=O)N2.c1(C(=O)NCC2(C(=O)OC)CC2)cc(C2CC2)[nH]n1 c1(N2CCCC(CC)C2)nc2cccnc2c(=NC2CC(=O)N(C)C2)[nH]1 c1(C(=O)NCCN(C(=O)C2=CC(O)CCC2)CCC)cc(Cl)c(Cl)c(Cl)c1 N1(C(=O)NCC2(c3ccccc3)OCCO2)CCN(C(c2ccsc2)C#N)CC1 CC1(C)CC(N=c2nc(C(F)F)c3cc(F)ccc3[nH]2)CCO1 c1(C(=O)NC(C)C(=O)N(CC(C)(C)N)C)ccccc1Cl N1(C(CC2(COCC)CC2)=O)CCC2(CC1)CN(C(c1sc(CO)nc1C)=O)C2 C(CC(=O)NCC(C)C(C)(F)F)(C(F)(F)F)NC(c1c(OC)ccnc1)=O c1(CC)ccc(F)c(C(=O)NCCC2(CNC(c3nnc(S)n3C)=O)CC2)c1F c1(N2C(CN(CCC)C(C3CCCC4CC34)=O)CCC2)ncc([N+](=O)[O-])c(C)n1 C=CC(C)(O)CC(=O)NCCC1(OC)CN(C(=O)CC2CC3CCC2C3)C1 C1(C(=O)NC2CC(CNC(c3ccnc(F)c3O)=O)C(O)C2)CC(C2CC2)=NO1 c1(NC(C)=O)ccc(S(=O)(=O)NC(=O)NCCCc2ccc(F)c(F)c2)cc1 C(CCC)(CCCNC(CCC#CC)=O)NC(c1cccnc1C(F)F)=O C12(NC(C=COCC)=O)CCCCCC1N(C(c1cccc(F)c1C)=O)CC2 C1(C(=O)NC2CN(C(C(N3CCNC3=O)C)=O)C2)CCc2nc[nH]c2C1 N1(C(C=C(C)C(C)(C)C)=O)CC2(C1)CN(C(C1CC(C#N)C1)=O)CC2CO N1(Cc2ccc(C3(C)C(C)(C)C3)cc2)C(=O)CN(CCF)C1=O N1(C(C2C(C#C)C2(C)C)=O)CCN(C(=O)CNC(=O)Cc2ccco2)C(CC)C1 c1(C(N2C3CC(NC(Cc4n(C)ncc4)=O)C(C3)C2)=O)cnn2cccc(Cl)c12 c1(-c2cn(CCOCC(=O)N(c3ccncc3)C)nn2)cc(F)cc(F)c1 N1(C(CCN(C(=O)C(C2CCC2)OC)CC=C)=O)CCC(O)CC1 C1(CNC(c2c(C)cco2)=O)COCCN1C(=O)CC1CCCS1(=O)=O C(=O)(C(C)(C)C(O)C(C)C)N(C(CC)CNC(=O)CCCCCOC)C Cc1cc(C(=O)NC(C(=O)NCCC(F)F)C2CCCO2)oc1C Cc1cc(C(N2CCC(O)C(F)C2)=O)cc(C)n1.C12CCOC(C1)C(=O)N2 CN(C)S(=N)(=O)N1CCCC1C(=O)NC1CC2CCC1C(NC(=O)C(C)(C)C)C2 C1(NC(CCC(C)NC(C(COC)(C)OC)=O)=O)CC2(C1)CC21CC1 c1(NC(C)=O)cnc(O)c(C(N2CCOCC(NC(=O)C(C)CCN(C)C)C2)=O)c1 C1(CCC(=O)NC2C(C(=O)OC)CC2)CCCN(C(=O)CC2CC(SCC)C2)C1 c1(NC(N2CCC(Cc3cccc(F)c3)CC2)=O)cccc2cnccc12 c1(OC)ccccc1OCCC(=O)CN(C(=O)CCC1CC1)CCNCC(=O)OC C(CCN=c1nc(N2CCS(=O)(=O)CC2)c2c([nH]1)CCCCCC2)SCC.CC COn1cnc(C)c1C(=O)N(C1CN(C(=O)COc2ccccc2Cl)CC1F)C N1(C(CCCN(C)C(c2c[nH]c(=S)cn2)=O)=O)CCC2(CCOC2=O)C1 C1(C(N2C(CNC(=O)Cc3csc(S)n3)CC(F)C2)=O)CCCC2(CC2)C1 c1(CN=c2scc(CC(=O)Nc3cc(C)ns3)[nH]2)ccc2nc(Cl)sc2c1 C(CCN=C(NCC)NC(C1CC2CC1C2)C)Cc1ccc(OCCOC)cc1 C1(NC(C(C)(N(C)C(C2CCCC(O)C2)=O)C2CC2)=O)CC2CCCC(C1)C2 CC1CN(C(=O)CC2CCOC2)CC1CNC(c1ccc(-c2ccncc2)o1)=O c1(C(=O)NC2CCC(NC(C3CC(CC)OCC3)=O)C2)c2c(c[nH]c1=N)CCC2 c1(C(N2CCC(O)(c3cc[nH]n3)C2)=O)ccc(-c2nnc(S)o2)cc1 C1(C(N(CCCC#C)C)=O)(OC)CCN(C(C2CC(C(C)C)=NO2)=O)CC1 N1(C(C=Cc2ccc(C)o2)=O)CCC(C)N(C(=O)CCc2ccn(C)n2)CC1 Cc1cc(CC(=O)NC2CCN(C(c3ccco3)=O)CC2)n(-c2ccccn2)n1 C1(C(=O)NCC2OCCN(C(C)=O)C2)CC2CC(CN2)O1 C(=O)(C#CC1CCCCO1)NCC1CCN(C(Cn2ccc(C)cc2=O)=O)CC1 c1(C(CC(=O)NCCN(C(=O)Cc2ccns2)C)C)c[nH]c2ccccc12 N1(C(Cc2nc(C)oc2)=O)CCC(CNC(=O)C(c2ccccc2)N(C)C)CC1 Cc1cc(O)ncc1C(N1C2CCC1C(CNC(C1CC(=O)NC(=O)N1)=O)C2)=O C1(C(N2CCC(F)(C(=O)OC)C2)=O)CC2(CC(NCc3ccc(F)c(O)c3)C2)C1 c12ccccc1NC2=O.CC(C)C#CCNC(=O)C(c1cccnc1)N CCC(CC)CC(=O)N1CC(O)(C2CCCN2C(C23CCCC2(C(=O)OC)C3)=O)C1 C1(NC(=O)C2=CCCS2)CCN(C(c2cnc(O)c(Cl)c2)=O)CC1F c1(C(N2C(C(=O)NCCCC(F)(F)F)CC(F)C2)=O)cc(Cl)c2cc[nH]c2c1 N1(C(C(C(C)C)OCC)=O)CC2(CNC(=O)Cn3cccc3)CCC1CC2 Cc1cn(C)nc1C(=O)N(CCCNC(=O)C(C)CC1CCCC1)C(C)C C1(S(N)(=O)=O)(C(=O)NCC(C)Oc2ccccc2F)CCC1.C12CN(C1)CCN2 C1(C(=O)NC(c2ccc(F)cc2)C(C)C)CC2CC2N1C(=O)CN1CCNC1=O c1(N2CC(CNC(C(C)OCCOC)=O)N(C)CC2)cnc2ccccc2n1 Cn1c([N+](=O)[O-])cnc1C(N1CC2C(NC(C3CCC4CC3C4(C)C)=O)C2C1)=O C(=O)(C1c2c[nH]nc2CN1C(c1ncoc1C(C)C)=O)N(CCCC)C CC(C)(C)C(CC(F)(F)F)C(=O)OCCOC1CCCC1=O c1(C(=O)NCCCN(C(C(C)OCC=C)=O)CCO)cncc2nc(C)[nH]c12 N1(C(C2(CCCC)CC2)=O)CCCC(COC)(NC(=O)C=Cc2ccco2)C1 Fc1ccc(CC2CC3CCC(C2)N3CC2Cc3ccccc3S2)c(F)c1F N1(C(C(C)(C)C)=O)CCC(NC(c2cc(-c3ccco3)ccn2)=O)C(F)C1 N1(C(c2cn(CC)nn2)=O)CC(OC)CC(NC(c2cnn(CC(F)F)c2)=O)C1 c1(CCC(=O)NC(CNC(c2cn(C)nc2)=O)C2CC2)ccc(C(N)=O)cc1 C(=O)(CC(F)(F)F)NC(C)C(=O)N(C(C)CCNC(C1CC1CF)=O)C C=C=CCC(=O)NCCN(CCCN(C)C)C(c1cc(-c2ccn(C)n2)on1)=O C#CCC(CC#C)C(=O)NCC1CC(CNC(c2cc(N)cc(F)c2)=O)C1 c1(C2CNCC(C(C)C)(C3CCC3)N2)cccc(F)c1.CN=[N+]=[N-] c1(C(=O)NCCN(C(=O)C(c2ccc(Cl)cc2)(F)F)C)ccc(C(C)(F)F)cn1 CN1Cc2ccc(C(N3CCOCC(CNC(=O)Cc4cccs4)C3)=O)cc2C1 CC(CCNC(=O)CCSCc1ccccc1)CCNC(C1(O)CCOC1)=O c1(N)cccc2c1CCS2(=O)=O.c12ccc(cc1)N(C)CC2.N1(CC)CCOC1=O N1(C(C2(CC=C)CCCN2C(c2coc(COC)n2)=O)=O)CCC2(CCCO2)C1 n1(C(C(=O)NC(CNC(C=C(CC)C2CC2)=O)CC)C)ccnc1C CC(CS(C)(=O)=O)C(=O)NC1CCCC1CNC(=O)CC(C)(C)C C1(CC)CCCC1NC(=O)CNCC(C1CCC1)NC(c1sccc1OC)=O.C1CCC1 N1(C(C(C)SCC)=O)CCN(C(c2cn(CC)nn2)=O)C2CCCC12 Nc1ccc(C(=O)NCC2CCCN2C(c2coc(C(F)(F)F)n2)=O)nc1N c1(C2(C(=O)NC3C(C(=O)NCC4OCCN(C)C4)C3)CC2)ccc([N+](=O)[O-])cc1 C(=O)(C1=CCCOC1)N1CC(C)C(CCNC(=O)CCc2cccc(Cl)c2)C1 C=CCCC(F)(F)C(=O)N1C(=O)CC(CC2CC2)N(C=O)OCCC1 CC(C)CC(C)(C)C(=O)NC(C)C(C)C(=O)NC1(C)CCSCC1 C(=O)(CCC(=O)Nc1nccs1)NCC(C1CCC1)NC(c1ccc(CC)s1)=O CS(=O)(=O)c1ccc(NC(=O)Nc2nccc(NCCN3CCOC3=O)n2)cc1 N1(C(C)=O)CSCC1C(C(=O)Cc1ncc(C)s1)=O.C1(CN(C)C)(N)CC1 N1(C(c2nnn(C)n2)=O)CC(NC(c2nnc(Cl)cc2N)=O)C(C)(C)C1 CC1(C)CC(CNC(c2cc([N+](=O)[O-])n[nH]2)=O)CN1C(c1ccc(CF)cc1)=O C1(F)(CNC(COC(C)=O)=O)CCN(C(c2cnncc2C)=O)CC1 C1(CC#C)(C(=O)N(C2CSC2)C)CCN(C(c2ccncc2Cl)=O)C1 N1(CCNC(C(C2N(C(COCC)=O)CCC2)(C)C)=O)CCN(C)CC1 c1(OC)ncc(C(=O)NC2CCC2NC(C2CC(C(F)(F)F)C2)=O)c(C(F)F)n1 N1(C(COc2cc(C)on2)=O)CCCC(CCNC(=O)C(C)C(C)C)C1 CCC(CC)(CC)C(=O)NCC(C(=O)NC(c1csnn1)C)N(C)C C1(C(C)O)CCCN1CC.C(=O)NC(C(C(=O)O)c1ccsc1)=O Cc1cccc(C(F)C(=O)NCC(C)CN(C)C(c2c(C)nsc2C)=O)c1 CCC(F)(F)CC(=O)N(CCNC(=O)Cn1ccc(=O)cc1C)CCOC c1(-c2occ(CC(=O)Nc3nc(Cl)c(C(=O)O)s3)n2)c(F)cccc1F CC(C)CC(C)CC(=O)NCC1(F)CCN(C(C2(C)CC2(F)F)=O)C1 O=[N+]([O-])C1CCC2(CC1)NC(=O)N(CN1CC3(CCC3)C1CO)C2=O C1(NC(C2(COC)CC2)=O)CCOC2(CCN(C(=O)CNc3nccs3)CC2)C1 C1(NC(c2cnc(S)nc2)=O)C2CN(C(C3CC3F)=O)CC12 c1(NCC2CCC(CC)O2)cc(NCC(N2CCC(O)CC2)C)ncn1 Cc1ncc2n1CCN(C(=O)CCNC(C1CC(=O)CCO1)=O)C2 C1(C(N2CCCC(NC(c3cccnc3O)=O)CC2)=O)CCc2nc(O)[nH]c2C1 CCCC(F)C(=O)NC1CCCCC1NC(c1ccc(CCC#N)cc1)=O N1(C(CC(C=C)(C)O)=O)CCC2C(C1)NC(=O)CN2C(=O)Cc1ccc(C)o1 N1(C(c2c(C)csc2)=O)CCC(CCNC(=O)C2=CC(O)CCC2)C(F)(F)C1 CC(C)(CCNC(=O)C(=O)NCCSc1nnnn1CC(F)F)S(C)(=O)=O N1(C(CC(C=C)(C)O)=O)CC(CNC(c2ccoc2C2CC2)=O)OC2COCC12 c1(-c2c(OCC)ccc(CC)c2)ncnc2ccc(N(CC(C)O)C)cc12 C1(NC(c2c(OC)nccc2)=O)CC2CCC1N2C(=O)Cc1csc(C)n1 C12(C(=O)NCCC3(NC(c4n(C)c(O)nc4)=O)CCC3)OCCCC1C2(F)F C(CCN=c1ccnc(NCCNCCCN2CCOCC2)[nH]1)OC C1(CNC(CCOCCN(C)C)=O)CCC(C)(C)CN1C(C1CCNC1=O)=O Cc1cc(Br)ncc1NC(CC(N)=O)c1ccccc1 c1(-n2cc(CNC3(CC=C)CCCC3)nn2)cccc(F)c1 N1(C(C(C2CCCC2)OCC)=O)CCC2(C1)CN(C(=O)C#CC1(C)COC1)CCO2 C1(C(=O)NC(C(=O)NC(C(=O)NC)C(C)OC)C2CC2)CC(C)CC(=O)N1 Cc1nc2ccccc2c(C)c1C(N1CC(NC(=O)CC2CCC2)CC1C)=O c1(C(=O)NCC(CC(C)C)(C)NC(=O)COC(C)(C)C)occ2c1CCOC2 CC1CC(C(=O)NCC2=CCCN(C(=O)COc3ccccc3)C2)CC(C)C1 C1(O)(C(=O)NCC2C(CNC(c3c[nH]c(=N)s3)=O)C2)CCSCC1 C1(C(N2CCN(C(C3OCCN(C)C3)=O)CC2)=O)CCC(C2CCCO2)O1 c1(CC)conc1CC(=O)NC1(CNC(=O)C(C)Cc2cnco2)CCOC1 c1(C(N2CCC(OC)CC2)=O)cc(=NC(=O)c2cc(Cl)c(C)c(Cl)c2)[nH][nH]1 N1(C(c2ccc(=NC)[nH]c2)=O)CCN(C(=O)CCC2CCOC2)CC1C#N CN1CCC(O)(CNC(=O)C(Cc2cc[nH]n2)NC(=O)CC2CCN(C)C2=O)C1 CC(C)(C)C(CO)C(=O)NC1CCCC1NC(c1c(Br)cnn1C1CC1)=O c1(C(N2CCC3C(NC(=O)C(Cl)=CCl)C32)=O)cc2c[nH]cnc-2n1 C1(CC)CCN(C(=O)OC(C)(C)C)C1C.C12(CSC1)NC2 CC12CC(CNc3nccc(N4CCC(C)(CC#N)C4)n3)(CO1)C2 c1(OC)cc(C(=O)NCC2CCCC2NC(c2cc(C)ns2)=O)sn1 C1(NC(C(CCC)C)=O)CC(F)CN(C(c2cnn(CCN(C)C)c2)=O)C1 C1(CNC(C(CC#C)NC(=O)CC2CCCN2C)=O)CC2C=CC1CC2 CCCC(CCC)CC(=O)N(C1CN(C(=O)CSc2ccc(C)cc2)C1)CCO C=C1CCC(C(=O)NC(C(=O)NCc2cccc(Cl)c2)C2CC2)CC1 c1(C(N2CC(F)(C(=O)NCCC3CCC(C)O3)C2)=O)ncncc1N C(=O)(CCC1=NNC(=O)CC1)NCC1N(C(C(COC)NC(C)=O)=O)CCOC1 C(=O)(C(O)(C(F)(F)F)C1CC1)N1CCC(CNC(C=CCCC)=O)CC1 C1(NC(c2c(C(C)(C)C)ccs2)=O)CC(F)CN(C(c2ccc[nH]2)=O)C1 N1(C(=O)OC(C)(C)C)CCCC1C=CC(N1CCOCC1C(C)(C)C)=O c1(OC)cc(C(N2CC3CN(C(=O)CCS(C)(=O)=O)CC23)=O)ccc1O C1(C(=O)NCC(C)(C2CC2)NC(C(CC)=CCCC)=O)CN2CCCN1CC2 c1(C(=O)NCCCNC(C2C(C)CC(=O)N2)=O)cc2cc(Cl)c(Cl)cc2[nH]1 c1(C(C)NC(C)=O)cccc(C(=O)NCC(O)Cc2ccccc2C)c1 C1(C(=O)NCCC(C)N(C(C(CC)=CCCC)=O)C)CCCOC1C c1(C(N2C(CNC(C3C(=C)CCC3)=O)(CO)CCC2)=O)ccc(OC)c(Cl)c1F c1(C(C)(C)OC)nc(=NC2CCCCC2NC(c2cnn3c2CCC3)=O)s[nH]1 C(C)(CCNC(=O)Cc1cnoc1)NC(C1C(=C)C1)=O c1(SCC(N2C(C(C)NC(c3cnc(CC)[nH]3)=O)CCC2)=O)ccc(Br)cc1 C(CC)(C1CCCc2ccccc21)N(C(C(c1ccc(N)cn1)C)=O)C Cc1ccc(C(c2cccs2)NC(=O)CN2CCCC2)cc1 Cc1cc(C(N2CC(N(C)C(c3cnc(N(C)C)o3)=O)C(F)C2)=O)ccn1 O=C(C(O)CN1CCOCC1)NC1CC(CNC(=O)CC2C=CCCC2)C1 c1(OC)cc(CN=c2[nH]c(CN3C(CO)CCC3C)cs2)cc(O)c1O C1(C(N(CCCCC(=O)NCc2cnnn2C)C)=O)CCc2nn[nH]c2C1 N1(C(=O)CN(C2CCC2)C)CCC(CC(=O)NC(C(CC)C)CO)(COC)CC1 c1(C(=O)NC2(CNC(C3CCC3)=O)CCC2)ccc(Br)nc1.N(C)CCO C(=O)(C(C)(C)C1CCCCC1)N(CCNC(=O)CC1CCCO1)CC c1(C(N(CCOC)CCNC(=O)C2=NOC(C)C2)=O)cc2c(s1)CCCCC2 c1(C(=O)NC2C(NC(C(CCSCC)NC(C)=O)=O)C2)ccc(S(N)(=O)=O)o1 CC1(C)CN(C(=O)C(N2CCC(O)C23CCSC3)=O)c2ccccc2S1 C1(NC(CN(CCC#C)C)=O)CC2(CCCN(C(=O)CCCc3nccs3)C2)C1 c1(C(N2CC3C(CNC(CC(C)C4CC4)=O)(C3)C2)=O)cccc2ccnn12 c1(OC)ccc(C(N)CC(=O)NC(C)C(c2ccc(Cl)cc2)O)cc1 C=CCCCCC(=O)N1C2CCC1C(CNC(=O)CS(=O)(=O)N1CCCCC1)C2 c1(C(N2CC=CC(NC(CC(=O)N(C)C)=O)C2)=O)c(C(F)(F)F)cccc1Cl CC1(C)CCCN(C(c2cccnc2N)=O)C1CNC(C1(C#N)CCC1)=O N(C(=NCCCNS(C)(=O)=O)NC1CSC1)C(c1c(F)cccc1F)C c1(C(N2CCC(O)(CN(C(=O)C=C3CCC3)C)C2)=O)cnn2ccc(O)nc12 C1(CC)C(C(=O)N(CC(=O)NC(C)C)C)CCCN1C(=O)CCCCCCSC CC1(CCNC(=O)CSCC(F)(F)F)CCN(C(=O)CN2CCC2)C1 c1(CN2CCC(CNC(c3cccc(CC)c3)=O)C2)ccc([Si](C)(C)C)cc1 Cc1ccc(C=CC(=O)NC2(C3CCCCN3C(C3CC(F)(F)C3)=O)CC2)o1 Cc1cc(O)c(F)cc1NC(=O)C(O)C1CN(C(c2ccc3cc[nH]c3c2)=O)C1 C(=O)(C(C#N)C(C)C)NC1(CNC(C(=O)NCCCOC)=O)CC1 N1(C(c2c(CC)[nH]nc2Cl)=O)CCC(C)C(CNC(C2(O)CCOC2)=O)C1 c1(NC(C2CCCN(C(=O)CCc3cncc(Br)c3)C2)=O)ccnc(Br)c1F CCC(CC)C(=O)NC12CC(NC(c3cc(Cn4cccn4)on3)=O)(C1)C2 N#Cc1cc(C(=O)NC2CC3(C2)CC(NC(c2ccccc2I)=O)C3)ccc1F N12CCC(C1)n1cc(nn1)Cn1c(ncc1)C2=O.N1(Cc2ccno2)CCCC1 Cc1cc(Br)c(NC(C2CSCCN2Cc2ccc(O)c(F)c2F)=O)nc1C C(C(C)(C)C(=O)N(C1CCOC1)C)NC(C(CC)SC)=O c1(C(=O)NCC(C2CC2)NC(C=Cc2c(C)cccc2)=O)ncc(C#N)cc1Cl C(=O)(CC1OCc2ccccc21)N(CC(CC)NC(c1csc(Cl)n1)=O)C N1(C(C2C(C#C)C2)=O)CCC2(CCCC2NC(=O)C(O)(C2CC2)C2CC2)CC1 CC(C)C(C)(C)C(=O)NC1CCC1CNC(=O)CCCOC(C)(C)C N1(C(c2c(C)ocn2)=O)CCCN(C(C2CC3CCC(C2)C3)=O)CC1C c1(C(=O)NCCCC(CCC)NC(c2ccco2)=O)cnn2ccc(OC)cc12 CCC(C)CCCC(=O)N(CC(C)(C)CNC(=O)C(C(C)O)NC(N)=O)C c1(C(=O)NCCC(CNC(C2N(CC)CCCC2)=O)OC)ccc(C#N)c(C)c1 c1(C(=O)OC)ccccc1NC(C12CCC(CC1)C2)=O.C1CCCC1C c1(N2CC3(CCN(C(C4C(C)(C)CCC4)=O)C3)C2)ccc2c(n1)CCC2=O C#Cc1ccc(F)cc1C(=O)NC1(C)CC(NC(=O)CCc2cccn2C)C1 c1(NC(C2=CNN3C2=NC(=O)NCCC3)=O)nc2ccc(Cl)c(Cl)c2s1 c1(CC(=O)NCC(C)(CSC)N)ccc(C(F)(F)F)cc1.CCC(O)C=O C1(C(N2CCN(C(c3cccnc3)C)CC2)=O)CCCC2(C1)CC2(F)F N1(CC(=O)NCC(CNC(C2CC(C)(F)C2)=O)O)CCN(C2CC2)C1=O c1(N2CCC(NC(=O)C(F)C3CCC3)(CF)C2)ccncc1[N+](=O)[O-] Cc1nn(CC(F)F)cc1C(=O)NCC1(O)CCN(C(C2(Cl)CC23CCC3)=O)C1 CCCC(O)C(CO)NC(=O)C(CCC)NC(c1nccn1CC)=O CC1(C)CC(CNC(C2C(C)(C)C2(C)C)=O)N(C(C2NC(=O)OC2(C)C)=O)C1 c1(C(N(C)CC2CCN(C(c3ncoc3C3CC3)=O)C2)=O)cnc2ccoc2c1 CC(C)CC(C(=O)Nc1ncccc1N)ONC(c1ccccc1O)=O N1(C(C(=O)NC(=O)NC)C)CCOC(NC(C2CCN(C3CCSCC3)CC2)=O)C1 c1(OC)ccc(Br)c(CN2CCC(C3OCCO3)CC2)n1.C12CCCC1C(=O)N2 C1(C=C)(C(=O)NCC(CC=C)NC(c2nc(C)n(C)c2C)=O)CCOCC1 c1(OC)ccc(CO)cc1C(=O)NC(C1CCN(C(=O)Cc2ccsc2C)C1)C C1(O)(CCNC(C(C)N(C(C)=O)C)=O)CCCN(C(C2(CO)CCCC2)=O)C1 CC1CC(C(N2CC(CNC(=O)CCc3ccn(C)n3)(SC)C2)=O)CCS1(=O)=O N1(CCNC(C2C(C)(C)COC2)=O)CCCN(C(c2cc([N+](=O)[O-])c[nH]2)=O)CC1 c1(CC(N2CC(SC)C(NC(=O)CC3(CO)CC3)C2)=O)ccc(O)c(F)c1 c1(NC(C2CCCCCN2C(=O)Cn2cncn2)=O)cccc2[nH]ccc12 C1(N(C(c2ccn(CCCC)n2)=O)C)CN(C(c2cnc(CC)s2)=O)CC12CC2 N1(C(CCCCOC)=O)CCN(C(=O)C(=O)C2CC2)CC1CCO C1(N(CC#C)C(=O)C2CC2)CCN(C(C2(CN(C)C)CCC2)=O)CC1 C1(NC(C(C)n2ccnn2)=O)CCCN(C(=O)Cc2csc(S)n2)C1C c1(C(=O)NC2(CC(=O)N(CC)CC)CCC2)cc2ccccc2[nH]1 N1(C(C2C(C)CCC2)C(=O)NCc2ccco2)CCNC(=O)C1(C)C CCC(C(O)C(F)F)N1CCOCC1.C12(CC3(CCC3)C1)n1cc2nn1 C=CCC(C(=O)N1CCC(CNC(=O)CC2(O)CCC2)(OC)C1)c1ccccc1 C1(C(=O)OC)CC(OC)CN(C(c2nc[nH]c2C(C)(C)C)=O)C1.C1C(=O)N1 N1(C(c2c(C)ncc(N)c2)=O)CC2CC(NC(=O)C#CC(=O)N(C)C)CC2C1 O(C=C(C#N)C(=O)N(C1CCN(C(C2CC(C)C2(C)C)=O)CC1)CC)CC C#CC1CCCC(NC(C2CCCCCC2NC(c2ccc(NC)cn2)=O)=O)C1 C(=O)(C(F)CC(C)(C)C)NC1CC=C(C(=O)NCc2nn(C)c(=O)o2)C1 Cc1ccn2cnc(C(N3CCN(C(=O)CC4OCCCO4)C(CO)C3)=O)c2c1 C(=O)(CCCCCNC(c1ncccc1SC(C)C)=O)NCC(CC(C)C)N(C)C CC(C)CCC(C(=O)NCC(F)C(C)(C)O)NC(=O)C(O)Cn1cncn1 C1(C(=O)NC(C(=O)NCC2C(=C)C2)CCOCCO)CC2(C1)CC(C)C2 c1(CNc2c(Nc3cc(F)cc(Cl)c3)ccc(Cl)c2)c[nH]c2cc(Cl)cc(Br)c12 C(=O)(CC(C1CC1)NC(=O)CC1CC(C)=NO1)NCCOCC(=O)NC C1(C(=O)NCCC2N(C(Cc3cc(OC)no3)=O)CCSC2)CC(C)OC(C)C1 C1(CNC(c2cccc(NC(C)=O)n2)=O)CC2(CO1)CN(C(c1cnsc1)=O)C2 CC1(CNC(c2cnc(NC3CC3)s2)=O)CCN(C(=O)CCc2ccccc2)C1 Cc1cnc(C(=O)N(C2CCN(C(=O)COc3cccnc3Cl)C2)C)cn1 c1(C(N2CCN(C(CCC)=O)C(CCOC)C2)=O)ccc2c(c1)NC(=O)C(C)O2 c1(C(=O)NCCN(C(C(CC)COC)=O)C2CC2)cnn2c1OCC1(CC1)C2 C1(C(=O)NCC2CC(F)(F)CN2C(=O)CCOC2CC2)COCCC1(F)F N1(C(c2ncc(OC)cn2)=O)CC(NC(C2NC(=O)OC2C)=O)C(C)(C)C1 N1(C(c2ccc(C)[nH]2)=O)CCCC12CCN(C(=O)CCc1cocn1)C2 C(C(C)(C)CC(=O)N(C(CO)C(C)C)C)NC(C1C(=C)C1)=O N1(C(c2n(C)nc(O)c2)=O)CC2(C)CN(C(c3c(C(F)F)cnn3C)=O)CC2(C)C1 C1(C(=O)NC2(C)C(NC(c3cc(C)on3)=O)CCC2)CCCC12CCC2 Cc1nn2c(C(=O)NCC(C)(C)CNC(c3ccc(C)nc3C)=O)c(C)nc2s1 CCC(CNC(=O)Cc1ccc(C)cc1)C(=O)NC1(C(F)F)CCCC1 N1(CCCC2(c3n(-c4c(C)cccc4)nnn3)CC3(CC3)C2)CC(=O)N(C)C1=O C1(C(C)NC(c2cnc(C(C)C)[nH]2)=O)CCCN(C(=O)C(C)(C)OC(C)C)C1 N1(C(c2cc(C)no2)=O)CC2(CCC2)CC1C(=O)NC(c1cnn(C)c1)CO c1(C(=O)NCC2CCC(CNC(C(C)OCC=C)=O)CC2)n[nH]c2ccccc12 C1(NC(C(COC)CC(C)C)=O)CCN(C(c2n[nH]cc2Cl)=O)CCC1(F)F Cc1c(C(=O)NC(CNC(=O)C(C)(C)C2CCCO2)C2CCC2)cnn1CCO N1(C(CCCC(CC)CC)=O)CCC2(C=C(C(=O)NCCn3cnccc3=O)C2)C1 N1(C(c2c(C)ocn2)=O)CCOC(C(N2CCN(C(C)C)CC2C)=O)CC1 c1(C(=O)NCCC2N(C(CC(C)C(F)F)=O)CCSC2)cccc2nsnc12 N1(C(c2ccnc3cc[nH]c23)=O)CCC2CN(C(C3(C(F)(F)F)CC3)=O)CC2CC1 C1(NC(C2(NC(=O)OC)CCCC2)=O)CN(C(=O)CCC(C)(C)OC)CC12CC2 c1(C(=O)NC(C)CCNC(=O)C(c2cccc(F)c2)O)cccc(O)c1F Cc1ccc(Br)c(C(=O)NCC2N(C(=O)C3CC3)CCC2(C)C)c1 S(=O)(=O)(c1ccc(N2CCC(NC3CCCCC3)CC2)nc1)N(CC(C)CO)C C(c1ccc(O)cc1)=CC(N1C(C(C)NC(c2c(C)scc2)=O)CCCC1)=O c1(C(=O)NCC2N(C(C3N=C(C)SC3)=O)CC(F)C2)ccc2ncsc2c1 c1(OC)ncc(C)c(C(=O)NC(C)C(C)NC(=O)CCc2ccc(F)c(F)c2)c1Cl c1(C(=O)NC2CC3(C2)CC3C(=O)NCC2CC(F)(F)CO2)occ2c1CCC2 c1(C(=O)Nc2cccc(C(C)C)c2O)ccc2c(c1)CCNC2 C1(C(=O)OC)C(C)CCN1c1nnc(C[N+](=O)[O-])n1CC(c1nnc(C)n1C)OC CC(C#N)CCC(=O)N1CCC2NCC2C1 CCCCC(O)C(=O)N1C(CC(N2CCCCC2CCOC)=O)C2CCCC12 CN1C(=O)C(NC(=O)NC2OC3CCC2CC3)c2cc(Br)ccc21 C=CCC(CC)C(=O)NCCC(C(C)C)NC(C1(OC)CCOC1)=O c1(C(=O)NCC(C2CC2)NC(C=CC(C)(C)SC)=O)cnn2c1CN(C)CC2 C1(NC(CC2N(C(c3ccc(C(C)=O)o3)=O)CC2)=O)Cc2ccccc2C1OC C1(NC(=O)C(F)CC2CCOC2)CCN(C(=O)CSCc2ccccn2)CC1 C=CCCC(F)(F)C(=O)N1CC2CCC2(CNC(C2CC(C)(C)CN2C)=O)C1 C(CC(O)C(=O)NCCN(C(C1CCN(c2cnn(C)c2)C1=O)=O)C(C)C)SC C1(C(=O)NCC(=O)NC(C(=O)NCCN(C)C)(C)CO)CCCCN1C C1(N(C(CNC(=O)C(c2cnccc2C)CC=C)=O)CC(C)C)CCS(=O)(=O)C1 C12(CNC(COC(C)C)=O)CC(C1)C(NC(c1ccc(O)nc1)=O)CO2 c1(Oc2ccc(C(=O)CN3CCCC3)cc2)cc(F)c(F)c(F)c1 C(CC)(CC)(CCC(=O)OC)NC(C=CC)=O.C1=CCNC1=O c1(C(N2CCC(O)(c3cn(CC(=O)NCC)nn3)C2)=O)cc(F)cc2c1CCC2 C(C)(CCC(=O)NCC1(CN=[N+]=[N-])CC1)NC(c1ccc(CC)nc1)=O Cc1nc(NCC(C)(C(C)C)NC(=O)CCNC2CC2)c(C)c(O)n1 c1(NC(c2c(-n3ccc(C)n3)cccc2)=O)nc(C)ccc1F C1(CC(=O)N(C2CCN(C3CCCCC3)C2)CC)C2CN(CCNCCO)CC12 C1(N(C(CN(CCC)C(=O)C2CC2)=O)C)CC(C(=O)OCC(C)C)C1 C(CNC(=O)Cc1cc[nH]n1)(C(C)(C)C)NC(c1cc(COC)[nH]n1)=O c1(C(=O)NCC2CC(F)(F)CN2C(=O)C2CC2)ccc(F)c(Cl)c1F C=CC(CC)CC(=O)N1CCC(N=[N+]=[N-])(C(=O)NC(C)CN(CCCC)C)C1 N1(C(CCCC#N)=O)CCCC(CC(=O)NCC2CC3C=CC2C3)CC1 c1(OC)csc(C(N2CCN(C(=O)CC3CCCC3)CC2)=O)c1OC C(=O)(C(C)CC(=O)N1CCC(F)(C(=O)NCCN2CCCC2)CC1)OC c1(C(=O)NC2CC(F)(CNC(C3(F)C(C)(C)C3(C)C)=O)C2)ccc2cccnn12 c1(OC)cc(C#N)ccc1NC(c1cc(F)cnc1C)=O C1(NC(C(c2c[nH]c3ccccc23)C)=O)CC2CCC1N(C(C1(C)CC1)=O)C2 c1(C(N2CC(C)N(C(=O)CN(C)C3CC3)CCC2)=O)cc([N+](=O)[O-])cnc1O c1(C(=O)OC)nc(=NCC2(NC(C3CC(C)CO3)=O)CCSC2)cc(C(C)(C)C)[nH]1 Cc1oc(Cl)nc1C(=O)N(CC(N1CCCC(C)C1)=O)CC(C)C N(C1CCOc2ccccc21)CC(=O)OCCc1ccc(Br)cn1 c1(C(=O)NCC(CC(=O)OC)C2CC2)c(C)c(O)nc2ccccc12 Cc1ccc(SC(c2ccccc2)Cc2nc(C)nn2CC2CCOCC2)cc1 C1(C(=O)NCCCCC)CC2CC(C1)N(CC1(c3ccccc3)COC1)C2 C(=O)(C(C)N(OC)C(=O)C1CN(C(=O)CC2CCCCC2)CC1(F)F)OC C(c1cncc(OC)c1)=CC(=O)NCC1CCC(NC(c2ccc(COC)[nH]2)=O)C1 C1(NC(C=CC(C)(C)C)=O)CC(F)CN(C(C2CC3C=CC2C3)=O)C1 c1(NC(CC2CCN(C(C3CC(C)(CC)C3)=O)C2)=O)cc2c(cn1)NC(=O)CO2 c1(CC(=O)N(C)CCNC(c2cc(Br)co2)=O)cnn(C(C)(C)C)c1 N1(C(C(=O)N(C2CCN(c3ccc(NC=O)cc3)C2)C)=O)CC2C=C(Br)C2C1 c1(OC)ccc(CC(=O)NCc2ccc(-c3ccccn3)cc2)nc1 Cc1cc(C(F)F)nn1CC(=O)NC1CCN(C(c2ncc(F)cn2)=O)C1 C(=O)(C1=NOC2(CCOC2)C1)NCC(N1CCN(C(C(CO)OC)=O)CC1)C c1(CC)c(C(=O)NC(CNC(=O)CC2CC(OC)C2)CO)[nH]c(C)c1C(C)=O C1(c2ccc(C)cc2C)CN(N2CCC(C3=NOCC3)C2)CCO1 Cc1c(C=CC(N2CCC(CNC(c3sccc3Br)=O)C2(C)C)=O)cnn1C C1(C(C)C)CCC(C(=O)NC2CC(CNC(c3cn(CCCF)nn3)=O)C2)CC1 C12(CCNC(c3c(C)ccnn3)=O)CCC1CN(C(=O)C=C1CCC(C)CC1)C2 c1(C(N2C(C(C)(C)CNC(c3ccc(Cl)o3)=O)CCCC2)=O)cc2sccc2s1 CC1=NOC(C)(C(c2nnnn2CS)NCC2CC2)C1.C1(C2CCC2)CCCO1 C1(F)(CNC(C2CCOC2)=O)CCCN(C(c2cnn3c2OCC3)=O)CC1 Cc1cccc(C(N2CCSCC2C(=O)NCC(C2CC2)C2CC2)=O)c1 Cc1[nH]nc(C(C)C)c1C(N1CCC(C)(CNC(c2cc(C(N)=O)c[nH]2)=O)C1)=O OCCC(N=c1cc(NCC(F)(F)C(F)F)nc(C(F)(F)F)[nH]1)c1cccnc1 Nc1ccc(Br)cc1C(=O)NC1CC(F)(CNC(=O)Cc2ccoc2)C1 c1(NCC2C3(CC(NC(=O)OC(C)(C)C)C3)C2)nnc2ccccc2n1 N1(C(C(COC)(F)F)=O)CCOCC(NC(c2ccc(NC(C)C)cc2)=O)C1 N1(C(C(CCNC(c2cc(F)c[nH]2)=O)OC)=O)CC(F)(F)C(F)(F)C1 C1(NC(CCN(C)CCO)=O)CN(C(=O)C2=CCCCO2)CCC12CCC2 N(C(=NCCC)NCCC(C)(O)c1ccccc1)CC1C(=C)C1 CC1(CNC(=O)CN2CCCOC2=O)CCCN1C(=O)C=C1CCC1 C1(NC(=O)CCCN2CCCC2)CC2(CCCCN2C(c2ccc(Cl)nc2)=O)C1 CCC(O)C(C)C(=O)N1CCC(C)(CNC(C23CC2CCC3(F)F)=O)CC1 CC(C)C(C(=O)N1CCC=C(Cl)C1)C(C)NC(=O)CN1CC(C)(C)C1 CC(C)C(C)(O)C(=O)NCCCCCOCCn1cc(-c2nc(C(=O)O)co2)nn1 Cc1cc(COC(C2(O)CCC2C)=O)ccc1C#N C(=O)(CS(=O)(=O)CC(C)C)C(C(CC=C)CC1CCCC1)=O.ONC N1(C(CCN(C)CCO)=O)CC(F)CC1CN(C(=O)CN1C(=O)CNC1=O)C C12(C(=O)NCC3C4CN(C(C5C(CC(C)C)C5)=O)CC43)CCCCC1NC(=O)C2 c1(CSCC(=O)NCC(CNC(C2(CC)CCCC2)=O)O)cccc(C)c1 CN1C(=O)CCC1C(N1CSCC1C(=O)NCC(O)CN1CCCC1)=O Cc1ccc(O)cc1NC(C1(CNC(=O)C=CC(F)(F)F)CCCC1)=O c12ccc3ncccc3c1C(C)c1noc(n1)-c1ccc-2s1.C#Cc1ncc[nH]1 Cc1ccc(C)n1CC(=O)NCC(C)CN1CCCC1.C1CCC(=O)NC12CC2 C(=O)(C(F)(F)CCN(C)C)NC(CC)(C)CNC(=O)CCCOC1CCOCC1 C(=O)(C1=NOC(C)C1C)NC(C(=O)NCC(CC)(C)OC)CCOCCO C1(C(=O)NCCCC(=O)N(C)CC2(OC)CCCC2)(OC)CCCCC1 C1(C(N2C3C(NC(c4scc(C(=O)OC)c4)=O)C(C3)C2)=O)CC2(C1)CC1(CC1)C2 c1(SC)ccc(Cl)c(C(=O)NC2CC(F)(CNC(=O)CC3CCCS3(=O)=O)C2)c1 CCC(C)C(O)C(C)C(=O)NCC1CCC(C(N2CC(F)(CC)C2)=O)CC1 N1(C(C(c2ccccc2)C)=O)CC=CC1CNC(c1cccnn1)=O C(CNC(CCC(N)=O)=O)(CC(=O)NC1CC1)OCCOCCCO c1(C(C)C(=O)NCC2C(O)C(O)CN2C(C2CC2F)=O)cc(Br)ccc1F C1(NC(c2cnc(C)s2)=O)CCN(C(c2cc(C#N)co2)=O)C1(C)C CN1CCCC(O)(CC(=O)NCCCCN(CCCNC(=O)CCCF)C)C1 CCCCCC(O)C(=O)NC(C)(C)C(=O)NC1CCN(S(C)(=O)=O)C1 CCC(CC)(C(=O)N1CC2CCC(NC(c3cnn(C)c3OC)=O)C2C1)C(C)C C(=O)(C1=CCCOC1)NC1C(CNC(Cc2ccc(OC)nc2)=O)CC1 C1(C(N(CC(CNC(CC(CC)SC)=O)(C)C)C)=O)CCC(F)(F)CO1 N1(C(=O)OC(C)(C)C)CCC(NC(c2ccc(F)c(F)c2)=O)C(F)(F)CC1 c1(CC(=O)OCC)cccc(NNC(=O)Nc2ncn(CCOC)n2)c1 CC(C)C(C)(O)C(=O)NC1CCN(C(C2CC(=O)N(CCF)C2)=O)CC1 CCCCC(F)C(=O)N1C(C(=O)NCC2(C(=O)NC)CC2)CC1C CCC(CC)CC(=O)N1CCC(NC(=O)C(C(C)C)NS(C)(=O)=O)CC1 C(=O)(C1CCc2c(Cl)cccc21)N1CCCC(C)(NC(CC(C)C2CC2)=O)C1 N1(C(c2cccc(C(=O)NC)c2)C(=O)Nc2ccccc2)CCS(=O)C(C)(C)C1 C12(C(N3CC(=C)C3)=O)CC(CN(C(C3CCCSC3C)=O)C1)C2 N1(C(CC2(C=C)CCC2)=O)C2CCC1CN(C(c1cc(C3CC3)n(C)n1)=O)CC2 C1(=O)C(C)(C)CN1C.c1(OC)cc(NC(=O)CNC(=O)CCOC(C)=O)on1 C(=O)(C(CC)CCCC)N1CCC(CNC(CC=CC)=O)(CO)CC1 N#Cc1cccc(CC)c1.c1(C(C)NC(C(CCO)C2CCCC2)=O)csc(C=O)c1 C(=O)(C(C)S(N)(=O)=O)NCC1N(C(CN(C(C)C)C)=O)CCCC1 CN1CCN(C2CCCC2C(=O)Nc2cnn(Cc3ccccc3)c2)CC1 Cc1nc2c(N3CCCC4(NC(C5CC5(Cl)Cl)=O)CC4C3)ncnc2s1 C(=O)(CCCCNC(=O)C(F)C1CCOC1)NCC1(SC)CC(O)C1 C1(c2nnc(C)o2)CCCN(Cc2ccccc2-c2nnc(C3CC3)o2)C1 c1(OC)csc(C(=O)N(CCCCNC(c2cc(CC3CCC3)c[nH]2)=O)C)c1 c1(OC)cc(Cl)c(C(=O)OC)cn1.c1ccc(Cl)cc1C=O.C12CN(C1)NC(=O)C2 CC(C)C#CC(=O)NCC1CN(C(c2ccc(C(F)(F)F)cc2)=O)CCO1 S(=O)(=O)(c1c(Cl)cccc1Cl)N1CC(NC(c2ccc(F)c3[nH]ccc23)=O)C1 c1(OC)cccc(COC(C)C(=O)N(CC(C)NC(c2cnccc2Cl)=O)C)c1 c1(C(CC)(C)C)ccc(C(=O)NC2CN(C(=O)CN(C)CCO)C3CC23)cc1 C1(C(=O)NC2CCC(NC(C(c3cccnc3)OC)=O)CC2)OCC2COCCC12 C#CCC(CC(=O)NC1CCOC(=O)CC1)NC(=O)CC1CCC(C)(C)O1 N1(C(C2CN(CCC)C(=O)C2)=O)CCCC(C)(CNC(c2cnc(C)[nH]2)=O)C1 C1(C(=O)NCC2C(NC(CCc3scc(C)n3)=O)C2)CC2C=CC1C21CC1 c1(C(N(C(CNC(C(n2cnc(C#N)n2)C)=O)C)C)=O)ccc(F)c(CO)c1 N1(C(c2c(CC)occ2)=O)CCC(CC)(NC(C2CCNC2=O)=O)CC1 C(=O)(C(CC(C)C)N(C)C(c1cc(C(N)=O)co1)=O)NCC(C#C)C(C)C Cc1ccn(CC(N2CCN(C3CN(C(C4COC(=O)C4)=O)C3)CC2)=O)c(=O)c1 N1(C(CN(CCC)C)=O)Cc2ccccc2C(CNC(=O)C(C)(O)C(C)C)C1 C(=O)(CCCC(C)(F)F)NC(CNC(c1n(OC)cnc1C)=O)CC(F)(F)F Cc1nc(C=CCS(=O)(=O)Oc2ccccc2)[nH]c1C N1(C(C(C)OCCC#C)=O)CCCC(C)(CNC(=O)Cn2ccnc(O)c2=O)C1 C1(CNC(C=Cc2c(C)ncs2)=O)C2CCCC1N(C(=O)C(C)c1ccsc1)C2 N#Cc1ccc(=NCC(=O)NC(CNC(=O)CCC(F)(F)F)CO)[nH]c1 C=CCCCCCCCC(=O)NC(C)C(C(C)C)NC(c1ccc(C)c(N)c1)=O C1(C(=O)NCC2CC2NC(c2ccco2)=O)(NC(CSCCCC)=O)CCC1 c1(N2C(C)CC(CNC(C3(COCC)CC3)=O)C2)ncnc(Cl)c1[N+](=O)[O-] C(C1(C)CCOCC1)=CC(=O)NC(C)CC1CN(C(c2nnn(C)n2)=O)C1 N1(C(C(CC)NC(C)=O)=O)CC(C)(C)CC1CNC(c1cn(C)nc1C1CC1)=O c1(C(N2CC(C(N3CCCC(C)(Cc4cccs4)C3)=O)C2)=O)ccnc2[nH]cnc12 Cc1ccc(C(N2CC3(NC(c4scnc4Cl)=O)CC2C3)=O)c(F)c1F CC1CN(C(=O)CC2CCCC2O)CC1CC(=O)N(C)Cc1cn[nH]c1 c1(NC(C2CCN(C(=O)C=CC3CCOC3)C2)=O)cnccc1CO C1(C2CN(C(c3cccc(C)c3N)=O)C2)(NC(C2CC(CC)C2)=O)CC1 C(CCCCC(=O)N1CC2CC(NC(c3cnn(C4CC4)c3Cl)=O)C1C2)SC CC1=C(C)CC(C(N2CCC(CO)(NC(C3C(C)(C)C3(C)C)=O)C2)=O)CC1 C1(CC)CC(NC(=O)C(C)C)CCN1C(=O)OC(C)(C)C.N1(C(=O)N)CCCCC1 C1(OC)CCCN(C(c2cccc(CCOc3nc(C)sc3C)c2)=O)C1C C(=O)(C1=C(Cl)CCC(C)C1)NC(COC)CNC(c1c(C)ncn1O)=O C1(NC(c2cn(C)nc2Br)=O)CC2CC1N(C(C1COCCOC1)=O)C2 c1(C(N2C(CNC(C=Cc3occ(C)n3)=O)CC2)=O)cc2c(Cl)cccc2s1 C1(NC(c2cc(N)cc(O)c2)=O)CN(C(=O)CCCCO)CC2(CCC2)C1 C#CCC(C)(C(=O)NCC1(CC)CCOC1)NC(C)=O Cc1ccc(F)c(C(=O)NCC(C)NC(=O)CSc2cccs2)c1F c1(OC)cc(C(N2CCCN(C(=O)CCC3CCCCN3C)CC2)=O)cc(C)n1 N1(C(C2C(C=C)C2)=O)CCN(c2cccc(NC(=O)C(C)N(CC)CC)c2)CC1 C(=O)(C(C)C(=O)NC(C)CCCNC(=O)CCN(C1CCCCC1)C)OC Cc1cc(N2CCCC2C(=O)NCCCOc2ccccc2)nc(C)n1 c1(OC)nccnc1C(=O)NCC1CCC1NC(=O)CSc1ccccc1O N1(CCCC)CCCC1C(N1CC(C(C)NC(=O)C(C)SC2CCCC2)C1)=O C1(CC=C)(NC(=O)C(C)SC(F)(F)F)CCCN(C(=O)C(C(C)C)SC)C1 C(CC(=O)NCC1CN(C(c2cc(C)n(C(C)C)c2C)=O)C1)(C(N)=O)NC(C)=O Cn1nc(I)cc1N1CCC(C(=O)OCc2nc(-c3cncc(N)c3)no2)CC1 N1(C(C(C)(C)NC(C(C)Nc2ccc(C)cc2)=O)=O)CCOCC(C)(C)C1 CCN(C(C)C)N(Cc1cnn2c1CC(C(C)(C)C)CC2)C1CC1 c1(C(=O)NC2CC(CNC(C(c3cccc(F)c3)C)=O)C2)ccc(C(F)F)cn1 C1(C(N2CCCC(C(=O)Nc3nc(C4CC4)n[nH]3)C2)=O)CCC2(CC2)C1 N1(C(C(c2cnn(C)c2)C)=O)CCOCC(C)(CNC(=O)CN(C)CCO)C1 N1(C(C(C)OCCC=C)=O)CC(CNC(=O)C(C)SC(F)(F)F)(OC)C1 c1(CNC(c2c(C)c[nH]c2)=O)nc(C(N2CC3CC2CS3)=O)c(C)o1 N1(C(CC2(N(C(C(CC=CCC)C)=O)C)CC2)=O)CC(C)=CC(C)C1 C1(c2n(CC=C)nnn2)(Nc2cccc(NC(C)=O)c2)CCN2CCCCC12 CCCC(C)(O)CC(=O)NC1CC(N(c2ccccc2)C(=O)CNC=O)C1 C(=O)(CC(C)P(C)(C)=O)NCC(CCNC(c1c(OC)cnc(Cl)c1)=O)OC C#CCCCC(=O)N1CC(NC(c2cc(C)n(C)n2)=O)C(F)C1 N1(C(c2c(C)ccc(C)n2)=O)CC(NC(=O)CC2CCC2(C)C)C2(CCC2)C1 C1(NC(c2c(C)csc2)=O)CCC2(CC1)CN(C(c1cnnn1C)=O)C2 N1(C(C2C(C)CCC2)=O)CC=C(C(=O)NCc2ncsn2)C1 Cc1ccc(CC(=O)NCCC(C)N(C)C(c2ccc(CO)c(F)c2)=O)cc1Cl N1(C(CCC2(C)CC2)=O)C2CCCC1CC(NC(C1CCCCC1C(N)=O)=O)C2 C1(CC=C)(NC(CCC(=O)OCC)=O)CCN(C(=O)CCCN(C)C(C)=O)C1 C1(C)(C(=O)NC2CN(C(C(CCC)(C)O)=O)CC2C)Cc2ccccc2C1 Cc1cc(C(=O)NCC2(C)CCC(NC(=O)C(C)C(C)(F)F)CC2)cc(C)c1C c1(C(N2CCC(O)(CCNC(C3CCC3(F)F)=O)C2)=O)nnn2ccccc12 C1(C(=O)NCCC2(NC(=O)C3=CCCCO3)CCC2)CCn2c(O)nnc2C1 C#Cc1ccc(C(=O)NC(CN(C(=O)CC2CNC(=O)C2)CC)CC)cc1F c1(C(N2CCC(NC(C3(Sc4ccsc4)CC3)=O)C2)=O)ccc2c(c1)CCO2 N1(C(c2ccc(NC)cc2)=O)CCC2(NC(c3cnc[nH]c3=N)=O)CC2C1 C1(NC(C(=O)NC(C)C)=O)(NS(C)(=O)=O)CCCCC1.C12OCCC1C(=O)NC2 c1(C(=O)NC2(C(=O)NCC)CC2)cnn2c(C)cc(C)nc12 C1(C)(NC(CN(CCC)C(c2ccncc2O)=O)=O)CCOC1C CC1(C(=O)Nc2ccc(CCN=c3[nH]nc(O)s3)cc2)CC2CCC(C1)S2 C(=O)(C(CCC(C)C)NC(N)=O)NCc1cn(CC2(OCC)CCCC2)nn1 c1(OCCC)cccc(C(=O)NCC(C)(C)CN(C(C2CC(CF)C2)=O)CC)c1 c1(NC(C)=O)cccc(C(=O)NC2CN(C(c3cc[nH]n3)=O)CCC2F)c1C c1(C(N(CC2N(C(CC(=C=C)C)=O)CCC2)CC)=O)ncc(F)c2ccccc12 c1(CC(=O)NC(C(C)NC(C=C2CCC(C)C2)=O)(C)C)n[nH]c2ccccc12 CC1C(NC(c2csc(C(F)F)n2)=O)CCN1C(C1CC(F)(CO)C1)=O C1(N(C(C2CC(NC(c3nc(C)sc3)=O)(CO)C2)=O)C)CCCC1(C)O C1(N(C(N(C2CN(C(c3ccccc3)=O)C2)C)=O)C2CC2)CCCC1(C)O N1(C(CCSCC)=O)CCC(C(=O)NCCCc2cnn[nH]2)C1CC C(=O)(C1CCc2scnc21)N1CCC(CCNC(C(C=C)O)=O)C1 CCC(C)CC(C)C(=O)N(CCCNC(c1ccc([N+](=O)[O-])cc1)=O)C N1(C(C(CN(C)C)N(C)C)=O)CC(=O)NCC1C(N1CCSC2(CCC2)C1)=O C1(NC(c2ccc(C)cc2N)=O)CN(C(=O)CSCC2CCCO2)C2(CCC2)C1 c1(CC(=O)NC(CCNC(C(CC2CC2)OC)=O)C)c(C)nc(C)nc1O c1(C(N(C)CC2OCCN(C(C(CCOC)C)=O)C2)=O)cccc(C#CCO)c1 N1(C(C2CC(Cl)(Cl)C2)=O)CCC2CN(C(C34CCCC3C4)=O)C2C1 c1(C(N2CCC(C)C2C(=O)NC2CCCC2)=O)cc(=O)n(C)cn1 CCC(O)C(C)(C)C(=O)N1CC2(CC(NC(=O)C(C)(C)COC(F)F)C2)C1 Cc1cc(C(=O)NC2CC2CNC(C2(CO)CCOCC2)=O)cnc1C(F)(F)F C1(CNC(c2ccccc2)=O)CC2CCC1N2C(C12COC(CF)(C1)C2)=O C(=O)(C#CC1CCCCO1)N1C(CNC(c2ccc(OC(C)C)nn2)=O)CCC1 C1(C(=O)NCC(C)(C2CC2)NC(c2cnccc2Cl)=O)CC2C=CC1CCC2 c1(C(=O)OC)ccc(C(N2CCC(N)CC2C)=O)c(F)c1 C1(C(=O)NC(C2(O)CCCCC2)C)(NC(c2cc(O)nn2C)=O)CCN(C)C1 c1(C(=O)NCC2OCCCN(C(C(CC(=C)C)C)=O)C2)cc(C#N)ccc1O CC(C)(C)CC(O)CC(=O)NCC1OCCC1C(N1CCC(CO)C1)=O Fc1ccccc1-n1nnnc1NC1(CC2CC=CC2)CC1.C1(C)CC1 Cc1cn(CC(O)C(N2CCC(CCN(C3CCC3)C)CC2)=O)c2ccccc12 S(=O)(=O)(c1ccc(NC2CCCCCC2F)c(Br)c1)N1CC(CC)OCCC1 N1(C(CC(C)NC(C2CC(O)C2)=O)=O)CC2(C)CC1CCO2 c1(CC(=O)NCC2C(C(=O)NC3C(C#C)C3)C2)cc(OC)cc(OC)c1 C(=O)(C1=CCCOC1)N(CCOC)CCNC(C1CC(C)CO1)=O N1(C(c2ccc(OCC)cc2)=O)CC(NC(c2coc(N(C)C)n2)=O)CC1(C)C CC(O)(CNC(c1cn(C2CC2)nn1)=O)CNC(c1cn(C2CCOC2)cn1)=O C1(C)(NC(CCN2CCN(C)CC2)=O)CCN(C(C2COCCO2)=O)CC1 n1(CC(=O)NCC2CN(C(C(F)=CCC)=O)CC23CC3)nc2c(n1)CCCC2 CC1(C)CC(NC(=O)C(F)=CC2CC2)CN(C(=O)C(=O)Nc2ccc(F)cc2)C1 c1(-c2cn(C(C)CNC(=O)CO)nn2)ccc(C(C)(C)C)cc1 C1(C(=O)Nc2ccc(C)cc2O)C2C(CN1Cc1cc(O)cc(O)c1)C2(C)C c1(N2CC(CCNCC(O)CC(=O)OC)(OC)C2)ccc([N+](=O)[O-])cc1C#N CC1CCCC1(C(N1CCC1(C)C)=O)NC(c1ccsc1C#N)=O C(C(C)(C(C)C)NC(c1cncc(C(C)(C)C)c1)=O)NC1CCN(C(C)=O)C1 c1(NC(=O)NC(C)CN2CC3CCC2C3)nnc(S(=O)(=O)NCCNC(C)=O)s1 CCC(CC)CCCC(=O)Nc1ccc(C(=O)NC(C)C(C)(C)COC(C)=O)nc1 c1(C(=O)NCC(CC)(CC)NC(C(C)SCC)=O)ccc2nc(C)n(C)c2c1 c1(C(C(=O)NCCCOC)N(c2cc(C)ccc2F)C)cc(OC)cc(Br)c1 N1(C(Cc2nnc(C)o2)=O)CC(CC(=O)NC2CCOC2)C2(CC2)C1 CC1(C)CCN(C(c2cc(-c3cccc(Br)c3F)no2)=O)CCS1 c1(C(N2CCN(C(C(CCC)C)=O)C(CC)C2)=O)cc(O)c(O)cc1O Cc1ccc(CC(=O)NCCCN(C(=O)C(C)CC2CCC2)CCO)cc1 c1(C(N(C(C)CNC(=O)CCOCC(F)F)C)=O)cc(C(C)(F)F)n[nH]1 C=C(Cl)CCC(=O)NC(CCSC)C(=O)Nc1cncc(CC)c1 c1(C(=O)NCC2(O)CCN(C(Cc3nc(NC=O)sc3)=O)C2)ccc([N+](=O)[O-])[nH]1 C1(NC(CCN(CCC)C)=O)CN(C(C2CCC(N=[N+]=[N-])C2)=O)CC2(CC2)C1 C1(C)(CC)CCC(C(N2CC=CC2C(=O)NC2COCC2N(C)C)=O)O1 c1(C(=O)NC2CN(C(CS(CC)(=O)=O)=O)CC2O)cc2cc(Cl)ccc2o1 C1(C(=O)NCC2C3CN(C(c4cc[nH]n4)=O)CC23)CCOCC12CCC2 N1(C(CC(C=C)C)=O)CCCC(NC(c2ccc(SC(F)F)cc2)=O)CC1 c1(NC(CC(=O)NC2(COC)CN(C(C=CCC)=O)C2)=O)ccc(C)c(C)c1 N1(C(C(C)NC(N)=O)=O)CCC(O)(CCNC(C23CCN(CC2)CC3)=O)CC1 C(CCN=c1[nH]c(=NC(C)C(C)C)[nH]c2cc(OC)ccc12)OC.C1CCN1 C(C1CCCCC1)=CC(=O)N(C)CC1(CNC(=O)Cc2coc(C(F)F)n2)CC1 N1(C(CS(CC)(=O)=O)=O)CC23CCCC2(C1)CN(C(c1onc(Br)c1C)=O)C3 C1(NC(C2OCCC(=O)C2)=O)CN(C(=O)CCc2cc[nH]n2)C2CCCC12 N1(C(C(C)O)=O)CC2CCN(C(c3csc(C(=O)N(C)C)n3)=O)CC12 c1(C(=O)NC(CC(=O)OC)C)n[nH]c2c1CN(C(C1NC(=O)CC1C)=O)C2 C(=O)(C=CS(=O)(=O)CC)N(C)CC1CCCCN1C(=O)C(F)=CC1CC1 N1(C(C2(CNC(c3ccc(C(F)F)o3)=O)CCCO2)=O)CCOC(CCO)C1 Cn1cc(C(=O)NC2CCC(NC(C3CC3(C)C(F)F)=O)CC2)cc1Br N1(C(CCCNC(=O)NCOC2CC2)=O)CC2CCN(C(=O)CC34CCCC3C4)C(C2)C1.OCF CC1ON=C(C(=O)N2CC(NC(c3c(F)ccc(O)c3F)=O)C3CC3C2)C1C CCCCCC(O)C(=O)NC1CCN(C(c2ccc(CO)s2)=O)C1C(C)C N1(C(Cc2c(C)con2)=O)CCC2CCN(C(=O)C3=CCSC3)C2C1 c1(Cc2ccc(C)s2)nc(-c2ccc(Cl)cn2)nn1-c1nc(Br)nn1C N1(C(C2CCC(C(=O)N(C)C)O2)=O)CC2CC(NC(C3(C)CC3)=O)CC1C2 Cc1ccc(Cl)c(C(N2CCC(C(C)(C)CNC(C3COC(C)C3)=O)CC2)=O)c1 N1(C(C=C(C)C)=O)CC(N(C(=O)CC2COC(C)(C)CO2)C)C2(CC2)C1 Cc1cccc2c1CN(C(=O)Cc1ccccc1NCc1c(F)cccc1Br)C2 c1(C(=O)NCC2(NC(=O)CN3CCc4ccccc43)CC2)n[nH]c2ccc(F)cc12 c1(C(=O)NCC2N(C(CC=C(C)C)=O)CCCC2C)cc2ncccc2[nH]1 N1(C(C2N(CCC)CCC2)=O)CCOCCC1.C1CC(=O)NCC(=O)N1 N1(C(C2(O)CCC2)=O)CCCC(C2(NC(C3CC34CCC4)=O)CC2)C1 c1(OC)cccc(C(N2CCN(C(c3ccc(C)c(F)c3)=O)CC2CO)=O)c1N Cc1ccc(F)c(C(=O)NCC#CCNC(=O)CC2=CCCC2)c1O c1(C(N2CC(CNC(C3N(C)C(=O)NC3)=O)OCCC2)=O)cccc2c1COC2 c1(C(N2CCC(N(C(=O)CC3CCCC(O)C3)C)C2)=O)ccn2nccc2c1 c12c(C)nc(nc1O)CNC(=O)CC2.c1(CC(COC)CO)ccc(F)c(F)c1 C1(NC(=O)CCC(=O)c2ccccc2)CC2CCC1N(c1nnn(C)n1)C2 C1(CC(=O)N(C)Cc2cnco2)CCN(C(C2CCC(=O)O2)=O)C1(C)C C1(NC(C(CCC)C)=O)CC(O)CN(C(=O)CCc2cccnc2F)C1 C1(NC(=O)Cc2ccc[nH]2)CCN(C(C2(c3cccc(F)c3F)CC2)=O)CC1F C(c1ccccn1)=CC(=O)N(CC)CC1CCCN1C(c1ccc(Cl)s1)=O C1(CNC(CCNS(C)(=O)=O)=O)CCN(C(=O)C(C)(C)C#N)CC1 C(=O)(C(O)C(C)(C)CC)N1CC(C(C(=O)NC2(C=C)CCCC2)O)C1 C1(C(N(C)CC2CCN(C(c3n(C(C)C)ccc3)=O)C2)=O)CCS(=O)(=O)C1(C)C CC1C(NC(C2(O)CCCCC2)=O)CCCN1C(=O)CCc1cnn[nH]1 CC1(C)CCCC(CC(=O)NC2CC(C)(NC(=O)CNc3ncccn3)C2)O1 C1(CN(c2ccccc2)C)CCN(C(c2scnc2Cl)C(=O)NCCCF)C1 c1(NC(C2CCN(C(=O)NC(c3ccccc3)C)CC2)=O)cc2ncsc2[nH]1 N1(C(C(=O)NCC)=O)CCN(C(c2ccn(CCO)c(=O)c2)=O)CC1COC CCC1(CNC(=NCCCCl)NCCc2nccc(C)n2)OCCc2ccccc21 Cc1ccc(CNC(=O)OC2CCC(OC(C)(C)C)CC2)c(I)c1F C1(CC(=O)NCCC(C(C)C)[N+](C2CCOC2)(C(=O)CN)[O-])CCC(C)(C)CO1.O Cc1cc(=NCC2CCOC(C)(C)C2)[nH]c(NC2CC23CCC3)n1 Cc1cccc(CNCCc2cn(C3CCC(C(OC(=N)O)=O)C3)nn2)c1F CCCCCCCCCCC(=O)N(C1(C(=O)N(C)CC)CC1)C1CC1 C(C(=O)NCc1ccsc1C(=O)NCc1nn[nH]c1CO)(C(C)C)SC N1(C(C(C(CC)O)C)=O)CCC2CN(C(c3cc4nc(C)sc4[nH]3)=O)CC2CC1 c1(C(N2CCC(OCCCCF)C2)=O)cc2ccccc2cn1.N1(C)CCC1C=O CCC(CCCC(=O)Nc1cnccc1C)NC(C1(C)CCCCC1)=O CCC(CC(F)(F)F)C(=O)N1CC(CNC(c2c[nH]nc2C2CCC2)=O)C(C)C1 C(=O)(C(CNC(C1CCC(=O)N(C)C1)=O)C(C)C)N(CC(CC)C)C c1(C(N2CC(N(C(CSCC=C)=O)C)C2)=O)cnc2n1CC(C)CC2 c1(OC)ccc(F)c(CN2CC3CN(Cc4c(C)cccc4Cl)CC3C2)c1OC N1(C(C(CCC)OCC)=O)CCC(C(=O)N(CCCO)C)C1(C)C c1(C(C)OCCCn2cc(CC3CCOC3)nn2)ccc(Cl)nc1 Cc1cnc(C(=O)NCC2CCCCCN2C(=O)C(C)SC(F)(F)F)cc1C CCC(C)C(C(=O)N1CC2CCC2(C)C1)N(C(=O)CN(C1CC1)CC)C CCCCCC(CC)C(=O)N1CCC(C)(NC(c2ccc(OC)nc2F)=O)C1 N1(C(C2(C)CCC2)=O)CC2(C=C(C(=O)NC3CCC(O)C(O)C3)CO2)C1 C(=O)(C(F)C(C)C)Nc1n(C(C)C)cnc1.C12CC(C1)C(=O)NC2 C(=O)(C1CCCn2cnnc21)N(C)CC1CN(C(=O)COCCCF)CCO1 C(CCCCCC(=O)N1CC2(COC(=O)C2)C1)N(C)C(C1CC2C=CC1O2)=O C(=O)(C(=O)C(C)(C)C)N(CC)CC1CCCCN1C(=O)C(F)n1cccn1.NCC C12(C(=O)NC3CCC3)CC=CC(C1)OC2.c1(NC(CN(CC)CC)=O)ccccc1 C1(COC(N2CCC(Oc3cnccn3)C2)=O)OC(=O)CC12CNC2 C12(NC(C(C(=O)N(C)C)(C)C)=O)CN(C(=O)CCCC3CC3)CC1CS(=O)(=O)C2 N1(C(CN2C(C)CC2)=O)CC2CC2(NC(c2ccc(CNS(C)(=O)=O)cc2)=O)C1 C(C)(c1ccccc1C)=CC(N1C(CNC(C2CCCS2)=O)CC(COC)C1)=O C1(NC(c2c(C)con2)=O)CC(=O)N(C2CN(C3CC3)C2)C1.C12CCCN1C2 c1(C2(NC(=O)Nc3cscn3)CCN(CCOC)C2)ccc(F)cc1F CCCCCCC(C)C(=O)N(CCC(=O)NCC1=CCCCC1)C Cc1cnn(CC(N2CC(=C(F)CNC(=O)C(C3CCCCC3)F)C2)=O)c1 c1(C(=O)NC(C2(O)CCN(C(CC=C)=O)C2)C)cc(C#N)ccc1C C1(C(N2CC(C)N(C(=O)CC3NC(=O)NC3=O)CC2)=O)CCc2nc(O)[nH]c2C1 N1(C(CNC(C)=O)=O)CCCC(O)(CNC(=O)CCc2nccs2)CC1 N1(C(C2(SCC)CC2)=O)CCCOC(CCNC(=O)CC2CCCCC2(F)F)C1 C1(CC(=O)N(C2CN(C(=O)Cn3cc(Br)cn3)C2)C)C=CCCC1 N1(C(Cc2nc(C)[nH]n2)=O)CC(N(C)C)C(C(C)C)C1.c12cc(n(C)n1)CNC2=O c1(SCC)cccc(CC(N2CCN(C(=O)C(C)C(=O)OC(C)(C)C)CC2)=O)c1 CP(C)(=O)c1ccc(C(=O)NC2CCN(C(C3OCCCO3)=O)C2)cc1 C(=O)(C1CCc2c(Cl)cccc21)N1CC2C(CNC(C3(CC)CCCCC3)=O)C2C1 CC(C)(C)S(=O)CCCN=C(NCC1CCCCO1)NCC1C=CCC1 c1(OC)c(C(N2CC(NC(=O)Cc3ccc(Cl)nc3)CCC2C)=O)cccc1F N1(C(CC(C=C)c2ccccc2)=O)CC2(CCN(C(C3(C#N)CCCC3)=O)C2)C1 C(CCC(C)C)(C(=O)NCC1C(=O)NCCC1C)NC(C)=O C1(C(N2CCC(CNC(=O)CCCc3ccccc3)C2)=O)CCc2nn[nH]c2C1 C(CC(CC)C(=O)N1CC(O)(CNC(=O)COc2cn[nH]c2)C1)=CC c1(OC)cc(CCNC(=O)N(c2occc2C)CC(O)C(C)C)c(F)cc1O Cc1cc(C)c(C(N2CCCN(C(=O)C(F)(F)C3CC3)CCC2)=O)c(S)n1 C=CC1(C(=O)NCC2CCOC(C)(C)C2)CCN(C(=O)CC2CCC2)C1 c1(CC(=O)NC(C)C(CO)NC(=O)CC2CCC(=O)N2C)c[nH]c2ncccc12 N1(C(C(CC)SC)=O)CCCC(F)(CNC(=O)C=C(Cl)Cl)C1 N1(C(CC2(CS(C)(=O)=O)CC2)=O)CC2CC1(C(=O)NC1CCOC1=O)C2 c1(C(=O)OC)cncc(C(=O)NCC(C)CN(C(=O)CNC(C)=O)C)c1C C1(C(=O)NCC(C2CCN(C(c3nnc(C)s3)=O)CC2)F)CCCNS1(=O)=O C(=O)(C(C)(F)C(C)(C)F)NC(CC)CNC(=O)CCC(=O)c1cnn(C)c1 C1(CC(N2C(CNC(C(C)NC(C)=O)=O)CCC2)=O)CC(=O)NC1=O C1(NC(CC2(C(=O)OC)CC2)=O)CCC(C(=O)Nc2scc(C)c2OC)CC1 Cc1nccnc1C(=O)N(C1CCCN1CC(=O)NC(C)C)C1CCCC1 C12(CNC(C(C)NC(=O)CC(C)(C)C)=O)CC(CO1)N(C(=O)CSCC(N)=O)C2 c1(N2C(C)(C(=O)Nc3ncc(C)nc3Br)CC2)nc(Cl)c2c(ccn2C)n1 CC1(C)OCC2CC12C(=O)NC1COCCC1NC(c1csnc1Br)=O CC(CCC(C)(C)C)C(=O)N1C(C(=O)NC2(C3CC3)CC=CC2)CCC12CC2 C1(CNC(c2cnc(C(C)C)[nH]2)=O)CN(C(=O)C(c2ccccc2)F)CC1(F)F C(=O)(C1=NN(CCO)C(=O)CC1)NC1C(C)CN(C(C2CCC2)=O)CC1 Cc1c(C(N2CCC(OCCNC(C3CCCN3C(C)C)=O)C2)=O)ccn1C Cc1cnc2cc(C(=O)NCC(C)(C)CNC(=O)CCN(S(C)(=O)=O)C)ccn12 CCC(CC(F)F)C(=O)NCC1(CCNC(c2n[nH]c3c2CCSC3)=O)CC1 C(=O)(C(C)(C)C(C)(C)O)NC1CC(CCNC(C(C)OCC)=O)C1 c1(C(=O)NC2(C)CC(NC(C(CC=CC)C)=O)C2)ccnc(Cl)c1NC c1(OC(C)C(N2CCCC2C(C)(C)CNC(=O)CC#N)=O)ccccc1C#N c1(C2CCN(C(C(C)Cc3ccc(Cl)cc3)=O)CC2)cccc(C(=O)O)c1F C(C)(C)(CCCNC(c1ccnnc1O)=O)NC(C(CN(CC)CC)F)=O C=CC(C)(CC)C(=O)NC1CCC1NC(=O)Cc1ccc(Cl)cn1 c1(C(C(=O)OCC)OC(c2c[nH]nc2CC)=O)ccccc1Cl C(=O)(C1=C(Cl)CCC(C)C1)NC1CCCN(C(c2c(OC)c[nH]n2)=O)C1 c1(NC2CCC3(CN(Cc4[nH]c(C)c(Br)c4C)C3)O2)nccc2oc(Br)cc12 c1(CNC(CC2(C=C)CCC2)=O)cnn(C)c1C(=O)NCC1CCC(=O)N1 C1(C(=O)NCC(CNC(C=CC(C)(C)C)=O)(C)F)CCCC2(CCC2)O1 c1(CN(C(c2cc(Cl)ccc2F)C(=O)NC2CCOC2)C)nc2ncccn2n1 CCC(CC)C(C)C(=O)NC(C)Cn1cc(-c2ccnn2C(C)C)nn1 N1(C(C(C)C(F)F)=O)CCC(C2(NC(=O)COCC3CCCO3)CC2)CC1 c1(CC(=O)NCCCN(C(c2ocnc2C)=O)CC)cccc2c1OC(C)(C)C2 S(=O)(=O)(c1cc(C)cnc1NCC1(OCC)CC1)NC1CCC(CCCC)CC1 N1(CCc2c(OC)cccc2)CCC(NC(C2CCCN2N=O)=O)CC(C)(C)C1 C1(OC)CN(C)C(C)(C(=O)NC2CN(C(=O)CCc3cncs3)C2)C1 CCCC(C)(O)CC(=O)NC(C1CCN(C(=O)C(O)CC2CCCC2)C1)C C(=O)(C1CCCc2nnn(C)c21)N(CC(CNC(c1onc(C)c1C)=O)O)C C=CCC(CC(C)C)C(=O)N1CC2CCCN(C(=O)CCC3CCCCO3)C2C1 Cc1cc(OCC(N2CCC(CN(C)C(c3cc(C(C)(C)C)no3)=O)C2)=O)no1 C(=O)(C(O)C(F)(F)F)NC1C(CNC(=O)CCCOc2cccnc2)CCCC1 N1(C(C(CC(CC)C)NC(c2ccc(C(C)C)o2)=O)=O)CCCC(C2(C)CC2)C1 N#Cc1cc(C(N2CC3(CC3C(=O)Nc3cnc(C4CC4)nc3)C2)=O)ccc1Br C1(NC(CC(CC)OC)=O)CN(C(c2ccns2)=O)C2CCCC12 C(CCC(F)(F)F)N(C(=O)CCCN(C)C(C1CCCOC1)=O)C C1(C(=O)NCCC2N(C(c3c(C(C)C)ncs3)=O)CCC2)CCC2(CCOC2)O1 C1(OC)CC(NC(C2CC(=O)NC(C)C2)=O)CN(C(c2ncnn2C)=O)C1 c1(C(N(C2CCN(C(C34CC(C)C3C4)=O)C2)C)=O)cccc2c1CCC2=O C1(C(NOCC(C(C)C)O)=O)CCC2CCC1N2C(=O)CCc1cnco1 CC1CCCn2ncc(C(=O)NCC3CC(NC(C4(F)CC4C)=O)C3)c21 CC1Oc2cc(NCC(O)COCc3ccccc3)ccc2NC1=O n1(CC(C)O)cc(C(=O)NC2C=CCN(C(c3cc(F)cs3)=O)C2)ccc1=O C1(C(C)C)C(NC(=O)C(F)C(C)C)CCN1C(c1csc(SCC(N)=O)n1)=O C1(CC=C)(NC(C2CC23CCCC3)=O)CCN(C(=O)CS(=O)(=O)NC)CC1 C1(NC(c2nc(C)[nH]n2)=O)CN(C(c2ccc3nnnn3c2)=O)C2(CCOC2)C1 C1(NC(CC(C)(C)N(C)C(C2CCCC(C#N)C2)=O)=O)CCOC12CCCC2 c1(C(N2CCCC(N(C(=O)CCc3cncs3)CC)C2)=O)ccc(NC)c(F)c1 C1(C)(C(N(CC(=O)NCC(=O)NCC=CC(CC)C)CC)=O)CC2C=CC1C2 c1(-c2ccc(SC)s2)ccc(OC(C)(C)C)cc1.N12CCC(C1)CC2=O C1(NC(CC(C)(C)O)=O)CC(C2CCN(C(=O)Cc3cc(F)ccc3Cl)C2)C1 CC(C)CCCCC(=O)NCCCN(C(C1CNC(=O)N1)=O)C1CC1 C1(CC(=O)N(C)CC2CC2c2cncs2)COCCN1C(=O)C(F)=C1CCCC1 N1(C(C2N(C)CC2)=O)CCCCC1CCC(N1CC(F)(F)C1C1CC1)=O CC1CCC(C)(C)N1C(C1CCN(CC2CCC(C)(C)O2)CC1)=O C(=O)(CC1NC(=O)c2ccccc21)NCC1CC(NC(c2c(N)nccc2)=O)C1 CCC(CC(=O)NCCCCN(CCCNC(=O)CC1CC(F)(F)C1)C)C1CC1 c1(C(N(CC(C)N(C(CCSCCCC)=O)C)C)=O)[nH]c2ccc(C)cc2c1C c1(C(=O)NCC(CC)NC(C2CC3(CC3)CO2)=O)cncnc1C1CC1 C1(C(N(C(C)CNC(c2nocc2Cl)=O)CC)=O)CC(C)=NO1 c1(-c2n(C(COC)C)nc(C(C)C)n2)cc(Br)c2cccnn12 CC(C(=O)NCC1CC1C(=O)NCCN1CCC1)C(C)(C)C CC1CN(C(c2cn(C3CC3)nc2C2CC2)=O)CCC1NC(C12CCC(C1)C2)=O c1(CC)cccc(C)c1C(=O)NCC1(C)CCCC1NC(=O)C1=CCCC1C N1(CCNC(CCN(CC#C)C(C2CC2C)=O)=O)CCCC1=O C1(NC(C(C)NS(CC)(=O)=O)=O)C2CCC(C2)C1C(=O)Nc1c(C)cccc1C N1(C(C2(C)CCOC2)=O)CC2(CCN(C(=O)C(N3CCCC3)C3CC3)CC2)C1 CC(C)(C)CC(C(=O)NCC1CCCCO1)NC(c1cccn2ccnc12)=O c1(C(C(=O)NCC(C)N(C(C2CCOC2C)=O)CC)=O)cc(F)ccc1C c1(C(N2C(C(C)NC(=O)C(=O)NCC(F)F)CCCC2)=O)nnc(O)nc1O C1(C(=O)NC(c2cc(C)on2)C)CC2CCCC2N1C(=O)C=CC1CCCC1 Cc1ncccc1C(=O)N(C1CCCC1)CC1CC(NC(C2CCCN2N=O)=O)C1 C(CN=c1[nH]c(N2CCn3cnnc3C2)nc2cccc(F)c12)OC(C)C CC1CN(C(Cn2cc(CNc3c[nH]nc3-c3ccc(Cl)s3)nn2)=O)CC(C)O1 CCCCCC(C)CC(=O)N1CC2(CCC2NC(c2cnn(C)c2SC)=O)C1 C=CCCCC(=O)N1CC(SC)(NC(=O)C=CCOCC(F)(F)F)C1 C1(N2CCC(n3cc(CCCC(C)O)nn3)C2)(CCO)CCCCC1 C(=O)(C(C)C(CC)CC)N1C(C(=O)NC(C2CCCC2)C=CC)CCCCC1 C(C(C)(C)CC(=O)NC1CN(C(=O)CSC)CCC1F)SC C1(N(C(c2c(CCC)n[nH]c2)=O)C)CCCN(C(C2(C)CC(F)(F)C2)=O)CC1 N1(C(CCCCN(C)C)=O)CC2(CC(C(=O)Nc3cnn(C(C)(C)C)c3)CO2)C1 N1(C(C2(COCC)CC2)=O)CC(O)CC1(C)C(=O)NC(c1ncn(C)n1)C c1(NC(C(C(=O)N(C)CC2CC3CC2C3)OC)=O)cc(C)cc(C)c1 C(=O)(C(C)(C)CCNC(C1COC(=O)N1C)=O)NCC1CCN(C(C)=O)C1 C1(NC(C2CCCC(C)(C)C2)=O)CN(C(=O)CC2CC(=O)C2)Cc2ccnn2C1 N1(C(Cn2cc(-c3n(CC)ccn3)nn2)=O)CCC(F)(F)CC1C(=O)OC c1(NC(CC(C)C2CCOC2)=O)cnc(O)c(F)c1 N1(C(C2N(C)CCOC2)=O)CCC(C2(O)CN(C(C3CC34CCCC4)=O)C2)CC1 c1(-c2nnc(NC(CCC)CC(=O)OCC)o2)ccc2cnoc2c1 CON1CCC(C(=O)NC(C2CN(C(c3ccc([N+](=O)[O-])[nH]3)=O)CCO2)C)CC1 N1(C(C(COC(C)C)(C)C)=O)CC2CC(NC(c3ccc(C(N)=O)nc3)=O)C1C2 N1(C(COCCOC)=O)CCC(C(=O)NC2(OC)CCSC2)CC1C C1(CNC(C(C2CC(NC(C(N3CC(C)C3)C)=O)C2)F)=O)CCC(=O)C1 c1(C(=O)NCC23C(CN(C(c4scc(COC)c4)=O)C2)C3)cnc(Cl)c(N)c1 c1(C(N(CC(=O)NCC2CC2CN(C)C)CC)=O)cc(CC)cs1 C(=O)(C1=C(Cl)CCCC1)NCC(CCC)NC(c1ccn(CC)c(=O)c1)=O c1(OC)cc(NC(=O)NNC(=O)Cn2ncc3ccccc23)c2ccccc2c1 N1(Cc2c(C)cccn2)CC2CN(C(c3ccc(Cl)nc3Cl)=O)CC2C1 N1(C(c2nccc(C)c2)=O)CC2(CC2)CC1C(N1CCSCC1C)=O C1(CC)CCC(C(=O)NCC(C)(C)NC(c2cc(C)ns2)=O)C1 C(CCCCN(C)C(c1cncs1)=O)NC(C1C(C(c2ccccc2)C)C1)=O C(CN=c1cc[nH]c(=NCCCN2CCC3CC23)[nH]1)N1S(=O)(=O)CCC1 c1(C(=O)OC)cc(N2CCC(C)(NC(c3ccc(Cl)s3)=O)C2)nc(C)n1 c1(C(=O)NC2CN(C(c3cccc(NC)n3)=O)CC2F)cc2n(c1)CCCC2 CC1CC(C(=O)Nc2cncnc2)N1C(=O)CNc1ccccn1 c12ncnc(Cl)c1C(=O)NC1(CO)CN2C1.c1(C(=O)OC)ccnc(N(C)C)n1 N1(C(c2n(C)cnc2)=O)CCN(C(c2ccc(C(C)(C)C)s2)=O)C2CCC12 C1(C(=O)NCc2n(C(C)C)cnn2)C=CCCN1C(=O)CC=CCO N1(C(CC=C=C)=O)CCC2(CCOCC2)C(NC(=O)C(C)CCCOC)C1 c1(C(=O)OC)ccc(C(C(=O)NC2CCOC2)N(C2CC(CO)C2)C)o1 C1(C#CC(=O)N2CCOCC(NC(=O)CCc3nc(C)cs3)C2)(CC)CC1 C1(NC(C2(C(C)C)CCN(C(c3c(C)ocn3)=O)C2)=O)CCCCC1N=[N+]=[N-] N1(C(c2ccc(OCOC)cc2)=O)CCCC12CCS(=N)(=O)CC2 c1(CNC(=NCc2n(C)ncc2)NCCC2CCCO2)cnc(C2CC2)nc1 Cc1nn(C)c(C)c1-c1cn(CC(N2CCCC(OC3CC3)C2)=O)nn1 N1(C(C2CCCC(OC)C2)=O)CCOC2(CCCN(C(C3CNC(=O)O3)=O)C2)C1 N1(C(CNC(c2cc(CC)ncn2)=O)=O)CC2CC=CC1C2.C1C(=O)N1 C(=O)(C1=CCC(C)(C)CC1)NC1CN(C(c2nc(OC)c(C)s2)=O)CC2(C1)CC2 C1(C(=O)NCC(CC)(C)OC)CC(=O)CN1C(c1cc(C(C)C)sn1)=O C1(C(N2CCCC(CN(C(C3CCC(=C)CC3)=O)C)C2)=O)CCOC2(CCC2)C1 c1(C(=O)NC2CN(Cc3c(F)cccc3F)CC2O)c(F)cc(F)cc1Cl Cc1nnc(O)c(C(=O)NCC2CC3CN(C(c4cc(CO)on4)=O)CC23)c1C N=c1[nH]c(C(=O)C(=O)NCC(c2ccccc2)NC(=O)C2=CCC2)cs1 C1(O)(C(N2C(CNC(C3CC4CCC3C4)=O)CCC2)=O)CCCCCC1 S(=O)(=O)(c1c[nH]ccc1=NCC(CO)C1CCC1)NCCCC=C C#CC1(C)CCCN(C(=O)C(N2CCC3(Sc4ccccc4)CCCC23)=O)C1 CC1(C#N)CN(C(=O)C(Cc2ccoc2)NC(c2cnn[nH]2)=O)C1 Nc1[nH]c(=O)c(Cl)nc1C(=O)NCC1CCCCC1NC(c1cnns1)=O c1(OC)c(Cl)ccc(Cl)c1C(=O)NC1CCCCC1NC(=O)CC1CCCC1O N1(C(N=c2cc(C)n(CCO)[nH]2)=O)CCc2cc(F)cc(F)c2C1 n1(C(C)(C)C(=O)NCC2(NC(C3CC(C#N)C3)=O)CCOC2)cc([N+](=O)[O-])cn1 C(C)(CC(C)NC(=O)C(F)(F)c1ccc(Cl)s1)NC(C1CN(S(CC)(=O)=O)C1)=O C1(C(=O)NCCCN(C(=O)C(=O)CC(F)(F)F)CC2CCCC2)C2CCC(=O)C12 N1(C(C(C=C)c2ccccc2)=O)CC2(CNC(=O)C=CC(C)(C)C)CC1CO2 c1(CC(N2C(CNC(C3N(C)CCOC3)=O)CC2)=O)cccc(C(F)(F)F)c1Cl c1(CNCC2(C(=O)Nc3ccc(Cl)c(Cl)n3)CC2)cc(F)ccc1Cl C1(NC(c2ncc(Cl)n2C)c2n(CC)nnn2)CCOC2(CCCC2)C1 C1(NC(CCNC(C)=O)=O)CCCN(C(=O)Cc2ccccc2C)CC1F c1(COC(C(c2cnn(C)c2)N(C)C(=O)OC(C)(C)C)=O)ncc(F)cc1F C1(NC(=O)OC(C=CC(=O)NC(C2CCCCC2)C#C)C)CC2CC2CC1C C(=O)(CC(C(N)=O)NC(=O)OC)OCCC(C)C c1(OC)cc(N)ccc1C(=O)NCC(CO)NC(=O)C(C)CN1CCOCC1 N(C1CCc2c(OC)cc(F)cc21)c1cccc(OCCC)c1 C=CC(C)CC(=O)NCCC(C)N(C)C(C1C(C(=O)OC)C1(C)C)=O C1(O)(CNC(Cc2cnc(C)[nH]2)=O)CCCN(C(C2CN3CCCC2C3)=O)C1 C1(O)(C(C(=O)NCCCOCCSC)F)CN(C(=O)CC2CNC(=O)O2)C1 C(CCC(=O)N1CCC(C(=O)N(CCCN(CC(C)C)C)C)O1)OC(C)=O N1(C(C)=O)CCCCC1C(N1CC(CNC(=O)C(C)Cc2ccco2)(OC)C1)=O C(=O)(C(C)CC(F)(F)F)NCCC1N(C(CC(=O)OC)=O)CC(OC)C1 c1(C(=O)NCCC(CNC(C(c2ccc(F)cc2)C)=O)O)ccnnc1S CC(C)(C#N)CC(=O)N1CCC(O)(CNC(=O)COc2ccc(O)cc2)C1 C1(N(C(CONC(C2(C(C)=O)CCC2)=O)=O)C)CCCC1C n1(CC)c(C(=O)NCC(C)(CO)NC(=O)CCCc2ccccn2)cnc1O c1(CC(N2CCC(N(C)C(C3(O)CCOC3)=O)CC2)=O)ccc2c(c1)CCC2 C12(CNC(C3CC(CC)C3)=O)CC1CN(C(c1ccc(O)nn1)=O)C2 c1(CCC(N2CCC(N(C(=O)CC3CCC3)CCO)C2)=O)ccc(Br)c(F)c1 c1(CC(=O)NC2CCN(C(CC3COCC(C)O3)=O)CC2)ccc(F)c(Cl)c1F C(=O)(CS(=O)(=O)CCO)NC1CC(C)N(C(=O)C=CSc2ccccc2)CC1 Cc1cc(CNC(c2csc(C(C)OC)n2)c2nnnn2C2(C)CC2)nc(Br)c1 N1(C(CC2(OCC)CCC2)=O)CCC(C)CC1NC(c1cccc(SC)c1)=O N1(C(Cc2n(C)nc(-c3ccsc3)n2)=O)Cc2ccc(F)cc2C1 c1(OC)cccc(C(F)(F)C(=O)NC2CCCC2NC(=O)Cn2nnnc2C)n1 C1(NC(Cc2c(C)cc(Cl)cc2)=O)C2CC3CN(C(C4CCNC4=O)=O)C1C3C2 N1(C(C2C(C)C2)=O)CC(CNC(=O)CC2=NNC(=O)C2)C2(CCOCC2)C1 N1(CCC(=O)N(CC(C)NC(=O)CCCC2CC2)C)CCC(F)C1 c1(C(=O)NCCCN(C)C(c2ccc(F)cc2)=O)ccc(F)c2[nH]c(=N)sc12 C#Cc1ccccc1CC(=O)NCCOCCN(C)C(C1(C)CCNC(=O)C1)=O N1(C(C2(C=C)CC2)=O)CC(OC)C(NC(=O)CCCOc2cccc(F)c2)C1 c1(NC(C)=O)ccc(NC(=O)C(=O)NC2CCCC2)cc1C.c12cccnc1NC2 c1(C(N(CCNC(C(CO)OC)=O)CC2CC2)=O)cc(O)nc(N(C)C)n1 Cc1c(CCC(N2CCC(C)(NC(=O)C(C)Cn3cccn3)C2)=O)cnn1C CC1CN(C(c2cc(Br)sn2)=O)CC1(C)CNC(c1cc(C(N)=O)c[nH]1)=O N1(C(C(CN(C)C)N(C)C)=O)CC(N(C)C(C23CC(CO)(C2)C3)=O)C(C)(C)C1 C#Cc1cc(F)c(C(=O)NC2CCN(C(=O)CN(C)C3CC3)CC2C)cc1F N(C(=NCCCCCCSC)NCc1noc(C)n1)CC1C(OC)CCC1 C(=O)(CCCCCC(C)O)NCC(C(C)(C)C)NC(c1c(CC)[nH]c(=N)s1)=O C1(NC(c2cccc(-c3ccsc3)c2)=O)CN(C(=O)CC2CC2)CCC1CO N1(C(C2(COC)C=CCN2C(=O)Cc2ccsn2)=O)CC=C(CO)CC1 CCCCCCCCC(=O)NCC(C)CN(C)C(c1nc(O)c(C)s1)=O C1(C(N(CC)CC2CCCCO2)=O)CCC(NC(=O)Cn2cnnn2)CC1 C1N=C(NCC(F)F)NCC(=O)N2CCC12.C1(NC)CCOCC1.CS n1(CC)cnc(C(=O)N(C2(CC(=O)NCCc3ccnn3C)CC2)C)n1 C=CCC(CC)C(=O)NCC1CC(OC)CN1C(c1cc(Br)sn1)=O c1(CNC(=O)CN2CCNC2=O)ccc(Cl)c(F)c1F.C12CCCN(CC1)C2=O CC1CC(NC(C2(C(N)=O)CCC2)=O)CCN1C(=O)CCc1ccsc1 C(=O)(C(CC(=C)Cl)NC(c1cncc(F)c1C)=O)NCC=C=C O=C1OC2CC(C(=O)Nc3ccc(F)c(F)c3F)CC2O1 c1(OC)ccnc(F)c1C(N1CCCC(C(C)NC(c2ccn(CC#N)n2)=O)C1)=O CN1CC(O)CC1(C)C(=O)NCc1cc(C(=O)NCC2=CCCC2)on1 C1(C(=O)NC(CC(C)N(c2ccccc2)C)C)C2CN(CC3CCOC3)CC12 N1(CC#C)CC(c2nnnn2CCCF)(NC2CCNC(=O)CC2)CCC1=O C1(C(N(CCCNC(c2c(C)nn(C(C)(C)C)c2)=O)C)=O)CC(C)(C)CN1C c1(C(=O)NC(CNC(C(c2ccnn2C)C)=O)C)cc2c(nn1)CCCC2 C1(C(=O)NC(CCCC=C)C2CC2)CC12CCN(C(=O)C1=CCSC1)C2 C1(C(N(CC(C)N(C(C(C2CCCCC2)OC)=O)C)C)=O)C(C#N)C1(C)C c1(C(N2CCCC(N(C(COCCCC)=O)CCF)C2)=O)cnn2ncccc12 CC1CN(C)C(=O)CN1N1CCCC1CNS(C)(=O)=O Cc1ccc(Br)cc1CC(=O)NC12CC1CN(C(=O)C(C)Cc1ccco1)C2 N1(C(CC2(OCC)CC2)=O)CC(NC(c2ccn(C)c2)=O)CC(O)C1 C=CCCC(CC(C)C)C(=O)N1CCC(NC(c2n[nH]c3c2CC(C)(C)C3)=O)C1 c1(CC(=O)N(C2CCN(C(c3nc(C4CC4)no3)=O)C2)CC)cccc(C)c1C C12CCOC1C(=O)N2.C(=O)(CCCc1ccsc1)NCCNS(C)(=O)=O c1(C(=O)NC2CCCC(NC(C3N(C)C(=O)OC3)=O)C2)nccc2ccncc12 N1(C(C(CCC)OCC)=O)CCN(C(C2CC(O)C2)=O)CC1C(F)F C=Cc1ccc(C(=O)NC2COCC2NC(=O)C(CC(C)C)NC(=O)CCC)cc1 CC(C(=O)NCC1CCC2(CN(C(C3(C(C)(F)F)CC3)=O)C2)O1)C(F)(F)C(F)F c1(N)ncnc2sc([N+](=O)[O-])cc12.CC(C)CCC(=O)NCC(N1CC(CN)C1)=O C1(C2CC2)(C(N2CCCC(CCOC)C2)=O)CN(C(=O)C(C)(C)CC#N)C1 CCCCS(=O)(=O)NCC(=O)N(C)CCNC(=O)C(c1cnn(C)c1)OC c1(C(N(CC(CC)NC(=O)C(C)(C)CO)C)=O)cnc2ccc(C)cc2c1 C(c1ccccc1C)=CC(=O)N(C(CN1CCN(C(CC)=O)CC1)C)CC N#Cc1cc([N+](=O)[O-])c[nH]c1=NCCCCNC(c1ccc(C(F)F)cn1)=O c1(C(=O)NC2C3C(C)N(C(=O)CO)C2C3)cc2c(cc1Br)OCCO2 c1(OCC)nc2ccccc2cc1C(N1CC2CC1(CNC(=O)C(C)SC)C2)=O C1(NC(C(C)N(CC)CC)=O)C2CN(C(c3cnoc3-c3cnn(C)c3)=O)CC12 Cc1ccc2c(C(=O)NCC3CCN(C(C4(F)C(C)(C)C4(C)C)=O)C3)onc2c1 c1(NC(CCc2c[nH]c(=N)[nH]2)=O)cnc2ccccn12.C12CC3CCC1N3C2=O CC1CN(C(=O)COC2CCN(C(C3(C#N)CCC3)=O)C2)CCN1C1CC1 N1(C(C(C)=C2CCC2)=O)CCC(N(C(=O)CC2CCC(C(F)(F)F)O2)CCO)C1 c1(C(=O)NCCc2cn(-c3cc(Cl)cc(Cl)c3F)nn2)[nH]cc2c1CCCC2 C(=O)(C1=CC2(CCOC2)C1)NCC(C1CC1)NC(c1c(C)nc(CC)nc1C)=O C1(NCC(=O)OCC)CCc2[nH]c(=NCCCN3CCCC3)ccc2C1 c1(C(=O)NCCCN(C(c2c(CC(C)C)n(C)nc2)=O)C)cccc2ncnn12 CCCCC(C)C(=O)NCC1CC(O)(CNC(c2cnc(CC)nc2C)=O)C1 N1(C(C=CC(CC)C)=O)CC(CNC(c2cc3ccncc3[nH]2)=O)C2(CCC2)C1 c1(CN2CCC(NC(c3ccc(Cl)o3)=O)CC2)ccc(O)c(O)c1O CCCC(C(=O)N1CCC(NC(C2COC(=O)N2C)=O)CC1)S(N)(=O)=O C1(C(=O)NCC(C)N(C(C2CCC2CC(=O)NC)=O)CC)C2CN(C)CC12 C(CC1CC1)(C(=O)NC1CCSC1)NC(=O)CCC1CC1 C1(CC)CN(C(c2c(C)coc2C)=O)CCC1NC(=O)C(C)NC(=O)C(C)(C)C N1(C(c2c(C)cc(N)cc2)=O)CCCN(C(=O)C(C)NC(=O)C(C)(C)C)CCC1 C1(C(=O)NC(C(C)C)CNC(=O)Cc2csc(Cl)n2)CC(C)(C)OC1(C)C C(CC(CN)NC(=O)C(F)(F)F)OC.C(=O)(C(C)NC)NC(C)(C)C.C1(=O)CC(Cl)C1 C(CCCOC)(C(=O)N(CCF)CCOC)NC(C(C=C)CC)=O C12(C(=O)OC)CCC(CC1)N(CCC(=O)Nc1cc(Cl)ccc1Cl)C2 Cc1c(C(=O)NCC(C)NC(=O)C(CC(C)C)n2ccnc2)nn2ccccc12 C(CC(C(=O)N(C)Cc1cccc(C)n1)NC(C1CC2(CSC2)C1)=O)OC c1(C(C(=O)NC2C(C)N(C(=O)CSC3CC3)CC2)CO)cc(Cl)cc(Cl)c1 CC(C)CC(C)(CNC(C1CCC(=O)N1)=O)NC(=O)C(O)CC(N)=O N1(Cc2scc(CC)c2)C(=O)CCN(CC2CCCSC2)C1=O C1(NC(C(C)OCC)=O)CCCN(C(=O)Cc2cc[nH]n2)CCC1 N1(C(C(CC)n2cncn2)=O)CC=CC(C(=O)NCCn2ncnn2)C1 C=CCCC(=O)NCC(CNC(c1cn(C2CCCC2O)nn1)=O)CO C=CCCC(O)Cc1ccc(NC(N2CC(C(=O)NC)C2)=O)cc1 c1(-n2cc(-c3nc(C)sc3)nn2)c(NC(=O)CC2CC3C=CC2C3)cccc1Br Cc1ccc(CCC(=O)NC2CCC2C)o1.C12(CCCC1)C(=O)NC2 CC1(C)CC(O)(CC(N2CCC(O)(CNC(C3CCC(=O)N3C)=O)C2)=O)CO1 C1(N(C)C=NCCc2cnnn2C)CCCC12CNC2=O c1(C(c2n(CC)nnn2)NCCCCF)cccc([N+](=O)[O-])c1C c1(C(N2CC(C(C(=O)Nc3cn(CC)nc3)OC)C2)=O)cc[n+]([O-])cc1 C1(NC(Cc2c(C)nc[nH]2)=O)CCCCN(C(c2ccoc2Cl)=O)C1 C1(C(N(C2CC(C(=O)OC)C2)C)=O)CCN(C(C2CCCC(C#N)C2)=O)C1(C)C C(=O)(CC(C(F)F)NC(c1ccnnc1O)=O)N1C(CC)CC(C)C1 C1(O)(SCCCCNC(=O)OC(C)(C)C)C(NC(C(=O)NC(C)C)=O)CCC1O CC1CN(C(=O)CCCC2CCC2)CC(C)N(C(c2cc(N)cc(F)c2)=O)C1 N1(C(COCCCCCC)=O)CC2(CCN(C(=O)CC3CCCCN3C)CC2)C1 c1(C(=O)NCC(CNC(=O)C=CC(F)F)OC)cc(C2CC2)oc1C C1(NC(c2cc(CNC(C34CSCC3C4)=O)cs2)=O)CCN2CCC1C2 C(C)(C)(CC(=O)N1CCOC(C2CN(C(=O)CN(C)C(C)C)C2)C1)OC C(=O)(C(C)(C)C1=CCS(=O)(=O)CC1)NC1CCCCC1NC(CNC(=O)NC)=O C(=O)(CC(F)(F)C(F)F)N1CC(NC(C(C(=O)OC)(C)F)=O)C1 N1(C(C(CCC)OC)=O)CC2CCC(C(=O)NCC3C(C)(C)C3(C)C)(C2)C1 C1(C(N2CCCC(NC(C3(Cc4ccc(Br)cc4)CC3)=O)C2)=O)C(F)(F)C12CC2 C1(C)(C(N(CCOC)CCNC(=O)Cc2nocc2C)=O)CC=CCC1 C1(NC(C(C)OCC)=O)CC2CC(NC(=O)CCc3ccccc3)CC12 CN1CCN(C(=O)C(C2(O)CCCC2)F)CC1C(=O)NCC12CCC(CC1)O2 C(=O)(C1=NOC2(CCOC2)C1)NCC1(C)COCCN(C(C=C(CCC)C)=O)C1 C1(C(=O)Nc2cnn(CC(F)(F)F)c2)C2CN(C(C3CC4CC4C3)=O)CC12 CCC(C)(CC)C(=O)NCC1CC(NC(C2(CC(=O)OC)CCCC2)=O)C(O)C1 CCC(C(=O)N(C)CCNC(C1CN(C(=O)CCCNC(C)=O)C1)=O)C(C)C N1(C(c2sccc2I)C(=O)Nc2ccc(OC)cc2)CC2CCC1C(O)C2O N1(C(CCC(C)SC)=O)CC(C)CN(C(=O)Cc2c[nH]c(=N)nc2O)CC1C C1(NC(C(c2cccs2)NC(c2cnn(CC)c2C)=O)=O)CCC2(CCC2)C1 N1(C(CCCOCC=C)=O)CCC2(CC1)CCN(C(C1C3CCC13)=O)CC2 C1(C)(CN(C(=O)CC2(CNC(C3(C(C)(C)O)CC3)=O)CC2)C)CCCO1 CCCCC(C)(F)C(=O)N1CCC1Cn1cc(CN2CCS(=O)CC2)nn1 CCC(C(=O)N1CCN(C(c2csc(C)c2C2CC2)=O)C(CO)C1)C(C)(F)F N1(C(CC(C)C)=O)CCC(NC(=O)CN(C)C(c2ccsc2)=O)C1(C)C c1(C(N2CCC(NC(Cn3nnc(C)n3)=O)C2(C)C)=O)nn2cccnc2c1Cl c1(NC(=O)NCC(C2CCC2)OCC)ccccc1 S(=O)(=O)(c1ccc(Br)c(C(=O)O)c1)N1CCCC(C(N2CCCC(C)CC2)C)C1 C1(C)(NC(c2c(C)cco2)=O)CCCN(C(=O)CC2NC(=O)NC2=O)C1 C12(C(=O)NC(CCNC(c3n(C(CC)C)ncc3)=O)C)CCOC1CC(=O)NC2 N(C(=NCCF)N1CCC(c2cccnc2)C1)Cc1nc(COC)on1 Cc1cc(C(=O)NC2CCCN(C(C3(CO)CCCCC3)=O)C2)c(Br)cn1 c1(NC)cc(C(=O)NC(CNC(c2occc(=O)c2OC)=O)CO)cc(Cl)n1 C1(NC(=O)NC23C(C)(C)OCC2C3)CCc2c[nH]nc2C1 c1(C(N2CC3N(C(c4cc(O)ccc4Br)=O)C3C2)=O)cc(F)ccc1[N+](=O)[O-] c1(NC(=O)NC(c2ccc(C)o2)C)c(C)nn(C)c1OC(F)F c1(C(N(CC(CN(C(C=Cc2c(C)ncs2)=O)C)O)C)=O)[nH]cc2c1CCCC2 N1(CC(=O)N(C(CCC)C(=O)OC)C)CCCC(F)(F)C1 c1(CNC(C2C(CNC(=O)CC3COCC3O)CC2)=O)ccccc1F Cn1ccc2cc(C(=O)NCC3CN(C(C4CC4CN(C)C)=O)C3)cnc12 c1(C(C(=O)NC2(CN(C)C(C3SCCS3)=O)CC2)=O)cccn1C C1(NC(C2C(C)C2)=O)CC2CC1N(C(C1(c3ccc(F)cc3)CCCCC1)=O)C2 c1(NC(C=CC(=O)N(C)C)=O)ccc(F)c(NC(=O)CSCCC#N)c1 c1(NC(CC(C=C)c2ccccc2)=O)ccc(N)c(O)c1.C12CC(C1)CNC2=O c1(C(=O)NC(C(C)NC(C2CCCN2C(N)=O)=O)CO)cc2n(c1)CCOC2 N1(C(C2C(C)(C)C(=O)C2)=O)Cc2[nH]nc(C(=O)NCCCc3cnccn3)c2C1 CC1(CNC(=O)Cc2ccc(CO)cc2)CCCN1C(c1ccsc1Cl)=O Cc1cc(C(=O)NCCCCCCN(C(=O)CC(C)(C)C#N)C)cc(C)c1F C1(NC(c2ccsn2)=O)CC2CC1N(C(c1cc(O)cc(F)c1)=O)C2 c1(C(=O)NC(CN(C(c2c(CCC)nco2)=O)C)C)cc2cccc(C)c2[nH]1 C1(CCCC(=O)NCC2CC(NC(c3c(C)cno3)=O)C2)CCC(C)C1(C)C C1(C(=O)NCCCNC(c2ccc(C)cc2)=O)COCCC12CN(C(=O)C(Cl)Cl)C2 N1(C(CCC=CC(C)C)=O)CCC(C(=O)NCCc2ocnc2CO)C1C CC(C)(C)CCCCC(=O)N1CC=C(CCNC(C2(n3cccn3)CC2)=O)CC1 C1(CNC(c2ccc(OC)s2)=O)CC(NC(=O)CCc2ccc(Cl)nc2)C1(C)C c1(C(=O)NC(CNC(C(CC)Sc2nc(=N)[nH][nH]2)=O)(C)CO)ccc(C#N)n1C c1(C(C)(F)F)ncncc1N1CCOCC1CC1CC1 c1(OC)cccc2sc(NC(C)CSC(F)F)nc12 Cc1ccc(C(=O)NCC2CN(C(c3c(C(F)(F)F)cccc3N)=O)C2)cc1C C(=O)(C(C)S(N)(=O)=O)N(CC(CC)NC(=O)CC12CCC(CC1)C2)C c1(C(=O)NCCC2CCC(NC(C(C=C=C)C)=O)C2)cnc(OC)nc1C(F)F c1(OC)ccc(NC(C2(C)CN(CC3CCC(C(C)C)CC3)C2)=O)c2cn[nH]c12 N1(C(c2cccc(C)c2)=O)CCCN(c2nnc(-c3cccnc3)s2)CCC1 Cc1[nH]nc(C(=O)NC2CCC2CNC(c2ccc(CO)c(Cl)c2)=O)c1[N+](=O)[O-] C1(CNC(C2CN(C)C2)=O)CC2(C1)CN(C(=O)C(O)Cc1cccc(Cl)c1)C2 CCCCCCCCC(=O)N1CCN(C(c2cnc(C(=O)OC)s2)=O)CC(O)C1 c1(OC)n[nH]cc1C(=O)N(CCCNC(C1CCC1C(C)(C)C)=O)C N1(C(c2cnc(OC)s2)=O)CC2CC2(CNC(C2CCOC2)=O)C1 N1(C(=O)OC(C)(C)C)C2CCC1CC(C(=O)N(CC(F)(F)F)CC(c1nccs1)=O)C2 n1(C(N2CCC(N(CCO)Cc3cnc(C(F)(F)F)s3)C2)=O)cc(CO)nn1 C=Cc1cncc(C(=O)NC(C2CCN(C(C3CCC(C)(C)CO3)=O)CC2)C)c1 c1(CC(=O)N(CC(C)NC(c2ccnc(F)c2F)=O)C)cc(F)cc(F)c1 S(=O)(=O)(c1nc(NC2CCc3c(nnn3C)C2)ccc1Br)NC(C(CC)CC)C C1(C(=O)NCCCCCNC(c2c(C(=O)OC)n[nH]c2)=O)CCCN(C(C)=O)C1 c1(C(=O)NC2C(C)(C)C(CNC(=O)Cc3cnsc3)C2)cc2sccc2[nH]1 c1(C(=O)NCC(CCNC(Cc2cc(C)sc2)=O)O)cc2c(Cl)cccn2n1 C(=O)(CCCCCC#N)NCc1ccc(CNC(c2ccc(OC)nc2)=O)cc1 C1(O)(C(C)NC(C2CC2c2ccc(Cl)s2)=O)CN(C(C2CC(O)C2)=O)C1 CC(C)CC(O)C(=O)NC1COCCC1NC(C1CC2(C1)CC(O)C2)=O C1(CNC(=O)NC(COC)C)CCC=CN1N(CC(=O)OCC)C.C(=O)OC N1(C(CN(C(COC)=O)C)=O)CCCCC(NC(C2CCN(OC)CC2)=O)CC1 C1(CC)CN(C(C2(c3c(C)cccc3Cl)CC2)=O)CCN1C(=O)C(C)CC(N)=O C(CNC(C1(F)CCCCC1)=O)(CC(F)(F)F)NC(c1c(Cl)cc(C)s1)=O C1(C(C(=O)NC)F)CCN(C(c2cnn(C(F)F)c2)=O)C1 C(=O)(C(F)(F)CC1CCCO1)NCC(C)(C1CC1)NC(C1CC(O)C1)=O C1(C(=O)NC(C)C(C)(C)C#N)CCCCCN1C(=O)CCCN(C)C C1(NC(c2n(C(C)C)ncc2)=O)COCCN(C(=O)C(C)(C)Br)C1 c1(CNC(Cn2c(C)ccn2)=O)cccnc1C(=O)N(CC(F)Cl)C N1(CC(=O)NC(CNC(CC2N(C(C)C)CCC2)=O)(C)CO)CCNC(=O)C1 C1(C(=O)OC2CC(=O)N(C)C2=O)COc2ccc(F)cc2C1 N1(C(c2c(C)nc(C3CC3)o2)=O)CCCC(C2CC2NC(=O)CNS(N)(=O)=O)C1 Cc1c[nH]c(C(=O)NCCn2cc(C(=O)NCC(C)(O)C(F)F)cn2)c1C C(=O)(C1=CC(O)C(NC(C2CC(C)(C)C2)=O)C1)NC(COC)C1CC1 C1(C(=O)NC2CCCC2CNC(c2cnc(Cl)s2)=O)(COC)CC1(F)F c1(N(N2CCCN(C)CC2)C)nc(=N)[nH]c(=NC(CF)C2CCC2)[nH]1 C1(c2nnnn2C2CCC2)(NC2C(CC(=O)OC)CNC2)CCN(C)CC1 Cc1nc2ncccn2c1C(=O)NCCNC(=O)C(Cc1ccc(O)cc1)C1CC1 Cc1cc(C(=O)NC2(C)CCN(C(=O)CN3CCC(CO)CC3)C2)c2n[nH]cc2c1 N1(C(Cc2ccc(C)s2)=O)CC(N=c2[nH]cnc3cnn(C)c23)CC2(CCC2)C1 C(=O)(CC(C(C)=O)C(=O)NOCc1cccc(C2(O)COC2)c1)OCC C1(C(=O)NCC(CC)C)(CCOC)CCN(C(c2ncc(C)cc2C)=O)CC1 C1(NC(C(C)Cc2ccccn2)=O)CCCCC1NC(c1cnco1)=O c1(C(=O)NC(CCNC(CCCNC(C)=O)=O)C)cc(Cl)c2cc(Cl)ccc2n1 CCC(C)(COC)C(=O)N1CCC(CNC(=O)C(C2CCCO2)C2CC2)C1 C(CC1CCC1)(C(=O)N=c1ccn(CF)[nH]1)NC(c1cc(CC2CC2)on1)=O C1(NC(c2noc(C)c2Br)=O)CCCC(NC(=O)CC2(O)CCC2)CC1 C1(C(=O)NC(C(C)C)C(=O)N(CCCCCO)C)CCC2(CC1)CC2 c1(C(C(C)C)N(Cc2snc(OC)c2Cl)CC2CC2)c(C)cccc1Cl CCN=c1[nH]c(C(N2CCCC(C)(CNC(C3CC3CCOC)=O)C2)=O)cs1 N1(C(C(CC)CC)=O)CCC2C(CCCN2C(c2c[nH]c3cc(Cl)ccc23)=O)C1 C(=O)(CCC(N)Cc1ccccc1)N1CC(CC(=O)O)C1 Cn1ncc2ncc(-c3nc(CCOC)nn3CCc3ccccc3F)cc12.CCF C(=O)(C(C)(C)CC(C)C)N1CC(CC(C(=O)NCCC(C(C)C)OC)F)C1 CP(C)(=O)C(C(F)(F)F)NC1CCC(O)CC1 C1(C(=O)NCCC2CCN(C(c3cn(CC)nn3)=O)CC2)CCC2(CCC2)C1 c1(C(N2CCCC(C(=O)NCCc3ccc(C)s3)C2)=O)cc(Cl)ccc1O c1(CCC(=O)NC(C(=O)NCC(=C)CC)c2cccs2)cncnc1 C1(OCc2c(C(=O)OC)nco2)CN(C(=O)CC2CN(C(C)=O)C2)CCC1(C)C C(C(CC1CCCC1)C(=O)NCCCC(=O)NC1CC(=O)NC1=O)N(C(C)C)C C1(C(=O)NC(C2(O)CCN(C(c3cc(Cl)c(Cl)s3)=O)C2)C)CCC2(CCC2)CO1 C(=O)(C(CCCc1cc(OC)no1)NC(=O)C(CN(C)C)N(C)C)OC c1(C(N(CCOC)CCNC(c2c(C)ccn2C)=O)=O)cc(C)nc(O)n1 C1(CNC(c2cc(C)no2)=O)CCN(C(=O)C(C)NS(C)(=O)=O)CC1C c1(C(=O)NCC2OCCN(C(CCCCC#C)=O)C2)sc2[nH]cnc(=O)c2c1C Oc1ncnc2ncn(-c3ccc(-c4ccc(Cl)c(F)c4)cc3)c12 N1(C(CCC(C)C)=O)CCN(C(C2(c3cnn(C)c3)CCCO2)=O)CC2(CC2)C1 Cc1cc(C2CCCN2CCCC(F)(F)OC(=O)Nc2ccccc2Br)ccn1 c1(CNC(C2(C)CCCN2CC)=O)cnn2c(C)cccc12 n1(CC(C)(C)C)ncc(Cl)c1C(=O)NC1CCC(NC(=O)CSC(F)F)CC1 C(=O)(CP(C)(C)=O)NC(C)(CNC(C1CCCN1c1ccncn1)=O)CO C(C(C)(C)C(=O)N1CCC(NC(C2CCC2(C)C)=O)C1)OC(C)(C)C CCCC(CC)C(=O)NC1(C(=O)NCC2CCCN2C)CC(CO)C1 C#CCC(C(=O)NC1CN(C(=O)COc2ccccc2)CC1O)C1CC1 C1(C(=O)NC(CC#C)C(=O)NC)C2CC3C(C2NC(C2CC(C)=NO2)=O)C13 N1(C(C(=O)NC2C=CC(C(=O)NC)C2)=O)CCOc2c(OC)cc(C)cc21 N1(C(c2c(C)cc(C)o2)=O)CCC(NC(c2nn(C)c(C)c2Cl)=O)C2(CCC2)C1 N1(C(CNC(CC(C)(C)C)=O)=O)CCCC2CN(C(c3sccc3F)=O)CCC12 c1(NC(C(CC)N(CC)CC)=O)ccc(N=S(C)(C)=O)s1.C12(CCC1)C(=O)N2CC c1(CC)oc2ccccc2c1C(=O)NCC#CCNC(=O)CC1CCC(C(N)=O)O1 CCCCC(CC(=O)NCC1(O)CCCC1)NC(=O)C=CC1CCOC1 c1(C2(C(=O)NCCCN(C)C(C3C(C)C3C3CCOCC3)=O)CC2)cccnc1 C1(CC(=O)NC2CCN(C(c3c(CCC)n[nH]c3)=O)C2)(OC)CCCCC1 c1(CC)cccc(C(=O)NC2CCC(CNC(C3(CO)CC3)=O)C2)c1N C(C(CCCC)N(C(=O)C=CCC1CCOCC1)CC)NC(C(F)=CC)=O C123CCC(CC1)(C2)SCCN3.C1(CCC)(OC)CCOC1 c1(C(N2CC(CC(=O)Nc3cc(C(F)(F)F)ncn3)C2)=O)cc(Cl)ccc1Br C1(NC(c2cc(-c3ccc(Cl)cc3)ns2)=O)C2CN(C(=O)CC3C=CCC3)CC12 N1(C(c2cn(CC)nn2)=O)CCCC(COC)(NC(C2CCC2(F)F)=O)C1 C(=O)(C(O)CC(C)(C)C)N1CC(CCCC)N(C(c2coc(Cl)n2)=O)CC1 N1(C(c2cncs2)=O)CC(C2CN(C(c3ccc(CC4CC4)cc3)=O)C2)C1 N1(CC(=O)NC(CC)CN(C(C2CCS2(=O)=O)=O)CC)CCC(=O)NC1=O C1(CC(=O)Nc2cnc(I)cn2)CN(C(c2cccs2)=O)CCO1 N1(C(Cc2n(C)ccc2)=O)CC(NC(=O)CC(=O)NCC2CC2)CC12CCOC2 N1(C(C2(C#N)CCC2)=O)CC2COCC(C1)C2NC(=O)CSC1CC1 C(=O)(C(CCC)CC(C)C)NC(CCCC)CNC(c1cnccn1)=O c1(C(N(CC(CNC(C(C)C2CCC2)=O)O)C)=O)ccc2c(c1)C(=O)C(=O)N2 c1(C(=O)NCC(CNC(=O)CCCn2ccnn2)OC)csc(Cl)c1 N1(C(C(N2CCSCC2)C)=O)CCCC(NC(c2ccc(F)c(Cl)n2)=O)CC1 C1(OC)CS(=O)(=O)C2CN(C(=O)Cc3ccc(Br)nc3)C12 CC1CCCN(C(=O)CC2CN(C(C3CCC3)=O)C(C)(C)C2)CC1 Cc1nc2c(o1)CCCC2CC(=O)N1CCC(NC(C2CC23CCC3)=O)C(F)C1 CCC(O)C(F)(F)C(=O)NC1CN(C(c2cnc(C3CCCO3)s2)=O)C1 C1(C(N(C)CC2CN(C(c3cnn(C(F)F)c3)=O)C2)=O)OCC2COCCC12 c1(C(=O)NC2CCCN(C(C(CC(=C)C)OC)=O)C2)ccc2nonc2c1 c1(C(N(CC(C)CNC(=O)C(=O)NCC2CC2)C)=O)cn2c(n1)CCC2 c1(C(=O)NC2CC(C(C)NC(Cn3ncc(CC)c3)=O)C2)n[nH]cc1[N+](=O)[O-] c1(C(=O)NCC(CC(C)C)NC(c2ncc(F)cn2)=O)cccn2nnnc12 C1(CNC(C2(C)CCCOC2)=O)CN(C(=O)CCOCC(F)F)C2(CCC2)C1 c1(C(N(C(CNC(C2C3CC4C(C3=O)C24)=O)C2CC2)C)=O)ccc2cnnn2c1 N1(C(=O)C=CCc2ccccc2)CC2(C1)CN(C(C1(c3cccc(F)c3)CC1)=O)C2 c1(C(=O)OC)cccc2c1CCNC2.C123CCC(CC1)(CC2)COC3=O Cc1nn2cc(C(=O)NCC3(C)CCCN3C(=O)CSC3CCCCO3)nc2s1 Cc1cc(C)c(C(=O)NC2CC(CNC(=O)CCn3ncn(C)c3=O)C2)cc1C C12CC13CN(C3)C2=O.c1(NC(CC)=O)ccn(C2CN(C(=O)OC(C)(C)C)C2)n1 N1(C(CCN(CCCCC)C)=O)CCC(C2(NC(=O)CCCNC(C)=O)CC2)C1 Cc1cc(C(=O)NC2CCN(C(=O)Cn3cccc3)C23CC3)ncc1S(N)(=O)=O C1(CCCC)CN(C(C2CC2C2CC2)=O)CCN1C(=O)Cc1csc(Cl)n1 C1(C(N(C)CC2N(C(c3onc(C)c3C)=O)CC(F)C2)=O)CCC(C)(C)OC1 c1(NCC(C)(C)NC(=O)CCc2ccc(F)cc2F)sc2ccccc2c1C=O N1(C(CN(C(=O)CN2CCC(O)C2)CCOC)=O)CCC2(CCOC2)CC1 Cn1ncc2c1CC(C(=O)NCC1(NC3C4COCC34)CC1)CC2 N1(C(Cc2c(C)n(C)nc2)=O)CCN(C(=O)C=CCN2CCCC2)C(C)C1 c1(C(=O)NCc2ccc(C(N3CC(C4CCCO4)C3)=O)s2)ccccc1C1CC1 c1(C(=O)NC2(CCCNC(c3cccc(C(C)C)n3)=O)CC2)cc(O)cc(=O)o1 Cc1ccc(C=CC(=O)NC2C3CN(C(C45CCC(CC4F)C5)=O)CC23)c(C)c1 CC1(C)CC(C(=O)NC2CCC(N=[N+]=[N-])C2)N(CC(=O)O)C1.N1(C)CCOCC1 CCC(CN(C(=O)C(C)NC(=O)Cn1cc(CC)cn1)C(C)C)CC N1(C(CS(C)(=O)=O)=O)CCN(C(c2cc3c(s2)CCC3)=O)C(C(F)F)C1 N1(C(c2n(C)nc(O)c2)=O)CCN(C(C2CN(C(=O)OC(C)(C)C)C2)=O)C2CC12 N1(C(C(CC=C)C(C)C)=O)CC=C(C(C)(C)C(=O)N2CC3CC(C2)C3(C)C)C1 N1(C(n2c(CC)ncc2)=O)CCCN(Cc2cnn(CCO)c2)CC1 c1(-n2cc(NCC3CC(NC(CC4CCC(=O)C4)=O)C3)nn2)cc(F)ccc1Cl C(=O)(CC(C(C)C)NC(C1(CCC)CC1)=O)NC(C=C)C(F)(F)F CCC(CNC(C1C(C(C)=O)C1(C)C)=O)(CC)NC(=O)C(C1CCCC1)OC c1(C(=O)NCC2CC(F)(CNC(C3CCN(C)C3=O)=O)C2)cccc2sncc12 C1(CC(=O)NCCNC(C(C)c2cccs2)=O)CC2OCCC2O1 N1(C(CS(C)(=O)=O)=O)CC(NC(=O)CCCCc2ccccc2)C(C2CC2)C1 c1(C=O)cccc2c1CCC2.CCC(C)C(C)N(C(=O)Cn1ccnn1)C C12(CC(=O)NCCCNC(C(C)C)=O)CCC1CN(C(c1c[nH]c(=N)o1)=O)C2 N1(C(CC2CCC(C)C2)=O)CCC2(CC1)C(NC(=O)CC1CN(C)C1)CS2(=O)=O Cn1c(CC(=O)NC(Cn2cncn2)C(=O)NCc2ccccc2)nnc1S c1(C(=O)NCC2(NC(=O)Cc3ccoc3)CCOC2)cnc2sccc2c1 C1(C(N(C)C)=O)CCN(S(=O)(=O)N2CCC(CSc3cnccn3)CC2)CC1 c1(COC(C2CCC3CN(C)CC32)=O)ccc2oc(O)nc2c1 C(=O)(CCNC(CC)CC)NCCCC.C12(CC1)N(C(C)C)C2=O c1(CN(C(C2CC2NC(c2cccc(O)c2)=O)=O)CC)c(O)ccc(Br)c1O C1(CNC(CCc2cc(C)[nH]n2)=O)CC(NC(=O)C=Cc2scnc2C)C1(C)C c1(OCC(=C)C)ccccc1C(=O)NC(C)(C)CCCNC(=O)C(O)C(C)OC c1(C(=O)NCC(F)CNC(c2cnc(S)[nH]2)=O)ccc(F)c(CC2CCC2)c1 c1(C(=O)NCC2CC3CN(C(C(C)CC4CC4)=O)CC32)ccc([N+](=O)[O-])n1C C1(CN(C(C2CC3(CC3)C2)=O)CC)CCC(CNC(=O)CC2CC(=O)C2)O1 N1(C(C2C(CC(C)(C)C)C2)=O)CCCCCC(NC(=O)CC2CCC(=O)O2)C1 C#CCC(CC#C)C(=O)NC1CN(C(C2(SC)CCC2)=O)CC1N1CCCC1 C(C(COC)CC(=O)NC1CC(O)CN(C(=O)CCCc2cnccn2)C1)OC c1(C(=O)NC(CC)CN(C(=O)C(CCO)OC)CC)ccnc2c1cnn2C c1(CNC(c2cc3cc(Cl)ccc3o2)C)c(Cl)c[nH]c2nccc1-2 C(=O)(C1=C(Cl)CCOC1)NC1C2N(C(C(CCSC)NC=O)=O)C(CC2)C1 N1(CC)CCC(NC(=O)CCCn2cc(C3CCCC3)nn2)C(C)C1 c1(C(N2CCN(C(CN(C(CC(C)F)=O)C)=O)CC2)=O)cc2[nH]ccc2s1 C(=O)(C(F)(F)CC1CC1)N(C1CCN(C(C2COC(=O)C2)=O)CC1)CC(C)C C#CCCC(O)C(=O)N1CCC(CN(C)C(C2(F)CC2)=O)C1 C1(CC(=O)NCC2CCC(NC(C3CC(C)C3)=O)CC2)CCC(C)(C)CO1 c1(C(=O)NCC2C(NC(C(CC)(F)F)=O)CCC2)ccc(F)c(C(C)=O)c1 C1(CNC(Cc2cc(C)sc2)=O)(NC(c2ccc(C#N)s2)=O)CCCCC1C CC1CN(C(=O)C(C2CCCCCCC2)O)CC(C)N1C(c1cnsn1)=O S(=O)(=O)(c1cnc(N2CCC(OC(F)F)CC2)c(Cl)c1)NCC1CCCC(C)C1 N1(C(COC(C)C)=O)CCOCC(CNC(=O)CCc2ccc(Cl)c(F)c2)C1 Cc1ccc(NC(=O)N(c2cccc(F)c2NC(c2ccccn2)C)C)c(C)c1 C12(C(=O)NC(c3occ(C(=O)NC(CSC)CO)n3)C)CCC(OC)C1C2 c1(CC(=O)NC(C2(C(=O)NC(=O)Cc3ccco3)CC2)C)cccnc1Br Cc1csc2ncc(C(=O)NC(C)C(C)(C)NC(=O)C(C)(F)F)c(=O)n12 N1(C(c2n(C(C)C)ncc2)=O)CC(CNC(=O)Cn2cccnc2=O)C(C)C1 CC1(C)CC(NC(c2ccoc2)=O)CCN(C(=O)Cc2ccc(Cl)s2)C1 C1(C(C=O)(C)C)CCCN(C(C2(C)CCN(C)C2)=O)C1.C(CCCCC1CC1)OC c1(C(=O)NC(CN(C(C(CC)OC)=O)CC)C)sc(C)nc1C(F)(F)F Cn1cncc1CNC(=O)Cc1csc(N2CCCC2=O)n1.C12(CCC1)CC(=O)N2 Cc1noc(C)c1CCC(=O)NCC1COCCN1C(C1CCCC1(F)F)=O Cn1ncc(C(=O)NC2CN(C(C3(CF)CC3)=O)CC3(CC3)C2)c1S(C)(=O)=O c1(C(=O)NCC(CNC(C2(COC(C)C)CC2)=O)O)ccn2nccc2n1 C1(NC(c2c(C)ocn2)=O)C(C)(C)C(NC(=O)C(O)CC2CCOCC2)C1(C)C c1(OCCCOC)ccc(C(=O)NC(C)CCNC(=O)CCC=C(C)C)cn1 C(C1=CCN(C(=O)CCc2nc(C)c(C)o2)CC1)NC(c1c(SC)cccc1)=O C1(NC(C(CCC)O)=O)COC2C(NC(=O)CCc3c(C)noc3C)COC12 C(c1ccccc1C(F)(F)F)=CC(=O)NC(CSC)C(=O)N(C)CCO C1(NC(C(CC#C)NC(c2nn(C)cc2C)=O)=O)CC(C)N(C)CC1C C(=O)(C1CCCc2n[nH]cc21)NC(C(C)NC(=O)CCCCN(C)C)CO C#CCCCCCNC(C1(CC)C=CCN1C(C1SCC=C1C)=O)=O Cc1cc(C(=O)NCC(CNC(=O)CCc2ccccn2)CO)nc(O)n1 C1(C(=O)Nc2cc(F)cc(I)c2)CN(C(c2sccc2I)=O)CC(F)(F)C1 C(=O)(CC(C)(C)CC(=O)NC1CC(O)CN(C(=O)C2CCc3c[nH]nc32)C1)OC C1(NC(C(C)C2CC2)=O)Cc2ccccc2C1NC(c1cnsn1)=O C(=O)(CCC(C(=O)N1CCOC(CN(C(=O)CC(=O)N(C)C)C)C1)N(C)C)OC c1(C(N(CC(=O)O)Cc2ccccn2)=O)cccc(SCc2n[nH]cc2Br)c1 n1(C(C)C)cnc(C(=O)NC2CC(C(F)C(=O)NC(CN3CCCC3)CO)C2)n1 c1(OC)cc(-n2nc(CCO)nc2C2CCCN(CC(F)(F)F)C2)ccc1F C1(C(N2CCC(CF)C2)=O)(NC(=O)C(O)CC2CCCC2)CCCCC1 C(=O)(CC1=NNC(=O)C1)NCC1CN(C(c2nc(CC)oc2)=O)C(C)CC1 C=CC1(CC(=O)NCC2CCN2C(c2cscn2)=O)CCC1 c1(C(N2CCC(CNC(c3ccc(C(C)=O)[nH]3)=O)C2)=O)[nH]cc2c1CCCC2 c1(C(C)(C)C)ccc2oc(CN(C(N)=O)CC3CC34CCOC4)cc2c1 N1(C(c2cc(F)cc(C)c2O)=O)CCC=C(C(=O)NOC2CC2)C1 CC(C)(C)CC(O)CC(=O)NCCCN(C(=O)CC(F)(F)F)Cc1ccccc1 C1(C(=O)NC2CN(C(c3c(OC)scc3)=O)CC2O)CN2CCCCC2CO1 C1(CC(=O)OC)C2CCC(C2)N1C(C(=O)NCC1CCOC1)c1ncco1 c1(C(N(CCC(C(C)C)NC(C(C(=C)Cl)(C)C)=O)C)=O)ccc(S(=O)CC#N)cc1 C(=O)(C(Cc1ccccc1)S(C)(=O)=O)N1CC(NC(CC=CC=C)=O)C(F)C1 C1(C(=O)NCC2(NC(COCCOCC#C)=O)CCOC2)CC2CCC(C1)N2C C12(NC(C(CC)=CC)=O)CCC(CC1)N(C(=O)C(C(C)(C)C)OC1CCCC1)C2 N1(C(c2c(OC)cccc2Cl)=O)CCC(C2CCN(C(=O)COCC(C)C)C2)C1 N(C(=NCCC=C(C)C)NCC1(N2CCOCC2)CCCCC1)CCSC CC(O)CCCC(=O)NC(C)CCN(C(=O)C1=NNC(=O)C1)C C(=O)(CCCCCN=[N+]=[N-])N.CC(C)CC(C(=O)N1CCCN(CC)CC1)N(C)C Cn1cc(C(C(F)F)NCCC2(C)CCN2C(=O)OC(C)(C)C)nn1 Cc1cc(N2CCC(C(C)NC(=O)CC(C)C(F)(F)F)C2)ccc1[N+](=O)[O-] c1(C(=O)NCC2CCN2C(=O)Cc2ccc(Br)cn2)nc2ccccc2s1 C=C(Cl)CC(C(=O)N1CC(C#N)(SC)C1)NC(=O)CC1CCCOCC1 C(C)(C)(C(C)NC(=O)C(=O)NCCC1CCOC1)OC Cn1ncc2c(N3CC4(CC4)CC3CNC(C3(C(F)F)CC3)=O)ncnc12 c1(C(=O)NC(C2N(C(CSCC)=O)CCCC2)C)cc(OC)cc(OC)c1 c1(C(=O)NCc2cccc(NC(C3C(C)COCC3)=O)c2)ccc(F)c(N)c1 c1(CNC(CC(=O)Nc2cc(CSC)c(Cl)cc2)=O)nc2cnccc2s1 N1(C(C(c2ccccc2Cl)C)=O)CCC(NC(=O)C=CC(C)(C)NC(C)(C)C)CC1 N1(C(CC2N(CC)CCOC2)=O)CC(O)(C2(CNC(=O)CNC(C)=O)CC2)C1 C1(CCNC(C(COC)(C)C)=O)CN(C(C2(SC)CC2)=O)C(C)(CSC)C1 N1(C(c2cc(OC)ns2)C(=O)NCCCSC)CCS(=O)(=O)C2(CCCCC2)C1 O=C(C1CCOc2ccccc21)NCC1CCCCN(C(C2CCC(=O)O2)=O)C1 n1(CC)nnc(C(N2CCCC(C(C)NC(=O)C=CCO)C2)=O)c1C CC1CN(C(c2ccc(CC#N)cc2)=O)CCCN1C(C1CCC1C(F)F)=O O=C(CC1=CCOCC1)NCC1CN(C(=O)CCc2ccncc2)CCO1 CC1CCCn2ncc(C(=O)NC3CCCCN(C(=O)CCc4ccco4)C3)c21 N1(C(c2c(CC)nn[nH]2)=O)CCC2(CC(NC(=O)C(C)=CC(C)(C)C)CO2)C1 C(=O)(C(C)(C)CNC(c1csc(=N)[nH]1)=O)NCc1cnc(CC)[nH]1 N1(C(C(c2cn(C)nc2)(F)F)=O)CCCCC1CNC(=O)CC1CCNC1=O C(c1cccc(F)c1F)=CC(=O)NC(C1CN(C(C2(C)CCCN2C)=O)C1)C Cc1cnc2c(cnn2CC(=O)NC(CNC(=O)CCc2cnn[nH]2)C2CC2)c1 c12cccc(F)c1C2NC(N(C)CC1(N(C)C)CCC1)=O.c1(C)ccccc1 N1(C(C(C)NC(COC)=O)=O)CCC(N(C(c2cc(CO)c(C)o2)=O)CC)CC1 C1(NC(C(C=C)O)=O)CC2CCC(C1)N2C(=O)C(COC)CC Cc1ccc(C(=O)NC(C)CCCNC(C2CC2c2cnc[nH]2)=O)c(N)c1 Cc1cc(C(F)(F)F)cc(F)c1.N12CC(F)CC1C2=O.c12ccnc(c1)CN2 C1(N(C(C(C)OCC)=O)CC)CCCN(C(c2ccnn(C)c2=O)=O)CC1 N1(c2cc(C)nc(N3CC4COCC4(C)C3)n2)CC(N)C2(CCC2)C1 C(CC(=O)NC(C(=O)N(CC(O)COC)C)c1cccs1)OCC#C C(CC(F)F)(C(=O)N1CCC2(CCO2)C1)NC(=O)CC1CC(CF)C1 C1(C(=O)NC(CN(C(c2cnn(C3CCC3)c2)=O)CC)C)CCCN1C c1(C(=O)NC(C(C)C)(C)CNC(=O)C(C)CSC(F)(F)F)cc2ccccc2o1 O(NC(=O)CS(=O)(=O)NCC)C(C(=O)N1CC(CC=C)C1)CC(C)C c1(C(=O)NC2CN(C(C3CCCC(C)C3)=O)C2)ccn2c1CS(=O)(=O)CC2 c1(C(=O)OCC)cc([N+](=O)[O-])ccc1S(=O)(=O)N1CCc2cc(Cl)ncc2C1 n1(CC)cnc(C(=O)N(C2CCN(C(=O)C=CSCc3ccco3)C2)C)c1 C1(O)(C(C)NC(C=CCC)=O)CCN(C(=O)CSCc2cccs2)CC1 C(=O)(CC1=CCCCC1)NC1CCN(C(c2c(C)cccc2N)=O)CC1 N1(C(C)C)CC2CC(N3CCC(CC(N4CCCC(C)CC4)=O)CC3)C1C2 c1(OC)ccc(CCC(N2CCCCC2C(=O)NCC#N)=O)cn1 c1(C(N(CC(C)N(C(C(CC)SC)=O)C)C)=O)ccc(N(C)C)c(OC)c1 CCCCCC(O)C(=O)N1CCCC(C)(C(=O)NCC2CCS(=O)(=O)CC2)C1 C1(C(=O)NC2CC3CN(C(C(COC)(F)F)=O)C2C3)Cc2cc(F)cc(F)c2O1 C1(NC(C=C(COC)C)=O)C2CCN(C(=O)C=Cc3nc(C)cs3)CC12 C1(C(=O)NCC(C)(O)CNC(C2COC(=O)N2)=O)CCOC2(CCCC2)C1 c1(-c2cc(NC(c3cnc(OC)c(C)c3)=O)ncc2)cccc(C#N)c1F c1(C(N2CCCC(N)C2)=O)cc([N+](=O)[O-])ccc1NCC1COC1 C1(C2CCC2)(C(=O)NC2CN(C(C(c3cn(CC)nc3)=O)=O)C(C)C2)CC1(F)F c1(C(=O)NC(C2CCCC2)CNC(c2c[nH]c(C(F)(F)F)n2)=O)ccc(Cl)nn1 C1(OC(c2nc(-c3cc(Br)ccc3F)cs2)C)CCC(F)(F)CC1 N1(C(CSC(C)C)=O)CC(C(=O)NCC2=CCCC2)C(C(C)C)C1 c1(N(CCCNC(c2c(C)scn2)=O)C2CC2)nc2c(cc1C#N)CCCC2 CC1CCN(C(=O)CNS(=O)(=O)N(C)C)C1CNC(=O)CCC=CBr Cc1nnc2n1CC(C(N1CC(CNC(=O)CCC(C)c3cccs3)C1)=O)CC2 C1(C(N(CCC(N2CCC(C)(OCC)C2)=O)CCCO)=O)CC2(CCO1)CC2 Cc1ccc(C(C)N(C(=O)CCCn2cccc2)C)nc1.C12CCCN(C1)C2=O C1(C(=O)NC(CC)CN2CCCC2)CN(C(C2(CC)CCCCO2)=O)CC1(F)F C1(CC(=O)NCC(CCOC)(C)C)CN(C(C2COC(=O)N2)=O)C(C)(C)C1 C(CC(=O)Nc1nnnn1C1CC1)(C(F)(F)F)NC(=O)CN1CCC(O)CC1 C1(c2ccccc2)(CC(=O)NCC(C)N(C(C(CC)SC)=O)CC)CCOCC1 c1(NC(C2C(CC)CCN2C(=O)C(C)OCCOC)=O)ccc(O)c(Cl)c1 C(=O)(C(C)C1=CCCC1)NCC1CC(NC(c2c(CC)c[nH]n2)=O)C1 c1(C(N2CCC(C(=O)NCCCc3ccccc3Cl)C2)=O)n[nH]c2c1CCC2 C(CCC(=O)NCC1CC1CNC(=O)CCc1cnn[nH]1)SC c1(OC)cc(C=CC(=O)NCC(O)CNC(c2cncc(SC)c2)=O)ccc1O c1(N(C(C)CNC(=O)Cc2cc(OC(F)F)no2)C)ncc(Br)cn1.CCC N1(C(C(CC)(C)Cl)=O)CC2CCCC2(CNC(c2ccncc2C2CC2)=O)C1 CC1CCCCC1(CO)NC(C12CC(CN1C(=O)CN1CCC(F)CC1)C2)=O Cc1nc2ncccn2c1C(=O)NCC1CCN(C(c2ccc(Br)c(O)c2)=O)C1 n1(CC)nnc(C)c1C(=O)NCCCCC(C)NC(=O)C(C1CCC(=O)N1)C C1(NC(c2nc(NC(C)=O)sc2)=O)CN(Cc2cc(C)on2)CCCO1 c1(C(=O)NCC(CC)NC(C2(C)CC(C)=NO2)=O)cc(C(F)(F)F)ccc1OC c1(C(=O)NCC(CNC(c2cc(C)sc2)=O)C)ccc(Cn2cncn2)cc1 C(=O)(CS(=O)(=O)C1CCCC1)NCC1(C)N(C(CC(CC)CN(C)C)=O)CCC1 C(=O)(C1CCc2nccn21)N1CCC(NC(=O)CCOCNC2C(O)CC2O)C1 C#Cc1cccc(C(=O)NC2(CNC(c3ccsn3)=O)CCC(C)(C)CC2)c1F C(=O)(C(CCNC=O)CC(C)C)N(C(CC)C(=O)OC(C)(C)C)CC(C)C.OC c1(C(=O)NC2CCN(C(C(C=C)O)=O)CC2F)cc2sccc2cn1 CC(F)(C(=O)N1CCC(NC(=O)CCCSC(C)(C)C)C(CO)CC1)C(F)(F)F N1(C(C2CCN(CC)C2)=O)CC(C(=O)Nc2c(C)noc2C(C)C)C(CC)C1 C(=O)(C(C#N)C(C)(C)C)NC1CC2(CC(CNC(c3c(C)cco3)=O)C2)C1 Cc1cccc(C(=O)NC2CCCN(C(=O)COc3ccc(F)c(Cl)c3)C2)c1F C=CC1CN(C(=O)COCC2CCOC2)CC1NC(=O)CNC(=O)CCC(C)C C1(OC)(CNC(=O)CSC)CCN(C(=O)C(Cc2ccccc2)SC)C1 N#CCCCC(=O)N1CCOCC1CCNC(C1(c2ccncc2Cl)CC1)=O c1(C(=O)OC)ccc(NCCN(C)C(c2ccc(S(C)(=O)=O)cc2)=O)c(C#N)n1 C#CC1CC(NC(=O)C(C)(C2(C)CC2)NC(=O)CSCCC)C1 Cc1ccc(Cl)c(O)c1C(=O)NC1CC1CNC(c1ccc(F)cc1C1CC1)=O C(=O)(CN=c1ccc(Cl)n[nH]1)N1C(CNC(c2n3c(nn2)SC(=C)C3)=O)CCC1 C1(NC(=O)CC2OCCO2)C2CCC(C2)C1C(=O)NCC12CCC(CO1)C2 CCC(CC)(CC)C1C(=O)N1.c1(CNC(C)=O)[nH]c(OC)nc1Cl c1(C(=O)OC)cccc(C(C)=O)c1.c12ccc([nH]1)C(=O)N(C)C(C)CNC2=O N1(C(CCSC)=O)CCC(C(=O)Nc2cc(C)ccc2OC(F)(F)F)C(C)(C)C1 N1(C(CCC=C)=O)CCOC2(CCN(C(C3CC3(Cl)C(=O)OCC)=O)C2)C1 N1(C(C2C(C=C)C2)=O)CCSCC1CCNC(=O)C=CCOC1CC1 Cc1ccc(-c2nc(CC(=O)NCc3ccsn3)cs2)s1 CCCCCC(=O)NCC(C)N(C(=O)C(CCC)NC(N)=O)C C(=O)(C1CCCc2ccccc21)N1C(CCC)CN(C(=O)CCC(F)F)CC1 c1(C(=O)NC(C2CCN(C(c3cnsc3)=O)CC2)(C)C)ncc[nH]c1=O c1(C(=O)NCCC(C(C)C)NC(=O)C2=C(Cl)CC2)c(F)cccc1[N+](=O)[O-] C(=O)(CC(C(C)OC)NC(c1c[nH]c(=O)cn1)=O)NC(C(=O)NC)CCC1CC1 c1(C(N2CCC(C)(c3cn(C4CCNCC4O)nn3)C2)=O)nccc2cc[nH]c12 CC1CC2(CCN(C(=O)CC3CCC(=O)NC3)CC2)CN1C(C1CCCCO1)=O CC1(C)CC(C(N2CCC3(CC2)CC3)=O)CN(C(C2CCC([N+](=O)[O-])CC2)=O)C1 N1(CC(N)=O)CCCCC1C.CC(C)C(Cc1nccn1C)N c1(CSC)ccc(-c2nc(Cc3ccccc3F)nn2Cc2ncccn2)cc1 C1(C(=O)NCc2ccc(N(C)C)c(F)c2)CCOCC12CCCC2 C1(NC(C2(NC(C(C(C)C)F)=O)CCN(C)C2)=O)CC2CCCC(C1)C2 CC12CCC(=O)N1C(C(=O)NC(CNC(c1ccncc1F)=O)CO)CS2 C(C(CO)C(C)(C)C)NC(c1cc(CNC(c2c(C)cc(C)s2)=O)[nH]n1)=O c1(CN=C(NCCOC)NC2CC2C)ccc(C#N)c(F)c1 C1(C(=O)NCC(C2CC2)NC(CCCc2onc(C)n2)=O)CC(C)(C)CO1 N1(C(C2CC(=C)C2)=O)CC2CCCC2(CNC(c2cc(CC3CCC3)c[nH]2)=O)C1 C1(NC(c2c(C)cccc2C)=O)CN(C(c2cn(CCO)nn2)=O)CC(F)(F)C1 c1(C(N(C(C)C)CCNC(=O)COCCF)=O)c(O)nnc2c1CCCC2 Cc1cc([N+](=O)[O-])cc([N+](=O)[O-])c1N1CC2(C1)C(NC(=O)C(C)O)CCS2(=O)=O c1(CNC(=O)NC2CCN(CCC)C2)nn(C)cc1Br C#CCCCCCC(=O)NCC1(C)CCCC1NC(c1ccccc1OC(F)F)=O C1(CCOC)CN(C(=O)C(c2ccccc2)OCC(F)F)CCN1C(=O)COC C(CO)(CC(F)(F)F)NC(=O)Cc1ccc(Cl)cc1 C1(CNC(c2c(C(C)C)occ2)=O)CCCCC1NC(=O)COC1CC1 c1(OC)ccccc1OCC(=O)NC1(CN(C(=O)CC(C)C2CCCO2)C)CC1 c1(N2CCC(CNC(=O)C(c3ccccc3)F)C2)cc(C(F)(F)F)nc(Cl)n1 c1(C(N2CCOC(C(=O)NCC3(C(=O)OC)CC3)C2)=O)cc(Br)ccc1I c1(NC(C#CC)=O)ccc(C(N2CCCC2c2ccncc2)=O)nc1 N1(C(COCCC#C)=O)CC(F)(F)CC1CCNC(c1ocnc1C(F)(F)F)=O CC(CCC(C)(C)C)NC(=NCC1CCN1C1CC1)NCc1ccccc1Br c1(CC(=O)NCCN(C(=O)CC2CCCCC2C)CCC)n[nH]c2c1CCCC2 C12(NC(CNC(C)=O)=O)CCCC1N(C(=O)CC1CC3CCC1C3)CC2 N1(C(=O)Nc2cc(C)sc2)CCS(=O)(=O)CC1C1CCC1 CC(O)(CC(=O)NC1CN(C(C2CC3(CCC3)C2)=O)C1)C1CC1 CC1(CC(=O)NC2CCC(C(N)=O)C2)CN(C(C2CC2c2ccco2)=O)C1 N1(C(c2scc(OC)c2)=O)CCC2C(CCCN2C(=O)CCc2cnoc2)C1 c1(C(N(CCC(=O)NCC2CCN(CC)C2)C2CC2)=O)ccc(C)cc1 c1(CC(N2CCC(C)(NC(C(C=C=C)C)=O)CC2)=O)cc2cccnc2nc1C C(C(CC(C)C)NC(=O)C(C)CCc1ccccc1F)NC(C1(C(=O)NC)CC1)=O c1(C(=O)OC2CCN(C(=O)COc3ccsn3)C2)ccc2oc(O)nc2c1 C1(CNC(c2cnc(C)nc2C)=O)C2CCCC1N(C(=O)Cc1csc(C)c1)C2 C1(CC)CCCN(C(=O)CC(COC)NC(=O)Cc2cccnc2O)C1 N1(C(C2(OC)CC2)=O)CCCC(C2CCCCN2C(=O)CCCSC(C)(C)C)C1 c1(CN2CC(CNC(c3ccc(C)s3)=O)OCC2)c[nH]c2cnccc12 c1(N2CC(NC(C(C)(O)C(F)(F)F)=O)C(F)(F)C2)ccn2ncc(Br)c2n1 CCCCC(=O)C(=O)N(CC(C)(C)CNC(C1CCOC(CCC)C1)=O)C N1(C(c2ccn(CC)n2)=O)CCC2(CCCCN(C(=O)C(C)c3ncco3)C2)C1 C1(NC(C2(CC#C)CCCO2)=O)CN(c2nnc(CO)s2)C2(CCOCC2)C1 c1(OC)cc(-n2nc(C3CC=CCC3)nc2Cn2c(C)csc2=O)ccc1Cl Cc1cccc(F)c1C(N1CCC(F)C(NC(c2cc(Br)c[nH]2)=O)C1)=O c1(COC)nc(NCc2cc(Br)ccc2C)cc(=NCCC2CCCN(C)C2)[nH]1 c1(C(N(C(CNC(c2ccc(OCC#C)cc2)=O)C)C)=O)cccc(S(C)=O)c1 N1(C(Cc2ccc(CC(C)C)cc2)=O)CCN(C)C(CNC(=O)C2=CCCC2)C1 N1(C(C=C(CC)CC)=O)CC2CC(CNC(c3ccc4occc4c3)=O)CC1C2 N1(C(C2C(=C)C2)=O)CC(C)(C)C(NC(=O)CCSCCC)C(C)(C)C1 S(=O)(=O)(c1cccc(=NCCNS(C)(=O)=O)[nH]1)NC1C(SC)CCC1 Cc1ccc2[nH]c(C(=O)NCC(C)CNC(C34COC(CCO3)C4)=O)cc2c1 c1(CC(=O)O)cn(CCSC2CCC(C(=O)O)C2)nn1 N1(C(c2coc(C(F)F)n2)=O)CC(C(N2CCC(c3cc[nH]n3)C2)=O)C2(CC2)C1 C1(C(C)NC(C=CC)=O)CCCN(C(c2cc(O)n(CC)n2)=O)C1 C12(C(=O)NC(CC=C)CNC(=O)C(CO)N(C)C)CCC(CC1)CC2 CC(C)CC(=O)NC(CC1CCC1)C(=O)N(C(C)CN1CCCCC1)CCO c1(SCCCC(N2CC(C(C(=O)OC)CN(C)C)OCC2)=O)ccc(F)cc1 N(C1c2ccccc2CC1NC(C1(NC(N)=O)CCCCC1)=O)C(C=CCC)=O N1(C(CCC(C)NC(CC(CC)SC)=O)=O)CC(=O)NC(C2CC2)C1 C1(C(N(C)CC2(NC(c3ccnnc3O)=O)CC2)=O)CC1C1CCCC1 CC1COC2(C1)CN(C(C1CCC(NC(c3ccnn3C(F)F)=O)CC1)=O)C2 n1(CCC)nnnc1C(c1cnoc1)NCC1(Oc2ccccc2)CCCC1 N1(C(CCNC(C(=CC2CCCC2)C)=O)=O)CCCC(C)C1C(N)=O C1(NC(C(C2CCC2)OCC)=O)CN(C(=O)CN(S(C)(=O)=O)C)CCC1F C12(C(=O)NC(C(=O)OC)C3CC3)C(NC(=O)C(C)N3CCCC3)C3CC1C2C3 N1(C(C(=O)NC2CC2)CC2CCC2)CCC(C2OCCO2)CC1C(F)(F)F C1(CN(c2nnc(CC)o2)CC)CCCN(C(=O)CSc2cnn(C)c2)C1 C1(C(N2CC(n3cc(-c4ccc(F)c(Br)c4)nn3)C2)=O)CCCC(C(F)F)CC1 N(C(=NCCN(C)C)NCc1noc(-c2ccccc2)n1)C1CCC(SCC)C1 C(CCCCC(=O)Nc1cccc(CO)c1)N(C(C(n1ncc(C)c1)C)=O)C c1(CC)nc(C(=O)NCCNC(=O)C(C)C2CCOC2)co1 C12(NC(c3ccn(CC)n3)=O)CC1CN(C(=O)C(c1ccc(Cl)cc1)(C)O)C2 c1(-n2ccc(C(=O)NCC(C)CNC(c3cnnn3C)=O)n2)ccc(Cl)c(F)c1 Cc1cnc(Cl)c(NC2(c3nnnn3C3CCCCC3)CCCC(C)C2)c1 CC1C(NC(=O)CC2CCC(=O)NC2)CCCN1C(c1ccc(C(=O)O)nn1)=O c1(CC)ccc([N+](=O)[O-])cc1C(=O)NC1CN(C(c2cc(C)c(C)o2)=O)CC1C C1(NC(C=C(COC)C)=O)CCOCC1CC(N1CCC(c2cc[nH]n2)C1)=O C(=O)(C(C(C)C)NC(C)=O)NC(C(=O)NC1CC(OCC)C1)C1CCCC1 CCCC(O)CC(=O)N1CC(=C(F)CNC(c2nncn2C)=O)C1 c1(C(N(CCNC(C(C2CCCCC2)C)=O)C)=O)cn(C)nc1Cc1ccco1 C(=O)(CCCCCCCBr)N1CCC(CCNC(CN2C(=O)CCCCC2)=O)C1 Nc1cc(C(N2CCC(NC(C3CC=CCO3)=O)C2)=O)ccc1-n1cnnc1 C1(CCO)(NC(C2CC(CCC)C2)=O)CN(C(c2scnc2C)=O)C1 CCC(CC)C(O)CNC(C1CCC(CNC(C2CCCC(C)(C)C2)=O)O1)=O N1(C(CC(C)O)=O)CC23CCCC2(C1)CN(C(=O)C=Cc1ccncn1)C3 C1(COC)CC(CNC(c2ncccc2CO)=O)N(C(=O)CCSC2CC2)C1 c1(OC)ncc(Cl)cc1C(N1CCC(NC(c2cn(C3CCOC3)cn2)=O)C1)=O Cc1cc(C(=O)NC(C2CCCN(C(=O)Cc3cn[nH]c3)C2)C)cc(C)c1F N1(C(C(C)OC(C)=O)=O)CCC2(C=C(C(=O)NCC3CC=CCC3)C2)C1 Nc1ccc(C(=O)NC2CCCC(NC(=O)Cn3ccnn3)C2)nc1Br C1(C(N(C2CCCC2)CCNC(C2(C)CC2(Cl)Cl)=O)=O)CCn2cncc2C1 S(=O)(=O)(c1ccccn1)N(c1nc(OC)c(F)cn1)C1CCNCC1F c1(NC(C23C(CN(C(c4ccc(Br)s4)=O)C2)C3)=O)cccc2cccnc12 c1(OC)ccc(Cl)c(CN(CC(=O)O)C(C2CC(F)CN2C(C)=O)=O)c1F N1(C(CCC#CC)=O)CCCC(F)(CNC(c2ccc(CC(C)C)nc2)=O)C1 c1(CC(=O)NC2(CNC(=O)CC34CC(C3)C4)CCC2)ccc2ccccc2c1 C#CC1CCN(C(=O)C(CCOCC)NC(C2CCCN2CC)=O)C1 C(=O)(CCCC(F)(F)CO)N1CCN(C(C23C(C)OC(CO)(C2)C3)=O)CC1 C(=O)(CC1COc2ccccc21)NC1CC(CNC(Cc2cn(C)nc2)=O)C1 C12(C(N3C4CC(CNC(CC(C)C)=O)C3CC4)=O)CC3CC(CC(C3)C1)C2 N1(C(C(C)c2cccs2)=O)CC2CCC1CC2NC(=O)CCC(N)=O C1(CNC(C2C3CC4C(C3)C24)=O)C2CCCC1N(C(c1cn[nH]c1)=O)C2 S(=O)(=O)(c1ccc(Cl)cc1F)NCC(=O)NC1(C2ON=C(C(=O)OC)C2)COC1 C12(NC(C(CC)SC)=O)CN(C(c3cnccc3Cl)=O)CC1CS(=O)(=O)C2 c1(C(c2n(CCC)nnn2)NCc2cc[nH]n2)cnc(C(C)C)nc1 CC1CN(C(C2C(CNC(C34CC(C#N)(C3)C4)=O)C2(C)C)=O)CC1(C)CO CN(S(=O)(=O)N1CCCCC(S)C1)C.c1(N(C)C)ccc(C(F)(F)F)cc1 C(C1CCCc2ccccc21)ONC(CNC1(N)CCOC1)=O C(=O)(C1CCc2nccn21)NC(C)(CNC(C1CSC1)=O)C1CCC1 Cc1cccn(CC(N2CC3(CCC3NC(C3CC=CCO3)=O)C2)=O)c1=O CS(=O)(=O)c1cc(C(=O)NCC2CCC2NC(=O)Cc2ccccc2)ccc1F C1(OC)CN(C(=O)Cn2cc(C(OC)OCC3CC3)nn2)C(C)(CN(C)C)C1 N1(C(C(CC)SC)=O)CCC2(CC1)CCN(c1cc(Nc3nncs3)ncn1)CC2 C12(CNC(c3nc(CC(C)C)sc3)=O)CC1CN(C(=O)CCCc1ccsc1)C2 C1(C(=O)NC(C)=O)CCCN(C(c2cnccc2-n2cccn2)=O)C1.C1C=CC1 Cc1cccc(CCC(N2CCC(O)C2C(N)=O)=O)n1 CCCCCCOCC(=O)NC1CC(N(C(=O)C(C)(C)OCC=C)C)C1 C(C(C(=O)NC(CNC(c1ccc(Cl)nc1N)=O)CC)C(C)(C)C)OCC=C C1(C(N2C3CN(C(c4c(CC)non4)=O)C(CC3)C2)=O)COc2ccccc2C1 C1(C(=O)NCC(CO)NC(CCC)=O)(COC)CCCCCC1 CC(CN(C)N1CCOCC2(CCOC2)C1)c1cccc(C(F)(F)F)c1 C1(C(=O)NC)(COC)CC=CC1.C1(OC)CC1NC(=O)CC(=O)NC1CC1 c1(C2(C(=O)NCC#CCNC(c3cn(C)nc3)=O)CC2)ccc(Cl)cc1Cl C(=O)(C(C)CC(F)(F)F)NCC(C(=O)N1CC(CC(=O)OCC)C1)O N#Cc1ccc(OCC(=O)Nc2cc(N3CCCC3)nc(Cl)c2)nc1 C1(NC(CC2CC(=C)C2)=O)CCCN(C(=O)C(O)C(F)F)C1C C1(C(=O)NCC2C(NC(c3ccncc3)=O)CCCC2)CCCC12CC2 N1(Cc2c(C)c(F)ccc2)CCC2CC(Nc3nnnn3C)CCC2C1 c1(C(N2CC(C)CC(CNC(C(CCC#C)O)=O)C2)=O)ccc(F)c(Cl)c1F C(=O)(C1=C(Cl)CCC1)NC1CC(C)(NC(c2c(C)coc2C)=O)C1 c1(C(C2C(C)(CO)C(=O)OC2C(C)(C)C)=O)cc2ccncc2cc1F N1(C(C=CCN(C)C)=O)CC(NC(=O)CC2CCC(C)(C)O2)C(C(F)F)C1 C1(C(CNC(C(C=C)C)=O)O)CCN(C(C2(C)CC2(Cl)Cl)=O)CC1 C1(NC(c2ccccc2)=O)CCC12CCN(C(=O)CCN1CCCCC1)CC2 c1(C(N2C(CNC(c3cc(C4CC4)no3)=O)COCC2)=O)cc(F)ccc1O c1(-n2c(C)ncc2)nccnc1NC(=O)NC1CC(CC(N)=O)C1 C1(C(N2CC(NC(c3ccc(C)c(Cl)c3)=O)C(F)C2)=O)CCC2C(C1)C2(F)F N1(C(c2csc(C)c2C)=O)CC(=O)NCC1C(=O)Nc1cccc(C(N)=O)c1 CCCC(C(O)C(=O)N(C)Cc1cnn[nH]1)NC(C1OCCCC1(C)C)=O C(=O)(N=c1[nH]n(C)c2ccc(I)cc12)C1N(CCC)CCCC1 c1(C(=O)NCCCCC(C)NC(=O)C=CS(C)=O)cc(Cl)cc2cccnc12 c1(C(N(CCNC(c2c(CC)scn2)=O)C(C)C)=O)ccc(C2CCOC2)cc1 C(=O)(CCC(=O)c1ccc(Br)cc1)N(C)CC1CCCCC1F C1(C(N(CCCNC(c2ccc(OC)o2)=O)CCO)=O)CCCNS1(=O)=O C1(NC(C)=O)CC(NC(=O)NCCS(=O)(=O)N2CCCC2)C1(C)C C(C(O)CC(F)(F)F)NC(C1(NC(C2CNC(=O)C2)=O)CCN(C)C1)=O N1(C(C=CC(CC)C)=O)CC(C(=O)NCCn2ccc(=O)cc2)C2CCCC12 c1(OCCC(=O)NC2CN(C(c3ns[nH]c3=O)=O)C2)ccc(Cl)cc1 N1(C(CC(CN(C)C)O)=O)CCC(NC(c2ccnc(CO)c2)=O)C12CCC2 Cc1cc(F)ccc1CCNC(=O)CC1CCCCOC1 c1(C(N2CCC(C)(NC(C3CC4(F)CC3C4)=O)C2)=O)cccc2occc12 CC1CCc2ncc(C(N3CC4C(CNC(c5ccc(Br)o5)=O)C4C3)=O)n2C1 C(CC(C)C(=O)NC1CC(C)(C(=O)NC2(C)CS(=O)(=O)C2)C1)OC CCC(O)CC(=O)N1CC(O)CC1c1cn(-c2ccc(Br)nc2)nn1 N1(C(CCCC#C)=O)CC(=O)NCC1C(=O)NCC(C)(C)CC(C)C N1(C=O)CCCC(N(CC=C)CC=C)C1.C(=O)(C(CC)c1ccccc1)NC N1(C(c2c(C(C)=O)ccs2)=O)CCC(C2CC2)(NC(c2cc(C)ncn2)=O)C1 C(CC(C)(C)CNC(c1cc(C(N)=O)no1)=O)NC(C1(OCC)CCOC1)=O c1(NCCC(C)OC)[nH]c(=NCc2cc(C)nn2C)nc2c1ncn2C(C)C c1(C(=O)Nc2cn(C)nc2-c2ccccc2)ccc2ncccc2c1Cl Cc1cc([N+](=O)[O-])ccc1NCC1CCC(NC(C2CC(C)CO2)=O)C1 CCC(CCc1ccccc1)=CC(=O)N(c1cnn(CO)c1)C c1(C(=O)NC(C(C)N(C(C)=O)CC)C)ccc(NC(C2(CF)CC2(F)F)=O)s1 C1(NC(C(CCC)N(C)C)=O)CN(C(c2ccnc(Cl)c2OC)=O)CCC1O c1(C(N2C(C)(CC)CC(NC(C3CNC(=O)N3)=O)C2)=O)c[nH]c2c(C)cccc12 C=CC1(C(=O)NCCc2cnn(C)c2)CCN(C(=O)C(O)CC(C)C)C1 C12(C(N(CC(CC)NC(C34CCC(C3)C4)=O)CC)=O)CC3CC1C2C3 C1(S(C)(=O)=O)(C(=O)NC2CN(C(CC(C(C)C)C)=O)CC2F)CCCC1 C=C=CCCC(=O)NC(c1nocc1C(=O)NCC1CCCO1)C C12(C(N3CCC(C)(NC(c4c[nH]cc(F)c4=O)=O)CC3)=O)CCCCC1C2(F)F C#CC1(NC(=O)CC2(NC(C3CCCN(C)C3)=O)CCCCC2)CCCOC1 C1(CC)CC(O)C(O)CC1C(=O)NOCC(=O)NCc1c(C)cnn1C C1(C(N2CCCC(CCNC(C(CC)CC)=O)CC2)=O)CC2(CCC2)CCO1 c1(C(N2C(C(=O)NC(CC)CN3CCCCC3)CC2C)=O)cc(C)nc(C)n1 Cc1ccc(C=CC(N2CCCC(CCNC(c3cncc(N)n3)=O)C2)=O)cn1 c1(OC)ccc2c(n1)N(CC1(c3c(F)cccc3Cl)CC1)CC2 S(=O)(=O)(c1cccnc1NCC1CC(O)CN1C)NCc1n(CC)c(C)nc1 C=CCC(C(=O)NCC1(CNC(=O)C=Cc2cnn(C)c2)CC12CCC2)C(C)C C(=O)(C1CCCc2nncn21)NCC=CCNC(=O)C1=CC(O)CCC1 N1(C(C(C)NC(=O)OC)=O)CCC(OCCNC(=O)CC2CCC2)CC1 N1(C(C2(CC=C)CC2)=O)CC(CNC(c2cc(COC)cs2)=O)CC(C)(C)C1 CCCC(C#N)C(=O)N1CCCC(CCNC(c2cc(O)nc(N(C)C)n2)=O)C1 CCCCC(CC)C(=O)NCC1(F)CCC(NC(C2CCOCC23CCC3)=O)C1 N1(C(c2cn(C)nc2C(F)F)=O)CC(NC(c2ncn(C)n2)=O)CC2(CCC2)C1 c1(OC)ccc(Cl)c(Cl)c1C(N1CCCC(NC(=O)CC2CCCCO2)C1)=O CCCCCCCCC(=O)N1CC2CCN(C(=O)CC3C(C)C3(F)F)CC2C1 N1(C(C(COC)N(C)C)=O)CC(C)N(C(=O)C(n2cc(Cl)cn2)C)C(C)C1 n1(C(C)C)cc(C(=O)NC(C2CCCCC2)C(C)NC(c2nc(Cl)cs2)=O)cn1 C(=O)(C1=CCC2(COC2)OC1)N1CCC(=CCNC(c2cccc(O)n2)=O)CC1 N1(C(C2CCC(=O)OCC2)=O)CCC(CNC(C2CC3(CC3)CO2)=O)C(F)(F)C1 C1(C(N2C(CNC(C34CC(C)C3C4)=O)CC2)=O)CCCCN1Cc1cccc(F)c1 Cc1ccnc(C)c1C(=O)NC1CCOC1C(=O)NCc1ncsc1C c1(C(=O)NC)ccc(NC(=O)NC2CC3CC2(CO)C3)c(C#C)c1 C1(C(N(CCCNC(c2cnc(N(C)C)o2)=O)CC)=O)Cc2c[nH]cc2S1(=O)=O Cc1nc(NC(c2nc(C(=O)N(C(C)CO)C(C)C)cs2)=O)nc(Cl)c1Br Cc1cc(C(F)(F)F)nn1CC(=O)N(C)CC1(NC(=O)C=CC2CC2)CC1 c1(OC)ccc(CC(=O)NC(C2CCN2C(c2ccncc2Br)=O)=O)c(OC)c1 S(=O)(=O)(c1cccc(N2Cc3cnn(CCO)c3C2)n1)N1C(C)(C2CC2)CCC1 C(=O)(C1=CCC(C)(C)CC1)NC(CNC(C1CN(C(=O)OC)C1)=O)(C)C1CC1.C(CO)O C#CC1CCC(C(N2CCC(C(C)NC(=O)COc3ccccc3C)C2)=O)CC1 C1(CNC(Cn2ncc(C)c2)=O)CN(C(=O)C=CC(C)(C)C)CCCO1 C1(CC=C)(C(=O)NCC(F)C(C)(C)O)CCCN1C(=O)C(C)NC=O CC1(C)CC(=O)NCC1c1noc(C2CCN3CC23)n1.C1CC1.C1CC1 Cc1ccc(C(=O)C(=O)NCC2CCN2C(=O)Cc2nc[nH]n2)s1 CC(C)(C)CC(C)(C)C(=O)NCC1(C)CN(C(C2(F)CC=CCC2)=O)CCO1 c1(-c2c(F)ccc(OC)c2OC)ccc2c(C(=O)Nc3cnsc3)c[nH]c2c1 C(C(CC(C)C)C(=O)NC1(CNC(c2nn(C)c(N)c2C)=O)CCC1)OC C1(C(=O)NCCCC2OCCN(C(C3OCCN(C)C3)=O)C2)CC12CCOCC2 C(=O)(CCC1=CCCCC1)NCC1C(N(C)C)CN(C(C2CCS(=O)(=O)C2)=O)C1 Cc1nc(O)[nH]c1C(=O)NCC1CC(NC(C2(SC(F)F)CCCC2)=O)C1 C(CCCC(=O)N1CCC(C)(CCC)C1)N(C(C(C)=CCC)=O)C C#Cc1cccc(CC(=O)N(CCNC(c2ccc(COC)c(C)c2)=O)CC)c1 c1(C(N2C3CN(c4ncc(I)cn4)CC23)=O)ccc2cc(O)ccc2n1 N1(C(C2C(C)(C)NC(=O)C2)=O)CC2CC(NC(c3c(Cl)cccc3Cl)=O)CC2C1 N1(C(c2c(C)con2)=O)CCC(C(C)(C)C)(CNC(=O)CC2COCCO2)C1 C1(CNC(c2ccc(NC)cn2)=O)CCCCN(C(c2nccc(SC)n2)=O)C1 CC1=C(C(=O)NC2CN(C(c3snc(Cl)c3Cl)=O)CC2F)SCCO1 c1(NC(C(C)C)CCO)ncccc1S(=O)(=O)NC(CN(C)C)Cc1ccccc1 c1(NC(c2n(CC=C)nnn2)C2(SC)CC2)ccc(-n2ccnc2)cc1 C1(C(N(CC(CC)NC(=O)COCCOC)CC)=O)(COC)CCC12CCC2 C1(NC(=O)Cc2csnn2)CCC2CCN(C(c3cnns3)=O)C12 N1(C(COCC)=O)CC(NC(=O)C(C)C(F)F)CCC1C.c12cn(nn1)C2 CC(CN(C)C(=O)OC(C)(C)C)CC(=O)Nc1nc(-c2ccccn2)cs1 C1(NC(c2cc(C)nn2C(C)(C)C)=O)CN(C(=O)Cn2cncc2C)CC2CC12 C1(C(N2CC(C3(NC(CC(COC)(C)O)=O)CC3)C2)=O)CC2C=CCC(C1)C2 N1(C(CCC=CC(C)C)=O)CCCC2(C1)CN(C(=O)C1=NOC3COCC13)C2 Cc1cccc(C(CNC(c2cc(C#N)c[nH]2)=O)NC(c2nscc2C)=O)c1 C1(NC(C2(COC)CC2)=O)CC(CO)N(C(=O)CCCN(C)C)C1 CP(C)(=O)CC(=O)NCCOC1(C(N2CCC(OCCF)C2)=O)CC1 N1(C(CCn2ncc(C)c2)=O)CCC(CNC(c2nnc(O)cc2C)=O)C(C)C1 CN1C(=O)OCC1C(=O)NCC1CCN(C(c2c[nH]nc2C(F)F)=O)CC1 CCCCS(=O)(=O)NCC(=O)NC(C)CC(C)NC(=O)CNc1ccc(C)cc1 c1(C(N2CC(C)C(O)CC2)=O)c[nH]c2cc(-c3cccc4c3OCCO4)cnc12 N1(C(CCCOCCC)=O)CC(O)CCC1C(=O)Nc1cccc(OCF)c1 C(=O)(C#CC1CCCOC1)N1C(C)CCN(C(Cc2c(C)cc(F)cc2)=O)CC1 C(=O)(CC(O)Cc1ccccc1)N(CCCN(C(=O)C(O)C1(CO)CC1)C)C C(C(COC)CC(=O)NC1CC(O)CN(C(=O)CCOCCCOC)C1)OC N1(C(C2(C#C)CC2)=O)CC(OC)CC(NC(c2cccc(Cl)c2N)=O)C1 C#Cc1cc(NC(C2CCN(C(C3(COC)CCCO3)=O)C2)=O)ccc1C CC1CC(=O)NC1C(=O)NCc1cccc(NC(C2CC(O)CN2C)=O)c1 C(C(C)(C)CC(=O)N1CCCC(C(C)(C)C)C1)N(C)CC1(C(=O)OC)CCC1 C=Cc1cncc(C(N2CCC(C(=O)N(CCN=[N+]=[N-])C)C2CC)=O)c1 Cc1ccnc(C(=O)NC(C)CCN(C(=O)C(F)CC2CCOC2)C)n1 N1(C(C=C(CC)C)=O)CCC(N(C)C(c2cc(C3CC3)[nH]n2)=O)C1 C1(C(=O)NCC2CCCN(C(C(C(C)(C)C)=O)=O)C2)CCCC2(CCC2)O1 c1(C(=O)NC(C)C(CO)NC(C2CC(C)(F)C2)=O)cccc(N2CCCCC2)c1 C=C(C)CCCC(=O)NC1CC(O)(CNC(=O)C(c2cc(F)cc(Cl)c2)OC)C1 C1(CNC(Cn2cc(C)c3c2cccc3)=O)CC2CCC(C1)N2C(C1CCC1)=O Cc1cc(=NCc2nccs2)[nH]cc1S(=O)(=O)N1CCC1C1CCCC1 n1(CC(=O)NCC(CN(C)C(C2CC2(F)F)=O)O)nc2n(c1=O)CCCCC2 C(C(=O)N1CC(C(F)(F)F)C1)(C1CN(C(C2(OC)CCC2)=O)C1)OC CCCC(C(O)C(=O)N1CC2(CCN2C)C1)NC(=O)C(CN(C)C)CC Cc1nc2cc(C(=O)NCC3CNCCN3Cc3ncco3)ccc2o1 c1(CN(C(c2c(N(CCCOC)C)ccs2)=O)C)nc2c(C)cccc2o1 c1(OC)ccc(C(=O)NC2CC(NC(=O)C(c3cncnc3)C)C2)nn1 Cc1c(C(=O)NC(C(=O)NCC(C)(C)O)C2CCCO2)ccn1C c1(C(N2CC(C(C)NC(C(C)NC(=O)NC3CCCC3)=O)C2)=O)cnc(Cl)s1 c1(C(C)(C)C(=O)N2CC(CNC(=O)CC3COCC3O)C2)cc(Cl)ccc1F N1(C(C(C2CCCOC2)OC)=O)CCN(C(=O)Cn2cc(C#N)cn2)CC1C N12Cc3cccc(C)c3C1c1nc(-c3cccc(OC)n3)nn1CCC2.CCOC CCS(=O)CC(=O)N1CCC(NC(=O)C=Cc2ccc(-c3ccccc3)o2)C1 C#CCC(CC(=O)N(CCNC(c1ccnc(C)c1)=O)C(C)C)c1ccccc1 N1(C(Cn2c(C)c(Cl)cn2)=O)CC2CC(NC(=O)CC3CCCC3(F)F)C1C2 n1(CC=C)c(C(=O)NC2CC23CC(NC(=O)C(C)=CCC)C3)cc2ccccc12 C(=O)(C(C)P(C)(C)=O)N1CC(C)(NC(C(CCC)c2ccccc2)=O)C1 Cc1cc(C(=O)NCCC2CCN(C(=O)C(C)C3CCC3)C2)c(Br)c(C)c1 C(=O)(C(CNC(=O)CCCOC)C(C)(C)C)N1CC(C(=O)NCC)C1 c1(C(N(CC(CN(C(C(C2CC2)SC)=O)C)O)C)=O)ccc(CN=[N+]=[N-])cc1 N1(C(CCNC(C)=O)=O)CC(=O)NCC1C(=O)NOCC=CCl C(C)(CNC(c1ccc(C#N)s1)=O)(C(C)C)NC(c1cnc(C(C)=O)s1)=O c1(OCCN(C)NCC)cc(C(=O)C(F)(F)F)ccc1OC(C)C n1(CC(=O)N(CCCNC(C2CC23CC3(F)F)=O)C)cc(Br)ccc1=O C1(NC(C(C2CCCC2)NC(C)=O)=O)CCCCN(CC(c2nccs2)C)C1 N1(C(CC(CC)OC)=O)CCC2CN(C(=O)CCCc3c(C)noc3Cl)C2C1 Cc1cc(OCCC(=O)N(C)CC2CCN(C(=O)C(C)CC(C)C)C2)cc(C)c1 C=CC(C)CC(=O)N1CC(C)(OCCC(=O)NCCCc2cccs2)C1 c1(C(N2CC(C)C(CNC(C3SCCS3)=O)CC2)=O)ccc(F)c(S(N)(=O)=O)c1 C(=O)(C(C1=NOCC1)N(C)Cc1ccncc1)NCCCC Cc1cccc(CN(C)CC2(NC(=O)CC3CCCOC3)CC2)c1Cl c1(C(N2CCSCC2)C(=O)NCSc2cccc(Br)c2)cc(Br)ncc1[N+](=O)[O-] C(=O)(C(C)CCCC(C)C)N(CCN(C(c1ccnc2ccnn12)=O)CC)CC S(=O)(=O)(c1cccc(Cl)c1F)NCC(CC1Cc2c3c(ccc2)N(CC3)C1=O)O C1(COC(c2c(C(=O)OCC)csc2)=O)CC(C)CN1C(=O)CCC(=O)OC N1(C(c2cc(CC)ncc2)=O)CCCCC(N(C)C(c2cccc(OC)n2)=O)C1 C1(C)(C(=O)NC2(c3cc[nH]n3)CC2)CCN(CC(c2ccccc2)OC)C1 n12cc(nn1)C2.N1(C(c2cnc(Cl)s2)=O)CCCC1CC(F)(F)F.C(CO)N N1(C(c2c(OCC)n[nH]c2)=O)CCC(NC(=O)CSc2ccccc2O)C(O)C1 c1(SC)nc(NC2C3CC2CN(C(=O)CC2CCCCO2)C3)cc(Cl)n1 c1(OC)ccc(CC(N2CCC(NC(C3CC(CF)C3)=O)C2C)=O)c(OC)c1 c1(CC)cccc(C)c1C(N1CCC(SC)C1)=O.C1CCN(C)C(=O)N1C(C)C c1(CCC(=O)N(CC(C)NC(C2(C)ON=C(C)C2)=O)C)cccc([N+](=O)[O-])c1 N1(c2ccc(OC)cc2)CCC2(CC1)CNC(=O)C2.c12c(F)cc-1cc2F C1(O)(CN(C)C(C2CC(F)C2)=O)CCN(C(=O)CSc2cn[nH]c2)C1 n1(CC(=O)NCC(C)NC(C2C(F)(F)C23CC3)=O)nc(O)ccc1=O N1(C(CC2(N(C(=O)Cc3c[nH]nc3C)C)CC2)=O)CC(=O)N(C)C(C)C1 C1(F)(C(=O)NCCNC(CC)=O)CCCN(C(=O)C2=CC(C)(CC)C2)C1 C1(C(N2CC(NC(CCC(C)C)=O)C(F)C2)=O)CCOC2(CCCCC2)C1 C1(NC(c2nn(C)c(O)c2)=O)CC2CCC(C1)N2C(c1cncc(CO)c1)=O C1(CN(C)C(C2(F)CC(N(C)C)C2)=O)CCCCN1Cc1ccncn1 C(=O)(C(F)CC1CN(C(=O)C(O)CC2CCC2)C1)N(CC(=O)OC)CCO C(=O)(C1=COCCC1)NC(C1CC1C(=O)NCCC1CC1)C c1(OC)c[nH]nc1C(=O)NC(C1(O)CN(C(=O)CN(C(=O)C(C)C)C)C1)C C12(C(=O)NCc3nc(C)c(C)[nH]3)CCCC1N(C(c1nocc1Cl)=O)CC2 N1(C(c2cc(C)[nH]c2C)=O)CCC(CCNC(C2(C)CCN(C)C2)=O)CC1C N1(C(CCN(CC(C(C)C)C)C)=O)CC(NC(=O)CCC2CC2)C(N=[N+]=[N-])C1 C=CC(C)CC(=O)N(CCNC(=O)CCCOc1ccc(F)cc1)C(C)C C1(C(N2CC(CC)N(C(=O)CCc3nccn3C)CC2)=O)OCCOC12CCC2 n1(C2(C(=O)NCC3C(NC(CCCOC(C)C)=O)C3)CC2)cnc2ccccc12 C1(NC(C2(C)CC2)=O)CCN(CCNC(c2cc(CN(C)C)n[nH]2)=O)C1 C(CN=C(NCc1cnc(-c2ccccc2)o1)NC1(CF)CC1)N(CC=C)C c1(C(N2CC(C)(C)C(NC(=O)CSc3ccccn3)C2)=O)cccc2nonc12 N1(CC)CCC(N(CC=CCSC)C(C2CC(C)(F)C2)=O)CC1 Cc1nccnc1C(=O)N(C1CC(NC(c2ccnc(OC3CCOC3)c2)=O)C1)C CC(CC(=O)NCCC1CC(NC(=O)Cn2cnc([N+](=O)[O-])n2)C1)C(F)F N1(C(CC(C)N(C)C)=O)CCCC(CCNC(c2nc(C3CC3)cs2)=O)C1 c1(C(N2CCC3CC2CN3C(c2ccsc2)=O)=O)ccc2nonc2c1 c1(N2CCN(c3ccnc(NCP(C)(C)=O)n3)CC2)ccc2c(c1)CCCS2(=O)=O C1(C(=O)Nc2ccc(CN3CC(N4CCCC4)C3)cn2)CCCC(CO)CC1 N1(CC2(NC(C34CC(C(C)C)(C3)C4)=O)CC2)CCN(C(=O)CN2CCCC2)CC1 c1(CNC(=O)NCC(N2C(C)C(F)(F)CC2)=O)cnc2[nH]cnc2c1 N1(C(c2c(N)cncn2)=O)CCCC(CC(=O)NCc2ccc(Cl)cn2)CC1 CC(CCC(C)(C)C)C(=O)NC1(CN(C(=O)CCN2CCOCC2)C)CC1 C1(NC(C(CCCC)C)=O)(NC(=O)C(C)CCCC=O)CCC(F)(F)CC1.OC N1(C(c2c(OC)ccnc2)=O)CCOCC(NC(=O)C(C(C)C)C2CCC2)C1 C(CC(C(C)(C)C)NC(c1cccn(C)c1=O)=O)N(C)Cc1cccc(F)c1Cl N1(C(c2n(CC)ccn2)=O)CCCC2CN(C(=O)CSCc3cscn3)CCC12 N1(C(c2nccc(-n3cccn3)n2)=O)CCC(C(=O)NCC2CC2)CC1.C1CN1 CC1COCCN(C(C23CCCC2CCN3C(=O)CN2CC3CC3C2)=O)C1 Cc1ccc(C(F)C(=O)N(CCCN(C(=O)Cc2cnccn2)C)C(C)C)cc1 c1(CC(N2CC(C)N(C(=O)Cc3c[nH]ccc3=O)CC2)=O)cc(F)c(Cl)cc1F N1(C(CCc2cn(C)nc2)=O)CC2CN(Cc3cc(C#N)ccc3F)CC2C1 CC(C(=O)NCC(C)(O)CNC(C1CCC(O)CC1)=O)C(C)(C)C C1(C(=O)NCCCC(=O)NC2CCC(=O)N2)CCN(C(=O)NC2CC2)CC1O c1(CC(=O)NC(CN(C(c2cc(CC)n(C)n2)=O)C)C)cccc(CC)c1OC Cc1cnc(C(N2CCC(CCNC(=O)CCCC(N)=O)C2)=O)c(F)c1 CCCCC(C)(F)C(=O)NCc1ccc(C(=O)NCC2CC23CC3(F)F)nc1 Cc1cc(Cl)cnc1CN(C(c1cn(CC(C)(C)C(=O)O)nn1)=O)C1CC1 CCC(CO)(C(=O)NC1(CCCC(=O)NC2CC2CN(C)C)CCC1)OC C1(C(N2CCCN(C(C(C)C3CCOC3)=O)CC2)=O)CC(=O)C12CCCC2 c1(C(N(CCN(C(=O)CC=Cc2ccccc2)C(C)C)C)=O)cc2cscc2s1 CC1CN(C(c2cnc3cccnn23)=O)CC(C)N(C(C2COCCN2C)=O)C1 N1(C(C2C(C)C2C)=O)CC2CCC1CN2C(c1ccc2scnc2c1)=O C12(NC(c3ccc(CC)cn3)=O)CCCC1CN(C(C1(CCF)CCC1)=O)C2 CCC(C)CC(=O)N1CC(NC(c2ccc(C3CC3)s2)=O)C(CC2CC2)C1 Cc1cc(C(=O)NCC2CCCN2C(=O)COc2ccc(C)c(C)c2)c(C)cn1 N1(C(C(C)SCC)=O)CC(NC(c2nc3cccnc3s2)=O)C2(CCC2)C1 C1(C(N2CCCC(NC(c3cc(C(F)F)no3)=O)C2)=O)CCCC2(CCC2)C1 C1(NC(=O)CC2CC2)CN(Cc2cn(-c3cccc(F)c3)nn2)C2CCCC12 N1(C(C2(C)N(C(c3cccc(CC)n3)=O)CCC2)=O)CCC(C)(CC2CC2)CC1 N1(C(c2cc[nH]c2)=O)CCN(C(=O)C(O)Cc2cccc(Cl)c2)C2CCC12 c1(CCC)ccc(C(N2CC3CC2C3NC(C2(C3CC3)CC2)=O)=O)cc1N C1(C(N2CC(CNCC)C2)=O)Cc2ccncc2C1.C12CCCN(C1)CC(=O)N2 C1(CNC(c2c(C)ncnc2O)=O)C2CCCC1N(C(C1CC(C)OC1C)=O)C2 C(=O)(CC(C)C(C)C(C)C)N(CCCNC(=O)C(c1cnn(C)c1)O)CC C1(n2c(-c3cnn(CCO)c3)nc(C(C)C)n2)CCC(F)(F)CC1 C1(C)(N(C)C(C2CCCC2)=O)CCCN(N2CCC(C=O)C2)C1.N1CCOCC1 C1(F)(CNC(C(CC#C)C)=O)COCCN(C(c2cc3sccc3n2C)=O)C1 c1(C(=O)OC)cc(O)cc(S(=O)(=O)N2CCC(C)C(c3ccccc3)C2)c1 c1(CC(=O)C2CC2)ccccc1.C1(C2CC2CCCO)CCCO1 c12ccc(cc1)CN(C)C2=O.c1(C(=O)NCC2C(C)C2)cccc(C2CC2)c1 C1(C2CC2)(CN=c2[nH]nc(COCC)s2)CCN(C(c2cc3occc3[nH]2)=O)C1 c1(C(=O)NC(C)CNC(=O)C(c2cccn2C)=O)cc(C(N)=O)cc(F)c1 Cc1cc(Cl)cc(Cl)c1OCC(N1CCN2CCCC2C1)=O C1(CC#C)(C(=O)O)CCN(C(=O)NC2C3CC2(C(C)(C)C)CO3)C1 CC1(C)CCCC(O)(C(=O)NC2CCC2NC(c2cccc3nccn23)=O)CC1 c1(NCc2cc(OC)ns2)ccnc(CNC(=O)CN(S(C)(=O)=O)C)c1 c1(C(=O)NC2CN(C(c3ncc(OC)cn3)=O)C3C2C3)cc2occc2s1 c1(C(=O)NC2CC(CCNC(C(C)(C)SC)=O)C2)n[nH]c(C)c1Br C1(NC(c2c(C)csc2)=O)CCN(C(c2cc(Cl)ns2)=O)CCC1CO C(C(=O)NCC1C=CCN1C(c1cnn(CC(C)C)c1)=O)(C(C)(C)C)SC c1(OC)ccc2c(c1)CC(C(=O)NCCCCCN(C)C(C1(C(N)=O)CC1)=O)O2 c1(C(=O)NCCC(=C)CNC(=O)CCOC)coc2ccc(C(C)(C)C)cc12 c1(CCCC(=O)NCC2CCN(C(c3c(N)non3)=O)C2)ccc(F)cc1 Cc1noc(C)c1CC(=O)NC1CN(CCCNC(=O)CCSCC(C)C)C1 N1(C(C(C)CCN(C)C)=O)CC2C3CCC(C2C1)N(C(C1CCC2(CCC2)C1)=O)C3 Cc1ccc(C(C(=O)NCC2CCCO2)N(CC(C)CO)C)c2cccnc12 c1(C(N2CC(CNC(C3(OC)CCC3)=O)(OC)C2)=O)cn(C(C)C(F)F)nc1C Nc1ccc(C(N2CC3CC2C3NC(c2cnn(CC3CCCO3)c2)=O)=O)c(Cl)c1 N1(c2nc(=N)nc(N(C)Cc3cccnc3)[nH]2)CCC(C2CCCN(C)C2)CC1 C12CCN(CC1)C2=O.C(=O)(CC(F)(F)F)N(CC)CC1CC1(c1ccccc1)F C12(C(N3CCC(N(C(=O)Cc4cscc4C#N)C)C3)=O)CCC(CO)(CC1)CC2 Cc1cc(=O)ccn1CC(=O)NCC1(O)CCN(C(=O)CCc2cn(C)cn2)C1 c1(N2CCC(CNC(C(C)CCN(C)C)=O)C23CC3)ncnc2c1nnn2C C1(C#N)(C(=O)NCC(CCOC)NC(C2CC(C)=NO2)=O)CCCCC1 N1(C(c2cc(CCNC(=O)CCc3cccs3)on2)=O)CCN2C(=O)OCC2C1 C(C(C)(C)CC(=O)NCc1cc(CO)n[nH]1)NC(CC1C(C)OCC1)=O C1(NC(c2ccc(C)nc2O)=O)CN(C(=O)C(C)(C)CF)Cc2nccn2C1 NC(=O)C(F)CC(N)C(=O)NC(c1ccc(Br)cc1)c1ccc(F)cc1 N1(C(c2cc(C)oc2CO)=O)CC(C)(C)CC1Cc1cn(CCCF)nn1 c1(CN(C)C(C2CCCC2)=O)ccc(CNC(C2CCCN2C2CC2)=O)nc1 N1(C(c2c(CC)nn[nH]2)=O)CC(NC(=O)C(c2ccccc2)C)C(SC)C1 c1(CNC23CC(C(=O)NC(C)C(C)(C)O)(C2)C3)c[nH]c2ccc(Br)cc12 N1(C(C(=O)NC)C2CC(CC3CCC3)C2)CCN(CC(C)F)CC1 Cc1ccnc(Oc2ccc(NC(c3cnc(C)[nH]3)=O)cn2)c1 c1(CNC(=O)C(C2(O)CN(C(C3(O)CCC3)=O)C2)F)ccc(CCCCO)o1 c1(CC(C(=O)N(C(c2cn(C3(CN)CC3)nn2)C)C)=O)cccc(Cl)c1 C[Si](C)(C)c1ccc(CNC(CCCc2nnc3n2CCCC3)=O)cc1 C1(C(N2CC(C)(NC(c3c(C(=O)OC)cccn3)=O)C2)=O)CCC2C1C2(F)F n1(CC(=O)N(CC(C)NC(c2cn(C(C)C)nn2)=O)CC)cc(C2CCC2)cn1 C=CC1OCCC1C(=O)OC(c1nc(C)cs1)C CC(C)CC(O)C(=O)NCCCCC1CN(C(=O)C(C(C)C)c2cccnc2)C1 C(C)(C)(CC(F)C(=O)N1CCCC1CCO)NC(C(CC)CN(C)C)=O CCCC(C#N)C(=O)N1CC(CNC(c2cnc(C3CC3)nc2)=O)C(O)C1 CCC(CC)C(C)C(=O)N(C(C)C(=O)NCCC1CCCCC1O)C1CC1 CC1(C)CCCOC1CNC(=O)N(Cc1ccsc1)CC12CCC(CC1)C2 CC1(C#N)CCCN(C(=O)C(C)(C2CCC2)NC(c2nsnc2O)=O)C1 c1(C(=O)NCC(C(=O)OCC)CC)cc2cc(C)cc(C)c2[nH]1 CC1CC=C(C(=O)NCC(O)CCNC(=O)C=CC(F)(F)F)CC1 C1(C2CCC2)(CNC(c2cccc(=O)o2)=O)CCN(C(=O)CC2CCOC2)CC1 N1(C(CCC)=O)CCCC(C(N2CCC(N(C)C(c3cc(Cl)n(C)n3)=O)C2)=O)C1 CC(C)C(CNC(c1csc(O)n1)=O)NC(=O)CC1(n2cncn2)CC1 N1(C(c2ccc(C(F)(F)C(F)F)cn2)=O)CC2CC1CN2Cc1ccccc1 c1(C(=O)OCC2C(C(=O)OCC)C2)cc2ccccc2nc1O N1(C(C(C(C)OC)NC(c2ccncc2N)=O)=O)CC(C)C(C)C1C Cc1cnn(C)c1C(=O)NCC1CCN1C(C1C2CCC1(c1ccccn1)C2)=O c1(C(=O)NCCC(C)NC(=O)C(C)Cc2ccco2)ccc(F)c2cnccc12 CC1(C)CCN(C(=O)CC2CC3C=CC2CC3)CC1CNC(=O)CNC=O c12cccnc1CNC2=O.Cc1oncc1C(N1CC(C2CCCO2)C1)=O c1(OCC(N2C(C(C)NC(=O)C3=NNC(=O)C3)CCC2)=O)cccc([N+](=O)[O-])c1 C1(F)(C(=O)NC(C2CCOC2)C#C)CCCN(C(c2cccc(F)c2F)=O)C1 C(=O)(CCCCC(C)(C)C)N(CC(=O)NCC(=O)NC(CC#CC)CO)C1CC1 C12(NC(Cc3nc(C(C)(C)C)sc3)=O)CCC(C1)N(C(c1ccc(O)nn1)=O)C2 c1(C(=O)NC(CN(C(=O)CC2=CCOCC2)C)(C)C)cnn2c(Cl)cccc12 C1(NC(CC2CC(CC)C2)=O)CCC(NC(C2CCC(C(N)=O)C2)=O)CC1 c1(C(=O)NC2CCC(CNC(=O)CC3CCCOC3)C2)cn2cccc(Cl)c2n1 C1(NC(C2CCSC2)=O)CN(C(C2CS(=O)(=O)C2)=O)CC2(CC2)C1 C1(C)(C(=O)NC(CCC)CCCNC(c2ccc(C)o2)=O)CCS(=O)(=O)CC1 C1(NC(C2(C(C)C)CC2)=O)CC2(C1)CN(C(=O)CSc1ccccc1F)C2 c1(C(=O)NC2C3CCC(C3)C2CO)ccc2c(c1)OC(F)(F)O2 CCC1CCOC(=O)C1.C(=O)(CCCNC(N)=O)OCc1ccccc1 C1(C(=O)NC2CN(C(Cn3nc(C)c(Cl)c3C)=O)C2)CCc2ccccc2O1 N1(C(C(CC)N(C)Cc2ncnn2C)=O)CC(NC(=O)C2CC2)CC(C)C1 c1(C(=O)NC2(C)CCN(C(C=CS(C)=O)=O)C2)cc(F)c(Br)cc1F c1(C(=O)NC2CCC(N(C(CCC=C)=O)C)C2)c(C)ccnc1C C(=O)(C1CCCc2n[nH]cc21)NCC1C(C)CCN1C(=O)CCc1cnoc1 c1(C(=O)NC2(CNC(=O)C=CC3CCCCCC3)CC2)cc2cc(O)ccc2[nH]1 c1(C(=O)NC(CNC(C2CCC(=O)N2C2CC2)=O)C2CC2)cc2cnccc2o1 CC1(C#CC(=O)N2CCOC3(C2)CN(C(=O)C#CC2(C)CC2)C3)CCCO1 CC1CC2CCC(C(=O)NC(C)CCCCNC(C3CC3(Cl)Cl)=O)CN2C1 c1(C(N2C(CCC(=O)NCC(C)O)CCC2)=O)ccc(O)nc1 c1(C(N2C(C(=O)NCCc3ccc(Br)cc3)CC(F)C2)=O)c(Br)ccc(F)c1F c1(CNC(=NCCCc2ccc(CO)cc2)NCC2CC2)ncnc2[nH]cnc12 N1(C(c2c(C)onc2)=O)C2CCC1C(CNC(=O)Cc1csc(Cl)c1)C2 Nc1cc(C(=O)NCC(CNC(=O)C(O)C2CCCC2)S(C)(=O)=O)cnc1Cl CCCCCCC(C)C(=O)NC1(C)CCCN(C(=O)CC2C(=O)ON=C2C)C1 c1(C(=O)NCC(C)(CO)NC(CC2(C=C)CC2)=O)cn2cccc(C)c2n1 c1(-c2n(-c3c(CC=C)cccc3)nc(-c3ccc(N)cc3)n2)ncc(F)cc1N c1(SC(CC)C(=O)NC(c2ccc(CO)o2)=O)ccccc1SC(F)F CC1CCC(CNC(=O)Cc2cccc(F)c2F)N(C(=O)CSCCC#N)C1 C1(CCCC)CN(C(C2NC(=O)C3CC23)=O)CCN1C(=O)C1=CCCC1 CCCC(C(=O)NC1CCCN(C(=O)CC(C)C2CC2)CC1)S(N)(=O)=O c1(SC)ccccc1C(=O)NC1(C)CCN(C(=O)CC2CCOC(C(C)C)C2)C1 c1(CNC(CN(CC)CC)=O)cc(C(N2CC(F)(C(=O)OC)C2)=O)no1 c1(C(=O)OCc2c(C)ccc(C(=O)OC)c2)ncc(F)c2ccccc12 C1(NC(CSCCNC(Cc2cc(C)[nH]n2)=O)=O)CC(O)CC1O Cc1cnccc1C(C)C(=O)NC1CCCCC1N(C)C(c1cccs1)=O C1(C(N2CCN(c3ncc(C)c(C)n3)C(C(C)C)C2)=O)CCOC2(CCCC2)C1 c1(C(=O)OC)cc(Oc2ccc(C)nn2)cnc1C.c12ccc(cc1)n2C n1(CCC(N2C(CNC(C(C)OCC)=O)CC(O)C2)=O)cnc(C)cc1=O C(=O)(CCCC(C)(C)C#N)NC1CCCC(CNC(C2=NOC(C)C2)=O)C1 C12(NC(C3C(C)CCC3)=O)CC(CNC(c3cc(Br)c[nH]3)=O)(C1)OC2(C)C C12(C(=O)OC(C(=O)OCC)CCc3ccccc3)CCC(CO)(C1)OC2 Cc1cc(C#N)nc(NC23CCCC2CN(C(c2cn(C4CCC4)nn2)=O)C3)n1 c1(NCC2CN(CC)C2)ccc(S(=O)(=O)NCC2CCOC(C)(C)C2)c(Br)c1 c1(C(C)(C)OCC)cn(CCOCCNC(=O)CCn2ccnn2)nn1 c1(C(C(=O)NC)N(C)NC(=O)C2CC2)ccc(N2CCOCC2)nc1 c1(OC)ccc2c(c1)C(CCN(C(CO)C(C)C)C)=CC2=O N1(C(CN(c2ccccn2)C)=O)CCC(O)(CCNC(=O)C(C)(C)N(C)C)C1 CCCN=C(NCCN(C1CC1)C(C)C)N1CCC(F)(c2cc[nH]n2)CC1 c1(N2CC(C)C(NC(C34CCCCC3C4(F)F)=O)CC2)ccc2nnnn2n1 C#CCC(O)C(=O)NC1CC(NC(=O)C(F)(F)c2ccsc2Cl)C1 N1(C(C(=O)NCc2ccnn2CC(F)F)=O)CCOCCC1C1CC1 C(=O)(C#CC1CCC1)NC1C(CNC(c2c(COC)cccc2)=O)CCCC1 C1(C(=O)NCC(C(C)(C)C)NC(C(CC)CN(C)C)=O)CC2(CCCCC2)C1 N1(C(c2cn(CCOC)nc2)=O)CC2(CCCC2NC(=O)C(CC2CC2)OC)C1 O=C(C(C1=CCCCC1)N1CCSCC1)NC(c1cccs1)C1CC1 N1(CC(=O)NC(CN(C(=O)CNC=O)C(C)C)C)C(=O)c2ccccc2S1(=O)=O c1(OC)c(C(N2CC=CC(NC(=O)CC(C)N(C)C)C2)=O)[nH]c2ccccc12 [N-]=[N+]=NC1CN(C(C23CC(CO2)C3)=O)CC1NC(C1CCCCN1N=O)=O c1(C(=O)NCC2(F)CC(NC(c3ccc(NC)cn3)=O)C2)cc2ccsc2n1C c1(C(=O)NC2CC3CN(C(C(C)O)=O)CC32)cc(Br)c2c(c1)[nH]c(=N)n2C c1(OC)ccc(CN2CCNCC2C(=O)NCc2ccc(Br)nc2)c(Br)n1 N1(C(CC=CCC)=O)CC2CCC(C1)N2C(=O)Cc1nnc(S)n1C c1(CC)c(C(N2CC(CCCCNC(=O)CCSC)C2)=O)oc2ccccc12 N1(C(C2CC3(CC(OC)C3)C2)=O)CCCN(C(C23CC(C)(CO2)C3)=O)CCC1 N(C(=NCCCF)NCc1nc(C2CCCO2)n[nH]1)Cc1ccc(CO)c(F)c1 C12(CCNC(C3(C)CC(=C)C3)=O)CCC(C1)N(C(c1cnn(C(C)(C)C)c1)=O)C2 C1(C(=O)NC2CCN(CC)CC2)C2CC(O)C(C2)N1C(C1CC2C=CC1O2)=O c1(OCCCC(=O)N(CCCNC(C2C(COC)C2)=O)CC)cccc(C)c1C c1(NC(c2ccnc(C)n2)=O)ccc(NCc2scnc2Cl)c(F)c1 c1(CC)cc(NC(c2cc(-c3ccn(C(C)C)n3)[nH]n2)=O)ccn1 C(CC(C(C)(C)C)NC(=O)C1=C(Cl)CC1)N(C(CCCN(C(C)C)C)=O)C C1(NC(CSC(C)(C)C)=O)CN(C(=O)C(O)Cc2ccccc2)CCC1CO C1(CC(F)F)(C(=O)NCCCC(C)NC(C2CCC(C)(C)O2)=O)CCOCC1 C1(C)(CNC(C2(C=C)CCC2)=O)CCN(C(=O)CN(CC)CC)C1 N1(C(C=CC=CC)=O)CCCCC1C1CCN(C(=O)C(C)n2cnnn2)CC1 N1(C(C(C)OC)=O)CCN(C(=O)C=CSc2nc[nH]n2)CC(C)(F)C1 C#CC1(C(=O)N(CCCCCNC(C2(N(C)C)CCC2)=O)C)CCOCC1 c1(NC(C2(C(=O)NOC3CCC3)C(C)(C)C2)=O)cc2occc2[nH]1 C1(C(NC(CC2CC(CC)C2)=O)C2CC2)CN(C(=O)C(C)(C)CC2CC2)CCO1 C1(CC)CCCCC1C(=O)NCC(C1CCC1)NC(=O)COC(F)(F)C(F)(F)F Cc1cc(C(N2CC3(NC(c4sccc4Cl)=O)CCC2CC3)=O)cc(C)c1N C1(CNC(c2c(CCC)n[nH]c2)=O)CCC2(CN(C(c3[nH]ncc3C#N)=O)C2)O1 C1(NC(C=CC(=O)N(C)C)=O)(CO)CCN(C(C2COC(=O)O2)=O)C1 CN1CC(O)CCC1C(=O)N(CC(N1CC2CC2C1)=O)C1CC1.n12cc(nn1)C2 N1(C(c2c(C)nn[nH]2)=O)CCCCC1CNC(c1ccc(Br)nc1)=O N1(C(Cn2ncc(C)c2)=O)CCC(F)C(NC(c2nc(C)oc2C)=O)C1 c1(C(C(=O)NCC(C2CCC2)NC(C2(C)CC2(F)F)=O)O)ccccc1F c1(C(N(CCC(=O)NCC(=O)OCC)C2CC2)=O)nnn(C)c1N Cc1ccc(C(=O)NCCCC2CCCN2C(C23COCC2C3(F)F)=O)nc1C C(=O)(CCCNC(=O)CC1(N(C)C)CC1)N(C)Cc1cscn1 C(=O)(CCCC(C)SC)N1CC(N(C(CSc2cnc(OC)nc2)=O)C)C1 C=CCCC(C(=O)NC)N1CCC(O)(C(F)(F)CO)CC1 CCC(S(=O)(=O)NC(C1CCC(F)(F)C1)=O)c1ccccc1 CCN=C(NCC(C)(C)CC(=O)ONC)N(C)CC(=O)OC(C)C C(=O)(C1=C(C)CCCC1)N(C1CCN(C(c2cc(C(C)=O)[nH]n2)=O)C1)CC C1(NC(C)=O)C(NC(C2CC(C)=NO2)=O)CC1O N1(C(c2n(CC=C)ccn2)=O)C2CCCC1CC(N=c1[nH]c(Cl)ncc1CC)C2 N1(C(c2c(N)cn(C)n2)=O)CC2CCCN(C(C34COC(CCO3)C4)=O)C2C1 N1(C(c2nc(C(C)OC)oc2)=O)CCOC2(CCCNC2)C1 c1(OC)ccc(O)c(C(N2CCOC(C)C2)C(=O)O)c1 c1(CC(=O)NCc2cn(CCCC)nn2)cc(C)cc(F)c1.C(COCC)S c1(C(N2CCC(CN(C(=O)C(C)(C)C)C)C2)=O)cccc2c(O)nncc12 c1(C(N(CCNC(c2c(CC)n[nH]c2)=O)CC2CC2)=O)cccc(OC)c1OC N1(C(C(=O)NCSc2cccc(Cl)c2)CC2CCC2)CC2CC(N)C2C1 CC(CCNC(=O)Cc1ccccc1)CCNC(=O)CCn1cccn1 C1(CN(C)C(=O)C2CC2)CCN(C(C2CC(N)C2)=O)CC1 C(C)(CC(C)NC(C(C)=CCNC(c1csc(C(c2ccccc2)=O)n1)=O)=O)OC N1(c2nc(COC)nc(C)c2)CC2CCC1C1CN(C(C3CC3(C)Br)=O)CC21 C1(C)(CNC(C2CCN(C)C2)=O)CCCN(C(=O)CCCNC(=O)C(C)(C)C)C1 N1(C(c2c(C)oc(Cl)n2)=O)CCC(C)(C)C(CNC(=O)CSc2ccccn2)C1 C1(NC(C=CC=CC)=O)CCN(C(C2(C(F)(F)F)CCCC2)=O)CC1O CC(C)(CCNC(=O)CSc1nc[nH]n1)C(=O)NCC1CCC(CO)O1 C12(NC(C(CCN(C)C)O)=O)CCCC(NC(=O)CCc3ccc(N)cn3)(C1)C2 c1(C(N2C(C)CC(CNC(CN(C)CC)=O)C2)=O)cc(Br)cc2c1OCO2 C(=O)(C1=CCCCC1C)N(CCOC)CCNC(=O)Cc1ccc(OC)cc1 C(CO)(C(F)(F)F)c1nc(-c2cnccc2C(=O)O)no1.CC(F)F N1(C(COCC=C)=O)CCC(C)C(CNC(=O)Cn2cccn2)C1 CC(=Cn1ccnn1)C(=O)NCC1CN(C(=O)CNS(=O)(=O)N(C)C)CCO1 C(=O)(C(CC1CCC1)NC(C1CCCCC1)=O)NCC1CC(=C)C1 CC1(C)C(=O)CC1C(=O)NOCC(=O)NCCC1(COC)CCCC1 C(=O)(C#CC1CCOC1)N(CC)CC1CCCCN1C(c1ccsc1)=O c1(OCCO)ccc(=NCc2cc(Cl)cnc2Br)[nH]n1 N1(c2nc(=N)nc(N3CCCCC(C(C)C)C3)[nH]2)CCOC2COCC2C1 c1(C(=O)NCC2(OC)CN(C(C3N(CC)C(=O)CC3)=O)C2)cnc2[nH]ccc2n1 C=C(C)CC(C)C(=O)NCC1CCN(C(c2ccc(N3CCCC3)cc2)=O)CC1 CCS(=O)(=O)CC(=O)NNC(=O)C(C)(C)CCCCNC(C1CCCCO1)=O N1(C(Cc2nc(NC=O)sc2)=O)CCN(C(=O)Cn2nnc(=O)[nH]2)C2CC12 c1(C(=O)NCCC2CCCCN2C(=O)CN2CC=CC2)csc2ccncc12 c1(C(=O)NC2CCCC(CNC(=O)C(F)=CCCF)C2)ccc2ncccc2n1 Cc1cc(C#N)cc(C)c1C(N1CCC(O)(C2(NC(=O)C=C3CCC3)CC2)C1)=O C(C(C)CC(=O)N1CCCCC1C(=O)NCCS(C)(=O)=O)OC N1(C(CC(CC)CN(C)C)=O)CCC(NC(c2cc(C(N)=O)[nH]n2)=O)CC(C)(C)C1 S(=O)(=O)(c1ccc(NCCS(N)(=O)=O)cc1Br)NCc1nnc(COC)s1 C1(C(C)NC(C2CC2(C)C(F)F)=O)CCCN(C(=O)Cc2cc[nH]c(=N)c2)CC1 CC(C)(CCN=c1nc(C(C)(C)C)nc[nH]1)NC1CC1.C12(CC1)C(=O)NC2=O CCC1=C(C(=O)N(C)CCOCCNC(c2c(C)[nH][nH]c2=N)=O)CCCO1 N1(C(CCCC(=O)OC)=O)C2CCC1CN(C(=O)C(C)C(O)CC)C2 C1(C(=O)NCc2cn(CC)nn2)C(C)OCCN1C(=O)C#CC(C)(C)C N1(CC)OCC(NC(=O)CNC(C2(C)CCCCO2)=O)C1=O CC1COCC(C(=O)NC(CC2CCCC2)C(=O)NC(CC2CC2)CO)O1 N1(C(C(C(=O)OCC)OC)=O)CCC(C)C(NC(=O)C(C)(C)N(C)C)C1 c1(C(=O)NCC(=O)N(CCCNC(C2CSCCS2)=O)C2CC2)cccc(O)c1 c1(C(N(C2CN(C(C(C)OCC=C)=O)CC2(C)C)C)=O)cccc2nn(C)nc12 CC(C)(CCCNc1cc(C(N)=O)ncn1)NC(=O)CCc1ccco1 c1(C(=O)NC(c2cncc(C)c2)CO)ccc2cnc(C)n2c1 c1(CC)onc(C(N2CCCC2C=CC(N2CCCCC2C2CCC2)=O)=O)c1C C1(NC(CCCCCC)=O)CN(C(C2CSCCS2)=O)Cc2ccnn2C1 C(=O)(C(C)(C)CC(=O)NC(C)(C)CNC(=O)CCN1CCC(F)C1)OC N1(C(C23CC(OC)C2C3)=O)CCC(NC(=O)CS(N)(=O)=O)C12CCC2 C=CC(C)CC(=O)N(C)CC1CN(C(c2coc(C(C)(C)C)n2)=O)CCO1 S(=O)(=O)(c1cnc(Cl)c(Cl)c1)NCCCc1ccn(C)n1 C1(CCNC(=O)CN2CCSCC2)CCCN(C(c2ccc(F)cn2)=O)CC1 c1(C(CC(F)F)NC(C(C2CN(C(=O)OC(C)(C)C)C2)OC)=O)cncc2c1CCC2 c1(C(N(CCNC(=O)C(C)(C)CCSC)CC)=O)cccc2occc12 C1(O)(CNC(C=Cc2ccc(C)o2)=O)CCCN(C(c2c[nH]nc2Br)=O)C1 c1(CNC(c2c(C)cnnc2)=O)ccc2cc(F)ccc2n1.C12(COC1)NC2 C1(C(=O)ON2CCOCC2)CCCCC1C1CCN(CC(F)F)CC1 Cc1ccc2c(c1)CCC(C(=O)OCc1cn(C(c3ccccc3)(C)C)nn1)O2 N1(C(CC2C=NN(C)C2=O)=O)CCOC2(C1)CN(C(=O)C=CC1CCCCC1)C2 N1(CC(CC)OC)CCC(C(C)NC(=O)CC2OCCC2C)CC1 CCC(C)CC(=O)NCC1(c2ccccc2)CC(NC(=O)CCN2CCC2)C1 C(=O)(C1=CC2C=CC1C2)N1CC2C(CC(=O)NC3CC3)C2C1.CC1C(=O)N1 c1(C(=O)NCCCC(C)NC(=O)CCC2CC2)cccc(C2(F)CC2(F)F)c1 c1(OC)cc(CC(N2CCC(O)C(NC(c3cocc3C)=O)C2)=O)ccc1C Nc1cc(F)ccc1C(N1CCCC1CCCNC(=O)C(O)C(F)F)=O C1(CC)CN(C(=O)C(C)C)CCN1C(=O)CNS(=O)(=O)NC N1(C(CC(=C)Br)=O)CC(CCNC(c2ccc(OC)nn2)=O)OC(C)C1 C(CN=c1nc(N2CCC(CN(C)C)C2)c2ncccc2[nH]1)c1cc(C)[nH]n1 C1(CC(C)NC(C2CC2(F)F)=O)CCN(c2nc(C3CC3)ns2)CC1 C1(C2C(NC(C3CC34CC4)=O)CCO2)CCN(C(c2cc(C3CC3)on2)=O)CC1 C(=O)(C1=C(Cl)CCOC1)N1CC(CC(CNC(C2OCCN(C)C2)=O)(C)C)C1 c1(OC)cc(C(=O)NC(C(C)NC(C23CCC2CC3)=O)C(C)C)ccc1Cl N1(CCC)CCCCC1C(N1CCC(F)(CNC(c2coc(C)n2)=O)C1)=O C(=O)(CCC(=O)NCC1CC(NC(C2CCCNC2=O)=O)C1)NC c1(C(C(=O)NC2(OC)CC2)NC(CS(CC)=O)=O)c(C)cccc1Br C12(C(N3CC(CC)(CO)C3)=O)COCC1CN(CCCCCc1ccccc1)C2 C(=O)(C(C(C)CC)N(C)C)N(C12CC(C1)C2)CC N1(C(C2C(OCC)C2)=O)CCN(C(CNC(C2(C#N)CC2(C)C)=O)C(F)F)CC1 C1(N(C(CC2CC(NCC)C2)=O)C)CCN(C(=O)C(C)(C)COCC(F)F)CC1 Cc1cc(Cl)ccc1CNc1cc(-c2ccccc2C(=O)N(C)C)ccn1 c1(C(=O)NCC(C)(C2CC2)NC(=O)Cn2nccn2)cc(F)ccc1Cl C(=O)(C(F)C(C)(C)O)N(CCC(=O)NC(C)CN1CCOCC1)CC=C C1(CNC(Cn2ncc(C)c2)=O)(CO)CCN(C(=O)COc2ccc(F)cc2)C1 c1(NC(C2CCC(CC)N2C(=O)C=CC(C)C)=O)cc(F)c(O)cc1C n1(CC(=O)NC2C(C)CCN(C(c3c(C)nc[nH]3)=O)C2)ccc(=O)n(C)c1=O Fc1ccc2c(c1)C(NCC(=C1CCOCC1)Br)CO2.C1CO1 n1(C)cc(Br)ccc1=O.C=C1CCC1(C(=O)OCC=CCOC(C)=O)C(=O)O c1(CC)nccc(-c2nc(CN3CCCCC3)nn2C(c2cccc(Cl)c2)C)n1 C(=O)(C(C(C)(C)C)NC(N)=O)NCC(C)N.CC(CC1CCCC1)C=O C(=O)(C1CCCc2cncn21)N1CCC2(CN(C(C3C(=C)C3)=O)C2)C1 N1(C(CC2(C=C)CCOCC2)=O)CC(NC(=O)Cc2ccc(C)o2)C(C2CC2)C1 c1(C(N2CC(C(C(=O)NC3(CC)CCC(C)C3)O)C2)=O)ncc(F)cc1F O=C(C1=CCOC1)NC(c1ccccc1)CNC(c1cncnc1C1CC1)=O c1(OC)ccc(NC(=O)C(C2CCN(CC3CN(CC(C)C)C3)CC2)C)c(C)c1 c1(C(=O)NC2C(NC(c3cc(C)c(O)cc3)=O)CC2)cc(P(C)(C)=O)cs1 C1(C(C(=O)NC2(CC(N)=O)CCC2)NC(c2cn[nH]c2)=O)CCCCC1 c12ccccc1NC2=O.n1(CCOC)cnnc1C(=O)NOC(CC)CC c1(OC)ccc(F)c(C(=O)NCC2CC3CCC2N3C(=O)CN2CC(C)C2)c1F O=C(CCCCCF)NCC1C2CCC(C2)N1C(C1CCCOCC1)=O N1(C(C2CSCN2C(C2CC2C(F)F)=O)=O)CCCC2(CC(O)C2)C1 c1(C(N2CCCC2C2CC2(F)F)C(=O)NC2CCOCC2)nc(F)ccc1Br Cc1cccc2c(C(=O)NC3CCN(CC(N)=O)CC3C)c[nH]c12 c1(C(=O)NCCN(C(c2ccc(F)cn2)=O)CC)cccc(C)c1O c1(CN(C(=O)CNC(=O)CC2CC2)CC)cccnc1 C1(NC(CCC2(NC=O)CCCC2)=O)CCN2CCC1C2.C1C(=O)N1 Cc1c[nH]c2ncc(C(N3CC(NC(c4cc(C#N)c[nH]4)=O)C(C)(C)C3)=O)cc12 C1(OCCCNC(C2CC3CCC3C2)=O)CCN(C(=O)C=C2CCCC2)CC1 Cc1ccc(OCCC(=O)NC2CCC2NC(=O)C(C)n2cncn2)c(C)c1 C(C1CCCCCC1)=CC(=O)NCC1CCCC(NC(c2n(CC)ccn2)=O)C1 C1(CCCC)CCC(N=c2nc(N3CCC4(CCN(C)C4)C3)c3sccc3[nH]2)C1 C1(N(C(c2sc(Cl)nc2C)C(=O)NC2COC2)CC)CCC(CC2CC2)CC1 c1(OC)cc(N(C)C)ccc1C(=O)NCCCCCCNC(=O)C#CC1(C)CC1 Cc1cccc2c(=O)c(C(=O)NCC(C)NC(=O)CC(F)F)c[nH]c12 Cc1ccc(Cl)c(C(=O)NCC2(O)CCN(C(=O)C(C#N)C3CC3)C2)c1 c1(C(=O)NC)cc([N+](=O)[O-])ccc1N1CCN(CCOC(C)C)CC1 C1(NC(C=C(C)C(C)C)=O)CC(c2ccccc2)CO1 N1(C(CCC#C)=O)CCC(C(=O)N(CC)Cc2ccccc2)CC1(C)C N1(c2n(CCC#C)c(-c3ccc(Br)c(C)c3)nn2)CCc2c(I)n[nH]c2C1 C1(NC(C=CC(=O)NC2CCCC2)=O)C2CCC(C2)C1CN(CCCC)C1CC1 C1(C(C)C)(CNC(c2cccnc2)CNC(=O)OC(C)(C)C)CCCCO1 c1(N2CCN(C(C(=O)NCCCC)COCC(C)C)CC2)nsc2ccccc12 C(=O)(C#CC1CCOC1)N.N1(CCNC(CNC(C(C)C)=O)=O)CC2CC2C1 c1(C(N(CC(C)CNC(C2(c3ncco3)CCC2)=O)C)=O)nc2ccccc2[nH]1 C1(O)(CN(C(=O)Cn2cc(C3CC3)nn2)C)CCN(C(=O)Cn2cnnc2O)C1 CCCC(CC(=O)NC(C)C(N)=O)NC(C1C=CCC1)=O N1(C(c2cc(C)[nH]n2)=O)CCC(C)(C)C1CC(N1CC(OCC(N)=O)C1)=O Cc1cc(Br)ccc1CNc1c[nH]nc1C(=O)NCC1COCCO1 CC1=CC(C)CN(C(=O)NCc2cccnc2N(C)C)C1 c1(CC(C)N(C(c2c(C)c(I)c[nH]2)=O)CCO)cccc([N+](=O)[O-])c1 Cc1cccc(NC(c2nnnn2CC(F)F)C=Cc2ccccc2)c1 N1(Cc2n(C)ccn2)CCN(C(C2CCC(Cc3cccs3)CC2)=O)C2CC12 C(=O)(C(C)(C)C#N)NCCOCCCN(C(C1C(CC)C1)=O)C C1(NC(C(CCC)OCC)=O)CCCN(C(c2ccc(C#N)o2)=O)CC1 N1(C(CC=C)=O)C2CCC1CN(C(=O)C(C1CCOC1)NC(C)=O)C2 C1(C(N2C(CCC)CCC2)=O)CC(C)(C)CCN1C(c1cc([N+](=O)[O-])c[nH]1)=O CC1CCCCC1(C)C(N1CCC(C(=O)Nc2ccccc2)C(C)C1)=O C1(C(N(CCCNC(=O)CC2CSCCS2)C)=O)CCc2nnc(O)cc2C1 c1(C(=O)NC(C2CN(C(C3CN4CCN3CC4)=O)C2)C)ccc2c(c1)ncn2C C(=O)(CCCCC#N)NCc1c(C(N2C(C)CCC2)=O)cco1 c1(CC)nc(N2CC(CC(C)NC(c3ncccc3C)=O)C2)[nH]c(=N)n1 C12(NC(C3C(NC(c4cccc(C)c4F)=O)CCOC3)=O)CC3CC(CC1C3)C2 C1(C(=O)NCC2(C(=O)NC(c3ccn(C)n3)C)CCCO2)CC(=O)CCO1 C(=O)(N=c1cnn(C2CCOC2)[nH]1)N(CCC#N)CC C(=O)(C(O)CC[S+](C)C)N(CCNC(CC(C(C)C)O)=O)CC1CC1 c1(C(N2C(CC)CCC2C)=O)ccc(C#N)c(C)c1 C1(C(N(CCOC)CC2CC2)=O)CCN(C(=O)C(CO)C(C)(C)C)O1 Cc1nccc(C(=O)NCC2CCC(NC(c3ccnnc3Cl)=O)C2)n1 N1(C(C(C(CC)C)N(C)C(C2CC3CCC3C2)=O)=O)CC2CCC(C1)C2C#N C(CCCCC(=O)NCC(CO)NC(c1cccc(F)c1C(F)F)=O)OC c1(C(=O)NCC(CC=C)NC(=O)CC2C=CS(=O)(=O)C2)ccc2nn[nH]c2c1 c1(C(=O)NC(CNC(C(C(C)C)F)=O)C2CCC2)cc(F)cc(Cl)c1N CC(C)CC(C(=O)OCc1cc(C(C)C)co1)C(C)C C1(C(N2CC(NC(=O)CC(=O)N(C)C)CC(C)(C)C2)=O)CC2OC(C)(C)OC2C1 c1(CNC(c2n(CC)ccc2)c2nnnn2C2(C)CCCC2)cnc(N(C)C)cn1 C1(NC(CC2CC(C)N(C(=O)CC3CC4(CC4)CO3)C2)=O)CCOC2(CCC2)C1 N1(C(C(CC)(C)CNC(=O)CCc2cnccn2)=O)CCC(=C(F)F)CC1 Cc1c(C(=O)NCCC(C)NC(=O)CC(c2cccc(F)c2)C)ccn1C c1(C(N(CCCNC(C(C)C(F)F)=O)C2CC2)=O)n[nH]c2c1CC(F)(F)CC2 N1(C(C(CC#C)NC(c2cc(CC)nn2C)=O)=O)CC2CC(O)CC1C2 c1(C(=O)NCC2CC(NC(c3c(C)cc(C(F)(F)F)s3)=O)C2)ccc([N+](=O)[O-])[nH]1 N1(C(CC2CN(C)C2)=O)CCCN(C(C2(C(C)(F)F)CCC2)=O)CCC1 C1(C(=O)NCC(C)NC(c2cc(CC)nnc2C)=O)CCCN1S(=N)(=O)N(C)C c1(C(N2CCC(C)C2CNC(C2C=CCC2)=O)=O)cc2n(n1)CCCO2 C1(N)CN(C(=O)C(c2ccccc2F)=O)C2CCCC12.C(CO)(C(=O)C(N)=O)N CCC(CNC(c1cccc(F)n1)c1nnnn1CCOC)(CC)CO Cc1ccc(C)c(CC(=O)NCCNC(=O)C(c2cccc(Br)c2)C)c1 C12(C(=O)NCC(CN(C(c3c(CC)occ3C)=O)C)O)CCC(CC1)C(C)(C)O2 C1(C)(CNC(C2N(CCC)C(=O)CC2)=O)CCN(C(C2(CCO)CC2)=O)CC1 C(=O)(C1=C(CC)OCCS1)NCC(CC)(CC)NC(=O)CC(C)(F)F N1(C(C(CC)NC(N)=O)=O)CC2CCC(NC(=O)Cc3ccoc3)CC2C1 n1(CC)nc(C)c(CC(N2CC(OC)CC2CNC(=O)CC(O)C(C)C)=O)c1C C(=O)(CCCCCn1cc(C(C)(C)O)nn1)N(C)CC1CCN(C)C1=O C12(C(=O)NC3(C)CCN(C(c4cc(C5CC5)on4)=O)C3)CCC(CC1(F)F)C2 c1(CC(=O)NC23CC(NC(C(Cc4ncn(C)c4)O)=O)(C2)C3)cc(F)ccc1O CCCC(C(=O)NCCOCCCNC(c1ccoc1Br)=O)c1ccccc1 CC1OC2(C)CC1(C(=O)NCCC1CCN(C(=O)COc3ccccc3)C1)C2 C=CCC(CNC(C1CC(CC2CC2)C1)=O)NC(c1ccc(C2CC2)s1)=O N1(C(CCc2cncc(C)c2)=O)CCCCC12CCCN(C(=O)C(Cl)Cl)C2.C([O-])C c1(C(N2CCCC(N(C)C(C3CCC(F)(F)CO3)=O)C2)=O)ccn2ccccc12 N1(C(C2(OC)CCSC2)=O)CC2(CCCC(CNC(=O)CCOC(C)C)O2)C1 N1(C(c2scc(OC)c2)=O)CC(C)(C)CC1CNC(c1cc(C)sc1C)=O c1(C(N2CCN(C(C(CCC)C(C)C)=O)C(C)CC2)=O)cccc2c1C(=O)CC2 N1(C(c2nc(CNC(C3C(C(=C)C)OCC3)=O)oc2C)=O)CCN(C)C(C)(C)C1 CC1(C)CC(=O)NC1C(=O)OC1CCC=CCC1 CC(C)CC(O)C(C)C(=O)N1CC2(CC(NC(=O)C(=O)N=S(C)(C)=O)CO2)C1 C1(CNC(C2CC2F)=O)CC(F)(F)CN1C(c1ccc(F)s1)=O N1(C(C(C)=CC2CC2)=O)CCN(C(C2CCCN2C)=O)CC(C)(C)C1 C(=O)(C#CC1CCOCC1)NC(CNC(C(c1cccc(C(F)(F)F)c1)CC)=O)C c1(NC(C2C3(CC(NC(C4CCCN(C)C4)=O)C3)C2)=O)nccn2cnnc12 C12CCC(CC1)C(=O)NC2.C1(NC(C(C)N(C)C)=O)(CO)CCCCC1 c1(-n2cc(C(=O)OCCN(C)C)nn2)cccc(OC2CC2C(C)(C)OC)c1 N1(C(c2cc(C)c(C)nc2O)=O)CCC2CCC(C1)N2C(C12CC(C)(CO1)C2)=O N1(CC(=O)N(C2(C(C3CC3)NCC3CC3C3CCCO3)CC2)C)CCNC1=O C1CC2CCC(C1)N2S(=O)(=O)C1CCCCC1.Nc1cccnc1C=O c1(CNC(c2ccc(Cl)cc2)C(N2CCC(CCC)C2)=O)ccc(F)cc1 c1(C(N(CC(=O)OC)Cc2nc(C(F)(F)F)cs2)=O)cnn2c1CNCC2C(C)C C(=O)(C1CCCc2nn[nH]c21)N(C1(CNC(=O)CN2CC3CC3C2)CCCC1)C Cc1scc(C(=O)NCCCOCCN(C)C(C2(C#N)CC2C)=O)c1C C1(OC)CN(C(=O)C(=Cc2c[nH]cn2)F)CC1C(=O)NC1CCC(=O)NC1 C1(CNC(C2(OC)CCC2)=O)CC(NC(=O)C=Cc2ccncn2)CCO1 C(=O)(CS(=O)(=O)CC(=O)N(C)CC1CCN(C(c2ocnc2C(F)F)=O)C1)OC CC(C)CCCC(C)C(=O)NC(C)CNC(=O)Cc1ccc(F)cn1 C1(NC(C=CC(C)(C)C)=O)C2CC3CN(C(C4(CN5CCCC5)CC4)=O)C1C3C2 C1(C)(NC(Cc2c(C)occ2)=O)CCCN(C(=O)CCCc2ccsc2)C1 C(CN=c1cccc(S(=O)(=O)NCCn2cc(C#N)cn2)[nH]1)N(C(=O)OC)C Cc1nc(C(N2CCCC(c3nc(C)c(C)[nH]3)C2)C(=O)NC(C)(C)C)nn1Br CC(CNC(c1ccc(N(C)C)cn1)=O)CN=c1[nH]cc(C#N)c2ccsc12 C(=O)(CC(O)C(Cl)(Cl)Cl)NC1CCCCN(C(CCCCOC)=O)C1 N1(C(COCCCC#C)=O)CCCC(CCCCNC(C2CCN(C)C2)=O)C1 CCCCC(CC)CCC(=O)NCCC(C)N(C(=O)CC1CC(=O)NC(=O)C1)C N1(C(c2cn(CC)nn2)C(=O)NCc2ccnn2C)CC(C(F)(F)F)CC1CO c1(C(N2CC(C(N3CCC(Br)C3)=O)C(F)C2)=O)cc([N+](=O)[O-])ccc1Cl C(N=c1[nH]c(N2CCOC(CC(N)=O)C2)nc(=NC)[nH]1)c1cc(COC)no1 C1(CC(CNC(=O)C(c2cn(C(C)C(=O)O)nn2)N2CCOCC2)O)CC(F)(F)C1 C1(NC(C2(COC)C=CCC2)=O)CC(OC)CN(C(=O)C(CC(C)C)OC(C)=O)C1 C1(C(N(C2CCN(C(c3cc(F)ccc3F)=O)C2)C)=O)CC(C)(C)CCO1 Cc1cn2ccc(C(=O)NC(C)(C)CNC(c3cc(C)n(C)c3C)=O)cc2n1 C(=O)(CCCC(=O)NCC1(COC)CCN(C(C2(CF)CCC2)=O)C1)NCCC c1(N2CCC(CNC(c3c(OC(C)=O)ccc(F)c3)=O)C2)nc2ccc(C)cc2s1 Cc1nccc(C(=O)NCC2CC(NC(=O)CCC3NC(=O)NC3=O)C2)c1N C1(C(C(C)NC(=O)CC2(F)CCC2)NC(COCC(=C)C)=O)CCCCC1 C(C(=O)NCC(C)CNC(c1ncn(C)n1)=O)(C(C)C)NC(=O)OCC C1(C(N(C(C)CNC(c2c(C(F)F)cnn2C)=O)C)=O)CC12CC(C)(C)C2 C=CCC(CC)C(=O)NCC1CN(C)CCN1C(c1cnc(C2CC2)nc1O)=O C=CC(C)(CC)C(=O)N1CC2CC(NC(=O)C(C)Cc3cccc(F)c3)C2C1 C(=O)(C(CN(C(=O)Cn1ccnc1)CC)C(C)C)N(CC(C)O)CC C1(C(N2C(CNC(CCc3c(C)cccc3)=O)COCC2)=O)COCC(C)(C)O1 CN1C(=O)CCCC1C(N1CCCC(CCO[Si](C)(C)C)C1)=O.C1(=O)CCC(=O)N1 N1(C(C(CC)SC)=O)C(C)CC2CN(C(c3ccc4sc(C)nc4c3)=O)CC12 C=CCC(CNC(=O)CC(C)(C)c1cccs1)CO c1(C(=O)NCCc2ncoc2CNC(C2CN(CCF)C2)=O)cscc1F c1(C(=O)NC(CNC(C2(CC)CCC2)=O)C2CC2)cccc(C2CC2)n1 c1(NC(C2(CCNC(c3ccc(C)cn3)=O)CC2)=O)cnc(Cl)c(C)c1 N1(C(c2ccc3cccnc3c2)=O)CCOC2(CCN(C(C3(Br)CCC3)=O)C2)C1 Cc1cc(C(N2CC(C(C(=O)N(C)CCN3CCOCC3)N(C)C)C2)=O)c(C)nn1 C1(NC(C(CCF)NC(c2cn(CC)nc2C)=O)=O)CCC(=O)N(C)C1=O CC1(C)CN(C(=O)CCn2cnccc2=O)CC1NC(c1cc(C(N)=O)no1)=O c1(C(=O)NC2C(NC(C(c3c(C)noc3C)C)=O)CCCC2)cc2n(c1)CCC2 N1(C(c2c(CC)ncnc2)=O)CC(NC(c2cc3scnc3[nH]2)=O)CC2(CC2)C1 C(=O)(CC(C(F)(F)F)NCC)N(CC1(F)CC(C)C(OCC)C(=O)NC1)C C=Cc1cc(C(=O)NC2CCCN(C(=O)Cc3cc(C)nc(O)c3)C2)cc(F)c1 c1(CC(N2CCC(C)(CNC(c3c(SC)nn(C)c3)=O)C2)=O)cc(Cl)ccc1Cl C=CC(CC)CC(=O)N1CCN(C(=O)C(C)CC)CC1C(C)(C)C Cc1nc(NCc2cc(C3CC3)n[nH]2)cc(N2CCC(n3nccn3)CC2)n1 c1(CN2CCC(NC(c3c(C)nn(CCO)c3)=O)C(O)C2)cnc2occc2c1 C(=O)(CCN=c1[nH]ccs1)N1C(CNC(c2nccc(C)c2)=O)CC(F)C1 c1(C(=O)NCC(CCNC(C=CCC)=O)O)cc(Cl)ccc1OC(F)(F)F c1(CC)cc(C)ccc1C(=O)NCCC1CC(NC(c2c[nH]cc(C)c2=O)=O)C1 c1(CN(C(C(C)NC(C(C)SCC)=O)=O)CC)ncc(F)cc1C N1(C(C(C)=C(C)C)=O)CC(F)(F)CC1CNC(c1c(Br)noc1C)=O Cc1ccc(OCCCCNCc2ccncc2C(F)(F)F)c(F)c1 C1(O)(CNC(c2cc(C(=O)OC)no2)=O)CCCN(C(=O)C(C)Cc2cnc[nH]2)C1 Cc1nc(C(=O)NC2CC(F)CN(C(C3CCC(O)CC3)=O)C2)c2n1CCCC2 C(=O)(C(C)(C)CS(C)(=O)=O)N1CC(OC)C(NC(c2cc(Cl)n(C)n2)=O)C1 c1(OC)cccc(F)c1-c1cccc(NC(=O)CC2SC(=N)NC2=O)c1 c1(NC(=O)CC2CCC(NC(c3c(O)cccc3F)=O)CC2)cc(Cl)c(Br)cc1Cl C(N=c1[nH]c(C#N)c(Cl)s1)C1C(C(F)(F)F)CCN(C(c2n(C)ccn2)=O)C1 C#CC1(NC(C2(CC)CN(C(=O)CN(C)CCOC)C2)=O)CCC(C)CC1 N1(C(CN(C)C)=O)CCOCC1CC(=O)NCc1cccc(F)c1 c1(C(=O)NCC(C)=CC(=O)NCCCn2cc[nH]2)c(C)oc(C)c1S(N)(=O)=O C1(NC(CSCC=C)=O)CC2CC(NC(c3cccc(C(C)(C)C)n3)=O)CC12 c1(C(=O)NCCC(=C)CNC(=O)C(C)(C)C2CC2)nc(C(F)(F)F)oc1Br c1(C(=O)NCC(C(C)C)NC(=O)CCc2ccc[nH]2)cccc2occ(Br)c12 C1(CCC(=O)NC2CC(C)(NC(=O)CC#N)C2)NC(=O)NC1=O C1(CCNC(CNC(c2c(CN)coc2)=O)=O)CCCCC1O N1(C(C(c2c(C)noc2C)C)=O)CC2CC(NC(c3cn[nH]c3)=O)C1C2 Cc1ccccc1C=CC(=O)NC1CCOC1C(=O)Nc1cncnc1O CC1CC(CNC(C2(P(C)(C)=O)CC2)=O)CN1C(c1coc(C2CC2)n1)=O n1(CC(=O)NCC(CNC(=O)C(O)CN2CCCC2)OC)ncn(C)c1=O C1(C)(CC(=O)N(CC(CN(C(=O)CCNc2ccccn2)C)O)C)CC1(F)F C1(CNC(C2(OC)CCSC2)=O)COC(C)(C)CN1C(=O)COCC1CCC1 c12nccnc1N2.C1(C(N2CCC(NC(C3CCCC3)=O)C2)=O)(CO)CC1(F)F Cc1ncc(C=CC(=O)NCC2(C)CC(NC(C3CC3Cl)=O)C2)s1 N1(C(=O)NC(C(=O)N(C)CS(C)(=O)=O)C)CCCCC1c1cccc(O)c1 CC(C)CS(=O)(=O)NC1CC2(CCO2)C1 C1(CC(N2CCC(C(C)NC(c3cnco3)=O)C2)=O)CCCC(F)(F)C1 Cn1cnc(C=CC(N2CCC(C(F)CNC(c3cc(F)c[nH]3)=O)CC2)=O)c1 Cn1nc(C(F)(F)F)cc1C(N1CCC(C(N2CCC(C)(C)C2)=O)C1)=O C=C(C)CC(C(=O)NC1CC2CC(OC)C2C1)NC(C1CC(=C2CC2)C1)=O N1(c2n(CCC#C)c(C(c3ccccc3Br)C)nn2)CC2(C1)CC(C)(O)C2 C1(C(N2CCC(N(S(C)(=O)=O)C)C2)C(=O)NC(CC)C)CCC2COCCC2C1 C1(CC(C)C)COCCN1C(=O)NCC(c1cn(C)nn1)(C)C C(CNc1c(-n2c(C(C)OC)nnn2)ccc(OC)c1)(CCS(C)(=O)=O)OC CC1CN(C(c2ccnc(C(F)(F)F)c2)=O)CCC1NC(=O)CCOC1CCC1 C1(F)(CNC(CC2CC(=C)C2)=O)CC(NC(=O)Cc2cnccn2)C1 C1(C(C)C)CN(C(c2cscc2Br)=O)CCN1CC1CCC(C)CC1 c1(-c2cc(C(N(CC(C)N(C)C(C3CCCS3)=O)C)=O)sn2)ccc(Cl)cc1 C1(NC(CCOCCOC)=O)CC2(CCN(C(c3cc(Cl)ccc3C)=O)C2)C1 c1(CC)ccccc1C(C12COCC(C1)C2)NC(=O)C(=O)Nc1cccs1 c1(C(=O)NC2(CC=C)CN(C(=O)CCN(C)CCC)C2)nc(Cl)sc1Br C=C(Cl)C(C)(C)C(=O)NCC(O)CN(C(=O)COCCOC(C)=O)C CN1CCCC(CC(=O)NC2CCCC2CN=c2[nH]nc(C3CC3)o2)C1=O C1(N(C(=O)CC2CC3(CC3)C2)C)CN(C(=O)CC2CCSC2)CC1c1nccn1C c1(CC(=O)CC2N(C(C=CCOCCOC)=O)CC=C2)ccc(C(=O)OC)nc1 c1(CCC)n[nH]cc1C(=O)NCC(CC)NC(=O)CC(C)N(C)C C1(C(=O)NCC(C)(C)NC(=O)C(F)C2CCCC2)CCCN1C=O C(CS(=O)(=O)CC(=O)NCC(C1CCN(C(=O)CC2CC(OC)C2)CC1)C)OC C1(CNC(c2c(OC)scc2)=O)CCCCN(C(c2cnn(C3COC3)c2)=O)C1 C1(C)(C(NOc2c(CC)ccnc2)=O)C=CCN1C(=O)C(C)O c1(C(=O)NCC(CNC(COCCC(C)C)=O)O)n[nH]c2ccc(Cl)cc12 C(=O)(C(CC(F)F)NC(C1CC(F)C1)=O)NC1(C)CS(=O)(=O)C1 C1(N(C(C2C(C)=CCS2)=O)C)CN(C(=O)C=CC2CCC2)CC12CC2 C1(CC(=O)NCC=CCNC(=O)CCc2nc(C(F)(F)F)n[nH]2)CC2CCC1O2 C1(OC(C)C)CCCN(C(=O)C(CNC(=O)CC2CCCCO2)CC2CCCC2)C1 C1(C(N2CCC(=C)CC2)=O)CN(C(=O)C=CCC(C)(C)SC)CC(C)(C)C1 N1(C(CC(=C)Br)=O)CC(CNC(=O)COC2CCOC2)C2(CCC2)C1 c1(C(=O)NCCOCCC(=O)NCC2COCC2O)cnc2scnc2c1 N1(C(CCC=CCC=C)=O)CC2CC1CN2C(c1nccc(OC)c1OC)=O N1(C(c2c3cccc(C)c3ncc2C#N)=O)CCCC2NC(=O)C(C)(C)C12 c1(C(=O)NC(C)CN(C(=O)CNC(=O)Cc2cnn(C)c2)C)ccc(Cl)nc1 N1(C(CC(C(C)C)O)=O)CC2C3CCC(C2C1)N(C(c1ccc(C(F)F)s1)=O)C3 C1(CCNC(C2C(C)CC2)=O)CN(C(c2n[nH]cc2Cl)=O)CCS1(=O)=O C(c1ccc(C(N)=O)o1)=CC(=O)NCC1(CNC(CC(C)F)=O)CC1 C1(CNC(CCOCCN(C)C)=O)CC(F)CN1C(c1cc(=O)n(C)o1)=O CCC(C)(C)CC(=O)NC(C)C(C)NC(c1ncoc1-c1cnn(C)c1)=O C1(OCC)CCCCN(C(=O)CCCn2cc(Cc3ccc(SC)cc3)nn2)C1 N1(C(c2ccc(C(N)=O)o2)=O)CCCC(CNC(=O)CCF)CC1 c1(C(N2C(C)(CNC(C3CCOC(=O)N3)=O)CCC2)=O)cc2c(nc1N)CCC2 N1(C(c2c(C)ncs2)=O)CCOC(NCCCO)C1.C1C(=O)N(C)CCO1 C1(NC(CSC)=O)CCCN(C(=O)CCCOC(C)(C)C)C1C.C1CO1 N1(C(C(C)=C(CC)C)=O)CC(NC(=O)Cn2nnc(-c3ccsc3)n2)CC(O)C1 N1(C(CC(=C)C)=O)CCC2(CCN(C(=O)C(C)C(F)F)CC2)C1 C#CC1CCN(C(C2(C(C)NC(c3nc(C)oc3C)=O)CC2)=O)C1 N1(C(CCC=C(C)C)=O)CC2(C1)SCCC2NC(=O)C(c1c(C)noc1C)C Cc1ccc(O)c(NC(C2CCC2C(N)=O)=O)c1 c1(C(=O)NC(C2CCN(C(C(C)=C3CC3)=O)C2)(C)C)ccc(C(C)=O)cn1 Cc1oc2ccccc2c1NC(=O)NCC1(S(=O)(=O)CCN2CCOCC2)CC1O N1(C(C2CC=C(C)CC2)=O)CCC(C2CC2)(CNC(=O)Cc2ccnc(C)c2)C1 c1(-c2cn(CCC(C)C)nn2)ncc2ccccn12 C1(C(=O)NC2CC(CNC(=O)C3=CCCOC3)C2)CCn2c(O)nnc2C1 N1(C(C(C(=O)OCC)(C)C)=O)CCC2(CC(NC(C3CCC(=O)N(C)C3)=O)C2)C1 c1(OCC)ccc(-c2cnc(C(=O)NCCSC(C)(C)C)cc2C)c(C)n1 N1(C(C=CC)=O)CC(CN(C(c2cnoc2-c2cnn(C)c2)=O)CC)C2(CCC2)C1 O=S(=O)(c1cc2cc(F)ccc2s1)NCCc1nc2n(n1)CCCC2 N1(CC)CCC(C2(O)CCC2)CC1.c1(CC=O)ccsn1.C1CCN1C c1(C(=O)NCc2cc(C)nc(CO)c2)cc([N+](=O)[O-])ccc1C CC1CCC(CNC(=O)C(Cc2cn[nH]c2)NC(=O)C(C)CO)C1 c1(C(N2CC(CNC(=O)NC(C)C)C(C)(C)CC2)=O)c(F)cccc1[N+](=O)[O-] C1(NC(COCCC=C)=O)C(C)CN(C(=O)CN(C)Cc2sccc2C)CC1C C1(NC(=O)CC2COCCO2)CC2(C1)CC(C(=O)NCC13COC(CF)(C1)C3)C2 CCCCCC(=O)NCc1nc(CNC(=O)C(CCSC)OC)cs1 c1(N2C3CC(=C)CC2CCC3)nc(=NCCC2(OCC)CCC2)[nH]c2c1COCC2 CC1COC(C)(C)CN1C(Cc1ccccc1)C(=O)NCP(C)(C)=O c1(C(C(=O)NCCCNC(C2CC23CC3)=O)O)ccc(F)c(Cl)c1 Cc1[nH][nH]c(=NC(=O)C2C=CC(NC(c3ccc4n[nH]cc4c3)=O)C2)c1Br C1(CNC(c2cccc(SC)c2)=O)C(C)CCCN1C(=O)CCC1CCC1 N12CCC(CC1)n1cc(nn1)C2.C1(NC(=O)COCC2CC2)CC(F)C1.C1(C)CC1 C1(C(NOCCC(C)C)=O)CN(C(=O)CCc2cccnc2)CCC1(C)C C1(C(=O)NCCC2CC2C)(COC)CCN(C(C2CCCCN2C)=O)CC1 CC(C)(C#CC(=O)NC(CC#N)c1cccs1)CNC(C1CC1F)=O C1(NC(C(C(C)O)(F)F)=O)CC2(CCCCN2C(c2cnncc2O)=O)C1 c1(OC)ncccc1CC(=O)NCC1CN(C(c2cccc(C(C)(F)F)c2)=O)C1 c1(NC(C(C2OCCC2COC)NC(CC)(C)c2nccs2)=O)ccccc1Cl c1(C(=O)NC2CCC(NC(Cc3cc(OC)ncc3)=O)C2)ccc(S(C)=O)cc1 Cc1nccc(C(=O)NCC23CC(NC(c4cc(CO)oc4C)=O)(C2)C3)c1C N1(C(C2N(C(C)=O)CSC2)=O)CCCCC1CNC(=O)CCCc1cccs1 C1(CCC)CN(C(c2cccc(COC)c2)=O)CCN1C(=O)C(C)C(F)F c1(OCCCC)cccc(OC(=O)C(CC)SCC)c1 c12ccc(OC)c(c1)CN(C)C2C(=O)NC.c1(SC(C)CC#N)ccccc1 C(=O)(CCSC)N(CC(=O)NCC(F)F)CCOC N1(C(C=C(C)CN2CCOCC2)=O)C2CCC1C(NC(=O)CSC(C)(C)C)C2 C(=O)(C1=CCCN(C(=O)CCCOC)C1)NC(CC#C)C(N)=O C(C)(C)(CCCCC(=O)N1CC2CC(NC(c3cnc(C4CC4)[nH]3)=O)CC2C1)OC c1(C(=O)NC2CC(C)N(c3cc(C4CC4)ncn3)CC2)occ2c1CCOC2 N1(C(C2CCCC(=O)N2)=O)CC2(CCC2NC(=O)C(=C2CCCCC2)F)C1 N1(C(CC(CC)(F)F)=O)CCOCC12COCCN(C(=O)CCC(C)O)C2 C1(NC(C=C(CC)CC)=O)CCN(C(C2CN(CP(C)(C)=O)C2)=O)CCC1(F)F c1(C(=O)NCC(C)NC(c2nnn(COCC)c2N)=O)ccc2c(c1)CN(C)C2 CN1C(=O)CCC1(C)CNC(C1C=CCN(C(c2ncncc2N)=O)C1)=O N1(C(CCCC#CC)=O)CCC2(CC1)CC2CNC(C1(COCC)CC1)=O O=C(N1OC2C=CC1CC2)C1CCN1C(C1(F)CC=CCC1)=O N1(C(=O)COCCN2CCOC2=O)CCC(CO)C1c1ccccc1 Cc1ncc(Cl)cc1CC(N1CCC(NC(=O)CC2CNC(=O)C2)C(O)C1)=O c1(CC(=O)NC(CC)CNC(=O)Cn2nc(Cl)ccc2=O)c(C)cc(C)cc1C c1(CC(N2CC(CCNC(=O)C=Cc3cn[nH]c3)OCC2)=O)cc(F)ccc1O c1(C(N(CCCCN(C)C(C2(N(C)C)CC2)=O)C)=O)cnc2c(Br)c[nH]c2c1 Cc1cc(C(N2CCC(O)(CCNC(C3(C)CCC3)=O)C2)=O)c(C)cc1Cl c1(C(=O)NC2C(CNC(C(C)n3ccnc3)=O)COC2)ccc(P(C)(C)=O)o1 C1(C(=O)NC(C)(CNC(=O)CSCc2ncnn2C)CO)CCCS1(=O)=O CC1(C(=O)NC2CC(C)(NC(=O)CCc3cncnc3O)C2)CCC(=O)NC1 C1(C(=O)NCC(c2ccccc2)NC(=O)CCS(C)=O)(NC(C)=O)CCCCC1 C(=O)(C1=CCCOCC1)NCC1CCC(NC(c2c[nH]c3nccc-3c2)=O)CC1 N1(C(C2CC(NC(C3(COC)CC3)=O)C23CCC3)=O)CCCN(CCO)CC1 CC1CC(N=c2[nH]c(N(C)Cc3cnn4c3CN(C)CC4)nc3c2CSC3)CS1 c1(CNC(=NCCCOC)NC2CCC(C)(C)CC2)ccc(S(=O)(=O)CCO)cc1 Cc1ccc2c(c1C(=O)O)CCCN2C(C1CCC(=O)N1C1CC1)=O c1(N2CCC(NC(c3cc(C)c(C)[nH]3)=O)C(C)C2)nc2ccc(N)cc2s1 c1(C(=O)NCCCNC(c2cc(-c3cccnc3)on2)=O)sccc1F C1(C(=O)NC(CN(CCC)CC)C)CC2CC1CC2NC(c1ncnc(C)c1C)=O c1(SC)nccnc1C(=O)NCCC1(NC(=O)CC2C=CCC2)CCCC1 c1(OCC(=O)NCCNC(COC)=O)ccc(NC(=O)CS(C)(=O)=O)cc1 N1(C(CC(C)N2CCCC2=O)=O)CCN(C(=O)CSCC(F)(F)F)CC12CC2 c1(C(=O)NCC(C)CN(C)C(C2CC(F)(CO)C2)=O)ccc2nn[nH]c2c1 c1(COc2cccc(CNC3C(C(=O)NCCCCO)C3)c2)cnc(Cl)c(F)c1 n1(C(CC)CC)nc(-c2cccnc2)nc1C(C(C)(F)F)c1ccccc1 c1(CCNC(CCOC2CN(C(c3cnc(C(C)C)o3)=O)C2)=O)ccc(F)nc1 N1(C(C=CCC)=O)CC2CC(NC(c3cc(Br)n(C)c3)=O)C(C2)C1 O=C(C#CC1CCCOC1)N1CCC(CCNc2ncnc(Cl)c2F)C1 CC1CCC(CNC(=O)COCC2CCCO2)N(C(c2cnc(C3CC3)o2)=O)C1 C1(CC)CN(C(c2cc(O)nc(C)n2)=O)CCN1C(C1CN(C2CCOC2)C1)=O c1(CCC(C)C)n[nH]c(=NCC2CC(NC(c3ccc(NC(C)C)cc3)=O)C2)o1 C1(CNC(c2cc(C(C)(F)F)ccn2)c2n(CCC)nnn2)CC=CCC1C C1(CC(=O)NCC2CCN2C(=O)C=Cc2cnccn2)COC2CC1C2 c1(C(N(CC(CNC(CC(CC)SC)=O)(C)C)C)=O)cc(C)ccc1N N(C(=NCCCN1CCOCC1)NC1CCC(F)CC1)CC1CCC(C)(C)CO1 N1(C(Cc2c(C)cn(C)n2)=O)CCC(C)C(C)(C)C1 N1(C(C(CC)C)=O)CCN(C(=O)CCc2nc(C(C)(C)C)no2)C(COC)C1 C(=O)(C1=NOC2(CCC2)C1)NC(C)(C)CNC(=O)CCCc1ccccc1Cl C1(c2nnnn2C2COC2)(NCc2n(CC)cnc2)CCN2CCC1C2 Cc1cc(=O)ccn1CC(=O)NCCCC1CN(C(=O)CC2(O)CCC2)CCO1 O=C(CCCCC1CCC1)NCC1(F)CN(C(c2c[nH]nc2F)=O)C1 N1(C(C(C)C)=O)CCC(NC(c2c(F)ccc(F)c2O)=O)CC(C)(C)C1 C1CCCCC1(F)F.CCC(C)C(=O)NCCNC(=O)CN(CCCOC)C1CC1 C1(C(=O)NCC2C(CNC(c3c(CC)noc3)=O)C2)CC12CCC(F)(F)CC2 CCCC(C(=O)NCCCCC1CC1C)NC(=O)CCOC(C)(C)C C(C1=CCN(C(=O)CCC2CCCN(C)C2)CC1)NC(Cc1c(C)noc1Cl)=O c1(CNC(C(C2CCN(C(=O)CCc3ccoc3)C2)C)=O)ccc(=N)[nH]c1 N#Cc1ccc(C(=O)NCC(F)CNC(c2cc3c(s2)CCC3)=O)c(F)c1 C(=O)(CCS(C)(=O)=O)NCC(=O)N(C1CCC(NC(C(CCC)C)=O)C1)C C1(C(C)NC2CC3(C2)CC3F)CCCC(C)(C)CC1 C1(CNC(CCC(=C)Br)=O)CCN(C(c2noc(C)c2C(=O)OC)=O)CC1C N1(C(c2ccc(OC)cc2I)=O)CC(C(=O)O)C2(C1)CN(C(=O)C(C)C1CC1)C2 N1(C(C2C(CCC)C2)=O)CC2(C)CC1(C(=O)N(C(CC)CC)C1CC1)C2 Cc1oc(C(C)C)cc1C(=O)NC1CC1NC(C1CCN(S(C)(=O)=O)C1)=O N1(C(C=C(C)Cl)=O)CCCCC(NC(c2cc(Cl)c(Cl)cc2O)=O)CC1 C1(CNC(N2C(C)CC(C(=O)OC)C2)=O)CCCCCC1C1CC1 c1(Cn2cc(C(CCC)NC(=O)CCc3cc[nH]n3)nn2)cc(Cl)ccc1C c1(Nc2c(Br)cc(OC)c(C)c2)ccc2ccccc2c1C N1(C(C(CCSC)O)=O)C2CCC1C(CNC(c1oc(C)nc1C(F)(F)F)=O)C2 c1(OC)cncc(C(=O)NC2COCC2NC(=O)CSc2c(C)n[nH]c2C)c1C C1(CC(N2CCC(O)C(O)C2)=O)C2CCCC2N1C(C1CCC(=O)N1)=O C1(NC(CCC(=C)C)=O)CC2CC(NC(=O)CNC(=O)NCC3CC3)CC12 c1(C(=O)NCC2C3CN(C(C4CC(C)OC4)=O)CC32)c(Cl)nc2ccccn12 CCC(C(=O)NC1(CCNC(c2ccc(F)c(F)c2)=O)CCCC1)C(C)(C)CC C1(C2CCCN(C(c3ccno3)=O)C2)(NC(c2cc(C)nnc2O)=O)CC1 Cc1cc(NC(c2nn(C)c(C)c2Br)=O)ccc1NC(=O)C(C)CC1CC1 C1(CNC(c2c(SC)snn2)=O)CC12CCN(C(=O)C(C)(C)N(C)C)CC2 N1(C(c2ccc(OC)c(Cl)n2)=O)CCC2(C1)CN(C(=O)Cc1cc[nH]n1)C2 C1(C(N(C2CCN(C(C(C)N(CC)CC)=O)C2)CC)=O)(N(C)C)CCCSC1 n1(CC(=O)N(CCCN(C(CC(COC)(C)O)=O)C)C)ccc2ccc(F)cc12 C1(NC(C2N(C(C3N(CC)CCOC3)=O)C3C(C2)C3)=O)C2CCCC1COC2 C(CC(C)CC(C)(C)C)NC(c1c(CNC(c2ccc(C)c(C)c2)=O)noc1)=O c1(CC)nc(C)[nH]c1C(=O)NC1CCCCC1CNC(=O)C(N1CCCC(C)C1)=O C(C(C)(C)C(=O)NCC1CC(O)CN1C(c1ccccc1Br)=O)N(C)C N1(C(C2CC(CC(C)C)C2)=O)CCCC2(C1)CN(C(=O)Cc1ccsc1)CCO2 C=C(C)C(C)(C)C(=O)NC1COCCN(C(c2cnn(C3CCCC3)c2C)=O)C1 c1(C(N2CC(CNC(C3CC(=C)C3)=O)C3C2C3)=O)cc(Br)cc2ccccc12 CCC(C(=O)NC12CC(C(=O)NC3(CCO)CCOC3)(C1)C2)C(C)(C)CC c1(C(=O)NC2CC(C)(NC(Cn3ncn(C)c3=O)=O)C2)cc(Br)cnc1C(F)F N1(CCC2CC(C)OCC2)C(=O)CN(Cc2ncc(Br)s2)C1=O c1(C2C(NC(C3C(NC(CNC(=O)NC)=O)C3)=O)C2)cncc2ccccc12 CC(C)CC(C)C(=O)NCC(C)NC(=O)CCC1C(=O)ON=C1C c1(NC(CCN(C(CC(OCC)OCC)=O)C)=O)c(C)cccc1Cl c1(OC)cc(C(=O)NCC2CC2NC(C23CC2COC3(C)C)=O)cc(C)n1 c1(N(CC(C)NC(C2CS(=O)(=O)CC(=O)N2)=O)C)ncc([N+](=O)[O-])cc1Cl c1(C(=O)NC(C(=O)NCc2onc(COC)n2)CN(C)C)ccc([N+](=O)[O-])o1 c1(C(=O)NC23CC(C(=O)NCCc4cc[nH]n4)(C2)C3)cc([N+](=O)[O-])c(O)cc1F Cc1cc(F)cc(C(=O)NCCC2CCCN(C(c3cc(CF)on3)=O)C2)c1N C1(F)(C(=O)NCC=CC(=O)NC(C2CCCO2)CO)CCCCC1 C(=O)(C1=COCCO1)N1CCC(C)(NC(c2c(C)nsc2)=O)C1 C(CCC(C)C(=O)NCC=CC(N1CC(=O)NCC1C)=O)OC c1(C(=O)NC(CCCC)CNC(C2CCCS2)=O)ccc(-n2cccn2)c(F)c1 CCC(CC)C(C(=O)NC1CC(O)(CNC(=O)CC2C(C)(C)C2(C)C)C1)OC CC1=C(C(=O)NC2CCN(C(=O)C=CC3CCCO3)C2(C)C)CCC1 c1(C(C)C(=O)NCCC2CCN(C(C3CN(C)C3)=O)CC2)noc2ccccc12 Cc1cn(CC(=O)NC2CC2CNC(c2nnsc2C2CC2)=O)c2ccccc12 C1(NC(C(C)SCCCC)=O)CCCN(C(c2ccc(C)c(C)c2)=O)C1C c1(CC)oc(C)cc1C(=O)NC1CCC(CNC(=O)C(CCO)N(C)C)C1 CC1SCCN(C(c2cc(C(=O)NC3OC4CCC3C4)nn2C)=O)C1C C1(NC(CC=C)=O)CC1C1CCN(C(c2cc(OCC)nn2C)=O)CC1 C(=O)(C(C)(C)CN(C)C)NCC(C)(CNC(=O)CC1CC(C)C1)OC Cc1nccc(C(N2CCN(C(=O)C=CSc3nc[nH]n3)C3CC23)=O)c1O O=C(CCCCO)Nc1cccc(CNC(C2CC23CCOC3)=O)c1 C1(C)(C(N(C2CCN(C(C)=O)C2)CCC)=O)CCN(C(c2cc(CC)no2)=O)C1 C(=O)(C(C)CC(C)CC)NCCOCCOCC.c1(O)cccc(OC(F)(F)F)c1 C(CC(C)C)(C(=O)NCc1ncccc1C(=O)N(C)CC1(O)CCC1)OC C=CCC(CNC(=O)CN(C)C(C)C)C(=O)NCC1CCOC(C)(C)C1 c1(C(c2nnnn2C)Oc2cccc(NCCCOC)c2)ccc2cc[nH]c2c1 C(C(=O)OC)(C(C)C(C)(C)C)N1CCC(N(C)CC2(C)CC2)(CO)C1.C(C)C N1(C(c2c(CC)cco2)=O)CCCC1(C(=O)NC(c1nc[nH]n1)CC)CC c1(OCC)ccc(C(N2CCC(N(C)C(c3ccc(C)cc3Br)=O)C2)=O)cc1O C(=O)(C1=C(Cl)CCCCC1)NC1(CC(N)=O)CCN(C(C2CC(C)(O)C2)=O)CC1 C1(CNC(=O)C=Cc2nccs2)CN(C(c2ccn(CCF)n2)=O)CCCO1 c1(C(N2CCN(C(C(CC(C)C)F)=O)CC2)=O)ccc2c(c1)N(C)CCO2 CC(C)CC(C(=O)NC1CNCC(C(=O)NCC(F)(F)F)C1)C1CCCCC1 N1(C(C2N(CC)CCCC2)=O)CCN(C(=O)CCS(C)(=O)=O)CC(O)C1 c1(C(N2CC(NC(C34OC(C)C(C3)C4)=O)C2)=O)ccc2ccccc2c1 Cc1cccc(Cl)c1C(=O)NCCOCCN(C)C(c1nscc1N)=O Cc1[nH]nc(CNC(=O)C=CCNC(=O)CC2CCCCO2)c1C N1(C(C2(CC#C)CCCO2)=O)CCCC(N(C(=O)C=CC=C(Cl)Cl)CCO)C1 c1(C(=O)NCC2(O)CN(C(c3cc(SC)c(C)o3)=O)C2)cnn2c1N(C)CC2 C(CN=c1[nH]nc(-c2ccon2)s1)C1N(C(C23C(C)OC(C)(C2)C3)=O)CCCC1 C1(C(=O)OC)CN(C(=O)CNC(=O)CCCF)CC1C N1(C(c2n(CC=C)ccc2)=O)CCCN(C(c2cc(OC)nc(F)c2)=O)CC1C C1(CNC(C=C(C)C2CCC2)=O)CCN(C(=O)CC2CCOC2)CCC1(F)F C1(C(=O)NCCCCC2(NC(c3ncn(CC)n3)=O)CC2)CCC(C)(C)C1 CC1c2c[nH]nc2CCC1C(N1CC(CNC(c2ccc(C#N)nc2O)=O)C1)=O Cc1cccc2nc(C(=O)N(C)CCN(C(=O)CCn3ccccc3=O)C)cn12 Cc1noc(C(=O)NCCCCCNC(=O)C(F)(F)c2csc(C)c2)n1 C(=O)(C#CC1(CC)COC1)NC1CC(C(C(=O)NC(CCC)C2CC2)F)C1 C=CCC(CNC(C1CC(C)N(C)C1)=O)C(=O)N1CCC(O)(C(C)C)C1 C1(OC)CC(CNC(=O)CCSC)N(C(c2cc(CCCO)on2)=O)C1 C1(C(N2ON=C(CCNC(CSCCCC)=O)C2)=O)CCC(N=[N+]=[N-])C1 C1(NC(c2ccn(COC)n2)=O)CN(C(c2ccc[nH]2)=O)CC1n1ccnn1 C(C(C)(O)CC1CCC1)NCC(CC)NC(=O)OC(C)(C)C CC1CCN(C(=O)C=CC(=O)NC2CC2)C1C(=O)NCCS(C)(=N)=O c1(C(=O)NCC(=O)NCC(COC)C)ccn(C)c1 C1(F)(CNC(C2CCCO2)=O)CCN(C(c2cccc(-c3ccoc3)c2)=O)C1 C1(CC#C)CCCCN1C(=O)CN(C)Cc1ccc(CO)cc1 C1(C(=O)NCCOCCN(C)C)CCN(C(C2CCCC(=O)N2)=O)CCO1 CC1=NNC(=O)C1CCC(N1CC2C(NC(=O)COc3cccc(F)c3)C2C1)=O Cc1cc(Cl)c(C(N2CCS(=O)(=O)C(CCNC(=O)CC=CCCO)C2)=O)cc1C CN1CCOC(C(=O)NCCCOCCCNC(c2cnn(C)c(=O)c2)=O)C1=O C(C(=O)N1CCC1(CO)CO)(C(C)(C)C)NC(c1c(CC)noc1)=O c1(C(N2CC3(CN(C(C(C)OC)=O)C3)C2)=O)cc(Br)cc2c1CCN2 CC(C)CCCCCC(=O)N1CC2CCC2(CNC(C2(C#N)CCCO2)=O)C1 N1(C(C(CO)OCC)=O)CCCC1(C)CNC(=O)C(C1CCCCCC1)O c1(-c2nnc(C(CC)NC(=O)NCCS(=O)(=O)NC)o2)ccccc1Br C1(C(=O)OC)CCC2(C1)CN(C(=O)Cn1cc(-c3cncc(Cl)c3)nn1)C2 c1(C(=O)NC23CC(CS)(C2)C3)cccc(C(N)=O)c1F.CC(C)CCCOCC c1(C(C(=O)NCC2CCOC2)N(N2CC=C(C)CC2)CC)ccnc(F)c1F C(=O)(C(C)(F)C(C)(C)F)N1CCN(CCCNC(C(C)c2cccs2)=O)CC1 N1(C(c2scc(C)c2)=O)CC2CCOC2(CNC(=O)C(O)C2CCC2)C1 S(=O)(=O)(c1ccc(NCC2CCC2CO)c(Cl)c1)NCc1c(C)scc1 CCC(CC(=O)NCC1CC(NC(=O)Cc2ccsc2C)C1)C(C)C CC1CN(C(=O)CSCc2cscn2)CCCN1C(c1nc(Cl)sc1Cl)=O C(CCCOCCO)NCCCN(C(C1CC1OC(C)(C)C)=O)CC C1(N(C(c2c(C)cno2)=O)C)CC2CCC(C1)N2C(=O)CCS(C)=O C(CNC(=O)CCn1ccnn1)(C(C)(C)C)NC(CCSCCC)=O C1(NC(COCC)=O)CCCC12CN(C(=O)CCn1ccnn1)C2 C1(c2ccc(OCOC)nc2)NC(=S)N(c2cccc(C)c2C)C2=C1C(=O)NCC2 C(=O)(C1=Cc2ccccc2C1)NC1C(NC(c2c(OC)noc2C)=O)CCC1 c1(OC)ccc(OCCSC(=O)NNC(=O)Nc2nn(C)cc2C(F)(F)F)cc1 C(=O)(CCCCC1CC1)N1CC(CC)(NC(C2(CCOC)CCCC2)=O)C1 N1(C(C2(C(C)C)CCN(C(C=C(C)C(C)C)=O)C2)=O)CC2CC(O)CC1C2 c1(C(=O)NC2CC(=O)N(C3CN(Cc4cocn4)C3)C2)c[nH]c(=O)c2ccnn12 c1(C(=O)NCCC2(CNC(C(COC)C)=O)CC2)cn(C)c(=O)cn1 Nc1ccc(F)c(C(N2CCN(C(=O)CN3CCS(=O)(=O)CC3)C3CC23)=O)c1 C(=O)(CCC(C)(C)NC(=O)CN1CCOCC1)N1C(CCN(C)C)CCC1 C1(C)(CNC(CCCCC=C)=O)CN(C(C2CSCCS2)=O)C(C)(C)C1 c1(OC)cc(-c2cnnn2C2CCOCC2)cc(OC)c1OC Cc1cc(C(=O)NC(C)CNC(c2csc(Cc3ccccc3)c2)=O)nc(O)c1 c1(OC)cc(OC)nc(C(=O)NCC2(C)CCN(C(C3NC(=O)CC3C)=O)C2)n1 Cc1ccc(Cl)c(OC(C)C(N2CCC(CNC(c3cc(C#N)cs3)=O)C2)=O)c1 c1(C(=O)NCCC2(O)CCCN(C(=O)CC(F)(F)F)C2)cnnc2ccccc12 c1(C(=O)NCC2N(C(c3c(C)nc(Br)o3)=O)CC2)ccc2c(c1)C=CCC2 c1(C(=O)NC(C2CCN(C(C3CCC(F)(F)C3)=O)CC2)C)cc(Cl)cc(Cl)c1O c1(C(N(C)CC2CC(C)(C)CO2)=O)cccnc1N.C12(CC1)CC(=O)NC2 N1(C(C(C(C)O)C)=O)CCOC2(CCCN(c3ncc4c(Br)cccc4n3)C2)C1 c1(C(=O)NC(C(=O)NC2CCC(=O)NC2=O)CC2CCC2)ccn2ccnc2c1 C1(CNC(C=CCCC(C)C)=O)CN(C(C2(F)CCC2)=O)CCC1C(F)(F)F CC1(C)CC(C(F)(F)F)CN(C(C(=O)NCCO)C(c2cc(F)c(F)c(F)c2)O)C1 C(=O)(C(CC)CCc1ccccc1)NC(CCCCNC(=O)COC(C=CC)=O)C N1(C(C(c2ccc(F)cc2)OC)=O)CC(NC(c2sccc2C(C)C)=O)C(C)C1 CC1(C)CC(C(N2CCC(C(=O)NCC3CCCC(=O)N3)CC2)=O)CCO1 N1(C(C(C)SCC)=O)CC(C(N2CCCC(F)(F)C2)=O)C2(CC2)C1 C(CC(=O)N1CCC2CC12)(CC(C)C)NC(C1(OC)CC(CO)C1)=O C(c1cccc2ccccc12)=CC(N1CCCCC(NC(=O)C=CCF)C1)=O N1(C(C(N=c2ncn(NC(=O)OC(C)(C)C)[nH]2)=O)=O)CCNC(=O)c2[nH]ccc21 CC(C)C1=NOC(C)(C(N2CC3CCC2CN3C(C2CN3CCC2CC3)=O)=O)C1 O=S(=O)(c1cccc(=NC2CCN(CCF)C2)[nH]1)N1CCCC1P1(=O)CCCCC1 N1(C(CCCC(=O)OC)=O)CCC2(CCN(C(C3CC3F)=O)CC2)C1 c1(CNC2CCCC(C(=O)NCc3cn[nH]c3)C2)cc(Cl)cnc1F O=C1NC2(C(=O)NC3CC(NC(C4(n5ccnn5)CC4)=O)C3)CC3CC1C2C3 C(=O)(C1(C)CCOc2ccccc21)N(C)CCNC(C1CC2C=CC1O2)=O c1(CC)nn(C)c(CC)c1C(=O)NCC(C)(C)CN(C(=O)CCCC#N)C C(=O)(CCCC(=O)N1CCC(CC(N2CCCCC2C(C)C)=O)C1(C)C)OC CCC(CC(=O)N1CCC(NC(=O)CN(C(=O)C(C)C)C)C(C)(C)C1)C(F)F C12(C(N(CC(C)(C)CO)C)=O)CC(C)(CN1C(C1CCC(=O)C1)=O)C2 c1(C(=O)O)ccnc(N2CCCCC2)n1.C12CCN(C1)C(=O)CCC1CC(C1)O2 Cc1ccc2c(-c3nc(C(=O)Nc4ccc(I)nc4)cs3)c[nH]c2c1 C1(=O)C(CC(C)C)CN(C)C(=O)CCNC(=O)C(C(C)O)N1.CN N1(C(C(C)n2cncn2)=O)CCC(NC(C2(C3CCCCO3)CC2)=O)C(C)(C)C1 C1(OC)CCn2cc(C(=O)NCC(O)CNC(c3cc[nH]n3)=O)nc2C1 C(CC(C(=O)N(C)CC1CCN(C(=O)C(C)SC)C1)NC(C)=O)SC Cn1nnc2ccc(C(=O)NCC3CN(C(=O)CCC(N)=O)CC(C)(C)C3)cc12 c1(C(=O)NC(CN(C(C(CC(C)C)O)=O)C)C)cc2ccsc2n1C Cc1cc(C(N2CCC(CNC(c3csc(Br)c3Cl)=O)C2)=O)[nH]c1C N1(C(=O)CC2CC3C=CC2CC3)CC2OCCN(C(=O)C=CC(F)(F)F)C2C1 CC(CCO)C(=O)NCc1ccc(CN(C(=O)C=CC2CCOCC2)C)cc1 C1(=O)C(O)C(C)(C)N1.C(C)(C)(C(=O)NCc1c(NC(=O)NC(C)C)scn1)SC CC1CCCN(CCN2CCCC(C(C)NC(=O)Cc3noc(C(C)C)n3)C2)C1 Cc1cc(F)c(C(=O)NC2CCN(C(c3cccc(F)c3Br)=O)CC2O)cc1F c12cc(ccc1Cl)-c1cccc(c1)C(=O)NCC2OC.C(CC(=O)O)NCC1CC1 C1(CCC)CCC(C(=O)NC2CC(NC(=O)C=CC3CCOC3)C(O)C2)CC1 N1(C(C(CC)(C)C#N)=O)CCC2(C1)CN(C(=O)CC1COC(C)(C)C1)CC(C)O2 C(=O)(C(CCOCC)NC(=O)CC1CC=CCN1C)NCC1CC(=C)C1 c1(C(=O)NCC2C(NC(C3(COCC)CCCCC3)=O)C2)ccc(OC)nc1Cl C=CCC(CC(F)F)C(=O)NCC1CC(F)(CNC(=O)C(C)(CC)CO)C1 c1(CNCc2cc(CO)on2)cnn(C(C)C)c1.CN1C(=O)N1 C(CC(=O)N1CCN(C)C2(CC2)C1)(C(C)(C)C)NC(C(C)=C1CC1)=O N1(CC(N)=O)C2CCCC1CC(SCc1nc(C)c(Br)cc1)C2 c1(NC)ccccc1C(=O)NCCC(O)CNC(=O)C=CCCC(C)C N1(C(CC2ON=C(C)C2)=O)C(C(=O)NC2(CO)CC(O)C2)CCC1C1CC1 CC(C)CCCCC(=O)NCC1C(CNC(=O)C(C)CC2CC2)C1(F)F c1(C(=O)NC2COCC2C(=O)Nc2ncccc2CO)cnc(O)nc1O C1(NC(C=Cc2scc(C)n2)=O)C2CCN(C(c3ccc(C)s3)=O)CCC12 c1(CCN(C(CC(CC)OC)=O)c2ncncc2OC)ccc2ccccc2c1 C1(NCC(c2c(OCc3ccc(F)cc3)ccc(Cl)c2)F)CCC12CCCCC2 c1(C(N2CC(NC(C34CCCCC3C4Br)=O)C2)=O)sc([N+](=O)[O-])cc1Cl C(N=c1[nH]c(Cl)nc2c1SCC2)c1ccc(C(=O)OC(COCC)C2CC2)cc1 c1(C(=O)NC2(C)CCN(C(c3cc(C)oc3C)=O)C2)ccnc2ccc(F)nc12 C12(C(=O)OCC)C3C4C1C1C2C3C41NC(=O)N(C1CCCCN1)C C(=O)(C(Cc1cn(Cc2cc(CF)on2)nn1)NC(c1cc(CO)on1)=O)OC C1(C(N2CCCC(CCC)(NC(c3csnn3)=O)C2)=O)Cc2cc(F)ccc2O1 c1(C(N(CC(CC)NC(=O)CC2CCC(=O)O2)C)=O)cc([N+](=O)[O-])ccc1C NS(=O)(=O)c1ccc([N+](=O)[O-])c(C(N2CCC(CNC(=O)C(F)(F)CO)C2)=O)c1 N#Cc1ccc(Br)c(F)c1NC(C1CC2CC2N1C(=O)CSC1CCCC1)=O C1(NC(C(CSC)O)=O)(CO)CCCN(C(=O)C(c2cccc(C)n2)(F)F)C1 CCCCC(C)C(C(=O)NCC(=C)C)N1CCc2cc(C(N)=O)ccc2C1 N1(C(Cc2onc(-c3cccc(OC)c3)n2)=O)CCN(C2CC2)C2(CCOC2)C1 C1(CCNC(CN(CC)CC)=O)CCCN(C(c2c(C)oc(C)c2C)=O)CC1 c1(OCCC)ccc(C(=O)NCCN(C(=O)Cc2csc(S)n2)CC)cc1N N1(C(N(C23CC(COc4ncc(C#N)cc4F)(C2)C3)C)=O)CCc2sc(Br)cc2C1 Cc1ccc(C(=O)NCC(=O)NCCN(C(=O)CC(C)N2CCCC2=O)C)s1 C12(CNC(=O)C(F)Cc3ccccc3)CCC(C1)N(C(=O)COCCF)C2 N1(C(C2(OCC)CCC2)=O)CCC2(CC1)CCN(C(=O)C(C#N)CC)C2 C1(NC(C=C(C)C(F)F)=O)CC2CC1N(C(=O)C(c1cnn(C)c1)O)C2 c1(CC(=O)NC2CC3CC(NC(c4cc(C)oc4C)=O)C2C3)cc2ccccc2s1 Cc1cc(C)c(C(N2CCC(N(C)C(C3CC(CCO)C3)=O)C2)=O)cc1C CCC(CC)C(F)C(=O)N1CC(CNC(C2CC(C)(C)C2)=O)C2(CC2)C1 N1(CC(N2CC(C(C(=O)NCc3cnc(CC)s3)O)C2)=O)CCOCC1=O C1(C(=O)NC(C(C)C)(C)CO)CN(C(C2CCC(C(N)=O)C2)=O)CC1(F)F C1(C(=O)Nc2nc(C)c(C)s2)C2CCC(C2)C1NC(c1cnnc(O)c1)=O CCCC(C(=O)NCC(C)CNC(c1cc(Cl)no1)=O)c1cc[nH]n1 c1(SCC(=O)NCCC(C)(C)NC(CCC=C=C)=O)cc(=O)n2ccsc2n1 C1(CNC(C(F)=CC)=O)CC(F)CN1C(=O)C(C)Cc1ccccc1Cl C(C)(C(=O)NCCC1(O)CN(C(=O)CCCSC)C1)(C1(C)CC1)OC C(=O)(C(O)CC[S+](C)C)NCC1(C)CCN(C(c2nnc(C(C)C)s2)=O)C1 N1(C(c2scc(Cl)c2Cl)C(=O)NC(C)C)CCN(C)CC1CCO c1(C(C(=O)NC2(CN(C(C3CCC4CC34)=O)C3CC3)CC2)(F)F)ccc(Cl)cc1 Cc1cccc(O)c1C(N1CC2CN(Cc3cccnc3)C2C1)=O CCCC(C)(C)C(=O)NCC(O)CCNC(C1CC(C(F)(F)F)(OC)C1)=O c1(C(=O)NC(C)(C)CCNC(C2CC23CC3(F)F)=O)nccc2cccnc12 C(=O)(CC(C)C(=O)N(C(C)(C(=O)NC1CC(C)OC1=O)C1CC1)C)OC N1(C(CCNC(=O)OC)=O)C2CCC1C(F)C(NC(=O)CC(F)(F)C(F)F)C2 c1(CN(C(c2cc(C(C)C)on2)C(=O)NC2COC2)CCC)ccccc1F N1(C(C)C(=O)N(C2CC=CCC2)C)CCN(C)CC1 CS(=O)(=O)c1ccnc(NCC2CCCCN2C(=O)CC2NC(=O)NC2=O)n1 Cn1cc(C(N2CCC(NC(=O)C=CSc3nc[nH]n3)C2)=O)cn1 c1(OC)cc(C#N)ccc1OCCC(=O)NC1CN(CC(O)CO)C1 C1(C(=O)NC(CSCC)C(=O)NC(C)C(C)F)OCCC1(C)C C1(C)(CNC(C(CCC)N(C)C)=O)CCCN(C(=O)Cc2cc(C)cs2)C1 CC(C)CCCC(=O)N1CCCCC1C1(C(=O)N(CCCO)CCO)CC1 C1(C(N(CCOC)CCNC(=O)CC2(C)CC2(Cl)Cl)=O)C2CCC1CC2 C1(C(=O)NCCNC(C2(NC(=O)OC)CCCCC2)=O)OCCOC1(C)C c1(C(N2CC(C)(C(=O)NC(CCC)c3ccco3)C2)=O)[nH]cc(C)c1C Cc1cc(C=CC(=O)NCC2CCN2C(=O)C(c2cnn(C)c2)C)ccc1F c1(C(N2CC(NC(Cc3n(C)ncc3Br)=O)C2)=O)cc2ccccc2cn1 NS(=O)(=O)CCCC(=O)N1CC(O)C(O)C1CNC(C1CC2CC2C1)=O c1(C(N(C2CN(C(c3cc(Br)cc(Br)c3)=O)C2)C)=O)noc2c1CCCCC2 C1(C(N2CCCC(OCCNC(C3CN(C)C(=O)N3)=O)C2)=O)(OCC)CCOCC1 c1(C(=O)NC2CC(O)(CNC(C3(CC)CCCC3)=O)C2)ccc(S(N)(=O)=O)nc1 N1(C(CNC(=O)NC)=O)CCC2(CC1)CC2(CO)CNC(c1ncccc1C)=O C1(C(=O)NCCC(C)NC(c2ccc(C(C)C)o2)=O)COC(C)(C)O1 C#CCCCCCCC[N+](C(=O)C=CC1CCCN1C(c1ccc(C)nc1O)=O)([O-])NC c1(C(=O)NC2CC(CCOCC)C2)cnc(N)cn1.C12(CCCC1)C(=O)N2 C1(CNC(C(C)OCCOCCOC)=O)(OCC)CCCN(C(=O)C(N)=O)C1 C1(C(=O)NCC2(C#N)CCC2)(COC)CN(C(c2ccc(C)o2)=O)C1 CCC(C)(C)CCCC(=O)Nc1cc([N+](=O)[O-])ccc1F.N(CCOC)(CCO)CC N1(C(C2C(C)(C)CO2)=O)CCC2(CCCN(C(c3n[nH]c(C4CC4)c3Cl)=O)C2)C1 c1(OC)ccc2c(c1)CC(C(=O)N(CCCNC(=O)Cc1cccc(O)c1)C)O2 Cc1ccc2scc(C(N3CCC(C)C(NC(=O)Cc4cscn4)C3C)=O)c2c1 c1(CN(C)CC2CCN(C(=O)C(=O)NCCCO)C2)ccc(Cl)c(Cl)c1 Cc1cc(F)cc(C)c1C(=O)NCC#CCNC(C1CC(C(F)(F)F)C1)=O C1(C(=O)NCCc2cc(C)sc2)CC2CCC(C1)N2C(=O)C(N1CCNC1=O)C C#CC1CN(C(=O)CC2C(=O)N(C)N=C2C)CCN1C(c1cc(C)nc(OC)n1)=O CC1CCCC=C1C(=O)NCCCCCNC(=O)Cn1ccc([N+](=O)[O-])n1 Cc1ccc(C#N)cc1S(=O)(=O)N1CCC2C(CCN2C(c2cc(C)[nH]n2)=O)C1 C12(C(=O)NC3CCC(NC(C(CC)CC(F)F)=O)C3)CC3CC(C1)CC(O)(C3)C2 c1(CC)nnc2ccc(=NC(CN(CCCC(=O)OCCO)C)C(C)C)[nH]n12 C1(CNC(C2OCCN(C(C(C#C)(C)C)=O)C2)=O)CCC2(CCC2)O1 C#CC1(O)CC(C(=O)NC2C=CC(C(=O)NC(C)C(C3CCCCC3)OC)C2)C1 CCCCC(C)(F)C(=O)NCCOC1CCN(C(c2cncc(F)c2Cl)=O)C1 C1(C(N2C(CCC(=O)NC3CCC(CC)O3)CCCC2)=O)CN2CCN1CC2 S(=O)(=O)(c1ccc2[nH]c(=NCC(C)N(C)CC)sc2c1)NCC(CC)CO N1(C(c2ccc(C(=O)O)o2)=O)CCOC(C(=O)NOCC2CCCC2)CC1 C1(C(N2C(CC)CN(C(C3CCN(C)C3=O)=O)CC2)=O)CCc2ccnn2C1 c1(C(=O)NC2C(NC(CC3(OCC)CCC3)=O)COC2)ccc(CC)c(F)c1 CCC(CCC(=O)N1CC(F)(C(=O)NCC(C2CC2)C2CC2)C1)OC CCC(C)C(C(=O)N1CC(C(C)OC)(NC(=O)C=CC(C)(C)C)C1)OC C#CC1(NC(c2coc(CNC(c3n[nH]c4c3COC4)=O)c2)=O)CCC(C)(C)C1 c1(CC(N2C(C(=O)NC(C)CCF)C=CC2)=O)ccc(O)cn1 C1(NC(=O)C=CCF)CC2CC1N(C(c1csc(-c3cnc[nH]3)n1)=O)C2 c1(CN(C)C)noc(CN(C)C(C2CCN(C3CNC3)C2)=O)n1 C1(NC(C2(CC)CCC2)=O)COCCN(C(=O)CCS(N)(=O)=O)C1 n1(CCC(=O)NCC2(F)CC(NC(C3(C#C)CC3)=O)C2)nc(C)c([N+](=O)[O-])c1C N1(CCC(N2CCN(c3ccc(Cl)cc3)CC2)=O)CCC(F)C(O)C1 C1(NC(c2ccc(CN=[N+]=[N-])s2)=O)C2CN(C(c3cccs3)=O)CC12 Cc1ncc(C(=O)N(CCCNC(=O)Cc2ccc(C(N)=O)nc2)CCO)n1C c1(NC(c2ccnc(F)c2)c2n(CCC)nnn2)ccc2c(c1)CN(C)C2=O CC(CCCNC(=O)CC1CC1(Cl)Cl)NC(C1(O)CCOC1)=O Cc1ncccc1CC(=O)NCC1C2CN(C(c3ccc(C4CC4)cc3)=O)CC12 c1(C(=O)NCC2(CCNC(C34CCC(C3)C4)=O)CC2)coc2c1COC2 c1(C(=O)NCC(C)NC(C(c2cccc(C)c2F)O)=O)cc2n(c1)CCOC2 c1(SC)cc(C(=O)N(C(C)CNC(=O)C=Cc2ccc(C)s2)C)cc(Cl)c1 n1(CCC(=O)NCC2(OC)CN(C(c3cc(C)c(C)o3)=O)C2)cc[nH]c(=O)c1=O c1(OC)cc(CO)ccc1C(=O)NC1CCN(C(=O)Cc2cccnc2)C(C)C1 C(=O)(CCCCCC(C)O)NCCCN(C(C(CC)c1cccnc1)=O)CC c1(NC(C2CN(Cc3ncc[nH]3)CCC2O)=O)ncc(I)cc1[N+](=O)[O-] C(=O)(CC(C)C(C)(C)C)N1C(CC)C(NC(=O)CCN(C)CCO)CCC1 C(=O)(C1=C(C)CCCC1(C)C)NCC(CC=C)NC(=O)C=C1CCOCC1 c1(CSC)cc(C(N2CC3(C2)CN(C(C2(C)CCC2)=O)C3)=O)ccc1F N1(C(=O)Nc2c(C)nn(-c3ccccc3)n2)CCc2cc(Br)cc(F)c21 c1(NC(C2(CSC)CCC2)=O)cc2[nH]ccc2cc1C#N CCCC(C(=O)N1CCCC1C1(O)CN(C(c2ncn(C)c2C)=O)C1)OCC N1(C(C(C)O)=O)C(CNC(c2ccc3c[nH]nc3c2)=O)CC2COCC12 Cc1cnc(C(N2CC(CNC(=O)CCn3cc(C)cn3)C2)=O)c(F)c1 N1(CC(N2CCN(Cc3ccc(C)c(F)c3)CC2)=O)CC(=O)Nc2ccccc2C1 N1(C(C)=O)Cc2occ(C(N3CCOCC3C3CC3)=O)c2C1.c1cnn(C)c1C#N C(=O)(C(C)(C)C(N)=O)NCC(=O)NCCC(C)(F)F C=CCC(CNC(=O)CC1CC1c1ccccc1)NC(=O)C(C)=CC(C)(C)C O=C(C1Cc2ccccc21)N1C2COCC1CC(NC(C1(C(F)F)CC1)=O)C2 N1(C(c2c(C(C)(C)C)[nH]cn2)=O)CC(C2CC2C(N2CC(S(C)(=N)=O)C2)=O)C1 c1(C(N(CC(C)C(N2CC(F)(C#N)C2)=O)C)=O)ccccc1CO c1(CC(=O)N(CCCNC(C2(C(C)C)COC2)=O)C)csc(-c2ncccn2)n1 c1(C(=O)NC2(C)CCN(C(c3c(C)cnn3C)=O)CC2)cnc2c(c1)NCC2 C1(c2n(CCC(=O)OC)nnn2)(OC)CN(C(C)C(=O)N(C)C(C)C)CC1C C1(C(C)(C)C)C(=O)N2C3C(CCC3)(CC2)CN1.S(=O)(=O)(CC)N(CC(=O)NC)C C12(O)CCN(CC1)C2=O.C1(CC(=O)OC)(NC(C(C)OC)=O)CCCC1 C1(C(N2C(COC)(CNC(=O)COCCCN(C)C)CCC2)=O)CC2C(C1)C2(F)F CC(C)CCCC(C)C(=O)NC(C1(O)CCN(C(C2CCCC2(C)C)=O)CC1)C Cc1nc2ccc(C(N3CC(C)CN(C(=O)C4=CCC4)CC3C)=O)cc2nc1C N1(C(C)=O)CCOCC1C(=O)NC(Cc1ccccc1)CCNC(c1cccs1)=O c1(C(=O)NC(CC=C)CNC(c2cnn(CC(F)F)c2)=O)ccc2ncccn12 S(=O)(=O)(c1cccc(=NC(C)CCO)[nH]1)N1CCC(C)C(C(=O)OC(C)(C)C)C1 C1(C(=O)NCC(C)(C)NC(=O)CSc2nc[nH]n2)CCCCC1C1CC1 C(=O)(CCCS(N)(=O)=O)N1CCC(N(CCC)C(c2cc(F)cc(F)c2)=O)CC1 C12(C(N3C(C=C)CC3)=O)CC(CO)(CN1C(=O)C(CCC)OC)C2 N1(c2nc(C(F)(F)F)cc(C)n2)CC2C3CCC(C2C1)N(C(c1cnoc1C)=O)C3 N1(C(C(c2ccc(C)s2)C)=O)CCOC(CC(=O)NCc2cncn2C)C1 N1(C(c2c(CC)nnc(C)c2)=O)CC2CCC1C(CO)C2 C12(NC(c3nccc(COC)c3)=O)CCCC1N(C(=O)Cc1cccs1)CCC2 Cc1cc(F)cc(C)c1C(N1CC2(C1)SCCC2NC(C1(CCN(C)C)CC1)=O)=O C(CC1=CCN(C(C2CCC2OC)=O)CC1)NC(C1(OC)CCOCC1)=O N1(C(CC2CC(=C)C2)=O)CC(C2CN(C(c3cncc(F)c3)=O)C2)C1 C1(F)(C(N(C(C(C)SC)C)C)=O)CCN(C(=O)CC2CCC(=O)NC2)CC1 C1(=O)C(C)CC(=O)NCC2CN1CC2C.c1(CCC(=O)OC)nncn1C C1(C(N2CC(NC(=O)Cc3cncn3C3CC3)(CO)C2)=O)OCC2CCCC12 C(=O)(C(=O)CC(C)C)NC(C1CCCC1)C(=O)NCCCc1cc(C)no1 N1(C(c2cc(CC)nn2C)=O)C(CNC(c2sc(C)nc2C)=O)CC2CCCC12 C(c1ccc(C(N)=O)cc1)=CC(=O)NC1CC(CCNC(c2nc(C)sc2)=O)C1 N1(C(C(CCC)F)=O)CCC(C)C(CC(=O)Nc2cn(C)nc2C2CC2)C1 N1(C(C(C)NC(C)=O)=O)CCCC(O)(CN(C(=O)CCc2ccncc2)C)C1 c1(OC)cc(CCC(C)NC2CCCC(n3cnnc3)C2)cc(F)c1 n1(CC)nc(C)c(C(N2CCCC2CN(C)C(c2ccc(F)cc2F)=O)=O)c1Cl C#CCC(C)(C(=O)NCc1nc(C)sc1C)NC(=O)C(O)C(F)(F)F C=CC(CCC)CC(=O)NCC1(OC)CCN(C(c2c(C)nn(CC)c2Cl)=O)C1 Cc1cc(C(=O)NCCCCCCNC(C2(C#N)CC2C)=O)c(Br)cc1F C1(NC(=O)C2=CCCC2)CS(=O)(=O)CC1NC(=O)CN1CCCCC1 Cc1cccc2[nH]c(C(N3CCN(C(c4ccc(F)cc4N)=O)C4CC34)=O)cc12 CC(O)CCCNC(c1coc(CNC(C2(C(F)(F)F)CC2)=O)n1)=O C1(NC(C(C)(C2CC2)OC)=O)CCC2CN(C(c3ncc(Cl)s3)=O)CC2C1 c1(C(=O)NCC2C(CNC(C3CNC(=O)N3)=O)C2)cnc2n1CCOC2 C1(C(=O)NCC(C(C)C)NC(C2(C)COC2)=O)CCc2cnnn2C1 c1(C(=O)NC2CC(NC(c3ccc4c(n3)CCC4)=O)C2)ccc(F)c2occc12 c1(C(C(=O)N(CC(C)NC(c2c(CC)scc2)=O)C)(C)C)nc2ccccc2s1 c1(C(CCC(=O)N(C(CCNC(C(C(C)C)O)=O)C)C)=O)ccc2c(c1)CCC2 C1(NC(=O)Cc2ccsc2)CN(C(c2occ3c2CCCC3)=O)CC(F)(F)C1 N1(C(=O)Cc2cccs2)CC2CN(C(c3cc4scnc4[nH]3)=O)CCC2(CO)C1 CC1CCOCC1C(N1CCCC1C=CC(=O)NC1CCCC1(C)C)=O Cc1cccc2c1CCOC2C(=O)N(CCCN(C)C)CCNC(=O)CCCF C1(C(=O)NCC2(Nc3cc(OC)ncn3)CCOCC2)CCN(C)C(=O)C1 Cc1ccc(CC(C(=O)N2CCN(C(=O)C(N)=O)CC2C)C(C)C)cc1F C(=O)(CC1=NN(C)C(=O)C1)NC1CC(CCNC(C2C(C(=C)C)OCC2)=O)C1 c1(C(=O)Nc2cc(OC(C)C)n[nH]2)ccc2ncc(-c3cc(O)ccc3F)n2c1 C1(CNC(C23CC(NC(CC(CC)SC)=O)(C2)C3)=O)COCC(=O)N1C c1(C(=O)NCCn2cc(CCC(=O)O)nn2)cc(F)c(F)cc1Cl N1(C(Cn2c(C)cc(C)n2)=O)CC(C)CCC1CNC(C1(CO)CCOCC1)=O c1(C(=O)NC(C2CCN(C(C3(C)CCOC3)=O)C2)C)cc(N)cc([N+](=O)[O-])c1 N1(C(CC2OCCOC2(C)C)=O)C2CCC1CC2.CNC(=O)OC(C)(C)C N1(C(C=CC(CC)C)=O)CCOC2(C1)CN(C(c1cc3ncccc3s1)=O)C2 c1(CNC(=O)CCc2cnn(C)c2)cc(C(N2CCC(C(C)(C)OC)C2)=O)on1 c1(-c2nnc(N3CCSC(C)C3C)n2C)nc2cc(Br)ccc2s1 CNS(=O)(=O)NCC(=O)N(C(C)C)CC1CC1NC(=O)CCCOc1cccnc1 N1(C(CS(CCOC)(=O)=O)=O)CCC(C2(NC(=O)CNC(C3CCC3)=O)CC2)C1 C(CCN=C(NCc1cncnc1)NC1CCC(c2ccccc2)C1)SC CC1OC(C)CC1CC(=O)NCCOCCN(C)C(C1(CO)CC(F)(F)C1)=O N(C1CCCn2nc(C(C)C)nc21)C(c1cc(C)ncc1)=O CCC(CCCC(=O)N(C1CCN(C)CC1C)C)NC(C1(n2cccn2)CC1)=O C(CNC(=O)CN(C1CC1(F)F)C)(C(C)(C)C)NC(CN1CCN(CC)CC1)=O c1(C(N2C(CNC(CC(CCC)CC)=O)CC2)=O)cc(OC)c2c(c1)OCO2 C1(NC(Cc2c(C)nc(Cl)cc2)=O)CCC2CN(C(C3CCOC3)=O)CC2C1 C(=O)(C1=CS(=O)CCC1)N1CC(=CCNC(=O)OC(C)(C)C)C1 N1(C(c2ccc(CNC(=N)N)cc2)=O)CCOC2(C1)CN(C(C1CCC1)=O)C2 c1(OCC(=O)NCC2C(C)(C)CN(C(=O)C3=CCC3)C2)cccc2ccccc12 C(CC(=O)NC1(c2nc[nH]n2)CC1)(C(F)(F)F)NC(C(CC)(C)NC(C)=O)=O C1(NC(CC2CC(OCC)C2)=O)CCN(C(c2cccc(N)c2F)=O)CC1O C(=O)(CC(C)(C)C)NC1CCN(C(C(C)NC(=O)C=CBr)=O)C1 CCCCC(C(=O)NCCC(O)C(C)C)NC(=O)CN1CCCCC1C c1(C(N2C(C(C)NC(c3c(C)cno3)=O)CCC2)=O)ccc(Cl)cc1F N1(C(CC(=O)OCC)=O)CC2CCCN(C(C3CC(F)(F)C3(F)F)=O)C2C1 c1(CNC(C2(C)CC(C)OCC2)=O)nc2c(s1)CN(C(=O)C(C)(F)F)CC2 n1(CC#C)c(C(N2CCN(C(=O)COC)CC2CCO)=O)cc2ccccc12 CC(C)(F)CCC(=O)NC12CCOC(CNC(C3CS(=O)(=O)CCO3)=O)(C1)C2 CC(CC(=O)NCC=CCNC(=O)COCC(F)F)n1ccnc1 CC1=C(C(=O)N2CCN(c3ncnc(Cl)c3CO)CC2)C(C)(C)CCC1 Cc1nn(C(C)C)cc1C(=O)NCCN(C(C1(O)CC1(C)C)=O)C1CC1 C1(C(N(C(CC)COC)C)=O)C(C)OCCN1C(=O)C(C)SC(C)C N1(C(c2ccc(SC(C)C)cc2)=O)CC(NC(C2CCC(=O)C2)=O)CC12CCC2 C1(C(N2C(C(=O)OC)C=CC2)=O)CCN(C(C2CC=CC2)=O)C12CCC2 C12CCC1CC2.C(=O)(CC(C)OC)N(CC(C)NC(CCOCC#C)=O)C C1(C(=O)O)(NC2C(OCC)C2Cn2nc(C)cc2C)CCN(C)C1 c1(C(=O)NCCC(C)NC(C=CCOC)=O)c2c(nn1-c1ccccc1)CCCC2 n1(CC(=O)N(C(C)CN(C(=O)CCc2cnc[nH]2)C)C)cc([N+](=O)[O-])cn1 C1(C(N2CCC(O)(Cc3cn(CCC=C)nn3)C2)=O)CC12CCOC(C)C2 N1(C(C(CC=C)(C)C)=O)CCCC2(C1)CN(C(c1ccc(C)c(F)c1F)=O)C2 C(=O)(CCCCC(C)=O)NCC1CCC(N(C(c2c(C)cnn2C)=O)CC)O1 C1(NC(CCSCCCC)=O)CCCC12CN(C(c1cc[nH]c3nccc1-3)=O)C2 C(CN=c1nc2scnc2c(N2CC=CCC2)[nH]1)OCC(=O)N(C(C)(C)C)C1CC1 Cn1nnc2c1CCN(c1nc(N3CCS(=O)C(C)(C)C3)c3c(n1)CSC3)C2 Cc1ccc(CCC(=O)NC2C3CN(C(C4(C)C=CCCC4)=O)CC23)cc1F N1(C(N)=O)CCC(C(N2CCCC(N(CCO)Cc3nccnc3N)C2)=O)CC1 c1(CC)cc(C(=O)NC2CC(NC(C3CC34CCCC4)=O)C2)nn1C c1(C(N(C(CNC(CCC)=O)C)C2CC2)=O)ccc(Oc2ccccc2)cn1 C(=O)(CC(CC1CC1)NC(=O)CNC(N)=O)N(CCCCO)C C12(C(=O)NCCN(C(c3cn(C)[nH]c3=N)=O)C3CC3)CCN(CC1)CC2 C(C)(CCC(=O)N1CC(C)CC1C(N1CCC(C)(C(N)=O)C1)=O)OCC c1(CC(N2CC(NC(=O)C(O)C3CCCC3)C2)=O)cc(C(F)(F)F)no1 N1(C(c2c(C)cccc2)=O)CCCN(C(c2coc(Br)c2)=O)C(CO)C1 CCCC(C(=O)OC)C(=O)N1CCC1CC(N1CCC(OC2CC2)C1)=O C12(CNC(C(C)(C3CCC3)NC(C3C(C)CCO3)=O)=O)CCC(CO1)C2 C1(CN(C(C2CC(OC)C2)=O)CC)CN(C(c2cc(CCOC)[nH]n2)=O)CCO1 C1(CC(C)C)CCN(C(=O)CNC(=O)CNC(c2ccc[nH]2)=O)C1 Cc1c(C(=O)NCC(C)N(C)C(c2sc(F)cc2Cl)=O)ccn1CCO CC(C)C(CCNC(C1CC1Cl)=O)NC(C12CC3CC1C2C3)=O C1(NC(CCC=C(C)C)=O)CCC2CN(C(=O)C(c3ccc(Cl)s3)C)CC2C1 C1(C(=O)NC2C(CC)COCC2)(C(=O)O)CCS(=O)(=O)CC1 C1(NC(C)=O)CN(C)CCC1N1CCN(C)CC1c1ccccc1 Cn1cc(C(N2C3CCC2C(CNC(C2COC(=O)N2)=O)C3)=O)ncc1=O CC(C)C(C)C(C)CC(=O)N(C)CCNC(=O)C(C)(C)CC1CC1 c1(NC(C(=O)NC2(NC(=O)OC(C)(C)C)CC(COC)C2)=O)cc(F)cc(Br)c1 C1(C)(C(=O)NCc2c(C(=O)NCC(C=C)OC)c[nH]n2)COC(=O)N1 N1(C(C2CCCS2)=O)CCCC(F)(C(N2C3CSCC2C3)=O)C1 C(=O)(CCCc1ccc(C(C)=O)s1)N(CCNC(C1C(C=C)C1)=O)CCC CN1CCC2CN(C(c3ccncc3Cl)C(=O)Nc3ccccc3)CC2C1 Cc1nc(=NC(=O)C2CCCC2NCc2ccc(F)c(F)c2Br)s[nH]1 CC1=C(C(=O)N2CC(CC(C)NC(c3ccc(C(C)(C)C)s3)=O)C2)CCS1(=O)=O c1(C(N2CCN(CCNC(=O)CCCC(F)F)CC2)=O)nccc2ccncc12 C12(NC(c3ncc(OC)cn3)=O)CCC(C1)N(C(c1cc(C3CCC3)[nH]n1)=O)C2 c1(C2(CN=c3cc(-c4c(F)ccc(F)c4)nc[nH]3)CC2)ccc2oc(O)nc2c1 N1(C(c2sc(Br)nc2C)C(=O)NCCCOC)CC(CO)C(C)(C)C1 c1(C(N2CC(NC(C(C(C)C)C)=O)C3(C2)CC3)=O)cc(F)cc2ccoc12 N1(C(CC)=O)CCCN(C(=O)CCCCCCSC)C(C)C1 N1(C(c2nncc(OC)c2)=O)C2CCC1(CNC(c1cc(C)on1)=O)CC2 C12(C(N3CCC(C)(NC(C(CCC)NC(N)=O)=O)C3)=O)COCC(C1)OC2 N1(CC(=O)NCC2N(C(C(CCC#C)O)=O)CCC2)C(=O)c2cccnc2C1=O C1(NC(CN(C)C(=O)OC(C)(C)C)=O)CCCC1NC(c1cnc(C(F)F)s1)=O c1(CC)ocnc1C(=O)NCC1(F)CC(NC(=O)C(C)OCCC(C)C)C1 c1(OC)ncc(C(=O)N(CCCN(C)C(C2CCCCC2F)=O)C)cc1C N1(C(c2n(C)c(C(F)(F)F)cc2)=O)CCC=C(C(=O)Nc2cc(F)c(F)c(F)c2)C1 N1(C(CC2CCC(=O)C2)=O)CCCC(CC(N2CCC(OC3CC3)CC2)=O)C1 CCC(CCCC(=O)NC1CCC(C)(C)CC1)NC(=O)C1=CCCCC1 C(=O)(C(C#N)(CC)CC)N1CC2CN(C(c3c(OCC)cc(Cl)s3)=O)C2C1 C1(NC(=O)CCc2ncc[nH]2)CN(C(c2ccc[nH]2)=O)CCC1c1ccccc1 C1(C(=O)NC(C=C)CO)(SC)CN(C(=O)CN2CC=CC2)C1 N1(C(C(COC)C)=O)CC(C)(C)CC1CC(=O)NCCC1CC(C)=NO1 C1(C(=O)OCC)CN(c2nccc(C#N)n2)CC(C)O1 c1(C(=O)NCCC(C)NC(c2nnc(O)nc2O)=O)ccc(C(F)F)c(F)c1 C1(CNC(CC=CC=C)=O)CCCC(NC(c2nncn2C(C)C)=O)C1 CCC(CC)C(C)C(=O)NCc1n[nH]cc1C(=O)NCCC1COCCO1 C12(CC)CN(C(c3cnc(C(C)C)nc3)=O)C(CNC(=O)CCOC(C)C)(C1)C2 CC(C)C(CO)C(=O)NCCCN(C(C1(C)CCCN(C)C1)=O)C(C)C CCCC(O)CC(=O)NC(CO)C(C)NC(c1cnn(CCN(C)C)c1)=O C1(CC(=O)N(C(C)CNC(=O)CC2CC(=O)NC2=O)C)C2CC3CC(C2)CC1C3 C(=O)(C1CCCc2n[nH]cc21)N1CCN(C(c2c(NC)scn2)=O)CC(O)C1 c1(C2N(C(=O)Cn3cnnc3O)CC2)cccc(F)c1.C1(C2CCCO2)C(=O)N1 C=C1CCC(C(N2CC(OC)CC2CNC(=O)CNC(=O)CC)=O)CC1 c1(C(N2CCC(CCNC(C=CC(C)(C)C)=O)C2)=O)ccc2nc(O)n(C)c2c1 c1(CC)ccc(NC(=O)CCC(C)NC(C2CCN(OC)CC2)=O)cc1C c1(C(=O)NC(C)CNC(C2CC2F)=O)cn(CCN(C)C)nn1 C=CC1CCN1C(=O)CN(C(=O)C(CC)OC)CC(C)C C1(C(N2CCCC(NC(CCCC#CC)=O)(CO)C2)=O)CCC2(CC1)CC2(F)F C1(C(N(C2CCCN(C(CC(=C)C)=O)C2)CC)=O)CCCCC1(C)C C1(C2CCN(C(=O)Cc3cc(C(F)(F)F)n[nH]3)C2)(NC(C(C=C=C)C)=O)CC1 C=CC(C)(C)CC(=O)NC(C)(C)C=CC(=O)NC1CCN(C)CC1C N1(C(C(=O)c2ccco2)=O)CCC2CCC(C1)N2C(C1CCCCCCN1)=O C1(CNC(=O)NC(c2cocn2)CC)CCc2n[nH]c(C)c2C1 N1(C(C2CCCOC2)=O)CC(CNc2cc(NCC3CC3)ncn2)OC2CCCC12 Cc1ccccc1C=NOCc1sc(C2CC2(F)F)nc1C C(=O)(CCCCC(F)(F)F)NCC1CCC(C)(C)CN1C(C1CC12CCC2)=O Cc1cccc2c1CCCC2Nc1nnc(C(=O)NCCCO)n1C(C)C C(=O)(C(F)(CNC(C1CC(=O)NC1(C)C)=O)C(C)C)NC(C(=O)NCC)CC c1(C(=O)NCCN(C(C(CCC)NC(N)=O)=O)C2CC2)c(N)cc(F)cc1Cl C1(NC(C2(C(F)F)CC(=C)C2)=O)CC2CC1N(C(=O)Cc1cc[nH]c1)C2 C1(N(C(CCSCCC)=O)CCC)CCN(C(C2CN(C3CCOC3)C2)=O)C1 N1(C(C2CCC(CC)N2)=O)CCC2(CCCN2S(=O)(=O)c2cc(Br)ccc2Cl)CC1 CC(C)C(C)CN(C(=O)C(=O)Nc1cnn(-c2ccccc2)c1)C N1(C(CCC2CC(OC)C2)=O)CC(NC(c2conc2C)=O)C2CCCC2C1 N1(C(CC=C)=O)CC2CC1CCN2C(c1cc(Cl)c(Br)cn1)=O C(CC(=O)NCC1(C)CCOCC1)(C(F)(F)F)NC(Cc1c(C)cnn1C)=O c1(C(N2CCC(C3N(C(C=CC=CC)=O)CCCC3)C2)=O)cc(F)c(Cl)cc1Cl N1(C(c2cc(CNC(=O)Cc3cn[nH]c3)[nH]n2)=O)C2CCCC1COC2 c1(C(N2CC(OCCNC(C(N3CCN(C)CC3)C)=O)C2)=O)c[nH]nc1[N+](=O)[O-] c1(SC)nccc(=NC(=O)CN2CCN(c3ccc(C(F)(F)F)cn3)CC2)[nH]1 Cc1cc(O)c(Cl)cc1C(=O)NC12CCN(C(c3c(Cl)cccc3Cl)=O)CC1C2 C1(C(=O)OC)CCC(C2CCCCC2)CN1C(C1(c2ccco2)CC1)=O C1(CC(=O)NCC(COCC)C)CN(C(=O)Cc2c(C)cnn2C)CCC1C N1(C(Cc2cc(CC)no2)=O)CCN(C(c2csc(C(F)(F)F)n2)=O)C2CCC12 N1(C(=O)CCCc2cccnc2)CCC2(CCN(c3ccc(-c4cn[nH]c4)s3)C2)C1 N1(C(C(C)Sc2ccccc2)=O)C2CN(CC3CCCC(C)C3)CC12 C#Cc1ccc(C(N2CCC(C(=O)NCC3C(C)(C)C3(F)F)CC2C)=O)nc1 C#CC1CCCCN1C(c1ccc(CNC(=O)C(O)C(C)C)nc1)=O Clc1cc(CN2CC(n3cnnc3-c3ccccc3)C2)on1 C(=O)(CP(C)(C)=O)NCC1(C(=O)NCCN(CC2=CCSC2)C)CCCO1 C1(NC(c2c(C)nco2)=O)CCCC12CN(c1nncs1)C2 C(=O)(CC(C)(O)c1ccccc1)NCC(CC)NC(=O)COCC1CCCCO1 c1(C(N(CCNC(Cc2nc(C)sc2)=O)C(C)C)=O)cc2cccnc2cc1F n1(CC)nc(C(=O)NCCC(C)NC(=O)C(C)CN2CCCCC2)ccc1=O CCCC(C(=O)N(C)CCC1CCN(C(=O)C(C)(O)C(C)C)CC1)S(N)(=O)=O C(CCN=c1[nH]c(=NCCC(OC)OC)[nH]c2c1CSC2)N1CCOCC(=C)C1 Cc1ccc(N2CCCCC2)c(CNc2c(SCC3CCC3)cccc2Cl)c1 c1(C(N(CC(CN(C(c2[nH]cc(CC)c2)=O)C)O)C)=O)cc(OC)c(C)o1 c1(OCC(N2C(CNC(CCOCC)=O)CCC2)=O)ccc(CO)cc1 CN1CCN(C(c2cccc(C#N)c2)C(=O)NCCC2(C)CC2)CC1(C)C C(=O)(CC(C)C(C)(C)C)N1CCC(OCCNC(c2nc(OCC)sn2)=O)C1 Cc1cccc(CCC(=O)NC(C)(CNC(=O)C(=O)N(C)C)C2CCC2)c1Cl c1(CC)nnc2n1CCCC2C(=O)NCC(C)CNC(c1ccc(OC)s1)=O C1(CN(C(C(CC)O)=O)C)CN(C(=O)CCC2OCCO2)CC12CC2 N1(C(CC(C)(C)SC)=O)CCC2(CC(NC(=O)C(C)(C)c3cc[nH]n3)CO2)C1 C=CC1(C(=O)NC2CC3CC2N(C(c2cc[nH]c2C2CCC2)=O)C3)CCCCC1 C1(NC(C(C#C)(C)C)=O)CC2CN(C(c3ccc4cncn4c3)=O)CC2C1 N1(C(c2nc(C)c(C)[nH]2)=O)CCC(O)(CNC(c2cc(Cl)cnc2O)=O)CC1 C#CC1CCCC(NC(=O)C#CCNC(=O)CC2(O)CCC2)C1 N1(C(C2OCCN(C)C2)=O)CCN(C(=O)CCCCCC#N)C2CCC12 C(C(C)NC(c1ccc(C(C)(C)C)s1)=O)(C(C)C)NC(C(C)=C1CCC1)=O CCC(C)CCC(=O)N1CCN(C(=O)C(CCSC)OC(C)=O)C(CF)C1.C(C)=O N#Cc1ccc(C(=O)NC2C3CN(C(c4coc(Cl)n4)=O)CC23)c(O)n1 Cc1cc(O)n2ncc(C(N3CCCC3CN(C(=O)Cc3cnsc3)C)=O)c2n1 C(C(C)C(=O)NOCC(=O)OCCN(C)C)NC(C1CCC(=C)CC1)=O C1(C(=O)NC2(CNC(C3CCC(C)S3)=O)CCCCC2)COCCN1C=O N1(C(C2N(C)C(=O)NC2)=O)CCC(C2CCN(C(=O)C(C)(C)CCC#N)CC2)C1 c1(C(=O)NC2(C3CN(C(Cc4ncc(C)s4)=O)C3)CC2)noc2c(F)cccc12 C1(NC(Cc2ccc(C)o2)=O)CN(C(=O)CSc2nnnn2C)C2(CCC2)C1 c1(C(=O)NC2CCC(CNC(c3nnn(CC)c3C)=O)C2)ccc(Br)cc1N c1(C(=O)NCCCN(C(CCOC)=O)CCO)ccc2n[nH]c(C)c2c1 C=CCC(F)(F)C(=O)N1CCSCC1c1nn[nH]n1 CCCCCS(=O)(=O)CC(=O)N1CCC(C(C)Nc2ccc(S(C)(=O)=O)cn2)C1 c1(CC)ccc(Cl)c(C(N2CC(NC(C3(CSC)CCC3)=O)C(O)C2)=O)c1 C12C3CCCC3N1C(=O)C2.CC1(C(=O)NCCOCCF)CCC(=O)C1 Cc1onc(Cl)c1C(=O)NCC(C)N(C(=O)COc1ccc(F)nc1)C C(CCC(=O)NC(C(=O)N(C1CC1)CC1CC=CCC1)C1(O)CCC1)N(C(C)C)C C1(CC(N2CCC(N(C(=O)Cc3ccn(C)c3)CC)C2)=O)CCCCC1(F)F C12(CS(C)(=O)=O)CC1CN(C(=O)Nc1cccc(SCCN3CCOC3=O)c1)C2 C(C(=O)NOCc1nc[nH]n1)=CCCN(C(=O)COCC1CC1)C C1(C(=O)NCC2CN(C(Cn3ncn(C)c3=O)=O)C2)CCCN2CCCC12 C=C(CNC(=O)CCc1ccccc1)CCNC(C1(C#N)CC1)=O c1(OC)ccc(C2(C(=O)NC(C)C(C3CCCCC3)N(C)C)CCCC2)c(C)c1 c1(OC)ccc(C(=O)CCC(=O)N(c2ccc(Cl)cc2)Cc2cccnc2)cc1F c1(C(=O)NC2(CCNC(CSC)=O)CCC2)cc2sccc2n1CSC1CC1 C1(CC)C(C(=O)N(CC(O)CN(C)C(c2cc(Br)n[nH]2)=O)C)CCN1C C(=O)(CC1OCc2cc(Cl)ccc21)NC1CN(C(CSCCCC)=O)C(CO)C1 c1(C(N(C(CNC(=O)C=CCO)C2CC2)C)=O)ccc2c(c1)C(=O)NCC2 C(N=c1[nH]c2c(c(=NCC3CC3Cl)[nH]1)CCCCCC2)c1cccc(CSC)c1 c12ccc(cc1)C(=O)N1CC(C1)CC(C)NC2=O.CCCS(=O)(=O)NC1(C)CC1 C1(CC(=O)N(C2CCCC2)CC#C)C2CCCC2N1C(C1CC(CC2CC2)C1)=O N1(C(CC(CC)CC)=O)CCC2CC(NC(=O)CCCCF)CCC2C1 C(CC1=CCCCC1)NC(C1C(NC(C(CCSC)O)=O)CC=CC1)=O Cc1cccc(C)c1C(=O)NC(C)CNC(c1cc(Br)n[nH]1)=O C1(CC)(OC2CC2)CCCN(C(=O)COCCC(=O)NCCOc2ccon2)C1 c1(C(C(=O)NC(C(C)NC(Cc2ccc(C)o2)=O)C)F)ccc(C(F)(F)F)cc1 C1(CNC(C(C)CO)=O)CCCC2CN(C(C3CCCC3)=O)CC12 CCCCCC(C(=O)N(C)CC1CN(C(=O)CCC(C)OCCOC)CCO1)C(C)C C12(CCNC(=O)CCCF)CCC1CN(C(c1ccc(Br)cc1O)=O)C2 C1(C(=O)NC(C2CCCC2)CNC(C2(SC)CCC2)=O)Cc2nccnc2C1 c1(-c2c(OCC)ccc(F)c2)nnc2ccc(N(CCCSC)C)nn12 c1(C(C(=O)NCC23C(CN(C(C(CCC)OCC)=O)C2)C3)=O)cc(F)ccc1C C1(CC(=O)NCCC2CC(NC(C3(Cl)CC3(F)F)=O)C2)CCc2nnnn2CC1 C1(CNC(=O)C=CCO)CCC2(CO1)CC(NC(c1csc(Cl)n1)=O)C2 c1(N(C(=O)C=CC2CCCC2)CC(N2CCCC(CCCO)C2)=O)ccc(O)cc1 C1(c2nnnn2C2CC2)(Nc2cncc(NC(C)=O)c2)CCN(C)C(C)C1 N1(C(C2C(CC(C)C)C2)=O)CCCCC(CNC(=O)Cc2cc3n(n2)CCO3)C1 CCC1C(=O)Nc2ccc([N+](=O)[O-])cc2-c2ccc(NC(C3CC3(C)C)=O)cc21 C(C(C(C)C(C)C)NC(C1(CC(F)F)CCC1)=O)NC(CCOC(C)=O)=O c1(C(N2CC=CC(NC(C3OCCN(CC)C3)=O)C2)=O)cc2ccc(C)cc2[nH]1 N1(C(C=C(C)c2ccsc2)=O)CCC(CNC(c2cc(Cl)n(C)n2)=O)C12CC2 C1(N2CCCC2=O)CC1C1CCCCC1.C12CC=CCN1C(=O)COC2=O CCCCCCCC(F)C(=O)NCc1cc2n(n1)CCN(C(C1CC13CC3)=O)C2 Cc1ccc(O)c(CC(N2CC(NC(C3(C)CCCCCC3)=O)CC2(C)C)=O)c1 Cc1cc(C(=O)N(C(C)CNC(=O)COCc2cc(C)no2)C)nc(O)n1 c1(OC)ccc(C(=O)NC(C2CCCCN2C(=O)CN2CCCC2)C)nc1 C123CC(CO1)N(C2)C(=O)CCCCCONC3=O.C=C(C)CNC(C)=O c1(NC2CC(CNC(c3c(C)nc(CCC)o3)=O)C2)cc2c(cn1)C(=O)CCC2 c1(SCC(N2CC3C(NC(C4ON=C(C)C4)=O)C(C3)C2)=O)ccccc1[N+](=O)[O-] C(=O)(C1=CSCCO1)N1CCC(O)(CNC(c2cccnc2N2CCCC2)=O)C1 C1(CC(=O)N(CCC(=O)N(CC(C)C#N)CC)CC)COCC(C)O1 C(=O)(CC(F)(F)Br)N1CCC(C(C)(C)NC(Cc2cc(C)ns2)=O)C1 c1(C(=O)NC2CCCN(C(C3(SC)CC3)=O)C2)ccc(-c2nnc(C)o2)c(F)c1 CC1CN(C(C2CC3C(C2)C3(F)F)=O)CCN1C(c1ccc(Cl)nc1)=O C1(C(=O)OC)C2C3CC4C1C1C2CC3C41.C12=NC=CC(=NCC3CN(CCO3)C1)N2 C(=O)(C(C)C(O)CC(C)C)N1CCC(CNC(C2C(CC)C2)=O)(CO)CC1 CC(C)CC(C)CC(=O)N1CC2(CCCC2)C1C(=O)NCC1CCCCO1 c1(C(=O)NCC(C)N(C)CC2CCC3CC3C2)ccc2sccc2c1 N1(C(C#CCNC(c2c(C)nns2)=O)=O)CC(C#N)(CCF)C1 C(=O)(CCCC(CC)NC(C1C2CCC(C2)C1C)=O)Nc1cn(CCC)nc1 N1(C(C(C(C)NC(c2c(C)non2)=O)C)=O)CC2OC(=O)N(C)C2C1 N1(C(c2c(CC)nccc2)=O)CC2(CC(CNC(=O)COC3CC=CC3)C2)C1 c1(C(=O)O)ccc(F)c(CN2CCCC2C(=O)NCC(O)C(F)(F)F)c1F Cn1ncc(C(F)(F)F)c1C(=O)NC1CCCCC1NC(C1CC1F)=O C1(NC(c2n(CC=C)nnn2)c2occc2Br)CCOC(c2cccc(Cl)c2)C1 CC1(C)OC(C)(C)C1(O)CNCc1csc(-c2ccccn2)n1 C(=O)(C1=NOC2(CCC2)C1)N1C(C)C(NC(=O)C(=O)NCC(F)F)CC1 C1(C2N(C(Cn3cc(NC(c4cc(OC)ns4)=O)nn3)C)CC2)CCCCCC1 CCCC(C)(O)CC(=O)N(CC(=O)NCC(N1CCCC1)=O)CC(C)C C(=O)(C(C)(C)CCCF)N1CCC(C(C(=O)NC(C)C(O)C(F)F)F)C1 N1(C(c2cn(CC=C)nc2)=O)CCN(C(=O)C(C)(C)C2(C)CC2(F)F)CC1CF C(=O)(C(C(C)(C)C)NC(=O)C(=O)C(C)(C)C)NC(CC(=O)NC(C)C)C N1(C(C2(C#N)C(C)(C)C2)=O)CC2(C1)CN(C(C1C3CC4C(C3=O)C14)=O)C2 C(N=c1[nH]cnc(Cl)c1COC)C1(CCNC(=O)COC(F)(F)F)CC1 c1(C(N(C2CCCN(C(=O)C(C)CO)C2)CC)=O)cc(C(F)(F)F)cc(F)c1 N1(C(c2c(C)cc(C(=O)OC)o2)=O)CCC2C(NC(=O)C=C3CCCC3)C2CC1 N1(C(=O)Nc2cc(C)ncn2)C2CCCC1CC(N)C2 C(=O)(CC(C)C(=O)OC)N(C1CCN(CCC(=O)OCc2ccccc2)CC1)CC c1(C(=O)NCC(C2CC2)NC(C2N(CC)CCC2)=O)ccc2nn[nH]c2c1O N1(C(C2CSCCN2C(=O)C=CC2CCCC2)=O)CC(CO)C2(COC2)C1 c1(C(=O)NC(C2CCCC2)CNC(C2(C)C(C)C2)=O)cc2n(n1)CCCO2 N1(CC(C2CCCCC2)C)CCC2(CC1)CC2NC(=O)CCl c1(CC(=O)NCC(CCNC(CCC=C)=O)=C)ccc2c(c1)CCC2 CN1C(=O)NCC1C(=O)NC1CC(CNC(=O)CC2(O)CCCCC2)C(O)C1 C1(CC(C)N(CC2=NOCC2)CCc2ccccc2)CCOCC1 N1(C(c2c(C)con2)=O)CC2CC(C1)CN(C(c1cc3ccnn3cn1)=O)C2 N1(C(c2cc(SC)oc2C)=O)CCC(C2CC2)(CNC(=O)C(C)(C)SC)C1 N1(C(COC(C)=O)=O)CCC2(CCN(C(c3n[nH]c(C(C)C)c3Br)=O)C2)C1 N1(C(c2cc(CNC(C(c3cnccn3)C)=O)[nH]n2)=O)CC2OCC(C)C2C1 C1(NC(Cn2ncc(C)c2)=O)CC12CC(NC(C1CCC1(F)F)=O)C2 S(=O)(=O)(c1ccc(C)c(C(=O)OC)c1)N(CC)Cc1sc2ccccc2c1Cl N1(C(CC=CCC)=O)CCOC(CN(C)C(C2(C#N)CCOC2)=O)C1 C12(C(=O)NC3CCC(N(C(=O)CS(=O)(=O)NCC4CC4)C)CC3)COCC(C1)OC2 c1(C(=O)NCC(C)NC(=O)C(c2ncc(Cl)n2C)(F)F)cc2cc(Cl)ccc2o1 N1(C(CNC(CC2C(NC(=O)OC(C)(C)C)CCC2)=O)=O)CCCC(N=[N+]=[N-])C1 c1(C(N(CC(CC)NC(=O)CN2CCOCC2)CC)=O)cc2n(n1)CC(O)CO2 C1(CC(=O)NCCN(C(=O)CCn2cncn2)CCOC=O)CCCC1CCC c1(OC)cc(N2CC(Nc3cnccn3)C(C)C2)nc(COC(C2CCC2)=O)n1 c1(C(N(CCCNC(CC(C)OC)=O)C(C)C)=O)cc(C2CC2)cc(F)c1 C12(C(=O)NC(CC)CNC(=O)Cc3cncc(C)c3)CCCC1NC(=O)C2 C1(C(C2(C)CCC2)NCCCCNC(C=CC)=O)CCC(=O)N(CC(F)(F)F)C1 c1(CCC)n[nH]cc1C(=O)NCC1CC1.C1C(=O)NCCCO1 CCCC(C)CC(=O)NC1(C)CCN(C(=O)C=Cc2cccc(Cl)c2)C1 N1(C(C(C(C)O)NC(c2cnc(O)c(F)c2)=O)=O)Cc2ncsc2C1 N1(C(CC=C)=O)CC(C(=O)OC)CC1(C)CC.c12ccnc(c1)NC(=O)C2(F)F c1(CNC(=O)C=C2CCCCC2)ccc(CCNC(C2CC23CCOC3)=O)cc1 C=CCCCC(C(=O)NCc1ccc(C#N)cc1)NC(=O)CCc1ccn(C)c1 N1(C(C(COC)O)=O)CC2CN(C(c3ccnc(OCCO)c3)=O)CC2C1 C1(F)(C(N2CC3C(CNC(c4ccn(C)n4)=O)C3C2)=O)C(C)(C)C1(C)C C1(NC(c2cncc(OC)c2)=O)CN(C(C2CC3CC3C2)=O)CCC1(C)C c1(-c2cc(-c3n(CC)nc(Cc4cnn(C)c4)n3)n[nH]2)c(F)cccc1F.C1(C)CC1 c1(C(=O)NC2C(C(C)C)CN(C(c3ccc[nH]3)=O)CC2)noc2cc(F)ccc12 C1(CNC(CCOC)=O)(NC(=O)CCc2cc[nH]n2)CCCCC1C N12CCN(CC1=O)CC2.CC1(C)C(NC(C2(N)CCC2)=O)CC1O Cc1cc(C2CC2)nc(N2CC(O)CC2CNC(c2ccc(C#N)cn2)=O)n1 c1(OC)ccc(-c2ccc(NC(=O)CCOC3CCNC3)c(F)c2)cc1F c1(C(=O)NC(C(C)C)C(C)NC(c2cn(C)ccc2=O)=O)ccc(O)c(CO)c1 C1(NC(c2c(C(C)(C)C)ccs2)=O)CCOCC1NC(c1ccc(CO)cn1)=O c1(OC)ncc(C)cc1C(N1CC2(NC(=O)C(C)SC(F)(F)F)CC1C2)=O CC1OC(C)C(C)N(C(=O)NC(c2nccn2C)C)C1C c1(C(=O)NC2CN(C(C(CCSC)O)=O)CC2(C)C)cnc2[nH]nnc2c1 c1(C(N2CCC(CCCNC(CC3C(C)C3)=O)CC2)=O)ccnc(Cl)c1N c1(Cn2c(N(C3CCSC3)C)nnc2C2CCOC2)ccc(S(N)(=O)=O)cc1 c1(OC)ccnc(O)c1C(N1CC(CNC(c2nccc(C)n2)=O)C(O)C1)=O C1(N(C(=O)Cn2[nH]cnc2=N)C)CCCN(C(=O)CCOc2cccnc2)C1 N1(C(c2c(C)nns2)=O)CCC(C)(CNC(c2cn(CC(N)=O)nn2)=O)C1 c1(C(=O)NCC(C2CCCC2)NC(=O)C(C2CCOCC2)=O)ccc(CO)nc1 c1(C(N(CC(N2CC(CO)CC2CO)=O)CC)=O)cc2occc2[nH]1 N1(C(C2CCCC23CC3)=O)CC2CCCC(C1)N2C(c1c(F)ccc(F)c1O)=O C1(CNC(C2C(CC)CCC2)=O)CCCC12CCN(C(C1C=C1C)=O)CC2 c1(N2C(C)CC(NC(c3ccc(SCC)cc3)=O)C2)ncc(F)c(COC)n1 c1(N(C)C)ccc2c(c1)CN(Cc1ccc(-c3ccc(N)cc3Br)s1)CC2 Cc1nnc2n1CC(C(N1CC(=C(F)CNCc3ccc(CO)o3)C1)=O)C2 N1(C(C(C)n2cncn2)=O)CCN(C(=O)CC2CC(F)(F)C2)C(C2CCC2)C1 C1(CC(=O)NCC(C)(CO)OC)CCN(C(=O)C2=CCCS2)CC1 c1(C(c2nnnn2CCCF)NC(c2ccc(C)o2)CC)ccc(OC)nc1 c1(C(N(CCOC)CCNC(c2ccncn2)=O)=O)cc2ccc(OC)nc2[nH]1 c1(COC)c[nH]nc1C(N1CCCC1C(=O)NC1CC(N2CCCC2)C1)=O C1(=CC(=O)Nc2c(C)[nH]cc2)CCN(Cc2ccc(C3(O)COC3)cc2)CC1 c1(CC)cc(C(N2CCCCC2c2cn(Cc3ncon3)nn2)=O)c(C)o1 CC1COC2(C1)CN(C(C13COC(C1)C(NC(c1ccon1)=O)C3)=O)C2 C1(CC(=O)NC(CNC(c2cnc(OC)s2)=O)C)CSc2ccccc2O1 CC1(c2cn(CC3CCCO3)nn2)CCN(C(C2CC3CC(O)C2C3)=O)CC1 NS(=O)(=O)C1CCC(C(=O)NCC=CCNC(c2ccc([N+](=O)[O-])cc2O)=O)CC1 CCCCC(C(=O)NCc1cc(C)no1)NC(=O)CN(C)C1CC1 N1(C(C=CC)=O)CC2ON=C(CNC(=O)Cc3c(Br)cnn3C)C2C1 c1(CC)cc(C(N2CC(CNC(=O)C=CBr)C2)=O)ccc1F c1(CC)cc(C(=O)OC2COCC2OCC(N2CC(C3CCOCC3)C2)=O)no1 c1(C(N(C(CCOc2c(N)cccc2)=O)CCC)C)nc2c(s1)CCCC2.OC C1(C(CN(C)Cc2ccc(O)cn2)F)CCN(C(=O)CC2CC3CCC2C3)CC1 C(=O)(C(C)CCCC(C)C)NC1CC2CN(C(c3ncc(C)nc3)=O)C(C1)C2 CC1CN(C(c2c(O)cccc2Cl)=O)CCC1CNC(C1CCCC(F)C1)=O N1(C(CC(COC)(C)O)=O)CC(NC(c2c(C)nsc2C)=O)C(C2CC2)C1 C(=O)(C1=CCCCO1)N1CCCC(C(C)(O)CNC(c2ncsc2CC2CC2)=O)C1 C1(CC(=O)NCC(N(OC)C)=O)CCN(C(=O)C(=O)C(C)C)C1(C)C c1(C23C(C(N4CCC(N(C(CCC)=O)C)C4)=O)(CCC2)C3)ccc2occc2c1 c1(C(=O)NCC(C)OCCO)n[nH]c2c1CN(C(=O)C1=CCCCC1)C2 Cc1cc(P(C)(C)=O)oc1C(=O)NCC(F)CNC(=O)CCC1CCC(=O)N1 Cc1cncc(C)c1C(=O)NC(Cc1ccco1)C(=O)NCC1CC12CC2(F)F C1(CC(N2CC(C)(OCCCN(C(=O)COC)CC)C2)=O)CCCC(C)O1 C1(C(=O)NCCCc2c(C)noc2)(CNC(=O)CCC2CCCCO2)CC12CCC2 c1(OC)cccc(C(C)C(=O)NC(C)C(C)NC(=O)CSC)c1 C(=O)(C1CCCc2nn[nH]c21)NC1C(C)N(C(=O)COCCN(C)C)CCC1 N1(C(c2c(CC)cc(Cl)cc2)=O)CC2(CC(NC(=O)C(C)(Cl)Cl)CO2)C1 N(C(=NCCC1CC1)NCc1cnc(Br)n1C)CC1CCCC(C)C1 C1(C(=O)NCC(C)NC(c2cocn2)=O)CCCCC1P(C)(C)=O C(CCCCC(=O)N1CC(O)CC1(C)C)N(C(C1C(CC)CCO1)=O)C c1(OC)ccc(C(C)C(=O)NC2(C)CCN(Cc3cccc(Br)n3)C2)c(C)c1 C(=O)(C(C)(C)CO)N1CC(N(C)C(C2CCC(C(F)(F)F)O2)=O)C1 N1(C(COCCC)=O)CC(O)C(O)C1CNC(=O)CC1OC(C)(C)OC1=O c1(C(N2CCC(C(=O)Nc3cccc(O)n3)C(O)C2)=O)cc(Cl)ccc1[N+](=O)[O-] S(=O)(=O)(c1ccccc1S(=O)(=O)NC)NCCc1n(CC)nnc1C C(CC(C)C)(C(=O)NC1CCCCC1)ONC(c1ccc(NC)cn1)=O C1(C(=O)NCC2CN(C(C)C)C2)(NC(C(C)C2(O)CCC2)=O)CCSC1 C1(C(=O)OCCC#CC)Cc2ccsc2CN1C(=O)NC(C)(C)C C1(NC(CSCCC)=O)CCN(C(=O)CC23CCCC2C3)C12CCC2 c1(C(=O)NCC(CNC(CNC(=O)OCC=C)=O)F)c(F)cc(F)cc1Cl c1(CCC(=O)NCC(C)N(C2CCN(CCC)C2)CC)ccc(O)nc1 c1(C2(C(=O)NC3CC(CNC(=O)Cn4cnnn4)C3)CC2)ccc(Cl)c(F)c1 C1(CNC(C(C)(C)F)=O)C(C2CC2)CCN1C(=O)CCC(=O)Nc1nnc(C)s1 N1(C(C(C(C)C)NC(N)=O)=O)CCCOC(CNC(C2COCCO2)=O)C1 CC1CCCC=C1C(=O)N1CC(C(O)C(=O)NCc2nnnn2C2CC2)C1 CCC(C)C(O)CC(=O)NC(C(=O)NCCC(F)(F)CO)c1ccoc1 C(=O)(N1CC(C)(O)CO1)C1(C)CC(NC(CCCN(C(C)=O)C)=O)C1 C1(CC)C(=O)NCCN1C(c1n[nH]c(Cn2cc(C(C)(C)OC)nn2)c1Br)=O C=CCC(C)C(=O)NC(C)C(C1CCCCC1)NC(=O)CCCNC(=O)C1CC1 N1(C(c2ccc(C(C)=O)nn2)=O)CCC2(CCCC2NC(c2ccccn2)=O)C1 N1(C(C2(NS(C)(=O)=O)CC2)=O)CCN(C(C2(C)C=CCC2)=O)CC(C)(F)C1 CC#CCC(CO)NC(C1CCCC1CNC(C1(CC2CCC2)CC1)=O)=O C1(NC(c2ccc(C(N(C)C)(CC)C3CC3)nc2)=O)CCC12CN(C(=O)C=CCO)C2 c1(N(C(C)=O)C)cccc(C2(C)CC2)c1.C1C(C2CC2)NC(=O)C=CC(=O)N1.C1(C)CC1 c1(NC(=O)NCc2c(C=O)[nH]cc2)cc(NC)cc(F)c1.C(=O)(COC)N c1(CN(c2cc(NCc3ccns3)ncn2)C)cccc(Cl)c1Cl C(CCCC(C)NCCOc1cccnc1)NC(C(C)NC(=O)CC(C)(C)OCC#N)=O.C C1(C(N2CCCN(CC(N3CCOCC3)=O)CC2)=O)CC2(CCC2)CCO1 O=C(N=c1c(Br)c[nH]cc1I)C1CC(F)CN(S(=O)(=O)C2CCOCC2)C1 c1(C(=O)NC2CCC3CC2CN3C(C2CC(Cl)(Cl)C2)=O)coc2ccc(F)cc12 C1(NC(c2cc(C)ns2)=O)CN(C(C2CC(=O)NC(=O)N2)=O)CCC1C(F)(F)F c1(C(C)N(CCCO)C)cccc(S(=O)(=O)NC2CCC2CN)c1 C12(CNC(C3C(C(=O)NCC#C)C3)=O)CC1CN(C(=O)CSc1nc(C)no1)C2 N1(C(C(C)(C)N(CC)CC)=O)CC2CN(C(=O)CN(C(=O)OCC)C3CC3)CC2C1 Cc1nc(C(F)(F)F)sc1CC(=O)N(CCCN(C(=O)CC1CCCC1C)C)C Cc1ccc(F)c(C(=O)NC(CC(C)C)C(=O)N(C2CCOC2)CCF)c1 C=C(C)CC(C(=O)NCCc1cnn(C)c1C)NC(=O)CNc1ccccn1 S(=O)(=O)(c1c(C)cc(C)cc1C)NCC1C(CC(=O)NC(CC#C)C)C1 c1(C(=O)NCC(CNC(CCC#C)=O)F)cc(F)ccc1-n1ccnc1 c1(-c2cccc(C(=O)NC(C(CC)(C)C)C)c2)ccc(C)c(N)c1 CC1(C)CCCCC1NC(=O)CCC1CCCN1C(C1CN2CCC1CC2)=O C(CCCC(=O)N1CCC(F)(CNC(C2(Cl)CC2(C)C)=O)C1)N(C(C)=O)C N1(C(CC(=O)OCC)=O)CC2(CC(CC(=O)NC3(CO)CCOC3)C2)C1 CC1(C)CC(=O)NCC1C(=O)NCC=C1CCN(C(=O)CCP(C)(C)=O)CC1 CC(O)C(F)(F)C(=O)NC12CC1CN(C(=O)C(F)(F)Oc1ccc(Cl)c(F)c1)C2 N1(C(C2C(C)CCC2)=O)CCC(C)(CCNC(C23CCC(C2)C3)=O)C1 C1(NC(c2cnn(-c3ccccc3)c2F)=O)CCCN(C(=O)CCF)C1 c1(NCC(=O)NC(C)C(N2CCSCC2)=O)cc(F)c2ncccc2c1 C1(C(=O)NCc2n(C)nnn2)N(C(c2cnc3n2CCC3)=O)CCC1(C)C C#Cc1cc(C(=O)NC2CCCCC2NC(C2CCC(C)(C)C2)=O)ccc1C Cc1ccc(C(F)(F)F)cc1S(=O)(=O)C(N1CCC(c2nc(=N)[nH][nH]2)C1)=O C12(NC(C(CCSC)O)=O)CCCC1CN(C(=O)CC=Cc1ccccc1F)C2 c1(OC)cc(CC2NC(=O)N(C(C3CCC3)=O)C2=O)ccc1Nc1ccc(F)cc1 N1(CC(=O)N(C2CCN(c3ccccc3)C2)C(C)=O)CCC(OCc2cc[nH]n2)C1 CC(C)C(C(=O)NC1CCN(C(C2(C)CCC2)=O)CC1F)C(C)C C(=O)(C1=CNC2=NCCC2=C1)N1CC(NC(CC2ON=C(CC)C2)=O)C(C)(C)C1 C1(CNC(CC(C=C)CC)=O)CN(C(C2CC(CC(F)(F)F)C2)=O)CCC12CCC2 N1(C(C=Cc2occ(C)n2)=O)C2CCC1CN(C(c1ccc[nH]1)=O)C2 C(=O)(C1CC(=O)c2ccccc21)N1CCC(F)(C(=O)OC(C)(C)C)C1 N1(C(CSCC#C)=O)CCC(C(CNC(=O)CCc2ccon2)OC)CC1 CS(=O)(=NC(=O)CCn1ccc(C(F)(F)F)n1)c1ccc(C#N)cc1 CC1CC(CNC(=O)NC2CC2CF)CC(C)O1 c1(NC(C=CC(C)NC(c2ccc(CO)nc2)=O)=O)ccc(O)cc1Cl CC1COCCN1C(C1CCN(C(C2SCCS2)=O)CC1)=O C1(C(C)C)CCN(C(C2CCCOCC2)=O)C(CNC(c2cc[nH]n2)=O)C1 N1(C(C(CCO)N(C)C)=O)CC2CS(=O)(=O)CC2(CNC(c2cnco2)=O)C1 Nc1ncc(C(=O)NCCNC(c2ccc(CN3CCOCC3)cc2)=O)cc1Cl c1(OCCOC)cnccc1C(N1CCOCC1N(C(=O)C(C)CSC)C)=O CC(Cc1cnn(C)c1)C(=O)NC1CN(C(=O)COc2ccsn2)C1 N1(C(CNC(C(C)(C)OC(C)C)=O)=O)CCC(O)C(C)(C)C1 C1(O)(C(=O)NC2C3(CC(NC(c4scc(C)c4)=O)C3)C2)CCCC(C)(C)C1 N1(C(C2(C(=O)OCC)CC2)=O)CCC(C)N(C(C2CCC3CCCCN23)=O)CC1 C1(CCNC(c2ncn(CC)c2)=O)C(C)CCCN1C(=O)C1=COCCC1 c1(CCN2CCC(c3cccc(CSCSS(C)(=O)=O)n3)CC2)ccccc1C1CC1.SC c1(C(N2CC3(C2)CN(C(=O)COCCCF)C3)=O)cnc2c(c1)COC2 c1(C(N2CCCC3(C2)CN(C(C2CC=CC2)=O)C3)=O)ccc2cc[nH]c2c1F c1(N2CC3CN(C(c4cnc(C)nc4C)=O)CC3C2)nc(Cl)nc2c1CCOC2 C1(C(N2CC(NC(c3cn4c(n3)CCC4)=O)CC(C)C2)=O)C2CCCCCCC12 N(C1CCc2c(Br)cccc21)C(=O)NC1C(c2c(C)cccc2)(C)C1 C(=O)(CC(F)(F)C(F)F)N1CC(CC=C)(NC(c2nonc2CC)=O)C1 C1(CNC(CC=CCNC(CCCOC)=O)=O)COCC(C)O1 Cc1cc(CSC)on1.C1(=O)C(F)CC2CN(C2)C(=O)C(C)N1C(C)C C1(NC(CN(CC)CC)=O)CCC(CN(C(=O)CNS(N)(=O)=O)C)CC1 O(N=C1CCCCCC1)CC(N1CC(OC)(CNC(=O)C(O)CN(C)C)C1)=O C1(C(=O)NCC2CN(C(c3sc(Br)cc3Cl)=O)CCO2)CCCC2(CC2)C1 C1(C(N(C(CC)(C)C)C2CC2)=O)CN(C(=O)C(c2cnn(C)c2)C)CCN1C N1(C(CSC)=O)CCc2[nH]nc(CNC(=O)C(C)Oc3cccc(F)c3)c2C1 N1(C(c2c(C)c[nH]n2)=O)CC(NC(=O)Cn2nnc(=N)[nH]2)C2(CCC2)C1 N1(C(C=Cc2ncn(C)c2)=O)CC2CC(C1)N2C(=O)CC1CC(C)(C)CO1 N1(C(=O)C(F)(F)Nc2ccc(F)cc2)CC=C(c2ccc(Cl)cc2)CC1 C(=O)(C(=O)C(F)(F)F)N1CCC(OCCNC(C(n2nnc(C(C)(C)C)n2)C)=O)C1 c1(NC(C2(NC(C(C)CCN(C)C)=O)CC(F)C2)=O)cnc2[nH]ncc2c1 C12(COC)CC(C(=O)NC3CC(C)N(C(=O)Cc4c(C)noc4Cl)C3)(CO1)C2 C1(CC)CN(C(C2CN(S(N)(=O)=O)C2)=O)CCC1NC(c1coc(C(C)C)n1)=O Cc1nc2ccc(C(=O)NC3CC4CC3N(C(=O)CC35CCCC3C5)C4)cc2o1 c1(CSC)nc(C(=O)N(CCOC2(C(=O)NCC(C)CCC)CC2)CC)c(C)o1 N1(C(C(CC)N2CCCC2=O)=O)CCC(C#N)(CC)CC1 N1(C(c2c(C(C)(C)C)noc2)=O)CC(=O)N2CCCCC2C1 c1(C(N(C(CN(C(C(C)SCC)=O)C)C)C)=O)cc2c(cn1)OCCO2 Cc1c(C(=O)CNC(=O)C(c2ccc(Cl)cc2)C2CC2)sc2ccccc12 N1(C(C2N(C(C)C)CCC2)=O)CCN(C)C(C(N(C)C[Si](C)(C)C)=O)C1 c1(N(c2ccccc2)C)ncnc2c1ncn2C.C12CCN(C1)C(=O)N2 c1(C(N(C(C)C)CCN(C(=O)CC(F)(F)C(F)F)C)=O)ccc(N=[N+]=[N-])cn1 CC(CS(C)(=O)=O)C(=O)N1CC2(CCCN2C(=O)CC(Cl)Cl)C1 Cc1ccc(C(=O)NCC2(C(=O)NC(C3NC(=O)NC3=O)C)CCCC2)nc1 Cc1nncc(C(=O)NCC23CC(C2)C(NC(=O)C(O)C2CC2)CO3)c1C N1(C(C(=O)NCc2ccccc2)C2CCSC2)CCn2c(cc3c(Cl)cccc23)C1 c1(C(=O)NCC(c2cccc(C)c2)NC(C(CC)F)=O)cccc2nn[nH]c12 C1(C(=O)NC2(CC=C)CN(C(=O)NCC3CC(OC)C3)C2)CC12CCCC2 c1(SC)cccc(C(=O)NCC(C2CCN(C(=O)C=C3CCC(C)C3)CC2)O)c1 Cc1nc(N2CC3C(CNC(c4cncc(C#N)c4)=O)C3C2)cc(O)n1 c1(CC(C)NC(=O)C=CCNC(C2CC2F)=O)cccs1 N1(C(C2C(NC(c3cc(O)nc(O)n3)=O)CCC2)=O)CCS(=O)(=O)CC1CCO C1(C(=O)NC2(CNC(c3c(CC)nc(C)s3)=O)CCC2)CCCC2(C1)CC2(F)F c1(OC)cccc(NC(=O)CN2CCC(NC(c3nc(C)cs3)(C)C)CC2)c1 N1(C(C(C)(C)C#N)=O)CC2CC1CC2NC(=O)CN(c1cccs1)C(N)=O c1(C(=O)NC(CC=C)CNC(c2cc(OC)n[nH]2)=O)cc(O)ccc1OC(F)F C=C(Cl)CC(C(=O)N1CCCCCO1)NC(C12COCC1C2)=O c1(C(=O)NC2(C)CCN(C(c3ccn(C)c3)=O)C2)cccc(F)c1Br C1(C(=O)OCC)CC(C)(C)CN1C(c1nccc(Cl)c1C)C(=O)NC1(C)CC1 N1(C(c2sccc2Cl)=O)CC(CO)C2(C1)CN(C(c1cscc1C(F)(F)F)=O)C2 C(=O)(C(CCC)C(C)C)NCC1(F)CCN(C(COCC(=C)C)=O)C1 Cc1ccccc1NC(N1CCN(C(=O)NC23CCC(CO2)C3)CC1)=O CC1CN(C(=O)C2=CCCS2)CCC1NC(c1cnc(N(C)C)c(Cl)c1)=O Cc1csc2ncc(C(=O)NCCn3cc(-c4cccc(N)c4)nn3)n12 C12(NC(CN(CCC)C)=O)COCCC1CN(C(c1cnoc1C1CCC1)=O)C2 c1(C(C(=O)N(CC(C)O)CCNC(CCC(=O)OC)=O)C)cc2ccccc2o1 N1(CC)CC(CNC(C2(C(=O)NCC3(C(=O)NC)CC3)CC2)=O)CC1C c1(C(N2CCCN(C(C(C)C3CC3)=O)C(C)C2)=O)cc2c(n1C)CCOC2 C1(CNC(c2ccc(OCF)nc2)=O)CCCCCN1C(C1C=CCS1)=O C(=O)(C1=C(C#N)CCC1)NC(C(=O)N(C)Cc1ccoc1)CCF N1(C(c2c(C)cc(O)nc2)=O)C2CCC1CC(NC(C1CCC3(CCC3)CC1)=O)C2 N#CC1(C(N2CCC(F)C(NC(=O)CN3CCOCC3)C2)=O)CC2(CC2)C1 Cc1cc(C(=O)NCC2N(C(=O)CCC=CC(C)C)CCC2(C)C)cc(C)c1C Nc1ccnc(C(N2C3CCC2C(CNC(c2ccn(C(F)F)n2)=O)C3)=O)c1Cl Cc1nc2c(C(N3CCCC3CNC(=O)CCCN(C)C(C)C)=O)ccnc2[nH]1 CC1=NOC(=O)C1CC(N1CCOC(CNC(c2cn(C)cn2)=O)C1)=O c1(C(=O)NC(CCOC)C(=O)NCCCC(=O)OC)cc(Cl)ccc1-n1ccnc1 N1(C(c2cnc(CC)s2)=O)CCC2(CCCN2C(C2OCCC2C)=O)C1 CC(C)C(O)C(=O)NCC12CC1CN(C(c1ccc(CO)cn1)=O)C2 C1(C(=O)NCC2CCCN(C(=O)Cn3cncn3)CC2)Cc2cccc(F)c2O1 C1(CNC(CC=CCC)=O)CC(F)(F)CN1C(C1CC2OC1C1CC21)=O CC(C(O)C(F)F)NC(C1(NC(=O)C#CC2CC2)CC(F)C1)=O N1(C(C2(C)C=CCN2C(C2CC3CC3C2)=O)=O)CCCCCCC1 c1(C(N2C3(CNC(C4CC=CCC4)=O)CCC2CC3)=O)c[nH]c2cc(F)ccc12 C12(CNC(CN(C(C(n3ncc(C)c3)C)=O)CC3CC3)=O)CCCC(CO1)C2 Cc1ccn(C(C)C(=O)N2CC(CCCCNC(N)=O)C2)n1.C12CCOC1C(=O)N2 CCC(CC(=O)N(CCCCNC(C1CCCN(S(C)(=O)=O)C1)=O)C)C(C)(C)C c1(C(=O)NCC(CC)NC(C(C2CCC2)OCC)=O)oc(Br)cc1C CC1(CNC(=O)CC23COCC(C2)C3)CCCN(C(C23CCCC2C3)=O)C1 C1(O)(C(=O)NCC2(O)CCN(C(CC3(C(=C)F)CCC3)=O)C2)CN2CCC1CC2 c1(OCC(=O)NCC2(C)CCC(NC(=O)C=CCO)C2)cccc(F)c1F c1(OCC(=O)N(C(CCNC(C2CCC(CC)C2)=O)C)CC)ccc(F)nc1 C(C)(C)(CC(=O)NCC(C)(O)CSC)NC(C(CC)SC)=O C1(NC(C2C(=C)CC2)=O)CCC(C)N(C(c2cnc(N3CCCS3(=O)=O)s2)=O)C1 C1(C(N2CC3(N(C(C(C4CCCCCC4)=O)=O)CC3)C2)=O)CC2(CCC2)CCO1 C1(CNC(C(Cc2cc[nH]n2)NC(=O)C=CC(F)(F)F)=O)C2CCCCC12 c1(OCCOC)nccc(NC(CNC(=O)C2=CCCC2)C(C)C)c1F N1(C(COCCCOC)=O)CCCC12CCCN(C(c1cc(C)oc1C)=O)C2 c1(NC2CCCCCN(C(C3N(C)CCCC3)=O)C2)nc(Cl)nc2[nH]c(O)nc12 N1CCCCC1c1nn[nH]n1.C=C1CC(C=O)(COC)C1 c1(C(=O)NCCOC2CCN(C(CC=CCC)=O)C2)cc2ncccc2o1 N1(C(C(c2ccoc2)NC(CCC2(C#N)CCC2)=O)=O)CCC2CCCC12 Cn1cc(C(F)(F)C(=O)NC2CCC2NC(=O)CC2CC=CC2)cn1 C#CCC(CC#C)C(=O)NC1CN(C(c2cnc(C(C)(C)C)o2)=O)CC1O C1(C(=O)NC2C(C)N(C(C3CCCCC3)=O)CCC2)CC(c2ccncc2)=NO1 CCCC(O)CNC(C1C=CCN1C(c1[nH]ccc1COC)=O)=O C1(CCC)CN(C(=O)C(F)(F)C(O)C2CC2)CCN1C(c1cnccc1Cl)=O Cc1cc(N)c(C(N2CCCCC2CNC(=O)Cn2cnnc2)=O)nc1C C1(NC(c2ccc(SC)o2)=O)CC(F)CN(C(=O)CC2CC2(Cl)Cl)C1 C1(NC(c2cn(C(C)C)cn2)=O)CC(=O)N(C)C1.C1(OC)CC(C2C(=O)N2)C1 C(Cn1cccn1)(C(=O)NC1CCC2CC12)NC(C=CC(C)(C)C)=O n1(CC)ccnc1C(=O)N(CCC(=O)NCC(Cl)C(C)(F)F)C(C)C C1(CN2CC(C(=O)O)CC(CC)C2)Cc2ccccc2C1(C)C C1(NC(c2c(C)cc(F)c(Cl)c2)=O)CC1C1CCN(C(=O)Cc2cnc[nH]2)CC1 C(=O)(C#CC1CCCOC1)NC1(CO)CCN(C(CC2CCN(C)CC2)=O)CC1 N1(C(C2N(C(=O)NCC)CC2)=O)CCN(C(=O)C(CC(C)C)OC)C(C)C1 N12CC3CCN(C3C1)CC2=O.C1(NC(=O)Cc2c[nH]nc2O)COC2(CCC2)C1 C1(C(=O)NCC(CC)O)C2CCCC2CN1C(C1CCC1C)=O CC(C)C(C)(O)C(=O)NC(C)C(CO)NC(C1(F)CCCC1)=O C1(CC(=O)N(C(C)CNC(c2ccc(CSC)o2)=O)CC)CCOCC1 C1(C(N2C(C)(CCC)CC2)=O)CN(C(=O)CC2CCOC2C)CCC1(C)C N1(C(c2oc(C)c(CO)c2)=O)CCN(C(C2OCCC2C(F)(F)F)=O)CC1C CCC(CC(=O)N1CC(C2CN(C(c3c(CC)nc(C)n3C)=O)C2)C1)C(C)C c1(C(=O)NCCCCNC(Cn2c(C)ccn2)=O)ccc(Cl)cc1N Cc1cc(C(C)C)nc(=NCCNC(C2(C)C=CCCC2)=O)[nH]1 c1(OC)ccccc1OCC(=O)NC(C1CCN(C(c2ccnnc2Cl)=O)C1)C c1(CCC(=O)N2CC(c3cccc(C(=O)O)c3)C2)nc2cnccc2[nH]1 N1(c2cn(C3CC(C(=O)NCC(CC=C)(F)F)C3)nn2)CCCC(OC)C1=O C1(CNC(C2(NC(C3C=C(C)CS3)=O)CC2C)=O)CC12CCOCC2 Cn1cc(C(CO)NC(c2cc(CNC(=O)C(F)C3CCCC3)on2)=O)cn1 N1(C(=O)CCc2ccccn2)CCOC2CN(C(C3(F)CC3)=O)CC12 C1(NC(CC=C)=O)COC2(C1)CN(C(=O)C(CO)C(F)(F)F)C2 CCCC(C)C(=O)NC1(C)CN(C(C23CCC2C3)=O)C1 N1(C(C(C)n2cccn2)=O)CCC=CC1C(=O)Nc1cnc(N(C)C)nc1 N1(C(c2c(Cl)cn(CC)n2)=O)CCC2(CC1)CC(C)N(C(=O)C(C)C(C)C)C2 Cc1cccnc1C(=O)N(CCC(C(C)C)NC(c1cc(CO)oc1C)=O)C CC1CCCCC1CCNC(C12CC(NC(=O)CCC3OCCO3)(C1)C2)=O C(=O)(C(C)N=[N+]=[N-])N(CCC(=O)N(CC(O)CO)C)C(C)C CCCCCCCNC(C1(CNC(C23CCCC2C3)=O)CCCC1)=O c1(OC)ccc(C(N2CC(NC(=O)CCC3CCCO3)C2)=O)c(F)c1 N1(C(C(C)=CC2CC2)=O)CCCC(C)(NC(C2CCC3CC2CO3)=O)C1 c1(C(N2CCOC(C3CC3)C2)C(=O)NC)cccc(CNc2nc(Br)cs2)c1 c1(C(N2CCC(N(C(C(CCCCC)O)=O)C)CC2)=O)cnc2ccccc2c1 N1(C(C2C(C)=CCS2)=O)CC(CNC(=O)C(O)CC(N)=O)C2(CC2)C1 C1(C(=O)NC)CCN(C(=O)CC2(C(N(CCC)C3CC3)=O)CC2)C1C.C(C)C Cc1cnn(C)c1N(C(=O)C(CCOCCO)NC(=O)CCOC1CCC1)C c1(C(N(C)CC2CCCN2C(=O)Cc2ccoc2)=O)cnccc1Br C1(CCC(=O)NCC2(C)C(C)(C)C2)CCCCN(C(c2cccs2)=O)C1 N1(C(C=NOC)=O)CCC(C)(C)C(NC(=O)COc2ccc(Br)cc2)C1 N1(C(CN(C(=O)OC)C)=O)CCC(C2CCCN(C(c3sccc3C)=O)C2)C1 C1(CNC(C(Br)=C(C)C)=O)CCN(C(=O)CCn2ccc(C)n2)CC1CO c1(CC(=O)NCC2(F)CCCN(C(c3c(C)cno3)=O)C2)c[nH]c2cccnc12 n1(CC(=O)NCC2C(CC(=O)NCC=C)C2)ncnn1 CN1N=C(CC(=O)N2CCCC(NC(C3(n4cncn4)CC3)=O)C(F)C2)CC1=O C1(CC(=O)NC(C(=O)OC)C2CCC2)CN(C(=O)CC2CCCN2C)CCO1 c1(CNC(=O)NC(COCCCNC(C(=C)C)=O)(C)C)ccc(OC)c(Br)c1 N1(C(c2ccc(F)cc2)C(=O)NCCSC)CCC2(CCCNC2)C1 C(CN=C(NCc1ccc(C)n1C)NC1CCCC(F)(F)C1)SC Cc1ccc(C(N2CCCCC2CCC(=O)NC(C)CCC2CCCC2)=O)nc1 c1(CCC(=O)NCC2C(NC(C3(CCOC)CC3)=O)CC2)ccc(O)nn1 c1(C(=O)NCC2C(C)CCN(C(=O)CC3(C)CC3)C2)cc(F)cc2c1C(=O)CC2 N1(C(C2(COC)CCC2)=O)CCCC(C2CCN(C(=O)CC(C)(C)O)CC2)C1 CC(CS(C)(=O)=O)C(=O)NC1CCCCN(C(=O)NC(=O)C(Cl)(Cl)Cl)CC1 C(CC1=CCN(C(C2CN(C)CC2C)=O)CC1)NC(C(C)(C)OC)=O CC1C(NC(c2cn(C(F)F)cn2)=O)CCN1C(C1CC1C#N)=O N1(C(CC)=O)CCC2(CC1)CN(C(C1CCCC(C(F)(F)F)O1)=O)C2 c1(C(=O)NC(CC(=O)N(CC#C)CC2CC2)CC)c[nH]c2cnccc12 S(=O)(=O)(c1cccnc1C(F)(F)F)NCCc1c(C)nn(C)c1C C1(O)(C(C(N2CC=CC2CNC(C2CNC(=O)N2)=O)=O)F)CCCC1 Nc1c(C(N2CCC(NC(=O)C3=CSCS3)C(O)C2)=O)sc2ccccc12 C1(C(N(CC(CC)NC(=O)Cc2c(C)cnn2C)C)=O)CC(C)CC(=O)N1 C1(CNC(CCNC(C(c2ccn(C)n2)C)=O)=O)CCCCC1CO c1(C(=O)NC(C(=O)NC(C2C(C(=O)OC)C2)C)Cc2cc[nH]n2)cc(F)ccc1O N1(C(CN(C(CCCCC)=O)C)=O)CCn2ncnc2C1 c1(C(=O)NC(C2CN(C(=O)CN3CCCC3=O)C2)C)cc(-c2ccccc2)cs1 O=C1CCC(CC(=O)NC2(C3CN(C(c4snnc4C4CC4)=O)C3)CC2)C(=O)N1 N1(c2nnc(-c3c(C)ncs3)s2)CC2CCCC(NC(=O)COC(C)(C)C)C2C1 c1(C(C)(F)F)cccc(C(N2C(C(=O)Nc3nccc(C(F)(F)F)n3)CC2)=O)n1 C1(NC(C(N2CCCCCC2)C)=O)CC12CC(NC(c1c[nH]ccc1=N)=O)C2 N1(C(c2ccn(C)n2)=O)CC2C3CCC(C2C1)N(C(c1ccc(S)cc1)=O)C3 C1(CNC(C(OCC)OCC)=O)(CNC(C2CC2CF)=O)CC(F)(F)C1 [N-]=[N+]=Nc1cc(C(=O)NC(c2ccccc2)C2CCC2)ccn1.C12CC1C2 N1(C(C=CCOC)=O)CCN(C(=O)C(c2cnn(C)c2)O)C(COC(C)C)C1 C1(CC(=O)NC(C)CNC(=O)Cc2nc(=N)[nH][nH]2)CCCCC1F c1(C(N(CCC(C)NC(c2cnc(SC)s2)=O)C)=O)ccc(OCOC)cc1 C(=O)(CCCS(C)(=O)=O)NCC(C)(CNC(C1CCCCS1)=O)OC O=C1CCc2cc(C(N3CCCC(NC(C4C=CCC4)=O)CC3)=O)ccc2N1 C(C(C)C(=O)N(C)CC1CCCN1OC(C)=O)N(C(C1(CC#C)CC1)=O)C C=CCCC(CC(C)C)C(=O)NC1(CC(=O)NCC2CCN(CCF)C2)CC1 C12(CN(c3cccc(C)c3)C(=O)C(=O)NC(=O)C(N)CN=[N+]=[N-])CCCC1NCC2 C(=O)(C1CNC(=O)c2ccnn21)NCC1(NC(C(C)OCCC#C)=O)CCCC1 Cc1ncc(Cl)cc1NC(=O)CSCCNC(=O)C(c1cnn(C)c1)C N1(CCNC(C(n2ccc(C)n2)C)=O)CCN(C(=O)CC2(n3cncn3)CC2)CC1 c1(C(N2C3CN(Cc4ncc(OC)cc4F)CC32)=O)cnc2c(ccn2C)c1 C1(C#N)(C(N2C(C3CCN(C(c4c(C)ccnc4)=O)C3)CCC2)=O)CC12CCCC2 c1(OC)cccc(SCC(N2CCOCC2CN(C)C(C2(O)CCCC2)=O)=O)c1 c1(C(=O)NC2(COC)CCN(C(=O)CCOC(C)C)C2)cccc([N+](=O)[O-])c1 c1(C(=O)NC2(C)CCN(C(CC=CC=C)=O)C2)cc2c(Br)c(F)ccc2[nH]1 c1(C(c2n(CC=C)nnn2)N(C2(c3cccc(Cl)c3)CC2)C2CC2)cccc(I)c1 c1(OCCC(=O)NCC(C)NC(CSCCC)=O)ccc(Cl)c(C)c1 CCC(CC)(CC)C(=O)NC1CCC(F)(CNC(c2ccc(C)cc2N)=O)C1 N1(C(C=CC=CC)=O)CC(NC(C2(C)CCCS2)=O)C2CCCCC12 CC1=C(C(=O)NC2(CNC(C3(N(C)C)CCCC3)=O)CCC2)C(C)(C)CCC1 C1(C(=O)NC(CN(C(=O)Cc2nnc(C)o2)CC)C)OCCOC1(C)C CCCC(C)CC(=O)N1CC2CC2C1CNC(=O)Cc1ccccc1OCC c1(C(=O)NC(CCCC)CNC(=O)C=CCOC)cnc(OC)c(Cl)c1 c1(COCC(=O)Cc2ccccc2F)nc(C2=NOCC2)no1 N1(C(c2c(C)[nH]cc2)=O)CCc2ccccc2C(NC(=O)C2=CC3CCC2C3)C1 Nc1[nH]c(=NCCC2CCCN2)ccc1[N+](=O)[O-] C1(C(=O)NC(c2ccc(F)c(F)c2)C)CC2(CNC2)CO1 C1(C(N2C(CNC(c3cc(CF)on3)=O)CC(OC)C2)=O)CC2CC(=O)C1C2 C(CN=c1nc(C)c([N+](=O)[O-])c[nH]1)NC(C1(C)C(CC)CCC1)=O c1(NC(C2=NOC(C)(C)C2)=O)cn2c(n1)CCC(C(F)(F)F)C2 c1(C(c2n(C)nnn2)NCc2cnc(C(F)(F)F)s2)cncc(C(F)(F)F)c1 c1(OC)cc(C(=O)NCC(C)NC(C2(C)CCCNC2=O)=O)cc(Cl)c1 CN1CCN(C(=O)CNc2cccnc2)CC1C1CN(C(=O)C#CC2(C)CC2)C1 CCCC(C)(C)C(=O)N1CCCCC(CNC(C2CCCN2C)=O)C1 c1(OC)nc(N2CCC(CCNC(c3scnc3C(C)C)=O)C2)cc(C)n1 CCCC(CCCO)C(=O)N1CCC2(C1)CN(C(c1cnnn1C)=O)C2 n1(CC(=O)NC2CC3N(C(CC(=O)OC)=O)C(CC3)C2)cnc2sccc2c1=O c1(C(N2CC(CC(C)NC(CNC(CCC)=O)=O)C2)=O)c[nH]c2c(F)cccc12 c1(C(N2CCCC(CCC(N)=O)C2)=O)ccc(-c2nnco2)cc1 N1(C(c2cnc(C(F)F)s2)=O)CC2CC(C1)N2C(c1cnn2ccsc12)=O c1(C(N2CCC(N(C(C(COC(C)C)(C)C)=O)C)C2)=O)n[nH]c2c(C)cccc12 C1(C(N(C2CCS(=O)CC2)C)=O)CC(C)(C)CCN1C(=O)CC1CCCOC1 N1(C(C2CN(C)C(=O)N2)=O)CCC2(CCCN(C(C3(Cl)CC3(F)F)=O)C2)C1 C1(C(N2CC(NC(CSCC#C)=O)C(C(F)F)C2)=O)CCCCN(C)C1=O CN1CCC(C)(C(=O)N(C)CC2CN(C(=O)C(F)(F)C(O)C3CC3)CCO2)C1=O N1(C(C2CC(C)(NC(C3CC4C=CC3O4)=O)C2)=O)CCCN2CCCC2C1 C(CCc1ccc(Br)cc1)(C(=O)NCC1CCCO1)N(C)CC1C(C)(C)C1 Cc1ccc(S(=O)(=O)NC(C)(C)C(c2ccc(O)cc2)=O)cc1C Cc1[nH]c(C#N)cc1C(=O)NC(C)CCC(=O)NC(c1cc[nH]n1)C N1(C(C(C)=C2CCCC2)=O)CCCC(NC(c2ccc([N+](=O)[O-])o2)=O)C(F)C1 c1(C(N2CCC(F)(CNC(C3CCCO3)=O)CC2)=O)cc(Cl)c(F)c(Cl)c1 C(=O)(CCS(=O)(=O)c1ccccc1)NC1(CNC(C2(C)CC(C#N)C2)=O)CCC1 C=C(C)C1OCCCC1C(=O)NCC1CN(C(=O)CC2OCCO2)C(C)(C)C1 Cc1oncc1C(=O)NCC(=O)NC1CC1CNC(C1CCNC1=O)=O c1(C(C)C(=O)NC(C)C=CC(=O)NC(C)(C)Cn2cccn2)ccn(C)c1 C1(CC(=O)NCCOC)CCCN1C(c1ccsc1Cl)=O c1(C(N2CCC(NC(c3n[nH]cc3C3CC3)=O)C2)C)cc(Cl)ncc1Cl c1(CN(C(=O)CCn2cc(-c3ccsc3)nn2)C)cccnc1Cl Cc1cc(Br)cc2cc(C(N3CCCC3CN(C(=O)C=C3CC3)C3CC3)=O)oc12 CCN=c1[nH]cc(C(=O)N(C)CC2CCN(C(C3CC3F)=O)C2)s1 Cc1coc(C)c1C(N1CCN(CN2CCN(C(=O)C(C)N(C)C)CC2)CC1)=O C(C(C)(O)CNC(c1csnc1C(F)F)=O)NC(C(c1cnn(C)c1)C)=O CCC(F)(F)CC(=O)NCC1CN(C(=O)C(C)N(C)C)CC1C(F)(F)F C1(CNC(=NCC)NCc2cccs2)CCC2(CCC2)C1O N1(C(C2N(C(C3NC(=O)C(F)C3)=O)CCCC2)=O)CCC(F)(F)CC1 Cc1cc(Cl)c(C(N2CC(NC(c3coc(C(C)(C)C)n3)=O)CC2C)=O)cn1 N1(C(C=CC)=O)CCC2C(COC2C(N2CCOC(C(=O)OCC)C2)=O)C1 c1(CC(=O)NCC(C(C)C)NC(c2cc(N)ccc2Cl)=O)ccc2nsnc2c1 C1(CNC(c2n[nH]c(C)c2O)=O)CC2(C1)CN(C(=O)CCCN1CCCCC1)C2 C1(CNC(c2ccc(C)o2)=O)CC2(CO1)CN(C(C13CCC(C)(CC1)OC3)=O)C2 c1(C(=O)NC(C)CONC(=O)c2ccsc2)nccc2[nH]ccc12 OCCC(N=c1[nH]c2c(c(=NCc3cocn3)[nH]1)COC2)c1ccccc1 c1(OC)ccc(-c2cn(C3(C(N4CC(C)CCC4C)=O)CC3)nn2)c(Cl)n1 Cc1nn(CC(=O)NC2CC3(C2)CC3C(=O)N(CC(C)O)CC(C)O)c(=O)o1 C1(NC(CCC(=C)C)=O)CC2CC1CN(C(c1ccc(Cl)cc1C(F)F)=O)C2 C#CCC(C)(C(=O)N1CCC(CC(C)O)CC1)NC(c1cc(CC)[nH]n1)=O N1(C(CN(CC(C)C(C)(C)C)CCC)=O)CC2CCC2(CC(=O)NC2CC2)C1.CC CC1NC(=O)CCC1CNC(=O)C(N1CCC(Cc2nccs2)C1)=O c1(N(CCCNC(c2cc(CCC)c(C)s2)=O)C)ncnc2cc(Br)sc12 c1(C(C)=O)cccc2c1ccn2CC(=O)N(C)CC1(NC(C2C(C)C2C)=O)CC1 N1(C(c2c(CC)cno2)=O)CCC2(CCN(C(C3CCCC(O)C3)=O)CC2)C1 C1(C(=O)NCc2scc(CNC(C=C(C)C(C)C)=O)n2)CC=CCO1 C(CCCCCNC(=O)C=CCCC(C)C)NC(Cc1c(C)ocn1)=O CC1COCC(C)N1C(C1CC(F)CN(Cc2cccc(-c3ccccc3)n2)C1)=O c1(N2CCC(CCNC(C3C(CC)CCC3)=O)CC2)cc(Cl)nc(C2(C)CC2)n1 c1(CC(=O)NCCCN(CCCCNC(CC(=C)C)=O)C)c(C)noc1C Cc1n[nH]c2cc(C(=O)NCC3CN(C(C4CCCCO4)=O)CCN3C)ncc12 N1(C(c2n(CC#C)ccc2)=O)CCC(C)(NC(c2cc(C3CC3)on2)=O)C1 c1(C(=O)NCC2(OC)CN(C(C34CC(C#N)(C3)C4)=O)C2)ccc(F)c(O)c1 C1(N(C)C(=O)OC(C)(C)C)CC2CC1N(C(C1CCC(C(=O)N)CC1)=O)C2.C1(C)CC1.N N1(C(C2CC(C)OC2)C(=O)Nc2ccccc2)CCn2ncc(S(C)(=O)=O)c2C1 C1(OCCOC)CCCCC1NC(N1CCCC1(C)C(F)(F)F)=O c1(N(C)C)ccc(-c2cn(CC3CCCN3C(N3CCCCCC3)=O)nn2)cc1 C1(CC(=O)NCc2ncc(C)[nH]2)CN(C(c2cc(CC3CC3)[nH]n2)=O)CC12CC2 C1(CC(N2CCCC(OCC#C)C2)=O)CC(C)(C)CN1C(=O)CCc1cnco1 N1(C(=O)Cc2cccs2)CC2CCC1CN2C(c1cccc(C2CC2)n1)=O CC1OC2(CO)CC1(C(=O)NC1CCC(CNC(=O)C=C3CCN(C)CC3)C1)C2 C(=O)(C(C(C)C)C(C)C)N1CCC(C(C)NC(CCc2cc(C)nn2C)=O)CC1 N1(C(C2(C(CC)=O)CC2)=O)CCCC(NC(=O)CCC(=O)Nc2nccs2)C1C c1(C(=O)NC(C)CCNC(=O)Cc2ccc(O)cn2)cccc2ncnn12 c1(C(=O)OCC)cc(Br)c(C)cc1NC(C1CC(=O)N(CCOC)C1)=O C1(NC(=O)CCOc2ccc(F)cc2)CN(C(C2CCC2)=O)CC(F)(F)C1 C1(n2ccc(C)n2)CCCN(Cc2ccnc(C(=O)OC(C)(C)C)c2)C1 C1(CNC(=O)C(F)C2CCC2)CN(C(=O)Cn2cccn2)CCC12CCOCC2 C1(C(=O)NCCN(C(c2ncccc2N)=O)CC)CN(CC)CCO1 C=C1CC(C(=O)NCc2cn(Cc3cscn3)nn2)(COC)C1.C(=O)N c1(CC(=O)NCCC2CC(NC(=O)C(O)CC(F)(F)F)C2)cnn2c1CCCC2 S(=O)(=O)(c1cc(C(=O)NCC2CCN2C(C2(C)CC=CC2)=O)ccc1OC)NC Cc1cnc2cc(C(N3CC4(CC4)CC3CNC(C3CNC(=O)N3)=O)=O)ccn12 Cc1nc2cc(NC(=O)CC3CCCN3C(=O)CS(C)(=O)=O)cnc2[nH]1 CC1(C)C2CCC1(C(=O)O)C(NCc1c[nH]c3cnccc13)C2 c1(S)ccc2ccccc2c1.N1(C2(NCC(C)(C3CC3)OC)CC2)CCO1 CC1CCOC(C(=O)N(CC(=O)NCC(C)(C)n2cccn2)CC2CC2)C1 C1(NC(c2ccc(C)c(F)c2)=O)CC12CCN(C(C1CC=CC1)=O)CC2 CC(C(=O)NC(C)CC1CN(C(c2cccc(CN=[N+]=[N-])c2)=O)C1)C(C)O c1(NC(=O)NC(CC(N2CCC(NC(CC=C)=O)C2)=O)C2CC2)ccc(F)cc1 Cc1ncccc1CC(=O)NCCCC1CCCN1C(=O)C(C)C1(O)CCC1 C1(NC(c2cccn3cnnc23)=O)CN(C(=O)Cc2cnc[nH]2)C2(CCOC2)C1 C=CC1(CC(=O)NCC(C)(CC)OC)CN(C(=O)C=C(C)C2CC2)C1 O=C(C1=NOC2(CCN(C(c3cncnc3)=O)C2)C1)Nc1cccc(I)c1Br n1(CC)nnc(C)c1CNC(=O)C(O)CCNC(=O)CC1CCC(=O)NC1 Cc1noc(C)c1S(=O)(=O)NC1CC2CN(Cc3cc(F)cc(Cl)c3C)CC2C1 C(=O)(C#CC1(CC2CC2)COC1)N(C1C2CN(C(CC(CC)CN(C)C)=O)CC21)C c1(C(N(C)CC2(CNC(C3CNC(=O)N3C)=O)CC2)=O)csc(S(N)(=O)=O)c1 Cc1cccc2c1OC(C(=O)NCCNC(C1(c3ccc(Cl)cc3)CC1)=O)C2 Fc1ccc(Oc2ccccc2)c(SCc2c[nH]c(C(F)(F)F)c2)c1 N1(C(c2nn(C)c(C#N)c2)=O)CC2(CCCC2NC(c2cc(N)c(F)cn2)=O)C1 Cc1ccc(CCC(=O)N(CC(O)CN(C(=O)C=CC2CC2)C)C)o1 C1(NC(=O)Cc2cncs2)COC2(CCCN(C(=O)Cn3cccn3)C2)C1 c1(-c2n(C)cnn2)cccc(CNC(c2cnc(CN3CCC(CO)C3)s2)=O)c1 N1(C(c2c(OCC)ccc(C)n2)=O)CCC2CC2(NC(=O)Cn2cccn2)CC1 C1(CCNC(c2cc(OC)no2)=O)CCN(C(C2(C)CNC(=O)C2)=O)CC1(F)F C1(CC=C)(NC(=O)C(C)S(N)(=O)=O)CCN(C(=O)CCc2nc(C)cs2)CC1 c1(OCCOC)ccc(CCC(N2CCOC(CN(C(=O)C(F)F)C)C2)=O)cc1 c1(C(=O)NCCC(C(=O)N(CC(O)CO)C)OC)ccc(O)c(F)c1 C(C(C)C)(C(C(=O)Nc1cccc(Cl)c1OC)N1CCCC1c1cn[nH]c1)OC c1(CN(C(C)(C)C)CC2CC2)ccc(Cl)cc1.C1(N)CCCNC1 CCCCC(C(=O)N1CCC1C(C)O)NC(c1cccc(F)c1O)=O C(=O)(C(C)(O)CCC)NC1(CC)CN(C(C(C(=O)NCCC)F)=O)C1 C(CC(=O)NCCOCC1CCCC1)(C(F)F)NC(CCc1n(C)cnc1)=O C(C1CCOCC1)=CC(N1CCCC1CC(=O)NCCC(F)(F)CO)=O c1(CC(NC(=NC)NC(C2CCOC2)C2CC2)C#C)cccc(F)c1 CN1CCN(C(=O)CCC2CC3CCC2C3)C(CNC(=O)CC(C)(C)C#N)C1 C(=O)(C(O)C(F)F)N1CC(CCCCN)C1.c1(CC)ncccn1.C1C(=O)C1=O Cn1cncc1C(O)C(=O)NC1CCN(C(C2(CC#N)COC2)=O)C1 c1(OCC)cncc(C=C(C)S(=O)(=O)NCCc2cc(Cl)nc(=N)[nH]2)c1 CC1(CNC(C2CCOCC2)=O)CCN(C(C2SC3C=CC2CC3)=O)CC1 Nc1c(F)ccc(Cl)c1C(=O)NC1CCN(C(=O)Cn2cnnc2O)CC1 CCCC(C(F)F)NC(=O)CC1CCC(NC(=O)C(c2ccc(F)cc2)F)C1 c1(SCC)cccnc1C(N1CCCC1CCNC(c1cn(C2CC2)nn1)=O)=O C1(C(=O)NCCC(C)OC)CC(C)(NC(=O)C(C2CCOCC2)F)C1 N1(C(C2C(=C)C2)=O)CCN(C(c2ccccc2C(C2CCC2)=O)=O)C2(CCC2)C1 C1(OC)(CNC(=O)CC(C)c2cccnc2)CCN(C(c2ncccc2N)=O)C1 c1(C(=O)NC2(C)CCN(C(=O)COCC3CCCO3)CC2)ccc([N+](=O)[O-])cn1 CC1CC(NC(=O)C=Cc2ccsc2)CN1C(c1cc(C(C)(C)C)n(C)n1)=O c1(C(N2CC3CC3C2)=O)cc2ncc(-c3c[nH]nc3C(F)(F)F)cc2[nH]1 C1(NC(c2c(C(C)C)n[nH]c2)=O)CCC2(CCN(C(C3(C)C=CCCC3)=O)C2)C1 c1(OC)nc(Cl)ccc1S(=O)(=O)Nc1cnc2ccnn2c1 c1(C(C(=O)NCC)N(CC)Cc2ccc(C)o2)ccc(Br)c(C)c1 C=CC1(C(N2CCC(C(C)C(=O)NC3CC(=O)N(O)C3)C2)=O)CCOCC1 C(=O)(C(CCC(N)=O)NC(N)=O)N1CCCC(CNC(C(C)CC(N)=O)=O)C1 C(=O)(C(C)CC(N)=O)N1C(C(C)NC(c2c(C)oc(-c3cccs3)n2)=O)CCC1 c1(C2CCN(C(Cc3c[nH]c(=N)s3)=O)C2)cc(N)c(NC(=O)C(F)(F)F)cc1C c1(CNc2c(NCc3nc(CC)sc3)cccc2)cccc2c(C(=O)O)n[nH]c12 C(=O)(C1=CS(=O)(=O)CCC1)N1CCN(C(CN(CC(C)(C)C)C)=O)C(C(F)F)C1 C#Cc1cccc(CC(=O)N(C(C)C(C)C)CCC)c1.C1(CC)CC(=O)N1C(C)C c1(C(C)C)ccc(C(=O)NC(CNC(c2n[nH]cc2C2CC2)=O)C2CC2)c(F)c1 c1(C(N2CCC(N(C(CN(CCC#C)C)=O)CC)C2)=O)cccc2c1CCC2 N1(C(C=C(C)C(C)C)=O)CCCCC1C(C)NC(=O)CCc1ccc(C)cc1 CC(C)(O)C(F)C(=O)NCC1(F)CC(NC(C2CC3CCC(C2)O3)=O)C1 C(=O)(C(C#N)C1CC1)NC(C1CCCN1C(=O)CSS(C)(=O)=O)C C#Cc1cc(C(=O)NC(C)(CNC(c2cc(COC)on2)=O)CC)cc(F)c1 C1(CNC(Cc2ccc(CC)cc2)=O)CCCCN(C(C2CCCN(C)C2)=O)C1 N1(C(c2n[nH]c3c2CCC3)=O)CCC2(CC1)CN(Cc1ccc(Cl)cn1)CCO2 Cc1nc(C2CCC2)sc1CC(=O)N(CCCCNC(=O)CN1CCCC1)C c1(C(N2CC(CCCNC(C=CC)=O)OCC2)=O)ccc2oc(C)nc2c1 c1(C(=O)NC(c2ccncc2Cl)C)ncccc1N1CCOCC1 C1(N(C(CCCOCCC)=O)CC)CCCN(C(=O)CC2CCCC2C)CC1 C1(NC(c2c(C)snc2)=O)CCC2(CC1)CN(C(c1ccc(CO)cc1)=O)C2 N1(Cc2cc(C)n(CC(=O)OCC)c2C)CC(C)(C)OCC1C(=O)OC CC(C)C(C)C(CNC(c1cn(C2CCCC2)nn1)=O)NC(=O)CCC1CCC1 Cn1nc(CC(N2CCCC2CCCNC(C23CC(C2)C3)=O)=O)cc1Cl C1(CNC(C=CCCC)=O)CN(C(=O)CSc2cccc(OCC)c2)CCO1 C1(O)(CN(C(c2c(C(C)C)ocn2)=O)C)CCN(C(C2CC2(C)C(C)C)=O)CC1 C1C(CCN=c2[nH]cnc3c(F)c(F)ccc23)N1.CC(C)(C)OC(=O)CCN C(CNC(=O)CCC1CC(F)(F)C1)(CC(C)C)NC(CCN(C(CC)CC)C)=O c1(C(=O)NC(C)C(N2CC3(CCNC3=O)C2)=O)cc2ccccn2c1 c1(OCC)oc(C)nc1C(=O)NCC(C)(CC)NC(c1ccon1)=O c1(OC)cc(C)c(CNCc2conc2CSC)cn1 N1(C(CC(COC)C)=O)CC2(C(=O)NCc3nc(CO)n[nH]3)CC1CCO2 C(=O)(C1CCOc2ccccc21)NCC1(C)CC(NC(c2cc(C)c(C)s2)=O)C1 c1(OC)cncnc1C(=O)NCC1CC1C(=O)N(C(CO)C1CC1)C C(=O)(CC(O)(C(F)(F)F)c1ncco1)N1C(CNC(C2SCCCS2)=O)CC1 Cc1ccc2c(NC(C3CC3NC(c3cc(C)c(Br)cc3C)=O)=O)cccc2n1 N(C1c2ccccc2CCC1C)C(=O)Nc1c(C)n2c(nc1)ccn2 C1(C)(NC(c2ccc(C(C)C)cc2)=O)CCCN(C(=O)C2=COCCC2)C1 Cn1nc2ccccc2c1-c1nc(-c2ccccc2Br)no1 CCC(C)(C)C(CC(=O)Nc1ccccc1-c1nc[nH]n1)c1ccccc1 C(CC(=O)N)SCCC.C1CC(=O)N1CC(C)C.C1(CCCF)(C(CC(C)C)=O)CC1 c1(CN2C(C(N(CCC#C)C)=O)CSCC2)cc(Cl)cnc1Br C1(C)(C(=O)NCC(CCCC)NC(=O)Cn2cnnc2)CC=CCO1 CCC(CC(=O)N1CC(C)(C)CC1CNC(C1(C)CC1)=O)C(C)(C)C C1(C(N2C(C(C)O)CC2)=O)CCC(C)(C)N(Cc2cn(CCCF)nn2)C1 O=C(C1=CCCN(C(c2ncco2)=O)C1)NCC1CC2CCCC2C1 N1(C(c2c[nH]c3cccnc23)=O)CCc2c(F)cc(F)cc21 Cc1ncc(CNC(C23CC2CN(C(=O)CCc2ccsc2)C3)c2cccs2)cn1 c1(C(=O)NCCCNC(=O)CSC(F)F)ccc(C2CCOC2)cc1 CS(=O)C=CC(=O)N1CCCC1CNC(C1CCCN1C1CCCC1)=O c1(C(=O)NC(CN(C)C(C2CC2CF)=O)(C)C)ccc(F)nc1F C(=O)(C1=NN(c2ccc(C)cc2C)C(=O)C1)NCC1C2CN(C(CC)=O)C1C2 c1(NC(c2occ(C)c2)=O)cccc(NC(C2CCCN2CCC(C)C)=O)c1 N1(CCC)CCN(C(=O)CCC2CCCN(C(C3CCCS3)=O)C2)CC1 c1(C(=O)NC(CN(C(C(F)=CC)=O)CC)C)c[nH]c2cc([N+](=O)[O-])ccc12 c12ccc3c(c1)CN(C3)C2=O.C1(OCC)CCN(Cc2cccnc2)C1 C(=O)(C(CC(C)C)NC(=O)CC1CN(C(c2scc(C)c2Cl)=O)CCO1)NC c12cn(nn1)C(C)C(=O)NC2.C1(N)CC(CF)C1.S(C)(=O)(=O)NC c1(N(C(c2c[nH]c(=NCC=C)s2)=O)C)ncnc2cccc(C)c12 N1(C(c2ccc(CC)nc2)=O)CC(C(=O)NCC=CBr)C(C)(C)C1 C1(NC(C(C)C2CC2)=O)CCN(C(=O)Cc2ccco2)C12CC2 N1(C(C=CCN(C)C)=O)CC(CNC(c2cnc(C(C)(C)C)o2)=O)C2CC12 C(=O)(CS(=O)CCC(F)(F)F)NC1(C2CCN(C(c3ccn(C(C)C)n3)=O)C2)CC1 N1(C(c2c(SC)nn(C)c2)=O)C(CNC(C2CC2[N+](=O)[O-])=O)CC2CCCC12 N1(C(C2N(C)CCC2)=O)CC(=O)CC1C(=O)NCC1(C)CCOCC1 C#CCCCCCC(=O)NCC1CCN1C(c1c(C)ccc(Cl)c1F)=O C(=O)(C(F)(F)C(O)C(C)C)N1CCC(NC(c2[nH]cc(S(=O)(=O)NC)c2)=O)C1 Cc1c[nH]nc1C(N1CCC1CC(=O)NCC1(N(C)C)CCSC1)=O CCC(CNC(c1n[nH]c2ccccc12)=O)(CC)C(=O)NCCC(C)CCO c1(NC(CC2N(C(C(C)=CC=C)=O)CCC2(C)C)=O)ccc2occc2c1 c1(OC)cccc(C(C)(C)C(=O)N2CCC(C(=O)NCc3ncc(CO)s3)C2)c1 c1(C(=O)OC)ccc(C(=O)OC)c(NC(N2CCOC3(CCSC3)C2)=O)c1Cl CC1(O)CCC(CC(N2CCC(CF)(NC(c3cc4n(n3)CCO4)=O)C2)=O)CC1 c1(C(=O)OCc2c(OC)cc(Cl)nc2)cnc2c(c1)c(C)nn2C C1(NC(C(C)OCCC#C)=O)CC1C1CCN(C(c2cnc[nH]c2=N)=O)CC1 N1(C(CCc2c(C)noc2)=O)CCCCC(C(=O)NCCCCN=[N+]=[N-])C1 Cn1ncc2nc(Cl)nc(NCC3CN(C(c4ccc5nonc5c4)=O)C3)c12 N1(C(C2(CC=C)CC=CC2)=O)CCCCC(C(N2CCCC(N(C)CC)C2)=O)C1 C(=O)(C(CC)(CC)CC)N1CC(CCC)N(C(=O)C=Cc2ccccn2)CC1 C(=O)(C(CO)C(C)(C)C)N1CCC=C(CNC(c2sc(C)c(O)n2)=O)C1 N1(C(c2cc(C)c(Cl)cc2)=O)CCCC2CN(C(=O)C(=O)Cc3ccccc3)CC12 c1(NC)ccc(C(N2CC(NC(=O)CC(C)C(C)C)CCC2C)=O)c(Cl)c1 C1(NC(C2C(C)(Br)C2)=O)CCCOC12CCN(c1cnc(C#N)cn1)CC2 N1(C(CC=C)=O)C(C(=O)NCCn2cc(COC)nn2)CC1C N1(C(C(C(CC)CC)C)=O)CCCCC12CC(NC(C1CCCC1)=O)C2 c1(C(=O)NC(CC)CNC(=O)CCc2ccc(OC)cc2)ncc2n1CCCC2 CC1(C(N2CC(O)(c3cn(CS(=O)(=O)CCCC4CC4)nn3)C2)=O)COC(=O)OC1 N1(C(CCCOCC)=O)CCOC2(CCCN(C(=O)C3=C(CC)OCCS3)C2)C1 C=C1CC2(C1)CC(C(N1CC(N(C)C(c3cc(Cl)cc(Cl)c3)=O)C3(CC3)C1)=O)C2 C#Cc1ccccc1Oc1ccc(C(=O)Oc2cc(C3CC3)ncn2)cc1 C1(CNC(C2CC(=O)N(O)C2)=O)CN(C(=O)CSc2cccc(F)c2)CC1(F)F C1(C)(C(N2CCCC(N(C(COCCCC#C)=O)CC)C2)=O)CCCCC1(F)F c1(C(=O)NC2C=CC(CNC(C3CCOC3)=O)C2)ccc2c[nH]nc2c1 C1(CC(N2CC(n3cc(Cc4cccnc4)nn3)C2)=O)CCCCO1 N1(C(C(CN(C(CCC(C)(C)OC)=O)C)C)=O)CCOC2(CCC2)CC1 N1(C(=O)CCOc2ccc3ncccc3c2)CCCc2c(F)ccc(Br)c21 Cc1ccc(C(=O)NC2CC(CNC(=O)C(C)C3CCC3)C2)c([N+](=O)[O-])c1 c1(C(=O)NC2C(CNC(C(C(CC)C)O)=O)CC2)cc2occ(Br)c2[nH]1 C(N=c1[nH]c2c(c(=NC3CC(C(N)=O)C3)[nH]1)SCC2)c1nc(CC)sc1 N1(C(C(c2ccco2)NC(C(C2CCC(=O)N2)C)=O)=O)CCC12CCCC2 c1(C(N(C)C)=O)cnc2n1CCN(C(c1ccn(CCO)c1C)=O)C2 N1(C(CCN(C(=O)OCC)C)=O)CCC2(CC2NC(c2cccnc2CC)=O)C1 c1(C(=O)OCCC2CC(C)CC(C)(C)C2)cccc2c1OCC2(C)C Cc1cc(C(N2CCC(C(c3ccccc3F)=O)CC2)=O)sc1Br c1(C(c2n(CC)nnn2)NCc2cc(C)c(C(=O)OC)s2)cc(Cl)c(C)cn1 N1(C(C#CC2(C)COC2)=O)CCC2(CNC(=O)COC3CCCC3)CCCCC12 c1(C(N(CCNC(=O)C(C)(O)CC(C)C)CC)=O)nccc2ncccc12 N1(C(c2ccc(CC)[nH]2)=O)CCC(O)(C(C)NC(=O)Cn2ccnn2)C1 c1(CC(C)C(=O)NCC(F)CNC(=O)C2=CCSC2)ccccc1Br CC(c1ccco1)=CC(=O)NCc1ccc(CCNC(=O)C(F)C2CCC2)cc1 c1(C(=O)NC(CNC(C(c2ccc(F)cc2)OC)=O)C)ccc2nc(O)cn2c1 C1(CNC(c2n[nH]c(CC)c2Cl)=O)CCN(C(C2CCCC2(C)C)=O)C12CC2 Cc1coc(C)c1C=CC(=O)NC1CC1NC(=O)Cn1cnc([N+](=O)[O-])c1 C1(OC)CCC2(CCN(C(=O)CN(c3ccccc3)Cc3ccccc3Br)C2)C1 N1(C(c2cc(C)n(C(F)F)n2)=O)CCCC2(C1)CN(C(C1CCCS1)=O)CCO2 Cc1coc(C(=O)NC2CCCC2c2cn(CC3CCC(=O)O3)nn2)c1C#N c1(C(N2C(CNC(CC(C)C)=O)COC(C)(C)C2)=O)cc2cc(F)c(F)cc2[nH]1 N1(C(c2cnn(CC)c2Cl)=O)CC(NC(=O)COc2ccsn2)C2(CCC2)C1 C(=O)(CS(=O)(=O)CC(C)C)NCCC1(O)CCN(C(C2C(C)=CCS2)=O)C1 N1(C(C2CC(OC)C(OC)C2)=O)CC2CC(C1)N(C(c1cc(OC)n(C)n1)=O)C2 CN=c1nc(C(=O)NC2CC(CNC(=O)CCC=CBr)C23CCC3)cc(C)[nH]1 N1(C(CC(Cc2cccs2)NC(c2c(C)c(O)ccc2)=O)=O)CCC(F)(F)C(F)C1 c1(CCC(=O)O)ccc(CNC2CCCCC2n2ccnc2)nc1 C1(CCNC(C2CCCC2O)=O)CC2CCC(C1)N2C(c1cc(CCO)on1)=O c1(C(N(CC(CN(C(Cn2cc(C(=O)NC)nn2)=O)C)O)C)=O)cc(C)c(C)s1 c1(C(=O)NCC2C(CNC(CCCOC(C)C)=O)C2)[nH]ncc1C#N N1(C(CSCCOC)=O)CC(C(N2CC3CCC3(C)C2)=O)CC(C)C1 N1(CC)CC(=O)NCC1c1ccccc1.C(C(C)(C)C(=O)O)S C1(SC(c2ccc(OC)cc2)CCC)CCC(C)N1C(=O)CC(=O)OC C(CC1=CCN(C(C2CCN(C)C(=O)C2)=O)CC1)NC(c1ccc(C)nn1)=O N1(C(CSCCCC)=O)CCC(F)(CNC(c2ncnc(OC)c2F)=O)CC1 c1(C(N2CC(CCNC(c3c(C)nsc3)=O)OCC2)=O)cc(C)c(C#N)c(C)c1 C(C)(CCC(=O)NCC1(OCC2CCC2)CC1)OC C1(CC)CCCN(C(C23COCC2C3)=O)C1C(=O)NC(c1ncc[nH]1)CO C1(C2(C)N=N2)CCCN(C(C2CCCN2C(c2c[nH]c(=N)s2)=O)=O)C1 N1(C(C(=O)NC2CC2)CCc2ccccc2)CCC2(CCCOC2)C1 N1(C(COc2cccc(C)c2)=O)CCC2(CC1)CCN2C(c1ccoc1)=O Cc1cnn2c1N(C(=O)CC(C(F)F)NC(=O)CC1CSC1)CCC2 C1(C(=O)NCC(C)N(C(COCCOCC#C)=O)CC)CCc2n[nH]cc2C1C N1(C(CC(=O)N(C)C)=O)CC2OCC(NC(C3CC3c3cccc(F)c3)=O)C2C1 CC1C(C(=O)N2CCN(C(c3ccncc3F)=O)CC2C)=Cc2ccccc21 N1(C(C(C=C)(C)CCOC)=O)CCCC2(CCN(C(=O)C(F)(F)C(C)C)CC2)C1 CC(=O)CCCCC(=O)NC1CC(NC(=O)CCc2ccc(C)c(Cl)c2)C1 c1(C(=O)NCC2CCCC(NC(C(C)=C3CC3)=O)C2)oc2ccc(Cl)cc2c1C N1(C(c2cn(C(C)C)nc2)=O)CC2CC(C1)CN(C(=O)CCC(F)F)C2 O=C(CC(F)(F)C(F)F)NCCSCC(N1CC(C2CC2)(CO)C1)=O c1(C(=O)NC(C(N2C(CC=C)CC(O)C2)=O)C2CCCO2)ncn2c1CCC2 CC(C)(CCC#N)C(=O)NC1CC1NC(c1ccc(C2CCOC2)s1)=O c1(C(=O)NC(CC)CN(C)C(C2(OC)CCC2)=O)cnc(OC)c(Cl)c1 CON(C)C1CCN(CCC(=O)N(c2ccc(C#N)cc2Br)C)CC1 C1(CNC(C=CCC)=O)CCN(C(=O)CCc2cncn2C)C12CC2 C1(NC(c2sccc2CC2CC2)=O)CN(C(=O)CN2CCOCC2)C2CCCCC12 c1(C(=O)NCC(COC)(C)SC(C)(C)C)ccc(S(=O)(=O)NCCO)cc1 N1(C(C=CC(C)(C)NC(C2CC23CCOCC3)=O)=O)CCC2(CCCCO2)C1 CC(C)CC(C)CC(=O)NC1CCC(CC(=O)NC2CC3CCCC3C2)CC1 Cc1ccc(-c2nc(C(CCS(C)(=O)=O)NC(=O)N(C)C)cs2)c(Cl)c1 C1(COC)CCN(C(C2CC(NC(C3(C)CC3)=O)C2)=O)C1(C)C C1(CC)CC(C(N2CCN(C(=O)Cc3cnn(C)c3)CC2C(C)C)=O)CC(=O)N1 CCCC(C(=O)NCc1c[nH]nc1C(=O)NC1CNC(=O)C1)OCC C1(CN(C(c2n(CC)ncn2)=O)C)CCN(C(=O)C(N2C(=O)CCC2=O)C)CC1 N1(C(C(C2CC2)OC)=O)CCCCC2(CCN(C(=O)CNC(=O)CCCCO)C2)C1 C#CCCCCCC(=O)NCC(COC)NC(C1CCN(C(=O)OC)C1)=O C1(NC(=O)Cc2ccccc2O)CN(C(c2[nH]ccc2C2CC2)=O)C2(CCC2)C1 n1(CC(=O)NCCn2cc(C3CC3)nn2)nnc(C2CC2)n1 Cc1cc(C(N2CCC(F)C(NC(=O)CCCCCO)C2)=O)cc(C)c1F c1(OC)ccn2cc(C(=O)NCCCN(C(c3csc(C)c3)=O)C(C)C)nc2c1 c1(C(=O)NCCC(CNC(c2c(COC)cco2)=O)O)ccc(C2(C)CC2)cc1 CC1(C#N)CCCN(C(=O)C(=O)NCCc2ccc3c(c2)CC3)C1 c1(-n2c(-c3ccn(C4CCCC4)n3)nc(C(C)OC)n2)cc(C)ccc1Br N1(C(C2=CCCCC2C)=O)CC2(CCN(C(c3cc(F)c(O)c(F)c3)=O)CC2)C1 C(=O)(C(C(C)C)NC(c1ncc(F)cn1)=O)NC(C(=O)NCC)C C=CCC(C)(CC=C)NC(=O)C1=CCC(NC(=O)CC(CC)C2CCC2)C1 CC(C)C(CCN(C)C(c1cn(C(C)(C)C)nn1)=O)NC(c1ccno1)=O N1(C(C(CC)OCC2CC2)=O)CCOC(C(=O)NOCC(O)C(C)C)C1 c1(C(=O)NCCOC2CCN(C(C3(CC4CC4)CC3)=O)CC2)cnn2c1NCCC2 c1(C(N2C(C(=O)NC(CCC)CO)CC(F)C2)=O)ccc(OC(F)(F)F)cc1Cl C=CCCCC(=O)N1CCC1CNC(=O)CCNC(C1CCCO1)=O C1(C(N(CC#C)CC2CC2)=O)CCCCCCN1C(=O)C(C)OC(C)(C)C N1(C(c2scc(C)c2)=O)CCCCC(C(=O)NCC2OC(=O)CC2(C)C)C1 c1(C(N(CCC(C)NC(=O)C(C)(C)C)C)=O)ccc(N2CCCCCC2)cc1 C(=O)(C(C(=O)N1CC(CNC(C2(C)CCN(C)CC2)=O)(OC)C1)C(C)C)OCC C(CCC(C(=O)NC1C2CCCCC12)NC(=O)C(C)CC#N)OC c1(C(N2C(c3cn(CC(C)O)nn3)CCCC2)=O)ccn(CC(F)F)c(=O)c1 c1(C(N2CCC(C(C)NC(Cn3c(C)cnc3)=O)C2)=O)cnc2c(cnn2C)c1 c1(Cc2cnn(C)c2)nc(C)nn1-c1cccnc1CC.C1(C)(C(C)C)CC1 CCCCCC(=O)NCCOC1CCN(C(=O)CCC2CCCN(C)C2)C1 c1(C(=O)NC(C)CNC(=O)Cc2nccn2C)c(F)ccc2c1NCCC2 Cn1cc(C=CC(=O)NC(C)(CNC(=O)CC2CC23CC3)C2CCC2)cn1 n1(CC(=O)NCC2C(NC(CCCCCC#C)=O)CC2)c(=O)oc2ccccc12 c1(C(=O)NC(C)CNC(c2ccoc2CC(N)=O)=O)ccc2cc(Cl)ccc2n1 c1(C(N2CCC(CF)C2)C(=O)NCCOCC)cc(Cl)sc1C N1(C(C)=O)CCCC(N=c2[nH]c(=NCC3(S(C)=O)CC3)[nH]c3ccc(Cl)cc23)C1 CC1=C(C)CN(C(=O)CN(C)C(c2cnc(C)c(C)c2)=O)CC1 c1(OCC(=O)OC2CCN(C(=O)OC(C)(C)C)C2)cc(OC)cc(Cl)c1 C1(N(C(C(C)c2cccs2)=O)C)CCC(NC(c2cnc(Br)s2)=O)C1 C(C)(C(=O)N1CC(O)CO1)N(C(CCCCCOC)=O)CC1CC1 N1(C(=O)C=Cc2cc[nH]n2)CCCC(N(C(=O)CCSC2CCCC2)CCO)C1 c1(CN(C)CC2N(C(c3nc(CCCCC)sc3)=O)CCC2)cncc(C)c1 N1(C(CC(=O)NCC2C(NC(c3cn(CCOCC)nc3)=O)C2)C)C(=O)CCC1=O O=C(CCCCC(F)(F)F)NC12CC1CN(C(=O)Cc1ccc3n[nH]cc3c1)C2 N1(C(C2CCCC(OCCNC(C3CCOC3)=O)C2)=O)CC2CCC1C(O)C2O Cc1nc2ccc3nc(NC(C4CC5CCC4C5)C)sc3c2s1 c1(NC(C)=O)cc(F)ccc1C(=O)NCC#CCNC(=O)CC1(O)CCCOC1 c1(NC(C2(CC#C)CCCO2)=O)cccn(-c2ccccn2)c1=O Cc1nc(C(=O)NCCC(C)NC(c2nc(=N)cc[nH]2)=O)ccc1Br Cn1nc(C(=O)NCCOC2CCN(C(C3(Cl)CC3(F)F)=O)C2)cc1O CCCCC(C(=O)N1CCC(N(C)C(c2ccc(CO)nc2)=O)C1)ON=C(C)C N(C(=NCc1ccc(Nc2ccncc2)cc1)NCC1CCC1)C1C(C)(C)C1 C1(C(=O)NCCOC(C)C)(CN(C)C)CC12CCC2.N12CCCC1NC(=O)C2 c1(C(N(CCCN(C(C(C(C)C)O)=O)C)C)=O)cc(C(F)(F)F)cnc1N Cn1cc(C(N2CC3CC3(CNC(C3(CC4CC4)CCCO3)=O)C2)=O)c(CO)n1 N#CC1(C(=O)NC2CC(NC(C3CCCCC3)=O)C23CCC3)CC2CCC1CC2 c1(C(=O)O)ccc(CN2CC(O)CC2NC(c2ccccc2C(F)F)=O)c(F)c1 N1(C(C=C(CCC)C)=O)CC(NC(c2cc(C(C)C)on2)=O)C2(CCOCC2)C1 c1(C(=O)NC2CC(C)CN(C(=O)CN(C)C)C2)cc(Br)cn2ccnc12 C(=O)(CCCC(=O)NCC(CC)NC(c1cnc(O)c(Br)c1)=O)OCC c1(C(N)=O)ccc(C(=O)NC2C(C)C2)cc1.c12cn(nn1)CC1(CC1)N2.C1CC1 c1(C(=O)NC2(CC)CCN(C(c3cccnc3)=O)C2)csc2cccc(OC)c12 c1(C(C)C)cc(F)ccc1C(C(N1C(C)CCCC1C)=O)C CC1(C)CCOC(C(=O)NCC#CC(=O)NC(c2ccccc2)(C)C)C1 C1(N(C(=O)CC2CCCC2)CC)CCCN(C(=O)C(F)n2ccnc2)CC1 c1(C(=O)NCC2(NC(C=CCC)=O)CC2)cccn2ncnc12 c1(SC)ccccc1C(=O)NC1CCCC(NC(=O)CCCN(C)C(=O)C2CC2)C1 c1(COC)nc(OC)cc(N2CCC(C)(NC(C3CCCCN3C)=O)CC2)n1 C#Cc1ccc(F)c(C(=O)NCC2CC2NC(C2(Cl)CC2(C)C)=O)c1 c1(C(N2CC(CC)CC(NCc3ccc(F)cc3)C2)=O)cc(F)c(F)cc1O C1(CNC(c2ccn(CC)n2)=O)CC2COCC2N1C(=O)CCN1CCCCC1 C1(CC)CCOCCN1C(C1CCCN(CCOC)C1)=O.c1(N)ccc(O)cc1 C1(C(=O)NC2CN(C3C(CC(=O)N(CCC)CCC)C3)C2)CC(OC)(OC)C1 CC1C(NC(=O)Cc2cnnn2C)CCCN1Cc1cc(Cl)ccc1Cl Cc1ccc2c(c1)CCC2Nc1conc1C1CCCC1 C1(C(=O)NCC2OCCN(C(CCN(CCCCC)C)=O)C2)C(C2CC2)C1(F)F C(=O)(N=S(C)(=O)N(C)C)c1nc(CC(C)C)oc1-c1ccc(-c2nn[nH]n2)cc1 C1(C(=O)NC2C(CCOC)C2)CCN(C(=O)Cn2cncn2)C1C C(C(=O)NC1CC(CCNC(=O)C=Cc2ccccc2)C1)(C(C)C)OCC CCS(=O)(=O)C=CC(=O)N1CCC(C)C(NC(=O)CCOCc2ccccc2)C1 c1(OCCOC)cncc(C(=O)NCc2ccc(NC(C3CC3(C)C)=O)cc2)c1 N1(C(C(C(C)C)NC(=O)CNC(=O)C2CC2)=O)CCCC(O)(C2CC2)C1 c1(CCC)cc(C(C(=O)NCCSC)N(CCC(=O)NCC)C)ccc1C c1(C(N(C)C)=O)ccoc1-c1nc(C(C(F)(F)F)C2CC2)no1 CC(=Cn1ccnn1)C(=O)N(CCCNC(C1CC2(CC2)CO1)=O)C S(=O)(=O)(c1ccnc(NC(c2ccc3c(c2)CNC3)=O)c1)N(C)C N1(C(C=CC(C)C)=O)CC2C(C(=O)NCCn3cc(-c4ccccc4)nn3)C2C1 C1(NC(c2cc(C)ncn2)=O)CCSC12CN(C(c1cccnc1C1CC1)=O)C2 C1(CCC)(NC(C)=O)CCCN(C(c2cnn(C3CCOCC3)c2)=O)C1 N1(C(c2nnsc2CCl)C(=O)NCCCOC)CCC(F)(c2ccccc2)CC1 C(C(C)C(=O)N1CCC(N2CC=CC2)C1)NC(C=CCN(C)CC)=O N1(C(C2(C)CCCOC2)=O)CCN(C(=O)Cn2cccc(O)c2=O)C2(CCC2)C1 N1(C(C=CC(=O)OCC)=O)CCC(C)(C(=O)NC2CC(CCNC(C)=O)C2)C1 c1(COC)nc(C)c(C(=O)NCC2C3CC2N(C(c2c[nH]c(=NC)s2)=O)C3)s1 c1(C(=O)N)cc([N+](=O)[O-])cc(Cl)c1Cl.CC1(C)OC(C(=O)NC2(C)CC2)C(C)(C)O1 c1(-c2nc(-c3cnc(C(=O)C4CC4)s3)on2)cccn(C(F)(F)F)c1=O N1(C(C2CCN(C)CC2)=O)CCCCC2(CCN(C(=O)CC3(C4CC4)CC3)C2)C1 c1(-c2nccc(NCc3nc(C)sc3)c2)cncc(C#N)c1 C(=O)(CCN=c1[nH]cc(-c2ccc(C)cc2)s1)Nc1cc(Br)ccc1C.c1(SC)ccccc1 CCC(C)CC(=O)NC(CCC1CC1)C(=O)N1CCS(=O)C1C c1(C(C)NC(CN(CCOC)C(c2cc(OC)no2)=O)=O)cccnc1O C(C1CCCCC1)=CC(=O)NC1CC(C2CC2)(CNC(CN(C)C2CC2)=O)C1 N1(C(c2c(OC)n(C)nc2)=O)CC2CC(NC(c3c(C)nn(C)c3N)=O)CC1C2 C1(CCOC)(NC(=O)CC(C)O)CCN(C(=O)CCSc2ccccc2)CC1 C=CC(C)CC(=O)NC(C(=O)NCCC(C)(C)F)C1(O)CCC1 c1(NC(C(C)NC(c2cc(OCC)ncc2)=O)C(C)C)cc(C)c([N+](=O)[O-])cn1 N1(C(COC(C)C)=O)CCN(CCCCCNC(c2scnc2C2CC2)=O)CC1 N1(C(Cn2c(C)c(Br)cn2)=O)CC(C)(C)CC1CNC(=O)C(C)C c1(C(N(CCNC(=O)CC2(c3ccc(Cl)s3)CC2)C2CC2)=O)csc2cnccc12 CC1(C(=O)NCCNC(=O)CC(c2ccccc2)NC(=O)C(F)(F)F)CCCO1 N1(C(C2C(C)=CCC=C2)=O)CCN(C(c2ccc(Cl)cc2)=O)C(C(F)(F)F)C1 C1(NC(C2(C(=O)OCC)CC=CC2)=O)COC2C(NC(=O)CN(C)C)COC12 c1(CC)ccsc1C(N1CCC(c2n[nH]cc2CNC(=O)C=CBr)C1)=O C12(C(N3CCC(CC(=O)NCCCSC)C3)=O)CC3CC(CC(C3)C1)C2 C12(NC(C3CN(C)C(=O)C3)=O)CCC(C(=O)NOCc3cccnc3)(CC1)C2 N1(CC)CCN(C(=O)C(C)N(C(c2cn3c(n2)CCC3)=O)CC)CC1C N1(C(C2CCCC3(CCOC3)O2)=O)CCOC2(CCCN(C(=O)CCCF)C2)C1 c1(N2C(C)CC(NC(=O)CCCn3ccccc3=O)C2)ncnc2sccc12 c1(CN(c2ccc(C#N)nc2)C)cccc2c1S(=O)(=O)CCC2 N1(C(c2cc(OC)oc2)=O)CCC2(CC1)CN(C(=O)CC13CC(C1)C3)CC(C)O2 Cc1cccnc1CNC(=O)C(C)N(C(c1c[nH]c(C)c1)=O)C1CC1 CC(CC(F)(F)F)C(=O)NCC(C)N(C)C(C1CC2(CCCC2)C1)=O CC1CCCC=C1C(=O)N1CCOCC(CNC(c2cccc3c[nH]nc23)=O)C1 CS(=O)(=O)c1cncc(-c2ccc(C(=O)N(CC(F)(F)F)CCO)nc2C)c1 c1(OC)ccc(C)c(C(=O)NCCC23CCC(C2)N(C(=O)CNC(C)=O)C3)c1 c1(C(N(CCC(C)NC(C(C(C)C)SCC)=O)C)=O)cc2cc(C)ccc2o1 C1(C(=O)NCC#CC(F)(F)F)CC(O)CCN1C(C1CCC2CC1CO2)=O Nc1ccc(-n2cc(-c3cnn(C4CCC4)c3)nn2)cc1.C12CSCCN1C2=O C1(N(C)C(c2cncs2)=O)CC2CC1N(C(=O)C(c1ccccc1F)(C)F)C2 CC(C)(C(=O)NC1CCC(CNC(C2CC3CC3C2)=O)C1)c1cccs1 N1(C(c2ccc(C#N)nc2)=O)CCOC2(CCN(C(c3cnc(Br)s3)=O)CC2)C1 c1(C(N2CCCCC(N3CC(c4n(C)cnn4)C3)C2)=O)cccc2ccoc12 N1(CCNC(c2c(CC)cns2)=O)CCCN(C(c2cncc(C)c2Cl)=O)CC1 N1(C(C=C(C)C(F)F)=O)CCC(C(C)(O)CNC(=O)CC2CC=CCC2)CC1 c1(C(=O)NC(CNC(CC=CC=C)=O)C(C)C)cc(C)ccc1Cl C1(C(=O)NC2CC(C)(NC(c3nc(CC)oc3C)=O)C2)CCN(CCO)C(=O)C1 CN=c1ccc(C(N2CC(F)CC2CN(C)C(c2ccoc2C)=O)=O)c[nH]1 N1(C(CCC)C(C)C)CCCC(O)(Cc2nc(-c3cc(F)c(Cl)cc3Cl)no2)CC1 C1(CCNC(CNC(C)=O)=O)CCCCN1C(=O)C=Cc1ncc(C)[nH]1 C1(C(N2CC(N(C(=O)Cn3ccccc3=O)C)C2)=O)CCC(C2CCC2)CC1 c1(OC)cccc2c(N3C4CN(Cc5cc(C)c(Cl)c(C)c5)CC34)ncnc12 N1(C(Cc2n(C)cnn2)=O)CCCCC(NC(=O)CCn2ncn(C)c2=O)C1 C(=O)(C1=CNC2=NCCC2=C1)N1C(C)C(NC(=O)CC2CC2(Cl)Cl)CCC1 CC(CCCNC(=O)C(O)CF)NC(=O)CN1CCCCC1 N1(C(c2c(CC)ncs2)=O)Cc2n[nH]cc2C1C(=O)N1CCC(CCOC)C1 C(C(C)(C)C(=O)NCCC(C)N(C(=O)Cn1cnnn1)C)OCC CC1(C)CN(C(c2cnc[nH]2)=O)CCN(C(c2ncoc2Br)=O)C1 c1(C(N2CCN(C(C3CCc4c[nH]nc4C3)=O)CC2)=O)ccc2cccnc2n1 c1(NC(CC2(OC)CN(C(C3CCCN3C(N)=O)=O)C2)=O)ccc(F)cc1O c1(C(N(CCCN(C)C(C2CCCC2(F)F)=O)C)=O)ccc(C2CC2)nc1 C(CCN=C(NCC1=NOC2CCCC12)N1CCCC(CC=C(C)C)C1)OC N1(C(C2C3CC2N(C(c2cn(C4CC4)nn2)=O)C3)=O)CCc2ncccc2C1 C1(NC(c2n(CC=C)ccc2)=O)CCCC12CN(C(=O)C(F)CC(C)C)C2 Cn1cc(C(N2CCC(CCNC(c3ccc(O)cn3)=O)CC2)=O)c(O)nc1=O N1(C(C(CCC)OC)C(=O)NC(C)(C)C)CC2C(C1)C2(F)F C1(NC(c2scc(C)c2)=O)CCN(C(C2CCCC23CC3)=O)C(C)C1 c1(CCC(=O)NCCC(C)N(C(=O)C2=NNC(=O)CC2)C)ccc(C#N)cc1F CC1CCC(Cl)=C(C(=O)NC23CC(C2)N(C(c2ccc4nnnn4c2)=O)C3)C1 CCC(C(=O)OC)C(=O)NCC1C(C)CCN1C(c1cc(Cl)ccc1F)=O c1(C(C)C(=O)NC2CN(C(=O)CC3(O)CCOC3)C2)ccc(F)cc1 N1(C(C(F)OC)=O)CC2C(NC(c3ccc(C(C)(C)C)cc3)=O)CS(=O)(=O)C2C1 c1(C(C)NC(C(=O)N(C)Cc2nnc(C(=O)OCC)s2)=O)ccc(C)cc1F c1(C(=O)NC2COCC2NC(C2(C3CC3)CCC2)=O)cccc2sccc12 Cc1noc(C)c1C(C(=O)Nc1ccccc1)N(C1CC(C(N)=O)C1)C Cc1ccsc1COC(C1(c2ncccn2)CCOC1)=O C#Cc1ccc(C(=O)NCc2ccnc(C(=O)NC(C)(C)CO)c2)nc1 c1(CN(CC)CC)ccc(-c2ccc(Nc3cccc(O)c3)nc2)cc1 c1(C(N2C(C)CC(CC(=O)NCC(C=C)(C)C)C2)=O)c(C)nn(C)c1N C1(CNC(C(C)(F)F)=O)COC(C(F)(F)F)CN1C(C1CCCC1)=O c1(CC(=O)OCC)ccc2c(c1)CC(C)O2.C12CCCC1=NC1=NNC(CC)C1N2 N1(c2nnc(-c3n(C)ccn3)n2CC2CCCCO2)CCOC2(CCCC2)C1 c1(C(N(C2CCN(C(c3cccc(NC(C)=O)c3)=O)C2)C)=O)nc(C)ccc1C c1(-c2cn(CCCCCCNC(CC3C=NN(C)C3=O)=O)nn2)cc(Cl)ccc1F C(CCN=C(NCc1nnn(C)n1)NCC(O)Cc1ccccc1)OC(C)C N1(C(C2CCC(C)(CC)O2)=O)CC2(CC(CNC(c3cnc(C)[nH]3)=O)C2)C1 Cn1c(C(N2CCCCC2CCNC(C2CC(=O)NC2(C)C)=O)=O)cccc1=O C1(NC(C2(C)C(C)CCC2)=O)CCC2CN(Cc3ccncc3Cl)CC2C1 C1(C(N2CCCC(CNC(CCCOC(C)=O)=O)C2)=O)Cc2nn(C)cc2C(=O)N1 Cc1cccn2ncc(C(N3CCC4C(C3)CN4C(=O)C(=O)NCC3CC3)=O)c12 c1(C(=O)NC(C2(O)CN(C(C3COC3)=O)C2)C)cc(C(C)(F)F)ccc1C C(=O)(C(COC)NC(=O)CSc1ccccc1)NCCCN(CCCC)C C1(c2cn(CCC(=O)NCc3ccc(CO)o3)nn2)(COC)CCOC1 C(=O)(CCCCCN(C(=O)C=CC(=O)NC1CC1)C)N1CCC(C(CC)=O)C1 N1(C(c2cn(CCC)nc2C)=O)CC2CC1CN2C(C)(C)C C(=O)(C(C)(C)C(F)F)NCC1CCC(NC(c2c(C)[nH]cc2)=O)C1 C(CCCN=c1ccnc(N2CCOC(c3ccc(Cl)cc3)C2)[nH]1)OC C1(CNC(C2C=CC=CC=C2)=O)CCCCN(C(C2CCOC2C(F)(F)F)=O)C1 c1(NC(C(C2CCCN(C(COCCC#C)=O)C2)C)=O)cc(C)ccc1O CC1=CC(C)=NS(=O)(=O)N1CC(=O)NC1CCN(C(=O)CCn2ccnc2C)C1 C1(C(=O)NC2C(OC)CC2)(CCOC)CCN(C(=O)CCc2csnn2)CC1 C1(SC)CCCC1C(=O)N(CCNC(=O)Cc1csc(=N)[nH]1)CC1CC1 c1(Nc2c(O)cccc2O)cn2ccccc2n1.O=C1C(F)(F)CN1 c1(CC)csc2c1CCOC2.c12c(C)nn(c1C)-c1ccc(F)cc1-c1nccn1-2 c1(OC)cc(CC(C(=O)NNC(C)=O)NC(=O)Nc2ccco2)ccc1C C1(C(N2CCC(C)(NC(c3c(C)ccnc3)=O)C2)=O)CCC(C)C(C)C1 C12(C(=O)NCC(CC)(C)C)CCC(CC1)N(C(=O)C(C)C1CCC1)C2 C1(NC(CC2CCCN(C)C2)=O)CCS(=O)(=O)C12CN(C(C1CC1F)=O)C2 Cc1nn(C)c(Cl)c1CC(=O)NC1CCCCC1CNC(=O)CCC1CCOC1 c1(OC)cc(C(N2C(C)CN(C(=O)C(O)CSC)CC2C)=O)c2occc2c1 C12(CNC(C3CCS3(=O)=O)=O)CCCC1N(C(=O)CSCCC(F)(F)F)CCC2 c1(C(N2CCCN(C(C(CC#C)O)=O)CC2C)=O)cc2cc(C)cc(Br)c2o1 C1(CN(C(=O)C(C#N)C2CC2)C)C2CN(C(c3ncn(C)n3)=O)CC12 Cc1cc(NC2CC2C(F)(F)F)[nH]c(=NCC(C)Cn2cccn2)n1 N1(C(c2cnoc2C2CC2)=O)CCN(C(=O)CCc2cocn2)C(CCO)C1 N1(C(C2C(=C)CC2)=O)CCN(C(c2cc(C3CC3)on2)=O)CCC1C c1(SCC)ccc(-c2nc(-c3cc(Cl)ccn3)nn2C(C)C(F)(F)F)cc1 c1(C(=O)NCC(C(=O)N(C2(CO)CC2)C)CC2CC2)cc2n(n1)CCO2 c1(C(N2CC(O)(C(=O)NCCc3n(C)ncc3)C2)=O)ccccc1C1CC1 C(=O)(CC(C)C(C)(C)NC(=O)C(C)C1(O)CCC1)NCc1c(CC)nco1 c1(CCCC)nc(CN2CCCCC2C(N2CC(F)CC2CNC)=O)c(Cl)[nH]1 Cc1nc2cncc(C(=O)NCC(C(C)C)NC(=O)C(F)OC(F)(F)F)c2[nH]1 c1(C(N2CCC(CN(C(C(C)S(C)(=O)=O)=O)C)C2)=O)c2ccccc2nn1C c1(C(=O)NC2(CC=C)CN(C(=O)CSCC3CCCCO3)C2)cc(C)sc1C n1(CCOCC=C)c(N(C2CC(c3cccc(Cl)c3)C2)C)nnc1-c1ncoc1C C12(C(=O)NC(C3CCCC3)CNC(C34CCCCC3C4)=O)CCCN(CCC1)C2 C1(NC(CC#C)=O)CC(O)(CNC(=O)CC2(C)CCC2)C1 C(CCCCC(=O)N1CCCC1C(C)(C)C(=O)NCCCN(C)C(C)C)OC c1(CNCC23C(CN(C(C(n4ncc(C)c4)C)=O)C2)C3)cc(O)ccc1Cl c1(C(C(=O)NCCSC)N(C(C)C(=O)OC)C)nn(C(C)C)cc1Br Cn1nccc1C=CC(=O)NCC1(CNC(C2C=CCC2)=O)CC1(F)F N1(C(Cc2ccn(CC)n2)=O)CCC(C(N2CC3C=CC3C2)=O)C1C(C)C C=C1CCC(C(=O)NCCCCN(C)C(C2(CC#C)CCCO2)=O)CC1 C1(NC(COc2c(OC)cccc2)=O)CN(CC(=O)N(C)C(C)C)CC12CCC2 C(=O)(CCCC(C)(C)C)NC(C1(O)CCN(C(C2(CC)CC(C)(C)C2)=O)C1)C c1(COCC(=O)N(C2CCN(C(=O)C(F)=CC3CC3)C2)C)cccc(CC#N)c1 Cn1ncc(CNC(=O)CC2NC(=O)NC2=O)c1C(=O)NC(CC1CCC1)CO C1(C(=O)NC)CCN(C(c2cc(C(F)(F)F)ccn2)=O)C1c1ccccc1 C(c1ccc(Cl)c(C)c1)=CC(=O)NCC(CNC(C1CC2CCCCC12)=O)OC C12(CC(=O)NCCN(C(C3(c4ccccc4)CC3)=O)CC)COC(C)(C1)C2 C1(C(=O)NC(CNC(=O)C=Cc2ncc[nH]2)C2CCC2)CCc2nnnn2C1 C1(CC(=O)NCCOCCC(=O)NCc2c(OC)nsc2)CCCNC1=O C(=O)(C(C)(C)CNC(=O)C(c1nccn1COC)N(c1ccccc1)C)NCC N1(C(C2(CC=C)CC2)=O)CC2CC(C1)N(C(=O)C(C)CC(C)(C)C)C2 C(=O)(CCC(C)C)N(CC(N1C(C)(CCC)CC1)=O)CCOCC C1(C(C)NC(CNS(CC)(=O)=O)=O)CCCN(C(c2cnn(C3CC3)c2Cl)=O)C1 N1(C(c2c(CC)cc(N)cc2)=O)CCN(C(C2CC(SC)C2)=O)CCC1C C1(C(=O)NC2CN(C(C(c3cccc(OC)c3)O)=O)CC2C)CCN(OC)CC1 CCC(CC)C(C)C(=O)NCC1(C2CC2)CCN(C(c2nccc(Cl)c2O)=O)C1 c1(NC(C(N2CC(C#C)C(OC)C2)=O)=O)nc2cnccc2[nH]1 C(C(C)(C)C#CC(=O)N1CCC(CO)C(O)C1)NC(COC(CC)(C)C)=O C(=O)(C1=CCCCCC1)N1CCCC(NC(=O)CCn2cnnn2)C1 c1(CC)nc2c(C(=O)Nc3cc4nncn4cn3)ccnc2[nH]1 C1(CC)C(NC(c2ccc(CO)s2)=O)CCCN1C(=O)C=CC1CCOC1 C(=O)(CCCCCCCCCO)NCC1(CNC(=O)C=CC2CCCC2)CCC1 C1(C(N2CC(O)(c3nn[nH]n3)C2)=O)(CC)CCCN1C(C12CSCC1C2)=O N1(C(C(C)S(N)(=O)=O)=O)CC2(C1)CN(C(=O)Cc1ccccc1[N+](=O)[O-])CCO2 N1(C(c2cnc(C(C)O)s2)=O)CC2(C1)CN(C(C1(CC3CCC3)CC1)=O)C2 N(C(=NCC(C)C)NC1CCOc2ccccc21)C(CC(C)=O)C(C)(C)C C1(C2CC2)(CNC(c2ccnc(CO)c2)=O)CCN(C(=O)C(=O)C(F)(F)F)C1 N1(C(=O)Nc2cc(C)c(Oc3ccccn3)cc2)CCOC(C)(C#N)C1 c1(OC)cccc(O)c1C(=O)NC1CCC(CNC(=O)C(O)CCN(C)C)C1 C(=O)(CCC(C(C)C)NC(=O)C(C)CC(N)=O)Nc1c(OC)ccnc1 C#CCC(C)(C)C(=O)NC(C)(C)COCCCNC(C1C2CCC(F)(F)C12)=O CC1(NC(=O)C2CC2)CCN(C(C23CCC(CO2)C3)=O)CC1 C1(CCCC)CCC(NC(=O)CCN(C(=O)CC2CCCN2CC)C(C)C)C1 c1(C(N2CCC(CCOCC)C2)C(=O)NCC=C)nc(Cl)cc(Cl)c1C c1(C(N2CCC(O)(C(C)NC(c3cc(C)[nH]n3)=O)C2)=O)cccc2sncc12 C1(N(C(CN(C2CCCC2)C)=O)CCOCC2CCCCN2)CCS(=O)(=O)C1 CCC(O)(CC)CCNC(C1CC(C)(NC(C2OCCCO2)=O)C1)=O C1(C2CCOCC2)(NC(C(COC)C)=O)CC1.c1(C2C(=O)N2)cnn(C)c1 c1(C(N(CCCCNC(C2(O)CCSCC2)=O)C)=O)c(F)ccc2cnn(C)c12 CCC(CNC(=O)CC=CC(C)(C)C)(CC)NC(c1cc(CCNC)n(C)n1)=O C(C(C(C)(C)C)NC(=O)CCNc1ccc(Cl)cc1)NC(C1(N(C)C)CC1)=O C1(NC(C2OCCN(C)C2)=O)C2CC1CN(C(c1cc(F)ccc1C(F)F)=O)C2 C1(CC)CN(C(C2CC(O)CN2C(=O)C(C)C(F)(F)F)=O)CCN1C C(=O)(CCC(F)(F)C(=O)N1CCC(CNC(c2ncsc2C)=O)C12CC2)OCC n1(CCC(=O)NC(c2cc(C(=O)NCC(Cl)C(C)(F)F)no2)C)cnc(=N)[nH]1 c1(C(N2CC3(CN(C(C(C)=C4CC4)=O)C3)C2)=O)cc(C)c(C)c2ncccc12 C1(CC=C)(NC(=O)OC(C)(C)C)CCCN(N2CC(OCC=C)C(O)C2)C1 N1(C(CC)=O)CCC(C(=O)NCC(=O)Nc2cccc(C)c2)C(C)(C)C1 C#CC12CN(C1)C2=O.c1(CC(=O)N(CC(C)C)C(C)C)cncnc1 c1(OC)c(CNC(=NCC2COC(C)(C)O2)NCC2CCCO2)c(C)nn1C c1(C2(OC)CC2)ccn2ncnc2c1.C1(C)(C(C)C)C(=O)NC2CC3CC2N1C3 c1(C(=O)NCC(CNC(COC)=O)C)c(C(F)(F)Cl)n[nH]c1C C1(NC(C(c2ccccc2)SC)=O)C2CC1N(C(=O)CCCn1cccn1)C2C c1(C(=O)NCC2C3CN(C(C(C)(F)F)=O)CC32)cc(Br)c2cccnn12 C1(CNC(COCCCC#C)=O)CCN(C(C2CC2C(=O)OCC)=O)C1 C1(CNC(c2cnsc2)=O)CC2(CCOCC2)CN1C(c1cc(F)ccc1Cl)=O C12(C(N3CC(O)(C(C)NC(=O)CN4C(=O)CCC4=O)C3)=O)CCCC1CCN2 n1(CC)cc(CC(=O)NCCc2ocnc2CNC(C2CC(=O)N2)=O)nn1 Cn1cc(C=CC(=O)NCCC2CCN(C(=O)Cn3cnc(=N)[nH]3)C2)nn1 C1(CNC(c2c(C)scn2)=O)(NC(c2cnsn2)=O)CC2CCC1CC2 c1(N(C)C(C2CC2)C2CC2)cnc(NC(=O)CN)nc1.C(=O)(C(C)(C)Cl)NCC1CC1 CC1NC(=O)CCC1NC(=O)CC1(C)CCN1C(C1CSC1)=O C(=O)(CC(C)(C)C(C)(F)F)N1CCC(CNC(CCc2c(C)ncs2)=O)C(C)C1 N1(C(CCN(CCCCC)C)=O)CCCC2(C1)CN(C(C1CC(C)OC1=O)=O)C2 C1(OCC)CC(C(=O)OC)N(CC2CN(c3ccccc3)C(=O)O2)C1 C1(=CC(=O)NCCC2(OC)CN(C(=O)C(O)CN(C)C)C2)CCN(C)CC1 C1(c2n(CCCC)nnn2)(NCC2(n3cnnn3)CC2)CCSC1C C1(Sc2ccc(C(C3CC3C(=O)OC)=O)cc2)CCC2(CCOCC2)C1=O C1(NC(C2(C=C)CCC2)=O)CN(C(c2ccnc(SCC)c2)=O)CCC1CO Cc1ccc(NC(=O)CC2(C)CCN2C(c2ccc(O)cn2)=O)c(O)c1 C(CCCCCNC(C1SCCS1)=O)NC(c1c(CC)scn1)=O N1(C(C=C(CC)C)=O)CC2(CNC(=O)C=Cc3scnc3C)CCC1CC2 N1(c2cccc(S(=O)(=O)N(CC3(C)C(C)=CC3C)C)n2)CCc2c(C)cc(Br)cc2C1 C(CC(C)(C)C(=O)NC1CCCN(C(c2ccc(F)c(O)c2)=O)CC1)OC C1(C(=O)OC)CC(C)N1C(C1CCC1CCc1ccccc1)=O Cc1cc(C(=O)NC2CCCC2NC(C2NC(=O)OC2C)=O)n(C)n1 N1(C(C(CC)SC)=O)CCOC(C(C)NC(=O)CC2(O)CC2)C1 N1(C(C)(C)C)CCCC12CCCC2O.N12CSCC1NC2=O C12(CNC(c3[nH]cc(CC)c3)=O)CCCCC1N(C(=O)C(C)CCOC)CCC2 C(=O)(N=c1[nH]nc2[nH]ccnc1-2)c1ncc(-c2cc(F)cc(C)c2O)nc1 C1(C)(C(N2CCC(C)(C(=O)NCc3ncc[nH]3)C2)=O)C(C)(C)C1(C)C CC#CC1CN(C(C2(NC(=O)Cn3cc(C)cn3)CCSC2)=O)C1 C(c1cccc(Cl)c1Cl)=CC(=O)NCCCNC(C1CC2C=CC1O2)=O N1(C(C(CC=C)N(C)C)=O)CCC2(CCN(C(c3cccc4nc[nH]c34)=O)C2)C1 C12(NC(C3C4CCCCCCC34)=O)CCCC1N(c1cc(O)ncn1)CC2 Cc1cnc(N2CCC3(CCCO3)C2)c(S(=O)(=O)N2CC(c3nncs3)C2)c1 c1(NC)cccc(C(=O)N(CCCN(C(=O)CCCn2ccnn2)C)C)n1 c1(C(=O)NCC2CC3CN(c4nccc(CO)n4)CC23)cc2ccc(Cl)cc2o1 Cc1cccc2oc(N3CCC(CCNC(=O)C4=NNC(=O)C4)C3)nc12 C(CNC(=O)COC1CC1)(CC(=O)N1CCC(C(F)(F)F)C1)OC C(=O)(C(C)(C)C(F)(F)F)NC(CNC(c1cn(CC(CC)O)nn1)=O)CO C1(C(=O)NCC2(OC)CC2)CCC(CNC(=O)CNC(N)=O)CC1 C1(C(N2C(C3(N(C)C(C4CC(O)C4)=O)CC3)CCC2)=O)CCC(O)CN1C N1(C(CC2(C)OCCO2)=O)CC(NC(C2CCCC(O)C2)=O)CC2(CC2)C1 c1(CC(=O)NCCNC(C2CCC(C)(CC)O2)=O)c(F)cccc1Cl c1(CC(=O)NC(C2CCN(C(c3cocn3)=O)C2)C)ccc(F)cc1Cl N1(C(CN(CC(C)C)C(C2CC3CC3C2)=O)=O)CCCC(C(C)(C)O)C1 c1(C(N2CCC(NC(C3CCCC3)=O)C2)=O)cc(C(F)(F)F)ccn1 c1(N2C(CN(C)C(c3cnn(CC4CCC4)c3)=O)CCC2)ncc(I)cn1 N#Cc1cc(C(=O)NCC23CC2CN(C(c2cc(C(N)=O)cs2)=O)C3)cc(O)c1 CC(C)(C#N)CCCC(=O)NC1(CCNC(=O)CC2CCCC(O)C2)CC1 N1(C(C2CC(CC)C2)=O)CCC2CCN(C(=O)C=C(C)c3ccccc3Cl)C2C1 Cc1nn(C2CCC2)c(Cl)c1C(N1CCC(CCOC(C)(C)C)(NC(N)=O)C1)=O C(C1=CCN(C(=O)CC2CCC3CC23)CC1)NC(C1NC(=O)OC1)=O C#Cc1cccc(C(=O)NC(CN2CCN(C(=O)CN(C)C(N)=O)CC2)C)c1 N1(C(C(CC)O)=O)CCn2nc(C)c(CNC(c3cc(=O)n(C)o3)=O)c2C1 N1(CC(C)OC)CCC2CCC(C1)N2C(c1csc(C)n1)=O CC(C)CC(C(=O)N1CCCC(CNC(=O)CC(O)CN(C)C)C1)C(N)=O Cc1nc(CN2C3CCC2COC3)cc(=NCc2cc(F)cc3c2CCC3)[nH]1 N1(C(C(=O)NCCC2CC2)CC2CCCC(F)(F)C2)CC2(CCC2)c2ccccc21 CC1CN(C(=O)C(O)C(C)c2ccccc2F)CCN1C(c1cc(C(N)=O)no1)=O Cc1cc(O)ncc1C(=O)NC1CCN(C(=O)CC(C)C2=NN=NCC2)CC1F C1(NC(Cc2cnc(C)[nH]2)=O)CN(C(=O)CCc2cn(C)nn2)CCC1(C)C c1(C(=O)OC)cc2[nH]c(CC3CCCN(C(N4CC5CCC(C4)O5)=O)C3)cc2s1 C1(NC(=O)CNC(=O)C2CC2)CCN(C(c2occ3c2CCC3)=O)CC1CO N1(C(CC2CC(CC)OCC2)=O)CC2CC(C1)N2C(=O)C(C)(C)CN(C)C Cc1cc(CNC(=O)CC2CNC(C)CO2)c2ccccc2n1 C(C(CNC(=O)Cc1cc(C)nn1C)C(F)(F)F)NC(CCC(C)OCC)=O C=C1CC(C)(CNC(=O)CSc2nc[nH]n2)C1.C12COCC1C(=O)N2 C1(C2CCN(C(=O)CN3CCCCCC3=O)C2)(NC(C(=C(C)C2CC2)F)=O)CC1 c1(OC)ccc(C(N2CCC(C(C)C(N3CCCCCC3)=O)CC2)=O)c(Br)c1 C(=O)(C1=CCCC1(C)C)NCC1(F)CC(NC(C2CN(C(C)C)C(=O)C2)=O)C1 Cc1scnc1NC(=O)C(=O)NCC(C1CCCCO1)(C)O c1(C(=O)NC2CN(C(c3c(C)c(=O)cc[nH]3)=O)C(CO)C2)cc2nnn(C)c2s1 C1(CNC(c2cc(C(C)=O)[nH]n2)=O)CC(O)CN1C(c1ccc(C(N)=O)cc1)=O C(CC(C(=O)NC(c1cccc(Cl)c1)CNC(=O)CCSC)N1CCC1)SC C1(c2cccc(OC)c2)CN(C(=O)Cc2ccc(Cl)cn2)CCN1C(=O)CO C1(C(N(C(CCNC(CN(C(C)C)C)=O)C)C)=O)CCc2cc(F)ccc2O1 N1(C(C(CSC)NC(=O)CC(CN(C)C)C(F)F)=O)CCn2c(C)nnc2C1 O=C1CC(CC(=O)NC2COCC2NC(=O)C=Cc2ccoc2)c2ccccc2N1 C(C(CC(F)(F)F)NC(=O)C(F)F)NC(C1CN(C(CC)CC)C(=O)C1)=O O=C1NC(=O)C2(CC(C(N3CCN(C(c4csc(Cl)c4)=O)C4CC34)=O)C2)N1 C(CCC1CC1)(C(=O)NCC(F)(F)C(N)=O)NC(CCCSC)=O CC1CN(C(C2C3CN(C(=O)CCc4cccc(O)c4)CC23)=O)CCC1=O N1(C(CNC(CC)=O)=O)CCC2(CC1)C(OC)CC2NC(c1ncn(C)c1C)=O Clc1ccccc1-c1ccc(C2CCN(Cc3cc(C4CC4)no3)CC2)cc1 Cc1ccc2occ(C(=O)NC3CN(C(=O)CNS(N)(=O)=O)CC34CC4)c2c1 C(CN=c1nc(C#N)[nH]cc1Cl)=CCNC(C(CC)C(C)O)=O c1(C(N2CC(=C(CNC(c3c(CC)scc3)=O)F)C2)=O)ccn2c1CCCC2 c1(N2CC3C(C(N4CCC(c5ccccc5)C4)=O)(C3)C2)ncnc2n[nH]c(Br)c12 N1(C(c2ccc(C(C)=O)cc2)=O)CCC(CNC(=O)C(C)Cc2cnc[nH]2)C12CC2 N#Cc1ccccc1SCC(=O)NC12CCCN(C(C3CCCC3)=O)C1C2 c1(C(N(C(c2ccc(-c3ccccn3)s2)=O)CC)C)cccc(C(F)(F)F)c1Br C1(NC(C2C(C=C)CC2)=O)COC2C(NC(=O)CC(C)CNC(C)=O)COC12 CN1C(=O)CC2CN(C(C3CCCN3CC(F)(F)F)=O)CCC12 CCCCC(O)C(=O)N1CC(NC(=O)C(F)F)C(C(F)F)C1 C#CCC(C)(C(=O)NC1CC2C=CC1C2)Nc1ccc(F)c(CO)c1 C1(C#N)(CC)CCN(C(C2(C)CCC(C)C2(C)C)=O)CC1 N1(C(C2C(CC)CN(C(=O)C(C3(O)CCCC3)F)C2)=O)CCC(C2CCCC2)C1 Cc1ccc2cc(C(=O)NC3CC3CNC(=O)CN3CCOCC3)sc2c1 c1(NC(C(=O)NC2CCC(SC(C)(C)C)CC2)=O)ccc2ncsc2c1 C(=O)(CCCC(=O)NC1(C(=O)NCC2CCOC2C2CC2)CC1C)OC Cc1cc(CN2CC(C(C)NC(c3ccn(C4CCOCC4)n3)=O)C2)no1 c1(CCN2CCN(CC3CCC(C)(C)O3)CC2)cc(Cl)cc(Br)c1 C1(NC(CCCOCCOCC)=O)CCCC1(C)N(C(=O)COCC)C c1(C(N(C(c2cn(CCN3CCOCC3)nn2)C)C)=O)cnn2c1OCCCC2 C1(CNC(C(C)(C)OC(C)C)=O)CCCC(CNc2ccns2)C1 CCCC(C)(CCC)C(=O)N(CCCNC(=O)C(C)(O)C(F)(F)F)C C=C(C)CCCC(=O)NC1CC(C(=O)NCC(CC(C)C)OC)CC1O C(=O)(C1=CCC(C)(C)CC1)NCC1CC(NC(CC(=O)NCC#C)=O)C1 CCC(C)C(C)CNC(C1(C)CN(C(C2(n3cccn3)CC2)=O)C1)=O N1(C(c2c(C)nc(C)s2)=O)CC(=O)NCC1c1ccccc1 C12(CNC(C=C(C)Cl)=O)CCC(CN(C(=O)CCNC(=O)OC(C)(C)C)C1)C2 N1(C(c2cccc(SCCC)c2)=O)CCC(NC(=O)C(F)=C2CCC2)CC1C N1(c2c3ncn(C(CC#C)CO)c3ncn2)CC(C(N)=O)S(=O)(=O)C(C)(C)C1 C(=O)(C(F)C(C)CNC(c1ccc(O)cc1)=O)NCc1cc(OC)nn1C N1(C(COCC#C)=O)CC(NC(=O)C(F)C(F)(F)F)CC12CCC2 CN1CCCCC1CC(=O)N(C1(c2ccccc2)CCN(C(=O)C2CC2)C1)C1CC1 C1(NC(CCNC(=O)NC)=O)CCN(C(=O)COC)C12CC2 c1(C(=O)NCC2CN(C(C3(COC)CCOCC3)=O)CC2C)cc(N)cc(F)c1 N1(Cc2ccc(Cc3cccc(C#N)c3)cc2)C(=O)NC2(CCC2)C1=O c1(CC(=O)NC2CC(NC(C(Br)=C(C)C)=O)C(O)C2)cccc(C)c1C C1(C(=O)NC(C#C)CC2CCCC2)(CNC(C2C=CCC2)=O)CC12CCC2 C1(NC(C=COCC)=O)CCCN(C(c2ccc(-c3ccc(O)nn3)cc2)=O)C1 C(=O)(C(C)(C)C(O)C(C)C)NCCCCC(=O)N(CCCC)CCN(C)C N1(C(C(C(C)NC(=O)CCc2nc(=N)[nH][nH]2)C)=O)CC(C2=NOC(C)C2)C1 c1(C(N2C(CNC(=O)COC3CCCOC3)CCC2)=O)ccnc2[nH]nnc12 C1(CCOC)CN(C(=O)C(F)F)CCN1C(C12CC(CN1C1CC1)C2)=O N1(CC)CC(C(=O)NCc2cc(C(N3CC(CCO)C3)=O)n[nH]2)CC1=O c1(C(=O)NC(CC(C)Nc2cc(CC)ncn2)C)cccc2cnnn12 c1(CC(=O)NC2(C)CCN(C(CNC(=O)OCC)=O)C2)coc2ccc(C)cc12 N1(C(C(C)Cc2ccncc2)=O)CCOC(CNC(c2ccccc2CO)=O)C1 C(N=c1[nH]cnc2c(C(N)=O)cccc12)C1(C)CCCN(C(C(OC)OC)=O)C1 N1(C(C2(C)CC(=C)C2)=O)CC(N(C)C)C(CNC(=O)C(C)c2ccsc2)C1 C12(C(=O)NCC3N(C(c4c(Cl)cn(C)n4)=O)CC4(CC4)C3)CCCCC1OCC2 C1(CNC(CCC(=O)OC)=O)(NC(C2CCC(C(C)C)O2)=O)CC2CCC1CC2 C1(C)(COC)CC(NC(C2CCS(=O)(=O)N2)=O)CN1C(c1cn(C)nc1C)=O N1(C(CCOCCOCCCC#C)=O)CCN(C)C(NC(=O)C(O)CC(N)=O)C1 C1(CNC(C(CC#C)C)=O)CCN(C(=O)CCSCc2ccccc2)CC1(F)F C12(NC(c3csc(-c4ccccc4)c3)=O)CC1CN(C(C1CC1C(F)F)=O)C2 C1(C(C)C)(C(=O)N(C)CCN2CCCC2)COC1.C1=CCNC1=O c1(CNC(C=CCN(C(CCn2ccc(C)n2)=O)C)=O)ccc(C)c(C)n1 C(CCCC(=O)NCc1ccnnc1O)OCCC=C c1(CCCC(=O)N2CC(CO)C2=O)ccccc1Br.C=CCCC1CC1 C1(C(N2C(C)(C(=O)OC)CC2)=O)C2CCCC2CN1C(=O)Cc1ccon1 C1(CC)(NC(C2(CCNC(=O)C3=COCC3)CC2)=O)CCCCC1 Cn1c(C(N2CCC2CNC(=O)CSc2ccsc2[N+](=O)[O-])=O)ccc1C#N c1(C(N(CC(CN(C(=O)C(C)(C)n2cncn2)C)O)C)=O)n[nH]cc1C1CC1 N1(C(N2CC(C)(CC(=O)OC(C)(C)C)C2)=O)CCC(C)(NS(CC)(=O)=O)CC1 C(=O)(C1=CCOCC1)N(CCCCNC(CC1(CNC(C)=O)CCCCC1)=O)C C1(C(N2CC(F)(CNC(=O)CC3CNC(=O)O3)C2)=O)CCCC1C1CC1 C1(C(N(C2CN(C(=O)CCCc3ccncc3)C2)C)=O)CCS(=O)(=O)N1 C(N=c1[nH]c(NCC(c2ccccc2)C)nc2c1CCCC2)c1ncc(C)cn1 N1(C(C)CNC(c2cc(C)nn2C)=O)CCCCCC1.C12(C(=O)N)CSCC1C2 N1(C(c2c(OC)ccc(C)n2)=O)CC2CCCN(C(C3CC3C)=O)C2C1 CC1CCC(OCC(=O)NC(c2cn(-c3cccc(O)c3)nn2)C)CC1 C(C(C(=O)NCC1C2CCC(F)(F)C12)C(C)(C)C)NC(COCCC=C)=O C1(C(=O)NCC2N(CC(=O)OCC(=O)N(C)CC)CCC2)CN(C)CCO1 C1(C(=O)Nc2cnc(Cl)c(Cl)c2)CCc2nc(-c3cccc(O)n3)sc2C1 C12(C(=O)NC(CC(C)C)CNC(C34CCC(CC3)C4)=O)CCCC1CC(=O)C2 N1(C(C(CCC#C)NC(=O)C(C)CC=CCC)=O)Cc2cccc(F)c2C1 C(C)(C)(CC(C)(C)C)NC(C1CCN(C(CCC(C)CN(C)C)=O)C1C)=O c1(C(=O)NCC2CC(NC(=O)CC3(O)CCCCC3)C2)cc(=O)c2cc[nH]c2s1 c1(CC)cccc(C)c1NC(=O)C(c1ccoc1)N(C1CCSCC1)C C1(NC(C(C(C)C)OCC(C)C)=O)CN(Cc2cc(C(C)C)on2)CCC1C C(CC1=CCN(C(C2CC2C)=O)CC1)NC(C1N(C(C)=O)CC(O)C1)=O C(C(O)C(=O)N1CC(OCCNC(=O)C(COC(C)=O)N(C)C)C1)SC C(CC(CC)C(=O)NC(C(C(=O)CC(=O)Nc1c(N)cccc1)=O)C1CC1)=CC C1(C(=O)Nc2nc(O)cc(C(=O)NC)n2)CCCC2CCCCC12 C(=O)(C(C)C(O)CCC)NCCCN(C(C(F)=CC)=O)CC C1(NC(c2ccc(C)c(C)c2)C)CCc2nnnn2CC1 CC1CCC(CNC(c2coc(CO)c2)=O)CN1C(c1cncn1C)=O O=C(C#CC1CCC1)NCC12CC1CN(C(=O)CCC1CCC(C(F)(F)F)O1)C2 N1(C(c2c(C)ncs2)=O)CC2(CNC(=O)C(c3ccccc3Cl)(C)C)CC1CO2 C(N=c1[nH]c(=NC)[nH]c(=NCC(CSC)SC)[nH]1)c1ccc(OC)c(Cl)c1 C(=O)(C(=NOC)c1ccco1)NCC12C(CN(C(c3c(C#C)cccc3)=O)C1)C2 C1(NC(CC2(C)CC2(Cl)Cl)=O)CC2(C1)CC2C(=O)Nc1ccccc1 C1(NC(C=CCN(CC)CC)=O)(CF)CCN(C(=O)CS(=O)(=O)NC)C1 N1(C(C(CC)O)=O)CCC2CC2(C(N2CCC(C)(C3CC3)C2)=O)CC1 N1(C(c2cn(C3CCCCC3)nn2)=O)CCC2C(C1)CN2C(C1C2COCC12)=O C1(CNC(C=COCC)=O)CCCC(CNC(c2cnn(C3CCC3)c2)=O)C1 CC1(NC(C2CC3CC3C2)=O)CC(NC(c2ccsc2-c2nn[nH]n2)=O)C1 Cc1nc2c(C)cc(C(N3CCCC(CO)(NC(=O)CCCF)C3)=O)cn2n1 c1(CC)ccccc1NC(C1(CCNC(C2CCCC2O)=O)CC1)=O CC(C)(C(=O)N1CCCC1)C1=CCN(CC(=O)NC2C3CCC(F)(F)C23)C1 CCCC(CCC)CN=c1cc(C)[nH]c(=NCc2ccnc(C)c2)[nH]1 C(=O)(CC(C)C(F)F)NC(=O)C(F)(F)CC1CCC1.C(CCN)OC Cc1ccc(CN(CCC(=O)NC2CC(NC(=O)COC3CCC3)C2)C)c(C)c1 c1(NC(C2(CCCNC(C(CC=C)Cc3ccccc3)=O)CC2)=O)ccc(N)c(Cl)c1O N1(C(c2n(C)nc(Cl)c2)=O)CCN(C(=O)CC2(n3ccnc3)CC2)C2CC12 C(=O)(C1=CCC(C)CC1)Nc1ccc(NC(CSCCC(C)C)=O)cc1F c1(OC)ccc(OCC(=O)NC2CCC2CNC(=O)C(C(=O)OC)OC)cc1 C(=O)(C1=C(C)CCC1)NCCCN1CCC(C(=O)NCC(COC)O)C1 CCC(=O)NNC(=O)C(C)OC(=O)Cc1cnn(C)c1C C1(CCNC(CCC#C)=O)CCN(C(c2cccc(-n3nnnc3O)c2)=O)CC1 c1(C(=O)NCC(CCCC)NC(C(CC=C)NC(C)=O)=O)ccn2c1CCCC2 Cc1nnn(CC(=O)N(CCC(C)NC(C2(CO)COC2)=O)C)n1 c1(CC(=O)NCC(C)N(C(c2cc(C3CC3)nn2C)=O)CC)sc(O)nc1O C1(CC(=O)NCC(O)CNC(=O)CC(F)(F)F)NC(=O)CNC1=O c1(OC(C)C(N2CC3CCN(C(=O)COC4CCC4)C3C2)=O)c(F)cccc1F N1(C(CCOCCOC)=O)CC(NC(C2(NC(C)=O)CC2)=O)C(C)C1 S(=O)(=O)(c1ccc2oc(=O)ccc2c1)NC(C1(F)CCC1)C C1(C(=O)NC23CC(CNC(CSCC(=O)OC)=O)(C2)C3)CCN(C)C(=O)C1 C1(NC(c2nc(C)nn2C)=O)CCC2(CC1)CN(C(C1CC1F)=O)CCO2 n1(CC)cc(C(=O)NC2C=CCN(C(c3cc(OC)ns3)=O)C2)c(C)n1 Cc1ccc2onc(CC(N3CCC4CCN(C(=O)CO)CC34)=O)c2c1 C1(NC(CSC)=O)CC2CN(C(=O)CNS(=O)(=O)Cc3cnoc3C)CC2C1 n1(C(C=C)C)nc(-c2ccccc2Cl)nc1C1=NOC2OCCCC12 N1(C(CC2(C)CC2)=O)CCCC(NC(C2Cc3nncn3C2)=O)CCC1 N1(CC#C)CCN(C(=O)C(C)NC(C2CCC2CF)=O)CC1=O c1(C(N2CCCC(N(C(=O)COC3CCC3)CC)C2)=O)cc2ccncc2s1 c1(OC)ncc(C(=O)NCC2CN(C(C3COC3)=O)C2)cn1 N1(CC2C(C)CC2)CCC(Sc2ccc(CC(=O)O)cc2)CC1 C=C(C)c1cn(CCC2CN(C(=O)CCNC(=O)NC3CC3)C2)nn1 CCCS(=O)(=O)C1CCCC1N=c1[nH]c2c(c(=NCCC3CCCC3)[nH]1)CSC2 N1(c2nc(N(C)Cc3ccc(C#N)o3)nc3c2CSC3)CCC2(CCCOC2)C1 c1(C(=O)NCC(C)N(C(c2c(C)cc(SC)o2)=O)C)cc(C)cc(C)c1 C1(CNC(C2(C=C)CC2)=O)(NC(=O)CC2CCCOC2)CCC(F)(F)CC1 CCC(F)(F)CC(=O)N1CCCC1Cn1cc(CO)nn1.c1(N)ncncc1C C(=O)(C1=CCc2ccccc21)NC(CN(C(c1scc(C)c1C)=O)C)C N1(C(C(C)Cc2ccco2)=O)CC2COCC(C1)N2C(c1cc(C#N)c[nH]1)=O c1(CC)c(N2CC3C(NC(=O)CN4CCCCC4)C3C2)nc(C)nc1Cl c1(OC)cc(C(N2CCC(NC(=O)C3=CCC3)C(O)C2)=O)c(Cl)cn1 N1(C(=O)NCC(=O)NCc2ccc(C(C)=O)cc2)CC2(C(=O)O)CCC1C2 CC(CCN(C(=O)CSS(C)(=O)=O)C)NC(=O)NC1CN(C(N)=O)C1 CC1(C)CN(C(c2cc(-c3cccs3)on2)=O)CC(CNC(C2CCCO2)=O)O1 C(C(C(=O)NCC1CN(CC)C(=O)O1)C(C)C)NC(c1n(CC)nnn1)=O N1(C(C)C)CCC(C(=O)NC(C2CCCN(C(=O)C(=O)NCC3CC3)C2)C)CC1 n1(CC(=O)NC2CCN(CC(=O)Nc3cn(C4CCOC4)nn3)C2)cnc(Br)n1 c1(-n2c(-c3cc(SC)c(C)o3)nc(C3CC3)n2)cc(Cl)cc(Br)c1F C(=O)(C1(C)CCn2c(C)nnc21)NC1C2CN(C(CS(CC)=O)=O)CC1C2 C(c1ccc(F)c(Cl)c1)=CC(=O)NC1CCCC1NC(C1CSC1)=O c1(C(=O)NCCN(CCOCCO)C(C23CCCCC2C3)=O)nccn2ccnc12 c1(CC(=O)NCCN(C(=O)CC2COCCO2)C)csc(-c2ccsc2)n1 C1(C(C)(C)C)=NNC2=NC(C)(C)C1=NOC1(CCCCC1)NS2 N1(C(c2c(CNC(C3CCN(CC)C3)=O)ccs2)=O)C2CCCC1CN(C)C2 N1(C(C(CC#C)O)=O)CC(C2CCCN(C(c3ccc(C)c(C)c3Cl)=O)C2)C1 C1(OC)CN(C(=O)C2=COCC2)CC1C(=O)N(C(C(N)=O)C1CC1)C N1(CC#C)CCC(C(=O)NC2(CNC(=O)C(=C3CCCCC3)F)CCOC2)CC1 CC1(CNC(=O)CCC=O)COCCN(C(C2(C)CCCCOC2)=O)C1.C1(O)CC1 N12CCN(C)CC1C2.N1(C(C(C)n2cccn2)=O)CCC(N2CCC(O)C2)CC1 c1(OC)ncc(F)cc1C(=O)NCC1CC1NC(=O)Cc1ccc(C)cc1 N1(C(C(C2CC2)OCC)=O)CCC(C)(CNC(c2c[nH]nc2CC(F)(F)F)=O)C1 N1(C(CCCC(CC)CC)=O)CC23CCCC2(C1)CN(SC(=S)N(C)C)C3 N1(S(C)(=O)=O)CCCC(C(N2CCC(NC(=O)C(=Cc3c[nH]cn3)F)C2)=O)C1 N1(C(C(CSC)OC)=O)CC(C(N2CCC(C)=C(C)C2)=O)CCC1(C)C C1(CCC)(NC(C2CC23CCC3)=O)CCCN(C(c2cc(NC)ccc2Cl)=O)C1 C12(C(N3C(CNC(C(CSC)O)=O)CC(C)(C)C3)=O)CCC(C)(CC1)OC2(C)C Cc1[nH]c(C(=O)NC(C2CCCCC2)CNC(C2CCCCNC2=O)=O)c(C)c1C CCC(C)CCC(=O)N1CC(N(C(=O)CC2(C#N)CC2)C)C(O)C1 C(CCC(C)C)(C(=O)NCC1CCOC1C)NC(CC1(C(=C)F)CCC1)=O N1(C(CCC=CC)=O)CCC2(CC1)OCCC2NC(=O)C(C)NC(C1CCC1)=O CC1(C)CC(NC(c2c[nH]c(=S)cn2)=O)CN(C(=O)CNC=O)C1 C1(OCC)CCCN(C(=O)C(CCF)NC(=O)CC2CCSCC2)C1 Cc1ncc(C(=O)NC2CN(C(c3cnsc3)=O)CC2C)n1C(F)F C1(C(=O)NCCCCN(CCCNC(C=C(C)C(C)C)=O)C)CCN(C)C1 C1(C(=O)NCC2CCC(NC(c3ncn(C(C)(C)C)n3)=O)C2)CC(S(N)(=O)=O)C1 N1(C(C(C=C=C)C)=O)CC2(CC2)CC1CC(=O)NCC(c1cccs1)C Cn1c(C(=O)NC(C2CCCCC2)CNC(=O)C(O)Cc2ccco2)cc(Cl)c1Cl N1(C(C2C(OC)CC2)=O)CCC(C2CC2)(CNC(c2ccnn2CC(F)F)=O)C1 c1(C(=O)NC(CNC(C2(CC)CCC2)=O)C2CC2)snc2ccccc12 C(=O)(CCCC(=O)C(C)(C)C)NC1(NC(C(C)CCCc2ccccc2)=O)CC1 C(C(C)(O)CC(=O)N1CCC(Cn2cc(-c3ccc(Cl)cc3)nn2)C1)SC C1(C)(CNC(CC=CC=C)=O)CCCC1NC(=O)Cc1cccnc1F C=CCCCCC(C(=O)NCc1ccco1)N(C1COCCC1O)C CC1=CCC(C(=O)NCC2(C)CCCN2C(=O)C=Cc2cc(C)no2)CC1 c1(CC)nc(NCC(C2CC2)N(C(=O)Cc2cc(C)on2)C)c(C#N)cc1C N1(C(C(CCC)CNC(=O)C2=NNC(=O)C2)=O)CCC2(CC(CO)C2)C1 c1(C(N(C(C(N2CCCC2C2CCCC2)=O)C2CC2)C)=O)nnc(O)nc1O C1(OC)CC(C(=O)NCCC2CCCC23CC3)N(C(=O)C#CC2CC2)C1 C#Cc1ccnc(C(N2CCC(C=C)(C(=O)NC3CCCC3)C2)=O)c1 N1(C(c2c(C)cc(CC)o2)=O)CC=C(CC(=O)N2CC(OC)C(OC)C2)CC1 N1(OC)CCC(C(=O)OC)C2(CCC2)C1.C12CCC(C1)NC(=O)N2 C(C)(C)(CC(=O)N(CCCCC(C)C)C)NC(C1C(CC)OCC1)=O C1(CNC(C2(F)C(C)OCC2)=O)(NC(C2CCCCCC2)=O)CCCCC1C C#CCC(C)(C)CNc1ncc(OCC(C)C)cn1 C=CC(CC)CC(=O)NCC(=C1CCN(C(=O)CC2CC(C)(C)C2)CC1)F CN(C)S(=O)(=O)N1CCN(C(C2CCC(C(=O)NCC3CCOC3)CC2)=O)CC1 c1(C(=O)NCC(C)(C2CC2)NC(c2ncccn2)=O)cc(O)ccc1N Cc1ccc(Cl)c(C(N2CC(NC(c3n[nH]cc3C3CCC3)=O)CC2(C)C)=O)c1 C1(CC)OCCCC1C(=O)NCCCCCN(C(c1csc(C)c1N)=O)C(C)C C1(C(=O)NC2(CO)CCCN(C(c3c[nH]c(=NC)o3)=O)C2)CCC([N+](=O)[O-])CC1 C1(C)(CC)CCCN(C(C2(C)CCCN2C(C2CCCC(=O)CC2)=O)=O)C1 C(=O)(C1=NNC(=O)CC1)NC1C(C)CN(C(=O)CCSCc2ccccn2)CC1 CC(C(=O)NC(=O)C=CCNCC1CC1Cl)n1cncn1 CC(CC(=O)N1C(C(=O)NCCN(C)C)CCC1C1CC1)C(C)(C)C C1(C(N2CCC(CC(N3CC(CC(C)N(C)C)C3)=O)C2)=O)CCCCC(=O)C1 N1(C(C(CC)(F)F)=O)CCN(C(=O)CN2C(=O)CCC2=O)CC12CC2 c1(CCC(=O)NC2CCCC2NC(c2ccc(C(F)F)o2)=O)nnc(O)nc1O c1(C(N(C2CN(C(c3cn(C(F)F)cn3)=O)C2)C)=O)ccn(C)c1 c1(C(C(=O)N(CC(C)NC(=O)C(C)Cc2ccncc2)CC)C)ccc(C)cc1 C1(CNC(c2ccnc(C)n2)=O)CC2CCC(C1)N2C(=O)CC1CCS(=O)(=O)C1 Cc1ncc(CCC(=O)NC(C2CN(C(c3cc(Cl)cc(Cl)n3)=O)C2)C)c(O)n1 C(C(O)CC(=O)N1CC(O)(c2cc[nH]n2)C1)C(=O)Cc1ccsc1 C#Cc1ccccc1CNC(=O)CC(C)CNC(c1ccc(C(F)F)o1)=O CC1(C)C(=O)CC1C(=O)NCC1(C)CCCN1C(C12COCC1C2)=O C1(COC(C(C)CC2CCC(F)(F)CC2)=O)C(=O)Nc2ccccc2S1(=O)=O CC(CN(C)C)CCC(=O)N1CCC2C(C(=O)NCCC(=O)NCCO)C2C1 C1(NC(CC2CCC(=O)N2)=O)CCOC(C(=O)NCc2nncs2)C1 Cc1[nH]c(C)c(C(N2CC(CNC(C3CCCOC3c3ncc[nH]3)=O)C2)=O)c1C CN=S(C)(=O)c1cccc(C(=O)NCC(C)(C)NC(=O)CC2OCCC2(C)C)c1 c1(OC)ccc(CC(=O)NCCNC(c2cn(C)nc2CC(F)(F)F)=O)c(Cl)c1 N1(C(C2ON=C(C)C2)=O)CCCC(NC(C2(S(N)(=O)=O)CC2)=O)C1C C#Cc1cccc(C(=O)NCC2CC(C(=O)N(C3(CO)CC3)C)CO2)c1C CCCC(C)(CCC)C(=O)NC1(CNC(c2cnn(CCO)c2)=O)CCCCC1 C1(C(N(C)CC2CC2(C)C)=O)CC=CCN1C(c1cccnc1)=O C1(C(C)NC(c2c(C)snc2)=O)CCCN(C(=O)CC2CCN(C)CC2)C1 c1(N(CCNC(=O)CC2CCCCO2)CC)cc(C)cc(C)c1O C1(CNC(c2nc(NC(C)=O)sc2)=O)CN(C(=O)C=CCF)CCC1C C1(C(=O)NC(C(=O)OC)C2CCC2)CCC2(CC2)N1C(=O)C(C)N1CC(C)C1 N#Cc1ncc(C(N2CCOC(CCCNC(=O)CCNC(=O)CO)C2)=O)s1 c1(CCCC)cc(C(=O)NC(CNC(c2nnn(C)c2C)=O)CCOC)c(C)o1 C(=O)(C(O)C1=CCCCC1)NCCC(C(=O)NCCCC(C)OC)(C)C c1(N2CC(C(C)NC(=O)CC3COCCO3)C2)ccn2ccnc2n1 c1(C(N2C3C(NC(c4cc(C)[nH]c4)=O)C(CC3O)C2)=O)cc2ccc(Cl)cc2o1 C1(NC(Cc2cn(C)nc2)=O)CCN(C(c2nocc2C2CC2)=O)CCC1(F)F C(C(C)(O)C(=O)NCC(C1CC1)N(C)C(c1c[nH]nc1C(F)F)=O)OC c1(CCC(=O)NC(C(CO)NC(COC)=O)C)ccc(COCCC(C)C)cc1 c1(CCC)nc(C)c(C(N2CCCC2Cn2cc(COC(=O)C(C)O)nn2)=O)s1 C(C)(C1CCCCC1)=CC(=O)NCC(c1ccccc1)N(C(C=CCC)=O)C Cc1ncsc1CC(=O)NC(C1CC=CCC1)C(=O)NCCn1cc(Cl)cn1 C1(C2CCCCC2)(CNC(=O)NC2CCC(C(=O)OC)C2)CCCCC1 C1(OC)CN(C(=O)Cn2ncn(C)c2=O)CC1NC(c1ccc(Cl)o1)=O C1(n2cccn2)(NC(CCOCC)=O)CCN(C(=O)C(CCSC)OC)CC1 c1(CC)onc(C)c1CN1CCOC(c2ccc(NC)nc2)C1 C(C)CCCCCO.C(CC(=O)NCCOC)N(C(C)=O)C c1(SCC(=O)NCCC(CNC(=O)CC2CCOC2C)OC)ccc(C)cc1C C12(CCC)CN(C(=O)C(=O)NCc3ccc(C)c(O)c3F)CC(CO)(C1)C2 c1(C(N(C(CCNC(CC(C)C)=O)C)C)=O)cncc(-n2cccn2)n1 C(C)(C)(C(=O)NCC(C1CCC1)OC)SCCCC.c12ocnc1C(=O)NC2 N1(C(c2c(C)cco2)=O)CCN(C(=O)C2CC2)C(c2cn[nH]c2)C1 C1(C(N2CCCC(C)C2CCO)=O)CCC2CCC1N2C(=O)C=Cc1ccsc1 c1(C(=O)NC2CCC(NC(C3(C)CCN(C)C3=O)=O)CC2)cnc([N+](=O)[O-])n1C C1(C)(C=O)CCCN(C(=O)CSCC(N)=O)C1.C(=O)(C(C)(C)C)NCCCC C(C)(CN=c1[nH]cnc(Cl)c1Br)N(C(C(C)CCN(C)C)=O)C N1(C(C2C(CC)OCC2)=O)CCN(C(c2ccc(CO)s2)=O)CC12CCC2.C(C)(=O)N N1(C(C2(OC)CCC2)=O)CCC(CCNC(=O)C(F)=C(C)C2CC2)C1 C1(C(N(C)Cc2n(CC)ccn2)=O)CCCC(NC(=O)C(C)c2ccco2)C1 c1(C(=O)OC)cccc(S(=O)(=O)N(C)CC2CCN(C)C2)c1 c1(C(=O)NC23CCN(C(=O)Cc4cocn4)CC2C3)cnc2ccccn12 S(=O)(=O)(C1(CNC(c2cccc(C(C)(C)O)c2)=O)CCC1)NC(C)(C)C C(C(CC(=O)N(CC(C)(C)O)C)NC(c1csc(F)c1)=O)OC c1(N2CCC(C)(OC)C2)nc(N2CCC(CN(C)CC)C2)c2ccc(C)cc2n1 Cc1sc(O)nc1C(=O)NC(C(=O)NC(c1nc[nH]n1)C)c1ccco1 N1(c2c(C(=O)OC)cccn2)CCC2(CCCCN(C(c3n[nH]c(C)n3)=O)C2)C1 C(C(=O)N1CC(CNC(c2cccs2)=O)C(C(F)(F)F)C1)(C(C)(C)C)N(C)C c1(OC)cc(F)ccc1N1CCN(C(=O)Nc2ccc(CCN(C)C)cc2)CC1 c1(OC)ncnc(C(=O)NCC(F)CNC(c2cn(CCO)nc2C)=O)c1F N1(C(COc2cccc(C)c2)=O)CCC(NC(C2(C)CCCS2)=O)CC(O)C1 C12(CNC(CCC(C)C)=O)CC(CO1)N(C(=O)C(F)n1cccn1)C2 C1(C)(CNC(C2CN(C(C)C)C2)=O)CCN(C(c2c[nH]nc2-n2cnnn2)=O)C1 Cc1ccc(NC(=O)CNC(N2CCCCC2CN(C)C)=O)c(F)c1 Cn1cc([N+](=O)[O-])c(=NCCOCCNC(=O)C(C)(C)CF)[nH]1 C1(C(=O)NCC2(C)CCCN(CCn3ncccc3=O)C2)CN2CCCN1CC2 C(CC1=CCCCCC1)NC(C1CCC(C(C)C)N1C(C1CCC(=O)N1)=O)=O C12(CNC(C3C(=O)NCC3)=O)CN(C(c3ccncc3C3CC3)=O)CC1CCO2 C(=O)(C(O)CC(F)(F)F)N1CC(SC)C(NC(C23CC(C(C)(C)C)(C2)C3)=O)C1 c1(C(N(CC(C)N(C(=O)CC2CC(F)(F)C2)C2CC2)C)=O)ccc(O)c(F)c1F c1(C(N2C(CNC(C3CCNC(=O)C3)=O)CC(OC)C2)=O)ccc2c(c1)CCN2 Cc1ncc(NC(C2CCN2C(c2ccnc(F)c2Cl)=O)=O)cc1Br Cc1ccc(=N)[nH]c1C(N1CCC(C)(CNC(C2(C)CC=CCC2)=O)C1)=O c1(CNC(C2N(C(C(C)OC(C)C)=O)CCC=C2)=O)ccc(F)cc1F C=C(C)C(CC(=O)N(C1CCC(NC(C2CCC(F)(F)CC2)=O)C1)C)OCC N1(C(CCCC(=C)C)=O)CCC2CN(C(=O)CSCc3ccncc3)CCC2C1 CC(C)(C)C(CNC(c1cn[nH]c1)=O)C(=O)NCCC1CCCC12CC2 C1(C(N2CC(N(C(C3CC(OCC)C3)=O)C)C2)=O)COCCO1 C1(C(C)C)CN(C(c2ccc(-c3cn[nH]c3)cn2)=O)CCN1C(=O)C(C)C1CC1 C1(CCC)(NC(=O)C(c2ccccc2)C)CCCN(C(C2CC3CCC2O3)=O)C1 Cn1c(CN2CCC(CO)C(O)C2)nc2cc(Br)ccc12 N1(Cc2c(C)non2)CCC2(CN(C(c3cc(Cl)ccc3[N+](=O)[O-])=O)CC(C)O2)C1 n1(COC)ncc(CNC(C2CN(Cc3ccc(OC)cn3)CC2O)=O)c1F c1(C(=O)NCC2(C)CCN(C(C3CCCC4CC34)=O)C2)c(Cl)oc2ccccc12 CC1(NC(=O)CCc2nnc(C3CC3)o2)CCCN(C(c2coc(Br)c2)=O)C1 C1(OC)CC(CNC(=O)C(C)(C)c2ccn(C)n2)N(C(c2cnc(C#N)s2)=O)C1 N1(C(C2C(NC(CN3C(C)CCC3)=O)COC2)=O)CC2CCCC2C1 N1(C(c2ccc(C)o2)=O)CCn2c(C(=O)Nc3c(C)ccnc3Br)cnc2C1C N1(C(c2c(SC)ccc(N)c2)=O)CC2CC(NC(c3[nH]c(C)cc3C)=O)CC1C2 N(C(=NCCc1ccc(F)c(F)c1)NCC(F)F)C(CF)Cc1cccnc1 C=CC(CCC)CC(=O)NCCC1(CNC(C2Cc3ccccc3O2)=O)CC1 c1(SCC)conc1C(c1nnnn1C1CCCCC1)NC(=O)CO N1(C(c2c(C)n(CCO)cc2)=O)CCN(C(c2cncn2C)=O)C2CCC12 C1(O)(CNC(CC2(C)CC2(F)F)=O)CCCN(C(c2cnsc2)=O)CC1 N1(C(C2N(C)CC2)=O)CCCC1C(N1CCC(c2ncc[nH]2)C1)=O C(=O)(C(=O)N=S(C)(C)=O)NCC(C)(C)NC(C1CCCN1CC1CCCC1)=O C(C)(CC#C)(C(=O)N(C(C)CN(C)C)C)NC(COCCC#C)=O C1(NC(c2ccc(C)s2)=O)CC2CCC(C1)N2C(C1CCOCC1)=O C1(C2CCCCC2)(C(C)(C)C)CC1.c12ccnc(n1)NC(=O)NCCO2 c1(C(N2CC(OCC)C(CNC(=O)Cc3n[nH]c(=N)s3)C2)=O)cc(C#N)cn1C c1(CS(N2C(C(=O)NC(COC)CO)CCC2C)(=O)=O)ccc(F)cc1F c1(OC)ccc2[nH]cc(C(=O)NCC3COCCN3C(=O)CNC(=N)N)c2c1 c1(OC)ccc(Br)cc1C1(C(=O)NCCN(C(=O)C2=CCSC2)C)CC1 c1(N(C(=O)CN2CCOC2)C)ccc(Br)nc1[N+](=O)[O-] N1(C(C(C(C)C)SCC)=O)CCCCC2(C1)CN(C(c1cnn(C3CC3)c1)=O)C2 S(=O)(=O)(c1nccs1)NCCC1CCN(C(C2CCC(C3CC3)CC2)=O)CC1 N1(C(C(C)=CC=C)=O)C(C(=O)NC2(CO)CCC2)CCC1C(C)C c12ccc(c(C#N)c1)[nH]c2=O.C1(CN(C)C)CCC(OC(F)(F)F)C1 CN1CC(NC(=O)C(CC2CC2)NC(=O)CN2CSCC2=O)C2(CC2)C1=O c1(C(=O)NC2CC3C(NC(c4ccccc4)=O)C3C2)ccc(F)c(F)c1 C(=O)(C(=O)C(C)(C)C)N1CCCC(C(=O)Nc2c(C(C)C)nsc2)C1 N1(CC(=O)NC(CNC(CC(CC)C)=O)C(C)C)C(C)=CC(C)=NS1(=O)=O N1(C(CC)=O)CC(C2CCCN(C(=O)C=CCN(C)C)C2)C1 N(C(=NCCCF)NCc1ccccc1Cc1ccccc1)C(C)C c1(C(N2CCC3(C(NC(=O)C4CC4)CC3)CC2)=O)ccc2c(=O)ccoc2c1 C1(C(N(CC=C)CCN(C)C)=O)CCN(C(c2ccc(CC)s2)=O)C(C)C1 c1(C(=O)NC(CN(C(c2ccc(OCC(C)C)nc2)=O)C)C)ccc(F)cc1Cl Cc1nccc(N2CC3CC2(c2cccc(OC(F)(F)F)c2)C3)n1 CC1(NC(C2(CF)CC2)=O)CCCN(C(C23CCCC2(C(N)=O)C3)=O)C1 C1(NC(COCCC)=O)C2COCC1CN(C(C1CC3CC(=O)C1C3)=O)C2 N1(C(Cc2nc(C)oc2)=O)CC2(CCN(C(C3CCCCC3C(F)(F)F)=O)C2)C1 c1(C(=O)NC2C(C)CN(C(=O)C=CC(F)(F)F)CC2)ccc2nn[nH]c2n1 C1(NC(c2c(C(=O)OC)cc(Br)c(O)n2)=O)CC2(CCC(C)(C)CC2)C1 C(=O)(C1CNc2ccccc21)NCC1(c2ccc(C)cc2Br)CC1 CCC(CNC(=O)C(C(C)C)NC(=O)Cn1ccnn1)C(C)(F)F c1(OC)ccc(Cl)c(C)c1C(=O)NC1CC(CNC(C2(N(C)C)CCC2)=O)C1 c1(C(=O)NCC2C(C)CN(C(c3cscn3)=O)CC2)ccc(C#CC2CC2)cc1 C1(NC(CC(=O)NCC2CC2)=O)CCOC12CCN(C(=O)C=CI)CC2 c1(C(=O)NC2CCC(C)(NC(C(CC)O)=O)CC2)cn2cccc(F)c2n1 C1(NC(C(CC)(F)F)=O)CCN(C(c2ncc(OC(C)=O)cn2)=O)C12CC2 C1(NC(C(C)Cn2ccnc2)=O)CC1C1CCCN(C(=O)CC(C)(C)N(C)C)C1 N12CCCCC3(C1)CN(C3)C2=O.CC(C(C)C(=O)OC(C)(C)C)C(C)(C)C C1(NC(CC(=O)NCC#C)=O)CCCN(C(=O)CCc2nc(C(C)C)no2)C1C c1(NC(C(N2C(NCCOC)C(C)(C)CC2)=O)=O)ccnc2c1ncn2C C1(C(=O)NCCc2c(C)[nH]nc2O)CCCCCN1C(C1CCS(=O)CC1)=O C1(N(C(=O)COCC(F)(F)F)C)CCC2(CC1)CCN(C(=O)CC1C=CCC1)C2 C(=O)(C1=CCC(C(F)(F)F)OC1)NCCN(C(c1n(CC)ccc1)=O)C1CC1 C(CCC(=O)NCCN(CC(C)O)C(c1cnn(C(F)F)c1)=O)OC(C)C c1(C(N(C2CCCC(CNC(CN(C)C)=O)C2)C)=O)cncc2c1CCC2 Cc1c(C(=O)NC2CCN(c3nccc(C(C)(C)C)n3)C(C)C2)cncc1Cl C1(CNC(CC=C)=O)CC2(CO1)CN(C(=O)CCCC(OC)c1ccccc1)C2 c1(CCC(=O)NC2CN(C3(n4cc(Cl)cn4)CC3)C2)ncccn1 c1(CSC=CC(=O)NC2(CN(C(C3(F)C(C)C3)=O)C)CC2)cccc(Cl)c1 Cc1cc(OC(C)C(=O)NC2(NCC(=O)O)CC2)cc(C)c1.c12ccc(cc1)o2 C(CCCCCNC(C1C2CCCCC12)=O)NC(C1C(C)C1C)=O C1(C(=O)NC2(CNC(C3CC3C3CC3)=O)CC(OC)C2)CC2CCC1C2 C1(C(C2CC(CC(=O)O)OCC2)=O)CCC2C(=O)N(c3ccc(F)cc3)C(=O)N12 CC(C)C(C(C)NC(c1cc(C(N)=O)c[nH]1)=O)NC(=O)CS(=O)(=O)N(C)C c1(C(=O)NCCCN(C(=O)C(C)(F)C(=O)OC)CC)c(F)ccc(C)c1Cl C#CC1CN(C(C2CCCN2C=O)=O)CCN1C(=O)C=CCOCCOC c1(C(N2CCN(C(C=C3CCC(C)(C)CC3)=O)CC2)=O)noc2c1CCCCC2 c1(C(N(CCN(C(=O)CC2CC3(CC3)C2)C)C)=O)cnc(C(F)F)nc1 C(=O)(C(CO)C(C)(C)C)NC(C1CC(NC(CC(=C=C)C)=O)C1)C C1(C(CNC(=O)CNC(N)=O)NC(=O)C=CCO)CCCC1.C(CCO)N(C)C c1(C(C)C(=O)NCCCN(C(=O)C(C)CC(C)(F)F)C)cc2ccccc2o1 C1(CNC(C2C(=C)C2)=O)C(C2CC2)CCN1C(c1ccccc1C(C)(F)F)=O C(CC(C(C)(C)C)NC(C1CC=CC1)=O)N(C(C(C1(O)CCCCC1)CC)=O)C c1(C(N2CCCC(F)(CNC(c3ccc[nH]3)=O)C2)=O)coc2c(F)cc(Cl)cc12 c1(NC(c2nc(NC(=O)CCn3cncn3)sc2)=O)cccc(F)c1Br C12(C(=O)NC(C(=O)OC)(C)C)CCC(CC1)N(C(c1cc(O)ccc1F)=O)C2 C(C)(CCCCNC(=O)CN1CCN(C2CC2)C1=O)NC(c1cc(OC)no1)=O S(=O)(=O)(c1cncc(C(F)(F)F)c1)N1C(C(=O)NC(CSC)C)CCC1C c1(NC(C=CC(=O)NCCCCN(C(C2C(C(=O)OC)CC2)=O)C)=O)ccccn1 c1(CC(=O)NC(C)C(C)NC(c2nc(Cl)ccc2Cl)=O)ccc(Cl)c(Cl)c1 N12CCN(C3CC13)CCc1ccc(cc1)C2=O.C12(COCC=C)CC(C1)C2 C1(CN2CCCC(C)(C)C2)CCCN1NC(=O)C(=O)Oc1ccc(F)cc1 N1(C(C2(CC#C)CCCO2)=O)CC=C(C(=O)NC2CCCC(C3CC3)C2)CC1 N1(CC(=O)N(C(C2CCCC2)CNC(=O)C(O)CNS(C)(=O)=O)C)CCCC1=O c1(C(=O)NC(C)CCCNC(=O)C(O)CC(F)(F)F)ccc2ccccc2c1 c1(C(=O)NCCCCCN(C(=O)CC(C)(C)C(F)F)C)ccc2c(n1)CCO2 C(N=c1[nH]c2c(c(=NCC(C)CO)[nH]1)CCC2)c1c(C)nsc1 Cc1c(C(N2CC(NC(C34CC(F)(C3)C4)=O)C2)=O)cc(S(N)(=O)=O)cc1[N+](=O)[O-] c1(NC(c2c(O)ccc(C)c2)=O)ccc2c(c1)COC(=O)N2 CCC(CNC(=O)C=Cc1ccc[nH]1)(CC)C(=O)NC1CC1C N1(C(C(n2ccc(C)n2)C)=O)CCC(CNC(=O)CCc2cncnc2)C1C CC1CN(C)C(C)CN1C(=O)C1=CCN(C(=O)CCC2CCCN2C)C1 c1(C(N2CC(CNC(c3cc(C)sn3)=O)C(C)CC2)=O)ccc(C)c2c1CCC2 C1(CC(N2C(CN(C)C)CCC2)=O)(NC(=O)CSc2n[nH]c(O)n2)CCCCC1 N1(C(c2cn(CC)nn2)C(=O)NCCCC)CC(C2(O)CCC2)C12CCC2 CC1(C(N2CC(CCO)(C(=O)NCCc3cccnc3)C2)=O)CCCS1 c1(NC(C(C)N(C(C2(CC#C)CC2)=O)C2CC2)=O)cncnc1C N1(CC)CC(C(=O)NC2(CCNC(=O)CC3CCC(=O)N3)CCC2)CC1=O c1(OC(C(=O)N(CC(C)N(C(c2c(C)con2)=O)C)C)(C)C)ccc(Cl)cc1 c1(C(=O)NC2CCN(C(CCCNC(=O)OC)=O)C23CC3)cnc2nccn2c1 c1(OC)ncnc(Cl)c1NC(C1C2CC1N(C(=O)C=CCN1CCC1)C2)=O C1(C(NOCCC(=C)C)=O)(NC(c2csnc2Cl)=O)CC1(C)C C1(NC(C(CNC(C)=O)(C)C)=O)CCCN(C(=O)CC2C=CCC2)CC1 n1(CC(=O)NCC2CCN(C(C3(CC)CCOCC3)=O)C2)nnc2c1CCCC2 c1(CC(=O)NC2CN(C(C=CCOC)=O)CC(F)(F)C2)ccc2c(c1)CCCO2 CCCCCCC(C)C(=O)N1CCC2CCC(C1)N2C(=O)C(C)CCO C1(CNC(C=CC=CCC)=O)CCCN1C(c1cc(C)[nH]n1)=O CC1CCSCCN1C(=O)CCN(C(=O)CCn1cnnn1)CC1CC1 N1(C(C2(CF)CCN(C(CCCCCC)=O)C2)=O)CCC2(COC(=O)N2)C1 C(=O)(C#CC(C)(C)C)NC1C(CNC(c2[nH]cc(C(C)=O)c2C)=O)C1 C1(NC(c2c(Cl)cc(C)nc2)=O)CCN(C(c2nccs2)=O)C12CCCC2 CCC(C)CC(CO)NC(=O)Nc1csc(CNC(=O)C#CC(C)C)c1 C1(N(C(C2CN(C)C(=O)N2)=O)C)CN(C(=O)COc2cccc(O)c2)CC12CC2 c1(C2CC(C(=O)NCCN(C(CC(CC)C3CC3)=O)C)C2)ccc(F)cc1F c1(N(CCCC)C)ccc(C(=O)NCCC(C)N(C(=O)C(C)(C)COC)C)cc1 N1(C(c2occ(C)c2)=O)CCC(F)(CNC(C2CCCCN2C(N)=O)=O)CC1 C(=O)(C(O)C(C)(C)C)NCCCNCC(=O)N(C(C(CC)C#N)=O)C1CC1 c1(C(c2nnnn2C2CCCC2)NC2C(O)COC2)ccc(CC2CC2)cc1 C(=Cc1ccccc1)=CC(=O)NC(C(N1CC(C#CC)C1)=O)Cc1cn[nH]c1 N1(C(C2(CCNC(C(CC=C=C)COC(C)=O)=O)CC2)=O)CCC(O)C(F)(F)C1 C12(CNC(c3cnc(COC)s3)=O)CN(C(=O)C(F)C(C)(C)O)CC1CCO2 C(=O)(CCC(CC)NC1CC1)N1CC(SCC)C(C2(C(=O)N(C)OC)CC2)C1 CC1(C)CCC=C(C(=O)N2CCN(C(C3C(F)(F)C34CC4)=O)CCC2C)C1 c1(C(=O)NC(CNC(CC2C(C)CCC2)=O)C)c(F)c(F)cc(F)c1F c1(NCC(C)S(N)(=O)=O)cc(S(=O)(=O)NCC2(N(C)C)CCOC2)ccc1C#N C(c1cc(F)c(F)c(F)c1)=CC(=O)Nc1ccc(NC(=O)C2CC2)cc1.C1C(=O)N1 c1(CSCCN(C(C(F)OC)=O)CCCN(C)C)cccnc1.C(=O)(C1CC1)N C#CCCC(O)C(=O)NCCCN(CCC)C(C1CCCCC1c1nc[nH]n1)=O C#CC1(C(N2CCC(C=O)CC2)=O)CCCC1.c1(C(N(CC)C)=O)cn(C)nc1C C(=O)(C(C)CC(C)C)OCC.O1NC(=O)C(C)NC(=O)C1 c1(CNC(CC2CC(=O)NC2)=O)cccc(CNC(=O)Cc2ncc(Cl)s2)c1 c1(N2CCC(C(C)NC(CCCOCCOC)=O)C2)ncc2c(ncn2C)n1 N1(C(C(C(C)(C)C)O)=O)C2CCC1CN(C(C1OCCCO1)=O)CC2 C1(CNC(=O)COc2cn[nH]c2)CC2(CCC2)CN1C(C1C=CCCC1)=O c1(C(=O)OC)cc2c(cc1NC(=O)CSC1CCCC(OC)C1)CCC2 Cc1cnn(C(C)C(=O)NCCOCCNC(=O)CSc2cn[nH]c2)c1 N1(C(C(=O)NC(C)C)=O)CCC2CCN(C(=O)C=Cc3scnc3C)CC2C1 C12(NC(CCC(=O)NCC)=O)CC(CNC(C3(C)CC3(Cl)Cl)=O)(C1)OC2C c1(C(N2CCC(CN(C(C(C)c3ccco3)=O)C)CC2)=O)cc2n(n1)CCCN2 Cn1ncc2ncnc(NC3CC3C(=O)Nc3ccc(F)c(CO)c3)c12 CCCC(CC(=O)OC(C)(C)C)C(=O)N1CCC1Cn1cc(C2(C)CCCO2)nn1 C1(C(=O)NCC(CCCC)NC(=O)Cn2nnnc2C)CCCC(=O)NC1 C1(O)(CC(=O)NC(CCN(C(C2(C#C)CC2)=O)C)C)CCCC1 n1(CCC(=O)NC(CC)CN(C)C(C2COC2)=O)sc2ccccc2c1=O C1(N(C(=O)CC2CC2C2CC2)CCC)CCN(C(=O)C=CC=O)CC1.OCC c1(C(CCC)C)nc(-c2cncc(CO)c2)n(C2CC(C(=O)N(C)C)C2)n1 N1(C(c2cc(C)n(C)c2)=O)CCCCCC1CNC(=O)C(c1cnccn1)C c1(CC)cccc2sc(NC(=O)NCCc3ncc(-c4ccc(F)cc4)o3)nc12 C1(NC(C(CC)OC)=O)CCN(C(c2cc(C)n(C)c2)=O)CC(O)C1 CC(C(F)(F)C(F)(F)F)=Cc1ccccc1.C1(N2C(=O)NC3(CC3)C2)CCSC1 C1(C(=O)NC2C(NC(CCOC)=O)C2)CCS(=O)(=O)N1C N1(C(C=CCC(C)(C)NC(C(C)OCC=C)=O)=O)CCN(C)CC1CCO N1(C(C(C2CCCCC2)OC)=O)CCN(C(C2CN(C)C2)=O)C(C(C)C)C1 N1(C(CCN(CCCCC)C)=O)CCC2CCC(C1)N2C(=O)CCCSCC C1(NC(C(C2CCN(C(COCCOCCOC)=O)C2)(C)O)=O)(CO)CCN(C)C1 Cc1nc(NS(N)(=O)=O)sc1C(N1CC(NC(C2CN(C(C)C)C2)=O)CC1C)=O Cc1ccc(N)c(C(=O)NC2CC(NC(c3cc4c[nH]nc4s3)=O)C2)c1 c1(NC(C(=O)NCC2ON=C(C(N)=O)C2)=O)cncc2cccnc12 N1(C(C(CC)(CC)CC)=O)CC2CCC(C1)C(NC(c1ccc(Cl)c(C)c1)=O)C2 c1(NC(C2(CN)CCO2)=O)ccc(-c2cnco2)cc1 c1(CC(=O)NCCCN(C(c2c(C)cnnc2O)=O)C)ccc2cnccc2c1 c1(C(=O)NCCCCNC(COc2ccc(C)cc2)=O)nn(C)c2c1CCC2 C=CC1(CC(=O)NCC2CC(NC(=O)C(CC(C)C)OC)C2)CCCCC1 c1(CC)nc(C)[nH]c1C(N1CCC(C)(CNc2nccc(OC(C)C)n2)C1)=O C=C(C)C1CN(C(c2cccc(NCC(O)CNC(=O)C(C)(C)C)n2)=O)CCO1 c1(OC)ncc(Cl)cc1C(=O)NCC1CCCN(C(=O)CC2(O)CCCCC2)C1 N1(C(C(c2nc(C)sc2)=O)=O)CCOCC(CNC(C2(C)CC3CC3C2)=O)C1 C1(C(=O)NCC(C)(CO)NC(=O)Cc2n[nH]c(C)n2)(CC)CNC(=O)C1 c1(OCC)cc(C(N2CC3CC3(NC(=O)CCc3cnc(C)s3)C2)=O)oc(=O)c1 c1(C(N2CC(C)C(CNC(C3COC(=O)N3)=O)CC2)=O)n[nH]c2c1CCSC2 CCC(C(=O)OC)C(=O)NCC(C)CN1CCN(C(=O)CCc2cnc[nH]2)CC1 N1(C(C=CC=CC)=O)CCCC(NC(C2CCCC2(C)C)=O)C1C N1(C(C2CCN(CC)C2)=O)CCOC2CN(C(C3(C#N)CCCCCC3)=O)CC12 Cn1cnc2[nH]c(C(N3C4CCC3CC(CNC(=O)C(O)C(F)F)C4)=O)cc12 C(=O)(CC(C)C(F)F)NC(CN(C(c1nc(-c2cnn(C)c2)oc1C)=O)CC)C S(=O)(=O)(c1ccc2nc(N(CCS(N)(=O)=O)C)sc2c1)NC(C(C)CO)C C(CCC(C)(C)NC(c1cnc(OC)s1)=O)NC(CC=C)=O c12ccccc1S2.C(C(CNC(c1scnc1C(F)F)=O)CO)NC(CC=C)=O C1(C(=O)OCc2n(CC)cnc2)CC2CCC(C1)O2 C1(C(=O)OC)C2CN(C(c3cnn(-c4ccc(F)cn4)c3)=O)CC12 Cc1cc(N(CC(C)NC(c2ccc(F)cc2)=O)C)nc(C(C)(C)C)n1 c1(C(N2C(c3ccc(C)cc3)C(C)C2)C(=O)NC(C)(C)C)cc2sccc2n1C c1(NCC2CC(NC(COC(C)(C)C)=O)C2)cccnc1 c1(CNC(=O)NC(C(c2ccccc2Br)OC)C)ccc(C)nc1O c1(NC(C)=O)cccc2c1CC(=O)N2.C1(=O)CCCCC(=O)c2ccccc2N1 C1(NC(c2cc(COC)oc2C)=O)CCN(C(C2CC(O)(C#N)C2)=O)C(C)C1 N1(Cc2cn(CC)nn2)CCCC(NC(C2CCCCC2)=O)C1 CC1(C)CCC(CNC(c2cccnn2)=O)N(C(c2cnns2)=O)C1 c1(C(=O)NC(C2(O)CCN(C(C(C=C)C)=O)C2)C)ccc2cc[nH]c2n1 Cc1ccc(C(N2CCC(N(C(=O)C#CC(C)(C)C)CCO)C2)=O)c(=O)n1C C1(CNC(C2(C)CC2(Br)Br)=O)CC(NC(=O)CC2CCC2)CC1O C1(C(=O)NCC2(OC)CC2)CC(O)CN1C(=O)CC(C)OC C1(C)(C(=O)NCC(CCOC)NC(=O)Cc2ccc(C)cc2C)CC2CCC1O2 c1(COC)ncc2c(n1)CC1CCC2N1S(=O)(=O)C1CCN(CC(F)F)C1 Cc1ccc(C(=O)NC2CC3CC(NC(c4ccc(C#N)cn4)=O)C2C3)c(O)n1 Cc1nc(O)[nH]c1C(=O)NC1(C2CCCCN2C(=O)CC2C(C)(C)C2(C)C)CC1 C=CC(CC)C(=O)N1CCC(CN(C(=O)Cn2c(C)ccc2C)CC)CC1 C(=O)(C1=CCC2(COC2)OC1)N1CCC(C)(CNC(Cc2cccc(C)c2)=O)C1 CC1CCCC=C1C(=O)NC1CC(C)CN(C(c2nnn3c2CCCC3)=O)C1 N1(C(c2c(C)n[nH]c2)=O)CC(N(C)Cc2cccc(C(F)(F)F)c2C)C(C)(C)C1 c1(C(=O)NCC2CC(CNC(c3ccccn3)=O)CO2)cncc(Cl)c1Cl c1(C(Cn2cc(CC3CCN(C(C4(C=C)COC4)=O)C3)nn2)C)ccc(F)cc1 N1(C(c2cn(C)nc2)=O)CCN(Cc2conc2C(F)(F)F)CC1 c1(NC(CC2(C)CC2)=O)cccc(SCC2CC2CNC(=O)COC(F)F)c1 c1(CCC(=O)NCCNC(c2cc[nH]c2)=O)nnc(-c2ccoc2)o1 c1(C(N(C(c2ccccc2OC)C(=O)OCC)C)=O)ccc(CC)c([N+](=O)[O-])c1 C1(CC)(NC(=O)Cc2occc2C)CCN(C(C2(C(C)C)CCOCC2)=O)CC1 C=C(C)CCCNC(C1CCN(C(C2CC2NC(C)=O)=O)C1)=O N1(C(C(CC#C)(C)C)=O)CCCC(C2(NC(C3CN4CCCN3CC4)=O)CC2)C1 c1(Cn2cc(C3(C(=O)NCC4CN(CC)C4)CC3)nn2)cccc(C(F)(F)F)c1 C1(NC(c2c(C)ccn2C)=O)CN(C(=O)C2=COCCO2)CC1N=[N+]=[N-] c1(C(C(C)C)NC(=O)CN(C(C)C)Cc2cc(CO)[nH]n2)cccc(Cl)c1 N1(C(c2cn(C(C)C)nc2)=O)CC2CC3CC2C1C3NC(=O)C(F)C(C)C c1(CC)onc(C(=O)NCCc2cn(CCCCC(=O)O)nn2)c1C C1(C(N(C)Cc2cnco2)=O)C(C2CC2)CCN1C(=O)CCOCC(C)(C)C c1(C(=O)NCC2N(C(C=CC(CC)=CC)=O)CC2)nc2sc(C)cn2c1C Cc1cncc(C(=O)NC(c2cn(C)nn2)C(=O)NCC2CC2Cl)c1 c1(C(=O)NC(C(=O)OC)Cn2cc(Cl)cn2)ccc2c(c1)nnn2C Cc1ccc(N)c(C(=O)N(CCCCNC(c2cnn3ncccc23)=O)C)c1F N(C(=NCC1CCCC12CC2)NCC(N1CCCCC1)Cc1cccs1)C(CC)C c1(C(=O)NCCC2(NC(=O)CCNC(c3ccoc3)=O)CC2)ccc2ccnn2c1 C=C1CC2CC1CN2C(C1(CC2(C)CC(F)(F)C2)CN(C(N2CCCC2)=O)C1)=O C12(CNC(c3ccc(C(F)F)o3)=O)CC(C(=O)Nc3cccnc3)(C1)C2 c1(C(N2CCC(O)(CNC(C(CCC)O)=O)C2)=O)c(F)ccc(Br)c1C Cc1ccc(CC(=O)NCCCCNC(=O)C(C)(C)c2ccccc2)cc1 CCC(C)C(CC(=O)NCc1ccnc(O)c1)NC(C1CC(=O)CS1)=O c1(CC(=O)N(C(C(=O)NCC=C)C)C2CC2)ccc(Br)c(OC)c1 c1(NC(=O)CCC=CCC2CN(C(CC(CC)C)=O)C2)ncc(C#N)cc1Cl c1(-n2cc(C(C3CC3)OC)nn2)ccc(F)c(C(=O)NCC2CNC(=O)CO2)c1F Cc1ccc2c(c1)CCC(C(=O)NC(C)CNC(C13CC(F)(C1)C3)=O)O2 N1(C(C(C)(O)C2CCC2)=O)CCN(C(=O)Cc2cccc(F)c2F)CC1CO C(C(CC(C)C)C(=O)NC(C)(C)CC(=O)NC1CCC2CCCC1O2)SC N1(C(c2nc(C)n(C)n2)=O)CCCCC12CN(C(C1CSCCS1)=O)C2 C(C)(C(C)(C)C(=O)N1CCCC(C(N)=O)C1)NC(C(C(=O)OC)NC(C)=O)=O C1(CC)Cc2ncc(NC(C3CCCN3C(=O)OC(C)(C)C)C(=O)NC)cc2C1 C(CCCCNC(c1cc(C(N)=O)c[nH]1)=O)NC(C(c1ccccc1)C)=O CC1(CNC2CCC(CNC(=O)OC(C)(C)C)O2)CS(=O)(=O)CCO1 c1(-c2onc(C(N(CC(CC)NC(C(CC)OC)=O)CC)=O)n2)ccccc1F C(=O)(C1=CC2CCCCCC12)N1CCC(CNC(=O)C=CC=C(Cl)Cl)C(F)(F)C1 C1(O)(C(C)NC(=O)C=CCO)CCN(C(=O)CC2CSCCO2)CC1 CN1CCC(C)(C(N2CCOCC2CNC(c2ccsc2Br)=O)=O)C1=O Cc1ncc(CC(=O)NCC2C(C)CCN2C(=O)CC2(C)CC2)c(O)n1 C1(C#N)(C(=O)NCC(C(=O)NCC(C(C)O)C)C)CCCOC1 CC1CN(C(C2CCN(C)CC2)=O)CC1CNC(c1ccc(-c2cccs2)o1)=O N1(C(c2n[nH]c(C)c2O)=O)CCC2(C1)CN(C(=O)CC=C(Cl)Cl)C2 N1(C(c2cnc(C)o2)=O)CCCC(C)(C)C1CNC(=O)CCc1c(N)cnn1C S(=O)(=O)(c1ccc(NC2CSCc3ccccc32)nc1)N(CC(C)(C)C)CC c1(CC(=O)NC(C2CCN(C(c3cncc(CC)c3)=O)C2)C)cc(C)ccc1C c1(C(=O)NC2CC(CNC(C3(C)CCCC3(F)F)=O)C2)ccc2c(c1)CNC2=O S(=O)(=O)(c1ccccn1)N1CC(NC(c2cc(OC)c(O)cc2)=O)C(C)C1 Cc1cc(C)c(NC(=O)C(N2CCCCC2(C)C)C(C2CCCC2)OC)c(C)c1 CCC(C)(C)N.N1(CC(=O)N(CCOCCCOC)CCN(C)C(C)C)CCC1C c1(C(=O)NC2C(CC)N(C(=O)CC3=NNC(=O)C3)CC2)c(Cl)ccc(Cl)c1O C1(O)(CCNC(C2CCN(CC(C)C)C2)=O)CCN(C(=O)C(F)=CC2CC2)C1 c12ccc(cc1)NC(=O)C(c1ccco1)NC2=O.C1(C(=O)O)CC2CC2C1 c1(CC)cn2c(n1)CCC(C(=O)NC1(C3CN(C(=O)C4CC4)C3)CC1)C2 C1(C(=O)NCC2CCN(C(c3ncc[nH]3)=O)C23CC3)CCCC2(CCC2)O1 c1(C(=O)NCC2(C(=O)NCC(C)C)CC(=C)C2)ccccc1SC(C)C(=O)NC C1(NC(C(CCNC(c2ccn(C(C)C)n2)=O)OC)=O)CN(C)CCN(C)C1 CC#CCC(C(=O)NCC1CC[Si](C)(C)C1)NC(=O)C(O)Cn1cncn1 C1(C(=O)NCCC(C)CO)C2CC3C(C2NC(C24CCN(CC2)C4)=O)C13 C1(C(=O)NCC(C(C)C)O)CCCOCC1.C1(=O)CC(=O)C2CN12 Cc1cc(Cl)c(Cl)cc1Nc1cc(OC2CCOC2)cc(C(=O)O)c1 Cn1nc(C(N2CC(NC(=O)CCCn3cccn3)C(F)C2)=O)cc1O N=c1[nH]c2cc(C(N3CC(NC(=O)C(O)CC(N)=O)CC(F)C3)=O)ccc2s1 N1(C(c2occ(C)c2C)=O)C(CNC(c2coc(Cl)n2)=O)CC2CCCC12 N1(C(Cn2nc(C)oc2=O)=O)CC23CCCCC2(C1)CN(C(C1CC1(Cl)Cl)=O)C3 N#Cc1cccc(C(C(F)F)NC(c2ccccc2Cl)=O)n1 c1(OCC)ccccc1C=CC(N1CC=CC(NC(c2sccc2F)=O)C1)=O C1(N(C(=O)NC(C)(C)C)Cc2ccc3ccccn23)Cc2nc3ccccc3n2C1 C1(NC(C(C)OCCC#C)=O)CC(C)(CNC(c2ccccn2)=O)C1 C1(C(C)C)CN(C(=O)C(C)C)CCC1NC(=O)C(C(C)C)N1CCCCC1 Cn1c(C(=O)NCC2COCCN2C(C2CC(C)(C)C2)=O)cnc1[N+](=O)[O-] C=CCCCCC(=O)N1CCN(C(c2nn(CC)nc2C)=O)CC1c1cn[nH]c1 c1(C(N2C(CN(C(c3n(C)nnc3)=O)C3CC3)CCC2)=O)nn(C)c(Cl)c1Cl C1(CCC)CN(C(=O)CCC2CC2(F)F)CCN1C(=O)Cc1nnc(C)o1 CC(C(=O)NC12COC(CNC(=O)CN3CCC(CO)CC3)(C1)C2)C(F)F Cc1nn(CC(C)C)c(Cl)c1C=CC(=O)NCCNC(=O)CCC1NC(=O)NC1=O c1(C(=O)NCC2CN(C(C3(C)C(SC)CCC3)=O)CC2(C)C)ccnc2[nH]nnc12 N1(C(C=CCC(C)C)=O)CCOC2(CC2)C1.C1(C(=O)O)CCCC(CCC)CC1 N1(CCCN(C)C)CCCC(C(=O)N(C(C)(C)C)CC2CCOCC2)CC1 c1(C(N(C)Cc2ccc(CNC(C3CC3(F)F)=O)cc2)=O)cnc2cccnn12 N1(C(C(CC#C)C)=O)CCCC2(CCCCN2C(C23CCCC2(C(N)=O)C3)=O)C1 C1(C(=O)OC)CCCCN1CCC1CC1.C1(C)(C)C(=O)N1C(=O)OC(C)(C)C N1(C(CN(C(C(CCC)OC)=O)CCOC)=O)CCC(C)(CN(C)C)CC1 Cc1cccc(CN2CCOCC2C(=O)Nc2cccc(I)c2Br)c1Cl C1(c2n(CCCC)nnn2)(NC(c2ccccc2C)C(C)C)CSCSC1 c1(CC#C)cc(NC(=O)CC(N2CCN(C(=O)OC(C)(C)C)CC2)C)nn1C C1(C(=O)NC2C(C)CN(C(C3(CO)CCC3)=O)CC2)CC(F)(F)CCC1(C)C CC(CN(C)C(c1coc(C(C)NC(c2ccnnc2)=O)n1)=O)C(C)(C)C C=Cn1ncc(C(N2C(C(N3CC4CC3(C(N)=O)C4)=O)CCC23CC3)=O)c1N Cc1ccc(CC(=O)NCC(C)CNC(=O)C(C(C)C)N2CCCCC2)c(C)c1 C(C)(C(C(=O)NC1CCC(OCF)CC1)C(C)C)NC(c1ccc(C)cc1C)=O C1(S(C)(=O)=O)(C(=O)NC(CCCNC(CC(C)C)=O)C)CCCCC1 C12(NC(c3[nH]cc(C(C)=O)c3)=O)CCCC1CN(C(=O)CC1CNC(=O)O1)C2 C1(O)(CCNC(C(c2ccccc2)C)=O)CCN(C(=O)CSc2n[nH]c(O)n2)C1 C1(NC(C2C(CNC(c3c(NC)scn3)=O)CCO2)=O)CCCC(F)(F)C1 C1(CC)CCN(C(=O)CCOC2CC2)C(C(N2CCC=C(C)C2)=O)C1 c1(NC(C2OCCN(Cc3scc(C)c3)C2)=O)ccc(C(N)=O)c(F)c1 N1(C(C(C(C)C)SCC)=O)CCC(CCOC)(NC(=O)C2=COCCO2)CC1 c1(-n2c(C(C)Cc3ccccc3)nc(C(CC)O)n2)ccc(S(N)(=O)=O)cc1 c1(CC)cc(CC)nc(NC2(CNC(=O)C(CC)OC)CCCCC2)n1 N#CC1(C(=O)NC2CCC(CCC(=O)NC3CNC3)C2)CC=CC1 C1(OC)CN(C(c2cncs2)=O)C(C)(CNC(=O)CC#N)C1 CN1CCC2CCN(C(=O)Cc3cc[nH]n3)C2C1.C12(CCCC1)CCC(=O)NC2 C1(O)(CC)CCC(NC(c2cnn(C3CCOCC3)c2)=O)C1 C(C(=O)N1CC(C(C)NC(=O)C(C)C)C1)(C(C)C)NC(CC(C)C)=O C1(NC(C(=O)N(C2CC(N)C2)C)=O)CN2CCC1(C)CC2 C1(CC)CN(C(=O)Cc2c(Cl)cnn2C)CCN1C(=O)CS(C)(=O)=O N1(C(CC(=O)NC2CC2)=O)CCC(NC(c2cccc(F)c2Cl)=O)C(O)C1 C(C)(CNC(=O)CNC(C1CCCCC1)=O)(CC(C)C)NC(c1c(C)ocn1)=O C(=O)(C(C)(C)C1CC1)NC(CN(C(C(C)NC(=O)OC(C)(C)C)=O)C)C C1(NC(CC2CCN(CCC)CC2)=O)CC(O)CN(C(=O)C(COC)NC(C)=O)C1 C1(C(N2CCN(CCOC)CC2)=O)CN(C(c2cncnc2O)=O)CC1(F)F CCC(CC)C(C(=O)NC)N(CCN1CCOC(C)C1)Cc1cccs1 c1(CC(=O)NCCCCCCNC(C(C)n2ccnc2)=O)ccc2[nH]ccc2c1 C=CC1COCCN1C(=O)CC1CCCC1NC(C1(O)CCCC1)=O C(=O)(C(C(F)(F)F)C(F)(F)F)N(CC(C)NC(C1CC12CC(C)(C)C2)=O)CC Cc1cc(C(c2nnnn2CCCF)NCc2cncnc2O)c(Br)cc1F c1(OCCCC(=O)NC2(CCC)CC2)ccccc1F.C12CCCC1NC(=O)C2 Cc1cnc(C=CC(=O)NC2CCCC2N(C(=O)COC(C)C)C)[nH]1 C1(n2cc(-c3ccc(OC)nc3)nn2)CC2CC(SC3CCCCO3)CC12 C(CCC(O)C(=O)NCc1cnn(C)c1O)NC(c1ccc(SC)o1)=O CCC(CC(=O)NC(C12CCC(CC1)C2)CN(C)C)CC(=O)N(CC(=O)NC)C N1(C(c2cc(CC)no2)=O)CC(CNC(=O)CCc2cnc(O)[nH]2)C(C)C1 C(CNC(c1ccnc(OC)n1)=O)(CC(C)C)NC(C(CC)OC)=O CC(CCNC(=O)CC1(C)CCCO1)CCNC(c1coc(Br)n1)=O C1(CNC(C(C(=O)NCC2(CCC)CCC2)CC)=O)CCC2(CCC2)O1 N1(C(CSc2n(C)cnn2)=O)CCC(NC(c2csc(C(N)=O)n2)=O)C(F)C1 N1(C(c2ccn(C)c2)=O)CCC(NC(=O)Cc2ccsc2)C12CCC2 CCC(C)N=c1[nH]c2c(c(=NCC3=COCCO3)[nH]1)CC(C)CC2 c12cc(ccn1)C(=O)N1CC(C1)NC2=O.c1(OC)ccc(NC(C2CCC2)=O)s1 C1(NC(C23CC(C)C2C3)=O)CCCN(C(=O)CCC2(O)CCC2)C1C C1(c2nn[nH]n2)(N(CC(C)C)C(C2CCC(=O)O2)=O)CCOC1C c1(C(N2CCC(NC(C(C(C)(C)C)SC)=O)(CF)C2)=O)cnn2c1NCC(C)C2 C1(NC(C(C)Oc2ccc(Cl)cc2)=O)COCC(C)(C)O1 C1(N(C(CC(C)N(C)C)=O)C)CCCCC1NC(=O)Cc1cnco1 C=C(Cl)CC(C(=O)NCC(C)(C)C1CCCC1)NC(=O)C(C)CO N1(C(CC(=C)C)=O)C2CCCC1CN(C(c1cccnc1NC(C)C)=O)C2 C1(N(C)C(c2cccnc2O)=O)CCCN(C(c2cnc(Cl)s2)=O)CC1 N=C1NC(=O)C(CC(N2CC3C(CNC(=O)Cn4cc(C5CC5)cn4)C3C2)=O)S1 C1(NC(Cn2ncc(C)c2)=O)CCCCN(C(C2C3CC(=O)CC23)=O)C1 c1(NCCC2(CC(=O)NC(CC)(CC)CC)COCCO2)nc2cc(F)ccc2s1 N1(C(c2ccc(F)s2)=O)CC2(CC(C(N3CCC4C(F)(F)C4C3)=O)CO2)C1 C1(C(=O)NC(C2CCN(C(C(CC=C)(F)F)=O)C2)(C)C)CCc2ncncc2C1 N1(C(C(C)C2CC2)=O)CCC2C(C3CCCN3C(=O)CN(c3ccccn3)C)C2C1 C1(NC(C2CCN(C(N)=O)CC2)=O)CCn2c(O)nnc2C1 CC1CCCC(CC(=O)N(C2CN(C(=O)C(F)(F)CN(C)C)C2)C)C1 N1(C(C2OCCN(C)C2)=O)CC2CCCC2C1C(=O)NCCC1(C)CCCO1 c1(CCC)nnc(S)n1CC(N1CCN(C(C2(COC)C=CCC2)=O)CC1)=O C(CCCCNC(=O)Cc1cnc[nH]1)N(C(=O)CSCc1ccccc1)C O=C(C1=CCOC1)NCC(O)COc1ccccc1.C12CCC13CC23 C1(NC(C)=O)CCC(C(=O)NCC2CN(C(=O)CC(C)(C)F)C2)CC1 N1(C(c2c(OC)cccc2)=O)C2CCC1C(CNC(c1cc(C)nc(O)n1)=O)C2 Cc1nn2c(c1C(N1CC(NC(=O)C=Cc3ccsc3)C1)=O)CCCC2 c1(OC)ccc2c(n1)NC(C(=O)N(C1CCN(C(=O)C(F)CC3CC3)C1)C)C2 C(=O)(C(CC(=C)Cl)NC(c1ccn(CC)n1)=O)N(CC#C)C1CC1 C(CC(C)(C)CC(=O)NC(C1(O)CCCCC1)C(N1CCCCCCC1C)=O)OC C1(C(=O)NC(C2CC(NC(c3ccncc3F)=O)C2)C)CCCCN1C C(C(C)(C)CC(=O)NCCCOCCNC(=O)C(C(C)C)C1CC1)OC.C(N)(=O)N C#Cc1ccc(C(N2CC(O)(C(C)NC(c3cnn(CCF)c3)=O)C2)=O)cc1F C1(CC)CN(C(C2CCCC2NC(=O)CN(C)C)=O)CCO1 C1(C(=O)NCC)CC2CCC1N(C(=O)CCc1ccccc1C)C2 c1(CC)ccc(CC(=O)N(CC(O)CN(C(=O)C(C(C)OC)N(C)C)C)C)cc1 C1(C(=O)NC2(C)CC(NC(c3ccncc3Cl)=O)C2)CCc2nc[nH]c2C1 C(=O)(CCCC(C)(C)C)N(C1CCCN(C(CN2CCCC(CC)C2)=O)CC1)C N1(C(CCC(C)OC)=O)CCC2(CCOCC2)C(NC(=O)CC2CC(SC)C2)C1 N(C(=NCCCOC)NCC(=O)NO)C(C#C)CCC.c1(SCC)nccs1 c1(C(=O)NCC23C(CN(C(CC(C)C)=O)C2)C3)cc([N+](=O)[O-])c(Cl)cc1F C(=O)(C1=NOC(CNC(c2cccc[n+]2[O-])=O)C1)N(CC(C)(C)O)CCC N1(C(C(C=C)OC)=O)CCC12CN(C(=O)CC1CCCN1C)C2 CCC(C)(C(=O)OCc1cccc(C(N2CCOCC2C)=O)c1)OC n1(C(COC)C)cc(C(C)NC(c2cc(-c3cnn(C)c3)[nH]n2)=O)nn1 N1(C(C2CCN(C(C)=O)CC2)=O)CC(NC(C2CCC3(CC3)C2)=O)CC(C)(C)C1 C[Si](C)(CCCN1CCCC1C(=O)NC1CC1)C1CC1 c1(CC(=O)N(CC)CC2CCCN2C(=O)COC(C)C)ccc(F)c(Cl)c1F c1(C(=O)NC2CN(c3c(OC)c(Cl)ncn3)CC(C)C2)cc2ccc(O)nc2s1 O=C(C1=CCCCCC1)NC1CC12CCC(NC(c1coc(Cl)c1)=O)CC2 c1(CC(=O)NC(CC(=O)OCC)C)cc(F)cc([N+](=O)[O-])c1 c1(C(=O)NC2C(C)N(C(C3CNC(=O)C3)=O)CCC2)nc2cc(O)ccc2[nH]1 c1(C(N(CCC(C)NC(c2cn(CC)nn2)=O)C)=O)cccc(N)n1 C1(NC(c2ccc(CC)cc2)=O)CCN(C(c2scnc2CC)=O)CC1O CCC(C(F)(F)F)NC(CC(C)c1nccs1)c1nnnn1C1CC1 c1(CCNC(=O)NCC(CC)(C)c2ccccn2)ccc(F)c(OCC)c1 C(C1=CCCN(C(=O)C(=O)C=Cc2ccccc2)C1)NC(=O)OC(C)(C)C C1(CCCNC(CC2N(C)CCC2)=O)CN(C(=O)CCC(=O)N2CCC2)CCO1 c1(-c2c(C(N3CCC(O)(C(F)(F)F)C3)=O)ccs2)cnc(CO)cn1 Cc1cnccc1C(C)C(=O)N(CC(=O)NCc1ccc(C(C)(C)C)o1)CC1CC1 C1(C(=O)NC2C(NC(CC(C)C)=O)CCC2)COc2ccc(F)cc2C1 c1(C(N2CC3C(C(=O)NCC(CC)CC)(CC3)C2)=O)ccnc2ccccc12 C1(OC)CCC(C)N(C(C23CC2CCN3C(=O)C(c2ccn(C)c2)C)=O)C1 C1(C(=O)NC(C=C)(C)C)CN(C(C2CC23CCOC3)=O)CC12CCC2 c1(OC)ccc2cc(NC(=O)NC(C)Cc3cnccn3)ccc2c1 C=CC(C)(O)C(=O)NCC1(OCCNC(=O)CN(C2CCC2)C)CCC1 C(c1cccc(O)c1)=CC(=O)NC1(CNC(=O)CC2(O)CCCOC2)CC1 C1(COC)(NC(=O)C(C)OCCN(C)C)CCN(C(=O)CCS(C)(=O)=O)CC1 C(=O)(C#CC1CCCO1)N1CCC(F)(CNC(=O)C=Cc2cnc[nH]2)C1 c1(C(N(C2CN(C(COC(C)=O)=O)CC2(C)C)C)=O)ccc2cncn2c1 c1(COC)noc(CNC(C2(NC(=O)CCC3CC3(C)C)CC(C(F)(F)F)C2)=O)n1 c1(OC)cc(CNC(C2CC2CNC(=O)COCCCF)=O)on1 N#CC1=C(C(=O)NCCOCCCNC(c2cnc(O)c(Cl)c2)=O)CCC1 C1(OCC)CN(C(=O)C(C)(CO)OC)CC1NC(=O)CN1CCCCC1 c1(NC2CC(C)CN(C(=O)NCCCl)C2)ccc2cccnc2c1 C1(CC#C)(C(=O)N(C)CCN(C)C(C2CN(C3CCC3)C2)=O)CCOC1 N1(CC(N2C(C)(C(=O)NC3CCCC3O)CCC2)=O)CCCCCC1=O CCC(CC(=O)N1CC=CC1(C)C(=O)NCC1(O)CC(C)(C)C1)C(C)C n1(CCOC)nc(-c2ccc(F)cc2)nc1-c1ccc(CC(C)C)s1 C1(NC(c2c(OCC)ccs2)=O)CC(NC(C2CC=CCC2)=O)CC1O N1(C(C2(C(C)C)CCN(C(=O)C(C3CC3)C3CC3)C2)=O)CC(CO)OCC1C CCCN=C(NCC(C)C)NCCCSCc1cc(C)on1 Cc1cc(CN2CCC(C#N)(NC(c3cc(O)ccc3F)=O)C2)c(C)cc1Br c1(C(=O)NCCC(C)N(C(=O)C(C)CC(F)F)C)cnc2sccn12 CCCCCCCC(=O)N1CC(O)CCC1C(=O)NCc1ccn(CCF)n1 c1(CC)cc(C(=O)NCC(C)C(N2CCOC(C)C2)=O)nn1C C=CCCCC(=O)NCC(C1CCCN1C(c1cc(-c2ccco2)c[nH]1)=O)(C)C N12CCOCC(C)(C1)CNC(=O)C(C)C2=O.N1(C(CNC(C)=O)=O)CCCC1 N1(C(C2C(=C)C2)=O)CCCC(CNC(c2ccc(CC(C)C)cc2)=O)C1 C1(NC(COc2ccc(C#C)cn2)=O)CC2CN(C(=O)C(F)C(C)C)CC2C1 N1(C(C(CC=C)CC)=O)CCC2C1CCCN2C(=O)CNC(=O)NC C(=O)(C1CCCc2ncnn21)N1CCC(NC(C)=O)CC1 C1(C(C)C)(C(=O)NC(CCO)C(C)C)CCCN1C(c1csnn1)=O N1(C(C(C)SCC)=O)CC=C(CNC(=O)C(C(C)C)n2cccc2)CC1 c1(C(=O)NC(C2OCCN(C(c3scc(OC)c3)=O)C2)C)ccc(S(N)(=O)=O)o1 C1(NC(c2cn(CCO)nn2)=O)CC2(CCN(C(=O)C=C3CCSCC3)CC2)C1 CC(C)(CC1CC1)C(=O)NC1CCC(C(=O)NOC2CCCC2)C1 C1(F)(C)CCN(N2CCn3c(Br)cn3C2)CC1.c12c(ccc(C)c1C)c2=O.CO C1(C2(CCC=C)OC2)(CNCCCc2nc[nH]n2)CN(C=O)C1.C(C)(C)(C)O c1(NCc2ccc(C(C)C)o2)ncnc2sc(NC(=O)OC(C)(C)C)nc12 N1(C(c2cc(C)oc2C)=O)CCc2ccccc2C1CNC(c1cn[nH]c1)=O C(C)(C(=O)N1CCC(CNC(C2COCCN2CC(F)F)=O)CC1)(C(C)C)OC Cc1nn(C)c(Cl)c1CCNC(=O)N(c1ccc(Br)cc1)C CC1CCC(S(C)(=O)=O)CN1C(c1ccc(-c2csnn2)cc1)=O N1(C(CCc2nnc(C)n2C)=O)CC2ON=C(CNC(=O)Cn3ncnn3)C2C1 C(c1cccc(Br)c1)=CC(=O)NCC1CCC(C)N(C(C2OCCO2)=O)C1 Cc1cc(C)c(C(=O)NCC2CC(C(=O)NC(CO)CC(C)(C)C)C2)cn1 c1(CC(=O)N(C(CNC(C(CC)C)=O)C2CC2)C)ccccc1CN1CCCCC1 c1(C(=O)NCCCN(C)C(c2cc(C3CC3)[nH]n2)=O)n[nH]c(CO)c1Cl Cc1ccc(CN2CCC(n3cc(CNC(C)CC4CC4)nn3)C2)cc1 c1(C(=O)NC2(CNC(CCN(C(C)=O)C)=O)CC2)cc(C2CC2)cs1 C1(NC(Cc2ccc(C)cc2)=O)CS(=O)(=O)CC1NC(C1CC1C)=O CC(C)CC(O)C(C)C(=O)NC1CCOC1C(N1C2CCC(C2)C1CO)=O c1(C(N2C(CNC(CN(C(C)=O)C)=O)CCC2)=O)cnc(C(C)(C)C)nc1C N1(C(C(CC)SC)=O)CC(C)CN(C(c2ccc3nc[nH]c3n2)=O)CC1C N1(C(CC(=O)OC)=O)CC2CC2(C(=O)N(C(C)CO)C2CC2)C1 c1(C(N2CCN(C(C(CC)=CC)=O)CC2COC)=O)cnc(O)c2ccccc12 CC1CN(CC(F)F)CC1(c1nnnn1C(C)(C)C)NC(c1c(Cl)cccc1Cl)=O c1(C(=O)NCC2N(C(C(CC)c3cccnc3)=O)CC2)cc(C2CC2)ccc1C C(=O)(C(O)P(C)(C)=O)NC(C(C(C)C)NC(Cc1ccc(C(C)C)cc1)=O)C c1(C(=O)NC2CC3(C(C(N(C4CCCCC4)CC)=O)C3)C2)ccc(C)nc1C C1(NC(c2cc(C(C)C)on2)=O)CC2CC1CN(C(c1ccn(C(F)F)n1)=O)C2 N1(C(c2cnc(C(C)C)o2)=O)CCCCCCC1C(=O)NCCCOCCCO Cc1c(NCCc2sccc2Br)ncnc1N1CCN2C(=O)CC2C1 c1(OC)cc(C(N2CCC=C(C(=O)NCCN(C)C)C2)=O)cc(OC)c1O C(=O)(C1=CCC2(COC2)OC1)NCCC1N(C(C(C)=CC2CC2)=O)CCC1 c1(CNC(c2cc(CC)oc2C)=O)ccc(CNC(C2(C)CC(C)C2)=O)c(F)c1 CC#CCC(C)N=c1[nH]c(N(C)CCc2ccccn2)nc2c1SCC2 C12(CNC(c3cccc(OC)c3)=O)CCC(C1)N(C(c1cnn(C)n1)=O)C2 C(C)(CNC(=O)Cc1csc(C)c1)(CC(C)C)NC(C(CC)OCC)=O C1(N2CC(CCN3CCC(C)C3)C2)CC2CCC1N(C(=O)C(C(C)C)N(C)C)C2 N1(C(c2cc(C(=O)OC)ncc2)=O)CCCC(CO)(NC(=O)CC(C)N(C)C)C1 C1(CC(N2C(C)CC(NC(Cn3nc(C)oc3=O)=O)C2)=O)CCC(C)(C)CO1 C1(NC(c2ccc(I)cc2F)=O)CN(C(c2cccc(F)c2F)=O)CCC1(F)F c1(NCC2(NC(C3CC4C=CC3C4)=O)C(C)CCCC2)ncnc(Cl)c1[N+](=O)[O-] n1(CCOC)nccc1C(=O)NCC(C)(O)CNC(=O)CC(C)C1CCCC1 C(=O)(C(C)CC1CCCC1)N(C)CCc1nccs1.C12CC(C1)C(=O)NC2C C1(NC(c2c(CNC(=O)C(F)=CC3CC3)cc[nH]2)=O)CC2CC3C(C2)C13 C1(CC)CN(C(c2n[nH]cc2Cl)=O)CC(C)S1(=O)=O C1(C#N)(CC(=O)NCC(CNC(c2ccnc(C(C)C)n2)=O)(C)C)CCOCC1 O=C1CCC(CC(N2CCCC2C2(CNC(=O)C3=NOCC3)CC2)=O)CN1 C(Cc1cc[nH]n1)(C(=O)NC1(N2CSCC2=O)CC1)NC(C(C1CCCCC1)C)=O CC1CC(NC(c2ccc(N)c(F)n2)=O)CN(C(=O)C(=Cc2cn(C)nn2)F)C1 Cc1ccc(O)c(C(N2C3CCC2C(C(=O)NC2(CF)CC2)C3)=O)c1 N1(C(C2CCC(C3CCC3)CC2)=O)CCC2OCCN(C(=O)COC3CC3)C2C1 n1(CC)nccc1C=CC(=O)NC1(COC)CCN(C(C2(SC)CC2)=O)C1 N1(C(c2c(CCC)nco2)=O)CCCC(NC(=O)C(C(C)C)NC(=O)C2CC2)C1 N1(C(c2nc(OCC)sn2)=O)CC(CO)C2(C1)CN(C(=O)CS(N)(=O)=O)C2 CCCCC(CC(=O)NCC1(C#N)CCCC1)NC(c1csc(C)c1C)=O C(CC(CNC(=O)CC1(C)CCCC1)NC(C1CC1(C)C)=O)OC C1(C(=O)NC(C2(O)CCC2)C(=O)O)CCN(Cc2nc(CC3CC3)no2)CC1O N1(C(C2CN(C(C)C)C(=O)CC2)=O)CC(CO)C2(C1)CN(C(c1cc[nH]n1)=O)C2 C=CC1(CC)CN(C(=O)CCSc2nnc(-c3cnccn3)n2CC)C1 C(=O)(C(C)CC(=O)OC)NC(C(=O)NC(CCOC)C)CC1CC1 C#CC(CC(C)(C)C)NC(=O)CC(C(C)C)NC(=O)C(C1(O)CCCC1)F N1(C(C(C)S(N)(=O)=O)=O)CCC(CNC(=O)CCC(F)F)C(F)(F)CC1 Cc1cc(C(=O)NCCCCC(C)NC(C2(F)CCS(=O)(=O)C2)=O)ccc1N c1(OC)ccc([N+](=O)[O-])c(CNC(=O)C(N2CCC(N3CC(O)C3)C2)=O)c1 c1(CC(=O)Nc2ccc(F)cc2Cl)cn2cc(-c3cccc(CO)c3)ccc2n1 N1(C(C(N2C(=O)CCC2=O)C)=O)CCN(C(=O)Cn2ncnn2)CC1 CC(c1ccccc1C)=CC(=O)NC1CCCCN(C(c2cc(Cl)ns2)=O)C1 c1(NCC(=O)NC(C)C(C)(C)NC(c2c[nH]nc2C2CC2)=O)ccc(F)cc1F Cn1ncc2cc(C(N3CCC(C(N4CC5CC5C4)=O)C(O)C3)=O)cnc12 N1(C(C2CCN(c3nnc(C)o3)CCC2CO)=O)Cc2ccccc2C1 c1(C(N2CC(CCNC(C3(OC)CC3)=O)OCC2)=O)cnn2c1OCC(O)C2 N1(C(CCCOCC)=O)CCN(C(C2ON=C(C)C2C)=O)CC1c1nccn1C C1(C2CCN(C)CC2)(C(=O)NCCCN(C(=O)CCCC(C)(C)C)C)CC1 N1(C(C(CC=C)CC)=O)CCC(C)(C)C(C(=O)NCCN2CCC2)C1 c1(CC)cc(C(=O)NCC(C)CNC(C2CCCC(C)(C)C2)=O)c2c(c1)CCO2 C(CCC(C)C)(C(=O)N1CC2(CCC(CNC(=O)CC3CCNC3=O)O2)C1)OC N12CCN(CC1)C1CC1C2=O.C1(OCC)COCC1n1cc(-c2csc(C)n2)nn1 CCC(CC(=O)NCC1(NC(C2(CO)CCCCC2)=O)CCC1)OC C(=O)(CCCC(=O)NC(Cc1ccco1)C(=O)NCc1nn[nH]n1)N(C)C c1(NC(C2CCCN(C(C(C)N(C)C)=O)C2)=O)ccc(C(C)(C)C)c(Cl)c1 C(c1ccccc1C#N)=CC(=O)N(C(CNC(Cc1c(C)nn(C)c1)=O)C)C C1(C#CC(=O)N(CCC(C)NC(c2cc[n+]([O-])cc2)=O)C)(CC)COC1 c1(NC(=O)C2=CCC2)ccnc(-n2cncn2)c1.C12CCCN1C(=O)C2 c1(C(C(N2CCCC(c3cn(CC(=O)OC)nn3)C2)=O)C)ccc(F)c(OC)c1 c1(CN(C)C(=O)NC(C(N)=O)C2CCC2)cc(C(F)(F)F)c[nH]1 c1(C(N2CCC(C(C)(C)NC(=O)CNC(=O)C3CC3)C2)=O)cccc2c1C(=O)NC2 Cn1nc(C(=O)NCC(C2CCC2)NC(C23CC(CO2)C3)=O)c2c1CCC2 N1(C(C2CC3(CC(=C)C3)C2)=O)CCN(C(C2CCC=CO2)=O)CC12CCC2 C(=O)(CCCC(=O)N1CCCC(NC(=O)CC2C(C)(C)C2(C)C)C1)NCC C1(NC(C(c2n(C)nnc2)(F)F)=O)CC(C)(C)C1OCc1ccccc1 C1(C(=O)NC(c2cccs2)C)CC(C)(C)CCN1C(c1cnn[nH]1)=O c1(C(=O)NCC2CN(C(=O)C=Cc3cc[nH]n3)CCO2)cc(F)cc2nn[nH]c12 CC1C(C(=O)NC2CCC(C(=O)NC3(C)CC(O)(CO)C3)C2)CCN1C C(=O)(C1=CCCC1(C)C)NC(CC)CNC(c1cnc(OC)c(C)c1)=O c1(CC(=O)NCC2CN(C(C3C(c4n(C)ncc4)OCC3)=O)C2)ccc(Cl)cn1 CC1(C)C(CO)CN1C(=O)CC1CC(F)CN1C(=O)CSCC(=O)N(C)C CC1CC(NC(c2cc(N)cc(O)c2)=O)CN(C(=O)CCSc2ccccc2)C1 CC(C(=O)NC1(CCNC(=O)CCc2cncs2)CCC1)N1CCC1 C1(NC(c2c(C)cns2)=O)CCN(C(C2CCSCC2)=O)CCC1CO N1(C(CS(CC)=O)=O)CCN(C(=O)COc2ccc(Cl)c(C)c2)C(C2CCC2)C1 c1(C(=O)NC2CC(NC(C3CC(C)C3)=O)C2)c[nH]c2ccc(Br)cc12 N1(C(c2cncc(NC)n2)=O)CC2(C1)CN(C(=O)Cc1cnn(C(C)C)c1)C2 CCCC(C(=O)NC)OC.c1(CN2CC(C(C)OC)C2)nccnc1C(F)(F)F N1(C(CC(CCC)O)=O)C2CCCC1CN(C(c1c[nH]nc1C(F)F)=O)C2 C1(C(N(C(CCSC)C)C)=O)CC12CCN(C(c1ccc(C)nc1C)=O)C2 C1(C2CC2)(CNC(c2cc(OC)nn2C)=O)CCN(C(=O)CC(C)C2CC2)C1 c1(C(N2CCC(C)(NC(C3(C=C)CC3)=O)C2)=O)cc(C)c2c(O)nc(O)nc2n1 C1(CCNC(=O)CC2CCOC2)CCCN(C(=O)C=Cc2ncc[nH]2)CC1 C1(NC(c2cnc3sccn23)c2n(CCOC)nnn2)CCCCC12CCC2 C(=O)(CCC(=O)NCC(C)(O)CNC(c1nnc(S)n1C)=O)N(C)C N1(C(c2cc(C(C)C)no2)=O)CCN(C(C2(C)C=CCCC2)=O)CC(O)C1 Oc1ncccc1CNC(=NCc1ccco1)NC1CCN(C(=O)C(Cl)Cl)C1 C1(NC(c2ncc(C)nc2)=O)CCCN(Cc2nc(C)c(C)o2)CC1 N1(C(C2C(C)=C2)=O)CCCC2(NC(C3CCC4(CCC4)O3)=O)CC2C1 c1(C(N(C)CCNC(=O)CCc2ccccc2O)=O)c2c(nn1C)CCCC2 Cc1cc(C(=O)NCC(C)NC(C2C3(CC3)C23CC3)=O)c2ncccc2c1 CC1CCC(C)(NC(C2CN(C(C3CCN(C)C(=O)C3)=O)CC3(CC3)C2)=O)CC1 Cc1ccc(CC(=O)NCC2CCN(C(=O)CCc3cn(C)nn3)CC2)c(F)c1 O=C1CC(C(N2CCC(C3CCCN3C(=O)CCCCC3CC3)C2)=O)CCCN1 NC(=O)CCC(=O)N1CCC(NC(=O)C=CCOC2CCOCC2)C1 c1(C(N(C2CCCC(NC(c3ccc(CCC)s3)=O)C2)C)=O)cc(N)nc(Cl)c1 C(=O)(CCCCCC(=O)NCC1CCCC1NC(=O)C(C)C(C)O)OCC C(C1CCOCC1)=CC(=O)NCC(C(=O)N(C(C#C)C)C)N(C)C CC1CC(NC(=O)Cc2ccc(CO)cc2)CN1C(=O)COc1cccc(Cl)c1 S(=O)(=O)(c1c[nH]ccc1=NC1CC(N)CC1O)N(C)CCOCCN(C)C c1(OC)cc(Cl)c(C(N2CC3CCC2CN3C(C2CC2C2CC2)=O)=O)cc1OC N1(C(C2CCC(CC)CC2)=O)CC(NC(C2CC(=O)N(OC)C2)=O)CC12CCC2 C1(C)(C(N2CCC(C(C)NC(C3C(=C)C3C(=O)OC)=O)C2)=O)CC(F)(F)C1 Cc1ncnc(C)c1CC(=O)NC(CNC(c1cnc(Cl)s1)=O)C(C)C C1(O)(C(C)NC(=O)OCC)CCN(C(=O)Cc2n[nH]c(C)n2)C1 c1(OC)ccc(OC(C)C(=O)NCC(C2CCCN2C(C2CCC2)=O)(C)C)cc1 CC1(CNC(C2(C)CC2Br)=O)CCCN(C(C2CC(=O)N2)=O)C1 c1(C(N2CC(C)CC(NC(c3cc(C)cc(Cl)c3)=O)C2)=O)c[nH]c2nccc-2c1 C1(C(CNC(CCCCC)=O)=O)CN(CC2CCOC2)CC(C)(C)C1 N1(CC)CC(NC(c2conc2CNC(=O)CC2CCCC(=O)C2)=O)CCC1=O c1(OC)ccc([N+](=O)[O-])cc1CNC(=O)C(c1ccccc1F)(F)F CC(O)CCCCCC(=O)N1CCCC(CNC(C23CC(C2)C3)=O)C1 c1(C(N(C(CNC(c2c(CC)cco2)=O)C)C)=O)ccc2c(c1)CCCO2 C1(CNC(=O)CCC2CCCO2)CCC(NC(c2ccnn2C2CCC2)=O)CC1 Cc1sc(Cl)nc1C(N1CC2CC2(NC(c2cc(Cl)ccn2)=O)C1)=O c1(CNC(C(C)(C)OCC)c2nnnn2C2(C)CC2)cccc(CS(N)(=O)=O)c1 C(C(C)(C)CNC(c1cnn(-c2ccccn2)c1)=O)N(C(=O)CN1CSCC1)C N1(C(C(=O)NCC(F)Cl)=O)CCc2ccccc2C(O)C1 CC(C)CCC(=O)N1CC(CF)(NC(=O)C(N2CCCCC2=O)C)C1 Cc1[nH]nc2ccc(C(=O)NCC3CCCN(C(C4CC4Br)=O)C3)cc12 C1(NC(C=C(C)C(C)C)=O)CN(C(=O)C(C)NS(=O)(=O)c2cccs2)CCC1O c1(C(=O)NCC(C)N(C(=O)COCCF)C)cn(C)c(C(F)F)n1 N1(C(c2c(SC)scc2)=O)CCOCC(NC(=O)CN2CCCC2C)C1 CCC(CC)CC(F)C(=O)NCC1CCN(C(=O)COCC(C)(C)C)CC1 CC(CC(=O)N1CCN(C(=O)C#CC2CCC2)C2CCC12)CC(F)(F)F c1(OCC)c(NC(=O)NCC(=O)Nc2cc(C)cc(C)c2)cccc1F c1(CNc2ccc(NC(C(CSC)(C)C)=O)cn2)cc2cnccc2[nH]1 N1(C(c2c(C)nsc2)=O)CCN(C(C2CS(=O)(=O)C2)=O)CC1C(F)F C1(N(C(CCOCCC)=O)C)CCN(C(c2csc(COC)n2)=O)CC1C C(N=c1nc(N2CC3CC2CS3=O)c2ccccc2[nH]1)N1C(=O)CCC1=O N1(C(C2C(C)CCCC2)=O)CCN(C(=O)C(C)(C)Nc2ccccn2)CCC1C N1(C(C=C(C)c2ccco2)=O)CC2CCC(N(C(=O)C(C)n3cccn3)C)C2C1 C1(C(=O)NC(c2c(C)noc2C)C)N(C(=O)CC2CC(F)(F)C2)CCC1(C)C CC(CNC(=O)C=CC1CCC1)(C(F)(F)F)c1ccc(Br)cc1 N#Cc1cncnc1N1CCC(CNC(=O)CC2COCCN2CC2CCCC2)C1 N1(S(=O)(=O)CCN2CCOC(c3ccccc3)C2)CC(C(=O)NC2CC2)CC(F)C1 N(C(=NCC1CCOC1=O)NC(c1ccccc1)C1CCCO1)C(C)C1CC1 Cc1nc(C2CC2)sc1C(=O)N(CC(C)NC(C1CC12CCCC2)=O)C C1(C(C(=O)OC)O)(NC(=O)C(C)NCC(C)(C)CO)CCCCC1.c12coc-1c2 CCS(=O)CC(=O)NC(C)(C)C=CC(=O)NCc1n[nH]c(C)n1 C#Cc1cncc(NC(=O)C(O)C2CN(C(=O)Cc3cc[nH]n3)C2)c1 N1(C(CCCCCCC)=O)CCC(NC(=O)C=CC=C(Cl)Cl)C2(CC2)C1.C=CCCO O=CN1CCCC1C(=O)NCCC1CCN(C(=O)CC2CC(OC(F)F)C2)C1 CN1C(=O)Cc2c(NC3CC34CCN(C(c3cnco3)=O)CC4)ncnc21 CCC(C)C(C(=O)Nc1cccc(C(F)(F)F)c1)N(C(C(=O)NC)C1CCCC1)C C(=O)(C(C)(C)C(=O)NCC(CNC(=O)CCc1nccn1C)OC)OCC N1(C(c2c(CC)cco2)=O)CCC2(CCCC(CNC(=O)CNC=O)O2)CC1 N1(C(C(CC)COC)=O)CCN(C(=O)C2=CCSC2)CC1CCOC N1(C(c2cc(COC)on2)=O)CC(NC(c2ccnnc2)=O)CC12CCCC2 N1(C(c2ccc(SC)s2)=O)CCN(C(C2CCOC2(C)C)=O)C(CCO)C1 CN1CC2CCCC2N(C(=O)NCCC(F)CN=[N+]=[N-])CC1=O CC1CCCc2cc(C(N3CCC(=CCNC(=O)C(C)C4CCC4)CC3)=O)nn21 C(=O)(CC(C)CC(=O)OC)N(CCC)CC1CCN(C(=O)C(C)(C)CO)CC1 c1(OC)cc(NC(c2cccc(NCc3ccc(F)nc3)c2)=O)ccc1Br CCC(O)C(C)(C)C(=O)N1CCCC(C)(CNC(c2cc(C)nn2C)=O)C1 c1(C(N2C(C(N3CCCC(C#N)C3)=O)CC3CC32)=O)cc2ncccc2[nH]1 Cc1cc(Cl)c(C(=O)NC2CC3CC2N(C(=O)CCc2cn[nH]c2)C3)cc1C Cc1cc(C(=O)NC2CCCCC2CNC(c2cc(C)n(C)n2)=O)ccc1F C1(NC(C2CCOC2)=O)(CO)CCCN(C(=O)CCC2CCCCO2)C1 c1(C(N2CC(C(C)(C)O)(CNC(c3nc(C)c(C)s3)=O)C2)=O)ccc(Cl)nc1N N1(C(C2CCN(C)C(=O)C2)=O)C2CCCC1CC(NC(C1C=CCC1)=O)C2 c1(C(=O)NC2C(CCC)CN(C(C3C=CCC3)=O)C2)cnc(C)cc1C C12(CNC(c3cc(=O)cc(Cl)[nH]3)=O)CCC(C1)N(C(=O)CCc1ccncn1)C2 C1(C)(C(=O)NC(CCCNC(c2c(CCC)n[nH]c2)=O)C)CCC(C)=C(C)C1 CC1CC(C(=O)NCC2CN(C(c3occc3-c3ccccc3)=O)C2)CO1 C12CN(CC13CC3)C2=O.N#Cc1c[nH]c(C(=O)NCC2(N3CCOCC3)CC2)c1 Cc1cc(C(=O)NCc2nc(C(=O)NC3COCC3N(C)C)co2)no1 CC(C(N)C(=O)NS(C)(=O)=O)NCC1CC(COc2ccccc2)C1.C1(=O)CN1 c1(C(=O)NC2CCC(NC(C3(COC)CCCO3)=O)CC2)cc(=O)c(O)c[nH]1 c1(C(=O)NCC(C(=O)NC)Cc2ccc(F)cc2)cc(C(=O)O)c(F)cn1 Cc1oc2ccccc2c1C(=O)NC1CC1NC(=O)CCc1cc[nH]n1 N1(C(CCCCC)=O)CCC(C2CCN(C(=O)C(c3cnn(C)c3)C)CC2)C1 Cc1cc2ncc(C(N3CCC4(CCCN4C(=O)Cc4cnc[nH]4)C3)=O)cn2n1 C1(N(C(CN(C)CC)=O)C)CCCCN(C(c2cc(NC(N)=O)ccc2Cl)=O)C1 c1(OC)ccc2[nH]cc(C(N3CCC(ONC(c4sccc4Cl)=O)C3)=O)c2c1 C1(NC(c2n(CC)ccc2)=O)CC(O)CN(C(=O)Cn2cc(Cl)cn2)C1 C=CC(C)(C)C(=O)NCCC1(NC(c2cnn(CCC)c2C)=O)CC1 C(C(=O)NCCC1COCCN1C(=O)CN1CC=CC1)(C(C)(C)C)SC C1(C)(C)CN(C(=O)CCCCCF)CCO1.Cc1cnc(C(=O)NCC)nc1 C(=O)(CCS(C)=O)N(C)Cc1cn(CCCC(=O)OC(C)(C)C)nn1 c1(NC(CCc2cn(C34CCC(CC3)C4)nn2)=O)cccc2nc[nH]c12.CSC CCCC(C(=O)NCCCc1cc(C)no1)NC(c1ccc(C#N)o1)=O c1(C(N2CCC(C(C)NC(=O)Cc3cc[nH]c3)C2)=O)c(F)cc(C#N)cc1F C1(NC(c2c(C)cn(C)c2)=O)CC2CCC(C1C)N2C(c1ccoc1)=O n1(CCC)nnc(CC(=O)NCCC(C)NC(C2(NC(C)=O)CCCC2)=O)n1 c1(C(=O)NC(CC(C)NC(=O)CC2(C)CCCC2)C)cnc2c(N)cccc2c1 C1(C)(C(N(C)CC2COC(=O)N2)=O)C=CCN1C(C1CCCC1O)=O N1(c2nnc(C(C)(C)C)o2)CCN(C2CCCN(C(C3CC(=O)CO3)=O)C2)C(=O)C1 C(Cc1ccccc1)(C(=O)N1CC(O)(CCNC(=O)CCc2nc[nH]n2)C1)OC c1(C(N2CCC(N(C(=O)CNS(=O)(=O)C3CC3)C)CC2)=O)ccccc1S(C)=O CC1CN(C(C2CS(=O)C2)=O)CCC1NC(=O)C1=CSCS1 CC1(C(=O)NOC2CC3C=CC2C3)CCCN1C(=O)CN1CCCC1=O C1(c2nnnn2C2CCOC2)(NCc2c(C)noc2)CCCCC1 N1(C(c2cnc(OCC)s2)=O)C2CCC1CN(C(c1cscc1F)=O)CC2 N1(C(CC2CC(=O)NC2)=O)CC(NC(=O)COc2cccc(F)c2F)C2(CC2)C1 C1(NC(C(C)NS(C)(=O)=O)=O)CCCOC12CCN(C(c1cscn1)=O)CC2 CC1(C)CCC(C(N2CCOC3CC23)=O)CN1C(C1C2CC3C(C2=O)C13)=O C1(C)(C(=O)NCC2OCCN(C(CCc3n(C)c(S)nn3)=O)C2)COC(=O)OC1 c1(C2(NC(c3n(CC=C)nnn3)c3occc3C)CC2)ccc(OC)cc1 C12COCCN1CCNC2=O.c1(CNC(c2cc[nH]n2)=O)ccc(Cl)o1 C(=O)(C(CC)C(=O)N1CCC(C)(C(=O)N(CC(O)CO)C)CC1)OCC C1(C2CC2)(C(=O)NCC(CC)NC(c2cnn(C)c2F)=O)CC=CC1 C1(CNC(C(C)NS(CC)(=O)=O)=O)CC2(CCN(c3cc(C)nc(C)n3)C2)CO1 N1(C(CSCC=C)=O)CCN(C(C2CCC(NC(=O)C(C)C)CC2)=O)C2(CCC2)C1 N1(C(C2CC(O)(CNC(=O)C#CC3CCCC3)C2)=O)CC2CCCC2C12CC2 c1(C2(NC(=O)CC3CN(Cc4sncc4Br)C3)CCC2)ccccc1 C=CCC(C)(C)CC(=O)N(C(=O)C(N1CCC(N(C)C)C2(CC2)C1)=O)C N1(C(CC(CC=C)NC(=O)CCCN(C)C(C)C)=O)CCC(O)CC12CC2 N1(C(CCCNC(Cc2c(C)nccc2)=O)=O)CC(C)(C2CCC2)C1 C1(NC(C2CC2F)=O)C2CC(CN(C(c3ccc(CCO)cc3)=O)C2)C1CO CC(CNC(c1cocc1C(N)=O)=O)C(=O)NC1(C)CCCC1 C1(C(=O)NCCC2(O)CCN(C(COCCSC)=O)C2)CCc2ccccc2O1 C1(CNC(=O)CSC2CC2)CC(F)(F)CN1C(C1CCCC(C2CC2)O1)=O Cn1nc(C2CC2)c(Br)c1CNCc1cnc2sccn12 O=C(N=c1cc[nH]cc1O)C1CC2(CC2)CN1C(=O)CN1C(=O)C=CC1=O C1(CNC(c2cnc(OC)s2)=O)CC12CCN(C(c1cc[nH]c(=N)c1)=O)CC2 CC(O)CC(C(=O)O)NC(c1ccc(SC(F)(F)F)cc1)=O.C1C(=O)N1 Cc1cc(C(=O)NC2CCN(C(=O)CC3CCCN3C)CC2(C)C)c(O)c(C)n1 c1(C(N2CCCN(CC(C)(C)O)CC2)=O)ccc2ncc(=O)[nH]c2c1 CC(O)C(F)(F)C(=O)N1CCOC(CC(=O)NC2(CO)CCCCC2)C1 N1(C(C(c2ccc(F)cc2)(C)F)=O)CCCC(CNC(c2cnsn2)=O)C1 c1(-c2nc(C(CC)C(C)C)on2)cnn2c1NCC2 N1(C(c2ccc(-c3ccc(C)s3)o2)=O)CCN(C(C)C)C(=O)C1 N(C(=NCCCC(F)F)NCCOCc1cc(C)ccc1Br)C(CC)C Cc1nc(Br)sc1C(N1CCN(C)CC1)C(=O)NCC1CC1 C(=O)(C1=CCCC1)N1CCC(C(N)=O)C1.CC(C)C(C)n1cccn1 C1(NC(CCSCCCC)=O)CC(CNC(=O)CCCc2cncs2)C12CCC2 c1(C(=O)OC)cccn(CC(=O)NC2CCCCC2CNC(C2CCC2)=O)c1=O C#Cc1cc(F)c(C(N2CCC3(C2)CN(C(=O)C(C)(CC)CC)C3)=O)cc1F Cc1oc(-c2nn[nH]n2)cc1C(F)(F)F.N12CCCCC1c1cn(nn1)CC2=O c1(CC(=O)NCCN(C(=O)CC2CCOC2(C)C)C)ccc2nc[nH]c2c1 C(=O)(C1CCCc2nncn21)NCC(CC(C)C)NC(CN1CCC(C)C1)=O c1(C(=O)NC(CNC(c2cc(C)c(C)nc2)=O)(C)C)cc(F)cc2c1NCCC2 N1(C(CCCc2onc(C)n2)=O)CCN(C(=O)C=CS(C)=O)CC1CC(F)F N1(C(C(C2CCC2)OC)=O)CCN(C2CN(C(=O)C(Cc3ccsc3)OC)C2)CC1 N1(C(CCN(C(C(C)(C)O)=O)CCCO)=O)C2CCC1CC(F)C2 c1(C2CCN(CC#C)CC2C(=O)O)cnn2ccccc12.N1(C=O)CC(OCC)C1 N1(C(C(C)CS(C)(=O)=O)=O)CC2(CCCN(C(=O)CCOC3CCCOC3)C2)C1 C=CCCC(C)(C)C(=O)N1CCC=C(C(=O)NCc2cn(C)nn2)C1 C1(C(C)C(=O)NCC2CCCN2C)CCN(C(=O)Cc2ccn(C)c2)CC1 N1(C(C2C3CCN(C(Cc4c(C)ncs4)=O)CC32)=O)CCCc2cccc(F)c21 N1(C(C2CC(=O)NC2)=O)CCC2(C1)CN(C(c1cc3cn[nH]c3cn1)=O)CCO2 Brc1cc2ncnc(NCC3CC4(CC4)C34CC4)c2s1 c1(C(=O)NC2CN(C(C(C)NC(CC)=O)=O)CC2CSC)c(F)ccc(O)c1F N1(CC2(NC(c3c(C)onc3)=O)CC2)CCN(C(C2CCC(F)C2)=O)CC1 N1(C(c2cccc(OCC)c2)=O)CCC(F)(CNC(C2SC3C=CC2C3)=O)CC1 c1(OC)cc(Br)cc2[nH]nc(C(=O)Nc3ncccc3CN(C)C)c12 CN1CC=C(CC(=O)N2CC3(CCCC3)C2C(N2CCC(CC(N)=O)C2)=O)CC1 c1(OCCOC)cccc(Br)c1Nc1cc(C)c(Cl)cc1I.C1CO1 CC(C)(CC1CCC1)C(=O)N1CC(c2ccc(N)cc2)C1 c1(OC)cc(C(=O)N(C)CC2CCCN2C(=O)CCC2CC2(C)C)n(C)n1 C1(C(=O)NC(CC)(C)CC)CC=CCC1NC(c1[nH]cc(C)c1C)=O C(CC)(CC)(CCNC(=O)C(C)N(C)Cc1ccccc1C)NC(CCCC)=O C1(O)(C(CC)C(=O)NC2CCC2CNC(C2(C(=O)NC)CC2)=O)CCCCC1 c1(C(N(CCC(C(C)C)NC(c2ccc(F)s2)=O)C)=O)cccc2c[nH]nc12 CC(=NOCC#N)C(=O)N(CC(=O)NCC(O)C(C)O)C(C)C c1(C(=O)NC(C2CN(C(=O)Cc3cnccn3)CCO2)C)nccc2nn[nH]c12 C1(CCC=C)(C(=O)NCc2ccc(C)nc2)CCN(C(=O)C(C)NC(=O)NC)C1 C1(C(N2CC(O)(CNC(C3(NC(C)=O)CCCC3)=O)C2)=O)CCOC2(CCC2)C1 C(=O)(C(C)(C)C(F)F)N1CCC(C(CNC(C(C=C)OC)=O)O)CC1 C(=O)(CC(C)(C)C(F)F)NCC1(OC)CCN(C(c2cc(OC)c(O)cc2)=O)C1 C1(CNC(c2ncc(OC)nc2)=O)CN(C(=O)C(C(C)O)NC(C)=O)CCCO1 C(=O)(CC(F)(F)C(F)(F)F)NCCCC(c1ccccc1)NC(=O)CC(=O)NC1CC1 c1(C(N2C3CC(NC(C=C(C)C(F)F)=O)CC2CC3)=O)ccc(F)c2occc12 N1(NC(CC2CCC(C)O2)=O)CC(C)CC(C)(C)C1.C12(CC1)CC(=O)N(C)C2 C#CC1CC2(CC(C(N3CCCCC(NC(=O)CC(C)(C)C4CC4)C3)=O)C2)C1 Cn1nc(Br)c2ccc(C(=O)NC3CCCCN3)cc12.c1(N)ccc2nc(O)[nH]c2c1 C1(O)(C(C)NC(c2cnn[nH]2)=O)CCN(C(=O)CC2C=CS(=O)(=O)C2)CC1 c1(C(N2C(C(N(C)Cc3c(C)occ3)=O)CCCC2)=O)ccc2cc[nH]c2n1 c1(OC)ccc2cc(C(N3CCCC(CNC(C4CC4F)=O)C3)=O)ncc2c1 c1(C(=O)NCCCN(CC(=O)NC)CC)ccc(CCC(N)=O)cc1 N1(C(=O)CC=C(Cl)Cl)CCN(C(=O)C(O)CF)C(C2CC2)C1 c12cnn(c1)CNC(=O)C2.N#CC(C(=O)NCCNC(=O)OC(C)(C)C)C1CC1 N1(C(COCCCOC)=O)CC2C(NC(=O)COCc3ccncc3)C2C1 c1(C(N2CCCC2CN(c2ncccn2)CC2CC2)=O)cc(Cl)ncn1 CC#CCC(C(=O)N(C1CC(C)CC(C)C1)C)NC(C1CCCCC(=O)C1)=O CCCCC(CC)CC(C(=O)NCC)N1CCOC(CC)(CC)C1 Cc1ccc(NCC(=O)N(C(C)CCNC(=O)CC2CC(C(F)F)C2)C)cc1 Cc1cc(C)c(CC(=O)NC(C)CN(C)C(c2cnc3nccn3c2)=O)c(O)n1 C(C)(CCCCNC1CN(C2COC2)C1)N(C(=O)CCC(C)c1ccccc1)C N1(C(c2cc(C)[nH]n2)=O)CC2CCOC2(CNC(=O)C(C)(C)CC(F)F)C1 N1(C(c2ccc(CC)nc2)=O)CC2CCCC1C2CNC(C1(C(C)(F)F)CC1)=O c1(OC)cccc(C(=O)NC(C)C(C)(C)NC(=O)CC2CC(F)(F)C2)n1 c1(C(=O)NCC(C2(O)CN(C(c3cnco3)=O)C2)(C)C)ccccc1C1CC1 N1(C(C(C)=CC)=O)CC(NC(=O)C(O)Cc2ccccc2)C(O)C1 c1(C(=O)NCC(=O)N(CC(C)NC(=O)CC2CCCC2)C)cccn2cnnc12 Cc1cc(C(=O)OC(C)C)nn1CCO.C(C)(C(=O)OCC(=O)O)NC(N)=O CC1(C)CN(C(c2cncnc2)=O)CC(C)(C)C1NC(c1n[nH]c2c1COC2)=O Cc1cc(C(=O)NCCCN(c2ncc(Br)c(O)n2)C)cc(O)n1 C=CCC(CNC(c1cscc1C(C)C)=O)NC(C1CC1C)=O Cc1nc(O)[nH]c1C(N1CC(C(C)(C)O)(CNC(c2cc(O)ncn2)=O)C1)=O c1(C(=O)NC2C(CNC(CCn3ccc(C)n3)=O)C2)ccc2c(c1)C(=O)CCC2 C1(CNC(=O)NCC(CN(CC)CC)F)CCCN1C(C)=O C1(NC(C(C=C)O)=O)CCN(c2ccnc(C(C)CC)n2)CC1C CCCCC(C(=O)N(CC(O)CN(C)C)C)N(C1CC(C(=O)OCC)C2C1C2)C C(C(C)(O)CNC(=O)C(Cn1cncn1)NC(=O)CCCNC(C)=O)OC C1(C(=O)NC2CN(C(CCCCSC)=O)C2)CC(C)(C)CCO1 C#Cc1ccc(C(=O)NC2CCC2CC(=O)N(C(C)C(N)=O)CC)cc1C C=C(C)C(C)(C)C(=O)N1CCC(C=CC(N2CCC2C(N)=O)=O)CC1 N1(C(CC2(C=C)CC2)=O)CCCC(C2CCN(C(=O)C3=CCC3)C2)C1 C1(NCCNC(CCCCCCC)=O)CCc2nc(N3CCOCC3)ncc2C1 N1(CC(=O)NCCC(C)NC(=O)C(C(C)(C)C)N(C)C)CC(=O)N(C)C1=O N1(C(C(c2ccccn2)C)=O)CC2CCCC2(CNC(=O)C(O)CNC(C)(C)C)C1 C(C1=NOC2CN(C(=O)C=CC=C(Cl)Cl)CC12)OC.C12(CCC1)C(=O)NC2 CON=CC(=O)NC(CNC(C1CC1(F)F)=O)C1CCC1 Cn1ncc(C(=O)OC2CCC(OC3CCC3)CC2)c1C(F)(F)F c12cccc(c1)N2.C1(NC(C=CCCC)=O)(CO)CCOC1.c1(=O)c(=O)[nH]1 C(CCN=C(NCC)N1CCC(F)(c2cc(C)cc(F)c2)C1)=CC=C Cc1ccoc1S(=O)(=O)NC(C1CCNCC1F)=O C(=O)(C(C)(O)CNC(=O)C(c1cnn(C)c1)NC(c1nnsc1C)=O)OC C(=O)(C(CC(F)(F)F)c1ccccc1)N1CC2C(COC(C)(C)C)C2C1 c1(C2N(C(c3nccc(Cl)c3F)C(=O)NCCOC)CCC2)c(C)cc(C)cc1C C1(CNC(N2CC(C(=O)NC)C2)=O)CCC(=O)N(C)C1=O c1(OC)cc(C(=O)NC2CCCCN(C(c3ccsc3)=O)C2)c([N+](=O)[O-])cc1F CON=C(C(=O)N1CCOCC(NC(=O)C(c2ccccn2)C)C1)c1ccco1 C1(NC(CC2CC(CC)C2)=O)CCC(NC(=O)CC(c2ccc(F)cc2)O)CC1 N1(C(=O)OC(C)(C)C)CC=C(C(C)(C)C(=O)Nc2[nH]nc3c2CCCC3CCO)C1 c1(N(C2CN(C(C(C)n3cnnn3)=O)C2)C)ncncc1Cl c1(C(=O)NCCC(=O)NC2CC3CCCC3C2)ccc2ccccc2c1 C12(C(=O)NC3CCCN3C(=O)OC)CCC(NC(CCC#C)=O)(CC1)CC2 C1(CC(=O)NC2CC(CCNC(C(CC)F)=O)C2)Cn2ccnc2NC1=O c1(CC(N2C(CCCNC(C3CC=CCO3)=O)CCC2)=O)ccc(O)c(F)c1 c1(C(=O)NCC2CC(F)(CNC(C(CC)C(=O)OC)=O)C2)cc2scc(C)c2[nH]1 C1(C(C)=O)CC(C)CN(Cc2cn(-c3cn(C)nc3I)nn2)C1 c1(C(N2CC(CC)C2C(N2CCCC(O)C2)=O)=O)c[nH]c2c(OC)nccc12 C(=O)(C1=CS(=O)CCC1)NC1C(NC(C2(OC)CCCC2)=O)CCC1 C(=O)(CC1=CCCCC1)N(CCC(N1CCCC1C1CC1)=O)C.CO C1(OC)CC(C)CN(C(C2(N(C)C(c3[nH]cnc3C)=O)CC2)=O)C1 c1(C(=O)NC2CC(CNC(C(C=C=C)C)=O)OCC2)ccc(Cl)cc1C N1(C(CSc2nc(C)[nH]n2)=O)CCC(C(F)F)(CNC(=O)C(C)CC2CC2)C1 c1(OC)cc(F)ccc1C(N1CC2CC2(CNC(=O)CSc2nc[nH]n2)C1)=O C1(C)(CC)CC(NC(c2cc(-c3ccoc3)on2)=O)CN1C(c1cccn1C)=O C1(CNC(CC(=O)NCC#C)=O)CN(C(=O)CCCN(C)N=O)C2(CCCC2)C1 C1(CNC(C#CC(C)C)=O)(NC(=O)CN(C)S(N)(=O)=O)CC2CCC1CC2 C1(CC)(NC(=O)CCCCCCN)CCCN(C(c2cc(C3CC3)[nH]n2)=O)C1 C1(SC)CCC(C(N2CC(CCO)(NC(c3cnc(C)cn3)=O)C2)=O)CC1 c1(NC(Cc2c(C(C)=O)cccc2)=O)ccc(NC(c2ccco2)=O)cc1Br C1(NC(C)=O)CC2(CCCN(C(=O)COC(c3ccc(COC(C)C)o3)=O)C2)C1 C12(CCNC(=NCCC)NC3CC3COC)CC3CC(CC(C3)C1)C2 CC(CC(=O)NC12CC(C(N3CCC(N(C)C)C3)=O)(C1)C2)CC(C)(C)C C(=O)(C(F)CC(C)(C)C)NCC1CC(CNC(c2c(CCC)cccc2)=O)C1 c1(C(=O)NCC(F)(F)Cl)ccc(F)c(Br)c1F C1(C(=O)NC(C)CNC(=O)CCCCN2CCOC2=O)Cc2cccc(F)c2O1 c1(C(C)=O)nc(Cl)cc(=NCC2CCC(Nc3cc(C)nc4ncnn34)C2)[nH]1 C=CC1(C(=O)NC2(CNC(=O)CC(C)(C)C3CC3)CCCC2)CCOCC1 c1(NC(=O)NCC2(C)CCCC2)c[nH]c2cc([N+](=O)[O-])ccc12 c1(C(=O)NCCCC2(NC(C3ON=C(C)C3)=O)CC2)cccc(C)c1F C1(CNC(C(CC)C)=O)CC2CCC(C1)N2C(C12CC(CCC(F)(F)F)(C1)C2)=O C1(C)(C(NOCC(=O)NCC2CC(N(C)C)C2)=O)CC=CC1.C(COC)S c1(C(N(CCN(C(c2ncoc2C)=O)CC)CC)=O)cnc2sccc2c1 CN1CC(C(=O)NCC23CC(NC(c4csc(Cl)n4)=O)(C2)C3)CC1=O C(c1nc(C)co1)=CC(=O)NC(CCCNC(CCCn1ncc(C)c1)=O)C Cc1noc2cc(C(=O)NCCC3(O)CN(C(c4cnn(C)c4)=O)C3)cnc12 C(=O)(C#CC1(C)CC1)NCC12CC(CNC(c3c(C(=O)OC)cccc3)=O)(OC1)C2 C1(C(=O)OC)CN(C(CN(CCC#C)C)=O)CC1NC(C)=O.C12CCN(C1C)C2=O C=CC(C)(O)CC(=O)NC(CO)C(C)NC(C1CCOC1)=O N1(C(c2cnc(COC)s2)=O)CC2(C1)CN(C(=O)C(C)NC(=O)C(C)(C)C)C2 Nc1cc(C(=O)NCCCOCCCNC(C2CC2C2CCC2)=O)nc(O)c1Cl CC(C)(C)C(=O)C1(C(=O)N)CCC1.c1(C(N2CC(C)C2)C2CCCO2)cccnc1 CCC(C)(C)C(=O)C(=O)NCC1(C(=O)Nc2cccc(F)c2C)CCC1 c1(C(CC)C)cn2c(n1)CN(CCC(C)(C)N(C)C)CC2 c1(C(CCC)OC(=O)C(C)N(C(=O)C(C)C)C)ccc(Cl)cc1 CCC(O)C(C)C(=O)NCC1CC1CNC(c1n[nH]cc1Br)=O N1(C(c2c(CCC)occ2)=O)CCC(F)C(NC(=O)C(=C2CCCCC2)F)C1 CC(CC(F)F)C(=O)NCC1CC(F)CN1C(c1coc(CO)c1)=O c1(C(=O)NCCN(C)C)cc(Cl)cc2c1CCC2.c12ccc(cc1)oc2=O CN1CC2(CC(NC(c3occc3CNC(C3CN(C4COC4)C3)=O)=O)C2)C1 N1(C(CCNC(=O)OCC)=O)CCCC(N(C(=O)C(C)(COC)OC)C)C1 C1(NC(CCC=CCC=C)=O)(CF)CCN(C(c2snnc2C2CC2)=O)C1 C1(CNC(C(CC)OC)=O)CC2CCC1N(C(c1ccc(C#N)c(Cl)c1)=O)C2 N1(C(C(C)OCC=C)=O)CCC(C(=O)N(CCC(=O)NC2CC2)C)CC1C.OCC CCC(C#N)(CC)C(=O)NCC1C=CC(NC(=O)C(C)Cc2ccncc2)C1 C(CCN(C(=O)C(C)OCCOC)C)(C(C)(C)C)NC(C(COCC)(F)F)=O C1(CNC(c2c(C)nc(Br)o2)=O)CN(C(=O)OC(C)(C)C)C2(CCC2)C1 c1(C(N2CCCN(C(c3c(C)n(C)nc3)=O)CC2)=O)csc2ccccc12 Cc1[nH]c(CNCc2ccc(Br)nc2F)c(C)c1-c1ccc(OC(=O)C2CC2)cc1 c1(NC(C(c2cn(C)nc2)NC(=O)CNc2ccccn2)=O)cnn2c1OCC2 C12(C(=O)NCC#CCNC(C(C(C)C)NC(C)=O)=O)CCCN1CCC2 N1(C(CCN(CC)CC)=O)CC(N(C)C(c2ccc(C)cn2)=O)C(O)C1 c1(C(=O)NCCC(C)(C)NC(C2CCN(C)CC2)=O)c(O)ccc(Cl)c1F c1(OC)ccc(C(=O)NC(C)(C)CC(=O)NCC(C)(C)C#N)cn1 c1(OC)ncc(NC(C2CN(C(=O)C(F)(F)C3CC3)CC2(F)F)=O)cc1C c1(C(=O)NC(CC(C)NC(c2n(CCC)ncc2)=O)C)cc(F)cc(F)c1 N1(C(C2CC(N(C)C)C2)=O)CCC(C(=O)NC2CCCCCC2)C(O)C1 N1(CC(C)OC2CCCN2C)CCC(CN(C)C)CC1 C1(CCC)CCN1C(C(=O)NC1COC1)c1cccs1 N1(C(c2n(C(C)C)ccc2)=O)CC(C2CCCN(C(=O)CC3CCOC3)C2)C1 CC1(C)CN(C(=O)CC23CC(C2)C3)CCC1NC(=O)C=Cc1nc[nH]n1 c1(C(N(C2CCN(C(C3COC(C)C3)=O)C2)CC)=O)cc2occc2[nH]1 C#CCC(CC#C)C(=O)N1CC(c2nnc(C)o2)C1.C1(Cc2cnc[nH]2)C(=O)N1 C=CC1(CC(N2CCC2CO)=O)CN(C(c2ccccc2C)=O)C1 c1(C(=O)NC2C(N(C)C)CN(C(=O)C(=O)N(C)C)C2)nc(Cl)ccc1N c12cccc(c1)NC(=O)Cc1cn(nn1)CCCO2.O=C(O)CCCC(=O)O c1(C(N2CCCN(CCNC(=O)CCCCCF)CC2)=O)cc2n(c1)CCCC2 CN1CC(C)(C)CC1CC(N1CCCC(O)(CNC(C2CCC=CCC2)=O)C1)=O C1(C(N(CC(=O)NC(c2ccccc2)CF)C)=O)CC(C)(C)C1 c1(C(=O)NCC(CN(C(=O)CCC2CCC(=O)N2)CC)(C)C)cc(O)nc(Cl)c1 C1(NC(C(C)(C2(C)CC2)OC)=O)CCC(CCC(=O)N(CCCO)C(C)C)CC1 C(CC(=O)NOCCC1CC1)C1CCN(C(c2c(C)cns2)=O)C1 C1(CNC(CSCCN(CC)CC)=O)C(C)CCN1C(=O)CCC(=O)NC C12CCC(CC1)CC1N(C2C(=O)NC)CC1.C(C)(C)(C)OC(CC(F)F)=O CC1C(NC(=O)CC2CCCCCCC2)CCCN1Cc1ccsc1 CC1Cc2cc(Br)ccc2CN1C(c1ccc(=O)n(-c2ccccc2F)n1)=O N(C(=NCc1ccnn1C)NCC1(SC2(C)CCCOC2)CCC1)C(C)C1CC1 C1(NC(CC(=C)C)=O)CCCCC12CCN(C(=O)C(F)CC)C2 N1(CC)CCN(C2(C(=O)Nc3cnc(C(C)=O)cn3)CCC2)CC(O)C1 c1(C(=O)NC2CC(O)(CNC(C(C)C#N)=O)C2)ccnc(CN(C)C)c1 C1(NC(COC2CN(C(C)=O)C2)=O)CC2CCC1N(C(=O)C(F)n1ccnc1)C2 C1(N(C(=O)Cn2ncnn2)CCF)COCC1NC(=O)C=CCN1CCCCC1 C1(CNC(C(C=C)OC)=O)CN(C(=O)Cc2cnn(C)c2)CC1(F)CO CCCC(C(=O)NCC1CCCCN1C(c1oc(C)nc1CC)=O)OCC C1(CNC(C=C(C)C)=O)CCC(C)(C)CN1C(=O)C(c1ccccc1C(F)(F)F)O c1(C(C(N2CC3C(O)C3C2)=O)F)cc(I)cc(I)c1 c1(N2CCC(NC(c3ccn(CC)n3)=O)C23CCC3)nc2ccc(OC)nc2s1 CC(CO)(CO)C(=O)NCC1(O)CCN(C(c2ccc(-c3ccncc3)o2)=O)C1 C=Cn1ncc(C(N2CCC(C(=O)NCC3(C)CCC(=O)N3)C2)=O)c1N C(=O)(CCCCC(=O)NC1CC(F)(CNC(=O)CC2CCC3(CCC3)O2)C1)OC C=CCN=C(NCC(CC)C(C)C)N(C)Cc1nnc(SC)s1 N1(C(CCNC(C)=O)=O)CC(NC(c2nccnc2N)=O)CC(C)C1 N1(CCC(=O)NC(C(C)C)(C)CNC(C2(C)CC=CCC2)=O)CCP(C)(=O)CC1 C12(C(=O)NC3CC(C#C)C3)CC(COC)(CN1C(=O)CC=C(C)C)C2 CC1(C)CN(c2ccn3ccnc3n2)CC(CNC(=O)Cc2ccsc2)O1 c1(CC(=O)NCC(CC)NC(=O)C=CCN(C)C)ccc2nsnc2c1 c1(C(=O)NCCCN(C(=O)Cc2cncnc2)C)nccc2ccn(C)c12 C1(NC(CC2C(CC)C2(F)F)=O)CCCN(C(=O)CSc2n[nH]c(O)n2)CC1 c1(C(C)N(CC(C2CCOCC2)N)CC2CC2)nccn1C c1(CC)nc(C(=O)NCC(CNC(C2CCN(S(C)(=O)=O)C2)=O)OCCO)co1 C1(Nc2c(C)nsc2)CCCN(CC2CCCOC2)C1 c1(C(=O)NC2CCCC(CNC(C(CC(=O)OC)C)=O)C2)ccc2nonc2c1 c1(CC)cn2c(n1)CCC(C(=O)NCCCc1nnc3n1CCS3)C2 C(=O)(CS(=O)CCC(F)(F)F)NC1CCCC(NC(c2c(C)cc(Br)o2)=O)CC1 N1(C(c2c(CC)ocn2)=O)CCCC2CN(c3cnc(C#N)c(C#N)n3)CCC12 C1(NC(C2C(CCC)CCC2)=O)CCCC12CN(C(=O)C(C1CCCC1)OC)C2 c1(C(=O)NC(CN(C(C2C(C)C2C)=O)CC)C)cc(C(F)(F)F)ccc1Cl c1(C(=O)NCC2C(NC(c3coc(Cl)c3)=O)C2)cc2ccc(Cl)cc2s1 c1(-c2cncc(C(=O)NCCCCC)c2)c(OCOC)cccc1F Cc1occc1C(=O)NCCCOCCN(C)C(C1CC(C)(F)C1)=O C1(NC(c2cccc(C)n2)=O)COC2(CCCN(C(=O)C(O)CN(C)C)C2)C1 c1(C(=O)NCC2N(C(c3cc(CCC)oc3C)=O)C3C(C2)C3)cncc(Cl)c1Cl N1(C(CCSCCCC)=O)CC2COCC(C1)C2NC(=O)C=CC1CCOCC1 C1(C(=O)NC(CCOC)CNC(c2occc2CN(C)C)=O)CCN(OC)CC1 Cc1ccc2nonc2c1C(=O)NC1(CO)CCN(C(C2CCOC2)=O)C1 C1(CC)CN2CCC1NC2=O.c1(NC)sc(Br)nc1C1CC1 c1(C(N(C)CC2(CNC(C3CC3(F)F)=O)CC2)=O)ccc(=O)n(CCF)n1 N1(C(c2c(C(C)C)ncs2)=O)CCC(C(F)(F)F)C(CNC(C2(F)CC2)=O)C1 Cc1cccc(-n2nnc(C(=O)NC3CCN(C(=O)CSC(F)(F)F)C3)c2C)c1 N12CC3CC(C1)N(C3)C(=O)CSCc1ccc(cc1)C2=O.c1(CC)ccccc1 C1(N(CC(=O)NCCCCOC)C(C2C(CCC)C2)=O)CCCCC1 c1(C(=O)OC)ccc(Br)cc1S(=O)(=O)N1CC(c2cccc(F)c2)C1 c1(CC(=O)NC2C(CNC(C(C(CC)O)C)=O)CCCC2)noc2ccccc12 CCCC(CCCNC(C1(N2CCOCC2)CCCC1)=O)NC(C1C2COCC12)=O C(CC(C(=O)NCC1COCC(C)O1)NC(C1COCCN1C)=O)SC N1(C(c2nn(C)c(F)c2)=O)CC(C2CN(C(C3CC3c3ccnn3C)=O)C2)C1 c1(C(=O)NCC2CCN(C(=O)C=C3CCCCC3)CC2)ccc(OC(F)F)c(F)c1 c1(-c2cn(CCC(=O)NCC(C(=O)NC)C(C)C)nn2)cccc2nc(O)[nH]c12 N1(C(C(CCC)F)=O)CCC(C(=O)N(C)CCC2CC2)C12CC2 C1(CC)CCN(C=O)C1(C)C.C1(C(=O)OC)CC1C1CCC1 c12ccc(nc1)OCC(=O)N2.C1(C(CNC(C)=O)OC)CCOCC1 c1(OC)ccc(F)cc1C1CCCN1CC(C1CC1)C(=O)O c1(OC)cccnc1C(=O)N.N1(C(c2c(C)occ2)=O)CCOCC1CN(C)C C(C(C(=O)N(C(CO)C(C)C)C)C(C)C)NC(C(COC)COC)=O Cc1ccc(CN(C(=O)CCOCCNC(C2CCCCO2)=O)C)nc1 N1(C(C(=O)NC(c2ccc(Cl)s2)COCC)=O)CCC(CC(C)C)CC1 c1(C(N(C2CN(C(CC(COC)C)=O)CC23CC3)C)=O)ccc([N+](=O)[O-])n1C N1(C(c2ccnc(Cl)c2F)C(=O)NCc2cccnc2)CCOCC(C2CC2)C1 C(=O)(C#CC1CCOCC1)N(CCCCC(=O)NCC1(O)CCCOC1)C c1(CNC(C2(CC)COC2)=O)cnn2c1CN(c1ccc(C(F)(F)F)nn1)CC2 C1(N(C(c2cnc(CC)o2)=O)C)CN(C(C2CCCN2C)=O)CC1(C)C c1(C(=O)NCC2(CNC(=O)C(F)F)CC2(F)F)ccc2c(c1)COC2=O CC(C)CCC(F)C(=O)N1CC(N(C(=O)CCc2ccncn2)C)C(F)C1 c1(C(=O)NCCCC(C)NC(C=C(C)c2ccsc2)=O)cccc2nsnc12 N1(C(C2OCCN(C)C2)=O)CCN(C(C2(F)CCCCC2)=O)CC1C1CC1 c1(C(N2C(CC(N3CCOCC3CO)=O)CCC2)=O)cc2c(F)cc(F)cc2[nH]1 C1(NC(c2ccnc(C)n2)=O)CCN(C(C2CCC2)=O)C12CCC2 n1(CC(=O)NC2C(CNC(c3c(COC)noc3)=O)C2)cnc2ccc(C)cc12 N1(CCCN(CCOC)CCO)CCN(Cc2ccccc2C)CC1 c1(C(N(CCOCCN(C)C(=O)C2CC2)C)=O)cc2c(F)cccc2[nH]1.C1(=O)CN1 C#CCC(C)(CC)C(=O)NC1CC1NC(=O)CCCC#CC C1(C(N2CCC(CF)CC2)=O)C2CC(NC(=O)C(F)(F)C3(O)CCC3)CC12 C=CCCCCC(=O)NCCc1n[nH]cc1C(=O)N(C)Cc1ncn(C)n1 c1(N2CC3ONC(=O)C3C2)nc(N2CC3CC2C2CC32)c2ccsc2n1 C(CCN=C(NCCOCCOC)NCc1cncs1)OC C1(NC(CC)=O)C(C)CCN(C(=O)C(CC)n2ccc(C3CC3)n2)C1C C1(CC(N)=O)CCCN(C(=O)N(CC2CC2)CC2CCC3(c4ccccc4)CC23)C1 Cc1ccnnc1C(=O)N(CC(CO)(CO)NC(C1CCSC(C)C1)=O)C C1(NC(Cc2c(OC)nccc2)=O)CCN(C(c2cccc(F)c2N)=O)CC1F N1(C(Cc2c(C)noc2C)=O)CCOCC(C(=O)NC(C)CCO)C1 C1NC(=O)COC1.C(C(C)(C)NC(C)(C)C)N(S(C)(=O)=O)C N1(CC(C2CCC2)NC(c2cnn(C)n2)=O)CCCS1(=O)=O c1(NC(c2csc(NC(c3ccc(Br)nc3)=O)n2)=O)cccc2ncsc12 c1(C(=O)NCCSCC(=O)N(CC(C)OC)C)ccc(=O)n(C)n1 c1(C(N2CC(N(C(=O)C(C)(F)c3ccccc3)C)C2)=O)ccccc1OC(F)F C(CC(C(C)C)NC(=O)CCCCn1ccnn1)OC.C(=O)CCN(C)CCO C(=O)(C(CNC(=O)CC(C)C)CC1CCCC1)NC1(CC=C)CC1 C(=O)(CCCN=[N+]=[N-])N1CC2C(CNC(C(C)OCC3CCCO3)=O)C2C1 c1(C(N2C3(CCN(C(C4C(C=C)C4)=O)C3)CCC2)=O)ccnc2cc(F)cnc12 N1(C(CCC)=O)CCC12CN(C(=O)CC1CSCCO1)C2 C1(C(N2C3CN(C(C4(O)CCCCC4)=O)C(CC3)C2)=O)COc2ccccc2O1 CC(CN(C)C)CC(=O)N(C1CCN(C(c2cc(CO)[nH]n2)=O)C1)C C1(C(N(C(CC)C2CC2)C)=O)CC1C1CN(C(C2(C#N)CCOCC2)=O)C1 C(=O)(CC1=Cc2ccccc2C1)NCCNC(C(C1CCC(=O)N1)C)=O C1(OC)CCC(NC(C2(NC(c3nccn3C)=O)CCSC2)=O)CC1 C1(NC(CN(CC(C)(C)C)C)=O)CCCN(C(C2(OC(C)C)CC2)=O)CC1CO c1(C(=O)OC)ccc2c(c1)CN(C(C1(C#N)CCC1)=O)CC2 C1(C2CN(C(C3Cc4cscc4C3)=O)C2)(NC(c2cc(C3CC3)ns2)=O)CC1 c1(C(N(C(CSC)C)C)=O)c(CNC(C2(C#N)CCCO2)=O)nnn1C c1(C(N2C(CCCCC(=O)N3CC4CCC3C4)CCC2)=O)cccc2c1CCC2 c1(C(=O)NCC(C)(O)CNC(c2coc(Cl)n2)=O)cnc2c(=O)[nH]ccc2c1 C(=O)(C1Cc2ccccc21)N1CC(C)CC(C(=O)NCC(C)OC)C1 n1(C(C)C)nc(C(N2CC3(NC(C4CCS4(=O)=O)=O)CC2C3)=O)cc1C(N)=O N1(C(c2cc(OC)nn2C)=O)CC2(CC(C(=O)Nc3cnc(Br)cc3C)CO2)C1 C=CCCCC(C(=O)NCC1=CCN(C)CC1)NC(=O)C(n1ccnc1C)C C1(NC(C2CCCO2)CC)CCC2(CCC2)C1.c12nnnn1C2 N1(C(C(C)SC(C)C)=O)CCC(NC(=O)C(C)OCCC(C)C)C1C c1(CC)c(C(=O)NC2CN(C(c3cncnc3)=O)CC2(F)F)cccc1Br C(=O)(CC(F)(F)F)N(C)Cc1cccc(CN(C)C(c2nnnn2C)=O)c1 C(=O)(C(C)C(C)NC(=O)CC1COCCO1)NCCc1cn(CC)nc1 C(CCCCC(=O)N(C(C(=O)NCC(c1cccnc1)O)C1CC1)C)OC C1(OC)(CNC(C2CC(SC)C2)=O)CCN(C(=O)CSc2nncs2)CC1 N1(C(=O)NC2CCN(c3ncccn3)C2)CCCC(Cn2ccnc2)C1 C1(NC(C(c2cnn(C)c2)NC(C(C)C2CC2)=O)=O)CCCC(O)C1O C=CC(C(=O)N(C)CCOCCNC(c1n[nH]cc1F)=O)c1ccccc1 c1(C(N(C(C(=O)NC(CC#C)C(N)=O)C)CC)=O)ccc(C=C)cc1 C1(NC(CC=CC=C)=O)CN(C(=O)CC(C)F)C2(CCCCCC2)C1 N1(C(c2c(C)cco2)=O)CCC2CCN(C(=O)CCCc3cccnc3)CC2C1 OC1c2ccccc2CC1N(c1ncnc(NCc2ccccc2)n1)CCO C12(CNC(C(c3ccco3)OC)=O)CN(C(=O)COCC3CC3)CC1CCO2 c1(CC)cc(OCC(=O)NC2(C)CCN(C(=O)CC=CC(C)(C)C)C2)ccc1Cl CC1C(=O)CCC1CC(N1CCC(CN(C(=O)C(C2(O)CCCC2)F)C)CC1)=O Cc1ccc(SC(C)C(=O)NCCC2CCN(C(c3ns[nH]c3=O)=O)CC2)cc1 Cc1nc(C)c(C(=O)NCCC(O)CNC(c2ccc(-c3cscn3)nc2)=O)s1 c1(C(=O)NCC2CCC(C)N(C(c3ccoc3)=O)C2)cc2sccc2cn1 C(=O)(N1CC2COCC2O1)C1N(C(CC(C)F)=O)CCCCC1 Cn1cc(NC(=O)CC2CNC(C)(C)C2)c(O)nc1=O C(N=C(NCc1cnc(C(C)O)s1)NC(C)C)C1CCN(CCOC)C1 c1(NC(C(c2n(C)ccc2)=O)=O)ccc([Si](C)(C)C)cc1.C12CN(CCS1)C2=O C(=O)(CN=c1ccnc(NCC)[nH]1)N(C)CCn1cc([N+](=O)[O-])cn1 N1(C(CC(C)N(C(c2nc(CC)oc2)=O)C)=O)CC2CC(C1)C2(C)C c1(C(=O)NCC(c2ccccc2)CNC(C(F)=C(C)C)=O)cc(C)c(C)[nH]1 C1(C(=O)NC2(CF)CCN(C(c3cccc(Cl)c3F)=O)C2)C2CCC(F)(F)C12 c1(C(=O)NC2(C)CCN(C(=O)CN3CCCC3)C2)ccnc2c1CC(=O)N2 c1(C(N(CCNC(=O)CCn2cc([N+](=O)[O-])cn2)C2CC2)=O)cc2sc(Cl)cc2[nH]1 N1(C(c2c(OC)nn(C)c2)=O)C(C)C2CC1C2NC(=O)CCc1nc(C)c(C)[nH]1 C1(C(N2CC(=CC)C2)=O)CC(C)N1C(C1(C)CC=CC1)=O C1(C(=O)NCCOCC(N2C(C)(COC)CCC2)=O)CC2CC1CC2O N1(C(CCC=CC)=O)CCC(CCO)(CO)C1 C(C(C(=O)N1CC(C)(C)CC1C)C(C)(C)C)NC(c1c(OC)scc1)=O C(CN=c1[nH]c(=NC2COC(N(C)C(C)=O)C2)[nH]c2c1COCC2)SC C1(CNC(C(C)CO)=O)CCC2(CCC2)C1NC(c1ccc2occc2n1)=O C1(C(=O)NC)CC2CCC1N(C(=O)OC(C)(C)C)C2.N1C(=S)NCC1 C12CCCCN1C2=O.C(=O)(C(C)N(C)C1CC1)NCCC1(OC)CC1 c1(C(=O)NC2CN(C(c3cnn4ccsc34)=O)CCC2O)nc2cnccc2s1 c1(CNC(C(N(C(COC)=O)C)C(C)C)=O)cc(CO)n(C)n1 C1(CNC(c2ccoc2)=O)CCCCN1C(=O)C(c1ncccc1Br)(F)F C1(NC(C(C)n2cccn2)=O)CC2CC1N(C(c1ccn(C)c1)=O)C2 c1(CC)c(C(=O)NC(CN(C)C(c2cnco2)=O)(CO)CO)cccc1C C(=O)(CCCC(CC)CC)N1CC(C#C)(C(N2CCC(OCC)C2C)=O)C1 C1(CNC(CCC#CC)=O)CCCCCN1C(=O)CNC(=O)Nc1ccccc1 C1(CC(=O)NCC(COC)O)CC(C)(C)CN1C(=O)CC1CNC(=O)C1 C1(C(N(CC(CNC(CCOCC)=O)C)C)=O)CCCCC1n1cccc1 C1(CCOC)CN(C(=O)CSCCC(F)(F)F)CCN1C(c1nc(=N)cc[nH]1)=O C1(NC(=O)CN(C2CCCC2)Cc2cn(C3CCCCC3)nn2)CC2CCC1O2 CC1(C)COCC(C(N2CCC(CCNC(c3cc(Cl)ccc3F)=O)CC2)=O)O1 C1(CNC(c2c(CC)nns2)=O)CC2CC(C1)N(C(c1c[nH]nc1F)=O)C2 c1(C(C)=O)cc(C(=O)NC2CC2CNC(=O)CSc2nccn2C)co1 N1(C(c2c(I)ccc(C)c2)=O)CCc2cc(-c3ccnc(C)c3)ccc2C1 c1(CNC(CN2C(C)CC2)=O)csc(CNC(=O)CCC2CCCO2)n1 N1(C(c2cc(C)[nH]n2)=O)CCN(C(=O)C(C)SC(F)(F)F)CC1c1ccccn1 c1(OC)ccc(CNC(=NCCOC)NCC2CCC(=O)N(C(C)C)C2)c(C)c1 N1(C(c2c(=N)[nH][nH]c2)=O)CCC2(CCC2)C(NC(C2CCCC(F)(F)C2)=O)C1 c1(C(=O)NCC2=CCN(C(c3c(C)nc(N)cn3)=O)CC2)cccc2nn[nH]c12 N1(C(CC=C=C)=O)CCCC2CN(C(C3(OCC)CCSCC3)=O)CCC12 Cc1cnnc(O)c1C(N1CCC2(NC(C3CCC(C(N)=O)CC3)=O)CC2C1)=O C1(COC)C=CCCN1C(=O)C=CC(C)NC(C1(COC)CCCCO1)=O S(=O)(=O)(c1cc(C(=O)N=c2ccn(C3CC3(F)F)[nH]2)ccc1Cl)NC(=O)CC1CC1 CC(C(=O)OCc1ccccc1)C(C)NC(=O)OC1CCCC1 c1(CC)ccc(C(=O)NC2CC(C)N(C(=O)CCC(C)CN(C)C)C2)c(C)c1 NC(=O)CCCCC(=O)NC(CC1CCCC1)C(=O)NCC(=O)NCCO CCC(C(=O)N(C(C(=O)NC(CN(C)C)C(C)(C)C)C(C)CC)C)C(C)(C)CC CC(C)(C(=O)N1CCN(c2nncs2)CC1)C(O)c1ccccc1Cl N1(C(COCC=C)=O)CC(CNC(=O)C(C=C)c2ccccc2)CC1(C)C C1(O)(CC)CCCN(C(=O)CC2COCCN2C(c2ccncc2O)=O)C1 CCC(CC(=O)NCCC(O)C(C)C)N(C(=O)C(c1ccn(C)c1)C)C c1(C(=O)N)ccc(CN2CCCCC2)s1.CCC(=O)NC(C)CNC(=O)OC C(CC1=CCN(C(C2(O)CCCCC2)=O)CC1)NC(CC(C)(O)C1CC1)=O C1(NC(=O)CCn2cccc2)CCCC(NC(c2ccc(C(F)(F)F)s2)=O)C1 CC1(C)CCc2cc(C#N)c(N3CC4CC3(C(=O)Nc3cnc(Cl)[nH]3)C4)nc21 Cc1sc(C(N2CCC(C)(NC(c3cc4sccc4[nH]3)=O)C2)=O)c(C)c1C CN1CCCC1C(=O)NCCOCCNC(C1CC1(F)Cl)=O C1(NC(Cc2cccc(OCC)n2)=O)CCCN(C(C2CCCN2C)=O)C1CC C1(CC=C)(C(=O)NCCCc2ccco2)CCCN1C(c1cn(C)c(C)n1)=O C(C)(C)(CC(F)C(=O)NCC1C=CCC1)NC(C(COC)C)=O C1(c2cn(CCCC(C)(F)CNC(c3c(C)nns3)=O)nn2)CCCNC1=O N1(C(c2ccc(C)c(O)n2)=O)CCC(C)(C)C(CNC(C2CC2C(C)C)=O)C1 N1(C(c2cccc(C#C)c2)=O)CC2CC(C1)CN(C(c1cnn3c1CCC3)=O)C2 N1(C(c2c(C)con2)=O)CC2CCN(C(c3cnn4c3CCC4)=O)CC2C1 n1(CC(=O)NCC(CNC(C2(CC)CCC2)=O)(C)C)nnc2c1CCCC2 Cc1ccc(C(N2CC=CC2CNC(C2(C)CCC(=O)N(C)C2)=O)=O)c(N)c1C N1(C(C2CCC(C)(C)C2)=O)CCOC(C)(CNC(=O)Cc2csnn2)C1 C1(C2(O)CNC2)(C(=O)NC(c2c(C)cccc2)C)CC1 c1(CC(N2CC(OC)(CNC(=O)C=CC(=O)NC3CC3)C2)=O)ccc(Cl)cn1 N1(C(c2c(C)cn(C)c2)=O)CC2CCN(C(c3cnc4[nH]ccc4n3)=O)CC12 C1(C(=O)NC(CC(=O)NCCc2c(C)cncc2)C2CC2)CCOC(=O)CC1 CCC(C)(COC)C(=O)NCCOCC(N1CCCC(O)C1)=O Cc1cccc(C)c1N(C(C(=O)NCC1CCOC1)C1CCOC1)C(C)C N1(C(CCC=C)=O)CC(C)CCC1C(=O)Nc1cccc(C(C)F)c1 c1(C(C(=O)NCC(=C)C)N(C)CC2CSC2)cnn2c1CCC2 c1(NC)ccc(C(=O)NC2CCN(C(C3CC3c3cnc[nH]3)=O)C2(C)C)cc1F c1(C(N2CC3C(CCNC(COCCN(C)C)=O)(CC3)C2)=O)occ2c1CCC2 Cc1cc(CNCC2CC(O)CN(C(=O)Cc3ccncc3)C2)cc(C)n1 Cc1cc(C(=O)NC2CCN(C(C3CCC(=O)N3)=O)CC2C(C)C)c(N)c(Cl)n1 N1(C(c2nc(CC)oc2)=O)CCC(=CCNC(C2(n3nccn3)CC2)=O)CC1 C(N=c1cc(NCc2ccc(Cl)cc2C(=O)NC)nc[nH]1)C1C(CCC)C1 c1(CC(N2CC(NC(CCC3CC(OC)C3)=O)C(O)C2)=O)ccc(F)c(C)c1 C1(C(=O)NC(C)CC2CN(C(=O)CC3CCCSC3)C2)CCn2cncc2C1 CC1=C(C(=O)NCC2CC(C)N(C(=O)CCc3cnccn3)C2)CCCC1 O=C1Cc2cc(CC(=O)Nc3ccc(N4CCC(O)CC4)cc3)ccc2N1 C12(CNC(CC3(C)CC3)=O)CCC(CC1)N(C(c1cn(C3CCOC3)nn1)=O)C2 CC1=C(C)CC(C)(C(=O)NCC2CN(C(C3CCCCC(=O)N3)=O)CCO2)CC1 C1(CC)(NC(c2ncsc2C(C)C)=O)CCCN(C(=O)CCOC2CC2)C1 Cc1nn(C)c(Cl)c1CNC(c1cccc(OC)c1)=O.C12(CCC1)CC(=O)N2 C(=O)(CN=c1ccc(Cl)n[nH]1)NCCC1CCN(C(C(CCC)N(C)C)=O)CC1 N1(C(Cc2n[nH]c(=N)s2)=O)CCCCC(CCC(N2CC(F)CC2CO)=O)C1 c1(CCC(C)C)noc(CN(C(c2csc(Br)n2)C(=O)NCCCO)C)n1.C1(C)CC1 Cc1c(C(=O)NC(C)C(C)n2cncn2)cnc(F)c1Br C(=O)(C(O)C(C)(C)C)N(CCCN(C(=O)CC1CCCOCC1)CCO)C N1(C(C(C)(Cl)Cl)=O)CC2CCC1CC2NC(C1(C(F)(F)F)CC1)=O c1(C(N2CC(NC(=O)C(O)c3ccco3)C3(C2)CC3)=O)cccc2nc(O)[nH]c12 C1(C(=O)NC(C2N(C(CNC(C)=O)=O)CCC2)C)CCN(c2cnn(C)c2)C1=O C1(O)(CNC(C2C(CC(C)(C)C)C2)=O)CN(C(C2CC3CC3C2)=O)C1 C1(C(=O)OC)C(O)C(O)CN1C(=O)Nc1cncc(Br)c1 n1(CC(=O)NC(CNC(c2ccnnc2)=O)C2CCC2)cc(Cl)c(O)nc1=O c1(C(=O)NCCCn2c(C)ncc2)cccc2[nH]ccc12.N12CCC(F)(CC1)C2=O C(=O)(C1=CCC(C)(C)CC1)NCCC1CC(NC(CCOCCC)=O)C1 c1(C(=O)NCC(C2CCCCC2)C)cc(C2CC2)nn1-c1ccc(Br)cc1 Cc1c[nH]c2cc(C(=O)NC3CCN(Cc4c(F)cccc4I)CC3F)ccc12 C1(C(N(C2CCCN(C(C(F)=C(C)C)=O)C2)CC2CC2)=O)CCc2c[nH]nc2C1 C1(CNC(c2cnn(CC3CCC3)n2)=O)CCN(C(c2coc(Br)n2)=O)C1 c1(NC(=O)N(CCOCC(F)(F)F)CC2CCOC2)c[nH]nc1[N+](=O)[O-] CCCCCCCCCC(=O)NC12CC1CN(C(C1CN=C3N=CNN3C1)=O)C2 C12(CN(C(=O)C(C3CC3)C3CC3)C)CC(CO1)N(C(=O)CC(=O)OC(C)(C)C)C2 CC1CCC=C1C(=O)NC1CN(C(c2cc(Br)c[nH]2)=O)C(C)(C)C1 C1(NC(c2c(C)coc2C2CC2)=O)CN(C(c2cnsn2)=O)C2(CCC2)C1 CC(C)(C(=O)N1CC2CC2(CNC(c2c[nH]nc2C(C)(C)C)=O)C1)C(N)=O C1(C)(NC(COCC#C)=O)CCN(C(C2CC2c2ccccc2)=O)C1 C=CC(CCC)CC(=O)NC(CNC(c1ccc(CC)[nH]1)=O)CC(C)C c1(C(N2CCCC(NC(C(CCC)O)=O)C2)=O)ccc2sc3ccccc3c2c1 c1(C(N2CC(C(N3C(c4ccc(C)cc4)CCCC3)=O)C2)=O)cccc(Cl)c1C c1(NCC(CC)(C)COC)ncnc(NCCc2cnccc2Br)c1C C1(CCC(=O)NCCC(=O)NC(C(=O)NC(C)C)C)CCC(C(N)=O)C1 c1(C(=O)NCc2c(C(=O)NCC3(O)C(C)OCC3)occ2)ncn2ccccc12 c1(CC)ccc(C(=O)NCC2CN(C(=O)C(C)C)CCC2C)cc1[N+](=O)[O-] Nc1c(C(N2CCC2CF)=O)ccc(F)c1Br Cc1ccc(C(=O)NCC2C3CN(C(c4nc(Cl)cs4)=O)CC23)c(F)c1F Cc1ccc(CCNC(=O)CN(C)C(c2ccc(C)s2)C)cc1 N1(C(c2cc(CC)on2)=O)CCCN(C(=O)CN2CCCC2CO)CCC1 C(=O)(CCC(C(N)=O)N(C)C(N1CCN(c2cccc(Cl)c2)CC1C)=O)OCC C1(C(=O)NC(C2CCCC2)CNC(Cc2cc(C)sc2)=O)C2CCC(C2)S1(=O)=O c1(NC(c2c(C3CC3)ccc(OC)c2)=O)cccc(S(C)=O)c1 C1(O)(c2onc(CC(=O)Nc3c(C)ccc(OC)c3)n2)CC2(CCC(N)CC2)C1 C1(CNC(C=CC)=O)CCCCCN1C(=O)C(C(C)C)n1ccc(C)c1 c1(C(N2CCCCC(NC(C#CC3(C)CC3)=O)C2)=O)cnc2c(n1)CCCC2 C(=O)(CCCCCC(C)C)NCCCC(C)NC(=O)Cc1ccn(C(F)F)n1 n1(C(=O)NCC2CCC(NC(C3(CCC=C)CC3)=O)C2)ccc2cc(F)ccc12 C1(C(N(CC(CC)NC(c2cnn(CC)c2C)=O)C)=O)C=CC=CC=C1 C1(C)(C(N(C2CN(C(=O)CCCCC#N)CC2O)C)=O)Cc2ccccc2C1 c1(C(=O)OC)c(NC(C2CC(F)CN(C(c3ccc(=O)oc3)=O)C2)=O)cccc1Cl C(=O)(CC1=CCCCC1)N1C(C2(NC(C(c3cccc(C)c3)C)=O)CC2)CCC1 c1(CC(N2CCCC(CNC(C=CS(C)(=O)=O)=O)C2)=O)cccc2ncccc12 C12(CNC(CCOC)=O)CCC(CN1C(=O)CCc1cccnc1OCC)C2 O=C1CCCCC(C(N2CCCCC2CC(N2CCCC2)=O)=O)N1 c1(C(=O)NC23COC(CNC(C4CC4(Cl)Cl)=O)(C2)C3)c(F)cc(F)cc1F Cc1ccc2c(C(N3CC4CN(C(C5CCNC(=O)C5)=O)CCC34)=O)onc2c1 C1(NC(c2ccc(CSCC)cc2)=O)CCCN(C(c2conc2C)=O)CC1F N1(C(c2cccc(C)c2O)=O)CCC2(CCC2NC(=O)CN2CCC2C)CC1 CCC(F)(F)C(C)(C)NC(C1C=CC(NC(C2CN(C3CCC3)C2)=O)C1)=O c1(OCCC(=O)NC2CC2NC(c2cc(Cl)ncn2)=O)ccc(F)c(F)c1F C(=O)(CC(F)(F)CC(=O)OC)N(C1CC(NC(c2c[nH]c(=NCC)s2)=O)C1)C C1(N(C(C=CC=CC)=O)C)CCCN(C(c2cncn2C(C)C)=O)C1 C(N=c1[nH]c(Cl)ncc1Cl)C1CCN(C(c2cnc(C)s2)=O)CC1C c1(C(=O)N(C(C)COC)C)cccc2ccoc12.C#CCC1C(=O)N1 Cc1ccc2c(c1C(=O)NCC(O)CNC(=O)C1=CCCCC1C)CCCN2 C1(NC(CN(CC#C)C(C2CCNC2=O)=O)=O)CC(O)C(O)C1 c1(C(=O)NC2CCC2)cccnc1CNC(C1CCCCC1F)=O CCC(C)(C(=O)NCC1CN2CCC1C2)NC(C1CC2(CC2)C1)=O C1(C(=O)N)CC2COCC12.C123CC(C1)(C2)NC(=O)C=CC(=O)N3.C1CC1 c1(CC(=O)NC2CC(NC(c3cccc4nncn34)=O)C2)ccc2c(c1)COC2 c1(C(N2CC(Nc3ccnc(C)n3)C(F)(F)C2)=O)cc([N+](=O)[O-])c(F)cc1F c1(C(N2CCC(Oc3c(C#N)cccc3)C2)=O)c(Cl)ccc(F)c1F C1(CNC(c2c(C)nsc2)=O)CC2(CCC2)CN1C(c1ccc(F)c(N)c1F)=O C=C(C)C1OCCC1C(N1CCC(CO)(NC(c2cncc(CC)c2)=O)C1)=O CC1=CC(C)=NS(=O)(=O)N1CC(=O)NC1CC2(C1)CC2NC(=O)C(C#N)C(C)(C)C c1(NC(=O)NCCNC(C(C)N(CC)CC)=O)cn2c(n1)CCCC2C n1(CCC(=O)NC2CCN(C(c3c(C)nns3)=O)C23CC3)ccc2ccccc12 c1(C(=O)NCC2CC(NC(COCC)=O)C2)ccc(F)cc1OC N1(C(C(C)=C(CC)C)=O)CCC(NC(=O)Cc2ccc(F)cc2)CC1C N1(C(C=C2CCN(C)C2)=O)CCOC2(C1)CN(C(=O)CCn1cnnn1)C2 N#Cc1c(N2CC3(CN(C(=O)CC4CC5(CCC5)CO4)C3)C2)cccc1F N1(C(C=C(CCC)C)=O)CCCC1C(=O)NCCn1ncnn1 C1(C)(CNC(c2c(OCC)cccc2)=O)CC(F)(F)CN1C(C1CC2CC2C1)=O C(C(O)CC(F)(F)F)NC(CC1CCCC(NC(c2cc(C(C)C)on2)=O)C1)=O N1(C(CC(CC)C)=O)CCCC2C1CCN2C(=O)C=CC=C(Cl)Cl C(=O)(N=c1[nH]n(C)cc1I)NCC(CO)OCC Cc1csc2c(C(=O)NC(C)CC(C)NC(C3(C#N)CCSCC3)=O)ncnc12 N1(C(C2(OC)CC2)=O)CCCC(C(=O)NCc2nonc2C)CC1 c1(C(=O)NCCC(CNC(c2csc(S)n2)=O)O)c[nH]c(=O)c2ccnn12 C1(C(=O)NCC(CC(C)C)NC(=O)CCc2cncnc2)CN2CCC1CC2 C1(NC(C(C)c2ccsc2)=O)CC2(C1)CC(CNC(=O)C=CCO)C2 S(=O)(=O)(c1ccc(C)c(C)c1)N(CC(N1CCCC(NC(CSCC)=O)C1)=O)CC C(c1cc(F)cc2c1OCOC2)=CC(N(OCC)C(C)C)=O c1(COC(=O)C=Cc2ccc(Br)o2)cnc(Br)c(Cl)c1 C#CC1CN(C(C2(C#C)CN(C(=O)CCn3ccnc3)C2)=O)CCO1 C1(=O)CCCC(=O)N2CCCC(CC2)N1.C(=O)(C(C)(C)C)N(C)C C1(C(=O)NCC2CC(F)(CNC(c3c(CC)csc3)=O)C2)CC(OC)C1(C)C Cc1ccc(C)c(C(N2CC(CNC(c3csc(Cl)c3)=O)CCC2C)=O)n1 c1(SC)ccc(Br)c(CN2CC(n3cc(CO)nn3)C2)c1 C1(NC(CC(C)SC)=O)CC2(C1)CC(NC(=O)Cc1c(Cl)cccc1Cl)C2 c1(C(N(CCCO)CC)=O)cccc2c1CCN(Cc1ccc(F)c(F)c1C)C2 c1(C(=O)NCC(COC)NC(c2cc(CCO)on2)=O)ccc(-c2ccco2)o1 N1(C(c2ccn(C)c2)=O)CCC2C(NC(c3cccc(F)c3O)=O)C2CC1 c1(C(c2nnnn2CCSC)NC(CC(=O)NC)C)cc(Cl)c(Cl)n1C N1(C(CNC(CCC)=O)=O)CCCC1C(=O)NCc1ncc(CCO)s1 N1(C(C)=O)CC(O)CC1C(N1CC2(N(C(=O)CSc3ccccc3)C)CC1C2)=O C1(CC)CNC(=O)CN1C(c1sccc1CNC(c1cnnc(O)c1)=O)=O Cc1nn(C)c(N2CCCC2)c1CNC(C1(O)CC(CN)C1)=O N1(C(c2cc(OC)c(Br)s2)=O)CCC(C)(Cc2cncc(Br)c2)CC1 c1(C(C)O)cn(CC(=O)NCC2(NC(c3cc(Cl)no3)=O)CCCC2)nn1 CC(CC1CCC1)C(=O)NCC1CC1C(=O)NCCNC(=O)CO N1(C(C(C=CCCC)O)=O)C2CCC1CN(C(c1cccc(CCO)c1)=O)C2 C(CNC(C1CCOC1C)=O)(C(=O)NCCNC(=O)C1CC1)OC C1(C(=O)NC2C(OC)CN(C(c3cc[nH]n3)=O)C2)CC(=O)NC(=O)N1 C(=O)(C1CCc2c[nH]nc21)NCC1(O)CCN(C(CC(C)(C)C(F)F)=O)C1 c1(CSC)cccnc1C(=O)N(CCNC(C1CC2CCC1C2)=O)C1CC1 C1(F)(C(N2CC(NC(c3cccc(F)c3Cl)=O)C(O)C2)=O)CCC2CCCCC12 C1(CNC(CC(C)(C)SC)=O)CC(C)(C)CN1C(C1CCN(C(C)C)CC1)=O C1(CC(=O)NCC2(NC(C3CC3C(F)F)=O)CCCC2)CCCOC1 C(C(=O)N1CC=CC(NC(C2(OC(C)C)CCCC2)=O)C1)(C(C)(C)C)OC c1(C(N2CCOCC2CO)=O)cc2c3c(ccc2[nH]1)N(C(=O)CC1(O)CCC1)CC3 N1(C(c2ncn(CC)c2)=O)CCC2CN(C(=O)CCC(CF)CF)CCC12 N1(C(c2cc(C)oc2)=O)CCCOC(CCNC(=O)Cc2cc(F)cc(F)c2)C1 C1(C2N(C(CN(C(C)=O)C)=O)CCC2)CCCN(C(c2ccnn2C)=O)C1 C(=O)(C1CCc2ccc(Cl)nc21)N1C(CNC(=O)C2=CCCCCC2)COCC1 c1(C(=O)NC(CNC(COC(C)C)=O)(C)C)coc(C(N)=O)c1 C(=O)(C1=CCCCCC1)NC12C(CN(C(c3sc(CCC)c(CC)c3)=O)C1)C2 c1(C(N(C(C)CNC(=O)C=CC2CCOC2)C)=O)cc(-c2cccnc2)n(C)n1 CC1CN2CCN1C(C(N1CC(CNC(C3CCS(=O)(=O)C3)=O)CC1(C)C)=O)C2 N#CCCCCCC(=O)N1CCN(C(c2ccc(Br)s2)=O)C(CO)C1 c1(CN2CC3C(CNC(CC4N(CC)C(=O)CC4)=O)C3C2)ccccc1[N+](=O)[O-] C1(C(=O)NC(CC)C)COC(CNC(=O)C(C)CC2CCCC2)C1 C(=O)(CC(C(F)F)N1CCOCC1)NC1C2(CC(NC(=O)C3=CCOC3)C2)C1 Cc1ccc(C(=O)NCC2CN(C(c3cccc(Cl)c3C)=O)C3CC23)cc1C N1(C(CCCC#C)C(=O)NC(C)C(=O)OC)CCOCC12COCCN(C)C2 CC(C)C(C#N)C(=O)N1CCC(CCNC(c2nncn2C)=O)CC1C c1(C(=O)NC(CN(C(c2cc(C(C)C)ccc2F)=O)CC)C)cnc(N)c(N)c1 C=CC(CC)CC(=O)NC1CCN(C(c2ncsc2C)=O)CC1CC N1(C(CCOC)=O)CCC(O)(CCCNC(=O)C(C)(C)C(N)=O)CC1 CC1COCCC1O.C1(=O)C(N(C)C)CN1.c1(CC(=O)N)cccn1C C(=O)(C(C(=O)NCCNC(C1CN(C(c2ccccc2)C)CCO1)=O)OC)OC N1(C(CCn2c(C)ncc2)=O)CCN(C(=O)CCc2ccccc2)C(C)C1C S(=O)(=O)(c1cccnc1NCC1CCCCO1)NCCCCC=C CC(C(=O)NC(CCF)C(=O)NC(CCO)C1CCCC1)C(F)(F)F N1(C(c2ccc(OC)s2)=O)CC2(CC1CNC(c1occ(C)c1C)=O)CC2(F)F C1(N(C(c2csc(CO)c2)=O)CCF)CCCN(C(C2CC3(CC3)C2)=O)C1 N1(C(Cc2cnc(C)s2)=O)CC2CN(C(=O)CCC(C)(C)C(=O)C3CC3)CC2C1 CC#CCCC(=O)N(CCNC(=O)Cc1cc(C)sc1C)Cc1ccccc1 N1(C(c2n(C)c(SN(C)C)nc2)=O)CC2CC(NC(=O)CC3CC4COCC4C3)C1C2 Cc1nn(C)cc1C1=NOC(C(=O)NC2CCN(C(=O)Cn3ccnn3)CC2)C1 c1(-c2[nH]cc(C(=O)NC(CNC(C(C)OC)=O)CO)n2)ccc2c(c1)OCCO2 C1(C(N(CCCNC(=O)Cc2ccnnc2)C)=O)CSCC(=O)N1 C=CC1CN(C(=O)CN(C)CCC)CC1NC(c1ccc(-n2ccnc2)nc1)=O C1(CC=C)(NC(=O)CNC(N)=O)CN(C(=O)C(CC)n2cncn2)C1 C1(CNC(C2CC2(Cl)Cl)=O)CCN(C(c2csc3nnsc23)=O)C12CC2 CCC(C(=O)NC1CC(NC(C2(O)CCOC2)=O)C1)n1ccc(C2CC2)n1 C(CC(F)F)(C(=O)NC(C)CCCCCO)N(C(C(CC)C)=O)C C12(CNC(C(N)=O)=O)CN(C(c3ccc4cnoc4c3)=O)CC1CCO2 C1(NC(CC(n2ccc(C)n2)C)=O)CCN(c2snc(C)c2C#N)CC(C)(C)C1 C1(NC(CCCCNC(N)=O)=O)CCN(C(=O)Cn2cc(C(C)O)nn2)CC1F C1(NC(C(CCC)OC)=O)CC2CCC(C1F)N2C(c1ncccc1C(F)F)=O c1(C(CC(=O)OC(C)(C)C)NC(C2CC3CCC3C2)=O)ccc(Cl)cc1 C1(C(=O)NC2CCN(C(=O)NCC(F)(F)F)C2)C2CCN1CC2 C(C(C(C)C)NC(=O)COC)CC.C1(=O)C(C)=CCNC(=O)CN1.OC c1(NC)ccc(C(=O)NCC(C)(CNC(=O)C(C2CC(F)(F)C2)OC)OC)nc1 CCCC(C(=O)N1CC(O)CC1CC(=O)Nc1cnc(C(C)C)nc1)NC(C)=O c1(OCC)ccccc1OCC(=O)NCC1CCN(C(c2nn(C)cc2Cl)=O)C1 C1(NC(c2c(C)scn2)=O)CCCC(NC(C2(C)CCNC2=O)=O)C1 c1(C(=O)NC2(C)CCN(C(C3N(C(C)=O)CCC3)=O)C2)c[nH]nc1S(N)(=O)=O c1(C(=O)NC(C2CCN(C(c3cnc(-c4ccccc4)[nH]3)=O)C2)C)cc(N)ccn1 N1(CC(=O)NC(COC)C(=O)Nc2cncc(C(N)=O)c2)CCN(C)CC1 C(=O)(CC(C(F)(F)F)NC(=O)CC(C)CN(C)C)N1C(C=C)CCCC1 c1(C(=O)NCC2N(C(CN(C)CC)=O)CC(OC)C2)cnn2ncccc12 C(=O)(CCC(=O)C1CC1)NCCCCCNC(CC(CC)c1ccccc1)=O C1(C(=O)OCC)CC(F)(F)CN1C(c1ccccc1)=O.c1(C(=O)OC)noc(C=O)n1 c1(C(=O)NCC2CN(C(C(C)SC)=O)CC(C)(C)C2)ccc(S(C)(=O)=O)cc1Cl C1(NC(c2c(F)ncc(OC)c2)=O)COC2(C1)CN(C(=O)CCC(C)(C)C)C2 N1(C(C(C)SC)=O)CC2C(CNC(=O)CCc3ccc(OC(C)(C)C)cc3)C2C1 c1(CCC(=O)NCCN(C(=O)CC(O)C(C)C)CC)c(C)nc2ccnn2c1C C(=O)(CCC(C)(C)C(=O)N1CCC(C)C(N(C)C(C2(SC)CCC2)=O)C1)OCC Cc1ccc(C(=O)N(CC(O)CNC(C2CC23CCC3)=O)C)nc1 C(=O)(NNc1cccc(Cl)c1Br)n1cccc(OC(C)C)c1=O C12(CNC(C(C)O)=O)CCC(NC(c3cc(F)ccc3O)=O)(CO1)C2 CCC(CNC(=O)C(C)CNC(C1OCCOC1C)=O)(CC)OC CC1CC(CCNC(c2cc(O)cc(Cl)c2)=O)CCN1C(=O)Cn1cnnn1 N1(c2snc(SC)n2)CCC(NC(C2(C)CCCCNC2=O)=O)C(C)(C)C1 C(=O)(CCCC(C)(F)F)NC1CC(CNC(C(CC)O)=O)C1 O=C1COC2=C(C(C(=O)O)(NCc3cc(Br)no3)N=CC(c3ccccc3)=C2)N1 C=CCCC(C(=O)NC1CC(=O)N(O)C1)NC(=O)C(C)CSC C1(CN(C(C2CCCO2)=O)CC)CCN(C(=O)C#CC(=O)N(C)C)CC1 C1(NC(c2nc(C(C)OC)oc2)=O)CC2CC1CC2C(N1CCCC(C#N)C1)=O C1(CC(=O)NCCN(C(=O)Cc2c(C)cccc2Cl)CCC)CCOC(C)(C)C1 Cc1nn2c(c1C(N1CCC1CNC(c1cccn(CC)c1=O)=O)=O)CCCC2C N1(C(C2OCCN(C)C2)=O)CCN(C(c2csc(Cl)n2)=O)C2COCC12 C(=O)(C(c1cccs1)NC(=O)C(=O)NC1CC1)NCC(Br)=C(C)C C12(CC)CN(C(=O)C(O)CF)C(CNC(=O)COc3ccc(OC)cc3)(C1)C2.C(C)=O N1(C(c2n(CC)ccn2)=O)CCCC1(C)CNC(C1CCOC1C)=O C(C(C)(C)CC(=O)NCCCC1CCCCC1)NC(c1c(OC)cnnc1)=O N12CC3CCCC3(C1)C(=O)NOC(CC#CC)C2=O.C(c1ccccc1)=CC C1(NC(C=Cc2c(C)ccs2)=O)CC(O)CN(C(C2(C)CCCC2)=O)C1 C(C1=CCCOC1)N(C1CCN(C(C(C)(C)c2ccno2)=O)C1)C(=O)C1CC1 c1(CC)ccccc1C(N1CCC(CO)(CNC(=O)Cc2c[nH]nc2O)C1)=O c1(CCC)cc(C(=O)N(C)CCNC(c2c[nH]cc2C2CC2)=O)c(C)o1 c1(C(=O)NCCCCN(CCCNC(C2CCC(COC)C2)=O)C)ccc[nH]c1=N N1(C(CCC)=O)CC(NC(=O)C(C)NC(=O)Cc2ccccc2)CC(C)(C)C1 CC1C(C)N(C(=O)CN(C)S(=O)(=O)N(C)C)CCN1C(c1ncoc1C1CC1)=O CCC(C)(C)C(=O)C(=O)N(C1CCN(C(c2nc(C)oc2OC)=O)C1)CCCC c1(C(=O)NC(CCCNC(c2cn(C)nc2Cl)=O)(C)C)coc2cc(O)ccc12 CC1CCCC(C(N2CC(CCCCNC(C3(CO)CCCCC3)=O)C2)=O)C1 N1(C(C=CC=CCC)=O)CCC2(CCCN2c2ncc([N+](=O)[O-])cc2F)C1 c1(OC)ccc(OC)c(C(F)(F)F)c1.c12ccc(cc1)CC(=O)N1CCC2C1 N1(C(CN(CCC)CC)=O)CCC(C(=O)NC(C)CC2CCC(=O)O2)CC1 c1(OC(CC)C)cc(C(N2CCC(CNC(C3CCC(C)S3)=O)CC2)=O)ccn1 CC(C)(C(F)(F)F)OCC(=O)NCC1CC1NC(=O)CCc1cccc(Cl)c1 c1(C(=O)NC2CCN(C(C(=O)N(C)C)=O)CC(O)C2)ccccc1C#CC1CC1 CC(C)CC(CC(C)C)C(=O)NC1C2CCN(C(=O)C(C)N3CCC3)CC12 N1(C(C2(CC)CC2(F)F)=O)CCCCCC1CNC(c1cc(C)cc(Cl)c1)=O Cc1cc(C(=O)NCC2CCN2C(=O)C=CCOc2ccccc2)cnc1O C1(C(=O)NC2CCCC(NC(C3CCCS3(=O)=O)=O)C2)(OCC)CCCCCC1 c1(C(N2CC=CC(NC(C3C(C=C(C)C)C3(C)C)=O)C2)=O)ccccc1N=[N+]=[N-] c1(C(N2CCCC(N(C(=O)C=C(Cl)Cl)C)CC2)=O)cc2ccccn2c1 c1(SC)cncc(C(=O)NC(CO)CCCNC(c2cnn(C)c2)=O)c1 Cc1ncc(CNC(=O)CNC(=O)COCCOc2cnn(C)c2)o1 Cc1cccc(C)c1-n1cc(CC(C(=O)O)NC(C2CN(C)CC2C)=O)nn1 C1(N(C(=O)C(CC2CCCC2)OC)CC)CCN(C(c2ccc(O)nc2)=O)CC1 C=CC(C(F)(F)F)NC(=O)CC1CC(O)CN1C(=O)CCc1ccsc1 N1(C(C2C(CC)C2)=O)CCN(C(c2cc[nH]n2)=O)CC1c1cn[nH]c1 c1(OC)cc(C)cc(CN2CC(CC(=O)Nc3ccnc(F)c3F)C2)c1O Cc1cc(O)ccc1C(=O)NCC1CCN1C(=O)C(C)n1cnnn1 c1(C(=O)NCCN(C(=O)C2=C(C)OCC2)CC)csc2ccc(F)cc12 c1(NC(=O)NCC(C)CC(F)(F)F)nn(C)c2nccnc12 c1(C(=O)NC(CNC(C2(OC)CCCC2)=O)C)sc2cccc(F)c2c1Cl c1(CC(N2CC(C)CC(C(=O)NC(c3ccncc3)C)C2)=O)ccc2c[nH]nc2c1 c1(Oc2c(Cl)ccc(C)c2)ccc(C#N)cc1Cl C(CC)(C(C)(C)O)(c1cccnn1)NCc1nccc(C(=O)OC)n1 Cc1ccn(C)c(=NC(=O)N2CCC(C3CCCO3)CC2)n1 CC#CCC(C(=O)NC1CN(C2CCC2)C1)NC(=O)C(COC(C)=O)CC(C)C N1(C(c2c(CC)n(C)nc2)=O)CCCC(N(C)C(c2occc2C)=O)CC1 C(=O)(CCN=c1ccc(C)c[nH]1)NCC(CC)NC(c1cccc(Cl)c1C)=O N1(C(c2cc(C)cc(C)c2N)=O)CCN(C(=O)CCNS(C)(=O)=O)CC2(CC2)C1 C1(C(=O)NCCN(C(=O)OC)C)CC2C=CC1N(C(c1cc3ccccn3n1)=O)C2 C1(NC(COC(CC)C)=O)CCCCCC1NC(c1nc[nH]c1C(C)(C)C)=O c1(C(=O)NC(CC)(CNC(=O)CC2CCC(=O)N2C)CC)ccc2cnnn2c1 c1(OC)ccc(C(N2CC=CC2C(=O)Nc2nc(Br)cnc2OC)=O)cc1C#N N1(CC)CCC(N(C)C(=O)N(Cc2ccccc2C)Cc2cccs2)CC1 C1(C(=O)NCC2N(C(C3CC=CC3)=O)CCN(C)C2)CCn2cnnc2C1 C(COC)(C(C)C)(c1n(CCOC)nnn1)NCC(C)(C)OC.C(CF)O CC1CN(C(=O)CC23COC(C)(C2)C3)CC(C)N(C(=O)CC(O)C(C)(C)C)C1 N1(C(CCCCCOCC)=O)CCC2(CC1)CC2CNC(C1(F)CCOCC1)=O C1C(=O)N=C2C=C(N(C)N2)O1.C1(C(N(CCC)C(C)C)=O)CCN(CC(F)(F)F)C1 c1(C(=O)NCCC2CN(C(C(=C)Cl)=O)CC2C)ccc(C)c(C)c1 C#Cc1cn(C)nc1C(=O)N(CCCCCNC(C1CCCO1)=O)C CC1(O)CCN(CC(N2CC=CC(NC(=O)CCN3CCOCC3)C2)=O)C1 N1(C(C(C)Oc2ccccc2)=O)CC(CNC(=O)C=CCn2cncn2)C(F)(F)C1 CCN(Cc1cccc(Cl)c1)N1CCN(CCCC2CC2)CC1 C1(CNC(c2c(C)cc(C)o2)=O)CN(C(c2cn(C)nc2C(C)C)=O)CC1(F)F c1(C(=O)NC2C3(NC(C4CCCN(C)C4)=O)CCC(C2)C3)ccn2nncc2c1 C1(CNC(C(CCCC)C)=O)CCN(C(=O)CNC(=O)CC(C)C)CCC1(F)F C1(CNC(c2csc(Cl)c2)=O)CC2CCCC(C1)C2(F)F c1(NC2CC3CN(C(C4CC(CC)(CC)C4)=O)CC32)cc(C)ccc1[N+](=O)[O-] CC(C)C(CO)ONC(=O)C1CC1C(C)N(C(=O)C=CC1CCC1)C1CC1 c1(CC)c(C(=O)NC2CN(C(=O)C(F)(F)CO)CCC2O)oc2ccc(Cl)cc12 C1(C(C)(C)F)CCN(C(c2cc(Br)sn2)=O)CC1 N1(C(c2c(C(C)C)nns2)=O)CCN(C)CC1CNC(=O)C(O)Cn1cncn1 C1(C(N(C(C)CNC(c2cn(C)c(C(F)F)c2)=O)C)=O)CC(C(C)(C)C)=NO1 CC1CN(C(C2CCSCC2)=O)CCC1CNC(c1ccccc1C(F)(F)F)=O Cc1cc(CNC(=O)CC2CCSCC2)oc1C S1(=O)(=O)CC(=O)N1.C(CC(C)CCO)NC(CCNS(C)(=O)=O)=O C1(C(=O)NCC2CC(NC(C3CCC3)=O)C2)Cc2c(F)cccc2O1 Cc1nc(CC(=O)NC2CC(NC(=O)CCS(C)=O)C2)c(C)s1 N1(C(C2COc3ccccc3C2)=O)CCCC2CN(C(C34CSCC3C4)=O)CC12 C(CC(=O)N1CC2(CC(N(C)C)C2)C1)(C(F)F)NC(C(CC#C)O)=O C1(CC)(CCC(=O)NCCn2cc(-c3sccc3C)nn2)CC(F)(F)C1 C1(C(=O)NCC(C)NC(=O)C(O)C(C)(C)C)CC2COCC(C1)C2(F)F c12cccc(n1)CNC2=O.N1(c2snc(C)n2)CCCC(CO)C1 Cn1nnc(=NS(=O)(=O)c2ccc(C(=O)OC(C)(C)C)cc2)[nH]1.C1COC(=O)N1 Cc1nsc(C)c1C(N1CCC(C(C)C(=O)NCC2CCC(C)CC2)CC1)=O C1(CNC(C(C)(C)F)=O)C2CCC(C2)N1C(c1ccc(Cl)c(O)c1)=O C1(NCC(c2ccc(C(F)(F)F)cc2)(C)C)CCC(C=C2SC(=S)NC2)C1 C1(N(C(=O)CC2CC(=O)C2)CC)CCN(C(C2(SC)CC2)=O)C1 C1(NC(=O)NC(C)(C)C(=O)Nc2ccccn2)CCNC(=O)CC1 C1(CC(=O)N(CCCN(C)C(C2CC2c2ccccc2)=O)C)CCCNC(=O)C1 c1(C(=O)NC(CN(C(CC2C(CC)C2)=O)CC)C)cnc2scnc2c1 C1(OC)(CNC(=O)Cn2nccn2)CCN(C(C2CNC(=O)C2)=O)C1 C1(NC(Cc2c(C)noc2)=O)CCCN(C(=O)Cn2cnnc2)CC1 C#Cc1ccccc1CNC(=O)C(C1CCCO1)NC(C1CN2CCN1CC2)=O C1(C)CCC(NC(=O)CCO)C1.C1(C(=O)NCCNC(C)=O)(OC)CCCC1 CC(C)C(C(C)NC(c1coc(Cl)n1)=O)NC(c1cn(CC2(C)COC2)nn1)=O C1(NC)CCCC12CC2.CCC1C(=O)N2CCC(C2)C(=O)N(CC)N1CC Cc1nc(C#N)ccc1C(=O)N(C)CC1(CNC(c2cc(CF)on2)=O)CC1 c1(C(=O)NCC(CNC(CC(COC)C)=O)(C)C)cccc(N)c1O N1(C(CCSCCCC)=O)CCCC(O)(CCNC(C2(F)CC2C)=O)C1 CCCC(C(O)C(=O)Nc1c(OC)noc1C)NC(=O)C(C)(F)C(=O)OC N1(C(c2c(C)nco2)=O)CC(NC(c2ncnc(O)c2Cl)=O)CC(C)(C)C1 c1(C(=O)NC2CC(NC(C3(F)CC3Cl)=O)C2)nsc2cc(Br)ccc12 c1(NC(c2nnnn2-c2cccc(OC)c2N)CC)ccc(Cl)cc1CCOC C#Cc1cc(F)c(C(N2CCC(NC(c3ccsc3Cl)=O)C(C)C2)=O)cc1F c1(OCC#C)cccc(NC(c2nnnn2CC(F)F)c2ccnn2C2CC2)c1 C12(NC(CC=C)=O)COCCC1CN(C(=O)CCc1cn(C)nn1)C2 C(CCC(C)C)(C(=O)N(C)CCc1cccs1)NC(c1c(C)coc1)=O c1(OC)ncnc(N2CCCC(CO)(NC(C3CCCC3C(N)=O)=O)C2)c1OC N1(C(C2C(C=C(C)C)C2(C)C)=O)CCN(C(c2ccsc2C)=O)C2(CCC2)C1 N(C(=NCC1CN(C(=O)OC)CCO1)NC1CCCCC1)C(CC)C.c1cnccn1 C1(NC(=O)C=C2CCCCC2)CCC2CC1CN2C(c1cnc(S)[nH]1)=O c1(C(=O)NC2C(NC(=O)C(O)CCCc3ccccc3)C2)nnn2c1CSCC2 C#Cc1ccc(Cl)c(C(=O)NCC(C)NC(=O)C(C)(CO)NC(C)=O)c1 c1(C(=O)NCC(C2CC2)NC(CSc2nc(C)[nH]n2)=O)n[nH]c(C)c1F Cc1ncnc2c1CC(C(N1CCN(C(=O)CP(C)(C)=O)C(C(F)F)C1)=O)CC2 N1(CC(N2CCC(C(C)NC(=O)C(Cl)=CCl)C2)=O)CC(=O)NC1=O CN1CCC(C(=O)NCC2CNC(=O)C2)(NC(=O)CS(C)(=O)=O)C1 Cc1ccc(-c2n[nH]c(CN(CCCNC(=O)CC(C)(C)F)C(C)C)n2)cc1 c1(CN2C(CC(=O)Nc3cc(C)c(Br)cc3F)COCC2)ccc(O)c(C#N)c1 c1(C(C(=O)NC(C(C)C)CCNC(=O)C(C)c2cc[nH]n2)=O)cc(F)cc(Cl)c1 C1(CNC(c2n(C)nc(CNC(=O)C3=C(Cl)CC3)c2)=O)CCCOC1(C)C CCCC(CCCNC(c1c[nH]nc1CC)=O)NC(C1ON=C(C)C1C)=O Cc1cccc(-c2cn(C3CC(C(=O)N(CCCF)C)C3)nn2)c1N(C)C Cc1cc(F)ncc1-c1noc(C2CCCN(C(=O)NC(C)(C)C)CC2)n1 N1(C(C2N(CCN(C)C)C(=O)CC2)=O)CC2CCN(C(c3cc(Br)n[nH]3)=O)C2C1 CCCC(CC)C(=O)NC(C)(CNC(C1(CF)CC1)=O)CC(C)C N1(C(c2n(CC)nc(C)c2)=O)CCCN(C(c2cn(C(C)C)nn2)=O)CC1CO N1(C(CC)=O)CCCC(C2CN(C(=O)COc3ccc(C)cc3)C2)C1 C1(C(N2CCC(N(C)C(c3cc(C4CC4)no3)=O)C2)=O)OCCC1(C)C c1(C(N2CCC(C(=O)NCC3CCC(=O)NC3)CC2)=O)ccc2ncsc2c1 c1(C(=O)NCC2C(C(=O)NC(CC)C(C)C)C2)csc(C)c1C c1(C(=O)NCC(C)(O)CNC(C2CCSC2)=O)cc2cccc(Br)c2[nH]1 c1(C(N2C(C(C)NC(=O)C=C3CCC3)CCC2)=O)cncc2[nH]ccc12 c1(CNC(C2(C(=O)Nc3cc(OCC)ncn3)CC2)=O)ccc([N+](=O)[O-])c(O)c1 c1(C(N2CC3CC3(NC(C34CCCC3OCC4)=O)C2)=O)n[nH]c2c1COC2 C1(CC)CN(C(=O)C(C)N(C)C)CCN1C(c1ccc(OC(F)(F)F)cc1)=O N1(C(c2c(C)c(F)ncc2)=O)CCOC2(C1)CN(Cc1cccc3c1OCC3)C2 CCCCC(O)CCC(=O)N1CC2(C1)CN(c1cnc3ccc(C)cc3c1)C2 N1(C(CSCCOC)=O)CCC2CN(C(=O)CNC(c3cccs3)=O)CCC2C1 C(=O)(NNc1cc(CC(N)=O)ccc1Br)C1N(C(=O)OC(C)(C)C)CCC1 C(C(O)CN=c1nc(C2CCCC2)[nH]s1)NC(C)=O.C1(C)(C)C(=O)N1C1CC1 CC[Si]1(CC)CCN(C(C2(C)CCOCC2)=O)CC1 c1(C(=O)NC(C2(CNC(=O)CC(C)c3ccccc3)CC2)C)ccccc1OC C1(C(N2CCC(C(C)NC(C3CC3F)=O)C2)=O)CCC(=O)N1C1CC1 N(C(=NCc1ccnc(OC)c1)NCC1(n2cccn2)CC1)C(C#C)C C1(C(C(=O)NC2C(NC(c3c(C(C)C)n[nH]c3)=O)CC2)=O)CCCCCCC1 C1(NC(CNC(N)=O)=O)CN(C(=O)CC2CC3(COC3)C2)CC1S(C)(=O)=O N1(C(C2=NOC(C)(C)C2)=O)CC(NC(c2cn(C3CC3)nn2)=O)CC12CCCC2 CC(C)(C)C1=NOC(C)(C(=O)NC2CC3CCC2(NC(=O)COC2CCC2)C3)C1 N1(C(c2c(F)ccc(C)c2)=O)CCOCC(C)(CNC(C2C3(CC3)C23CC3)=O)C1 CCC(CC)(C(=O)N1CCC(O)C(C(N2CCCCC2CO)=O)C1)C(=O)O n1(CC)cc(C(=O)NCC(C)NC(c2sccc2F)=O)c(C(F)(F)F)n1 c1(CC(=O)NC2(CF)CCN(C(c3cc(Cl)no3)=O)C2)ccc2c[nH]nc2c1 C1(CNC(CCCC)=O)CCN(C(=O)Cc2ccc(OC(F)F)cc2)C12CCC2 C(C(C)(C)C(C)(F)F)OC(=O)C(C)C1(C(C)(C)NC(=O)OC)CC1 N1(C(=O)OC(C)(C)C)CC=CC1C(=O)NC(C)C(=O)O C1(F)(CNC(=O)C(O)C2CCCC2)CN(C(=O)CN2CCCC2)C1 CC(C)CS(=O)(=O)CC(=O)N(C1CCN(Cc2c[nH]c3cc(F)ccc23)C1)C c1(C)[nH]c2ccc(F)cc2c1C.C1(C(=O)NO)(Cc2cn(CC(=O)OC)nn2)CCCC1 n1(CC)ncc(C(N2CCCC2C(C)NC(C2(O)CCC2)=O)=O)c1Br c1(C(CNC(C2CCC3(CCC3)C2)=O)NC(C(C)SCC)=O)cc(F)cc(Cl)c1 c1(C(N(CC(C)CNC(c2cc(N)c(F)cn2)=O)C)=O)cc2ncccn2n1 c1(C(N(C2CCN(C(=O)CCn3ccnn3)C2)CC#C)=O)csc(CO)n1 C12(NC(CCSCCC)=O)CCN(C(c3cncc(N(C)C)c3)=O)CC1C2 c1(C(=O)NCC2N(C(C3C(C=C)C3)=O)CC2)cc(N)ccc1CC(=O)OC C1(C(N2CCN(C)CC2CNC(C2CSCCS2)=O)=O)CNC(=O)CC12CCC2 c1(OCCOCCCC)cc(NC(C(C2(OCC)CC2)=O)=O)ccn1.C(=O)(C#C)N C(=O)(CCS(N)(=O)=O)NCC1CC(F)(CNC(C2N(C(=O)NC)CCC2)=O)C1 Cc1[nH]c(=N)[nH]c(=NCCn2ccc(O)nc2=O)c1Cl C(CC(=O)NC(CO)(CO)CO)(C(F)(F)F)NC(C(C(CC)C)C)=O C(=O)(C1=CCCCO1)NC(C1CCN(C(c2ncn3c2CCC3)=O)C1)C C1(CC(=O)NC(CC=C)CNC(=O)CN(C)C(N)=O)CCC(C)(C)C1 c1(C(=O)NCC23C(CN(C(C4(Cl)C(C(C)=O)C4)=O)C2)C3)ncnc2sccc12 CC(C)CC(CNC(c1cn(CC(F)(F)F)nn1)=O)NC(=O)C(F)C(C)C c1(C(N2CCC(CN(C(=O)Cc3csc(Cl)c3)C)C2)=O)cc(F)c(C#N)c(F)c1 N1(C(CC2C(NC(c3ccccc3)=O)CCC2)=O)CCC(CO)(CC2CC2)C1 N#CCCCCCC(=O)N1Cc2occ(C(N3CC(C4CCCC4)C3)=O)c2C1 c1(C(=O)NC2CCN(C(Cc3scc(CC)n3)=O)C(C)C2)ccc2ccsc2c1 c1(C(N2CC(C(C)NC(C3C(C=C)C3)=O)C2)=O)cc(OC)cc(Br)c1N CC1CCN(C(c2cn(C)c(O)n2)=O)C1CNC(c1cncc(C(N)=O)c1)=O CC1(C)OCCOC1C(=O)NCCCCn1cc(-c2cncs2)nn1 CC(C)CC(C)C(=O)N1CCCC(N(C(=O)C(C)OC2CCCCC2)C)C1 c1(C(N(CC(C)NC(C2(N(C)C)CCOCC2)=O)C)=O)ccnc2ccnn12 C(=O)(CC1=CCN(C)CC1)NC1CN(C(C(COC)N(C)C)=O)C(CO)C1 c1(OC)cc(C(=O)N(C)CCNC(C2CSCN2C(=O)C(C)(C)C)=O)ccc1F C1(NC(C2ON=C(C)C2C)=O)CN(C(=O)Cc2c(C)cccc2C)C2(CCC2)C1 C(=O)(C(O)CC(N)=O)NCC1(O)CC(CNC(c2cnn(C)c2C(F)F)=O)C1 C(=O)(C1CCc2cccc(F)c21)NC1(C)CCCN(C(c2c(C)csn2)=O)C1 c1(CC(C)C)nccc(C(=O)NCC2(C)CCN(C(C3(F)CCOC3C)=O)C2)n1 N1(CC(COC)O)CCN(C(=O)C(c2ccc(F)cc2)=O)C(C)C1.C(=O)C1CC1 N1(C(c2n(CC=C)ccc2)=O)CCC2(CCN(C(=O)CN3CCC(C)C3)C2)C1 c1(C(=O)Nc2c(C)nc(C(C)(C)C)s2)c(Br)cc(Br)c2ccccc12 C(C(C)(C)CC(=O)NC1CCCC1n1cc(-c2c[nH]c(C)cc2=O)nn1)OC c1(C(N(C(CNC(CN(CCOC)C)=O)C)C)=O)ccc(F)c(OC)c1F C1(CNC(COC)=O)COC(C)(C)CN1C(=O)Cc1cnsc1 C1(C(=O)NC(CNC(c2csc(-c3ccco3)n2)=O)C2CC2)CCC2CC2CC1 C1(O)(CC#C)CC(C(=O)NC2C=CC(C(=O)NCCc3ccncc3)C2)C1 c12ncccc1SC(C)CN(C)C2=O.C1(C(N)=O)(NC(C2CCC2)=O)CCC1 N1(C(C2N(C)C(=O)CC2)=O)CCOCC(C(N2CC(F)CC2C(N)=O)=O)C1 c1(SCC)ccc(C(N2CCN(c3cccc(O)n3)CC2)=O)c(Cl)c1 c1(CC(C)NC(c2c(C)nn(CCC)c2C)=O)ccc2c(cnn2C)c1 CCC(C)(C(=O)NCC1(O)CC(C(=O)NC)C1)OC c1(OCC)cnccc1C(N1CCC(NC(C2CC3CC3N2C(C)=O)=O)C1)=O Cc1cc(C)c(CNC(N2CCOC(C3CC3)C2)=O)o1 Cc1nnc2n1CCC(C(=O)NCC(O)CNC(=O)C(c1ccccc1F)(F)F)C2 c1(-n2c(C(=O)NCC(C)CN(C)C(C3CC34CCC4)=O)cnc2)cccc(Cl)c1 C(C1CCN(C(C2CC3CC3C2)=O)CC1)=CC(=O)N(C1(C)CC1)C c1(SC(C)C)ccc(C=CC(=O)Nc2cc(C(F)(F)F)ccc2C)cc1 n1(CC=C)nnnc1C(C1(C2CCCO2)CCC1)NCC1(CC#N)CC1 C1(CC=C)(NC(=O)CC(C)(O)CCC)CC2CCC(C1)N2c1ccncn1 N1(C(CC(=O)OC)=O)CCC(NC(c2cc(Cl)cc(Br)c2O)=O)C(C)(C)C1 c1(C(CNC(=O)CCSC2CCCC2)NC(C2CC2F)=O)ccccc1 CCC(C)C(C(=O)NCCCn1cc(C)cn1)NC(=O)CCCN(C)C(C)=O Cc1cc(F)cnc1C(N1CCCCC1CCCNC(=O)Cc1ccc(Cl)cc1)=O C1(n2ccnc2)(C(=O)OC)CN(CC(=O)N(C)C(C)C)C1 C1(NC(=O)CCC2CCC2)CC(NC(C2C3(CC3)C23CC3)=O)CC1O CN1C(=O)C(=O)N(CC(=O)NC2(C3CCCN3C(C3C4CNC(=O)C34)=O)CC2)C1=O C(=O)(CCCCC(N)=O)N1CCCC(CN(C(Cc2ccc(SC)cc2)=O)C)C1 c1(-c2c(OCC(=O)NC3C(C)(O)CCCC3)ccc(F)c2)cc(F)c(Cl)cc1F C1(C(N(C)CC2COCCN2C(c2ccnc(S)c2)=O)=O)CCCCC2(CC2)C1 Cc1nc2ccccn2c1CC(=O)NCC1C2CN(C(=O)CN(C)C(N)=O)CC12 C1(C(=O)NCCN(C(C)C)C(C2(C3NC(=O)NC3=O)CC2)=O)CC2C(C1)C2(C)C C1(CC)CC(C(=O)Nc2ccc(C(=O)NC(C)C)nc2)CCO1 C(C(O)CNCC1(COC)CCC1)(OCC)OCC N1(C(C2N(C)CC(C)(C)C2)=O)CCC2CCN(C(=O)C3=CCCC3(C)C)C2C1 C1(N(C(c2cnc(C)n2C)=O)C)CC2CC1N(C(c1cccc(C(F)F)c1)=O)C2 c1(C(N2CCC(C(C)NC(=O)CN3CCC(C)(O)C3)C2)=O)ccn2nnnc2c1 C1(C(N(CCNC(c2cc(CC(C)C)[nH]n2)=O)CC)=O)COC(C)(C)C1 c1(CSCC(=O)NCCC(C)NC(=O)Cc2ccccc2)csc(=N)[nH]1 C(=O)(CC(C)CC(C)C)N(C(CNCCC)C1CC1)C.N12CCCC(C1)C2=O c1(C(=O)NC(CNC(c2ccc[n+]([O-])c2)=O)C2CC2)cccc2c1COCC2 C(CC)(CCCC(=O)NCC1COCC1O)NC(CSCCCC)=O C=CCCCC(C(=O)NCC12CC(CN1C)C2)NC(=O)Cn1ccc(C)c1 C1(NC(CSCCCC)=O)CCC2CN(C(=O)CC3CCCN3C(C)=O)CC2C1 CC1CCN(CCC(=O)NC2CC2NC(=O)CC2CC(=O)NC2=O)CC1 C1(C(=O)NCCCCC(N)=O)CCN(C(=O)CC2(O)CCOC2)C12CC2 C(C(=O)NCc1nc(Cl)ccc1F)(C1=NOCC1)N1CC2C(C)(C2)C1 N12CC(CC3(CCOCC3)C1)C2=O.CC(C)C(O)C(=O)N1CCC(C)C1 N1(C(C2OCCN(C)C2)=O)CC2(CC2)CC1CNC(=O)C(F)(F)c1cnccn1 N1(C(C(CC)(F)F)=O)C(CC(=O)NCCS(C)(=O)=O)C2CCCC12 C1(O)(C(=O)NC(C2CN(C(C3CCc4nc[nH]c4C3)=O)C2)C)CCCC(C)(C)C1 C(CNC(=O)CC=CC(C)(C)C)(C(C)(C)C)NC(c1cc(CC)[nH]n1)=O c1(C(=O)NCC2C(NC(C(C(CC)C)C)=O)CCC2)cccc2sccc12 C1(CCNC(c2cccnn2)=O)CCCN(C(=O)CSc2ccccc2F)C1 c1(COC)cccnc1C(=O)NCC1(CNC(c2nocc2C)=O)CC1(F)F C1(C(N2CCC(C(N3CCC(OCC#C)CC3)=O)C2)=O)CCC2(CCC2)O1 N#Cc1cc(C(N2CC(F)CC2C(=O)N(CCc2ccccc2)CCl)=O)ccc1O N1(C(C(CC#C)C)=O)CCC2(CCCN2C(=O)CN(C)C(C)=O)C1 C1(NC(c2ccc(OCCC#C)cc2)=O)CCN(C(C2(CC)COC2)=O)CC1O CC1C(CC(N2CCCC2CNC(=O)Cn2nnnc2C2CC2)=O)CC1(F)F c1(CC)c(NC(C2CC23CC(NC(=O)C#CC(C)C)C3)=O)cnn1CC CC1CCCC(CC(=O)NC(c2cccc(Cl)c2)C)O1 CC(C)CC(C(=O)NCc1cnc(=N)[nH]c1)NC(c1nnc(O)nc1O)=O C(CO)(C(C)(C)CO)NC(C1(CNC(CC(C=C)C)=O)CCC1)=O C1(COC)(NC(=O)CCC2CCOC2)CCN(C(=O)C#CC2(C)CC2)CC1 N1(Cc2conc2C2CC2)CCN(CC(=O)OCc2scc(CC)c2)CC1 c1(C(=O)NC(C)CCCNC(c2ccc(F)cc2)=O)ccc(OC(F)F)c(Cl)c1 N#Cc1ccc(C(=O)NCC2OCCC2C(=O)N(CC(O)CO)CCO)o1 C(=O)(CCCCCC(C)O)NCC(CN(C(C=CC(CC)C)=O)CC)(C)C C1(NC(C(CC)C#N)=O)CC(CNC(C2CCCC(O)C2)=O)C12CCC2 CC1CC(C(=O)N(CCCn2cc(COCC(N)=O)nn2)C)CO1 c1(C(=O)NCC2(CCNC(C(CSC)C)=O)CC2)ccc2n[nH]cc2n1 c1(N2CCC(CN(CC=C)C)C2)ccnc(N(Cc2sc(C)cc2C)CC)n1 C(CC(=O)N1CC2CC1CN2C(C)C)(C(F)(F)F)NC(CCCSC)=O N1(C(C2C(C#C)C2)=O)CC(NC(C2(n3cncn3)CC2)=O)CC(F)C1 C1(C(N2CCC(CNC(c3c(Br)cn(C)n3)=O)C2)=O)SC2C=CC1CC2 C(CC(C(C)(C)C)NC(=O)C(C)(Cl)Cl)N(C(=O)CCC1CCCC1)C c1(OC)cc(C(N2CCC(CO)C(NC(=O)C(C)(C)CSC)C2)=O)ccc1F c1(C(=O)OC)c(NC(C2(F)CCN(Cc3cnc(Cl)c(I)c3)C2)=O)sc(C)c1C C1(C(N2CC(C(=O)NCCSCC)C2)=O)CCOC1(C)C c1(CC(=O)OC)ccc(C)c(NC(C2CC2(C)C(F)F)=O)c1 C1(CN(C)CCO)CCN(c2cc(N3CCCC(c4nncs4)C3)ncn2)CC1 n1(CC)ccnc1C(=O)NC12CC(CNC(c3cnsc3)=O)(C1)C2 C1(C(=O)NCC(C)N(C(=O)C=C(CC)CC)CC)CCC2(CC2)N1C(=O)OC N(C(=NCC1(OC)CCCC1)N1CCC(C(=O)NC)CC1)C(C)C.c1(SC)ccc(Cl)cc1 NS(=O)(=O)CCC(=O)N1CCCC1CNC(=O)CC1CC(O)C12CCC2 CCC(C)CC(=O)NCc1cn(Cc2ccccc2)nn1.N12CCC(C1)CC2=O C1(C2CC2)(NC(c2cccc(=O)o2)=O)CCN(C(c2onc3ccccc23)=O)C1 c1(CC)cnccc1C(=O)NC(CCF)C(=O)NCC1CCN(C(N)=O)C1 C(=O)(C#CC(C)(C)CNC(c1cccn1C)=O)NCc1cc(OC)nn1C C1(Cn2cc(CC3(NC(CNS(N(C)C)(=O)=O)=O)CC3)nn2)CCC(C)(C)NC1 c1(C(c2nnnn2C(C)(C)CC)NC(CC)(C)C)nc2ccc(Br)cc2o1 N1(C(c2c(CC)n[nH]c2)=O)CCCC(C(=O)NC2CC(CC(C)(C)C)C2)C1 n1(CCC(=O)NCC2C(CNC(CNC(C)=O)=O)C2)nc(O)c2ccccc12 C1(NC(CC(CNC(=O)CCc2nncs2)OC)=O)CN(C)C(=O)C12CC2 CCCC#CC(C)(C)NC(=O)C(C)NC(=O)CC1CCC(C)CO1 C1(CS(N)(=O)=O)CCCCC1(c1nnnn1C1CCCC1)N1CCCC1.CC(F)F C(=O)(C1=NNC(C(F)(F)F)C1)N1CCC(N(C(C(CC)OCC)=O)C)CC1 C1(C)(CNC(CC2(C=C)CC2)=O)COCCN(C(c2cnc(Cl)n2C)=O)C1 n1(CC)ncc(C(=O)NC(Cn2cncn2)CO)n1.C12(CC(CO)C1)C(=O)N2 C(=O)(C1Cc2ccccc21)NC1C2CN(C(C3NC(=O)CC(C)C3)=O)C1C2 CCCC(C(N)=O)NC(=O)CCC1(C)CCCN1C(=O)C=Cc1cscn1 Cc1cc(C(=O)NC(CNC(C2CC2(C)C(F)F)=O)C(C)C)cc(C)c1F O=C(C#CC1CCCCC1)N1CC2CC1(C(=O)N(CC(F)F)C1CCC1)C2 CC(C)CS(=O)(=O)CC(=O)NC12CCC(CC1)N(C(=O)CC(O)C(C)C)C2 C(=O)(CCCCc1ccccc1)NCC(C)(C)CNC(C1(C)CC1(F)F)=O C1(NC(c2c(Cl)cnc(C)n2)=O)CN(C(=O)CCc2cc[nH]n2)C2(CCOC2)C1 C1(NC(C2CCCC(=O)N2)=O)CCN(C(C23CCC(CC2)CC3)=O)CC1F c1(CNC(C(CCC)O)=O)cnn2c1CN(C(c1sccc1CN(C)C)=O)CC2 c1(C(=O)NCCCCC(=O)NC2C=CCN(CC3CC3)C2)ccnc2cc[nH]c12 C1(C(=O)NCC2CC(C(=O)N3CC(CCO)C3)=NO2)(OCC)CCCSC1 C1(NC(CCOC(CC(C)C)C)=O)CCN(C(=O)C=Cc2cnc[nH]2)C12CCC2 c1(NC(=O)CSCCN(CC=CC#C)C)ccc(OC)cc1 C(=O)(NN1CCCC1C(=O)NC(CO)C1(C)CC1)c1cc(C)on1 C1(NC(=O)CSC2CC2)CCC2(CC1)CCN(C(=O)C(F)(F)c1ccccn1)CC2 C(CCCCC(=O)N1CC(NC(=O)CP(C)(C)=O)C1)=CC C1(C(=O)NCC2(CO)CC(C)C2)CCN(C(C2CC3CCC2C3)=O)C1(C)C C(=O)(CCS(=O)(=O)N(C)C)N1CCC(N2CCN(C(CCSC)=O)CC2)CC1 c1(C(N(C(c2ccc(CCC)s2)C(=O)NCCC2CC2)C)C)cc(Cl)ccc1Cl N1(C(C(C)=C(CC)C)=O)CCCC(N(C(c2cc(SCCO)oc2C)=O)CC)C1 N1(C(CCOCC#C)=O)CCOC(C(=O)N(CC(=O)NCC=C)C2CCC2)C1 CCCC(C)(O)CC(=O)N1CCCC(C)(CNC(C2CN(C)CC(C)O2)=O)C1 C(C(=O)N(CCCN(C(=O)CC(c1cccs1)N(C)C)C)C)(C(C)C)NC(C)=O c1(C(=O)NC2(C)CCN(C(C=Cc3n(C)ccc3)=O)C2)nc2cnccc2s1 Cc1nc(CCNC(=O)CONC(=O)NCCOC(C)(C)C)c2ccnc-2[nH]1 CC(C)C(CO)CCNC(=O)C=CCC1(NC(=O)Cn2cnnc2)CCC1 C1(NC(C2C(c3c(C)cccc3)C2)=O)CCN(Cc2nccs2)CC1O c1(C(=O)NCC2CC(NC(C(C(CC)C)C)=O)C(O)C2)cccn2ccnc12 N1(C(C2(C)CC2)=O)CCC2CCN(C(=O)CCC(=O)NC3CC3)CC2C1 C(CC(C)(C)CBr)(c1n(C(C)C)nnn1)Nc1cccc(N2CCC2)c1 c1(OC)ncc(F)c(=NCc2ccc(C(N3CC4CC4C3)=O)[nH]2)[nH]1 Cc1cc(NC(=O)C(C)(C)C)sc1C(=O)NC1CC1CNC(=O)CC1CCCO1 Cc1ccnc2sc(C(=O)N(C)CC3(CNC(=O)C4=COCC4)CC3)c(C)c12 N1(C(c2c(C)[nH]nc2Br)=O)C2CCCC1CC(NC(=O)Cc1ccoc1)C2 CCC(C)C(C(=O)NCCC1CC(C)(C)CO1)N(C)C(c1n[nH]c2c1COC2)=O c1(SC)c(C(=O)NC2CCOC(c3cccs3)C2)cccc1Cl c1(C(=O)OC)cc(OC)cc(C(N2CCC(C)(NC(=O)C(C)(C)CSC)C2)=O)n1 Cc1ccncc1C=CC(N1CCC(F)(CNC(=O)CC2OCCO2)C1)=O C1(O)(CCC)CN(C(=O)C(C)(C2(OC)CC2)NC(c2cnc(OC)s2)=O)C1 C(=O)(C(CN(C)C)C(C)C)N1C(CC=C)(C(=O)NCc2cc(C)sc2C)CCC1 C(C(CC(F)(F)F)NC(=O)C=Cc1ccccc1)NC(C=C(CC)CC)=O N1(C(C(C)C)=O)CC2CC1CC2CNC(C1CC(CCO)C1)=O c1(C(=O)NC(CN(C(C(C)NC(CC)=O)=O)CC)C)ccc(F)c(SC)c1 CC(CC(=O)NC(C1CCCCCC1)CNC(c1nocc1Cl)=O)C(F)F C1(CNC(C=C(COC)C)=O)C(C)CCCN1C(c1cc(C)sn1)=O N#Cc1cc(F)c(F)cc1NC(C1CC(F)CN1C(c1sc(Br)cc1Br)=O)=O CC(C)CC(CNC(=O)CN1C(=O)CNC1=O)NC(c1coc(CO)c1)=O Cc1cc(C(=O)NCC(O)CNC(C2CN(C)C(=O)N2)=O)cc2ccoc12 N1(C(CC2C(C)=CC=CC2)=O)CC(C)CCC1S.c1cc(=N)[nH]cc1Br c12ccc(cc1)C(=O)NC2.C(C(CCCSC)OC)NC(=O)C(COCC)OCC C1(C2CC2)(NC(c2csc(C)c2C)=O)CCN(C(=O)Cc2cccc(F)c2)C1 C1(COC)(CNC(=O)CCCC2CCC2)CCCN1C(c1ocnc1C1CC1)=O n1(CC(=O)NC(C2CN(C(=O)C(O)CC3CC3)C2)C)c(O)nc2ccccc12 c1(OC)cc2ccccc2cc1CN1CCC(O)C(C(=O)Nc2cnc[nH]2)C1 c1(NC(=O)NCC(CC)C(F)(F)F)ccc2c(c1)CCCS2 c1(C(N(C)CC2N(C(CCN(C)CC)=O)CCOC2)=O)cc2ccccc2[nH]1 c1(C(=O)NCCCN(C(C(CCC#C)O)=O)C)cccc2c1CCCN2 n1(CC)nc(NC(=O)CCC2CCCN2C(c2c(OC)nsc2OC)=O)cc1C c1(C(=O)NC2CCC(OC(C)(C)C)CC2)ccc([Si](C)(C)C)cc1 C1(C(N(CC(=O)NCCC2CCC(C)O2)CC)=O)CC2(CSC2)C1 C(=O)(C(C)(C(C)C)OC)N(CC(CC)NC(=O)C=Cc1ccco1)CC C12(C(=O)NCCCCN(C(C3N(CC)CCC3)=O)C)CCC(OC)C1CC2 C(=O)CC(C)CC(C)C.Cc1cc(O)ccc1CN=c1[nH]c(CN2CCCC2)cs1 c1(C(N2CCC(F)(C(=O)NCc3nccnc3Cl)C2)=O)cc(Cl)c2cn[nH]c2c1 c1(C(N(CC#CC)C)=O)cnc(CNC(=O)C#CC2CC2)nc1 CCCN=C(NCCSc1ncc[nH]1)NCC(c1cc(Cl)ccc1OC)(F)F C1(NC(CCCC=C)=O)CCN(C(=O)C(C)OCc2ccccc2C)C1(C)C C1(NC(CC(CNC(C(CC)N(CC)CC)=O)OC)=O)C2CCN(CC2)C1C c1(N(C2CCCCCC2O)C(c2c(C)scc2)=O)ncnc2c(Br)c[nH]c12 n1(Cc2c(NC(N)=O)cccc2)c(=O)ccn(CC2CCCC2)c1=O C1(CN(C(=O)CN(C(=O)COC2CCC2)C2CC2)CC)CC2C=CC1C2 N1(C(C(n2ccc(C)n2)C)=O)CCN(C(=O)Cc2ncccc2C)CC2(CC2)C1 C1(CNC(CSCCCC)=O)CN(C(=O)C(O)C2CC2)CC(C)(C)C1 c1(OC)ccc(CC(=O)NC2CN(Cc3nccnc3Cl)CC2O)cn1 Cc1nn(C)c(C)c1CCCNC(=O)Cc1ccoc1.C1(=O)CN1C1CC1 N1(C(c2cccnc2F)=O)CC(CO)C2(C1)CN(C(=O)C1=CC3(CCOC3)C1)C2 c1(OC)ccc(NNC(=O)N(c2cccc(C)c2F)CC2CC2)c(OCC(N)=O)c1 C1(NC(C(=O)N(C)CC2CCC(C)CC2)=O)CC2C(=O)N(C)CC(=O)N2C1 C12(NC(C(C3CCN(CCC#C)CC3)C)=O)CCC(C1)OC2C c1(C(N(C2CN(C(=O)CCn3ccnc3)CC23CC3)C)=O)cc2ncccc2[nH]1 S(=O)(=O)(CC(=O)NCCOCCCNC(=O)C(F)(F)c1cnccn1)NC N1(C(CC2CCC(=O)O2)=O)CCCCC1CCCCNC(C1CCC(F)(F)C1)=O C1(CC(=O)N(CC(C)CNC(C2(C(N)=O)CCC2)=O)C)CCCCC1 O=CN1CCCC1C(N1CC=CC1C(=O)NC1CC(c2ncc[nH]2)C1)=O CC(CC(=O)N1CCC(C)(NC(=O)CSC(C)(C)C)CC1)P(C)(C)=O C(c1ccc(Cl)c(Cl)c1)=CC(=O)NCCN1CCN(C(C(C(C)O)(F)F)=O)CC1 C=C1CC(C(F)(F)F)(C(=O)NCC2CCN2C(=O)CSc2cnn(C)c2)C1 CC1=C(C(=O)NC2(CN(C)C(c3nc(C)nn3C)=O)CC2)CCC(C)(C)C1 C1(CCNC(C(C)NC(CC)=O)=O)CCCCN1C(=O)CCc1ccc(C)s1 Cc1nc2ncc(C(=O)NC3CC3CNC(=O)Cc3nncn3C)c(=O)n2[nH]1 CC(C)(C#N)CCC(=O)NCC1CN(C(C2Cc3cccnc3C2)=O)C(C)(C)C1 C1(C(=O)NCCCOC)(CC)CN(C(=O)C(C)=C(C)CC)C1 CCC(C)(C)CC(=O)N1CCCC1C(=O)NCc1oc(COC)nc1C N1(C(CCC#C)=O)CCN(C(C2C=CC2C(=O)OC)=O)CC1CC(F)F c1(CC)nc(C)c(C(N2CC3C(C(=O)NCCSC(C)(C)C)C3C2)=O)o1 C1(CC(=O)NC2CC(CCNC(=O)Cc3csnn3)C2)CCC2(CC1)CCC2O N1(C(=O)Cc2csc3ccccc23)CCN(C(c2ccoc2Cl)=O)C2CCCC12 C1(C(=O)Nc2cncc(C)c2)C2CCCC2CN1C(C1CNC(=O)N1)=O Cc1cnc(C(N2CCCOC(CCNC(=O)Cc3cn[nH]c3)C2)=O)cc1Br N1(C(c2[nH]cc(CC(C)C)c2)=O)CC2CN(C(=O)C(N3CCOCC3)C)CC2C1 C1(CC)CC(CC(=O)NC2C3CC2N(C(=O)C(N2CCCC(C)C2)=O)C3)CCO1 c1(C(=O)NCCCOCCN(C)C(C23CCC(C2)C3)=O)ccnc(OC(F)F)c1 C1(OC)CCCC(CNC(=O)C(C)(Cn2cccn2)NC(=O)CCC(C)C)C1 c1(-c2nc(Cc3nc(C)[nH]n3)n(C3CCCC3(C)C)n2)nccn2nccc12 c1(NC(CC2CC(NC(C(C(=O)OC)(C)F)=O)C2)=O)ccc(S(N)(=O)=O)c(O)c1 c1(SC)cc(N2CCOCC2C(=O)NC(c2ccccc2OC(F)F)C)ncn1 CCCCS(=O)(=O)CC(=O)N1CC2CC1CN2C(c1c(Cl)ccc2c[nH]nc12)=O c1(C(N2CC(C)C(NC(=O)C3=CCSC3)CC2)=O)ccc(C#N)cc1O N1(C(C(c2cccc(Cl)c2)OCC)=O)CCC(NC(c2nc(C)n(C)n2)=O)C1C c1(C(N2CC(N(C(CCCC)=O)C)C2)=O)cnc(OC)c(C)n1 N1(C(C2C(=C)C2)=O)CCCCC(CNC(c2ccncc2Oc2ccccc2)=O)C1 N1(C(C2ON=C(C(C)C)C2)=O)CCCC(C)(NC(=O)Cn2ncc(Cl)c2C)C1 c1(OC)cc(S(=O)(=O)N2CCCC(Cc3nccs3)C2)cc(Cl)c1O N1(C(c2ccc(CC)cn2)=O)C2CCC1C(NC(=O)Cn1cc(C)cn1)C2 c1(C(=O)NN2CCNCC2CO)cccc(Br)c1C.c1(CCO)ccc(I)cc1 c1(C(=O)NCCCN(C(=O)C(c2cccnc2)O)C)cc(=O)c(Br)c[nH]1 C(C)(CCC(=O)NCC(C)CNC(c1occc1Br)=O)OC C12(CNC(C3CCCCS3(=O)=O)=O)CCCCC1N(c1ncc[nH]1)CC2 C12(CNC(C3CC3(Cl)Cl)=O)CCC(N(C(C3CCC3)=O)C3CC3)(CO1)C2 CC1(C(=O)NC2CC3CCC2N3C(C2CC(Cl)(Cl)C2)=O)OCCc2ccccc21 N1(C(C2C(C(C)C)OCC2)=O)CC2(CCCC2NC(c2cc([N+](=O)[O-])sn2)=O)C1 C(CSC)(C(=O)NCC1OCCC1C(=O)NC1COCC1N(C)C)OC N1(C(C2(C=C)CC2)=O)CCC(C2CCN(C(=O)C(C)SC(F)(F)F)CC2)C1 c1(C(=O)NC(C(C)NC(CNC(C)=O)=O)CO)cccc2cccc(Cl)c12 C1(CC=C)(NC(c2csc(S)n2)=O)CCN(C(C2CCCC23CC3)=O)C1 CC1CCC(NC(=O)Cc2ccccc2CO)CN1C(C1CC1C(N)=O)=O N1(C(c2n(C(C)C)ccn2)=O)CC2CC(NC(C3CCCOC3)=O)C2C1 c1(C2(NC(=O)NCC(C)N(CC)CC)CCC2)cccc(C#N)c1 c1(CCC(=O)NC(CNC(C2C(CC)OCC2)=O)C(C)C)cccc(N(C)C)c1 C1(NC(COCCN(C)C)=O)CC12CCN(C(C1(C)CCN(C)C1)=O)C2 CC1(C)COCCC1CN(C(=O)CC(C(F)F)n1cccn1)CCO c1(C(N(CCC(C)NC(COC(C)C)=O)C)=O)cnc2c(c1)c(O)nc(=O)n2C Cc1ccc(C(=O)NC2CC(C(=O)Nc3ccc(Cl)c(Cl)c3)C2)c(I)c1C C1(NC(=O)Cc2cccnc2O)CCCCC1CNC(c1ccc[n+]([O-])c1)=O Cc1cc(F)cnc1C(=O)NC1(CCCC(=O)N2CC(CC(N)=O)C2)CCC1 C(=O)(C1CCc2cc(F)ccc21)NCCCN(C(COCCC=C)=O)C1CC1 c1(C(=O)NC2CCCN(C(c3nnc(CC)s3)=O)CC2)c(O)nnc(C)c1C C1(NC(C2(CC)CCC2)=O)CCN(Cc2cccnn2)CC1O S(=O)(=O)(c1ccc(Cl)cc1C(F)F)N1CC(C)CC(C)C1.c12ccc(cc1)CN2 Cc1cc2c(C(=O)NCCC3CN(C(=O)CCc4cnn(C)c4)C3)nccn2n1 CCC(CC(=O)NCC1(O)CCN(C(c2cc(N)ccn2)=O)CC1)C(C)(C)C C#Cc1ccc(C(N2CCCC2CN(C(=O)C(O)C=C)C)=O)cc1Cl N1(c2nnc(C)s2)CC2CC1CN2OC.C1(C=O)CC12CC(O)C2 C(=O)(C(CO)NC(=O)C1CC1)N(CC(CC)NC(=O)C(CC)C1CCOCC1)C N(C1c2ccc(OC)cc2CC1(C)C)C(=O)NCCc1ccc(C(=O)OC)s1 c1(CC(=O)N(C2CCN(C(=O)C(F)(F)c3cccnc3)C2)C)ccc(F)cn1 C1(C(=O)NCc2nc(C(=O)NC(C3CCOCC3)C)sc2)C=CC(=O)N=N1 C1(NC(CCCNC(C)=O)=O)COC2C(NC(c3nc(C)c(C)s3)=O)COC12 N1(C(CCC2CCN(C)C2)=O)CCN(CC(C)(C)NC(C2CC2[N+](=O)[O-])=O)CC1 Cc1nonc1C(=O)NC(C)(C)CCNC(=O)CC(C)NC(C1CCCCC1)=O Cc1c(C(=O)NCC(O)CN(C(=O)Cc2cccc(C(N)=O)c2)C)cccc1F c1(C(=O)NCCC(C)NC(C2(C)CCCOC2)=O)c(O)cccc1Cl N1(C(C(C)CNC(=O)C=CCF)=O)CC2C3CCC(C3)C2C1 n1(CC(=O)NC(C)C(C)(C)NC(=O)CCC23CCC(CC2)C3)ncc(C#N)c1N N1(C(C=CC)=O)CC2(CCC(C(N3CCCCC3CO)=O)O2)C1 c1(OC)cccc(C(C)=CC(=O)NC2(CNC(=O)C3=CCCC3)CCC2)c1 C(=O)(CCCCCC#N)N(CCNC(C1(OC)CC(C)CC(C)C1)=O)C1CC1 CC1CN(C(=O)CC2COCCO2)CC1(C)CNC(=O)C=Cc1ccsc1 c1(NC(C2C(CC)N(C(C3CCC(=O)CC3)=O)CC2)=O)cnn2c1CCCC2 c1(CCN(C)Cc2cccc(Br)c2)ccc(CO)c(F)c1 C=CC1(CC(=O)NC(C)CC(C)(C)O)CN(C(C(C)(CC)CC)=O)C1 CN1CCC(CCC(=O)NCC(C)(CO)NC(c2ccc(F)s2)=O)C1 c1(CC)cc(CC)[nH]c(=NCCC(C)NC(=O)C(N2CCCCCC2)C)n1 C1(C(=O)NC(C(=O)NC(C)Cn2cccn2)c2cccs2)CCCC1C1CC1 C(=O)(CCCC(F)(F)F)N1CC(C(C)NC(=O)C=Cc2cnc[nH]2)C1 CCCCC(CC)CC(=O)NC1CCC1CNC(c1ccc(Cl)c(N)c1Cl)=O C(CC(C(=O)Nc1nccs1)N1CCC(n2cccn2)CC1)N1C(=O)CCC1 c1(CC)ccc(C=CC(N2CCC(CF)(NC(c3cc(OC)cs3)=O)C2)=O)o1 C1(CS(=O)(=O)OC)CN(C(C2CC=CC(n3cc(SC)nn3)C2)=O)CCO1 c1(C(=O)NC(C2CCCN2C(=O)C(N2CCC(C)C2)=O)C)n[nH]c(C(C)C)n1 c1(C(=O)Nc2cnc(F)cc2C(=O)NCC(O)C(F)(F)F)ccc(O)c([N+](=O)[O-])c1 Cc1coc(C)c1C=CC(=O)NCCC1(C)CCN(C(=O)C(C)C2CC2)C1 c1(C(=O)NCC2N(C(C#CC(C)C)=O)CC(C)CC2)ccc2cnoc2c1 Cc1cc(CNC(C2CCC(CNC(c3ccsc3C)=O)C2)=O)sn1 c1(CS(=O)(=O)NC(C2(n3ncc(C)c3)CCC2)=O)ccc(C(C)C)nc1O O=S(=O)(c1ccnc(N2CCC(C3CC(O)CN3c3ccccc3)CC2)c1)C1CC1 C#CC1(NC(C2CCC(CNC(=O)C(C)SCCC)CC2)=O)CC2CCCC12 C#CCCCCC(=O)NCCN(CCOC)C(C1CCCCC1O)=O C12(C(=O)NCCNC(=O)COc3ccccc3C3CC3)COC(CCF)(C1)C2 c1(C(=O)Nc2scc(-c3c(C)noc3C)n2)cc(F)ccc1O N1(C(c2cc(C)cc(Cl)n2)=O)CCC2(CC1)CCN(C(C1C(C)(C)C1(C)C)=O)C2 c1(C(=O)NC2C(CNC(c3c(C#N)ccs3)=O)C2)ncnc2sccc12 Cn1cc(CNC(=O)N(C2CC2)Cc2ccon2)c(CC(C)(C)C)n1 C1(C(=O)NCCCCC(C)NC(=O)C(C)Cc2cnc[nH]2)CCc2c[nH]nc2C1 C1(C(=O)OCC(=O)NCC(c2c(OC)cccc2)(C)C)Cc2c(C)cccc2O1 C(C(C)(C(=O)N(CC(c1nn[nH]n1)C)C)NC(=O)CCCn1cncn1)SC Cc1cc(F)ncc1NC(C1(CNC(=O)C(O)Cn2cncn2)CC12CCC2)=O N1(C(C(COC)OC)=O)CCC2CCN(C(=O)Cc3cnc(OC)c(C)c3)CC12 N1(C(C(N2CCSCC2)C)=O)CCN(C(=O)CCCc2cncs2)C(C2CC2)C1 S(=O)(=O)(c1ccc(I)cc1)N1CCN(C(COc2c(C#N)ccc(F)c2)=O)CC1 c1(C(N2CC3C(NC(C(C)SCCCC)=O)(C3)C2)=O)cnn2c1CC(F)(F)C2 c1(C(=O)NC2C3(NC(C(C)OC)=O)CCC(C2)C3)nc2ccccc2cc1Cl N1(C(C2(CC=C)CCC2)=O)CCC2(CC1)CC2C(=O)Nc1cc(C)ccc1Br N1(C(c2cccc(CC)n2)=O)CC=C(CNC(C2CCC=CCCC2)=O)CC1 C1(C(=O)NCC(C2CC2)NC(C2CC2c2cccs2)=O)C2(CC2)C12CC2 C1(CCC(=O)N(C2CC3CC3C2)C)CCCC(NC(=O)COC2CCCCC2)C1 c1(CNC2CCCC(C)C2)cn(C)c(=O)c2cnccc12 CC1CCc2n[nH]cc2C1C(=O)NCC1CCCN1C(=O)Cn1ccc(=N)[nH]1 c1(CNC(c2cc3c[nH]cnc-3n2)=O)cccc2c1CCN(c1ncns1)C2 C(C(C)CC(=O)N=c1cc(C2CC2)n(C)[nH]1)NC(C(CCC(C)C)F)=O C1(CNC(CCCC(=C)C)=O)CN(C(c2cccn2C(C)C)=O)CCC12CCC2 N1(C(C(CC)N(C)C)=O)C2CCC1CN(C(C1CC(=O)N(C)C1)=O)C2 c1(C(N(CCCN(C(C(C)OCCC#C)=O)C)C)=O)cc(C(C)(F)F)ccn1 C1(C(N(CCN(C(=O)CCSCC(N)=O)C(C)C)C2CC2)=O)CC2OC1C1CC21 C1(NC(CC(C)NC(N)=O)=O)CC(CNC(c2cncnc2)=O)C(O)C1 C1(C(N2CCC(NC(C(C)(C)OC(C)=O)=O)C2C)=O)CCC2(CCC2)CC1 C1(C(=O)N(C(=O)CC2CC3(CC3)C2)C2CC2)(Cc2c(C(C)C)n[nH]c2)CCN(C)C1 CC1(C)CCCCC1NC(=O)CC1CCCN(C(C2CC(=O)C2)=O)C1 CC(CSc1ccccc1)C(=O)NC1CC(C)(CNC(=O)C(C)(F)F)C1 C12(C(=O)NCCOCCCNC(c3n[nH]c4c3CCC4)=O)OCCCC1C2(F)F C1(C)(C(=O)NCCn2c(C)nnc2)C=CCN1C(=O)C(C)n1cccc1 c1(C(=O)OC)cc(C(N2CC(CC(C)NC(=O)Cc3ncc[nH]3)C2)=O)cc(C)c1 C1(C(=O)NC(C(=O)OCC)C2CC2)CCC2CCC1N2C(=O)CN(C)C c1(CC)nn2c(c1C(=O)N(C(C)C(C)C)C(c1cn(CCCF)nn1)C)CCC2 CC1(C)CCCC(NC(C23CC2CN(C(C2(C(N)=O)CC2)=O)C3)=O)CC1 c1(OCC(N2CC3C(CNC(C4(O)CCCC4)=O)C3C2)=O)ccc(Cl)c(F)c1 c1(C(=O)NCC(C(C)C)NC(=O)Cc2cnccn2)ccc(N)c2ccncc12 N1(C(C(C)OCCC=C)=O)CCCC2(C1)CN(C(=O)CCc1ccon1)CCO2 c1(N(C(C(=O)NC(C)CNC(=O)C=CCOC)C)C(c2ccco2)=O)cncnc1 CCC(CC)(CC)C(=O)N1CC2CC1C2NC(C1ON=C(C)C1C)=O CCC(CC(=O)NCC1(OCC)CCCCC1)NC(C1(COCC)CCCC1)=O N1(C(C(CCC)=CCC)=O)CCC2(NC(=O)C3=CCN(C)C3)CC2C1 N1(C(CC2CC(=C)C2)=O)CC(CCNC(c2cnc(N(C)C)nc2)=O)C(C)C1 c1(C(N2CC(CNC(C(C)(Cl)Cl)=O)OCC2)=O)cc(S(=O)(=O)NC2CC2)c[nH]1 C1(CF)C(=O)N1.c1(OC(=O)CC2CC(O)C2)ccccc1.C12(CC1)C(=O)N2 c1(CC(N2C(CNC(CCSC)=O)C=CC2)=O)c[nH]c2cc(Cl)ccc12 C1(Cc2cn(NC(C=C(C)C(=O)O)=O)nn2)CCC2CCC12 N1(C(C2(C#C)CCCC2)=O)CC(C)OC2(CCN(C(=O)COC(F)(F)F)C2)C1 C1(NC(C(=C)Cc2ccccc2)=O)COCCN(C(=O)CSC)C1 C1(C(C)NC(c2cscc2C(F)F)=O)CN(C(=O)CCN2CCOCC2)CCO1 c1(C(N2CCCC(CNC(Cc3ccc(SC)cc3)=O)C2)=O)cn2ccnc2s1 c1(C(=O)NCc2cnc(C)s2)cccc2c1CN(C(c1ccncc1C)=O)CC2 c1(C(=O)NCC(C)NC(C(CCC)C)=O)ccc2cc(C)ccc2n1 c1(CC(=O)OCc2csc(SCc3ccccc3)n2)ccc(F)c(Br)c1 NC1CCOCC1CNCC(F)(F)Cn1cccn1 c1(C(N2CC(NC(C3(NC(C)=O)CCOCC3)=O)C(C)C2)=O)csc([N+](=O)[O-])c1 C(=O)(C(C)CC(F)F)NC1(C2CCC(NC(CCCC)=O)CC2)CC1 C1(NC(C(N(C)C)C2CC2)=O)CN(C(c2cc(F)c(F)c(F)c2)=O)CC2(CC2)C1 C1(CC(=O)N(C)CC2CCN(C(C(n3cc(Cl)cn3)C)=O)C2)CC2C=CC1C2 N1(CC(=O)OC)CCN(C(C(=O)NC(C)C)C(C)C2CCC2)CC1C c1(OC)cccc(C2=NOC(C(N3CCC(CN=c4cc[nH]cc4C#N)C3)=O)C2)c1 O=CN1CCCC1C(=O)NC(N(c1ccccc1)CC12CC(C(F)(F)F)(CO1)C2)=O N1(C(=O)OC)CCCC(C(N2CC3C(NC(C4SCCCS4)=O)C3C2)=O)C1 N1(C(C2CCCCCC2)=O)CCC2CCN(C(c3nccc4occc34)=O)C2C1 N1(C(c2ccn(COC)n2)=O)CCOC2(CCN(c3snc(Cl)c3C#N)CC2)C1 N1(C(CCCCC=C)=O)CC(C(N2CCOC(C(C)(C)C)C2)=O)C2(CCC2)C1 C12(NC(C(=O)N(C(C)C)Cc3nc(Br)cs3)=O)CC(C)(C1)OC2(C)C C1(C)(CC)CC(NC(c2c(F)cccc2F)=O)CN1C(c1cncnc1C)=O C(=O)(C(O)C(F)(F)F)N1CCCC(CCC(C)(C)NC(CCSCCC)=O)C1 c1(CC(=O)NC(C(=O)NC(c2cnn(C)c2)CC)C)csnc1C.C(COC)S C[Si](C)(C)c1ccc(COC(C23CCC(O)(CC2)C3)=O)cc1 c1(C(C(C)NC(=O)NCCCCc2ccccn2)OC)ccccc1F c1(C(=O)NCCC(C(=O)NCc2ccnc(O)c2)OC)cc(C)nc(O)c1 N1(C(c2c(CC)cccc2)=O)CC2CC(C1)N(CC(N1CC3CCC1C3)=O)C2 c1(CC)cnc(F)c(-c2cccc(N3CCN(C(=O)CCOC)CC3)c2)c1 N1(C(c2nc(CC)oc2)=O)CCC(NC(=O)CSc2cccc(OC)n2)C12CC2 NC1C=CCN1C(C(=O)NCCCF)c1csnn1 c1(C(N2CCN3CCN(CC3C)CC2)=O)coc2cc(O)ccc12.CCCOC C1(C(=O)NCCC(=C)CO)CC(C)(C)CN1C(=O)CC(C)(F)F CON(CCC(=O)NO)C(=O)c1coc(CC2CC2c2ccccc2)n1 c1(CC(=O)NC23C(n4cc(C5(SC)CC5)nn4)CC(CC2)C3)ccc(C#N)c(Cl)c1 N1(C(C=CC(=O)OCC)=O)CCC=C(C(=O)NOCC(C)(C)O)C1 N1(C(COCCCCC)=O)CCCC1C1(NC(=O)C(=O)NCC2CC2)CC1 N1(C(CC2(C)CCCC2)=O)CCC(O)(CNC(c2coc(C3CC3)n2)=O)C1 N(C1CC(C)n2ncnc21)C(c1n(CCC)cnc1)c1nnnn1C1(C)CC1 CC(C)CCCCC(=O)N(C1CCC2CN(C(C3(C)CCSCC3)=O)CC12)C N1(C(C(c2n(C)ccc2)=O)=O)CC=C(C(=O)NC2CCC(C)(C)C2)CC1 C1(C(=O)NC(C2CCCC2)C#C)CCCC(NC(=O)CCCOCC)C1 N1(C(C2CC(C)(C)C2C(F)(F)F)=O)CCC(CO)(NC(=O)Cc2cc[nH]n2)CC1 C(C)(CO)(C(=O)N(CC(C)(C)C#N)C)NC(CCC)=O C(C(CC1CC1)C(=O)Nc1cnccc1SC)NC(C(C1CCC1)OC)=O C(N=c1[nH]c(NCC2CC(F)(F)C(=O)N2)nc2c1CCC2)C1(C)CC(C)(C)C1 N1(C(CC(=O)OCC)=O)CCC(C)C(NC(=O)CC(C)C2CCCO2)C1C C(=O)(CC(C)CC(C)(C)C)NCC(CC=C)C(=O)N1CCN(CC)CC1C c1(C(N2C(C(=O)NC(c3ncccc3F)C)CC3CC32)=O)c[nH]c2nccc-2c1 C(N=c1[nH]c(N2CCCC2)nc2c1CSC2)c1c(F)ccc(OC)n1 c1(CNC(C2CC(n3cc(C(C)(C)O)nn3)C2)=O)cnc(C(=O)O)s1 C1(NC(c2cc(C)no2)=O)CCN(C(=O)Cn2ccc(=O)n(C)c2=O)CC1(C)C c1(C(N(C(C)CCNC(C2CCC(C)O2)=O)C)=O)cccn(C2CCC2)c1=O CC1C(NC(=O)COC2(C)CCC(C)C2)CCN1C(=O)CCc1ccccc1 N1(C(CCOCCC)=O)CCCC(C(C)N(C(=O)CC=C(Cl)Cl)CC)C1 c1(NC(C(CC)OC)OC)nc(C(=O)O)n2ccccc12 N1(C(C=Cc2n(C)ncc2)=O)CCN(C(=O)CCc2cncs2)C(CO)C1 N1(C(CC2C(C)=NNC2=O)=O)CC2(C(=O)NCC3(C)CNC(=O)O3)CC1CCO2 CCC(CCCO)N=c1[nH]c(N2CCOCC2)nc(=NCc2cnn[nH]2)[nH]1 C1(NC(C2(CC)CCCCO2)=O)CC=C(C(=O)N2CCCC(CN(C)C)C2)C1 N1(C(C(N2CC3CCC(C)(C)C3C2)=O)=O)CCC(O)C(F)(F)CC1 C(=O)(C1=NOC(C)C1C)NC1C(SC)CN(C(C2CCCOC2)=O)C1 c1(CN(C)CC2CCN(C(CCCCC=C)=O)C2)ncccc1C#N n1(CC(=O)NCC(COC)NC(CC2C(CC)C2)=O)cc(Cl)c(C)n1 c1(C(=O)NCc2[nH]cnc2C)cc(Cl)ccc1N(C)C(C1CCCN(CC)C1)=O c1(CC(=O)NC2CN(C(C(c3ccc(C)cc3)=O)=O)C(C)C2)cc(O)nc(O)n1 C(CCCCC(=O)N(CC(C)NC(=O)CC1(N(C)C)CC1)CC)=CCCC C(C(O)CC(F)(F)F)NC(=O)NCc1noc(-c2cccc(F)c2)n1 Cc1cccc2c1OCCCC2NC(N1CCC(F)C1)=O C#CCC(C(=O)NC(=O)CCC)NC(C1CC(C)(C(=O)OC)C1)=O N#Cc1ccc(O)c(NC(=O)C(Cn2ccnn2)NC(c2c[nH]cc2C2CC2)=O)c1 c1(OC)ccc2[nH]cc(C(=O)NC3CCOCC3NC(C3CSC3)=O)c2c1 C1(C)(CC)CCC(CNC(=O)C(C)(CO)NC(c2csnc2OC)=O)O1 c1(C(N(CCOC)CCNC(c2cc(C)sc2C)=O)=O)cncn(C)c1=O N=c1nc(Cl)cc(C(N2CCCC(CNC(=O)CCN3CCCCC3)CC2)=O)[nH]1 Cc1nn(C)c(C(=O)NCCC2CCCCN2C(=O)C(C)C2CC2)c1Br CCC(CC)C(C)C(=O)NCC1(F)CCCN(C(c2c(C)cncc2O)=O)CC1 Cc1c(NC(=O)C(=O)NS(=O)(=O)Cc2cccc(Cl)c2)cccc1Cl C(=O)(C1=CCCOC1)NCC1N(C(CN(C)C(c2cccs2)=O)=O)CCC1 CC1CCC2(CC1)CCN2C(=O)C(=O)NCc1ccc(F)c(Cl)c1 C1(C2CCC2)(C(N(C(C)CN(C(=O)CCCn2cncn2)C)C)=O)CC1 N1(C(C=CC(C)(C)SC)=O)CCCCC1C1CCN(C(c2ccc(Cl)s2)=O)C1 C1(C(N2CCN(C(C3C(C(C)O)C3)=O)CC(O)C2)=O)CC(c2cnn(C)c2)=NO1 c1(CN2CCC(CC(CC)C)C2=O)cccc(N)c1F N1(C(C(C)Cn2cccn2)=O)CC2(COC(CNC(c3ccccc3O)=O)C2)C1 Clc1ccccc1-n1nnnc1COC(c1ccco1)CC1CC1 c1(C(=O)OC)ccc(O)c(C(=O)NC2CC2CNC(c2csc(Br)c2)=O)c1 Cc1cc(C(=O)NCC#CCNC(c2ncc(Br)cn2)=O)c(C)n1C1CC1 Cc1cc(=NC(=O)CN(C(C)(C)CO)C(c2cccc(F)c2C)=O)[nH]o1 c1(CN(C2CC3CNC2C3)C(C2COC(=O)O2)=O)c(F)cccc1F N1(C(CC(C)OC)=O)CCC2(C(=O)Nc3ccccc3)CC2C1.[nH]1c(O)nnc1O C(=O)(C(C)(C)CC(F)F)NC1C(NC(c2onc(COCC)n2)C)CCCC1 c1(C(=O)NCC2(C)OCCN(C(C=NOC)=O)C2)cccc2c1CCS2(=O)=O C1(O)(C(C)NC(CN(C(=O)OC)C)=O)CCN(C(=O)Cn2cnccc2=O)C1 C1(CCNC(=O)CCc2ccc(C)o2)(OC)CN(C(c2ccoc2)=O)C1 CCS(=O)(=O)CC(=O)N1CC2C(C(=O)Nc3c(C)cccc3C)C2C1 C1(CC)CCCN(C(c2cc(C3CC3)n(C)n2)C(=O)NCC2CCCO2)C1 C1(C(=O)NC(C)CC2CN(C(=O)C=CCN(C)C)C2)CCCC(C(C)C)C1 c1(C(N2C(CCNC(c3c(C)cnnc3)=O)COCC2)=O)ccc(Br)c(F)c1 C1(C(N2CC(CCC=C)(C(=O)NC3CCN(C)C3=O)C2)=O)COCCN1C c1(NC(C2C3CN(C(C(CCC)CCC)=O)C2C3)=O)ccc2c(c1)OCCO2 c1(C(=O)NCC#CC(=O)NC(CO)C2CC2)c[nH]ccc1=O N#Cc1cncnc1C(N1CC(CO)(NC(C2CCN2S(C)(=O)=O)=O)C1)=O C1(CNC(C(Cc2cn[nH]c2)NC(C(=O)N(C)C)=O)=O)CCNC(=O)C1 c1(C(C(C)NC(=O)NCc2c(I)ccnc2F)OC)cc(Cl)cc(Cl)c1 C1(NC(c2nc(C)oc2C)=O)C(C)(C)C(NC(c2cc(Cl)ccc2F)=O)C1(C)C CCC(CC)CC(F)C(=O)NC(C)CC(=O)N(C)CC1CCCN(C)C1 c1(C(N2CC(CC(=O)OC(C(C=C)NC(C)(C)C)=O)C2)=O)ccc(C(F)(F)F)cn1 c1(C(=O)NCC2(C)CC(NC(C(CCOC)C)=O)C2)cc([N+](=O)[O-])c(C)s1 C1(CCC)(NC(=O)Cc2cc(Cl)cs2)CCCN(C(=O)CCc2cc(C)no2)C1 CC(CF)C(=O)NCC(C)(C1CC1)NC(=O)CSS(C)(=O)=O C1(NC(c2cccs2)=O)CN(C(=O)Cc2ccc(Br)cn2)CC2CC12 c1(N(CCCc2ccccc2Br)C)nc2ccc(Cl)cc2c(=NCC2CC23CC3)[nH]1 C1(C(=O)NC2CCN(C(CN(C)C)=O)C2)(N(C)C)CCCCC1 CC(=O)CCCC(=O)NC1CCCC(C(=O)Nc2c(C)ncn2C)C1 c1(C(N2CC(OC)(CNC(C3CC4CC3C3CC43)=O)C2)=O)scc2c1OCCO2 C1(C(N2CCC(C)(CNC(=O)Cc3ccsc3)C2)=O)C2CCC3C(C2)CC13 CC1CN(C(C2C3CCCC23)=O)CCC1N(C)C(c1cn(C)ccc1=O)=O CS(=O)(=O)c1cnn(CCNC(=O)C(=O)NC2CC2(F)F)c1 c1(CN(C(C(=O)NCCOC)C2CC2C)C)cc(Br)nn1COC CCC(CC)(O)C(=O)N1CCOC(CN=c2nn[nH]n2-c2ccccc2)C1 CC1CCCC=C1C(=O)N1CCC2CN(C(c3ccc(F)cc3Cl)=O)C2C1 N12CCOC3(CCS(=O)(=NC(=O)CC1=O)CC3)C2.CC(C)(C)C(=O)NCC1CCCS1 N1(C(c2n(C)ccc2)=O)CCC(CO)C(NC(C2(C)CCCNC2=O)=O)C1 C1(C(=O)NC(CCNC(CCS(=O)(=O)NC)=O)C)Cc2ccncc2N1 C(=O)(C1=C(C#N)CCC1)NCC1CCCC(NC(c2ccc(C)s2)=O)C1 CC1(C)CCN(C2CC2)C(=O)CC(=O)NC1=O.C(CCO)SC1CC1 C(=O)(CC(C)C(C)C)N1CCC(C)(C(NOCCCC)=O)CC1 C1(C(N2CCCC(NC(CC(CC)CN(C)C)=O)C2=O)=O)CNC(=O)CC1(C)C C(C)(C)(CCCNC(c1[nH]ccc1CNC(c1c(C)nsc1N)=O)=O)OC Cc1nn(C)c(NCC(c2ccccc2)Oc2ccc(Cl)cc2)c1C#N c1(CCC(=O)NCC(C(C)C)NC(C23CCCN2CCC3)=O)ccc(Cl)c(F)c1 c1(C(=O)NCCCN(C(CCC(CC)OC)=O)CC)cc2nccnc2cc1F CC1(C)C2CCC(C2)C1C(=O)NCC(C)(C1CC1)NC(=O)C=CC(F)(F)F C1(C(N2CC3CCC2C3)=O)CCCCN1C(=O)Cc1ccc(Cl)cc1 C1(C(=O)NCC2(C)CC(NC(c3cnco3)=O)C2)CC2C(C1)C2(F)F c1(NC(N2CC(CCC)C2)=O)ccn2nccc2n1 CC(C)C(F)(F)CC(=O)N1CCC1CNC(C1CCN1S(=O)(=O)C1CC1)=O N1(C(c2ccn(CCNC=O)n2)=O)CCC(OCC(=O)SCC)C1.C1CCO1.OC C(C(=O)NCc1ccc(F)cc1)(C(CC)CC)N1CCC(CN(C)CC)C1 c1(NCC2CCN(C(C3C(COC)C3)=O)C2)ncccc1C(=O)OC C(C1=CCN(Cc2cccc(C(F)(F)F)c2N)CC1)NC(C=CCC)=O C(=O)(C1COc2ccccc21)NC1CCCC(NC(C(CSC)(C)C)=O)C1 CCC(CC)(CCC(=O)NCCCC(C)(C)NC(c1nocc1CC)=O)[N+](=O)[O-] C(=O)(C(CNC(=O)C(C1CCC1)OC)CC1CCCC1)NC(CN(CCCC)C)C C(c1ccccc1)=C(OC)C(=O)NC1CCCC1CN(C(=O)CC(C)O)C C1(CNC(Cn2ncc(CC)c2)=O)CN(C(=O)C=CC(=O)N(C)C)CC1(F)CO c1(C(N2CC(CNC(CC(CC)O)=O)N(C)CC2)=O)ccc2c(C)[nH]nc2c1 C1(N(C(c2cn(CC=C)nn2)=O)C)CCCN(C(c2ccc(OCC)nc2)=O)C1 c1(NC(C2CNCCN2Cc2cc(Br)ccc2F)=O)ccnc(Cl)c1I N1(C(CONC(Cc2scc(C)c2)=O)=O)CCOC2COCCC12 Cc1oc(C(=O)OCC2(C)OCCCO2)cc1-c1ccccc1 c1(C(=O)NC2(CF)CCN(C(C(C)OCC=C)=O)C2)cc(=O)c(Br)c[nH]1 c1(C(N2CCC(C(C)NC(=O)C=CCN3CCCC3)C2)=O)nc2ccccc2[nH]1 c1(NC(=O)C(N2CCCC2c2ccc(F)cc2)=O)nc2ccc(F)cc2s1 N1(C(C=C(C)C)=O)CC(CC(=O)NCC2CC(F)C2)C2(CC2)C1 C1(C(=O)NCC(C)N(C(c2c(Cl)c(C)n(C)n2)=O)C)CC(C(C)(C)C)=NO1 N1(C(Cc2ccc(C)o2)=O)CCN(C(=O)CC2=CCCC2)C2CCCCC12 c1(C(=O)NC2CCN(C(C(CC)N(CC)CC)=O)C2C2CC2)scc2c1OCCO2 C#CCCC(C(=O)N1CC(C)(CF)C1)NC(c1cnncc1)=O C(=O)(C1=NOC(C2(O)COC2)C1)N(CC(CC)NC(c1cnnc(Cl)c1)=O)C C1(CSCC2OCCC2)CCCC2(CNC2)O1 CC1CN(C(=O)Cc2ccc(F)c(Cl)c2)CCN1c1ccc(F)cc1 C=CC1(C(=O)NCCCCC(C)NC(=O)CC(C)(O)C2CC2)CCOCC1 S(=O)(=O)(c1cnn2ccc(=NCC(C)(C)C3CC3)[nH]c12)N(C)CC1CCCC1O c1(CC)conc1CC(=O)NCC(CC)NC(=O)C(F)(F)C1CCOCC1 N1(C(Cc2cnc(C)s2)=O)CCC2CN(C(c3cccc(Br)c3F)=O)CC12 C1(NC(c2nc(CC)oc2)=O)CN(C(c2c(Br)cncc2Br)=O)CC12CC2 CC(C)C(O)C(F)(F)C(=O)N1CC(NC(c2ccc([N+](=O)[O-])o2)=O)CC2(CC2)C1 C(=O)(N=c1cnc(I)c(Cl)[nH]1)C1N(C(c2ccc3ncn(C)c3c2)=O)CC1 Cc1cc(Cl)ccc1OCC(=O)N(CC(C)NC(C1CCC(C)(C)C1)=O)C C(C1CCCCC1)=CC(=O)NCC=CC(=O)NCc1nc(C)oc1 Cc1c(C(=O)NC2(C)CC(NC(=O)CCS(=O)(=O)N(C)C)C2)cccc1F C1(NC(C2C3CN(C(c4coc(C5CC5)n4)=O)CC23)=O)CCN2CCC1C2 N1(C(C2(CC#C)CCCO2)=O)CCC2(CCCN(C(=O)Cc3nccn3C)C2)C1 N1(C(c2cc(C)nc(Cl)c2N)=O)CC2CC(O)C1C2NC(c1c(OC)csc1)=O C(=O)(CC(F)(F)C(F)F)N(CC(=O)NC1(C#C)CCOC1)C1CC1 c1(C(=O)NCC2C=CC(NC(c3cnsc3)=O)C2)ccc(F)c(O)c1 N1(C(c2c(C(=O)OC)ccnc2)=O)CCCC(C)(C=CCCN(C)CCOC)C1 N1(C(c2nn(CC)c(C)c2)=O)CCC(CNC(c2cccc(C)c2Cl)=O)C1(C)C c1(C(=O)NCC(CNC(c2ccc(C(C)=O)o2)=O)O)cccc2ncnc(O)c12 N1(C(C2CCCN(C(C)C)C2)=O)CCC2(CCCN2C(=O)C=Cc2cscn2)C1 C12(C(=O)OCC)CCC(NC(c3cc(Cl)cnc3F)=O)(CC1)C2 c1(C(C(=O)NC(CCNC(c2c(C)cno2)=O)C)O)ccc(F)c(Cl)c1 C1(C(CNC(CC2(C=C)CCC2)=O)(C)O)CCN(C(C2CCCCC2)=O)CC1 O=S(=O)(c1cnc(N2CCOCC(O)C2)c(Cl)c1)NCC1COCO1 C1(NC(c2c(C)nc(O)s2)=O)CCN(C(c2cc(Cl)ccn2)=O)C1(C)C C1(C(=O)NC)(NC(=O)CC(C)(C)n2cc(-c3ccc(C)s3)nn2)CCCCC1 CN1CCC(NC(=O)NCCCNC(=O)CO)C1c1cccs1 C1(c2ccccc2Cl)(C(=O)NC2C(NC(C3(CCC=C)CC3)=O)C2)CCCCC1 C(c1nc2ccccc2s1)=CC(=O)NCCN(C)C(C1CCC=CCC1)=O C1(C(=O)NCCc2c(C(NOCCC(C)O)=O)c[nH]n2)C2CCCC(=O)C12 C#Cc1cnn(C)c1C(=O)NC(CC(C)C)C(=O)NCC12CCC(CO1)C2 c1(C(=O)SC)ccc(NC2CCNC2c2ccccc2)c(F)c1 c1(C(N2CC3C(C(N(CCOC)C)=O)(COC3)C2)=O)cn2cccc(C)c2n1 c1(NC(CC)(CNC(=O)CC2CC=CCN2C)CC)ncc2ccnc-2[nH]1 C1(NC(CCCOC(C)C)=O)COCCN(C(=O)CC=CCc2ccccc2)C1 C(=O)(CC(=O)N1CC(Oc2ccccn2)C1)N(C)CC1(CO)CCCO1 c1(OC)ccc(C(=O)NCC2CCCCN2C(=O)C=CC(C)C)cc1C(F)(F)F C12(C(N3CC(C=C)C(NC(=O)CCCCC)C3)=O)CCC(NC)(CC1)CC2 CCC(C)CC(=O)N1CCCCC1CCn1cc(CN(CC)CC)nn1 c1(-c2cn(C(C)=O)nc2)ccc2[nH]cc(C(=O)Nc3cc4ccoc4s3)c2c1 Cc1cc(NCC2CCN(C(C)C(C(=O)CC(C)(C)C)=O)C2)nn1C.C1C(=O)N1 C1(CCNc2nccc(N3CCC(CC)(CO)C3)n2)CCC2(CCOCC2)CO1 c1(C(=O)NC2(C)CN(C(=O)C(F)(F)Cc3ccccc3)C2)cc2ccccc2o1 CN1CCN(C(=O)CC2CC3(C2)CN(C(=O)C(F)(F)CO)C3)CC1C(C)(C)C N1(C(CCc2cnn(C)n2)=O)CCCCCC(NC(c2n[nH]cc2C2CC2)=O)C1 c1(OC)cnc(Cl)cc1C(=O)NC1CC(CNC(=O)C2=C(Cl)CCC2)C1(C)C c1(CN2C(C(N3CCC(O)C(F)C3)=O)CC(F)C2)c(Br)cccc1[N+](=O)[O-] C1(CNC(C(C2CCCCC2)C)=O)CN(C(c2cnc(O)n2C)=O)CC1O C12CCN(C1)CC(O)COCC2.c1(NC(C2CCCC2)=O)ccccc1 c1(OC)ccc(Cl)cc1C(=O)NCC(C)(C)CN(C)C(C1CCOC1C)=O C(CC(=O)NC(CO)C(C)(C)C)(C(C)C)NC(C1(COC)COC1)=O Cc1scc(C(N2CCC(N3CCN(C(C4C=CCCC4)=O)CC3)C2)=O)c1N C(CC(C)(C)C(=O)NCC(C)O)NC(c1c(C)cccn1)=O N1(C(C(C)OCCC=C)=O)CCC(CNC(c2coc(Br)n2)=O)(OC)C1 c1(C(=O)NC2CCC(N(C(c3cc(C)sn3)=O)C)C2)c(Cl)ccc(C)c1N C(=O)(C(O)C1=CCCCC1)NCC(CC)(CC)C(=O)NCC1CCCC12CCC2 c1(OCCC(N2CC(O)(CNC(C3C(C)(CC)C3)=O)C2)=O)ccc(C)cc1C Cn1nncc1CC(=O)NCC1(O)CN(C(=O)CC2(C)OCCO2)C1 CCN=c1cc(C(=O)NC2(CNC(=O)C(F)(F)c3csc(C)c3)CCC2)cc[nH]1 c1(C(N2CCN(CCNC(COC)=O)CC2)=O)cc(=O)c2ccccc2o1 C1(NC(c2c(NC)scn2)=O)COCCC1NC(=O)CCOCCOC C1(CNC(C2C(C)(C)COCC2)=O)CCN(C(C2(O)CCCC2)=O)CCC1(F)F C(CCN=C(NCCC(C)(C)C)NC1C(C)(C)C1(C)C)SC c1(C(C(=O)NCC2CCC(NC(c3ccoc3Cl)=O)C2)O)ccc(F)c(Cl)c1 O=C(C#CC1CCCO1)NCC1(O)CCN(C(=O)CCc2ccc(O)cc2)C1 c1(CC(=O)NC2C3CN(C(C(C(C)(C)C)SC)=O)CC32)ccccc1S(N)(=O)=O N1(C(C(C(C)C)N(C)C)=O)CC2OCC(NC(=O)CCc3cccc(F)c3)C2C1 Cc1ncnc(C)c1CC(N1CCC(OCCNC(=O)C=CC2CCCC2)C1)=O C1(NC(C2CC(=O)NC2)=O)CCCC12CN(C(=O)CSCC1CCCO1)C2 c1(C(N(CC(=O)Nc2ccc(Cl)c(Cl)c2)C)=O)cccc(S(C)(=O)=O)c1 N1(S(=O)(=O)Cc2ccccc2)CCCC(OC2(C(F)F)CCOCC2)C1 c1(C(N2CCC(C(N3CC(C)(OC(C)=O)C3)=O)(CC)C2)=O)ccnc(O)c1F Cc1cc(C(=O)NCCNC(=O)CCC2NC(=O)NC2=O)n(-c2ccccn2)n1 C(=O)(CC1=CCN(C(=O)C(C)C(F)F)CC1)NC(C)C(=O)NCCF CC(C)C(CCCC(=O)O)NC(c1ccc(Sc2ccccc2Cl)cc1)=O CC1=C(C)CC(C)(NC(=O)CC2C3CCC(C3)N2C(c2ccncn2)=O)CC1 C1(CNC(=O)CCc2cnco2)CC2(CCOCC2)CN1C(=O)CCCC1CC1 c1(CN2CC(C(=O)Nc3ccc(I)c(Cl)c3)C(O)CC2)ccc([N+](=O)[O-])cc1Br Cc1ccc(C(N2CCC(C)C(NC(=O)CCSC(F)(F)F)C2)=O)cc1C#N Nc1cccc2c1ccn2CC(=O)NCC1CC1NC(=O)Cn1ccnn1 n1(CC)ccnc1-c1cn(CCCCCNC(C2CCOC2CC)=O)nn1 c1(C(CC)NC(C(COCC)n2cc(COCC)nn2)=O)nnc(C)n1C c1(C(=O)NC(CCC(=O)NC(CC)CC(=O)OC)(C)C)ccc(F)c(O)c1 c1(CNC(C(CC)C)=O)ccc(CN(C(C2CCN2S(C)(=O)=O)=O)CC)c(F)c1 c1(C(=O)NC2CC(O)C2C(=O)O)cccc(C(F)(F)F)c1 N1(C(CS(C)(=O)=O)=O)CCC(NC(=O)Cc2cn3c(n2)CCCC3)C12CCC2 C1(CC(=O)NC(C2C(C(=O)NC(CC(=O)OC)C)C2)C)CCCCC1O N1(C(Cc2nc(OCCCC)sc2)=O)CC2CN(C(=O)OC(C)(C)C)CCC12 Cc1cc(F)cc(C(=O)N(C2CN(C(c3c(O)cccc3F)=O)CC23CC3)C)c1C Cc1nc2cc(C(=O)NC(C3CN(C(=O)Cc4cnc[nH]4)C3)C)ccc2o1 Cn1nc(-c2cccnc2)cc1C(=O)NC1CC1NC(=O)CC1CCCC1O CC1(NC(=O)CCc2cc(F)ccc2F)CCN(C(C2CCCCN2N=O)=O)CC1 C1(CNC(C2C=CCN(C(c3cnn(C)c3Cl)=O)C2)=O)CC2(CCC2)CO1 C1(CN(C)C(c2cn(C)nn2)=O)COCCN1C(=O)C(c1ccccn1)O N1(C(c2c(CC)n(C)nc2)=O)CCC(NC(C2(C)CC2C)=O)C(C(N)=O)C1 N1(C(c2cc(SC)n[nH]2)=O)CC2(C1)CN(C(c1cccc3scnc13)=O)CCO2 Cc1cc(C)c(C(N2CC(CNC(c3cnc(C)o3)=O)C3(CCC3)C2)=O)c(C)n1 N1(C(C(C)=C2CC2)=O)CC(CNC(=O)COCC2CCOCC2)CC12CCC2 C1(CCC)(NC(=O)CN(C)C2CC2)CCN(C(c2c(C)nn(CC)c2C)=O)CC1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCC(CO)NC(C(C(C)(F)F)(C)C)=O C1(C(N2CCC(NC(C3(F)C(C)C3)=O)C2c2ccccc2)=O)CCC2(CC1)CC2 C(=O)(C(C)C(=O)OC(C)(C)C)NCC1(C(C)NC(CCC=C)=O)CC1 C1(O)(Cn2cc(CSC)nn2)CCN(C(=O)C(=O)CC2CCCO2)C1 CC1(C)CC=C(C(=O)N2CCCC(CNC(c3ccc(O)cc3)=O)C2)CC1 Cc1ccc(CC(=O)NCCOCCNC(c2occc2C)=O)c(Br)c1 C(=O)(CCN=c1[nH]c2ccccc2s1)NC1C(CNC(CCC(N)=O)=O)CCC1 C1(C(=O)NCC(C(=O)NC)O)CC(C)CN(C(=O)CC(C)(C)O)C1 c1(CC(=O)NCC2(NC(c3ccc(C(F)F)o3)=O)CCOC2)csc2nccn12 CCCCC(CC(=O)N1CCC(C)(CCO)C1)NC(c1ccc(O)nc1C)=O C1(C(N2CCC(C)N(C(=O)Cc3cnn(C)c3)CC2)=O)CCC2(CC1)OCCO2 N1(C(C(=O)NCCOC)=O)CCCN(C(=O)Cn2cc(Br)c(C)n2)CC1 C1(NC(CCC(=O)NCCC)=O)CCN(C(=O)C(OC)OC)CCC1CO C=C(Cl)CC(C(=O)NCC(O)CC(=O)OC)NC(C1CCN1CC)=O C1(C)(C(=O)NC2C3(CC(NC(C4OCCN(C)C4)=O)C3)C2)Cc2ccccc2C1 c1(C(=O)NCCC2(NC(c3ccc(C)s3)=O)CC2)cc(O)nc2cnccc12 CC1(C)COC(C)(C(=O)NC2CCCN(C(=O)CCCc3ccncc3)C2)CO1 c1(C(=O)NC2(CF)CCN(C(c3nccs3)=O)C2)cc2c(s1)CCCC2 C1(CC=C)(C(=O)Nc2cccc(C3CC3)c2)CCCN1C(C1(OC)CCC1)=O c1(C(N2CCN(C(C3CC(C)CC(C)C3)=O)CC2)=O)cc2cc(O)ccc2[nH]1 N1(C(c2cc(C)sn2)=O)CCN(C(c2ccc(SC(F)(F)F)o2)=O)CC1COC CCCC(CC)C(=O)NC1CCC(C)N(C(=O)Cn2nnc(C)n2)C1 c1(CC(=O)NC2CC2C(=O)Nc2cnc(Cl)c(Br)c2)cccc2sccc12 C1(F)(CNC(c2ccn(CCC)n2)=O)CCC(CNC(C2CC2[N+](=O)[O-])=O)C1 c1(C(=O)NCCC(C)N(C(C(C)N(CC)CC)=O)C)c(CO)ccn1C.C(=O)C1CC1 Cc1ccc(C)c(C(N2CCC2C(=O)N(C2CCCC2C#N)C)=O)c1 N1(C(Cc2ccc(OC)cc2)=O)CC2(CNC(=O)C=C3CCCC3)CCC1CC2 c1(C(=O)NC2C(NC(CSCCC)=O)CCOC2)ccc2nncn2c1 CCCCCC(O)CC(=O)N(C(C)CCNC(=O)CC1CCCN1C(C)=O)C Cc1nccc(Cl)c1C(N1CC(Cn2cc(-c3ccnn3C(C)(C)C)nn2)C1)=O c1(CNC(C)=O)nc(CNC(=O)C(c2ccccc2)C)cc(O)n1 N1(C(c2c(COC)scc2)=O)CCC(CF)(NC(c2nc(=O)n(C)[nH]2)=O)C1 c1(CC(N2CCN(Cc3ccc(C(F)(F)F)nc3)C3CC23)=O)cc(F)ccc1Cl N(C(=NCCC1=CCCCC1)NC(c1ccco1)C)Cc1nc(COCC)on1 CCC(CC(=O)N1CC(C(N2CC(C)(C)CC2C)=O)C(C)(C)C1)C(F)F C1(C(=O)NCCC(C)NC(Cc2c(C)coc2C(C)C)=O)CC12CCOCC2 c1(CC(=O)N(C2C3CN(C(c4c(C)nc(CC)o4)=O)CC32)C)ccc(O)cc1C c1(C(=O)NC(C)CCNC(C2(C(F)F)CCC2)=O)ccc(Br)nc1O C(=O)(C1=CCC(NC(c2scnc2CC)=O)C1)NC(C#C)C1CC1 c1(C(N2CCC(NC(CNS(CCCC)(=O)=O)=O)C2)=O)c(C)cccc1F c1(C(=O)NC2(CN(C)C(C3CCC(F)C3)=O)CCC2)cc(O)ccc1Cl c1(C(N(C2CN(C(=O)COC(F)F)CC2F)C)=O)cc(F)cc2nn[nH]c12 C1(CC)CN(C(c2ccc(OCC(=O)OC)cc2)=O)CCN1C(C1CC(O)C1)=O N1(c2cccc(C)c2)CC2CCCCC2C1C.N1(C(C(CCC)F)=O)CC(C(=O)N)CC12CCC2 c1(CCC(=O)NCC(CC=C)NC(C2C=CCC2)=O)ccnc(Cl)c1 N1(C(CCC=CC)=O)CCCC(NC(=O)Cc2cc(C)no2)CC1 c1(C(N2CC3C(CNC(C(CC)C(C)C)=O)C3C2)=O)cc(C)c(C)c2ncsc12 Cc1c(C(=O)NCC2CCCN(C(=O)CN3C(=O)CNC3=O)C2)ncn1C N1(C(c2cn(CC)nc2C)=O)CC2(CC2)CC1C(=O)NC(C)(C)CC1CCC1 C1(C)(C(=O)NC(C2CC(NC(C3CCNC3=O)=O)C2)C)CC=CC1 N1(C(CCN(C)CCO)=O)CC2CC(N(C(=O)CCc3ncco3)C)C1C2 N1(C(C(C(C)C)SC)=O)CCC(C)N(C(C2CC23CC(O)C3)=O)CC1 Cc1cc([N+](=O)[O-])c(Cl)cc1NC(C1CC(F)CN1Cc1cncc(C)n1)=O C1(C(=O)NC2CC(NC(c3cn4cnnc4cn3)=O)C2)C2CCN(CC2)S1(=O)=O C(CCC(O)C(=O)NCC1(C(C)(F)F)CC1)NC(C1CC(C)C1)=O C12(NC(C(C)OCCN(C)C)=O)CCCC1N(C(=O)C=CC1CCCO1)CCC2 c1(C(=O)NC(CC2CCN(C(C=COCC)=O)CC2)C)nnc2n1CCCCC2 Cc1oc(C(=O)NC2C3CN(C(=O)C(C)(C)C)CC23)cc1CO c1(OCC(=O)NCC(CNC(Cc2nnc(C)o2)=O)O)ccc(CO)cc1.C(CF)O n1(C(CC)C)nnnc1C1C2(CCC2)N1.C(C)(C)(C)OCCSC C1(CNC(=O)Cn2nnc(=O)[nH]2)CN(C(=O)C2=COCC2)CC1C(F)(F)F O=C(CCCc1ccncc1)NC1CC(NC(C2CCOC2C(F)(F)F)=O)C1 C(=O)(C(CC(F)F)N(C(=O)C=Cc1cc[nH]c1)C)N(CCC(N)=O)CC C12(NC(C3CC(O)(CC#C)C3)=O)CCN(C(=O)CCC3CCCC3)CC1C2 C1(CCCCN(CCN(CC)CC)C)CN(C(=O)CCCCCO)CCC12CCC2 CC#CC1(C(N2CCC2(C)CC(=O)NCC(=O)NOC)=O)CCCC1 c1(C(N(C2CCN(C(C3CC(C)C3)=O)CC2)CC2CC2)=O)cnc2[nH]ncc2c1 CCC(CC)(CCNC(=O)CSC)Nc1csc(C(C)C)n1 Cc1ccc(C(=O)NC2CCCCN(C(c3ccn(CC#N)n3)=O)C2)cc1F c1(-n2ncc(CNC3CCCC(NC(CCC(C)C)=O)C3)c2)cc(Cl)ccc1F c1(C(=O)NCC2CN(CCN(C(C)=O)C)CC23CC3)cc(F)c(C)cc1Cl N1(C(C=C(CCC)C)=O)CCC(CN(C(=O)C(C)(C)c2cc[nH]n2)C)C1 c1(COCC)nc(-c2ccnnc2)n(C2CCCCC2C)n1 C(CCCCC(=O)N(C)CCc1cnn(C)c1)N(C(C1CCCC(C)C1)=O)C N1(C(C2C(CC(C)C)C2)=O)CCOCC1C(=O)NCc1cnn(CCO)c1 C1(F)(CNC(C(n2cc(Cl)cn2)C)=O)CCN(C(C2CCC(=O)N2C)=O)CC1 c1(N(C(C2CCCO2)(C)C)C(N(C)CCO)=O)ccccc1[N+](=O)[O-] c1(C(N2C3C(NC(c4ccc(COC)o4)=O)C(C3)C2)=O)cc2sccc2[nH]1 c1(C(=O)OC)cc(NC(c2[nH]cnc2CNC(C2(C3CCCO3)CC2)=O)=O)n(C)n1 C(=O)(C1CCc2nccn21)N1CCC(C(NOCC=C)=O)C12CCC2 N1(C(CC(c2cccs2)NC(C)=O)=O)CCN(C(C2(C)CC=CC2)=O)CCC1C C1(NC(C(CC)(F)F)=O)CCCN(C(C2(C)CC3CCC2C3)=O)CC1 CCC(C)(C)CCCC(=O)NCCCNC(C1CC2(C1)CC(C)(C)C2)=O c1(C(=O)NCC2CC(NC(c3ccc(CC)[nH]3)=O)C2)cc(OC)cc(Br)c1C CC1(NCC2CCN2C(=O)CCCCOc2ccc(Cl)c(F)c2)CCCNC1=O O=C(C(O)CC(F)(F)F)NCCC1(O)CN(C(c2cc(Cl)cs2)=O)C1 CC(CNC(C(=O)NCC(F)F)=O)CN1CCCC1.C12(CCC1)C(=O)N2C1CC1.CO C1(NC(c2c(C)[nH]nc2Cl)=O)CC1C1CCCN(C(c2cn(C)nc2C(F)F)=O)C1 C1(C(=O)NC23CC(NC(c4c(COC)cco4)=O)(C2)C3)CN2CCN1CC2C c1(CC(C)NC(=O)C(=O)N(C)Cc2cncs2)ccc(F)c(F)c1 C1(F)(CNC(C(C2CCC(=O)N2)C)=O)CCN(C(c2cc(C(N)=O)cn2C)=O)CC1 N1(C(c2c(CC)[nH]cc2)=O)CC(NC(C2CCC(F)(F)C2)=O)C(CC2CC2)C1 CC1CN(C(c2ccc(=O)n(C)n2)=O)CC1(C)CNC(c1ccc(Cl)cc1F)=O N1(C(C(C2CCCC2)OCC)=O)CCOCC1CNC(=O)CC1COC2CC1C2 C1(CNC(C2C(C(=O)OC)C2)=O)CC(C(=O)NCC(C)C#N)C1 N1(C(C2C(CCC(C)C)CCC2)=O)CCCC(C(=O)NCCOC(C)(C)C)C1 Cc1ncnc(C)c1CC(=O)NCC1CC1CNC(c1ncccc1F)=O N1(C(C(C)(Cl)Cl)=O)CC2CS(=O)(=O)CC2(NC(c2cnc[nH]2)=O)C1 c1(CNC(C(CC)NC(=O)CSC)=O)n[nH]c2c1CCC2 Cc1nc(NC(=O)C(O)Cc2cn(-c3ccsc3)nn2)sc1C(=O)N(C(C)(C)C)C N1(C(CCOCC#C)=O)CCCC1(C)CNC(=O)CNC(=O)OCC CC1CCN(C(C23CCCC2C3(F)F)=O)CCN1C(c1n[nH]c(C(C)(C)C)n1)=O c1(OC)nn(C)cc1C(=O)N(C)CCN(C(=O)C(O)C(C)c1ccc(C)cc1)C C1(OCCNC(C=CC(=O)N(C)C)=O)CCN(C(C2CC23CCC3)=O)CC1 C(CN1CC(C)OC(C)C1)(CN=C(NCC1(C2CCC2)CC1)NC(C)C)OC C1(CNC(C(=O)NCC(CC(C)C)NC(C(CC)SC)=O)=O)CC=C(C(C)C)CC1 C1(CC)CCN(C(=O)C(O)C(C)(C)C)C(C(=O)NCCNC(C)=O)C1 c1(NC2CC(NC(C(CC)C(C)O)=O)C2(C)C)cc2nnc(C)n2cn1 C(=O)(CC(C)C(=O)NCC1CCC(C)CN1C(c1ccc(C)cn1)=O)OC N1(C(c2c(C)ncs2)=O)CC(F)CC1C(=O)Nc1c(Br)cnn1C CCC(C(=O)N(C(C)C(=O)NCC(F)(F)CC1CC1)C)C(C)(C)CC N1(C(COCC(C)(C)C)=O)CC(CNC(c2cnc(N)c(CO)c2)=O)CC1(C)C N1(C(CCCNC(C)=O)=O)CC2(C1)CN(C(C1CC(Cl)(Cl)C1)=O)C2 n1(CC)cnc2[nH]c(=NCC(C)C(F)F)nc(N3CCC(CC(C)(C)C)C3)c12 c1(CC)ccc(C(=O)NC(C)(C)CCCNC(=O)C(N2CCNC2=O)C)c(Cl)c1 CC(N=S1(=O)CCCC1)c1cc(-c2ccc(N(C)C)cc2)ccn1 C1(C(=O)NCC2C3CC2N(C(=O)CN(C)C(C)=O)C3)(CC)CC(F)(F)C1 Cc1nnc(O)c(C(N2CC(NC(=O)C(C)(O)C3CCC3)CC3(CC3)C2)=O)c1C c1(C(N2C(CC)CN(C(=O)CC(C)(C)COC)CC2)=O)ccc2c(c1C)CCC2 c1(C(C(=O)N(CCCN(C(C(C2CCCC2)OC)=O)C)C)(C)O)ccc(Cl)cc1 N1(C(C(CC)NC(c2ccc(C#C)o2)=O)=O)CCC(C2=NOCC2)C1 C1(NC(C2CCN(C(N)=O)CC2)=O)COC2(C1)CN(C(=O)C(O)C1CCCC1)C2 C(=O)(C#CC1(C)COC1)N(C1CN(C(c2c(C(C)C)occ2)=O)CC1(C)C)C C1(C(C)C)CN(C(=O)CNC(c2cc(Br)ccc2Br)=O)CC(c2ccccc2)O1 c1(CC)cc(C(N2CCCCC(NC(C3(COC)C=CCC3)=O)C2)=O)c(C)nn1 c1(C(CC)C(=O)N(CCCNC(=O)C(C)Cc2ccco2)C)ccc(Br)cc1 C(=O)(C(C)(C)CS(C)(=O)=O)NC(CCN(C(C(C)NC(CC)=O)=O)C)C Cc1cccc(OC(C)C(=O)NCC(C)(C)NC(c2csc(C(N)=O)n2)=O)c1C C1(C(=O)NC2CCCN(C(C(C=CC)O)=O)C2C)CCOCC12CCCCC2 c1(C(NC(C23C(CN(C(=O)CN4CCOCC4)C2)C3)=O)CCl)ccccc1[N+](=O)[O-] Fc1ccc2c(c1)CCN(c1nc(Br)cs1)C2 c1(C(=O)NC(CC)CN(C)C(C2CC3(CCOC3)C2)=O)nccc2[nH]ccc12 Cc1cc(C2(C(=O)N(C)CC3CCCN(C(C4CC4(Cl)Cl)=O)C3)CC2)cc(C)c1 c1(OC)ncc(C(=O)NC2(CNC(=O)Cc3cn(C)nn3)CC2)cc1Br c1(OC)ccc(CNC(C23CC2CN(C(N2CCN(C)CC2)=O)C3)=O)cn1 CC(C)CCC(F)C(=O)NCCO.C1C(C)(C)OCC(=O)N1CC(C)(C)C CCC(C)(C)C(O)C(=O)N1CC(CCNC(=O)Cc2ccccc2)C1 N1(C(c2n[nH]c(C)c2F)=O)CCC(CNC(=O)CN2CCS(=O)CC2)C12CCC2 C(CC)(CCCO)NC(CN(C(=O)CCCN(C)C)CCOC)=O C(=O)(CC=CC(=O)OCC)N(CC(=O)NCC)C.C12CC(C1)C(=O)NCC2 c1(C(N2CCCC(C)(CNC(c3cn(C)nc3O)=O)C2)=O)nc2ccccc2[nH]1 C1(O)(NC(N2CC(F)(F)C2)=O)CCN(C(=O)COc2ccccc2)CC1 C(C1CN(C(C2CC23CCC3)=O)CC1C(=O)NC1CCN(CC)CC1)=CC C1(NC(C=C(CC)C)=O)CCC(NC(=O)C(c2cncc(F)c2)(C)C)CC1 CCCC(C(=O)N1CCC(C(=O)NC(c2cc(C)on2)C)(CC)C1)NC(N)=O C#CCC(C(=O)OC)NC(=O)C(C1CC1)NC(=O)CC1CC1(C)C C1(C(=O)NCC(CC)C)CCCN(CC2CC(O)CN2)C1 C1(NC(C=C(C)C(C)C)=O)CC(CO)N(C(=O)C(C)Oc2cccc(Cl)c2)C1 C1(C(=O)NC(C2CN(C(c3ccc(N)c(Cl)c3)=O)CCO2)C)CN2CCN1CC2 c1(N(CCN(C(c2c(OC)ccnc2)=O)C)C)ncnc2sc(C)nc12 c1(C(=O)NCC(CNC(C(C)C2CCC2)=O)F)nc[nH]c2ncc(Br)c1-2 C(C(N=c1[nH]ccn2c(C(C)C)nnc12)C(C)C)NC(C1CC(C)(CC)C1)=O N1(C(C(CCC)n2cc(-c3cccc(Cl)c3F)nn2)=O)CCOCC1(C)CC c1(C(N(CC(CC)NC(=O)CC2CCCO2)C)=O)coc(CC2CC2)n1 c1(SCC(=O)NCCN(C)C(c2cn(C3CCCCC3)nn2)=O)n[nH]c(=N)s1 Cc1cc(=O)n(CCC(N2CCCC(CCCCNC(=O)CCCF)C2)=O)cn1 C1(NC(=O)CC2CCCCO2)CCC2CC1CN2C(c1ccon1)=O c1(C(N2CC(CC=C)(NC(=O)C(C)C(O)C(C)C)C2)=O)cc2c(nc1O)CCC2 C1(C(N2CC(CNC(COC)=O)(OC)C2)=O)CCCCCCC1 N1(C(C(C)OC2CCCC2)=O)CCC2(CN(C(c3ccncc3Cl)C)C2)C1 N1(C(c2c(CC)noc2)=O)CCCC(CNC(C2(CO)CCCC2)=O)CC1 N1(C(c2cc(C)oc2C)=O)CC2CCOC2(CNC(C2CCN(C)S2(=O)=O)=O)C1 C1(NC(c2noc(C(F)(F)F)n2)=O)CC2CN(C(C3CC34CCOCC4)=O)CC12 C(=O)(C(CC)CC)OCCCC.c12ccccc1CC(=O)OC1CCN(C1)C2=O CC1CN(C(c2cnc(S)nc2)=O)CC(C)N(C(c2ccc(Cl)c(F)c2N)=O)C1 N1(C(C(C)SC)=O)CCCCC1CCCOCCNC(C1(C)CC1)=O c1(NC(=O)CC2CN(C(c3cccnc3Cl)=O)C2)cc(Cl)ncc1Br CC(CC(=O)NC1(CC(N2CCC(CCO)C2)=O)CCCCC1)C(F)F C1(NC(c2c(C)ccn2C)=O)COC2C(NC(C3NC(=O)C4CC34)=O)COC12 Cc1ccc(CNC(=O)C(C)NC(=O)CN2CC3CC3C2)c(O)c1 N1(CCNC(=O)C=Cc2nccs2)CCCN(C(C2CCC2c2nc[nH]n2)=O)CC1 c1(C(=O)NCC2C(NC(c3c(C(=O)OC)ccs3)=O)CCC2)ccnc(F)c1Cl c1(C(=O)NCC2CCN(C(c3n[nH]cc3Cl)=O)C2)cn2cccc(Br)c2n1 Cc1cnc2n1CC(C(=O)N(CC(C)CNC(=O)C=Cc1cn(C)nn1)C)CC2 C1(C(=O)NC23CC(CNC(c4n(CCC)ccc4)=O)(C2)C3)CCC(C)(F)CC1 C(=O)(C1CCOc2c(F)cccc21)N1C2CN(C(COC(C)(C)C)=O)CC1CCC2 c1(NC(c2ccc(OC)cc2OC)=O)cc(P(C)(C)=O)ncn1 N1(C(CC2N(C(C)C)CCC2)=O)CCCC(C(N2CCCCC2)=O)C1 C1(CN(S(C)(=O)=O)C)COCCN1C(C1C2CCC1NC2)=O C(=O)(C1=NNC(=O)C1)NCCN(C(c1nc(C)c(C)s1)=O)CC C1(C(=O)NCc2c(C(=O)NCc3c(C)nccc3)nco2)CC(C)(C)CN1C Fc1cccc(OCc2cccc(Br)c2Cl)c1Br c1(-n2c(-c3c(C)cco3)nnc2N(C2CN3CCC2CC3)C)cc2n(n1)CCCC2 N1(C(CC2CCCC(C)(C)O2)=O)CCC2CCC(NC(C3(F)CCCCC3)=O)C12 CC(Cc1ccc(F)cc1)(C(=O)O)NC(c1cc(C(F)F)no1)=O c1(OC)cc(C(=O)NCC2CN(C(=O)C(=Cc3cccs3)C)CC2C)ccc1O c1(CC(=O)NCC(C2CCOC2)NC(=O)Cc2cnc[nH]2)ccc2c(c1)OCO2 C1(C(CNC(CC(C)F)=O)C)CCN(C(C2(n3ccnc3)CCCC2)=O)CC1 C(=O)(CC(C)C(F)(F)F)NC1CC(CC(=O)NC(COC)(C)C)C1(C)C C=CCC(C)(C)CC=O.C1CCN(C(=O)C(C)C)CC(O)C1 N1(CC(=O)NC(CNC(C(C(C)C)N(C)C)=O)C(C)C)CCc2sccc2C1 c1(OCC)ncccc1CC(=O)NCC1(F)CC(NC(=O)C=C2CCC2)C1 C1(C(N2CCCCC2)=O)(CC)CN(C(CNC(C(C)OCCSCC)=O)=O)C1 N1(C(CCSCCCC)=O)CC(C(=O)NC(=O)C(CCC)OC)CC1(C)C N1(C(c2c(Oc3c(NC)cc(C)cc3)cccc2)=O)CCC2(C(=O)O)CCCC12 S(=O)(=O)(c1csc(NC(=O)OC)n1)N(c1ccccc1)CC(CC)O c1(C(=O)NC23CC(NC(C4C(OC)CCC4)=O)(C2)C3)c(C)ncnc1C N1(C(c2c(NC)nccc2)=O)CC(CCNC(C2(CF)CC2)=O)OC(C)C1 N1(C(C(CC#CC)NC(C23CSCC2C3)=O)=O)CC2(CCC(=O)N2)C1 c1(C2(C(=O)Nc3n(COC)ncc3)CC2)ccc(OC)c(OC)c1 c1(C(=O)NC2CC3CC2CN3C(C2CC2F)=O)csc2c1CCCC2 C1(NC(C2(NC(c3cc(Cl)cn3C)=O)C(C)C2)=O)CCCN2CCCC12 C1(OC)CCCCC1C(=O)NC(C)CNC(C)=O CN1CCCC1(C)C(N1CC(NC(c2ncnn2C2CCOCC2)=O)C1)=O C1(C(=O)NC(C2(O)CN(C(=O)CCC3CCCC(=O)N3)C2)C)CC(F)C(=O)N1 C=CC(C(F)(F)F)NC(C1C(NC(=O)C(C)NC(=O)C2CC2)C1(C)C)=O c1(NC2CC(C)N(C(c3cnc(Cl)s3)=O)C2)ncc(C#N)cc1Br C1(NC(CNC(CCNC(C)=O)=O)=O)CC2CC(NC(c3cccnc3)=O)C1C2 C(=O)(C1CCCc2n[nH]cc21)N1C(C)(CNC(CCOCC(C)C)=O)CCC1 n1(CCC)nnnc1C(CC)(C1CC1)NC(C1CCOC1)NC(C)=O.OC C(=O)(C1COc2ccc(Br)cc21)NC(CCCNC(CSCC=C)=O)(C)C CC12COC(C(N3CCC(N4CCN(C(C5(F)CCOC5)=O)CC4)C3)=O)(C1)C2 C12(C(=O)NC3CC(n4cc(C(CC)O)nn4)C3)CCCC(CC1C(=O)OC)C2 N1(CC(=O)NC(CNC(C=CC=CC)=O)C)C(C)=CC(C)=NS1(=O)=O Cn1c(O)nc2cccc(C(N3CC(CCNC(C4CCCC(O)C4)=O)C3)=O)c12 C(=O)(C1=CCCCC1)N1CC(C=C)(C(N(C2CN(CCOC)C2)C)=O)C1 N1(C(c2c(CC)onc2)C(=O)NC(C)C(=O)OC)CCC(F)(CO)C1 CC1(C(N2CCCC(CNC(=O)Cc3ccc(F)cc3)CC2)=O)CCNC(=O)C1 Cc1cc(C#N)ccc1C(=O)N(C1(C(=O)N(CC(O)CO)CC)CCC(C)C1)C1CC1 C1(N(C(CCC2(NC(C=NOC)=O)CCC2)=O)C)CC2CCC1CC2 C(=O)(C#CC1CCCCC1)NC1C(C)N(C(=O)CC2=CCCCC2)CCC1 C(=O)(C(F)CCC(C)C)NC1CN(C(Cc2nc(C)oc2)=O)CC(O)C1 N1(C(COC)=O)CCCCC1C(=O)NCC(C)(C)CO CCCCC(O)C(C)C(=O)C(CC(C)N(C(=O)C(O)CCC)COC)N N1(CC(=O)NCC(C)(C2CC2)NC(c2cnco2)=O)CCNC(=O)C1 c1(C(C)NS(C)(=O)=O)ccc(C(=O)Nc2cc(-c3ccc(O)nc3)cs2)cc1 C1(OC)CC(NC(C2CC2(F)Cl)=O)CN(C(c2ccc(CS(C)(=O)=O)o2)=O)C1 c1(N2CC(C)C(NC(C3(C(F)F)CCOCC3)=O)C2)c(Cl)cncc1[N+](=O)[O-] n1(C(C)C)cnnc1CC(N1CC(CCNC(c2cc(C(C)(C)C)n[nH]2)=O)C1)=O n1(CCC)cc(C(=O)N(CC(C)NC(C2CCCC2O)=O)CC)nn1 N1(C(c2n(CC)ccc2)=O)CCN(C(c2cnoc2-c2ccc(C)o2)=O)C(C)C1 Cc1nc(C(N2CCC(CNC3CCCC3N3CCCCC3)C2)=O)co1 C(CC1=CCC2CC1C2(C)C)OC(c1c(C(C)C)n(-c2cccc(Cl)c2)nn1)=O Cc1nc(Cl)ccc1C(N1CCCC(n2cc(CN3CCOCC3)nn2)CC1)=O C1(C2CN(C(=O)CC3CCCC(C)(C)C3)C2)(NC(=O)NC(C)C(=O)OC)CC1 c1(CC2CN(C(C)(C)C)C2=O)c[nH]c2cc(F)ccc12.Cn1cncc1CCN c1(C(N2CCC(O)(CNC(=O)CCn3ccnn3)C2)=O)cnc2ncccc2c1 C(=O)(C(CO)C(C)(C)C)NCc1c(CCNC(C(C(C)C)OC(C)=O)=O)ocn1 N1(C(CC2CCC(NC(=O)CCC3CCCCO3)CC2)=O)CC(N(C)C)C2(CC2)C1 C1(N(C)C)(CNC(c2nncn2C)=O)CCOCC1.C1=CCNC1=O c1(C(N(CC(C)(C)NC(C2C(CC)OCC2)=O)C)=O)nc(C)n(C)c1C N1(C(CC)=O)CCC2(C1)CN(C(=O)C(C)NCS(=O)(=O)Cc1ccccc1)C2 N1(C(C2CC(C)(NC(CC3CCCN(C)C3)=O)C2)=O)CCN2CC(O)CC2C1 c1(C(C(=O)NCC(Cn2cc(CCNC(C)=O)nn2)(C)C)C2CC2)ccc(Cl)cc1 c1(C(N2C(CNC(C3CC4(CCC4O)C3)=O)CC2)=O)cnc2ccccn12 C12(C(=O)NCCNC(CCc3c(C(=O)OCC)cccc3)=O)CCCC1C2(F)F C(c1cccnc1)=CC(N1C(CNC(C2(CCOC)CC2)=O)CC1)=O CC(F)CC(=O)N1CCC(CCNC(=O)CCCF)C1 c1(OC)ccc(S(=O)(=O)N2C3CC2CN(Cc2ccc(F)cc2O)C3)cc1OC C(=O)(C(O)C(CCC)NC(c1cc(C(F)F)[nH]n1)=O)N1CCC(F)(CCC)C1 c1(CC)ncc(C(=O)NCC2CC(NC(c3nnsc3C)=O)C(O)C2)cn1 Cc1nc([N+](=O)[O-])cn1CC(N1CCN(C(=O)C(C)C(C)C)C2CC12)=O C#Cc1ccc(C(N2CCC(CC(N)=O)(NC(C3CC3COC)=O)CC2)=O)cc1 C1(N(C)C(C2(C3CCCO3)CCC2)=O)CC2CCC(C1)N2C(C1CCSC1)=O N1(C(COCCCOC)=O)CC2CC1C2CNC(C1CCOC1C)=O C(=O)(C1=NOC2(CCOC2)C1)NCC(N(C(CCC=C)=O)C)C1CC1 C1(C(=O)NOCC(F)F)(CNC(=O)CCNC(c2ncc[nH]2)=O)CC(F)(F)C1 C12(C(N(CCC)CCNC(C34COCC3C4)=O)=O)CCCC1(C(N)=O)C2 CC1(C)CCC(C(=O)NCC2OCCC2(C)C)(NC(C23C(=O)C4CC2C3C4)=O)C1 c1(C(=O)NCC(CNC(C2C(COC)C2)=O)OC)cc(C)nn1C1CCOCC1 C1(SC)CCC(C)N(C2CCN(c3cc(C)nn3C)C2=O)C1.c12cnnc(c1)C2 Cc1cccn(CC(=O)NCC2CC(C)CCN2C(C2CCCC23CCC3)=O)c1=O CC1CN(C(=O)NCCc2cnco2)CC(C)(C(F)F)O1 C1(CN(C(=O)CC2C(NC(C3CCS(=O)CC3)=O)CC2O)C)CCC(C)(C)C1 C(=O)(CCCC(=O)N(CCCC(=O)NC1CCCC1C(N)=O)C)OC c1(OC)ccc(C2CC2)c(C(=O)NCCC(C(C)C)NC(=O)C2=C(Cl)CCC2)c1 c1(C(N(CCNC(=O)C(C)CCOc2ccccc2)CC)=O)cc2n(n1)CCO2 Cc1ccc2oc(N3CCCCC3CNC(C3C4C5CCC(C5)C34)=O)nc2c1 N1(C(c2c(C)cc(C3CC3)cc2)=O)CC2CCC1CC2NC(C1CC1(C)C)=O c1(C(=O)NCC(CC)NC(=O)CCCc2nccs2)cnc(C)[nH]c1=N C1(CNC(c2c(OC)n(C)nc2)=O)CCC(C)N(C(C2OCCN(C)C2=O)=O)C1 C1(C(N2CCC(NC(c3ccc(=O)oc3)=O)(CF)C2)=O)Cc2cc(F)ccc2O1 CCCC(C(=O)NCC(O)CC(=O)NC(CC)(CC)CC)OCC C1(C(=O)NCC2C(C)CCN(C(c3c(C)onc3Cl)=O)C2)CC2(C1)CC1(CC1)C2 C1(CNC(c2c[nH]c(=N)o2)=O)CCCC(NC(=O)C(c2ccccc2)O)C1 C1(OC)CC(NC(=O)C(C)C)CN(C(C2CCCCN2C(C)=O)=O)C1 c1(OC)ccc(OC)c(C(N2CCCC(C(C)NC(=O)C(F)=C(C)C)C2)=O)c1 c1(NC(C)=O)ccc(CC(=O)NC(C)CNC(c2c(C)ncn2C)=O)cc1 N1(C(C(CC)n2cncn2)=O)CCC(C(=O)NCc2ccc(Cl)nc2)C(C)(C)C1 N1(C(C(C)Cc2ccccc2)=O)CCN(C(c2cncc(O)c2)=O)CC(C)(F)C1 c1(C(=O)NC(C)(C)C2CCC2)c[nH]nc1CCNC(=O)CCc1ccsc1 C1(C(N2CC3C(CC)(C3)C2)=O)CC2CCCC2N1C(=O)C=NOC c1(C(C(=O)NCC(=C)C)N(c2ccccc2)CCN(C)C)nn(CC)nc1C C1(CC)CN(C(C23CC(CCO2)C3)=O)CCN1C(=O)Cn1nc(C)cc1C C=CCC(CNC(=O)CNC(=O)C(C)(C)C)NC(C1(c2ccccn2)CC1)=O CCCCC(F)C(=O)N1CCC(C)(NC(C2CCCN2C=O)=O)CC1 C12CN(CCN1C)C2=O.C1(C(C)C)CCCC(NC(C2CCC3(CC3)C2)=O)C1 N#CC1CCCC(C(N2CCCN(C(c3ccc(C4CC4)s3)=O)CC2)=O)C1 C1(CC(=O)NCC2(COC)CN(C(=O)CN3CC(C)(OC)C3)C2)CCCCN1C c1(C(=O)NC23CC2CN(C(C2CCCC(F)(F)C2)=O)C3)ccc2c(O)n[nH]c2c1 N1(C(C(CC)CC)=O)CCCC(NC(c2csc(C(N)=O)n2)=O)C1C c1(CNC(c2ncn(C)c2)=O)ccc2ncccc2c1.C12CN(C1)C2=O C12(C(N(CCOCCCOC)C3CC3)=O)COCC1CN(C(=O)CC1CCC1)C2 CC1(CNC(=O)CCOCC(F)F)CC(NC(C2(O)CCC2)=O)C1 c1(C(=O)Nc2cccc3nc(C)[nH]c32)cc(C)cc2c1NCCC2C N1(CC(=O)NCC2CC(C)(CNC(=O)C(F)n3ccnc3)C2)CC2CCC1C2 c1(COC)nn(C)c(Cl)c1C(=O)NCC1COCCN1C(c1ccsc1C)=O c1(CC)cccc(C(n2cnnc2CN2CCN(CC3CCOCC3)CC2)C)c1 C1(C)CC(C)CN(C(C2(CF)CC2)=O)C1.Cc1cc(COCC(=O)N)on1 S(=O)(=O)(c1ccc(NC(C)C(C2CCCCC2)O)cc1Cl)NCC(C(C)C)(C)C Cc1cc(C(=O)NC(CNC(=O)C=CSc2nc[nH]n2)C(C)C)co1 Cc1cc(C2CC2C(=O)N(CCC(C)NC(c2cn[nH]c2)=O)C)on1 c1(C(=O)NCC2(NC(c3[nH]c(=NC)sc3)=O)CCC2)c(C)nc2cccnn12 C=C1CCC(C(=O)NCc2nocc2C(=O)NC(C)(CO)CCF)CC1 N1(C(C(CSC)O)=O)CCCC(O)(CNC(c2cnc(CO)nc2C)=O)C1 N1(C(Cc2ccc(OCC)cc2)=O)CCCC(NC(=O)C(F)C2CCCC2)C1C C12(CNC(CSCC)=O)CC1CN(C(=O)CN(c1ccncc1)C)C2 C(CCC(C)C(=O)N1CCCC(NC(c2nonc2N)=O)C1)OC C1(C(=O)NC(CC=C)CC)(CC)CCN(C(C2CCCCC2O)=O)CC1 c1(C(N2CCC(O)(CNC(CC3(C)CCC3)=O)C2)=O)ccc2c(=O)ccoc2c1 c1(OC)noc(-c2nc(C3CCCC3)nn2-c2ccoc2)c1Br C1(CNC(C2CCCS2)=O)CC2CCC1N2C(c1cc(Cn2cccn2)on1)=O C1(C(=O)NC2CC(NC(=O)CCCn3cccn3)C2)(OC)CCOC1 c1(NCc2cccc(F)c2)cccc2nonc12.C12CCCN(C1)C(=O)N2C N1(C=O)CCCC1(C(=O)NOCC(F)(F)F)CC.CCCC(C)OCC N1(C(C2CCN(C(C=CC3(C)COC3)=O)C(C)(C)C2)=O)CCCC12CCNC2=O C1(CC(N2CC(C)C(NC(c3cnn(C4CCC4)c3)=O)C2)=O)CCCCC1(F)F c1(C(N(CC(CC)NC(=O)C(c2cnn(C)c2)OC)C)=O)[nH]c(C)nc1C N1(Cc2c(C)nc(-c3ccc(OC)cc3)s2)C(=O)CCN(CC2C3CCC23)C1=O c1(C(=O)NC(CC2CCOC2)C(=O)O)ccc(C(F)(F)F)c(Cl)c1Cl C1(C(N2CC(CN(CC(C)C)CC)C2)=O)C2CC(O)C(C2)N1C(=O)CSC c1(C(N2C(C(=O)NCc3ccc(O)cc3)CC3CC32)=O)cc(O)ccc1Cl c1(C(N2C(CNC(C3CC(OCC)C3)=O)CC3CC32)=O)ccc2cncn2c1 C(=O)(CC(C(F)F)N(C)C1CC1)N1CCC(NC(=O)CC(C2(C)CC(=C)C2)=O)C1 C1(C(N2CCC(F)(C(N3CCC(c4nn[nH]n4)C3)=O)C2)=O)CCCC2(CC2)C1 C1(CNC(Cc2cn(CC)nc2)=O)CCCCN(C(c2nnc(C)s2)=O)C1 C1(C(=O)NC2(c3cccc(C)c3)CC2)CN(C(c2cscc2F)=O)CC1(F)F c1(C(=O)NCCN(C(=O)C(O)C2CCC2)CC)n[nH]c2ccc(C(F)(F)F)cc12 C(=O)(CC(O)CC(C)(C)C)N1CCCCC(N(C(C(=O)NCC)=O)C)C1 N1(C(c2[nH]nc(OC)c2Cl)=O)CCC2CCN(C(=O)C(c3ccc(C)o3)C)C2C1 c1(C(=O)NC2CCC(N(C(c3nccc(C)n3)=O)C)C2)cc(C(C)C)nc(O)c1 c1(CN(C(C(N2CCCC(N(CCOC)C)C2)=O)=O)C)ccc(C#N)cc1 c1(CNC(C(C)OCCCC)=O)nc2c(s1)CN(C(c1[nH]c(O)nc1C)=O)CC2 C#CCC(C)(C)C(=O)NCC(CC=C)C(=O)N1CCC(n2cncn2)C1 CC1Cc2n[nH]cc2CN(C(=O)C(=O)N(C)C)C1.c1(CC)ccc2c(c1)CCCC2 c1(C(=O)NC2CCCN(C(c3c(CC)oc(C)c3)=O)C2)ccc2ccccc2n1 N1(C(CC2C(C)(C)C2(C)C)=O)CCCC2CN(C(=O)C#CC3CCC3)CCC12 C1(CNC(=O)COC(F)(F)F)CCN(C(C2(CO)CCCC2)=O)C12CCC2 CC(C)CC(C(=O)NCC1CNC(=O)CO1)NC(c1cccc(=O)o1)=O c12ccc(cc1Cl)s2.c1(C(C(C)(C)NC(C(=O)OC)=O)=O)ccc(O)cc1 c1(C(=O)NCC(CN(C(C(CC)(F)F)=O)C)O)cccc(F)c1C CN1CCC(c2ncc(C(=O)NC3CCC(NC(c4ccc[nH]4)=O)C3)[nH]2)CC1 C(=O)(CCC(=O)NC(CO)C(=O)NC(C1CCCC1O)C)NCCC Cc1cc(C(=O)NCC(O)CC(=O)NC(C)(C)C(O)CO)cnn1 N1(C(C2(C)CCC(F)(F)C2)=O)CC2(CCCN(C(c3ncccc3Cl)=O)C2)C1 C1(NC(c2ccsc2)=O)CC12CCN(C(c1ccc(Cl)c(F)c1F)=O)CC2 C1(NC(COCCCC#C)=O)CCN(C(=O)Cn2ccnn2)C2CC12 C1(NC(CCc2c(OC)cccc2)=O)CC(F)CN(C(=O)CCC2CC2(F)F)C1 C(=O)(C1=C(C)CCC1)NCCCC(C)(C)NC(c1c(COC)cccc1)=O C(=O)(C(CCC(N)=O)n1cc(CCNNS(N)(=O)=O)nn1)N(CCO)CC c1(C2CC2)cc2c(Cl)nccc2o1.C1(NC(C(C)SCC)=O)CNCC2(CC2)C1 C1(S(C)(=O)=O)(C(=O)NCCN(C(=O)CC2CCCS2(=O)=O)C)CCC1 c1(OC)cc(N)c(Cl)cc1C(=O)NCC(C)(CC(C)C)NC(=O)C=CS(C)=O CC(C)C(C(=O)NC12CC1CN(C(=O)CCCCC1CC1)C2)c1ccccc1 C1(Nc2ccc(Oc3c(C)ccc(OC)c3)cc2)CCCCC1C1CC(F)(F)C1 c1(C(=O)NC2(CCO)CN(C(C3(COC)CC3)=O)C2)ccnc(-n2cncn2)c1 CC1CN(C(c2cnc(O)o2)=O)CC(CCNC(C23CC(F)(C2)C3)=O)O1 CC1(C)CC(NC(=O)CCC2CCC(=O)N2)CN(C(C2(C(F)(F)F)COC2)=O)C1 Cc1cnc(C(N2CC3C(CNC(c4c(Br)ncn4C)=O)C3C2)=O)c(C)c1 N1(C(CCC=C)=O)CC(C(F)(F)F)OCC1CNC(=O)Cc1cccc(O)c1 C1(C(=O)NC(COC)(C)C)CN(Cc2cc(Br)cc(Cl)c2F)CCC1(F)F C(=O)(C1CCC(=O)c2ccccc21)N1CCC(NC(c2cc3n(n2)CCC3)=O)C1 N1(c2c(C#C)cc(F)cn2)CC2CCCC(C1)N2CC(=O)NC [N-]=[N+]=NC1(C(=O)NC23CCN(CC2)CC3)CCN(C(c2coc(C3CC3)n2)=O)C1 N1(C(C=CCCC(C)NC(C2COCC(C)O2)=O)=O)CCc2ccsc2C1 N1(C(c2cnn(C)c2F)C(=O)NC)CC(C)OC(C)(C)C1.c12ccccc1n(C)s2 C1(C(=O)NCCc2cc[nH]n2)CCCC(NC(C2COCCO2)=O)CC1 N1(C(C(C)NC(CC)=O)=O)CCCC(NC(N(CC(C)NC)C)=O)C1 N1(C(Cc2nnc(C)s2)=O)CC(F)(F)CC1CNC(=O)CCC1CCOC1 c1(C(N(C)CC2CCN(C(c3c(C)scc3)=O)C2)=O)ccnnc1NC1CC1 c1(NC(C2CC3CC3N2C(c2sc(Br)cc2Br)=O)=O)cc(Cl)cc(Cl)c1F c1(CC(=O)NCC2N(C(c3cccc(OCC)c3)=O)CC2)ccc(C)c(F)c1 CCC1(C)CC(=O)N1.C1(C(=O)OC)CC(=O)N(C)C1c1ccc(OC)cc1 CC(N=c1ccnc(C2CC2)[nH]1)C1CCN(C(c2ccc3c(c2)CC3)=O)C1 N1(C(c2cc(C)sn2)C(=O)Nc2ccsc2)CCCc2c(CC3CCC3)cccc21 C1(NC(=O)Cn2ccnn2)CCN(C(=O)C2=CCCC2)C12CCCC2 c1(CC(C(N2CC(NC(C(C)NC(N)=O)=O)C(F)C2)=O)C)cccc([N+](=O)[O-])c1 C1(C2CCN(C(c3nccc(OC)c3OC)=O)CC2)(NC(C(CC)O)=O)CCC1 C(=O)(CC(C(F)(F)F)NC(c1cc(Cl)n(C)n1)=O)NCC1(CC)CC1 C1(OC)CCC2CN(C(=O)CCCCNC(=O)CC3C(=O)NN=C3C)CC12 c1(C(=O)NC(CNC(c2ncn(C(C)C)n2)=O)C)ccccc1F c1(C(N(C)C)C)ccc(C(=O)Nc2ccccc2COC(C)(C)C)cc1 C1(CC#C)(C(=O)NC(CNC(C2CCCN2S(C)(=O)=O)=O)C(C)C)CCCO1 c1(CCC(N2C(C)CC(CNC(C3CC(O)C3)=O)C2)=O)cc(Cl)cc(Cl)c1 Cc1c(C(=O)NCC2C(C)CCN2C(=O)CC2CC3(CC3)C2)ccn1C(C)C C(=O)(C(O)CC[S+](C)C)N(C)CC1CCN(C(C2(CCC=C)CC2)=O)CC1 C(=O)(CC(C)C(C)C)NCCC1(NC(COCCCC#C)=O)CC1 C1(OC)CC(NC2(C)CCN(C(=O)OC(C)(C)C)C2)C12CCCO2 C1(CCOC)(C(=O)NCCCCOC)CCN(C(C2CC3CC3C(=O)N2)=O)CC1 C1(CNC(c2cnc(NC(C)=O)s2)=O)CN(C(=O)C2=NOC(C)C2)CC12CCC2 c1(-c2ccc(CN3C(C)(COC)CCC3)s2)cc(C(F)(F)F)ncc1F Nc1ccc(CCC(=O)NCC2(NC(=O)CNC(=O)CC3CCCC3)CC2)cc1 C1(CCNC(C)=O)CSCCN1C(=O)CC1CCCOC1.c12cn(nn1)C2 CCC(C)(CC)C(N)=O.C12(NCc3nnn(C)n3)COCC1Cn1c2nnn1 C=CCC(CC)C(=O)NCCCOCCN(C(=O)C(c1cc(C)cc(C)c1)O)C C1(N(C)Cc2nccc(C)n2)CC(=O)N(c2cnn(C)c2)C1=O.c1cnn(CC)c1 c1(SC)cccc(CNC(c2nnnn2C2CC2)c2ccno2)c1 CC(C(=O)N(CCCNC(C1(N(C)C)CCCSC1)=O)C)C(=O)N1CCCCC1 C1(CC(C)C)CNC(=O)N1.C12(CC(=O)OC)COC(C(C)N(C)C)(C1)C2 C(=O)(CCC(=O)c1ccncc1)N(CC(O)CNC(c1ccnn1CCF)=O)C N1(C(=O)OC(C)(C)C)CCC(CN(CC(C)(C)C2CCCC2)C2CC2)C12CCC2 c1(C(N2CCC(O)(C(C)NC(C(C)N(CC)CC)=O)C2)=O)ccn2nccc2c1 N1(C(C(CC)N(C)C)=O)CCCC2(C1)CN(C(c1cccc3nnn(C)c13)=O)C2 c1(OC)ncnc(C(N2CCC(NC(C3(C#N)CCCC3)=O)C(CO)C2)=O)c1F C1(OCCOCC(=O)NC2CCC2)CC12CCN(C(c1cnc(S)[nH]1)=O)CC2 C(=O)(C(F)CC(C)(C)C)NC1(COC)CCN(C(=O)Cc2ccc(C)s2)C1 C(=O)(C(C)(C)C1=CCN(C(c2ccsn2)=O)C1)NCC(C)Cc1cn[nH]c1 c1(CC(C)C)ccc(C(C(C)C)NCc2sc(-c3ccccc3F)nc2C)cc1 Cc1n[nH]c(=NCC(CNC(c2ccc(F)nc2)=O)C(F)(F)F)o1 N(C(=NCc1cc(C(F)(F)F)cs1)NCc1nnc(SC)s1)C(CC)CC C1(CNC(c2sc(CC)c(C)c2)=O)CC(C)(C)CN1C(C1CCCC(C)(C)C1)=O Cc1cc(NC(C2CC(F)CN(C(=O)Cc3cnc(C)s3)C2)=O)cc(Br)c1 CC(CC(=O)NCC(c1ccccc1F)NC(=O)C#CC1CCC1)C(C)(C)C C1(C(N2CC(N3CCNC3=O)C2)=O)CCC(C2CC2)N1C(C1CC(OC2CC2)C1)=O CC1(C)C2COC1(C(=O)NCCCCC1CCN(C(C3(O)CCC3)=O)CC1)C2 C1(NC(=O)Nc2cccc(O)c2)CCCN(C(c2cnccn2)=O)C1 N1(C(c2n(CCC)nc(C)c2)=O)CCOCC(CNC(c2cnsc2)=O)C1 Cc1cnc(C(=O)NC2C3CC2CN(C(=O)CCc2nc(=N)[nH][nH]2)C3)cc1C c1(C(N2CCN(C(c3ccc(OC)[nH]3)=O)CC2C(C)C)=O)csc(S(N)(=O)=O)c1 Cc1nnc2n1CC(C(=O)NCC13CC1CN(C(C1CCC(F)(F)C1)=O)C3)C2 c1(C(=O)OC)cc(NC(=O)NCC2(C)CCCCO2)cc(O)c1 N1(C(CCC#C)=O)CCC2(CC2C(=O)NC(CN(C)C)C(C)(C)C)C1 C(=O)(C(O)C1=CCCCC1)NC1CC(C(ONC(=O)CCc2cccnc2)C)C1 O=S1(=O)C=C(c2ccccc2F)CCC1Nc1ncccc1F C1(C(C)(C)O)CCCCN1C(C1(NC(=O)CC2(O)CCCCC2)CCC1)=O C=CCC(C(=O)NCc1cc[nH]c1C(=O)NCC(C)CCC)C(C)C C1(NC(Cc2nc(C)sc2)=O)C2CC(NC(=O)C(C)(C)C3CCCO3)CC12 n1(CCC)ccc(C(=O)NCC(C)(O)CNC(c2ccc(CCC)[nH]2)=O)n1 N1(C(C(C(C)(C)C)CNC(C2(Cl)CC2(F)F)=O)=O)CCN2C(=O)OCC2C1 c1(C(=O)NCC2(C)CCCN(C(C(C)=O)=O)C2)ccc2oc(C)nc2c1 N1(C(CC2C(CC)C2)=O)CCOCC(NC(=O)CNC(CCC)c2cccs2)C1 CC1(C)CN(C(=O)C2=COCC2)CC1CNC(=O)C=Cc1cnccn1 S(=O)(=O)(c1ccc(NCCCF)c2cnccc12)NC(C1C(CC)OCCC1)=O CC1CCC(NC(=O)NC(N)=O)N(C(c2cccc(NC(N)=O)c2)=O)C1 c1(C(N2CCC(NC(c3nc(C)oc3)=O)C2)=O)cnc2ccoc2c1 Cc1ccc(C(=O)NCCC23CCC2CN(C(c2cnc(S)[nH]2)=O)C3)c(C(C)C)n1 C(=O)(C(C)(CCC)CCC)N1CCC(OCC(=O)NC(CC#C)CO)C1 N1(Cc2cccc(OCOC)c2)CC2CN(C(c3cccc(I)c3F)=O)CC12 Cc1cnc(N(CC(C)CNC(c2ccc[nH]2)=O)C)nc1S(C)(=O)=O Cn1ccc(C=CC(N2C(C(=O)NC(C)(C)CNC(N)=O)CCC2C2CC2)=O)c1 c1(C(N(CC(CC)NC(=O)CC2CCCOC2)C)=O)ccc2cnccc2c1 C1(C(=O)NCCCCCN(C(c2cc(OC)no2)=O)C)CNC(=O)C(C)(C)C1 c1(NC)ncc(C(=O)NCC2CCN(C(C3CCC3C)=O)C2)cn1 C1(CC(C)O)COCCN1C(=O)Nc1ccncc1F c1(COCC(c2ccccc2)C)nc(-c2nc[nH]n2)no1.N12CCC1NC2=O C(CCC(=O)NC1(CCNC(=O)C(C)NC(C)=O)CCCC1)OCC C1(N(C(CCSCCCC)=O)C)CCC(NC(c2cc(COC)cs2)=O)C1 C1(C2(O)CN(C(=O)CC(C)F)C2)(CNC(CCc2ccc(C)c(C)c2)=O)CC1 c1(C(=O)OCC)ccc(CN(C)CCc2ccccc2F)cc1.N12CCCC1C2=O C1(C(=O)NC2C(NC(C3(C=C)CCC3)=O)CCOC2)CCc2nc(C)[nH]c2C1 c1(C(=O)NC(CNC(C(C=C)O)=O)C2CCC2)cccc(C(F)(F)F)c1 C(=O)(C(O)CCC(C)C)NCC(Cn1cc(CCCc2cccnc2)nn1)OC C1(CNC(CNC(C)=O)=O)CC2(CCN(C(=O)C=C(C)c3cnn(C)c3)C2)CO1 Cc1noc2nc(C3CCCC3)cc(C(=O)NC3CC3NC(C3CSC3)=O)c12 c1(C(C)OCC)nc(C(C)SC2CCOCC2)n(-c2ccnc(C(F)(F)F)c2)n1 c1(C(=O)NCC2C(CNC(C3(COC)CCOC3)=O)C2)cnc2c(cnn2C)c1 c1(OC)ccc2cc(C(N3CCC(NC(=O)C(=O)N(C)C)CC3C)=O)[nH]c2n1 c1(NC)cc(C(=O)N(CCCNC(=O)C(C)C(F)F)CCO)cc(Cl)n1 c1(SC)nccnc1C(=O)NC1C=CCN(C(=O)Cn2cccnc2=O)C1 C(=O)(C(C)(C)CC#N)N1CCCC(N2CCN(C(c3cnn(C)n3)=O)CC2)C1 c1(C(N2C(CC(=O)NC)CC2)=O)cc(CNC(c2nocc2C)=O)no1 Cc1ccc(-n2cc(CCCCNC(c3cc(CC(C)C)on3)=O)nn2)nc1 c1(CC(N2CC(C)(NC(C3CN(C(=O)NC)C3)=O)C2)=O)cc(C(N)=O)cc(O)n1 C1(C(N2CCOC(C3CC3)C2)=O)CCCCCCN1C(C1C2CC3C(C2=O)C13)=O C1(NC(CC2(C)CCOCC2)=O)CCN(C(c2ccc(O)c(N)n2)=O)CC1F C1(CC(N2CC(CC(C)NC(C3(CSC)CC3)=O)C2)=O)CCCC(F)(F)C1 CCCC(C)(CCC)C(=O)NC(CNC(=O)COc1cccc(O)c1)C(C)C N1(C(=O)N)CCCCC(CC(=O)CCCC#N)C1.CC(C)(C(=O)OC)C1CCOC1 N1(C(C=Cc2cn(C)nn2)=O)CCC(C2CCCN(C(c3ccoc3)=O)C2)CC1 C1(C(C)C)CC(C(=O)N(C)Cc2cn(-c3ccccc3Cl)nn2)CCO1 c1(C(=O)NCCN(C(=O)CC2(CO)CC2)CC)ccc(COC)nc1C N1(c2nc(C)cc(OC)n2)CC(NC(=O)CN2CCCCCC2)C2CCCCC12 C1(=O)CCOCC(C)N1C1CN(C(=O)Cc2nc[nH]n2)C1.C(C(C)C)OC C1(C)(CC)C=C(C(=O)N2CC3CC2CN3C(=O)Cc2ccc(O)c(C)c2)C1 c1(NC(C(C2CCOC2)N(C)Cc2ccccc2)=O)c(F)cc(C#N)cc1Br c1(CNC2CCC(C(=O)Nc3ccc(O)cc3Br)C2)c(F)ccc(Cl)c1Cl N1(C(Cc2cccc(C)c2)=O)CCCC2(CCN(C(C3CC4(CCC4)C3)=O)C2)C1 N1(C(CNC(CCC)=O)=O)CC=CC1CNC(c1cc(CCCO)on1)=O C1(C(=O)NCCNC(COC)=O)OCCC1CNC(C1CC12CC2)=O C1(NC(c2c(CC)oc(C)c2)=O)CCN(C(=O)CC2CSCCS2)CC1(C)C C1(CC)CCN(C(=O)CC2(C)CC2)C1C(=O)NCCC1CC(C)=NO1 c1(OC)cccc(CN2CC(NC(c3ccc(C(=O)OC)o3)=O)C(F)C2)c1 c1(CC)ncc(CNC(C2(NC(=O)CC3CCCC3O)CC=CC2)=O)s1 n1(CC(=O)NC2C(NC(C(C)c3cc[nH]n3)=O)CC2)ccc2ccc(Br)cc12 c1(C(N2C(C(=O)O)CSCC2)=O)sc2sccc2c1Cl N1(CC)CC(C(=O)NC2CC(CCNC(=O)CNC(=O)C3CC3)C2)CC1=O Cc1nc(CC(C)C)oc1C(=O)N(C(C)CCNC(=O)CNC(N)=O)C N1(C(CC2(OC)CCC2)=O)CC2CC1CN(C(c1c(C)ccc(F)c1O)=O)C2 C(=O)(CN=c1ccc(Cl)n[nH]1)N1CC2CN(C(C3CCCC4(CCC4)O3)=O)C2C1 N1(C(c2nc(CC)oc2)=O)CC(OCCCNC(=O)C2=NOCC2)C(N=[N+]=[N-])C1 C1(NC(c2cc(OC)ncc2)=O)CCCCCN(C(=O)C(C2CCCCC2)=O)C1 C1(C(=O)Nc2cccc(C)c2)CN(C(C23CC(C)(C2)C3)=O)CC(C)O1 C1(C#N)(C(N(CCCN(C(=O)C(C)(C)c2cnco2)C)C)=O)CC2CCC1CC2 c1(CC(C)C)cccc(C(N2CCCC(NC(C3CC=CCO3)=O)C2)=O)c1 c1(NC(CC(=O)N(CCCNC(C2(CC)CC2)=O)CC2CC2)=O)ccc(C)cc1 C12(C(=O)NCCC(C)(C)NC(c3ccc([N+](=O)[O-])[nH]3)=O)CCC(C)(CC1)CC2 CCCCC(O)CC(=O)NCCN1CCCN(C(c2coc(C3CC3)n2)=O)CC1 C1(CC(N2C(CN(C(CCOCC)=O)C)CCC2)=O)CCC(=O)CC1 c1(OC)cc(C(N2CCCC(NC(C3CC(C)C3)=O)C2)=O)ccc1C CN1CCC(C#N)(C(=O)N(C2CC(NC(=O)C(C)(F)F)C2)C)CC1 C1(C(N(CCN(C(=O)CN2CCN(C)CC2)CC)CC)=O)CC2CC1CC2=O c1(C(=O)OC)c[nH]c(C(=O)OC)c1.C12COCC1n1cc(nn1)N2C c12cc(ccc1O)NCC2.C1(CC(F)F)(OC)CCC1 CCC(C)(C)C(O)C(=O)NCC1(CNC(c2cc(CO)[nH]n2)=O)CC(F)(F)C1 CC(CC(=O)NC(CNC(=O)COc1c(F)cccc1F)C1CC1)CC(F)(F)F Cc1ccc(SCC(=O)NCC(C2CC2)NC(=O)CCc2cccs2)cc1 C(=O)(C#CC1CCOC1)NCC1OCCCN(C(Cn2c(C)nnn2)=O)C1 N1(C(CC)=O)Cc2ccccc2C(CNC(c2cnc(O)n2C)=O)C1 N1(C(C(CCC)C#N)=O)CCCC12CCN(C(C13CCOC(C)(C1)C3)=O)C2 C1(C(=O)NCC(C)(CO)NC(=O)Sc2ccccc2)CN(CC#N)c2ccnn2C1 N1(C(CCSCC)=O)CCC(C2CCN(C(c3cnsc3)=O)C2)C1 C1(C(=O)Nc2ccc(C#C)cc2)CCCCCCN1C(=O)CN1CSCC1=O N1(C(c2c(NC)cccc2)=O)CCOC(C)(CNC(=O)CCn2ccnc2)C1 C=CCCC(F)(F)C(=O)NC(CCC)CCCNC(c1[nH]nnc1C1CC1)=O c1(C(=O)NC(CNC(c2[nH]nc(OC)c2Cl)=O)C)ccc(C)c(F)c1Br c1(CNC(C2CCN(C(=O)OCC)C2)C(F)(F)F)nccc2c(C)cccc12 N1(CC(=O)NCCC(C)C)CC(C(=O)OCc2ccccc2F)Oc2ccccc21 c1(C(=O)NC(C)CN(C)C(C2C3(CC3)C23CC3)=O)cc([N+](=O)[O-])cc(Cl)c1Cl N1(C(CCCNC(C)=O)=O)CCN(C(=O)CSCC(F)(F)F)C(CCO)C1 c1(OCC(=O)N(CC(C)NC(CSCC#C)=O)CC)ccc(F)nc1 C1(CN(C(N(CC)CC2CC(F)(F)C2)=O)C)COC(C(F)(F)F)C1 C1(CNC(C(CC)OC)=O)CC2CCCCC2N1C(=O)COCCC(C)C C12(CC(=O)N(C3CCCN(C(=O)CS(=O)(=O)N(C)C)C3)C)CC3CC(CC(C3)C1)C2 Cn1nc(C2CC2)cc1N.C12(C)CCCN1C2=O.c1(C)cccc(O)c1 c1(OCCC(=O)OCc2c(C)oc(-c3ccc(F)cc3)n2)cc2c(s1)CCC2=O CCC(C)(CCNC(C1CCC(O)CC1)=O)NC(=O)C=Cc1cncn1C C(=O)(C1=C(C2CC2)N(CCC#N)C(=S)NC1c1cnc2c(cnn2C)c1)OC c1(C(=O)NCCOC2CN(C(CC3(C)CCOC3)=O)C2)cnn2c1OCC(F)C2 c1(-c2nc(CCCCc3scc(C)n3)nn2CCF)cc(C(F)(F)F)ccc1F C1(C(=O)NC(C2(O)CCN(C(c3cnc(N)cn3)=O)C2)C)Cc2ccccc2O1 C1(CC(=O)NC(C#C)CCC)CCCN(C(c2cnccc2C)=O)C1 CCCC(C(=O)OC)C(=O)NC1(C(N2CCC(F)(F)C(C)C2)=O)CCN(C)C1 c1(C(N2CCN(C(CCC3OCC(C)(C)C3)=O)CC2)=O)cnc(S(C)(=O)=O)s1 O=C(CC1CCc2ccccc21)NC1(CNC(C2CC2C2CCCC2)=O)CCC1 c1(CC(=O)NC2(CNC(C3CC(F)C(=O)N3)=O)CC2)c(F)cncc1Cl C1(C(=O)NC(C)C(C)NC(c2cc(=O)n(C)cn2)=O)CC(c2ccncc2)=NO1 N1(CCC)CCCC(C(=O)NC2CCCC2NC(=O)C(C2CC2)C2CC2)C1 N1(C(CC(CC)C2CC2)=O)CCN(C(c2csc(C(C)(C)C)n2)=O)CC1CO C(=O)(CCC(C)(C)F)C(C(C)N1CCC1CNC(=O)C(c1ccccc1)F)=O.N c1(C(=O)NCC2(F)CCC(NC(C3CC(F)(F)C3)=O)C2)cnc2[nH]cnc2c1 Cc1cn(CC(=O)NC2CCN(C(C3CCC3(C)C)=O)C23CCC3)c(=O)nc1O C(=O)(C1=CCSC1)N(C1CC1)CC1(O)CN(C(C2(N(C)C)CC2)=O)C1 C1(N(C(=O)CCc2cnco2)CC)CCCN(C(=O)CCc2cccnc2)C1 Cc1nn(C)c(C(=O)NC2COC3C(NC(C4CSCCS4)=O)COC23)c1Cl CC1CN(C(=O)CCc2nccs2)CC(C)N(C(c2ccc(C3CC3)nc2)=O)C1 C(=O)(C(C)(C)CC(=O)N1CCC(CN(C)C(c2nccc(F)c2Cl)=O)C1)OC c1(C(N(C(C)CN(C(=O)C(C)C=Cc2ccccc2)C)C)=O)nnc(O)cc1O c1(OC)cccc(C(C2CCCO2)NC(c2cc(-n3cccn3)ccn2)=O)c1 C(C(=O)N1CCC(C(N2CC3CC3(CO)C2)=O)(C(C)C)C1)(C(C)C)OCC c1(CC)cnc(C(=O)NCCC(=O)NCC(CSCCCOC)OC)cn1 N1(C(C=C(C)C2CC2)=O)CCOC(CCNC(C2CCN(C)C2)=O)C1 N1(C(C(CNC(C(C(C)C)C)=O)(F)C(C)C)=O)CCc2cccnc2C1 N12CCOCC1C2.C1(CCn2cc(C3(C)CCC3)nn2)C=CCOC1 C=CCC(CN)C(=O)n1c2nnc1s2.C(C)(C)(C)OC(=O)N(C)C C(=O)(C#CC(C)C)NCCCN(C(=O)CC1CCC2CC12)CC c1(C(=O)NCCC(C(=O)NCC2N(CC)CCC2)OC)ccc(O)nc1C C12(C(=O)OC)CCCCC1(C(N1CCCC(NC(=O)C(F)=C(C)C)CC1)=O)CC2 CCC(C)CCCC(=O)N1CCC(C(C)NC(=O)CCCC(N)=O)C1 CCCC(CC(C)C)C(=O)NC1CCCCC1NC(c1ccncc1C1CC1)=O C(=O)(C1c2c[nH]nc2CCC1C)NCCC(C)NC(=O)Cc1cc(Cl)ccc1Cl C#Cc1cncc(NC(C2(F)CCN(C(=O)CCc3nc(O)n[nH]3)C2)=O)c1 C1(C(=O)NCCCCCCNC(c2cccc(C)n2)=O)Cc2nn[nH]c2C(C)C1 C(=O)(CC(C)(C)C(F)F)NC(C)CNC(c1ccc(F)cc1)=O C(=O)(N(O)C(C)C)NC(c1cnn(CC)c1)CC c1(OC)ccc(CC(N2CCCC(NC(C3CCNC3=O)=O)CC2)=O)c([N+](=O)[O-])c1 CC(C)(O)C(F)C(=O)NCCC(=O)NCC(O)C(F)F C1(C(CC)(C)C)CCC(C(N2CCC2CNC(C2CC2(C)C)=O)=O)CC1 CC1CC(CC(N2CC=CC2(C)C)=O)CN1C(=O)CCc1cnn(C)c1 Cc1ncc(C(=O)NCC2(F)CCN(C(=O)CN3CC(=O)NC3=O)C2)n1C c1(C(N2CCC(C)(NC(C(C3CCOCC3)OC)=O)C2)=O)cncc(C#N)c1 CC1CC(C(=O)NCc2ccncc2F)CN(C(C2C=CCS2)=O)C1 OCC1(CCNC(C(Cc2ccc(Br)s2)C(=O)O)=O)CCC1 C(C(CO)(CO)NC(=O)C=CC=Cc1ccccc1)N(C(C1(CC)CCOC1)=O)C C1(C(=O)NCC2CC(C(C)C)=NO2)(CC)CCN(C(c2c[nH][nH]c2=N)=O)CC1 c1(NC(C(C)(C)C(=O)OC(C)(C)C)c2nnnn2C)ccc(F)cc1CSC N1(C(c2occ(C)c2C)=O)CCCC(CNC(c2cccc(C(N)=O)n2)=O)CC1 c1(C(=O)NCC2CN(C(C3(CC(C)=O)CC3)=O)CC2C)cc(F)cc(Cl)c1 C(CC(C(C)C)NC(c1csc(CS(C)(=O)=O)n1)=O)N(C(c1c(C)snn1)=O)C C(=O)(C(C(C)(C)C)NC(=O)C(=O)NCNC1CCNC1)OC c1(C(=O)NCCC2(CNC(C3C(CC)C3)=O)CC2)cc2n(n1)CCCC2O CCCCC(O)C(C)C(=O)NC1(CCC)CCN(C(=O)CC2(CO)CCC2)CC1 N1(C(C2(C(C)(C)C)CCCC2)=O)CC2CN(C(C3CCCO3)=O)CC2(C)C1 Cc1cc(C(=O)NC2(CF)CCN(C(C3(CO)CCCC3)=O)C2)cc(C)c1F C(CC(C)CCNC(C1CCC(C(C)C)CC1)=O)NC(C1(CC=C)CCCN1)=O c1(CO)ccc(Cl)nc1C.CCCC(C(=O)N1N2CCC(CC2)C1)OCC c1(C(N(CCN(C(C23C(C)OC(CC2)C3)=O)C)C)=O)ccc2cccc(F)c2n1 CCCCC(C(=O)NCC1(F)CCN(c2cc(OC(C)CC)ncn2)CC1)C(C)C C1(NC(=O)CC2(O)CCC2)CCC(O)CN(C(C2OCCOC23CCC3)=O)C1 N1(C(CC)=O)CC(NC(=O)Cc2ccc(C3CCC3)cc2)CC1(C)CC Cc1nc(C)c(C(=O)NCC=CCNC(c2cc([N+](=O)[O-])c[nH]2)=O)c(C)n1 N1(C(C(C(C)C)CO)=O)CC(C)OC2(CCN(C(C3CC(C)(C)C3)=O)C2)C1 C1(NC(c2cn(CC)nn2)=O)CCC2CCC1CN2C(=O)C(C)SC c1(C(N2CCC(N(C(CCC(=C)Br)=O)C)C2)=O)cc(-n2ccnn2)ccc1F C1(NC(N2CCOC(C3CC3)CC2)=O)CC[Si]2(CCCC2)CC1 c1(C(N2CCCC(CCNC(C3COC(=O)O3)=O)C2)=O)ccc(Cl)nc1O N1(C(CCC(=O)NC)=O)CC2CCC(NC(=O)Cc3cccnc3OC)CC2C1 c1(OC)ccc2c(CNC(=O)C(N3CCCC3c3ccccc3)=O)c[nH]c2c1 C1(C(=O)NC2(C)CC(F)(F)C2)CC(NC(=O)CC2CCCNC2=O)C12CCC2 N1(C(CC2(NC(C)=O)CC2)=O)CCC(CCC(C)(C)NC(=O)C(O)C(C)C)CC1 C(CNC12CC(C(=O)NC)(C1)C2)(CC(F)(F)F)NC(c1c(OC)ccnc1)=O c1(NC(C(C)C)=O)cc(-c2ccc(NCC3CCSCC3)s2)cc(C2CC2(F)F)c1 c1(C(CNC(C=CC(C)NC(CN(CCC#C)C)=O)=O)O)ncc[nH]1 C1(CCC(=O)N(CC#C)CCO)CCCN(C(=O)Cc2cncs2)C1 Cn1ncc2ncc(C(N3CC(CO)(NC(=O)Cc4ccsc4)C3)=O)cc12 C1(C(N(CCCNC(C2C(CCC)C2)=O)C2CC2)=O)CS(=O)(=O)CC(=O)N1 CCC(O)C(C)(C)C(=O)N1CCC1CNC(c1c(-c2ccco2)c[nH]c1C)=O c1(CC(=O)NC2CCN(C(CCNC(COC)=O)=O)C2)c(C)cc(N(C)C)cc1C N1(C(CCNC(COC)=O)=O)CC(CNC(=O)CC2CC(C)=NO2)CC1(C)C C#CCCCCCC(=O)NC1CCC1CNC(=O)Cc1cnccc1OC C1(NC(C2(NC(C)=O)CCCCC2)=O)CC2CN(C(=O)Cc3cc[nH]n3)CC12 C(N=c1nc(NC2CC(C)n3ncnc32)c2c([nH]1)CSC2)c1[nH]c(=NC)sc1 S(=O)(=O)(C(F)(F)F)NC(=O)C=CC1CC1.C1(CC=C)(O)COC1 C(c1ccc(F)cc1F)=CC(=O)N(CCCNC(=O)CC1CC1(C)C)C(C)C c1(CN(C)C(c2cccc(-c3ccn(-c4ccccc4)n3)n2)=O)ccc(F)cc1 c1(C(N2CC3=C(CN(C(C(CC)COC)=O)C3)C2)=O)cc(F)cc2cccnc12 c1(NC(C=CCN(C)C(c2cccnc2C2CC2)=O)=O)c(C(N)=O)cnn1C c1(CC(=O)NC2CC(F)(CNC(C(C)=C3CCC3)=O)C2)ccc(C)c(Cl)c1 C1(NC(c2ccc3cc[nH]c3c2)=O)CC2CC1CN(C(=O)C=CCO)C2 C1(=CC(=O)NCC(CCCC)NC(=O)C(CC)CC)CN2CCC1CC2 c1(OCC(N2CC(C)C(NC(C3CC4(CCC4)C3)=O)C2)=O)ccc(Cl)cc1Cl N1(C(C2C=CC(NC(C3CCC=CCC3)=O)C2)=O)CC2(CCC2)C12CCC2 C1(NC(CCCOCC=C)=O)CN(C(c2cc3sccc3s2)=O)C(C)(CC)C1 C(=O)(CP(C)(C)=O)NCCN(CCOC)C(c1cnc(COC)nc1)=O C=CCCCCCC(=O)N1CC(NC(=O)Cc2ccnc(C)c2)CC1(C)C C1(C)(C(N2CC(OC)(CNC(=O)C(C)CCN(C)C)C2)=O)C(C)(C)C1(C)C CC1(C)CCCN(C(=O)Cc2ccccc2Cl)C1CNC(c1ccc[n+]([O-])c1)=O c1(CN(c2ccccc2)C(C2C(C)(C(F)F)C2)=O)cn2c(n1)CCCC2 Cc1c(NC(C2CCCN(C(=O)C(C)CO)C2)=O)cccc1[N+](=O)[O-] CC1=NOC2(C1)CC(c1nc(-c3ccccn3)nn1C1CCOC1C(F)(F)F)C2 C1(C(N)=O)C2CCC(C2)C1NC(c1ncccc1NC(=O)CC1CCCC1)=O C(C(C)(O)C(=O)N1CC(NC(c2c(-c3cccnc3)noc2C)=O)CC1C)OC C1(NC(CSC)=O)CCCC(NC(=O)CSc2nncn2C)CC1 N1(C(C2(OCC)CCSCC2)=O)CC2(CNC(C3(C)CCCS3)=O)CCC1CC2 N1(C(c2n[nH]c(C)c2N)=O)CC2CC(NC(c3ccn(C(C)(C)C)n3)=O)C2C1 C(=O)(CCCC(=O)NCCC1CCCN(C(=O)Cc2nc(C)sc2C)C1)OCC C1(C(=O)NC2CN(C(Cc3n(C)ccn3)=O)C2)C(C2CC2)C1(F)F c1(NC(c2c(OC)c(F)ccc2)C)nc(Cl)nc2c(F)cc(C)cc12 C1(CNC(c2cncc(OC)c2)=O)CCN(C(=O)C(CO)N(C)C)C(C)C1 C(N=c1ccnc(-c2ccccc2)[nH]1)C1C(NC(=O)CC2CC2(Cl)Cl)C1(F)F C1(C)(C(N2CCN(CCn3cc(C(CC)O)nn3)CC2)=O)CCCCCC1 CC(CC(=O)N1C2CCC1CC(NC(=O)Cc1nc(C3CC3)cs1)C2)P(C)(C)=O N1(CC(=O)N(C(CNC(=O)C(F)CC2CCOC2)C2CC2)C)CCOCC1 N1(C(c2ccc(CC3CC3)o2)C(=O)NCCCC)CC(c2ccccc2)C(C)(C)C1 Cc1c(NCC(F)(F)Cl)cnn1C c1(CC)nc(C(=O)NC2CC(NC(c3cnc(OCC(F)F)nc3)=O)C2)c(C)o1 C(=O)(C(CC(=O)NCCCOCCCOC(C)(C)C)NC(C1CC1)=O)OC C#CC1(CNC(=O)C(C)(CO)NC(=O)CN2CCC(OC)C2)CCCC1 C(=O)(CC(C=C)CCC)N1CCC(C(C(=O)NCCSCC#C)C)CC1 CCC(CO)C(=O)N(CC(C)(C)NC(c1ccnn1CCOC)=O)C CN1CCN(CCCNC(CC(N2CCCCC2c2ncc[nH]2)=O)=O)CC1 c1(CC)ccc(F)c(NC2c3ccc2o3)c1.c1(SC)nnnn1CCOC C(C)(C)(CCC(=O)NC(C1CCCC1)C)NC(c1cc(OC)ns1)=O C1(NC(=O)CCc2ccc(F)cc2)CCCC12CN(C(C13CC(CO1)C3)=O)C2 c1(CC)nc(C)[nH]c1C(=O)NC1CCC1NC(C1(F)CCOC1C)=O c1(NC)ccc(F)cc1C(N1CC(CNC(C2COC3(CCC3)C2)=O)C1)=O C1(C(N(C2CN(C(=O)COC(F)(F)F)C2)CC)=O)CCc2ncnc(C)c2C1 C1(CC)(NC(=O)CCCCCO)CCCN(C(c2ncccc2C)=O)C1 n1(CC2CCN(C(=O)NCCC3CCCNC3)CC2)cnc2ccccc12 N1(C(c2c(CC)non2)=O)CCN(C(=O)C=Cc2csc(Br)c2)CC1C CC1(C)OCCOC1CC(=O)NC(CNC(=O)C(C)(C)c1ccccn1)C1CC1 C(=O)(C(C)C(C)c1ccco1)NC1(CNC(CSCCCC)=O)CCCC1 N1(C(CNC(c2csnc2Br)=O)=O)CC2CCC1CN2C(C1(c2cc[nH]n2)CC1)=O N1(C(CC(C)SC)=O)CCC(C)(C)C(CNC(c2n[nH]c3c2CCOC3)=O)C1 C1(CNC(N2CCCOC(c3ccc(Br)cc3)C2)=O)CC23CCCC2(C1)C3 c1(C(=O)OC)ccc2[nH]c(=NC(C)CCSC)oc2c1 Cn1cc(C#N)cc1C(=O)NCCCC(O)C(=O)N1CC(c2ncc[nH]2)C1 C(N=c1[nH]nc(CC(C)C)s1)C1OCCN(C(C(=Cc2cn[nH]c2)C)=O)C1 N(C1CCCc2ccc(O)cc21)C(=O)CCNC(c1cn(C)nc1)=O Cc1cn2c(n1)CCC(NC(=O)NCc1ccc(Br)c(C)c1C)C2 c1(NC(=O)NC2CN3CCC2C3)ccc([N+](=O)[O-])c(Cl)c1 C1(NC(C(CC)CCOC)=O)CN(C(C2(C)CC(F)(F)C2)=O)CC2(CCC2)C1 C(=O)(C(O)CCCNC(c1ccc(C(N)=O)[nH]1)=O)N1CCN(C(C#C)C)CC1 Cc1cc(C#N)cc(C)c1NCCC(O)C1CCCC1 CC(C)CS(=O)(=O)CCC(=O)N(CC(C)CNC(=O)CSc1cccc(O)c1)C N1(C(C(n2ncc(C)c2)C)=O)CC(NC(c2cc(F)cs2)=O)C(n2ccnn2)C1 c1(C(=O)NC(C2CCOC2)CNC(c2cnc(C)o2)=O)c(C)nn(C)c1C(F)F C1(CNC)CCC(C(F)(F)F)CC1.n12ccnc1CNC(=O)NCC2 C12CCCC(C1)N2.N1(CC2(C)CC2)CCN(C(=O)OC(C)(C)C)CC1 C(C(C)(C)CCNC(c1ccc(C(C)(C)C)o1)=O)NC(C=CC(=O)N(C)C)=O c1(SCC(=O)N(CC)CC2(CCN)CC=CCC2)ccc(OC)c(OC)c1 CC(=O)CCCC(=O)N1CCN(C(c2ccnnc2O)=O)CC1c1ccncc1 c1(C(N2C(CNC(CCCN(C)C)=O)C(C)(C)CC2)=O)ccc2occc2c1 C12(NC(c3c(OC)ncc(Cl)c3)=O)CCCCC1N(C(=O)CCC(C)(C)F)CC2 C1(C(=O)NC(CC)C2CC2)CCN(C(=O)CCc2ccn(C)c2)CC1O C(=O)(C(C(=O)NC1(CNC(=O)C(F)C2CCC2)CCCC1)C(C)C)OCC c1(C(=O)NCCCN(C(C(C)c2ncco2)=O)C)cnc(N)c([N+](=O)[O-])c1 N1(CC)CCOC(C(=O)NCC(O)CCNC(c2ccccc2C2(C)CC2)=O)C1 c1(C(=O)NCC(CNC(c2c(C)snn2)=O)CO)ccc2c(c1)CC(=O)NC2 N1(C(CCC2(C)N=N2)=O)CC(NC(=O)CC(C)(C)C(F)F)CC12CCOCC2 C1(C(N2CC(C)(C)C(NC(=O)C=CC(F)(F)F)C2)=O)Cc2c[nH]cc2S1(=O)=O c1(C(N2CC(NC(CC(COC)C)=O)C(C)C2)=O)c(C)nn2cc[nH]c(=O)c12 C(CN=c1cc2n([nH]1)CCC2)(c1ccc(-c2nn[nH]n2)cc1)OC N1(C(c2c(C)csc2Cl)=O)CC(C2CCCN(C(c3ccc(Cl)[nH]3)=O)C2)C1 C1(C(=O)NCCN2C(=O)C2CCNC(C)=O)(CC)CCNC1=O.OCC C1(S(N)(=O)=O)(C(=O)NCC2N(C(Cc3c(C)n(C)nc3)=O)CCOC2)CCCC1 c1(C(N2C(CNC(=O)CCC3CCCO3)CCC2)=O)ccncc1Cl c1(C(C2(c3ccccc3)CC2)=O)ccc2ncccc2c1.N12CCOC(C1)C2 Cc1cc(C(=O)NC(C2CN(C(=O)C(C)OCCC(C)C)C2)C)cc(C)c1 c1(C(=O)NCCN(C(C(C(C)C)(C)O)=O)C)cc(O)nc2c1CCCC2 c1(C(=O)NCCN(C2CCCC2)C(c2ccc(CSC)o2)=O)ccc(O)nn1 c1(C(N2C(CN(C(CN(C3CC3)CC)=O)C)COCC2)=O)cc2ccncc2[nH]1 c1(C(=O)NC(CNC(c2cc(C)oc2C)=O)(C)CC(C)C)cc2c[nH]cnc-2n1 N1(C(C(COC)C)=O)CCC(NC(=O)C(=Cc2cnn(C)c2)C)C12CCCC2 C1(C(CC(C)(C)C)=O)CCN(N2CC3(CCCC3)C2c2cccs2)CC1 c1(CC)cc2c(CC(=O)NCC3(OC)CN(C(C4(F)CC4)=O)C3)csc2s1 c1(C(=O)OC)cc(NC(N2CCC2CC(=O)NC2(C)CCOC2)=O)n[nH]1 c1(C(C)C(=O)NCC(C)(C)CNC(=O)CCC2CC2C)ccc(F)c(F)c1 c1(C(=O)NC(CC(C)NC(c2cc(CCOC)on2)=O)C)cnc2n1CCCC2 C1(C(=O)NCC(C)NC(c2ccc(O)nn2)=O)C2CCC1(c1ccc(F)cc1)C2 C1(C(N2CCN(Cc3cccc(Cl)c3)CC2)=O)C2CC3C(C2=O)C13 C1(C(=O)NCC(C2(O)CCN(C(=O)C=Cc3cnc[nH]3)C2)C)(CC)CCOCC1 C1(NC(C=CCN(C)CC)=O)CCN(C(c2cc(O)nc(Cl)c2)=O)CC(C)(C)C1 C(=O)(CN=S(C)(C)=O)NCC(C)(CO)NC(C1CC1c1ccccc1F)=O C(=O)(C(CC(C)C)C(C)C)N1CC(OC)(CNC(=O)Cc2cccn2C)C1 C(=O)(CCCC(C)C)NC1CCN(C(C(C)OCc2cccc(C)c2)=O)C1 c1(-c2cn(CCC(=O)NC(CCC)CCC)nn2)cc2c(s1)CCC2 c1(OC)ccc(OC)c(C2CCN(CC(N3CC(O)CCC3CO)=O)CC2)c1 c1(OCC(=O)N(C2CCC(NC(C3(C)CC3(F)Cl)=O)CC2)C)ccc(F)cc1 c1(C(=O)NC(C)Cc2cn[nH]c2)cc(Oc2ccccc2)cn1C CC1CC=CCC1NC(=O)C(C1(O)CCC1)NC(=O)C=CC(F)(F)F CCCCCCC(C)C(=O)NC(Cc1ccccc1)CCOC C1(Nc2ccnc(C(N3CCCC(C(C)NC(C)=O)C3)=O)n2)CCC(=O)NC1=O c1(C(=O)NC(C(C)NC(c2cnc(C(=O)OC)s2)=O)C)ccc(C)cn1 CCC(CC(=O)NCC1CN(C(C2CCCN2N=O)=O)C2(CCC2)C1)CC(C)C c1(OC)ncc(Cl)cc1C(=O)NCC(C)CNC(C1CC(N2CCOCC2)C1)=O C1(C)(NC(CCSCCCC)=O)CCCN(C(c2nc(Br)cnc2N)=O)C1 C12(C(=O)NC(c3ccccc3)Cc3ccccc3)CC3CCC(N3)C1C2 Cc1cn2cccc(NC(C3CC4CCN(C(=O)CCOC(C)C)CC34)=O)c2n1 c1ccccn1.c1(C2CN(C(C(C)OCC)=O)C2)nc(C(=O)NOCCC(C)O)co1 c1(C(=O)NC2C3CN(C(c4c(C)noc4C)=O)CC32)ccc2c(ccn2C)c1 c1(C(=O)NC2C(CNC(C(N(C)C)C3CC3)=O)CC2)cn2c(n1)SCC2 N1(C(CC=CC=C)=O)CCC(C(C)(C)NC(c2csc(C(C)=O)c2)=O)CC1 Cc1scc(C(N2CCN(CCNC(=O)CC3(C)CC3(F)F)CC2)=O)c1C1CC1 Cc1cc(C(=O)NCCC(C)NC(C2(CCC3CCCCC3)CCC2)=O)n(C)n1 c1(C(=O)NCC2(C)N(C(CC(=C=C)C)=O)CC(F)(F)C2)c(C)cc(C#N)cc1C C1(NC(C=CCC)=O)CCCC(N(C)C(c2cnc(-c3cccs3)o2)=O)C1 C1(C(=O)NCCCC(=C)Cl)(CC)CCCN(C(c2cc[nH]c2)=O)C1 c1(C(c2n(CCCC)nnn2)NCC2C(C(C)(C)C)CCO2)cnn(C)c1CC C=CCC(C)(CC)C(=O)N1CC(CNC(c2ccc(O)nc2Cl)=O)C(F)(F)C1 N1(C(C(C)=C(CC)C)=O)CCN(C(=O)C(F)Cc2ccccc2)C2CCC12 c1(OCCC#C)ccc(C(=O)OCC2(CO)COCCN2)cc1 c1(CC(=O)NC2(CNC(C(C)c3cncs3)=O)CC2)ccnc(O)c1 C12CC(F)(F)CN1c1noc2n1.C1(CCC(N)=O)CCS(=O)(=O)C1 Cc1cccc(F)c1CC(=O)N(CC(C)N(C(=O)COc1ccccc1F)C)C CC(C)(CN(C(=O)CC1(C)CC1(Cl)Cl)CC(=O)NCc1ccccc1Cl)C(=O)O c1(C(C)C(=O)NC2(CNC(C3CCC(C)O3)=O)CCC2)ccc(Cl)c(Cl)c1 C(=O)(C1=C(C2(C)CC2)N(c2ccccc2C)C(=S)NC1c1sccc1Cl)OC C1(CNC(C2CCC(CC)O2)=O)CN(C)CCN1C(=O)CC12CCC(CC1)OC2 c1(C(=O)NC(C2CN(C(c3ccc(C)nc3C)=O)C2)C)ccc([N+](=O)[O-])cn1 N1(C(C(=O)N(C(C)C)C)=O)CCC(NC(=O)OC(C)C)CC1.C(C)(CO)N C(=O)(C1CCc2c[nH]nc21)N1CCCCC(NC(c2c(N)sc(C)c2C)=O)C1 C(C(N=[N+]=[N-])C(=O)N1CC(C(=O)NCC(F)C2CCC2)C2(CC2)C1)OCC C12(CCc3n(-c4ccc(OC)cc4)nc(CCN(C)C)n3)CCCC1OCC2.OC C1(C(=O)NCC2CC(NC(C3CC(F)(CO)C3)=O)C2)CCCCCC1(F)F c1(C(=O)NCC(C)NC(C2CCn3nncc3C2)=O)cc2cccc(Cl)c2s1 C1(CNC(C)=O)CN(C(=O)Cn2cc(C(F)(F)F)c(C)n2)CCN1C O=C1CC(CCC(=O)NC2(CF)CCN(C(c3ccn(O)c(=O)c3)=O)C2)=NN1 N1(C(COCCC=C)=O)Cc2n[nH]cc2C1C(=O)NCCCc1ccn(C)n1 c1(C(=O)NCC2CN(C(CSC)=O)C(C)C2)ccc(C)c(O)c1 C(C(C)(C)C(=O)NCC(c1cn(CC2COCCO2)nn1)C)NC(C)=O Cn1cc(C(N2CC(F)(CNC(C3CCC(C)(C)OC3)=O)C2)=O)n(C)c1=O c1(C(N2CC(NC(C(C)C#N)=O)C(CO)C2)=O)cc2cnccc2o1 c1(C(=O)NC(CNC(C2C(COC)C2)=O)(C)C(C)C)cccn2ncc(Br)c12 c1(OC)cccc(C(N2CCC(N(C)C)CC2)C2CC2)c1Cl C12(CNC(c3ccns3)=O)CC1CN(C(=O)Cn1ncc(Br)n1)C2 c1(C(=O)OC)cc(C(N2CC(O)CC2C(=O)Nc2sccc2CO)=O)cc(F)c1 Cc1ccc(C(=O)NCC(C)NC(=O)C(c2cccc(Br)c2)(C)C)c(N)c1 C(C1CC(C)Oc2ccccc21)NC(c1c(OCC(C)C)cccc1)=O C1(O)(C(=O)NCC2C(C(=O)NCc3n(CC)cnc3)C2)CCOC1(C)C C1(C(N(CCN(C)C)CC)=O)CCN(C(c2cc[n+]([O-])cc2)=O)CC1O C1(C(=O)NCC2CCN(C(C(C)(C)OCC)=O)C2)CC(F)(F)C1(F)F C(=O)(C(C)(C)CCC#N)NCCC1(CNC(C(n2c(C)cc(C)n2)C)=O)CCC1 Cc1nc(N2CCC(C(C)NC(=O)C(F)C3CC3)CC2)c2scc(C)c2n1 N1(C(CC2C=NN(C)C2=O)=O)CCCC(F)(C(=O)NCC(C)(O)CO)C1 c1(C(=O)NCC(CNC(C(C)=O)=O)(C)O)csc(C)c1Br c1(C(=O)NC(CC)CN(C)C(c2cnc(-c3ccco3)[nH]2)=O)ccc(CO)nc1 C(=O)(CC1=CCCCC1)NC(C1CN(C(C2(C(=O)NC3CC3)CC=CC2)=O)C1)C C1(C)(C(=O)NC(C(=O)N2CCC(C(=O)OCC)C2)C(C)C)C=CCCC1 C(=O)(C(CO)C(F)(F)F)N1C(C)CC1C(N1CC2CC1C2)=O C=CCC(CNC(C1CCCN1C(=O)C(C)(F)C(C)(C)F)=O)CC(C)C C(=O)(C(C)(C)CCC(=O)NC1CC1NC(C1COCC1(C)C)=O)OC N1(C(C2(C)CCOC2)=O)CC2(C1)SCCC2NC(c1csc(-c2cnc[nH]2)n1)=O c1(C(=O)NC23CC(C(=O)NC4(c5ccsc5)CC4)(C2)C3)cc2ccccc2[nH]1 CC1CC(C)(C(=O)NCCn2cc(CNC(C3CCC(=O)O3)=O)nn2)CCO1 N1(C(C2CC=CC(n3cc(C4C5COCC45)nn3)C2)=O)CCCCC(F)(F)C1 C1(CNC(c2c(C)n(C3CCOC3)nn2)=O)CCC(C)CN1C(=O)CC1CC1 C1(C(=O)NCC(CC)C#N)(CC)CCCN(C(=O)C=CC2CCC2)C1 C1(C(C)NC(c2scnc2C(F)(F)F)=O)CCN(C(=O)CNC=O)CC1 C1(NC(CCC=C(C)C)=O)CCC(C)N(C(c2cnn(C(C)(C)C)c2C)=O)C1 C1(NC(c2ccn(CC#N)n2)=O)COCCN(C(=O)Cc2ccc(F)cc2Cl)C1 CC1(C)CN(C(C2CCCC(F)C2)=O)CCC1C(=O)NC1CCCC1F Cc1nccnc1C(C)NC(=O)C(C1CCCN(C(=O)CC2(C)CC2)C1)C C(C(=O)N1CC2C(NC(c3sccc3Br)=O)C2C1)(C(C)(C)C)N(C)C Cc1cccc(OC(C)C(=O)NC(C)CCNC(=O)C(=O)Nc2ccccc2)c1 C1(C2CCN(C(C3CCCN3C3CC3)=O)CC2)(NC(c2c(C)nn(C)c2)=O)CC1 c1(NC(=O)CSCCOCCNC(C2(F)CSC2)=O)ccc2c(c1)OCCO2 N1(C(CS(CC)=O)=O)CCC(C2CC2)(CNC(=O)Cc2coc(C)n2)C1 C1(OC)CC2CC1CN(C(=O)C(F)CC(C)(C)NC(=O)CCn1ccnn1)C2 C(=O)(C(C)(CC(F)(F)F)c1ccccc1)N(C(C)CNC(C1CC(NC)C1)=O)CC c1(CC(=O)NCC(C2CC2)NC(C2CCN(C)C2)=O)csc2c(F)cccc12 c1(SC)cccc(NS(=O)(=O)NC(=O)C(C(c2ccccc2)N(C)C)C2CC2)c1 C1(C(=O)NCC(=C)F)CC2C=CC1N(C(=O)C=Cc1ccccc1)C2 C(c1cocn1)=CC(=O)N(CC(C)NC(C1CC2(CC2)C1)=O)C CCCCC(F)C(=O)N1CC2CC1CN2CC(O)COCc1ccccc1 c1(C(=O)NCC2CN(C(CCc3cccc(C)c3)=O)C3C2C3)nnc(O)nc1O c1(C(=O)NCC2N(C(CN(C)C)=O)CC(C)(C)CC2)ccc(Br)c(Cl)c1F c1(OC)ccc(C(=O)NC2CC23CC(NC(C2CCCOC2)=O)C3)cc1O c1(C(N2C(C)C(NC(=O)COC3(C)CCCC3)CC2)=O)coc2c1CS(=O)(=O)C2 O=C1C2CC3C(C2)C13C(N1CC(O)C(O)C1CO)=O.N1CCCC(CCCO)C1 Cc1cnc(OCC(=O)NC2C=CCC2)nc1 N1(C(C2(CC)CCC2)=O)CCN(C(=O)CC2CC(=O)C2)CC(C)C1 n1(CCC)nccc1C(=O)N(CC(N1CC(N2CCOCC2)C1)=O)C(C)C C(=O)(N=c1[nH]oc(-c2ccc(Cl)cc2)c1C#N)N1C(C)(C(=O)NCC=CC)CCC1 c1(OC)ccc(C2CCCN2C(c2ccccc2SCc2cccs2)=O)cc1F C1(CC(=O)NC2C3CN(C(c4c(CC)nns4)=O)C(C3)C2)CC2(CCCC2)CO1 c1(SC)ncc(N)c(C(=O)NCC2CCCC2NC(c2cc(C)ncn2)=O)n1 C=C(Cl)CC(C(=O)NCCc1cccs1)NC(=O)CSC(C)C c1(C(N2C(CN(C(CSc3nc(C)[nH]n3)=O)C)CCC2)=O)nccc(N)c1Cl N(C(=NCCC1CC(F)C(=O)N1)NCC1CCCCO1)CCOC C1(C(=O)OC)CC12CN(C(=O)CC(C)CNC(=O)CNC(C)=O)C2 C(=O)(C1CCCc2cccnc21)NC(CNC(CCC(=O)NCC)=O)C(C)C C(c1ccc(OC(F)F)c(NC(=O)CN2CCC(=CC=CC#N)CC2)c1)=CC C1(NC(c2ccccn2)=O)CCC2CCN(C(c3ccc4cccnn34)=O)C1C2 CC1C(NC(C2CC=CC2)=O)CCCN1C(c1cc(NC2CC2)ncc1Cl)=O C1(C(=O)N(Cc2nnn(C)n2)C2CC2)CCCN1NC(=O)CCC1CCCO1 Cc1ccc(Br)c(F)c1C(=O)NC1(CNC(C2(C#N)CCC2)=O)COC1 c1(CC(=O)NC2C(NC(c3c(C(C)=O)cccc3)=O)C2)c[nH]c2cc(Cl)ccc12 C1(NC(C2(NC(=O)C(F)F)CC(O)C2)=O)CC2(CNC(=O)O2)C1 c1(NC(=O)CCCOC(c2cnn(C3(C(F)(F)F)CC3)c2)=O)ccc(F)cc1 c1(-n2c(C(COC)C)nc(-c3cc[nH]n3)n2)ccc2ncccc2c1 N1(C(C(n2ccc(C)n2)C)=O)CC(C(N)=O)C2(CC2)C1.c12occc1C(=O)N2 O=C1NCC2C(C(N3CC(C(C)NC(c4ccc(C(N)=O)[nH]4)=O)C3)=O)C12 c1(N2CCC(NC(=O)CC3CC4(CC4)CO3)C2)cc(C(F)(F)F)nc2ncnn12 C(=O)(CCCCC(N)=O)N(C(C)CN(C)C(c1cc(-c2ccco2)c[nH]1)=O)C c1(C(N2CC3(C(C(=O)Nc4ccno4)C3)C2)=O)c(F)cncc1F C12(NC(C3C(=C)C3)=O)CC(CNC(c3cc(COC)[nH]n3)=O)(C1)OC2C CC1(C(=O)NCC(CO)NC(=O)C(C2CC2)C2CC2)CCC(F)(F)CC1 c1(NC(c2ccn(CCC)n2)=O)ccc(NC(C2COCCOC2)=O)cc1C c1(C(=O)NCC(C2CCOC2)NC(CCC=C)=O)ccccc1SC(F)F C(=O)(C(C)(C)CC(=O)N1CCCC(CNC(=O)CC2(C)CC2)C1)OCC CC1OCCCC1C(=O)NCCCN(C(=O)CCOC1CCCC1)C C12(NC(c3n(CC)c(O)nc3)=O)CCC(C1)N(C(=O)COC1CCC1)C2 CC(CC(=O)c1ccccc1F)C(=O)NC(C)CN(C(=O)Cc1c[nH]nc1O)C c1(C(=O)NC(CNC(C(C)SC)=O)C(C)C)ccccc1NS(=O)(=O)C1CC1 c1(C(=O)NC2CC(C)(NC(C(CCC)CC)=O)C2)ccc(OC)c(F)c1N c1(C(=O)NCC2CN(C(C3(CC(C)C)CC3)=O)C(C)C2)cc2n(n1)CCO2 CC(C)CC(CNC(C1(CCF)CCC1)=O)NC(C1CC1C(N)=O)=O C(=O)(CCCCCCNC(C)(C)C)NC1CCCC(C)O1.C12CC1OC(=O)N2 NS(=O)(=O)c1ccc(C(=O)NCC(CNC(=O)C2=CCCCO2)C(F)(F)F)o1 N1(C(C(C)OCCCC)=O)CCCC(C)(NC(c2ccc(=O)n(C)n2)=O)C1 C(=O)(C1CCCNc2ccccc21)NC(CNC(Cc1nnc(C)s1)=O)C c1(C(=O)NCC(CNC(=O)C=C2CCC2)O)n[nH]cc1C1CCC1 c1(C2(C(=O)NCCN3CC(NC(=O)CCC4CC4(F)F)C3)CC2)ccc(F)cc1Cl N1(C(CCC=C)=O)CC(C(=O)NC(C)CN2CCCC2)C2(CC2)C1 c1(C(=O)NC2CCC(N(C(C(C)SCC)=O)C)CC2)c(C)[nH]c2ccc(Cl)cc12 Cc1cc(C(N2CC=C(C(=O)Nc3cnn(C)c3)C2)=O)nnc1C N1(C(c2n(CC#C)ccc2)=O)C(C)CN(C(=O)C=C(Cl)Cl)CC1C N1(C(C2C(C)(C)CO2)=O)CC(CO)C2(C1)CN(C(c1cncc(Cl)c1Cl)=O)C2 c1(CC(C)(C)C)ccc(C(=O)NCCC(O)CNC(=O)C(CO)N(C)C)cc1 c1(C(=O)OC)nc(C(=O)NCCC(C)N(C)C(C2CC(CO)CO2)=O)cs1 C(=O)(C1=C2CCCN=C2NN1)NCC1(O)CCN(C(CN2CC(CC)C2)=O)C1 N1(C(c2cc(N)c(Cl)cc2)=O)CCOC2CC(c3nn[nH]n3)CCC12 c1(C(=O)NC(CCC)CNC(=O)C(CC)NC(N)=O)cc(C)n(C)c1C C=CC1(O)CCN(C(C2CCCN(C(c3cncc(OC)n3)=O)C2C)=O)C1 C1(NC(CCCC#C)c2nnnn2CC(F)F)C2CCC1CC(C(N)=O)C2 C1(N(C(C2C(C)CC2)=O)CCO)CCN(C(C2(N3CCCC3)CCC2)=O)CC1 c1(C(=O)NCCCOCCNC(C(C(CC)CC)C)=O)n[nH]c2nccc(Cl)c12 C=CCC(C)C(=O)NC12CC(CNC(c3ccccc3OC)=O)(C1)C2 c1(NC(c2cccc(CO)c2)=O)cncc(CO)c1.C12CC(C1)NC2=O C12(C(OC(C3C(C=C)CC3)=O)=CC)CC1CN(C(c1csc(-c3cnc[nH]3)n1)=O)C2 C1(COCCCCCC(=O)NCc2cncn2C2CC2)CCCCC1CC=O c1(OC)ccc(C(c2cn(CC(=O)NC(C3(O)CCC3)CC)nn2)C)cc1 N1(C(C(COC)C)=O)CCCC1(C)CNC(c1ccc[nH]1)=O c1(C(=O)NCC(C)CNC(c2csc(=N)[nH]2)=O)cccc(C(F)(F)F)c1 C(N=c1ncc(F)c[nH]1)C1CC(C)N(C(=O)CS(=O)(=O)N2CCOCC2)C1 C(=O)(CC1=CCCCC1)NCC(=O)NCC(CC(C)C)NC(C1(CF)CC1(F)F)=O C1(NC(CNC(COCCOCC)=O)=O)CN(C)CCC1O C1(NC(C23CC(SC)(OC2)C3)=O)CN(C(=O)CSC(C)C)CC1C1CC1 c1(OC)ccc(F)c(C(=O)NC2CC2NC(=O)C(O)CC2CC2)c1F Cc1cc(C(=O)NC(CC2CC2)CC(=O)NCCCCN2CCC2)c(C)o1 CC1(c2ccccc2)CN(C(c2nnc(C(F)(F)F)s2)=O)CCO1 N1(C(C(N2CCNC2=O)C)=O)CCC(CF)(NC(c2cncc(CO)c2)=O)C1 Cc1ccc2ncc(C(N3CC(F)(F)CC3CCNC(=O)C(O)C(F)F)=O)n2c1 C(=O)(CC(C)(C)CC(C)=O)N1C2CC(CN(C(c3c(Cl)cn(CC)n3)=O)C2)C1 c1(CNC(=O)CC2CCCC(NC(C3SCCS3)=O)C2)cc2n(n1)CCC2 c1(C(C(=O)NCCC2N(C(C(C)NC(C)=O)=O)CCC2)C)ccc(Cl)cc1 C1(C(=O)NCC(CNC(COCCOCC)=O)OC)CCOCC1(C)C c1(CN(c2cc(N(CCCCC=C)C)ncn2)C)c(C)nn(CC)c1C CC1(C)CCc2c(C(N3CCCC(CNC(=O)Cc4cscn4)C3)=O)n[nH]c2C1 C=CCC(C)(O)C(=O)N1CCC(C(F)(F)F)C(C(=O)OC(C)(C)C)C1 c1(C(=O)NC(COC)CNC(C2(C3CC3)CC2)=O)nnn(CCOC)c1C C1(C(=O)OC)(NCCN2CCP(C)(=O)CC2)CCCC(C)C1 N1(C(CC(C)C)=O)CCOCCC1C(=O)NCC(C)(O)C1CCC1 C(=O)(C1=CC2CCC=CCCC12)N1CC(Nc2nccc(C(C)(C)C)n2)C1 N1(C(C2OCCN(CC)C2)=O)CC(NC(C2(C)CC2Br)=O)Cc2ccccc21 C(CC(N)=O)(C(=O)NCC1CCC(CO)CC1)NC(C(CC)O)=O Cc1ccc(F)c(CC(=O)NCC2CCCCN2C(=O)Cc2ccn(C)n2)c1 C(=O)(C1=CS(=O)(=O)CCC1)N1CC(CNC(c2cc(CC)sn2)=O)CC12CCC2 N1(C(C)CC2CC2)CCC2(CC1)CC2(C)C(N1CCN(C2CCOCC2)CC1)=O c1(C(N(C2CCN(c3nc(C#N)c(Cl)s3)C2)CCC)=O)nn(C)cc1[N+](=O)[O-] c1(C(=O)NC2C3(CC(NC(C4CC(=C)C4)=O)C3)C2)c(F)ccc(Br)c1Cl c1(C(N2CC(SCc3cn(CCCN(C)C)nn3)C2)=O)ccncc1F C1(=O)C(F)CC(=O)N(CC)CCCN1.N1(C(=O)OC(C)(C)C)CCC1CC Cc1[nH]c(=NCc2cccc(O)n2)sc1C(=O)Nc1cccc(Br)n1 Cc1nsc(C(=O)NCC2COCCN2C(=O)CC(C)(C)C)c1N N1(C(COCCOC)=O)CCC(F)CC1C(N1CCSCC1C)=O C1(CC)CCCN(C(c2cnc(C)nc2C)=O)C1C(=O)NC(c1cnn(C)c1)C C1(C(N2C(C(=O)OC)CSC2c2cccc(Cl)c2)=O)CC(c2nn[nH]n2)CCO1 CCCC(CC)C(=O)N(C(C)CN(C)C(c1cc(=O)n(C)cn1)=O)C c1(NC(C(CC)(C)O)=O)ccc(NC(=O)CCCN2CCCC2)c(F)c1 c1(C(N2CCCC(N(C(=O)CC3CCC(=O)N3)CC)C2)=O)ccc(S(N)(=O)=O)s1 C1(C(=O)OC)C(CC)CCCN1C(=O)C=CCNC1CC1.C1CC(=O)N1 c1(C(=O)NCC2N(C(c3c(C)snc3)=O)CC(F)(F)C2)c(C)sc2ccccc12 Fc1ccc(C(c2nnnn2C2CC2)NCc2ncccn2)cc1Cl C(c1ccc2occc2c1)=CC(=O)NCC(CNC(C1C(C(C)C)C1)=O)(C)O Cc1cccc(C(=O)NCC(CC2CC2)C(=O)NC)c1N.C1(C)CCCS1 C1(C(=O)NCC2(O)CN(C(c3ccc(C#C)o3)=O)C2)CC(OC)C12CCC2 c1(C(N2CCCC(O)(CNC(CC(=O)NCC)=O)C2)=O)cn(C)c(=O)cc1OC c1(C(=O)Nc2c(CN(C(C)=O)C)cccc2)c(C)nn(C)c1Cl C1(CC)CN(C(c2cnc(O)cc2C)=O)CCC1NC(=O)CCc1ccco1 C(=O)(CCCC(C)(C)NC(c1ccc(C(N)=O)o1)=O)NCC(C(C)C)C Cc1cc(F)ccc1C(N1CCCC1)=O.c12ccc(cc1)C(=O)N(C)C2 CC(Cn1ccnc1)C(=O)NCC(F)CNC(c1ccn(C)n1)=O C(=O)(C(C)O)N(C(C)C)CCN(C(c1cccs1)=O)CC#N c1(C(=O)OC)ccc(N2CC3CC(OCc4ccccc4)C3C2)nc1C Cc1[nH]c(=N)sc1CC(N1CC=CC(NC(c2ccc(C(N)=O)[nH]2)=O)C1)=O CC1CC(C(N2CC(c3ccccc3)(NC(C3CC4CCC3C4)=O)C2)=O)CCO1 Cc1ccsc1CC(=O)NC(CN(C(=O)C=CCO)C)Cc1ccccc1 c1(C(COC)OC)cccc(CN(C)C(c2noc(C)n2)C)c1 c1(C(=O)OCC)cc(-c2sc(C(C)C)cc2-c2cnn3c2NCC3)no1 C1(C2CCCCC2)(C(N(C(CCNC(C(C(C)C)OC)=O)C)C)=O)CC1 c1(C(=O)NC2CCN(C(C3(OC)CCCSC3)=O)CC2F)csc2ccccc12 N1(C(C(C)(c2ccccc2)OC)=O)CCC2(CCC2)C(CNC(=O)CCCF)C1 c1(CC(=O)NC2C(CNC(CNC(CCC)=O)=O)CC2)c(CC)n[nH]c1CC C1(NC(c2c(C)cc[nH]2)=O)CCN(C(C2CCC(C(F)(F)F)CC2)=O)CC1C C1(CCC(=O)N(CC(CC)NC(c2c(CC)nns2)=O)CC)CCC(=O)NC1 c1(OC)ccnc(OC)c1C(=O)NC1CC2CC1N(C(=O)C(C#N)C(C)C)C2 CCC(C#N)(CC)C(=O)N1CC(NC(=O)C(C)Cc2ccncc2)C(O)C1 CCC(C(=O)NCCCN(C(c1sc(=N)[nH]c1C)=O)CC)C(C)O c1(C(=O)NC(C)C(=O)N(CCN=[N+]=[N-])CCO)cccc2ccnn12 c1(CCC(=O)NC2CN(C(c3nc(C)nn3C)=O)CC2O)nc2ccccc2[nH]1 c1(C(=O)NCC=CCNC(C(C2CC2)SC)=O)csc(=NC)[nH]1 C(=O)(C(F)n1ccnc1)NCC(=O)NCc1ncc[nH]1 N#Cc1ccc(CC(N2CC3CC3(CNC(=O)CC3NC(=O)NC3=O)C2)=O)cc1 C1(C(c2n(CC)nnn2)NCC2CC(CC(C)(C)C)C2)C(C)(C)C1(C)C c1(-n2ncc(C(N(CC(C)CNC(=O)CC(C)O)C)=O)c2)cccc(Cl)c1 N1(CC(c2ccc(C)cc2)NC(=O)OC(C)(C)C)CCOC(C)C1CO CCC(C)C(CC(=O)NCCS(=O)CC)NC(=O)C(CC1CC1)OC c1(C(=O)NCC(C2CC2)NC(C2CCC(C(N)=O)O2)=O)ccc([N+](=O)[O-])s1 C(=O)(C(C)(F)C(C)(C)F)NC1C(C)CCN(C(c2cc(N)c(F)cn2)=O)C1 N1(C(c2cc(OC(C)C)ncc2)=O)CC2(C1)SCCC2NC(=O)C(C)C1CCC1 Cn1nc(C(=O)NC2COCCC2NC(=O)Cn2cnnc2)cc1C(F)(F)F C=CCCC(C)(C)C(=O)NCC1CN(C(=O)CC2CCN(OC)CC2)CCO1 C1(C(C)C)CN(C(c2ccc(Br)cc2)=O)CCN1C(C12CC(C(=O)N(C)C)(C1)C2)=O C1(C(N(C2CC(C)(C)C2)C)=O)CC2(CC2)CN1C(=O)Cn1cccc1 Cc1nc(C2CCCCO2)sc1C(=O)NC1CC(C)(CNC(c2cc[nH]n2)=O)C1 CCCCCCC(CNC(c1ncoc1C(F)(F)F)c1nnnn1CCC1CC1)CC N1(C(CCCC(=C)C)=O)CCC2(CC1)CC2NC(=O)CCN(C)CCO c1(C(N2CCC(C)CC2CNC(C2CC2C#N)=O)=O)cc2c(nc1N)CCCC2 c1(C(N(CC(CNC(C(COC)(C)C)=O)C)C)=O)cc(OC)ccc1F c1(C(N2CCCN(C(C34CC(C)C3C4)=O)CC2)=O)ccc2nn[nH]c2c1 c1(CC)cc(C(=O)NC2CCN(C(C3(CC)CC=CCC3)=O)CC2O)ccc1F C1(C)(CNC(C(CCC)O)=O)CCN(c2nc(OC)ncc2Br)CC1 CC(C)C(CNC(c1occ2c1CCOC2)=O)N=c1[nH]nc(C(N)=O)s1 C1(CS(=O)(=O)N(CCN(C)CCO)CCO)CC(C)(C)CCO1 N1(C(C2C(=C)CC2)=O)CCC(c2cn(Cc3cc(-c4ccco4)on3)nn2)C1 C(C(CC(C)C)NC(c1c[nH]cc1Br)=O)NC(CCCOCC=C)=O O=C1CN(C(C2(CC(F)F)CC2)=O)c2ccccc2N1.c12ccc(cc1)CO2 c1(C(=O)NC(CNC(C(CCC)C)=O)C)cccc(C#N)n1 c1(C(N(CCCCC(=O)NCCC=CCCC)C)=O)c[n+]([O-])c(C)cn1 c1(-c2cncc(NC(c3cc(Cl)ncc3Cl)=O)c2)ccc2c(c1)C(=O)C(=O)N2 CC(C)CC(C)C(=O)NC(CNC(c1cccc(O)c1Cl)=O)CO c1(CN2C(C(N3CCOC4CC34)=O)CC(=C)C2)cnc(Cl)cc1OC C1(C(=O)NCCNC(C2CC(=O)N(CC(F)(F)F)C2)=O)CCC2(CCC2)CO1 C(=O)(C(C(C)O)NC(C1CCCN1CC1CCN(CCC)C1)=O)OC Cc1cn2c(n1)C(C)CC(C(=O)NCC1CN(C(C3OCCCO3)=O)CC1O)C2 c1(C(=O)NCC(=O)NCC(N2CCC(O)CC2)=O)ccc(F)c(Cl)c1 C(=O)(CCC(=O)NN(C)C)N1C(C)CN(C(c2cnc(CCCC)s2)=O)C(C)C1 Cc1nc(C)c(C(=O)NC(c2nc(C(F)(F)F)n[nH]2)C)c(C)n1 c1(C(=O)NCC(C2CCCC2)NC(c2c(CC)occ2)=O)ccn2ccnc2c1 C1(NC(=O)Cc2cscn2)CCCC(NC(c2ccc(-c3ccsc3)nc2)=O)C1 N1(C(CC2CCCN(C(c3cc(C)nn3C(C)(C)C)=O)C2)=O)CCN(C)C(O)C1 C12(NC(=O)CSC(F)F)COCCC1CN(C(=O)CCOc1cccnc1)C2 Cc1c(C(=O)NCCC(O)CNC(=O)CC2CCCOC2)sc2[nH]cnc(=O)c12 N1(C(C2CCC(C(F)F)CC2)=O)CCN(C(=O)CCc2cn[nH]c2)C(CCO)C1 C12(C(=O)NCCN(C(CCC3CC(C)C3)=O)C3CC3)CCCC(C1)OC2 CC(CC(=O)N1CC2C(C1)N2C(c1csc2ccc(Cl)cc12)=O)CC(C)(C)C C(C(CO)(CO)NC(CC=CCC)=O)N(C(=O)C(COC)OC)C c1(CCC)cnnc(C(N2CC(CC(C)(C)COC)C2)=O)c1.C12CC(C1)NC2=O c1(C(N(C(C)C)CCN(C(=O)C(c2ccccc2)F)C)=O)cncc(CO)c1 O=CC#CC1CCCC1.C(=O)(NOCCC1CC1)N(CC(F)F)C1(C)CC1 C(CCCC(=O)NCCCCC(=O)N(C)C(C)C)OC CC(C)(C)C(=O)NC1CC1C(=O)NCC1COC(=O)N1 c1(C(N2CCC(N(C(=O)C(F)C(C)C)CC(C)C)CC2)=O)cncc(Cl)c1C C(C(=O)N1CCC(C)C1C)(C(C)C)NC(CCCOC(C)=O)=O Cc1noc(C(N2CC(COC)CC2CNC(=O)CCCc2cnn[nH]2)=O)c1C C1(NC(CC2CC(=O)NC2=O)=O)CCN(C(c2cc3scnc3[nH]2)=O)CC1CO C(C1=NOC2CN(C(c3nocc3C(C)(C)C)=O)CC12)NC(COCCC=C)=O C(=O)(C(C)(C#N)CC)N1CCC(C(C(=O)NCC(C2CCC2)OCC)C)CC1 N1(C(Cc2cc(C)[nH]n2)=O)CCC(C(=O)NCc2nnnn2C)C(C)(C)C1 c1(C(=O)NC(C(C)(C)NC(CC(C)C2CC2)=O)C)ccc(=O)n(C)n1 C(=O)(CCCC(C)=O)NCC1(C(=O)NC(C)COC(F)(F)F)CC(=C)C1 N1(C(=O)C(c2ccccc2)n2ncnn2)CCCN(C(=O)CCCCCO)C(CO)C1 C(C(=O)NCC(O)C1CC1)(C(C)C)NC(C1(CC)CCCC1)=O c1(C(=O)NCC(CC(C)C)NC(Cc2cc(C)sc2)=O)c(C)nn(C)c1C C(=O)(CCCC(F)F)N(CCCOCCN(C(C1CC(C(=O)NC)C1)=O)C)C C1(NC(C2C(C)(CC)C2)=O)CC2(CCN(C(=O)CC3=CCCC3)CC2)C1 C1(CNC(C=CC=CC)=O)(CNC(=O)COCC2CCCO2)CCCCC1 N1(C(c2ccc(SC)cc2)=O)CCOC2CN(Cc3c(O)cccc3Br)CC12 N1(C(CC2N(C(CCC(CC)OC)=O)CCC2)=O)CCCNC(=O)C1C N1(C(C(C(C)C)CO)=O)CCC(C)N(C(c2ccc(-c3ccncc3)o2)=O)CC1 Cc1cc(C(N2CCCC(N(C)C(c3cc(Cl)no3)=O)C2)=O)c(Br)s1 N1(C(c2c(C)cco2)=O)CC(NC(C2CCC(N(C)C)CC2)=O)C2(CC2)C1 N1(C(C(C)S(C)(=O)=O)=O)CC2CCN(C(c3cc(Cl)c4ccccc4n3)=O)CC2C1 c1(CCC)cc(C(N2CCC(CNC(=O)C(C)COC(C)=O)C2)=O)n(C)n1 CC(C)CC(C(=O)NCC1(F)CC(NC(c2ncoc2Br)=O)C1)C(C)C C1(OC)(CNC(C2CCC2(F)F)=O)CCN(C(=O)CC(=O)NCC(F)(F)F)C1 N1(C(CC(C)OC)=O)CCC2(CC1)C(NC(=O)CC1(CO)CC1)CS(=O)(=O)N2C N1(C(COCCNC(c2c(CC)cncc2)=O)=O)CCCC2(CC1)CC2 c1(C(=O)NCC(C(C)C)NC(=O)C(C)C(C)(C)C)cnc(N)c([N+](=O)[O-])c1 CCC(CC(=O)NCCC1CN(C(c2nc[nH]c3ncnc2-3)=O)C1)CC(C)C C1(CCCCNC(c2c(C)occ2)=O)CCCN(C(=O)CC(C)N(C)C)C1 C(S(=O)(=O)CCCCc1ccccc1)c1ccc(OC(C)CC#N)o1 C1(C(N2CCC(F)(COC)C2)=O)Oc2ccccc2OC1Cn1cnnc1 N1(C(C2C(=C)CC2)=O)CC2(CCC2)CC1CNC(C12CCC(C1)OC2)=O C1(Cc2cn(CCN(C)C)nc2)C2CN(CC(O)CNC=O)CC12.C1(C)CC1 C(N=c1cccc(S(=O)(=O)N2CCC3CCCCC3C2)[nH]1)c1c(C)noc1C N1(C(C(CC)n2cccn2)=O)CCOCC(NC(C2CC(C)(F)C2)=O)C1 c1(OCC)n[nH]cc1C(=O)NC1(CCNC(=O)Cc2cnnn2C)CCC1 C(N=c1[nH]c(=NCc2nnc3c(=O)[nH]ccn23)[nH]c2c1CCC2)C1CCC(=C)CC1 c1(C(N2C(C(=O)NCc3ccc(F)cc3F)CC(O)C2)=O)c(Cl)cc(Br)cc1Cl C1(CCN(C(=O)Cn2cc[n+](C)c2)C)CCN(C(c2cncc(F)n2)=O)CC1 C(=O)(C1=CCN(C(C2(C(C)(C)O)CCC2)=O)CC1)NC(CCOC)C N1(C(C2CC3(CC(=C)C3)C2)=O)CCCN(C(=O)CCC2CCCOC2)CC1C C1(C(=O)O)CCN(Cc2cncc(F)c2Br)C(C2CC2)C1 C(=O)(C1CCCc2nncn21)N1CCN(CCN(C(=O)CCS(C)=O)C)CC1 c1(C(=O)NC2CCCN(C(CCCOCC=C)=O)C2)ccc(O)c(C(C)=O)c1 c1(CN2CCC(NC(c3ncsc3Br)=O)C2)ccc([N+](=O)[O-])cc1Br c1(C(=O)NC2CC(NC(CCOCCCOC)=O)C(O)C2)ccc2n[nH]cc2n1 N1(C(=O)NCc2cncs2)CCCC(F)(Cc2cc(N3CCC(F)CC3)cs2)C1 c1(C(N2CCN(C(CC3CN(C)C3)=O)C(CF)C2)=O)ccc(N)c(Cl)c1O C(=O)(CCCC(C)(F)F)N1CCC(NC(CCOc2c(OC)ccc(Cl)c2)=O)C1 CON(CCO)C(=O)C1CCC(NC(=O)C2=C(C)CC2)C1 C(=O)(C1CCCc2cncn21)N1CCC(N(C(C2(OC)CCCOC2)=O)C)CC1 Cc1n[nH]c(C)c1C(C)C(=O)N(C(CNC(c1cncc(Br)c1)=O)C1CC1)C Cc1ccc(S(=O)(=O)NC(=O)CCc2ccccc2N)cc1C C1(C#CC(=O)NCC2CCCC2NC(=O)CC2(C)CCOCC2)(CC)CC1 C=CCC(C(=O)N1CC(C)(NC(c2nn3cc(C)nc3s2)=O)C1)C(C)C C1(C(C)C)CN(C(C2CCC(N(C)C)CC2)=O)CCN1C(=O)C(=O)N(C)C C1(NC(C2CC(C)C2)=O)CC2(CCCN(C(=O)CNc3cccnc3)C2)C1 C(=O)(C(CNC(C1CC(F)(CF)C1)=O)C(C)(C)C)NCc1n(C)cnc1 c1(C(=O)NCC2CC3CCC2N3c2ncncc2I)ccc2ncccc2n1 N1(C(C2CCCCC(=O)N2)=O)CC2CCCN(C(=O)C(F)=CC3CC3)C2C1 CC1CCC(NC(c2ccc(C(F)(F)F)[nH]2)=O)CN1C(c1ncc(Cl)nc1Cl)=O c1(CCC(=O)NC2CCC(CNC(C)=O)C2)c(C(=O)OCC)nc2n1CCC2 Cc1c(C(=O)NC2(CC(N3CCC(C(=O)N(C)C)C3)=O)CC2)ncn1C c1(C(=O)NCc2ccc(C(=O)NCC(C)C(C)(C)C)o2)ccn2cncc2c1 CCCCCCC(CC)NC(=O)CC1CC(F)CN1C(C1(C)CC2CCC1C2)=O CCC(CC(=O)N1CC2CC2(CNC(=O)CCOCCCCN)C1)SC C1(SCC(=O)OC(C)(C)C)CN(C(=O)OCc2ccc(C)c(Cl)c2)CCC1(F)F c1(C(=O)NCC2(NC(c3cc(C(F)(F)F)cc(F)c3)=O)CC2)cc2cccn2cn1 Cc1cc(C(=O)NCCC(C)N(C(=O)C(n2ccc(C3CC3)n2)C)C)ccc1Cl C12Cc3ccccc3N1C2=O.N1(c2ncc(C(=O)OCC)cn2)CCN(C#N)CC1 n1(CC)ncc(C(=O)NC(Cn2cncn2)C(=O)OC)c1Cl C(C)(N(C)N1CCC2(CCC(O)CC2)C1)c1cccc(OC)c1 CN1CCOCC1C(N1CCCC1(C)C(=O)NC1CCCC1C#N)=O C1(NC(Cc2ccc(C)s2)=O)CC2CCC(C1)N2C(=O)COC1CCOCC1 C1(CC(=O)NCc2c(CC)scn2)CN(C(=O)CCc2cnn[nH]2)CCC1C C1(CCNC(c2c(CC)nc[nH]2)=O)CCCCN1C(=O)CCOCCN(C)C Cc1ccc(C(N2CC(NC(=O)Cc3sc(O)nc3O)C(C)C2)=O)c(O)c1 N1(C(C(C=CC)O)=O)CCN(C(c2cccc(F)c2Cl)=O)C(CC)C1 Cc1ccnc2c(C(=O)NCCN(C(c3ccn(C(C)C)n3)=O)C(C)C)cnn12 C(C(C)N=c1[nH]nc(C(N)=O)s1)(c1cccs1)NC(C(C)N(C)C1CC1)=O N1(C(C)CNC(c2ccoc2Cl)=O)CCN(C(=O)CCC2CCOC2)CC1 c1(C(C)C)ncc(C(=O)NC(C)CC2CN(C(=O)CC(=O)N(C)C)C2)s1 C(=O)(C(CNC(c1ccc(CC)nn1)=O)CC1CCCC1)OCC CC1CCC(CNC(=O)CSc2cccc[n+]2[O-])N(C(=O)C=CC2CCCC2)C1 C1(C(N2CCCC(CN(C(c3cc(C)sc3)=O)C)C2)=O)CC12CCOCC2 c1(N(C(CC)C)C)cc(NCc2ccc(O)c(Cl)c2)nc(C(F)(F)F)n1 CCCC(CCC)C(=O)NCC1(CNC(C2CCN(C3CCSC3)CC2)=O)CC1 C(=O)(C(CC(C)C)N(C(=O)COC)C)NCCCNC(CC)=O c1(N2CCC(C)(NC(C(CCC)NC(N)=O)=O)CC2)ccc([N+](=O)[O-])c(SC)n1 Nc1cc2c(cc1C(N1CCC3CN(C(C4CCCOC4)=O)C3C1)=O)CCC2 C1(C2CCCC2)(C(=O)NC(C(C)(C)O)CS(C)(=O)=O)CCNC1=O N1(C(c2oc(CC)c(C)c2)=O)CC(NC(=O)C(COC)OC)CC12CCC2 CCCCCC(=O)N1CCC(CCOC)(NC(=O)CCCn2ccccc2=O)C1 c1(OC)c(C(=O)N(C2CC2)Cc2cccc(F)c2)ccc(I)c1F c1(CCNC(=O)Nc2ccc(NC(C)=O)cc2)c(C)cnnc1O O(NC(=O)C(O)CCCNC(c1ccoc1C(C)C)=O)C(C(=O)OC)(C)C c1(C(CC)C(=O)N(CC(O)CN(C)C(C2CCCC2CC)=O)C)cccc(Cl)c1 C#CCCC(C(=O)NCC1CC2CCC(C1)C2)NC(c1cc(C)[nH]n1)=O N1(C(C(CCCCC)F)=O)C2CCCC1CN(C(=O)C(c1ccccc1)=O)C2 c1(C(N2C(CNC(C(CC)c3ccccc3)=O)CCC2)=O)ccc2ccccc2n1 C(C(C)(C)CC(=O)NC1(CCCCO)CC1)NC(C1N(CC)CCOC1)=O c1(CC(C(=O)NC2CC(OC)C2)NC(=O)C(C)C(C)C)cnn(C)c1O c1(C(=O)NC(CN(CCOCC)C)C)ccccc1OCc1ccc(Cl)cc1 c1(OC)nc(C(N2CCCC(F)(CNC(C34CC5CC3C4C5O)=O)C2)=O)cc(C)n1 Cn1ccc2cc(C(=O)NCCC3CCCN(C(=O)COC(F)F)C3)cnc12 C#CC1(NC(C2CC2CNC(=O)CC2CC(C)(C)CO2)=O)CCOC1 C1(C)(C(=O)OC(C)(C)C)CC12CCN(C(=O)Cc1ccccc1O)CC2 C(=O)(CC(C)(C)CN(C)C)NCCC1CCCN(C(C2(CC)C=CCC2)=O)C1 NC1CCc2cc(-c3ccc(NC(=O)C(F)(F)F)cc3)ccc2C1.C1CC(=O)N1 c1(C(=O)NCC(C)N(C(c2c(C)[nH]cc2)=O)C)ccc([N+](=O)[O-])c(N(C)C)c1 C(=O)(CC1NC(=O)c2ccccc21)NCCN(C(=O)Cc1ccn(C)n1)CC Cc1cccc2c(C(c3ccc(Cl)cc3)NC(C3(c4nn[nH]n4)CC3)=O)coc12 Cc1ccc(C(=O)NC2CCCC2NC(C2(C)COC(=O)OC2)=O)cc1Cl N1(C(CSCCCC)=O)CC(C)(CNC(=O)COc2cc(C)on2)CC1(C)C CCC(C)C(O)CC(=O)NC(CNC(C1(C2(O)CCC2)CC1)=O)C1CC1 C(=O)(CC(C)(C(F)(F)F)NC(C)=O)NC(CCCC)COC CC1CCN(C(c2nc(Cl)cs2)C(=O)NCC(F)F)CC1NC(=O)OC(C)(C)C c1(CC(=O)NC2CC3CN(C(=O)CC(C4CC4)C4CC4)CC23)cc2ccccc2s1 C(=O)(C(C)(O)C(C)C)N(CCOC)CCNC(=O)C(c1cccc(C)c1F)O c1(C(N(CC(C(=O)NCCCOCC)OC)C)=O)ccc(CC2CC2)nc1 N1(C(COCCC)=O)CCOCC(CNC(=O)CC2CCC(C)(C)CO2)C1 N1(C(CC(C)(O)c2ccc(Cl)cc2)=O)CCC(NC(=O)C=C(Cl)Cl)C(CO)CC1 c1(C(N2CC(OC)C(NC(c3ccc(C(F)(F)F)o3)=O)C2)=O)ccc(N)c(F)n1 C(=O)(CCCC1CC1)NC1(CC(=O)NC2CN(CCN(C)C)C2)CCC1 C1(C(=O)NCC(CN(C)C(C2(F)CC2C2CCCCC2)=O)O)(CF)CCOCC1 CCCC(CNC(=O)C(c1ccoc1)OC)NC(c1c[nH]nc1C(F)F)=O C(=O)(C1=NOC(C)C1)N1CCC(OC)(CNC(=O)CC2(OC)CCCCC2)C1 N1(C(C2(N=[N+]=[N-])CCN(C(C(CCC)F)=O)C2)=O)CCCC2(CC(O)C2)C1 c1(OC)cc(C(=O)NCC2CCCN2C(c2c[nH]c(C)c2)=O)c(C)cc1[N+](=O)[O-] C1(C(N2C3CN(C(N)=O)C(CC3)C2)=O)CCc2nccn2CC1 c1(C(=O)NCCC2N(C(C(C)=CC)=O)CCC2)cccc(OC)c1O N1(C(C2(CO)CCCCC2)=O)CCC(F)(C(N2CCC(F)(CO)C2)=O)CC1 c1(C(N2CCCC(NC(C3CC(=C)C3)=O)C2C)=O)cccc(SC)c1[N+](=O)[O-] CC(C)(CCCCNC(=O)C(O)Cc1ccccc1)C(=O)NNC(=O)C(C)(C)O Cc1ccc(C(=O)NCC23CC(NC(C4OCCOC4C)=O)(C2)C3)cc1C C(=O)(C(CC(F)F)NC(C1CC(C)(C)CO1)=O)NCc1cc(C)ns1 C1(NC(CC2CC(NC(CC3(OCC)CC3)=O)C2)=O)CCC2(CCC2)C1 C=CCCCCCCC(=O)N1CC(OCCNC(c2n[nH]c3ncccc23)=O)C1 N1(C(C(C)C)=O)CCCN(C(=O)CCc2nnc(S)nc2O)CC1C(C)C C1(NC(c2cn[nH]c2)=O)C2CCC1N(C(=O)CCc1ccncn1)C2 O=C(CC1=CCCCC1)NC1CCN(C(=O)Cn2nnnc2C2CC2)CC1F C1(CNC(C2=C(C)OCC2)=O)CN(C(C2CC3CCCN(C2)C3)=O)CC(C)(C)O1 n1(CCCN(C)C)cc(CCNC(C2(F)CCCC2)=O)nn1.n12cc(nn1)C2 c1(C(N(C2CCN(C(c3cnc[nH]3)=O)C2)CCC)=O)cnc(NC)cn1 c1(C(N2CC3C(NC(=O)Cc4c[nH]nc4O)(C3)C2)=O)cc2ccnc(Cl)c2[nH]1 N1(CCNC(c2c(CC)nns2)=O)CCN(C(C2CCC23CC3)=O)CC12CCC2 O=C1CC2CC(C(N3CC(O)(c4cccnc4)C3)=O)C1O2 Cc1cc(C(=O)NCC2(CNC(=O)C(C)Cc3cccnc3)CCCC2)oc1C N1(C(c2cn(C(C)C)nc2)=O)CC(CNC(c2ccn(C)n2)=O)C(F)(CO)C1 C1(CNC(C(C)n2cncn2)=O)CC2CCC1N2C(c1ccc(=O)n(C)n1)=O c1(C(C)OC(C2CCCC(n3ccnc3)C2)=O)ccc(C#N)cc1F C1(NC(c2c(OCC)oc(C)n2)=O)CN(C(=O)C(C)(O)CC)CC1S(C)(=O)=O C1(C)(C(N2CCC(N(C(Cn3c(CCC)ncc3)=O)CC)C2)=O)CC(C)(C)C1 c1(NC(C=CCNC(C(C=CC)O)=O)=O)cnn2c1OCCC2 C1(OCCCC)CCOCC1NC(C1(C(=O)NCC)CC1)=O c1(CC)cnc(OC(C)(C)CN(CC(=O)NC(C)C)C)nc1 c1(CC)nc(C(C)NC(C2CCS2(=O)=O)=O)no1 c1(COC)cc(=NCC2CCC(NC(=O)CCCC3CCCCC3)C2)[nH]cn1 CCCC(C)(C)CC(=O)NCC(CNC(C12CCCC1C2(F)F)=O)S(C)(=O)=O CCC(CC)C(C(=O)N1CCCOC(CNC(C2(C)CC2)=O)C1)OC C1(NC(COCc2n(C)ncn2)=O)CC2CCC1N2C(=O)CC1CC1C1CC1 CN1CC(C)(C)CC1C(=O)NC1CCCCN(C(C2(C)CCC(=O)N2)=O)C1 c1(C(N2CCC(C)C2CNC(C2CCC(O)C2)=O)=O)cccc(C#N)c1 C(=O)(C(C(=O)N1CCC(NC(=O)CCCOc2ccccc2)C1)C(C)(C)C)OCC N1(C(COCCC)=O)CC2CCC1C1CN(C(c3csc(C)n3)=O)CC21 c1(OC)ccc(C=CC(=O)NCC2CC(NC(c3csc(CO)n3)=O)C2(C)C)nc1 CCCCCC(C)CC(=O)N1CC(C(O)C(=O)NCC2CCC(=O)NC2)C1 CN1CC(NC(c2ccc(CNC(c3cccnc3C3CC3)=O)cn2)=O)C(=O)N1 c1(C(=O)NCC(C)(C(C)C)NC(CCC(C)SC)=O)cc2ccccc2nc1C C1(OCCC(=O)NCCCCC)(OCCNC(c2ccsc2)=O)CCOCC1 C1(OC)CCCCC(CNC(c2sccc2CNC(=O)OC(C)(C)C)=O)C1 CC1CCN(C(=O)CCCc2nccs2)C(CNC(=O)CC2CCC(=O)NC2)C1 c1(NC)ccccc1C(=O)NCCC1CC(C(=O)Nc2ccsc2C(N)=O)C1 N1(C(CSCC#C)=O)CCC(NC(=O)CN2CCn3ccnc3C2)CC(O)C1 CC(CCCCCO)NC(=O)C(C1CCCO1)NC(=O)CCc1ccccc1 c1(CC)nc(C)c(C(N2CC(CNC(c3c(Cl)cnn3C(C)C)=O)CC2C)=O)s1 Cn1cccc(C(=O)NCC2CCCCN2c2nnc(-c3ccccc3)o2)c1=O CC1C2C(CCN2C(=O)CC2(O)CCCC2)CN1C(c1csc(S(C)(=O)=O)c1)=O C1(C(N2CC(C3(NC(C4CSC4)=O)CC3)C2)=O)CCOC2(CCCC2)C1 CC1CN(C)CCN1N1CCN(C(=O)CCCCCS(N)(=O)=O)CC1=O C(=O)(C1CCCc2ncccc21)NC(CC)(CNC(C1NC(=O)CC1C)=O)CC Cn1cnc2c1CCC(C(N1CC(NC(C3CCCC(=O)N3)=O)C(O)C1)=O)C2 Cc1cc(=NCCC=CBr)[nH]cc1S(=O)(=O)NC(C1CCCO1)CO C1(C(N(c2nc(CC)cc(C)n2)CCC)=O)CC12CCc1ccccc12 c1(CNC(N2CCC(F)(F)C(Nc3ncc(Br)s3)C2)=O)ccccc1[N+](=O)[O-] c1(CC(=O)N(CCC(C)NC(c2c(SC)cccc2)=O)C)cc(F)cc(F)c1 c1(-c2ccc(CNCc3cc(OC)cc(O)c3)cn2)ccc(C)c(Br)c1C c1(-n2c(NC(=O)NC)nc(-c3ccc(Cl)s3)n2)ccc2nccnc2c1 S(=O)(=O)(c1ccc(C(=O)NCC(CNC(=O)C=Cc2c[nH]cn2)OC)cc1)NC C(=O)(C1=C(Cl)CCOC1)NC(C)(C)C(=O)Nc1cc(Br)ccc1F c1(C(N(c2cc(N(C)C)ncn2)C2CC(N)C2)=O)ccc2nn(C)cc2c1 Cc1c(C(C(=O)NCCC2(C)CC2)N(C2CC2)Cc2ccccc2)n[nH]c1C1CC1 Cc1ccc(C(N2CCN(CC3(NC(c4cc(C#N)c[nH]4)=O)CC3)CC2)=O)cn1 C12(CNC(CSCC=C)=O)CCC1CCN2C(c1cccc(NC(C)=O)c1O)=O C(CCC1C(=O)NC2(CC(=O)N1)CC2)OC.C1(CNC(C)=O)CC(O)C12CCC2 Cc1cc(=O)n(C)cc1C(=O)NCC(O)CNC(c1cn(CCO)nn1)=O c1(COC)ocnc1CNC(=O)CN(C)C(C1CCC(Oc2ccncc2)C1)=O C1(NC(CSC(C)(C)C)=O)C2COCC1CC(NC(C1(C(C)(F)F)CC1)=O)C2 N1(C2CCN(CC)C2=O)CCC2(CCN(C(C3(N4CCOC4=O)CC3)=O)C2)C1 N1(C(C2OCCN(CC)C2)=O)CCN(C(c2ccn(C(C)(C)C)n2)=O)C(CO)C1 CC1CCC(CNC(c2ccc(C(F)F)nc2)=O)N(C(c2c[nH]c(=N)o2)=O)C1 c1(C(=O)NC2CC(C(C)NC(Cc3cc(C)[nH]n3)=O)C2)ccccc1Br c1(CN(CC(CC)NC(C2CCN(C)S2(=O)=O)=O)C)cc2c(cc1OC)OCO2 C(CN=c1[nH]nc(C2CC2)o1)(CC(C)C)NC(C1CCN(C(C)=O)CC1)=O C1(N(C(c2c(C)snn2)=O)C)CN(C(c2cnn(-c3ccccc3)n2)=O)CC1O c1(OCC)nc(Cl)ccc1C(N1CCC1CNC(=O)CC1CCC1(C)C)=O c1(C(N2CCC(CC=C)(NC(=O)CCC(=C)Cl)C2)=O)cc2c(O)cccc2[nH]1 c1(NCC(CC)N(C)C)nc(=NC2CCC3CC2C3(C)C)[nH]c2c(C)nn(C)c12 c1(C(=O)NCC2CN(C(C3C(C#C)C3)=O)CC2C)nn(CC)cc1[N+](=O)[O-] N1(C(C(CC)SC)=O)CCC2C(CCCN2c2cc(CC)nc(CC)n2)C1 c1(C(N(CCN(C)CCF)C)=O)cc(C)cc(Br)c1 N1(C(COC2(C)CC=CC2)=O)CCCC(NC(C2CCC23CCC3)=O)CC1 CC(O)(CNC(=O)CCCC1CC1)CNC(C1CCCCC1)=O Cc1nnc2n1C(C(=O)NC(C)CCNC(c1cccc3c1CCCC3)=O)CC2 C1(NC(=O)CC2C(c3cn(C)nc3)C2)(CO)CCN(C(=O)C=Cc2ccco2)C1 C1(NC(c2c[nH]c(=N)o2)=O)CC2(NC(C3C4CCC(=O)C34)=O)COC1C2 C#CC(CNC(=O)CCN(CCCCC)CCOC)C(C)C.C12CCCN1C2 CC1(C)CC2(CC(CS(=O)(=O)NNC(N3CCCN(C(=O)C4CC4)CC3CO)=O)C2)C1 C12(CNS(N(OC)C)(=O)=O)CCCCC1N(CCc1cccc(Br)c1F)CCC2 c1(C(=O)NCC2CCCN(CC3CCCO3)C2)cc(F)c2nc(O)ccc2c1 C1(CCC(=O)N(CC(N)=O)CC(N)=O)CCN(C(=O)C(c2ccc(F)cc2)F)CC1 C(CC)(C(=O)NC1(CNC(c2cc(CSC3CCCO3)on2)=O)CC(OC)C1)CC C1(NC(c2ccncc2O)=O)CC(F)CN(C(c2ccc(OCCO)nc2)=O)C1 N1(C(c2c(CC)c(C)sc2)=O)CC2C3CCC(C2C1)N(C(=O)C(F)(F)C1CC1)C3 n1(CC(N2CCC3(C(NC(C(C)C(C)(C)C)=O)C3)C2)=O)cc2ccccc2n1 N1(c2cccc(S(=O)(=O)NCCN(OC)C)n2)CCc2ccc(C#N)cc2C1 c1(C(=O)NC2C(NC(C3(C)CCOC3)=O)CCC2)c[nH]c2cnccc12 N1(C(CC(n2ccc(C)n2)C)=O)CCC(C)(C)C1CNC(=O)CC1CCOC1 Cc1nc(C)c(CC(N2CCCC(C)(NC(=O)C(C)c3ccsc3)C2)=O)c(O)n1 c1(C(=O)NCCNC(C(CC(=C)C)C)=O)cc2c(Br)cccc2s1 C1(C(N2C(C(N(C)C)=O)CC2)=O)C=CCN(C(c2cc[nH]c2)=O)C1 c1(C(N(C(C)CNC(c2nc(Cl)oc2C)=O)CC)=O)ccc(F)c(C#N)c1 C(=O)(C1CCSc2ccccc21)NCC1(NC(C(C(C)(C)O)F)=O)CCOCC1 c1(C(=O)NC2CCC(F)(CNC(C(C)NC(C)=O)=O)C2)ccc(Br)c(N)c1 C1(CNC(=O)CC2CCOC2=O)CC(NC(=O)C(F)(F)C(F)F)C12CCC2 Cc1nccc(CCC(=O)NCCC2CC(NC(=O)CCCN(C)C)C2)n1 N1(C(C2C(OC)CN(C(CCCCCC)=O)C2)=O)CCCC(C2(C)CC2)C1 c1(C(N2CC(CC=C)(NC(=O)CCN3CCC(F)C3)C2)=O)coc2c1CS(=O)(=O)C2 n1(CC)c(C)cc2c1CCCC2NC(=O)Cc1c(C)oc(C)c1S(N)(=O)=O C1(C(=O)NC2C(C)CCN(c3nc(C)cc(OC)n3)C2)Cc2ccccc2C1 c1(C(N2CCCC(N(C)C(C3CC(=O)CCO3)=O)C2)=O)[nH]nc2ncccc12 c1(CCC(=O)NC(C)CCCCNC(C2OCCCO2)=O)nnc(O)nc1O C(=O)(C1CCc2c[nH]nc21)NCCCCNC(c1cncc(OC)c1)=O c12cccc(c1)NC2=O.C1(CNCCC(=O)NC2CC2)C2COCC12 C12(CNC(C3CCN3C(=O)COC3CC=CC3)=O)CCC(CC1F)C2 C1(C(N2C(CC)COCC2)=O)CC(C)(C)CCN1C(=O)Cn1ncccc1=O C1(COC)(NC(=O)CCC2CC2(C)C)CCN(C(C2C(C)OC(C)C2C)=O)CC1 C(=O)(C1Cc2ccccc21)NC1C(NC(Cc2cnc(C)s2)=O)CC1 C(=O)(CCCC(F)(F)C(F)(F)F)NC1COCCN(C(C(C(C)C)C#N)=O)C1 c1(C(N2CCOCC(NC(C(C)S(C)(=O)=O)=O)C2)=O)coc2c1CCCC2 C1(C(N2C(C)CC(NC(COC(C)C)=O)C2)=O)CCCCC1(F)F C#Cc1ccc(C(=O)NCCC2CCCCN2C(C2CC(SC)C2)=O)cc1C C12(CNC(C(F)=C(C)C)=O)CCC1CN(C(C1(c3cccs3)CC1)=O)C2 c1(CC)cnc(C(=O)NC(CNC(c2cc(COC)nn2C)=O)C2CCC2)cn1 C1(C(=O)NC(CC(C)(C)OC)C)CN(C(C2CC2Cl)=O)CC12CCC2 CC(CNC(=O)CC1(C#N)CC1)(C1CC1)NC(=O)CNC(=O)OC1CCC1 c1(NC(c2cscn2)C)[nH]c(=NC2CCCC(O)C2)nc2c1cnn2C C1(C)(CNNCc2cc(NC(CCCC=C)=O)ncn2)CCC(OC)CC1 C1(C(=O)NC2(C3N(C(C(C)CF)=O)CCC3)CC2)CCS(=O)(=O)C(C)C1 C#Cc1ccc(C2CCCN2C(C)=O)nc1.C1(C)(Cc2ccccc2)C(=O)N1 c12cnc(nc1C(F)(F)F)C(=O)NCC(CO)NC2=O.c1(CO)ccsc1C1CC1 C(=O)(C(C)(C)C#N)N(C(C(C)CSc1ccccc1)=O)C1(C=O)CCC1.C1(N)CC1 C(CCCN=[N+]=[N-])NC(COCCN(C(C1C(CC)C1)=O)C)=O C1(CC(N2C(C=C)CC2)=O)CC(C)(C)CN1C(=O)CS(=O)(=O)NC c1(OC)cc(C(c2nnnn2C)NCCc2ccncc2F)ncc1C O=C(N=c1cccn[nH]1)C1CC(O)CN(Cc2ccnc(-c3ccncc3)c2)C1 C1(C(N2CCCN(C(=O)NCC3CCC3CO)CC2)=O)COc2ccccc2O1 CCC1=NOC(CC(=O)N(CC(C)NC(=O)C=C(C)c2ccco2)CC)C1 C1(C(=O)NCC(CCC)NC(=O)Cc2cc(C)sc2C)CCc2nc(C)[nH]c2C1 C1(c2nnnn2C2COC2)(NCCCC(C)(C)F)CN2CCC1C2 C(=O)(C1=CCC2CCC1N2C(C1(C)CC1)=O)N1CCCC(COCC)C1.C(CF)O C1(C)(NCCC(C)CCCCl)C(C)(C)C1(C)C C1(C2(NC(c3cccc(F)n3)=O)CC2)CCCCN1C(C1CCC=CCC1)=O CC(C)(F)C(C)(F)C(=O)NCC(=C1CN(C(=O)Cc2cnc3cccnn23)C1)F N(C1CCCc2c1n[nH]c2C)C(c1cc(C)n(C)n1)c1nnnn1C CC1COCCCN1C(=O)C(CC(N)=O)NC(=O)Cc1ccon1 C(N=c1[nH]c(=NC2CC(N(C)C)C2)[nH]c2ccsc12)c1c(Br)cn(CC)n1 C=CCC(CNC(=O)CSc1n[nH]c(O)n1)NC(=O)CC1CCC(C)O1 N1(C(C2(COC)CC=CC2)=O)CC(N(C)C(C2CCCO2)=O)C(C)(C)C1 c1(C(N2C(C)CN(C(C3(C)CC3Br)=O)CC2)=O)ccc2ncsc2c1 N1(C(c2cn(C(C)C)nn2)=O)CCOCC(NC(C2(CCF)CCC2)=O)C1 S(=O)(=O)(c1csc(C(=O)NC(C(C)NC(C23CCC(CC2)C3)=O)C(C)C)c1)NC N1(C(C=C(C)C)=O)CCCC(C(C)(C)C(=O)N(CCCCN(C)C(C)C)C)C1 C1(NC(C(=O)NCC)=O)COC2C(NC(C3CNC(=O)N3)=O)COC12 c1(C(=O)Nc2c(-c3ccc(N(C)C)s3)nccc2)cc2cccnc2cn1 c1(C(=O)NC(C)CN(C(=O)CCc2nccs2)C)sccc1S(N)(=O)=O N1(C(c2c(CC)cco2)=O)CC2CCCC(NC(=O)CNc3nccs3)(C2)C1 c1(CC)c(C(=O)NCC2CC2C(=O)N(CCCO)CC)cccc1C N1(C(COC(CC)(C)C)=O)CC(OC)CC1C(=O)NCc1cccc(=O)o1 C1(C(N2CC(CNC(C3C(OC)CCC3)=O)C2)=O)(CO)CCOCC1 c1(C(N2CC(NC(c3n(CCOC)ncc3)=O)C(O)C2)=O)cc(O)ccc1C c1(C(CC)O)nc(-c2nnn(C(C)(C)C)n2)n(C2CC2C)n1 c1(OC)cc(CC(=O)N(C)CCN(C(=O)C(C)(C)CF)C)cc(F)c1 c1(CCNC(CC(C)C)CNC(=O)OC(C)(C)C)ccc(F)cc1F S(=O)(=O)(c1ccc(NC)cc1)N(CC#CC1CCCCO1)C.C1CC1 C(=O)(C(C)C(F)(F)C(F)F)N(CC(C)NC(=O)CCc1nc(C(C)(C)C)no1)C c1(SC)cc(C(=O)NC2CC(CNC(c3[nH]cnc3C)=O)C2(C)C)c(C)o1 C1(CC(N2CCC(C(F)(F)F)C2)=O)CC(O)CN1C(C1CCCCC1)=O Cc1nnc(NC(c2cnn(C3CCOC3)c2)c2nnnn2CC2CCCO2)s1 C1(CNC(N(CCCC2CCCO2)C)=O)CC(C(=O)OC(C)(C)C)C(O)C1 c1(CC(N2CC(NC(C3CCC(C(=O)OC)C3)=O)(CO)C2)=O)cc(C)nn1C c1(C(N2C(C)CC(CNC(C(CC#C)CC#C)=O)C2)=O)cnc2cnccc2c1 c1(SCC)cccc2[nH]ccc12.Nc1cncc(Cl)c1C(N1CC2CC1CC2C)=O C1(C)(C(=O)NCC2C(C)CN(c3ncns3)CC2)CCCNS1(=O)=O N1(C(C2(CC#C)CC2)=O)CCC(N(C)C(C2CC2C2CC2)=O)CC1 c1(CC(=O)NCC23C(CN(C(C(C(C)C)C)=O)C2)C3)ccc(C#N)cc1F c1(C(CCC)NC(C)CCOC(C)=O)nnnn1C(C)(C)C C=CC(C)CC(=O)NC(CCOC)C(=O)N(C)CC NS(=O)(=O)C1(C(=O)NCC2(F)CCC(NC(C3CCNC3=O)=O)C2)CCCC1 N1(C(C(CC)CC)=O)CC2CN(C(c3cc(C(=O)OC)ccc3Cl)=O)CC2C1 C(=O)(C1=C(Cl)CCOC1)N1CC(CCNC(c2ccc(F)s2)=O)OCC1 C(=O)(C1=CNC2=NCCC2=C1)NCC(C)NC(C1C(CCC)CCC1)=O C1(NCc2cc(Br)c[nH]2)CC2CN(C(=O)C(n3ccc(-c4cccs4)n3)C)CC2C1 C(=O)(C(C)(C)C(C)O)NCC1(OC)CN(C(=O)C(C)CN2CCOCC2)C1 Cn1c(N(CC(=O)O)CCN2CCC(OCC(F)(F)F)CC2)cnc1S c1(C(=O)NC(CNC(CC2(C=C)CCC2)=O)C(C)C)ccc(O)nc1Cl C=CC(CCC)CC(=O)NC(C(=O)NCC1([Si](C)(C)C)CC1)C1CCCC1 C1(C(N2CCC(CCNC(c3cnco3)=O)C2)=O)CC2CCC(C1)S2 c1(C(N2C(C(C)NC(CC)=O)CCC2)=O)cnc2ccncc2c1 CCCC(O)C(=O)N1CCC(CCN(C(=O)CCc2c(C)noc2C)CC)CC1 N1(C(=O)OC(C)(C)C)CCC(NC(=O)CC2CC2(C)C)C(O)C1 C(CCC(C)C(=O)NC1CC(NC(c2ncoc2C)=O)C1)OC C1(C(N2CC(C=C)(CC(N3C4COCC3C4)=O)C2)=O)C2CCC(F)(F)C12 N1(CC(=O)N(CCC(=O)NCC2(O)CSC2)CCO)C(=O)CNC1=O CN1CCCC(C(c2nnnn2C2CCC2)NC2CC2)C1c1cccc(Cl)c1 c1(C(=O)NCC(CC=C)NC(=O)C(F)(F)CC2CCCO2)cn(C)nc1C C1(C(=O)NCCc2c(C)nc[nH]2)C=CCN(C(c2nocc2Cl)=O)C1 Nc1ncnc2c1ncn2CCNC(c1ccccc1-c1ccc(F)cc1)=O C(CC1=CCN(C(=O)CN2CCOCC2)CC1)NC(=O)CC(C1CC1)C1CC1 c1(OCC(=O)N(CC(C)NC(C(C)OCC#C)=O)CC)cccc(Br)c1 c1(C(N(CCC(C)NC(=O)CCN(S(C)(=O)=O)C)C)=O)coc(C(F)F)c1 c1(C(=O)NC2C3(CC(NC(C(C)NC(C)=O)=O)C3)C2)cncc2c(O)nccc12 S(=O)(=O)(c1ccc(Cl)nc1)N1C(CC)CN(C(=O)C(c2ccc(O)cc2)C)CC1 C1(C(=O)NCC(C)(C)NC(C2CCN(CCC)CC2)=O)CCc2n[nH]cc2C1C c1(C(C(=O)NCCCN(C2CCC(C)C2)CC)(C)C)cc(Cl)ccc1F N1(C(C(CC=C)C)=O)CCC2C(NC(=O)Cc3ccsn3)C2C1 C1(COC)(NC(=O)CC=Cc2ccc(C)cc2)CCCN(C(C2CCSC2)=O)C1 C1(CC)C(CC(=O)N(CCCN(C(=O)C=Cc2cnc[nH]2)C)C)C1(F)F N1(C(=O)Cn2ccccc2=O)Cc2ccc(Br)cc2C1.C12CC(C1)C(=O)N2 c1(NC(CCC)=O)ccc(CNC(C2CCC2c2ccc(F)cc2F)=O)c(F)c1 n1(C(C(=O)NC(C2CN(C(c3snc(O)c3Cl)=O)C2)C)C)c(C)cc(O)cc1=O CC1CCC(CC(=O)NCC2CN(C(=O)CCC(C)SN3CSCC3=O)C2)OC1 N1(C(C)C(=O)N(C(C)CNC(=O)C(C)Oc2cccnc2)C)CCCCC1=O N1(C(C(C)(C(C)C)OC)=O)CCN(C(c2csc(C(C)(C)C)n2)=O)CC(O)C1 N1(C(C(=O)NC)=O)CC(CNC(c2c(-c3cccnc3)noc2C)=O)CC1(C)C C(=O)(C(F)(F)CCn1cccn1)N1CC2C(CNC(COCC(C)C)=O)(C2)C1 Nc1ncc(Br)nc1C(=O)NCC1CCC(NC(C2CN(C3CCC3)C2)=O)C1 C(=O)(C1=CCCN(C(C2CCCSC2C)=O)C1)N1CCC(C=C)(O)C1 N1(C(C2C(NC(C(CCC)NC(C)=O)=O)CCCC2)=O)CCc2oc(C)nc2C1 c1(C(N(C(CCNC(C(C)C2(O)CCC2)=O)C)C)=O)cc(C2CCCC2)nn1C C1(C)(CNC(Cc2cn(C)nn2)=O)CCCN(C(c2cc(Cl)ncc2F)=O)C1 C1(C(=O)NC(c2cnn(-c3cccc(C#N)c3)c2)C)CC2CCCCN2C1=O c1(OC)nn(C)cc1C(C)NC(c1cnn(C)c1)=O C1C2CCC1N(C(=O)C(C)(C)NC(=O)OC)C2.c1(OC)ccccc1NC(=O)NC N1(C(CN(C(COC)=O)C)=O)CCC(C)N(C(C2CNC(=O)C(C)(C)C2)=O)CC1 N1(CCc2ccc(C(=O)NCc3ccnc(Cl)c3F)cc2)C2CCC1CC(O)C2 c1(C(=O)NCC(=C2CN(C(=O)COC(F)(F)F)C2)F)cnn2ncccc12 C1(NC(C2CCCN(C)C2)=O)CC2CCCC(C1)N2C(c1ocnc1C(F)F)=O C1(NC(c2c(C(C)(C)C)c[nH]c2)=O)C2CC(NC(C3(C)C=CCC3)=O)CC12 CC(C)CC(C(=O)NCC(O)CCNC(c1ccc(C#N)o1)=O)C(N)=O c1(C(=O)NC2C3CN(C(C(C(C)(C)C)(C)O)=O)CC32)ccc([N+](=O)[O-])c(Cl)c1 c1(OC)cc(C)c(C(=O)N(C)CC2CCN(C(c3cnoc3C)=O)C2)cn1 C1(CC)CN(C(=O)CC2CCCO2)CC1C(N1CC2(CC2)C1)=O C1(N(C(C2CCCC2Nc2cnc(C)s2)C(=O)NCCCC)C)CC(=O)NC1=O C(=O)(CC(C(C)C)C(C)C)N1CC(OC)C(NC(=O)CCC2CCN(C)CC2)C1 c1(SC)ccc(CNC2CCCC(C(N3CCC3C)=O)C2)cn1 Cc1cn(CC(N2CCC(NC(C3CC3c3nccn3C)=O)C2)=O)c(=O)nc1O C1(C2CCN(C(C3CSCCS3)=O)C2)(NC(=O)C(F)CC2CC2)CC1 c1(C(=O)NCC(CC=C)NC(=O)CC)coc2c(C)cccc2c1=O C1(CNC(c2cc(OC)n[nH]2)=O)CC12CCN(C(=O)CC1CSCCS1)CC2 CS(=O)(=O)c1ccc(C(N2CC(OCCNC(C3(F)CCOC3)=O)C2)=O)[nH]1 O=C(CCCCCO)NCC1(NC(C2(N3CCOCC3)CC2)=O)CCOC1 N1(C(C2(CF)CCN(C(C#CC(C)C)=O)C2)=O)CC2(COC(C)(C)C2)C1 c1(C(=O)NC(C)CN(C)C(C2CCC2CF)=O)c(C(F)(F)F)ncn1O N1(C(CCN(S(C)(=O)=O)C)=O)CCN(C(C2(C#N)CC3CCC2C3)=O)CC(O)C1 CC1=CC(C)CN(C(C2C(C)CN2C(C2CCN(C)C2)=O)=O)C1 Cc1cccnc1CNC(=O)CC1CCC(NC(=O)C=CC2CCOC2)C1 C=CC1(C(N2CCOC(NC(=O)COCCOCC)C2)=O)CCCCC1 N1(CC(=O)NC(C#C)C)CCN(C(c2cnccc2OC)=O)CC1 C1(NC(c2ccc(C)c(C)n2)=O)C2CC(O)C1N(C(C1CC(C)(C)C1)=O)C2 c1(NC(=O)NC)ccc(C)c(C(=O)Nc2ccc(CC(N)=O)cc2)c1 N1(C(C2(CC#C)CCC2)=O)CCN(C(=O)CC(C)SC)C(C2CCC2)C1 N1(C(C2CN(OC)C(=O)C2)=O)CCC2CCC(C1)N2C(=O)C=CCO C1(CC(=O)N(c2ccccc2)C)COC2CC1C2.C1(C(C)C2CC2)CCC(C(=O)NC)O1 Cc1ccccc1C(C)CC(=O)N1CC(C)(NC(c2cc(O)n(C)n2)=O)C1 c1(Sc2cccc(NC(N3C(C(=O)OC)CCC3)=O)c2)ccc(NC(C)=O)c(C)c1 c1(C(=O)NCCN(C(C2CC(=C3CC3)C2)=O)CC)ccc(C2CCCO2)[nH]1 c1(NC(COC(C)(C)CNC(=O)COCCCF)=O)cccc(F)c1O C1(C(=O)NCC(C)NC(c2cnn3c2OCC3)=O)CC(S(C)(=O)=O)C1 C=CC1(CC(=O)NCCc2cccnc2F)CN(C(C2C(C)C2C)=O)C1 c1(NCCC(=O)NC(CC)C)nc(N2CC(O)CC(C)C2)cc(C)n1 C#Cc1cnc(C(=O)NCC2(CNC(=O)CC(=O)OC)CC23CCC3)c(C)c1 C1(C(=O)NCC(CNC(COCCC)=O)F)CCSCC1 N1(C(C2(NC(c3ncccc3O)=O)CCC2)=O)CC2C3CCC(O3)C2C1 C(=O)(C#CC1CCCCO1)N(C1CCCN(C(c2c(C)coc2)=O)CC1)C c1(SCC(=O)NCCC(C)(C)NC(CC=CC)=O)nc2ccc(C)cc2[nH]1 CC1CCN(C(=O)Cc2c(C)noc2Cl)C(C)C1NC(=O)C1=COCC1 N1(C(CN(C(C(C)C)=O)C)=O)CC2(CC2)CC1CNC(C1CC12CCSCC2)=O c1(C(N2C(COC)CC2)=O)cccc(C(C)(C)C)c1N.C12(CC(CF)C1)C(=O)N2 CCC(CN(C)C)CC(=O)NCC1CC1CNC(=O)C=Cc1cncs1 c1(C(=O)NC2C(OC)CN(C(=O)CC3CC3C(F)(F)F)C2)cncc2c[nH]nc12 CN1C(=O)NCC1C(N1CC2C(N(C(=O)CC3CSCCO3)C)C2C1)=O C(N=c1[nH]cnc(Cl)c1C#N)C1CCN(C(c2nc(C(C)OC)oc2)=O)C1 N1(C(COCCC)=O)CCC(C)C1CNC(=O)COCc1nc[nH]n1 CC(C(C)C(=O)NC1CN(C(C23CC4CC(CC(C4)C2)C3)=O)CC1O)S(C)(=O)=O c1(CNC(=O)CCC2CCCOC2)cc(C(=O)NCC(C)(C2CC2)OC)no1 C1(C(=O)NCC2CCCC2)CCCN(C(=O)CC2CCS(=O)(=O)C2)CC1 CCCC(C#N)C(=O)NCCCCc1cn(-c2ccc(C)c(Br)c2)nn1 c1(CC)cnc2ncnc(C(=O)N(C3CCCN(C4CC4)C3)CC(C)C)c(=O)n12 C1(NC(Cn2ccc(C)n2)=O)CC2CN(C(C3CN(C)CC(C)O3)=O)CC12 c1(C(=O)NC2(CC=C)CCNC2)cc2c(s1)CCCCCC2OCC C1(NC(CCN(CC)CC)=O)CS(=O)(=O)CC1NC(=O)Cc1ccc(OC)nc1 c1(OC)cccc(C2CCN(Cc3cc(Cl)ccc3N(C)C)C2)c1F c1(C(=O)NCC2(COC)CCN(C(c3cc(C)[nH]n3)=O)C2)nnc(O)cc1O CN1CC(C)(C)CC1C(=O)NC1CC2(C1)CC2C(N1CC2(CSC2)C1)=O CN1Cc2cc(C(N3CCCC3SCC(F)(F)F)=O)ccc2NC1=O C1(CC(=O)N(CCC(=O)NC(COC)CC)CC=C)CC=CCC1 c1(C2CCCN(C(=O)NC3CCN(C(C)=O)CC3)C2)ccc2sc(C)nc2c1 C(C(C)(C)C(=O)NCC1CCN1C(=O)CCn1cnc(=N)[nH]1)SC Cc1nc(C(N2CC(CC(=O)Nc3cccc(C(N)=O)c3)C2)=O)sc1C N1(C(C(=Cc2ccco2)C)=O)CCCC2C(NC(=O)C=CSc3nc[nH]n3)C12 N1(C(CNC(=NC)NCCCN2CC(C)OC(C)C2)=O)Cc2ccccc2C1 N1(C(c2nc(CCCC)sc2)=O)CCCC(C2(NC(C3(OC)CCSC3)=O)CC2)C1 N1(C(C2(COC)CC2)=O)CCC(CNC(=O)CCN(CC(C)C(C)C)C)C(O)C1 O(NC(=O)C(C)(C)CCNC(=O)C(=O)CCCC)CCCCCC=C c1(C(C)OC)nc(CS(C)(=O)=O)n(C(C)C(F)(F)F)n1 CCC(CC)(CC)C(=O)NCC(C)NC(c1ccc(CN2CCCC2=O)cc1)=O C1(NC(C(CCC)C)=O)CC2CCC(C1)N2C(C)C(=O)NC1CCCCC1 C(N=c1cc(NCc2cnnn2C)nc[nH]1)C1C(C)CC(C)O1 Cc1cccc(C(N2CCOC(C(=O)NC(c3ccc(Br)cc3)CO)C2)=O)c1O C1(CNC(C2C(C)CCCC2)=O)CCCN(C(c2ncccn2)=O)CC1 C(=O)(CCCCC(C)(C)OC)NC(CCOC)CNC(=O)C(C(C)C)NC(N)=O C1(NC(C=C(C)C(F)F)=O)CCCN(C(C2CC(=C3CCC3)C2)=O)C1 c1(CC)cc(C(=O)NCC2(NC(c3ccc(-n4ccnc4)cn3)=O)CC2)sc1C O=C(CC(F)(F)C(F)(F)F)NC1CCC12CN(C(c1cccc3[nH]ncc13)=O)C2 n1(CC)ncc2c1CC(C(=O)NCC(CC(C)C)NC(=O)C1=CCCC1)CC2 C(=O)(CC(C(=O)OC(C)(C)C)OCO)NC1(C)CC(NC(C(C)(F)F)=O)C1 N1(C(COCCC)=O)CCC(N(CCC)C(C2CC(F)(F)CS2)=O)CC1 Cc1ccc2sc(N3CC4CCC3CN4C(c3coc(Cl)c3)=O)nc2c1C Cc1nn(C(C)CC)c(C)c1C(=O)OC1C(=O)OC2CCCC12 c1(C(N(C2CN(C(=O)CCC3CCCOC3)C2)C)=O)csc2cccc(F)c12 C1(CC(C)(C)C)(CNC(C(F)F)c2cccs2)CCNC1 c1(OCC)ccc(Cl)c(C(=O)NC2(CCO)CN(C(=O)C(C)n3cccn3)C2)n1 c1(C(N2CC3(C(NC(=O)NCC(F)(F)F)C3)C2)=O)cccc2c1C(=O)OC2 C(N=c1[nH]c(N2CCOC(CCF)C2)nc2c1COC2)C1(C)COCCO1 CCCC(O)CCNC(C1(CNC(c2sccc2F)=O)CC(C)(C)C1)=O N1(C(c2cnn(CCC)c2C(F)(F)F)=O)CCN(C(=O)CC(=C)C)CC(CO)C1 C(CCC(C)(C)C(=O)NCC1(O)CCCC1(C)C)NC(C1CC(CC)OCC1)=O C1(O)(C(=O)NCCC(C)CCNC(c2ccc(CO)o2)=O)CN2CCC1CC2 c1(-n2c(C3C(CC)C3)nc(CC(C)OC)n2)cc(Cl)ccc1C N1(C(COCC)=O)CCC2CCC(C1)N2Cc1ccc(C#N)cc1F Cc1ccc(F)cc1NC(N1CCOC(C(=O)NC2CC23CCC3)C1)=O c12cn3c(n1)CN(CC3)C2=O.c1(CN2CCC(C)(OC)C2)c(F)ccc(Br)c1Cl c1(Nc2cccc(CNC(=O)Nc3c(C)coc3C)c2)ccc2c(c1)CCCO2 C(=O)(C1=CCCCC1C)NC(C(=O)NC(CC)C(=O)OC)C(C)C CCC(F)(F)C(=O)NCC(C)CNC(=O)C(=O)C=Cc1ccccc1 CC1N(C(C2(C(C)NC(c3ncccc3O)=O)CC2)=O)CCOC1(C)C c1(COC)ccc(C(=O)N(C(CC)C(=O)N2CCCC2CNC(C)=O)C)o1 c1(C(=O)NCC(O)CCNC(c2ccc(O)nc2Cl)=O)ccc2c[nH]nc2n1 C12(C(=O)NCCC(CCNC(C(C)OC)=O)C)CCC(CC1)C2.N12CCCC1C2 CCCCCC(C(N)=O)NCC1CCC1CNC(=O)N(CCOC)CC1CCCC1 c1(C(N(CCN(C(c2ccc(C(=O)OC)[nH]2)=O)C)C(C)C)=O)cc2n(n1)CCO2 c1(C(=O)NCC(N(C)O)=O)cc(CO)ccc1F.C12CCCC(C1)C(=O)N2 c1(C(N2CCN(C(CS(CCC)(=O)=O)=O)CC2)=O)cc2cccc(C)c2s1 c1(C(C)C)ncc(C(=O)NC2CN(C(=O)C(C)c3ccsc3)C2)n1C c1(CCC=C)ccc(C(=O)NCCN(C(C2CCCCN2C)=O)C2CC2)cc1 CN1CCc2ccc(C(=O)NC3C4CN(C(=O)Cc5ccc(Br)cc5)CC34)cc21 C1(CNC(=O)CCCc2nccs2)CN(C(=O)COC(F)F)CC(C(F)(F)F)O1 Cc1ncc(CCC(=O)NC2CCCC(NC(c3cc(CF)on3)=O)C2)c(O)n1 N1(C(=O)CC2COCCO2)CCOC2(CCN(C(C3CCCCO3)=O)CC2)C1 C1(CCNC(CC2C(C)C2(F)F)=O)CCCCN1C(c1cc(C(F)F)no1)=O N1(C(c2cc(CNC(c3ccc(OC)o3)=O)[nH]n2)=O)CCCCCCCCC1 C(=O)(CCOCCN(C(=O)C(C)=CC(C)(C)C)C)NCCNC(=O)NC C1(NC(C(CC)(C)O)=O)CN(C(=O)C=Cc2cncc(OC)c2)C(C)(C)C1 C1(C(=O)NC(C(C)NC(Cc2c(C)nn(C)c2)=O)(C)C)CCN(C)C(=O)C1 c1(C(N2CC(C#N)C(NS(=O)(=O)c3cccs3)C2)=O)[nH]nc2ncccc12 N1(Cc2cn(C(C)(C)C)nn2)CC2CC2(C(=O)NCC2CCC(=O)NC2)C1 C1(NC(C2CCOC2)=O)CCC2CN(CCN3C(=O)CCC3=O)CC2C1 C1(CCC(N2CCC(CCNC(CCNC(C)=O)=O)C2)=O)CCC(=O)NC1 C(=O)(C1=Cc2ccccc2C1)N1CCC(NC(c2ncc(F)cn2)=O)C(CO)C1 CC1C=C(C(=O)NC2CC(F)(CNC(c3ccc(F)cn3)=O)C2)CC1 Cc1ccc(C(=O)NCCNC(=O)C(O)Cc2ccccc2Cl)c2c1NCCC2 Cc1cc(=NC2CC=CCC2)[nH]c(N2CCSC(C(F)(F)F)C2)n1 C(=O)(C1=NOC2(CCC2)C1)N1C2CC(NC(Cc3ccc(C)cc3)=O)CC1CC2 CC1(C)COC(CCC(=O)NC2CC3(C2)CC3NC(c2coc(CO)c2)=O)C1 c1(OC2CCN(C(=O)OC)C2)cc(NC(=O)C(C)OC2CCCCC2)ccc1Cl N1(C(c2cn(CC)nc2)C(=O)N(C2CCC2)Cc2ccccc2)CCCC2CC12 C(CCCC)(CC(=O)NCC1(C)CCCC(=O)N1)NC(C(CC=CC)C)=O C1(CCC)CN(C(c2ncn(C(C)(C)C)n2)=O)CCN1C(=O)CC(C)O C(C(=O)NNC(=O)C1OCCCC1C1CC1)c1cc(C)[nH]n1 Cc1nc(Cl)sc1C(N1CCC(CC(=O)NCc2nccnc2Cl)C1)=O C12(CCNC(c3c(C)n(C)cn3)=O)CCC1CN(C(c1cc(Cl)ccc1F)=O)C2 c1(-c2cn(C3(C(=O)NCC(C4CC4)OC)CCOCC3)nn2)cc(N)cc(F)c1 N1(C(C(CCC)OC)=O)CC2CC(CNC(C3(N(C)C)CCC3)=O)C2C1 C1(NC(=O)C(C)(C)C2CCC2)CC(F)(NCC(CCCC)C2CCC2)C1.C1(C)C(=O)N1 CC(Cc1cnc[nH]1)C(=O)NCC1CC1C(=O)NCCCC(=O)NC1CC1 c1(COCCC)cccc(C(=O)NCC(c2cccc(OC(F)F)c2)N(C)C)c1 c1(CC(=O)Nc2cccc(C(N(C)C)=O)c2)cccc(N=c2nn[nH][nH]2)c1 N1(C(=O)NCCCN(C)C)C(NC(=O)OC(C)(C)C)CCC1(C)C c1(C(=O)NC2(C)CN(C(CC(COC)(C)C)=O)C2)ccn2c(C)ncc2c1 n1(CC)ncnc1C(N1CC(CC(C)(C)CNC(c2coc(N(C)C)n2)=O)C1)=O CC1(C)CC(=O)NCC1C(=O)NCC=CCNC(c1ocnc1C1CC1)=O c1(C(=O)NC(C(=O)NC(C#C)C(C)C)CO)cnn(C)c(=O)c1 c1(CC)noc(CC)c1CNC(C1OCCC1N1CCC(NC)C1C1CC1)=O C1(N)CC12CCN(C=O)C2.c1(CC)nc(C(=O)NCCNC(C2CCCC2)=O)cs1 CN(C)S(=O)(=O)N1CCN(C(C2CCN(C(=O)C=Cc3ccccc3)C2)=O)CC1 C(CC(C)(C)C(=O)NC1(C2CCCN2C(c2ccc(C3CC3)s2)=O)CC1)OC N1(C(C(C2CCCCC2)OC)=O)CCCC(CC(N2CCC(C(C)O)CC2)=O)C1 O=C1Cc2cnc(N3CCC(NC(=O)Cc4cccc(Cl)c4)CC3)nc2N1 CCCCCC(O)C(=O)NCC12CCC(CC1)N(C(=O)CC(C)(C)O)C2 c1(C(=O)NCC(C)NC(C(C)C2CCC2)=O)sc(Cl)cc1Br C1(CNC(C2(CCS(N)(=O)=O)CCC2)=O)CCCCN1C(C12CC3CC1C2C3)=O c1(C(=O)NCCN2CCN(C(C(C)C3CCC3)=O)CC2)cccc2c1CC(=O)N2 c1(C(N2CCC(NC(c3nc(C)oc3)=O)C(F)C2)=O)[nH]nc([N+](=O)[O-])c1Cl C1(CCC=C)CCCN(C(c2ncoc2C2CCCO2)=O)C1 Cc1c(C(=O)NC(CO)C(C)NC(C2(Cc3ccon3)CC2)=O)nn2ccccc12 c1(C(=O)NCCn2c(C)nc(C)n2)ccc2c(n1)CCN(C(=O)CCC(C)C)C2 c1(OC)cncnc1C(=O)NCCC1CCN(C(=O)Cc2cccn2C)C1 C1(C(=O)NCC2(NC(c3c(CC)non3)=O)CCC2)CCCC1S(C)(=O)=O C1(C(C(=O)NC2(c3ccon3)COC2)O)CCN(c2ncccn2)CC1 Cn1cc2c(n1)CC(C(=O)NCC#CCNC(=O)Cn1ccnn1)CC2 c1(N2C3C(NC(C(CC)c4cccs4)=O)CC(CC3)C2)nc2ncc(Cl)cc2o1 C1(CNC(C(C2CCCC2)OC)=O)(CO)CCN(C(C2(CC(C)C)CC2)=O)C1 C1(CCC(=O)N(CC(CC)NC(=O)C(C)(C)n2ccnn2)C)CC(C)(C)CO1 c1(CCC(=O)NCC(CC)NC(C2CC2C(=O)OC)=O)ccccc1Cl c1(NC(=O)CSCC2(O)CCNC2)ccccc1OC(F)(F)F CC1(NC(=O)COC2COC2)CCCCO1 C(=O)(CC(C)(C)CS(C)(=O)=O)N1CCC(C2C(NC(C3(C)CC3)=O)CCO2)CC1 N1(C(c2ncc(OC)nc2)=O)CC=C(C(=O)NCC2(O)CC(O)C2)CC1 c12ccc(Cl)cc1C(=O)N2.c1(N(C(C(C)OC(=O)CN(C)C)=O)C)ccccc1 CCC(C)CCS(C)(=O)=NC(=O)c1cnc(O)c2ccccc12 C=Cc1ccc(C(=O)NC(CN=[N+]=[N-])C(=O)NCCC2CCCC2(C)C)cc1 CC(CC(=O)NCC1CCN(C(C2CCC3(CCC3)CC2)=O)C12CC2)C(C)(C)C C(N=c1[nH]c(=NCC2CCCC2)c2ncccc2[nH]1)C1ON=C(C)C1 N1(C(C(C)C2(O)CCC2)=O)CC(N=[N+]=[N-])CC1C(=O)NCCS(C)(=O)=O c1(CC)nc(C(N2CC(OC)CC2CNC(=O)C(C)OCOC)=O)c(C)o1 CC(F)(F)C(F)(F)CC(=O)NC1CCCC1NC(=O)CCc1nc(=N)[nH][nH]1 c1(CC(N2CC(C)N(Cc3cnn(C)c3)CC2)=O)cc(F)c(Br)cc1F N1(C(C2N(CC)CCC2)=O)CCCC(O)(CCNC(=O)CCc2cccnc2)C1 N1(C(C)C)CCCC1CC(=O)NCCCCN(C)C(c1nc(C)no1)=O N1(C(C2(S(C)(=O)=O)CCC2)=O)CCN(c2ncnc(Cl)c2CO)CC12CCC2 C1(CC)CN(C(=O)Cc2sc(O)nc2O)CC1NC(c1ccn(C)n1)=O C1(CNC(C2CC(Cn3ccnn3)C2)=O)CCCC1C1CC1 N1(C(c2n(C)cnc2)=O)CC(NC(c2cnc(Cl)s2)=O)C(C#N)C1 c1(OC)cc(C(=O)NCCN(CC(C)O)C(=O)Cc2cn(C)nn2)cc(Cl)c1 c1(COCC)noc(C(N2CC(O)(C(C)NC(=O)Cc3cc(C)on3)C2)=O)n1 C(=O)(CCCCCC#N)NC1CN(C(c2cnc(C)c(N)c2)=O)CC1C c1(C(=O)NC2CC(SC(C)(C)C)C2)cccc(S(=O)(=O)CC(F)(F)F)c1 c1(CCC(=O)NC2C(CN(C)C)COC2)c(I)ccnc1O C(CC)(CCCC(=O)NCc1nn[nH]c1C1CC1)NC(CSCCC)=O c1(C2(C(C)NCc3ccnc(Br)c3)CC2)c(F)cccc1F C(=O)(CC(C(F)F)NC(=O)CC1(C)CCN1C(=O)C(C)(C)OC)OC C1(C(=O)NCCc2c(C)nn(C)c2)CCN(C(c2cc[nH]c2)=O)CC1O N1(C(c2ccn(CC)n2)=O)CC=C(C(=O)N(C)Cc2nccs2)CC1 Cc1cn(C)cc1C(=O)NCC1CCCC1C(=O)NCCc1cccnc1C CC1CC(NC(=O)CN(C)C(C2CCCC2)=O)CN1C(=O)C=Cc1cccs1 C(=O)(C1CCCn2cnnc21)NCC(CO)NC(CCNC(=O)NC)=O C1(NC(C2(SCC)CC2)=O)CN(C(=O)COCc2ccnc(O)c2)CCC1C N1(C(CC=C)=O)CCC2(CC1)CCN(C(=O)C=C(C)C1CCCCC1)C2 Cc1nc2c(N3CC4(C3)CN(Cc3c(Cl)ccnc3Br)C4)ncnc2[nH]1 C(C)(CO)(C(=O)NCc1coc(C)c1)NC(CC=CC=C)=O C1(CNC(C2(C=C)CCCC2)=O)CCC2(CCC2)C1NC(c1cccnc1C)=O c1(C(=O)OCCCC(C2CCC2)C2CCC2)csc(-c2ccccn2)n1 c1(NC2C3CCN(C(C)=O)C32)cc(NC(c2cn(C)cn2)=O)nc(C(F)(F)F)n1 C(CN=c1ccc([N+](=O)[O-])c[nH]1)C(C(C1CCOC1)NC(NNC(C)=O)=O)=O C(=O)(CC(C)(C)C)NCC(C)(CC)N(C(C(F)=CCC)=O)CC C1(CC(=O)NCC(C)NC(=O)C(C)NC(=O)Cn2cnnn2)CCS(=O)(=O)C1 N(C(=NCCCc1nnc2ccccn12)NSc1cccs1)C(C(C)C)C c1(C(=O)NC2(CCNC(C3CCC4CCC34)=O)CCC2)nccc2[nH]ccc12 N1(C(C(C2(O)CCC2)NC(COC(CC)C)=O)=O)CC2CC1CN2CCO C=CCCC(C(=O)NC1(c2ncc[nH]2)CC1)NC(C1CC(=O)N(C)C1)=O CN(C)S(=O)(=O)N(C)CC(N1CCCC(NC(C2CCCS2)=O)C1)=O c1(NC(N2C(C(=O)OCC)C(C)CC2)=O)ccc(OC(C)(C)CCl)cc1 n1(CCNC(C)Cc2cccs2)ccnc1C(c1nnnn1C(C)(C)C)OC C1(C(N2CCC(OC)CC2)=O)CCC(C2CC2)C1.N12CCC1(C)N(CC)CC2=O C1(CNC(=O)Cc2cnoc2)CC2COCC2N1C(c1ccc2cc[nH]c2n1)=O C(C1CCCCCC1)=C(C)C(=O)NC(C1CCOC1)CNC(c1cnn(C)c1)=O N1(C(C(C)n2ccnn2)=O)CCC2(C1)CN(S(=O)(=O)c1ccn(C)n1)C2 c1(OC)ccc(C(=O)NC2CC2CNC(C2(F)C(C)(C)C2(C)C)=O)c(N)c1 N1(C(C(C=C)CC)=O)CCC(NC(c2ccc(C)o2)=O)CC1C1CC1 c1(CC)ncnc(N(C2CNCC(F)(F)C2)C(=O)CCc2cn(C)cn2)c1F C(=O)(CCC(C)(F)F)NC(C(C)NC(c1c(C)cc(SC)o1)=O)C C=CCC(C(=O)NCCNC(=O)CCF)n1cc(C2(N(C)C)CCCCC2)nn1 c1(C(=O)NC2CC3C(NC(=O)CC(C4CC4)C4CC4)C3C2)ccnc2ccsc12 c1(CC(=O)NC2CCCN(C(c3cccn3C3CC3)=O)C2)c(Cl)ccc(O)c1Cl c1(C(=O)O)cnc2c(cnn2CCCN2CCCC2c2ncccn2)c1 C1(C(=O)NCCC2CCN(C(C3(CCC)CCC3)=O)C2)CC2COCC(C1)C2 N#Cc1ccc(CCC(=O)NC2(CO)CCN(C(C3CC3Cl)=O)C2)c(F)c1 C12(CNC(CCC=C)=O)CCCC1N(C(c1nn(C)cc1C)=O)CCC2 CCCCCCC(F)C(=O)NC1CN(C(=O)Cn2cc(F)ccc2=O)CC1F N1(c2ccc3c(c2)OCCCO3)CCN(C(=NCCC2CCCO2)NC2CC2)CC1 c1(C(=O)NC)ccc(C(N2CC3C(C2)C3(C)C)C(=O)NCCOC2CC2)c(Cl)c1 C(=O)(C(C)(O)CCC1CC1)NCCCC1(NC(Cc2n(C)nnc2)=O)CC1 C1(C(C)NC(c2cc(-c3ccccc3)cs2)=O)CCN(C(=O)C(F)(F)CO)CC1 C(CC(C(=O)NC1(CNC(=O)CCc2cn(C)nc2C)CCOC1)N(C)C)SC N1(C(C(C)OCC(C)C)=O)C2CCC1C(C(=O)NCc1ccsc1F)C2 O=C(C1=CSCCO1)NC1CCCCC1CNC(=O)COc1ccccc1 Cc1ccc(C)c(OCC(=O)N(C2CCN(C(=O)C=CC3CCOC3)C2)CCO)c1 c1(C(N(C)CCNC(=O)CCSc2ccc(Cl)cc2)=O)cccn(C)c1=O c1(-n2cc(-c3cc(=N)[nH]cc3)nn2)cnn2cnnc2c1 C12(C(N(C(c3nc4c(s3)CCCC4)C)C3CC3)=O)CCCC1CC(F)(F)CC2 CN(C)NC(=O)CCC(=O)N1C(C(=O)NC2CCC3(CCC3)C2)CCC1C Cc1ccc(C(=O)OCC(=O)NCCCc2ccc(F)cc2)cc1 C1(C(=O)NCCC)CCCN1CCC(=O)NCCC(C)(F)F C12(CNC(CCC)=O)CN(C(c3ccc(C4(C(N)=O)CC4)cn3)=O)CC1CCO2 N1(C(CC2N(C(C(C(C)C)C#N)=O)CC(C)(C)C2)=O)CCCNC(=O)C1C C(C(C)(O)CNC(=O)COCC1CCCO1)N(C)C(c1cnn(C2CC2)c1)=O c1(OCC)cccc(C(C(=O)NCC2CCCO2)N(C)C(c2ccco2)C)n1 CN1N=C(CC(=O)N(C)CC2CN(C(c3ccc(F)c(C#N)c3)=O)C2)CC1=O CC(C)CCC(C(=O)NCC1C(CO)C1(C)C)NC(=O)CC(C)O C12CCCN(C1)C2=O.C(CS(=O)(=O)NCC(=O)Nc1ccns1)OC(C)(C)C C1(F)(CNC(C2C(C(N)=O)CC2)=O)CCCN(C(C2CCSCC2)=O)C1 C1(C)(CNC(C(C)Cn2cccn2)=O)CCCN(C(c2ncc(Br)cc2O)=O)C1 c1(CCC)ccc(C(=O)N(CC(CC)NC(=O)CC2CCCO2)CC)cc1 Cn1nc(O)cc1C(N1CC(CNC(C2CCC(=O)NC2)=O)C1)=O C1(CC(N2CC3C(CC)C3C2)=O)C2CCCC2N1C(c1n[nH]c(C)c1O)=O CC(CN=c1[nH]c(-c2ccccn2)nc(=N)[nH]1)NC(c1ccn(C2CCC2)n1)=O C1(CCC(=O)NCC2(NC(C3CNC(=O)N3)=O)CCOCC2)CCC(F)(F)CC1 CCCCC(C(=O)NC)NC(C1(C=C)CCN(C(c2ccncc2N)=O)C1)=O C(=O)(CCC(=O)C(C)(C)C)NCCN(CCC)C(c1ccc(CN(C)C)nc1)=O N#Cc1cccc(Cl)c1C(=O)OCc1ccnc(O)c1 c1(C(N(CCCNC(=O)CCCc2ccc(F)cc2)C2CC2)=O)cc(Cl)ccc1F CC1CC(NC(C2COC3(CCC3)C2)=O)CCN1C(=O)CC(F)(F)F N1(CC#N)CC2CCC1CN2C(=O)CCNc1cc(F)cc(F)c1 C1(C)(C(=O)OCC)CCCN1N(CCO)CC1(O)CCN(C(C)C)C1 C1(C(=O)NC(c2ccccc2)C(=O)NC(CCCC)C)CC(F)C(=O)N1 C12(NC(c3cc(C)sc3C)=O)CCCC1CN(C(=O)C=Cc1cccs1)C2 c1(C(=O)NCCC(=O)NCCC2CCCCN2C(C2CC2)=O)cc2scnc2[nH]1 Cc1nn(C)c(=O)c(C(N2CCC(CNC(=O)CN3C(=O)CCC3=O)C2)=O)c1C c1(C(N2CCC(O)(CNC(C3(C)CCCC3)=O)CC2)=O)ccc2c(c1)COCO2 n1(C(C)C)cnc(C(N2CCCC2CNC(C2CC2F)=O)=O)n1 c1(C(=O)NCC(CN(C)C(c2cnc3sccc3c2)=O)O)cc2c(nn1)CCC2 C(N=c1nc(N2CCC(C#N)CC2)c2c([nH]1)CSC2)C1(C)CCC(=O)N1 C1(CNC(C2C(CNC(C3CCC(C)O3)=O)OCC2)=O)CC12CCOCC2 N1(C(CC(CC)O)=O)CCCC(CNC(c2ccc(-c3cnco3)cc2)=O)CC1 C1(NC(c2ccc(OCCC)cc2)=O)CC2CC(NC(=O)C(C(C)C)SC)C1C2 C(c1ccc(Cl)cc1Cl)=CC(=O)NCC(C)NC(C(CC=C)CC)=O C(=O)(CC1CCc2ccccc21)NCCCN(C(C)=O)C(C)C N1(C(c2ccc(CC)nc2)=O)CCCN(C(c2cccc(OC)c2N)=O)CC1C c1(NC(C)=O)ccc(C(N2CCN(C(=O)Cc3c[nH]nc3C)C3CC23)=O)cc1C C(C)(CCNC(C=C(CCC=[SH]C)C)=O)SC.C12(CC1)C(=O)N2 N1(C(c2n(CC=C)ccn2)=O)CCC2(CCCN2C(C2CC2F)=O)CC1 CCC(C)(C#N)C(=O)N1CCCC(N2CCN(C(C3(C)CC3)=O)CC2=O)C1 c1(C(N2CCC(CCCNC(C3C(C)(C)C3C#N)=O)CC2)=O)cc2occc2[nH]1 c1(CCNC(CCCOCC=C)c2nnnn2CC)c[nH]c2cc(Cl)ccc12 c1(C(=O)NCCC2CCCN2C(=O)Cc2cc[nH]n2)sc(F)cc1Br Cc1ccc(N(C(=O)C(C)NCCC2CCCC2(F)F)C)cc1 N1(C(C(C(CC)O)C)=O)CCC2(CCN(C(=O)CN3CCc4ccccc43)C2)C1 C(C)(CN=c1[nH]cnc2ccc(F)cc12)NC(C(CC(C)C)(F)F)=O c1(C(=O)NC2CC(CCC(N3C(C=C)CCC3)=O)C2)cc(C#N)nn1C S(=O)(=O)(c1cc(C(=O)NC2(C)CCCN(C(C3(C)CCC3)=O)C2)ccc1F)NC CC1CCC(C)N1CC(N1CC=CCC1C(=O)NC(C(O)CO)C1CC1)=O c1(C(N(CCNC(C(CCCOC)C)=O)C(C)C)=O)ccc2occc2n1 Cc1ncc(Cl)cc1C(N1CCC(CNCS(C)(=O)=O)C1)=O.C1CO1 C(CCN=C(NCc1c(NS(C)(=O)=O)cccc1Cl)N1CCC(C)C(F)(F)C1)SC C1(O)(CNC(C(C)(C)Cc2cnn[nH]2)=O)CCCN(C(C2CC3CCC2O3)=O)C1 C1(C)(C(N2CC(OC)(CNC(=O)Cc3cncn3C)C2)=O)C=CCCC1 C1(C(=O)NCC2(SC)CC2)CC(C)(C)CN1C(=O)Cn1nnnc1C1CC1 N1(C(=O)C=CC2CC2)CCC2(C1)c1[nH]cnc1CCN2C(C1CCCOCC1)=O c1(C(C)F)ccc(C(=O)N(C2CN(C(=O)C=Cc3ccncn3)C2)C)cc1 c1(C(N2CCC(C)C2CNC(=O)CCC2CCOC2)=O)ccc2c(c1)C(=O)NC2 c1(OCC=C)cccc(C(=O)OCCCN(C)CCOCC)c1 C1(CNC(C2OCCN(C)C2)=O)CN(C(C2CCCCCC2)=O)CCC1(F)F C(c1ccoc1)=CC(=O)Nc1ccoc1.C12CCC1C(=O)N2CC(Br)Br c1(C(=O)NC2CC(NC(Cc3c(C)ccs3)=O)C2)ccncc1N(C)C C1(NC(N(C(C)(C)C2CC2)C)=O)CCN(N2CCOC(C)(c3cnn[nH]3)C2)CC1 c1(C(=O)NC2CCN(C(CCC(C)C)=O)C2(C)C)nc2ncc(Br)cn2n1 c1(CC)ccc(C(N2CCC(C)C(CNC(C3CCN(C)CC3)=O)C2)=O)c(O)c1 C1(C(=O)OC)C2CC(CN(C(=O)C(C)(C)O)C2)N1C(=O)Cc1csc(NC=O)n1 C#CCCN=C(NCC(CCC)CCCC)NCC1CCCC1 c1(C(=O)NC(C(=O)NCCC(C)N(C)C)c2cccs2)cccc(=O)o1 C1(NC(c2cnn(CO)c2)=O)CCC2(CCN(C(c3n[nH]cc3[N+](=O)[O-])=O)C2)C1 C12CCCCC1CN2.C1(C(C#C)NC(=O)SC(C)(C)C)CCCCC1 c1(C(=O)NC2CC(F)(CNC(CC(OCC)OCC)=O)C2)cncc(CC)c1 c1(C(=O)NC(CC)(C)CC(=O)Nc2ccc(C)c(Cl)c2)ccc(Cl)cc1N N1(C(C(=O)NCC(C2CCC2)C2CC2)=O)CCCCC1CC(F)(F)F c1(CNC(C(=O)NCc2c(CC)nco2)=O)cc(NC2(C)CCCO2)cnc1F C(C(CC(C)C)C(=O)NC1CC2(C1)CC2C(=O)N(c1cccc(OC)c1)C)OC CCC(C)C(C(=O)N1CCCC(CCNC(c2sccc2SC)=O)C1)OC C1(C(=O)NC2(CO)CN(c3nnc(C)o3)C2)(COC)CC1(F)F N1(C(c2c(C)cno2)=O)CCC(CN(C(=O)Cn2[nH]cnc2=N)C)CC1 C1(OC)(CNC(C2CN(C)CC(C)O2)=O)CCN(C(c2nc(Cl)cs2)=O)CC1 Cc1ccc(F)c(C(N2CCC3CN(C(C4(C)CCC(=O)CC4)=O)CC23)=O)c1F c1(C(N2CCC(CNC(C(CC)(C)CO)=O)C2)=O)cc(C)c2c(O)n[nH]c2n1 CC1(C)CN(CCC(N2CC(C3(NC(=O)CCC(F)F)CC3)C2)=O)CCS1 N1(C(C2(C)C(C)CCC2)=O)CC2(CCCCN2C(=O)CCCCC2CC2)C1 c1(NC(CC2N(C(CSCCOC)=O)CCC2)=O)cccc2c1CCC2 N1(C(=O)Cc2cnsc2)CCCC2(C1)CN(C(C1C3CCC13)=O)CCO2 N1(Cc2c(C(=O)OCCC)ccs2)CC2CN(C(c3cccnc3C)=O)C2C1 CC1(C(=O)NC2(CC3CCC3)CC2)CC(O)CN1C(c1ccsc1)=O C(=O)(C(CCCC)N(C)C)N(CCCCCCNC(c1nc(CCC)oc1)=O)C C1(CN(C(CCNC(=O)NC)=O)C)COCCN1C(=O)CC(C)N(C)C CC12CC(C(N3CCC(CCCN4CCOCC4)CC3)=O)(C1)C1(CCC1)O2 C1(C(=O)NCC(CC)(C)OC)CC12CCN(C(c1sc(F)cc1C)=O)C2 N1(C(c2ncc(OC)cn2)=O)CC(NC(c2cc(Br)c(C)o2)=O)C2(CC2)C1 CCCCC(C(=O)NC1CCN(c2nnc(C)c(C)n2)C1(C)C)c1ccccc1 C(=O)(CCCCCC#N)NCC(C(=O)NCCN1CCC2CC12)N(C)C C1(C2CCCN(C(c3ccc(N)cc3O)=O)C2)(NC(CCC#C)=O)CC1 C(=O)(CCC(C)(C)O)NCC1CC(Nc2nccc(NCCC)n2)C1 CC1(CNC(=O)C(CNC(c2cn[nH]c2)=O)CC2CCCC2)CCCC1O C1(CNC(CC(c2ccc(C)cc2)C)=O)CC(F)(F)CN1C(=O)C(C)CF N1(C(c2ccc(P(C)(C)=O)s2)=O)CCC2(NC(=O)CCC3CCC3)CCCCC12 C1(NC(C(C)OC)=O)(CNC(=O)CC2=CCCCC2)CCC(C)(C)CC1 CC1(C(=O)NCCc2ccc(F)cc2)CCCN(C(=O)C(F)F)C1 N1(C(CC2CCN(C(C(=O)NC3CC3)=O)CC2)=O)CCC(O)C(F)(F)C1 c1(C(=O)NC(C2CCCN2C(=O)CCOC2CC2)(C)C)nc2cccnc2s1 N1(C(C2CC(SC)C2)=O)CCCCC(NC(c2cccnc2C2CC2)=O)C1 n1(CC)nc(C(C)C)cc1C(=O)NC(C1CCN(C(c2cn[nH]c2)=O)C1)C CCCCC(C)C(=O)NC1CN(Cc2cnc(Cl)cn2)CC1(C)C N1(C(C23CC(CC)(C2)C3)=O)CC2CN(C(C3(C)C=CCC3)=O)CC2C1 C12(C(=O)NCCCCC(=O)NC3CCOC3)CCCC1OCC2 CCC(CC)C(O)CNC(C1COCCC1NC(c1coc2c1COC2)=O)=O Cc1cc(C(N2CCCC(CO)(Nc3ncnc4sccc34)C2)=O)cc(C)c1F CN1CCCCC(C(=O)NCC(O)CNC(c2cc(C(F)(F)F)ncn2)=O)C1=O C(=O)(C(CCCS(C)(=O)=O)NC(=O)OC(C)(C)C)NCCSC Cc1cc(=NC2CCCN(CP(C)(C)=O)C2)[nH]c(NCCCn2ncc(N)n2)n1 Cc1nccc(C(=O)NCC(C)NC(c2ncsc2S(N)(=O)=O)=O)c1Cl C1(CCNC(C=CCN(C)CC)=O)CC(OC)CN1C(=O)CCc1nncs1 C(CC(C)(C)F)NC(C(C1CN(C(C2CC(F)(CF)C2)=O)C1)OC)=O CCC(CC)(CCNC(C1CCCC1C(F)(F)F)=O)NC(c1cnnn1C)=O N1(C(C2(COC)CCOCC2)=O)CC(NC(C2CC(C)(F)C2)=O)CC(F)C1 n1(CCNC(C(N)=O)=O)cc(C(=O)NC2CCC2O)cn1 c1(CC(=O)N(CCNC(C(C)=C2CC2)=O)C2CC2)sc(C)cc1C c1(C(=O)NCC2(CNC(C(N3CCN(C)CC3)C)=O)CCC2)ccc(Cl)nc1O C(=O)(CC(C)CC(C)(C)C)NC1CCN(C(c2cc(CCC)c(Cl)cc2)=O)C1C C#CCC(C)C(=O)N1CCCC1CN(C(=O)C(c1ccc(C(F)F)cc1)C)C CN1C(=O)COCC1CNC(=O)NC1CN(C(C2CCCCC2F)=O)C1 Cc1nnc(N2CCN(c3cccc(F)n3)CC2)n1C(c1cccs1)C c1(CCC(=O)NCC(CNC(Cc2ccc(C)o2)=O)C)ccc(=N)[nH]c1 C=CCCCCCCC(=O)NCC1CCCCN1C(C1(c2ncco2)CCC1)=O N1(C(c2c(C)[nH]c(=N)s2)=O)CCC2(CCC(NC(C3COC(C)C3)=O)C2)C1 C1(=O)C(N)CNS(=O)(=O)N1.C1CCOC1.CCC C(C(C(=O)N1CCC(C(C)NC(C2CCN(C)C2)=O)C1)C(C)(C)C)OCC(=C)C C=CC1CN(C(c2ccnc(C)c2)=O)CC1NC(c1cccc(N)c1C(F)F)=O c1(C(=O)NC(CN(C(C(C)OCCCC)=O)C)(C)C)ccoc1Br C1(C(=O)NCC(CNC(c2n(C)ncc2)=O)(C)O)CC2(CO1)CC(F)(F)C2 C1(C(N2C(CC)CN(C(=O)Cc3cccnc3O)CC2)=O)CN2CCCN1CC2 C(=O)(C(F)(F)CC)N1CCC(OCCNC(C23CC(CC)(C2)C3)=O)C1 c1(C(=O)NC(CSCC)C(=O)N(C)CC2CCOC2C)n[nH]c(C)n1 C1(CNC(c2cccc(OC(F)F)c2)=O)CCCN(C(=O)CCN2CCCC2=O)C1 c1(C(=O)NC(CC)CN(C)C(c2sccc2C(C)=O)=O)cc(Cl)c(N)c(Cl)c1 C(C(C(C)(C)C)NC(c1csc(C(C)(F)F)n1)=O)NC(c1cnc(CCC)s1)=O CC1CN(C(=O)CC2CCN(C)C2=O)CC(C(=O)N(C2CCCCC2O)C)O1 c1(OC)ccc(-c2ccc(CC(=O)N(C)CCc3ncccn3)cc2)cc1CO Cc1nc(NC2CC(C)N(C(c3[nH]nnc3C3CC3)=O)C2)sc1C(=O)OC(C)C c1(CC)oc2ccccc2c1C=CC(=O)NCC1CC1NC(=O)C=C(C)C C=Cc1cc(C(=O)NCCCNC(c2cccc(CCOC)c2)=O)cc(F)c1 C1(CC(=O)NCC(C)(CO)NC(Cc2c(C)scc2)=O)CCCN(C)C1 c1(NC(CC2CC(C)N(C(=O)CC3C(C)(C)C3(C)C)C2)=O)cc(Cl)cnc1O Cc1cccc(OCCC(N2CCCC(C(=O)Nc3ccc(Br)nc3)C2)=O)c1 c1(C(=O)NC2(CC)CCCN(C(=O)CCc3ccsc3)C2)nccc2occc12 C(=O)(C(C)(C)CCCF)N1CC1.CC1CN(C(=O)CN(C)S(N)(=O)=O)C(C)CO1 C(=O)(CCCCCCNC(C1CCCS1)=O)NCC(C)Cn1cccn1 Cc1nn(CCO)cc1C(=O)NC1(C(=O)N(C)CCc2cc[nH]n2)CC1(C)C C1(CC)C(NC(c2cc(C3CC3)on2)=O)CCCN1C(=O)C(c1ccc(C)s1)C N1(C(c2ccc(CC)nc2C)=O)CCC(NC(=O)C=C(C)C)C(F)(F)CC1 N1(C(C(C(CC)C)O)=O)CCn2c(C(N3CCC4(CCCCO4)C3)=O)cnc2C1 N1(C(C2(C)ON=C(C)C2)=O)CCC(C)(NC(C2CCCC(C(C)C)O2)=O)CC1 C(=O)(C1=NOC(CNC(=O)CC2CC3CC3C2)C1)NCc1c(C)nns1 N1(C(COCCC)=O)CC2(CCCCN(C(C3CC34CC(C)(C)C4)=O)C2)C1 Cc1c[nH]c(C(=O)NC(Cc2cnc[nH]2)C(=O)NCCC23CCCC2C3)c1 N1(C(c2ccncc2Cl)C(=O)NC)CCN(C2=NCC(C)S2)CC1 Cc1ccc(CCNC(=O)N(C)Cc2ccc(Cl)c(F)c2)cc1Cl c1(N2CC3(CC(NCc4c(C=C)cccc4)C3)C2)ncc2sccc2n1 C=C1CCC(CNC(C2CCN2C(=O)Cc2cnn(C)c2)=O)C1 N1(C(CCN(CCCO)C(c2c(CC)n[nH]c2)=O)=O)CCC(C)C(C)C1 c1(C(=O)NCC=CCNC(C(CC)OC)=O)cnn2c1OCCC2 N1(C(c2c(C(C)C)cco2)=O)CCC(C)(NC(=O)NC(=O)C(F)(F)F)C1 c1(COC)nccc(=NC(C)C2CCN(C(c3cnc(C)cn3)=O)CC2)[nH]1 c1(N(C(CNC(C2CCN(C(CC)=O)C2)=O)C(C)C)C(C)=O)scc(C)c1Cl.C C1(C(=O)NCC2CC3CN(C(c4scc(C)c4C)=O)CC32)CN2CCN1C(C)C2 Cc1cn2c(C(=O)NCC(C)N(C)C(C3(NC(N)=O)CC3)=O)c(C)nc2s1 C1(NC(c2c(CC)c[nH]c2)=O)CC2C1CCN2C(=O)CCC1C(=O)ON=C1C c1(C(=O)NC2CCCCN(C(C=C(COC)C)=O)C2)c(Cl)ccc2ncccc12 Cn1nnc2c1CCC(C(=O)NCCNC(C1CC3CCC1C31CC1)=O)C2 CCCCCC(O)CC(=O)N(C1CCCN(C(=O)C=C(C)C(C)(C)C)C1)CCF c1(OC(C(=O)NCC(CC=C)NC(c2ccoc2Cl)=O)C)ccccc1OC C1(CC(C)Nc2ccn(C3CCCNC3)n2)CCCCN1 C(=O)(C(C)NC(=O)CNC(C)=O)NC.C1(=O)CCC2(CCC2)N1 N1(C(C=CC(C)O)=O)CC(C2CC2)(C(=O)NCC2CCOCC2(C)C)C1 Cc1ccc(C=CC(=O)NC2C3CN(C(=O)CCc4nc(=N)[nH][nH]4)CC23)o1 c1(C(N2CCC(NC(CCCOC)=O)C23CC3)=O)nn(C)c2ccccc12 C=CC1(CC(=O)N(c2ccccc2OCCF)CC)CN(C(=O)COC(C)C)C1 N1(C(C(c2ccc(Cl)s2)C)=O)CC(F)(CNC(=O)C=CC2CCCO2)C1 C=CC1(C(N2CCC(C(=O)Nc3cnn(C)c3C(=O)OC)C(C)C2)=O)CCOCC1 C(C(=O)Nc1cc(C)ccc1C)(C(C)CC)N(C(CC=C)=O)C N1(C(C(COC)OC)=O)CCC(C)(C)C(NC(=O)Cc2cnns2)C1 C1(C(N2CC(C(N)=O)OCC2)=O)CCCC12CCN(c1ccnc3ccnn13)C2 c1(C2CC(=O)N(C3CCOC3)N2)ccc(F)c(C(=O)Oc2ccc(Cl)cc2)c1 C1(CNC(C(CC)(C)CO)=O)CCC2(CN(C(C3CSC3)=O)C2)O1 N1(C(C=CCC)=O)CCN(C(c2cncnc2CC)=O)C(CCC)C1 C12CCN(CC1C)C2=O.c1(NC(C2CC(C)(COC)C2)=O)cc[nH]c(=N)c1 C1(C(=O)OC)CCC(C(=O)NC2CCN(C(C)=O)C2)N(C(=O)C(F)C(C)C)C1 CCC(O)C(C)C(=O)NC(c1ccccc1F)CNC(c1cc(C)n(C)c1C)=O c1(C(N2C(CNC(C(COC)O)=O)CC(OC)C2)=O)cc2ncccc2cc1Cl c1(CC(C)N(C(CC)(C)C)C2CC2)cccc(F)c1F n1(CC(=O)NCCCC2CCCN2S(=O)(=O)CCBr)ncccc1=O C12(C(=O)NC3(C)CC(NC(Cc4c(C)noc4Cl)=O)C3)CCC(F)(CC1)C2 C12(C(=O)NCC3(NC(c4ccc(C=C)cc4)=O)CC(OC)C3)CCC(C1)C(C)(C)O2 c1(-n2cc(-c3ccc(OC)c(F)c3)nn2)c(F)ccc(Cl)c1N c1(CC)ncc(C(=O)NCCOCCNC(=O)Cc2nc(=N)[nH][nH]2)s1 C(C1CCOCC1)=CC(N1CCC(OCC(N2CC(C)(N(C)C)C2)=O)C1)=O C1(CCC)CCN(C(=NCCc2cccs2)NCC2CN(S(C)(=O)=O)C2)C1 CC1(C(=O)NC(CC(=O)NCCC2(C)CC2(F)F)C2CC2)CC(=O)C1 C1(NC(COCCOCC)=O)C(C(=O)NCC(C)CCO)C1(C)C c1(C(N(CC(COC)O)C)=O)ccc(CNC(C2CCN(C)C2)=O)nc1 N(C(=NCCOC)N1CCC(C2(O)CC2)CC1)C1CCCC(COC)C1 c1(OC)ccc(F)c(C(N2CCCC(CN(C(=O)C(Br)=C(C)C)C)C2)=O)c1F C(C(C)(C)CC(F)(F)F)(c1nnnn1C(C)(C)C)Nc1c(OCC)cccc1F CCCC(C(=O)N1CC(OC)C(NC(c2cc(F)n[nH]2)=O)C1)OCC CCCC(C)(C)CC(=O)NCC1(CO)CCOC1.C1(=O)CCOCCN1 CN1C(=O)OCC12CCN(C(c1cnn(-c3cccs3)c1)C(=O)NCCCF)C2 C12(NC(c3c(C)nc(O)[nH]3)=O)CCCN(C(C3(CC(F)F)CC3)=O)CC1C2 c1(C2CCN2)ccc(C2CCC2)cc1.n1(CC(C)C)cnnc1C1CC1 N1(C(C(C)NC(=O)Cn2cncn2)=O)CC=CC1CNC(=O)C(C1CC1)C1CC1 C1(CC)C(NC(=O)COCc2cccc(C)c2)CCCN1C(c1occc1C)=O Cc1n[nH]c(C)c1CCC(=O)NC1CCCC(C(=O)NCC2CCC(C)C2)C1 C1(CNC(c2c(CC)csc2)=O)CCCCN1C(=O)Cn1cc(C(C)(C)CO)nn1 Cc1nc2cc(C(N3CCN(C(=O)CCCF)CCC3C)=O)cc(Br)c2o1 c1(CC(C(=O)NCC(CN(C(=O)COC2CC2)C)(C)C)(C)C)ccc(C#N)cc1 N1(C(C(C)NC=O)=O)CCC(C)(C(=O)NC2CCCCC2N(c2cnccn2)C)C1 N1(C(C2(CNC(CCSCCC)=O)CCCO2)=O)CC2(CC(CO)CO2)C1 CC1CN(C(=O)C(c2ccccc2)O)CC(C)C1N=c1nc[nH]s1 C1(C(=O)NC(CNC(Cn2c(C)ncc2)=O)C)CC12CCC1(CC1)CC2 CC(C)CS(=O)(=O)CC(=O)N1CC(CNC(C2(F)CCCN(C)C2)=O)C(C)C1 Cc1ccc(C)c2c1OCCC2Nc1ccc(Br)cc1C(F)(F)F N1(C(C2CCN(C(C)=O)CC2)=O)CC2CC(NC(=O)CSC(C)C)C1C2 C1(CNC(CC(COC)(C)O)=O)CC2(CCC2)CN1C(=O)CCc1cc(C)[nH]n1 C(=O)(C(F)(F)Cc1ccc(Cl)cc1)N1CC(C(C)(C)C)C1 N1(CC(c2ccccc2Cl)C)CCC(C(=O)N(C)Cc2ccc(O)nn2)CC1 CCCC(CCC)CC(=O)NCC=CCNC(=O)CCc1ncc[nH]1 C(CCC(N)=O)(C(=O)N1CCN(CCc2ccccn2)C2(CCC2)C1)NC(C)=O c1(C(=O)NC23CC(NC(=O)C(O)CC(F)F)(C2)C3)cc(F)cc(F)c1O C1(NC(C(C)SCCCC)=O)CC(NC(C2CC=CCO2)=O)C(O)C1 Cc1c(C(=O)NC2CCCC(CNC(c3cc(F)ccc3F)=O)C2)cncc1Br N1(C(COCCOC)=O)CCCC1(C)CNC(=O)CCNC(c1ccco1)=O c1(OCC)nc(NCCC(C)(C)C2CC2)ncc1Cl.C1(=O)C(C(=O)OC)N1 N1(C(C2(C)CCOC2)=O)CCCN(CCNC(C2CCCN2C(N)=O)=O)CC1 c1(CC)c(N(C(c2cc3occc3s2)=O)C2CC2)ncnc1Cl.C1(C)(C)CC1 N1(C(C(C(CC)(C)C)=O)=O)CCC2CCCC(C1)N2C(C1COCC(C)(C)O1)=O C1(C(=O)NCC2N(C(CC(=O)OC)=O)CCCC2)Cn2c(C)nnc2CN1C c1(C(=O)NCC(CC)NC(c2[nH]nc(C(F)(F)F)c2C)=O)cc(C)ncc1C CS(=O)(=O)c1c[nH]c(=NC2CN(C(=O)COC3CCCC3)CC2C#N)cn1 C(=O)(C1CCc2ccccc21)N(CCNC(C1CCC(CC)CC1)=O)C1CC1 N1(C(C(CC)(C)OC)=O)CCN(C(c2ccc(-c3ccco3)o2)=O)CC12CC2 C1(NC(c2ccc(OC)nc2Cl)=O)C2CCC1CN(Cc1ccnn1C)C2 N1(C(c2cccc(F)c2F)=O)CCN(C(C2OCC3COCCC23)=O)CC(O)C1 Cc1ccc(S(N)(=O)=O)c(C(=O)NCCN(C(=O)C(C)NC(=O)C2CC2)C)c1 N1(C(CN(CCC)C)=O)CCOC2(CCCN(C(c3ccc(SC)cc3)=O)C2)C1 c1(C(=O)NCC2CC(NC(CC(=C=C)C)=O)C2)cc(Br)cc2scnc12 CC1(C)C(CC(=O)NCCC2(NC(C3CNC(=O)N3)=O)CCC2)CC1O N1(C(C)=O)CS(=O)(=O)CC1C(N1C2CCC1(CNC(c1cn(C)nn1)=O)CC2)=O C1(C(=O)NCCNC(C2(C)CCCOC2)=O)OCC2COCCC12 C(CCC(O)C(=O)NOC1CC1)NC(=O)CN1CC(F)(F)C1 CC(C)(CNC(=O)OC(C)(C)C)CC(N1CC(c2ccccn2)C1)=O C(=O)(C(C)(O)Cc1ccccc1)NC1C(CNC(c2n(C(C)C)ncc2)=O)C1 CCC(CC)C(C)C(=O)NCC1CN(C(=O)Cc2cc(F)ccc2OC)C1 Fc1ccc(F)c(CNCC2CC2c2cccnc2)c1F N1(C(c2c(C)nc(C(C)C)cc2)=O)CC2CN(C(c3cnoc3C)=O)CC2(C)C1 N1(C(C(CCC)O)=O)C(C(=O)N(c2ccc(O)cc2)C)CCC12CC2 C1(C(N2CC(CC)OCC2)=O)N(C(c2cc[nH]n2)=O)CC12CCCC2 C1(c2cn(CC(=O)N(CCOCCC=C)C(C)C)nn2)CCCC(=O)C1 Cc1cc(C)n2ncc(C(=O)N(C)Cc3nc4ccccc4o3)c2n1 c1(CC(N2C(CNC(C3C(C(=O)OC)CCC3)=O)CC2)=O)ccccc1[N+](=O)[O-] C(=O)(C1=C2CCN=C2NC=C1)N1CCC(C(C)NC(c2cncc(C#C)c2)=O)C1 N1(C(CN2CCCC2)=O)CC(C(=O)OC(C)(C)C)C1C(C)C.c1(CS)cccnc1 N1(C(C2(CC)CC2)=O)CCC(C)C(N(C)C(c2cc(C3CCCCC3)[nH]n2)=O)C1 c1(OCC(C)N)ccc(CN2CCC(NC(=O)NN(C)C)C2)cc1 c1(C(N2CC(CNC(C3(C(F)F)CC(=C)C3)=O)C2)=O)c[nH]c2cccc(OC)c12 CC1(CNC(=O)CC2CCCC(=O)N2)CC(F)(F)CN1C(=O)C=C1CCCC1 CCCC(CC)C(=O)N1CC(C(=O)NCCOCC(F)F)C(C)C1 C1(CN(C(C(CC)OC)=O)C)CN(C(=O)Cn2ncc(Br)n2)CCO1 C1(C(N(CCCNC(c2ccc(CSC)o2)=O)C)=O)CC2(C1)CC21CCC1 CCCCC(C)CCC(=O)NC(C)CN(C(=O)CN1CCCNC1=O)CC c1(OCC)ccc(Br)cc1C(=O)NC(c1nc(C2CC2)no1)(C)C N1(CCN(C(NOCCC(C)C)=O)C(c2ccsc2)C)CCc2sccc2C1 N1(C(CN(CC(C)C)C(C2CC3(CCC3=O)C2)=O)=O)CC2(CCC1CO)CC2 c1(CC)ncoc1C(=O)NC(C)(C)C(C)NC(=O)C=C(C)C(C)(C)C C(=O)(C(O)C(C)(C)CC)NC1CC2CN(C(C3(C(=O)OC)CCCC3)=O)CC2C1 C1(CN(C2CCNCC2)C(c2cc(C3CC3)[nH]n2)=O)CCCCC1n1cccn1 CCCCC(F)C(=O)NC1CCCCC1CC(=O)NCC1(C)CC2CC2C1 C=CC(CC)CC(=O)N1CC(O)CC1CNC(C1CCC(=O)N(C)C1)=O Cc1c(C(=O)NCC2CC2NC(=O)CCCc2nccs2)cccc1F C1(CC(=O)NCC)C(=O)NCCN1C(=O)C(=O)NCC1CCC(C(=O)OC)CC1 CC(CC(F)(F)F)C(=O)NC1CCC(CNC(c2ccc3[nH]ccc3n2)=O)CC1 c1(C(=O)NCC(CNC(c2cc(C)nc(O)n2)=O)F)ccnc2cc[nH]c12 Cc1nc(=NC2CCCCC2C(F)(F)F)s[nH]1.c12coc(n1)CNC2=O C#Cc1cccc(NCC(N2CCCC(NC(=O)CCCc3cccs3)C2C)=O)c1 N1(C(C=Cc2ccn(C)c2)=O)CCCC12CCN(C(C1CCC(C)(C)CO1)=O)C2 N1(C(c2c(C)ccs2)=O)CCC=C(C=O)C1.c1(NCC)cc(Cl)ccc1C(F)(F)F C1(C(=O)NCC2(OC)CC2)COCC1NC(C1(CO)CCCO1)=O CC1(CCNC(C2C=CCS2)=O)CCN(C(=O)COC2CC2)C1 c1(C(=O)NCCN(C(=O)C(c2ccc(F)cc2)F)CCC)cnc2[nH]cnc2c1 N1(C(C2N(C)CCC2)=O)CCCC(O)(CNC(c2ccc(C(F)F)cc2)=O)CC1 C1(N(C2CCCC2)C)(C(=O)O)CC12CCC2.C(C=C(Cl)Cl)N(CC(=O)O)CCO c1(C(=O)NC2CN(C(c3cncs3)=O)CC2O)cc(Cl)c2cc[nH]c2c1 c1(C(=O)NC2CN(C(c3c(C(C)C)ccs3)=O)CC2O)cc2c(F)cccc2s1 Cc1ccc(SCCC(N2CC(c3ccccc3Br)C2)=O)c2ccccc12 c1(CC)cscc1C(=O)NC1CCCC1CC(=O)NCC1SCC=C1C C1(CNC(C2(CC)CN(C(C3CC(O)CN3C)=O)C2)=O)COCC(C)O1 C1(NC(c2ccc(COC)o2)=O)CN(C(=O)C(F)CC2CCOC2)CC1C c1(CNC2CCCN(C(c3ccc(C)cc3O)=O)C2)cc([N+](=O)[O-])c(C)cc1C C1(C(N2CCN(C(C(=O)NC3(C)CNC(=O)C3)=O)CC2)=O)CCC(F)(F)CC1 c1(C(=O)NCC2CC(NC(C=CC=CC)=O)C2)c[nH]cc1Br C12(NC(c3c(OC)cc(C)s3)=O)CCCC(NC(c3cnc(Cl)s3)=O)(C1)C2 c1(C(N2CC(C)C(CNC(=O)C(=O)N(C)C)C2)=O)cc2cccc([N+](=O)[O-])c2[nH]1 N1(C(C2C3(CCN(C(c4c(C)ocn4)=O)C3)C2)=O)CC2CC(C(=O)O)C(C2)C1 N1(C(CCC=C)=O)CC2(CC(CC(=O)N(CC)CC3CCCCC(O)C3)C2)C1 Cc1cccc2c1CC(NC(=NCc1cc(C3CCCC3)nn1C)NC1CC1)C2 N1(C(CN(CC(c2ccccc2)(C)F)C(C)CC)=O)CCOCC1 Cc1cc(CNC(=O)CC2(CN)CCCCC2)nn1C Cc1cc(CNC(=O)C(=O)NC(c2cnn(C)c2)C)c(C)s1 CCC(C)(C)C(O)C(=O)NC1(CC(=O)NC2CCn3cncc3C2)CC1 N1(C(CCC(CC)OC)=O)CCC(C2CC2)(CNC(c2cccs2)=O)C1 N1(C(C(=O)N(c2cccnc2)CCOC)=O)CCC(c2ccc(C)s2)C1 C1(C(F)(F)C(=O)N(CCCNC(=O)CCOc2ccccc2)C)(OC)CCCC1 N1(C(c2ccc(C#C)o2)=O)CC2CC(NC(=O)C(N3CCN(C)CC3)C)C1C2 C1(CC)CCN(C(=O)C(CSC)OC)C(C(N2CCC2C)=O)C1 C1(=O)C(C(C)C)NC(=O)CNCC(=C)CCN1.c1(C(C)OC(C)=O)nccn1C c1(-c2cc(C)c(F)cc2F)n[nH]c2cccc(C(=O)Nc3cnnc(C)c3Cl)c12 C1(C(=O)NCC(CC)(CC)NC(=O)C(C)N2CC(C)C2)CC2C=CC1C21CC1 C1(CCCNC(c2ncn(CC)c2)=O)CN(C(c2nnsc2SC)=O)CCO1 Cc1ccc(C(=O)NCC2CN(C(=O)Cc3ccccc3F)C3CC23)c(O)n1 C(=O)(C1CCCn2cc(C)nc21)NCC1N(C(c2ccc(OC)c(N)n2)=O)CC1 N1(C(c2c(N)non2)=O)CCOC(CCNC(C2CC3CC3C2)=O)C1 C(CC(CNC(=O)C(C)(C)NS(C)(=O)=O)NC(=O)C(O)Cc1ccccn1)OC c1(C(=O)NCC2C3CN(C(COC(C)=O)=O)C2CCC3)ccc2cnccc2c1 C12(NC(C(CC=C)C)=O)CCCC1N(C(=O)CC1(OC)CCC1)CC2 CC1=NOC(CC(=O)NCC2(CC(=O)NCCc3cnc(C)[nH]3)CC2)C1 CC(C)C(F)C(=O)N1CCC(CNC(=O)C(c2ccccc2Cl)O)CC1 N1(C(c2cccc(C)c2O)=O)CCC(C2(NC(=O)C(n3cc(Cl)cn3)C)CC2)C1 Cc1cc(C(N2CCN(CCNC(c3ccc(F)s3)=O)CC2)=O)c2c(c1)CCC2 CC(CS(C)(=O)=O)C(=O)N(C(C)CN(C(=O)CCc1ccc(O)nn1)C)C CC1CN(C(=O)CC2(C)CCOC2)CCCN1C(c1ccc([N+](=O)[O-])nc1)=O C(c1cc(Cl)cc(Cl)c1)=CC(=O)NCC1(O)CC(NC(C(=O)N(C)C)=O)C1 CCC(CC(=O)N1CCCCC(C2CNC2)C1)CC(F)(F)F C12(C(=O)NCCC3CCN(C(C(COC)OC)=O)C3)CC3CC1C2C3(F)F n1(CC)cnc2c(NCc3nc(C)sc3C)nc(N3CCC(C)CC(C)C3)nc12 c1(CN(C(CCC2(NC(C(C)OC(C)=O)=O)CCC2)=O)C2CC2)cnn(C)c1 c1(C(=O)NCCC(C)N(C(=O)Cc2cc[nH]n2)C)cc(Cl)c(F)cc1N O(N(C(=O)C1CC(C)(C)CN1C(=O)CC(C)C(F)(F)F)C(C)C)CC N1(C(C2(CSC)CC2)=O)CC(CNC(C2(C)CC=CC2)=O)C(F)(F)C1 CCCCCCCS(=O)(=O)N1CC(Sc2ncc(-c3ccccc3)o2)C1 Cc1ccc(SCC(N2CCC(Nc3nccc(CC#N)n3)C2)=O)cc1 CC1(C)CC=C(C(=O)NC2CC2NC(C2CC3(C2)CC(C)(C)C3)=O)CC1 CCC(C)CC(C(=O)N1CCCCC1C)NC(=O)CC(C)(C)C(C)=O c1(C(C2CC2)NC(=O)C(N2CCCC(N3CCCCC3)C2)=O)ccc(F)cc1F C12(NC(C3CC(C#N)C3)=O)CCCC1CN(C(c1sccc1Cl)=O)C2 c1(OC)ccccc1NC(=O)C(c1cccc(Br)n1)N1CCC(C#N)C1 c1(NC(c2ccc(CN3CC4C(CC(=O)OC)C4C3)o2)=O)ccc2n[nH]cc2c1 N1(C(CC(CC)C)=O)CCC(c2ccccc2)(CNC(c2cc(C#N)no2)=O)CC1 N1(C(c2ccc(C(C)=O)s2)=O)CCOCC1CNC(=O)C(C1CCOCC1)C c1(C(=O)NC(CC)C(OC)OC)cc(S(=O)(=O)N2CCCCC2)ccc1N c1(C(N2CCCC(CNC(=O)C(F)F)CC2)=O)cc(S(=O)(=O)NCC2CC2)c[nH]1 c1(-c2nnc(C)o2)ccccc1C(=O)NC(CNC(C12CCC1C2)=O)CO N1(S(CC(=O)OC)(=O)=O)CC2(CN(C(=O)Cc3cccc(Br)c3)CC2CO)C1 C1(C(N2CCCC(CCNC(C3(C)CC3(F)F)=O)C2)=O)CCCC12CCOCC2 C(CN=C(NC1CCS(=O)(=O)C1)NCc1csc(-c2cccs2)n1)C1C(C)C1 c1(-n2cc(C(C)NCC(CC(F)F)c3ccccc3)nn2)cccc(C#N)c1 c1(C(=O)NC(CCC)CC(=O)NCCCOC(=N)O)cccc2[nH]ncc12 N1(CC)CCc2c(Sc3ccccc3Cl)cccc2C1=O.N12CCCC1C2 c1(N(CCCNC(C2CCC(C)C2)=O)C(C)C)nnccc1C#N Cc1cc(C(N2CCN(C3CN(C(=O)CC(C)(C)O)C3)CC2)=O)ncn1 C1(NC(C(C)C(F)F)=O)CN(C(c2cccc(OC3CC3)c2)=O)CC(C)(C)C1 C1(C(N2CCC(C(C)(C)NC(CCn3ncc(C)c3)=O)C2)=O)COCCC1(F)F c1(CNC(=O)NC2(C(CS)(F)F)CCC2)n[nH]cc1CC(=O)OC(C)(C)C.N(C)C c1(NCC=CC)[nH]c(=NC(C)CC2CCCCC2)nc2c1cnn2C C1(C(=O)NC(C(C)NC(=O)Cc2ccc(CO)cc2)C)CC2(CCCCC2)CO1 C(CCCCCCO)(C(=O)NC1CCCOC1)N(CC(=O)NC)CC c1(C(=O)NC(CN(C(C2N(C(C)=O)CC2)=O)C)C)cccnc1 C1(C(=O)NC2C(F)CCN(C(c3c(C)scc3)=O)C2)CCc2[nH]nc(O)c2C1 c1(C(N(CCOCCC(=O)N(C)CCC2CCCC2O)C)=O)cn(C)c(=O)cn1 c1(CC)cc(C(=O)NC(C)(CNC(C2CCS(=O)(=O)N2)=O)C2CCC2)ccc1F N1(C(c2cnc(C(C)C)s2)=O)CCC(NC(=O)CCSC2CCCC2)C(O)C1 CC1(C)CCC(C(=O)NC2CCN3CCOCC23)N(C(=O)OC(C)(C)C)C1 C1(NC(CCC(=O)NC)=O)CCN(C(=O)Cn2cnc(C(N)=O)n2)C12CC2 C(=O)(CCCCCCCCCO)N1CC2CN(C(c3c(CC)onc3)=O)C2CC1 CC1CN(C(=O)Cc2ccccc2I)CC1NC(C1CN(C(N)=O)C1)=O Cc1nn2c(c1C(=O)NCCCN(C)C(c1coc(Cl)n1)=O)CCCC2C c1(C(=O)NCC(N(C)C(C2CCC(C)(C)OC2)=O)C2CC2)ccc(Cl)c(C#N)n1 C1(C(=O)NCC2CCN(C(C=CCN(C)CC)=O)C2)CCCC2(CCCCC2)C1 c1(CC(N2CC3CC3(CNCc3ccc(O)nn3)C2)=O)cccc2ncccc12 N1(C(C(Cc2cn[nH]c2)NC(c2cnccn2)=O)=O)CC(F)(F)C1C1CC1 CN1CCN(C(C2CN(C(=O)COc3ccc(O)cc3Cl)CCO2)=O)C(CO)C1 C12(CNC(CC3CCC(C)C3)=O)COC(CNC(=O)C3=COCC3)(C1)C2 C12CC3CCC1(C3)NC(=O)Cn1nccc1-c1cn2nn1.c1(CC)cc(C)c(Br)o1 C1(C(N(C)CCNC(=O)Cc2ccno2)=O)CCCC(F)(F)CC1 Cn1cnnc1CCCC(=O)NC1COCC1NC(c1cc[nH]c1C1CC1)=O C1(C(=O)NC2CCN(C(=O)CN3CCCC3CO)CC2)CCCC2(CC2)C1 CC(F)(F)C(C)(C)C(=O)NC1COCCC1NC(c1ccon1)=O c1(-c2ccc(CNC3CON(CC)C3=O)cc2)ccc(-n2cccn2)c(C)c1 C(C)(C)(CC(F)C(=O)NCCc1cncs1)NC(C(C(C)C)SC)=O c1(C(N(C(C)C(N2CCC(c3cnco3)C2)=O)CCC)=O)cc2ccccn2c1 Cn1cc2c(C(N3CC(NC(=O)C4=NOC(c5ccccc5)C4)C3)=O)cccc2n1 Cc1ncoc1C(=O)NCC(=O)NCC(C)N(C(=O)CN1CCCC1=O)C C1(NC(C2(OCC)CCCC2)=O)CN(C(=O)Cn2ncccc2=O)CCC1CO C1(C)(NC(CC=CCNC(CCSCC)=O)=O)CCN(C)C1=O C1(NC(=O)CCC2CCCN2C(=O)CCc2cn[nH]c2)CCC(=O)NC1 c1(C(=O)NCC2N(C(CC(C(N)=O)NC(C)=O)=O)CCCC2)c(C)cc(O)cc1C C1(C(=O)NC(C(=O)NC(C)C(C)(C)CO)CO)CC2(CCC2O)C1 c1(NC(N(C(c2ncoc2C)C(F)F)CC)=O)ccc2nc(C(F)(F)F)[nH]c2c1 CCC(=O)NNC(=O)C(C)N.C(C(C)O)OCCCC C1(NC(C2CN(CCOC)C(=O)C2)=O)CCN(C(c2c[nH]nc2C)=O)CC1O C(CCC(=O)NC(c1n[nH]c(CO)n1)C)(C(C)C)NC(C(c1ccc(C)o1)C)=O C12(CC1)CNC(=O)CC(=O)NC(=O)C1C(C1)C2.N(C1CC1)(CC)CC CC1CCCC(C)C1NC(c1cc(CNC(C2CCN2C)=O)ccn1)=O C1(C(N2CC3C(CNC(C4C=C(C)CS4)=O)(C3)C2)=O)CC2CCCC2C1 C1(C)(NC(C2C3N(C(c4cnc(C)s4)=O)C(CC3)C2)=O)CN2CCC1CC2 C1(CCNC(c2nc(C)sc2)=O)CCCCN1C(c1cnnn1C)=O Cc1cn2c(n1)CC(C(N1CC(NC(c3c[nH]nc3Br)=O)CCC1C)=O)C2 N#Cc1ncc(Br)cc1NC(C1CCN(C(=O)C=Cc2cccnc2)C1)=O CCCC(CNC(c1c(C)nsc1N)=O)C(=O)NC(c1nc[nH]n1)C1CC1 c1(Oc2cccc(C(=O)NCCC(C)N)n2)ccc(Br)cc1F.C(=O)(CO)OCC N1(C(c2ccc(OC)cc2)C(=O)Nc2ccccc2)CCc2c(nccc2Br)C1 CN1CC(C(=O)NCC(C2CCCCC2)N)NC1=O.c1(O)ccccc1.C1(=O)C=CC1 C(CC(C(C)(C)C)NC(=O)CC1(C(F)(F)F)CC1)N(C)C(C1CC=CC1)=O C1(C2C(C(=O)NCC(C)(C)C3CCC3)C2)CCCN1C(=O)CSCCC#N N1(C(C2(C#N)CC2)=O)CC2CC1C2NC(c1sccc1F)=O CC1OC(=O)NC1C(N1CCCC(C(=O)NCC2C(CO)C2(C)C)C1)=O c1(NC2CC(NC(c3c(C)[nH]nc3Cl)=O)C2)ncnc2cccc(Br)c12 C1(C(=O)NC(CC=C)C2CC2)CC12CCN(C(=O)C=Cc1cc[nH]n1)C2 c1(C(N2CC(C)C2)=O)cnc2nc(NCC=Cc3ccc(C#N)cc3)ccc2c1 N1(C(c2cc(CC)c(F)cc2)=O)CCN(C(C2CCC3(CC3)C2)=O)CC(O)C1 N1(C(C)=O)CC2CCC(C1)N2C(c1cc2c(ccn2C)[nH]1)=O CP(C)(=O)c1cccc(=NCC2(c3ccc(O)cc3Cl)CC2)[nH]1 Cc1cc(C)c(C(=O)N(C(CNC(c2ccc(C(N)=O)[nH]2)=O)C2CC2)C)c(S)n1 C1(C(N2C(C)(C(=O)Nc3n(C)ncc3)CCC2)=O)CSC(c2ccccc2)=N1 C1(n2cc(C(N(C)C)=O)nn2)CCCN(C(c2cscn2)=O)C1 CCC1(CC)CCNN1.C(=O)(C(C)(O)COC)C(=O)C=Cc1cn(C)nn1 c1(-c2scc(CC(=O)NCCCN(C(CC(C)N(C)C)=O)C)n2)cccc(Cl)c1 NS(=O)(=O)c1ccsc1C(=O)NCC1CCC(NC(C2CC(F)(CO)C2)=O)C1 Cc1cccc2c1CC(C(=O)NCC1CN(C(C3(C)CCCCCC3)=O)C1)N2 C1(C(=O)NCC(C)NC(C2CCN(c3ccccc3)C2)=O)COC(C)C1 c1(NC(CC2CCN(C(C3C(C)=CCC=C3)=O)C2)=O)cc(C#N)ccc1I c1(C(N2CCCCC(NC(C3C(COC)C3)=O)C2)=O)ccc2nc(C)cn2c1 N1(C(c2c(CNC(CC3CC(C)(C)C3)=O)ccs2)=O)CC2CC=CC1C2 C1(NC(c2ccon2)=O)CCCCN(C(c2cc3ccncc3[nH]2)=O)CC1 N1(C(C2C(C)(C)CO2)=O)CC2CN(C(c3cccn4cnnc34)=O)CC2(C)C1 c1(C(=O)NCC2COCCN(C(C3(C)N(C)CCC3)=O)C2)coc(S(C)(=O)=O)c1 CCCCCCNC(C1CC(C(=O)OC)C1)=O.n12cc(cn1)CNC(=O)C2 C1(C(C(=O)NC2(CC(=O)OC)CC2)C)CCN(C(=O)C(C)(C)SC)C1 N12C(=O)NC(C(C(=O)OC)=C1c1cn(C)cn1)c1cc(N)c2cc1I.CCC CON=C(C(=O)N1CC=CC(NC(c2cc(C(F)(F)F)cs2)=O)C1)c1ccco1 C1(C(F)F)(NC(c2cscn2)=O)CCN(c2ccnc(CCC)n2)C1 C(=O)(C1CCCc2nc[nH]c21)NCC(C(C)C)NC(Cc1c(C)noc1Cl)=O C1(C(N2CC(N(C(=O)CC3(C)CCOC3)C)C2)=O)CC(OC(C)(C)C)C1(C)C N1(C(Cc2ccc(C)s2)=O)CCCC2(NC(c3cnn(C)c3F)=O)CC2C1 C1(CNC(=O)Cc2c[nH]nc2O)CC2C1CCN2C(=O)Cc1ccc(Cl)nc1 N1(C(C2CNC(=O)N2)=O)CCC2C(CCN2C(c2ccc([N+](=O)[O-])o2)=O)C1 C1(OC)CC(CC(=O)N(C)CCNC(=O)C(F)(F)Cc2ccc(F)cc2)C1(C)C C12(C(N3CCC(CN(C(=O)CC4(C)CC4(F)Cl)C)C3)=O)CC(CO)(C1)OC2(C)C Cc1cc(C(=O)N(C)CCNC(c2c[nH]nc2C2CCC2)=O)c(N)c(F)c1 CC(C)C(CC1CC1)N=c1[nH]c(=NCc2c(Cl)cncc2Cl)[nH]c2cccnc12 C1(C(N2CCC(NC(CCc3ccc(SC)cc3)=O)C2)=O)CN(S(N)(=O)=O)C1 c1(C(N2CC(N(C(=O)CCc3ccnn3C)C)C(O)C2)=O)[nH]nc2c1CCC2(C)C C(=O)(N=c1ccn(CC2CC2)[nH]1)C1N(C(C)(C)C)CC(O)C1.N12CCC1C2=O C(=O)(C(C(C)C)N(C)C)N1CC(O)(CN(C(C(C)NC(COCC)=O)=O)C)C1 C1(=CC(=O)OC2(C)CN(CC(=O)N(CCOC)CCO)C2)CCC(C)(C)CC1 N1(C(c2onc(COC)n2)=O)CCN(C(=O)C(CO)C(C)C)CC(O)C1 C1(CC)(C=O)CCCN1C(=O)N(C(C)CC)C.N1(C(=O)OC(C)(C)C)CCCC1 N1(C(C(COC)OC)=O)CC(OC)CC1CNC(=O)C(Cc1ccsc1)NC=O CC1(C)CC(CC(=O)NCC2CCN(C(c3cnc(C(F)(F)F)s3)=O)C2)CCO1 O=C(C1=NOC2(CCN(C(=O)COC(F)(F)F)C2)C1)NCc1cc(F)cc(Cl)c1 C1(CNC(C2(C)CC(F)C2)=O)CN(C(c2c[nH]nc2Cl)=O)CCO1 O(S(=O)(=O)c1ccccc1)CC(CC1C(=O)NC(c2ccc(Br)cc2)CC1)O c1(C(=O)NCC2CC(NC(c3cncnc3)=O)C2)cc2c(s1)CCSC2 C1(CNC(CCCC(C)=O)=O)CN(C(c2cc(N)ccc2F)=O)C2CCCC2O1 c1(N(CC)CC)nnccc1C(N1CCC(C)(C(=O)N(CCCOC)C)C1)=O Cc1cc(C(=O)N(C)CC2COCCN2C(=O)CCCC2CC2)ccc1F C1(NC(C2(C)CCSCC2)=O)CCN(C(C2CC=CCC2)=O)CC1CO N1(C(=O)NC(CC)CF)CCCCC1c1nc(O)n[nH]1 C(=O)(C(C)(F)CCCC)N1CCC(CN(C(C(C=C)(C)C)=O)C)C1 c1(C(=O)NCC(C2CCCC2)NC(C2C(C)OCC2)=O)ccc(CC2CC2)nc1 Cc1nccc(C(N2CC(N(C)C(c3nnn(C(C)C)c3C)=O)C(O)C2)=O)n1 C1(C(N2CCCC(CNC(=O)Cc3nccs3)C2)=O)CC1C1CCCC1 C12CN(C3CC13)CCCNC2.Cn1nccc1NC(C(C)NC(=O)CCCF)=O N1(CC(=O)NCCOCCOC)CCOCC1=O.C1CCCCN1C.c1(C)ccccc1 C1(C(N2CC(NC(c3coc4c3CS(=O)(=O)C4)=O)C2)=O)CCc2[nH]nc(O)c2C1 c1(C(N(C(CN(C(c2cncc(OC)c2)=O)C)C)C)=O)ccc2oc(C)nc2c1 N1(C(C2C(CC)CCC2)=O)CC(C(=O)Nc2cc(C#N)ccc2F)C2(CCC2)C1 c1(CNC2CC(C(=O)NCCS(=O)(=O)N(C)C)C2)ncc(Br)cc1F C(C)(CN=c1[nH]c(=NCCC(C)CCO)[nH]c2ccccc12)Oc1c(C)cccc1 CC(C(CC1CC1)C(=O)NC1CNC(=O)C12CC2)NC(C(n1c(C)ncc1)C)=O CC(C)(CO)C(C)(C)NC(C1CCCCN(C(=O)C=Cc2ccncc2)C1)=O C1(OC)CC(F)CN(C(=O)CC2CCCN2C(=O)CC2(C)CC2)C1 N1(C(C2N(CCC)CCC2)=O)CCC(C(N2CC(CO)C(C)C2)=O)(CF)C1 C1(=CC(=O)NCCC2(C)CCN(C(C(=O)NCC)=O)C2)CCC(C)(C)CC1 c1(OC)ccc(NC(C2(NC(=O)CC3CCOC3)CCSC2)=O)cc1 N1(C(C(C)(C2CC2)OC)=O)CCC(C(=O)NCCC(C)N2CCC2)C(C)C1 C1(C(N2CCOCC(F)(CNC(=O)C(F)F)C2)=O)CCOCC12CCC2 C#Cc1cccc(CN2CCN(CCCC(C)C)CC2)c1 c1(CCCC)ccc(O)c(CN2CC(F)(F)CC2CO)c1 C(=O)(C(N=[N+]=[N-])C(C)C)N1C(C(N2CC(COC(C)=O)C2)=O)CCC1 N(C1CC2(CN(C(c3ccc(C)cn3)=O)C2)n2ccnc21)C(CCCC(=C)C)=O Cc1cc(C(=O)NC2CC(CNC(=O)C(F)=C3CCC3)C2)c2[nH]cnc2c1 CC1(C)CN(C(c2cc(Cl)ns2)=O)CC(CNC(=O)Cn2cnc(=N)[nH]2)O1 C1(C(=O)NC(C)CC#N)CCCC(Nc2cc(-n3ccnc3)ncn2)C1 c1(C(=O)NCCCN(C(C2(CSC)CCCO2)=O)CC)cnnc2ccccc12 C(=O)(C(=O)CC(C)CC)NC1CCCC(C(=O)NC(CC#C)CO)C1 c1(C(=O)NCC(CC)N(C(=O)C(O)CCC(C)C)C)c(C)cc(C)cc1C CCCCCC(O)C(=O)NC(C)(CNC(=O)C=CCOC)CO CC1CC(=O)NCC1C(=O)NCCN1CCCN(C(=O)CCN2CCCC2)CC1 C=CCC(C)(C)CC(=O)NCCn1cc(C(=O)NC(CO)CC(C)(C)C)nn1 C1(NC(c2ccc(Cl)cn2)=O)C2CC3C(C2)C13C(=O)NC1CCCC(CO)C1 c1(C(=O)NCCOCCN(C(=O)Cc2cnccn2)C)ns[nH]c1=O Cc1nc2cc(C(=O)NCC(C)(CO)NC(=O)CC3CCC(=O)N3)cnc2[nH]1 Cc1cc(C(=O)Nc2cnc(F)cc2C(=O)NCc2ccc(O)cc2)ccc1O c1(CC(=O)N(C)C)ccc(Cn2cc(-c3ccc(CCN)cc3)nn2)cc1 C(=O)(CN1C(=O)Cc2ccccc21)N1CC(C(N(c2nccs2)C)=O)C1 C(N=c1nc(N(CCS(C)(=O)=O)C)c2c([nH]1)CCC2)c1c(O)ccc(C)c1 N1(C(c2c(COC)cccc2)=O)CC2CN(C(C3CC3(F)F)=O)CC2(C)C1 C#CC1(C(=O)NCCc2cccc(O)c2)CCN(C(c2nnn(C)c2C)=O)C1 c1(C(N2CCN(C(COCC(=O)NC)=O)CC(O)C2)=O)cccc2ccn(C)c12 N1(C(C(C)(C)NC(c2ccc(Br)cc2)=O)=O)C2CCC1C(N)C2 c1(C(N2CC(C(Cn3cc(CCOCC)nn3)F)C2)=O)ccc(C)cc1 CCC(C)C(O)C(C)C(=O)N1CC(C(N2CCC23CCC(O)CC3)=O)C(C)C1 N1(C(C2C(C=CC)CN(C(C3CCN(C)C(=O)C3)=O)C2)=O)CC2CC(O)CC2C1 C1(NC(N(CCC)Cc2cccc(Br)c2)=O)CC2CC3C(C2)C13 N1(C(COC2(C)CN(C(CCn3ccc(C)n3)=O)C2)=O)CCC(F)(CN(C)C)CC1 C1(C(=O)NCC(CC(=O)NCc2cnns2)C2CCC2)CC2(CCO1)CC2 c1(C(=O)N(CC2C(NC(c3ccc(NC)cc3)=O)C2)C2CC2)ccc2nncn2c1 c1(N2CCC3(CCN(C)C3)C2)nc(N2CC3(C)COCC3(C)C2)nc2c1COC2 C1(CC)C=CCCN1C(=O)N(CCN1CCCCC1)C1CC1 N1(C(COCCCCCC)=O)CCC(CNC(C2(O)CCC2)=O)C(C)C1 N1(C(C(C)N2CCC2)=O)CCN(C(c2ccn(CCO)c(=O)c2)=O)C(CCO)C1 C1(C(=O)Nc2c(C)c(I)ccc2)CC(=O)N2CCCCC12 C1(CC)CN(C(c2scnc2C(C)(C)C)=O)CCC1NC(=O)COC(F)(F)F O=C(NNc1ncnc(C2CC2)c1Br)N(CCCc1ccc(F)c(Cl)c1)CCO Cc1nc(Cl)ccc1S(=O)(=O)N1CCC(NC(=O)CC2COCC(C)O2)C1 S(=O)(=O)(c1ccc(NCCc2ccsc2)c(F)c1)NC(COC)C(C)C C(=O)(CCCC(CC)NC(C1(CN2CCC(OC)CC2)CC=CC1)=O)OCC N12CCC3C(C3C1)C2=O.N#Cc1ccc(C(N2C3CCC2(C(=O)NC)CC3)=O)[nH]1.CO N1(C(COCCSC)=O)CCC(C=CC(=O)N(CC(F)F)CCO)CC1 Cc1nccc(C(=O)NCC2CC2NC(=O)COCC2CCCOC2)c1N N1(C(C2ON=C(C)C2)=O)CCC(NC(c2cc(Br)no2)=O)C(C)(C)C1 CCCC(CCCNC(=O)COCC1CCC1)NC(c1cncc(OC(C)=O)n1)=O c1(C(C(=O)N(CC2(CNC(C(C=C)O)=O)CCC2)C2CC2)(F)F)ccccc1Cl C(=O)(C(C)CC(C)C)NC1CN(C(CCCOCCOCCOC)=O)CC1C C1(NC(c2cccnc2F)=O)CCCN(C(C2(C(=O)OC)CC2)=O)CC1 N1(C(C2C(CC)CCC2)=O)CC(C)(C)CC1CNC(=O)CC1CC(O)C1(C)C C(=O)(C(O)P(C)(C)=O)NCC(CNC(C=CCN(CCOC)C)=O)OC c1(N2CC(C)(CNC(c3c(OC)cc(Cl)nc3)=O)C2)ncc2cn[nH]c2n1 C1(C(=O)NCCCC(=O)NCCSC)C2CC1N(C(=O)CCn1ccnn1)C2 Cn1cc(C(=O)N(CCC(=O)N(C2CC(O)C23CCC3)CC2CC2)C)ccc1=O C(=O)(CCCCC(=O)NC)N1C(CC)C(C(=O)NCC(O)(C2CC2)C2CC2)CC1 Cc1nc2ccc(C(N3CC4CCCN(C(=O)C(C)CN(C)C)C4C3)=O)cc2o1 C1(CC(=O)NCCC(CNC(c2cnc(CC(C)C)s2)=O)O)CCCCC1F c1(C(=O)NC2COC2)ccc(F)c(Cl)c1.O=C1C(F)(F)COC2CCN1CC2 N1(CCNC(C(C)N(C(=O)C(F)=C2CCCC2)CCC)=O)CCCC(O)C1 c1(C(=O)NCCN(CCC)C(c2ccn(CC)c(=O)c2)=O)cc(C#N)ccc1C c1(C(N2CCC(F)(C(=O)Nc3cnn(C(F)F)c3)C2)=O)cccc(C2CC2)n1 CC1CCN(C(N)=O)C1.C(CC(=O)NCC(=O)N)N(C(C1(C(F)(F)F)CC1)=O)C C(CNC(=O)CC1(O)CCCOC1)(C(C)(C)C)NC(C(C)N(C(C)=O)C)=O C1(CNC(N(C(c2c(C)cccn2)C)C)=O)COc2ccccc2O1 C1(CCNC(C(CN(C)C)NC(c2cc(C(F)F)[nH]n2)=O)=O)CCCC2CC12 C(=O)(C1CCCc2n[nH]cc21)N1C(CNC(c2ccc(CC)cc2F)=O)C=CC1 CC1c2ccccc2CC1C(=O)NC1CCN(C(=O)C=Cc2cccn2C)CC1 C1(CC(N2C(CNC(CN(C)C3CC3)=O)CCC2)=O)Sc2ccccc2NC1=O N1(C(CC(=C)C)=O)CC(NC(=O)Cc2cncn2C2CC2)CC2(CC2)C1 c1(CCC)cc(C(=O)N(C)CCNC(=O)Cc2cccnc2C)ccn1 CCC(C(=O)N(CC(N1CCC(CSCC)C1)=O)C1CC1)N(C)C c1(OC)ccnc(C(=O)NCC(C)CC(=O)N2CCOC(CC(N)=O)C2)c1 CC#CC1CCN(C(=O)CC2CCCN(C(=O)CCCNC=O)C2)C1 N1(C(CSCC#C)=O)CC(O)(CC(=O)NCc2nccn2CC)C1 CC1=C(C(=O)N2CC(C(=O)NCC3(F)CCCCC3)CCC2C)CCC1 n1(CC(N2C(CNC(C3CCC(F)(F)C3)=O)C=CC2)=O)ccc2ccc(F)cc12 c1(C(N2CC3CC(CN(C(=O)CCCF)C3)C2)=O)nc(C(F)(F)F)n2ccccc12 C12(C(N3C4C(NC(CNC(C)=O)=O)CC(CC4)C3)=O)CC3CC(C(=O)N1)C2C3 C12(C(C)C)CCC(NC(C)(COc3ccccc3)CO)C1C2 CCCC(C(=O)N(CC(N1CCC1C(C)O)=O)C(C)C)NC(N)=O N1(C(CCC(C)=O)=O)CCC2(CC1)CC2C(=O)NC1COC(C2CC2)C1 CC(O)(CC(=O)N1CC2=C(C1)CN(C(=O)COCCCN=[N+]=[N-])C2)C(F)(F)F N1(C(c2c(CC)nns2)=O)C2CCC1C(C)C(NC(c1ncccc1SC)=O)C2 c1(C(=O)NC2CCN(C(C3C(CC)N(C)CC3)=O)C2)cc(O)nc2cnccc12 Cc1cc(N)ccc1C(N1CC(NC(=O)Cc2cnc(Cl)cc2C)C2(CC2)C1)=O C1(CCNC(C(C)(C)C2CCC2)=O)CCN(C(=O)C(N2CCCC2)C2CC2)CC1 C1(CNC(C2C=CC(C(=O)OC)C2)=O)COCCN(C(=O)C#CC(C)(C)O)C1 C(=O)(C(F)CC(C)(C)C)NC1CCCC(N(C(CC2CC(SC)C2)=O)C)C1 c1(CNC(c2nnc(COC)s2)c2nnnn2CCSC)ccc(F)nc1C C1(C(N2C(COC)C(C)(C)C2)=O)CNC(=O)CN1C(=O)Cc1scnc1C c1(C(N2C(C)CC(NC(=O)CC3(C)OCCO3)C2)=O)ccn2nncc2c1 N1(C(COCCC)=O)CC(F)(C(=O)NCC(C)OCCO)C1 c1(C(C2(n3cccn3)COC2)NCC(C)Cn2cccn2)nnnn1CCOC.C1CC1 C1(CN(C(c2ccco2)=O)C(c2ccccn2)=O)CCCN1C(=O)CC1CC1 C(=O)(C1=CS(=O)CCC1)N1CC(NC(=O)CC(c2ccccc2)N2CCC2)C1 CC(C)C(N=[N+]=[N-])C(=O)NCC1COC(CNC(=O)C(C)c2cncs2)C1 C1(C(=O)OC)(C(=O)OC(c2n[nH]cc2C(C)C)=O)CC(C)C1.OC c1(CC)cc(C)c(NC(=O)CSc2cccc(CC)c2)cc1C c1(NC(C(CC)OC(c2cc(Br)no2)=O)=O)cc(Cl)ccc1Cl N1(C(C#CC2(CC)CC2)=O)CCC2CN(C(c3cnc(C)cn3)=O)CC2C1 Cc1cc(C(=O)NCC2CCCSC2)c(C)o1 N1(C(c2ccc(C#N)[nH]2)=O)CCC2CCCC12C(N)=O.C1(CN=[N+]=[N-])C(=O)N1 C(=O)(CC(C(F)F)NC(=O)CCC(N)=O)N1CCC(NC(C)=O)CC1 c1(-c2ccc(NC(=O)NC(CSC)CO)o2)ccc(F)c(F)c1 c1(C(N2CCCC(CN(C(c3scc(C)c3Cl)=O)C)C2)=O)ccc(F)nc1F c1(C2(C(=O)NCC3C(CNC(CC=CC=C)=O)C3)CC2)ccn(C)n1 C1(C(=O)OC)CC(C(=O)N(C)CCNC(c2cccc(Br)c2F)=O)C12CCC2 C1(C(=O)NCC(C)(C)OCCO)CCN(C(C2CC2Cl)=O)C1 C(c1cccc(Cl)c1)=CC(=O)NC1(CC=C)CN(C(C2(C)CCCS2)=O)C1 C1(C(=O)NCC2CC2c2ncon2)CCC(C2CC2)N1C(c1cnsc1)=O c1(OC)ccc(CNC(C2CCN(C(c3cc(Cl)nc(Cl)c3)=O)C2)=O)cc1Br C1(NC(C2CNC(=O)O2)=O)CN(C(=O)Cc2cn[nH]c2)CC1C1CC1 Cc1nn2c(C(N3CCC(CNC(c4ncccc4Cl)=O)C3)=O)c(C)nc2s1 c1(C(=O)NC2(CC(=O)NCC3CC3(Cl)Cl)CCC2)nccc2[nH]ccc12 C(=O)(C(C)C(=O)N1CCOCC1c1ccc(C(=O)NCc2cc[nH]n2)n1C)OC C(=O)(CC(C)CC(=O)N1CCCC1CN(C)C(c1cccc(F)c1SC)=O)OC C1(CCCN2C(=O)CN(CC3(c4occc4)CCC3)C2)SC2=NCCN2C1=O C(=O)(CCCn1cc(CNC=O)nn1)OC(C)(C)C c1(CNC(C2(C)CC=C(C)CC2)=O)nc2c(s1)CN(C(c1ccoc1)=O)CC2 N1(C(c2cc(CC)[nH]n2)=O)CC2C(NC(c3cc(CC)sn3)=O)C(COC)C2C1 C1(NC(C(c2cccc(C)c2)O)=O)CCC(C)N(Cc2cc(C)on2)C1 C(=O)(C1CCCn2c(CC)nnc21)NC1CC(CNC(COCCC)=O)C1(C)C c1(C(=O)NCC2(F)CN(C(C34CCC(CC3)CO4)=O)C2)cc2ccc(Cl)cc2o1 N1(C(CCCN(CCC)CCC)=O)CC2(CC(NC(C3CCN(C)C3C)=O)C2)C1 C1(C(=O)NC(CNC(C2(CCCC)CCC2)=O)(C)CO)CS(=O)(=O)CC(=O)N1 CC(C)(C)C(=O)C(=O)NCC1CN(C(C2(Cl)CC2(F)F)=O)C1 C1(CCOC)(C(N2CCC(O)(CCNC(=O)C(C)(C)CF)C2)=O)CCN(C)CC1 S1(=O)(=O)c2ccc(cc2)N1.CC1(C)CN(S(C)(=O)=O)CCC1CO C(=O)(C(F)(CNC(=O)CCC1CC(OC)C1)C(C)C)NCC(C(CC)C)C N1(C(c2cn(CCCC)nn2)=O)CC2C3CCC(C2C1)N(C(=O)CNC(C)=O)C3 CCC(C)(C)CC(=O)NC1CC(CNC(=O)C(O)Cc2cccc(Cl)c2)C1 C=CC1(C(=O)NC2(C(=O)O)CCC2)CCC1 C1(C(N2CC(NC(C(C)(C)N(C)C)=O)C(F)CC2)=O)Cc2ccccc2S1 C=CCC(C)(O)C(=O)NCc1cccc(C(=O)NCC2(C)NC(=O)NC2=O)n1 C(=O)(C(C)N(OC)C(=O)CCCCC1CN(C(=O)CN2CCCC2=O)C1)OC C=CCN=c1[nH]cc(C(=O)NCCN(C)C(C2CC3CCCCC23)=O)s1 c1(C(N2CCN(C(c3c(C)nsc3)=O)CC2CC#N)=O)cccc2ccn(C)c12 C(Cc1ccccc1)(CCC(=O)O)NC(Cc1ccc(C)cc1)(C)O c1(C(=O)NCC2CCN(C(c3n[nH]c(CC)c3Cl)=O)C2)cc2cccn2cn1 CC(C)C(CCc1ccccc1)(c1nnnn1C1COC1)NCC1C=CCCCC1 N1(C(c2cc(C)cc(Br)c2)C(=O)NC(C(=O)OC)C)CCc2ccc(F)cc21 N1(c2n(CC)c(C3CCCCO3)nn2)CCC(F)(F)CC12CC2 N1(N(CC(C)(C)N(C)C)C)CCC(C)(C)CC1C=O.c1(C(=O)NCCF)ccncc1F CC(C)(O)C(O)C(=O)NC1(c2ccccc2)CCN(C(=O)Cc2nso2)CC1 c1(C(=O)NC(CCN(C(=O)C=Cc2cccs2)C)(C)C)ccc(C2CC2)cn1 CCCCCCC(C)C(=O)N(C1CCN(C(c2cnc(C3CC3)s2)=O)CC1)CC C12(NC(c3cc(CCC)ncc3)=O)CCCC1N(C(c1cc(Cl)cnn1)=O)CC2 C=Cc1cc(C(=O)NCC(C2CC2)N(C(=O)C(COC)CC)CC)cc(F)c1 N1(C(C2(C)CCCS2(=O)=O)=O)C2CCC1CC(CN=c1ncc(F)c[nH]1)C2 Cc1ccc(Br)c(CN2CCC(F)(C(=O)NC(C#N)C(N)=O)C2)c1 CC1CCCC(CC(N2CCC(CC(=O)NC34CCN(CC3)C4)C2)=O)O1 C1(C(N(CC(CO)(CO)NC(c2nccc(C)n2)=O)C)=O)CC(C2CCC2)C1 C1(NC(CCCOCCC)=O)C2CCC1N(C(C1CCCCN1C)=O)C2 c1(-n2cc(C(N(C)C)=O)nc2)cccc(NCC2CCC3(CC3)C2)c1 C(CCNC(C1COCC1C(N)=O)=O)(CNC(=O)C(C)c1ccco1)OCC CCC1=NOC(C(=O)N(c2cc(C)c(C)s2)C(C)C(N2CCC(N3CC(O)C3)C2)=O)C1 c1(OC)ccc(C(C)=CC(=O)NCCC(O)CNC(=O)CSCCN(C)C)cc1 C12(CC)CCN(CC1)C(=O)Cn1nccc1C(=O)N1CCC(C1)CC(=O)N2.NC C1(CC(=O)NCc2cc(OC)no2)CCCC(CNC(c2cnsc2C)=O)C1 c1(C(c2nc[nH]n2)NCCC=C)nnnn1CCOCC Cc1cnccc1C(=O)NCC(O)CN(C)C(c1cc(C)n(C)c1)=O CC(CC(=O)N1CC(S(C)(=N)=O)C1)CC(F)(F)F.c12cn(nn1)CO2 c1(C(=O)NC2C(CNC(C(C)CS(C)=O)=O)CCC2)ccc(F)c(O)c1F C(=O)(C(C)(O)CC(C)C)NCCC1(NC(C2CCN(CC)CC2)=O)CCC1 c1(C(=O)NCC(CC(=O)OCC)C)cc(I)ccc1O Cn1nnc2c1CC(C(=O)NCCC1(NC(=O)CC3(O)CCOC3)CCC1)CC2 CC1CC(NC(c2c[nH]nc2CNC(=O)CCc2csnn2)=O)C(C)CN1C C(N=c1[nH]c(=NCCNS(=O)(=O)N(C)C)[nH]c2c1COCC2)C1C(C(CC)OC)C1 C1(F)(C(=O)NC(C2CC(NC(C3CCC(C)CC3)=O)C2)C)CCCN(C)C1 C(=O)(CCCS(C)(=O)=O)N1CC(N(C(C2CC=C(C)CC2)=O)C)C2(C1)CC2 C1(C(=O)NC2C(OC)CC2O)CC2(CCN1C(=O)C(F)C(C)(F)F)CC2 c1(CC)cnccc1C(N1CC(NC(c2nc(Cl)sc2C)=O)C1)=O C(=O)(C(CC(F)F)NC(c1cc(C(N)=O)co1)=O)NCC(C)(O)C(F)F C(=O)(CC(C)n1ccnc1)NC(C1C(C(N(CCC(=O)OC)C2CC2)=O)C1)C C1(C(N2CC3C(CNC(c4c(CC)ccs4)=O)(C3)C2)=O)CC(C)CC(C)C1 c1(C(N2CCN(C(=O)Cn3ccnn3)C(C(F)F)C2)=O)cnc2ncccc2c1 c1(OC(C)C(=O)NC(C)(C)Cc2ccc(I)cc2)ccc(Cl)c(F)c1 C#Cc1ccnc(C(=O)NC(CC(=C)C)C(=O)NCc2ccn(C(C)C)n2)c1 n1(CCOC)ccc2ccc(C(=O)N(CCC(=O)O)CCO)cc12 Cc1cc(=NCC2(S(=O)(=O)N3CCOCC3)CC2)[nH]c(=NCC2OCCC2C)[nH]1 N1(C(C(C(C)C)NC(COCCOCC#C)=O)=O)CCC12CCOCC2 C1(C(N(CC(O)CNC(c2ccc(CO)nc2)=O)C)=O)CCc2nc(O)[nH]c2C1 c1(C(=O)NCC2N(C(c3ccc(SC)o3)=O)CC2)cc(F)c2cn[nH]c2c1 C1(CNC(c2ccc(CCF)cc2)=O)COCCN(C(=O)CC2CCCC2)C1 C1(NC(C2C(C)OCC2)=O)CCOCC1NC(c1coc(Cl)c1)=O CC(C)C(=O)C(=O)N1CC2C(NC(=O)C(C)Oc3ccc(Br)cc3)C2C1 C=C1CCN(C(=O)CC2CC=CC2)C(C(=O)NC2CC2C2CCC2)C1 c1(CN(C)CC2CCN(C(N3CCC(CO)CC3)=O)C2)ccc(S(C)=O)cc1 c1(OC2(C(=O)NC3CCC(NC(=O)COC4CC=CC4)C3)CC2)ccc(F)c(F)c1 c1(C(=O)NC2CC(N(C(c3scc(OC)c3)=O)C)C2)cccc[n+]1[O-].C(=O)N C1(C(=O)OC)CN(C(=O)C(F)(F)C2(NC(=O)OC(C)(C)C)CCNC2)CC12CC2 C1CCCCC(=O)NOC(=O)N1.CC(C)(C)CCN.C12CC1C(=O)N2 CC1CN(C)CCCN1C(=O)Cn1cc(CNC(C2(C#N)CCOC2)=O)nn1 C1(C(=O)NC2C(CNC(C3CC(C#N)C3)=O)CCC2)CCC(CC(F)(F)F)CC1 C1(NC(CC2(CC)CCC2)=O)CC(C(=O)N(C2CC(SC)C2)C)CC1O CN1CCCCC1C(=O)NNC(=O)NCc1ccc(OCC(F)F)cn1 C1(C(=O)NC(c2nc(C)[nH]n2)(C)C)(NC(=O)C(C)C2CC2)CCN(C)C1 N1(C(=O)CCCO)CCN(C(C2CC(F)(CO)C2)=O)C2CCCCC2C1 C(=O)(C1CCCc2nncn21)NC1C(CNC(=O)Cn2cnnc2O)C1 N1(C(C2CCN(CC)C2)=O)CC(C)C(C)(CNC(c2[nH]cc(C)c2C)=O)C1 C1(NC(C2C(C=C)OCC2)=O)CCN(C(c2c(N)cccc2F)=O)CC(C)(C)C1 C1(NC(Cn2c(C(C)C)ncc2)=O)C=CCN(C(C2CNC(=O)N2C)=O)C1 C1(C(=O)NC2C(OC)CN(C(=O)Cc3c[nH]nc3C)C2)COCC2(CCC2)O1 C1(C(N2CC(=C)C2)=O)CCC(CC2CC2)N1C(c1cnns1)=O C1(C(N2CCC(N(C(CCCN=[N+]=[N-])=O)CCO)C2)=O)CCn2cncc2C1 c1(C(=O)NCC(CN(C(=O)CC2CCCN(C)C2)C)O)cccc(CF)c1 Cc1c(Cl)c(C(=O)NC2CCC(NC(C34COC(CF)(C3)C4)=O)C2)nn1C Cc1cc(Cl)c(C(N2C3CCC2CC(NC(C2(CC#N)COC2)=O)C3)=O)cc1C N1(C(c2cc(CCC)nn2C)=O)CCN(C(C2(CC)CCCC2)=O)CCC1C CC(=O)CCCC(=O)N1CCC(C(=O)NOCCC(C)C)(C(C)C)C1 Cc1cccc2c1CCCC2NS(=O)(=O)c1c[nH]ccc1=NC1CCCC1C1CC1 N1(C(CSCCN(C)C)=O)CC(NC(c2c[nH]c(Br)c2)=O)C2CC12 c1(C(=O)NC(CC)CN(C(=O)C(C)OCC2CC2)C)cccc(CC(F)(F)F)c1 n1(C(C2CCCCC2)C)nc(-c2cccs2)nc1-c1ccon1 CC1CN(C(C2(C)CC3CCC2C3)=O)CCC1NC(C1CC2CCC1C2)=O c1(C(N2CCCN(C(CC3(OC)CCC3)=O)C(C)C2)=O)cnn2c1C(=O)CCC2 N1(CCOC)CC2CC(NC3CC(C)CN(SCC)C3)CC2C1 Cc1cc(F)c(C(N2C(C(=O)Nc3cnn4cccnc34)CC3CC23)=O)c(F)c1 n1(CC(C)C)ncc(C(=O)NC(C)C(C)NC(C2(c3cccnc3)CC2)=O)c1N C1(NC(CC=C)=O)CCCN(C(=O)C(O)Cc2ccccc2Cl)C1C c1(C(C)NC2CCN(Cc3ccsc3C(=O)O)C2)ccnc2cc(Cl)ccc12 c1(C(N2CC(O)(c3nnc(-c4ccccc4)o3)C2)C2CC2)cccc(Cl)c1 c1(C2(CC3(COC)CCCN3C(=O)OC(C)(C)C)CCC2)ccc(F)c(Cl)c1 N1(C(CCC)=O)CC2(CCC2)CCC1C(=O)NNC(=O)Cn1ccc([N+](=O)[O-])n1 C(=O)(C(C)(C)CNC(C1C2CC1N(C(C1CCCC(=O)C1)=O)C2)=O)NC C(=O)(C(C)(C)CC=O)NCC1CC1.c1(CC)cc(C)c(C(=O)N(CCC2CC2)C)o1 N#Cc1ccc(C2CC2C(=O)NCc2ccc(OC3CCC3)cc2)s1 c1(C(N(C2CCCCC2NC(C2(n3cncn3)CC2)=O)C)=O)c[nH]c(=S)cn1 C1(CNC(C(C=C)(C)O)=O)CC(C)(C)CN1C(=O)Cc1ccc(O)nc1 c1(C(=O)NC2C(NC(C3CC(=C)C3)=O)CS(=O)(=O)C2)cccc2c1oc(=O)n2C C1(NC(c2c(C)scc2)=O)CC(O)CN(C(c2ccccc2C(C)C)=O)C1 N1(C(c2nnc(C)s2)=O)CCOC(CCNC(c2c(C)nsc2N)=O)C1 Cc1coc(C)c1C(=O)N(C1CCN(C(=O)CCc2nc(C)no2)C1)C c1(CCNC(CN(CC(COCCC)O)C)=O)ccc(C)c(O)c1 n1(CC)cccc1C(=O)N(C)CCOCCN(C)C(C1(C)CC1C(F)(F)F)=O CC(C)CC(O)C(C)C(=O)NCc1cccnc1C(N1CC(O)CC1(C)CO)=O n1(CC)cnc2nc(N3CC4CSCC4C3)nc(N(CC#CCOC)C)c12 c1(N(C(=O)C(=O)NCC2(OC)CCCSC2)CCOC)cc(Cl)c(C)cn1 CC1OC2(C)CC1(C(=O)NC13CCC1CN(C(c1cccnc1N)=O)C3)C2 c1(-c2nnc(C(C)OC)o2)cccc(CNC(N2CCCCC2C(C)(C)C)=O)c1 N1(c2nnc(COC)n2CCCOCC(F)(F)F)CCC2C(C1)C2(F)F C(=O)(C1=NN(C(C)C)C(=O)CC1)NCC1N(C(c2occ(C)c2)=O)CC2(CC2)C1 C1(NC(C2C(C=C)C2)=O)CC(NC(C23CCC(OC)C2C3)=O)C(O)C1 C1(C(=O)NCC2CC(NC(CC(C)CN(C)C)=O)C2)CCC2(CCCC2)C1 C1(C(N2C(C(=O)Nc3c(C)nsc3)CCC2)=O)OCCCC1(C)C N1(C(CCSCC(C)C)=O)CCCN(C(c2cnc3nccn3c2)=O)CCC1 c1(C(=O)NC(CCCC)COC)ccc(F)cc1N c1(C(=O)NC(CN(C(=O)CSCc2nc[nH]n2)CC)C)ccc(C)nc1O C1(CC)C(C(=O)NCCCc2ncccn2)CCCN1C(c1c[nH]c(=O)cn1)=O CC1=C(C(=O)NC2CC3(C2)CC3C(=O)NCCC(C)C(C)C)COCC1 N1(C(C2C(C)(C)N(C(=O)C(F)CC3CCOC3)CC2)=O)CCc2cccc(O)c21 C(=O)(C(CC(F)F)n1cccn1)N1CC(OCCNC(C(C(C)C)F)=O)C1 C1(C(N)=O)(CNC(CC=CC=C)=O)CC=CC1.C12(CCC1)C(=O)NC2 Cc1cc(C(=O)NC(C(N2CC3(CCN3C)C2)=O)c2cccs2)ncc1N C1(C(F)(F)F)(OC)CCCN(N2CC3(CCOCC3)OCC2C)C1 c1(C(=O)NC2CN(C(C3N(C)CC(O)CC3)=O)CC23CC3)ccnc2c1CCO2 C(=O)(C(C)CC(C)C)N(CC(C)NC(C1CC(OC)C1)=O)CC C(C)(C)(C=CC(=O)C1C(C(N)=O)C1)COC(CNC(COCC=C)=O)(C)C C(=O)(C1=CC2CCCCC12)N1CCC(NC(c2ncc3ccccn23)=O)(CF)C1 c1(C(=O)NC23CCN(C(c4c(C)nc[nH]4)=O)CC2C3)cc2c(o1)CCCNC2=O c1(C(=O)O)ccc(CNC2CCC(N3CCOCC3)C2)cc1 C1(C(N(CCOC)C)=O)CCCCCC1NC(c1cc(C#N)cn1C)=O C(=O)(CCCC(F)(F)CO)N(C1CCCN(C(=O)CC2CCC(C)C2)C1)CC c1(CCCC)nc(C)c(C(=O)NCCOCCNC(=O)Cn2c(C)csc2=O)s1 c1(NC(C2CCCN(C(=O)Cc3cccnc3)C2)=O)cc(F)c([N+](=O)[O-])cc1F c1(SC)ccccc1C(=O)NCC=CCSCCNC(=O)CC1CC1 c1(C(N2CCC(NC(C(c3ccc(Cl)cc3)C)=O)CC2)=O)c(Cl)nn(C)c1Cl C1(NC(C2N(CC#C)CCC2)=O)CC2CC(C1)N(CCCC(=O)OC)C2 c1(C(N2C(CCNC(=O)COC(F)(F)F)CCCC2)=O)c(F)ccc2n[nH]cc12 N1(C(C2(C#N)CCCO2)=O)CC(F)(F)CC1CNC(=O)CCC1CCCCCC1 c1(CC)c[nH]c(C(=O)NC(c2ccccc2)CNC(=O)C=CCSC)c1 N1(C(CC(C=C)C)=O)CCC2(CC2NC(c2cc(C3CC3)no2)=O)C1 c1(OC)ccccc1C1(C(=O)N(C(C)CN(C)C(c2nc(C)sc2C)=O)C)CC1 c1(OC)cc(CNc2ccc(C(=O)Nc3nc(C)cs3)nc2)ccc1C c12ccc(Cl)c(c1)NC2=O.C1(O)(CC(=O)NC2CCCC2CCO)CCCOC1 C(CC(C)(C)C(=O)N1CCC(N(C)C)C(C)C1)NC(C)=O N1(C(=O)OC)CCCC(C(N2CC3CC3(NC(C3CCCN3C)=O)C2)=O)C1 Cc1cc(S(=O)(=O)N2CC(C)(C)OC(C)(C)C2)ccc1-c1cccnc1 C#Cc1ccc(C(=O)NCC2CCN2C(=O)C(C)N(C)C(C)=O)cc1 N1(C(CC2(C)CCCO2)=O)CCC2(CCN(C(c3cnc(N)c(Cl)c3)=O)CC2)C1 c1(C(N(C2CC(NC(C3C(=C)CC3)=O)C2)C)=O)cc(Cl)cs1 Cn1ccc(C(N2CC3CC2(C(N2CC(C)OCC2C(C)C)=O)C3)=O)cc1=O.C N1(CCNC(C2(C=C)CC2)=O)CCCC(O)C1.C12CC(CO1)C(=O)N2 c1(CC(=O)NCCC2(CNC(CSCC#C)=O)CC2)ccccc1C c1(C(=O)NCc2cc(-c3cccc4c3CNC4=O)[nH]n2)ccc2c(c1)C(=O)NCC2 C1(C2CN(C(C3CC3Cl)=O)C2)(NC(C2CCCCC2)=O)CC1 C1(OC)COCC1N=c1[nH]c(=NCC2CC3C(C2)C3(F)F)[nH]c2ccsc12 CCCC(C(=O)NC1C2CN(C(=O)CNC=O)CC12)S(N)(=O)=O CC1C(C(N2CCCC(CCCCNC(=O)CSS(C)(=O)=O)C2)=O)CCN1C c1(CCC(=O)NCCCN(C(C2(N(C)C)CC2)=O)C(C)C)cc(SC)c(C)o1 c1(C(N2C(CNC(C(CCCOC)C)=O)CC(F)C2)=O)cc(C)c(O)c(C)c1 C(CCC)(CCCNC(=O)CN(S(C)(=O)=O)C)NC(C(C)SC)=O N1(C(CCCC2C(C)C2)=O)CCN(C)CC1CC1CN(NC(=O)C2CC2)C1 N1(C(CC(CCSC)O)=O)CC(CNC(=O)CN2C(=O)CCC2=O)CC12CCC2 c1(C(N(C)Cc2ocnc2CNC(=O)CC2CCC(O)C2)=O)cnn(C)c1N c1(C(N2CC(O)CC(NC(C3CC4C=CC3C4)=O)C2)=O)c(Cl)ccc2ccoc12 C=CCCC(C)(C)CNC(c1cncn(C)c1=O)=O N1(C(C(C)S)=O)Cc2[nH][nH]c(=NC(=O)Nc3ccc(F)c4c3CCC4)c2C1 c12cccc(c1)CNC2=O.C(C(=O)NCC1(N(C)C)CC1)OCCOC N1(C(C2(C)C(C)(C)C2)=O)CC2CCCN(C(=O)CCc3cccc(Cl)c3)C2C1 Cc1cc(Cl)c(C(=O)NC2CN(C(=O)C(C)n3ccnn3)CC2O)cc1C C1(CNC(C=C(COC)C)=O)CCCN(CC(=O)NC2CCCC2)C1 Cc1cc(CC2CCN2C(=O)NCC2CCOC2)n(C)n1 CC1NC(=O)CCC1CNC(C1CCN(C(C2CCCCC2)=O)CC1)=O CC1CC2(CC(C(N3CCCC(NC(C4(Cl)CCC4)=O)C3)=O)C2)C1 C(C(C)(CC(=O)O)NC(c1ccc(C(C)(C)C)cc1OC)=O)OC c1(C(=O)NC(CSCC)C(=O)N(C)CC2CCCCC2)nc(C)ccc1C C#CCCCC(C(=O)OC)N1CCN(C(C#N)C(=O)c2cc(C)on2)CC1 CC1CC(NC(=O)C=CC2CCCN2C(=O)CSC(F)(F)F)CCC1(C)C C1(C(=O)NCC(N(C)C)C2CC2)CN(C(=O)CN2CCOC2=O)CCC1(C)C C1(NC(C2C(NC(C(CCC)OCC)=O)CCOC2)=O)CCC(N=[N+]=[N-])CC1 c1(CC(=O)NCC(C)N(C(C=Cc2nc(C)c(C)[nH]2)=O)C)ccccc1S(C)=O Cc1ccc(-c2cc(C)c(C(=O)NCC3CCCN3C(C3CCOC3)=O)s2)cc1 c1(C(=O)NCC(=O)N(CC(O)CNC(C2CCCS2)=O)C)ccc(Cl)cc1 N1(C(CC(C)F)=O)CCC2(NC(=O)CSc3cccc(F)c3)CCCC12 S(=O)(=O)(c1c(F)ccc(C)c1F)Nc1c(C(=O)OC)scc1C CC(CCCN=c1[nH]c(=NC)[nH]c(=NCC2(C(F)(F)F)CCC2)[nH]1)N(C)C C1(CC(=O)NCc2cccc(OC(F)(F)F)c2)CC2OCCC2O1 c1(C(=O)NC(C2CC3CCC2C3)C#N)cc(C(=O)O)c(Br)cn1 c1(C(=O)NCCOC2CCN(C(c3nc(CC)oc3)=O)C2)nnn2c1CCC2 N(C1COc2ccccc21)C(c1cc(C)ccc1C)(c1nnnn1C1CC1)CC c1(C(=O)NCCNC(C2(C(=O)OC)CC2)=O)nnn2c1CCC2 N1(C(Cc2c(C)n[nH]c2C)=O)CC23CCCC2(C1)CN(C(=O)CSC(F)(F)F)C3 C(=O)(CC(C)(C)C(F)F)NCC1CC(C)N(C(=O)Cc2ncsc2Cl)C1 C1(C(=O)NCCOCCN(C)C(C2(C)CCCS2)=O)(COC)CCOC1 Cc1cccc2[nH]c(CNc3cccnc3C(=O)Nc3c[nH]nc3Cl)nc12 Cc1c(C)n(C)c2cccc(C(N3CCCC(NC(C4(F)CC4(F)F)=O)C3)=O)c12 C1(COC)(CNC(c2n[nH]c(C)c2C)=O)CCCN1C(c1[nH]cnc1C)=O Cc1cc2[nH]c(C(=O)NC3C4CC3CN(C(c3ccc(F)cc3Cl)=O)C4)cc2o1 C=CC1OCCCC1C(=O)NCCC1CCN(C(=O)C=CC)C1 CCC(CCC(=O)NC(C)CC(C)O)OC.c12cccc(c1)NC2=O c1(SC)nc(N2CCC(NC(C3CCN(C)CC3)=O)C(C)C2)cc(Cl)n1 c1(-n2ccc(CC(=O)NCCn3cc(C4CCCCO4)nn3)n2)ccc(F)cc1 C(CC(=O)NC(c1cncs1)C)(CC(C)C)NC(c1c(C)nncc1)=O C(c1ccc(C(=O)NC2CN(C(c3ccsc3)=O)CC3CC23)nc1)=CC(=O)OC c1(OC)ccc(CNC(Cc2nonc2C)C(C)C)c(F)c1 C=CCC(C)C(=O)N1CCC(C(CO)NC(C2CC(C(F)(F)F)C2)=O)CC1 c1(C(=O)NCC2N(C(C=C(C)CN3CCCCCC3)=O)CC2)cncc(N)n1 CC(C)(C(=O)N1CC2(CCN(C(c3coc(CS(C)(=O)=O)n3)=O)C2)C1)S(C)(=O)=O c1(C(=O)NC(CNC(C(C)NS(C)(=O)=O)=O)(C)C)ncc(F)cc1N c1(CC(=O)NC2CC(N(C(=O)C(O)C(F)F)C)C2)ccn2cncc2c1 C1(CNC(c2cnc(CC)s2)=O)CCN(C(C2CC2c2sccc2C)=O)CC1C C=C1CC(C(=O)N(CC(C)N(C(=O)C(C)CNC(=O)O)C)C)(C(F)F)C1.CC Cc1csc(C(N2CCC(CC(c3ccccc3)C)C2)C(=O)NCCC2CC2)n1 c1(C(C(=O)NC2C(NC(C(CSC)(C)C)=O)C2)C)ccc(F)c(Cl)c1 Cc1nc(C)n(CCCC(=O)NCCC(C)NC(=O)C=CC(=O)N(C)C)n1 c1(C(=O)NC(C(=O)NC2(CCOC)CC2)CCF)cc(C)nc(C)c1 BrC1=CC=CCN2C1OCCC1(CC1)C2CCC C1(OC)CC(C)CN(C(C2(C)CC(O)CN2C(=O)C(C)=NOCC#N)=O)C1 c1(NCc2c(C)ncs2)[nH]c(=NCC2CCCC3(CC3)C2)nc2c1ncn2C(C)C CC(C)(O)C(C)(O)C(=O)NC1CCN(C2CCN(C(=O)C3CC3)CC2)CC1 CC(F)(F)C(F)C(=O)NC(C)(C(=O)NCCc1ccccn1)C1CCC1 N1(C(c2cnc(C)c(C#N)c2)=O)CCOC2(CCN(C(=O)C(C)(C)F)C2)C1 Cc1c(C(N2CCC(CCC(=O)NCC(O)CN(C)C(C)C)CC2)=O)ncn1C C1(CC)CN(C(c2ccc(OC)nc2Cl)=O)CCN1c1ncccn1 CC1CCCCC1C(N1CCC(C)(NC(c2cn(C3(C(=O)O)CC3)nn2)=O)C1)=O c1(OCC)cc(C(N2CCC2CNC(c2cnc(C)c(C)c2)=O)=O)ccc1Br c1(C(C(=O)NC)N(C(C)C(=O)NC)CC2CC2)cncn1C C(=O)(C1CCCc2ccccc21)NCC1N(C(C2C(C)(C)CC(=O)NC2)=O)CC1 CC(C)(CNC(C1CCCO1)=O)CCNC(c1ncoc1C1CC1)=O C#CCC(C(=O)NC(CCF)C(=O)NC(c1ncc(C)cn1)C)C1CC1 c1(C(=O)NC(CC)(C)CNC(C2CC2C(C)(F)F)=O)cncc(C#N)c1 C12(NC(c3c(C)cccc3Cl)=O)CCCN(C(C3CCCC(=O)N3C)=O)CC1C2 C(=O)(C#CC(C)(C)O)N(C)CC1CCCCN1C(c1cn(C(C)(C)C)nn1)=O c1(CC)ncc(C(=O)N(C2CCC(NC(c3nc(O)sc3C)=O)CC2)C)c(O)n1 C(N=c1[nH]cnc(Cl)c1OC)C1CCC(CNC(C(CC=C)N(C)C)=O)CC1 CC1(CNC(C2CC(NC(=O)Cn3ccnc3)CC2O)=O)CC2CCC1C2 C1(C)(CNC(C2(NC(=O)OC)CCCC2)=O)CCN(C(c2cnn(C)n2)=O)C1 c1(C(N2CC(C(C)NC(C(C)OCC)=O)C2)=O)cc(C#N)c(F)cc1F C1(CC(=O)NCCC(F)Cl)(NC(=O)CC2CCC(O)C2)CCCCC1 C1(NC(C(C2CC=CCC2)C)=O)CCCCC1c1ccc(F)cc1 C1(C)(C(ONC(C2CC(=O)OC23CCC3)=O)=O)CCCNCC1.CO N(C(=NCCc1ccsc1)NCC1CCOC1)Cc1n(C)nc(C(F)F)c1 C(=O)(CC(C)C(F)(F)F)NC1CC(C(F)F)(NC(C2(COCC)C=CCC2)=O)C1 CCCC(O)C(CO)NC(=O)C1=CCN(C(c2n[nH]c(C)c2C)=O)C1 N1(C(c2nn(C)c(C3CC3)c2)=O)CC(NC(=O)Cn2cnnc2)C2CCCCC12 N1(C(c2c(CC)n(C)cc2)=O)CC2CCCC1CN(C(=O)Cn1nc(C)oc1=O)C2 C1(C(=O)NCCn2ccc(C(=O)NCCC3C(C)C3)c2)CCC(=O)C(C)C1 N1(C(c2ccn(C)c2C(F)(F)F)=O)CCn2cc(C(=O)Nc3cn[nH]c3)nc2C1 N1(C(C2(C(=O)NC)CC2)=O)CC2(C)CN(C(C3(CCC)CCCC3)=O)CC2(C)C1 N1(C(CCC=C(C)C)=O)CCC2(C1)CN(C(c1cn3c(n1)CCC3)=O)CC(C)O2 N1(C(C(C)C2CC2)=O)CCC(CNC(c2ccn3ncnc3c2)=O)C12CCC2 N1(C(c2cc(Cl)ns2)=O)CCC2(C1)CN(C(=O)CCc1ccc[nH]1)C2 C1(NC(=O)CC2CC2(Cl)Cl)CC2CCC1(NC(c1cc(Cl)cs1)=O)C2 N1(C(C(=O)NCC#C)C)CCC(NC(=O)COC(c2cn(CC=C)nc2)=O)CC1 C1(c2cn(-c3nccc(C)n3)nn2)COCCN(C(c2occc2C2CC2)=O)C1 c1(CC(=O)NC2CC3CC2N(C(c2ccco2)=O)C3)ccc(Br)cc1F Cc1ccc(CC(=O)NCC2C3CN(C(=O)C(C)(C)CO)CC23)cc1Br CCC(CCC(=O)N1CC(Cn2cc(CC3CCOCC3)nn2)C1)OC c1(CC)cc(C(=O)NC2CCCC(c3ccc(Cl)cc3)C2)ccc1Cl C(CCN=C(NCCCN(C)C)NCC1CCC(C)O1)SC N1(C(c2ccc(OCC)nc2O)=O)CCC(=C(F)F)CC1 N1(C(c2c(CC)n[nH]c2)=O)CC(NC(C2(OC)CCS(=O)(=O)C2)=O)CC1C N(C(=NCCCCl)NCC(C(F)(F)F)N1CCOCC1)CC.c12ncc(s1)CN2 N1(c2nc(C)nc(Cl)c2)CC(NC(=O)C2=C(Cl)CC2)C2CCCCC12 C1(C#C)(C(=O)NCCCC#C)CCN(C(=O)C(C)C(C)C)C1 C1(N(C(c2c(C)nco2)=O)C)CCCN(C(C2CC2c2sccc2C)=O)C1 N1(C(CCC(C)(C)NC(C(n2ccc(C)n2)C)=O)=O)Cc2cccc(F)c2C1 c1(N(C(C2C(NC(CCOC)=O)CCC2)=O)C)cc(C)cc(F)c1 C#Cc1ccc(C(=O)NC(C)CNC(C2(C)CC2C)=O)cn1 c1(NC)ccc(C(N2CCC(CN(C(=O)C(C)CC3CC3)C)CC2)=O)cc1 C1(NC(C(=O)N(C)C)=O)CC2CCC1N2C(=O)C(F)(F)c1ncccn1 C1(C(=O)NCC(CC=C)CC(C)C)CN(C(c2cc(C)cc(C)n2)=O)CCC1(C)C N1(C(c2cc(C)[nH]n2)=O)CCN(C(=O)Cc2ccc(Cl)cc2Cl)CC1C(C)(C)C N1(C(=O)CCc2cncnc2)CCC2C1CCN2C(C1CCC(F)(F)C1)=O C1(C(N(CCCCN(C(Cn2ccc(C)n2)=O)C)C)=O)CC2(C1)NC(=O)NC2=O N1(C(C(C(=O)OC)F)=O)CCC2(CCC(NC(c3ccc(C4CC4)s3)=O)C2)C1 N1(C(CN(CC(C)C)C(c2ccn(C3CC3)n2)=O)=O)CCCC2(CC2)C1 N(C)(S(=O)(=O)N(C)C)CC(=O)NCC1N(C(C=Cc2nc(C)sc2)=O)CCC1 C1(N(C(C(C(C)C)SC)=O)C)CCCCN(C(c2ccc(C)nc2O)=O)C1 C1(C(=O)OCC2CCN(C3CC3)C2=O)CCN2CCOCC12 c1(CC(=O)NC2CCCN(C(C=Cc3n(C)ncc3)=O)C2)ccc(Cl)c(F)c1 C12(NC(C3(OC)CCCOC3)=O)CCC1CN(C(=O)CNC(=O)CC(F)(F)F)C2 c1(C(=O)NC(C)CNC(=O)C=Cc2nccs2)ccc(CCC2CC2)cc1 N(C1c2ccccc2CC1NC(=O)C=CC=C(Cl)Cl)C(c1cncn(C)c1=O)=O N1(C(Cn2nc(C)oc2=O)=O)CC(O)CCC1C(=O)N(CC(C)(C)N(C)C)C c1(C(=O)NC(CN(C(C(C2CC2)OCC)=O)CC)C)cc(I)c[nH]1 C(N=C1NC(C2CC2)N1)c1cc(OC)n[nH]1.C1(CN(C)C)CC12CC2 N1(C(c2n(CCOC)ncc2)=O)CCC(C)(NC(c2cc(Br)ccc2F)=O)CC1 CS(=O)(=O)c1nccc(Nc2cnc(F)cc2C(N2CCC(C#N)CC2)=O)n1 N(C1CCCc2cc(NC(c3ccnc(-c4ccccn4)n3)=O)ccc21)C(C)=O C12(C(N3CC(OCCNC(C(C(C)(C)O)F)=O)C3)=O)CC3CC(C(=O)N1)C2C3 CCCC(CCCNC(C1CC1Cl)=O)NC(=O)C=Cc1cncs1 c1(C(=O)NCC(C(C)C)NC(C2CN3CCC2CC3)=O)cnc2n1CC(C)CC2 N1(C(C2N(C(C=CCN(C)CC)=O)CC(O)C2)=O)CCC2(CCOC2)C1 c1(CC(=O)NC(Cn2cc(C3(C(C)=O)CCOC3)nn2)C)ccc(Cl)cc1Br CC1(C2CC2)CCN(C(=O)Nc2cncc(CO)c2)C1 n1(CC)nc(C(F)(F)F)cc1C(=O)NCCC(O)CNC(C1CC1(Cl)Cl)=O CC(CC(=O)N(C1CCN(C(c2nonc2N)=O)C1)CCO)C(F)(F)C(F)(F)F N1(C(c2c(CC)[nH]cc2)=O)CCCCCC1CNC(=O)Cc1cnn(CSC)c1 C(C)(C)(C(C)CC(=O)NCc1noc(C(C)C)n1)NC(CC(CC)SC)=O C1(NC(C2CCCCO2)=O)CCC(C)(C)CC1.CC1C(=O)NCCC2(CC2)CO1 CCCCC(CCCC)NC(C1C(C)OCCN1C(c1ccn(C)n1)=O)=O N1(C(CCCCN(C(C)C)C)=O)CC2(CC2)CC1CNC(=O)C#CC1CC1 C1(C(N(CCCOCCN(C(C2(SC)CC2)=O)C)C)=O)CCCC(C)(C)CC1 N1(C(C2=C(C)CC2)=O)CC(O)C(O)C1CNC(=O)C(C)OCCC(C)C CN(S(N)(=O)=O)CC(=O)NC1CC(N(C(=O)CCC2CC2(F)F)C)C1 c1(CC(=O)NC2CCN(C(C34OCC(C)(C3)C4)=O)CC2)ccc2c(c1)OCCO2 C1(CC)CN(C(=O)CCCF)CCC1NC(=O)CCc1ccncc1 N1(C(c2cn(CCCC)nn2)C)CC2C(C(=O)N)C2C1.C1(CC#N)CCNCC1 c1(C(=O)NC23CC(C(=O)OC)(C2)C3)c(C)[nH]c2ccc(Br)cc12 CCC(O)C(C)C(=O)N1CCCCC1CN(C)C(c1cnc(S)[nH]1)=O CC1CN(C(C2CC2(F)F)=O)C(C)CN1C(c1ccc(C2CC2)s1)=O C1(NC(C(n2cnc(C#N)n2)C)=O)CCC(F)(CNC(C2(F)CCC2)=O)C1 CON(C)C1CCN(C(=O)C(c2ccccc2)NC(C2CC3(CCO2)CC3)=O)CC1 c1(C(=O)NC(CN(C(c2c(C)nc[nH]2)=O)C)C)cccc2c1CCCN2 c1(C(N2CC(NC(C(C)C3CC3)=O)(CO)C2)=O)sc(C(F)(F)F)cc1Br S(=O)(=O)(CCC(F)(F)F)NC1CC2(CN(Cc3c(C)noc3C)C2)C1 N1(C(C(CCC)O)=O)CC2(C(=O)N(C(C)C(C)SC)C)CC1CCO2 c1(C(=O)NC(CCNC(=O)C#CC2CC2)Cc2ccccc2)ccc(F)cc1Cl N1(C(C(C)OCC#C)=O)CC(CNC(c2ccn(COC)n2)=O)C(C)C1 C1(CN(CCS(=O)(=O)N(CC)CC)C)(OC)CCCSC1 C1(CNC(c2cn(CCC)nc2C)=O)CN(C(C2C3CCC2CC3)=O)CCC1C CC(F)CC(=O)OCC(=O)NC(c1ccccc1)c1csc(Cl)n1 CCCC(C)C(=O)NCC(C1CCCCCC1)NC(=O)CCC1CCCO1 CCC(CC(=O)N(C1CCN(C(=O)OC(C)(C)C)C1)C)NC(C1(C)CC1)C C1(CNC(=O)CC2CCCOC2)CC2(CCN(C(c3coc(C4CC4)n3)=O)C2)CO1 c1(OC)ncc(C(=O)NC(C)(CNC(C2(CCF)CC2)=O)C2CC2)c(C)n1 c1(C(=O)NCC2(NC(CC3CCCN(C)C3)=O)CCOC2)cc(F)c(Cl)cc1Cl c1(OC)cc(C(=O)NCC2(O)CCN(C(=O)C(F)C3CCC3)C2)nc(Br)c1 N1(C(C2N(C(c3ccn(C)c3)=O)CC(O)CC2)=O)CC2(CCCCC2)C1 N1(C(CCCN(C(C)=O)C)=O)CC(O)CC1C(=O)N(C)C(C1CCCCC1)C N1(C(C2(CC=C)CN(C(c3scnc3C)=O)C2)=O)CCN(CC)C(C)C1 CCC(C)C(=O)NCC(C(C)C)NC(=O)Cn1cc(CCOC(C)=O)nn1 N1(C(=O)COC2CCOCC2)CCC2C(CCN2c2ncncc2I)C1 S(=O)(=O)(c1cccnc1N(CC(C)C#N)C)N(CCCN(C)C)C C1(C(=O)NCCN(C(=O)C(C)(C)C2CCOC2)C)CC(=O)OC1(C)C C1(CSc2cc(NC(C3C(C)C3)=O)ncc2)CC(F)(F)CN1c1nnc(C#N)s1 N1(C(C2N(C(C3N(C)C(=O)CC3)=O)CC=C2)=O)CC(F)(F)C(F)(F)C1 C1(C(N(C2CCCN(C(C3CC(=C)C3)=O)C2)CC)=O)CCc2ccccc2C1 C(=O)(C1=NOC2(CCOC2)C1)NCCn1cc(CNC(C(C)=C(CC)C)=O)nn1 CC1CCC(C(=O)NC2(CCNC(=O)CSC(F)(F)F)CC2)CC1 C1(CC(=O)NC2C(SC)CN(C(c3ccc(C)cn3)=O)C2)CC2CCC1CC2 C(=O)(CC(CNC(=O)CC(Cl)Cl)OC)NC(C(=O)OCCC)C Cc1nn(C)c(C(=O)NC23CC2CN(C(c2c(N(C)C)noc2C)=O)C3)c1[N+](=O)[O-] c1(C(N2CCC(N(C(C3CC(Cl)(Cl)C3)=O)CC)C2)=O)ccc2ccsc2c1 c1(CN2CC3(CC(NCc4c(OC)ncc(Cl)c4)C3)C2)ccc([N+](=O)[O-])cc1Cl N1(CC(=O)Nc2cccc(NC(C3(COCC)CC3)=O)c2)CCS(=O)(=O)CC1 N#Cc1c[nH]c2c(F)c(NCc3nc(-c4ccc(Br)s4)n[nH]3)ccc2c1=O c1(OC)c(C(=O)N(C)CC2CCCN2C(C2CC23CCOCC3)=O)cccc1Cl C1(NC(c2cn(CCC)nc2)=O)CC2CCC1N(C(=O)Cc1ccncc1Cl)C2 n1(CC)ncc(-c2nc(C(Oc3ccccc3)O)no2)c1CCOC(C)(C)C.CO C(=O)(CCCC(=O)NCC1(F)CCN(C(C)C)CC1)NCC(COCC)O c1(N(C(c2cn(-c3cccnc3)nn2)C(=O)NCC=C)C)cccc2nn[nH]c12 C(=O)(CC(C)C(=O)OC)N1C(C(N(C2C(OC)COC2)C)=O)CCC1 C(=O)(C(C)C(O)C(C)C)NC1CC(C(=O)NC2CCN(CC)C2)C1 C1(C(C(=O)N(CC(C)NC(C2(CCC)CCC2)=O)C)C)CCOCC1 Cc1cc(N)c(C(=O)NCCC(C)NC(=O)Cc2c(F)cncc2Cl)c(F)c1 C1(NC(C(C)NC(C)=O)=O)CC(C)(NC(=O)CCCc2nncn2C)C1 c1(OC)cncc(C(N2C=CC(NC(c3ccc(CN(C)C)cn3)=O)C2)=O)c1 Cc1ccc(C(F)(F)C(=O)OC(F)(F)F)nc1.C12CC(C1)NCCSCC2 C12CC(C1(C)C)C(=O)N(CCC1CC1)C2.C(C)(C)(C)O.C(=O)(NCC)N c1(OC)ccc(NC(=O)C(C)C)cc1Nc1ccc[nH]1.N12CC(C(F)C1)NC2=O N1(C(c2cnc(OC)c(Cl)c2)=O)CC(C)CN(C(C2(C)CCSCC2)=O)CC1C C1(COC)(CNC(C2CCCOC2)=O)CCCN(C(=O)COC2CCC2)C1 C1(OCc2cnn(-c3ccccn3)c2)CCCCC1.C1(=O)C(=O)NC(C)CN1C c1(N2CCCC(C(C)C)CC2)nc2c(c(=NC3CCN(C)C(=O)C3)[nH]1)SCC2 CC1CCC1C(=O)NCCC(=O)N1CC(Cc2ccco2)C1 CCCCCC(C)(C)C(=O)N1CC(NC(C2C=C(C)CS2)=O)C(F)C1 c1(C(=O)NCC(CC)NC(c2cccn2Cc2ccncc2)=O)[nH]cc(C)c1C C1(CC(=O)N(CCNC(C(C2CCOCC2)C)=O)CCOCCO)CCS(=O)(=O)C1 C1(NC(C2CCC(C)(CC)O2)=O)CCC2CN(C(c3ccc(F)s3)=O)CC12 C1(CC(=O)N(C)CC2(CNC(c3ccccn3)=O)CC2)CCCCCCC1 N#Cc1cc(C(F)F)cc(N2CCCC(Oc3ccccc3Cl)C2)n1 Cc1csc2ncnc(NC3CCCN(C(C45CCC(F)(CC4)CC5)=O)C3)c12 CC1=NNC(=O)C1CCC(N1CCC(NC(=O)C(C)C(C)C)CC1)=O CCCCCC(CC)C(=O)N1CC(NC(c2nc(Cl)sc2C)=O)CC12CCOC2 c1(C(=O)NC(CC)CN(C)C(c2cnnc(C)c2)=O)c[nH]c(=O)c2ccnn12 CC(C)(O)C#CC(=O)N1CCC(C(N2CCc3c(O)n[nH]c3C2)=O)O1 CS(=O)C=CC(=O)N(CCNC(C1CSCCS1)=O)Cc1cccc(Cl)c1 Cc1cc(C(N2CCC(N(C(=O)COC(F)(F)F)C(C)C)CC2)=O)c(C)s1 N1(C(c2c(C)nccn2)=O)CCC2C1CCCN2S(=O)(=O)CCC(F)(F)F N1(C(C=CC)=O)CCC(C2CC2NC(C2CC(CC3CC3)C2)=O)CC1 C1(COC)(NC(=O)C(F)C(C)(C)O)CCN(C(C2CCN(S(C)(=O)=O)C2)=O)CC1 c1(Nc2ccc(NC(C3N(C)C(=O)OC3)=O)nc2)ncc2ccsc2n1 c1(NCC2CCC(NC(CN(C(C)=O)C)=O)C2)cccc2c([N+](=O)[O-])cccc12 c1(OC)ncnc(OC)c1CNCC1CCCN1C(c1cccc(Br)c1O)=O N1(C(c2c(CC)c(F)ccc2)=O)CC(NC(=O)C=Cc2cnc[nH]2)C(F)(F)C1 c1(C(=O)NCC2C(NC(c3cncn(C)c3=O)=O)C2)cn2cccc(F)c2n1 Cc1ccc(NC(C2CN(C(c3cc4sccc4s3)=O)CCC2O)=O)c(C)c1 C(C)(C1=CCN(C)CC1)NC(CN(C(=O)Cc1cn(C)cn1)C(C)C)=O C1(NC(CNC(C2C(C)C2)=O)=O)CC=C(C(=O)N2CC(O)(CCO)C2)C1 N1(C(CCSC)=O)CCN(C2CCN(C(c3cnc(Cl)cc3Cl)=O)CC2)C(=O)C1 C1(O)(CNC(C=CCN(CC)CC)=O)CCCN(C(c2ccnnc2O)=O)CC1 N1(C(C=Cc2cn(C)nn2)=O)CC(C(NCP(C)(C)=O)=O)CC1(C)C C=CC1(CO)CCN(C(=O)C(CCC)NC(c2cn(CC)nc2C)=O)CC1 c1(NC(c2ccc(CNC(c3ccc(O)nn3)=O)cc2)C)ccc([N+](=O)[O-])c(O)n1 N1(C(c2cc(C)nnc2)=O)CCC2(CC2C(N2CCS(=O)(=O)CC2)=O)C1 CCCC(C(=O)NCC1CC(NC(=O)CC23CCC(CC2)C3)C1)OC C(C(C)(C)C(=O)NCCC1CC(NC(=O)CCc2cncc(F)c2)C1)N(C)C c1(C(N(C2CN(C(C(C)SC)=O)CC2(C)C)C)=O)c(C)ccc2n[nH]cc12 CS(=O)(=O)C1(C(N2CC(c3ocnc3CNC(c3cccnc3)=O)C2)=O)CC1 CN1CCN(C(c2cc(=O)n(C)cn2)=O)CC1CNC(=O)Cn1cccnc1=O C1(NC(C2(CC#C)CC2)=O)CN(C(C2C3CN(C)CC23)=O)CCC1C N1(C(c2cnc(SC)n2C)=O)CCN(C(=O)CNC=O)C(C)C1C N1(C(=O)COCC2CCCC2)CCC2CN(C(c3ccc4[nH]ccc4n3)=O)C2C1 C1(CNC(CN2C(C)CCC2C)=O)CC2(CCN(c3cc(=O)n(C)c(O)n3)C2)CO1 CN1CC2(CCN(CCCCO)CC2)C1=O N1(C(c2n(CC)ncc2)=O)CCC(C(N2CCOCC2CF)=O)(CO)C1 c1(C(N(C(C(=O)NC2CC(C(C)C)C2)C)C2CC2)=O)ccc(C#N)[nH]1 c12cc(C)ccc1NC2=O.C1(SC)CCCC(N2CCN(C(C)C)CC2)C1 C1(CNC(C(c2ccoc2)NC(c2ncc(C)nc2)=O)=O)CC2(CCCO2)C1 C1(C(C)NC(=O)COC2CN(C(=O)CC3(C)CC3)C2)CC(F)(F)C1 c1(O)c(F)ccc(Br)c1F.c12cccc(c1)C(=O)OCO2.c1(C(=O)OC)cncnc1 N1(C(c2c(C)oc(CO)c2)=O)CCOC2(CCN(C(=O)C#CC3CCOC3)C2)C1 C1(C(N2CCC(CCOC)CC2)=O)C2CCC1CN(C(C1(F)CCCC=C1F)=O)C2 N1(C(CNC(C)=O)=O)CCC2CC1CN(C(=O)Cc1c(Br)ccc(Cl)c1F)C2 C1(NC(c2n(CC)ccc2)=O)C2CCN(C(C3SCCS3)=O)CCC12 C1(NC(=O)C(Cl)(Cl)Cl)CN(C(=O)Cc2cc(F)cc(Cl)c2)CC(F)(F)C1 C1(C(=O)NC2CC(N(C)C(c3cc(C(N)=O)[nH]n3)=O)C2)COCCN1C C(=O)(C(C)(C)CN(C)C)NC(C1CCCN(C(=O)Cc2ccoc2)C1)C CC(CF)CC(=O)NC1(CO)CCN(C(=O)C(Cl)=CCl)C1 C(=O)(C1c2c[nH]nc2CN1C(=O)CC1CCC(O)C1)N(C)CCOC1CC1 c1(C(=O)NCC(C2CC2)NC(C2CC23CCOCC3)=O)cccc(Br)c1Cl c1(NC(c2cc(-c3c(OC)ccc(OC)c3)on2)=O)nc2c(s1)CC(O)CC2 n1(CCOC)cc(C(=O)NCC(CC)(CC)NC(=O)C(C)C2CC2)c(=O)cc1C c1(C(c2nnc(C(C3CCOC3)SC3CCC3)n2C)N)ccc2c(c1)OCO2 C(C)(CCCC(=O)N1CCCC(C)CC1)NC(C1(CCC)CC(=O)C1)=O N1(C(CCC(C)(F)F)=O)CC2(CNC(=O)C(CO)C(C)(C)C)CC1CCO2 C(=O)(C(F)C(C)(F)F)NC1CC(N(C(C=Cc2ccc(C)o2)=O)C)C1 Cn1ncc(S(N)(=O)=O)c1C(=O)NCC1(C)CCCN1C(c1cncnc1)=O Cc1cnnc(N(c2ncccn2)C(C2CNCC2F)=O)c1 c1(OC)c(Cl)cc(C(=O)NC2CC23CC(NC(c2c[nH]ccc2=O)=O)C3)nc1Cl Cc1ncc(C(N2CCC=CC2C(=O)NCc2ccc(C(N)=O)o2)=O)cc1C#N C1(c2nc(C(C)(C)C)no2)(CNC(=O)OC(C)(C)C)CCCCC1(C)C N1(C(c2cn(CC)nc2)=O)CCN(C(=O)Cc2ccc(Cl)c(Cl)c2)C(C2CC2)C1 c1(OC)ccc(C(=O)NC2(C)CC(C(=O)Nc3ccnc(C)n3)C2)c(F)c1F C(=O)(CC(F)(F)CC(=O)N1CC2CC(NC(c3cnsn3)=O)CC1C2)OC C1(CNC(=O)C(c2ccccc2)O)CC2(CO1)CN(C(=O)Cc1cc[nH]c1)C2 C(c1ccccc1)=NC(N1CC2CC1C2C(=O)NCc1ncccn1)=O c1(CN2CC(C(=O)Nc3cc(OC)c(Br)cc3)OCC2)cc(F)cc(C)c1O C(CC(C)(C)C(=O)NCCC1CCCC1(C)C)NC(C(C(=O)OC)C)=O Cc1ccccc1C(=O)N(C(C)CN(C(=O)Cc1cc[nH]c(=N)c1)C)C C(=O)(CC(C)(C)CC(F)F)N1CCC(C2(NCCNC(C(CC)N(C)C)=O)CC2)C1 CC1(C)CCC(CNC(c2cncc(Cl)c2)=O)N(c2ncc(I)cn2)C1 c1(CC(=O)OCC)ccccc1NC(c1n(CC2CC2)nnn1)c1cccs1.C(CSC)N c1(C(=O)NC2C(CNC(CCCC(N)=O)=O)CCC2)coc2c1C(O)CCC2.C1(C)CC1 CCC(C)CCCCC(=O)NCCCC1CCCN1C(=O)Cc1cncc(O)c1 O=C1OCc2cc(C(=O)NC3CCCCN(C(c4c[nH]c(=O)cn4)=O)C3)ccc21 N1(C(C2(SC)CCC2)=O)CCC2(CCC2CNC(=O)CC2CC2(C)C)CC1 C(=O)(C(F)C(C)(C)O)N(CC(N1CCCC(OCC)C1)=O)C1CC1 Cc1csc(C(N2CC(CNC(=O)C(=C3CCCCC3)F)C3CC23)=O)c1C C1(CN(C)C(c2ncn(C)n2)=O)CCCCN1C(=O)C(F)=C1CCCC1 N1(C(Cc2c(C)cnn2C)=O)CC2CCC2(CC(=O)NCCC(=O)NC(N)=O)C1 N1(C(CCC=C=C)=O)CCC(NC(=O)COc2cncc(Cl)n2)C(CO)CC1 C(=O)(C1=CCc2ccccc21)NC1CC2CN(C(=O)OC(C)(C)C)CC(C1)C2 c1(C(=O)NC(C)CC(C)NC(C2(N(C)C3CC3)CCC2)=O)cccc(=O)n1C c1(C(CC)OC)cn(CC(C)NC(c2ccnn2CC(F)F)=O)nn1 N1(C(C(C(C)O)C)=O)CCN(C(c2nccc3cc[nH]c23)=O)C2(CCC2)C1 N1(C(C2CC(CCC)OCC2)=O)CCCN(c2ccccc2)CC1 C1(NC(C(C)=C(C)C)=O)CC2CC(C1)N(C(c1cc(O)ncc1F)=O)C2 Cc1cc(C(N2CC(N(C)C(C3CC4CCC3O4)=O)C(C)(C)C2)=O)cc(N)c1Cl C1(NC(C(COC)(C)C)=O)CC2CC(C1)N(C(=O)C=Cc1ccc(F)cc1F)C2 Cc1ncc(C=CC(N2CCC(C)C2CNC(=O)Cn2cc(C3CCC3)nn2)=O)s1 c1(CC(C(=O)NC(CN(C(c2c(CC)n[nH]c2)=O)C(C)C)C)NC)cccc(C)c1 c1(C(=O)NC(C(=O)NCC(COC)C(C)C)C2CCC2)ccccc1C#N C(=O)(CC(O)(c1ccccc1)C1CC1)NCC(C(C)C)NC(C1(C)CC1C)=O c1(OCCOC)ccc(CNC(=O)C(=O)Nc2cnc(C(F)F)nc2)cc1 C(=O)(C1=C(C#N)CCC1)N1CCC(CCNC(Cc2c(C)scc2)=O)CC1 N1(C(Cn2ncc(C#C)c2)=O)CCCC(C(=O)NCC(=C)Cl)C1C N1(C(C=C(CCC)CCC)=O)CCOC2(CCN(c3ccc(C#N)nc3)C2)C1 C1(CNC(=O)NC(c2cccc3c2CCC3)C)CC2CC1C1CC21 N1(C(=O)NCc2ccc(C)s2)CCN(C(C2CC2F)=O)C(c2cn[nH]c2)C1 c1(C(N2CC(OC)(CNC(C3CCN(C(C)C)CC3)=O)C2)=O)cc2n(c1)CCC2 C1(C(N(C2CCN(C(c3nc(CCC)sc3)=O)C2)CC)=O)CCC(=O)NC1 c1(NC(CNC(C(C=C)OCCOC)=O)=O)ccc(CO)nc1 N1(C(C(CCC)O)=O)CC2CS(=O)(=O)CC2(NC(=O)C=CCN(C)C)C1 Cc1ccc(C(=O)NCC2(NC(c3ccnc(C(C)(F)F)c3)=O)CCCC2)nn1 C=CCC(CC=C)C(=O)NC(CC=C)C(=O)N(CC(C)O)C1CCC1 c1(C(N(CC(C)(C)NC(C2CC(C)(C)CCO2)=O)C)=O)n[nH]c2ccccc12 c1(C(=O)N(C23CC(C(N4CCCC4)=O)(C2)C3)c2ccncn2)cccc(F)c1 c1(N2CCC(=C)C2)[nH]c(=NCC(C)(C)OC(C)C)nc2c1cnn2C(C)C C1(CNC(C(C)CNC(=O)C(C2(O)CCCC2)F)=O)CC12CCOCC2 C#Cc1ccc(C(N2CC3(CC3)CC2CC(N2CC3(C)CC2CCO3)=O)=O)cc1C S(=O)(=O)(c1cccnc1)NCCCNC(=O)C(C)NC(C1C(C(=O)OCC)C1)=O C(=O)(CCC(C)(C)C(=O)OC)NC1CC(C)(CNC(CC(CCC)C)=O)N(C)C1 N1(C(C2C(OC)CCC2)=O)CCC(F)(F)C(CNC(=O)CNC(=O)CC(C)C)C1 C1(NC(C=CC(C)C)=O)CCCC(CC(=O)NCC2(F)CCOCC2)C1 C=C1CC(C(=O)NC2COCC2SC)(CNC(=O)Cn2ncnn2)C1 S(=O)(=O)(c1ccc(C2(CO)CC2)cc1)C(=O)NCC(C)(C)NC(=O)C1=CCCS1 C1(C)(C(=O)NCC(C(C)C)NC(c2ccccn2)=O)CC(C2CC2)=NO1 c1(-c2occ(C(=O)NC(c3ncc(F)cc3F)C)n2)c(Cl)cccc1Cl CC(F)(F)CC(=O)NCC(C1CCOC1)NC(=O)Cn1nnc(C2CC2)n1 Cc1cc(CC(N2CCC(C(C)NC(C3(N=[N+]=[N-])CC3)=O)CC2)=O)ccn1 Cc1c[nH]ccc1=NC(=O)C1C=CCN1C(C1CCCN(c2ncccc2Cl)C1)=O C(CNC(n1nnc(C2CC2)n1)=O)(CC(F)(F)F)NC(Cc1c(C)n[nH]c1C)=O c1(C(=O)NC2C(C)CCN(C(c3cccn3C)=O)C2C)cccc2c1nnn2C c1(CC(=O)NCCCOCCNC(C(C)C2CCC2)=O)ccc(C(N)=O)cc1 C1(C)(C(N2CC(O)(CNC(C3(OC)CCCOC3)=O)C2)=O)CCC(C)C1(C)C C(=O)(C1CCCn2nccc21)N1C2CN(C(c3cccnc3)=O)C(C2)C1 c1(C(N2C(C#N)CN(C(c3cc4ccccn4n3)=O)CC2)=O)cc2ccoc2cn1 CC1(C)C(CNC(C2CC(=O)CN2C(=O)CCc2nc(=N)[nH][nH]2)=O)C1(C)C c1(C(=O)OCc2ncoc2COc2ccc3c(c2)OCO3)cccc2ccnn12 c1(CC(=O)NC(CN(C(c2ccc(C#C)cn2)=O)CC)C)cnc2ncccn12 C1(NC(=O)COc2cccc(F)c2)CN(C(=O)CCCCc2cnn[nH]2)C2CC12 C1(NC(Cn2ncc(CC)c2)=O)CCCN(C(C2CCC=CCCC2)=O)CC1 Cc1sc(Br)c(C(=O)NCC(CNC(=O)CCC(C)C)C(F)(F)F)c1C CCC(CC(=O)N(C1CCCN(C(=O)CCCc2ccsc2)C1)CC)C1CCC1 N1(CCC)CCC(NC(=O)Cc2ccc3c(c2)CCC3)CC(C)(C)C1 c1(C(=O)NCC(C)(C2CCC2)NC(C2Cc3nccn3C2)=O)cc2n(n1)CCC2 c1(C(=O)NC2CC3CN(C(c4cn(CC)nn4)=O)CC32)cnn2ccn(C)c12 CC(C(=O)N1CCN(C(=O)C(C2CCCCC2)=O)CC1)S(C)(=O)=O N1(C(C2(C)CCN(C(C3CC(=O)CCO3)=O)C2)=O)CCC2CCCC12 c1(OCC)ccc(C(=O)CCC(=O)N(C(C)CN(C)C(c2cnsn2)=O)C)cc1 C1(C(N2CCC(c3ccon3)C2)=O)Cc2ccc(OCC(F)(F)F)cc2O1 O=C1C2Cc3ccccc3CN2C(=O)N1CC1(Br)CCOCC1 N1(C(C2C(C)OCC2)=O)CCOC2(CCC(NC(=O)CNS(C)(=O)=O)CC2)C1 CC(=O)CCCC(C)C(=O)NC1CC2CC1CN(C(=O)Cc1ccc(C)nc1)C2 C(C)(CCC(=O)NC1(CNC(c2cccnc2Cl)=O)CCOC1)OC c1(C(N2CC3C(CNC(C(C)C4CC4)=O)C3C2)=O)cc(S(N)(=O)=O)cs1 C1(C(N2CC(N(C(C(C3CCCO3)OC)=O)C)C2)=O)(COC)CCCC1 C1(N)C2CCC1(c1ccnn1C)C2.S(=O)(=O)(CCOC(C)C)N1CC1.CO C12(NC(CNC=O)=O)CCC(C1)N(C(=O)CSc1nnnn1CC(F)(F)F)C2 C1(C(=O)NCCC2CN(C(=O)Cn3cnnc3)CCCO2)CCn2cnnc2C1 c1(C(CC)NC(=O)C(C)N2CCC2C(=O)OC)ccc(=O)n(C)c1 C1(N(C2(C(=O)NOCCCF)CCCC2)C(c2ccncc2)=O)CCCCCC1 C(=O)(CCCCN(C)C(c1cncn1C)=O)N(C)Cc1cc[nH]n1 Cc1ccc(SCC(=O)NCC2CCCN2C(c2cn[nH]c2)=O)cc1Br c1(C(N(CC(C)N(C(CCN(C(CCC)C)C)=O)C)C)=O)cc2ccncc2s1 CC(F)(F)C(F)C(=O)NCc1cn(-c2ccc(N)cc2Br)nn1 Cc1ccc(C(=O)NCC(C)(F)CNC(=O)C(C)C)cc1F C12(NC(c3ocnc3C3CC3)=O)CCCCC1N(C(=O)CS(=O)(=O)C1CC1)CC2 c1(C(=O)NC2CC(NC(=O)CC(c3ccc(F)cc3)O)C2)ccnc2ncnn12 C(=O)(C(O)P(C)(C)=O)NCC1CC(OC)CN1C(c1cnn(C(C)C)c1C)=O CC(C)C(CNC(C1(C)CC1(C)C)=O)C(=O)N(C(C)CCO)C C1(C(N2CCC(Br)C2)C(=O)N(C2COC2)Cc2ccccc2)CC12CCOC2 c1(OC)ccc(Cl)cc1C(N1CC2CC1CC2NC(=O)Cc1ccnn1C)=O C=CCC(CNC(C1CCCN1CC(C)C)=O)NC(c1cc(CC(C)C)[nH]n1)=O c1(CC(=O)NCCN(C)C(c2ccc3nonc3c2)=O)cncc2ccccc12 C1(CC)CN(C(c2nccn2C)=O)CC1C(=O)NCCC1(C(=O)OC)CC1 C(=O)(CCCCCSC)NC(C1N(C(C2C(=C)CC2)=O)CCC1)(C)C C1(C(N2CCC(CCC)C2)=O)CN(C(c2cc(C#N)cnc2C)=O)CC(C)(C)C1 C1(NC(CCCOCC=C)=O)CCC(C)N(C(=O)Cn2ccsc2=N)C1 C1(O)(CNC(c2occc2C2CC2)=O)CCN(C(=O)CCSc2ccccn2)C1 C1(CNC(C(C=C)O)=O)CC12CCN(C(=O)CCCCC#N)CC2 C1(C(=O)NCC2(F)CC(NC(CCC3(C)N=N3)=O)C2)CCC(F)(F)C1 Cc1ncnc(O)c1C(N1CCC(C(C)CNC(C2(CO)CCCO2)=O)CC1)=O Nc1c(F)cc(C(=O)NC2(CNC(=O)CC3CCCC4(CC4)C3)CC2)cc1F n1(CC)cc(Br)c(C(=O)Nc2ccc(NC(=O)C(=O)NC3CCCC3)cc2)n1 C1(C)(C(N2CC(C(C)NC(CCSCC)=O)C2)=O)CCSCC1.NCC c1(CC)cccc(OCC(N2CC(O)(CN(C(=O)CCC(C)OCC)C)C2)=O)c1 Cc1cc(C(=O)NCC(C)(C)CN(C(=O)CCC2CCCCO2)C)cc(C)n1 N1(C(C(C)(C)CF)=O)CCC(C2(O)CC(NC(C3C=CCCC3)=O)C2)CC1 N1(C(C(CCCC)O)=O)CCN(C(=O)Cc2ccoc2)CC(C)(F)C1 c1(C(C(=O)NC(CNc2n(C)ccn2)(C)C)C2CC2)cccc(I)c1 c1(SC)ccc(-c2cncnc2C(N2CCN(C3CC3)CC2)=O)cc1F.CCCN CC(C)CC(CNC(=O)CCC1CCN(C)C1)NC(c1ccc[nH]1)=O Cc1cc(Cl)n[nH]c1=NCC1(C(C)=O)CCCC1C.CC C1(NC(c2c(OC)scc2)=O)CCN(C(=O)CC2CC3(CCC3)CO2)CC1F c1(C(N2CC(F)(CNC(c3c(C)nc(C(C)C)o3)=O)C2)=O)ncc2n1CCCC2 N1(CC)C(=O)CCC1CC(=O)NC1CCN(C(c2sccc2C(C)C)=O)C1C C1(NC(c2c(C)cnn2C(C)C)=O)CC2CCC1N2C(=O)CCC1(C)CC1 N1(C(C2C(CC)CCO2)=O)CC2(NC(=O)C(=O)Nc3ncc[nH]3)CCC1CC2 C1(CNC(c2c(C)onc2C2CC2)=O)C(C2CC2)CCN1C(=O)Cc1ccns1 Cc1c(C2CCCN2C(=O)C(=O)Nc2nccc(Cl)c2F)oc2ccccc12 C(=O)(C(C)(C)CCC(C(=O)NCCC#N)N1CCOCCC1C(C)C)OCC c1(CN(CC(O)COCCF)C(=O)NC)ccc(NC(CSC)=O)cc1 c1(C(N(CCF)CC2CC2)=O)ccc(F)cc1.n12cc(nn1)SCC2C C1(C(=O)NCC#C)CCCN(c2ncncc2C(C)C)C1 c1(C(=O)NCC(C(C)(C)C)NC(C2C(COC)C2)=O)cc(N)c(F)cc1F c1(C(c2n(CC=C)nnn2)NC(C2CC2)C2CC2)ccc(-n2cncn2)c(F)c1 N1(Cc2ccc(N(C)C)cc2O)CC2CN(C(c3ccc(F)c(Cl)c3)=O)CC2C1 c1(-c2nc(CNCCn3c(C(=O)OCC)cc(C)n3)on2)ccc(Cl)c(Cl)c1 C1(CC(=O)NC(CC#C)CCOC)N(C(c2ncc(CC)cn2)=O)CCC1(C)C c1(C(=O)NCCCN(C(C(=O)NC)=O)C2CC2)nc(Br)c[nH]1 N1(C(C2(OC)CC2)=O)CCC(CCCCNC(C2CC2C(C)C)=O)CC1 c1(C(=O)NC(CC(C)NC(c2cn(CCF)nn2)=O)C)cccc2nnn(C)c12 CCCCCCC(F)C(=O)NC(CNC(=O)CS(=O)(=O)N1CCCCC1)CO Cc1c[nH]cc(C(N2CCC(N(C)C(C3CN(C4CCC4)C3)=O)CC2)=O)c1=O C1(CC)COCCN1C(C1CC(=O)N(Cc2ccccc2)C1)=O c1(NCC2CCCN(Cc3c(N(C)C)cccc3)C2)ncnc2cc[nH]c12 c1(CCC)ncc(C(=O)N(CC(O)CN(C)C(C2CC(CC(F)F)C2)=O)C)s1 c1(C(C)C(F)(F)F)cccc(CNC2CCCC(CN)C2)c1 C1(CNC(C2(C(C)C)CN(C(=O)Nc3nccn3C)C2)=O)COC(C)(C)C1 c1(C(N(CC(O)CNC(=O)CN(C2CCCC2)C)C)=O)cc(=O)n(C)cn1 N1(C(CC)=O)C2CCC1CC(c1ccccc1)(NC(c1ccn(C)c1C1CC1)=O)C2 c1(CC(C)C)cc(C(=O)NC2CCC(NC(C3CC3C(N)=O)=O)CC2)cc(O)n1 O=C(CCCCC(F)(F)F)NCC1(F)CCN(C(C2CCCOC2)=O)CC1 C12(NC(CC=C)=O)CCN(C(c3cccs3)=O)CCC1C2 N1(C(C(CCC)n2c(COC)nnc2O)=O)CCOC(C(=O)NCCSC)CC1 c1(NC(C(N2CCC(F)(C(=O)OC)C2)=O)=O)ccc(F)cc1C(F)F C1(CNC(=O)Cn2cccn2)CCN(C(=O)CCOCC2CCCO2)CC1(F)F c1(C(N(C(C)CNC(=O)C(F)C2CCCC2)CC)=O)ccccc1N(C)C(C)C c1(NCC(N(C)C(C2(C)COCCO2)=O)C2CC2)ncc([N+](=O)[O-])cc1C(N)=O N1(C(c2c(C)scc2)=O)CCN(C)c2ncccc2C1 N1(NCC(CC)(C)OC)C(=O)CN(C(c2ccccc2)C2CCCCC2)C1=O C(CCN(C)C(c1ccc(O)o1)=O)(C(C)C)NC(c1cn(CC=C)nc1)=O N1(C(C)=O)CCC(C)(C)C(CNC(=O)C(O)CC2CC2)C1 C1(N(C)C(C2CC(C3CCC3)C2)=O)CCCCN(C(c2cccnn2)=O)C1 Cc1cc(C(N2CC(C(C)NC(c3cc([N+](=O)[O-])oc3C)=O)C2)=O)cc(C)c1F C1(N2CCN(C)CC2CC(N)=O)CCC12CCN(C(=O)C1CC1)CC2 CC1(C)NC(=O)CC1C(N1CCCCC1CNC(c1nc(Cl)c(Cl)s1)=O)=O c1(C(C)C)ccoc1C(=O)NC1CC1C(=O)NCC(C)CC c1(C(=O)NCC2N(C(CCCCOC(C)C)=O)CC2)cc(Cl)c2ccccc2n1 C12(CNC(C3C(C)(C)C3(F)F)=O)CCCC1N(C(c1coc(O)n1)=O)CC2 CC(C)CNC(=O)CNC(=O)CN(C)C(C1(Cl)CC1)=O C(=O)(CC(C)(C)CCOC)NC(CC)CN(C(=O)CC1CC1)C C(=O)(CC(=O)NC1CN(CCC(CC2CCNCC2)(C)C)C1)N(C)C N1(C(C(n2c(C)ccn2)C)=O)CC(O)CC1Cn1cc(CC(O)C2CC2)nn1 C(C)(C(C(=O)NC(C1CC=CCC1)C(=O)NCC(CO)C1CCC1)N(C)C)OC c1(C(N(C(CNC(c2ccc(Cl)s2)=O)C2CC2)C)=O)cn2c(n1)CCCC2 c1(C(N2CC(CC)N(C(=O)C(C)C3CC3)CC2)=O)cc(F)cc(OC)c1N N1(C(C2CN(C(C)=O)C2)=O)CCCCC1C1CCN(C(=O)C(C)n2cncn2)C1 C1(C(N2C(C(C)C)CC2)=O)CN(C(=O)C(C)C2(O)CCC2)CCN1C C(=O)(CCCCCCc1ccc(O)cc1)NCC=CCNC(C(CC)C(C)C)=O Cn1cnc(C=CC(=O)NCC2CCCC2NC(c2cc(C(F)F)ccn2)=O)c1 C1(CN(C)C(C2CC2c2cccnc2)=O)CC(F)CN1C(=O)C(Cl)=CCl CN1CC2CCC(N3CCCC3)C2C1.C1(C(C)(C)C)CNC(=O)N1 c1(NC(C2C3CC2N(CC2N(C)CCCC2)C3)=O)c(C#N)cnn1C(C)(C)C N1(C(CN(C)CC2CCC(C)CC2)=O)CC2CCCCCC12 C1(NC(c2csc(O)n2)=O)CC2(C1)CN(C(c1cnc(C(F)(F)F)cn1)=O)C2 c1(-n2ccc(C(=O)NCC(C)N(C(=O)C(C)(C)SC)CC)n2)ccc(F)c(Cl)c1 C1(CCC(=O)N(CCC(=O)NCc2cncs2)C)C(C)(C)CO1 c1(C(N2CCN(C(C(C)OCCOC)=O)C(C)CC2)=O)cccc2c1C(=O)NC2 N1(CCNC(=O)C(O)CF)CCCN(C(c2ccn(-c3ccccc3)n2)=O)CC1 c1(OC)cc(C(N2CC(C(=O)O)OCC2C)=O)ccc1CN1CCOCC1 N1(C(CC(C=C)CC)=O)CCOC2(CCN(C(=O)C(c3cccn3C)=O)CC2)C1 C1(C(=O)N(CC(CC)OC)C)(NC(CC=CCC)=O)CCSC1 Cc1cncc(C)c1C(N1CCC(C(=O)NCC2CC(O)C(O)C2)C(C)C1)=O c1(OC)cc(F)c(C(N2CC(NC(C3CCC(C)(C)C3)=O)CC2(C)C)=O)cc1N C1(NC(COCCOCC)=O)CC2CN(C(=O)CC3(O)CCC3)CCN2C1=O c1(CC(=O)O)ccc(-c2csc(C(N3CCCC3CC(=O)CCO)O)n2)cc1 C1(C)(CNC(C2C(CCOC)C2)=O)CN(C(=O)CSC(F)(F)F)CCO1 C(=O)(C1=NN(CC(C)C)C(=O)CC1)N1C(C)CC(CNC(C(CC)(C)O)=O)C1 C12(n3cc(CC4(CNC(N5CCCCC5)=O)CCCO4)nn3)CCCCC1C2 C(C(C(=O)NCCCOCCCOCC)OC)OC.c12ccoc1NC2=O.C=O C1(C(=O)NCCC2(NC(C3NC(=O)OC3)=O)CC2)CCC(C2CC2)C1 CC1CN(C(=O)C(CCC2CCC2)NC(c2coc(O)n2)=O)CC1(F)F C(C#Cc1cn(C2C=CCCC2)nn1)NC(c1noc(C)c1C)=O C(=O)(CC(C(F)(F)F)NC(C1CN(C)CC(C)O1)=O)NC(CC)CCO CCC(C(=O)NC1(CNC(C2(C)CC2(C)C)=O)CCCCC1)C(C)C c1(C(N2CC(O)(CCNC(C(C)OCC=C)=O)C2)=O)cc(O)c2ccccc2c1 C(=O)(CCF)N(CCNC(C1(COC)CCC1)=O)CC Cn1c(=O)oc2cc(C(N3CC4COCCC4(C(=O)OC(C)(C)C)C3)=O)ccc12 N1(C(C2(N(C(c3nc(C)c(C)s3)=O)C)CC2)=O)CCCC2(CCC2)C1 N1(C(C(=O)NCC(c2cncc(Cl)n2)(C)C)=O)CCCCC1c1ncc[nH]1 N1(C(C2(NC(C3CN(C)C3)=O)CC(O)C2)=O)CC(CO)C2(CCC2)C1 Cc1cccc(C)c1OCC(O)CN(C)C(c1ccnc(NC(=O)C2CC2)c1)=O C1(NC(c2ccnc(C3CCC3)n2)=O)CCCN(CCC2CCCC2(F)F)CC1 CCCCC(C(=O)NCCN1CC2CC2C1)N(C(=O)C(CCC)NC(=O)COC)C N1(C(C(N)=O)=O)CCN(C(C2CC3CCC3C2)=O)CC1c1cn[nH]c1 C(CCC(O)C(=O)N1CCOCC(C)C1)NC(c1ccc(CC)nc1)=O N1(C(c2c(Cl)cc(C)s2)=O)CC(NC(=O)C(Cl)=CCl)C(C)(C)C1 CC1(C)CC(NC(c2cc[nH]c2)=O)CN1C(c1ccsc1C(F)F)=O N1(CCc2ccc(OC)cc2)CCC(NC(=O)CC2CCC(C)(C)CC2)C(O)C1 c1(-c2cn(CC)c(=O)cc2)ccc2cc(C(N3CCCC(C)CC3)=O)cn2c1 N1(CC)CCOC(C(=O)NCC(C)(C2CC2)NC(c2ccc(CC(C)C)[nH]2)=O)C1 CC1CN2CCN1CC2C(=O)NCCCCC(C)NC(=O)Cc1ccsc1Cl CC1(C)COC(C(=O)NC2CCCN(C(C3COCCOC3)=O)C2)C1 N1(C(c2c(C#N)scc2)=O)CCCC2(NC(C3CCCOCC3)=O)CCCC12 c1(C(N2CCC(N(CCC)C(c3cccc(OC)c3)=O)C2)=O)ccc(N)c(N)n1 C1(NC(C(n2c(C)ncc2)C)=O)CCN(C(c2cn(C3CC3)cn2)=O)C12CC2 c1(NC(=O)CC2CCCN2C(c2cc(Br)ccc2F)C2COC2)cc(Cl)c(Br)cn1 CC(C(=O)N1CC(CN(C(=O)C=CBr)CCO)C1)C1CC(=O)C1 c1(SCC(=O)NCc2nc(CNC(c3n[nH]cc3Cl)=O)cs2)ccc(F)c(F)c1 C1(C(N2CCC(COC)CC2)C(=O)NC)CCC(F)(F)CC1.C1CN1 c1(C(N2CC=CC(NC(C3CCCCS3(=O)=O)=O)C2)=O)ccc(F)c(O)c1 c1(C(=O)NC(CNC(C2(CC(F)F)CCC2)=O)CO)cc2n(n1)CC1(CC1)C2 C(=O)(CC1=CCN(C(=O)C(C)(C)CCF)CC1)N1CCCC(C)(CCC)C1 c1(C(=O)NCC(C)(C)OCC(=O)NCC2(C)CCCCO2)cc[n+]([O-])cc1 Fc1ccc(CNc2nnnn2CC2CC3CC3C2)nc1 N1(C(CCCSC)=O)CCN(C(c2ccc(CCN(C)C3CC3)cc2)=O)C2CC12 CC(C(C)C(=O)N(CC(N1CCCCC1)=O)C)S(C)(=O)=O.C12(CCCC1)C(=O)O2 CCC(CNC(c1c(CNC(c2cc(C3CC3)[nH]n2)=O)nnn1C)=O)CCO C(CCCCC(=O)N1CC(C)OC(C)C1)N(C(CC(C)OC)=O)C c1(N(C2CCN(C(C3(CC=C)CCC3)=O)C2)C)ncncc1C#N n1(CCNC(c2ccc([N+](=O)[O-])[nH]2)=O)cnc2cc(Cl)ccc12 c1(CN(C(=O)C(=O)NC(C23CCC(C2)NC3)c2ccc(Br)o2)C)ccc(F)cc1 CCC(C)C(C(C(=O)NCCC1CC1)N(C)Cc1cccc([N+](=O)[O-])c1)OC CC1=CCC(C(=O)N(CC(O)CN(C(=O)C(C)(C)c2ccsc2)C)C)CC1 Cc1nnccc1C(=O)NC(C1CCCC1)CNC(C1(C2(C)CC2)CC1)=O N1(C(c2cc(C)c(Cl)cc2)=O)CCC(C)N(C(c2nocc2Br)=O)CC1 C(=O)(C1=C(Cl)CCCC1)N1C(CNC(C23CCC(OC)C2C3)=O)CCC1 c1(OCC=C)cc(N(CCCNC(=O)C=C(C)C)CCO)sn1 C1(NC(CN(C(C)C)C)=O)COCC1CNC(C1CCOC1)=O c1(CC(=O)NCC(CC)Oc2cccc(Br)c2)ccc([N+](=O)[O-])c(C)c1 CCC(C)(CC)C(=O)N1CCN(C(c2cccc(OC)c2N)=O)C(CCOC)C1 c1(NC(N2CC3CCCC(C3)C2)=O)cnc2[nH]cnc2c1 C1(OC)(CNC(=O)CN2CCNC(=O)C2)CCN(C(=O)CCCn2ccnn2)C1 c1(CNC(C2(C)CCN(C(C(C=CC)O)=O)C2)=O)ccc(O)c(F)c1 c1(C(C)C)ncc(C(N2CCC(NC(=O)C(C)OCCN(C)C)C2)=O)s1 C1(N(C(=O)CCCn2cncn2)CC#C)CCN(C(=O)C(C)c2ncco2)CC1 Cc1ccc(C(N2CC3CC(NC(c4cccs4)=O)C2C3)=O)c(C)c1 c1(NC(CSc2nc(NC(c3nn[nH]n3)=O)sc2)=O)c(Cl)cccc1Cl C(=O)(CCC(CF)CF)NCCN(C)CP(C)(C)=O.c12ccc(cc1)s2 O=C(CC(F)(F)C(F)F)NC1CC1CNC(c1ccn(CCC(F)(F)F)n1)=O N1(C(CCCCC=CC)=O)CCC2CCC(NC(=O)C(C(C)C)SCC)C1C2 C1(C(=O)NCC(C)(C2CCC2)NC(CC=CCC)=O)Cc2nn(C)cc2C(=O)N1 C(CC1=CCN(c2nccc(C)n2)CC1)NC(C(c1cc(C)cc(C)c1)C)=O N1(C(c2cccc(C)c2F)=O)CC2CCCC2(NC(c2cnnc(C)c2C)=O)C1 C1(C(NOCC2(C)CC2)=O)C(C)OCCN1C(=O)C(F)C1CCCC1 Cc1ccc(C(=O)N(C)C)c(C(=O)NCc2cc(Br)ccc2O)c1 N1(C(C(=O)NCCCC=C)=O)C2CCC1CC(F)C2 C1(C(=O)NC(CNC(c2cc(C(F)(F)F)n[nH]2)=O)C2CC2)CCn2ncnc2C1 C1(C(=O)NCC2(C)CC2)COCCN(C(C2OCC3CCCC23)=O)C1 C#Cc1cnc(N2CCC(CNC(c3cnc(F)c(F)c3)=O)C2(C)C)nc1 C1(C2CN(C(=O)CCCCn3ccnn3)C2)(OC)CC1.C1C(=O)NCCS1 N1(C(C(CC)COC)=O)CCCN(C(c2cc3sccc3[nH]2)=O)C(C)C1 c1(NCC2N(C(C3(C)CCC(=O)N3)=O)CCCC2)nccn2nnnc12 N1(C(CCC=CC(C)C)=O)CCC(CO)(CNC(C2(C3CCCCO3)CC2)=O)C1 c1(CCC(=O)NC2OCCC(CNC(=O)OC(C)(C)C)C2)c(Cl)cncc1Cl N1(C(c2ncc(C)cc2C)=O)CC(C)(C)OC2(C1)CN(C(c1[nH]cnc1C)=O)C2 C(c1ccc(C)nc1)=CC(=O)N(CC(CC)NC(C1CCC=CCCC1)=O)CC Cc1ccc(F)c(C(N2CC(NC(=O)CN(C3CCSC3)C)CC(O)C2)=O)n1 CCCCC(CNC(c1sccc1OC(F)F)=O)NC(C1(CF)CC1(F)F)=O CCC1CC(=O)NCC2CCCC2N1C.c1(C(=O)NC)ccnc(CO)c1 C1(CC(=O)NCC2(F)CN(C(C3CCCN3C3CC3)=O)C2)CCC(C(F)(F)F)CC1 Cc1ccn(C(=O)NC2(CCNC(=O)CSCC(F)F)CC2)c(=O)c1 Cc1cc(CC(N2CCC(CNC(c3cnn[nH]3)=O)C2)=O)no1 N1(C(COC(C)=O)=O)CC(CC(=O)N(C(C)CO)C(C)C)CC1(C)C Cc1nnn(CC(=O)NC(C(=O)NC(C2CCCO2)CO)C2CCCC2)n1 C1(NC(C2CCC(CCC)CC2)=O)CC1C1CCCN(C(c2cnc[nH]2)=O)C1 N1(C(CC2(OC)CC2)=O)CCC(F)(CNC(C2C3CC4C(C3)C24)=O)C1 C12(NC(=O)Cc3ccc(CO)cc3)CCCC1CN(C(=O)C1=COCC1)C2 N1(C(C(=O)NCC(F)F)=O)CCC2CN(C(c3ccn4c3CSCC4)=O)C2C1 CCCCCCOCC(N1CCC(OCCNC(C2CCCN2C)=O)C1)=O C12(NC(CCOCCOC)=O)CCC(NC(C3CCCC3C(F)F)=O)(CC1)C2 C(CCN=c1[nH]c(=NCc2cccnc2N(C)C)[nH]c2ccsc12)OCC N12CC(CCC1C)C2=O.c1(CC(C)NC(C2CC2C(N)=O)=O)cnccn1 c1(CC(C)C)ncc(C(=O)NCC2CCN2C(c2cn(CC(N)=O)nn2)=O)s1 c1(OC)cc(Cl)ccc1C(N1CC(CCNC(=O)COC)C1)=O c1(C(=O)NC(CC=C)CNC(=O)CCCCC=CC)ccc(N)c(Cl)c1O N1(C(c2ccn(CC)c2C)=O)CCN(C(=O)C(C)(COC)OC)CC1CC(F)F c1(C(N2CCC(N(C(c3cccc(OC)n3)=O)C)CC2)=O)ccc([N+](=O)[O-])s1 C1(OC)CN(C)C(C)(C(=O)N(C2CCN(C(c3ncc(Cl)s3)=O)CC2)C)C1 C1(N(C(CCOCCOC)=O)CC(=O)NC2CC2)CCN(C2CC2)CC1C c1(CC)cccc(CC(N2CCC(N(C(=O)Cc3nc(C4CC4)n[nH]3)C)C2)=O)c1 N1(C(Cc2c(C)noc2C)=O)CCC2(CCCN2C(C2CCC(C)(C)C2)=O)C1 c1(C(N2CC3N(C(C(CC)=O)=O)C3C2)=O)cc(F)c(Cl)c(Br)c1 Cc1cc2[nH]c(C(N3CCCN(C(=O)CC(=O)NCC4CC4)C(C)C3)=O)cc2o1 c1(CC(=O)OCC)cc(Cl)ccc1Nc1ccccc1.c12csc(n1)NC2=O C1(CNC(C2CC(=O)N(C3CC3)C2)=O)CC(NC(c2cccnc2)=O)C(O)C1 c1(NC(C2N(Cc3cc(C(=O)OC)cc(Cl)c3)CCOC2)=O)cc(Cl)c(O)c(Cl)c1 N1(C(c2cc3nc[nH]c3cn2)=O)CCN(C(c2cnns2)=O)C2CCCCC2C1 CC(C)C1=CCC(C(=O)NC2CCN(C(=O)C(c3cccn3C)=O)C23CC3)CC1 C1(NC(c2c(OCC)cccn2)=O)COC2(CCCN(C(=O)CC3(C)CC3)C2)C1 C1(N(C(C=CC(=O)OCC)=O)C)CCC(NC(c2ccnc(O)c2)=O)CC1 c1(NC(N2CCN(CCOCCO)CC2)=O)c[nH]c2c(F)c(F)c(F)c(F)c12 c1(C(=O)Nc2n(CC(C)C)ncc2)cccc([N+](=O)[O-])c1Cl N1(C(c2n(CC=C)ccn2)=O)CCCC2(C1)CN(C(=O)CC(O)CCCC)CCO2 N1(CC)CCOCC1CC(=O)NC1CN(C(=O)C=CSC)CC1C(N)=O N#CC1CC(F)(F)CN1C(C1CCCN(C(C2CCC(=O)N2C(F)F)=O)C1)=O c1(OC)ccccc1C(=O)NC1CCCC1C(=O)Nc1ccccc1N(C)C C(c1c(C)nn(C)c1Cl)=CC(N1CC(CNC(CC2CC(CC)OCC2)=O)C1)=O CCC(COC1CCCCC1)N=c1c(C#N)c[nH]c2c(C)cccc12 N1(C(=O)NCCN)CCC(O)C(O)C1.N1(C(=O)OC(C)(C)C)CC1C(=O)O C1(=O)CC2=CCN(CC2)C(=O)CC(=O)N2CC(C)N1CC2C.C(C)(C)(C)OC c1(C(=O)NC(CC2CN(C(C(CC)C)=O)C2)C)cc(Br)c(Cl)s1 C1(CC(C)CN)CCCCN1C(c1c[nH]nc1NC(=O)C(F)(F)F)=O N1(C(C2CN(C(CCCCOC)=O)CC23CC3)=O)CCC2(CCCC2)C1 c1(C(=O)NCC2N(C(C3(OC)CCCCC3)=O)CCC2C)cn2c(n1)SCC2 c1(C(=O)NCCCCC(C)NC(=O)C=C2CCN(C)C2)ccn2ccsc12 C12(C(=O)NCC3CC(C)N(C(C4C(C)(C)C4(F)F)=O)C3)CCC(F)(CC1)CC2 N1(C(CCC)=O)CCCC(C(=O)N(CCCNC(=O)C=Cc2cnc(C)s2)C)C1 C=C=C(C)CC(=O)NC(C)CN(C)C(c1cccc(Oc2ccccn2)c1)=O C(=O)(C1=CCN(C(c2cnn(C3CC3)c2C)=O)C1)NCCc1cc(C)no1 c1(OC)cc(NC(=O)Cc2ccccc2NCc2ccc(Cl)c(Cl)c2)cc(Br)n1 Cc1cc(=NCc2cccc3c2CCN3)[nH]c(N2CCCC(N(C)C)C2)n1 Cc1nn(C)c(C)c1CCC(=O)NCC1CC(O)CN1C(C12CC3CC1C2C3)=O c1(C(=O)NC)ccc(-c2cnn(CC3(C(=O)O)CCCCC3)c2)cc1F CC(C)=C=CC(=O)N1CC(O)CC1CNC(c1ccc(C2CC2)nc1)=O CCC(CC)CC(=O)NC1(CNC(C2CC23CCCOC3)=O)CCCC1 Cc1cc(F)c([N+](=O)[O-])cc1C(=O)NC1CN(C(=O)CCS(N)(=O)=O)CC1C Cc1cc(C(=O)N(C2CN(C(=O)C(C)(C)F)CC2F)C)c(S(N)(=O)=O)s1 N1(C(CC2CCCN(C(C(C)(C)CCCF)=O)CC2)=O)CCc2cccnc2C1 Cn1cc(C(C(=O)NCCO)NC(CC(F)(F)F)CO)c(=O)cc1OC1CC1 N1(C(C(C=C)O)=O)CCCC2C1CCN2C(c1cc(Br)cn1C(=O)C1CC1CCCC)=O Cc1nc(C(F)(F)F)oc1NC(C1CC(C)N1C(=O)OC(C)(C)C)=O c1(C(N2CC(NC(=O)Cc3ccc(Cl)cc3Cl)C3C2C3)=O)cncc2[nH]ccc12 Cc1cc(Br)cc2cc(C(=O)NC3CCN(C(C4CCOC(=O)N4)=O)C3)oc12 C#Cc1cc(C(=O)NC2(C)CCN(C(c3ccnn3C(F)F)=O)C2)cc(F)c1 C1(NC(c2cn(CC)nc2C)=O)C2CC1N(C(C1CC3(CCCO3)C1)=O)C2C CC(C(=O)N1CCC(CNC(c2ncn3c2CCC3)=O)C(C)C1)P(C)(C)=O CC1CCCC(N(C(CC2(C)CCOC2)C(=O)NCC2CCOC2)C)C1 CCCC(C)(O)C(=O)NCC1CCC1NC(=O)Cn1nnc(=O)[nH]1 c1(CS(=O)(=O)NCC=C)ccc(NC(=O)C(=O)NC(c2ccc(Cl)cc2)C)cc1 C1(C(N2CC(C=C)C(OC)C2)=O)CC2CCC(C1)N2C(=O)Cn1ncnn1 c1(CC(=O)NCC2(F)CC(NC(CCCN(C)C)=O)C2)c[nH]ccc1=O N1(C(COC2C(C)CCCC2)=O)CC=C(CCNC(=O)CCc2ccccn2)CC1 N1(C(=O)Nc2cc(SCCCCC)no2)CCC(c2ccccc2)C1(C)C Cc1cccc(OCC(=O)NCC2(O)CCCN(C(=O)C(O)CC(C)C)C2)c1F c1(CNC(CCC(F)(F)F)=O)scnc1C1CCCC1 CC(CCNC(=O)C(F)n1cccn1)CCNC(=O)C=Cc1nnc(C(C)C)o1 N1(C(C(C)SC)=O)CCC2(CC1)CCN(C(c1cc(C)c(C)nc1O)=O)CC2 N1(Cc2c(OC)nsc2)C2CCCC1CN(C(c1cncnc1)=O)C2 c1(C(=O)NCC2C(NC(c3nc(COC)oc3)=O)COC2)cc(N)ccc1Cl c1(C(=O)NC(C)CCCNC(=O)C(F)=C2CCC2)ccc(C(F)(F)F)cc1Cl c1(C(=O)NCC2CN(C(C(C(C)C)(C)O)=O)CC2C)cccc2c1NCCC2 N1(CC(=O)NCc2cccnc2)CC2CCC(C(=O)NC(=O)C3=CCOC3)(C2)C1 S(=O)(=O)(c1cccnc1NCc1cnccn1)N1CCCC(CCC)CC1 N1(C(c2ccn(CC)n2)=O)CCC(C2(O)CN(C(=O)C3=C(C)CCC3)C2)CC1 N1(C(=O)Cc2cnoc2)CCC2(CCCN(C(c3cccc4c3NCC4)=O)C2)C1 CC(O)(CNC(=O)CC1CCCO1)CNC(=O)CN(C1CCCC1)C CCCCC(CNC(C1CC1C(N)=O)=O)NC(c1oc(CCC)nc1C)=O c1(C(N2CC(CNC(C(COCC)(C)C)=O)OCC2)=O)cnc2n1CCOC2 C1(NC(=O)NCc2cn(CCC)nn2)CCCC(OC)C1 c1(C(=O)NC(C)(CNC(=O)Cc2cccs2)CO)ccc2oncc2c1 C1(C(=O)NCC2(COC)CCCN2C(c2cccnc2)=O)CC(C)CC(C)(C)C1 N1(C(c2c(CC)ocn2)=O)C(C(=O)N(C)CCNC(=O)CC)C2CC(O)C1C2 Cc1c(C(=O)NCC2CCCCN2C(C2CC(O)C2)=O)[nH]c2c1CCCC2 C(N=c1cccc(N2CC3CCC2CO3)[nH]1)c1n(C(C)C)cnn1 N1(C(c2cncc(OC)n2)=O)CCCC(F)(CNC(c2sc(C)cc2Cl)=O)C1 N1(C(c2ccn(CC(C)C)n2)=O)CC2(CCCC2NC(c2cnc(C(C)C)o2)=O)C1 N1(NC(c2ccc(C=C)cc2)=O)Cc2ccnn2CC1C.C12CCC1NC2=O N1(C(c2n(C=C)ncc2)=O)CC2CC(C(=O)NCc3cnc(O)nc3O)CC2C1 C1(C(N2CC(F)C2)=O)CCCC(F)C1.O=C1COCCN1 N1(C(C=CC2CCN(C(CCOCC(C)(C)C)=O)CC2)=O)CC2C(C1)C2(C)C c1(OC)ccc2oc(C(=O)N(CC(C)NC(=O)C(C)C#N)C)c(C)c2c1 C(CNC(c1ccon1)=O)(CC(=O)Nc1cccnc1)OC c1(CCC(=O)NCCN(CCOC)C(C2COCC(C)O2)=O)ccc(C)cc1C CC1CC(C)CN(CCNC(=O)NCCC2CCCCC2NC(=O)C2CC2)C1 c1(SC)ncc(Br)c(NC2(Cc3ccc(Cl)c(O)c3)COC2)n1 c1(C(N(C)CC2CCCN2C(C2CCC(=O)O2)=O)=O)cccnc1N(C)C N1(C(c2n(C)cnc2)=O)CCC2(CC(NC(C3CCC3)=O)C2)C1 c1(C(N2CCC(O)(CNC(c3c(C)c(Cl)cnc3)=O)C2)=O)cc2cnccc2[nH]1 c1(C(=O)NC(C2CCCC2)CNC(=O)CCOC2CC2)ncoc1C1CCCO1 N1(C(C(c2cccc(C)c2)Nc2cc(O)ncn2)=O)CCN(CCO)C(=O)C1 CC(C)C(F)(F)CC(=O)NC1CCN(C(c2cn(Cc3ccccn3)nn2)=O)C1 c1(C(N2CC3C(NC(C(CC(C)C)F)=O)C3C2)=O)cccc2nccnc12 C1(c2ccc(CC)cc2)CN(C(C2C(C)C2C)=O)CCN1C(=O)C1=CCC1 CC1(NC(c2snnc2C2CC2)=O)CC(NC(c2coc(Cl)c2)=O)C1 N1(C(C(C)CSC)=O)CCC2(CCCN(CC3(C(=O)NC(C)(C)C)CCC3)C2)C1 c1(OCc2nc(-c3cccc(F)c3)no2)ccc(Br)cc1.O=C1CCN1 c1(C(=O)NCC)ccco1.C1(C(=O)NC2(c3nc[nH]n3)CCC2)CC2CC2C1 C1(C(=O)NC(C)C(CO)NC(=O)Cc2ccsc2C)(CC)CC(C)(C)C1 C1(C(=O)NC2(C(=O)NCC3(CN(C)C)CCC3)CC2(C)C)CC(F)C(=O)N1 CCC(CCC(=O)NCCc1cccc(CNC(=O)C(=O)NC2CC2)c1)OCC Cc1cc(C(=O)NCCC2CC(NC(=O)Cc3cc[nH]n3)C2)ncc1F Cc1ccc(C)c(C2N(C(=O)NCC(c3ccco3)N(C)C)C(C)C2O)c1 c1(OC)c(C)cc(C(=O)N(C(C)C)CC2CCC3(CCC3)O2)cc1Cl N1(C(C(C)=CC)=O)CC(C(=O)Nc2ncccc2C2CC2)C(C2CC2)C1 c1(OC2CC(COCC(=O)N(CCNC(C3N(C)CCC3)=O)C)C2)ccc(F)cc1 C1(N(C(=O)CCc2nc[nH]n2)CC)CCCN(C(c2ncccc2C)=O)C1 C=CC(CCC)CC(=O)N1CCC(NC(c2ccccc2N2CCCC2=O)=O)C1 C#Cc1ccc(C(N2CCCC(CC)(NC(=O)CCNC(N)=O)C2)=O)nc1 N(C1COc2cccc(Br)c21)S(c1ccc(Nc2c(C)nc(C)s2)nc1)(=O)=O C1(CC)CN(C(=O)CC23CCC(CC2)CC3)CCC1NC(=O)Cc1csc(C)n1 CCCC(O)C(CO)NCc1ccc(CCC(F)(F)F)cc1 N1(C(CNC(c2c(C(C)C)onc2)=O)C)CCN(C(=O)CC2(O)CCOC2)CC1 c1(C(c2n(C(CC)C)nnn2)NCCCOC(N)=O)scc(C)c1NC(C)C N1(C(c2ccc(C#N)cc2Cl)=O)CCC2(CC1)CC(C(=O)Nc1cc(O)n[nH]1)C2 C=Cc1ccc(C(=O)N(C(C)(C)CC(N2CC3CC=CC2C3)=O)C)cc1 C1(OCC(=O)NCC23C(CN(C(C(C)c4cncs4)=O)C2)C3)CCC(F)(F)CC1 N1(C(C)=O)CCCCC1C(=O)NC1CCN(C(c2cc(Cl)n(C)n2)=O)C1C1CC1 C(=O)(C(C)(CNC(c1n[nH]cc1C#C)=O)CC)N1C(C#C)CCC1 Cn1nccc1C=CC(=O)NCCCNC(=O)CC1CCOC1 N1(C(C(S(C)(=O)=O)C2CC2)=O)CC2CCC(C1)N2C(=O)CCC1CCC(=O)NC1 n1(CCNC(C(F)=CCC)=O)cc(CC(C(=O)OC)C2CC2)nn1 c1(CC(N2C(CN(C)Cc3sccc3Br)CCC2)=O)ccc(Br)nc1 C1(C(=O)NC(C2N(C(c3nc(C(C)=O)sc3)=O)CCC2)(C)C)CC2CC2CC1C N12CCS(=O)(=O)C(C1)CCNC(=O)C2.c1(C(=O)OCC)ccnc(OC(C)=O)c1 c1(C(N2CC(N(C)C(c3ccsc3)=O)C3(C2)CC3)=O)ccnc2c1ncn2C CCC(CO)(C(=O)NCC1CC1C(=O)NCC1CN(C(C)=O)C1)OC C(=O)(C1CCCc2nccn21)NCC(CNC(c1c(C)cc(Br)o1)=O)O c1(C(=O)NC2C(N(C(CCN(C)C)=O)C)CCCC2)cc(C(F)(F)F)ccc1N c1(C(=O)NCC(CNC(CC=CCC)=O)C)cc2cccnc2s1 C(=O)(C(CC=C)C(C)C)NC(C1CCCCC1)CNC(c1nccc(C#C)c1)=O C1(C(=O)NCc2cc(OCC)no2)CN(C(C2(C)CCCN2C)=O)CCN1C C1(C(N2CC3C(CNC(=O)CCc4ccccc4O)C3C2)=O)CC2(CCC2)CO1 Cc1n[nH]c(C)c1S(=O)(=O)NC1CN(c2ncnc3c(Br)csc23)C1 c1(C(N2CC=CC(NC(c3cocn3)=O)C2)=O)c(F)ccc(I)c1F N1(C(C)C)CCCC1C(N1CC(C(C)NC(=O)C=CSc2ccccc2)C1)=O c1(OC)ccc(C(=O)NCC2CCC(C(F)(F)F)N(C)C2)nc1Br c1(CC)cc(F)ccc1C(=O)NCC1CCCC1NC(=O)C1=C(Cl)CCC1 C(C(C)(C)CC(F)(F)F)NC1N(Cc2ccc(OC)cc2)CC(OC)C1 c1(CC)ccc(OC)cc1C(=O)NCC1CCCN1C(=O)C(C1CC1)SC C1(CC(=O)NC(CN(C(c2ncn(C)n2)=O)CC)C)CCc2ccccc2C1 Cc1nc2c(n1C)CN(C(c1ccc(CO)o1)C(=O)NCC1CCCO1)CC2 O=C(C1=CCOCC1)Nc1cccc(C2(Oc3ccccc3)CC2)c1 Cc1csc(=O)n1CCCNCC1CCC(CNC(=O)OC(C)(C)C)C1 CC1=C(C(=O)NCC2CN(C(=O)C(C)CC3CCCO3)C(C)(C)C2)CCO1 c1(C(N(N2CCCCC2)C)=O)ccc(-c2cc(C(F)F)[nH]n2)cc1 C1(NC(c2ccc(C(F)F)cc2)=O)CN(C(=O)Cc2sc(O)nc2O)C2CC12 C(=O)(C1=C(C)OCCS1)N(C(CCNC(C1C(C(=O)OCC)C1)=O)C)CC C1(NC(C(C2CC2)OCC)=O)(CO)CCN(C(=O)CCN2CCCS2(=O)=O)CC1 Cn1nc(Br)c2ncnc(N3CCC(NC(c4ccnc(Cl)c4)=O)C(C)(C)C3)c12 C1(C)(C(NOCCC#C)=O)CC(O)CN1C(c1c[nH]nc1COC)=O c1(C(N2CCN(CCOC)CC2)CNC(CC=C=C)=O)cccc2cnccc12 C1(NC(c2nccc(C#C)c2)=O)CN(C(c2cscc2Cl)=O)C2(CCOC2)C1 C=CCCC(C)(c1nnnn1CCCC1CC1)NCC(C)(C)SC c1(CC(=O)N(CCCNC(C2(C)CC(F)(F)C2)=O)CC)c[nH]c(=N)nc1O C1(NC(C2C(C)C2)=O)CCN(C(=O)C=Cc2ccoc2)CCC1c1ccccc1 N1(C(C(CCC)CCC)=O)CCc2sc(CNC(=O)COCC3CC3)nc2C1 Cc1cc(C(=O)NCCC(C)(C)CNC(c2cnc(S)[nH]2)=O)cc(O)n1 N(C(=NCC1C(C)(C)C1(C)C)NC(c1cccs1)C)CC1(C#N)CCC1 c1(C(C#N)NCC(=O)Nc2c(C(=O)OC)cccc2)nc(Cl)ccc1Cl CCN=c1nc(C(=O)NC2CN(C(=O)C(C)=CC)CC23CC3)cc(C)[nH]1 c1(OC)ccc(Cl)c(C(N2CC(O)CC2CNC(c2ccc(OC)cc2)=O)=O)n1 C=CC(CC)CC(=O)N1CCCCCC1CNC(c1sncc1CC)=O c1(C(=O)NCCC(C)NC(c2cc[nH]c2-c2ccccc2)=O)ccc(F)cc1Cl N1(C(c2[nH]ccc(=N)n2)=O)CCN(C(=O)CCc2nccs2)C2CCCCC2C1 C(=O)(CC(CC(C)C)NC(c1ccc(C#N)s1)=O)NC1CCN(C(CC)=O)C1 N1(C(=O)CSc2ncccn2)CC2CN(C(c3ccc[nH]3)=O)CC2C1 N(C1CCCn2cnnc21)C(C(CCSC)NC(C1CC2CCCC2C1)=O)=O c1(NC(C2N(C(c3ccc(CC)cc3)=O)CC=C2)=O)ccc(S(N)(=O)=O)cc1Cl C=CCCC(CCC)(c1nnnn1-c1ccccc1Cl)Nc1ccc(COC)nc1 C(CCCC(=O)NC(C)CCF)NC(C(C)C1CCOC1)=O C(=O)(CC(C(F)(F)F)NC(c1ccc(F)c(C2CC2)c1)=O)OC C1(COC)(NC(=O)CCc2cnn(C)n2)CN(C(=O)Cc2ccc(C)o2)C1 c1(C(=O)NC2C(CNC(c3cc(N)c(Cl)nc3)=O)CCC2)ccc2cnnn2c1 C12N(CCC1(C)C)C(=O)C(=O)NC(=O)C21CCC1.Cc1cc(C(F)(F)F)ns1 N1(C(C(c2ccccc2)OC)=O)CCC(C2CC(NC(c3cc(C)c[nH]3)=O)C2)C1 C12(C(=O)NCCN(C(CCNC(=O)NC)=O)C(C)C)CCCCC1NC(=O)C2 C1(C(N2CC(C)(NC(c3coc(O)n3)=O)C2)=O)COCCN1S(C)(=O)=O c1(OC)cc(NC(N2CC(CO)C2(C)C)=O)c2cc(OC)ccc2n1 Cc1cccc2cc(C(=O)NCC3CN(c4cncc(Cl)n4)CCC3(F)F)[nH]c12 N1(C(C2CN(C3CCC3)C2)=O)CCN(C(C2(n3cccn3)CCC2)=O)C2(CCC2)C1 N1(C(C2CCC=CCCC2)=O)CCC(C)(C(N2C(C(=O)OC)CCC2C)=O)CC1 O=C(Cc1cccc(OC)c1C(F)F)NNC(=O)N=c1cc2n([nH]1)CCCC2.C1(N)CC1 CCC(O)C(C)C(=O)NCC1(O)CCN(C(c2cnc(C(C)=O)s2)=O)C1 N1(C(C=C(CC)C)=O)CC(CNC(C2(S(C)(=O)=O)CCOCC2)=O)C2(CCC2)C1 C(C)(C)(CCC(=O)NC1CCCC1(C)O)NC(CNC(=O)OC)=O N1(C(c2ncccc2Cl)=O)CCC2C(C1)CN2C(=O)CCSCc1ccccn1 N(C(=NCCc1cccc(C#N)c1)NCC1(Cl)CCCCC1)C1C(C=C)C1 N1(C(c2cc(C)no2)=O)CC(N(C)Cc2nnsc2Cl)C(C)(C)C1 C(CC(C(=O)NCC1(C(C)(F)F)CC1)NC(C12CC(F)(C1)C2)=O)N(C)C c1(CCC(N2CCN(C(=O)C3CC3)C(CC(F)(F)F)C2)=O)ccc2c(c1)OCCO2 c1(C(N2CCOC(CS)C2)=O)cnc(O)cc1C(=O)O.c1(C)cn(C2CC=CC2)nn1 C(=O)(C1CCOc2ccccc21)NCC1CC(NC(C(c2cn(C)nc2)=O)=O)C1 CC(=O)CCCCC(=O)N1CC2(CCCC2NC(c2sc(C)cc2C)=O)C1 N1(C(C(CCOCC)NC(=O)CC2C(=O)NN=C2C)=O)CC2(CC=CC2)C1 C1(CNC(C2C(CC)C2)=O)C(C)CCN1C(=O)CCN1CCNC(=O)C1 Nc1cccnc1C(=O)NC(CC1CCCC1)C(N1CCCC(F)C1)=O c1(C(CNC(C(CC)C)=O)NC(=O)Cc2cccc(Cl)c2)ccc(F)cc1 C(=O)(C(F)(F)CO)N1CC(CC(C)NC(c2cnc(-c3cnn(C)c3)s2)=O)C1 CCCS(=O)(=O)C(C)C(=O)N1CCCCC1CN(C(=O)C(C)c1cccs1)C C(=O)(CCCC(=O)NC1(C)CC(CNC(=O)CC(O)CC)C1)NCCC C(C(CNC1(c2nnnn2CCN2CCOCC2)CCOC1C)C(C)C)OC C12(CNC(CCCCCC)=O)COCCN1C(=O)CN(C(C1CCC1(F)F)=O)C2 C(=O)(C(Cc1cccnn1)N(C)Cc1ccsc1)NC(CC)C C(=O)(CC(C)(O)CCC)N1C(C(NOCCC)=O)CCC1 c1(CNC(CC2CCN(C(C(CC)C)=O)C2)=O)ccc(OC)nc1 C12CCN(C(=O)C(C)=CC1=O)O2.C=CC1CCN1C(C1CCCCC1)=O CCCC(O)CC(=O)NCC(CC)NC(=O)C(F)(F)C(O)c1ccccc1 N1(C(C(C)(C)C2CCN(C(=O)Cc3cc[nH]c3)C2)=O)CC(O)C(O)C1 Cc1n[nH]cc1CCNC(C1(NC(c2csnn2)=O)CC1(C)C)=O c1(N(C)CC2CC2)nc(N2CCS(=O)C3(CCC3)C2)nc2c1CCCCCC2 C1(C(=O)NC(C2CC3(CCC3)C2)C)CC2CC2N1C(C1CCN(C)CC1)=O C12(CC(=O)NCC(c3cncs3)NC(C(C)C3CCCO3)=O)CCC(CC1)CC2 c1(CC)c(C(=O)NC2(CNC(=O)C(C)C(C)(C)C)CC2)cccc1F Cc1nc(NC2CCN(C(=O)CC3CC4CCC(C3)N4C)C2)c2c(C)csc2n1 N1(C(C(CC=C)NC(C)=O)=O)CCC2(CC1)CC2C(=O)N(CCCF)C N1(C(C2(C)CN(C)C(=O)C2)=O)CCN(C(C2CNC(=O)N2C)=O)CC12CC2 C=CCC1CC(C)OC(=O)CNC(=O)N1.c1(CNC(=O)CCOCC)ccsc1 CCC(C)(C)C(O)C(=O)NCC(CC1CC1)C(=O)N1CC(C(F)(F)F)C1 C1(C(=O)NCC=CCNC(=O)CCc2ccsc2)CCC2CC2CC1 c1(C(N(CC(CN(C(C(C)NC(=O)NC)=O)C)O)C)=O)ccnn1C(C)(C)C Cn1cc2c(NC(C3(CNC(=O)OC(C)(C)C)CC(F)(F)C3)=O)ccnc2n1 N1(C(C2(COC)CCCC2)=O)CCC2C(C1)CN2C(c1cccc2scnc12)=O C1(OC)CCCCC1C(c1ccc(C2CC2)cc1)NC(c1cccnc1)C C1(CC(=O)NCC(CC=C)NC(=O)CCC2CCOC2)CC2C=CC1CC2 Cc1ccc2occ(C(=O)NCC34CC3CN(C(c3ccc(Cl)cc3)=O)C4)c2c1 CN1CC(O)CC1(C)C(N1CCCC(NC(c2cc(O)n(C)n2)=O)CC1)=O C1(NC(C(COC)C)=O)CN(C(=O)C(C2(O)CCCC2)F)CC1F C1(NC(c2c(C)cccc2C)=O)CC2CC(C1)N(C(C1CCN1C(C)(C)C)=O)C2 N1(C(C2C3N(C(C4(C(C)(C)O)CC4)=O)CC(C=C3)C2)=O)CCN2C(=O)NCC2C1 c1(C(N(CCCCN(C(C2(CCC)CC2)=O)C)C)=O)cnc(C#N)s1 C1(C(C)=O)CC(C(=O)NCC2(NC(=O)C(F)(F)c3nccs3)CC2)C1(C)C C1(O)(CN(C(COC)=O)C)CCCN(C(C2CCC(=O)N(C3CC3)C2)=O)C1 CCC(CCC(=O)Nc1cccc(CO)c1C)NC(=O)CCc1ccco1 c1(C(N2CC(F)CC(NC(c3n[nH]c(C4CC4)n3)=O)C2)=O)coc2ccc(F)cc12 N1(C(CCC(C)SC)=O)CCC(F)(Cc2ncc(-c3cccc(Br)c3F)o2)CC1 N1(C(C2=C(C)CCC2)=O)CC(NC(C2(Cc3ccccc3)CC2)=O)CC(F)(F)C1 CC1CC2(CCN(C(=O)C3=COCCC3)CC2)CN1C(C1CCCC(C#N)C1)=O c1(OC)c(NC(C2C3CCC2(c2ccccn2)C3)=O)cccc1C(F)F c1(C(N2CCCCCC2)C(=O)NC2CCCC2)cn2c(n1)CCCCC2 C1(c2n(C)cnn2)CCCC1NC(=O)N(N1CCOCC1)CC1(C2CC2)CC1 C1(NC(C(CCCC)O)=O)CN(C(c2cn(C(F)F)cn2)=O)C2(CCC2)C1 C1(NC(c2c(Cl)cc(C)s2)=O)CC2CN(C(c3conc3C)=O)CCN2C1=O C(CCS(N)(=O)=O)NC(C1C(OCCCC(=O)NCC)CC1)=O.OCC C1(NC(CC(C)C)=O)CCC(C)(C(=O)NCC2CN(C(N)=O)C2)C1 c1(C(N2CC(O)(C(C)NC(c3cncs3)=O)C2)=O)[nH]nc2c(=O)n(C)ccc12 CN1N=C(CC(=O)NC2CN(C(=O)CN3CCSCC3)CC3CC23)CC1=O CC1(C(F)(F)F)CCN(C(=O)COC(C2(c3ccccc3)CCC2)=O)C1 C(C)(CCC(=O)N1CCOC(CNC(c2cn(CCC(C)C)nn2)=O)C1)OC N1(C(CC(C)=O)C)c2ccccc2CC1C1(CN)CC1 c1(CNC(c2cccnc2O)=O)cc(O)nc(CNC(C2(CO)CCC2)=O)n1 c1(OC)ccc(C(=O)NC(C)CC2CCN(C(c3cccs3)=O)CC2)c(C)n1 N1(C(c2ccc(CC)nc2)=O)CCC(CNC(=O)CN(C2CCC2)C)(OC)CC1 c1(OC)ccccc1C(CNC(=O)C(C)NC(N)=O)NC(=O)CC1CCN(C)C1 c1(CCNCc2cc(C(=O)OC)[nH]c2)cncc(C)n1.C12CC1C(=O)NC2 C1(C(N2C(CNC(C(C)OCC=C)=O)CCCCC2)=O)CCc2nccn2C1 C1(CC)CN(C(=O)C(C(C)OC)NC(C2COC(=O)N2)=O)CC1F CN1CC(C(N2CCN(C(=O)CC3CS(=O)(=O)C3)C(CF)C2)=O)CNC1=O C12(C(=O)NCc3ccon3)CCNCCC1C2 N12CCC(C)C(C1)Nc1nsc2n1.C(=O)(C(C)(C1(C)CC1)OC)OC Cc1csc(C=CC(=O)NCC(C)N(C)C(C23CCC(CC2)C3)=O)n1 N(C(=NCCCCS(C)(=O)=O)N1CCC=C(C)C1)Cc1ccn(CC)n1 c1(CN(CCNC(c2nnc(C)o2)=O)CC)cccc(C(N)=O)c1 C(=O)(C1CCCc2ncnn21)NC1(C)CCCN(C(CCC#C)=O)C1 c1(-c2cn(-c3ccc(NC(C4CCN(C)C4)=O)cc3)nn2)cc2ccccc2o1 CCCC(C#N)C(=O)N1CC(NC(c2cc(-c3cnn(C)c3)on2)=O)CC1(C)C N1(C(COCC#C)=O)CC(NC(=O)C(CC#C)C2CC2)C(O)C1 N1(C(C(CC=C)CC)=O)CC2CCC1C(CNC(c1ccc(CCC)[nH]1)=O)C2 N1(C(CC2(NC(c3nc(C)c(Br)s3)=O)CCC2)=O)CCc2cc(F)c(F)cc2C1 c1(OC)ccc(C(=O)NCC2CC(OC)CN2C(C2CNC(=O)N2C)=O)cc1F c1(C(C2CC2)CNCC2(OC)CC(CO)C2)ccc(Cl)cc1 CC1(C)CCC(C(=O)NC2(C(=O)Nc3cc(F)ccc3O)CCSC2)CO1 N1(C(CN(C)C(=O)C2CC2)=O)CCCC12CCN(C(c1cc(N)c(Cl)cn1)=O)C2 N1(C(COc2c(C(C)C)cccc2)=O)CCC12CCC(C(=O)O)CC2 Cc1ccc([N+](=O)[O-])cc1C(=O)NC1CCN(CCCS(N)(=O)=O)C(C)C1 C(c1cccc(F)c1F)=CC(=O)N(C1CCCCC1NC(C1CC(C)=NO1)=O)C CC1(C)COC(CC(=O)NCCC2CN(C(=O)Cc3ccn(C4CC4)n3)C2)CO1 C(=O)(C(COC)COC)N(CC(C)(CO)NC(c1cnc(CC)[nH]1)=O)CC Cc1cccnc1C=CC(=O)NCCN1CCN(C(C2(C)C=CCCC2)=O)CC1 N1(C(CNC(c2n(CC)ncc2)=O)C(F)F)CCN(C(=O)CC2CCOC2)CC1 c1(OC)cc(N2CC3CC(NC(=O)C(C)=C4CCC4)C3C2)ccc1[N+](=O)[O-] C1(C(=O)NC2CCC23CN(C(c2cc(Cl)c[nH]2)=O)C3)CCc2nccn2C1 C1(CC)CN(C(c2ccn(C(C)C)c(=O)c2)=O)CCN1C(c1[nH]cnc1C#N)=O CC(O)C(C)(C)C(=O)NC1CN(C(C2CC(=O)N(CC(F)(F)F)C2)=O)C1 NS(=O)(=O)c1n[nH]cc1C(N1CCC12CN(C(c1ccnc(Cl)c1O)=O)C2)=O C1(F)(C(=O)NCc2cc(C(N3CCC(CF)CC3)=O)cs2)CCCCC1 N1(C(C2CC(C)SCC2)=O)CC2(CCN(C(c3cc4ccccn4n3)=O)CC2)C1 C(c1cncn1C)=CC(=O)NC1CCC(N(C)C(c2cccc(Br)c2)=O)C1 C(C)(C)(CC(=O)NC(C1CC2CCC1C2)C)NC(C(C)N(C)C)=O N(C(=NCCc1ccccn1)NCc1ccc(C(N)=O)cc1)CC(C)C1CCC1 c1(C(=O)NCC(C)N(C(C(C)OCC#C)=O)CC)cnc(CCC(F)(F)F)s1 C(=O)(CCC(=O)N1CCC(F)(CNC(=O)CC2CCC(C)(C)O2)C1)NC N1(C(C2C(=C)C2)=O)CCCC2(NC(c3cnc4ccccn34)=O)CC2C1 N1(C(c2c(C)nns2)=O)CCN(C(=O)C(C)C=Cc2ccc(F)cc2)CC1CF C1(CNC(CC=CCC)=O)CCCC(OC(=O)C(C2CCCC2)OCC)C1 C(=O)(CCC(C)(C)C#N)N1CC2C(NC(c3cc(OCC)no3)=O)C2C1 N1(C(Cc2scc(C)c2)=O)CC2CCC(NC(c3ncn(C(C)C)n3)=O)CC2C1 C12(N(C(CCN(C(=O)CC3C=CCCC3)C)=O)CCO)CCC(CC1)C2 C1(NC(C2(CCCC)CCC2)=O)CCCCCC1NC(=O)CC1CCN(C)CC1 c1(OC)nscc1C(=O)NC1CC(O)C1CC(=O)NCc1cnc(C2CC2)o1 C1(NC(c2cn(CC=C)nn2)=O)CCN(Cc2nc(O)n[nH]2)C(C)C1 CCC(CC)(CCC(=O)OC1CCCC(S(C)(=O)=O)C1)[N+](=O)[O-] C(=O)(C(O)C(F)(F)F)NCC(C)(C)CNC(C1(n2cccn2)CCC1)=O c1(C(=O)OCc2ccsc2)ccc(NC(N2C(CC)CCCC2)=O)cc1Cl c1(C(C)OCC)nc(C)c(C(=O)C2CC2)s1.N1CC(CNC(C)=O)(OC)C1 N1(C(C2C(C)CCC2)=O)CC(C2CN(C(c3cc(C(C)C)nc(O)c3)=O)C2)C1 CCC(C)(CNC(=O)C(F)(F)c1cccnc1)NC(c1csc(=N)[nH]1)=O C1(C(=O)NC2(CCCNC(c3c(C)ccnn3)=O)CC2)CCC2(C1)CC2(F)F Cc1ccnc(CNC(=O)N(C)Cc2nnn(C(C)C)n2)n1 CC1(C)CCOC1CNC(=O)C(CC1CCOCC1)NC(=O)CC1CCSC1 CCCCC(CC)C(=O)N1CCN(C(c2cc3ncccc3o2)=O)CC1C1CC1 O=C1COc2cc(F)c(C(N3CCCC(NC(C4CNC(=O)C4)=O)C3)=O)cc2N1 C1(C(=O)NC2C(CNC(CN(C)CC)=O)C2)CCCN1C1CCCC1 C1(CNC(c2ccc(C)cn2)=O)COCCN(C(C2(C)COC(=O)C2)=O)C1 c1(CN(C2CCC3(CCC3)C2)C=O)ccc(F)c(C(F)(F)F)c1 c1(OC)c(C(N2CCC(CNC(c3cccnn3)=O)C23CC3)=O)ccnc1Cl C1(C(=O)NC(CC)C2CCC2)CCN(C(=O)Cc2ccsn2)C1 O=[N+]([O-])c1cc(F)c(N2CCN(CC3CCNC3)CC2)c(F)c1 c1(C(=O)Nc2c(F)cc(O)cc2F)n[nH]c2c1CN(C(c1nc(Br)cs1)=O)CC2 c1(NCc2ccc(C)c(F)c2)ccc2ncc(-c3ccc(C(F)(F)F)nc3)n2c1 N1(C(c2nc(OCC)oc2)=O)CC(C2CN(C(=O)C(C(C)(C)C)NC(C)=O)C2)C1 c1(OC)ccnc(NC(=O)NCc2ccc(SC)cc2)c1.C123CCC(C1C2)O3 Cc1cc(-c2cn(C3CC3C(C3CCCOC3C)=O)nn2)c(C)cc1Cl CCC(C)(COC)CNC(=O)C=CC(C)NC(=O)C(c1cncnc1)C C(=O)(C1=CCC2CCC1N2C(C12C=CC(CC1)C2)=O)N1CC(OCC)(COC)C1 C1(C(=O)NC(C)(CNC(=O)CC2C=CCC2)C2CC2)CC2(C1)CC(F)(F)C2 N1(C(c2nnn(CC)c2C)=O)CCN(C(C2(C(F)(F)F)CCC2)=O)CC1CF C1(C)(C(=O)NCC(C2CC2)NC(c2c(OCC(C)C)nccc2)=O)CCCC1(F)F C(=O)(C(C)Cc1ccco1)NC1C=CC(=O)NC1.O(C(F)(F)F)CC(C)O CC1CCC(NC(=O)Cc2cccnc2)CN1C(c1cccc(F)c1N)=O CCCC(C)CC(=O)N(CC(=O)N(CC(C)OC)C)CCn1cc(C)cn1 c1(C(=O)NCC2(CNC(C(C)(C)C)=O)CC2(F)F)cnn2c(=O)cc[nH]c12 C(C(C(C)(C)C)NC(c1cc[nH]n1)=O)NC(C(n1ccc(C(F)(F)F)n1)C)=O C(C)(C)(CCC(=O)N1CCC(CO)C(O)C1)NC(c1n[nH]c(C)c1Cl)=O C1(C(=O)NCC(n2ccc(C)n2)C)CC2(CCC2)CN1C(=O)COC(=O)N(C)C N1(C(C=C(C)C(C)(C)C)=O)CCC(O)(CNC(=O)CCc2ccnc(Cl)c2)C1 C1(NC(=O)C(c2ccc(F)cn2)(F)F)CC12CCN(C(c1coc(Cl)n1)=O)CC2 c1(C(N2CCCC(OC)C2)C(=O)N(C2CCCC2)CC(C)C)cccc2ncnn12 c1(CC)ccoc1C(=O)NC(Cc1cc[nH]n1)C(=O)NC1CCCSC1 c1(C(=O)NCC2C(NC(c3cccc(CC=C)c3)=O)C2)ccc(OC)cc1Cl C1(C(N2CCC(n3nccn3)CC2)C(=O)NCCCC)CCC2(CC2)C1 CC1(C)CN(C(c2cc(N)c(O)c(F)c2)=O)C(CNC(=O)C(=O)NC2CC2)CO1 N1(C(c2c(CC)cco2)=O)CCC(C)CC1C(=O)NCC(C)(F)C(C)C N1(C(C=C(C)C(C)C)=O)CCCC(C(C)(O)CNC(=O)CCCn2ccnn2)C1 C#CC1(C(=O)NCCCC(O)CO)CCN(C(=O)C(C)CSC)C1 C1(CNC(C2C(C)N(C)CC2)=O)CC2(CCN(C(c3cncs3)=O)CC2)C1 N1(C(CC2C(C)(C)C2)=O)CC(C2CN(C(c3ccc(CO)c(F)c3)=O)C2)C1 C1(NC(Cc2nnc(CC)o2)=O)CCN(C(=O)CN2C(=O)CNC2=O)C12CCC2 C1(C#N)(C(=O)NC2C(NC(C3N(C(C)=O)CCCC3)=O)CCCC2)CCCOC1 N1(C(C(C)CF)=O)CCCCC1CCC(C)(C)NC(=O)C=Cc1ccncc1 c1(C(N2CC(C(=O)Nc3ccc(CC#N)cc3)C2)=O)cc(Cl)cc(Cl)n1 C1(NC(C(COC)O)=O)CC(NC(=O)COc2ccsn2)C(O)C1 c1(CC(=O)NC(C)CCCNC(c2c[nH]cc2Br)=O)noc2ccc(F)cc12 c1(C(c2nnnn2C2CCOCC2)NCC(C)(C)SC)cc2cccnc2o1 N1(C(c2cccnc2Cl)C)CC2CC(C(=O)Nc3ccc(=N)[nH]n3)CC1C2 C(=O)(C1=C(C)CCCC1(C)C)N1C2CN(C(CC(CC)(F)F)=O)C(CC2)C1 C1(NC(=O)NCC(c2ccccn2)(C)C)CCCCC1Oc1ccon1 CC1(CNC(c2cnoc2-c2ccc(Cl)s2)=O)CCCN(C(C2(F)CC2)=O)C1 C(=O)(C1=CC2CCCCCCC12)N1CCN(C(c2cccnn2)=O)CC(C)CC1 c1(CC)ocnc1C(=O)NC(C)C(=O)N(CCCN1CCOCC1)C c1(CN(C(=O)C(=O)N(CC(F)F)CCC2CCCO2)C)cccc(F)c1 C(C(O)CN(C(=O)CCC1CCCO1)C)N(C)CC1CCOC1 C1(C2CC2)(C(=O)N)CCC1.C1(C(NOCc2cn(C)nc2)=O)C2CCC(F)C12 c1(C(N2CCC(C(=O)NOC)(CC#C)C2)=O)n[nH]c2c1COC2 C1(CNC(CC2CC(CC)C2)=O)CC12CCN(C(=O)COc1cncc(C)n1)CC2 N1(C(c2c(C)nncc2)=O)CCC2CN(C(c3oc(Br)nc3C)=O)CC12 N1(C(C2N(CC)CC2)=O)C2CCC1(CNC(=O)Cc1c(C)cccc1Cl)CC2 c1(C(=O)NC(CNC(C(CC)C(F)(F)F)=O)(C)C(C)C)ccc2nccnc2n1 N1(CC)CCCC1C(=O)NC1CCCC1C(=O)N(C1CCCC1C)C c1(N(C(=O)CCCNC(=O)Nc2[nH]ccc2C)CC)ccccc1C C1(C(N2CCC(OCC(=O)N(CC(C)O)CC(F)F)C2)=O)CC(O)CN1C C(C(=O)N1CC2CCC2(CCNC(c2cscc2C)=O)C1)(C(C)(C)C)OC N1(C(c2c(C)nc[nH]2)=O)CCC2CC1CN(C(c1cn[nH]c1C)=O)C2 Cc1cc(CCC(N2CCCC(CNC(=O)C(C)(C)C3CCCO3)C2)=O)n(C)n1 c1(C(N(C(C(C)C)C)C)=O)occc1CNC(=O)CC1(N(C)C)CCC1 C1(NC(C(CC)CO)=O)CCN(C(=O)CC2CC(O)C2(C)C)CCC1CO Cc1csc(C(=O)NCCC(Cc2ccccc2)NC(=O)Cc2nncn2C)c1 C1(CNC(C(C)P(C)(C)=O)=O)CN(C(=O)C=CCN2CCCC2)CC12CCC2 C(=O)(C1=NOC(C)C1C)NC1(CO)CCN(C(c2c(C)n(C(C)C)nc2)=O)C1 CC1CCC(CC(=O)NCC2CC(F)(CNC(=O)CCc3cnc[nH]3)C2)O1 N1(C(C2C(C)CC(=O)NC2)=O)Cc2[nH]nc(C(=O)NCCCC3CC3)c2C1 N1(CC2CC(O)(CC)C2)CCOCC1CC(=O)NC(c1c(CC)ocn1)=O CC1CC(NC(C2CCC(F)CC2)=O)CN1C(C1CC(=O)N(C)C1)=O C(=O)(C(CNC(=O)C(C1CCCCC1)C)N(C)C)NCC(COC)O c1(CC)ccccc1CNC(=O)CC1CCN(C(=O)C=Cc2ccccc2)C1 C1(CCNC(CNS(C)(=O)=O)=O)CN(c2ncc(I)cn2)CCS1(=O)=O C(CCCCCC(=O)NC1CC12CCCCCC2)NC(c1cn(CC)nn1)=O N1(C(C(C)c2cncs2)=O)CC2(CNC(=O)CCCOC(C)(C)C)CC1CO2 C1(CC)CN(C(c2ccccc2Br)C(=O)NCCC#N)CCO1 c1(NCC2C(C)CN(C(c3ccc(=O)oc3)=O)C2)ncnc2c(Br)nn(C)c12 C=CCC(C)(C)CC(=O)N1CCCC(C)(C)C1C(=O)NC1CC1C1CC1 C(CC(C)C)(C(=O)NC1CCC1CNC(C1CC(OC(F)(F)F)C1)=O)OC c1(CN(C(=O)CC=CCNC(c2ccc(C3CC3)o2)=O)CC)cn(C)nn1 N1(C(C2C3CC(=O)CC32)=O)C(CC(=O)NCCn2ncnn2)C2CCCC12 N1(C(CC(CCCC)O)=O)CCC2(CCCN2C(=O)C(C)c2cccs2)CC1 n1(CCNC(C(C)C2CC2)=O)ccc(C(=O)N(C2(CC3CCOCC3)CC2)C)c1 C1(NC(c2cc(CO)ccc2F)=O)CC2(CCN(C(C3C4CCCC34)=O)CC2)C1 CC1ON=C(C(=O)N2CCN(C(=O)C=Cc3ccc(F)cc3F)CCC2C)C1C Cn1ncc(Cl)c1CC(=O)NC1CCC(F)(CNC(=O)Cn2nnc(=O)[nH]2)C1 C1(C(CC)C)CCN(C(=O)C=CC2CCCN2C(=O)CC2CCC(C)CC2)CC1 Cc1ncc(Cl)c(C(=O)NC2CCC(NC(C3CC34CC4)=O)C2)n1 N1(CC(=O)OC(=O)NC(C(=O)NCCOC)C)CCCC(NC(=O)C(C)C)C1 C#Cc1ccc(C)c(NC(c2ccc(CNC(c3coc(C(N)=O)c3)=O)cn2)=O)c1 CC(CCNC(=O)CCc1cccc(F)c1)CCNC(=O)CN(C1CCCC1)C c1(NC(C2CCCN(Cc3ccc(O)cc3Br)CC2)=O)ccc(I)cc1C(=O)O CC(C(=O)NC1CC(CC(=O)NCCCN(C)C)C1)=CC(C)(C)C N1(C(C2(COC)CCC2)=O)CC2CCC(C1)N2CC(=O)Nc1ccc(F)cc1Cl CCC(CC)CC(=O)N(C1CCC(NC(c2cccc(C(=O)OC)c2)=O)CC1)C Cc1ccc(O)c(CC(C(=O)CCCNCC)=O)c1.C1(CN)(NC(=O)C2CC2)CCOC1 CON=CC(=O)N1CCC(n2cc(CNC(=O)CSCC(N)=O)nn2)C1 c1(NC(C(C)N(C(COC(CC)C)=O)C2CC2)=O)cc(C)cc(Cl)c1 N1(C(COCc2c(C)cccc2)=O)CCC(NC(=O)CN=S(C)(C)=O)C(C)C1 Cc1cc(C)c(NC(=O)CC2C3CCCC3N2C(=O)C(C)C(O)C(C)C)cc1N C12(CC(=O)NCCCCC3CN(C(=O)C=Cc4cc[nH]n4)C3)CCCC1C2 C1(NC(c2cc(C(F)(F)F)n[nH]2)=O)CC2CCC1CN(C(C1CSCCS1)=O)C2 C(C)(CC(=O)NC1CCCC1NC(=O)CCOC1CCC1)SC C(CCC[Si](C)(C)C)N(C(C#C)C1CCC1)C1CCC1 C1(C(=O)NC2C(CNC(=O)CCC3OCCO3)CC2)CC2C=CC1C21CC1 C1(NC(C(C)C2CCC2)=O)CCCCN(C(=O)CCc2ccccc2)CC1 N1(C(C2CC(OC)(OC)C2)=O)CCC(CC(=O)NCC(F)(F)Cl)CC1 N1(CC(=O)NCC2(CNC(Cc3c(C)ncs3)=O)CCC2)CCCCCC1=O c1(NC(C2N(Cc3c(OC)ccs3)C3C(C2)C3)=O)cnc2c(Cl)cccn12 Cn1nc2c(c1C(N1CC(CCNC(C3CCCC34CCC4)=O)C1)=O)CSCC2 c1(N(CC(O)CO)C)cc(Br)ccc1S(=O)(=O)NCC1CCOCO1 c1(C(C(=O)NC2(C)CC2)N(CCC2=CCCCC2)C)cnc2c(c1)COC2 c1(C(=O)NC2CCC(C)(CNC(C3(COC)CCC3)=O)C2)cccc2[nH]ncc12 C(=O)(CCCCN=[N+]=[N-])N1CC2C(CCNC(C=CC)=O)(CC2)C1 c1(NC)nccc(C(=O)NCc2cc(C(=O)NC3CCCC(CO)C3)n[nH]2)n1 C(F)(C(=O)NCC1(CC(N)=O)CC1)=CCC.C1C(C)(C)OCC(=O)N1 Cc1cccc(CN(C2CC3CC3C2)C(=O)CC(F)F)c1.N12CCCC(C1)C2=O N1(C(C2CCCCO2)C(=O)NCCCOC)CC(C)CSc2ccccc21 C1(CNC(C(c2c(C)cccc2)C)=O)CN(C(c2nocc2C)=O)CC1(C)C C1(C(=O)NC(C2CCCN2C(=O)CC(C)(C)O)C)CCC2(CC1)CC2 n1(CC(=O)NC2CN(C(=O)Cn3cccc3)CC2O)c(C(F)F)nc2ccccc12 N1(C(c2c(C)scn2)=O)CCC(C)C1CNC(c1cnccc1Br)=O N1(C(CCCN(C(=O)OC)C)=O)CC2CC1CCC2NC(=O)Cc1ccon1 C1(C(=O)NCCCNC(C(C2CC(F)(F)C2)OC)=O)CCCN(C(N)=O)C1 c1(SCC(N2CC(O)(CNC(=O)CCC=CBr)C2)=O)ccccc1[N+](=O)[O-] C1(CNC(=O)C(C)(C)C=CCN)CC(CCC)CCO1 c1(C(N2CCC(NC(C3CC(OC)C3)=O)C2)=O)cccc2c1COCC2 c1(C(=O)NCC(C)N(C(CSCC(=O)OCC)=O)C)csc(CC)n1 c1(OC)ccc(C(N2CC3CC2CN3C(c2ncn(C)n2)=O)=O)nc1N N1(C(C(C)=C(C)C)=O)CCC(CNC(=O)Cc2sc(O)nc2O)C12CCC2 C(CC(F)CN=[N+]=[N-])NC(C=CC(=O)N(C1(CC(=O)O)CC1)C)(C)C C1(C(N2CC(NC(C3N4CC(C)N(CC4)C3)=O)C2)=O)CCOCC12CCC2 C1(O)(C(C(=O)NC(COC)C(=O)N2CC3CC2C3)F)CCCC1 C(=O)(CC(C)NC(C1CC(NC(c2cc(Oc3ccccc3)cs2)=O)C1)=O)OC C1(C(=O)NCC2CCN(C(CCCCCC#N)=O)C2)CC(=O)c2ccccc2C1 N(C1CS(=O)(=O)c2ccccc21)Cc1onc(-c2ccc(C(C)C)s2)n1 C1(CNC(CCc2ccc(C)cc2)=O)N(C(=O)C2=CCCC2)CCC1(C)C C=CC1COCCN1C(=O)CCN(C)C(C1CCC(=O)C1)=O C=CC(C)(C)CC(=O)N1CCCC1C(C)(C)CNC(=O)CCCC1CC1 C=C(C)CC(=O)N(CC(CC)NC(C1CCCC1)=O)C N1(C(C)C(=O)Nc2cn[nH]c2)CCCC(NC(=O)Nc2ccc(C(F)(F)F)[nH]2)C1 N1(C(CC(C)(C)NC(c2ccn(CC)n2)=O)=O)CC(C)N(C(C)=O)CC1C C1(N(C(c2ccc(C)n2C)=O)C)CN(C(=O)C(F)(F)C2CCCC2)CC1(C)C CC(C(O)C(F)F)NC(=O)C=CC1CCCN1C(c1ncccc1N)=O c1(C(=O)NC2C=CC(C(=O)Nc3ccc(COC)cc3)C2)ccc(C)cc1 C1(C2CCN(C(=O)C(C)Nc3ccc(Cl)cc3)C2)(NC(c2cc(C)ns2)=O)CC1 C1(CNC(c2ccn(COC)n2)=O)CN(C(=O)Cc2cnc[nH]2)CC12CCC2 C1(C(=O)NC(CC)(C)CNC(=O)Cn2ncnn2)CNC(=O)C(C)(C)C1 n1(CC(C(=O)NCC(C)NC(C=CC)=O)C)nnc2ccccc12 C(=O)(C1=CCc2ccccc21)NCC1(C)CN(CCCN(C)CC2CC2)CCO1 CS(=O)c1cc(C(=O)NC2CC(O)(CNC(C3CCC(=O)O3)=O)C2)cc(F)c1 C1(C(=O)NC(C2(O)CN(C(C3CC4CCCC34)=O)C2)C)(COC)CCOCC1 Cc1cc(C(N2CCC(NC(=O)C=Cc3cocn3)C2C(C)C)=O)ncc1C#N N1(C(C(C)NC(=O)NC)=O)CCC(NC(C2(C)CC3CCC2C3)=O)C(F)C1 CC(C)(CCn1cccn1)NC(=O)CCc1ncc[nH]1 CC(C(=O)NCCCCC(C)NC(C1CCC2(CCC2)O1)=O)S(C)(=O)=O CN1CCN(C(=O)C2=COCCO2)C(CNC(=O)C=Cc2cccnc2)C1 N1(CC(c2n(C)cnc2)CCl)CC(=O)N(CC2(c3cnn(C)c3)CC2)C1=O C(CCCN=c1nc2c(ncn2C(C)C)c(NCc2ccoc2)[nH]1)SC C(=O)(C1CCCc2nc[nH]c21)NCC=CCNC(C1=NOC(C)C1)=O C1(NC(=O)CCC(F)F)CCOC2(CCN(C(c3cn(C4CC4)nn3)=O)CC2)C1 C(C(C)(O)CC(=O)N1CCN(CC(=O)Nc2c(C)cccc2O)CC1)OC c1(CC(=O)NC2CC3CN(C(C(CC)CC)=O)C(C2)C3)ccc2c(c1)NC(=O)C2 N1CCCC1C=Cc1ccccc1.N1(C(c2ccccn2)C)CCOCC1 N1(C(CCC=CCC=C)=O)CC2CC2(NC(=O)CSc2ccccc2Cl)C1 C=CCCC(C(=O)NCCCCC(C)(F)F)NC(=O)CCCN=[N+]=[N-] N1(C(c2csc(C)c2C)=O)CC(C)CCC1CNC(c1ccc(C(N)=O)s1)=O CC1(C)C2CC(CN3CCCC3(C)C3CCOCC3)CC12 C1(COC)(NC(=O)C(=O)Nc2ncc[nH]2)CCCN1C(c1c(C)ncn1C)=O c1(C(N2CCC(=CCNC(C(C)SCCCC)=O)CC2)=O)coc2c1CCCC2 N1(C(CC(CC)C)=O)CCC2(CCCCC2NC(c2csc(S)n2)=O)CC1 Clc1ccccc1CNC1CCC(Nc2nccc(N3CCCC3)n2)C1 C(CC(C(=O)NCC1CCC(CCO)CC1)OC)OC.C1(C)C(=O)N1 c1(C(=O)NCC(CC)NC(=O)C(N2CCN(CC)CC2)C)cccnc1C C1(NC(=O)C=CCF)(CO)CCCCC1.C1CCCCNC(=O)C(C)NC(=O)N1 c1(C(=O)NCC(CNC(=O)C=CC(C)C)OC)c(Cl)sc(C)c1C C(C(=O)N(CC(C)(C)CNC(=O)C(C)(CO)NC(C)=O)CC)(C(C)C)OC Cc1noc(C)c1CC(N1CCC(CNC(C2(n3cc(Cl)cn3)CC2)=O)CC1)=O O=C(CC(C(F)F)n1cccn1)N1CC(N2CCN(C(=O)C#CC3CCC3)CC2)C1 c1(C(N2CCSC3CCC23)C(=O)NCc2ccccc2)cn2cc(F)ccc2n1 c1(NC(C(CCCOC)NC(C2OCCC2(C)C)=O)=O)cnc2ccnn2c1 C12(NC(C3N(C)C(=O)CC3)=O)CCOCC1CN(C(c1cc3scnc3[nH]1)=O)C2 CCCCC(=O)C(=O)N1CCC(C2CCCN2C(=O)Nc2cc(C)ccc2F)C1 CC1CN(C(c2ccoc2)=O)CCC1CNC(C1CCOC1)=O C(=O)(C(C)(C)N=[N+]=[N-])NCC(CC(=O)N(CC(F)(F)Cl)C)O c1(CC)cnc(C(=O)NC2C=CC(CC(=O)NC3CC4(CSC4)C3)C2)nc1 c1(NC(N2CCC(CC3CCCCO3)CC2)=O)cc(-c2cccc(F)c2)ccn1 C1(C(N(CC(COCC)O)C)=O)CN(C)CCN1C(c1cnc(O)c(C)c1)=O C1(C(=O)OC)CCCC(C(N2CC(NC(=O)Cn3ccnc3C)(CF)C2)=O)CC1 C1(C(=O)NC(C(=O)NC(C2CCCCC2O)C)CC2CC(CO)C2)Cc2nccn2C1 N1(C(C(CCCC)O)=O)CC2CCC1C1CN(C(c3cccc(CO)c3)=O)CC21 c1(CNC(C2CCC(CC)C2)=O)ccc(C(=O)NC2CCSC2)nc1 C(C(C(C)(C)C)NC(=O)C(C)(N(C)C)C1CC1)NC(C(c1ccc(CO)o1)C)=O N1(C(C=Cc2n(C)ncc2)=O)CCC2CN(C(=O)CCc3nccs3)CCC2C1 c1(C(=O)NCCC(C)NC(c2cccc3nonc23)=O)cc2ccncc2s1 c1(C(=O)NC(C(=O)OC)CC2CCC2)cc2ccccn2c1 N1(C(Cn2nc(C)oc2=O)=O)CCN(C(C2CCN(C)C2C)=O)CC(C)C1 N1(C(c2cc(SC)oc2)=O)C(C(=O)N(C)Cc2ccnn2C)CCC1C1CC1 N1(C(C2(OCC)CCOC2)=O)CC2(C)CC1(C(N1CC3CC3C3CC13)=O)C2 C=C(Cl)CCC(=O)NC1C(C(N2CCCC2C(C)(C)CO)=O)C1(C)C N1(C(Cc2nc(CC)sc2)=O)CCOCC1CN(C)C(C1(C)CCCOC1)=O N1(C(C2(C)ON=C(C)C2)=O)CCC(NC(=O)C2=CCCCC2C)C(CO)CC1 C(=O)(C1=CCOCC1)NCCCN(CCCNC(c1cnc(C(F)F)s1)=O)C N1(C(C(C=C)C)=O)CCN(C)C(C(N2CCC(C(C)O)CC2)=O)C1 N1(C(c2c(COC)noc2)=O)CCC(C)C1CNC(C1(OC)CCC1)=O Cn1ncc2ncc(C(=O)NCC34CCC(NC(C5CC5(Cl)Cl)=O)(CC3)CO4)cc12 C1(C(=O)NCc2c(S(=O)(=O)N(C)C)cccc2)CC(=O)NC2CCCCC12 N1(C(CN(C(C)=O)C)=O)C(C)CN(C(=O)CCC2CC3CCC2O3)CC1C c1(C(=O)NC2C(CNC(CCSC)=O)CC2)ccc(C2(F)CC2(F)F)cc1 CC1(C)C2CCC1(CC(N1CC(OCCNC(C3C4CCCOC34)=O)C1)=O)CC2 c1(CC)noc2ncc(C(=O)NC3CC4CN(Cc5sccc5Cl)CC34)cc12 CC1(C)CC2(CO1)CN(C(c1csc3ccc(Cl)cc13)C(=O)NCS)C2 Cc1ccccc1C1(NC(C2CC(c3cccc(Cl)c3)(O)C2)=O)CC1 C1(NC(c2cc(CC)nc(O)c2)=O)CN(C(=O)CCN2CCCC2)CC(C)(C)C1 C(=O)(CC(O)CC(C)(C)C)NC1CCCN(C(C2(CCCC)CCC2)=O)C1 c1(OC)ccc(Cn2nnnc2C(Cc2occc2Br)NCc2ccoc2)cc1 CC(CF)N=c1[nH]c(N2CCC(OC3CCOC3)CC2)nc2c1COCC2 CS(=O)(=O)c1cccc(Cl)c1NC(=O)CC(O)C1CCNCC1 Cc1cncc(C)c1C(=O)NC1C2CN(C(C3CCCN3C=O)=O)CC12 C1(O)(CCNC(C2(CCOC)CCC2)=O)CN(C(=O)C(C)C2CCC2)C1 N1(C(C2(C#N)C(C)C2)=O)CCN(C(=O)CC(=O)N(C)C)CC(C)(C)C1 c1(C(=O)NCC2CC(=O)N(C)S2(=O)=O)ccc2c(c1O)CCC2 c1(C(=O)NC2C(C)N(C(c3ccc(C(C)(C)C)nc3)=O)CC2)ccc(F)cc1F C1(NC(=O)C2CC2)CCCN(CC(N2CC(c3ccccc3)C(O)C2)=O)C1=O.C(=O)O c1(C(=O)NC(CCNC(CC(C=C)CC)=O)C)ccn2cc(C)nc2c1 Cn1ncc(C(N2CC(n3cc(C4(C(=O)O)CC4)nn3)C(O)C2)=O)c1C#N Cc1cccc(Cl)c1C(N1CC(NC(c2cncc(Cl)c2)=O)C(C)(C)C1)=O c1(-n2cc(NCc3ccc(C#C)cc3)nn2)ccc([N+](=O)[O-])cc1C1OCCO1 c1(COCC)nc(Cl)cc(=NC(C)CN(C)C(c2cn(CC3CCCC3)nn2)=O)[nH]1 C1(NC(CCOCCN(C)C(C2CCS(=O)CC2)=O)=O)CCCC(O)C1O C(CC(O)C(=O)NCCCc1nccs1)NC(c1occ(C)c1)=O C(N=C(NC1CCCC1)NC1CCN(C(=O)N(C)C)C1)c1c(C)ccs1 c1(C(N2CCC(C(N3CCC(CCOC)C3)=O)(CF)C2)=O)cccn(C)c1=O c1(OCC(=O)N(CC(C2CC2)OC)CC)ccc(F)c(Br)c1.C(=O)(C(C)CC(C)C)N C1(CN(c2ccc(Cl)cc2)C(CNC(CCC)=O)=O)CCCC(C)CC1 N1(CCN(C)C)CCC(N=c2[nH]c(N(C)Cc3c[nH]c(Br)c3)nc3c2COC3)C1 C(=O)(C#CC1CCOC1)N1CCC(C(CNC(Cn2c(C)nnn2)=O)(C)O)CC1 C(CC(=O)NC1(CC(N)=O)CC1)OCCN(C(CSCC#C)=O)C C1(F)(C(N2C(CNC(c3n(C)cnn3)=O)CCC2)=O)CCS(=O)(=O)C1 N1(C(c2c(C)nc(C)s2)=O)CC(C)CN(C(C2CC3C=CC2C3)=O)C(C)C1 CC1=C(CNCCC(C)C(=O)OC(C)(C)C)CCC1 c1(CCC(=O)O)ccc(Cl)c(CN2CCC(=Cc3ccccc3)CC2)c1 c1(C(=O)NCC2(OCCNC(CC(C)(F)F)=O)CCC2)cccc2c1CCN2 N1(C(C(C(CC)C)OC)=O)CCC2CN(C(c3ccc(N(C)C)nn3)=O)CC2C1 CC1(C)CCN(C(=O)CC2CCOC2=O)C1C(=O)NCC#CCCO CCCN=C(NCc1cc(C)on1)NC(C)C(c1ccc(Cl)s1)OC CC(C)CC(C(=O)NCC1CCC1CO)ONC(C1(C)CCC(=O)C1)=O c1(C(=O)NCc2cccc(CNC(C(C)=CC)=O)c2)ccc2nc(Cl)nn2c1 N1(C(c2ncc(CO)cn2)=O)CC2CC(C(N3CC(CO)C(O)C3)=O)(C2)C1 N1(C(c2c(C)non2)=O)CC2(CC(CNC(=O)CSc3ccccc3C)C2)C1 C(=O)(C(O)CC(F)(F)F)NC(c1cccc(NC(c2cc3sccc3s2)=O)c1)C C=C1CN2C(=O)CCC2(C(N2CC(N(c3ccncc3)CCO)C2)=O)C1 C(=O)(C(CC(F)F)SC)N(CC(CC)NC(c1coc(N(C)C)n1)=O)C Cc1csc(C(N2CCCC(CC(=O)Nc3cnccc3C3CC3)C2)=O)c1C c1(C(=O)NC2CCN(c3cccc(C)c3)C2=O)cc(C)c(Br)c(C)c1 N1(C(C(C)OC2CCOC2)=O)CCCCCC1CNC(C1(CC2CCC2)CC1)=O N1(C(C2(C)ON=C(C)C2)=O)CCCC2(C1)CN(C(C1OC(C)CC1C)=O)CCO2 N1(C(C2=C(CC)OCCS2)=O)CCC(C2CCN(C(=O)CN3CCOCC3)C2)C1 N1(C(c2ncc(C)cn2)=O)CCC2(CC1)CCN(C(=O)C(C)CS(C)=O)C2 C(C1=CCN(C(C2(C)CCCCC2)=O)CC1)NC(C1C(CC)CCC1)=O c1(C(=O)NCC(C)NC(c2cc(C(F)(F)F)no2)=O)cn2c(n1)SCC2 c1(C(N2CC(C)(NC(=O)CC3(C)CCS(=O)(=O)N3)C2)=O)cc(Cl)c(F)c(Cl)c1 C1(C(N(C)CC2CC2(C)C)=O)N(C(c2cnn[nH]2)=O)CCC1(C)C CC1CCn2cc(C(N3CCCC(F)(CNC(C4CC(O)C4)=O)CC3)=O)nc2C1 C#CCC(C(=O)N(C)CCN(CC)CC)NC(=O)C(C)n1ccnc1.N C1(CC(N2C3CN(C(c4n(C)ncc4)=O)C(C3)C2)=O)Cc2cccc(Cl)c2O1 C(C(=O)N(C)CCN1CCN(C(=O)CCOC)CC1)(C(C)C)OCC N1(C(C(CCC)C(C)C)=O)CCC2CCN(C(c3nn[nH]c3Cl)=O)CC12 c1(-c2cccc(C)c2)n[nH]c2c1CN(C(N1CCNC(=O)C1(C)C)=O)CC2 Cc1c(F)ccc(C(=O)NC2CCC(NC(=O)C(C)(C)CC(C)C)C2)c1C c1(NCCCN(C)C)nc(N(CC(F)Cl)C)nc2ccccc12 c1(C(N2CCC(C(=O)NC3(C(O)C(F)(F)F)CCC3)(CC)C2)=O)cn2c(n1)SCC2 Cc1ccnc2ccc(C(N3CC(O)(CCNC(=O)C4=CCOC4)C3)=O)cc12 Cc1ccc(C(N2CCN(C(=O)C3=CCC(C)C3)CC2C(C)C)=O)cc1CO Cc1cc(C2CC2)ccc1C(=O)NC1CC1NC(C1CN2CCC1CC2)=O N1(Cc2ccc(C)c(F)c2)CCCCC(NC(C2CCC=CCC2)=O)CC1 C1(C(N2CC(CNC(CC(C=C)(C)C)=O)C3C2C3)=O)Cc2cncn2C(=O)N1 CCC(CC)CC(F)C(=O)N1CC(NC(c2cncnc2)=O)CC(F)C1 c1(CC(C)C)cc(O)nc(C(=O)NCCCSCCO)n1 C1(NC(C(CCSC)O)=O)CCN(C(c2cc(N)cc(O)c2)=O)C(C)C1 C(=O)(C(C)CC1CCCCC1)NCC(C)NC(c1coc(-c2cnn(C)c2)n1)=O C1(C(=O)NC2CCCN(C(c3csc(C)c3C)=O)C2)SC2C=CC1CC2 C1(NC(CCCN(C(C(=Cc2ccco2)C)=O)C)=O)CCCN(C)C1=O Cc1cc(F)ccc1NC(=O)C(CC(C)C)ONC(c1ccc(F)s1)=O CCC(C(=O)OC)C(=O)N1CSCC1C(=O)NC1(C)CCC(C)(C)C1 C12(CNC(C3C(CC)OCC3)=O)CCCCC1N(C(c1csnc1C)=O)CC2 N1(C(CCNC(=O)CO)=O)C2CCC1C1CC1(NC(C1CC1(Cl)Cl)=O)C2 C1(CC=C)(C(=O)OCC)CCCN(C(CC2CCOCC2)C(=O)NC(C)CC)C1 C(CCCC(CO)NC(=O)C(COC)COC)NC(CC(=C)C)=O c1(C(=O)NCCCn2cnccc2=O)ccc(C(F)(F)F)c(F)c1 c1(C(=O)NCC(CN(C)C(C2CCC(F)(F)C2)=O)O)cc2cccnn2c1 CCC(C(=O)N1CCN(C)C(CNC(C2CNC(=O)CC2C)=O)C1)C(C)(C)CC C1(NC(c2cnc(C)s2)=O)CC(CNC(=O)C(C#N)C2CC2)C(O)C1 c1(OCC(=O)NC2CCN(C(C3(F)C4CCCC34)=O)CC2)ccc(F)c(F)c1 n1(CCC)cccc1C(N1CCCC1CC(=O)NC1CCOC1C1CC1)=O N1(C(CCCOC)=O)CCN(C(c2ncc(C(F)F)s2)=O)C(C(C)(C)C)C1 c1(OC)cc(C(F)(F)F)ccc1C(=O)OCCC(C)Sc1cccc(Br)c1 N1(C(C(CNC(C=CCNC(=O)OCC)=O)(C)C)=O)CC(CO)CC(C)(C)C1 CCCCCC(C)(C)C(=O)NCC1C=CC(NC(c2cc(F)ccc2Cl)=O)C1 C1(NC(C2CC3(CC(=O)N3)C2)=O)CCCC12CCN(C(C1CC(O)C1)=O)CC2 c1(CC(=O)N(c2ccc(OCC(F)F)cc2)C2CC2)cc(F)cc(Cl)c1 C(=O)(CC(C)CNC(=O)C=Cc1ccoc1)NCC1(SC)CC1 N1(C(C2CCCCC2)C(=O)OC)Cc2ccc(C(=O)OC)cc2C1 C12(NC(C3CN(C)C3)=O)CCC1CN(C(c1ccc(NCC(N)=O)cc1)=O)C2 C(=O)(C(CNC(=O)CC1OCCCO1)CC1CC1)NC(c1n[nH]c(CO)n1)C C1(CC)CCCCN1C(C1CCCC1OC)=O C1(NC(c2cc(OC)no2)=O)CN(C(=O)CCC2CCCCN2C)C2(CCC2)C1 c1(CNC(C(C)N2CCC2)=O)cc(O)nc(CNC(c2cccc[n+]2[O-])=O)n1 CCC(O)(C(=O)NCC1(C)CCN(C(=O)Cc2cc(Cl)cs2)C1)c1ccccc1 CCCCC(CN1CC(CC(C)N(C(=O)CC2CCOC2)CC)C1)CC C1(N(C(c2occ(C)c2)=O)C)CCC(NC(C2CC2c2ccsc2)=O)CC1 C(=O)(CC(C)(C)C)NC(C)C(=O)NC1(c2cn(Cc3ccccc3)nn2)CC1 c1(SC)ccc(C(N2CCN(C(C3CCCOC3)=O)C(C(C)C)C2)=O)c(Cl)c1 C(=O)(C(O)CCC(C)C)N1C(C(=O)N(CCN(C(CC)C)C)CC)CC(OC)C1 c1(OC)cnc(N(C2CNCC2C#N)Cc2csc(Br)n2)nc1C C1(C)(COC)CC(NC(=O)CCSC2CC2)CN1C(c1c[nH]cc(Cl)c1=O)=O C12(CCC1)C(=O)N2.n1(C2(C(C)NC(=O)CC3(C)CC3)CC2)ccnc1.C(N)=O Cc1c(Br)ccc(C(=O)NCCCNc2cccc(F)c2)c1F O=S(=O)(c1ccc2[nH]c(=NC(CF)c3ccc(Cl)cc3)sc2c1)NCCF O=C(C(O)CC(F)F)NCC1(F)CCCN(C(C2(C(N)=O)CC2)=O)C1 Cc1ccc(C(=O)NCC(=O)NCC(C(C)C)NC(=O)COCCF)c(C)c1 C12(NC(c3cccc(N)n3)=O)CCC(CC1)N(C(C1CCC3CC1CO3)=O)C2 N1(Cc2c(C(=O)O)c3c(s2)cccc3)CC2CS(=O)(=O)CC(C1)C2(F)F S(=O)(=O)(c1c[nH]c2ncncc12)NCC.C12(COC(C)(C)C1)C(=O)O2 c1(C(N2CC(O)(CN(C(C(CC#C)CC#C)=O)C)C2)=O)n[nH]c2ccc(F)cc12 c1(-c2cn(C3CCN(C(C4CCS(=O)(=O)C4)=O)C3)nn2)ccc(F)nc1 C1(NC(c2n[nH]cc2Cl)=O)CN(C(c2cnn3c2CCC3)=O)CC12CCOCC2 CCCCC(CC(=O)NCc1nccn1C)NC(C1CC1(Cl)Cl)=O c1(COC)nc(C(=O)NC2(CO)CN(C(=O)CNc3ccccn3)C2)co1 CC1(CNC(C2CCC(OC(F)F)CC2)=O)CCCN(C(c2c[nH]c(=N)s2)=O)C1 c1(C(=O)NC(CNC(CCCC#C)=O)CC(C)C)c(OC)cc(OC)cc1N Cc1ncc(C(=O)NC2(C3CCCN3c3nc(C(C)C)ns3)CC2)cn1 N=C1NC(=O)C(CC(N2CCN(C3CCCN(C(=O)CC4CC4)C3)CC2)=O)S1 CC1CN2CCC1C2=O.c1(C(N(C2CC(N(C)C)C2)C)=O)cscc1C#N S(=O)(=O)(c1ccc(Cl)c2nonc12)NC1C(C)CN(C(C2(C(N)=O)CC2)=O)C1 C1(C(N(C2(O)CCC2)C(C)C)=O)CCC2CCC1N2C(=O)C(C)CC(N)=O c1(C(=O)NC2CC(NC(C(CC)(F)F)=O)C(O)C2)ccc2cc(C#N)ccc2c1 N1(C(C2CN(C(C)C)C2)=O)CC2CCC2C1.C(Cn1cccn1)(C(=O)NCC)OC N1(C(CCC)=O)CCC2(CCCC2NC(=O)Cc2ccc3c(c2)CCC3)CC1 c1(OCC)cc(OC)c(Cl)cc1C(=O)N(C1CCC=CO1)CC.C(C(C)C)O CC(C)C(C(=O)NC1CCCC1CNC(=O)CCOC(F)(F)F)c1cccnc1 C1(CNC(=O)Cc2ncccc2Br)CCC2(CCC2)CN1C(=O)C=CCF C(=O)(CC(C(F)F)n1ccnc1)NCc1c(CNC(CNC(C)=O)=O)nccc1 Cn1ccc(=O)c(C(=O)NCCCOCCNC(=O)OC(C)(C)C)c1 C1(C(=O)NCC(C)N(C(C(C=CCCC)O)=O)C)CCc2nc(O)[nH]c2C1 C1(C(=O)NC2CCN(C(c3cc(Cl)ns3)=O)CC2C)(OC)CCC(C)(C)CC1 N1(CC(N2CCCCC2c2cc[nH]n2)=O)CCN(Cc2ccc(F)cc2)CC1=O N1(C(=O)CCN2CCCCC2)CC2=C(C1)CN(C(C13CCOC1CCOC3)=O)C2 C1(CC)C(C)CCN1C(C1CCCN(CC2CNCCC2C)C1)=O c1(CN2CC(C(=O)NCc3cccc(C)n3)SCC2)cnc(C)c(Br)c1 c1(CC)cc(Cl)ccc1C(N1CCCC1CNC(C1CSC1)=O)=O C1(C)(OC)CC2CC1CC2NS(=O)(=O)CC1CC2(C1)N=N2 N1(C(C2(NC(=O)CN3CC(C)(C)C3)C(C)CCC2)=O)CCCNC(=O)CC1 C1(CN)CCN(C(C2(OC)CC(C)(C)C2)=O)CCO1.C1(C(=O)OC)C(CO)C1(C)C Cc1csc2nc(CC(=O)NCC3(O)CC(CNC(C4CCC5CC45)=O)C3)cn12 c1(NC2C(C)CS(=O)(=O)C2)nc2c(c(=NCC3Cc4ccccc43)[nH]1)CCC2 C1(CNC(CNC(C)=O)=O)CN(C(=O)COc2cncc(Cl)n2)C2CCCC2O1 N1(c2nc(C)cc(OC)n2)CC(NC(=O)CC(C)(O)C2CC2)CC2(CCC2)C1 c1(C2C(CNC3(c4n(CCSC)nnn4)CC(C(C)C)C3)C2)ccc(C)cc1 Cc1cc(C)c(CN2CCC(n3cc(CNC(C4CCCO4)=O)nn3)C2)s1 C(=O)(CC1=CCCCC1)NC(C(=O)N(C1CCOCC1)CC)c1cccs1 N1(CC)CCOCC1C(=O)NCCCN(C(=O)C(n1ccnc1C)C)C1CC1 C1(C(=O)NCC2CC(OC)C2)C(C2CC2)CCN1C(c1ccoc1)=O c1(C(=O)NCC2CCCC(NC(C3(C)ON=C(C)C3)=O)C2)cccc(N)c1O C1(CN(C)C)(NC(C2CCC(NC(C3CCSC3)=O)C2)=O)CCCC1 CC(C)CCC(O)C(=O)N1CCC2(CC2)CC1C(=O)NCC=C(Cl)Cl c1(C(=O)OC)cc(N2CCC(CNC(C3CCOC3)=O)C2(C)C)nc(Cl)n1 c1(NCC2(C)COC2)cn(CC(c2cnn(Cc3ccccc3)c2)=O)nn1 c1(NC(CC2(CNC(C(CN(C)C)N(C)C)=O)CC2)=O)c(F)cccc1F Cc1cc(C(N2CC(F)(C(=O)Nc3cccc(Oc4nccs4)c3)C2)=O)cnc1O c1(C(=O)NCCOCCN(C(C2C(OC)C2)=O)C)cnn2cc(C)cnc12 C#CCCCC(C)(c1nnnn1C)NC1(C)CN(C(C)=O)CCO1 C1(COC(C)C(=O)NC2CC(CNC(C3CC3)=O)C2)COCCN1C c1(SC)nc(C)c(CCC(N2CC(NC(=O)COC3CCOC3)CC2C)=O)c(O)n1 Cc1nnccc1C(=O)NC(C(=O)NCC(C1CC1)N(C)C)c1ccoc1 C1(C(N(CC=C)CCC)=O)CCCN(C(=O)CS(=O)CC)C1C c1(C(N2C(C)(CNC(C(CCC)OC)=O)CCC2)=O)sc2ccc(Cl)cc2c1C c1(CN2CCC(NC(CCCn3c(C)ncc3)=O)CC2)cc([N+](=O)[O-])ccc1O c1(C(=O)NCC(C)CNC(C2(n3ccnn3)CC2)=O)cnc(N)c(CN(C)C)c1 N#Cc1cccc(C=CC(=O)NC2(CNC(=O)Cc3ccc(Br)nc3)CC2)c1 C=C(Cl)C(C)(C)C(=O)N1CCC(NC(C2(CCN(C)C)CCCC2)=O)C(F)C1 C=CCC(C)(C)CC(=O)NC1CS(=O)(=O)CC1NC(c1ccnc(C)c1C)=O c1(C(=O)NC(C)CN(C(=O)COC(F)F)C)ccnc(N2CCCC2)c1 c1(C(N2C(CNC(C(CC)OC)=O)CC2)=O)cc(-c2ccccc2)cnc1C CC(C)C1CCC(=O)N2CCCC(CC2)CC(CCC)C=CC(=O)N1 c1(C(=O)NCC(CCOC)NC(c2[nH]c(C3CC3)nc2C)=O)ccc(C)nn1 C(CC(=O)N1CCOC2CCCC12)(C(F)(F)F)NC(c1ncn(C)c(=O)c1)=O N(C(=NCC(C)c1ccc(F)cc1)NCN1CCCCCC1C(C)C)CC(C)C c1(N(C)C(c2cc(NC(=O)COC3CCCOC3)c(Cl)s2)=O)cccc(Cl)c1Cl O=C1CCC(C(=O)NC2COCCC2NC(=O)CCN2CCC(F)C2)=NN1 CC(c1cccc(C)c1)=CC(N1CCC1CNC(c1cn(C2CCC2O)nn1)=O)=O N1(CC(c2c(OC)cccc2)OC)CC(=O)N(CC2(C3CCCCO3)CC2)C1=O c1(OC)cc(C(=O)NC2(C)CN(C(c3c[nH]c(C#N)c3)=O)C2)cnc1O C=CCCCC(=O)NC(C)CCCNC(C1(CC(F)F)CC1)=O c1(CC)cccc(F)c1C(N1CCC(CO)C(NC(=O)CSC(F)F)C1)=O Cc1ccc(N)c(C)c1C(=O)NCC(F)CNC(=O)C(C)C(C)(F)F CC1=C(C)CC(C(=O)N(C2CCCCN(C(=O)COC3CC3)C2)C)CC1 c1(C2C(=O)N(C)CC2C)cc(F)cc(F)c1.c1(C(N2CCC2)=O)ccccc1F c1(C(=O)O)cc(C(=O)O)cc(C(N2CCC(OCCC)CC2)=O)c1.C(C)(C)O N1(C(C(C(C)C)NC(C)=O)=O)CC2CC(C1)N(C(=O)C(C)(C)OC(C)C)C2 CC(CC(F)F)C(=O)N1CCC(NC(=O)COc2ccccc2C(F)(F)F)C1C N1(C(CCC=CCC=C)=O)CC(NC(c2conc2C2CCCC2)=O)C(C)(C)C1 C1(NC(C2CCCC(C)(C)C2)=O)CCN(C(=O)CCc2ccsc2)CC12CCC2 CCC(CC)(CO)C(=O)N1CC2CC(C(=O)NOCCC(F)F)(C2)C1 N1(C(c2c(C(=O)OC)c[nH]n2)=O)CC2CCN(C(=O)C(CC)N(C)C)CCC2C1 c1(OC(C)(C)CNC(=O)C(F)C(F)(F)F)c(F)cccc1F.C1C(=O)N1 c12cnc(cn1)NC1CCN(C1)C2=O.c1(C=O)cnn(C(C)(C)C)c1Br.CO C1(CCOC)(C(N2CC(C)C(F)(F)C2)=O)CCN(C(c2c[nH]nc2OC)=O)CC1 c1(C(N2CCC(CC(=O)NC(C)C(F)(F)F)C2)=O)cc(Cl)nc(Cl)c1F c1(CC)[nH]nc(C(N2CCC(F)(CNC(=O)CCCC3CC3)C2)=O)c1Br C(N=c1nc2sccc2c(N2CCCCC(C)(F)C2)[nH]1)c1nn(C)c(Br)n1 C1(NC(=O)COC2(CC(F)(F)F)CC2)CN(C(c2cccs2)=O)CC1C(F)(F)F C(=O)(C(C(C)(C)C)NC(=O)CC(C1CC1)C1CC1)NCC1(CO)C(C=C)C1 N1(C(CC2(OC)CCC2)=O)CCCC(CCNC(C2CCC3(CC3)C2)=O)CC1 C1(CNC(CCC(C)CN(C)C)=O)CCCC1P(C)(C)=O CC1CN(C(C2C3CC4C(C3)C24)=O)CC2(CCN(c3nccnc3F)C2)O1 C1(CC)CN(C(=O)C(C)CC(=O)OC)CCN1C(c1cccc(C)c1F)=O c1(CCC(=O)NCCC(=C)CNC(c2ccnc(SC)c2)=O)ccc(F)nc1 N1(C(CNC(C(C)(C)C)=O)=O)CCC2(CCC(NC(=O)C(C)(C)S(C)(=O)=O)C2)C1 C=CCCC(O)CNC(C1CC1C(C)NC(c1c[nH]nc1C(C)C)=O)=O C1(CNC(C(F)OC)=O)COCCN(C(=O)Cc2cncnc2)C1 CC1(C)CCN(C(=O)C(F)OC(F)(F)F)C1CC(N1CCCC(O)(C(N)=O)C1)=O CC(C)C(CNC(=O)CN1CCCC1C)C(=O)NCCC=C1CCOCC1 c1(C(C)C)nn(C)c2c1CCN(CC1CCNC3CC13)C2 C1(N(C(C(C)OCCC=C)=O)C)CN(C(=O)Cc2c(C)noc2Cl)CC1(C)C C12(C(N(CCC)CC)=O)CC(CN1C(=O)C(C)(C)COC)C2 CC12CC(C(=O)NC3CCC(NC(C4CCCCC4)=O)CC3)C(CO1)C2 c1(C(N2C(CN(C(C3(C)C=CCC3)=O)C3CC3)CCC2)=O)ccc([N+](=O)[O-])cc1 c1(C(N2CC(CCCCNC(CCCOCCC)=O)C2)=O)c(C)cccc1Cl N1(C(c2ccc(OC)s2)=O)CCCN(C(c2cnn(CC3CCC3)c2)=O)CC1C Cc1cnc2n1CCCC2C(=O)N(C)CC1(O)CCN(C(=O)CSC2CC2)C1 CC(CC(C)C(F)F)NC(C1CCCCCN1C(c1ccc(=N)[nH]c1)=O)=O c1(CC)c(C(=O)NC2(CC(F)F)CCN(C(=O)CO)CC2)oc2ccccc12 c1(C(C)=O)c(C)[nH]c(C(=O)NC2CCN(C(c3ncc(F)c(OC)n3)=O)C2)c1C C1(CC(N2CCC(C(C)(C)NC(c3cnsn3)=O)C2)=O)(COC)CCCC1 N1(C(C=COCC)=O)CCC2CC1CN(C(c1sccc1OC)=O)C2 CP(C)(=O)CCC(=O)N1CCC(C(=O)Nc2ccc(C3CC3)nc2)C1 Cn1c(=O)[nH]c(C(=O)CNCC2CCC(OC(F)F)CC2)cc1=O C1(C(=O)NCc2ccc(CNC(C(C)NC(C)=O)=O)cc2)CC(=O)N(OC)C1 c1(C(=O)NCCc2nnc(C)n2C)ccc2c(c1)c(C#N)cn2C C1(CNC(c2csc(C3CCNCC3)n2)=O)(NC(C2CCCO2)=O)CCOCC1 C1(CC)(CC)CC(NC(=O)C#CC(C)(C)C)CN1C(=O)CN(C)C N1(CC(=O)NC2COCC2C(=O)NCc2ccco2)CCCCC1=O C(CC(CC)C(=O)NCC1(C)CCCN(C(=O)Cc2cncnc2)C1)=CC Nc1ccc(N)c(C(N2CC(F)(CNC(c3csc(-c4cn[nH]c4)n3)=O)C2)=O)c1 Cc1noc(N)c1C(=O)N(C1CCN(C(C2CC3CC2C3)=O)CC1)C C(CC1CCCC1)(C(=O)Nc1cc[nH]c1)NC(COCCOC)=O N1(C2(OC)COC(OC)C2)CCNC(=O)CC1C(F)F Cc1cccc(C(C)NC(C2CCCN(Cc3ccc(C(F)(F)F)cc3)C2)=O)c1 N1(C(c2cc(C3(C)CC3)n[nH]2)=O)CC2(CCC(CNC(=O)C(O)C3CC3)CC2)C1 N1(C(C(C)OC)=O)CCN(C(=O)C(F)(F)CCn2ccnn2)CCC1C Cc1nc(C(=O)NCC(C(C)C)NC(C2CC2c2ccccc2)=O)c(C(F)(F)F)s1 c1(NCC(C)N=c2cncc[nH]2)cc(Br)ccc1S(=O)(=O)NCc1ccco1 c1(C(=O)NCC2(C)CCCN(C(=O)CC3C=CCC3)C2)cc(C#N)ccc1O N1(C(C2(c3ccc(F)cc3)CC2)=O)CCN(CC2CCCCO2)CC12CCC2 c1(CNC(C(CN(C(c2n(CC)ccc2)=O)C)C)=O)ccc(C)nc1 c1(C(N2CCC(NC(C3CN4CCC3CC4)=O)C(F)C2)=O)ccc2nn[nH]c2c1 C1(CC(=O)NCC2N(C(COC)=O)CC2)SC(=N)NC1=O CC1(CCNC(C2CC(O)CC2O)=O)CCN(C(=O)COCCF)C1 c1(OC)cc(C)ccc1-c1cn(CCNC(c2ccc(-n3cccn3)cn2)=O)nn1 C1(CNC(C(C)Nc2scc(C)n2)=O)CCCN(C(C2(CC(C)C)CCC2)=O)C1 C1(NC(c2c(NCC)cncc2)=O)CCN(C(c2cc(O)ccc2F)=O)CC1C c1(CC)ccc(C(=O)NC(C)C(CO)NC(C2(C(F)F)CCC2)=O)c(C)n1 c1(CCNC(c2n(CCOC)nnn2)C2CCC(C)C2)cn2cccc(F)c2n1 C#CCC(C(=O)NCC#CC1CC1)NC(c1csc(CC)n1)=O Cc1nc2c(o1)CCN(C(C1CC(C)N1C(c1noc(C)c1C)=O)=O)C2 C12(CC3CCCC13)NC(C)C(=O)N2.CCC(C)(C)OCOC.C12CC1C(=O)N2 c1(C(=O)NC2(CCNC(C(C)c3ccsn3)=O)CCC2)ccc(N)c(F)c1F N1(C(Cc2c(C)cco2)=O)CCC2(C1)CN(C(C1CCCC1C1CC1)=O)CCO2 c1(C(=O)NCCOC2CN(C(C(C(C)C)SC)=O)C2)nn(C)c2ccc(F)cc12 CCC(C)(C(=O)NC(c1nc(C(N2CCC2CF)=O)co1)C)OC C1(NC(c2cc(-c3cn(C)nc3)no2)=O)CCN(C(C2(C)CC=CC2)=O)CC1O C1(NC(C(N2CCOCC2)C)=O)CC2CC(C1)N(C(C1CC1C)=O)C2 C(=O)(C(C)CC(C)(C)C)NC(CCCC)C(N1CC2(CCC2)CC1C)=O c1(COC)nc(CC2CCCCC2)n(-c2ccccc2F)n1 C1(O)(CCNC(CCC)=O)CCN(C(C2(C(=O)OCC)CC=CCC2)=O)C1 C1(C)(CCNC(C(C)Cc2ccncc2)=O)CCN(C(c2cncnc2)=O)C1 S(=O)(=O)(c1cccc(C2OCCO2)c1)N1CCC(N2CC(C)C3(C2)CNCC3)C1 N1(c2c(F)cnc(C)n2)CC2CCC(NC(c3cccnc3C(F)F)=O)CC2C1 N1(C(COCC(=C)C)=O)CC2CC2(CNC(=O)CC2CCCOCC2)C1 N1(C(C2CCC(=C)CC2)=O)CC(NC(=O)CCn2cccn2)CC12CCOCC2 C1(NC(C2(CCOC)CCN(C(=O)C(F)F)CC2)=O)CC2CCCCCC12 c1(-n2cc(CNC(C(C3CN(C(C)=O)C3)OC)=O)nn2)ccc(C)cc1F Cc1ccc(CNC2CCCC(NC(=O)CN3CCOCC3)C2)nc1Br C1(CC(=O)NCCN2C(C)CCC2)CCN(C(c2sccc2F)=O)C1(C)C CC(C)CC(CNC(C1(C)CCC(=O)N1)=O)NC(=O)CCSCc1ccccn1 Cc1ccc(C=CC(=O)NC(C)C(C)NC(c2ccc(Br)s2)=O)cc1C C(C1CCOCC1)=CC(=O)N(C)CC1CCCN1C(C1CCC1(F)F)=O c1(CC(=O)NCCC2(O)CN(C(C(C)N(C)C)=O)C2)ccc(Br)c(Cl)c1 C(CCCCn1cc(-c2ccn(CC(F)F)n2)nn1)SC.C1(C(C)C)CC(C=O)C1 c1(CC(C)CN2CC(O)C(F)C2)ccc(F)cc1.N12CCC(CC1)C2=O N1(C(C(C2CC(F)(F)C2)OC)=O)CCOCC(CNC(C2(OC)CCC2)=O)C1 C12(CN(C(C3CCC=CO3)=O)C1)C(=O)NC2.c1(CC2CC2)ncccn1 c1(C(=O)NC(C(C)NC(=O)CCc2cccnc2)CO)cc(Cl)ccc1O N1(C(c2c(C)ccs2)=O)CCCC(CCCCNC(C2OCC2(C)C)=O)C1 N1(C(C(C)N2CCC2)=O)CC2CCN(C(C3CCOC3c3ccncc3)=O)CC12 c1(C(=O)NCCC(C)N(C)C(C2C(F)(F)C23CC3)=O)cc2occc2s1 C1(COC)CC(CNC(c2csc(CO)n2)=O)N(C(=O)C(C)C)C1 c1(CN(CC(C)NC(=O)OC(C)(C)C)C2CC2)ccc(-n2cccn2)nc1 c1(C(=O)NCCNC(C(C)Cn2ccnc2)=O)cccc2sncc12.C12CC1C2 c1(C(=O)NCc2scc(CNC(C(CC)C)=O)n2)n[nH]c(C)c1O C(CCCC(C)NC(C1(F)CCCCC1)=O)NC(c1c(C)scc1)=O O=C(C1=C(Cl)CCCC1)NCC=CC(N1CCOC(CF)C1)=O c1(C(N2CC(CNC(C(C3(O)CCCCC3)CC)=O)C(C)C2)=O)ccn(O)c(=O)c1 C=C=C(C)CC(=O)OCCC.C12CCCCC1N(C)C(=O)N2 C#Cc1ccnc(C(=O)NC2CN(C(=O)CNS(=O)(=O)N(C)C)C(C)(C)C2)c1 C1(NC(c2[nH]cc(C#N)c2)=O)CCC2CCN(C(c3ccc4nc[nH]c4n3)=O)C12 C(CN=c1[nH]c(=NCCCCS(C)=O)[nH]c2c1SCC2)C1(OCC)CCC1 c1(N2CC(COC)OC(C)(C)C2)nc(C)cc(=NC(C)c2ccc(Cl)c(F)c2)[nH]1 C1(C(=O)OC(C)(C)C)CC(C(=O)NCCCn2nccn2)C1(C)C N1(C(C(=O)NC(c2ccncc2Cl)C)=O)CCC(C)C(N)C1 c1(C(N2CCC(F)(CNC(c3n(C)ccn3)=O)CC2)=O)ccc2ncncc2c1 c1(N(C2CCCN(C(C3(C)CC(=C)C3)=O)C2)CCO)nc(OC)c(F)c(C)n1 C1(C(=O)NC(CNC(C2(N3CCOCC3)CC2)=O)CC)CCC(C)O1.C=CCCN N1(C(C(C)OC)=O)CCCN(CCNC(=O)CCc2csnn2)CC1 c1(C(=O)NC2C3(CC(NC(c4cc(OC)no4)=O)C3)CC2)ccn2cccc2c1 C1(C(=O)NC(C(=O)N(C)CCn2ccnn2)Cn2cncn2)CC2CCC1C2 C12(NC(=O)Cc3cncc(F)c3)CCC(CC1)N(C(=O)C=Cc1cocn1)C2 N1(C(CCN(C2CCCCC2)C)=O)CC(CNC(C2CC3(CCC3)C2)=O)C(O)C1 C(N=c1[nH]nc(C(N)=O)s1)C1(C)CCCN1C(C1CCC2CC12)=O c1(OC)cc(C(N2CC(C)(CC(=O)Nc3cc(F)cc(F)c3)C2)=O)ccc1I CCC(CC)C(C)C(=O)NC1CC(C)(NC(=O)CC23CCC(CC2)OC3)C1 C1(C)(C(=O)NC)CCN(C(=O)N(C)CCF)CC1 C1(N(C(CNC(CCC)=O)=O)C)CCCC(NC(=O)Cc2nnc(S)s2)C1 C1(CN(C)C)(NC(=O)C(C2CC2)N(C(=O)C=C2CCOCC2)C)CCCC1 C(=O)(C(CC(C)C)C(C)C)N1CC=C(CNC(Cc2cc(C)sc2)=O)C1 C(=O)(CC(C(F)F)NC(C1CNC(=O)O1)=O)N(C1CCCC1)CC c1(C(=O)NC2CN(C(Cc3c(C)n[nH]c3)=O)CC2O)ccc2ccc(Cl)cc2n1 CC1CCCC(NC(=O)C(N2CC3(C(=O)O)CC2C3)=O)CC1.C1CCO1 c1(CC)ccc(F)cc1C(N1CCNCC1C(=O)NC)C(=O)NC1CCC1 c1(CCC(=O)NC2CN(C(C(C=C=C)C)=O)CC2C)c(C)nc(O)nc1C C12(CCCCC1C)C(=O)N2.C(CC(=O)NC)OC.S(C)(=O)(=O)N(CCN)C CCCC(C(=O)NC(Cc1ccco1)C(=O)NCc1cocn1)NC(C)=O N1(C(c2cn(CC)nc2)=O)CCC(C(=O)NCCn2cc(CO)cn2)C1C c1(C(=O)NCCN2CCN(C(C3(C4CCC4)CC3)=O)CC2)cc2c[nH]cnc-2n1 N1(C(c2c(C(C)C)nns2)=O)CCC2CN(C(C3CCSC3)=O)CC12 N1(CCOC)C2CCC1CN(c1nnc(-c3n[nH]c(C)n3)n1Cc1cccs1)C2 c1(SCC(=O)NC(CN(C(C2CC(C)(F)C2)=O)CC)C)nn(C)c(=O)n(C)c1=O N1(C(c2nnn3c2CCC3)=O)CC2CCN(C(=O)C(C3CCCCC3)F)CC2C1 c1(C(=O)NC2C(CNC(c3cn(CCC)nn3)=O)CC2)cncc2ccccc12 C1(NC(C(C)(C)C2CCOC2)=O)CCCCCC1NC(C1CS(=O)(=O)C1)=O C(=O)(C1=CCCOCC1)NC(C(C)NC(c1cc(C(F)F)ccc1F)=O)(C)C Cc1nc2sccn2c1C(=O)NC1CC12CCN(C(C1CC1C1CC1C)=O)CC2 CCC(CC)(CO)C(=O)NCCC1CCCN(C(=O)C(F)C2CCOC2)C1 C1(C(=O)NCC(C2CCC2)NC(c2ccc(C(F)(F)F)o2)=O)CC2CCC1C2 c1(C(N2CCC(CCNC(c3nc(C4CC4)cs3)=O)C2)=O)ccc(O)cc1 C1(C(N(C)Cc2ccc(O)nc2)=O)CC2(C1)CN(S(=O)(=O)Cc1ccccc1)C2 Cc1ccc([N+](=O)[O-])c(-n2cc(C(=O)NC(c3ccccc3)CO)nn2)c1 N1(C(C=CC)=O)CCCC2CN(c3ncc(C#N)cc3Cl)CCC12 N1(C(c2cc3cccnc3o2)=O)CCC2CCN(Cc3ccccc3)CC12 C(C(F)(F)C(F)(F)F)n1c(-c2csc(CO)n2)nc(C(CC)C)n1 C#Cc1ccc(C(=O)NC2CN(C(c3ccc(SC)s3)=O)CCC2C)nc1 C1(NC(N(C)Cc2ccc(C(=O)NC)s2)=O)CCOC(C)(CC(C)C)C1 N1(C(CC2C(=O)NC(=N)S2)=O)CC2CC1CN2C(=O)CCc1cncnc1 C1(CN(C(C=C(CCC)C)=O)C)CCCC(NC(=O)CSc2nc[nH]n2)C1 c1(C(=O)NC2CC(NC(CN(CCOC)C)=O)C2)cccc2[nH]nc(O)c12 C1(N(C(CC2(N(C)C)COC2)=O)CCO)CCCN(C(C2CCNC2=O)=O)CC1 CC#CCCCC(=O)NCC1(OC)CCN(C(=O)CCCCN2CCCC2)C1 N1(C(C2CC(C)CN(C(=O)C3=CC(C)(C)C3)C2)=O)C2CCCC1COC2 C1(NC(C(C(CC)C)OC)=O)CN(C(c2cccc(C(F)F)c2)=O)CC1N=[N+]=[N-] N1(C(N(C)Cc2ccccc2)=O)CCC2CCNC(=O)C2C1 c1(CC)ccc(F)c(C(N2CCC(C(F)F)(CNC(=O)CCCN=[N+]=[N-])C2)=O)c1 Cc1ccc(C(=O)OCCCC2(F)CCC2)c(N(C)C)n1 C1(CNC(c2c(C)ccn2C)=O)C(O)C(O)CN1C(c1cnc(CC(C)C)s1)=O c1(C(N(CCCNC(=O)C(C)CC2CC2)CC)=O)nc2ccccc2nc1C O=C(CCCC1CCCO1)NCCCNC(=O)Cc1ccccc1 C12(CNC(C3CCC3)=O)CCC(C1)N(C(=O)Cn1ncc(Br)n1)C2 C1(C2CCOCC2)(C(N2C(CN(C(C(C)C3CCC3)=O)C)CCC2)=O)CC1 N1(C(CCOC)=O)CC(C)N(C(C2CCCC(C)C2)=O)CC1C N1(C(C(C2CCC2)OC)=O)CC2(NC(c3cc(N)c(N)cc3F)=O)CCC1CC2 CC(CC(=O)NC1CC(O)(CNC(c2cc(C(N)=O)co2)=O)C1)n1cccn1 C1(NC(CC2N(C(C)=O)CCC2)=O)C2CC3C(C2NC(=O)CC(C)F)C13 CCC(COC)C(=O)NCCCC(=O)NC(c1cnn[nH]1)C O=NN1CCCCC1C(=O)N(C1CC1)CC1CCCN(C(C2(CCF)CC2)=O)C1 N1(C(C(C)OCC2CC2)=O)CC2CC1C2NC(=O)CCC(C)OCC(F)(F)F c1(C(=O)NC(C(C)(C)C)CNC(c2cccc(O)n2)=O)cc2sccc2n1C c1(C(C)C(=O)NCCOC2(C)CC2)ccccc1S(N)(=O)=O C1(CC=C)(NC(c2cn(C)cc2C)=O)CCN(C(c2cccc(N(C)C)c2)=O)C1 C1(OC)CCN(C(=O)CSCCNC(c2ccnc(SC)c2)=O)CC1C C1(C(=O)NC(C=CC(NOCC(=O)OCC)=O)(C)C)CCC2(CC2)C1 N1(C(CCN(CC(F)(F)F)C)=O)CCC(CO)(NC(c2cnc(Cl)[nH]2)=O)C1 c1(C(=O)NC(CNC(C2(C)CC2)=O)C2CC2)cccc(OC2CC2)c1 CC1CCc2ncc(C(=O)NC3CC3CNC(=O)CCc3csc(=N)[nH]3)n2C1 c1(C(=O)NC2C(C)COC2)coc2c1CN(C(=O)COCCF)C2 c1(C(N2C3CN(C(c4c(CC)nns4)=O)C(C3)C2)=O)nnc2ccccc2n1 C1(C)(NC(CN(CCC)C(c2ccncc2N)=O)=O)CC2CCC1C2 n1(CC(=O)N(C)CC2N(C(C3C(C)=C3)=O)CCC2)ccc2c(N)cccc12 Cc1ncc(Br)c(C(=O)NCCCN2CCN(C(C3CCC(=O)NC3)=O)CC2)n1 C1(NC(c2c(C)nccc2)=O)CC(N(C)C)C12CCC2 c1(CN(CCSC)C(c2ccccc2)C)c(Cl)cc(Cl)nc1C c1(NC(C2N(C(CN(c3ccccc3)C)=O)CC2)=O)ccc(-c2ccccc2)nn1 C(=O)(CCCC(=O)N(C(C)(C(=O)NC1CN(C)NC1=O)C1CC1)C)OCC c1(C(=O)OCC)cc(NCCCSc2ncc[nH]2)cc(Br)c1[N+](=O)[O-] c1(SC)cc(C(N2CC(C(C)NC(c3ccccc3C(F)(F)F)=O)C2)=O)c(C)o1 CCCC(C)(CC)C(=O)NCCN(C(=O)Cc1c[nH]c(=N)nc1O)C N1(C(C2N(CC)CC2)=O)CC(OC)C(NC(c2sc(CN(C)C)nc2C)=O)C1 C1(NC(CC2(OCC)CC2)=O)CC(c2ccccc2)(NC(=O)Cc2cc[nH]c2)C1 c1(C(N2CC(OC)C(NC(=O)C(F)C3CCC3)C2)=O)nnn2c1CCCC2 c1(C(=O)NC(CNC(c2cnc(OCC)s2)=O)C2CC2)cc(O)n(C)n1 C(=O)(C(F)C(C)C)OC(c1nnc(CO)s1)CCC C(C(=O)N(C)CCN(C(=O)C(C)OCC1CCCO1)C)(SC)SC C1(NC(C(CC#C)(C)C)=O)CN(C(=O)C2=C(C)OCCS2)C2(CCCCC2)C1 C1(C)(NC(c2nccc(CC)c2)=O)CCCCC1C(=O)Nc1cnn(CCOC)c1 N1(C(C(C(C)(C)O)F)=O)CCC2CN(C(C3CC3c3ccccc3)=O)CC2C1 N1(C(CNC(=O)OC)=O)CC2(C)CN(Cc3cccn3C(F)(F)F)CC2(C)C1 c1(C(=O)NC(C)CNC(=O)C=Cc2ccco2)cc(Cl)c2n[nH]cc2c1 c1(C(=O)NC2(C)CN(C(c3cc(OC)cc(OC)c3)=O)C2)cc2sc(F)cc2[nH]1 CC(CC(=O)NC(C1CCN(C(C2CC(O)CN2C(N)=O)=O)CC1)C)P(C)(C)=O CCC(CC(C)C)C(=O)N1CCC(C2CCCN2C(C2(CO)CCCC2)=O)CC1 C12(CNC(CSCCC)=O)CCCCC1N(C(=O)C(C)CCOCC)CCC2 Cn1cnc(C=CC(N2CCCC2CC2C(C)(C)C2(C)C)=O)c1 c1(CNC(C2CCCN(C(=O)Cc3cccs3)CC2)=O)cccc2occc12 C12(CC(=O)NC(CNC(CCn3ncc(C)c3)=O)(C)C3CC3)CCC(CC1)C2 Cc1nn(CC(C)C)c(C)c1CN1CCN(C(=O)NC(C)(C)C)CC1C(F)(F)F c1(C(N2C(C(C)(C)NC(CCCC)=O)CCC2)=O)cc([N+](=O)[O-])ccc1Cl CC1CC(C(=O)N2CCC(OCC(=O)NCCCC(F)F)C2)=NO1 CCCC(C)(O)CC(=O)N1CCOC(CCNC(c2occc2COC)=O)C1 c1(C(=O)NC(C)C(=O)NCC(c2ccccc2)C2CCC2)cnn(C)c1 C12(C(=O)NCc3ccc(C(C)NC(CCSC)=O)cc3)CCC(O)(CC1)CC2 N1(C(C2(N(C)C)CCC2)=O)CCC2C(CCN2C(C2(C)CCCCC2(F)F)=O)C1 Cc1nocc1C(=O)NCC(=O)NC(C(C)(C)C)c1cccs1 C(=O)(CC(C)CC(C)C)NCCC1(OC)CN(C(c2nnsc2N)=O)C1 c1(C(=O)NC2C(NC(c3cnn(CCC)c3C)=O)CCC2)ccc(C#N)cc1C c1(C(N(CCCNC(CCNC(C)=O)=O)C(C)C)=O)cc2cc(F)ccc2[nH]1 C1(C(=O)NCCC2(C(=O)NCCN3C(C)CCC3)CC2)CC(=O)OC1(C)C CC1CN(C(=O)CN(C)CCO)CCCN1C(c1ccc(OC(F)F)nc1)=O c1(OC)cc(C(=O)Nc2cccc(F)c2Cl)c(NCc2cc(Cl)cnc2C)cn1 N1(CC(=O)N(Cc2c(OC)cccc2)Cc2ccsc2)CC2(C1)CN(C)CCO2 CC1CC(C(=O)NC(C)(C)CF)CN(C(=O)Cc2ccnc(O)c2)C1 CC1(C)CCN(C(c2cnnc(O)c2)=O)C1C(=O)NC1CCCC1N=[N+]=[N-] Cc1ccc(N(S(=O)(=O)C(C)C)CC2CCCCO2)c(C)c1 Cn1cc(C=CC(=O)NC2(C)CC(NC(C3(CC(F)F)CCC3)=O)C2)cn1 N1(C(C2N(C(C)=O)CSC2)=O)CCCC(NC(=O)C=C(C)C2CC2)C1 C(=O)(C(C(C)C)OC)NCCCCN(C(C(c1cncnc1)OC)=O)C C=CC(C)(CC)C(=O)N1CC(CNC(=O)CC2CCC3(CCC3)O2)C(F)(F)C1 C=CC(CCC)CC(=O)NCC(CCOC)NC(c1c(F)cc(Cl)cc1F)=O CC(O)(Cc1ccccc1)C(=O)NCC(CC(F)(F)F)NC(c1cocn1)=O N1(C(C2C(=C)C2)=O)CCN(C(c2cccc(F)c2C)=O)CC1c1ccnn1C C1(C(NOCCC)=O)CN(C(=O)Cn2cnnc2O)CC12CC2 Cc1cc(Cl)c(C)c(C(N2CC(CO)(NC(=O)C=CC(C)C)C2)=O)c1N CC1(C)CN(C(=O)C(C2CCCCC2)O)CC1NC1CCNCCC1C c1(CNC(C2C(NC(c3ccoc3)=O)C2)=O)ccc(Br)nc1 c1(NCc2c(NC)nccc2)nc[nH]c(=NCC2(OC)CCCCC2)c1C Cc1cn2c(C(=O)NC3CCN(CC4CCCS(=O)(=O)C4)C3)c(C)nc2s1 CC(=O)CCCC(=O)N1CCC(C)C1CNC(c1ccc(C(C)C)nc1)=O NS(=O)(=O)c1ccc(F)c(NCc2cccc(I)c2O)c1 C=C(Cl)CCC(=O)NC1CN(C(=O)C(C2CCCC2)N(C)C)CC1CC1CC1 C(=O)(CCC(CF)CF)N1CC2C(C(N3C(C(C)C)CC(O)C3)=O)(C2)C1 C#Cc1ccccc1CNC(=O)CCC(C)NC(c1c(CC)noc1C)=O NC12CCOCC1CN(C(=O)C(=O)NCC(N1CCOCC1)=O)C2 C1(C)(NC(Cc2nc(COC)sc2)=O)CCN(C(=O)C(C)CN(C)C)C1 N1(C(Cc2ccc(C)o2)=O)CC(CCNC(=O)CC2(C#N)CC2)OC(C)C1 C12(CNC(C(C)NC(c3ccco3)=O)=O)CC(NC(C3CCCO3)=O)(CCO1)C2 C1(NC(C2(N(C)C)CCC2)=O)C2CC1N(C(C1CC1c1cccc(Cl)c1)=O)C2 CCC(C)C(O)CC(=O)N1CCCC(C)(C(=O)NC2CCN(C)C(C)C2)C1 c1(C(N2C(CNC(C3N(C(C)=O)CCCC3)=O)C=CC2)=O)nccc2n[nH]cc12 N1(C(C(C)=CC2CC2)=O)CCC(F)CC1C(=O)N(C1CC(C)C1)C N12CCN(CC1)C2=O.C(C(O)C(=O)NCC1CCC1)OC S(=O)(=O)(c1cccnc1NCCF)N(C1C(CCC)CCC1)C C(=O)(C1=CC2(CCOC2)C1)NC1CN(C(c2nc(C(C)=O)sc2)=O)CC1C1CC1 Cc1cccn2cc(C(=O)NCC3CCCCC3NC(=O)C(CO)C(C)C)nc12 CCCCCCCC(F)C(=O)N1CCN(C(C2COc3ccccc3C2)=O)CC1 C1(NC(c2nc(C)oc2)=O)CN(C(c2cnsc2)=O)CCC1C C(=O)(C(C)(CC)C(N)=O)NC1CCN(C(C2N(CCC)CCC2)=O)CC1 C(C)(C)(C(C)CC(=O)N1CCSCC1)NC(c1nc(C)oc1)=O C1(CNC(CC=C)=O)CC(C)CN(C(=O)CSCCC(C)C)C1 c1(C(=O)NC(CC)CNC(=O)C(c2ccccc2)SC)ccc2cnccc2n1 C(CC(C)(C)C)(C(=O)N1CC2C(NC(C)=O)C2C1)NC(c1cncc(NC)c1)=O c1(CC(N2CCC(CNC(C(F)=CCC)=O)C23CC3)=O)ccc2nc[nH]c2c1 c1(N(CCCCOC)C)cccc(S(=O)(=O)NC2CCS(=O)(=O)C(C)C2)n1 CC(C)CCC(=O)N(CC(N1CCC1(C)CC(=O)N(CC(C)C(C)C)C)=O)CCO c1(OC)ccc(CCC(=O)N2CCC2CNC(c2cocn2)=O)cc1OC C12(NC(CCCC#C)=O)CCC(Nc3ncncc3OC)C1CC2 C1(CC(C)C)CN(C(C2CCC(C)O2)=O)CCO1.c12ccc(cc1)CN(C)C2C C1(CC(N2CC(=C)C2)=O)CC(OC(C)=O)C1(C)C.C12CCN(CC1)C2=O CN1CCC(OCC(F)(F)F)CC1=O.C1C(F)C(c2ccccc2)NC(=O)N1 c1(C(N)=O)ccc(CCC(N2CCCC2c2cccc(Br)c2)=O)cc1 C1(NC(CN(CC(C)(C)C)C)=O)CC(CNC(c2cc[nH]n2)=O)CC1O c1(CC)c(C(=O)NC2CCN(C(C34CCCC3CC4)=O)CC2)oc2ccccc12 Cc1nc(N2CC3(CCCC3NC(C3CCC(=O)N3C)=O)C2)c2ccsc2n1 C=C(Cl)CC(C(=O)NCCCCN(C)C(C)C)NC(=O)CC1CCC(C)(C)O1 C(=O)(CS(=O)(=O)C(C)(C)C)NCC1CCC(NC(CCSCCC)=O)CC1 c1(CC(N2CCC(N(C(C=CC)=O)C)C2)=O)ccc(C(C)=O)cn1 C12(CNC(CC(C=C)C)=O)CCC(CNC(=O)Cc3cccs3)(CC1)OC2 C(=O)(C1CCc2nnc(C)n21)NCCC1N(C(c2cc(C)ns2)=O)CCSC1 c1(CC)cccc(NC(c2ccc(NC(=O)C(=O)N(C)C(C)C)nc2)=O)c1C C(=O)(C(F)(F)C(F)(F)C(F)F)NCC(CNC(CCC(CC)OC)=O)C N1(C(c2cc(C(C)C)[nH]n2)C(=O)NCCCC)CCC2C(C1)NC(=O)CCN2C C(CNC(C1COC(C)(C)C1)=O)(CC)(CC)NC(c1nc(CCC)oc1)=O c1(C(=O)NC2CC(C)(NC(C3CC(C(C)C)OCC3)=O)C2)cncc2nc[nH]c12 c1(C(N2CC(C)(CNC(C(CC)O)=O)OCC2)=O)cc2c(nnn2C)[nH]1 C#Cc1cccc(CC(=O)NC2CC3C(NC4(COC)CC4)C3C2)c1 C(=O)(CC(C)C(C)(C)C)NCC(C)(CC(C)C)NC(c1c(CC)sc(=N)[nH]1)=O C(=O)(C1=NOC(C)C1C)N1C(CNC(COc2cc(C)on2)=O)CC(C)(C)C1 N1(C(C=CCCC)=O)CCCC(C(N2CCCC2CC2CCC2)=O)C1CC C=CC(C)CC(=O)NC(CCOCCC)C(=O)NC1CC(CO)(CO)C1 c1(Cc2cc(NC(c3ccc(OC)c(F)n3)=O)ncc2)c(O)cc(F)cc1F C1(C(N2CC(OCCOC)C2)=O)CC12CCN(C(c1ccsc1C)=O)CC2 C1(C(=O)NC(CC(=O)NC)C)CCC(C(C)C)N1C(=O)CCn1cnnn1 CC1(C)C(C(C2CC2)NC(=O)NCc2ncoc2C2CC2)C1(C)C C(=O)(C1CCCc2sc(C)nc21)NC1CC(F)(CNC(C(C=C=C)C)=O)C1 C12(C(N(C)CC3(NC(c4ccc(C)nn4)=O)CC3)=O)CC(C)(C1)OC21CCC1 N1(C(CCCn2cc(-c3c(C)cccc3)nn2)=O)CC(C(=O)O)CC12CCC2 N1(C(C2(CSC)CC2)=O)CCC(F)(C(=O)NC2(CF)CC2)C1 C1(CC#C)(C(=O)NCC2CCCC2(C)C)CCN(C(c2ccc(CO)nc2)=O)C1 c1(CNC(=O)NCCn2ncc(C)c2)ccc2ncnn2c1 N1(C(C(CC)n2ccnc2)=O)CCC(C)(CNC(c2c(C)ncn2C)=O)C1 c1(C(C)NC)cc(OC)c(OC)cc1N(C(=O)C(=O)NCCC)C1CCC1 N1(C(c2cnc(C)s2)=O)CCC(C)(NC(c2ccccc2N2CCCC2)=O)C1 CC(C)(C(=O)NC1CCCC(CNC(c2c[nH]nc2C2CCCO2)=O)C1)C(F)F C(=O)(C(C)(C)CCCO)NCC1(OC)CN(C(=O)C(c2ccccc2)=O)C1 c1(OCC)cc(C(=O)NCC2CCC2NC(C2CC2(F)F)=O)ccc1C c1(C(=O)NCC(CNC(C(C)Cc2ccnn2C)=O)(C)O)ccc(C2CC2)nc1 C1(C(=O)NC2C(C)N(C(c3cnn(C)c3N)=O)CC2)CNC(=O)CC12CCOC2 c1(SC)ncc(N)c(C(=O)NC(C)CCNC(=O)Cc2cc(F)cc(Cl)c2)n1 C(=O)(N=c1cc(CCO)cn[nH]1)c1ccnc(N2CC3(CCC(OC)CC3)C2)n1 CC(C)CC(=O)C(=O)NC1(C(N2CCC(C(=O)N(C)C)C2)=O)CC1C C1(C(N2CC(OCCNC(C3CC4(CCC4)C3)=O)C2)=O)CCCC(C(F)(F)F)O1 C(N=c1ccnc(CC23COC(CF)(C2)C3)[nH]1)C(=O)NC1(c2ncccc2F)CC1 C(=O)(CC(C)(O)C(F)(F)F)OCC(=O)NCC1CC(NCc2n(C)ncc2)C1 c1(C(=O)NCC(CN(C)C(c2ccccc2F)=O)O)ccc(Br)c(F)c1 c1(OCC)ccc(C(=O)NC(c2ccnc(F)c2)C(=O)O)cc1 c1(C(C=O)(F)F)ccccc1OC.c1(CN(CC)C)cn(CC2CCCN2C)nn1 O=C(CC(C(F)F)n1ccnc1)NCCN(C(=O)COC1CC=CC1)CC1CC1 C1(C(N2C(COC)C=CC2)=O)CCC2(CC2)N1C(=O)CN1CCSCC1 N1(C(C(CCC)OC)=O)C2CCC1CC(F)(CNC(C1(CC)CCC1)=O)C2 Cc1cc(C(=O)NCC2(CNC(=O)C3=NOC(C)C3)CC2)c(C)n1C1CCCCC1 C1(OC)(CNC(=O)C=CCCc2ccccc2)CCN(C(C2(C)CC2C)=O)C1 C1(C(N2CC(CC(=O)NC(C)C)(C(=O)NCCN(C)C)C2)=O)CC2CC(=O)C1O2 c1(CC)cc(C(=O)NCCc2ocnc2CNC(c2nnsc2SC)=O)on1 c1(C(=O)NCCC(C)N)ccc(CNC(=O)CO)cc1.c1(C2CC2)cccs1 c1(NC(C2CCCN2C(=O)Nc2cncc(F)c2)=O)nc2ccccc2s1 C1(C(N2CC(OC)C(NC(c3cnc(SC)s3)=O)C2)=O)CC(S(C)(=O)=O)C1 C1(NC(C(CO)NC(N)=O)=O)CCCCN(C(c2ccncc2N)=O)C1 c1(OCC)cccc(NC(C2CC(F)CN2C(C2CC2C(C)(C)C)=O)=O)c1 c1(C(=O)NC2(CF)CCN(C(C=C(CC)CC)=O)C2)ncnc2c1cnn2C c1(C(N(C2CN(C(c3c(CC)csc3)=O)CC2(C)C)C)=O)cccn2nnnc12 C1(C(=O)Nc2cn(C)nc2)CC(NC(=O)CN2CCC(=O)CC2)CCO1 c1(C(=O)NC(CN(C(=O)CC2CC3CC3C2)C)(C)C)ccc(S(N)(=O)=O)s1 C1(NC(CSc2ccc(OC)cc2)=O)CN(C(=O)CC2CCN(C)C2)CCC1F Cc1ccc(CCC(=O)NC2CC2CNC(c2cn(C(C)C)nc2C)=O)c(C)c1 c1(N(CC(=O)NCC)C)nc(-c2ccccc2)nc(=NC(CC)CC#N)[nH]1 C1(c2nnnn2C2(C)CC2)(NCCc2cccc(CC)c2)CCOCCC1C c1(C2C(C(CN(C(C3CCCCC3)C(=O)O)C)OC)C2)ccccc1 CC(C(=O)NC1(C)CC(NC(=O)CCOc2ccc(F)c(F)c2)C1)S(N)(=O)=O CCCC(C)(CC)C(=O)NCC(C)(C)CNC(c1ccc(=O)n(CC(C)O)c1)=O N1(CC)CC(NC(=O)C(c2ccco2)NC(c2cc(CO)[nH]n2)=O)CCC1=O C#Cc1cncc(C(=O)NCC2CN(C(=O)CC(=O)NCC3CC3)CC2(F)F)c1 C1(CNC(CC(C)SC)=O)CCN(C(c2cc(Cl)nn2C)=O)C1(C)C N1(C(c2ccc(F)c(Br)c2F)=O)CCC2CN(Cc3ncc(Cl)cc3Cl)CC12 c1(C(C)=O)ccc(CC(=O)OC)cc1.C1(NC(=O)C(=O)NC)CCC1C(F)F n1(CC)cnc2[nH]c(=NC3CCS(=O)CC3)nc(N(CCCCOC)C)c12 C1(NC(C(C)NC(N)=O)=O)CCC(CNC(=O)CCCn2ccnn2)CC1 C(C(=O)NC1CCC1NC(c1ncoc1C1CCCCC1)=O)(C(F)(F)F)OC(C)=O c1(C(=O)NCC2C(NC(C=CC)=O)CCC2)ccc(C)c(C(C)=O)c1 c1(CNC(C2CC2F)=O)n[nH]cc1C(=O)NCC1C=CCCC1 CCC(CC(F)F)C(=O)N1CCOCC(NC(C2CCC(N=[N+]=[N-])C2)=O)C1 C1(NC(c2c(C)nc(CO)s2)=O)COC2(CCN(C(c3ncn(C)c3C)=O)C2)C1 C(CCCCCCCC1CC1)(C1CC1)CN(c1ccc(F)cc1)C C(c1cccc(C)c1)=CC(=O)N(CCNC(=O)CC(C)(O)C1CC1)CC N1(C(C2CC2C)=O)CCN(CCC(=O)NCC(=O)NCC(C)SC)CC1.CO C(C)(C)(C(=O)NCCCCCNC(C1CC(O)C1)=O)OCC C1(CC)CC(C)CCN1C(=O)CC(C1CC1)NC(c1cnnn1CC)=O c1(C(=O)Sc2ccc(C(C)(C)O)cn2)cc(Cl)nc(Cl)c1 c1(C(N2CCCCC(CNC(C=C(C)C(F)F)=O)C2)=O)ccn2c(O)nnc2c1 C1(CCCC)(C(=O)NC(CNC(=O)Cc2cncn2C)C2CC2)CCCC1 C(=O)(C(F)(F)CCn1cc(C2CCCNC2=O)nn1)NCC1(C)CCCC1 N1(c2c(Br)cnc(OC)n2)CC2(CCCC2NC(=O)C2=CC(C)(C)C2)C1 N1(C(CCOC(CC(C)C)C)=O)CCCC(N(C)C(C2(O)CCOCC2)=O)CC1 CCCCC(CNC(=O)CCC(C)OC)NC(C1CCCN1C1CC1)=O C1(NC(Cc2ccc(CC)cc2)=O)CN(C(C2CC(C)CC(=O)N2)=O)C(C)(C)C1 Cc1cc(C(=O)NC2(CNC(=O)CSc3cn[nH]c3)CC2)c(C)n1CC(F)(F)F c1(C(c2nnnn2CCSC)N)ncccc1OC.C1(CCO)CN1.C(CC(C)C)OC N1(C(c2cncn2C)C(=O)NCC)CCC(CN2CCCC3(CC3)C2)CC1C C1(C(C)C#N)CCN(C(C2C3CN(Cc4cc(Cl)ccn4)CC23)=O)CC1 C1(C(CNC(C=C(CCC)C)=O)O)CCN(C(=O)CCC(C)SC)CC1 C1(c2ccc(CC)cc2)CN(C(=O)CC2CC3CC2C3)CCN1C(=O)C(F)OC C#CCC(O)C(=O)N(CCCOCCNC(c1n[nH]c(C)c1O)=O)C N1(C(C2C(=C)C2)=O)CCCCC1CC1CCN(C(=O)CCC2CCOCC2)CC1 C12(CCCC1)CCC(=O)N2.C1(C(=O)OC)CC1(C)C(=O)NC(C)(C)CN(C)C Cc1cc(C(N2CC(NC(c3c(C)ncn3C)=O)CC(O)C2)=O)ncc1N N1(C(c2cc(C)n(C)n2)=O)C2CCCC1CN(C(=O)C(F)CC1CCOC1)C2 c1(C(=O)NC2(COC)CN(C(C3CCCSC3)=O)C2)ccc2nnc(S)n2c1 C(CO)(C(=O)NCC1(NC(=O)CN2CC(C)(OC)C2)CCCC1)NC(C)=O N1(C(CC(C(C)C)O)=O)CCC(C(=O)Nc2cccc(C(C)C)c2)C(C)(C)C1 c1(C(N2CCC2CNC(C2C(=O)NCCC2C)=O)C)cccc2ccccc12 N1(C(C2CCCN(C)C2)=O)CCC2(CC1)CCN2C(c1cc(Br)cnc1Cl)=O C#CCC(C)(CC)C(=O)NCC(C)(C)C#CC(=O)Nc1ccc(F)nc1 Cn1nc(Br)c2cnc(N3C4CCC3(CNC(C3CC35CCOC5)=O)CC4)nc12 CC1SCCCC1C(=O)NCCNC(c1cc(-c2ccc(Cl)s2)on1)=O c1(C(N2CCC3CN(C(C4C5CCCOC45)=O)C3C2)=O)cccc2nc(Cl)cn12 C(=O)(CC(C)(O)COC(C)=O)NCC12OCC(CNC(CCCOCC#C)=O)(C1)C2 c1(C(=O)NCc2cn(CC)nc2)cc(O)ccc1CN1CCCCC1C(=O)O C1(OC)(CNC(=O)C=Cc2sccc2Br)CCN(C(=O)Cn2cnnn2)C1 CCCCS(=O)(=O)CC(=O)NC1CC(NC(c2nc(C)ccc2Br)=O)C1 C1(CNC(CC=CCC)=O)CN(C(=O)COc2cc(C)on2)CC1(F)F C(C1(C)COc2ccccc21)NC(NNC(c1ccc(OCC=C)cc1)=O)=O C(c1ccncc1)=CC(=O)NC(C(=O)NCC1CCN(CC)C1)Cc1ccco1 C1(CNC(CCCNC(C)=O)=O)CCN(C(c2cc(C(F)F)nn2C)=O)CC1C C(=O)(C1CCc2nccn21)N1CCN(C(C2(C)CSC2)=O)CC1CF C#CCC(C)(CC)C(=O)NC1CCOCC1NC(c1cc(C)no1)=O C(=O)(CC(C)(C)CC=C)NCC1(C(=O)NCC=C)CC12CCC2 c1(CC(=O)NC2CN(C(Cc3csc4cc(C)sc43)=O)C2)cn(C)c(=O)nc1O C(=O)(CCC1(NC(c2ccon2)=O)CCC1)NCC1(CC(N)=O)CC1 C1(NC(COC(C)=O)=O)CCCC12CCN(C(c1cccc3nsnc13)=O)CC2 N1(Cc2c(C)ccnc2)CC2CCC(C1)C2NC(=O)C(C)O C(=O)(C1=NNC(C(F)(F)F)C1)NCC1C2CN(C(c3nn(C)c(Cl)c3)=O)CC21 c1(COC)cc(OC)ncn1.C12(CN(C(=O)CC3CC4CC4C3)C1)C(=O)NC2 Cc1ccccc1C(C)CC(=O)NCC1CCCN1C(=O)C(C(C)C)NC(N)=O N1(C(C(N2CCC(C(C)(C)C)C2)=O)=O)CCC(N(F)F)CC1 CN1C(=O)CCC1CC(N1CC=CC1CNC(c1ncc[nH]c1=O)=O)=O CCCC(CC)CCC(=O)N1CCOC(C(=O)NCCCCCCF)CC1 c1(C(N2CCC(C)(CNC(C(C)SC(C)C)=O)C2)=O)cc(S(N)(=O)=O)c[nH]1 c1(C(=O)NC(CNC(CCOCC)=O)(C)C)ccnc(OCCO)c1.CC(F)(F)F c1(NC(CN(C(c2cccc(Cl)c2Cl)C(=O)NC)C)=O)cccc2ccccc12 N1(C(COCCNC(=O)C2=COCCC2)=O)CCC2C(C1)C2(F)F c1(OC)ccc(-c2cnccc2C(=O)Nc2sncc2C(N)=O)c(OC)c1 c1(C(N2CCCN(C(c3cc(C(F)F)no3)=O)CC2)=O)cc2cccnn2n1 N1(C(C2C(O)CCN(C(CC(C(C)C)O)=O)C2)=O)CC(=O)NC(C)(C)C1 n1(CCC)cc(Cl)c(C(=O)NCCC(C)CCNC(c2cnn(CCC)c2)=O)n1 C1(c2cccc(F)c2)(NC(=O)C(F)F)CCN(C(=O)CC(O)C2CC2)C1 C1(NC(c2c(C)c[nH]c2)=O)CC(O)CN(C(c2cn(C)nc2-c2ccoc2)=O)C1 c1(C(=O)NCC2N(C(CNC(=O)OC)=O)CCCC2)c(Br)nc2n1CCC2 N1(C(C(CC)Sc2nc(=N)[nH][nH]2)=O)CC(N(C)C(c2cnc(OC)s2)=O)C2(CC2)C1 C(C1CC1)(C1CC1)=CC(=O)NCC(C(=O)NCC1CC1c1ccco1)OC C(C1CCCc2ccccc21)c1cn(-c2nc(C)cs2)nn1.FCF c1(C(C)Cn2cc(-c3ccc(C4CC4)s3)nn2)ccccn1 c1(N(C)CC2CCN(C(=O)CC3CC=CCC3)C2)ncncc1Cl N1(C(CN(CCOC)C(c2nocc2Cl)=O)=O)CCCN(C2CC2)CC1 c1(C(=O)NC2CC2CNC(=O)C(F)F)nc2c(cc1Br)OCCO2 C=CCC(CC(C)C)C(=O)Nc1ccccc1OCc1cccs1 c1(CN2CCN(C(c3c(C)c(F)ccc3)=O)CC2)cnc2[nH]ccc2c1 Cc1cc(C)n(C(C)CC(=O)NC(CCNC(=O)Cc2cnc(C)s2)C(C)C)n1 CC(CC(=O)N(C)Cc1ncon1)C(=O)c1cccc(Br)c1 c1(CC)cc(F)ccc1C(=O)NC(CNC(=O)C(CSC)c1ccccc1)CC Cc1cc(F)c(OC(=O)CCn2cnc(C)c2C)c([N+](=O)[O-])c1 Cc1ccc(NC(N2CCN(C(C)Cc3ccc(O)cc3)CC2)=O)c(C)c1C N1(C(c2ccn(C)c2)=O)CC2=C(C1)CN(C(C1CCc3ncsc3C1)=O)C2 CC1CC(=O)NCC1C(=O)NCC(C)(C)NC(=O)CCCn1ccnn1 C(=O)(C(C)(C)C(F)(F)F)NCC1CCCCN(C(C2(CCC#C)OCCO2)=O)C1 c1(CNC(=O)NC2CCCCC2)nc2cc3c(cc2[nH]1)CCCC3 c1(C(N2CCC(O)(C(C)NC(CCSCC)=O)C2)=O)cc(N)cc(S(C)(=O)=O)c1 N1(C(C2CC(O)(CNC(C=CC)=O)C2)=O)CCCCCCC1CC c1(C(N2CCC(CNC(C(C)NC(C)(C)C)=O)CC2)=O)csc2nccn12 C1(CCN(C(=O)NCCCOCC(F)F)C2CC2)CCCCN1C1CCCC1 C1(CC(=O)NC(C2CCOC2)C#C)(ON)CCCCC1.C(=O)(C(C)N=[N+]=[N-])N(C)N c1(CC(=O)NCC(=O)NCC2(Sc3ccc(F)cc3)CC(O)C2)ccnc(F)c1 c1(C(=O)NCC=CCCNc2cc(OCC)ncn2)cc2sccc2[nH]1 c1(C(N(CC(O)CNC(=O)CC2CCOC2)C)=O)c[nH]c(=N)c2[nH]ccc12 Cc1sc(C(=O)NC2(CNC(c3c(Cl)ccc(Cl)c3O)=O)CC2)cc1[N+](=O)[O-] O=C(C1=CNC2=NCCCN12)N1CC2CCN(C(C3CC4CCC(C3)O4)=O)C2C1 c1(C(N(CCCNC(c2cc(C)cc(O)n2)=O)CC)=O)nccc2ccncc12 c1(NC(C2N(C(NC=CC)=O)CC2)=O)sc(Cl)nc1C N1(c2snc(C(C)C)n2)CCCC2(CCN(C(=O)C3=CC4(CCOCC4)C3)C2)C1 C(=O)(CCCN(C(=O)C(C)CN(C)C)C)NCCCN(C(C)=O)CC N1(C(=O)Cc2ccc(O)cc2)CCCC2(C1)CN(C(c1cnn[nH]1)=O)C2 CCCCC(CC)CC(=O)NC1CC(CC(=O)NCCOCC)C1(C)C N1(C(=O)NC(C#C)C)CCC(C(C)(C)Cc2ccc(F)cc2)CC1 C(=O)(CCCC(=O)NC1CN(C(C2CC(C)(C(C)(C)C)C2)=O)CC12CC2)OCC C1(CC)CC(CC(=O)NCC2CCCN2C(=O)CN(C(=O)C(C)C)C)CCO1 N1(C(C2N(CC)CCC2)=O)CCC2CN(C(c3cc(C)cnc3N)=O)CC2CC1 CN1CCC2(CC1)CCN2Cc1cccc(Cl)c1O Cc1ccnc2nc(C(=O)NCCC3CCN(C(=O)CC4CCCC4)CC3)nn12 N1(C(C2C(CN(C)C)C2)=O)CCN(C(=O)CCC2(C)CC2)C(C2CCCC2)C1 c1(OC)noc(C)c1C(=O)NC1CN(C(=O)COCP(C)(C)=O)C2CC12 C1(OC)CCCN(N(C)C2CN(Cc3ccccc3)CC23CCC3)C1 N1(C(C(CCC)O)=O)CCC2(CC1)CN(c1nccc(C(C)(C)C)n1)C2C(C)C Cc1ccnc(N2CCCC2c2ccc(Br)s2)c1-c1ccc(C(C)C)cc1 C(=O)(CC(CC)NC(c1ccn(COC)n1)=O)N(CC#C)Cc1ccco1 c1(C(C(=O)NC(CC)CNC(=O)CCc2cnco2)C)ccc(OC)cc1C c1(C(=O)NC(CCNC(C(C)(C)ONC(=O)OC(C)(C)C)=O)C)n[nH]c(C)c1Cl CC(CC(N)=O)C(=O)N1CCC(CCNC(c2ncncc2N)=O)CC1 C1(CNC(c2cc(C)[nH]n2)=O)CCC2(CN(C(c3c(C)ncn3O)=O)C2)O1 c1(COC)ccnc(NC(=O)NC2(C(N3CCCC(C)C3)=O)CC2)c1 c1(CC(C(=O)O)NC(CC2CCC(C)C2)=O)cc(F)ncc1Br C(=O)(CCCC(C)C)N1C(CN(C(=O)C(C)Sc2ccccn2)CC)CCC1 N1(C(C(C)(F)F)=O)CCCC(N(CCO)C(C2CCN(S(C)(=O)=O)CC2)=O)C1 N1(C(C(CCC)OC)=O)CCc2nc(CNC(=O)C(CC(C)C)C(C)C)sc2C1 c1(C(=O)NC2CN(C(COCCCC)=O)C(C)C2)cc(Cl)c2ccccc2c1O N12CC3CC(C(C3)C1)C2C(=O)NSC(F)F.N1(CC(F)F)CCCC(F)(CF)C1 c1(C(N(C(C)CNC(c2cc(C)[nH]c2C)=O)CC)=O)cc(C)n(C)n1 C1(NC(c2cnc(CC)[nH]2)=O)CC(NC(c2ccnnc2C2CC2)=O)C12CCC2 C1(=CCNC(Cc2cc(C)on2)=O)CCN(C(C2(CC(C)C)CCNC2=O)=O)CC1 Cc1cccc(C(=O)N(CCNC(C2CC2C(=O)OC(C)(C)C)=O)C(C)C)c1F CC(C)C(C(=O)NCC(CC1CC1)C(=O)N(CC(F)Cl)C)C(C)C C1(C(C)(C)NC(C(C)NS(C)(=O)=O)=O)CCN(C(=O)Cc2cncn2C)CC1 C(=O)(C1=C(Cl)CCCC1)NC(CNC(c1ccc(C#C)nc1)=O)CC N1(C(Cc2cc(C)no2)=O)CC(N(C(=O)Cc2c(C)n[nH]c2C)C)C2(CC2)C1 C12CCCN(C1)C2.C1(CNCC=C(C)C)CCOC(C)C1 c1(C(=O)NC(C2CCN(C(COC3CN(C(C)=O)C3)=O)C2)C)cc(C)nn1C c1(N(C)CCN2C3CCC2CC3)nnc(-c2ccc(F)cc2)n1C CC(C(=O)NCc1ccc(C(N2CCCC2C2CCOC2)=O)o1)C(C)(C)C C(CC(C(=O)NCCOCCN=[N+]=[N-])NC(=O)C(C)CC1CCC1)SC C1(C(=O)OCC)C2CCC(C2)C1C.C1(=O)C(C)O1.C1CO1.C1CO1 c1(OC)ccc(C(N2CC3CC(NC(=O)C(C)C4CCC4)C2C3)=O)cc1O CN1CCCC(C)(C(=O)NCC(=O)NC2CC(C)(C)C2)C1 O=S(=O)(c1[nH]c(=NCC23CCCC(CO2)C3)ccc1Br)NCC(=C1CCOCC1)F C1(C(=O)NCC2C(CNC(CCC=C=C)=O)C2(F)F)CN2CCN1CC2C C1(NC(=O)C=CC2CCOCC2)CCCC(CNC(C2(C(F)(F)F)CC2)=O)C1 CC1(O)CCCCN(C(C2CCCCC2NC(c2cccc3occc23)=O)=O)C1 c1(C(=O)NCC2(CN(C(=O)CCn3cc(Cl)cn3)C)CC2)cc(F)ccc1F Cc1nc2ccc(C(=O)NCC(C3CCC3)NC(C3(CCN(C)C)CC3)=O)cc2o1 Cc1c(C(N2CCC(O)(C(=O)NCc3ccnn3C)C2)=O)cccc1F Cc1ccncc1C(=O)N(C1CCCN(C(=O)Cc2ccoc2)C1)C c1(OC)ccccc1SCC(N1CCCC(C(C)NC(=O)CN2CCCC2)C1)=O C(=O)(C(C)(C)S(C)(=O)=O)NCC1N(C(c2c(C(C)C)cnn2C)=O)CC=C1 N1(C(C=CC)=O)CCN(C(c2[nH]cc(C)c2C)=O)C(CC)C1 C(C(C)(CC)CC)(c1n(CCOC)nnn1)NC.C1(C(=O)OC)CCCC(C2CC2)O1 c1(N(C(=O)C2=CCCOC2)C2CC3CC2CN3)c(F)cc(OCC(F)F)cc1F c1(C(N2CC(N(C(C(C=C=C)C)=O)C)C(F)C2)=O)ccc(Cl)c(OC)c1F C1(C(=O)NCC(C)NC)CCN(C(=O)OC)CC1.C1(c2cccs2)C(=O)S1 C12(C(=O)OC)CN(CC(=O)Nc3cc(C)cc(C)n3)C(C)(CO1)C2 Cn1nc([N+](=O)[O-])cc1C(N1CC2(CC(NC(=O)C(CO)C(F)(F)F)CO2)C1)=O C1(C(N(C)CC2CCN(C(c3ccsn3)=O)C2)=O)Cc2c[nH]cc2S1(=O)=O N1(C(CC2CC(N(C)C)C2)=O)CCSCC1C(=O)NC1(CCO)CCC1 c1(C(=O)NCC(CC=C)NC(=O)C2=C(C)CCOC2)cc(C#N)ccc1F C(C(C(=O)N(C(C)CO)C)C(C)(C)C)NC(C1C(CC(C)C)C1)=O c1(C(N2C(C3(NC(C4CC5CC5C4)=O)CC3)CCC2)=O)nc[nH]c2ncnc1-2 N1(C(c2n(CC)cc(Cl)c2)=O)CC2(C1)CN(C(=O)CC(C)c1ccco1)CCO2 C(C1=CCCN(C(=O)CCC2CCCC2)C1)NC(=O)Cc1ccc(OC(F)F)cc1 C1(C(C)C)(C(=O)NCc2nc(Cl)n[nH]2)CCCN1C(c1cccnn1)=O O=C1NCC(C(=O)N(C2(C(C3CC(F)(F)C3)=O)CCC2)C2CC2)N1 C(CC(=O)N1CCC(NC(c2cccc(N)c2O)=O)CC1C)(C(F)(F)F)OC c1(CC)cc(C(=O)NCC2COCC2NC(C2CCN(C(C)=O)C2)=O)cc(O)n1 C(=O)(C1=NN(C)C(=O)CC1)NCC1CC(F)(CNC(c2cn(CC)nn2)=O)C1 C1C(C)(O)CC(=O)N(C)CCN(C)C(=O)C2CC(C2)C(=O)N1.CCOCC c1(C(N2C(C(N3CCC(CO)CC3)=O)CSCC2)=O)cccc(F)c1Br C1(C(N(CCCCCNC(=O)CN2CCCCCC2=O)C)=O)OC(C)(C)OC1=O C(c1ccc2c(c1)OC(F)(F)O2)=CC(=O)OCC(c1c(Cl)ccc(Br)c1Cl)=O c1(C(=O)NCC(C(C)C)NC(CC(c2ccc(C)cc2)C)=O)cc(Cl)ccc1F C1(CN(C)Cc2ccc(C(C)(C)C)s2)CCN(CC(c2ccccc2)O)CC1 c1(NC(C2C3CN(C(c4ccnc(C)n4)=O)CC32)=O)cc(F)c(F)cc1[N+](=O)[O-] C1(C(N2CC(O)(C(C)NC(C(C3CC3)OCC)=O)C2)=O)CCC(=C(F)F)CC1 c1(OCC)ccccc1C=CC(=O)NC12CC(NC(c3c(C)ncnc3O)=O)(C1)C2 C(N=c1ccnc(CO)[nH]1)C1C(CNc2cc(CC)nn2Cc2ccon2)C1 C=C(C)CCCC(=O)NC(C(=O)N1CCN(C)CC1CCO)C(C)(C)C C12(C(N(CCCCNC(C(C)Cc3ccccn3)=O)C)=O)C=CC(CC1)C2 Cc1c(Br)ccnc1C(=O)NCC1(F)CCN(C(=O)C(C)(C)OC(C)C)C1 C1(CC(=O)OCC)COCCN1C(C1CCN1C(c1cncc(F)c1)=O)=O C12(C(N3CC(CC)OCCC3)=O)CCCC1CN(C(c1ccc(O)cc1F)=O)C2 c1(C(=O)NCC2CC2NC(C2CCC2(F)F)=O)cccc(C(F)F)c1F C(CC)(CCC(=O)NCC(O)C(C)O)NC(C(C)OCCCC)=O c1(C(N2CCC2c2cn(C3CCC3)nn2)=O)cc(Br)ccc1C(F)F N1(C(C)C)N=C(C(=O)NC2CCN(C(=O)Cc3cccnc3)CC2F)CCC1=O c1(CC(=O)N(C(C)CCNC(C2CC(F)C2)=O)C)ccnc(O)c1 C(CCCNC(c1cccs1)=O)(c1ccccc1)NC(CC1(CC)CCC1)=O N1(C(C(C=C=C)C)=O)CCC2(NC(=O)CCCOCCOC(C)C)CC2C1 C1(C#N)(C(N2CC(C(=O)NCC(=O)NCCC(C)C)(COC)C2)=O)CC(C)C1 c1(CC(=O)OCC(=O)NCCN(CCCC)CC)cc(C(F)(F)F)nn1C Cc1oc(C#N)cc1C(=O)NCC(C)C(=O)NC1(C)CS(=O)(=O)C1 c1(C(=O)NCC2CCN(C(C3CN(C(C)C)C3)=O)C2)cc2[nH]ccc2s1 C1(C)(CNC(c2n(C(CC)(C)C)nnn2)c2noc(CC3CC3)n2)C=CCCC1 CC1(CNC(C2CCCN2C(=O)CCc2cc[nH]n2)=O)CCCCCC1 c1(C(=O)NCC(CO)NC(C(C)Cc2ccccc2F)=O)cc2cccnc2o1 C(=O)(C1=CCCOCC1)NC1CCN(C(c2n(CC#N)ncc2)=O)CC1O CCCCCC(=O)NC1CCN(C(=O)CCc2ccccc2F)C1CC1CC1 C1(C(N(C)CC2(Br)CC2)=O)CCCCC1CNC(=O)CN1CCSCC1 C1(C(N2CC(C)C(NC(=O)C(C)(C)CF)CC2)=O)CC2C=CC1C21CC1 C1(C(=O)NCc2c(C(N(CC(N)=O)CC)=O)nco2)CCC(C2CC2)C1 C1(C(=O)NCC(CCC)NC(=O)C(C)(O)C2CCC2)CCCC(F)(F)C1 C(c1cccc(N)c1)=CC(N1CCCC(Cn2cc(C(C3CCCO3)C)nn2)C1)=O C12(C(N3CCC(N(C(C(C)SC)=O)Cc4cnccn4)C3)=O)CC(C1)C(C)O2 C1(NC(c2c(C#C)c[nH]n2)=O)C2CC3C(C2)C13C(=O)N(CC)OC CC1(C)CC(C(=O)NCCOCCC(=O)NCC2CC3CCCC3C2)CCO1 c1(C(N2CCC(C(F)F)(CNC(C=CCOC)=O)C2)=O)ncc(Cl)cc1F c1(C(=O)NCC(CCNC(C(CC(=C)C)C)=O)O)cc(C)nc2cc(Cl)ccc12 CN1Cc2c(CNC(c3nn(-c4ccccc4)n(C)c3=O)=O)cccc2C1=O N1(C(C(c2ccccc2)OCC)=O)CC2(CCOCC2)C1.C1C(C)C(=O)N1 N1(C(c2n[nH]c(C3CC3)n2)=O)CC2CCN(C(=O)C(F)CC3CCCC3)C2C1 c1(N(C(C2CN(C(=O)Cc3cn[nH]n3)CCO2)=O)CCl)c(Br)cc(C(F)(F)F)cc1I C(=O)(C(C)CCC(=O)OC)NC(c1cnn(C)c1)C(=O)NCCCC=C CC1(C(N2CC3CC2C3C(=O)NCCC2CCC(=O)N2)=O)C=CCCC1 C(=O)(CC(C)C(F)(F)F)N1CCCC(C)(NC(Cc2ccc(SC)cc2)=O)C1 c1(C(=O)NC(C(C)C)C(C)NC(=O)CC2C(C)(C)C2(C)C)noc2ncccc12 N1(C(Cn2cc(-c3ccc(OC)nc3Br)nn2)=O)CC2CC(CO)CC(C1)C2O c1(C(=O)NCCC(C)(C)NC(C2CC=C(C)CC2)=O)cc2n(n1)C(C)CCC2 C1(NC(C2(OCC)CCCC2)=O)CN(C(=O)CC2(C3CC3)CC2)CCC1O C1(NC(C(CCSC)N)=O)CCC(C)(C)CC1NC(=O)NC(C)(C)C N#CC1CCN(C(C2(Cc3nccs3)CC2)=O)C1.c12cc(ccn1)NC2=O c1(C(=O)NC2CCCN(C(C3CC34CCSCC4)=O)CC2)scc2c1CCCC2 C1(NC(C2CCC(C(C)C)CC2)=O)CCCCN(C(C2(F)CCOC2)=O)C1 C1(C)(CCNC(c2c(C)onc2)=O)CCN(C(C2CCC(C(C)(C)O)CC2)=O)C1 N1(C(=O)NC2CCN(C(N)=O)CC2)CCCCC1NC(C(=O)NCC)=O c1(OCC(=O)NC(CC)CN(C(=O)C=CC2CCCC2)CC)cccc([N+](=O)[O-])c1 C1(C(=O)Nc2c(C(=O)OCC)ncs2)(CF)CCN(C(c2cc(C)c[nH]2)=O)C1 C=CCC(C)(C)CC(=O)NC1CCN(Cc2cc(C)cc(Br)c2O)CC1F N1(C(C(c2cccc(Cl)c2)(C)F)=O)CC2CC1CN2C(=O)CCc1ccoc1 CC1(C)CCCC(C(=O)NC2CCC(=O)NC2c2ccccc2)O1 c1(C(N(CCNC(C2CN(C)C(=O)C2)=O)CS(C)(=O)=O)=O)ccc(Cl)c(C#N)c1 C1(C(=O)NC(C2CC2(Cl)Cl)CNC(C)=O)C2CCC1(c1cnco1)C2 c1(C(C)C)c[nH]c(C(=O)NCC=CCNC(C2(SC3CC3)CC2)=O)c1 N1(C(c2cccc(CNC(C3C(C)OCC3)=O)n2)=O)CCOC2(CCC2)C1 C(=O)(C(O)CCC(C)C)NC1(CNC(c2nc(OC)c(F)cn2)=O)CCOC1 CCCC(CC)CCC(=O)N1CCC(OC2CCC2)CC1.C12CCN(C1)C2C n1(CC(C)(F)F)ccc(NC(N2CCC(N)C2)=O)n1 c1(C(=O)OCC(CCC(=O)N2CC(COC)OCC2)=O)cc(C)c(O)nn1 C(N(O)C(=O)Cc1cccc(Cl)c1)c1cn(C(C)C(=O)N(C)C)nn1 N1(C(C2N(C(C3N(C)C(=O)CCC3)=O)CC(O)C2)=O)CC2C=CCC(C2)C1 CC1(CC(N2CC(CNC(c3cn(C(F)(F)F)cn3)=O)C(O)C2)=O)CCCCC1 C1(OC)CCCC(NC(c2nc(-c3cnccn3)no2)C)C1 CC12CCC(C(=O)NCC3CCCCCN3C(=O)Cn3cnnc3)(CC1)CO2 N1(C(CCOCCOCCOC)=O)CC(NC(=O)C(F)(F)CO)C(C)C1 C1(C2CC2)(NC(CCCC=C)=O)CCN(C(c2noc3c2CCCC3)=O)C1 CC1(C)CCC(C(=O)NCc2nn[nH]n2)(NC(C2CCC3(CCC3)O2)=O)C1 Cc1ccnn1CC(=O)N(C1(O)CN(CC(C)CC#N)C1)C c1(CC)ccc(C(=O)NCC23CC(C2)N(C(=O)C(C)(C)CF)C3)cc1OC C1(C(=O)NC2(CC(=O)OC)CC2)CC=CCC1NC(C1(C#N)CC1)=O C12(CSC)CC(C(=O)NC3CCC(NC(=O)CC4CCCCC4O)C3)(CO1)C2 c1(C(N(C2CN(c3ccnc(-c4ccccc4)n3)C2)C)=O)onc2ccccc12 C1(CCCC)CN(C(=O)C(COC)CC)CCN1C(c1cn(C)nc1C(C)C)=O CC1(C)CC(CC(=O)NCC2CCCC2NC(c2cccc(O)n2)=O)NC1=O C1(CNC(C(C(C)C)NC(COC)=O)=O)COCCN(C(c2cc(C)c[nH]2)=O)C1 N1(C(CC(C)OC(C)=O)=O)CCC(NC(=O)C(=O)N(C)C)CC1 C1(N(C)C(c2ccc(CN=[N+]=[N-])o2)=O)CCCN(C(C2CC3CC2C3)=O)CC1 c1(C(N(C2CN(C(Cc3cc(C)[nH]n3)=O)CC2F)C)=O)cc2nccn2c(O)n1 C(=O)(CCCc1sccc1C)N1CC1C.C1(C(=O)NC)(CCOC)CC1 C12(CNC(C(C(CC)CC)C)=O)CCCC1N(C(=O)C=C1CCCCC1)CCC2 C(=O)(C1=NOC(C2(O)COC2)C1)N(CC(C)NC(C12CC(C1)C2)=O)C CC(C)S(=O)(=O)C(C)C(=O)N1CCC2CN(C(c3cc(Cl)n(C)n3)=O)CC2C1 Cc1cccc(C)c1C(=O)NC1CC1C(=O)OC(=O)C(C)N(C)C CCC(C=O)OCc1ccccc1.C1(C(=O)N(CCO)CC)CCC(=O)N1 C(CCCC(=O)NCc1ocnc1C(N1CCOC(C(C)C)C1)=O)OCC C1(NC(Cn2c(C)cc(C)n2)=O)CC2CC1CN(C(c1onc(C)c1F)=O)C2 C1(C(=O)NC(C2(O)CCN(C(=O)CNS(=O)(=O)C3CC3)C2)C)C2CCCCCC12 c1(C(C)OC)nc(C)c(C(=O)OC)s1.C1(=O)C(F)(F)Cn2cc(nn2)C2CC(C2)N1 c1(C=O)ccc(C(C)C)cc1SCC.C1(CCN(C)C)CC=CCC1 c1(CC)nc(C)oc1C(=O)NCC12CC1CN(C(c1csc(O)n1)=O)C2 c1(C(=O)OCC)cnn(C)c1C(=O)NC1CCCCC1CNc1nc(OC)c(C)s1 C(=O)(CCCC(CC)NC(=O)Cc1c(C)cnn1C)NCCCC=C C1(O)(CN(C)C(C2CC3CCC3C2)=O)CCN(C(C2(C3CCCO3)CC2)=O)C1 C1(C(N(C(C(=O)NC(C#C)(C)C)CC)C)=O)CC(=O)N(CC)C1 c1(C(N2CCC3(NC(=O)COC4CC=CC4)C(C2)C3)=O)cc(Cl)c([N+](=O)[O-])[nH]1 c1(C(=O)NC(C)CCNC(=O)C(c2cccc(F)c2)C)cnc2n(c1=O)CCS2 c1(C(N2C(CN(C(c3ccc(C=C)cc3)=O)C)CCC2)=O)cncc2[nH]ccc12 C=CCCCC(C(=O)NCC(C)C(F)(F)F)NC(C1COCOC1)=O c1(CNC23CC(C(=O)Nc4c(C#C)cccc4)(C2)C3)n[nH]c2ccc(Br)cc12 c1(C(C(N2C(CNC(CC=C)=O)C=CC2)=O)C)ccc(F)c(Br)c1 c1(CCCC(=O)OCc2ccncc2Br)c[nH]c2ncccc12 c1(C(C(=O)NCC)N(c2ccccc2)C(C)=O)cccc(Cl)c1 C(c1ccc(OC(F)(F)F)cc1)=CC(C)NC(N(OCC)CC)=O CC1=C(C(=O)N2CCCOC(CNC(C3(F)CCC3)=O)C2)CCO1 N(C1CCc2cc(F)c(F)cc21)C(c1cn(C)nc1)C(=O)NCC1CCOCC1 N1(C(CC(=O)N(C)C)=O)Cc2ccccc2C1CNC(=O)CCC(C)(C)F c1(CNC(CCNC(=O)OC)=O)c(NC(=O)NC(C)(C)C)cnn1CC(F)(F)F C(C)(CCC(=O)NCCOCCC(=O)NCC1(O)CCSCC1)OCC C1(NC(C(CSC)c2ccccc2)=O)CCCCC1NC(=O)C=Cc1cncn1C C1(NC(Cn2ncc(CC)c2)=O)CCC(C)(C)CC1NC(=O)CN(C)C1CC1 C(=O)(C1CCCCc2ccccc21)NCC1CC(NC(=O)CCc2cnco2)C1 C12(NC(CC(C)(C)F)=O)CCC(C1)N(C(=O)C(C)(C)N1CCCCC1)C2 CC(=O)C(C)CC(C)C(=O)N1CC(C(=O)NCC(O)CC(C)C)C2(CCC2)C1 C1(CNC(C(CCOC)C)=O)CCCCN(C(c2cc(-c3ccco3)c[nH]2)=O)C1 c1(OC)ccc(-c2n[nH]c(CN3CCCC3(C(=O)N(C)C)C(C)C)c2Br)cc1 c1(C(N(c2ccccc2)OC)=O)nc(NC(=O)C(C2CCCCC2)F)oc1C C(N=c1ccc2ncc[nH]c-2n1)C1(C)CCN(C(C2CC(F)(CO)C2)=O)C1 C(CCCCCNC(=O)CCOCCNC(C1CCOC(C(F)F)C1)=O)N(C)C Cc1cc(C(N2CC(O)CC2C(N2CCN(C3CCCC3)CC2)=O)=O)ccc1Br c12nocc1C(=O)NC2.C(CC(C)(C)C1CC1)OC.C1(C2CCCC2)C(=O)N1 C1(NC(C(=O)NCC2CC2)=O)CCCC2CN(C(c3nccc(Cl)c3F)=O)CC12 N1(C(C(C)(C)OCC)=O)CCN(C(c2cnncc2C)=O)C(Cc2nc(C)no2)C1 CC1(C)CC(NC(C2CC23CC(O)C3)=O)CN1C(c1ccc(C(N)=O)nc1)=O CCS(=O)(=O)CC(=O)NCC(CC)CC(=O)NC(CO)CCCO c1(CNC(C2(NC(c3n[nH]c(C)c3Cl)=O)CCOCC2)=O)ccnc(F)c1F C(=O)(C(C)CC(N)=O)NCC1(OC)CN(C(CC2(C(=C)F)CCC2)=O)C1 CC1CN(C(c2ccnc(N(C)CCOCCO)c2)=O)CCC1C(=O)O C(C(=O)N1CCCCCO1)C1(N(C(c2cc(C)c(C)nc2)=O)C)CC1 N1(C(C2CC(n3cc(CCC(C)=O)nn3)C2)=O)CCCN(CCO)C(=O)C1 c1(C(N2CC(CN(C)C(c3c[nH]c4cccnc34)=O)C2)=O)ccc2[nH]ccc2n1 Cc1n[nH]c(=NCC(C)(C(C)C)NC(=O)CC2CCNC2=O)s1 c1(-c2onc(C)n2)ccc(C(=O)NC(C)CNC(c2nocc2Cl)=O)cc1 C(CC(C)(C)CC(=O)NC1CCN(C(=O)CC2CCOC(C)(C)C2)C(C)C1)OC C1(NC(C2(c3ccn(C)c3)CC2)=O)COCCN(C(c2ccoc2)=O)C1 CC1CC(NC(=O)CC(C)(C)c2cccs2)CCN1C(c1cnc(=N)[nH]c1)=O CC1=NN(C)C(=O)C1CC(N1CCC1CNC(=O)CSC(C)(C)C)=O C(=O)(CCCCC(=O)NC)N1C2C(N(C(C(C=C)C)=O)C)CC(C2)C1 C12(C(=O)NC(CNC(C(C)NC(N)=O)=O)CO)CC3CC1C2C3 CC1(C(=O)NCC2(F)CCC(CNC(=O)C(F)CC3CC3)CC2)CCC(O)CC1 c1(C(=O)NC2C(NC(=O)Cc3cnc[nH]3)CC2)cnc2c(Br)n[nH]c2c1 C(=O)(C(O)CC(C)C)NC1CC(CNC(C(C(=O)OCC)C2CC2)=O)C1 C(=O)(CCCC(=O)NC1CC1)NC(C(=O)NCC1(O)C(C)CCC1)CO c1(OCCC(=O)NC(C)C=CC(=O)N(C)CCO)ccc(F)cc1Cl Cc1cc(C(c2nnnn2C2CCC2)NCCCCCCO)ccc1Cl c1(OC)cnc(F)c(C(=O)NCC(n2cc(-c3cnccc3Cl)nn2)C)c1 C1(C(N(C(CC(=O)NC)C)C)=O)CCN(C(=O)CCc2cnoc2)C(C(C)C)C1 C1(NC(C2C(CNC(Cc3cnc(C)s3)=O)CC2)=O)CCCN(C)C1 C1(CC)C(NC(c2cccnc2C)=O)CCCN1C(=O)CN1CCC(OC)C1 C1(C(=O)NCC(C(C)C)C)CC2CC2N1C(c1csc(Cl)c1)=O c1(SC)nc(N(C2CCNCC2(C)C)Cc2cncc(F)c2)cc(C)n1 C1(NC(c2c(C(C)C)cccc2)=O)CC2CCC(C1)N2C(C1(N=[N+]=[N-])CC1)=O N1(C(C(C)CCO)=O)CCN(C(=O)Cc2csc(NC=O)n2)CC(O)C1 C1(C(=O)NCCN(C)C(c2c[nH]nc2Br)=O)(OC)CC(C)CC(C)C1 Cc1cn2c(n1)CCC(C(=O)NC13CC(C1)N(C(C1CCCOC1)=O)C3)C2 C(=O)(C(C)CCO)NCC(C(C)C)NC(c1ccc[nH]1)=O c1(OC)cccc(C(N2CC3C(N(C(C(C4CC4)OC)=O)C)C3C2)=O)c1O C1(C(=O)NCC2OCCC(NC(C3(CC(C)C)CCC3)=O)C2)CCCS(=O)(=O)C1 C1(CCNC(C2CC(OC(F)F)C2)=O)CCN(C(=O)CSC2CCCCO2)C1 C1(C(N(CC(C)CNC(C2CC2C(C)(F)F)=O)C)=O)CS(=O)(=O)CC(=O)N1 C1(NC(c2ccc(C)c(O)c2)=O)CN(C(=O)CC2(C)CC2F)C2(CCOCC2)C1 CC(C)C(C(=O)NC1CCN(C(c2c[nH]nc2F)=O)C1)N1CCCCCC1 N12CCC(C1(C)C)NCC2=O.N1(C(=O)OC)CCC(CCC(=O)N(C)C)C1CO C1(N(C(c2c(CC)nco2)=O)C)C2CN(C(=O)CCOc3ccccc3F)CC12 N1(C(C(CCSC)O)=O)CCC(NC(C2CN(C)CC(C)O2)=O)CC1C CC(C(=O)NNc1ccc(Br)nn1)c1cccc(Br)n1 c1(-c2onc(C(c3ccc(OC)nc3)N)n2)ccc(OCc2ccccc2)cc1Cl C1(Cc2cn(Cc3c(CC)cco3)nn2)CCN(C(C2CCCCS2)=O)CC1 C1(NC(c2ccc(SC)cc2)=O)CN(Cc2cccnc2)CCC1(F)F N1(C(C(C)SCC)=O)CCC(C)(CCn2cc(CNC(N)=O)nn2)CC1 C1(O)(CCCC(=O)NCCNC(C2C(C)(C)C2N2CCC2)=O)CCCOC1 CN1CCN(C(=O)C(CNC(C2OC3CCC2C3)=O)N(C)C)CC1CO c1(C(N2CCN(C(C3C(=C)C3)=O)CC2C2CC2)=O)cc(S(N)(=O)=O)c(Cl)cc1Cl c1(CC(C)NC(=O)C(C)CC2CCCC2)ccc(CNC(=O)CNC=O)cc1 C#Cc1ccc(C(N2CCCC(NC(=O)C(C)N(C)C)C2C)=O)cc1 C1(C(N(C)CC2CN(C(=O)Cn3nnc(C4CC4)n3)C2)=O)CCCS1(=O)=O N12CCN(CC1)Cn1c2nnc1-c1cccc(F)c1.C1CC(C)CO1.CC CCC(CC(F)F)C(=O)N1CCCC(CCNC(c2cc3oc(Cl)cc3[nH]2)=O)C1 N1(C(CC#C)=O)CC2CCC2(CC(N2CCCC2C(=O)N(C)C)=O)C1 c1(NC(C2CC(=C)CN2C(c2cc(Cl)cs2)=O)=O)cccc2c([N+](=O)[O-])cccc12 C1(C(=O)NCC2N(C(c3cncs3)=O)CCC2)CC12CCOc1ccccc12 c1(OC)cc2c(c(S(=O)(=O)N3CCCCCC3C3CC3)c1)OCC2 c1(C(=O)Nc2ccc(-c3cnn[nH]3)cc2)ccc(O)cc1Cl c1(C(=O)NCC2CCN(C(=O)C(N3CCOCC3)C3CC3)C2)cccc(CO)c1 c1(CNC2CCC(OCC=C)CC2)ccc(F)c(OC)c1F c1(C(N2CC(OC)CC(NC(C(C=C)(C)C)=O)C2)=O)ccc2nn[nH]c2c1 N1(Cc2n(CC=C)c(-c3ncccn3)nn2)C(=O)C2c3ccoc3CCN2C1=O CC(C)(C)CS(=O)(=O)NCCc1c(Cl)cccc1Cl C1(C(N2CC(NC(=O)Cc3nnco3)C2)=O)CCCC12OCCO2 N1(CCNC(Cc2cc(C)no2)=O)CCN(C(C2CCCC23CC3)=O)CC1 c1(CC(=O)NCC(CN(C(C)=O)C)O)n[nH]c2ccc(Cl)cc12 c1(CC)ccc(C(N2CCC(NC(c3cc(COC)no3)=O)C2(C)C)=O)cc1F N1(C(C2N=C(C)SC2)=O)CCCCC2(C1)CN(C(=O)CCCN1CCCCC1)C2 NS(=O)(=O)CCC(=O)NCCCC1CCCN1C(c1ccc(NC=O)cc1)=O C1(C(=O)OCC)C(C(C)NC(=O)CCN(C2CCCC2)CC(C)C)C1(C)C CC(C)(C)S(=O)(=O)CC(=O)N1CCN(C(C2COC(=O)N2)=O)C2CC12 c1(C(=O)NCC(CC(C)C)NC(C2CCCC(N(C)C)C2)=O)cc2ccsc2[nH]1 Cc1ccc(C=CC(=O)NCC2(CNC(=O)C(C)O)CC(F)(F)C2)cn1 N1(C(c2cnc(C)nc2C)=O)CCCC2(NC(c3cnc(C)[nH]3)=O)CCCC12 Cc1cc(F)cnc1C(=O)NCC1CN(C(C2CCO2)=O)CC12CC2 N1(C(=O)OC(C)(C)C)C(C(=O)NC2(Cl)CC3CCC2O3)CCC12CC2 N(C1CCc2c(Cl)ccc(Br)c21)Cc1cnc(OC)nc1 C1(C(=O)NCCC2CCN(C(C3CC(C(=O)OC)C3)=O)C2)CCC(C)(C)OC1 c1(NCC(C)C(F)(F)F)ccc(S(=O)(=O)NC2CC2C2CCOCC2)c(Br)c1 C=CC1(CC(=O)NCCN(C(=O)CC23CCC(CC2)OC3)C)CCCCC1 c1(NC(C)=O)ccc(C(=O)NC(C)CNC(C2(C#N)CC=CC2)=O)c(Cl)c1 C1(N(C(c2ncc(C)s2)C)C)CCCCN1C=O.C1(ON)CN(C(=O)OC(C)(C)C)C1 N1(S(c2ccc(SCC)nc2)(=O)=O)CCCC2(CCN(C(=O)CC3CC3C)C2)C1 c1(NCCCC(N)=O)nc(N2CCSCC2)nc2scnc12 C1(NC(CCC2(C)CC2)=O)CC2CCC1N2C(c1ccc(OC2CCC2)cc1)=O C(=O)(CCCS(C)(=O)=O)NCC(c1ccccc1)CNC(CC(CC)SC)=O CC(C)C(C(=O)NC1CN(C(C2CCC2)=O)CC1C)NC(c1cccs1)=O N1(CCCNC(C2C(OC(C)(C)C)C2)=O)CCN(C(c2ccc(F)s2)=O)CC1 CCC(C)(C(=O)NC(C)C(=O)NCCC(C)N1CCC1)OC N1(C(c2c(C)n(C)nc2)=O)CC2CN(C(=O)C(c3cccnc3)C)CC2(C)C1 c1(C(=O)N(CC(=O)NCCO)CCCC2CC(O)C2)c[nH]nc1C(F)F c1(OCC)cc(Cl)c(C)cc1NC(=O)C(F)(F)CC(c1ccccc1)c1cccs1 c1(C(=O)NCc2ccc(OC)cc2OC(F)F)c[nH]c2nc(F)ccc12 Cc1cnc(Cl)c(C(N2CCN(C(=O)CC3(O)CCCC3)CC2C(C)C)=O)c1 N1(C(c2cc(C#N)sc2)=O)CCCC2(CCCN2C(c2ccc(Cl)nc2O)=O)C1 N1(C(Cc2ncc(C)s2)=O)CC(C2CN(C(c3cc(F)c(F)cc3O)=O)C2)C1 Cc1cnsc1C(=O)NCC(C)NC(c1ccn(C2CCC2)n1)n1cccn1 CCCC(C)(C)C(=O)N1CCC(C)(NC(C2CCC23CCOCC3)=O)C1 CCCC(CCC)CCCC(=O)N1CC(CCNC(=O)CN(C2CCSC2)C)C1 C1(C(=O)OC)CC(=O)CN1C(c1c(O)noc1C)=O c1(C(N2CC(C)C(CNC(C3CCCCO3)=O)CC2)=O)cccc([N+](=O)[O-])c1 Cc1cc([N+](=O)[O-])cc(Br)c1NC(=O)NCCC1CCOC(C)C1 CCC(C(=O)OC)C(=O)NCc1cc(C(=O)NCC(=O)NOC)on1 CN1CC(C(N2CCC(F)C(NC(=O)CCc3csc(=N)[nH]3)C2)=O)OCCC1=O Cc1ncc(CC(=O)NC(C2(O)CN(C(C3CC3[N+](=O)[O-])=O)C2)C)[nH]1 C1(CC(=O)NCCN(C(=O)CCNC(=O)CC(C)C)CC)CCC(=O)N1 C(=O)(C1=CCCOC1)NC(CCNC(C(C(C)C)N(C)C)=O)C c1(N2CCCC(CNC(=O)CC3CCCS3(=O)=O)CC2)c(Br)cccc1[N+](=O)[O-] c1(NCc2cc(C)ns2)cc(NCC(Cl)=CCl)ncn1 c1(CN2CC(C)C(n3cc(C4(C(=O)O)CC4)nn3)C2)ccc(F)cc1Cl CC(O)(CC(=O)N1CC(NC(=O)COCCCF)C(c2ccccc2)C1)C1CC1 C(=O)(C(C)(C)CC(=O)NC(C)CNC(c1ccccc1C(C)(C)C)=O)OCC Cc1cccnc1C(=O)NCC(CC(=O)NCC1CCNC1=O)C1CCC1 CC1(C)C2CCC1(C)C2C(N1CCC1CNC(c1cc(F)ccc1F)=O)=O c1(CC)cc(C(=O)NCC2CCC(C(=O)NCCC(C)(C)F)O2)n[nH]1 O(C=C(C#N)C(=O)N1CC(NC(c2cc(C3CCC3)no2)=O)C(C)(C)C1)CC C1(Nc2c(C)cnn2CO)COc2ccccc2C1C c1(CNCC(C)N(C(C(C(=O)NCC)(C)C)=O)C)nc(C)nc2sc(C)c(C)c12 N1(C(C2CN(C(=O)CO)C2)=O)c2cccnc2CC1c1ccccc1 C(C(COC)C(=O)NCC1CCCN(C(C2(N(C)C)CCCOC2)=O)C1)OC c1(OC)ccc(C(C(=O)NCC2CCCO2)N(C)C(CC(F)F)C)c(Cl)c1OC C1(NC(=O)Nc2c(C)cccc2)CC(F)CN(Cc2ccn(CCF)n2)C1 c1(C(=O)NC2C(NC(C(C)NC(C)(C)C)=O)CCOC2)cn2c(n1)CCC2 C(C)(C(=O)N(CCCNC(=O)CNC(=O)Cn1cncn1)C)=CC Cc1ccc(C(=O)NCC2CN(C(c3cnnn3C(C)C)=O)CCO2)c(C)n1 C#Cc1ccc(C(N2CCC3CC23C(=O)NC(CSc2nc[nH]n2)CC)=O)cc1 C1(NC(CCn2ncc(C)c2)=O)CC2CCC1CC(NC(C1(C)CC=CC1)=O)C2 C#CCCCC(C)C(=O)NCC12CCC(CNC(c3cnc[nH]3)=O)(CC1)CO2 CC1CC(NC(=O)Cn2cnnc2O)CN1C(=O)CN1CCS(=O)CC1 C1(C)(C(=O)NCCC(CC)(C)NC(C2COCCO2)=O)CCCN(C)C1 C1(OC)CCCN(C(=O)C(CC(C)C)ONC(c2cccc(F)c2)=O)CC1 C1(NC(c2ccoc2)=O)CCC12CCN(C(=O)C1=CSCCO1)CC2 c1(N(CC=C)C)nc(N(C2CC2)Cc2cccc(CN(C)C3CC3)c2)c2c(n1)CCC2 c1(N2CCC(NC(c3c[nH]nc3-n3cnnn3)=O)C2=O)ccc(Cl)c(Cl)c1 CCC(CC(F)F)C(=O)NCC1(NC(c2ccn(C(C)(C)C)n2)=O)CCOC1 C1(CNC(C(=O)NCC)=O)C(C)CCN1C(c1ccc(CC)o1)=O C1(C(N2C(CNC(COCCCCC)=O)CC2)=O)CCCC(F)(F)C1 C1(NC(CN(C2CCSC2)C)=O)CC(C2CCN(C(C3CC3F)=O)C2)C1 CC1C(C)N(Cc2cccc(C#N)c2Br)CCN1C(c1ccccc1)=O c1(C(C(=O)NCC(C)C)N(CCCOC)CC2CC2)nc(Br)ccc1OC n1(C(c2cccs2)C)nc(-c2ccnc(Cl)c2)nc1-c1sccc1Cl C1(CNC(c2[nH]cc3c2CCC3)=O)CN(C(=O)C(F)(F)CC2CC2)CCC1(F)F C1(N(C)CCNC(=O)NC2CC2C)C=CCC1 O=S(=O)(c1ccc(NC(c2ccc(F)cc2F)c2ncccn2)cc1Br)NCCF C(=O)(C(C)(C)C(C)C)NCC(C)(C1CCC1)NC(c1cc(CC)c(C)s1)=O C1(NCC2C(Cl)(Cl)C2)CCCCC1Cc1nc(-c2ccncc2)no1 Cn1cc(-c2nc(-c3cc[nH]n3)nn2C2CCSCC2)c(C(C)(C)C)n1 c1(-c2ccc(CN3C4CN(S(CCOC)(=O)=O)C(C4)C3)cc2)cccc([N+](=O)[O-])c1 CCCCC(C)(N=c1ccn(CCCC#N)[nH]1)c1nnnn1C1CCOC1 C1(CC(=O)NCCC2CCN(C(C3(CO)CC3(F)F)=O)CC2)CCC(=O)NC1 Cc1n[nH]c(=NC2=CC(NC(=O)C(N3CCCC(O)C3)C)C2)o1 C1(NC(C(C)NC(=O)NCCc2ccco2)=O)CCNC(=O)C1 c1(OC)cccc2[nH]c(C(=O)NCC3CC(NC(=O)C(C)c4ncco4)C3)cc12 c1(C(N2C(C)CC(NC(c3c(C)c(N)n(C)n3)=O)C2)=O)ccc2cncn2c1C c1(C(=O)NCC2CC(F)CN2C(c2cc(Br)n[nH]2)=O)csc2ccncc12 C1(CC(=O)NCCN(C(=O)CC=C(C)C)CC)CCN(C)C1=O C12CCN(CC1)C(=O)C2N1CCOCC1.C1(CNCCCC)CCCCO1 C1(OC)C(NC(C2(CNC(=O)C(c3ccn(C)n3)C)CCCC2)=O)CC12CCC2 N1(C(CCCOCC)=O)CC2(CCCCN(C(C3(Cl)CC3(F)F)=O)C2)C1 CC(C)(C(=O)NC1CCCCC1NC(=O)CCc1nc(C2CC2)no1)S(C)(=O)=O C1(NC(C(C(C)C)SC)=O)CCC2CCN(C(C3CC34CCSCC4)=O)C1C2 C1(C(=O)OCC)CN(C(c2cnc(Br)c(OCC)n2)=O)CCS1(=O)=O CC1(C)CC(=O)NC1CNC(=O)CNC(=O)C(F)n1ccnc1.C(=O)(C1=NOCC1)N CC1CCCC=C1C(=O)NC1C=CCN(C(=O)C2CC2)C1 C1(CN(C(=O)Cc2ccccc2C(F)(F)F)C)CCCCN1C(=O)CC1(C)CC1 C1(NC(C2N(C(c3c(C)n(C)cn3)=O)CSC2)=O)CC1C1CCCC1 C1(C(=O)NCCCCC#C)(NC(c2ccc(F)cc2)=O)CCN(C)C1 N1(C(COCCC=C)=O)CCCC(CCC)(NC(c2cccn2C)=O)C1 n1(CC(C)C#N)c(N2CC3CC2C3)nnc1C(C)(F)F C1(NC(c2ccncc2)C(=O)OC(C)C)CCCN(Cc2cccc(F)c2)C1 Cc1sc(C)c(C(=O)NCC2(NC(C34CC(F)C3C4)=O)CCOC2)c1C#N C(=O)(C#CC(C)(C)C)NC1CC(NC(C(C(C)C)c2cc(O)no2)=O)CC1O C=CC(F)(F)C(=O)NCCC(C)NC(C1C(CN=[N+]=[N-])C1(C)C)=O Cn1cncc1CCC(=O)NC1CCCC1NC(C1COCCO1)=O N1(C(CCC=CCC=C)=O)CC(OC(F)(F)F)C(NC(=O)C(C)NC(=O)NC)C1 Cc1ccc(C(N2CC3CC3(NC(C3(C4CCCO4)CC3)=O)C2)=O)cc1Cl c1(OC)ccc(Cl)cc1S(=O)(=O)N1CC2CCN(C(=O)OC(C)(C)C)C2C1 C(CN=c1cc(-c2ccccc2)nc[nH]1)NC(c1n(CC#C)ccc1)=O C1(C)(NC(CNC(=O)OCC)=O)CN2CCC1CC2.C(CC)(C=O)NC(=O)COC c1(OC(CC)C(=O)NC(C)(C)C(C)NC(=O)C(C)NC(=O)NC)cccc(C)c1 c1(C=O)ccc(-c2nncn2C)cc1.C1(C)(C(N(CCO)CC)=O)CCN1C(=O)OC N1(C(c2c(C)nc(COC)s2)=O)CCN(C(=O)CC(C)OC)CC1CO C1C(CC)(CNC(=O)OCC)C(=O)O1.C(C)(C)S N1(C(C=CCC)=O)CCN(C(c2coc(CO)c2)=O)CC1C(F)F C1(C)(C(N(C)CC2CC(O)C2)=O)COCCO1.c12cn(nn1)C1CN(C1)C2=O N1(C(C2(C=C)CCN(C(=O)CCn3cc(C)cn3)C2)=O)CCCC(C)(C)CC1 C(C(N=c1[nH]nc(CC)s1)C1CCC1)(OCC)Oc1ccc(C(F)(F)F)cc1 c1(C(=O)NCC(CCCC)NC(=O)C(C)SC(F)(F)F)nc(C)c(C)nc1C C1(CC)C(C(=O)NCCN2CC(C)(O)C2)CCN1C(=O)C=C1CCCCC1 CC1CCC(C(=O)NC2COCCC2O)CN1C(=O)Cc1cccc(F)c1 Cc1c(NCCC2CCCCO2)ncnc1NCCCCCF C#CCCCCC(=O)NCC1(OC)CCN(C(=O)CC2CCCN2CC)CC1 c1(C(C(=O)N(CCNC(CCc2onc(C)n2)=O)C(C)C)C)ccc(F)cc1 c1(C(N2C(C)CC(CNC(c3cccc(OC)n3)=O)C2)=O)ncc(Cl)cc1Cl C#CC1CCC(c2nc(-c3ccc(Cl)cc3)nn2C)CC1 N1(C(c2csc(C(C)=O)n2)=O)CC(C(N(CC(C)OC)CC)=O)OC(C)(C)C1 c1(CC)nc(C(F)(F)F)ccc1C(=O)NC1CC(c2nccn2C)C1 c1(C(C)C)ccc(C(=O)NCC2CN(C(=O)C(C)OCCN(C)C)CCO2)cc1 C1(CC)(CC)CN(C(c2ncc(C)cc2Br)C(=O)NC(C)CC)CCS1(=O)=O C1(CNC(c2c(OC)nsc2)=O)N(C(C2CC2F)=O)CCCC1(C)C C=CCC(CC(C)C)C(=O)N1CCN(C(=O)COCCF)CC1C1CCC1 c1(CNC(c2n(C)ccc2)=O)nc(CNC(C2C(C3CC3)C2(F)F)=O)cc(O)n1 Cc1cc(C)c(N2CC(C(=O)Nc3cc(I)ncn3)CC2=O)c(C)c1 N1(C(c2cc3n(n2)CC(F)C3)=O)CC2(CCCCN2C(=O)CC2CCC2)C1 Cc1cc(C(=O)OCC(c2ccc(O)c(Br)c2)O)ccc1OC(F)(F)F Cc1ccc(C)c(SCC(N2CC(NC(C3CCN(CC)CC3)=O)C(F)C2)=O)c1 N1(C(=O)NC2CN(c3c(C)cccc3)C2)CCc2sccc2C1c1ccc(Cl)cc1 c1(C(=O)NCC(C)(C(C)C)NC(C(C)SC)=O)cccn2nnnc12 c1(CCC(N2CC(O)(C(C)NC(C3CCCOC3)=O)C2)=O)cccc(N(C)C)n1 c1(C(N2CCC(OC)(CNC(c3ccoc3)=O)C2)=O)cc2c(F)cc(F)cc2[nH]1 C=CC(C)(CC)C(=O)N1CCC(OCCNC(c2cn(CCO)c(=O)nc2O)=O)C1 N1(C(CN(C(=O)OCC)C)=O)CCC(NC(=O)CCC2CCCCN2C)C(C)C1 C1(C(=O)NCCC2CCN(C(C(COC)N(C)C)=O)CC2)CCCCCN1C c1(C(=O)OC)ccc(C)nc1NC1CCN(C(c2cc(C)no2)=O)C1C CC1CCCCN1CC(=O)NC1C2CN(C(c3coc(Br)c3)=O)CC12 N1(C(c2cccc(CSC)c2)=O)CC(NC(=O)COC2CCCC2)CC(O)C1 C#Cc1cccc(C(=O)NCC(CO)NC(=O)C(c2cc(F)ccc2C)=O)c1Cl c1(CN(C(C(C)(C2CC2)OC)=O)C)ccccc1CNC(c1c(C)cnn1C)=O Cc1cnncc1CN(CCC(N1CCOCC1c1cn(CC(N)=O)nn1)=O)C c1(C(N2C(C)CCN(C(=O)C(F)OC(F)(F)F)CC2)=O)c[nH]c2cc(F)ccc12 Cc1nc2ccccn2c1C(=O)NC(C)(CNC(=O)C(C)C(C)(F)F)C1CCC1 N1(C(CCS(C)(=O)=O)=O)CCC2CCN(C(C3CCCC3O)=O)CC12 c1(C(=O)NCC2C(NC(CC(C=C)(C)O)=O)COC2)cccc2c1COCC2 c1(CC)cc(C(=O)N(CCCCCNC(=O)C(C)N2CCCC2)C)n(C)n1 Cc1ccc(-c2nc(C)sc2CC(=O)N(C)C)cc1.C12(CC1)C(=O)O2 c1(C(=O)NC2(C3N(C(CC4CC(OC)C4)=O)CCCC3)CC2)cc(Cl)c(F)c(Cl)c1 CS(=O)(=O)c1coc(C(N2C3CCC2CN(C(c2cc4scnc4[nH]2)=O)C3)=O)c1 C12(C(=O)NC(C)CC3CCN(C(C4(S(N)(=O)=O)CC4)=O)CC3)CCCC(CO1)C2 C1(C2CCC2)(C(=O)NCCNC(c2cc(C(N)=O)ncc2)=O)CCC1 C12(C(N3CCN(CC)C(C)C3)=O)CCCC1CCN2C(=O)CC(C)(C)C1CC1 Cc1nn(CC(N2CC(C)CCC2CNC(=O)CC(C)C)=O)c(C)c1Cl C1(CC(=O)N(C(C)(C)C)C2CC2)CCN(S(=O)(=O)CCc2ccno2)CC1 N1(C(C2CC(=O)NC(=O)C2)=O)CCC2CCCC12C(=O)NCc1nnc(O)o1 C1(C(N2CC(CNC(c3cn(CCC)nc3C)=O)C2)=O)CCc2[nH]nc(O)c2C1 c1(OC)ccc(CC(=O)NCCCn2cc(C(C)C(=O)O)nn2)cc1O c1(C(N(CCOC)CCNC(C2CC23CCOC3)=O)=O)cnc(C)nc1C C1(C(=O)NC2CC(F)(F)C2)C2CN(CC(N3CCC(O)C3)=O)CC12 N1(CC(=O)NCc2scc(CO)n2)CCC(CNC(C2C3CCCCC23)=O)CC1 c1(NCC2C(C(N(C)C3CC3)=O)CCC2)ccc(-c2ncco2)cc1F c1(C(=O)NC(CC)CNC(=O)CCC2CCC(=O)N2)cncc2[nH]ccc12 C(=O)(C(F)(F)CC(C)C)NCC(CC=C)NC(C1CC1Cc1ccccc1)=O C(=O)(C(CC(=O)O)c1ccc(Br)cc1)n1cc(C2OCCNC2)nn1.CC1(C(O)Br)CCC1 C1(C(N2CCC(NC(c3cc(C)on3)=O)C(O)C2)=O)CC(O)c2ccccc2O1 c1(NC(=O)NCC23CC(C(=O)OC)(C2)C3)c(Cl)c(F)nc(F)c1Cl c1(NC(c2nc(-c3c(C)ccc(OC)c3)sc2C)=O)ccc2scnc2c1 n1(CC(=O)NC2(C(F)F)CC(NC(C(C)(C)OC)=O)C2)c(O)nc2ccccc12 C1(C(=O)NCC2CCCN(C)C2)CCN(C(c2cccc(CO)c2)=O)C12CC2 Cc1ccc(C(N2CCN(C(C3CCC(F)(F)C3)=O)C3CC23)=O)cc1O O=C(C1=CCCCO1)NC1CN(C(=O)C(CO)c2ccccc2)CC1O Cc1ccccc1C(=O)N(CCCN(C(=O)CCC1CC12CC2)C)C C1(CC(C)CNC(=O)C#CC2CC2)CCN(C(=O)Cc2cc[nH]n2)CC1 c1(NC(=O)CC2CCCN(C(=O)CC3CCOC3=O)C2)cccc(F)c1F CCC(C(=O)NC1CC(C(F)C(=O)N(C)Cc2cncn2C)C1)OC C12(NC(c3c(Cl)cncc3Cl)=O)CCCC1N(C(=O)CC1CC1)CCC2 c1(C(N2CC3C(CNC(C(CC)=CC)=O)(C3)C2)=O)cc(C)c(Cl)c(C)c1 C1(C(N2C(C(=O)Nc3cc(O)nc(O)n3)CCC2)=O)CCc2nc[nH]c2C1 c1(N2CC3(C(NC(C4CC45CC5)=O)CCS3)C2)c(Cl)cncc1[N+](=O)[O-] CC1CN(C(=O)CC2CCCC2)CCC1N1CCCC1.C1(=O)CCCCCN1 N1(C(CCN(C(c2c(C)cnn2C)=O)CC2CC2)=O)CC(O)CC1(C)C C(=O)(C(=O)C(F)(F)F)NCC1CCN(C(C(C)CC2CCC2)=O)CC1 c1(C(N2C(C)C(NC(c3n[nH]cc3Cl)=O)CCC2)=O)cc([N+](=O)[O-])ccc1O c1(C(N2CCN(C(C3CCCCN3C3CC3)=O)CC2)=O)cnn2c1OCCC2 C1(C(=O)NC(COC)CNC(C2CC(OC)C(OC)C2)=O)CCn2c(O)nnc2C1 C1(NC(c2nnc(C)s2)=O)CCCC2CN(C(=O)C(c3ccccc3Cl)C)CC12 C12(NC(C(CC)F)=O)CCC(C1)N(C(c1ccc(F)cc1OC(F)F)=O)C2.C(C)(=O)O c1(NC(=O)NC(C)(CN)C2CC2)ccc2cccnc2c1 N1(C(c2cc(C)sn2)=O)CC(C(=O)Nc2cccnc2C)C(C2CC2)C1 C1(CCNC(=O)NC(c2cnn(-c3cccnc3)c2)C)COCC2(CCC2)O1 C#CC1(O)CCN(C(=O)C=CC2CCN(C(=O)C(CO)C(C)(C)C)CC2)C1 c1(C(=O)OC)ccc(NCCCNC(=O)CC2CC3(CCC3)CO2)c([N+](=O)[O-])c1 c1(C(N2CC(OCC)C(CNC(=O)Cn3cncn3)C2)=O)ccc(F)c(C)c1C N1(C(c2ccc(C#C)o2)=O)CC(F)(F)CC1C(=O)NC1(C)C(C)(C)C1(C)C c1(C(=O)NCC(C)(C2CCC2)NC(=O)CCS(C)(=O)=O)cccc2[nH]nc(O)c12 c1(C(CC)NCC2CC(=O)N(C)C2)cc(Cl)ccc1OC CC(C)(O)C(=O)NCCN(C1CCCCC1)C(c1ccsc1)=O c1(OC)nccnc1CSCc1cc(F)ccn1 O=C1NCC2(CCN(C(=O)CC3(NC(C4CC(CF)C4)=O)CCCCC3)C2)O1 N1(CCOCC)CCC(N=c2[nH]c(=N)[nH]c(=NCCCc3nc[nH]n3)[nH]2)CC1 N1(C(C(C)SCCCC)=O)CCCC(NC(C2CCOC(CC)C2)=O)C1 C1(CNC(C2=CCC(C)CC2)=O)CN(C(c2cc(Cl)ns2)=O)C2COCC2O1 N#Cc1cn(CC(N2CCCC23CCN(C(=O)C2=CCCC2)C3)=O)c(=O)nc1O c1(CC)cc(Cl)ccc1NC(C1(O)CCN(C(c2ccc(Cl)s2)=O)C1)=O C(=O)(C(C)C(F)(F)C(F)F)N1CCC(C(C)NC(C2(CC#C)CCOCC2)=O)C1 C1(NC(c2c(CC)nns2)=O)CCN(C(C2(N=[N+]=[N-])CC2)=O)CC1CC N1(C(CCOC)=O)CC(C)CCC1C(=O)N(C)CCc1cnn(C)c1 c1(C(=O)NCCN(CCC)C(c2cc(C3CCOC3)[nH]n2)=O)cn(CC2CC2)nn1 c1(C(C)OCC)nc(C(=O)NC2(C)CC(NC(c3snnc3C)=O)C2)cs1 C(c1ccc(C(N)=O)cc1)=CC(=O)N(CCCNC(C1C2CCC(=O)C12)=O)CC c1(C(=O)NC(C(C)N(C)C)C(=O)N2CCCC2)ncc(F)cc1N.C1(NC)(CO)CC1 C(=O)(CS(=O)(=O)CC(=O)NCC1CC(CNC(C23COCC2C3)=O)C1)OC N1(C(Cc2cnc(C)[nH]2)=O)CCCC(C)C1CCNC(=O)Cc1ccncn1 C1(NC(c2c(C)scc2)=O)C(CNC(c2cc(C(N)=O)[nH]n2)=O)CCC12CCC2 c1(OC)sc(C(=O)NCC2CC2CNC(c2ccnc(C)c2)=O)cc1Br N1(C(c2c(C(C)C)c[nH]c2)=O)CCCCC(N(C)C(c2cn(C)nn2)=O)C1 c1(C(C)(C)C(=O)NC2COCCN(c3ncc(C#N)s3)C2)csc2c1CCCC2 C1(NC(c2c(CC(N)=O)occ2)=O)CCCCCN(C(c2nc(Cl)sc2Cl)=O)C1 c1(C(=O)NCC(C)NC(C2C(COC)C2)=O)ccc(F)c(N)c1 c1(CNC(C2(COC)CC2)=O)ncccc1CNC(c1cnccc1C)=O N1(C(C(CC(N)=O)C(=O)OC(C)(C)C)=O)CCOc2ccc(Br)cc2CC1=O N1(C(CN(S(CC)(=O)=O)C)=O)CCOC2(CCCN(C(C3CCC=CO3)=O)C2)C1 Cc1cc(=NC(=O)C2CCN(Cc3cc(Br)ccc3F)CC2O)[nH]c(Cl)n1 Cc1ncc(CC(=O)NC(C2(C(=O)NCC3CCCN3C)CC2)C)s1 C(=O)(CCC1=CCCCC1)N1CC(C#C)(C(N2CCc3c[nH]nc3C2)=O)C1 C(CCCCC(=O)N1CCC(NC(c2csc(C(F)F)c2)=O)C1)OCC S(=O)(=O)(CC(=O)NCC(O)C(N1CC=CC(O)C1)=O)NC c1(C(N(C)CC2N(C(C3C(=C)CC3)=O)CCOC2)=O)cc(C)c(Br)cn1 CC1C(C)N(C(c2cc(Cl)nc(=N)[nH]2)=O)CCN1C(=O)CSc1ccc(Cl)cc1 C1(N(C(=O)CC2(OC)CCC2)CC)CN(C(c2cc(=O)cc[nH]2)=O)CC12CC2 C1(CNC(c2c(OC)nsc2)=O)COCCN1C(=O)CC(C)c1ccco1 N1(C(C2C(C)CC(C(F)(F)F)CC2)=O)CCCC2(CCN(C(=O)C(F)F)CC2)C1 c1(OC)ccc(O)cc1C(N1CC(O)(CNC(c2csc(Cl)c2Cl)=O)C1)=O c1(N2CCCC(CNC(c3cc(CC)cc(F)c3)=O)C2)ccc([N+](=O)[O-])cc1F CCC(C(=O)N1CC(NC(c2cnn(CC(=O)NC(C)C)c2)=O)C1)C(C)C C(C(C(=O)N1CCOCC1)NC(=O)C(n1ccnc1C)C)SCC.N C1(CCNC2(c3nnnn3C(C)C)CC(CC(C)C)C2)CCC(C)(C)C1 N1(C(c2cc(COC)n(C)n2)=O)CC2CN(C(c3cccc(CO)c3)=O)C2C1 CC(C(=O)NCC1CC2CCC1N2C(C1CCC(=O)N1C)=O)C(C)(F)F C(=O)(C(C)(C)O)NC(C)CCN(C(=O)Cc1ccoc1)C1CC1 N1(C(=O)C=Cc2cnn(CCF)c2)CCN(C(=O)CC2CC2)C(c2cccnc2)C1 c1(C(=O)NC(c2cccc(C)c2)CNC(c2occc2F)=O)ccc(F)cc1C c1(CC(=O)NCCCN2CCN(C(C)C)CC2)ccc(C#N)cc1 C1(OC)COCC1n1cc(C(=O)NCCC(C)NC(c2ccnn2C)=O)nn1 c1(C(=O)NCC(C)CNC(c2cn(C)c(O)n2)=O)cc(Cl)cc(F)c1N Cc1cc2c(C(N3CCCC(CO)(NC(c4cnns4)=O)C3)=O)ccc(C)c2[nH]1 C1(C(=O)NC2(COC)CN(C(C3CCC3(C)C)=O)C2)COC2(CCC2)C1 c1(CNC(CNC(C)=O)=O)ncccc1C(=O)N(C1CC(O)C1(C)C)C c1(CC)nocc1C(=O)NCC=CC(=O)N(C(C)CC(N)=O)C C1(C(=O)NCCCCNC(c2ncc(Br)s2)=O)CCCC(F)(F)C1 N1(C(C2CC(=C)CN2CC)=O)CCC(O)C(C)(C(=O)Nc2cc(Br)ccc2C#N)C1 C1(CCNC(c2c(CNC(C3CCN(C)CC3)=O)ocn2)=O)CCC(C)(C)CO1 c1(C(CC)C)ccc(C#N)c(N2CCC(N(C(=O)C(C)Cc3ccco3)C)C2)n1 c12ccccc1C(C(=O)NCCO)N(C)CCCCCOCC2.C1(S)CC1.C1(CC)CC1 N1(C(C2(OC)CC2)=O)CCC(C(F)(F)F)C(NC(=O)C=CC2CCC2)C1 CS(=O)CCC(O)C(=O)NC1C2CC1N(C(=O)Cn1nc3c(n1)CCCC3)C2 N1(C(c2c(C)scn2)=O)CC(CNC(c2cc(CO)c(C)o2)=O)C2(CCC2)C1 CS(=O)(=O)c1cccc(S(=O)(=O)N2CC(O)CC2c2cccc(Br)c2)c1 CC1(C(=O)OCc2ccc(-n3cccn3)cc2)CCNC1=O C1(C)(C(N2CC(CC)C(CNC(C3CCC(=O)N3)=O)CC2)=O)CC(C)OC(C)C1 C1(NC(CCSCC(N)=O)=O)CC=CCC1C(=O)NCC1(C(F)F)CCCO1 N1(C(=O)C=Cc2cccc(F)c2)CCN(C(=O)CN2CC=CC2)CC(CO)C1 C(=O)(CCCCCC#N)N1CCC(CC)C1C(N1CCCC(C)(O)C1)=O c1(C(N(C2CN(C(C3CCSCC3)=O)C2)C)=O)cccc(Cn2cncn2)c1 Cc1nc(CC(=O)N(CC(O)CNC(=O)CSCCCc2ccccc2)C)cs1 c1(CC(=O)NCC(C)NC(c2c(CC)ccs2)=O)cc(Br)c2c(c1)CCO2 C(=O)(C(F)(F)C(F)F)NC1CN(C(C(CC=C)N(C)C)=O)CC1F O=C(C(O)C(F)(F)F)NCCc1cccc(-c2cc[nH]n2)c1 N1(N2C(N(C(CC=CC=C)=O)C=O)CC2)CCCC(CCCCC)CC1.OC Cc1noc2ncnc(N3CCCC(C(C)NC(=O)CC(O)CN(C)C)C3)c12 C1(OC)CCCC1C(=O)NCC(C)N(C)C(C1CC(C)(C)C1)=O c1(CCNC(C(=O)NC(C)CC2(C)OCCO2)=O)nc(Br)cs1 C1(C(=O)NCC2CCC(NC(C(C)OCCN(C)C)=O)C2)COC2COCC12 CC1CCN(C(C2CC23CC3)=O)C(CNC(=O)Cn2cc(C3CCC3)nn2)C1 C(=O)(CC(CC1CC1)NC(=O)CN(C1CCSC1)C)N(c1ccc(O)cc1)CC CCC(C)C(O)C(=O)Nc1cccc(NC(=O)CN2CCCC2)c1 c1(C(=O)NCc2c(C(=O)OC)cccn2)cc(F)c(Cl)cc1F.C12CCCN1C2=O Cc1nc(C(C)C)nc(O)c1C(=O)NC(CCNC(=O)C(C)C1CCC1)C(C)C Cc1nc2c([nH]1)CC(NC(c1ccccc1I)c1nnnn1C1CCC1)CC2 Cc1c[nH]c(C(=O)NCC2(C(=O)NC3CC(CC(N)=O)C3)CCCO2)c1C c1(CNC(C2CC3(C2)CN(Cc2cccnc2)C3)=O)cc(Br)cc(Cl)c1F C(C)(C(CC(=O)NCC1CCOC1C)NC(C1CCC1C(F)F)=O)OC N1(C(COC(CC)(C)C)=O)CC(N(C(=O)CN2CCC(O)CC2)C)C(O)C1 C(=O)(CCC(N)=O)NCC1(NC(c2n(C(CC)C)ncc2)=O)CCOC1 N12CCC(C(C)C1)C2=O.N1(CC2CN(CC)C2)CCN(c2ccc(F)cn2)CC1 c1(CNC(C2(C)CCN(C(=O)CC3CCCOC3=O)C2)=O)ccc2c(c1)CC2 N1(C(c2c(OC)scc2)=O)CC2(NC(C3OCCC3C)=O)CCCC2(F)C1 C1(CN(C(=O)C(N2CCCC(F)CC2)=O)C2CC2)CCC2(CCCCCC2)O1 N1(C(CC2(CNC(CCC)=O)CC2)=O)CCC(CC2CC2)C1 CS(=O)c1ccc(C(=O)NCC2CC2NC(c2ccc(C3CC3)s2)=O)cc1 C=C(C)CC(C(=O)NC)N1CCC(C)C1C.c12ccccc1S2 C(=O)(C=C1SCC(=O)N1C)N1C(CC)CN(C(=O)C2=CC3(CCOC3)C2)CC1 c1(OCC(=O)NCC2C(NC(c3ccc(C)cn3)=O)CC2)ccccc1[N+](=O)[O-] N1(C(c2c(CNC(C(C(C)C)C3CC3)=O)cc[nH]2)=O)CC(CO)CC1(C)C c1(CC(=O)N(CC(CNC(C(CC)C)=O)(C)C)C)c[nH]c2cc(F)ccc12 c1(CCC(=O)NCC2CC(CNC(C=CCCC)=O)OC2)ccc(O)cc1 C1(C)(C(=O)NCC(n2cc(C3(C)CCCC3)nn2)C)CCCS1 N1(C(=O)C=CC2CCCCCC2)CC2CCN(C(C3C=CCCC3)=O)C2C1 Cc1cc(C(=O)N(C)CCOCCCNC(C2CC(OC(F)(F)F)C2)=O)sn1 c1(C(N2CCN(C(n3ccccc3=O)C)C3C2C3)=O)ccc2oc(O)nc2n1 c1(C(=O)NCCCOCCCNC(C(C(C)(C)O)F)=O)cn2cccnc2n1 Cc1cc(C(=O)NCC(C)CC(=O)NC2CC3CC3C2)nc(O)c1 n1(CCC(=O)NCCN(C(=O)CC2CCC3CC23)C)cc([N+](=O)[O-])cn1 N(C(=NCCC(C)C)NC1CC1(C)C)CC.C=C1C2C1C(=O)NC2=O c1(C(=O)NCC2CC(OC)CN2C(c2ccc(C)s2)=O)cc(C)c(C)c(F)c1 C=CCCCCCC(=O)N1CCN(CC=C(Br)C)CC1 N1(CCOCCOCCn2cc(CNC(C=C(C)C)=O)nn2)CC2CCC1C2 N1(C(C(c2cccc(C)c2)O)=O)C2CCC1CC(O)(CNC(=O)CCF)C2 c1(OC)ccccc1NC(=O)COC(CNC(c1snnc1C)=O)CO C1(C)(OCCC)CCCN(C(=O)CN(C(=O)Cc2ccc[nH]2)C)C1 C1(C(=O)NC2(CNC(c3c(C)cns3)=O)CCCCC2)CCCCN1S(N)(=O)=O CC1=C(C)CC(C)(NC(=O)CNC(c2ccc(C#N)n2C)=O)CC1 C(=O)(CC(C)C(C)(C)C)N1CCC(C=C)(C(=O)NCC(c2cnc[nH]2)C)C1 C1(C2CCN(Cn3nc(C(C)C)oc3=S)CC2)(c2n(CC)ccn2)CCOCC1 N(C(=NC)N1CCC(Oc2ccccc2)CC1)CC1CC(CCC)NC1 C1(CCNC(COCc2cccc(OC)c2)=O)CN(c2nncs2)CC(C)(C)O1 C(CC)(CC)(CCNC(=O)C(F)CC1CC1)NC(C(CCC)c1ccccc1)=O Cc1cc(F)sc1C(=O)NC(C)C(=O)NCC1CC12CCC2 CC(C)C(O)C(=O)Nc1ccc(C2CC2)cc1.C1C(C)NCCO1 c1(CC)cccc(C(N2CC(NC(=O)CCc3ccc(Cl)cc3)C(O)C2)=O)c1 C(C(=O)N=c1[nH]oc2ncccc12)C1C2CN(C(CCSC)=O)C1C2 C1(c2ccc(C)cc2)NC(=O)N(CCCNC(c2nnnn2C)=O)C1=O c1(NC(C2(F)CCCN(C(c3c(C)c[nH]c3)=O)C2)=O)ccnc2c1ccn2C c1(C(=O)NC(C)CN(C(=O)CC2C=CCC2)C)ccc(C(=O)OC(C)(C)C)cc1 C12(C(=O)NCC(CO)NC(Cc3cccc(OC)c3)=O)CC=CCN1CCC2 CC1CCN2C(C)C1NC(=O)CCC2=O.c1(C=O)cccc2c1CCO2.C1CC1 C1(C(=O)OC)C2CCC1CN(C(=O)CNC(=O)Nc1cc(Cl)cc(Cl)c1)C2 c1(C(=O)NC(CC)(CNC(c2cc(C)cc(C)n2)=O)CC)cc(C)nc(Cl)c1N C1(OC)(CO)CCCC(C)C1.c12oc(cc1C)C(=O)N(C)CCNC2=O C=C(C)C(CC(=O)NCCN1CC(CC(=O)NCCO)N(C)CC1)OC.O(C)CC CN(CCCC(=O)NCC1CC1NC(=O)Cc1cc2ccccc2o1)N=O C1(C(=O)Nc2ccc(SC)nc2)(CC)CCCN(C(c2ccn(C)c2)=O)C1 CC(F)(F)C(F)C(=O)N1CC=CCC1C(=O)NCC1Cc2nccn2C1 N1(C(C2CCN2C(c2cc(F)c(F)c(Cl)c2)=O)=O)Cc2ccc(F)cc2C1 C1(CC(=O)NCC(CC)NC(c2ccc(OC)c(C)c2)=O)CCCC2(CCC2)O1 c1(C(=O)NC23C(CN(C(CC(C)F)=O)C2)C3)cc(N)c(Cl)cn1 N1(C(=O)NCCC(CCC)C)CC(C(=O)O)C2(CC2)C1 N1(C(CN(C(C(C)C)=O)C)=O)CCC(C)(NC(C2(C(C)C)CCCO2)=O)C1 C1(NC(C(CCC)CC)=O)CCN(C(C2CC3(CCCCC3)C2)=O)CC(O)C1 CC(CCN=c1ccc(Br)c(S(=O)(=O)NC)[nH]1)N(C)C.CC(O)C1CCC1 O=C(C1=C2CCN=C2NC=C1)NCCN(C(C1CCCCC1)=O)Cc1ccsc1 C1(C)(C(=O)NCC2(C(=O)NC(C#C)CC3CCC3)CC(=C)C2)CCCC1O N(C(=NCC(C)(C)CC1CCOC1)NCC1CC1)C(c1ccc(Cl)c(F)c1)C N1(C(c2cc(C)[nH]c2)=O)CCCC(C(=O)NCCc2cc(C)ns2)CC1 C(=O)(C1=C(C#N)CCC1)NC(CC)CN(C(=O)C(c1ccc(F)cc1)(F)F)CC C1(C(=O)NCCN(C)C(c2cccc3c2OCCO3)=O)Cc2c(F)cccc2O1 C1(NC(C2CCCN2C(=O)Cc2ccc[nH]2)=O)(CO)CCCCC1 N1(C(COCCCC)=O)CCC(C2CC2)C1CNC(c1cncn1C(F)(F)F)=O Cc1c(C(C)C)cc(C(N2CCN(C(=O)CCCC#N)C3CCC23)=O)cc1[N+](=O)[O-] Cc1cc(NC(=O)C(C)(C2CC2)N(C)C(c2ccc(F)cc2)=O)cnc1C c1(CCC)sc(C(N2CC(CNC(=O)CC(C)O)C(O)C2)=O)cc1Br N1(C(C2(C=C)CCCC2)=O)CCCC(CCC)(CNC(=O)CCOCC(C)C)C1 c1(N2CC3N(C)C(CCC3)C2)nc(=NCC2(N(C)C)CC2)[nH]c2c1COC2 c1(C(=O)NCC(C)CNC(C2C(F)(F)C23CC3)=O)cnn(C(C)(C)C)c1Cl C1(C(CSCC)(C)C)CCN(C(=O)CCOC2CC2)CC1.C12CCCC1NC2=O c1(C(=O)OCC)c(N2CCCC(NC(=O)CC3(O)CCCC3)C2)cc(C)nc1O CCCCC(=O)C(=O)NC(C1(CNC(=O)C(CO)N(C)C)CC1)C N1(C(C2CC(SC)C2)=O)CC2CC(NC(=O)C(C)(O)C3CC3)C(C2)C1 c1(CNC(C2CCCN(C(=O)CSC3CC3)C2)c2cc(C)no2)ccsc1[N+](=O)[O-] N1(C(c2cc(C)oc2C)=O)CC2CCC1C(CNC(C1CC1F)=O)C2 C12(C(N(c3cccn3C)CCNC(C)=O)=O)CC3CC(C1)CC(O)(C3)C2 c1(C(=O)OC)ccc2[nH]c(C(=O)NCCNc3c(C)cc(C)cc3C)cc2c1 Cc1cc(C)c(CC(=O)NCCC2CC(NC(=O)COc3cccnc3)C2)s1 C1(c2cn(CCC3CN(C(C4OCC(C)C4)=O)C3)nn2)CCCC(F)(F)C1 CCC(CCC(=O)N1CC(CCOC)C1)NC(=O)Cn1cnnc1O N1(C(c2c(OC)cnnc2)=O)CCCC(CC(N2CCC2C)=O)CC1 NS(=O)(=O)CCCC(=O)N1CCC(O)C(NC(=O)C(O)c2ccsc2)C1 CCC(CCCC(=O)O)NC(=O)COCc1cn(C2CCC(C3CC3)C2)nn1 Cc1cn(C)nc1C(=O)NC1(C(=O)NC(C(N)=O)C2CCCC2)CC1C Cn1[nH]c(=NC(=O)CC2CC(O)CN2C(=O)C(c2ccccc2)F)cc1C1CC1 N1(C(CC2(C)OCCO2)=O)CCC(CO)(NC(=O)Cc2cc(C3CC3)no2)C1 Cc1ccc(C(N2CCN(C(c3cn(CCC4CC4)nn3)C3CC3)CC2)C)cc1 Cc1cc(C(=O)NC(C)CC(C)NC(=O)Cn2ncnn2)c2c(c1)CCCN2 CCC(C)C(O)C(C)C(=O)N1CCOC(CN(CC(=O)NC)C2CC2)C1 c1(C(=O)NC2(CNC(CCCC(=O)OC)=O)CCOCC2)cccc2c1CCC2 Cc1ccc(Cl)cc1C(=O)NC1(CNC(C2CCN(CC(C)C)C2)=O)CCCC1 N1(C(c2n(C)nc(CC)c2Cl)=O)CCCC(C2CCCN(C(=O)C(O)CC)C2)C1 c1(C(N2CC(OC)C(NC(c3ccnnc3)=O)C2)=O)n[nH]c(C(C)C)c1[N+](=O)[O-] C=CCCC(F)(F)C(=O)N1CCC1(C)CC(=O)NCCN1CCCC(O)C1 c1(C(C(N)=O)=O)ccc(CNN2CCN(C(=O)CCCCC3CC3)CC2)cc1 N1(C(Cc2ncc(C)o2)=O)CCC(CNC(=O)C(C)NS(C)(=O)=O)C(C)C1 C1(NC(C(=O)NCCNC(c2ccc(SCC)c(Br)c2)=O)=O)CCCCC(F)(F)C1 c1(C(N2CCC(F)(CNC(C3(CF)CCC3)=O)C2)=O)cccnc1F C=CCCCC(C)(C)C(=O)N1CC2CCC(C1)N2C(c1c(C)cc(C)nc1O)=O C1(C)(CNC(C2C(CC)CCC2)=O)COCCN(C(C2(C3CC3)CC2)=O)C1 c1(CN(C2CC2)CC2N(C(C=COCC)=O)CCCC2)ccc2ccccc2c1 C(=O)(CC(F)(F)C(C)C)N1CCCC(n2c(CCC)ncc2)C1 C1(CCNC(c2ccc(C3CCCCC3)o2)=O)CN(C(c2cccs2)=O)CCO1 CC(CS(C)(=O)=O)C(=O)N1CC(O)(CN(C)C(C2(CO)CCOCC2)=O)C1 c1(C(N2C3CC(NC(CSCCCC)=O)C3CC2)=O)nnc2ccccc2c1N C1(CNC(C(COCC)C)=O)CN(C(c2ccccc2OC(C)CC)=O)CCN1C c1(C(N2CC(NC(CC3(C)CC3(F)F)=O)C2)=O)ccc(C(=O)CF)cc1 c1(C(N2CCC(OCCNC(C(C)n3cncn3)=O)C2)=O)cc(C2CC2)nn1C c1(C(=O)NCC2C(N(C)C(C3CCN(C)C3=O)=O)CCC2)cc2n(n1)CCC2 Cc1nc(N2CC3CCCC(NC(c4cc(Cl)sc4Cl)=O)C3C2)ccc1[N+](=O)[O-] N1(C(CN(C(C(C)C)=O)C)=O)CCC2CN(C(=O)CN3CCN(C)C(=O)C3)C2C1 C1(C2CC(=O)NC2)CC(NC(=O)COC2CC(F)(F)C2)CCO1 CC1(C)COCC1CC(=O)NCC1(NC(=O)CC2CCCC2)CCCCC1 CCC(C)(CNC(C1CCC(=O)O1)=O)C(=O)N(C)Cc1nnc(O)o1 C1(CC(=O)NC(C2CN(C(C3C4CCC(=O)C34)=O)CCO2)C)CC2(CCC2)C1 c1(OC)cc(C(N2CCC(F)(CNC(c3cnn(C)c3)=O)C2)=O)c(F)cn1 c1(NC(=O)C2CC2)ccc(C2CCN(Cc3cccc(F)c3)CC2)nc1 CCC(CC(F)F)C(=O)NC1CN(C(C2(CC3CC3)CC2)=O)CC1O C(CC(C)(C)CC(=O)Oc1cc([N+](=O)[O-])sn1)OCC C1(C(=O)NC2CC(CC(=O)NC(CC(C)O)C)C2)CCC(C)(C)OC1 c1(CCOCC)nc(=NCC2(O)CCCN(C(=O)C(C)=C(C)C)C2)s[nH]1 Cc1cc(C)c(CC(=O)NCCCCCN(C(=O)CCC(F)F)C)c(C)c1 C1(C(=O)NCC2CCC(C(=O)Nc3ccc(OC)nc3)O2)CCOC(=O)CC1 Cc1cccc(CC(=O)N(C(C)CCNC(C2(S(C)(=O)=O)CC2)=O)C)c1Br Cc1ncc2cc(C(=O)NC(C)CC(C)NC(C3(O)CC(C)(C)C3)=O)ccn12 N1(Cc2ccc(C#N)cn2)C2CCC1CC(NC(c1ccc(I)c(F)c1F)=O)C2 c1(OCC)cccc2[nH]c(C(=O)N(C3CCN(c4ccc(C)cc4)C3=O)C)cc12 N1(C(C(=Cc2cn[nH]c2)C)=O)CCOC(CCNC(=O)CC2CCC(=O)N2)C1 C(=O)(CCCCCC(=O)NCCCN(C(=O)Cc1ncoc1C)CC)NCCC C(CC(C(C)(C)C)NC(C1CC1c1ccco1)=O)N(C(C(C=C)(C)C)=O)C C1(=CC(=O)N)CN2CCC1CC2.C1(OC)CN(C(=O)COCCF)CC1CNC(N)=O C(CCC)(C(=O)NC1CCC(OCC)C1)NC(CSCCCC)=O C(=O)(C1CCCc2n[nH]cc21)N(CC(C)CNC(=O)Cc1cccnc1Cl)C c1(N2CCN(Cc3c(C)nn(C)c3Cl)CC2CC#N)nc2ccccn2n1 Cc1nc(C)c(C(=O)N(CC(=O)N(CC(O)CN(C)C)C)CC2CC2)o1 c1(C(CC)=O)ccc(NCC(c2cccs2)NC(C2CCC(=O)N2)=O)c([N+](=O)[O-])c1 C=CCC(CC)C(=O)Nc1cc(C2CC3(C(C(=O)OC)C3)C2)cc(F)c1 c1(OC)ncccc1C(N(C)Cc1cccc[n+]1[O-])=O c1(C(C(=O)NCCCCNC(CC2CC(=C)C2)=O)=O)cc(Br)cs1 CCC(C)C(O)CC(=O)NC1(CNC(=O)CNS(=O)(=O)c2cccnc2)CCC1 CC1C(C(=O)NCCN2CCN(C(=O)CS(=O)(=O)N3CCCCC3)CC2)CCN1C C(C(CC(C)C)C(=O)NCc1ccc(C(=O)NC(C2CCCO2)C)nc1)OC c1(C(=O)NC(C#C)C2CC2)occc1CNC(=O)CSc1cccs1 N1(C(CCCCCCC)=O)CCC2(CC1)CC(NC(C1C3CCC13)=O)CO2 c1(C(N2CC3(N(C(c4nc(C)oc4C)=O)CC3)C2)=O)cc(F)cc(Br)c1F C(C(=O)N1CC(O)(C2CCCN2C(=O)COCC2CC2)C1)(C(C)(C)C)NC(C)=O CC(CCC(=O)N1CCC(CNC(=O)Cc2cncnc2)C12CC2)S(C)(=O)=O C1(C)(CC)CN(C(c2ccnn2C)C(=O)Nc2ccc(F)cc2C)CCO1 CCCC(C(=O)N1CCN(c2nc(C(N3CCOCC3)=O)c(C)s2)CC1)N(C)C C1(CNC(CCCC(C)=O)=O)COC(C)(C)CN1C(=O)CC1CCOC1=O c1(CN2CC2=O)cnc(Cl)c2ccccc12.n1(CCOC)cc(C(=O)OC)c(C)n1 N1(C(CCC2(NC(=O)CCc3ccsc3)CCC2)=O)CC(O)(C2CCC2)C1 C(=O)(C(CC1CCCC1)NC(=O)CC(C)C1CC1)NC1(COC)CC1 c1(NC(C2C(NC(c3ccc(N4CCCC4=O)cc3)=O)C2)=O)ccnc2ncnn12 N1(C(Cc2nc(C)oc2)=O)CC(CCNC(C2CCC(C(N)=O)CC2)=O)C(C)C1 N1(C(CC(C)F)=O)CCC(O)(C2(NC(=O)CC34CCC(CC3)C4)CC2)CC1 CC1(C)CCC(CC(=O)NCC(CNC(=O)CCNc2ccccc2)CO)OC1 Cc1cnc(C(N2CCOCC2CNC(=O)CCS(C)(=O)=O)=O)c(C)c1 N1(C(C(COC)(C)C)=O)CCCC(CO)(CNC(=O)CCC2(C)CC2(F)F)C1 C1(NC(c2cscc2F)=O)CC2CCC1CN(C(=O)C1CCc3c[nH]nc31)C2 N1(C(C(C2CCCCC2)C)=O)CC2CC(NC(c3ccc(Cl)s3)=O)CC1C2 c1(OC)cnc[nH]c1=NC(=O)c1ncccc1OC(=O)C=C1CCNCC1 C(=O)(C(C)(C)C(=O)N1CCC(F)(C(=O)NC(CC)C(C)(C)O)C1)NC n1(CC)nnc2c1CCC(C(=O)Nc1ncoc1CCCSc1ccccc1)C2 Cc1cc2nc(NC(=O)Cn3cnc4sccc4c3=O)sc2cc1C O=C(C1CCc2ccccc21)NCCC1CSCCN1c1nc2c(F)cccc2o1 c1(N2CCC(C(C)(C)C)C2)nc(NCCc2cccc(F)c2Br)c2ccsc2n1 n1(CC(=O)NCC2CC(NC(C(CCCC)O)=O)C2)ncc2ncccc12 N1(C(c2[nH]cc(C)c2)=O)CC(NC(C2SCCS2)=O)CCC1C C(C(F)(F)C(=O)N1CCOCC1)Oc1ccc(C(C)=O)cn1 N1(C(c2c(C)cn(C)n2)=O)CC2CC1CCC2NC(c1c[nH]nc1C(C)(C)C)=O Cc1cnc(C(N2CC(NC(C3CC4(CC4)CO3)=O)CC23CCC3)=O)cc1C#N N1(C(=O)NCC(C)Cc2ccc(Br)cc2)CCOC2C(C(F)(F)F)CC12 c1(C(N(CC2N(C(CSCC)=O)CCC2)CC)=O)nc2ncc(C)cn2n1 N1(C(c2ccc(-c3cnc4n3CCC4)cc2)=O)CCC2Cc3cccc1c3CC2 Nc1cc(F)c(O)cc1C(=O)NCC1(CNC(C2CCC(O)C2)=O)CCCC1 C1(NC(C(C)OC)=O)COC2(C1)CN(C(c1c(N)cccc1F)=O)C2 N1(CC)CCOC(C(=O)NC(C2CN(C(=O)CCC3CCCC(=O)N3)C2)C)C1 C1(C(N(CC#C)Cc2ccco2)=O)CCN(C(=O)C(F)C(C)(F)F)CCO1 Cc1ccc(C(N2CCN(C(CNC(=O)CSC(=N)N)C(F)F)CC2)=O)cn1 c1(NCC=C)ccc(C(C)(C)C)cc1NC(=O)Nc1cnc(C(F)F)nc1 C1(NC(c2ccn(CCF)n2)=O)CC2CC(NC(c3cnc(Cl)s3)=O)C1C2 C(=O)(C(C)C(C)COC)N1CC(OCC(N)=O)C1.C=C1CC2(C1)C(=O)NC2 Cn1cnc(=N)[nH]c1=NCC=C1CC(=O)N2CCCCC1C2 Cc1cccc2c(N(C(=O)C=Cc3ccc(F)cc3)CC3CCNCC3)ncnc12 C(=O)(CC1=CCCC1)NCCN(C(=O)C(c1cc(Cl)ccc1F)(C)C)CC(C)O Cc1ccc(CNC(C2CC2C(=O)Nc2onc(C)c2C#N)=O)c(F)c1 Cc1cc(C)nc(N2CC(NC(c3cn(CC4CCCOC4)nn3)=O)CC2C)n1 N1(C(CCC2CC(NC(C3(C)N(C)CCC3)=O)C2)=O)CC2CC3CC2C1C3 C1(NC(N(CC(=O)Nc2nc(C3CC3)cs2)CCC)=O)CCN(C)CC1 C1(CC)C2CCCC1N(C(c1cccs1)=O)C2.n12nc(C(C)C)cc1NC2=O c1(C(N(C)CC2CCCN(C(=O)C(C)(C)C#N)C2)=O)cc2c(nn1)OCCS2 C1(OC)CC2CCC(C1F)N2C(=O)CCCC(c1nnnn1C(C)(C)C)OC(C)=O CCCCN=c1[nH]c(=NCCc2cccnc2C)[nH]c2c1CSC2 C(=O)(C(CC(C)(C)C)NC(c1cc(=N)[nH][nH]1)=O)NC1CN(C)C(=O)C1 C(CN=c1[nH]c(C)cc(=NCC2CC(C(N)=O)=NO2)[nH]1)c1c(C)ccnc1 C1(CNC(C(C)Sc2ccccn2)=O)CN(C(=O)Cc2ccon2)CC1(C)C C1(N=[N+]=[N-])(C(N(C)OCC(F)F)=O)CCN(C(C2CC(=O)C2)=O)C1 C(CC1=CCCCCC1)NC(C1C(NC(c2c(CCC)nco2)=O)CC=CC1)=O c1(CC(=O)NC(C2CN(C(C(COC)(C)OC)=O)C2)C)cc(F)ccc1C C1(C(N2CC(OC)(CNC(c3cncs3)=O)C2)=O)Cc2c(C)cccc2O1 c1(C(=O)NC2CCN(C(c3cc(CC)on3)=O)CC2)cc(C)c(O)c(C)c1 CN1C(=O)CCC1C(N1CC(CCNC(=O)CC2CC2)C1)=O c1(C(=O)NCCOCCNC(CCC2CCN(C)C2)=O)[nH]nc([N+](=O)[O-])c1Cl C1(C(CC)NC(C2CCCN(Cc3ccccc3)C2)=O)CCOC(C)(C)C1 C1(C(=O)NC(Cn2cc(C(C=C)(C)O)nn2)C)CC2(CCNCC2)CO1 Cc1cc(C(=O)NCC2CC2NC(=O)CC2(n3cncn3)CC2)cnc1C(F)(F)F C(=O)(C1=NN(C)C(=O)CC1)NC1CCC(N(C(c2nc(CCC)oc2)=O)C)C1 C(CN=c1[nH]c(=NCCc2ncccc2F)[nH]c2c1SCC2)(C1CCC1)OC C1(NC(CC)C(N2CCC(C(=O)NCc3ccco3)(C(C)C)C2)=O)C(C)(C)C(O)C1(C)C C1(C2(O)CCN(C(=O)COCCF)CC2)(NC(CC(C)c2ccco2)=O)CC1 C(=O)(CCCC(C)=O)N1C(C(=O)NCC2(F)CCCCC2)(COC)C=CC1 c1(OC)cccc(C(=O)NC2CCCCC2NC(C2CCC(C3CC3)C2)=O)c1N C1(NC(c2cnc(OC)nc2)=O)CN(C(=O)COCC2CCCOC2)C(C)(C)C1 C(C1=CCN(C(=O)CCCC(OC(C2CCCC2C)=O)OC)CC1)OC c1(N2C3C(CNC(=O)Cc4ccoc4)C(CCC3)C2)cccc(F)c1[N+](=O)[O-] C1(C(C)N(C)C(C2CC(CCNC(=O)CC(C3CC3)C3CC3)C2)=O)CCOCC1 Cc1cc2c(cc1C)OC(C(=O)Nc1ccc(-c3nn[nH]n3)cn1)C2 CC1COc2c(C(=O)N(C(C)CCNC(=O)CCc3ccoc3)C)cccc21 CC1(C)C=C(C(=O)N2CC(NC(c3cc(-c4cccs4)[nH]n3)=O)CC(F)C2)C1 c1(C(=O)Nc2c(C(=O)NCCOCCOC)scc2)cc(Br)ncc1Br C12(CC(=O)NCC3C(CNC(c4nn(C)c(F)c4)=O)C3)CCC(CC1)CC2 c1(C(=O)NC2CCC(NC(c3cc[n+]([O-])cc3)=O)C2)coc2c1C(=O)NCCC2 C1(C(=O)NCC(C(=O)OCC)C)CCN(C(c2cnc(S)nc2)=O)CCO1 C1(OC)CC(CCNC(C2CCN(CCF)CC2)=O)N(C(=O)CC2CC(F)C2)C1 C1(C(=O)NCc2c(C(C)C)noc2)CN(C(C2(C#N)CCCOC2)=O)CCN1C c1(OC)cccc(CCC(=O)NC(C)CC(C)NC(c2ccsn2)=O)c1F N1(C(c2cncc(C)c2)=O)CCC2CN(C(c3cnc(C(F)(F)F)s3)=O)CC2C1 C1(C#N)(C(N(C(C(=O)NCCCC#C)(C)C2CC2)C)=O)CC(=O)C1 c1(C(C=CC(=O)N(C(CCC)C)CC)=O)ccc(Cl)cc1 C1(C)(C(N(C(C)C(=O)N2CCC2C(N)=O)CC)=O)CC(C)=NO1 C1(NC(CC2(C)N(C(c3cc(C)cc(O)n3)=O)CCC2)=O)CCn2nnnc2C1 c1(C(=O)NCC(CC(C)C)NC(C(C(CC)O)C)=O)nc(N)cc2ccccc12 CC1(CCCCCNC(C2(F)CC2)=O)CN(C(c2ccccn2)=O)CCO1 C1(CNC(C2(F)CCC(C)CC2)=O)CCC2CN(C(c3ccc(Cl)o3)=O)CC12 C1(C(=O)NCC(CSC)(C)C)C2CCC(C2)N1C(=O)C(C1CCCCC1)C c1(C(=O)NC2C(NC(C(CC)O)=O)C2)c(Cl)cc(Cl)cc1Br C#CCCCCCC(=O)N1CC=CC1C(=O)NCc1cc(F)ccc1Cl N1(C(Cn2c(C)c(Cl)cn2)=O)CCC2(CCCCC2NC(C2CC2(C)C)=O)C1 N1(C(C(CC)C)=O)CCCC12CCN(C(c1cc(C)c(C(=O)OC)o1)=O)C2 c1(N2CCCC(CSC)C2)nc(N(CCS(N)(=O)=O)C)nc2ccc(Cl)cc12 c1(NCCC(C)(C)NC(C2C(C)(C)CO2)=O)ccc([N+](=O)[O-])cc1F N1(C(CCc2nc(C)sc2)=O)CC(NC(=O)CCc2scnc2C)CC12CCC2 C1(NC(c2c(SC)ccs2)=O)CCN(C(C2(C)COCCO2)=O)CC1CO Cc1cc(C(N2CCOC(C(=O)NC(C)C(C)(C)CO)C2)=O)nc(C)c1 C1(CC)CN(C(C2CC2C(N)=O)=O)CC1C(=O)NCC(C)(C)OC c1(C(C(=O)NCC(C)(C)NC(C2(CC)COC2)=O)O)cccc(OC)c1 O=C(CCCC(=O)C1CC1)NC1CC(CCC(=O)NCCc2ccc(Cl)cc2)C1 C1(C(N2CCCC2C2(C(N3CC(OC)C(C)C3)=O)CC2)=O)(CC)CCCC1O C#CCC(C(=O)N1CC(C)(NC(=O)COCC(=C)C)C1)C1CC1 Cc1ccc(F)c(CC(N2CCC(C)(NC(C3CC34CC4)=O)CC2)=O)c1 c1(C(N(CCNC(CC2(C)CCCO2)=O)C2CC2)=O)cc(Cl)ccc1-n1cncn1 Cc1cc(C(N2CC3CC2(C(=O)NCc2cc(C)cnc2F)C3)=O)c(C)cn1 CC#CCCCC(=O)NC(CCOC)C(=O)NCCC(N)=O N1(C(c2cnc(CC)s2)=O)CCOC(CNC(=O)C=Cc2nccs2)C1 Nc1cc(F)cnc1C(N1CC2CCC2(C(=O)NCc2nc(O)cc(O)n2)C1)=O C1(CNC(C2CCCC(OC)C2)=O)CN(c2nc(C(N)=O)c(C)s2)CCCO1 CC1(C)CCCC(C(=O)NC(CNC(c2cscc2F)=O)CO)CC1 C1(C(=O)NC(c2ncnn2CC)C)(CNC(CCC)=O)CC12CCC2 c1(C(C(=O)NCCC#N)N(C(c2ccccc2)CC)C)cc(C)nc(C)c1 C(=O)(CCCC1CC1)N(CCNC(C(C)OC1CCCC1)=O)CC1CC1 C1(C(N)=O)(COC)CN(C(=O)CCNC(=O)NC2CCOC2)C1.C1(=O)CN1 C(C)(C(=O)N1CC(NC(=O)C(C)(C)CO)CC(F)C1)(C(C)C)OC N1(C(C2CC(OC)C2)=O)CCC(C(C)(C)NC(C2C3(CC3)C23CC3)=O)CC1 c1(C(C)C)nc(CC(=O)NCC(C)NC(=O)C(C)(C)N2CCCC2)cs1 CCC(C)C(C(=O)Nc1cncc(OC)c1)N(C)CC1CCCC(C)C1 N1(C(CCOCCC)=O)CC(CNC(c2cncn2C)=O)C(F)(F)C1 Cc1cc(=O)oc(C)c1C(N1CC2CC1C2NC(C1(Br)CC1)=O)=O C1(O)(CNC(=O)CCc2ccoc2)CCN(C(c2ccccc2SC(F)F)=O)C1 C1(OC)CC2(C1)CN(C(=O)C(c1cccs1)NC(=O)C(F)CC1CCCC1)C2 C(C(C)(O)CC(=O)NC1(C2CCCN2C(c2cnc(OC(C)=O)cn2)=O)CC1)OC N1(C(C(C(C)C)(C)C)=O)CC(NC(=O)CCC2(C)CC2(F)F)CCC(O)C1 c1(OCCOCC(OC(F)(F)F)=O)cc(C)cc(F)c1.CC(C)(C)OC=O.C1CO1 c1(C(=O)NC(CC)CNC(c2c(C)nn(C)c2C(F)F)=O)nn(C)c2c1CCC2 c1(C(=O)NC(c2ccccc2)CNC(C(C(C)C)O)=O)csc2ncnc(O)c12 N1(C(CCC2(C)CC2)=O)CCN(C(c2cccc3ncoc23)=O)CC(O)C1 N1(C(c2n(COC)ncc2)=O)CC=C(C(C)(C)C(=O)N2CCC(F)(C#N)C2)C1 c1(SC)cc(C)c(C(N2CC(NC(c3cscc3Cl)=O)C3CC23)=O)o1 N1(Cc2ncc(C)s2)CCC(NC(C2(N(C)C)CCCC2)=O)C(O)C1 c1(C(N(CC(CN(C(C2CC(C)=C(C)CC2)=O)C)O)C)=O)n[nH]c2c1CCSC2 C1(C(=O)NC2CCN(C(C(C)OCCOC)=O)CC2C)CCC(C2CC2)CC1 c1(C(C(=O)N(C(CNC(=O)CN2CCOCC2)C2CC2)C)F)ccccc1 N1(C(C(CC)n2ccc(C3CC3)n2)=O)CCOC(C)(CNC(=O)CCS(C)(=O)=O)C1 Cc1cc([N+](=O)[O-])ccc1C(=O)NCC(C(C)C)NC(C1CCC(=O)C1)=O Cc1cccc2cc(C(=O)NCC3CCCN3C(c3cc(Cl)ncc3O)=O)sc12 CCC(O)C(=O)N1CCC(C(=O)NC2CSC2)C1 c1(-n2cc(CN)nn2)ccc([N+](=O)[O-])c(C(=O)NC(C2CC2)C2CC2)c1 c1(C(=O)OC)ccc(C)cc1NCCCN(C(=O)C(O)C(C(C)C)OC)C N1(C(C)(C)C)CCN(Cc2nccc(-c3cccc(OCC(N)=O)c3)n2)CC1 c1(C(=O)NCC(CC)NC(c2conc2C)=O)c[nH]c2cccc(F)c12 C1(C(=O)NCC2C(C)CN(C(=O)C(N)=O)C2)CC2(C1)CC2(F)F N1(C(c2c(CC)cncc2)=O)CC2CCOCC2(NC(=O)CCCOC)C1 C1(CNC(c2ccc(F)nn2)=O)CCN(Cc2cc(Cl)c(O)cc2F)CC1(F)F C(=O)(C1=Cc2ccccc2C1)N1CC(CNC(c2n[nH]cc2Cl)=O)C(O)C1 CC1C(NC(=O)CCSC2CCCC2)CCCN1C(c1ccc(F)s1)=O C1(C(N2CCC3(CC3C(=O)NC3CC3)C2)=O)CCn2ccnc2C1 Cn1cc2c(n1)CC(C(=O)NC1CCC(CCNC(=O)CNC=O)C1)NC2=O CC(F)CC(=O)N1CCCC1C(C)(C)C(=O)N(C(C)CN(C)C)C c1(C(=O)NC2C(NC(CSCC(=O)OC)=O)C2)ccn(CC#N)n1 CC1CCC2(CC2)N(C(C2C=CCN2C(C2CC3CCC3C2)=O)=O)C1 c1(C(N(CCCNC(=O)C=Cc2ccc[nH]2)CC)=O)cc2cccn2c(O)n1 C#CCC(C)C(=O)N(C)CCNC(c1ccoc1I)=O C(=O)(C(F)(F)C(F)(F)F)NC(C1(O)CCN(C(c2nnc(C)s2)=O)C1)C c1(CC)nocc1C(=O)N(CC(CC)NC(=O)Cc1ncoc1C)CC N1(c2ncc(C)c(C)n2)CC2CCC(NC(C3CN4CCN3CC4)=O)CC2C1 CC1(C)COCC1C(=O)NC1CC2(C1)CC2NC(=O)CN1CCOC1=O C1(C(C)(C)C)CCCN(N2CC3(CCC3)C2)CC1 CN1CCOc2cc(CNC(C3(C(=O)Nc4cc(F)nc(F)c4)CC3)=O)ccc21 c1(C(=O)NC2CCCC2CNC(C23CC(CC(F)F)(C2)C3)=O)cc(CO)oc1C.C.C CON=C(C(=O)N(C)CC1(CNC(=O)C=CC(=O)N(C)C)CC1)c1ccco1 C(=O)(C(CC(C)C)NC(=O)OC)NCC1N(C(COCCC)=O)CCC1 Nc1cc(C(=O)NC2CCC2NC(c2n[nH]cc2Cl)=O)c2ccccc2c1 N1(C(Cc2ccc(C)cc2)=O)CCC(NC(c2cc([N+](=O)[O-])c[nH]2)=O)C(C)C1 C1(C(N(C(CNC(C2(CO)CC23CCC3)=O)C2CC2)C)=O)CC(=O)CC(=O)N1 c1(OCCC)cccnc1C(=O)NC(C1(O)CN(C(=O)CCC=CC)C1)C N1(C(CC(CC)OC)=O)CC(NC(C2CCc3ccnn3C2)=O)CC12CCC2 c1(C(N2C(C(C)C)CCC2C(=O)N(C)CC2CC2)=O)ccc2[nH]ccc2c1 c1(C(N2CCOCC(NC(C3C(=C)CC3)=O)C2)=O)cc(C)nc(Cl)c1N c1(CCC(=O)NCCc2c(OC(CSC)C)cccc2)ccc(Cl)c(Cl)c1 CC(C)(C)S(=O)(=O)CC(=O)N1CC2CCC1CN2C(=O)CC1CCOC1=O N1(C(c2nc(CCCC)sc2)=O)C2CCC1CC(CNC(=O)C(O)C(F)(F)F)C2 C1(O)(CCNC(C(C)CO)=O)CCN(C(=O)Cc2cncnc2O)C1 c1(C(N2CC(NC(c3cncs3)=O)C(F)(F)C2)=O)ccc2ccccc2n1 C1(NC(c2cnc(CC)nc2)=O)CCN(C(c2scc(C)c2C)=O)CC1F C(CC(C(=O)NC1CSC1)NC(C12CC(CC1CO)C2)=O)SC CCC(C)(CC)C(=O)NCC(C1CCCN1C(c1nn(C)cc1Br)=O)(C)C C12(NC(C3CCC(=C)CC3)=O)CCCC(CN(C(=O)CC(O)C3CCCC3)C1)C2 N1(C(C(C(C)C)NC(C)C)=O)CC2CCC1C(NC(C1(O)CC1)=O)C2 C=CC(C)CC(=O)NCCC(=O)NCC(Cc1ccccc1Br)CO c1(OC(C)C(=O)NCC(F)CNC(=O)CC2CC(=O)C2)ccc(Cl)cc1Cl C1(C(=O)NCCOC2(CNC(C3C(=C)C3)=O)CCOCC2)CNC(=O)CC1C C1(NC(=O)CCCc2cnn[nH]2)CCN(C(c2ccoc2Br)=O)CC1CO C(=O)(C(C)(C)C(=O)NCC(C)N(C(=O)CC1CC1(Cl)Cl)C)OCC C1(NC(C(c2ccnn2C)C)=O)CCC(NC(c2cn(C(C)(C)C)nn2)=O)CC1 n1(CC)cc(C(=O)NCC(C)(C)OCCNC(C2(C)CCCCO2)=O)c(C)n1 CCC(CNC(=O)C(C(C)O)NC(=O)C=CC1CC1)C(C)(F)F c1(C(C(=O)NC(C2CN(C(c3c(OC)noc3C)=O)C2)C)C)cc(C)cc(C)c1 C(=O)(CS(=O)(=O)c1ccccc1C)N1CC(NC(CC2CC(OC)C2)=O)C(F)C1 c1(CNC(=O)NCC2CCN(CCC)C2)ccnc2[nH]ccc12 C1(C(=O)NCC(C)NC(=O)C(O)C2=CCCCC2)CCc2nnnn2CC1 Cc1nc2ccccc2cc1C(N1CC2CN(S(=O)(=O)c3cccs3)C2C1)=O CC(C)(O)C#CC(=O)N(CCCNC(C1C2CS(=O)(=O)CC12)=O)C1CC1 C1(NC(C(CCC)OC)=O)(NC(N)=O)CCCN(C(=O)CCCN(C)C)C1 C1(O)(C(=O)NC2CC(NC(c3cnn4c3CCCC4)=O)C2)CN2CCC1CC2 c1(C(N2CCC3(CC2)CC3)=O)cccc(F)c1Sc1ccncn1 c1(NC(c2cc(CNC(C(CC#C)O)=O)no2)=O)cc(CO)ccc1C N1(C(C(=O)NCCOC)=O)CCC(NC(c2sccc2C)=O)C1 c1(C(=O)NCC(CN(C(C(CC)CC(F)F)=O)C)O)cccc2c(C#N)c[nH]c12 N1(C(c2cccc(N(C)C)c2)C(=O)NCC2CC2)CCC(F)C(O)C1 N1(C(c2ccc(COC(C)C)cc2)=O)CCC(O)(CNC(=O)C(C)O)CC1 C1(C(N(CC=C)CC)=O)CCN(C(=O)C(CO)N(C)C)C(C)C1 N1(C(c2ncc(OC)nc2)=O)CCCCC(C(=O)NC(C)C(C)(C)CN(C)C)C1 c1(C(C2CC2)NC(C(C2CCC2)NC(CC)=O)=O)cnn(C)c1.c1(C=O)nn[nH]n1 C1(NC(C(C(C)C)CO)=O)CN(C(c2ccc(=O)n(C3CC3)c2)=O)CC2(CCC2)C1 NC(=O)CCCCC(=O)N1CCC2(CC1)CC2NC(c1ccc(=O)oc1)=O C(=O)(C(O)CCC(C)C)NCC1CC1CC(=O)NCc1ncc(C)[nH]1 c1(C(N2CCN(C(C=CSC)=O)C(C)CC2)=O)ccc(C#N)c(F)c1Br Cn1cc(S(=O)(=O)NC2CCC3(CC2)OCCO3)ccc1=O N1(C(c2cc(CC)c(CC)o2)=O)Cc2nccn2CC(NC(C2CC2(Cl)Cl)=O)C1 CC(C)CCCCC(=O)NCCC1CN(C(c2cccn2C(C)C)=O)C1 N1(CCNC(C#CCNC(C=CCOC)=O)=O)C(=O)CNC1=O c1(C(N2CC(NC(CP(C)(C)=O)=O)C(O)C2)=O)cc(F)cc2nn[nH]c12 C(=O)(C(C)(C)C(C)C)N1CCC(CC=C)(NC(=O)C=Cc2ccc(C)s2)C1 S(=O)(=O)(c1ccccc1F)Nc1nc(CCOC)[nH]c1 N1(CCCCOc2ccccc2)CCC2(CC1)CNCCO2 Nc1ccc(F)c(F)c1C(N1CC(NC(=O)CC2(O)CCOCC2)C(O)C1)=O Cc1sc(Br)cc1C(=O)NCC(C1CCC1)NC(C1CCS(=O)CC1)=O C1(C(N(C(C)C)CC)=O)(NC(=O)CCCOC)CCN(C)C1.n12cc(nn1)C2 c1(C(CN(C(=O)CCC(F)(F)Br)CC)=O)ccc2nnc(C(F)F)n2c1 Cc1c(C(N2CCN(C(C3C4CCCC34)=O)CC2)=O)cc(Cl)cc1Cl CC(CCc1ccccc1F)C(=O)NC(C)CN(C(=O)CC1(C)CC(F)(F)C1)C C#CCC(C)(C(=O)NC(c1ccns1)C)NC(C1CC(F)(CC)C1)=O N1(C(C=CC(=O)N(C)C)=O)CC(F)(CNC(=O)C(F)(F)SCc2cnn(C)c2)C1 N1(C(CSCCCC)=O)CC2CC2(CNC(C2CC2F)=O)C1 CC(C)(COc1cccc(Br)c1)C(=O)N1CCC(NC(c2csc(C#N)c2)=O)C1 Cc1cccc(CCNC(=O)Cn2cc(-c3cncc(C(N)=O)c3)nn2)c1C S(=O)(=O)(c1cccc(=NCC(C)c2ccsc2)[nH]1)NC(C(CCC)C)CO C1(CNC(c2c(C)ncs2)=O)CCCC12CCN(C(C1CC(F)(F)C1)=O)CC2 N1(C(c2cccc(OC)c2OC)=O)CC2CCC1CN2c1nc(C#N)c(Cl)s1 CCC(CC)C(C(=O)NCC1CN(C(=O)C(Br)=C(C)C)CCO1)N(C)C c1(C(=O)NCC2(CCNC(C3COC3)=O)CC2)cccc(Cl)c1.c12cn(nn1)C2 C1(O)(C(=O)NC2CC3CC2N(C(=O)CC2CCCC2)C3)CC2(CCOCC2)C1 c1(CC)ncc2c(n1)CCC(C(N1CCCC(CNC(=O)C(C)(C)F)C1)=O)C2 C(C(C)(O)CC(=O)NCCCCCCn1cc(C2CCCC2O)nn1)OC CC1CC(NC(c2cc(OCC(F)F)ccn2)=O)CN1C(c1cscc1F)=O C1(CC)CCC(C(N2CCOC(CNC(=O)C(O)CSC)C2)=O)CC1 C1(NC(c2ncn(C(C)C)c2)=O)COC2(C1)CN(C(C1(C(F)(F)F)CCC1)=O)C2 N1(C(c2c(C)ccc(F)c2)=O)CC(C2CN(C(c3cc(C(C)(C)C)c[nH]3)=O)C2)C1 C=C=C(C)CC(=O)N1CCC(C2CCCCN2C(=O)C=CC(N)=O)C1 C(=O)(CC1=NNC(=O)C1)NCC1(CNC(CCC(=O)N(C)C)=O)CCCCC1 CC1CN(C(=O)C(C2(O)CCC2)NC(c2ccc(O)nn2)=O)C(C)C(C)(C)O1 C(=O)(C(F)(F)C(F)F)NC1CN(C(C2C(C(=O)OCC)C2)=O)CC1C(F)F C(=O)(NNc1cc(Br)ccc1F)N1C(Cc2cccc(OC)c2)CN(C)CC1 c1(C(=O)NCN2CCCC2=O)cccc(Cl)c1Cl.C1(C2c3cn2nn3)CCOCC1 C1(NC(COCCCOC)=O)CCCCC1CNC(c1ncc(SC)s1)=O C1(CC)(CNC(C2CC(O)CN2C(=O)CNc2cccnc2)=O)CCOCC1 C1(CC)CN(C(=O)CC(F)(F)F)CCN1C(=O)C(F)CC1CC1 C=CC(C)(C)N1CC(C(=O)OCCOC(C)(C)C)C1.C(C)=O c1(C(=O)NCCN(C(=O)CC2(C)CCOC2)CC)cnnc(-c2ccccc2)c1 CCC(CC(=O)NCCCc1cccs1)N(C(=O)C(CSC)OC)C c1(SCc2cncc(C)n2)ccc(C(=O)NCC(N2CCOCC2)=O)c(C)n1 c1(C(C)NC(C)C(c2cncn2C)=O)cccc2c1OC(F)(F)O2 C(=O)(C1=CCS(=O)(=O)C1)N1CC(CCCNC(c2c(C)coc2)=O)OCC1 C(=O)(CCCCCOC)NCC(CC)NC(c1nc(Cl)oc1C)=O C(C(CC(=O)O)c1cn(CCC(F)(F)Cl)nn1)NC(CC(=O)N(C)C)=O c1(N2C(C3CCN(C(CC(C(C)C)O)=O)CC3)CCC2)ncc2cccnc2n1 Cc1cc(C)n(-c2cncc(NC(C)C(=O)NCC3CC(N)C3)n2)n1 CC(C)(C)CCCCNC(=O)CC1CC(F)CN1C(=O)COC1CCCC1 Cn1c([N+](=O)[O-])cnc1C(=O)OCc1ccc(F)cc1 Cc1ccncc1C=CC(=O)NCC1CCCN(C(C2CC3CC3CC2C)=O)C1 N1(C(C(COC)C)=O)CCN(C(c2ccccc2-n2ccnn2)=O)CC(O)C1 c1(SCC(=O)NCCC(O)CNC(C2CCCCO2)=O)ccc(F)cc1 C#Cc1ccc(C(=O)NCC2(C3(O)CN(C(C4CC(=C5CC5)C4)=O)C3)CC2)cc1 C(C)(N=c1nc2sccc2c(NCC2CSCN2C(C)C)[nH]1)c1c(SC)cccc1 c1(C(N2CC(CNC(c3c(C)cc(C(F)(F)F)s3)=O)C2)=O)cnc2cc[nH]n12 c1(CCCOC(C(CC)Cc2cccc(Br)c2)=O)ccc(F)cc1C#N c1(C(N2C(C)CCC(NC(C3C(OCC)C3)=O)C2)=O)cccn2nccc12 c1(C(=O)NC2CN(C(C3CNC(=O)O3)=O)C(CO)C2)cc2ncsc2[nH]1 c1(CC)cccc(F)c1C(=O)NCC(C)NC(c1ccc(F)cc1)=O C1(C(NOCCC=C)=O)(CNC(c2cc(Cl)ns2)=O)CCCO1 C1(NC(COCCC=C)=O)CCN(C(=O)COc2ncccc2CC)CC1C C1(NC(CNC(CCCC)=O)=O)CN2C(C)(C1)C2=O.C(C)(C)(CCC=C)OC CCCCC(CNC(=O)Cc1ccns1)NC(c1cc(OC)cs1)=O c1(CC(C(=O)NC(C(CO)NC(C2(C(CC)=O)CC2)=O)C)C)ccccc1C c1(C(=O)NCC(CNC(c2cc(Cl)cc(C)c2N)=O)O)ccc2c(c1)CCC=C2 C(CC(CNC(=O)CSCc1ccncc1)NC(C1CC(C)(CF)C1)=O)OC c1(C(N2C(C(=O)Nc3cc(OC)cc(F)c3)CC3CC32)=O)ccn2cncc2c1 Cc1cc(N)c(C(=O)NC2CCC(NC(C3(C)CC4CC4C3)=O)C2)c(F)c1 CCCC(C(F)(F)F)NC(C1CCCN(C(c2cc(C)nn2CCC)=O)CC1)=O C1(C#N)(C(=O)NC(C2CCCN(C(CC3CC(=C)C3)=O)C2)C)CCCCC1 C12CC3(CC3)CN1C(=O)N(C)CCOC(=O)C2.C1(OC(C)(C)C)NC(=O)CC1(C)C N1(C(COC)=O)CCC(N(C(=O)CCCNC(c2ccsc2)=O)C)CC1 c1(C(N(C(CNC(C=C(C)C2CC2)=O)C2CC2)C)=O)c(N)sc2c1CCSC2 Cc1cc(CC(=O)NC(C)CCC(=O)NCC2(C#N)CCC2)c(C)s1 S(=O)(=O)(c1ccc(Cl)c2cccnc12)NC(C(c1ccc(C(C)=O)cc1)N)=O CC1CCc2[nH]nc(C(N3CCCC(N(C)C(c4cccc(=O)o4)=O)C3)=O)c2C1 C1(C(=O)NCCC(C)NC(=O)CCc2nc(C(C)(C)C)no2)CCCN1C1CC1 C(=O)(C1=CCCN(C(=O)C=CC(C(CCCCCC)C)(C)C)C1)OC(C)=O C1(C(=O)NC(C(=O)N(C(C)CO)C)Cc2cn[nH]c2)CC(=O)CC1(C)C c1(CC(=O)NCCc2cn(-c3cc(C)cc(N)c3)nn2)cccc2cccnc12 S(=O)(=O)(c1nccs1)NC1CCCN(C(c2cccc(Br)c2F)=O)C1 C1(CC(=O)NC2(C(N3C(C(C)O)CC3)=O)CC2)CC2CCC1O2 C(=O)(CCS(=O)(=O)CC(C)C)N1CCC(NC(CCC(C)SC)=O)C12CCC2 N1(C(C(CCC)OC)=O)CC(C2CC2)(NC(C23CCCC2(C(=O)OC)C3)=O)C1 C12(C(=O)NC3CC(CNC(C(Cc4c(C)n[nH]c4C)C)=O)C3)COCC1C2(F)F c1(C(c2nnnn2CSc2ccccc2)NC(CCSC)C)ccc(F)c(Br)c1 N1(CCNC(CCC2(NC(C(C)c3cccs3)=O)CCC2)=O)CCCCC1 c1(C(N2CC(NC(C(C)C3CCCO3)=O)(CO)C2)=O)cc2c(Cl)cc(F)cc2[nH]1 C(=O)(C(F)C(C)(F)F)NC1CCC(CC(N2C(C)(C(=O)OC)CCC2)=O)CC1 C=C(C)CN=C(NCc1cccn1C)N(C)CCOC C1(CC)CN(C(c2nn(C(F)F)cc2Cl)=O)CCC1NC(C1CC1CF)=O N1(CC)CC(C(=O)NC2CN(C(=O)CCc3nc(C)no3)C2)CCC1=O c1(C(=O)NCCC(C(C)C)NC(c2cscn2)=O)c(F)cccc1[N+](=O)[O-] N1(C(c2cc(C)nnc2)=O)CCN(C(=O)CCCCCF)CC1C1CCC1 C(=O)(CC1=CSC2=NCCN12)NC(CC(C)NC(=O)CCCc1cccs1)C CC(=O)CC(C)(C)C(=O)N1CCC(OCCNC(=O)CCCCN(C)C)C1 C12(CC(N3C(C(=O)OC)CC3)=O)CCC1CN(C(=O)CCC1CCCCC1)C2 c1(NCC(C(C)C)OC)ccc(S(=O)(=O)NC(c2cccc(C)c2)CF)c(Cl)c1 C(C(C)C)(C(O)C(=O)NC1(CCO)CN(C(c2c(OC)cccc2O)=O)C1)OC CCC(C(=O)NCC1CCCCN(C(=O)C(C)OC)C1)C(C)(C)CC c1(CC(=O)NCCC(C)NC(C(C(CC)C)NC(C)=O)=O)ccc([N+](=O)[O-])c(N)c1 N#CCCCCC(=O)N1CCC(NC(C2CC3CCC2O3)=O)CC1 c1(SCCSc2cccc(Br)c2)nc(C)sc1C(=O)NCC(C)(C)C.CC CCC(C)(C)C(=O)C(=O)NC1CCN(C(c2c(C)noc2C)=O)C1C Cc1cc(NC(c2sccc2CNC(=O)C#CC2CCC2)=O)cnc1Cl c1(C(=O)NCC(C(=O)N(CC(COC)(F)F)C)N(C)C)cccc(C)c1F N1(C(C2CCN(CC(C)C)CC2)=O)CCN(C(=O)CC2CC2(C)C)CC(CO)C1 CCCCC(C(=O)NCCC1CCCN1C(=O)C(C(C)(C)C)OC)N(C)C c1(C(N(C(C)CNC(=O)CCn2cccn2)CC)=O)cnn(CC)c1Br C(CC(C)C)(C(=O)N(CC(C)C(=O)NC)C)N(C(C1C(=C)C1)=O)C N1(C(C(Cc2cn(CCC(C)(C)C)nn2)O)=O)CC2(CO)CC2(COC)C1 O=C1C2S(=O)(=O)CCCN2C(=O)N1CCCc1ccc(Cl)cc1 c1(C(C)NC(=O)C=CC(C)NC(=O)C(C(C)C)N(C)C2CC2)ccncc1F C1(NC(=O)C(F)(F)C2CC2)CC2(C1)CN(C(C1(C3CCCO3)CC1)=O)C2 C1(NC(Cc2nc(C)sc2C)=O)CC(F)(F)CC1NC(c1c(C)nc(C)n1O)=O CN1CCC(C(=O)NCC2CCC(NC(c3cc(C(F)(F)F)cs3)=O)C2)CC1=O C(N=c1ncc(O)c[nH]1)C1N(C(C(CC(=C)C)c2ccccc2)=O)CCCC1 c1(N2CCC(CNC(C#CC(C)(C)C)=O)CC2)ccc([N+](=O)[O-])cc1F C(CNC(C12CC(F)(C1)C2)=O)(C(C)(C)C)NC(Cc1cc(C)no1)=O N1(C(C2CC(C#N)C2)=O)CCC(NC(=O)Cc2ccc(F)cn2)C2(CCC2)C1 CC(CCC(C)(C)C)C(=O)N(C(c1ccccc1)CNC(=O)CP(C)(C)=O)C c1(NC(c2cc(Br)ccc2F)c2n(CCOC)nnn2)nccc(Cl)c1C N1(C(CCCOCCOC)=O)CC2CC(NC(c3ccco3)=O)CC1C2 c1(C2(F)CN(C(C(=O)NC)C=Cc3ccc(C)s3)C2)ccc(F)cc1 C(CC1=CCCCCC1)NC(CC1CC(CNC(C2C(CC(C)C)C2)=O)C1)=O c1(CC(=O)N(C2CCCN(C(c3c(CC)nns3)=O)C2)C)ccc(C#N)cc1 C=Cn1nncc1C(=O)NC(c1ccccc1)CNC(=O)C=CCOCC c1(C(=O)NCC(CCCC)NC(C(C=C)(C)C)=O)c(F)ccc(C)c1Cl C1(CNC(N(C2CCNCC2)C(C)C)=O)CCCC(F)C1 CC1(C(N2CCCC(C(=O)NCC(N3CCCC3)=O)C2)=O)COCCO1 Cn1nc(CO)cc1SCC(=O)NCCNC(C1CC1OC(C)(C)C)=O c1(NCC2C(NC(c3cc(OCC)n[nH]3)=O)CCC2)c(C)ccc(OCC)c1N N1(C(C2CCN(C)C2=O)=O)CC2CCCC2(C(N2CCCCC2)=O)C1 Cc1cc(C(N2CCCC2(C)C(=O)Nc2cncnc2O)=O)ccc1Br c1(C(=O)NCC(C)=CC(=O)N(CCO)CCOCCO)ccn2ccnc2c1 N1(C(CCNS(CC)(=O)=O)=O)CC(C)CN(C(c2ccc(Cl)c(O)c2)=O)CC1C c1(C(C(=O)OCC)(F)F)ccc(F)cc1.C1(=O)C(C(C)C)n2cc(nn2)C2CN1C2 C1(OC(C)(C)C)CC2CC(NC(=O)NC3CCN(C4CC4)C3=O)CC12 c1(SC)ccc(C(=O)NCCN(C(c2cn3c(n2)SCC3)=O)C2CC2)c(Cl)c1 CC1(C(=O)NO)CN(C(c2ocnc2-c2cn(-c3ccncc3)nn2)=O)C1 C(C(O)CC(F)(F)F)NC(C(C(C)NC(c1cccc(CO)n1)=O)C)=O Cc1nc(C(=O)NC2CC(C(=O)NCC3CN(C4CC4)C3)C2(C)C)sc1C CCCCC(CNC(c1ccc(C(F)(F)F)o1)=O)NC(c1nocc1Br)=O c1(C(=O)NCC(CC)NC(=O)C(c2cccnc2)O)ccc2c(C)noc2c1 CCCC(CNC(=O)C(C)(C)C(=O)OC)C(=O)NCc1n[nH]c(CC)n1 c1(SCCC(=O)N(CCOCCN(C(=O)C=CC2CCCC2)C)C)ccccn1 C1(NC(c2ccc(OC)s2)=O)CCCCC1CNC(c1c(C)[nH][nH]c1=N)=O c1(C(N2CCN(Cc3ccc(OC)cc3)CC2)=O)ccnc(Cl)c1OC c1(C(N2C(CCNC(c3c(C)snc3)=O)CCCC2)=O)cc2c([nH]1)CCC(C)C2 c1(NCC2CC(NC(C(=O)OC)=O)C2)c(Br)ccc(F)c1I C12(C(N3CCC(Nc4nnc(-c5ccon5)s4)C3)=O)CCCC1C2(F)F C1(C(N2CC3(CCNC3=O)C2)=O)N(C(C2CC23CC3)=O)CC12CCCC2 C(C)(CNC(=O)Cc1ccn(CC)n1)(CC(C)C)NC(c1cccc(CC)c1)=O N1(C(c2nc(CNC(C(N3CCOC3=O)C)=O)oc2)=O)CCC2(CC1)N=N2 c1(C(N)=O)cc(C(=O)NCC(O)Cn2cc(CO)nn2)c[nH]1 C1(NC(CSCCCCC)=O)C=CC(CC(=O)NC(C)CC(C)O)C1 CCC(C)CC(=O)NCCCNC(=O)CCCN1C(=O)CNC1=O c1(C(=O)NCCCCCNC(Cc2c(C)ccs2)=O)c(C(F)(F)F)cncc1F N1(C(c2cnc(C)[nH]2)=O)CCC(C)C(NC(C2CCC(=O)N2C2CC2)=O)C1 CCC(CC(=O)NCC(O)CNC(=O)C(F)C1CCCC1)OC C1(NC(C2(CNC(C(CC=C)NC(C)=O)=O)CC3(CC3)C2)=O)CCOC(C)(C)C1 C1(C(=O)OC(C)=O)CN(c2ccc(C(F)(F)F)nc2)CCC1CO c1(C(=O)NC(C(C)C)CNC(=O)CC2CC(C)C2)ccc2c(=O)cc[nH]c2c1 c1(C(=O)NC(C2CCCN(C(CN(C)CC)=O)C2)C)ccc(C(C)(F)F)nc1O C1(=CC(N2CC3C(NC(=O)C=CCn4cncn4)C3C2)=O)CN2CCC1CC2 c1(C(N2CCC(CC=C)(NC(=O)C(O)CCSC)C2)=O)cccc(Cl)c1[N+](=O)[O-] C1(NC(CC2N(C)CCC2)=O)CCCCN(C(c2cncnc2)=O)CC1 CC(CNC(=O)C(C)(C)CO)N=c1ccn2c(Br)cnc2[nH]1 c1(OC)cc(CNC(=NCCCc2cccs2)NC(CF)CF)cc(OC)c1OC CCN(Cc1nn[nH]n1)N1CCC(c2cc[nH]n2)C(F)C1 N1(C(c2[nH]cc(CN(C)C)c2)=O)Cc2ccccc2C(NC(=O)C=CCF)C1 c1(SC)ccccc1NC(c1ccc(C)nn1)c1nnnn1C1CC1 C#CC1(NC(C23CCN(C(C4(SC)CC4)=O)CCC2C3)=O)CCCCCC1 Cc1noc(Cl)c1CC(=O)NCCN(C(c1csnc1Cl)=O)C(C1CC1)C1CC1 c1(C(=O)NCC2N(C(CC3(OC)CCC3)=O)CC=C2)cnc2[nH]nnc2c1 C1(NC(=O)C2CC2)CC(O)CN1OC.c12nc(cs1)C(=O)NC1CC(O)(C1)CC2=O C=C=C(C)CC(=O)N(C)CC1COCCN1C(=O)C(=O)Nc1ncc[nH]1 c1(CNCC2(OC)CCCCC2)ccc2ccc(Cl)cc2n1 C=CC1CCCCN1C(=O)C(C(C)(C)C)NC(C1CC(C)N(C)C1)=O c1(C(N(C)CC2N(C(C(CC)O)=O)CCC2)=O)ccc(OCF)cc1 Cc1oc(CNC(=O)CCCC#N)nc1C(N1CCC(C(C)CO)CC1)=O Cc1cn(C(C)(C)C(=O)NCC(C)NC(=O)CCc2nncn2C)cn1 C(CC(O)CCO)NC(C(C1CCCC1)NC(=O)CCc1ccccc1)=O c1(C(=O)NCC2CCN2C(=O)C=C(Cl)Cl)ccc(=O)n(CC(F)(F)F)c1 [N-]=[N+]=Nc1cc(F)ccc1CN=c1ccnc(N2CC=C(Br)CC2)[nH]1 CC(O)(CC(=O)N1CC(NC(=O)CC(c2cccs2)n2ccnn2)C1)C(F)(F)F C(CC(C)C(=O)N1CCCC1C(N1CC(C(C)C)C1C(C)C)=O)=CCC c1(SCC2(C(=O)OCC)CC(NC(=O)C(C)OC)C2)cccc(F)c1Br c1(C(N2CCCC(CN(C(c3c(COC)cc[nH]3)=O)C)C2)=O)ccc(O)nc1Cl N1(C(c2cccc(N(C)C)c2)=O)CCC2(C1)CN(c1nc(C3CC3)ns1)CCO2 C1(NC(C2CN(C)C(=O)CC2)=O)CCC2CN(C(=O)CN3CCOCC3=O)CC12 c1(CC)ncc(C(N2CCCC(NC(c3n[nH]c(COC)c3Cl)=O)C2)=O)c(O)n1 Cc1cc(C(=O)NCC23CCC2CN(C(C2C=CCCC2)=O)C3)cc(F)c1 CC(F)(F)C(CCc1ccccc1)C(=O)NCCNC(=O)CCC1CC1(C)C CC(C)C1=CCC(C(=O)NC2CC2NC(c2ccc(C3CC3)s2)=O)CC1 C1(Nc2ncn(C)c(=O)c2)(CNC(=O)C(=O)NC2CC2)CCC(F)(F)CC1 n1(CC(=O)NCCC2(NC(=O)CSC3CCC3)CCCC2)ncn(O)c1=O N1(C(c2cc(C)no2)=O)CCC(C)(CNC(=O)C(C)(C)C2CCOCC2)C1 CC1CN(C(C2(c3ccsc3)CC2)=O)CC1CNC(c1cn(C2CCC2)cn1)=O C(C(=O)O)(C(O)c1cccnc1)NC(=O)C(n1cc(Cl)cn1)F c1(C(=O)NC(C2(O)CN(C(C=CCC)=O)C2)C)cc(C)c(Cl)cc1C N1(Cc2ccc(OC)c(Br)c2)CC2(CCC(C(=O)NC3(O)CCOCC3)O2)C1 c1(C2(NC(C(C)n3cccn3)=O)CC2)ccc(Cl)cn1.C12CCN1C2=O C=CCCCC(C)(C)C(=O)N1CCN(C(C2OCC3COCCC23)=O)C(CC)C1 C1(NC(c2cn(CCOC)nn2)=O)C=CCN(C(=O)C(F)C2CCC2)C1 Cc1c(NC(C2CCCN(CCNC(=O)CC(F)(F)F)C2)=O)nn(C)c1 C1(CC)CN(C(c2occc2C)=O)CCN1C(C1CC1C(=O)OC(C)(C)C)=O C(C)(C)(CC(F)C(=O)N(CC(C)N(C)C(C)=O)C)NC(c1c(CC)cco1)=O c1(C2(C)CN(C(=O)NC3CC(OC(C)(C)C)C3)C2)c(C)nc2scc(C(F)F)n12 C(=O)(CCC(C)(C)C(=O)N1CCC(N(C(=O)Cc2ccon2)CCO)CC1)OC Cc1ccc(C(F)(F)F)cc1C(=O)NCC1CC1NC(c1ccc(F)s1)=O C1(C(=O)NC(C)C(C)(C)NC(=O)CS(=O)(=O)C2CC2)Cc2cc(Cl)ccc2O1 c1(CC)noc(C(N2CCC(N(C(=O)Cc3ccoc3C)C)CC2)=O)c1C Cc1cccc(C(=O)N(CC(C)C(=O)NCCC2CCCN2C)C)c1F N1(C(C(CCF)NC(=O)CCCCCO)=O)CC(C2CCCCC2)C1 C1(CCNC(Cc2nnc(C)s2)=O)CSCCN1C(=O)CSC(=N)N c1(C(=O)NC2CN(C(c3cncc(OC)n3)=O)C3C2C3)cc2n(c1)CCSC2 n1(-c2ccc(NC(C3N(CC)CCC3)=O)cn2)ccc2ccccc12 c1(C(=O)NC(C2OCCN(C(C(C)C)=O)C2)C)cc2nc[nH]c2cc1F c1(C(=O)NCC(CC(=O)N(CC(CC)CC)C2CC2)C2CCC2)ccc([N+](=O)[O-])o1 c1(C(N2CC3CN(C(c4c(C)c[nH]n4)=O)CC3C2)=O)ccc([N+](=O)[O-])cc1F N1(C(c2cn(CCC(F)(F)C(F)F)nn2)C(=O)NC)CCCC1C1OCCO1 c1(NC(CC2CN(C(=O)OC(C)(C)C)C2)=O)c2cccc1-2.C(C(F)(F)F)OCCO c1(C(N2CC(CNC(CCC=C)=O)N3CCC2C3)=O)ccc(=O)n2c1CCC2 c1(NC(C(=O)NCCc2ccc(OCCC)cc2)=O)scc(O)c1C#N C#CCCCC(C)C(=O)NC1C2CC1N(C(c1cnc(C3CC3)nc1)=O)C2 c1(C(C(=O)NCC(CNC(Cc2nc(C)[nH]n2)=O)C)(C)O)ccc(F)cc1 CCC(Cc1cccc(F)c1)C(=O)NCC(c1cn(C2COC2)nn1)(C)O c1(CC(=O)NC(CC(C)C)CNC(=O)C2CC2)ccc2nc(O)[nH]c2c1 C#CC1(C(=O)NCc2nonc2C)CCN(C(=O)Cc2c[nH]nc2C)C1 N1(C(C2CCCN(C)C2)=O)CCC2(NC(=O)CNc3ccccn3)CCCC12 CC(C)(CNC(=O)C(C1CCOCC1)N1CCCC1)Cn1cc(C2CC2)nn1 CC1(C)CC(NC(=O)C=CCO)CCN(C(C2CC3(CCCC3)CO2)=O)C1 C(=O)(C(C)C(F)(F)C(F)F)NC(CNC(C(CC)(F)F)=O)(C)CO c1(CC(N2CCN(C(CSCCCC)=O)C3C2C3)=O)c[nH]c2c(CC)cccc12 N1(C(C(CCCC)C)=O)CC2(C1)CN(C(=O)CCCOCCOC)CCO2 C1(CCC)CN(C(C2(CO)CC2)=O)CC1C(N(C)CC1CC12CC2)=O Cc1ccc(O)c(CN2CCCC(CC(=O)NCC3(C4CCCO4)CC3)CC2)c1 Nc1c(C(=O)NCC(c2ccccc2Cl)CO)cc(F)cc1Br C#CCCCC(C)C(=O)N1CC(NC(=O)C(C)CSC)C(c2cncn2C)C1 O=C(C1=CCCCO1)N1CCN(c2ncnc(O)c2Br)CC1 C(=O)(C1=COCCO1)NCC1(CNC(=O)CCc2cnco2)CC12CCC2 c1(N2CCC(C(C)NC(c3cnc(Cl)cn3)=O)C2)nc(C(F)F)nc(=N)[nH]1 C1(CCOC)(NC(=O)CCC2(C#N)CCC2)CCN(C(=O)C(CN(C)C)N(C)C)C1 C=CC1(C(N2CCC(C(C)C(=O)NCC(C)(C)C3CC3)C2)=O)CCOCC1 c1(CC(=O)NC(CNC(C2(C)CC2(F)F)=O)C2CC2)ccc(C(F)F)cc1 N1(C(C2C(OC)(OC)CC2)=O)CC(CNC(c2ncoc2C)=O)CC1(C)C CC1CCN(C(=O)CCCc2cncs2)C(C(=O)NCC2CCCCO2)C1 C1(C(=O)NC2C(NC(=O)CCc3ccsc3)C2)CCCC2(CCC2)O1 c1(C(N2CC(CNC(c3n(CC#C)ccc3)=O)OCC2)=O)cc(F)ccc1F c1(C(N)=O)ccc(C(=O)NCC(O)CNC(c2ccc(C3CCOC3)s2)=O)[nH]1 c1(CN(C)CC2(C)CC2(F)F)cc2cc(Cl)ccc2s1 CC(C)(O)CC(=O)NC1(CCC(=O)NC(C)(C)C)CCCC1 c1(OC)cc(C(=O)N(C(C)CN(C(=O)C=CC(C)(C)SC)C)C)c(C)cc1O C1(C)(CC)C=C(C(=O)NCC2CN(C)CCN2C(c2csc(C(C)=O)n2)=O)C1 C(C(=O)NC1CC(N(C(=O)Cc2ccccc2C)C)C1)(C(C)(C)C)OC C=C(C)CC(C(=O)NCCCNC(c1ccc(CC2CC2)s1)=O)NC(C)=O c1(C(=O)NC2CC3(C(NC(c4c(N)cccn4)=O)C3)C2)ccnc2c1CCC2 N1(C(C(n2c(C)cc(C)n2)C)=O)CCCC(C)(C(=O)NCCn2ccnc2)C1 N1(CC(C2CCCC2)OC)CCCCC(NC(c2csc3cncn23)=O)C1 C1(=CC)CCCC1(C)O.C(C(=O)N1CC(=O)NCC1)NC(=O)OCC C1(OC)CC(C)CN(C(c2ccnc(CNC(=O)CN(C3CCCC3)C)c2)=O)C1 N1(C(=O)CN2CCCC2=O)CC2(C(N3CCCC(CCO)CC3)=O)CCC1CC2 C1(C(=O)NCCc2ccc(C)s2)CC2CN(CCC(=O)Nc3nccs3)CC12 C1(NC(c2n(C)cnn2)=O)CN(C(c2cc(O)ccc2F)=O)C2(CCOCC2)C1 N1(C(c2scc(OC)c2OC)C(=O)NCCC)CCCC(C)(C)C1C(=O)OC C1(NC(CCCCOCCC=C)=O)CN(C(c2cccnc2)=O)C(C)(C)C1 N1(C(C(C)OCCC#C)=O)CCC2(CCOCC2)C(NC(=O)CC(C)CCC)C1 C(=O)(C(C#N)CC)NC(CCC)CNC(c1ccncc1OC(C)C)=O CCC(C(=O)OC)C(=O)NCCCOC.C12(CF)CCN(C1)C(=O)C(=O)N2 c1(OCC)cccnc1C(=O)NC(C)(C)CC1CC1.C12CCCN1C(=O)N2.OCC N1(C(c2cnc(C)s2)C(=O)NC)CC2(CCOCC2)C1Cc1ccc(Cl)cc1 c1(NC(C(=O)NC2(C)CC(CC)C2)=O)cnc2[nH]c3ccccc3c2c1 C(C(O)(C(=O)NC1CN(C(=O)CN2CCCCCC2)C1)C(F)(F)F)N(C)C C1(NC(C(F)=C(C)C)=O)CCN(C(=O)C(C)C2CC2)CC1F c1(C(=O)NC(CNC(C(C)SCCCC)=O)C2CC2)csc2cc(OCC)ccc12 C1(NC(Cc2c(C)cccn2)=O)CC(F)CN(C(C2CCC(=O)N2)=O)C1 CC1C(=O)NCCCN1C(C1CCOCCN1C(=O)CN1CC2CC2C1)=O C(=O)(C(C)(C)C(=O)NC1CCN(C(=O)COc2cnc(O)c(C)c2)CC1)OC N1(C(c2c(CC)ncs2)=O)CCCC2CN(C(=O)C(c3ccccc3C)C)CC12 c1(CN(C)C(C2CCCN(CC3(C(N)=O)CC3)CC2)=O)cc(=O)c2ccccc2[nH]1 C1(NC(C(C)Cn2cccn2)=O)CCN(C(c2ccc(Cl)c(Cl)c2)=O)C12CC2 c1(C(=O)NC(CCOC)CNC(c2cc(C)[nH]n2)=O)ccc(=O)n(C2CC2)c1 N1(C(CNC(C2CCCCCC2)=O)=O)CCOC2CCCCC12 c1(C(=O)NCCCOCCN(C(C(C2CCCCC2)C)=O)C)cscc1Cl Cc1ncc([N+](=O)[O-])n1CC(=O)Nc1cnn(C2CNC2)n1 CC1=C(C)CC(C(=O)NCC#CC(=O)NC2CC2CCN(C)C)CC1 CC1Cc2cc(C(=O)NC34CCC(C3)N(C(=O)CN(C)C3CC3)C4)ccc2O1 C1(CC)CCCC(C(N2CC(O)(CN(C)C(c3ncccc3F)=O)C2)=O)C1 c1(C(N2CCC(F)(C(=O)NC(CSC)C)C2)=O)nn(C#N)cc1C C(=O)(C(CCC(C)C)N=[N+]=[N-])N1CC(NC(C(n2ncc(C)c2)C)=O)C(C)(C)C1 C1(C(CC)O)CCCCN1C(=O)NC(C)Cc1ccc(NC(C)=O)cc1 N1(C(C(CC)n2cncn2)=O)CCN(C(c2cc(O)cc(=O)o2)=O)CC12CCC2 n1(CC)cc(Cl)c(C(=O)NC(C(C)NC(c2conc2COC)=O)C(C)C)n1 c1(C(=O)NCc2cc(C(N(CC(C)O)CCF)=O)on2)cc2occc2[nH]1 c1(C(N2C(CO)CC(NC(CC(C=C)(C)C)=O)C2)=O)ccc2oc(N(C)C)nc2c1 c1(CC)ccccc1NC(C1(Cl)CC1)=O.c12nocc1C2NC(=O)OC(C)(C)C C12(NC(COCCSC)=O)CCC(CC1)N(C(=O)CC1CCCS1(=O)=O)C2 n1(CCNC2(C(C)(F)F)CC2)ncc(NC(=O)OC)n1 c1(C(=O)NCCCN(C(C2CCCC(CF)C2)=O)CC)ccc(F)c(OC)c1F c1(C(=O)NC2CN(C(C(CC)C(C)O)=O)CC2(C)C)ccnc2[nH]ncc12 N1(C(c2cn3c(n2)CCCC3)=O)CCC2(CCCN2C(c2occc2Br)=O)C1 N1(C(C(CCC)=CCC)=O)CCn2c(CNC(C3CC3(C)C(F)F)=O)nnc2C1 C1(C(N2C(C)(CC(=O)NCC(CC)(C)Cl)CC2)=O)COCCC1C C(CCCC(=O)N1CCC(F)(CNC(C2C3CN(C)CC23)=O)C1)SC C1(CNC(c2cnc(CCOCC)s2)=O)CCC(C)CN1C(=O)CN1CC(C)C1 c1(SC)cc(C(=O)NCCC2(O)CCCNC2)cc(SC)c1 N1(C(c2nc(C)c(C)[nH]c2=O)=O)CCN(C(=O)CC2CCCC2)C2CCCC12 C1(CCNC(c2cc(OCC)no2)=O)CC(F)(F)CN1C(=O)C(N)=O C1(NC(c2[nH]cc(C(C(C)C)=O)c2)=O)CC2CC1CN2C(C1CC1C(N)=O)=O C1(NC(c2c(CCC)[nH]cc2)=O)CCC(CN(C(C2C(C)C2C)=O)C(C)C)CC1 C1(C(=O)NCCNc2ccccc2)(NC(=O)CCc2ccc[nH]2)CCOCC1 C1(CC(C)C)(CNC(C(=O)NCC(c2ccccc2)OCC=C)=O)CCCC1 C(=O)(C(C)C(O)C(C)C)NC(c1nc(C(=O)NCC(O)C2CCC2)co1)C CC1(C)CCC(C(=O)Nc2cccc(NC(C3CCC3(F)F)=O)c2)C1 CCC(CC)C(C)C(=O)N1CC2(CCC(CNC(=O)CN(C)C(C)C)O2)C1 c1(CCCC)nc(C)c(C(N2CCN(C(=O)C(CC)N(C)C(C)=O)CC2)=O)s1 N1(C(C(CC(C)C)C)=O)CCCN(C(c2csc(-c3ncc[nH]3)n2)=O)CC(CO)C1 c1(C(=O)NCC2(F)CN(C(C3C(CCC)CCC3)=O)C2)cccc(C(C)(F)F)n1 N(C1CCCc2sccc21)C(CCCCCO)c1n(C(C)C)nnn1 C1(C)(CC)CC1C(=O)NCC1CC(C(=O)N(CC(C)(C)OC)C)C1 CCC(CC(=O)N(C)CC1CN(C(C2OCCC2(C)C)=O)CCO1)OC C1(C(N2CCCC(OC)C2)=O)(OC)CCN(C(C)C(=O)NC2CCOCC2)CC1 C(=O)(C(C#N)C(C)C)NCC(c1ccccc1)N(C(c1[nH]cc(C)c1)=O)C c1(OCC)cnc(C(=O)NC(CN(C)C(C2CC2C(=O)OC)=O)(CO)CO)cn1 c1(OC)nccnc1C(=O)NC1CC(C)(OC(C)=O)C1.C12CCC(C1)C(=O)N2 C1(C(=O)NC(c2cn(-c3ccccc3CCO)nn2)C)CNC2(CC2)CO1 CC(C)CC(C(=O)Nc1cc(Cl)cnc1O)NC(=O)C(C)CC#N Cc1c(F)cc(C(=O)NC2CCCCN(C(=O)C=Cc3cscn3)C2)c(F)c1N Cc1ncsc1C=CC(N1CCCC1CNC(c1nnc(S)n1C)=O)=O C1(CN(C)C)CCC(C(N2CCC(N(C(=O)Cc3nc[nH]n3)C)C2)=O)O1 N1(C(c2c(C)nc(CNC(C(C(CC)C)C)=O)o2)=O)CC2(C(N)=O)CCC1CC2 N1(C(C(C)=NOCC#N)=O)CCCC(CCNC(=O)C=Cc2ccc(C)o2)CC1 C(=O)(C(C)(C)CC(=O)N1CC2CCCC2(NC(c2ccoc2C)=O)C1)OCC C#CCCCC(C)C(=O)N(C)CC1(O)CN(C(=O)COc2ccc(C)cc2)C1 c1(C2(C(N3CCC(NC(c4c(CC)c[nH]n4)=O)C3)=O)CC2)cc(F)cc(C#N)c1 c1(-c2ccc(CN(C(=O)COC3CCCNC3)C)o2)cc2ccccc2o1 c1(C(N2CC(CNC(CSCC=C)=O)C3C2C3)=O)nc(C)ccc1C C1(COCC(=O)NCC(O)CCNC(C2CCC2)=O)CCC(N(C)C)CC1 N1(C(COCCCC#C)=O)C(CNC(=O)C2=C(Cl)CCOC2)CC2CCCC12 N1(C(C2CCN(C(C(CC)(CC)CO)=O)C2)=O)CCc2c(O)noc2C1 C1(C(=O)NCC2C(NC(=O)CC3(CO)CCC3)C2)CCCCS1 CCN=c1ccc(C(=O)NCC(C)(C(C)C)NC(c2ccc(COC)o2)=O)c[nH]1 C1(NC(C(=C(C)C2CC2)F)=O)CC12CCC(NC(=O)C=C1CCN(C)C1)CC2 Cc1cc(C)c(CN(c2ncccn2)CCc2ccccc2)c(C)c1 O=C(N=c1nc(CC2CCCCC2)[nH]s1)Nc1cc(F)cc(F)c1 N1(C(C(C)n2cncn2)=O)CC2C(NC(c3ccc(C(F)F)cc3)=O)C2C1 c1(C(=O)NC(C2CCN(C(C3(CC)CCCO3)=O)C2)(C)C)cc(C)c(C)c(C)c1 Cn1nc(CNCc2cc(Cl)ncc2Br)c2ccccc2c1=O [N-]=[N+]=NCC(C(=O)N1CCS(=N)(=O)CC1)NC(=O)CC1CC2CC2C1 CC1CC(CNC(c2ccn(-c3cccnc3)n2)=O)CN1C(=O)CSCCC#N c1(OC)ccccc1C(C(C)NC(c1ccco1)=O)NC(c1ncc(F)cn1)=O N1(C(c2cnccn2)C(=O)NC(CC)C)CCn2c(nc3ccccc23)C1 CCC(CC(=O)NC1(CNC(C2(C(=O)N(C)C)CC2)=O)CC1)C1CC1 C1(C(N2CC(O)(CCNC(COC3(C)CCC3)=O)C2)=O)CC(C2CCCC2)C1 c1(C(N2C(C(=O)OC)CC2C)=O)cnc(COc2ccc(F)cc2)nc1 C(=O)(CC(C)(O)C(F)(F)F)N(CCCN(C(=O)C(C)(C)CC1CCOCC1)C)C c1(C(=O)NCCN(C(C(c2ccccc2)SC)=O)C)cc2cc(Cl)ccc2s1 C(=O)(C#CC1(C)CCCO1)N1C(C(=O)Nc2c(OC)n(C)nc2C)CC=CC1 C1(NC(c2cnc(C3CC3)s2)=O)COCCN(C(c2ccccc2Br)=O)C1 c1(C(=O)NCC(C)CNC(c2cnc(S)[nH]2)=O)cn(C(F)F)ccc1=O C1(C(=O)NCC2N(C(CCC(=O)N(C(C)C)C)=O)CCC2C)CCCCC1(F)F c1(CC(C(=O)NC(C)C(CO)NC(=O)CC2CC2)C)ccc(Cl)c(Cl)c1 c1(C(=O)NC(c2nocc2C(=O)NCc2ccncn2)C)cccc2cncn12 C#Cc1ccc(C(=O)NCCc2ccc(C(N3CCC(=C)CC3)=O)cc2)nc1 c1(SC)ccc(CNC(N2CCOCC2C2CCCC2)=O)cc1 C=C(C)CCCC(=O)NCc1nc(C2CCN(C(C3CC3(F)F)=O)CC2)n[nH]1 N1(C(C=Cc2c(C)ccnc2)=O)CCC2(CCCN2C(=O)COCC(F)F)CC1 CC(C)C(C)(CNC(C12COCC(C1)C2)=O)NC(c1cnc(C(N)=O)s1)=O CC1CC(=O)NCCN1S(=O)(=O)CC1CCC2CC2CC1 C=C=CC(C)C(=O)N(C)CC1COCCN1C(c1cn(CCO)nc1C)=O c1(N2CCC(CC(N)=O)C2)ccc(S(=O)(=O)NCC2(C)CCCS2)c(Br)c1 C=C(CNC(=O)COCc1ccccc1)CCNC(C1CSCCS1)=O c1(NC)ccc(Cl)c(C(=O)NCC2(C)CCCN2C(c2cnc3n2CCC3)=O)c1 C=CC(C)(CCOC)C(=O)NC(C)CCCNC(=O)CC1CCCNC(=O)C1 C1(CNC(c2c(CC)n[nH]c2)=O)CN(C(=O)C=CC2CCOCC2)C(C)(C)C1 N1(C(C=C(C(=O)NC2CC2)C)=O)CC(F)CC1CC(=O)N.CC=O C=Cn1nccc1C(=O)NC1CC(F)(CNC(c2ccc(CC(C)C)nc2)=O)C1 c1(C(c2ccnc(C3C(C)(N)C3(C)C)n2)C)ccc(Cl)c(Cl)c1 C(=O)(CCCN=[N+]=[N-])NC(C=CC(=O)Nc1c(C)n(C)nc1)C C1(C(=O)NCCCNC(=O)COC(F)F)CCCC(Nc2ccc(F)s2)C1 N1(S(CC)(=O)=O)CCC(C(N2CC(CCC(=O)Nc3ccon3)(OC)C2)=O)CC1 CCC(CC)CC(=O)NC1CCC1S(=O)(=O)NCCSC(C)(C)C c1(C(=O)OC)ccc(NC(C)=O)c(NC(=O)CC2CCCN2Cc2nccs2)c1 CCC(C(=O)NC(C1CCN(C(c2cnc3n2CCC3)=O)C1)(C)C)C(C)C C1(C(N2CCC(C3CCCCN3C(c3ccnnc3O)=O)C2)=O)C2CCCCC12 C(=O)(CCCCCn1cc(-c2ccn(C3CCC3)n2)nn1)N(C1(C)COC1)C CC(C)C(C)(CN=c1[nH]c(=NCc2c(S)cccc2)[nH]c2c1CCC2)N(C)C n1(CC(=O)NCC2CCCN(C(CC(CCC)O)=O)C2)cc([N+](=O)[O-])ccc1=O c1(OC)cccc(C(=O)NC(C)CNC(C2C3CCC2(c2ccncc2)C3)=O)c1 c1(NCCO)cc2c(cc1C)OCO2.N12CCC3(CC1)CC3C(=O)N(C)CCC2 c1(NC(C)=O)ccc2c(c1)CN(N1CCC([N+](=O)[O-])CC1)CC2 O(NC(=O)CCCC(CC)NC(c1cc(C(F)F)[nH]n1)=O)CC#C C1(C(N2C(CN(C(c3c(CC)ocn3)=O)C)CCC2)=O)CCCCC(C)(C)C1 N1(C(=O)CC2CCCCC2O)CC(C2CN(C(c3cnc4n3CCS4)=O)C2)C1 CC(CC(=O)NCCCCNCCCC(N1CCC2(C1)CC2(F)F)=O)CC(C)(C)C c1(C(N2CC(OCCNC(CC(C)CF)=O)C2)=O)cc(F)c(O)c(F)c1 c1(NC(N2CCCC2Cc2ccco2)=O)n[nH]c(C2CC2)c1Cl c1(C(N(CCCNC(CCOCCOC)=O)C2CC2)=O)ccc(C)c(P(C)(C)=O)c1 c12cc(cc(N)c1Br)NC2=O.N1(C(COC)=O)CC(OC)CC(F)C1 C1(NC(C(=O)N(C)Cc2ccc(C)cc2)=O)CC(O)CN(C(=O)OC(C)(C)C)C1 CC(C)CC(C)(C)C(=O)NCC1CCC(C(N2CCCCCC2C)=O)O1 O(NC(=O)CC=Cc1ccccc1)CC(=O)NCc1c(CC)nn[nH]1 C12(C3CCCO3)CC1CN(C(c1cnn(CC(F)F)c1)=O)C2.C(C)(CC=O)SCC Cc1cc2c(N3CCCC34CCS(=O)(=O)C4)ncnc2s1 [N-]=[N+]=NC1CCCN(C(c2cccc3c[nH]nc23)C(=O)NCc2ccccc2)CC1 N1(C(CC(=O)OCC)=O)CC2CCN(C(c3cc(CC4(C)CC4)c[nH]3)=O)CC12 C1(CNC(C(C)=CC)=O)CN(C(c2ccnc(C)c2)=O)CC(C)(C)O1 C1(O)(CN(C(=O)CC2CCCN(C)C2)C)CCN(C(=O)CC2CC2)C1 N1(C(C(C)(C)C(F)F)=O)CC2CC(NC(c3ccn4ccnc4c3)=O)CC1C2 c1(NC(=O)Cc2csc(=NCc3cccc4cc[nH]c34)[nH]2)ccc2ncsc2c1 N1(C(CNC(=O)Nc2ccc(-n3ccnn3)cc2)=O)CCC2(CC1)N=N2 C(CC(C)(C)CC(=O)NC1CCC(N(C)C(c2nnc(O)cc2C)=O)C1)OC c1(C(=O)NCC23C(CN(C(C(C)=C4CC4)=O)C2)C3)cc(C)cc([N+](=O)[O-])c1 c1(C(=O)OCC)cccc(C(=O)NCCc2ccc(CC(F)(F)F)cc2)c1O c1(NC(c2n(C(C)C)nnn2)c2c[nH]nc2C2CCCO2)ccc2c(c1)CCC2 C1(C(N(CC(COC)C)C)=O)CC(O)CN1C(C1(N2CCCC2)CC1)=O N(C1c2ccccc2CC1NC(C1CC1CF)=O)C(=O)Cc1cccnc1O c1(C(N2CCN(C(CS(CC)(=O)=O)=O)CC2CCO)=O)nccn2cnnc12 C1(C(N(C(C)CNC(C2CC2CF)=O)C)=O)CC(=O)c2ccccc2O1 C1(CNC(c2cnc(C)nc2)=O)COC(C)(C)CN1C(C1CCCN(C)C1)=O C(=O)(C1=C(Cl)CC1)NC(CC)(C)CNC(=O)CCc1ncco1 N1(C(=O)Cc2ccco2)CCC2CCC(C1)N2C(=O)CCc1ccc(O)c(Cl)c1 N1(C(CC)=O)CCCC(C(=O)NCC2CCC(NC(=O)COc3ccncc3)C2)C1 CC1CN(C(c2cncc(C(F)F)c2)=O)CC(C)CN1C(=O)C(CO)C(C)(C)C N1(C(Cc2cnc(C)s2)=O)C2CCC(C(N3CCCCC(CO)C3)=O)C1CC2 Cc1nc(=N)[nH]c(C)c1C(=O)NCCCC(C)NC(c1cccc(F)c1C)=O N1(C(C2C(C)C2)=O)CCOC2(C1)CN(C(=O)CN1CCCC(C(F)(F)F)C1=O)C2 C1(NC(C2(CO)CCCCO2)=O)CC2CC(C1)CN(C(=O)CCn1cccc1)C2 C1(OC)CC(C)CN(C(C2CCCN(C(=O)CC3CCC(=O)C3)C2)=O)C1 N1(C(c2cc(C)sc2C)=O)CCC(C)C(CNC(c2nccc(C)c2O)=O)C1 CC1(CNC(=O)CC2CCCC(C)(C)O2)CCC(NC(c2cnco2)=O)CC1 C1(C(N2C(CC(N3CC=C(C)CC3)=O)CC2)=O)CC12CCCCC2 Cc1nn(C2CCCC(NC(=O)NC3(n4cnnn4)CC3)C2)cc1NC(C)(C)C c1(C(n2cc(C(c3cncn3C)C(C3CC3)N)nn2)C)cccnc1.C1CC1 C(N=c1[nH]c(=NCCc2cnco2)[nH]c2ccccc12)c1n(C)ncc1Cl Cc1ncsc1C=CC(N1CCCCC1CCCNC(C12CC(F)C1C2)=O)=O O=C(CCCC(F)(F)F)NC1C2CCC1CN(C(c1ccnn1C(F)F)=O)C2 N1(CC)CCC(C(=O)NC(C)CCN(C)C(C2(CSC)CC=CC2)=O)C1 CN1CC(=O)N(CC(=O)NC2CN(C(=O)CSCc3ccncc3)C2)C1=O c1(C(=O)NCC2N(C(c3nc(OC)oc3)=O)CCOC2)cnn2c(=N)[nH]cnc12 N1(C(C2C(CC)C2)=O)CCN(C(=O)CNC(=O)OC)CC1c1ccccc1OC C1(CNC(C2CCS(=O)(=O)N2)=O)CC2(CCC2)CN1C(c1cn2ccsc2n1)=O N1(C(C2(CC)CNC(=O)C2)=O)CC2(C1)CN(C(=O)C(C1CC1)OC)CCO2 C1(NC(Cc2ncn(C)c2)=O)CN(C(=O)CC2=CCCC2)CC2(CC2)C1 C=CC(C)(C)CC(=O)NC1CCN(C(c2ccc(SCC)nc2)=O)C1(C)C N1(C(C(F)=C(C)C)=O)CCc2[nH]nc(CNC(c3ccncc3Br)=O)c2C1 c1(-c2nnc(NC(c3ccc(F)cc3F)=O)s2)cc([N+](=O)[O-])ccc1F Cc1cc(CC(=O)NC(C)(CNC(c2c(C)n[nH]c2C)=O)C(C)C)n(C)n1 n1(CC(=O)OC)cc(CC(=O)Oc2cocc2Br)cn1.C1(=O)CCN1C1CC1 c1(C(=O)NCC(C)NC(c2cc3cc(F)ccc3[nH]2)=O)n[nH]c2c1CN(C)CC2 CCCC(C)C(=O)N1CCC(C(=O)Nc2ccccc2C(C)(C)C)C1 c1(CN(C2CCCN(C(CC3CCN(C)CC3)=O)CC2)C)ccc2nccnc2c1 C1(C(F)(F)F)(C(N(C(C)CCNC(c2ncn(C)n2)=O)C(C=CC)=O)=O)CCCC1 C1(CNC(c2cn(CC3(C)OCCO3)nn2)c2nnnn2C2CC2)CC12CCOCC2.C.C.C(=O)C N1(C(CC(=O)OC)=O)CC(CNC(=O)C(C)CN2CCCCC2)OC(C)(C)C1 Cn1nnc(C(=O)NC2(C(N3CCC3C(N)=O)=O)CC2(C)C)n1 c1(C(N2C(CNC(c3c(C)scn3)=O)CCC(C)C2)=O)ccc2nncn2c1 C1(O)(C(=O)NCC2C(NC(c3cnc(C(C)C)s3)=O)CCC2)CCCC(C)(C)C1 CC1(CNC(=O)CC2(NC(c3ccncc3F)=O)CCC2)CCC(=O)N1 c1(C(=O)NC2(C)CC(NC(COC(CC)C)=O)C2)cccc(C)n1 N1(C(=O)NCCCOC(C)(C)C)CC(F)(F)C1C1CC1 c1(OC)ncc(Cl)c(=NC2CC(C)CN(C(=O)NC(C)(C)C)C2)[nH]1 C(=O)(CCCC(F)(F)C(F)(F)F)NCCN(C(c1occ(C)c1)=O)C CCC(C)(C)CC(=O)NCC(C)(CNC(c1nsnc1O)=O)OC CC1(NC(=O)Cc2nc[nH]n2)CCC(NC(c2cccc(CC3CC3)n2)=O)CC1 C(C(=O)NC1CCN(C(C2CCCN(C(C)C)C2)=O)CC1C)(C(F)(F)F)OC(C)=O C(N=c1nc2c(cnn2C)c(NCc2cccc(Cl)c2Cl)[nH]1)c1c(SC)csc1 N1(C(c2nccc(CC)c2)=O)CCC2CN(C(=O)CSCCC(C)C)CC12 n1(C(CC)C)ccc(=NC(=O)C(C)CNC(=O)CC2(CO)CCC2)[nH]1 N1(C(COCCCC)=O)CCCCC(N(C)C(c2ccnn2CCC)=O)C1 CCCC(C(=O)N1CCCC(CCNC(C2(CO)CCOCC2)=O)C1)S(N)(=O)=O N1(C(C(CC(=C)C)C)=O)CCCCC(C2CN(C(c3cncc(Cl)n3)=O)C2)C1 c1(C(=O)NC2C3CN(C(C(C)(F)F)=O)C2C3)cnc2c(n1)CCCC2 N1(C(c2ccc(C)cc2)=O)CCC2(CC2)CC1C(N1CCCCC(C(=O)O)C1)=O C1(NCc2nc(CC)on2)CC2(CCN(C(=O)Cc3cccc(OC)c3)C2)C1 N1(C(C(CC)F)=O)CCN(C)CC1CNC(c1sc(-c2ccccn2)nc1C)=O c1(C(=O)NC(C)C(C)(C)NC(C2CCC2(C)C)=O)ccc(CO)cc1F C1(NC(C(C2CN(C(=O)CCC3CCCC3)C2)OC)=O)CC12CCCCCC2 CC1=C(C(=O)N2CCC(CC(C)NC(C3(C(=O)N(C)C)CC3)=O)CC2)CCC1 c1(CC)ccc(NC)cc1.O1NC(=O)CN(C)C(=O)C1 C12(C)CC(NC(=O)C(O)C(C)SC)(CN1C(=O)C1=C(C)OCC1)C2.CO n1(CC)ncc(C(=O)NC2CCC(CNC(=O)CCC(C)SC)CC2)c1C C=CCN(OC)C(=O)CC1C2CN(C(c3cc(OC)n[nH]3)=O)CC12 C(=O)(C1=COCCC1)N(C)CC1(O)CN(C(c2csc(C3CC3)n2)=O)C1 c1(CN(C)CC2CCN(C(Cc3cccc(C)c3)=O)C2)cc2c(C)sc(C)c2s1 C(=O)(C(C)C(C)C(C)(C)C)NCC=C1CCN(C(C2(C(=O)OCC)CC2)=O)CC1 C1(NC(C2C(C)OCC2)=O)CN(C(c2cnn3cccnc23)=O)C2CCCC12 N1(C(C)=O)CCC=CC1C(=O)NC(CC)C(=O)ONC1C2(CC(C(=O)OC)C2)C1.O=C C1(C(=O)OC)CC(OC(=O)C(c2ccc(C(C)C)cc2)C)CCN1 N1(C(C(CC)C)=O)CCCOC(C(=O)OCCCC(=O)NC2CC2)C1 Cc1cc(C(=O)NC2CC(C)CN(C(=O)C(C)NC=O)C2)cc(O)n1 N1(C(c2nc(CC)sc2)=O)CC(NC(C2CC2c2cccnc2)=O)C(O)C1 C=CCN=c1[nH]cc(C(N2CCC(C)C(NC(c3ccc(C(C)C)s3)=O)C2)=O)s1 CC1=C(C(=O)NC2CCC(NC(c3cncc(C(F)F)c3)=O)C2)CCO1 C(=O)(C1=CCC2(COC2)OC1)NC(C(C)NC(=O)Cn1ccc(C(F)(F)F)n1)C N1(C(C2C(COC)CC2)=O)CC2CC3CC2C1C3NC(C1CCCC(O)C1)=O N1(C(C(CCC)F)=O)CCC(CNC(=O)CNC(=O)CNC(C)=O)C(O)C1 CC1CN(CCNC(=O)Cc2ncc(F)cc2N)CC(C(F)(F)F)O1 c1(OC)c(F)ccc(C(N2CC3CN(c4cc(C(C)C)ncn4)CC3C2)=O)c1F N1(C(C2C(C)C2C)=O)CCC2CN(C(C3CCS(=O)(=O)N3)=O)CC2C1 c1(C(N(C)C(N)=O)=O)cc(NC(=O)CC2CCC(C3CC3)O2)ccc1Cl C1(CC)C(=O)NCCCN1C(=O)CCN(C(c1cc(C)c[nH]1)=O)C1CC1 Cc1ccc2c(c1)c(CN1CC(CCO)(NC(=O)CCn3cncn3)C1)cn2C C(=O)(CC(C(=O)NCCC(C)CCNC(c1cnsc1)=O)NC(C)=O)OC c1(CC)ccc(C(=O)NCC(C2CCOC2)NC(=O)C(C)(C)n2cc(Cl)cn2)s1 C(c1ccc(F)cc1)=CCC(N1CC2C(CNC(CCSC)=O)C2C1)=O N1(C(CCN(C)CCO)=O)CCC(C2CC2)C1C(=O)NC1CC2(CCOC2)C1 CC1CSCC1NC(=O)C(=O)N(c1cccs1)CC1(c2ccccc2)CC1(C)C C(N=c1[nH]c(=NC2CCCC(C(C)C)C2)[nH]c2c1SCC2)c1nc(CC)sc1 N1(C(CCc2c(C)n[nH]c2C)=O)CCCN(C(C2CCN(C3CC3)C2=O)=O)CC1 c1(OC)ccncc1C(N1CCCC1C(C)(C)NC(c1nccnc1N)=O)=O CC(O)C(F)(F)C(=O)Oc1cccc(C(=O)NC2CC3CC2C3)c1 c1(C2C(C(N3CCCC(c4cn(C)nc4)C3)=O)CC2)ccc(Cl)c(Cl)c1F C1(NC(c2c(C)cncc2)=O)CCC2CN(C(c3cn4c(n3)CCC4)=O)CC2C1 C1(CNC(CCCCSC)=O)C2CCC1CN(C(C1CCS(=O)(=O)CC1)=O)C2 N1(C(C(C)=O)=O)CCC2(CC(C(=O)N=c3[nH]n(C)c4cc(I)sc34)C2)C1 N1(C(CCCOCC=C)=O)CCC(C(N2CC=CC(CO)C2)=O)(CC)C1 O=C1CN(CC(=O)NC2CCCCC2NC(C2CC3CC2CO3)=O)C(=O)N1 C1(c2cn(CC)nn2)CN(C(=O)CC(C)C2CCCO2)CCO1 C(=O)(C(C)(C)NC(C1CCN(C(=O)C(n2ccc(C)n2)C)C1)=O)OC C(=O)(CCC(C)NC(c1ncn(C)n1)=O)NCc1ncc(C)o1 C=CCC(C)(C)C(=O)NCc1occc1C(=O)NCc1nocc1C(C)C C1(NC(C23CC(F)(C2)C3)=O)CN(C(c2csc(-c3nc[nH]n3)n2)=O)CC12CC2 N1(C(C(CC)C)=O)CCCC2(CCCN2C(c2n[nH]c3c2CCC3)=O)C1 C1(NC(C(CC=CC)C)=O)(CC)CCCN(C(=O)COC2CCCOC2)C1 CC1(C)CC(=O)N(CC(=O)NC2C3CCN(C(c4ccn(C(F)F)n4)=O)C23)O1 C1(C(=O)NCC2OCCC(NC(CC3(C)CC3(F)Cl)=O)C2)CCC(C(N)=O)CC1 C1(C)(C(=O)NC(C)(C)C=CC(N2CCC2CC(N)=O)=O)CC(F)(F)C1 c1(C(=O)NCC2(C)CCCN(C(C3(CC)COC3)=O)C2)cc2c(=O)[nH]ccn2n1 N1(C(C2CC=C(C)CC2)=O)C2CCC1C(NC(c1cc(C)[nH]n1)=O)C2 c1(CC(N2CC3(CN(C(=O)CCc4cnn[nH]4)C3)C2)=O)cncc2ccccc12 C1(CNC(C2(C)CC2)=O)CC2CCC1N(C(c1cc(C(F)(F)F)cnc1N)=O)C2 c1(NC(=O)COC2CC3CCC2O3)cccn2ncnc12 C1(CC)CN(C(c2cc(C)c[nH]2)=O)CCC1NC(C12CC3CC1C2C3)=O N1(C(c2c(COC)nn(C)c2)=O)CCOCC(C(=O)NC(CO)C(C)(C)C)C1 N1(C(c2ccc(N)cn2)=O)CCC(NC(=O)CC2CC(O)C23CCC3)C(O)C1 c1(C(N(C)CC2CCN(C(c3c(C)nc(CC)o3)=O)C2)=O)cc(F)cc(Cl)c1N C12CCC(C)(C)N(C1)c1nnnn1C2.C1(C(=O)OC)CCC12CCCC2 CCCC(C(=O)NCC(CC)N(C(c1ccn(CCF)n1)=O)CC)C(C)C N1(C(COCCOC)=O)CC(C(=O)NC(C2CCCO2)(C)C)C(C(C)C)C1 C1(NC(C2CC(=C)C2)=O)CCN(C(=O)C(=O)N(C)C)CC1C C(CCO)(C(F)F)N(C(CNC(CN1C(C)CCC1)=O)=O)C C1(NCC#C)CCCN(C(=O)C(N2CCOCC2)C2CCOC2)C1 N1(C(C2(OCC)CCCC2)=O)CC2C(CNC(=O)CC3COCCN3C)C2C1 N1(C(C(C)NC(CC)(C)C)=O)CC(NC(=O)Cc2ccn(C)c2)CC1(C)C C12(C(=O)OCC)CC(CC(=O)NCCC(O)CNC(=O)CC3CCCC3)(C1)C2 C(CN=c1[nH]c(=NCCc2nc(C(C)C)cs2)[nH]c2ccsc12)N(CCOC)C N1(C(=O)C(=O)NCC2(CF)CCC2)CCC(c2cccnc2)C1 c1(C(C)C)c[nH]ccc1=NCC12CC(CNC(C3CC(=O)N(C)C3)=O)(CO1)C2 C1(NC(=O)Cn2cnnn2)CCCC(NC(c2cscc2F)=O)C1 c1(N2C(C(=O)Nc3cc(Cl)c(OCCBr)c(Cl)c3)CC(C)C2)ncc(C#N)cc1Cl Cc1ccc(C=CC(=O)NCC(C)CNC(c2c(Br)cnn2C)=O)s1 C1(C)(CC)CCC(C(=O)NC2CC2CNC(=O)CCc2cn[nH]c2)O1 c1(OC)ccc(Br)c2c1C(NCC1CCN(c3ccc(Br)cc3)C1=O)CC2 C(=O)(C1=CC2C=CC(C1)C2)N1C(C)(C)C(C(N2CC3CCCC3C2)=O)CC1 Cc1cc(C(=O)NC(CNC(=O)Cn2ncc(Cl)c2C)C(C)C(C)C)cc(C)c1Cl CC(C)CCC(=O)NCC(=O)N(CCNC(C1CCOC1C1CC1)=O)C1CC1 c1(C(N(C)CC2(NC(C(C(C)C)SC)=O)CC2)=O)cc(F)cc2cnccc12 O(NC(=O)C(CCC(C)C)NC(=O)C(C)NC(N)=O)C(CC)CC c1(OC)ccc(C(CN(C)C)NC(=O)NC(C(F)(F)F)C2CC2(C)C)cc1 C=CCC(C)(C)C(=O)N1CC(O)(CN(C)C(c2ccc(C(C)(F)F)nc2)=O)C1 C=CC1(C(=O)NCc2cnns2)CCN(C(=O)CC(C)C(F)F)C1 N1(C(C(C2CCC2)OC)=O)CCN(C(C2CC2c2ccsc2)=O)C(C2CCC2)C1 N1(C(C(CCC)CNC(C2CC2Cl)=O)=O)CCC2(CC(CO)C2)C1 Cc1cc(=NC(=O)CN2CCC(F)(F)C(CNC(=O)CC3CC3(C)C)C2)[nH]o1 C(CCO)(C(C)(C)C)NC(C=CCN(C)C(c1cnc[nH]c1=N)=O)=O N1(C(C(C)(C)CO)=O)CC2CN(C(C3(S(C)(=O)=O)CCCC3)=O)CC2(C)C1 CC1CN(C(c2ccccc2C2CC2)C(=O)NCCCC2CC2)CC1(C)CO c1(C(=O)NCCC2N(C(c3ccc(SC)s3)=O)CCC2)c2ccccc2nn1C N1(C(C(COCC)N=[N+]=[N-])=O)CCCC(C2CN(C(c3cc(=O)cc[nH]3)=O)C2)C1 Cc1nc2c(s1)CCCC2C(=O)NCCCNC(c1coc2ccc(O)cc12)=O c1(CCC(=O)NC(CN(C(C(C)OCCCC)=O)C)(C)C)cc(C)n(C)n1 n1(CC)cc(C(=O)NCC2(CN(C)C(C3CC3CN3CCOCC3)=O)CC2)nn1 C1(C(=O)OC)CC12CCN(C(c1cc(F)c(-c3nc(CO)cs3)cc1F)=O)CC2 CCCC(CCC)C(=O)N(CCNC(C1CCCC1C1CC1)=O)CCOC c1(C(=O)NCC2OCC(OC)(OC)C2)cc(O)n2ncc(Br)c2n1 C#Cc1ccc(F)c(C(N2CCCN(C(=O)CN(C3CCC3)C)CC2)=O)c1 c1(C(=O)NCC2(F)CC(NC(C3C(C)CCC3)=O)C2)c(F)ccc(F)c1N C1(C(=O)NCCCCC2CN(C(C(CC3CC3)OC)=O)C2)CCOC(=O)CC1 C12(CNC(=O)C(O)Cc3ccccc3)CC1CN(C(=O)CC1(CO)CC1)C2 c1(C(N2CCC(C)(C(N(CCN(C)C)C)=O)C2)=O)c(-n2ccnc2)cccc1Cl C1(NC(COc2c(C(C)C)cccc2)=O)CCCN(C(=O)C(C#N)C2CC2)C1C C(C)(C)(CC(=O)N1CCN(CCCNC(c2cc[nH]c2C2CCC2)=O)CC1)OC C#CCCCCCCC(=O)N1CC2CC1(c1cn(-c3ccccc3SC)nn1)CO2 Cc1ccc(N2CCC(NC(=O)C(=O)NCc3cn(C)nc3I)C2)cc1 c1(CC)ccc(Cl)c(C(=O)NC2(CF)CCN(C(=O)C(C)(O)C3CCC3)C2)c1 c1(C(C(=O)NC2CN(C(c3cc(C)cc(F)c3)=O)C2)C)cn(C)c2ccccc12 N1(C(c2c(CC)ccc(F)c2)=O)CCC2(NC(=O)Cc3cccnc3)CCCC12 C12(CCCC1C1CC1)CNC1CCC1CN2.c1(CNC(=O)OC(C)(C)C)ccccc1 C1(C(=O)NC(CCNC(C2CCC(CCCCC)CC2)=O)C)CC(C)CC(=O)N1 c1(CN2CCCCC(N(C(CN(C)C)=O)C)C2)cc([N+](=O)[O-])c(Br)cc1F C1(C(=O)Nc2c(CC)scc2)CN(C(=O)Cn2cc(Cl)cn2)CCC1O C1(C(=O)NC(c2nc(C(=O)NC3COCC(C)(C)C3)co2)C)CCC(=O)NC1C Cc1nc(C(N2CC3CC3(CNC(=O)C(C#N)C3CC3)C2)=O)c(=O)[nH]c1C CN1CC(C(=O)NC2(CCNC(c3nc[nH]c3C(F)(F)F)=O)CCCC2)NC1=O c1(C(=O)NCC2C(NC(C(n3ccc(C)n3)C)=O)C2)cc(Br)c(C)cn1 C(CCCC(=O)NC(C(=O)N(C)Cc1cnc[nH]1)c1cccs1)SC c1(CC(=O)NC2C3CN(C(c4c(OC)ccnc4)=O)CC32)ccc(F)c(F)c1F C12(C(=O)NC(C(C)F)C)CCCC1CCN2C(=O)C(c1cnn(C)c1)C C1(NC(C2C(C)C2C)=O)COC2(C1)CN(C(c1cnoc1-c1cccs1)=O)C2 C=CC(CC)C(=O)NC(C(=O)NCC1(OC)CCC1)c1ccco1 N1(C(CCc2onc(SC)n2)=O)CCC2(C(=O)NCc3cnn(C)n3)CCCC12 N1(CC)CC(NC(=O)C(CC2CCC2)NC(=O)C=Cc2cncs2)CC1=O c1(C(C(=O)NC(C2CCCN2C(C2CC(C)(O)C2)=O)C)C2CC2)ccc(F)cc1 C(N=c1[nH]c(=NC2CC(F)(F)C2)c2[nH]ccc2[nH]1)c1c(C)nc(C)s1 c1(SC)ccc(C)c(C(=O)NCC2(O)CCN(C(=O)Cc3ncc(F)cn3)C2)c1 C1(C(=O)NC(CNC(c2c(CCC(=O)OC)c[nH]c2C)=O)C)CN2CCC1(C)CC2 N1(C(CCC(C)NC(c2cnc(Cl)s2)=O)=O)CCC2C(O)CC12 c1(CC(C(=O)NCC(CNC(CC(=C)C)=O)C)O)ccccc1Cl Cn1cc2c(n1)CC(C(=O)NCC1CN(CC=CCl)CCCO1)CC2 Cc1coc(C(=O)NC2CCC(CCNC(=O)C(F)(F)c3sccc3Cl)C2)c1 N1(C(Cc2cc(CC)no2)=O)CCC(NC(c2nc(Cl)oc2C)=O)C(CO)CC1 C=C(C)CCCC(=O)NCC1CN(C(=O)COc2ccccc2Cl)CCO1 C1(CC(=O)NCC2CC2c2cccc(Cl)c2)CNC(C(F)(F)F)CO1 Cc1cc2cc(C(=O)NCC3CN(C(=O)C(C)(F)C(F)(F)F)C3)[nH]c2cc1Cl C1(CC(=O)NC2C(N(C)C)COC2)CCOC1(C)C S(=O)(=O)(c1ccsc1C(N1CCC(NC(=O)Cc2ccoc2)C1)=O)N(C)C Cc1ccccc1C(=O)NCC(=O)NCC(F)CNC(c1sccc1Cl)=O c1(C(N2CC(OC)C(NC(c3cnnc(C)c3)=O)C2)=O)cccn(C)c1=O c1(NC(C2C3(CN(c4c(Br)cnc(SC)n4)C3)C2)=O)c(C)[nH]c2ncncc12 N1(C(C2C3N(C(CN(C(C)C)C)=O)C(CC3)C2)=O)CCC2CC(F)(F)CCC2C1 c1(C(N(C(CNC(c2ccc(C)o2)=O)C)C)=O)cnc2c(c1)c(C)nn2C S(=O)(=O)(c1ccc(F)c(Br)c1)N1CCN(C2CCN(C(=O)C(F)F)C2)CC1 C1(CNC(=NCCC)NCCc2cncs2)COC2(CCCC2)O1 N1(C(COCC=C)=O)C(C(=O)N(C(C)C(C)(C)O)C)C2CC(O)C1C2 C1(C(C)C)C(NC(=O)C(C)Oc2cccnc2)CCN1C(=O)CCC=CC(C)C c1(OCC(N2C(C(C)C)COCC2)=O)ccc(Cl)c(C2=CC(=O)CC(C)(C)C2)c1 c1(C(N2C(C(C)NC(c3cnc(O)o3)=O)CCCC2)=O)cccc2oc(O)nc12 N1(C(Cn2c(C(C)C)nnn2)=O)CCCC(N(C)Cc2cc(F)c(Br)cn2)CC1 N1(C(c2c(C)cccn2)=O)CC2CCC(CNC(C3CC3C)=O)C2C1 C1(Cc2cn(C3C4(NC(C(C)(C)O)=O)CCC(C3)C4)nn2)CC2CCCCCC12 c1(C(N(CCNc2nccnc2C(=O)OC)CC)=O)ccnc2c1CCO2 Cc1[nH]nc2cc(NC(=O)CC3CC(C)(C)CN3C(C3CC3C3CC3)=O)ccc12 c1(C(N2CCCC(N(C)C(C3CC4CC3C4)=O)CC2)=O)c[nH]c2cc(O)ccc12 C1(NC(c2c(C(C)C)ocn2)=O)CC(NC(c2cnc(O)n2C)=O)C12CCC2 C(=O)(C1=CCC2(COC2)OC1)NC(CC(C)C)CNC(C1(C)CC1(C)C)=O C1(NC(C2CCN(C(C)C)CC2)=O)CCN(C(c2cnc(N)c(Cl)c2)=O)C1(C)C C12(S(=O)(=O)N1C)CCC2.C1(CC(C(=O)N(CC)CC)N)CNCCO1.C(C)(C)(C)S c1(C(C(=O)NC(=O)CCC(=O)c2ccc(Cl)s2)(F)F)cccc(Cl)c1Cl C12(C(N(C3CCN(C(C4CC5CC4C5)=O)CC3)CCO)=O)CCOC1CCOC2 Cc1nn(CC(=O)NC(C(C)NC(C2(O)CCC2)=O)C(C)C)c(C)c1[N+](=O)[O-] CC(C)(C)C(CNC(=O)CCC(F)(F)F)C(=O)NC1CCC2CCC12 c1(NC(c2cccc3nccn23)=O)cccc2ccoc12 C1(NC(C(c2cccc(F)c2)C)=O)CN(C(=O)CCCC(N)=O)CCC12CCC2 CCCCCS(=O)(=O)CC(=O)NCC(C)CN(C(=O)CC12CC(C1)C2)C C(C(C)(C)C(=O)NC1CN(C(=O)C(F)=CCCF)CC1C(F)F)OC(C)C CC(C)C(C(=O)NC(C)CNC(=O)Cc1n[nH]c(=N)s1)c1ccncc1 c1(OC(C)C)ccc(C(N2CCC2CNC(C2CCC(=O)N(C)C2)=O)=O)cc1N N1(C(CC2CC(C)(C)OCC2)=O)CCCC(C2CN(C(=O)CC3OCCO3)C2)C1 CN1C2CCCC1CC(CNC(=O)Nc1ccnn1C1CCCOC1)C2 Cc1cc(C(=O)NCCC2(C(=O)NCc3ccncc3)CCC2)cc(C(F)F)c1 c1(OC)cnncc1C(=O)NC(C1CCN(C(C2CCC(=O)N2)=O)C1)(C)C CC1CCC(C(N2CCC(C)(NC(c3cncc(O)c3Cl)=O)C2)=O)C(=O)N1 c1(C(N2C(C)CCC(CNC(=O)CN=S(C)(C)=O)C2)=O)c(F)ccc(N)c1F CCCC(C)CC(C(=O)Nc1ccc(Cl)cc1)N1CCN(CC2CCOC2)CC1 C(=O)(CCCCCF)N1CCC(CCNC(c2cccc(OC(C)(C)C)n2)=O)C1 C(CCC(C(=O)NCC1CCCO1)N1CCOC(C(=O)OC)C1)OCC C(C(=O)N1CC(NC(C2CCC(CO)CC2)=O)C(O)C1)(C(C)O)NC(C)=O CCCC(CC(C)C)C(=O)NC(CNC(C12CC(C)(C1)OC2C)=O)C1CC1 N1(C(CCN(C)CC)=O)CCC2CCN(C(=O)Cc3ccn(C)n3)CC2C1 C(CCCCCCO)NC(C(C1CCCN(C(=O)CCc2cncs2)C1)C)=O Cc1cc(NC(C2CCCC(C)O2)=O)ccc1NC(=O)COCCC(C)C N1(C(Cc2n(C)c(=O)ccc2)=O)CC2CCN(C(C3C4COCC34)=O)C2C1 c1(NC(C(C)C)CNC(=O)CCC2CCCCC2)ccc(C#N)cc1[N+](=O)[O-] Cc1cccc(C(=O)NC2(CCNC(=O)C(F)C(C)(C)O)CCCC2)c1C C(C(C)(C)C#CC(=O)Nc1ccc(O)cc1Cl)NC(CCCC#CC)=O c1(SC)cscc1OC.C12(CCC1)C(=O)NC(C)CN(CC)C2=O C(=O)(C(C)(C)n1cncn1)N(CC(=O)NCC1CCOC1)CCOC N1(C(=O)Cn2cnnc2O)CCN(C(=O)COCCCF)C(c2cn[nH]c2)C1 C1(C(=O)OC)CC(C(=O)OC)CC(C(N2CCC(C(C)N)CC2)=O)C1 Cc1cc(C(=O)NCC2CCCC(CO)C2)n(C)n1.N12CC3C(C3C1)C2=O.C1CC1 C1(C(N2CCC(C)(CC)CC2)=O)CCC(C)(C)N(C(=O)Cc2nc(=N)[nH][nH]2)C1 C(CC(C)C)(C(=O)NC1COCC1CO)ONC(c1cc(CSC)no1)=O c1(C(=O)OCc2ccccc2[N+](=O)[O-])cc(Cl)cc2c1OCCC2 CN1C(=O)CCc2ccccc2C(NCCCCCCN(C)C)C=C1 CCC(O)C(C)C(=O)N1CCC(OCCNC(c2cnn(CCO)c2)=O)C1 C1(C(N(CCOCC#C)C)=O)CCCC(NC(c2cc(COC)sn2)=O)CC1 C(C1CCCCCC1)=CC(=O)NCCCNC(=O)CC1CCCCS1(=O)=O C1(NC(c2cncc(-n3cc(CCOC(=N)O)nn3)c2)=O)CCCCC1(F)F C1(CNC(c2ccc(Cl)o2)=O)CC2(CO1)CN(C(c1cc(Cl)c([N+](=O)[O-])[nH]1)=O)C2 c1(OC)ccc(C=CC(=O)NC2CCC(N(C(=O)C(CO)OC)C)CC2)cc1O c1(C(=O)NCC(CC=C)NC(=O)CC2COCCN2C)cc2c(C)nn(C)c2s1 C1(CNC(COCCCCC)=O)COC(C)(C)CN1C(c1cccc(C)c1)=O N1(CC(=O)NC(C2(O)CN(C(c3cccc(F)c3F)=O)C2)C)C(=O)CCCC1=O Cc1ccc(CNC(C2CSCCN2C(c2cccc(OC(F)F)c2)=O)=O)nc1 C1(NC(C(c2c(C)n[nH]c2C)C)=O)CC2CC(C1)N(c1nnc(C#N)s1)C2 c1(CC(=O)O)ccccc1N(CCCC#N)C(C1CC1c1nn[nH]n1)=O CC(C)C(O)CC(=O)NCC(F)CNC(c1cc(-c2ccncc2)no1)=O C=CC(CC)CC(=O)N1CCCC(CNC(c2coc(-c3cn[nH]c3)c2)=O)C1 C1(C)(C(=O)NCCC2CCCN(c3ncc(OC)cn3)C2)CCCCCC1 c1(C(N2CCN(C(C)CNC(=O)Cc3ccns3)CC2)=O)cc2cccnc2o1 c1(C(=O)NCC(C(F)(F)F)N2CCOCC2)cc(=O)c2ccc(O)cc2o1 N1(C(CN2CCCN(CC(=O)O)C(=O)C2)=O)CCNc2cc(Br)ccc2C1 c1(OCCC)cccc(C(=O)NCCC2CCN(C(=O)C(C)c3ccsc3)C2)c1 C1(C(N(CCCNC(C(CSC)OC)=O)C)=O)CC2(C)CC1CO2 C12C3CN(CC13)C(=O)N2.C1(Nc2c(C(=O)OC)nn[nH]2)CCN(C2CC2)CC1 N1(C(C(C)Oc2ccc(C)cc2Br)=O)CCCC2CCCCC12 N1(C(=O)CC2CCC3(CCC3)O2)CCC2(CC1)CCN(C(c1ccsc1)=O)C2 c1(C(=O)NCC(CNC(CC(C(C)(C)C)O)=O)O)cc2c(F)c(F)cc(F)c2[nH]1 c1(CC=CC(=O)C2C(C(=O)NCC)C2)ccc(NC2(CC#C)CCC2)nc1 CC(O)(C(=O)N1CC(NC(c2ccc(C(F)(F)F)[nH]2)=O)C(F)C1)C(F)(F)F C(=O)(C1=CCc2ccccc21)NCCC(CCNC(CC(=O)OCC)=O)C c1(C(=O)NC2CC(CNC(C3C(C)(CC)C3)=O)C2)cc(C)nn1C c1(C(=O)NCC2(F)CCN(C(c3ncc(OC)nc3)=O)C2)ccc2c(c1)CCC2 c1(CNC(C2C3(CC(NC(CCSCCCC)=O)C3)C2)=O)cccc(C)c1C C1(NC(C2CCCN2C2CC2)=O)CC(O)CN1C(C1CCC(F)(F)C1)=O C(=O)(C(C)(C)C(=O)NCC(CC)NC(C1CC1C(C)C)=O)OC C1(N(C(C2CC(SC)C2)=O)C)CN(C(=O)C=C2CCN(C)C2)CC1F Cn1nc(C(N)=O)cc1NC(C12CC1CN(C(c1csc(C#N)c1)=O)C2)=O c1(CC(=O)OC)cccc(C(=O)NCC(CNC(C2(C)CC=CCC2)=O)OC)c1 c1(C(=O)NC(c2cccc(Cl)c2)CC)nnc(N2CCOC3CC23)n1CCC#N CC1CS(=O)CCN1C(=O)CCC(C)(C)NC(=O)CC1CCCOCC1 C1(CNC(CCCN(C)C)=O)C(C)CCCN1C(C1CCCCC1)=O N1(C(C(CO)N(C)C)=O)CCCN(CCNC(=O)C(F)CC2CCCC2)CC1 c1(C(N(C2CCC(NC(=O)CN(C3CCCC3)C)C2)C)=O)ccnnc1N(C)C C1(CNC(CSCCC)=O)CC2(CCC2)CN1C(c1sccc1C)=O C(C)(C(C)(C)C(=O)NCC(c1cccs1)C)NC(C(CO)NC(C)=O)=O CN1CC(C(=O)NC2CN(C(=O)C=Cc3ccc(=N)[nH]c3)CC23CC3)CCC1=O N1(C(c2c(C)cc(F)s2)=O)CCC2CC(NC(c3csnn3)=O)CCC2C1 c1(NC(N2CCC(=O)CC23CCC3)=O)cc(=O)[nH]c2c(F)cccc12 C1(C(=O)NCC(C)(C)CNC(=O)Cc2c(F)cncc2Cl)CCC2(C1)CC2(F)F N1(C(N2CCC(=C)C2)C(=O)NC(C)(C)CC)CC2CC3CC2C1C3 c1(C(=O)NC2C(NC(C(CC)OC3CCCC3)=O)C2)ccc(F)c(C(C)C)c1 CCCC(C)(CCC)C(=O)NCCNC(C1CN(C(C2C=CC=CC=C2)=O)C1)=O N1(C(C(=O)N(C(CC)CC)C2CC2)C)CCCC(C)(C(N2CCC3CC23C)=O)C1 c1(NC)c(C(=O)NCCN(C)C(c2c[nH]cc2C(C)C)=O)cccc1F C1(C(=O)NC(C)CCN(C(=O)CCc2ncco2)C)OCCN(C)C1=O c1(CNC(c2c(C)cc(Br)cc2Cl)=O)ccc2nc(O)oc2c1.C12CCN(C1)C2 c1(NC(C2C(NC(c3c(O)ccc(C)c3)=O)C2)=O)cc(Cl)c(Cl)cc1I C12(NC(=O)C3=COCCO3)CCCC1N(C(c1nc3ccccn3n1)=O)CC2 Cc1cc(C(=O)NCC(C2CCN(Cc3ccc(C)s3)CC2)=O)n(C)n1 CC(C)(CC(=O)NC12CC1CN(C(=O)CN1CCSCC1)C2)c1ccccc1 c1(C(=O)NCC2OCCN(C(CCC3(C)CC3(F)F)=O)C2)cccc2c1CCC2 C(=O)(CCC(=O)NC(C)CC(C)NC(=O)C=Cc1ccsc1)OCC N1(C(C2C(CCC)C2)=O)CCCC(C(=O)N(CC(CC)CC)C)C1 C1(O)(CN(C)C(C2(F)CCOC2)=O)CCN(C(=O)CCc2ccc(Cl)cc2)CC1 c1(C(=O)NCC2C(NC(c3cnc(C(=O)OC)s3)=O)COC2)nn(C)c(N)c1C c1(C(=O)OC)ccc(CNC(=O)C(C)C2CC2)cc1.C12CCOC1CCNC2=O C(=O)(CCC(=O)N1CC(NC(=O)Cc2c[nH]nc2O)CC1C)N(CCC)CCC N1(C(C(C)CC(N)=O)=O)CCN(C(c2c[nH]c(C(F)(F)F)c2)=O)C2COCC12 C1(C(C)NC(C2(N(C)C)CC2)=O)CCN(C(c2ccc(CO)cc2)=O)CC1 CC1(C)CC1(C(N1CC(C(=O)NC2CC2)C1)=O)NC(=O)C=CC1CCCC1 c1(C(COC)=O)ccc(OC(C)CCF)c(C)c1 N1(C(Cn2ncc(CC)c2)=O)CCCN(C(=O)CCCC(=O)N(C)C)CC1C Cc1cc(F)c(C(N2CCN(C(c3nccc(Cl)c3O)=O)C(CF)C2)=O)cc1F c1(C(=O)NCC2(F)CC(NC(=O)COC3CC3)C2)ccc2nnc(O)n2c1 C1(O)(C(=O)NC2(C)CN(C(c3cccc(OC(F)(F)F)c3)=O)C2)CCCCC1 C(=O)(CCC(C)C#N)N(CCOC)CCN(C(=O)CCn1cnnn1)C1CC1 N1(CC2CC3(CC(OC)C3)C2)CCC(=O)N(CC(C)(O)CNC(C)=O)C1=O C1(C)(NC(C2C(OC(C)=O)C2)=O)CCN(C(c2cc(CC(C)C)on2)=O)C1 N1(CCc2cn(C(C)(C)C)nc2)CC(CO)C(CO)C1 N1(C(CCCC(=C)C)=O)CC2OCC(CNC(=O)C(O)C(F)(F)F)C2C1 c1(CC)ccc(CC)c(C(=O)OCCC23CC(OC)(C2)C3)c1 C1(S(N)(=O)=O)(C(N(C)CC2CN(C(C3CCCCN3C)=O)C2)=O)CCC1 C1(CNC(Cn2ncc(CC)c2)=O)CCC2CN(C(=O)C(F)=CC3CC3)CC12 N1(C(CC(C)SC)=O)CCC(CCC(=O)NC2CN(C)CC2C)CC1 N1(C(Cc2c(SC)cccc2)=O)CCC2(CC1)CN(C(=O)CC1CCOC1C)C2 C#Cc1cccc(C(=O)NC2CC(CCNC(c3ncccc3F)=O)C2)c1F c1(C(N2CC(CC)N(C(C3(C)CC3(C)C)=O)CC2)=O)oc2cc(Cl)ccc2c1C C1(CNC(CCCC#C)=O)C(C)CCCN1C(=O)C(C)SCCCC N1(c2ccnc(CC)n2)CCCN(C(=O)NCCC2CCCN(C)C2)CC1 C1(NC(c2cc(CO)[nH]n2)=O)CCC2CCN(C(C3(CO)CCC3)=O)C1C2 N1(C(c2c(C)cccn2)=O)CC2CC(C1)CN(C(=O)CCCC(F)(F)F)C2 Cc1[nH]cc(C(N2CC(NC(C3CC4CSCC(C3)C4)=O)C2)=O)c(=O)c1Cl C1(N(C)C(C2(C)CC(C(F)(F)F)C2)=O)CCC(N(C)C(c2ccccc2)=O)C1 C1(CNC(c2ccncc2)=O)CSc2ccccc2O1 c1(C(N(CCC(C)(C)NC(=O)Cn2nccn2)C)=O)ccc(F)c(OC(F)(F)F)c1 C(=O)(CCCC(=O)NC1CCN(C(C2(C)CCNC(=O)C2)=O)C1)N(C)C N1(C(C2(CNC(=O)C=CCCC)CC(=C)C2)=O)CC2CC(CO)C(C2)C1 c1(CC(=O)N(CC(C)NC(CC(=C)C)=O)C)sc(C)cc1C N1(c2ncc(C)cn2)CC(NC(=O)C(C)(C)CC2CC2)CC(C)C1 CC(C(=O)NCC(O)CC(=O)N1CC(C(N)=O)C1)C(C)(C)C c1(C(=O)NC(C)CNC(c2csc([N+](=O)[O-])c2)=O)c(F)cccc1[N+](=O)[O-] c1(C(=O)NCC2(F)CN(C(CC3(C=C)CCC3)=O)C2)cn2c(n1)CCCC2 C1(NC(C2CC=CC(NC(C)=O)C2)=O)CC2(C1)CC(C)C2 C1(C(=O)NC2C(C)(C)CN(c3ncns3)C2)CC(c2ccccc2)=NO1 C(C(C)(COC)C(=O)N1CC(C(N)=O)(CNC(=O)CC2CCC(C)(C)O2)C1)OC N1(C(c2ccc(OC)cc2)=O)CCCC(NC(=O)CCc2cc(C)sc2C)C1C c1(CC(=O)NC(C2CCCN2C(C2CCSC2)=O)C)nc2ccccc2o1 N1(C(=O)OC(C)(C)C)CCN(C(N(C(C)C(F)F)C(c2coc(Br)c2)C)=O)CC1 Cc1cnc2c(C(N3CCCC(CNC(=O)C(F)n4ccnc4)C3)=O)cccn12 N1(C(C(C)C2CC2)=O)CC2(CCN(C(c3ccc(F)c(Cl)c3)=O)CC2)C1 C1(C(=O)NCC(C(C)C)NC(C(C)=C(CC)C)=O)CCC(C)(C)OC1 n1(CC(=O)NC2CN(C(C3(SC)CC3)=O)CC2C)c(C)cc2ccccc12 C1(N(C)C)CCCC(C(N2CC(O)(CN(C(=O)CC3CCOC3)C3CC3)C2)=O)C1 C(=O)(CS(=O)(=O)C1CC1)N(C1(CC(=O)N(C)CC2CCOC2)CC1)C C(=O)(C(F)CC(C)(C)C)NC(C(=O)NC(C)CCCCCO)C1CC1 N1(C(C(C)NC(=O)NCc2c(CC)c[nH]n2)=O)CCN(C(C)C)CC1 Cc1cnc(C)c(C(=O)NCCC2CCCN2C(=O)CC2CC(C)=NO2)c1 c1(OC)ccc(CC(N2CC(NC(c3ccc(O)nc3C)=O)C3(CC3)C2)=O)cc1Cl C(=O)(C1=NOC(C)C1C)N(C)CC1(O)CCN(C(C2(C)CCNC(=O)C2)=O)CC1 CCC(C)(C(=O)O)N(c1ccccc1)C(c1cn(-c2cccc(Cl)c2)nn1)=O c1(NC(C2(CNCc3ccc(OCC)c(C)c3)CC2)=O)cc(F)c(C)cc1Cl C(C)(CCC(=O)NC1(CNC(=O)C(C)(C)n2cccn2)CCCC1)OCC c1(OC)ccccc1CC(N1CCOCC1CNC(=O)C=CC(C)(C)C)=O C(=O)(C1COc2ccccc21)N(CC(C)NC(C1CCC(=O)N1C)=O)C N1(C(=O)OC(C)(C)C)CC2CCC(CNC(C3(C)CSC(C)(C)C3)=O)C2C1 N1(C(C(CCSC)NC(=O)C=Cc2cccnc2)=O)CCN2C(=O)CCC2C1 C(=O)(C1=NNC(=O)C1)N(CC(C)NC(C1(c2ccon2)CC1)=O)CC CC1(C)CC(C(N2CC=CCC2)=O)CCN1C(=O)CCn1cccc1 N1(c2c(C)c(Cl)ncn2)CCC2CCC(NC(=O)CCC3CCC(=O)NC3)C1C2 c1(C(N(C2CCC(NC(=O)C(O)C(C)(C)C)CC2)C)=O)nccc2ccccc12 C1(SC2C(CC)C2)CN(C(C2C=CCN2C(=O)OC(C)(C)C)=O)CCO1 c1(C(N2C(CNC(C3CC(OCC)C3)=O)CC(CSC)C2)=O)nn(C)c(C)c1Cl c1(C(=O)NC2CC3CC(NC(c4c(C)cno4)=O)C3C2)cc(Cl)cc(F)c1N C(=O)(CN=c1[nH]c(=NCC2CCC2C(F)(F)F)c2ccc(C)cc2[nH]1)NCC=C C=C(C)C1CN(C(C2CCN2C(C2SCC=C2C)=O)=O)CCO1 CC1OCCC1C(=O)NC1CC(CC(=O)N(C)C)C1.C1C(=O)N1 Cc1c(F)ccc(NC(=O)CC2CCN(C(=O)Cc3ccc(Cl)cc3F)CC2)c1Cl c12nc(no1)C2.C(C(=O)NCCn1cncn1)(C1CC1)OC n1(C(C)C)ncc2cc(S(=O)(=O)Nc3cccc(I)c3)ccc12 CS(=O)(=O)c1ccnc(NCC2CCCN(C(C3CCCC3O)=O)C2)n1 C1(CNC(C2N(C(CCc3n(C)ccc3)=O)CC=C2)=O)CC12CCOCC2 C(C1=CCN(C(=O)CCN2CCCC2)CC1)NC(c1cncc(CC)c1)=O CC(=O)CCCC(=O)NCC1CN(C(=O)CCSC(F)(F)F)C2CC12 C1(C(N2CCN(C(=O)C(O)c3ccsc3)C3C2C3)=O)CCc2ccccc2C1 C1(CC(=O)NC2(CNC(c3n(CC#C)cnn3)=O)CCCC2)CC(C)(C)C(=O)N1 N1(C(C(C)=C(C)C)=O)CCC(C(=O)NCc2ccnc(O)c2)CC1(C)C N1(C(C2(F)CCN(Cc3cc(OCC)c(Br)cc3)C2)=O)CCCC(F)C(F)(F)C1 C1(C(N(CC(CN(C)C(c2cc(C#N)cs2)=O)O)C)=O)CC2CCC(C1)S2(=O)=O C1(CNC(C(CCC)OC)=O)CC(C)CN(C(C2(Cc3cccnn3)CC2)=O)C1 c1(C(N2CC(C(N)=O)(CNC(C3C(C(N)=O)C3)=O)C2)=O)cnn2c1CCCC2 c1(NC(C(c2cnn(C)c2)NCC)=O)ccc(C)nc1OC.C1(C)CCOC1 c1(C2(N3CCOCC3)CC2)cccc(Br)c1.C1(C2CC(F)O2)CCCN1CCN CCC(C(=O)N1CCC(c2ccccc2)(CNC(=O)C2=COCC2)CC1)C(C)C c1(OC)c(C(=O)NC2CC(C(=O)NC3CC(N4CCC4)C3)C2)cnn1C C1(C(N(CCCCCC)C)=O)(CNC(=O)CC2(O)CCOCC2)CC(C)(C)C1 N1(C(C2(CC)CC(=O)C2)=O)CCC(F)(C(N2CCCC2CC2CC2)=O)C1 Cc1cccc(C(=O)NC(C)C(C)NC(c2cnc(C3CC3)[nH]2)=O)c1C#N c1(-c2ccc(NC(C34CCCC3NCC4)=O)nc2)cccc(Cl)c1F N1(C(C2=CC(C)(C)C2)=O)CCn2ncc(CNC(c3cccc(Cl)c3F)=O)c2C1 C12(CNC(=O)NC3(C)CCSCC3)CCN(CC1)C(=O)NC2.C(C)(C)(C)OCC N1(C(C2C(c3nc(C)[nH]n3)C2C)=O)CC2CCCC2(Nc2cnc(C#N)cn2)C1 C1(NC(=O)CCCN2CCCC2)C2CC3CN(C(c4cc5scnc5[nH]4)=O)C1C3C2 CC(CC1CCC1)C(=O)N1CC(O)C1.c1(C(=O)NOC2(C)CSC2)nc(=N)[nH][nH]1 C(=O)(CCCC(=O)NCCCNC(C1CCCCN1C)=O)N(C)C C1(Cl)(C(=O)NCC2C(NC(C3(C(F)F)CC(=C)C3)=O)CC2)CC2CCC1O2 CCC(CC(F)F)C(=O)NCc1nc(C2CCCCN2c2ncc(Br)cn2)n[nH]1 N1(C(CCc2n(C)cnc2)=O)C2CCCC1CN(C(C1CCCCS1(=O)=O)=O)C2 Cc1nc2sc1NC(=O)C(C)CN1CCC2CC1.C1(C(=O)C2CC2)CCCOC1 N1(C(COCCOCC)=O)CC(C(=O)NC2CC(OC3CC3)C2)OCC1C C1(C(=O)NCC2N(C(CCCNC(N)=O)=O)CCC2)Cc2ccc(F)cc2O1 Cc1[nH]nc2c1CCC(C(N1CC(NC(c3ccn(CCF)n3)=O)C(O)C1)=O)C2 C(Cc1ccco1)(C(=O)NCCC1CCCC1)NC(C1C(C(C)(F)F)C1)=O c1(C(N2CC(C)C(CNC(=O)CCC3CCCC3)CC2)=O)c(N)cc(Cl)cc1F CCCCCCC(=O)NCC1C2CN(C(c3nc(C)oc3C)=O)CC12 C(=O)(C(C)CC(F)(F)F)NC(CN1CCN(C(c2ccc(CCC)s2)=O)CC1)C Cc1cnc2n1CCC(C(=O)NCCCN(C(=O)COc1ccccc1C)C)C2 N1(C(c2cc(NC(C)=O)ncc2)=O)CCC2(CCCC2NC(c2csc(O)n2)=O)C1 Cc1ccc2nc(C(=O)N(C)CCN(C)C(C3CCCO3)=O)ccc2c1 c1(SC)cc(C)ccc1C(=O)NCC1CCCN1C(C1COC(=O)C1)=O c1(NCC)cncc(C(=O)NCC(C)N(C(=O)C(c2c(C)noc2C)C)CC)c1 C1(C(=O)NCC(CC)C)(COC)C=CCN1C(c1ccncc1OC)=O Cn1ccc2[nH]c(C(=O)NC3CC(NC(c4c[nH]c(=O)cn4)=O)C34CCC4)cc12 N1(C(C2CCN(C(CCC)=O)CC2)=O)CC2CC1CS2=O c1(C(N(CCCN(C(C=NOC)=O)C)C)=O)ccc(NC(=O)NCCOC)cc1 C1(c2n(-c3c(OC)cccc3)nc(C3CC34CC4)n2)CC2(CCC2(OC)OC)C1 C1(CN(C(=O)CC2(c3cncnc3)CCCC2)CC)CCN(C(=O)CC)CC1 c1(C(N2CC(CC(C)NC(COCCC)=O)C2)=O)ccccc1N(C)C(C)C C1(C2CC2)(NC(COCC)=O)CCN(C(=O)C(C(C)C)n2cccc2)C1 c1(CC)conc1CC(=O)NC1COCC1n1cc(-c2csc(C3CC3)n2)nn1 n1(CC)ccc(CC(N2CCC(CN(C)C(c3csc(=N)[nH]3)=O)C2)=O)n1 C#CCC(C)(C(=O)N=c1cc(OC)n(C)[nH]1)NC(=O)CC1CCC(C#N)C1 C1(C)(C(=O)NC2(C)CN(C(N)=O)C2)CCN(C(=O)C(F)=CC2CC2)C1 c1(C(=O)OCC)ccccc1CNC(=O)C(F)(F)c1nc(C)cs1 C1(CCN(C(=O)CCNC(c2ccncc2)=O)C)CCCCN1C(=O)CCCF CCCCCCCC(O)C(F)(F)C(=O)NC(C)CN(C(=O)CC(C)(C)OC)C C1(C(C)CNC(=O)Cn2ccnc2)CCN(C(=O)C(C2(O)CCCCC2)O)CC1 C1(COC)(CNC(=O)CCn2ccc(C)n2)CCCN1C(c1ccccc1)=O c1(C(N2C(C(=O)NC(C(=O)OCC)CO)CCC2)=O)ccc(=O)n(C)c1 c1(C(=O)NC(CNC(c2sc(C)c(O)n2)=O)C(C)C(C)C)ccc(C)c(Cl)c1Cl C1(C(=O)NC2CCN(CC)CC2)CCN(C(=O)CCC2CCCC2)C12CC2 C1(CC)(CC)CCN(C(=O)C(C)(C(C)C)NC(=O)C(C)N=[N+]=[N-])CC1 N1(CC(CC(C)C)C)CCOC(C)(CNC(c2cnc(C(C)(C)C)o2)=O)C1 C1(C(=O)NCCC(C)CCNC(=O)Cc2ccoc2)CC2CCC(C1)C2F c1(C(=O)NC(C2CCCCN2C(=O)C2=CSCS2)C)cccc[n+]1[O-] C#CCCC(C(=O)NC(c1ccc(C)cn1)C)NC(=O)Cn1ccnc1C C1(C(=O)C(CCNCCNC(=O)CN)C)CCSC(C)C1.C1(C(C)(C)C)CCCC1 C1(CC#C)(C(=O)O)CCN(C(C2CCCN(CCc3ccc(Cl)cc3)C2=O)=O)CC1 C1(O)(C(C)NC(C=CSC)=O)CCN(C(C2CC(C)CO2)=O)CC1 C(=O)(C(CC(F)F)NC(=O)CN(C)C(=O)C1CC1)NCC(C(=O)NC)CSC c1(C(=O)NCC(F)CNC(C2CC=CC2)=O)cn(CC(F)(F)F)c(=O)nc1O CC(CNC(N1CCOCC(C(=O)O)C1)=O)CC(F)(F)F c12cc(ccc1F)NC2=O.N1(C(CCOC)=O)CC2CC1CN2C(=O)OC(C)(C)C N1(C(C2CC3(C2)CC(F)(F)C3)=O)CCC2OCCN(C(=O)CC3(CO)CC3)C2C1 CC1=C(C(=O)NC(C(=O)NCC2=CCCCCC2)C(C)(C)C)CCC1 C1(C(=O)Nc2ncc(C(C)=O)c(C)n2)CC2CCC1CN2Cc1c(Cl)cccc1Cl C1(OC)C(O)CC1N=c1[nH]c2ccccc2nc1N(C)CC1CC1 CC1(C)CCC(C)(C)c2ccccc2N1C(c1cn[nH]c1)=O C1(N(C)C(C2CCC(NC(=O)CC3(C#N)CC3)C2)=O)CCCC1(C)O C(CCC(=O)NC(C)CCCNC(=O)CC1CN(C)C1)OCCOCC CCC(O)C(C)(C)C(=O)N1CCN(C(c2ccnc(S)c2)=O)C(CO)C1 N1(C(C(C=C)O)=O)CCN(C(c2cn(CC)nn2)=O)CC1CCO CC(C)C(C(=O)O)SC1CC1.N12CC3CC1(C3)Cn1cc(nn1)C2=O N1(C(C(C(COC)C)C)=O)CCCN(C(=O)Cc2cc(OC)ccc2Cl)CCC1 C1(C(=O)NC2CCOC(CSC)C2)(OC)CCN(C(c2ncccn2)=O)C1 C1(NC2CCN(C3CCCN(C(=O)OC(C)(C)C)C3)C2=O)CCN2CCOCC12 CC1(C)NC(=O)c2ccccc2C1NS(=O)(=O)c1ccc(Br)s1 N1(C(C2(CC)CCOCC2)=O)CC2CCC(CNC(=O)C3=C(Cl)CCOC3)C2C1 CCC(CC(=O)NCCCCC1CN(C(=O)CNc2nccs2)C1)C(C)C N1(C(C(=O)NC)c2ccoc2)CCCC(CO)(CN(C)C)C1.C1(=O)C(C)(C)CN1 c1(C(=O)NC(CCC)C(=O)NCC2CCC(C)C2)ncc(F)cc1C C(C(C)(COC)C(=O)N1CCC(C(C)C(=O)NCC2(N(C)C)CCC2)C1)OC N1(C(C(C)NC(=O)Cc2cccs2)=O)CCC2CCN(C(c3cnn[nH]3)=O)CC12 CCC(CC(=O)N1CC(CCNC(=O)C=Cc2cnc(C)s2)C1)C1CC1OC C12COC3C(COC13)NC(=O)N2.c1(NC(CSC)=O)c(F)cccc1Cl S(=O)(=O)(c1ccc(Br)cc1)N(C(CN(C1CCSCC1)C)=O)CC1CC1 C(CCC1CC1)(C(=O)NCc1ccc(O)nc1)NC(c1cn(CC)nc1)=O Cc1nn(C)c(Cl)c1CNC(C1CC1NC(=O)CCOc1cccc(C#N)c1)=O N(C(=NCCOC(c1ccccc1)C(C)C)NC1CSC(C(F)(F)F)C1)C(CC)C CCC(C(C)C)S(=O)(=O)NC(C1CC(C2CCC2)C1)=O c1(C(=O)NC(C=C)C)cc(O)cc(F)c1.C12(C)CN(C1)C(=O)CC2 c1(SC)nccc(=NCC(CC(C)C)NC(=O)CSc2c[nH]c3ccccc23)[nH]1 N1(C(C(=O)NCC)=O)CCC(CNC(=O)C(C)C2CC2)(OC)C1 C(=O)(CC(C)O)NCC(C)CNC(=O)CCF C(=O)(CC(C(F)F)NC(c1ccc(C)c(OC)c1)=O)N(C)CC1CCN(CC)C1 C1(CCNC(CNC(CCC)=O)=O)CC(F)(F)CN1C(C1OCC2CCCC12)=O C1(CNC(=O)CCc2cncnc2)CC2CCC(C1)N2C(=O)C1=C(Cl)CCCC1 C1(C2CCC2)(C)CC1(F)F.C1(N(C)C)CN(C(=O)CSCc2ccccc2)CC1N Cc1ccc(C(C)(C)C(=O)N(CCC(C(C)C)NC(c2csc(F)c2)=O)C)cc1 C(=O)(C#CC1CCOCC1)N(C1(C(=O)NC(C2CCCC2)C)CCC1)C1CC1 N#CC1CCCC(C(N2CCCC(NC(=O)Cc3cncnc3O)C2)=O)C1 c1(C(C(N2CCCC(CCNC(C3C(C)C3)=O)C2)=O)(F)F)ccc(=O)n(C)c1 Cc1cc(CC(=O)NC2(O)CCCN(C(=O)C(C)OC(C)(C)C)C2)ccc1Cl N1(C(C(C)OCC=C)=O)CCC(O)(CNC(c2cccc[n+]2[O-])=O)C1 N1(C(c2c(C)n(C)cn2)=O)CCN(C(=O)CCc2ccc(F)nc2)CC1C c1(C(N(C2CCN(C(=O)C)CC2)CC)=O)cc2n(n1)CCNC2=O.C#CCOC c1(OC)cc(Cl)c(Cl)cc1CNC1CC1C(=O)OC.c12cc(cc(C)c1)CN2 c1(CCCC(=O)N2CC(=C(CNC(C3CC(C)(F)C3)=O)F)C2)ccc(F)c(F)c1 Cc1ccc(C(=O)CN2CCN(C(c3ccsc3)=O)C(C3CCC3)C2)cc1Cl CON1CCC(C(=O)NC2CN(C(=O)CSC(C)(C)C)CCC2C)CC1 N1(C(CC(C)OC)=O)CCC(C)(C(=O)NCCC(F)(F)F)C1 CC1CCN(C(C2CCCC2(F)F)=O)C(CNC(=O)C(C)(F)F)C1 c1(NCC2OCCN(C(C3(COC)CCCO3)=O)C2)ncc([N+](=O)[O-])cc1F c1(CN(C(C(C)(C)c2ccccc2)=O)Cc2cnn(CCO)c2)ccccc1F C(CN=c1cnc(N(C)C(c2ccsc2)=O)c[nH]1)c1cccc(C(=O)OC)c1 C1(C)(C(N(CCCCN(C)C(C2CCC2)=O)C)=O)CCCNC1=O C1(NC(CCC(=O)NC)=O)CCC2CN(C(c3ccn(C)c3)=O)CC2C1 N1(C(C(C)C(c2ccccn2)C)=O)CCC2C1CCN2C(=O)C(C)Nc1ccccn1 C12(CNC(C(CC)NC(N)=O)=O)CC(CN(C(=O)OC(C)(C)C)C1)C2 c1(C(=O)NC(CCCNC(Cc2c(C)non2)=O)C)cc2c(C)ccc(F)c2o1 Cc1cc(C(=O)NCC2CCN2C(C2NC(=O)C3CC23)=O)nn1C1CCC1 C=Cc1cc(C(=O)NCC(C)N(C)C(c2csc(CCC)n2)=O)cc(F)c1 CC(C)(CNC(=O)C(c1ccoc1)NC(=O)CC1CCCC(=O)N1)C(N)=O C1(NC(CC(CC)(C)C)=O)CC2CN(c3cc(C)c([N+](=O)[O-])cn3)CC2C1 n1(CC(=O)NC(CCC(=C)C)C)cc(C(=O)OC)c2cccnc12 c1(C(C(=O)NC2COCC2F)N(CC(=C2CCCCC2)C)C)cnn(C)c1Cl c1(C(=O)NCC(CNC(c2c(CCC)nsc2N)=O)C)cccc2cncn12 N1(C(C(CCCC)N(C)C)=O)CCC2(CCN(C(c3ccnnc3C)=O)C2)C1 c1(C(=O)NC2CCCN(C(c3cnc(CC)[nH]3)=O)C2)cnc2ccnn2c1N N1(C(CCC=C)=O)CCOC2(CCN(C(c3cnc4cc(C)nn4c3C)=O)C2)C1 c1(C(N(CC(=O)NCC(=O)NCC)C(C)C)=O)n[nH]cc1CC C(C)(C)(CC(F)C(=O)NCCC(=O)NC)NC(C=C(CCC)C)=O C1(CNC(c2c(SC)cccn2)=O)CC(F)(F)CN1C(=O)CC1CC(C)(C)C1 c1(OC)cc(C(C)(C)C)cc(OC)c1NC(=O)C(C)(C)O C1(n2cc(-c3c(C(=O)O)ocn3)nn2)(NC(COCC(N)=O)=O)CCCOC1 CCCC(O)CC(=O)N(C1(C=C)CCOCC1)C.C12CCN(C1)C2=O CC1CCC(=CC(N2CCC3CC23C(N2CCSCC2C)=O)=O)CC1 N1(C(Cc2cc(C)sc2C)=O)CCCCC12CN(C(c1cc(C3CC3)oc1C)=O)C2 c1(C(=O)NC2CC(CCNC(C(C)CC(C)(C)C)=O)C2)ccc([N+](=O)[O-])c(N)n1 n1(C(C)C)ncc(C(=O)NC2CCCN(C(=O)CC3CCCCO3)C2)c1Cl N1(C(CC)CC)C(=S)NC(c2cc(OC)ccc2F)C2=C1C1(CCC1)NC2=O C1(CNC)(CO)CCCN(C(C2(NC(C(CCC)NC(N)=O)=O)CC2)=O)C1 C(C(=O)NC1(CNC(=O)C2=CSCCO2)CCC1)(C(C)(C)C)OC O=S(=O)(c1nc(N2CCC3(CCCCC3)C2)ccc1Br)NC1CC12CCOCC2 N1(C(c2c(C)c(Br)no2)=O)CCOCC(NC(C2(C)CCCS2)=O)C1 N1(C(CSCCCC)=O)CCC(C(C)(C)C)(CNC(c2cncs2)=O)C1 N1(C(CCC2CCCN(C(CCC(=O)NCCC)=O)C2)=O)CCCC(C)(O)CC1 c12c(C)[nH]c(c1C)CC(=O)N2.N1(C(C)=O)CCOCC1C1CCOC1 N1(c2nccc(SC)n2)CCCC12CCN(Cc1cccn3cnnc13)C2 CCC(CC(=O)NC(CCCOC)C1CCC1)NC(c1oc(C2CC2)nc1C)=O c1(C(N2CC(CNC(C(C)NC(CCC)=O)=O)N(C)CC2)=O)cc2nnn(C)c2s1 C#Cc1cn(C)nc1C(N1CC2(C)CC1(C(=O)NC1CCC(C)(C)C1)C2)=O C1(NC(CCC=C)=O)CCN(C(=O)C(c2ccc(F)cc2)F)C(C)C1 c1(C(=O)NCCC2(CNC(c3n(CC)nnc3)=O)CC2)cc2c(s1)CCCC2 CC1CN(Cc2ccc(Cl)cc2)CCC1NC(=O)NC1(C)CCC(=O)N1C C(=O)(C1=CCCC1C)N1CCC(C(=O)NCC2(CC)CCOCC2)C1C C1(NC(C=CC=CCCCCC)=O)CCN(C(c2ccc(C)cc2Cl)=O)CC1C c1(OC)cc(CN(c2cnn(C3CCCC3)n2)Cc2ccccc2)cc(F)c1 C(CCC(C)C)(C(=O)N(C)CC1CCOCC1)NC(CC(CC)C1CC1)=O C1(NC(C(CSC)O)=O)CC2CCC(C1)N2C(c1ccoc1C)=O c1(CN2CC(NC(CC(CC)O)=O)C(F)(F)CC2)ccc(C)cc1[N+](=O)[O-] C=CCCCCCCC(=O)NCCOCCC(=O)NCCc1cnc(C)[nH]1 C(=O)(C(C)(C)CNC(=O)C(C)CN(C)C(c1cncc(C)c1)=O)NCC C(=O)(C1CCc2ccccc21)N(C)CC1(NC(c2c(OC)cncn2)=O)CC1 CCCCCCNC(=O)CCC1CCN(C(=O)Cc2cn(C)nn2)C1 c1(C(N(C(C)CNC(=O)CCCc2nncn2C)CC)=O)cc(Cl)cnc1O N1(C(C2ON=C(CC)C2)=O)CCCC(CC)(NC(c2cc(C)c(N)cn2)=O)C1 c1(CN(C(N2CCC(C)C2)=O)CC)cncc(NC(=O)C(=O)N(C)C)c1 Cc1ccc2sc(C(N3CC4CC(C3)C4NC(=O)CN3CCCC3=O)=O)c(C)c2c1 C(=O)(C1=C(Cl)CCC1)N1CCC(OCCNC(=O)C(O)CN2CCCC2)C1 N1(C(C(CSCC#C)O)=O)CCC(C(=O)NC)(CNC(=O)C2CC2)CC1 C#Cc1cccc(NC(C)C(N2CCN(C(=O)C(F)n3cccn3)CC2)=O)c1 C1(NC(CSCc2cccc(C)c2)=O)CCC12CN(C(c1cc(Cl)cnc1C)=O)C2 N1(c2snc(CCOC)n2)CC(NC(=O)Cn2c(C)c(C)sc2=O)CC2(CC2)C1 O=C1CC(=O)NC(C(=O)NCC2(F)CC(NC(=O)Cc3ccncc3Cl)C2)C1 Cc1cc[nH]c1C(=O)N(C1CN(C(=O)C(F)n2cccn2)C1)C c1(N(C(=O)CN2C3COCC2C3)C(c2cn[nH]c2)=O)ccccc1F C1(CNC(c2cocn2)=O)C(C2CC2)CCN1C(c1csnc1Cl)=O C12(CNC(C(c3ccc(C)cn3)(F)F)=O)CCC1CCN2C(c1ccc(C)s1)=O C=CC1CN(C(=O)C(C)NS(=O)(=O)CCCC)CC1NC(c1ncccc1C)=O c1(CC)cccc(CC(=O)NCCN(C(c2cc(C)c(Br)o2)=O)CC)c1 c1(C(N2CCC(C(C)NC(=O)Cn3nccn3)C2)=O)cnc2[nH]nnc2c1 C(=O)(C1CCCc2nc[nH]c21)NCC1(F)CC(CNC(=O)CCOC2CC2)C1 CC1C(=O)CC1C(=O)NCC(O)CNC(C1CCCN1C)=O C1(C(N(CCC(C(C)C)NC(c2ncc[nH]c2=O)=O)C)=O)CC2COCC(C1)C2 Cc1ccc(C(=O)NC(C)C=CC(N2CC3(CC3)CC2CO)=O)cc1O C(CCC(=O)N1CCCC1CC(=O)NCC=CCl)NS(C)(=O)=O C1(CNC(C(n2ncc(C)c2)C)=O)CC(O)CN1C(=O)C=Cc1ncco1 N1(C(C=Cc2cc(OC)ns2)=O)CC2CN(C(c3cc(C)c(O)nn3)=O)CC2(C)C1 c1(OC)c(C(=O)NC(CNC(=O)Cc2ccoc2)C(C)C)cccc1C(F)F C(CCC(O)C(=O)NCCCSCCO)NC(C(CCC)NC(C)=O)=O N1(C(C(CC)CC)=O)C2CCC(C2)C1CC(=O)NC1C=CC(COC)C1 Cc1nn(C(C)C)cc1C(=O)NCCC1CC(NC(=O)C(C)OCCC(C)C)C1 C1(C(=O)NCC2CC(NC(C(CC(C)C)C)=O)C2)CN2CCN1CC2C C1(NC(C(C)(C)O)=O)CCN(C(=O)C(F)(Cl)c2ccccc2)CC1 c1(OC)ccc(C(=O)N(CC(C)NC(C2(C)CCCO2)=O)C)c(C)c1 c1(C(N2C(CO)CC(NC(C3CCCS3)=O)C2)=O)c(Cl)ccc2c[nH]nc12 C(=O)(C(O)CCCc1ccccc1)NC(CC)CNC(C1(N(C)C)CCC1)=O FC(F)(F)C(F)(F)C(F)(F)CCN=c1nc2scnc2c(NCC2C3COCC23)[nH]1 C1(CC(C)NC(=O)CC2(C)CC2(Cl)Cl)CCN(C(c2nnn(C)n2)=O)CC1 CC1(C)CCCC(N2CC(O)(c3nc(-c4cc(Cl)ccc4Cl)no3)C2)C1 C1(CCCNC(c2cccc(=O)o2)=O)CCN(C(c2ccncc2F)=O)CC1 C(=O)(C1=CCCCO1)NC1CN(C(=O)C2=CCCC2)CC1F C(=O)(C1=C(C#N)CCC1)N1CC(C)(CNC(C=CCCC)=O)C(C)C1 c1(OC)cccc(C2(C(=O)NC3CCCC(NC(C4CCSCC4)=O)C3)CC2)c1 N1(C(C2C(CC)(CC)C2)=O)CCC(=CCNC(C2(SC3CC3)CCOCC2)=O)CC1 Cc1ccc2[nH]c(C(=O)NC3(C)CCCN(C(c4sc(C)cc4C)=O)C3)cc2c1 CC(=O)CCCC(C)C(=O)NC1(C(N2CCC3(CCC(O)C3)C2)=O)CCCCC1 c1(C(=O)NC2(CC(=O)N(C3CC(C(=O)OC)C3)C)CC2)cnc(O)o1.C(C)(=O)O C1(C(=O)NC(CCCNC(c2cn(CC)nc2C)=O)C)COC2COCC12 C1(NC(C(CC#C)C)=O)CC(C2CN(C(=O)COC(F)F)C2)C1 n1(CC(=O)N(CC(CNC(CC(C)(C)OC)=O)(C)C)C)cccc(C)c1=O C1(C(c2cnn(C)c2)NCc2c(OC)ccs2)CCC(NC(=N)N)CC1 N1(C(C(Br)=C(C)C)=O)CCC(C(C)CNC(=O)C(C)Cn2cccn2)CC1 c1(C(N2CCC(C(C)N=c3nc(C(C)(C)C)[nH]s3)C2)=O)ccc2ccncc2n1 C1(NC(c2ccc(C)cc2)=O)CCC12CN(C(=O)CC1CCCCN1C)C2 N(C1CCCc2c1cnn2-c1ccccc1)C(=O)NC1C(CS(C)(=O)=O)C1 CC1=C(C(=O)N2CC(NC(=O)CC(C)N(C)C)C(C)C2)S(=O)(=O)CCO1 CCC(CC)(CO)C(=O)N1C2CCC1C(C(=O)NCC1C3CCCC13)C2 C(C(C)(F)C(C)(C)F)c1cn(C2(C)CC3(CC3)C2)nn1.C12COCCN1C21CC1 c1(C(C(=O)NCC2CCCO2)N(CC)CC)ccc(C2OCCO2)cn1 c1(COC)ccc(C(=O)N(C2CCN(C(C3C=C(C)CS3)=O)C2)CCO)s1 CC(C)CCCC(C)C(=O)N(CC(C)(C)CNC(=O)CCC1CCOCC1)C C1(CNC(C)=O)C2CCC1CN(C(=O)Cc1cncnc1)C2.C1CCCC(=O)N1 N1(C(C(C)NC(CC)=O)=O)CC2(CO)CC1(C(N1CC(C(CC)CC)C1)=O)C2 CCC(CCC(=O)NCC(O)C(F)(F)F)NC(=O)CNC(=O)CN(C)C n1(CC)nc(C)c(C(=O)NCC2CCCCN2C(=O)C(=Cc2c[nH]cn2)F)c1C C1(NC(Cc2c(C)nc(S)s2)=O)CC(O)CN(C(=O)COCC2CC2)C1 C(=O)(C1Cc2ccc(Cl)cc21)N1CC(CNC(=O)Cc2cncs2)OCCC1 Cc1ccc(F)cc1-c1nnc(CN2CCCC2CS(N)(=O)=O)o1 C(C1CC1)(C1CC1)=CC(=O)NCC(C)C(=O)NC1CCN(CC2CC2)C1 Cc1cccc2cc(C(=O)N(C(C)CN(C(=O)CCn3ccnc3)C)C)cnc12 CC1CN(C(=O)C(F)(F)c2cccnc2)CCN1C(=O)CC1CCCC1 N(C1CCCc2ccoc21)C(C1=CCN(C(CCC=CC)=O)C1)=O c1(C(=O)NC2CCC2NC(c2cccc(C3CC3)c2)=O)ccc2oc(S)nc2c1 CC(CC(C)(C)C)C(=O)N1CC(C)(C)CC1CC(N1CCOCCC1C)=O C(=O)(C(C)(C)C(C)NC(c1cc(C)c(CC)o1)=O)NCC(CCC)O C1(NC(CC(C)OC)=O)CCN(C(c2cnn(CC3CCC3)c2)=O)C12CCC2 n1(CC)nc(C(N2CCOCC2CNC(=O)C(c2cnn(C)c2)OC)=O)cc1C C12(NC(CCCc3onc(C)n3)=O)CCCC1CN(C(c1cc(C)c(C)o1)=O)C2 CC1CC(NC(c2cc(C(F)F)nn2C)=O)CN(C(c2nn(C)cc2N)=O)C1 C(CNC(N)=O)(CCNC(C1(N(C)C)CC1)=O)OC C(=O)(CCCC(C)(C)CC)N1C(CC(=O)NC(C#C)C)C2CCC1C2 N1(C(C=C(C)C)=O)CCC2(CC1)CN(C(=O)CCC1CCC(=O)N1)C2C(C)C Cc1cc(C(N2CC(F)CC2CNC(=O)CCC(C)C)=O)cnc1F C(=O)(C(C)(O)C(C)C)N(C(C(=O)NC(C(=O)OCC)C1CC1)Cn1cccn1)C C1(C#N)(C(N2CC(N(C(=O)Cn3cc(Cl)cn3)C)C2)=O)CC1(C)C CCCCC(CC)C(=O)NCC(C)(F)CNC(=O)CCC1CC(C)C1 N1(CC(=O)NC(C2(C(=O)NC(COC)C3CCC3)CC2)C)CCOCC1 N1(C(C(CC=CC)C)=O)CC2(CC(NC(C34CCC(OC)C3C4)=O)C2)C1 CCCCC(CNC(=O)CC(C)n1cc(Br)cn1)NC(=O)CCSC Cc1[nH]c(C#N)cc1C(=O)NC(C)CC(N1CCC(C)(C(N)=O)C1)=O C1(O)(CC(N2CCC(CCO)CC2)=O)CCN(C(=O)CCn2cncn2)CC1 c1(NC(CC)=O)ccccc1C(=O)NCC(C)=CC(N1CC=CC1CSC)=O N1(C(C2COCCN(C(C(n3ccc(C)n3)C)=O)C2)=O)CC2(CNC(=O)C2)C1 C1(CNC(COC2(C)CCCC2)=O)CCCC(NC(c2cccnc2)=O)C1 Cc1ccn(C)c1C(N1CCCC(CCCCNC(c2cc(Cl)ccn2)=O)C1)=O Cc1nc(NC(N2CCCCC(C)C2)=O)c2ccsc2n1 Cc1cnc(C(=O)Nc2ccc(CO)nc2)c(Cl)c1 C1(C(N2C(CO)CC(NC(COCC=C)=O)C2)=O)CN2CCC1(C)C2 c1(C(C)=O)ccccc1C(N1CCC(C(=O)NCC(CO)CO)C1)=O C12(CC(=O)N(C3CCCN(C(c4snc(C)c4N)=O)C3)C)CCCN1CCC2 N1(C(c2c(OCCOC)scn2)=O)C2CCC1CC(OCCOC)C2 Cc1cc(C(=O)N(CCCC(=O)NC2CCN(C(C)(C)C)C2)C)c(C)n1C CC(CCC(=O)N(C(=O)CCc1nncn1C)CC(F)F)N1CCCCC1 c1(C(=O)NC2(C)CCCN(C(C3(CC4CCC4)CC3)=O)C2)cnn2cnnc2c1 c1(C(=O)NC2CCCO2)ccc(NCC(CC)NC(=O)OC(C)(C)C)cc1 c1(C(=O)OCC)cnc(Cl)cc1NC(C1CC1NCc1ccc(Cl)nc1Cl)=O C1(CNC(C(F)=CC)=O)C(C)CCN1C(=O)CCc1cn[nH]c1 N1(C(CSCCC)=O)CC(NC(=O)C(C2(O)CCOCC2)(F)F)CC12CCOC2 C(C1=NOC2CN(C(=O)C=Cc3nccs3)CC12)NC(c1nncs1)=O CCC(CC)C(=O)NCCNC(c1ccccc1C(C)=O)=O.C12CCCN1C2 n1(CCC)nccc1C(=O)N(C1CC1Cl)CCNC=O.C1CO1 c1(C(N)=O)cocc1C(=O)NCC1CCCN1C(=O)CC1CC2(CC2)C1 C1(O)(CCNC(C2C(=C)C2)=O)CCN(C(C2(C)CS(=O)(=O)C2)=O)C1 C#CCCCCCCC(=O)NCC(CC=C)C(=O)NCCNS(=O)(=O)CC C1(NC(c2c(OC)ccs2)=O)CCCC(C(=O)NCC2(CCO)CCCC2)CC1 C(N=c1nc2sccc2c(N2CCn3c(C4CC4)nnc3C2)[nH]1)C1OCCSC1 CCCCCCCC(=O)NC(CO)C(=O)NCc1ccc(C)c(O)c1 Cn1cc(CC(N2CCCC2C(C)(C)NC(C2(F)CC=CC2)=O)=O)cn1 N1(C(C(CCC)OCC)=O)C2CCC1CN(C(C1CCC(C(=O)NCC)C1)=O)C2 c1(CNC(C(=O)NC2CC3(CC(N)C3)C2)=O)ccc([N+](=O)[O-])cc1Cl C1(NC(c2cc3nc(C)sc3[nH]2)=O)CCN(C(=O)COCCF)CC(C)(C)C1 c1(CN2CC(NC(c3ccc(I)c(Cl)c3)=O)C(F)C2)csc2ccccc12 C(=O)(C1=C(C)CCOC1)NC(CCC)CNC(=O)CC1CCSC1 c1(OC)cc(C(N2CCCC2CCCNC(=O)CSCC2CCCCO2)=O)sn1 C1(COC(C(c2cccc([N+](=O)[O-])c2)C(C)C)=O)CC2COCC(C1)C2 O=[N+]([O-])c1c(Br)cc(CNCC2(CO)CC23CCOCC3)cc1Br c1(C(=O)NCC(C)N(C)C(C2CC2c2ccncc2F)=O)c[nH]c(=O)cn1 C1(NC2(CCOC)CCOC(C)(C)C2)(CO)CC2CC(O)C(C1)N2C c1(C(CC)NC(=O)Nc2ccc(-c3cccs3)cn2)ccc(-c2cscn2)cc1 C1(CNC(C2(C)CC(C)C2)=O)CCN(C(C2CC(C(F)(F)F)C2)=O)CC1C N1(C(C(CC)(C)CO)=O)CCC(C)(C)C(CNC(c2ccc(F)cn2)=O)C1 C1(=O)C(C)(C)CN1C1CCNC1=O.C(=O)(C(C)CC1CCCO1)OC C(=O)(C1=NOC2(CCC2)C1)N(C12CC(NC)(CO1)C2)c1ccc(CC)cc1 C1(NC(C(=CC2CCCC2)C)=O)CC2CC(NC(c3cc(C(N)=O)co3)=O)CC12 c1(C(=O)NCC(CC)NC(C2C3CCC(F)(F)C23)=O)cc([N+](=O)[O-])cnc1N C(CC(O)CNC(=O)CSCCC(C)C)NC(C1C(=C)C1)=O C1(N(C(C2C(CC)C2)=O)CCO)CCN(C(=O)CC2CCN(C)CC2)CC1 CC(=Cn1ccnn1)C(=O)NCC1(O)CC(NC(=O)CC(=O)NCC2CC2)C1 C#Cc1cccc(OC)c1.N12CCOCC1N(CC)CCCNC2=O.C1(=O)CN1 C1(CC)CN(C(C2CCCCN2C)=O)CC1NC(c1ccc(C(F)(F)F)[nH]1)=O C(CCCC(=O)NC(C1CCCN1C(=O)C(C)C)C)(OC)OC C1(C(N2CC(O)CC2CO)=O)CCN(C(C2(O)CCCCC2)=O)C12CCC2 CC1CC(=O)NC1C(=O)NC1(C)CC(NC(c2[nH]c(O)nc2C)=O)C1 C1(OC)CCCN(C(C(=O)NC2CCC(F)(F)CC2)C(C2CC2)OC)CC1 C(=O)(C(O)C1=CCCCC1)NC(CCC)C(=O)NCC(C)(C)N1CCCC1 N(C1CCC(NC(=O)C(CC)(CC)OC)c2ccccc21)C(C=CCN(C)CC)=O C1(NC(C=Cc2scc(C)n2)=O)C2CCCC1CC(NC(=O)C1=CCCC1)C2 N1(C(c2cnc(C(C)OCC)s2)=O)CCC(C2(NC(c3cc(O)no3)=O)CC2)C1 N1(C(C2(C)CCCCCN2)=O)CC2CC(Cc3ccccc3)C(C2)C1 C1(CC=C)(NC(=O)Cc2c(C)cnn2C)CCN(C(=O)CN(C)CCC)C1 C12CCCCC1NC(=O)CCN2C.C1(C(=O)NC2CCOCC2)CCC(C)CC1 C1(CC)CN(C(C2CS(=O)C2)=O)CC1NC(c1ccc(C#N)[nH]1)=O c1(C(=O)NC(CNC(CC(=C)C)=O)(C)C2CCC2)cc(=O)n(C)cc1Br C1(CCCCNC(C(C)OCC(F)(F)F)=O)CCCN(C(=O)CO)C1 c1(N2CC(CNC(c3c(OCC(=C)C)cccc3)=O)SCC2)oc(C)nc1C#N C(CCCCC(=O)NCC1CN(C(=O)CC#N)CCO1)OCC C1(OC)CN(C(C2(C3CCCN3C(c3c[nH]c(C#N)c3)=O)CC2)=O)CC1O c1(NC(C(=O)N(C(c2ccccc2F)C)C)=O)ccc(C(F)(F)C(F)F)cn1 c1(NCc2cc(C)[nH]n2)nc(N2CCC(N(C)C)C(C)C2)nc2c1cnn2C NC(=O)C1=NOC(CNC(C2CC(F)CCN2C(=O)CCc2csnn2)=O)C1 N1(CCNC(C(C2CCSC2)N(C)C(c2cc[nH]n2)=O)=O)CCCCCC1 C#CCCCCC(=O)N(CC=C)CC1C(O)CCN1C(=O)OC(C)(C)C c1(CC(C(=O)Nc2ccc(ON3CCCC3)cc2)O)c(F)cccc1Cl Cc1ccc(C)c(C(N2CC(O)(CNC(c3onc4c3CCCC4)=O)C2)=O)c1C c1(CC(=O)NC2C(CNC(C(F)=CC)=O)C2)ccc([N+](=O)[O-])c(N)c1 CS(C)(=O)=NCC(=O)NCC1CC(CNC(C2(CCOCC#N)CCCC2)=O)CO1 C(N=c1cc(C)nc(N(C)CCC2CCCCN2C)[nH]1)C1(OCC)CCCSC1 C1(O)(CN(C(c2c(C)scn2)=O)C)CCN(C(c2ccncn2)=O)C1 C1(OC)CN(C(c2cn[nH]c2)=O)CC1C(=O)Nc1cncnc1C C1(CC(=O)NC(CCNC(C2(CCOC)CC(=O)C2)=O)C)(OC)CCCCC1 C1(NC(C=CSC)=O)CCOC2(CCN(C(C3CC3CC(C)C)=O)CC2)C1 c1(C(=O)OC(C(C)C)Cc2ccc(Cl)cc2)nc2ccc(Br)cc2s1 c1(C(=O)NCC2C(C)CN(C(C3CNC(=O)N3)=O)CC2)cnn2ccccc12 C(C(C(=O)N(C)Cc1cnc(C)s1)NC(=O)Cc1cnnn1C)OC c1(CC)cnccc1C(=O)NCC1C2CN(C(=O)CNS(C)(=O)=O)CC12 c1(C(=O)NCCN(C(c2c(C#N)cnn2C)=O)CC)ccc(=O)n(C)c1 C(=O)(CC(C)(C)SC)NC1(c2ccccc2)CC(NC(COC2(C)CCC2)=O)C1 N1(c2n(C)c(C3CC3)nn2)CCC(C2CC2)C1C(c1ccccc1)n1ccnn1 C(C)(C(=O)NC(C(N1CCC(OC(C)=O)C1)=O)c1ccoc1)(C1CC1)OC C1(CNC(C(CC)C(C)O)=O)CCC2(CCN(C(c3sc(C)nc3C)=O)CC2)O1 CCC(C)(CO)C(=O)N1CC(NC(=O)COc2ccc(F)cn2)C2(CC2)C1 C12(C(N3CCC(C(C)C)CC3)=O)CC(CO1)N(C(C1(C(C)(C)O)CC1)=O)C2 CC1C(C(=O)Nc2nc(N(C)C)n[nH]2)CCCN1C(c1ccc(CN(C)C)[nH]1)=O CC(C#N)C(=O)N1CC(N(C)C(c2cc(C3CC3)no2)=O)C1 C1(NC(C(C#N)C2CC2)=O)C=CCN(C(c2sccc2C(N)=O)=O)C1 C1(C(=O)NCCC2CCCN2C(c2cc[nH]n2)=O)CCCCC12CC2 C1(CC)(CC)CNC(=O)C(CC)OCC(=O)N1.c1(Nc2cc[nH]n2)ccccc1 c1(N(C(C2CCC(COC)O2)=O)CC2(O)CNC2)ncnc(C(F)(F)F)c1Br C1(CCNC(c2ccc(OC)s2)=O)CC2CCC(C1)N2C(C1C2COCC12)=O C1(CCC)CN(C(c2cnc(C(C)=O)s2)=O)CCN1C(=O)Cc1ccn(CC)n1 c1(C(C(=O)NCC2N(C(CCCOCCC)=O)CCC2)(C)C)cnccc1C CC1CCC(NC(c2cc(C(F)F)n(C)n2)=O)CN1C(C1(C#N)CC1(C)C)=O N1(C(c2c(C)coc2)=O)CC(C)(C)OC2(C1)CN(C(C1CSCC(=O)N1)=O)C2 C(=O)(C(C)(F)C(=O)N(CCCNC(=O)COCC1CCC1)C(C)C)OC c1(C(C(=O)NCC(CNC(c2n(CC#C)cnn2)=O)OC)C)cccc(OC)c1 c1(SCC)nccc(=NCCCc2n[nH]c(=N)s2)[nH]1.C12(CCOCC1)CNC2 c1(OCC)csc(C(=O)NCC(C)(C2CC2)NC(c2cc(OC)cs2)=O)c1 C1(C(=O)NCCCCCCNc2c(C(N(C)C)=O)cncc2)CCCCNC1=O n1(CC(=O)N(C)CC2CCCN(C(c3c[nH]nc3C)=O)C2)ccc2ccccc12 c1(C(=O)NCCOC2CN(C(C(C)n3cccc3)=O)C2)cnc(CN(C)C)s1 N1(C(C2(C)CCCOC2)=O)CCC(C2CCN(C(C3CC4CCC3C4)=O)CC2)C1 C1(CNC(c2c(C)coc2)=O)(NC(C2CCNC2=O)=O)CCCCC1 CC1(C)CCC(C(=O)NOCC2CCOC2)CN1C(=O)CC1CCCC12CC2 CCCC(C(=O)N(C(C)CNC(c1nsnc1O)=O)C)S(N)(=O)=O CS(=O)(=O)c1cc(NC(=O)CCCNC(=O)NC2CN3CCCN2CC3)cs1 C(=O)(CCCCCN(C)C)NCC(CNC(c1c(CC)con1)=O)CO O=C(CCC#Cc1ccccc1)NCC1COCC1NC(C1(CO)CC1)=O C(C)(CCC(=O)NC(C)C(CO)NC(=O)C(c1ccnn1C)C)SC C(C(=O)N(C)OCC)NC(=O)CC1CCCC1O.C(C(=O)OC)CCC c1(C(N2CCC(O)(CNC(C(CC)C(C)C)=O)CC2)=O)cc(N)c(Br)c(F)c1 N1(C(C2CC3CC3C2)C(=O)NCCCSC)C2CCC1CN(C(C)C)C2 c1(NCCOC(C)C)ccc(C(F)F)c(F)c1 C(=O)(C1CCCc2nn[nH]c21)NCCc1c(CNC(C(CC)(C)O)=O)nco1 C1(CCNC(C2C(NC(C3CC(CC(=O)OCC)C3)=O)C2)=O)CCC(C)(C)O1 CCN(OC)C(=O)C(CC1CC1)NC(c1ccncc1C)=O c1(OC)ccc(C(N2CCCC(O)(CCNC(=O)Cn3cnnn3)C2)=O)c(O)c1 c1(-c2cc(CNC(c3coc(Cl)n3)=O)n[nH]2)cccc2[nH]c(C(F)(F)F)cc12 N1(C(C(=Cc2ccccn2)C)=O)CC2CCC1C2NC(=O)C1=CSCS1 CCCCC(CNC(=O)C=C(CC)CC)NC(=O)CC1(O)CCOC1 c1(C(=O)NCCC2CN(C(CCC=CC)=O)CC(C)O2)ccc(Cl)c(C)c1Cl c1(C(N2CCC(=CCNC(c3cc(C)sc3)=O)CC2)=O)cc(F)cc(Cl)c1O c12sc3c(c1N2C(C)=O)CCC3.C1(C)C(=O)O1.c1(NCC(=O)N(C)C)cocn1 C12(CNC(c3c(N)c(F)ccc3)=O)CCC(CN(C(=O)C3=C(Cl)CCOC3)C1)C2 N1(C(COCC#C)=O)CC(NC(c2ccc(C(F)F)cn2)=O)C(C)(C)C1 C1(COC)(CC)CC(NC(C2C(CNC(COCC(=C)C)=O)C2)=O)C1 c1(CNC(C(=O)Nc2cccc(C3CCCN(C)C3)c2)=O)ccc(F)c(N)c1 Cc1cccc(Cl)c1C(=O)NC1CCC(NC(c2cc(Cl)ns2)=O)CC1 Cc1cnn(C(C)C(=O)NCC(C)(C2CCC2)NC(=O)CC(C2CCC2)C2CC2)c1 c1(C(=O)O)cc(C(=O)NC2CC2c2cccc(F)c2F)cc([N+](=O)[O-])c1 C1(CNC(C2C(C(C)(F)F)C2)=O)CCCC(NC(=O)CCc2csnn2)C1 N1(C(CCCOCC)=O)CCCC(NC(c2cn3ccsc3n2)=O)C1C N1(C(CCC(=C)Cl)=O)CCN(C(C2(C3CC3)CC2)=O)CC1C1CCC1 c1(S)cccc(Br)c1F.c1(C(=O)OC)ccncc1NC(C1(N(C(=O)CC)C)CC1)=O Cc1nc(CCCNC(=O)CC(C2CC2)NC(=O)C=Cc2cncs2)n[nH]1 c1(OC)ccc2cc(C(N3CCCCCC3CNC(=O)C(C)OC)=O)[nH]c2n1 C1(O)(C(=O)NCC2(NC(CC3(OC)CC3)=O)CCCC2)CCC(C)(C)CC1 C=C(Cl)CCC(=O)NCC(C)NC(c1coc(-c2cnn(C)c2)n1)=O CC1C(NC(C2C3(CC3)C23CC3)=O)CCN1C(=O)CN1CCN(C)CC1 C(=O)(CCCC(C)N(C)C)N1C(CN(C(CNS(CC)(=O)=O)=O)C)CCC1 Cc1cccc(C(O)C(N2CCC(NC(=O)Cc3nccn3C)C2)=O)c1 C(c1nc2ccccc2s1)=CC(=O)NC1CCC1NC(C1CCCCC(=O)N1)=O N1(C(CC)C(N)=O)CCCC(CCC(C)C)C1.C1(C(=O)N)(CN)CC1 Cc1cc(F)c(C(=O)NCC2(NC(=O)C#CC3CCC3)CCC2)c(Cl)c1 c1(C(N(C)CC2CC3CC3N2C(=O)C(O)C(C)(C)C)=O)c(F)cc(Cl)cc1F CCC(C)(C)C(O)C(=O)NCC(C)NC(c1coc2c1CCCC2)=O c1(C(N2CCCC(N(C)C(c3ncncc3F)=O)C2)=O)cc2ccsc2c(O)n1 C1(C)(CNC(c2c(C)n[nH]c2)=O)CN(C(C2CCOC2=O)=O)C(C)(C)C1 C1(CNC(C(C)SCC)=O)CN(C(c2cc(C(C)=O)[nH]n2)=O)CCC1(F)F NS(=O)(=O)c1n[nH]cc1C(N1CC=CC(NC(=O)CNC(=O)C(F)(F)F)C1)=O N1(C(C2N(c3ccnc(C)n3)CCCCC2)=O)CCCC(N=[N+]=[N-])CC1 N1(C(CC2(C)CCCO2)=O)CCN(C(=O)C(F)n2cccn2)CC1 N1(C(c2nccc(CC)c2)=O)CCC2C(CCCN2C(c2ncn(CC)n2)=O)C1 c1(NC(c2c(C(N(C3CC(OCC)C3)C)=O)c(C)co2)=O)cccc(OC)c1 C1(C(C(=O)NCC(C2CCCC2)NC(CN(C2CCCC2)CC)=O)F)CCCCC1 N(C(=NCCCOC(F)(F)F)NC1CC1C(F)F)CCC N1(C(C(CC)=CCCC)=O)CCC2(CCCCN(C(=O)C(C)(C)CC(C)(C)C)C2)C1 c1(C(N(C2CCN(Cc3nc(CC)sc3)C2)C)=O)cnn2cccnc12 c1(CC(=O)NC2C(CNC(CC(=C)C)=O)CC2)c(F)cccc1Br c1(C(=O)NC(CC)CN(C(=O)C(C)OCCOC)CC)cnc(C(C)(C)C)o1 c1(C(N2CC3(CC(NC(C4CCCCS4)=O)C3)C2)=O)cc(Cl)cc([N+](=O)[O-])c1O C(C(C)(C)C(C)(F)F)OCC.C1CC(=O)N1.C12(CC1)C(=O)N2C Cc1nn(C)c(C(=O)NC2CCC2NC(c2ccsn2)=O)c1Cl C=CCC(C)(C)CNC(=O)C(C1CCN(C(C2(CSC)CC2)=O)C1)F C1(N(C(=O)Cn2[nH]cnc2=N)C)CCN(C(=O)C=CC2CCOCC2)CC1 c1(C(C(=O)NC2CC(C)(NC(C(C)SC)=O)C2)F)ccc(C(F)(F)F)cc1 N1(C(CSc2n(C)cnn2)=O)CCCC12CCN(C(c1c[nH]c(C(N)=O)c1)=O)C2 c1(C(=O)NC2CC3CCCC(C2)N3C(=O)C(F)F)cc2nccc(Cl)c2s1 c1(NC2C(=C)C2)nc(=NCc2nc3cc(Cl)ccc3s2)nc(N2CCOCC2)[nH]1 N1(C(C(CC)C)=O)CC2(C)CC1(C(=O)NCCCC(C)O)C2 N1(C(Cc2c(C)non2)=O)CC(NC(=O)C(C)OCC2CCC2)CC12CCCC2 C1(C(=O)Nc2nn(C)c(C)c2Br)COC2(CCN(Cc3c(C)scn3)CC2)C1 c1(NC(C)=O)cnc(O)c(C(C(=O)CC2(C)OCCO2)=O)c1.C(CC1CCC1)N C1(CNC(c2c(CC)scc2)=O)CC2(CCC2)CN1C(=O)C(C1CCOCC1)C C1(C(N2CCC(N(C(C3CC(C(F)(F)F)(OC)C3)=O)C)C2)=O)CCCCNC1=O C#CCCCC(=O)N(C1C2CN(C(c3scnc3Cl)=O)CC12)C Cc1c(C(=O)NC2C(OC(c3ncccc3Cl)C)CCCC2)cnn1C(F)F c1(C(N2CC=CC(NC(CCc3c(C)n[nH]c3C)=O)C2)=O)ccc2nccn2n1 c1(C(N2CC(C(C)NC(CCNS(CC)(=O)=O)=O)C2)=O)ccc(C2CCC2)nc1 N1(C(C)C)CC(C(=O)NCC2CC(NC(c3cc(C(F)F)no3)=O)C2)CC1=O c1(CC(=O)NC2C3CCC2N(C(=O)C2=CCCC2)C3)ccc2nc(O)[nH]c2c1 CN1C2CCC1CC(C(N1CC(CNC(=O)CCc3nncs3)C3(CC3)C1)=O)C2 N1(C(C2N(CC)CC2)=O)CC(CO)(NC(c2n[nH]cc2CC)=O)C1 CC(C)C(O)CCN=c1[nH]c(=NCc2c[nH]nc2OCCO)c2ncccc2[nH]1 c1(CCC(N2CC(n3cc(-c4c(C)ocn4)nn3)C2)=O)ccc(Br)cc1 c1(C(=O)NC(CC(C)NC(Cc2c(C)n(C)nc2)=O)C)n[nH]c2c1CCSC2 Cc1ccc(C(=O)NCC2C=CCN2C(=O)Cc2nncn2C)cc1C C1(C(=O)NC(CCC)CO)CCN(C(c2c[nH]c(=NC)s2)=O)C12CC2 C(=O)(C1=CCCN(C(=O)CCN(CCCO)C2CC2)C1)N(c1cnc(C2CC2)o1)C c1(SCC(=O)NCC(C2CCC2)NC(CCC2CC(OC)C2)=O)ccccc1Cl C1(CN(C)Cn2cc(C(=O)NC)nn2)CC(C)OC1=O N1(C(N(c2cncc(-c3cncn3C)c2)C)=O)CC(F)(F)OC(F)(F)C1 C1(C(=O)NC2C(NC(C3(OC)CC3)=O)C2)CC(C(C)C)C1 c1(CCC)cc(C(=O)NC2(C3CCCN3C(=O)C(C3CCC3)OC)CC2)cc(O)n1 C(=O)(C(C(=O)N(C1CCCCC1NC(C12CC(C)(C1)C2)=O)C)C(C)(C)C)OCC C1(C(=O)NCC(CNC(c2ccc(CC(C)(C)O)s2)=O)O)CC=CCC1C CCCCCC(C)CC(=O)NC(C)CCNC(C1CNC(=O)CC1C)=O N(C1c2ccccc2CC1O)C(C(=O)NC1C(CC)(CC)C(OC)C1)=O N1(C(CC(=O)NCC#C)=O)CC=C(CNC(C2CNC(=O)N2C)=O)CC1 Cc1oc(C(C)C)nc1C(=O)N(CC(C)NC(C1CCN(C)C1=O)=O)C c1(C(N2CC3C(CCNC(CC=C)=O)(CC3)C2)=O)nc2ccccc2cc1Cl C(C1CCCN1C)=CC(=O)N(C1CC(C(NOCC2CC(=C)C2)=O)C1)C Cc1ncoc1CNC(=O)CC1(NC(c2cc(C)on2)=O)CC1 C1(N(C(c2cncnc2)=O)CC)CCCN(C(=O)C(C2CC2)C2CC2)C1 C1(O)(C(N2CCC(NC(C(=O)NCC)=O)C2)=O)CCSCC1 c1(C(=O)NC(CN(C(CC2C(C)OCC2)=O)C)(C)C)ccc(C#N)[nH]1 c1(C2C(C(N(C3CN(C(=O)C(F)(F)c4ccnn4C)C3)C)=O)C2)ccc(F)cc1 Cc1cnn(CCC(=O)NC2(CNC(=O)CN3CCCC3=O)CCOC2)c1 Cc1cc(CCC(=O)N(CCCNC(=O)CC2CCCC(C)(C)C2)CC)cc(C)n1 CC1(C)CCC1C(=O)NCC1(CNC(C2CS(=O)(=O)C2)=O)CCC1 c1(NCC2N(C(c3cc(NC(C)=O)cn3C)=O)CCCC2)ccc(C#N)c(Cl)c1 C1(NC(CC2CCN(C)C2=O)=O)CCCN(C(c2nccc(Cl)c2F)=O)CC1 c1(C(=O)NCC(C)(C)CNC(C23CCCCC2OCC3)=O)cccc2ccoc12 c1(C(=O)NCC2(O)CN(C(C3CC(=O)N3)=O)C2)ncc(Br)cc1F C(=O)(C=CS(C)(=O)=O)N1CCC(CNC(CNC(c2ccc(C)s2)=O)=O)C1 N1(CCC)CC(C(=O)N(CC(C)(C)NC(C23CCC2C3)=O)C)CC1=O c1(C(=O)NC2CCC(C)N(C(c3nccnc3N)=O)C2)c[nH]c2cc(Cl)ccc12 N1(C(CCSCCC)=O)C2CCC1CC(CNC(=O)C(C)(C)n1cnc(C)c1)C2 c1(OC)ccc(Br)c(C(=O)NC2C=CC(C(N3CC4CC3CO4)=O)C2)n1 C(=O)(C1=C(C)OCCS1)NC1C2CN(C1)C(=O)C(C)(C)S2.N1(CC)CCOCC1 Cc1cccc(-c2cc[nH]n2)c1F.C12CC(C1)N(C1CC1)C(=O)C(=O)OC(=O)CO2 CC(C)C(O)C(C)C(=O)N1C2CCC(C(=O)NCC3CCC(C)C3)C1CC2 C1(NC(C2CC3CC2C3)=O)Cc2ccccc2C1NC(=O)C(F)(F)C(F)F CCC(C)CC(=O)C(=O)NC1CCCCCC1C(N1CC2CC1CS2=O)=O C1(NC(C2(NC(CC3CCN(C)C3)=O)CCCCC2)=O)CCC(=O)N(C)C1=O C(=O)(C(C)OC1CCCC1)N(CC(=C)Cl)CSC C1(NC(C2C(C)=CCS2)=O)CCC(C)(CNC(=O)CN2CCNC(=O)C2)CC1 c1(C(N(C)Cc2cc(C)c(O)c(C)c2)=O)ccc2c(c1)CC(=O)N2C C12(CNC(CC3(C=C)CC3)=O)CC3CC(CC(C3)C1NC(=O)C(F)CC1CC1)C2 Cc1cn2c(n1)CCC(C(=O)NC1CC3CC(O)C1C3)C2 C1(C(N2CCC(C(N(C)C)=O)CC2)=O)CCC2CCC1N2C(=O)CCCCN=[N+]=[N-] c1(C(=O)NCC(CCC)NC(C2CCC(NC(N)=O)CC2)=O)cccc(Cl)c1 N1(NC2CN(C(C3CCC(C)S3)=O)C2)CCN(C(C2(S(N)(=O)=O)CC2)=O)CC1 S(=O)(=O)(c1c(Cl)cc(Cl)cc1Cl)N1CCC2(CCCN(C(C(C(CC)C)O)=O)C2)C1 N1(C(C2CCN(c3ccc(C)cc3)C2=O)=O)CCN(C)CC12CCC2 c1(C(C)=O)ccc(C(N2CCC(N(C(=O)CSCC3CCCO3)C)C2)=O)[nH]1 Cc1ccc(F)c(C(=O)NC(CCN(C(=O)CCCCC(F)F)C)C(C)C)c1O CCCC(C)(O)CNC(=O)CCOCNC(=O)C(C)N1CCCC1.C(CCN(C)C)O NC1CCCC12CCN(C(=O)Nc1cnn(-c3ccccc3)c1)CC2 C1(NC(=O)CCSC2CC2)CC=CCN1C(=O)C(O)CC1CCC1 c1(C(CC)NC(=O)Cc2ccccc2F)ccc(OCC)c(OC)c1 C=CCCCCCC(=O)NC(C)CC(C)NC(c1cc2sccc2[nH]1)=O N1(C(C2(COC)CC2)=O)CC(C(=O)Nc2cnccn2)C(n2ccnn2)C1 C=CC(O)(C(=O)NC1CN(C(c2ccc(CSC)o2)=O)CC1OC)C(F)(F)F c1(C(N2CC3CCN(C(c4cn(C)c(O)n4)=O)C3C2)=O)cc2ccc(Cl)cc2o1 c1(C(=O)NCC23CC(NC(CCC(C)SC)=O)(C2)C(C)O3)cc2c(ncn2C)[nH]1 C1(NC(C=CSC)=O)CC(NC(C2CC2c2cncn2C)=O)C(O)C1 C(=O)(C(CC1CC1)NC(c1ncoc1C)=O)NCC(C1CCC1)OC N12CCC(C)C(C1)CC2=O.c1(OC)ccccc1OCCC(=O)OC C1(C(N(CCOCC#C)C)=O)CCC(CNC(C2C3CCC(F)C23)=O)CC1 N1(C(c2cc(C)c(N)cn2)=O)Cc2nccn2CC(NC(C2CC2(C)C)=O)C1 Cn1cc(C(=O)NCCN(CCCN(C)C)C(C2CCO2)=O)c(-c2cccs2)n1 Cc1ocnc1C(=O)N(CC(N1CC(N(C(=O)CCNC(N)=O)C)C1)=O)C c1(OCC)cc(CNC(C(C2CCC2)OC2CCC2)=O)[nH]n1.C12CC(C1)NC2=O CC1(C)CC(CO)CN1C(=O)CCC1CCCN(C(c2sccc2Cl)=O)C1 N1(C(c2occ(C)c2)=O)CC2(CCN(C(=O)C=Cc3ccccc3Cl)C2)C1 N1(C(C(c2ccccc2)N(C)C)=O)CCC(CNC(=O)CC2CC=CC2)C1 CN1CCOC(CC2CCN2C(c2cccc(-c3cn(CCO)nn3)n2)=O)C1 C(=O)(CN=c1[nH]c2ccccc2s1)NCCN(C(C(COC)C)=O)C CC1CC(NC(=O)CSc2ccccc2)CN(C(=O)CCc2n[nH]c(=N)s2)C1 C(CCCCC(=O)N1CCN(C(c2n[nH]cc2C(C)C)=O)CC1)SC C(CCC(=O)NCC(O)CCC)NC(CCSCCOC)=O O=C1NCC2CCC1N2N1CCCC(c2n[nH]c(C3CC3)n2)C1 n1(CC)c(C(C)NC(=O)N=c2[nH]ncn2C)cc2ccccc12 N1(C(COCCCC(C)C)=O)CCC(NC(C2CC(CC(F)F)C2)=O)CC1C CC(CCCc1ccccc1)C(=O)N(c1ccc(I)c(Cl)c1)C1CCC1 c1(SC)cc(N2CCN(C(=O)CCc3ccccc3)CC2)nc(SC)n1 C(=O)(C(CC(F)F)NC(=O)C=Cc1cnccn1)N(C)Cc1ncco1 O=C(CCS(=O)(=O)c1ccc(F)c(F)c1)NCC(O)COc1ccnn1C(F)F C1(CNC(C(C)c2ncco2)=O)CC12CCN(C(c1ccoc1Cl)=O)CC2 C(C(CC(=O)Nc1cccnc1)C(F)F)NC(C(C)(C)N(C)C)=O C(=O)(C1Cc2c(Cl)cccc21)NCC1C(NC(c2ccnc(OC)n2)=O)COC1 C(Cn1cc(C(O)C(C)C)nn1)(CC(F)(F)F)NC(c1c(C(=O)OC)cnn1C)=O N1(C(CSc2ccc(C)s2)=O)CCC(N2C3CCC2CC3)C2(CC2)C1 N1(C(c2ccc(COC)s2)=O)CC2CCC1C2NC(=O)CC1CCCC1O Cc1ncsc1CCNC(=O)C=CCC(C)(C)NC(=O)CC1CCC2CC12 C(C1CCN(C(=O)CCC2CCCCO2)CC1)=CC(=O)NCc1ccc(C)o1 C=CCCC(C(=O)NCC(C)CC(=O)NC)NC(c1cnc2n1CCC2)=O c1(CCCC)sc(C(=O)NC(C2CCCN(C(=O)C=CCO)C2)C)cc1C N1(C(C=COCC)=O)CCC(C2CCN(C(c3cn(C4CC4)nn3)=O)C2)C1 CCC(C)(CN=c1[nH]c(N2CCC=C(c3ccncc3)C2)nc(=N)[nH]1)C(N)=O c1(C(N(CC(C)O)CCNC(C2(C)CCCCC2)=O)=O)ccc2c(c1)nnn2C C(C1=Cc2cc(Cl)ccc2OC1)NCCC(C)S(C)=O C1(NC(C(n2c(C)ccn2)C)=O)CCCC(NC(=O)C(C)NC=O)C1 O=C(CS(=O)(=O)CCO)NCCC1CCCN(C(C2CC3C=CC2O3)=O)C1 c1(OC(C2CCOCC2)=O)cc(N2CCCC2)ccc1F.C1(=O)CCN1C CC1(C)CC(C(N2CC(OCCNC(C3CC=CCC3)=O)C2)=O)CNC1=O N1(C(C(c2c(C)n[nH]c2C)C)=O)CCN(C(C2CC2(C)C(C)C)=O)C(C)C1 C(CC(=O)NC1CCOC1C)(C(F)(F)F)NC(CCCC=C)=O S(=O)(=O)(CC(=O)N1CC(C(O)C(=O)NCCCCCSC)C1)NC C1(NC(COCCSC)=O)CC2CCC1(CNC(C1CC1c1ccnn1C)=O)C2 C1(CCCOC)CCN(C(=O)CC2CC2COC)CC1.c12ncsc1C(=O)NC2 CN=c1[nH]cc(C(N2CCSCC2C(=O)NCC#CC#CCO)=O)o1 c1(C(=O)OCC(c2ccccc2)CC)c(C)ccc2nsnc12 c1(C(=O)NC2CCCN(C(CC=CCC)=O)C2)ccc2c(c1)oc1ccccc21 c1(C(N2CCC(C(CNC(C(CC)O)=O)(C)O)CC2)=O)ccn2cncc2c1 N1(C(c2c(C)con2)=O)CCN(C(c2ncncc2Cl)=O)C2COCC12 CCC(C)(O)C(=O)NCCN(CC(=O)OC)Cc1ccccc1Br C(=O)(C(C)CS(C)(=O)=O)N(C(CC)CC)CCNC(=O)CS(=O)(=O)CC N1(C(c2cnn(C)n2)=O)CCC2CC1CN(C(=O)CCn1cncn1)C2 C(=O)(C(CCS(C)=O)N(C)C)N(C1CN(C(C2(C)CCCNS2(=O)=O)=O)C1)C c1(CNC(C2C(NC(c3n(C)nc(C)c3F)=O)C2)=O)c(O)cc(F)cc1F CCC(CC)(CN=c1[nH]c(N2CC(=O)NC(C(C)C)C2)nc(=N)[nH]1)NS(C)(=O)=O C1(C(N(C2CC(NC(C3(c4ccncc4Cl)CC3)=O)C2)C)=O)CC2CCC1O2 O=C1Cc2c(C(=O)NCC(F)CNC(=O)C(F)n3ccnc3)ccnc2N1 N1(C(C2N(C(Cc3cncc(C)c3)=O)CC(C)CC2)=O)CC(O)(C2CCC2)C1 c1(CCCC(=O)NCCN(C(=O)Cc2ccc(OC)cc2)CC)ccc(Cl)cc1 N1(C(C2CC(C)=C(C)CC2)=O)CC2=C(C1)CN(C(=O)CCS(C)=O)C2 C(=O)(C1CCCc2sccc21)N1C(C)CN(C(c2c(C)nc[nH]2)=O)C(C)C1 C(CC(N)=O)(C(=O)NCC1(F)CCCN(C(=O)NC2CC2)C1)NC(C)=O c1(CNC(=O)NCc2c(C)nn[nH]2)c(OC(F)F)cccc1Br CC(C)C(C)(O)C(=O)NC1CN(C(=O)Cc2ccon2)C(C)(C)C1 S(=O)(=O)(c1ccc(Br)cc1N1CCC(C)(OC)C1)NC1CN(CC)C(C)(C)C1 c1(C(C)NC(C2C(OC)C(O)C2)=O)ccc(CN=[N+]=[N-])cc1 C#CCCCCCC(=O)NC1CCN(C(c2cnoc2C)=O)C1(C)C c1(C(=O)NC2(CC=C)CN(c3ncc(F)c(OC)n3)C2)ccc2occc2n1 N1(C(C(CCC#C)O)=O)CC(NC(c2ccc([N+](=O)[O-])s2)=O)C(C2CC2)C1 C1(CF)(NC(C2CCN(C(CCC)=O)C2)=O)CCN(C(=O)CCc2cncnc2)C1 C(=O)(C1Cc2c(Cl)cccc21)N1CC(C)(CNC(CC2(CSC)CC2)=O)OCC1 C1(CNC(c2ccn(C)n2)=O)CC2COCC2N1C(c1ccccc1)=O C1(CN(C)C(N)=O)CCCN(C(C2CC23CCCC3)=O)CC1.C12(CCCC1)C(=O)N2 Cc1cnn(C(C)C)c1NC(=O)NC(C1CCOC1)CO C1(C(N2CC(n3cc(CN(CC(C)(C)C)CC)nn3)C(C)C2)=O)CC(=O)NC(=O)N1 C(=O)(C(O)C(C)(C)CC)NCC1N(C)CCN(C(Cn2cc(C(=O)OC)nn2)=O)C1 N1(C(COCC)=O)CCC(N2CCN(C(c3csnc3Br)=O)CC2)CC1 N1(C(c2cc(OC)ns2)=O)CCC(C2CCN(C(c3ccnn3C)=O)C2)CC1 N1(NC(c2scc(CSC)n2)C2(c3ccccc3)CCC2)CC(CC)OC1=O N1(C(CCN(CCC)C)=O)CC(CC(=O)NCC2CCOC2(C)C)CC1C c1(C(c2nnnn2-c2ccccc2)NCC(C)OC)cc(F)c(F)c(F)c1 c1(OC)ccc(N2CCNCC2)cc1NC(c1cnc(-c2nn[nH]n2)cn1)=O c1(-c2nc(CCCCCC)nn2C(c2ccncc2)C)ccc(F)cc1Cl c1(CCNC(c2nnnn2Cc2cccs2)C(C)C2CCCO2)occc1Br c1(C(=O)NC2CCN(C(C(CC)(C)O)=O)CC2)ccc(-n2cncn2)c(C)c1 N1CCC(C(=O)NC(c2ccon2)=O)C1.CC(C)(C)OC(=O)NC1CC1CF Cc1ccc2c(C(N3CC(C)N(C(=O)CC4CC4)CC3C)=O)n[nH]c2c1 C1(N(C(C(C=C)O)=O)C)CN(C(c2cccc(OCC(F)(F)F)n2)=O)CC12CC2 N1(C(CNC(C)=O)=O)CCCCC(NC(=O)COc2ccccc2C(C)C)CC1 Cc1cc2c(CCNC(CCS(N)(=O)=O)C(=O)N(C)C)csc2s1 c1(NC(=O)C(F)C2CCCC2)ccc(C#N)cc1.C12CC(C1)C(=O)NCCN2C Nc1c(C(=O)NCCN(C2CCCC2)C(C2CC3CC23)=O)cccc1F N1(C(c2n(CC)nnc2)=O)CCCC1(C)C(=O)NCC(C)(C)C1CCC1 c1(-c2ncc(NC(CCS(C)=O)c3nnnn3C3COC3)s2)ccc(Cl)cc1Cl C12(CNC(C3CCCN(C)C3)=O)CCC(CNC(C(CC)C(C)C)=O)(CC1)CO2 n1(CC(=O)NCC2CC(C)(C)N(C(C3CCOC3)=O)C2)nc2c(n1)CCCC2 Cc1cc(C(N2CC(CNC(=O)CCN3CCOC3=O)C3CC23)=O)cn(C)c1=O CC(C)CC(C)(CNC(C1CN2CCC1CC2)=O)NC(=O)C(C)OC(C)(C)C Cc1oc(-c2cccs2)nc1CC(N1CCOC(CN2CCCC2)C1)=O c1(C(=O)NCCN(C(c2cn(CCC)nc2C)=O)C)cnc(O)c2cccnc12 N1(C(C2(C)CCN(C)C2)=O)CCC(CO)(CNC(C2C3CCN2CC3)=O)CC1 c1(OC)ccc(CCNC(=O)C(N2CCOCC2CN2CCOCC2)=O)c(C)c1 C1(C(N2CC(O)CC2CO)=O)(COC)C=CCN1C(c1sccc1C#N)=O C#CCCC(=O)NC(C1CC1C(=O)NC(c1nn[nH]n1)C)C N1(C(CN(S(C)(=O)=O)C)=O)CCCC(NC(C23CC(C)(C2)C3)=O)CC1 C1(NC(CCCCN(C)C)=O)CCN(C(=O)Cn2cnnc2O)CC1CO C(=O)(C(O)CC1CCOCC1)NCCCN(C(=O)C(O)Cc1cn(C)cn1)CC c1(C(N2C(CCOC)CN(C(=O)C=C(C)Cl)CC2)=O)cnn2cc(C)cnc12 O=C(N=c1ncnc2[nH][nH]cc1-2)C1CC12CCN(Cc1cccc(F)c1O)C2 C1(NC(c2c(OC)ncc(Cl)c2)=O)CN(C(=O)CSC(C)C)C2(CCC2)C1 c1(C(=O)NC2(c3cn(CCN(C)C)nn3)CC2)cccc(C2CCOC2)c1 C(CC(O)C(=O)NCC(CC(C)C)NC(C1(C(=O)OC(C)(C)C)CCCC1)=O)SC c1(-c2c(C(=O)NCc3c(C)ccc(F)c3)nccc2)ccc2ncccc2c1 N1(C(c2ccc(N)c(F)c2)=O)CCN(C(=O)Cc2ccccn2)C(CO)C1.OC(F)F N1(C(c2occc2CO)=O)CC2CCC2(CC(N2CCC3(CC2)CC3)=O)C1 N#Cc1cc2ccccc2n1CC(=O)NCC1C=CCN1C(C1COC1)=O CC1CN(C(=O)C(C2CC2)N(C(=O)Cc2ccccn2)C)CCS1=O C1(CN(C(=O)CNC(=O)CC(F)(F)F)C)CCCCN1C(C1(C)CC=CC1)=O c1(N2CCC(NC(C3CN(C)C3)=O)C(F)C2)nc2ccc(O)cc2s1 Cc1cc(C(N2C3CCC2(CNC(c2nc(Cl)sc2C)=O)CC3)=O)cc(N)c1 N1(C(c2nc(C(C)C)oc2)=O)CC2CC1C2NC(=O)COc1ccsc1Cl c1(C(C(N2C(CNC(C(C)(C)OC)=O)C=CC2)=O)C)ccc(C(F)(F)F)cc1 C12(NC(C=CC=CCC)=O)CCC(CC1)N(C(c1cccc(C)c1Br)=O)C2 c1(C(=O)NCCC2(NC(C3C(C(C)(F)F)C3)=O)CCC2)ccc2nccnc2c1 C(c1ccncn1)=CC(=O)Nc1csc(C(N)=O)n1.C1C(C)(O)CNC(=O)CN1C C1(CC(=O)NC2C3CC2N(C(=O)COCC2CC2)C3)CCS(=O)(=O)C1 C1(OC(C)C)CN(C(=NCCOCS(C)(=O)=O)NC2CC2C)C1 c1(OC)cc(O)ncc1C(=O)NC(C)(C)CCNC(c1cc2n(c1)CCC2)=O C12(NC(CCC(CC)OC)=O)CCCCCC1N(C(=O)C(O)C(C)C)CC2 c1(CC)ccc(C(=O)NCC2CC(F)(CNC(C3CC3(F)Cl)=O)C2)c(N)c1 Cc1nnc(CCCC(=O)NCC2CC(C)N(C(C3(C(N)=O)CCC3)=O)C2)n1C c1(C(N2CC(CC(C)NC(C3C4CN(C)CC34)=O)C2)=O)cnc(S)n1C C1(C(N(C2(CC(=O)NCCCCC#C)CC2)C)=O)CCCCC1O C(CC(=O)N1CCC(C(C)(C)O)CC1)(C(C)CC)NC(CCCCC#C)=O c1(SC)cccc(C(N2CCCC(NC(c3cn(CC)cn3)=O)C2)=O)c1O N1(C(C(CCN(C)C)NC(=O)C#CC(C)(C)C)=O)Cc2cccc(O)c2C1 CCCC(CC(C)C)C(=O)N1CCC(C(=O)N(C2CCCC2)C)C(C)C1 C1(NC(c2sc(C)cc2OC)=O)CCN(C(C2CCC(C(=O)OC)O2)=O)C1(C)C c1(C(=O)Nc2cccc(SCCO)c2)[nH]c2ccc(Br)cc2c1Cl c1(C(=O)NCCCNC(c2ccc(O)nc2)=O)cc(F)c(Cl)c(Cl)c1 N1(C(C=CC(C)C)=O)CC(NC(c2ccc3nn(C)cc3c2)=O)CC12CCCC2 c1(C(=O)N(CCNC(=O)CC2(O)CCOCC2)C2CC2)ncnc2c1CCCC2 C1(CC)CCc2[nH]nc(C(=O)NCC3CN(C(=O)C(F)C4CCC4)CCN3C)c2C1 CN1C(=O)CCC1C(N1CCCC1C1(O)CN(C(c2cc(CO)nn2C)=O)C1)=O c1(NCC(=O)NCC2(F)CCC(CNC(C(CCC)O)=O)C2)c(C)cccc1Cl C1(C(N(CC(CC)C)C)=O)CCN(C(C2CCCOCC2)=O)CC1 c1(C(=O)NC(CNC(Cc2c(C)non2)=O)C2CC2)ccnc(C2CC2)c1 C1(OC)CN(C(c2sccc2F)=O)C(C)(CNC(c2ncsc2C(C)C)=O)C1 C1(CNC(CCSCC)=O)CCC(NC(C2CC2C(F)(F)F)=O)CC1 O=C(C1=CCCOCC1)NC12CCCC1N(C(c1cnns1)=O)CC2 O=C1CCN(CC2CC3(CCC3)C2)C(=O)N1Cc1cc(Br)ccc1F C1(OC)CC(C2C(=O)N2)C1.C1(SC)CN(C(C)=O)C1.C12CCN1C2=O c1(C(N2CC(CNC(=O)CC3COC(=O)C3)C2)=O)cc([N+](=O)[O-])ccc1O N1(C(c2ccc(C(C)C)o2)=O)CCCC(O)(CNC(c2nnn3c2CCC3)=O)C1 C1(CC)CN(C(C2CCCOC2)=O)CCN1C(c1cc(OC)ns1)=O C(=O)(C1=NOC2COCC12)N1CCN(C(CCCC#N)C(F)(F)F)CC1 C(=O)(C#CC1CCOC1)N1CCC(C(N(c2cccc(F)c2)C)=O)OCC1 C1(C(=O)N(C)CCC2CCCO2)(OC)CCN(C(c2oc(C)nc2C)=O)C1 CC(CC(=O)NCC12CCC(CC1)O2)C(C)(C)NC(=O)C1=NOCC1 CC1CCC=C1C(=O)NC(c1ccccc1)c1ccccc1.C12CSCN1C2=O c1(C(=O)NC2CC(C)(CNC(C3(NC(C)C)CC3)=O)C2)c[nH]c2c(Cl)cccc12 CCC(CCC(=O)NCCOc1ccncc1)NC(=O)C(C)CC(F)F C1(CC)CNC(=O)CN1C(=O)C(CC(C)C)NC(=O)CC(O)C1CCCC1 CC1=C(C)CN(C(=O)C(CNC(C2CC2(C)C(C)C)=O)N(C)C)CC1 c1(OC)ccc2c(=O)c(C(=O)Nc3ccccc3OC(F)F)c[nH]c2c1 CS(=O)(=O)c1ccc(Br)c(C(=O)NC2(C3CN(C(C4CC4F)=O)C3)CC2)c1 C1(=O)C(O)(C(F)(F)F)N1.CC(C(C)(C)NC(=O)C1CC1)OC(F)F Cc1nc(C(C)C)ncc1C(=O)NC1CCN(C(C2(C3CC3)CC2)=O)CC1O C1(CC(=O)NCCN(CCC)C(C2CCCCCC2)=O)CCC(F)(F)CC1 C(=O)(CCCCC(=O)NC1CC(CO)N(C(=O)CCNS(C)(=O)=O)C1)NC c1(CSCC(=O)NCC(C2CC2)NC(=O)C=Cc2cn[nH]c2)cccc(Cl)c1 c1(C(N2CC(C)C(NC(c3ccc4c(c3)CCN4)=O)C2)=O)c(F)ccc(C#N)c1F C1(CC)CC(O)CCN1C(=O)CC1(C)CCN1C(=O)CN1CCCC1 c1(NC(=O)NC2CN(C(COCc3c(C)noc3C)=O)C2)nn(C)cc1[N+](=O)[O-] C(=O)(C(CCF)NC(c1nc[nH]n1)=O)NC(C)CN=[N+]=[N-] N#Cc1ccc(=NCC=C2CC(C(=O)N)C2)[nH]c1C(F)(F)F.N1(CC)CCCC1 C1(C(N(CCNC(c2ccc(F)c(O)c2)=O)CCOCCO)=O)CCCC12CCC2 C1(NC(C2(C=C)CCOCC2)=O)CCN(C(=O)CC2CCCN(C)C2)CC(O)C1 CCCC(C(=O)NC(Cc1cn[nH]c1)C(=O)Nc1cccc(F)c1)C(C)C C1(C(=O)NCCCCC)CC(=O)CN1C(C1CC=CCO1)=O c12ccc(o1)CCC(C)=CCNC(=O)CCOC2=O.N(CC)(CC)CC C(=O)(CCCCCN(C(=O)CC1CNC(=O)O1)C)NC(c1ccco1)C C1(CNC(CCCOCC=C)=O)CCCN(C(=O)Cc2c(Cl)cnn2C)C1 CN1CCn2nc(C(=O)N(C3CCCC3)CCc3nn[nH]n3)cc2C1 N1(C(C2C(NC(c3cnn[nH]3)=O)C3CCC2C3)=O)CCC(C2CCC2)C1 c1(C(N2CC3CC(NC(C4(CCF)CCC4)=O)CC3C2)=O)ccn2cncc2c1 Cc1cc(NC(C2(CNC(=O)CC3CCCN3C)CC2)=O)cc(C)c1O c1(C(=O)NCC2(CNC(c3ncn(CC)c3)=O)CC2)cccc(N2CC=CC2)c1 Cc1cc(C=CC(=O)NCC(C(C)C)NC(=O)C(C)OCC(C)C)on1 N1(C(C(c2ccc(F)cc2)C)=O)CCCC(CO)(CNC(=O)C2=CSCS2)C1 C1(C)(CC)CC(NC(C2CC=CC(NC(=O)CCC3CC3(C)C)C2)=O)CCO1 C1(N(C(C(CCC)N(C)C)=O)CC)CCCN(C(c2nn(C)cc2C)=O)CC1 c1(OC)ccc(C=CC(=O)NC(C)CN(C(=O)C(F)CC2CCC2)C)c(OC)c1 c1(NCCc2c(OC)ccc(F)c2)ccc(S(=O)(=O)N2CCSCC2)cc1Cl Cn1ncc(C(N2CC(NC(=O)C(O)C(F)F)C3(CC3)C2)=O)c1S(C)(=O)=O C(=O)(C(F)(F)C(F)(F)F)NC(C(C)(C)NC(c1cc(C)[nH]c1C)=O)C CC(CO)C(=O)NC(C)(CNC(c1csc(-c2ccccc2)c1)=O)C1CC1 c1(C(C(=O)NC(C2CCCN2C(=O)Cc2cocn2)C)(C)C)ccc(Cl)cc1 N1(C(C2C(C)CC2)=O)CCC(C)(C)C(C(=O)NCC2(O)CCSC2)C1 c1(C(=O)NC2CCC(N(C(c3cc(C)no3)=O)C)C2)cnc2nccn2c1 Cc1ncc2c(n1)CCC(C(=O)NC1CCC1NC(=O)CCC(=O)N(C)C)C2 C(=O)(CC1=CCCC1)NCC1C(C)CCN1C(=O)CCOC1CC1 c1(C(N2CC(N(C(c3c(C)scn3)=O)C)C2)=O)ccc2c(Cl)ccnc2c1 C1(NC(Cc2cc(C)n(C)n2)=O)CCN(C(c2nnn(C)c2C(F)F)=O)C12CC2 C1(C(=O)NCC(C(C)C)NC(c2nccc(C(F)F)c2F)=O)CC12CCSCC2 C1(C(N2CCC(C)(NC(C3(O)CCOCC3)=O)C2)=O)CC12CCOCC2 C1(NC(=O)CC2CCOC2)CCN(C(=O)CNC(C2CCC2)=O)CC1CO c1(NC(=O)NC(C2CCN(CC(CC)OC)CC2)C)cnc(C(C)(C)C)nc1C N1(CCC(CC)(C)C)CCC(=O)N(Cc2ccc(CC(C)C)cc2)C1=O CCCCNC(=O)CN(CC(N)=O)CC1CC1 N1(C(CC(C)(C)N(C)C(C2(C)CCCOC2)=O)=O)CCn2ccnc2C1 C#CC1CCN(C(=O)C(CC)N(C(=O)Cc2csc(C)n2)C2CC2)C1 c1(C(N2CCC(c3c(C)ccnc3)C2)C(=O)NC2(C)CC2)c(F)ccc(F)c1Cl S(=O)(=O)(CCC(=O)NCC(F)CNC(=O)C(C)OC1CCCC1)NC c1(CC(CC)NCc2ccc(C)o2)ccc(OC)c(OC)c1 C#Cc1ccc(C(=O)NCC2CC2NC(=O)Cn2cc(Br)c(C)n2)c(C)c1 CCC(C)C(=O)C(=O)NCC(C)N(C)C(C1CC2(CC(=O)C2)C1)=O N1(C(C(C)OCC#C)=O)C(C(=O)NC(C2CC3(CCC3)C2)C)CCC12CC2 C1(NC(C23CC(NC(C(CC)OC)=O)(C2)C3)=O)CCCC(C(C)(C)C)C1 N(C(=NCCCC(F)F)N1CCC(OC(C)C)C1)CC1C(=C)C1 N12CCCCC1C2=O.N1(C=O)CCC(C)(CNC(=O)C=CCN2CCCCC2)C1.CN C(=O)(CC1OCc2ccccc21)N1CCC(CCNC(CC(C)O)=O)C1 N1(CC(=O)NC(C)CCNC(=O)CCc2ccsc2)CC(=O)Nc2ccccc21 N1(C(C2C3CCCCC23)=O)CC(C2CC2)(C(N2CCOC3CC23)=O)C1 C1(C(=O)OCC)CCCCC1NCc1cc(C(F)(F)C(F)(F)F)on1 c1(C(=O)NC(CNC(C(C(C)C)NC(CNC(C)=O)=O)=O)C)c(O)nnc(C)c1C C1(c2cn(CCc3cn(C)nn3)nn2)CCC(N)CC1 CC1CCC(CO)(NC(=O)CCN(C)C(c2cccc(CC#N)c2)=O)C1 N1(C(C(CC(N)=O)O)=O)CCOC2CN(C(=O)CC3CCC(F)(F)C3)CC12 C1(C(=O)OC)Cc2c(F)cccc2CN1C(C1OCCN(C)C1=O)=O Cc1oc(C(N2CCC(CNC(C3(CC#N)COC3)=O)C2)=O)cc1Br Cc1cc(C#N)nc(NCc2ccc(-c3cnc(O)nc3O)nc2)n1 N1(c2nc(C(=O)OC)c(C)s2)CC2CC(NC(c3nc(Cl)oc3C)=O)CC2C1 c1(C(N2C(C(=O)NCCC(CC)(F)F)CC2)=O)ccc(C)c(F)c1 CC1=C(C(=O)N2CCC(CC(=O)N(C(C)C)Cc3cnccn3)C2(C)C)CCO1 N1(S(CCOC)(=O)=O)CCC2CNCC12.C1(C)C(=O)N1 c1(C(=O)NCC2(C)CC(NC(C3CC4CC4C3)=O)C2)cccc2[nH]ncc12 N1(C(C2(CC)CCCC2)=O)CC(N(C(=O)Cc2n[nH]cc2Br)C)C(O)C1 C1(CC=C)(C(=O)NCC(=O)OC)CCN(C(=O)CCCOCCC)C1 c1(CC)nn(C)c(CC)c1C(=O)NCC1(CNC(C2CCCC(O)C2)=O)CCC1 N1(CC(=O)NC(C(=O)N(CC)CC)C(C)(C)C)CCC2OCCCC2C1 N1(C(C(C)n2ccnc2)=O)CCC2(NC(=O)Cc3ccc(O)nc3)CCCC12 Cc1ccc(Cl)cc1NC(=O)C(C1CCN(C(C2C(C)(C)C2(F)F)=O)C1)F C1(NC(C(C)Cc2cnc[nH]2)=O)CCC2(CC1)CC2NC(C1CN(C(N)=O)C1)=O c1(C(=O)NCC2(Nc3nnc(C)c(C)n3)CCCCC2)cnc2ncc(Cl)cn12 N1(CCCCC(C)C)CC(=O)NC(c2cnn(-c3cc(F)ccc3F)c2)C1 c1(NC(C2N(C(c3cc(CC)c(Br)cc3)=O)CC=C2)=O)ncc2c(n1)CCNC2 c1(NC(C(CC2CCC2)NC(C=C2CCC(C)CC2)=O)=O)cnn2cccnc12 c1(C(N(CCCCNC(C(C)NC(C)=O)=O)C)=O)c(Cl)ccnc1F Cc1oc(-c2ccccc2)cc1C(=O)NCC(C(C)C)NC(=O)C=CC(F)(F)F CCS(=O)(=O)CC(=O)NC1CCCC1(C)CN(C)C(c1ncnc(C)c1C)=O C(=O)(C(C)CS(C)(=O)=O)N1CC2(N(C(COCCCCCCOC)=O)CC2)C1 C1(C(=O)NCCN(C(=O)CC2CCCC(C#N)C2)C(C)C)CC2CCC1C21CC1 Cc1cc(C2CC2)ccc1C(N1CCC(C)(CNC(c2cnc(=N)[nH]c2)=O)C1)=O N1(C(c2cscc2Cl)C(=O)NCc2ccc(C(=O)OC)o2)CCC(C#N)C1 C1(CNC(c2c(CC)occ2)=O)C2CN(C(=O)Cc3csc(C)n3)CC12 C12(C(=O)Nc3cc(SC)n[nH]3)CC1CN(C(c1ncoc1C)=O)C2 Cc1c(Cl)ccnc1C(=O)NCCN(C(c1csc(O)n1)=O)C(C)C C1(C(=O)NC(c2ncccn2)CC)CC[Si](C)(C)CC1 C(CCC(=O)NC(C)CNC(=O)C(C)(C)C1CC1)NC(=O)OC CC1CN2CCN1CC2C(=O)NC1CCCCC1CNC(C12CCCC1C2)=O C1(C(N(CCOCCNC(CCCCOCCC)=O)C)=O)CC2(C1)CC(O)C2 N1(C(C(CO)OC)=O)CCC(N=[N+]=[N-])(C(=O)NC2CC=C(C(C)C)CC2)C1 c1(C(=O)NCC2(OC)CN(C(C3CCC(F)C3)=O)C2)cnn2c1CCC2 C1(C(N2C(CCC)COCC2)=O)CC(C)(C)CCN1C(C1CC(=O)CCO1)=O c1(C(=O)NC(C)CN(C)C(C2CCCCS2)=O)ccnc(C2CCC2)c1 c1(C(N2C(C(C)(C)NC(c3cn[nH]c3)=O)CCC2)=O)cc2n(n1)CC(F)C2 N1(C(C(C2CCC2)OC)=O)CCN(C(=O)CCc2conc2C)CCC1C c1c(C)cc(C)oc1=O.C=CC(C(=O)NC1CN(C(=O)CC(C)C)C1)c1ccccc1 Cc1cccc2cc(C(=O)N(C3CCC(CN(C)C)CC3)C)nn12 Cc1cccc(N)c1C(=O)NC1CCCC(NC(=O)C=CBr)CC1 CCCCC(CCC)NC(=O)C(=O)Nc1cccc(CSCC)c1 C1(CNC(C(CSC)(C)C)=O)CN(C(=O)CC(F)(F)F)CCC1C c1(NC(C2CC3(CC3)CN2C(C2CC=CCC2)=O)=O)cc(Br)cc2[nH]ncc12 Cc1cnc(CC(=O)N(CC(C)N(C)C(c2cocc2Br)=O)C)o1 c1(OC)ccc(C=CC(N2CCC(NC(c3ccc(SC)o3)=O)C2)=O)c(C)c1 c1(CN(C)C)ccc(C(CO)NCc2cncc(C(F)(F)F)n2)cc1 C(=O)(C(C(F)(F)F)C(F)(F)F)N1C2C(CNC(C(C(C)C)O)=O)CC(CC2)C1 c1(NC(C2CCN(C(Cc3cc(C)on3)=O)C(C3CC3)C2)=O)cnc2ncnn2c1 N1(C(Cc2c(C)cccc2C)=O)CCC2CN(C(c3ccnnc3S)=O)C2C1 N1(C(C(CC=C)C)=O)CCN(C(c2cc(C)c(C)o2)=O)C(C2CC2)C1 C1(CNC(CC2(OC)CC2)=O)CCC(C)(C)CN1C(=O)CN(c1ccncc1)C c1(NCC2CCCN(C(C=CCOC)=O)CC2)ncc2c(n1)CCCCC2 C1(NC(c2c(C)cc(C)s2)=O)CCCCCN(C(=O)CC=CC(C)(C)C)C1 Cc1cc(CO)cc(N2CCCC(C(=O)NCCOC(F)F)C2)n1 C=CCC(CC)C(=O)NCCOCCCNC(=O)CC1CCC(C)(C)CC1 C12(C(N3C4CCC(NC(C5N(C)CCC5)=O)C(C4)C3)=O)CCC(C#N)(CC1)CC2 CC(C)C1C(C)CCN1.C(CCCCSC1(Oc2ccccc2)CC1)OC c1(C(=O)NC(CNC(C(C2CCC(=O)N2)C)=O)(C)C)cc(=O)n(C)o1 c12cccc(c1)C2.c1(C(N2CCC(NC(C=CC)=O)C2)=O)occ(C)c1C C(=O)(CC(O)C(C)C)NC1C2CCN(C(CCc3cc(C)[nH]n3)=O)C21 C=CC(CCC)CC(=O)NCC1=CCN(C(=O)CN2C(=O)CCCC2=O)CC1 C(=O)(C(F)(F)C1=CCOCC1)N1CCC(CC)C1CNC(=O)CCC1(C)CC1 N1(C(c2c(C)nc(C3CC3)s2)=O)CCN(C(=O)C(C)C#N)C2CS(=O)(=O)CC12 c1(CC2(C(N(C)CC3(N(C)C(c4c[nH]c(=N)s4)=O)CC3)=O)CC2)cccc(Br)c1 C12(NC(C=CCCC)=O)CC(CNC(=O)C(N3CCN(C)CC3)C)(C1)OC2(C)C c1(C(=O)NC(c2ccccc2)C(=O)NC)ccc(OC)cc1OC(C)C#N N1(C(CC=CC)=O)CC(OC)CC1(C)CNC(c1cocn1)=O C1(C(=O)NC(CN(C(c2cc(C)n(CC)n2)=O)CC)C)CCCN(C)C1 c1(C(C(=O)NC(C)CC)N(CCCOC)C)sc(C(=O)OC)cc1C Cc1cccc(OCCC(=O)N(CCNC(C2C3CNC(=O)C23)=O)C2CC2)c1C c1(SCC(=O)NCC(C2CCCC2)NC(=O)CCn2cccc2)ccncc1 C=CC(CC)CC(=O)NC1CN(C(c2cc(C(F)(F)F)cnc2N)=O)C(C)(C)C1 Cc1cc(CC(=O)NC(C)CC(C)NC(c2cnsn2)=O)ccc1CO CCCCC(CNC(c1cc(CC)c[nH]1)=O)NC(c1cc(C)nn1CC)=O N1(C(C(C)N(C)C)=O)CC(C(N)=O)(CNC(C2CC2(F)F)=O)C1 CCC(C)(C)C(C)NC(=O)C(C)(C1CC1)N(C(=O)Cn1ccnc1)C c1(C(=O)NCC2(CNC(C(CSC)O)=O)CC2(F)F)cc2c(F)ccc(F)c2[nH]1 C(=O)(CCCCNC(=O)CN1CCOCC1)N(C1CCOCC1)C C12(NC(C3C(C)OCCC3)=O)CCCN(C(c3cc4n(n3)CCC4)=O)CC1C2 N1(C(c2c(Cl)cc(C)s2)=O)CCC(C)C(NC(C2CC3CCC2CC3)=O)C1 C1(CNC(CC2(C)CCS(=O)(=O)N2)=O)CCCC2(CN(c3nccnc3F)C2)O1 S(=O)(=O)(c1ccc(NC(CC(N)=O)C2CC2)c(F)c1)NCCC1C(C)OC(C)C1 N1(C(c2ccsn2)=O)CCC2C1CCN2C(c1ccc[nH]1)=O C#CCCCCCCCNC(=O)CC(C)CNC(=O)C(C)n1cccn1 C=CC1(C(=O)NCC(CCCC)OC)CCN(C(=O)C(C)CC(=O)OCC)CC1 N1(C(c2c(OC(C)C)nccc2)=O)CC2CC(C(=O)NCCC(N)=O)C(C2)C1 C1(NC(=O)CSCc2cccs2)CC2(C1)CC(CNc1nccnc1C#N)C2 CC(C)CCCCCC(=O)N1CCC(C)C1C(N1CC(C(C)(C)C)C1)=O C1(C)(CNC(c2c(Cl)nc(OC)s2)=O)CN(C(c2cnc(C)nc2C)=O)CCO1 C1(C(N(C2CCN(C)CC2)C)=O)CCC(O)CN1C(c1nnc(S)n1C)=O C=CC(C)(C)CC(=O)NC(C)CCN(C(=O)C(F)C1CCCC1)C O=C(CC1=CCCCC1)NCC1CCCC(NC(=O)CCCn2ccnc2)C1 C1(CNC(=O)CO)CC(F)CN1C(c1cnn(-c2nccs2)c1)=O CN1CCC(C(N2CCCC(CF)C2)=O)(NC(c2sccc2CO)=O)C1 C1(C(=O)NC2CCCC2NC(=O)CSCCC(C)C)(OC)CCCC(C)(C)C1 N1(C(C(COC)N(C)C)=O)CC=CC(NC(C2(C(=O)OC)CCC2)=O)C1 N1(c2n(Cc3ccc(Cl)cc3)c(Cc3cc[nH]n3)nn2)CCOC2(CCCC2)C1 C1(CC)CCCCN1C(=O)CN(C(c1cn(C(C)C)cc1C)=O)C(C)C.C(C(F)F)S c1(C2(O)CN(C(C3CCNC(C(F)(F)F)C3)=O)C2)c[nH]c2ccccc12 Cc1cncc2nc(CNC(=O)CC3(C4(O)CNC4)CC3)cn12 CC1(C)CCC1C(=O)NCC(C1CCCC1)NC(c1cnc(C(N)=O)s1)=O CN=c1ccc(Br)c(C(=O)NC(C)CN(C(=O)CCC(C)C)C(C)C)[nH]1 c12c(cccc1NC(=O)CC(C)(O)c1ccccc1)NC1N(CCC1)C2=O.CCSCC C(=O)(CC(C(=O)N1CCC(C2CCCN2C(c2ccns2)=O)CC1)N(C)C)OC N1(C(CCNC(=O)OCC)=O)CCCC(c2cccc(OC)c2)C1 C1(C(C)(C)C)CC(CNC(=O)C(F)C(C)(C)O)CN(C(C23CC(C)(CO2)C3)=O)C1 C=CCC(CC)C(=O)N1CCN(C(=O)CN2CC(C)(OC)C2)C(C2CCC2)C1 Cc1ccc2c(C)c(C(=O)NCC34CC3CN(C(=O)CCC3CC3)C4)[nH]c2c1 c1(C(C(=O)NC2CCC2)N(C)CC2(CC)CCC2)ccc2c(c1)oc(=O)n2C C1(C(N(C(CNC(=O)Cc2ccno2)C2CC2)C)=O)CC12C(=O)Nc1ccccc12 C(=O)(C(CO)C(F)(F)F)N1CCC(C(C(=O)NCc2c(OC)c(F)ccc2)(C)C)C1 C(=O)(CC(c1cccs1)NC(c1ccc(CC)s1)=O)OCC C1(N(C2C3CCCC23)C(C=CC)=O)CCC2(CC1)CNC2 C(CC(C)(C)C(=O)N1CCCOC(CNC(C2NC(=O)OC2(C)C)=O)C1)OC C1(CNC(=O)NC(c2cnsc2)C)CCOC1c1cnn(C(C)(C)C)c1 C(C1=CCN(C(C2(C)CC2(F)F)=O)CC1)NC(C(CC)Oc1ccccc1)=O C(CCCC(=O)N1CCCC1)N(C(C(C)(C)OC(C)=O)=O)CC(C)C C1(C(N(C(C)C)CCNC(C2CCC(F)C2)=O)=O)CCn2ncnc2C1 C1(CC#C)(C(=O)NCCCCCNC(c2cnc(C(C)OC)[nH]2)=O)CC=CCC1 N1(C(c2ccc(CC#N)cc2)=O)CCC12CN(C(c1coc(Cl)n1)=O)C2 C1(NC(c2c(C)cno2)=O)CCCC(NC(c2c(Br)noc2C)=O)C1 C1(C#CC(=O)NC2COCCN(C(=O)CC(C)C3CCCO3)C2)(CC)COC1 c1(CC(C(=O)O)C(C2CCCCC2)C(=O)NC2CCOCC2)csc2ccccc12 C1(C2CCOCC2)(C(N(C)CCNC(=O)C(C)(C)C(N)=O)=O)CCOCC1 N1(C2CN(C(C3C(CCC)C3)=O)C2)CC(NC(=O)CCn2ccc(C)n2)CC1=O C1(CC)CCCN(C(=O)C(C)NC)C1C(=O)NC1CC1NC(=O)NC Cc1cccc(C(C)(C)C(=O)N2CCC(C3CC(C(F)(F)F)(CN)C3)C2)c1 C1(C(N(CC(C)(C)C#N)C)=O)CC12CCN(C(C1COC(=O)C1)=O)CC2 N1(C(=O)Oc2ccccc2)CCS(=O)(=O)N2CCOCC12 CC1(C(N2CC=CC(NC(c3ccncc3F)=O)C2)=O)CCC2(CC1)OCCO2 C12(C(=O)OC)CC(COC(c3[nH]c4ccc(C)cc4c3)=O)(C1)OC21CCC1 c1(C(=O)Nc2nc(C)c(C(N3CCCC3C(F)(F)F)=O)s2)ccc2cc[nH]c2c1 CCCCCCCCCC(O)C(=O)N1CCCN(C(=O)Cn2cnnn2)CCC1 C1(CC(=O)N(CCOCC=C)C)COCCN1C(=O)CC1(O)CCCOC1 C1(O)(CCC)CCN(C(c2c(CNC(=O)C(C)NC(C)=O)nnn2C)=O)CC1 N1(CC)N=C(C(=O)NCC(O)CCNC(=O)CC2CSCCS2)CCC1=O Cc1nc(C(=O)N(C)CCc2ccccn2)c(=O)[nH]c1C C1(OCCN(C)C)CCN(C(=NCC2CC3CCC3C2)NC2CC2)C1 c1(C(N2CCC(NC(C(C)SCCCC)=O)C2)=O)cccc(C)c1[N+](=O)[O-] N1(C(CSCCCC)=O)CC2CCC1C(CNC(=O)C(O)CC(=O)OC(C)(C)C)C2 CC1CCN(C(=O)C(=O)NC2CC(NC(=O)C(C)O)C2)CC1 c1(CC)cc(CC(=O)NC2CC(C)(NC(c3cc(CSC)on3)=O)C2)on1 N=c1nnn(CC(=O)NCC2CC2NC(c2cn(CC(F)(F)F)nn2)=O)[nH]1 CC12CN(C(c3ccc(OC(F)F)cc3F)=O)CC1CN(C(C1CNC(=O)N1)=O)C2 C1(CNC(C(C=C)O)=O)CN(C(C2C(C)C2C)=O)CCN1C c1(C(=O)NC2CC(N(C(CC(c3ccc(F)cc3)C)=O)C)C2)c[nH]ccc1=O CC(CCCc1ccccc1)C(=O)NCCNC(=O)C(F)(F)c1csc(=N)[nH]1 c1(C(=O)NCc2c(C(=O)NC3CCCC(SC)C3)con2)ccc(O)nc1C N1(C(CC23C(CN(C(C#CC(C)C)=O)C2)CC3)=O)C2CCC1CC(CO)C2 C(C1CN(C(c2cccc(C)n2)=O)CC1C(=O)N(C1CCC1(C)C)C)=CC N#Cc1cc(N2CC(CCCCNC(c3csc(Cl)c3)=O)C2)nc(C(F)(F)F)n1 Cc1ccc(C(C)C(=O)NC(C)(C)CNC(c2sccc2F)=O)s1 Nc1ccc([N+](=O)[O-])cc1C(N1CCC(NC(=O)CC2CCOC2)C1)=O C1(C(=O)NCCN(C(=O)C=C2CCCC2)CCC)CCCN(c2nccn2C)C1 CC(C)CC(CC(C)C)C(=O)N(C)CC1(NC(=O)CN2CC(C)(C)C2)CC1 Cc1ccnc(CNC(C2CC3CC3N2C(=O)CC2CCOC2)=O)n1 C1(NC(C2CC(=C)C2)=O)CCCCC12CCN(C(C1CCCN1C(C)=O)=O)CC2 c1(CCNc2nc(C)nc(N3C(C)CC4CNCC34)c2)ccc2ncccc2c1 C(CN=c1[nH]cnc2ccc([N+](=O)[O-])cc12)NC(=O)CC(c1ccon1)C1CC1 c1(C(N2CC(OC)(CNC(=O)Cc3coc(C)n3)C2)=O)cc(C)cc2c1CCC2 Cn1ncc(C(=O)NC(C)(CNC(c2ccc(C3CC3)cn2)=O)C2CC2)c1F C(=O)(CS(=O)(=O)C1CC1)N1CC(CNC(c2cc(F)cnc2O)=O)C(O)C1 c1(CNC(=O)OC(C(c2ccccc2)NC(=O)NCC)C(C)C)ccccc1F N1(C(C(C)=O)=O)CC(F)(F)CC1NC(=O)N(c1ccccc1C)Cc1ccccc1 C(=O)(C1CCCc2nncn21)NCC1C(NC(c2ccc(CC)cc2N)=O)CC1 CC(C(=O)NN1CCCCC1=O)N(C1CC1)CCc1ccc(Cl)cc1 C1CCC(O)C(=O)NCCOCC(=O)N1.c1(CSC)cnsc1 n1(CC(=O)NCC(CCNC(C(C)Cn2cccn2)=O)O)sc(=O)c2ccccc12 c1(NC(C(C)N(C(c2c[nH]ccc2=O)=O)CC)=O)ccc(N)cn1 Cc1ncc2n1CC(C(=O)NC(C)CC1(O)CCC1)CC2 N1(C(C2C(C(C)(C)C)C2)=O)CCCCC(NC(c2ccc(C3CC3)cn2)=O)C1 c1(C(N(CCN(C(c2sccc2F)=O)CC)CC)=O)ccc2c(c1N)CCCC2 N1(C(C(C)SCCCC)=O)CCN(C(=O)C#CC(C)(C)O)C(C)C1 C1(C(N(C)CC2(O)CN(C(=O)CCCn3cncn3)C2)=O)CCCCC1OC N1(C(C2CN(C(C)=O)C2)=O)CC2COCCC2(NC(=O)C(O)Cc2ccccc2)C1 c1(CC(=O)NCCCNC(=O)Cc2cn[nH]c2)c(F)cccc1F c12ccc(cc1F)CN2C(=O)OC.c1(OCC2CC2)ccccn1 c1(-n2cc(CNC(CC(C)SC)=O)nn2)cnccc1C Cc1cc(Br)c2nc(C(=O)OCc3ncc(Cl)s3)cn2c1 C(CNC(C1CC1C1CC1)=O)(CC(C)C(C)C)NC(C12CC(C(C)C)(C1)C2)=O C1(C(=O)NCC(C(C)O)(C)C)CCC(C)(C)N(C(=O)C(C(C)(C)C)N(C)C)C1 c1(OC)cc(C(=O)NCC(F)CNC(=O)C(C(C)O)N(C)C)cc(Cl)c1O N1(C(C(=Cc2ccccc2)CC)=O)CC(NC(c2cc(C)cc(C)c2)=O)CC1(C)C C1(CC)CCC(O)(C(=O)NC2(CNC(c3cnn(CC)c3Cl)=O)CCCC2)C1 N1(CC(=O)NC(C(C)C)(C)CNC(C2CC=CC2)=O)CCS(=O)(=O)CC1 C(=O)(CC(C)(O)CCC)N(C1CCN(CCCC)CC1)C1CCC1 CCC(C)CCC(O)CN1CCN(C(=O)OCC(C)(C)C)C(C)C1 C1(NC(CCC2CCC(=O)NC2)=O)CC2CN(C(c3ccc[nH]3)=O)CC12 Cc1cc(C(=O)N(C2C3CN(C(c4nocc4Br)=O)CC23)C)cn1C(C)C Cc1cc(Br)cnc1C(=O)N(C)CCN(C(=O)CC1OCCC1(C)C)C C1(CC(=O)NC2(CNC(C=C(CC)C)=O)CCC2)COC(C)(C)C1 CCCCC(C)C(=O)NC1(COC)CCN(C(=O)CC2COC(=O)C2)CC1 C=C(C)C(C)(O)C(=O)NCC1CCN1C(=O)C(C)=CC C(=O)(C1CCCc2nn[nH]c21)NCC1CC(NC(C#CC(C)(C)C)=O)C1 c1(OC)ccccc1CC(=O)NCC(C)CNC(=O)CCC1CC1(F)F c1(CC(=O)N(C2CCOC2)C)ccccc1CC(=O)O.C1CCN1 N1(C(C(CCOC)(C)C)=O)CCN(C(c2cc(C(F)F)cs2)=O)C2CCCCC12 C(=O)(CCNC(=O)C(C)N(C(=O)CCC1CCCO1)CC)OCC#C N1(C(C(c2cccc(OC)c2)OC)=O)CCOCC(NC(c2cc(C)[nH]n2)=O)C1 N1(C(C2CC(NC(c3c(C)cn(C)c3)=O)C2(C)C)=O)CCS(=O)CC1C c1(CC)ccc(NC(C2CC(C)N2C(=O)C(=O)C2CCCC2)=O)cc1OC c1(NCc2cn(C3N(C(C=CCSC)=O)CCC3)nn2)ccc2cnc(C)n2c1 C12(NC(C(C)OC3CCCC3)=O)CCCC1N(C(c1cc(C#N)on1)=O)CC2 C(=O)(C1=CNS(=O)(=O)N=C1C)N1C(C)CCC(CNC(C(CC)OCC)=O)C1 c1(C2(CN3CC(C)C(n4cc(-c5ccc(F)c(F)c5)nn4)C3)CC2)cc(N)ccc1Cl C(=O)(C(O)CC(F)(F)F)NC1CC(CNC(c2nsc3ccccc23)=O)C1 N1(C(C(C)(C)c2ccno2)=O)CCCC(CNC(c2ccccc2O)=O)C1 c1(CC)ccc(C(=O)N(CCCCCNC(=O)Cc2cnccn2)C)c(F)c1 c1(C(=O)NCC(CNC(CCC(C)OC)=O)OC)ccnc(C)c1C C1(C(N2CCC(OCCNC(C(C)(C)C(N)=O)=O)C2)=O)CCOC2(CCC2)C1 N1(C(C(C)=O)=O)CCOC2(CCCN(C(c3cc(C)n(C4CC4)c3C)=O)C2)C1 CCC(C(=O)NCC1CCCN1C(C1CCC=CO1)=O)C(C)C N1(C(C2C(C(=O)OC)CC2)=O)CCC(N(C)C(c2coc(CC(C)C)n2)=O)C1 Cc1ccc(O)c(C(=O)NCC2(F)CC(NC(C3CC(C)(C)CO3)=O)C2)c1 c1(C(N2C(CNC(COC3CCC(C)CC3)=O)CC2)=O)cc2ncn(C)c2cn1 c1(N(C(C)=O)C(C2CCCO2)=O)cnc(NC(Cc2ccccc2)CCCO)nc1C CCCC(O)CC(=O)N(C1CCCCN(C(c2ccc(O)c(CC)c2)=O)C1)C c1(CC(=O)N(C(C(=O)N(C(C(C)SC)C)C)(C)C2CC2)C)ncccc1F C=C(C)CN=C(NC(c1cc(OC)ns1)C)N1CCC(NC(C)=O)C1 c1(C(C(=O)NC2CCN(C(c3nn[nH]c3Cl)=O)CC2)(F)F)cc(Cl)ccc1F c1(C(=O)NC(CCC)C2CC2)sccc1CNC(=O)CCc1ncnn1C c1(OC)ccc(OC)c(CCC(=O)N(C2CN(C(C3(C#N)CC3)=O)C2)C)c1 CCC(C)CCC(=O)NC(C)(C(=O)NCC(C1CC1)OC)C1CCC1 c1(CC)noc(CC)c1CC(N1CCCC1CCCNC(=O)CNS(C)=O)=O C(=O)(C1CCC(C)(C)c2ccccc21)N(CCN(C(c1scc(C)c1C)=O)C)C C1(C#CC(=O)NC2CN(C(C3(C)CC(OC)CN3CC(C)(C)C)=O)C2)(CC)CC1 C1(C(C2(O)CCOCC2)C)NC(=O)N(CCc2nccs2)C1=O c1(NC(C2CCN(Cc3cc(OC)c(O)cc3)CC2O)=O)cc(C)cc(C)c1C C(=O)(C(O)CC[S+](C)C)N1CCC(N(C(=O)COCC2CCC2)C)C1 Cc1cn2c(n1)CC(C(N1CCCC(CNC(=O)CC(C)N(C)C)C1)=O)CC2 Cc1cc(N2CCC(C)(CCO)CC2)c(S(N)(=O)=O)cc1[N+](=O)[O-] c1(C(C)C(=O)NCCC2(NC(C34CC(C)C3C4)=O)CCCC2)ccccc1Cl c1(C(N(C2CN(C(=O)COCC3CC3)CC2O)C)=O)cnc2c(F)cccc2c1 C1(n2c(CC)ncc2)CCN(CCCOC2CCCC2)CC1 C1(CC(=O)NC2CN(C(c3ccc(C)o3)=O)CC2O)(C(F)(F)F)CCC(=O)NC1 N1(C(CC(=C)C)=O)CCN(C2CCN(C(=O)C(C)Sc3ccccn3)CC2)CC1 S(=O)(=O)(c1cccc(N2CCCC(CS(N)(=O)=O)C2)n1)NCCC(=O)NCCCC C1(CC(=O)Nc2n(CC)ncc2)COCCN1C(=O)C(C1(O)CCCC1)F C1(C)(CNC(c2ccc(CCC)s2)=O)CCN(C(=O)C(C)(C)N(C)C)CC1 c1(CC23N(C(=O)CCCC4CC4)CCC2CCCC3)cc2ccccc2c(O)n1 C(N=c1[nH]c(=NCCCCS(N)(=O)=O)[nH]c2c1COC2)C1CC(C(C)C)C1(C)C C(=O)(N=c1ccn(C2CC(c3ccc(C#N)cc3)C2)[nH]1)Nc1cccc(SC)c1 C1(CNC(C(c2cscn2)N(C)C)=O)CN(C(=O)CC2CCCC(C)O2)CCO1 CCCC(O)CN(C)C(C1CCC(NC(C2C(OC)C2(C)C)=O)C1)=O Cc1cc(C(N2CCC(C)(NC(=O)Cn3cc(C#N)cn3)C2)=O)ncc1Br C1(C(=O)NC(CC)CNC(c2ccnn2CC2CCC2)=O)CC2C=CC1C21CC1 C(CCCC(=O)N1CC2C(CNC(=O)Cc3ccc(F)cc3)C2C1)N(C(C)=O)C c1(NC(C)=O)cc(C(N2CCC(N(c3nnc(C)s3)C)CC2)=O)ccc1F N1(C(C(C=C)OC)=O)CC2(C1)CN(C(c1cnn(C)c1SC)=O)CCO2 c1(OC)cccc(C(=O)N(C2CCN(C(C3CCCC34CC4)=O)CC2)C)c1O C(Cc1ccccc1)(C(=O)NCCCC)OC(C1CCCNC1)=O CCCCCC(C)CC(=O)NC1CC(F)CN(C(c2cc(OC)ccc2N)=O)C1 Nc1nc2c(cc1C(=O)OCc1ccc3c(c1)CC(=O)N3)CCCC2 N1(C(CC(CC2CC2)NC(c2ncc(OC)nc2)=O)=O)CC2(CNC(=O)C2)C1 Cc1cc(C)c(C(=O)N(C2CCN(C(C3(c4nccs4)CC3)=O)C2)C)c(S)n1 c1(OC)cc(C(F)(F)C(=O)NC2CC(CNC(=O)CN(C)C(N)=O)C2)ccc1C C1(CNC(c2ccc(CC=C)s2)=O)CCCCN1C(=O)C(C)CC1CCCC1 C(C(C)(CC(C)C)NC(c1cnc2n1CCC2)=O)NC(c1c(C)sc(Cl)n1)=O Cc1c(C(=O)NC(C)(CNC(C2CC2(F)F)=O)C(C)C)nnn1C C(=O)(CCC(=O)N1CCCC(N(C(=O)CCC(F)F)Cc2ccccc2)C1)OC c1(C(=O)NCC(CO)NC(CCN(C)C(=O)OC(C)(C)C)=O)n[nH]c2c1CSCC2 C(C)(CC(=O)N1CC2(C1)CN(C(=O)C(N)=O)C2)(C(F)F)N(C)C C(N=c1[nH]c(C(=O)Nc2cncc(-c3ccoc3)c2)cs1)c1cc(C)[nH]n1 c1(C(=O)NCCC(C)NC(=O)Cc2nnc(O)s2)cc(Cl)cc(Cl)c1 C1(C(=O)OC)CCC(C(N2CCCC2CCNC(=O)C(C)SC(F)(F)F)=O)CC1 N1(C(C(C=C)(F)F)=O)CC2CCC(C(=O)NCC(CC)CC)(C2)C1 N1(C(CC2CC(C(C)(C)C)C2)=O)CC2COCC(C1)C2NC(=O)Cn1cccn1 C1(NC(CC=C)=O)CCC(C)(CNCCC(N)=O)C1.c1(=O)c(=O)[nH]1 N#CC(C(=O)N1CCCC1CNC(=O)C(c1ccccc1)O)c1ccccc1 N1(CC(CC)OC)C(=O)CN(CCCc2cccc(OC)c2)C1=O C1(c2n(C(CC)(C)C)nnn2)(NCC)CC2CCCCC12.c1nnnn1CCOC N1(S(=O)(=O)c2cc(C(F)F)on2)CCc2cc(F)ccc2C1 C(=O)(CCC(C)N(C)C)N(C(C(=O)NCc1cnn(C)c1O)C1CC1)C c1(Cc2onc(C3(SC)CCOC3)n2)[nH]nc2c1CNCC2(C)C C(c1ccccc1)=Cc1cn(CC(C)NC(C2CCN(C)C2=O)=O)nn1 C1(C(N2C(C(N3CC(F)C(F)C3)=O)C=CC2)=O)C2Sc3ccccc3C12 c1(C(N(CCNC(c2cnn(CCOC)c2)=O)CC)=O)cc(Cl)sc1Cl C(=O)(C1CC(=O)c2ccccc21)N(C(C)CNC(=O)Cn1cc(Br)cn1)C c1(CNC(C2(F)CCN(C(CC3CC(=O)NC3=O)=O)C2)=O)ccc2nc[nH]c2c1 c1(CCC(=O)NCCN(C)C(C2CC2Cl)=O)ccc2ncsc2c1 C(=O)(C1=CCCOC1)NC(C12C(CN(C(=O)NCC(c3ccccc3)C)C1)C2)C C1(NC(c2ccc(C)cc2Cl)CC(=O)OC)CN(S(=O)(=O)N2CCOCC2)C1 Cc1c(C(=O)NCCC2CCC(NC(c3ocnc3C3CC3)=O)C2)c(Cl)nn1C C(=O)(CCCC(=O)N(C)C)NCC=CCNC(CCC=CC(C)C)=O S(=O)(=O)(c1cc(Br)c(F)cc1F)NCC1N(Cc2c(OC)ccc(Cl)n2)CCC1 CC1(C)C(CNC(C2(NC(C3(C)CC4CC4C3)=O)CCSC2)=O)C1(F)F N1(C(c2cn(C)nc2)=O)C2CCC1CN(C(=O)C(c1ccc(O)cc1)C#N)C2 c1(OCC(=O)NCC(C)(C)Cn2cc(C3(C)CCCO3)nn2)ccc(F)nc1 CC(N(C)N1CCCC(C2CCOCC2)C1)c1cn(C)nn1 CC(C)CC(C(=O)NC(CC(N(C)C)NCC1CNC(=O)CO1)C(C)C)C(N)=O CC(C)(C(=O)NCC1(F)CC(NC(=O)CCc2cnc[nH]2)C1)C1CCCO1 C1(NC(CCCC)=O)CCCC(C(=O)N(C2CCCOC2)CC)C1 c1(CC(N2CC(C)N(C(=O)CCS(C)=O)CC2)=O)c[nH]c2nccc(Cl)c12 c1(NC(=O)Cc2ccccc2C(=O)Nc2ccc(O)nc2)ncnc2[nH]c(Br)nc12 CCN=c1[nH]cc(C(=O)NC2CCC(CN(C(=O)CCCC3CCC3)C)CC2)s1 c1(CC)cccc(OC)c1C(=O)NC12CC(NC(c3cc(Cl)cnn3)=O)(C1)C2 c1(CC(=O)NCC(CCC)NC(C2CC(O)C2(C)C)=O)cccc(F)c1F C(=O)(C(O)CC(N)=O)N1CC(C(=O)NC2C(OC)CCC2)C(c2cncn2C)C1 c1(C(=O)OCc2ccccc2)ccnc(OCCCS(=O)(=O)NC(C)=O)c1 c1(C(=O)NC2CC(NC(C3C4CNC(=O)C34)=O)C2)cc(Br)ccc1F C=CC1(C(=O)NC2CCC(C)(CNC(=O)CN(C)C)C2)CCOCC1 c1(CN(C(=O)C(c2ccc(F)cc2)(C)O)CC)ccc(O)c(C)n1 C(=O)(CCP(C)(C)=O)N1C(CN(C(=O)C=Cc2ncc[nH]2)CC)CCC1 c1(OC)ccc2c(c1)C(NC(=O)NC13CCCCC1OCC3)C(=O)N2C C1(CNC(C2(NC(CCCOC(C)=O)=O)CCOCC2)=O)CC1C1CCCC1 c1(C(=O)NCCOC(C)(C)CNC(C2C=CCCC2)=O)cc(Cl)cnn1 c1(CC)c[nH]nc1C(N1CC(O)(C(C)(C)CNC(=O)Cn2cncn2)C1)=O c1(C(=O)NC2CSCC2c2ccccc2)cc2n(n1)CCNC2 CC(C(=O)NCc1ccc(CNC(c2cnc(S)[nH]2)=O)c(F)c1)C(C)(C)C c1(C(N2CCC(C(C)(C)C)C2)C(=O)NC(CC)(C)C)nn(C)c2ccccc12 Cc1cn2cc(C(N3CCCC(CO)(NC(C4CC(F)C4)=O)C3)=O)cc(C)c2n1 c1(C(N2CCC(NC(CCC=C)=O)CC2C2CC2)=O)ccnc2c1ncn2C Cc1cc(C(N2CCC(O)(CCNC(c3ccco3)=O)CC2)=O)c(Cl)cc1F C(N=c1cc[nH]cc1S(=O)(=O)NC1CCN(CC(F)F)C1)c1cc(OC)c(F)cc1 c1(NC(C2C=CCN2C(=O)Cc2cccs2)=O)ccc(O)c(=O)cc1 Cc1cc(NC(=O)CCC2CCCN2C(=O)Cc2ccccn2)cc(C)c1 N1(CC(=O)Nc2nc(C(N3CCC3C(C)C(=O)N(C)C)=O)oc2)CCN(C)CC1 N1(C(C2CCC(C)N2C)=O)CCC(F)(F)C(CNC(=O)COCCN(C)C)C1 c1(OC)nc(C(N2CCC(NC(=O)CCc3cn[nH]c3)CC2C)=O)cc(O)n1 CC1Cc2cccc(C(=O)NC3(CNC(=O)C4=C(Cl)CCOC4)CC3)c2O1 C(=O)(C(C)CC(C)C)N(CCCNC(C(=Cc1cnc[nH]1)C)=O)C1CC1 CCCCC(C)(F)C(=O)NCC1CCCCN(C(c2cn(C)nc2C)=O)C1 N1(C(c2ccc(C)cn2)=O)CCCCC(NC(C2CCN(CC(F)(F)F)C2)=O)C1 N1(C(C(COCC)C)=O)CC(C)(C)CCC1CNC(c1csc(C(F)(F)F)c1)=O C(CS(=O)(=O)CC(C)C)N(C(=O)NC1CC(OCC)C1(C)C)C N1(C(C(C)C2(O)CCC2)=O)CC2(CCN(C(=O)Cc3ccccc3CO)CC2)C1 C=C1CCC(C(=O)NC2CC3(C2)CC3NC(=O)CNC(=O)OC)CC1 CC1CC(C(=O)NCCN(C(=O)CCN2CCC(O)CC2)CC2CC2)CC(C)C1 c1(CC(=O)NCCCCCCNC(C2N(C)CCC2)=O)ccc2cccnc2c1 c1(CNC(N2C3CN(C(c4n(C)ccc4C#N)=O)CC32)=O)cc2ncccc2[nH]1 CC1=C(F)CN(C(C2C=CCN2C(c2cc(C)nc(C)n2)=O)=O)CC1 c1(C(N(CCC)CCNC(=O)C(CC)NC(N)=O)=O)cn(C)c(=O)cc1OC CCCCC(O)C(C)C(=O)NCC(C)CN(C)C(c1cnc2cc[nH]c2c1)=O N1(C(=O)C=CC2CCCC2)CCOC(C)(C2CC2)C1.CC1(C)C2C1C(=O)N2 c1(CNC(C2CC(F)CN2C(C2CCCS2)=O)=O)c[nH]c2ccc(Br)cc12 N1(C(c2c(CC)n[nH]c2)=O)CC(O)CCC1C(N1CCC(n2cncn2)C1)=O N1(C(C2CCC(CC)O2)=O)CC(CNC(c2cc(C3CC3)on2)=O)CC1(C)C N1(C(c2ccc(C)c(C)n2)=O)CC(NC(C2COC(=O)N2C)=O)CC(C)(C)C1 c1(C(=O)NC2CC(CNC(C3(C)CCCCO3)=O)C2)cc(N)ccc1F c1(CC2ON=C(CC)C2)cccc(F)c1OS(=O)(=O)CCCc1cccs1 C1(NC(C2(C)CCCS2)=O)CC(NC(=O)CN2CCCCC2=O)CC1O N1(C(c2cnc(C)[nH]2)=O)CC(CNC(c2n[nH]c(C)c2Br)=O)C2(CCC2)C1 C1(NC(c2ccsc2C(F)F)=O)CC2CN(C(=O)C=Cc3ccc(Cl)cc3)CC12 N1(C(C2CCC(OC)C2)=O)CCC2(CC1)CC2NC(c1cnc(N(C)C)s1)=O CCC(CN(C)C)C(=O)NC(C)CCN(C)C(c1ccc(CNC(C)=O)cc1)=O c1(CNC(C(c2ccsc2Br)N(C2CCC2)C)=O)cccc(Br)c1 c1(SC)nc(N2CCOC(C(C)NC(C3(C4CCC4)CC3)=O)C2)cc(C(F)F)n1 N1(C(CCCCCNC(N)=O)=O)CC2CC(NC(=O)CC3=CCCCC3)CC2C1 CCCCC(O)C(=O)N1CCCC1C1(O)CN(c2c(CC)ncnc2CC)C1 N1(C(CC(C(=O)OCC)(C)C)=O)C2CCCC1CC(NC(=O)Cc1cn[nH]c1)C2 c1(C(=O)NCCC(=O)NC2CC2(F)CO)c(F)cccc1F C1(NC(CCOCCN(C)C)=O)CCC12CN(C(=O)CCn1ccc(O)nc1=O)C2 C1(C)(C(C)(C)C)CC(C(=O)NC2CC2NC(C2CC3CC3C2)=O)C1 N1(C(C(CCOCC)NC(=O)C=CC(F)(F)F)=O)CCCCC(C)(F)C1 C1(N(C(CCNC2C(CC)C2)=O)C)CCN(C(C2CN(C(C)=O)C2)=O)CC1 C1(NC(CC=CC)=O)CC(CNC(c2c[nH]nc2OCC(F)(F)F)=O)C12CCC2 c1(C(N(C2CCOC2)C)=O)cc(NCc2cccs2)cc([N+](=O)[O-])c1 c1(C(N(C2CCN(C(C(COC)C)=O)C2)C)=O)cncc2[nH]ccc12 CC(C)(CC(F)(F)F)C(=O)NC1CCC1NC(=O)CCc1cccnc1Cl C(=O)(CC(C)C(C)(C)C)N1CCC(O)(CNC(c2c(CC)ccs2)=O)C1 C1(C(=O)NC(c2nc(=O)o[nH]2)C)(N(C(=O)CC#N)C2CC2)CC1(C)C C(=O)(C1=NOC2COCC12)N(C1CN(C(=O)CCn2cccn2)CC1(C)C)C C1(NC(CCNC(CC(C)C)=O)=O)CC(CNC(=O)CC=C(Cl)Cl)C12CCC2 c1(C(N2C(CNC(c3cnn4cc[nH]c34)=O)CCC2)=O)cccn(O)c1=O c1(OC)ccc2c(c1)N(C(=O)NCCN1CCCOC(C)C1)CCCC2 N1(CCCC=C)CC2CCC1C1CN(C(c3cc(C)ccc3[N+](=O)[O-])=O)CC21 c1(-c2cnc(CNC(c3ncc(C#C)nc3)=O)nc2)ccc2c[nH]nc2c1 C1(O)(CCNC(=O)Cc2cc[nH]c2)CCCN(C(=O)Cc2ncc(Cl)s2)C1 CCC(CC(C)C)C(=O)NCCN(C(C1C(F)(F)C12CC2)=O)Cc1ccccc1 N1(C(C2(C(CC)=O)CC2)=O)CCCC(CN(C)C(C2CCC(C)(C)C2)=O)C1 C1(C(=O)NCC2CCN(C(C34CCC(F)(CC3)C4)=O)CC2)CCCCC(F)(F)C1 c1(COC)ccc(C(c2nnnn2CCCC2CC2)NCCc2c[nH]nc2C)o1 C(=O)(CC1COc2ccccc21)NC(CNC(C(C(=O)OCC)(C)C)=O)C c1(N2CC3C(C(F)(F)F)(C3)C2)nccc(-c2ccncc2)n1 c1(C(=O)NC(C(C2CC2)OC)C)cc(CCNC(C2CC2(F)Cl)=O)on1 c1(CCC(=O)NCC(CC)NC(=O)C(CC)NC(N)=O)c(C)noc1C CC1=C(C(=O)N2CC(NC(=O)CCc3ccc(O)nn3)CC2(C)CO)SCCO1 C1(CC(=O)NCC(CNC(Cc2n[nH]c(=NC)s2)=O)(C)O)CCCC12CC2 c1(CC)nc(C(=O)NCCCC(=O)NCc2nnc(O)o2)co1 c1(NC(CCc2cc(C(=O)OCC)ncc2)=O)sc2ccccc2c1C#N CCCCC(CNC(=O)C(c1ccc(Cl)cc1)=O)NC(c1cnn(C)c1)=O CC(C)C(C(=O)NC1CC(NC(=O)COc2cnccc2Cl)C1)c1ccccc1 CCCC(CC)CC(=O)NCC(CNC(c1ccc(CO)c(Cl)c1)=O)CO c1(C(N2C(CNC(C(C(C)OC)N(C)C)=O)COCC2)=O)cnc(CO)nc1C N1(Cc2nc(C)on2)CCN(C(c2ccc(SC(F)(F)F)o2)C)CC1C C1(C(CNC(C(C)SC)=O)F)CC2CCC(C1)N2C(C)C C1(OC)CC2N(C1)C2=O.C1(CNC(=O)C(C2CC2)N(C)C)CC2(CC2)CO1 CN(C)S(=O)(=O)NCC(=O)NCC1C2CN(c3nc(C(C)(C)C)ns3)CC12 N1(C(C(C)OC)=O)CCCC(C2CC2NC(c2cccc(C)c2F)=O)C1 C1(NC(C=CCNC(Cc2ccn(C)c2)=O)=O)CCCC(C)(C)C1 C1(C(NOCC=C)=O)C(NC(c2occc2C(C)C)=O)CC1O Cc1sc(S(N)(=O)=O)cc1C(N1CC2CCN(C(C3CS(=O)(=O)C3)=O)C2C1)=O c1(CCC(=O)NCC(CC)(C)NC(C2(CF)CCC2)=O)ccc(OC)c(O)c1 C1(NC(c2cc(COC)c(F)cc2)=O)CCCCN(C(c2cc(CF)on2)=O)C1 C(=O)(C1CCc2nccn21)N1C(C(N2C(CCN(C)C)CCC2)=O)CNC(=O)C1 NS(=O)(=O)c1cccc(-c2ccc(=NCC3CC=CCC3)[nH]c2)c1 Cc1ccc(C(=O)NCCOCNC(C2CC2(C)C(F)F)=O)c(Cl)n1.C1CCO1 C1(C(=O)NC(C2CN(C(c3n[nH]c4c3CCC4)=O)C2)C)CCCCS1(=O)=O C12(NC3(CNC(=O)NCCC(C=C)(C)C)CC(N)C3)CC3CC(CC(C3)C1)C2 C1(CNC(C2N(C(C)C)CCC2)=O)CCCCN(C(=O)C(C)c2cccs2)C1 C1(C(=O)NCCC(C)(C)NC(c2ccnn2C2CCCCC2)=O)CCC12CCC2 N1(C(COc2ccc(OC)cc2)=O)CC2CC1CC2NC(=O)CC(C)F C(=O)(CCCCC(c1nnnn1C1CC1)(C1CC1)NCC)C1C(=C)COC1 c1(C(N2CC(NC(c3ccc(OC)c(O)c3)=O)C(F)C2)=O)cc2ccccc2o1 Cc1ccc(C(N2CCCCCC2C(N2CCN(C)C(C3CC3)C2)=O)=O)c(C)n1 N1(C(c2ccc[n+]([O-])c2)=O)CC2(CCCN(C(c3ncncc3Br)=O)C2)C1 N1(C(C(CC=C)OC)=O)CC=C(CC(=O)NCC2(O)CC3C=CC2C3)CC1 c1(C(=O)Nc2nnc(CC3CCNCC3)s2)ccn2c1CCC2 N1(C(c2c(C)[nH]c(C#N)c2)=O)CCC2(CC1)CC2C(=O)NC1CCCC(O)C1 c1(OC)ccc(CC(N2CCCC2C2CCN(C(=O)CC(C)(C)C)CC2)=O)cc1 c1(CN2CC(CC(=O)Nc3nc(Cl)c(Cl)nc3CO)C2)c[nH]c2ncc(Br)nc12 C1(N(C2CCN(CC)CC2)C(=O)CC2CCN(C)C2=O)Cc2nnc(C)n2C1 CC(C)(C)C(=O)C(=O)NC1CCN(C(c2occc2Cl)=O)CC1C(N)=O S(=O)(=O)(CC(=O)NC1(CNC(C2CC3CCCC23)=O)CCC1)N(C)C C1(C(=O)OCc2ccc(N3CCOCC3)nn2)C2Cc3ccc(Br)cc3C12 Cn1nc(-c2cccnc2)cc1C(=O)NC1CC1NC(=O)Cc1ccon1 CC#CCC(CO)NC(=O)CC(C)CNC(c1ocnc1CCC)=O C1(C(=O)NC)CCCCN1C(c1c(C2CC2)noc1C)C(=O)NC1CC1 c1(C(N2CC(NC(CN(C)CC)=O)C(CO)C2)=O)ccc(C)cc1O C(=O)(N=c1ccn(CC(=O)OC)[nH]1)C1C(C=CC=CC)CN(C(=O)CCCOC)C1 C1(C)(CNC(CN(C(C)C)C)=O)CN(C(=O)CCN2CCNC(=O)C2)C(C)(C)C1 Cc1ccc2c(c1)CN(C1CCN(C(=O)OC(C)(C)C)C(C)C1)CCO2 N=c1ccc(C=CC(=O)NCC(O)CNC(=O)COC2CCOC2)c[nH]1 c1(NC(C(N2C(CC)C(O)CC2)=O)=O)cc2[nH]cnc2cc1NC(C)=O c1(C(=O)NC(C2(O)CN(C(CC(C(=O)OC)C)=O)C2)C)cc2c(Cl)cccn2n1 C(c1c(Cl)cccc1Cl)=CC(=O)NCC(CNC(C(C)(Cl)Cl)=O)O C12(C(=O)NC(CNC(C3CCN(CC(C)C)CC3)=O)CO)CCCCN1CCC2 c1(CN=C(NCCP(OC(C)C)(C)=O)NC2CCCCC2C)c(F)ccc(Cl)c1F CC(C)(C(=O)NCc1cc(C(=O)NC2CCN(C(C)(C)C)C2)n[nH]1)C(F)F Cc1nc(NCc2nc(-c3ccncc3)cs2)cc(=NCC2(C)C=CCCC2)[nH]1 N1(C(C23N(C(C(OC)OC)=O)CCC2C3)=O)CC(=O)OCC1c1ccccc1 c1(OC)ccc(CNC(=O)C(C2CC=CCC2)NC(=O)C(=O)NC(C)C)nc1 C1(NC(=O)C(c2ccccc2)O)CC2CC(C1)CN(Cc1ccc(F)cc1Br)C2 C1(NC(=O)CC23CC(C2)C3)CCN(C(c2ccc(O)nn2)=O)CC1O CC1=C(C(=O)N2CCC2C(=O)Nc2cc(C(C)(C)O)ccn2)CCO1 c1(-c2scc(NC(c3cc(OC(C)=O)ncc3)=O)n2)cccc([N+](=O)[O-])c1 C1(NC(COC2C(C)CCCC2)=O)CCSC12CN(C(=O)C(C)(C)C1CCC1)C2 c1(OC)c(C)ccc(C(=O)N(C2CCCC2)CCNC(c2csc(O)n2)=O)c1F C1(CNC(C2CC(SC)C2)=O)CN(C(c2c[nH]nc2C(F)F)=O)CC1(C)C C1(c2n(CC(=C)C)nnn2)(N(C2CCC(C(=O)NC)CC2)C)CCN(CC)CC1 c1(CC(=O)NC2C(NC(c3c(CCC)nns3)=O)CC2)ccc(F)cc1F C#CC1(CC(=O)NCC2(O)CC(NC(=O)Cc3nnc(C)o3)C2)CCC1 C1(NC(c2snc(Cl)c2Cl)=O)CC12CCN(C(=O)COCc1ccccc1)CC2 c1(C(=O)NCC2(F)CCN(C(=O)C3=COCCC3)CC2)cc2n(n1)CC1(CC1)C2 C(CC(=O)NOCCC(F)(F)F)(C(C)(C)C)NC(c1c(CC)nn[nH]1)=O C1(N(C(c2cccn2C)=O)Cc2cccc(OC)c2)CC(C)(C)OC1=O C1(CNC(C2OCCN(C)C2)=O)CC12CCN(C(C1CC3(CCO1)CC3)=O)CC2 C1(C(=O)NC2C(NC(CC(C)CF)=O)COC2)CC2CC(C1)CC(F)(F)C2 Cc1n[nH]cc1CC(=O)NC(C)(C)CN(C(=O)CCOCC1CCC1)C C(=O)(C1=CCCC1)N1CCC(SCC(=O)N(CC(=O)N(C)CC)C2CC2)C1 CC(c1ccccc1)=CC(=O)NCC(c1cccc(C)n1)O CCC(C)(CCNC(=O)C(C)OC)NC(=O)C=Cc1ccnn1C C(CC(C(=O)N=c1ccn(CCOC)[nH]1)NC(=O)C(C1CCOCC1)O)=CC N1(CC(=O)NC2CCC(NC(C(C3CC3)OC)=O)C2)C(C)=CC(C)=NS1(=O)=O C1(NC(C(CC)C(C)C)=O)CC2(CCCN(C(=O)C#CC3(CC)COC3)C2)C1 C1(N(C)C)(CNC(C2C=CCN2C(c2ccnnc2O)=O)=O)CCCCC1 c1(C(=O)NCC2N(C(c3cncc(C(C)(C)C)c3)=O)CC2)c(O)cccc1O N1(C(C(CC#C)O)=O)CCCC(NC(c2ccc(CCO)cc2)=O)C1C C1(CNC(C2CCS(=O)(=O)C2)=O)CC2(C1)CN(C(=O)C(c1ccc(F)cc1)F)C2 C1(C(N2CCC(CCC(=O)NCC3COC(=O)N3)C2)=O)(OCC)CCOCC1 O=C(C#Cc1ccc(Cl)cc1)N(C1CC2CNC1C2)CCc1ccc(Br)s1 CCCC(C)(O)C(=O)N(C1CC(NC(=O)CCCc2ccc(C)cc2)C1)C Cc1ccc(C(=O)NCC2CCCCN2C(c2c(F)ccnc2Cl)=O)c(Cl)c1 c1(NCc2c(C)cnc(N)c2Br)c[nH]c2c(F)cccc12 Cc1ncnc(C(N2CCC(C(C)(C)NC(c3c[nH]cc(F)c3=O)=O)C2)=O)c1C c1(N2CC(C(C)NC(=O)CCC[N+](=O)[O-])OCC2)ncc([N+](=O)[O-])cc1C#N c1(C(=O)NC2(CNC(=O)CC3(O)CCOC3)CCC2)sc(Cl)cc1Cl CCC(CC)CCC(=O)NCCOC1CCN(C(=O)C(COC)OC)CC1 c1(C(C)C)ccc(C(N2CCCC2COC(C)(C)C)=O)nc1Cl C(c1ncco1)=CC(N1CCC1CNC(=O)C(c1ccccn1)O)=O Cc1c(N)ccc(C(=O)NC2CS(=O)(=O)CC2NC(c2coc(O)n2)=O)c1F C=CCC(C(=O)OC)NC(C1C2CN(C(=O)CCCCNC(C)=O)CC12)=O C1(C(N2CC(F)CC2C(N)=O)=O)CCCN(C(c2c(Cl)cncc2Cl)=O)CC1 CCCCCCCCC(=O)N1CC2(C1)CN(C(C1CC(OC)C1)=O)C2 CC1CCC(NC(c2ccc[nH]2)=O)CN1C(c1cc(Cl)ncc1O)=O Cn1nc(Br)c2ncnc(NCC3CC(CNC(=O)CCn4cnnn4)CO3)c12 N1(C(C=C(C)C(C)C)=O)CC(N(C)C(c2[nH]c(C(F)(F)F)nc2C)=O)C2(CC2)C1 c1(OC)cccc2cc(C(=O)NC(C)CC(C)NC(=O)C(O)CN3CCCC3)[nH]c12 C1(CCC)CCC(C(=O)N(C2CN(C(=O)CC3CCOCC3)CC2F)C)CC1 C(=O)(CC(C(=O)Nc1ccc(F)nc1)N1CCCCC1)OC C1(NC(CCN(C)CC)=O)C(CNC(=O)Cc2ccccc2Cl)CCC12CCC2 c1(CC)cc(C(=O)Nc2cccc(NC(=O)CN3CCCCC3C)c2)oc1CC N1(C(C2(C)N(C(c3c(CC)nn[nH]3)=O)CCC2)=O)CCC2(CCOCC2)C1 N1(C(C2N(C(C(C)C)=O)CCCC2)=O)CCN(C(=O)C#CC2CC2)CC(C)(F)C1 c1(C(=O)NCC2CC(O)CN2C(=O)CC2(n3cccn3)CC2)nc(Cl)ccc1Cl S(=O)(=O)(C1CN(CC(F)F)C1)NC1CC1.CC1CCCN(C(=O)C(=O)N2C(C)C2)C1 c1(SC)ccc(C=CC(=O)NCCC2(O)CN(C(=O)CC(=O)N(C)C)C2)s1 C1(C(=O)NC2(CNC(c3c(C)n[nH]c3)=O)CC2)CC2CCCC12 C12(C(CN(C)CC3(OC)CC(C)C3)=O)CC3CC(CC(C3)C1)C2 Cc1cc(C)c(C(=O)NCCC2CCN(C(=O)CC(C)n3cccn3)C2)s1 C=CC(F)(F)C(=O)NCC(CNC(=O)CC1(OC(C)C)CC1)OC1CCCC1 C1(F)(CNC(C2(Cl)C(C)(C)C2)=O)CCN(C(c2cnccn2)=O)C1 C1(O)(CNC(c2cn(C3COCC3F)nn2)=O)CCN(C(=O)Cc2cnsc2)C1 c1(-c2cc(Nc3nc(C#N)c(F)cc3)sc2)ccc2[nH]nc(Br)c2c1 c1(N(C(C(C(C)C)n2cncn2)=O)CC(C)C)ccc(Cl)c(Cl)c1 C1(CC)(NC(=O)C(C)Nc2ccccc2)CCCN(C(=O)Cc2ccc(C)o2)C1 CON=C(C(=O)N1CCCC(N(C(=O)CSC(F)(F)F)C)C1)c1ccco1 CCC(C)(O)C(=O)N1CCC1CNC(=O)Cn1nccc1C N1(C(C(CCC)C)=O)CC(C(N2CCC(C)(N3CCC3)CC2)=O)CC1(C)C c1(CC(=O)NC23CC2CN(C(C2(C(F)F)CC2)=O)C3)nsc2ccccc12 C(=O)(C#CC1CCOC1)N1CC(C(=O)Nc2cc(C)cnc2O)(COC)C1 CCC(C)C1C(=O)N1.C(=O)(C1=CCCCC1)C(C=C(C#N)N)=O.C1(NC)CCC(O)CC1 c1(N(N2CCC3CC23C(N2CCCC2CC(N)=O)=O)C)cccnc1O.C N1(C(C(CC)(C)C)=O)CCC2(NC(=O)Cc3cncnc3)CCCC12 C1(C(N(CC(CC)(C)OC)C)=O)(CF)CCN(C(c2ccsn2)=O)C1 N1(C(CCCCCOC)=O)CCC2(CC1)OCCC2NC(c1nocc1C)=O C(=O)(CCC(C)(C)F)N(C1CCCC(N(C(Cc2scc(C)n2)=O)C)C1)C c1(C(N2CCN(C(c3ccc[nH]3)=O)CC2c2cn[nH]c2)=O)cc2c(s1)CCOC2 C1(c2cn(CC3N(Cc4n(C5(C)CC5)ncc4)CCC3)nn2)C2CCCOC12 N1(C(c2cc(CC)[nH]n2)=O)CCC(NC(=O)C(C)CCC(C)(C)C)C2(CCC2)C1 C1(CNC(c2n(CC)cc(Cl)c2)=O)N(C(=O)C(C)=C2CCCC2)CCCC1(C)C N1(C(CC=CC)=O)CC2(CC2)CC1CNC(=O)CCc1ccc(F)nc1 C1(NC(C(C)SC)=O)COC2(CNC(=O)C(c3ccc(C)cc3)(F)F)CC1C2 c1(C(=O)NCC=CCNC(C(C)n2ccnn2)=O)cn(-c2ncccn2)cn1 c1(C(N2C3C(C(=O)NCCC4C(C)CCCC4)C(C3)C2)=O)cc(F)c(F)cc1Cl N1(C(C(CCC)C#N)=O)CC2CCC(NC(=O)C(C)(C)OC(C)C)C2C1 c1(CC)cccc(C(=O)NC(C2CCN(C(c3cccnc3)=O)CC2)C)c1C N1(C(Cc2nc(C(C)C)sc2)=O)CCC(C)C1CNC(=O)CC1CCC(C)CO1 C1(NC(=O)Cc2cc(C3CC3)on2)CN(C(=O)C2=C(Cl)CCC2)CCC1O C1(C(N2CCC(C(O)CNC(=O)C(C)CC#N)CC2)=O)(COC)CCOCC1 S(=O)(=O)(c1ccc(C(=O)O)cc1)N(c1nccn1Cc1ccccc1)C C=CCCC(O)CN(C)C(C1(C)C=CCN1C(=O)Cc1c(C)noc1C)=O CCN=C(NC(CCONS(=O)(=O)CCOC)C1CC1)Nc1c(C)ccnc1C Cc1cccc(OC(C)C(N2CC3CC3(NC(=O)Cc3cc[nH]c(=N)c3)C2)=O)c1 c1(C(=O)NC2CCN(Cc3cc(F)cc(Br)c3Cl)C2)noc2c1COCC2 O=C1CCC2C(C(N3CC4CC4C3C(=O)NCc3ccc(C(N)=O)o3)=O)C12 c1(C(C(=O)N(C(C)C)CCNC(=O)CC2CCC2)(F)F)ccc(C(F)(F)F)cc1 C(=O)(C1CCCc2n[nH]cc21)NCCC(C)N(C(c1sc(CC)c(C)c1)=O)C CC(CC(C)(C)C)C(=O)NC1CCC1CC(N1CCC(O)(CO)CC1)=O C(=O)(C1=C(C)OCCS1)N(CCC(=O)NC(CC)CC)CCO N1(C(Cc2c(C)noc2Cl)=O)CCC(NC(=O)CC2(C)OCCO2)C(CO)C1 CC1CCC(NC(c2cn3c(n2)SCC3)=O)CN1C(c1nnn(C(C)(C)C)n1)=O C(=O)(CCCCCOC(C)C)N1CCC(N(C(C2CC(OC)C2)=O)C2CC2)CC1 C1(NC(c2cc(Cl)ns2)=O)CCCC(CNC(C2(Cc3ccccc3)CC2)=O)C1 c1(CNC(c2cc(C)c(O)c(C)c2)=O)ccc2c(c1)CN(C(c1ncc[nH]1)=O)C2 c1(NC(=O)NCC2CC3C(C2)C3(F)F)nc2c(s1)CC1(CCCC1)CC2 n1(CC)ncc(NC(=O)C(O)CCNC(=O)C=CC2(C)COC2)c1C C1(C(=O)NCC(CNC(C(C)(C)Cc2cccc(Cl)c2)=O)(C)O)NC(=O)OC1(C)C C#Cc1cccc(C(N2CC3CC(C2)C3(C)C)C(=O)Nc2ccccc2Cl)c1F O=C(CC1=CCCC1)NCC1C2CN(C(=O)CCNS(=O)(=O)CC)CC12 c1(-c2cn(C)nc2)nc(C2CCCCC2)nn1CCCn1ccnc1 C1(NC(CCN(CC=C)CC)=O)CC(NC(c2cccc(C=C)c2)=O)C12CCC2 c1(CN2CCCN(C(c3c(OC)cc(O)nc3)=O)CC2)cccc2c1ncn2C Cc1ccn2nc(C(=O)NCC(C)(C)NC(c3cnnc(C4CC4)c3)=O)nc2n1 c1(C(N2CCCC(N(C(CNC(CC)=O)=O)C)C2)=O)cc2occc2[nH]1 C12(C(=O)NCC3CCN(C(c4ccoc4)=O)C3)CC3CC1C2C3 CCC(C)(C)C(C(=O)N1CCOCCC1c1cn(CCCOC)nn1)N(C)C CCCCC(CNC(c1ccc(-c2cccs2)s1)=O)NC(c1nc(O)sc1C)=O C1(F)(CNC(c2cnc(O)s2)=O)CCN(C(=O)C(c2ccc(Cl)cc2)O)CC1 c1(CN(C(=O)C(c2c(F)cccc2F)(C)O)C)cccc(S(N)(=O)=O)c1 c1(C(C)=O)ccc(NC(C2CCC(NCc3ccc(Br)cc3C)CC2)=O)cc1Cl Cc1cnc(C)c(C(=O)NC2(CCO)CN(C(c3cn[nH]c3)=O)C2)c1 C1(CNC(C(C)(C)C)=O)CC2(CCC2)CN1C(C1CC=CCC1C(F)(F)F)=O N1(C(c2n(CC(C)C)ncc2)=O)CC2CCC(NC(=O)Cc3cn[nH]c3)CC2C1 C=CC(CC)CC(=O)NCCCCC1CCCN(C(=O)Cc2cn[nH]c2)C1 c1(C(=O)NC2C(NC(c3cc(C(C)=O)on3)=O)CCC2)c(C)[nH]c(C)c1C c1(OC)c[nH]c(C(=O)N(CCNC(C2CCOC(C)C2)=O)C(C)C)cc1=O c1(C(=O)NC)ccc(C(=O)NCCC2(O)CN(C(=O)C=CCCC=C(C)C)C2)cn1 N1(CC)CCN(CC(=O)OC)CC1.C1(C)C(=O)N1C(C)=O.c1(CCCS)cccs1 C1(CC=C)(C(=O)OC)CCN(c2nc(CO)cs2)C1.c12ccc(cc1)c(=O)[nH]2 C(c1ccc(C)cc1C)=CC(=O)NCC(CC=C)NC(=O)C(C)(O)C(C)C C(=O)(CC(C)(C)CC(F)F)N1CC(NC(c2nc(C)c(C)[nH]2)=O)C(C)C1 C1(CNC(c2c(CC)[nH]c(=N)s2)=O)C(C)CCCN1C(=O)C(O)C(C)C c1(C(C)C)cc(C(=O)NC2CC23CCN(C(=O)CCCF)C3)cc(O)n1 Cc1cc2ccc1On1cc(cn1)CNC(=O)N2.c1(OC(C)C)ncccn1 N1(C(c2cnccc2Cl)=O)CCC2CCN(C(C3(F)CC4(CCC4)C3)=O)CC2C1 N1(C(C=COCC)=O)CCC2(CCC(CNC(C3CN(C)C3)=O)O2)CC1 C(=O)(C1=CCS(=O)(=O)C1)NC1CN(C(CS(C)(=O)=O)=O)CC1F C1(c2cn(C(C)C(N3CCC(CO)C34CC4)=O)nn2)CCCCCCC1O c1(CCNC(c2n(C(CC)C)nnn2)CC(C)C)cccc(Cl)c1Br c1(OC)c(CN)cnn1C.C1(C(=O)OC)CCCN1C(=O)CC1CCCN1C(C)=O C1(CCC(=O)NCc2ccoc2)CCCN(C(=O)CCCn2cccc2)C1 N1(C(C(C(C)C)(C)O)=O)Cc2ccccc2CC1CNC(=O)CC1CCN(C)C1 Cc1oc(C)c(C(N2CC(NC(=O)CCc3cnoc3)C(C)C2)=O)c1C c1(C(N2C(CNC(C34CC(OC)C3C4)=O)COCC2)=O)cccc(C)c1F C1(NC(c2nnc(C)s2)=O)CC(O)CN(C(=O)Cn2cc(C3CC3)cn2)C1 C1(C#N)(C(=O)NC(C)(C)CCNC(=O)COC2CCCCCC2)CCCCCC1 C1(C(N2CCC(NC(Cn3nnc(=N)[nH]3)=O)(CF)C2)=O)CCc2nc[nH]c2C1 C1(C(=O)Nc2ncc(C(=O)OC)s2)CC(F)(F)CN1Cc1cccc(OC)c1O C=C(C)C1OCCC1C(=O)NCCNC(c1c[nH]nc1C)=O N1(C(c2c(C)n(C)nn2)=O)CCN(C(=O)CC(C)NC(c2ccccc2)=O)CC1C c1(NC(C=Cc2nnn(C)n2)=O)csc2c1CCCC2 C(=O)(CC(C(C)C)OCC(C)C)N1CCC(NC(C2CC(CC)(CC)C2)=O)CC1 C1(CNC(COCCOCC)=O)CNCCN1C(C1CN(C2CCOC2)C1)=O c1(C(C)(C)C)cc(CC(N2CCC(c3cn(Cc4ccc(Cl)s4)nn3)C2)=O)no1 CCCCC(CC)CC(=O)N1CCCC(Nc2nc(C)nc(Cl)c2C)CC1 c1(C(=O)NC(C)CNC(C2CCOC(=O)N2)=O)ccc2c(c1)NC(C)CC(=O)N2 C(c1ccc(F)cc1)=CC(=O)NC1CCC(NC(c2cccn2C2CC2)=O)CC1 N1(c2ncnc(=N)[nH]2)CCCC1C1CCCCN1C(=O)CC(=O)c1ccco1 c1(NC(=O)NC)cccc(NC(C)C(N2CCCC(n3cc(C4CC4)nn3)C2)=O)c1 c1(C(=O)NC(CN(CCC)CC)C)ccnc(NC(=O)C(C2CCCC2)SC)c1 c12cccc(c1)CCC1CN(C1)C2=O.n1(CC)cc(-c2ccccn2)nn1 CC1(C)CCCCC1CNC(=O)CCC1CCN(C(C23CCC(C2)C3(C)C)=O)C1 N1(C(COCC(=O)NC)=O)C2CCC1C(CNC(=O)COC1CC(C#N)C1)C2 C1(C(=O)NCC(CO)NC(C)=O)CCN(C(c2cc(CO)on2)=O)CC1 C1(NC(C2CCC(C)O2)=O)CCC(CC(=O)NCCc2cnn[nH]2)CC1 CCCCC(C)C(=O)NC12CC1CN(C(c1coc(C(F)F)n1)=O)C2 c1(CN2C(C(=O)Nc3cc(C)cc(O)c3)CC(O)CC2)cc(C#N)ccc1Cl c1(C(C)NC(=O)NCC(=O)N(CC(C)C)CC#C)ccccn1 N1(C(C2(n3ccnc3)CC2)=O)CCC(n2nccn2)CC1 CC(C)S(=O)(=O)CC(=O)N(C(C)CNC(c1ncoc1C(F)(F)F)=O)C N1(C(CN2CCN(C)CC2)=O)CCN2CC1C2=O.C1(SC2CC2)C=CS(=O)(=O)C1 C1(CNC(c2ncccc2Cl)=O)C2CN(C(C3(CF)CC3)=O)CC12 C(=O)(C1CCCc2sccc21)NC(C)CNC(C1(C2CCC(=O)NC2)CCC1)=O C(=O)(C(=O)N=S(C)(C)=O)NC(CCCNC(CN1C(C)CCC1C)=O)(C)C C(=O)(C(F)C(C)(F)F)N1C(C2(C(=O)NCc3n(C)cnc3)CC2)CCC1 C(=O)(CCCC(=O)N1CC(=O)NCC1C(=O)NC1CN(CCF)C1)OC CS(=O)(=O)c1ccnc(N2CCC3NC(=O)CCC3C2)n1.c12nccc(n1)N2 N1(c2ncc(C)cn2)C2CCC1CC(CNC(=O)CC1(O)CCCN(C)C1)C2 Cc1cnc2ccc(C(=O)NC3(CNC(C4(Cl)CC4(C)C)=O)CC3)cn12 Cc1ccncc1CC(=O)NC1CC(CNC(=O)CSCc2cccnc2)C1(C)C c1(SC)cccc(C(=O)NCC2C=CC(NC(c3ccc(C4CC4C)o3)=O)C2)c1 N12CCCCC1C2=O.c1(CNCC(C)CN2CCOCC2)scnc1C(F)(F)F Cc1nc(CC(N2CCCC2CCNC(c2csc(C3CC3)n2)=O)=O)cs1 C12(C(=O)NC3CC4(C(NC(C5C6CCC(=O)C65)=O)C4)C3)CCCC1C2(F)F N1(C(c2cn(CC(C)C)nc2)=O)CCCN(C(c2cnc(C(C)O)s2)=O)C(C)C1 Cc1cncc(C)c1C(=O)NCC(C)(C(C)C)NC(C1CC2CCC1CC2)=O C1(F)(CC)CCN(C(=O)C(n2cc(-c3nn(C)cc3C)nn2)C)C1 N1(C(C(C)=C2CC2)=O)CCC(C(=O)N(C2CC2(C)C)C)C1 c1(CC(C=O)NC=O)ccc(C)c(C)c1.n1(C2CC2)cc(-c2c(C)nsc2C)nn1 c1(OCCC(=O)NCC(C(C)C)NC(Cc2nc(C)sc2)=O)ccccc1O.CN CCCC(CCCNC(=O)COCC(=O)OC(C)(C)C)NC(c1cc(C)n(C)c1)=O C=C1CCC(C(=O)NCCC2CCN(C(C3CC(OC(C)(C)C)C3)=O)C2)CC1 C1(NC(C(C)OCCC#C)=O)COC2(CCN(C(c3ccnnc3O)=O)CC2)C1 CCC(C)CCCCC(=O)NCCCOCCC(=O)NCCCCC(C)(C)C c1(C2(C=O)CCC2)nccc(Nc2cccc(CS(N)(=O)=O)c2)n1.NC N1(C(c2c(C)ncnc2)=O)CC2(NC(c3cccn3C)=O)CCC1CC2 Cc1ccc2sc(C(=O)NC3CC3NC(c3ccc([N+](=O)[O-])c(C)c3)=O)cc2c1 N1(C(C(CNC(=O)OC)C)=O)C(C(=O)NC(C2CCCC2)C)CCC12CC2 C1(NC(c2c(SC)scc2)=O)CCCCC1NC(c1[nH]c(C)nc1C)=O O=C(N=c1cnn(-c2cccnc2)[nH]1)NCC12CC(C1)C(c1ccccc1)O2 Cc1csc(C(C)C(=O)NC(CNC(=O)CN2CCC(C)C2)CO)n1 N1(C(C(C)OCC)=O)CCCC(N(C(=O)C(c2ccccc2Cl)C)C)C1 CC(C)CC(C(=O)NC1CCOC(CNC(C2(F)CCC2)=O)C1)C(N)=O C12(C(=O)NC3CCC(C)N(CCCc4cccc(F)c4)C3)CCCN(CCC1)C2 CC(CCN1CCCCC1)C(=O)N1CCC1C1CCCCC1 C12(CC(=O)N(C)CC3N(CC)CCC3)CCC1CN(C(=O)Cc1csc(C)c1)C2 c1(OC)cncc(NC(C2CCCC2CNC(c2cnsc2)=O)=O)c1 C1(C(=O)NCC(=O)NCc2c(C)nn[nH]2)CCN(C)CC1 c1(C(=O)NC(CCC2N(C(COCCOC)=O)CCCC2)(C)C)cc2ccsc2s1 c1(CC)cc(C(N2CCC23CC(c2ccsc2)C3)=O)nc(C(F)(F)F)c1 c1(COC)noc(COCC(=O)N(CCN(n2ncnn2)C)C2CC2)n1 c1(SCCC(N2CCCC(N(C(C(CSC)O)=O)C)C2)=O)ncnc2[nH]cnc12 Cn1cccc(C(N2CCOC(CCCNC(C3C4(CC4)C34CC4)=O)C2)=O)c1=O C=CCCCCC(=O)N(CC(C)O)CCNC(=O)C=Cc1cn(C)cn1 C(=O)(CCCCCC(C)O)NC1C(CNC(c2ccc(CC)cn2)=O)COC1 N1(C(C)C)CCC(C(=O)NC(C)(CNC(C2CC2F)=O)CO)CC1 CC(C)C(C)C(CNC(c1occc1Cl)=O)NC(c1ccc(C(F)(F)F)nc1)=O C12(NC(CC3ON=C(C)C3)=O)CCC1CN(C(=O)Cc1nccs1)C2 N1(C(CC2C(C)C2)=O)CCCC12CCN(C(c1cc3c(s1)CC(C)(C)C3)=O)C2 C(c1ccc([N+](=O)[O-])cc1)=CC(=O)NCC1CCCN1C(C1OCCOC1(C)C)=O C(C(C(C)(C)C)NC(c1cc(C(F)(F)F)ncn1)=O)NC(C1(CC#C)CCC1)=O c1(OC)cccc(NC(=O)CCN(CC2CC2)CC2CCCO2)c1 N1(C(c2c(CC)n[nH]c2)=O)CC(C)CN(C(c2cn(C)c(=O)c(C)n2)=O)C(C)C1 CC(CN1CCOCC1)N=c1ccc(NS(=O)(=O)c2ccccc2)n[nH]1 O=C1CC2(CCN(C(=O)C(c3cccc(Oc4ccccc4)c3)(F)F)C2)CN1 c12cc(Br)ccc1S(=O)(=O)N2.c1(CN(CCOCCC)C(C)C)cccc(Cl)c1 Cc1noc(C(C)C)c1C(=O)NC1CN(C(=O)C#CC2CC2)CC1F c1(C(N2CCC(N(CC#C)C(C3(CC)CC3)=O)C2)=O)ccc2cn(CC)nc2c1 CCC(O)C(F)(F)C(=O)NC(C)CC1CN(C(c2cc(=O)n(C)cn2)=O)C1 CCC(CCC(=O)NCCc1ccncc1F)NC(=O)C=Cc1ccsc1 CC#CCCC(=O)NC1CC(CNC(=O)CCCCC2CCCCC2)C1 C(=O)(C(C)(C)C(=O)NC)NC1CCC(C(N2CCC2(C)COC)=O)C1 CCC(C)(CNC(=O)CCC1CCCN1C(=O)C=CC1CCC1)CO C1(C(=O)Nc2c(OC(C)C)ccc(C#N)c2)CCc2cncn2C1 CC12CC(C(N3CCCCC3CNC(=O)CCNS(C)(=O)=O)=O)(C1)C1(CCC1)O2 c1(Nc2ccc(NC(C3CNC(=O)O3)=O)cn2)ccc2nccnc2c1 C1(C(N2CCC(N(C(Cc3ccc(OC)cc3)=O)C)C2)=O)Cc2ccccc2C1 c1(C(=O)OCC)[nH]nc(NCC2=CCCC2C(=O)OC)c1Cl C1(C(=O)NC(C#C)C(C)C)CC(F)CCN1C(c1n[nH]cc1C)=O c1(NC(C)=O)ncc(S(=O)(=O)NC2CN(C(c3nccs3)=O)CC2F)s1 N1(S(CCC)(=O)=O)Cc2[nH]nc(C(=O)NCc3ccc(OC(F)(F)F)cc3)c2C1 c1(C(=O)NCC(CC)NC(c2ccsc2OC)=O)cc(OC)cc(C)n1 C=CCC(CC(C)C)C(=O)N1CC(NC(c2nn(CC)cc2[N+](=O)[O-])=O)C(C)C1 c1(NC(C(C2CCN(CCC3CCCN3C)CC2)C)=O)ccccc1[N+](=O)[O-] CC1CCCN(C(=O)CCn2ccnn2)C1CNC(=O)CN1CCN(C)CC1 C1(CNC(C=Cc2c(C)nccc2)=O)(NC(=O)C=CC(C)(C)C)CC2CCC1CC2 CCC(C)C(O)C(C)C(=O)N1CCC(N(C(=O)CCc2csnn2)CC)C1 Cc1cc(C(=O)NCC(C2(O)CN(C(c3cn(C)nc3Cl)=O)C2)(C)C)cc(C)c1F C1(C(=O)NCC(C)(C)CNC(=O)C(F)F)CC12C1CC3CC(C1)CC2C3 c1(-n2ccc(C(=O)NCC(CC)NC(=O)C(C)SC3CC3)n2)ccccc1C C1(OC)CN(C(=O)COCC2CC2)CC1NC(=O)C(C1CCCCC1)O CC1CCN(C(C2(c3ccccn3)CC2)=O)CC1NC(=O)C(C)NC(N)=O c1(N(CCC)CCNC(=O)C(C)C2CCC2)ccc([N+](=O)[O-])cc1 C1(N(C(C(C)(C)c2ccccc2)c2nnnn2C2(C)CC2)C)CC2CC3C(C2)C13 N1(C(CNS(CC)(=O)=O)=O)CC(NC(=O)Cn2cc(C3CCC3)nn2)C(C)(C)C1 Cc1nc(Cl)ccc1C(N1CC(O)CC1C(=O)Nc1cnc(Cl)c(Cl)c1)=O CC1CCN(C(C2CC(CF)C2)=O)CCN1C(c1nonc1N)=O Cc1ncn(C)c(=O)c1C(N1CC(O)(CNC(C2(C#N)CC3(CCC3)C2)=O)C1)=O C1(OC)CC2(C1)CC(C(=O)NCC(C(C)(C)C)NC(C1CCC(F)(F)CC1)=O)C2 C=C(C)C(C)(C)C(=O)N1CC2CCC2(CCNC(=O)Cc2coc(C)n2)C1 N1(C(CC(CC)(C)C)=O)CCCN(C(C2(c3cccc(Cl)n3)CC2)=O)CC1C N1(C(C2(CC)CC2)=O)CCc2nc(CNC(c3ccncc3F)=O)sc2C1 C(c1c(Cl)cccc1Cl)=CC(=O)NCC(CNC(c1c(C)snc1)=O)CO Cc1nsc(N2CCC(NC(=O)CC3CC=CCC3)C2)n1 CCCCC(O)C(=O)NC1CN(C(=O)CCN(c2ccccc2)C)CC1O c1(NCc2onc(COCC)n2)ccc2[nH]cc(CC(=O)OC(C)C)c2c1 N1(C(C(CCC)(F)F)=O)CC(C(N2CCC(O)(C(F)F)C2)=O)CC(C)(C)C1 c1(C(N2CCC(C)(NC(CSc3ccc(C)cc3)=O)C2)=O)cc(N)c(F)cc1C C1(C(N(CC(C)NC(C=CCC)=O)C)=O)CC(=O)NC(=O)C1 C(=O)(N1CCCCCO1)C1CCC(C(=O)NC(C)(C)C)N1Cc1c(C)ccnc1 N1(C(CC2(OC)CCC2)=O)CC2(CC(NC(c3ccccn3)=O)c3nccn32)C1 C1(C(=O)NC2(CC=C)CN(C(c3cccc(C4CC4)n3)=O)C2)CC2C=CC1CCC2 c1(C(N2CC(C(C)(C)O)(CNC(CCCCCC)=O)C2)=O)cc2n(n1)CCCO2 c1(CC)cc(C(=O)NC2CN(C(=O)NC)C2)n[nH]1.C12(CCCC1)N(C)C2=O c1(N2C(C(CC)C)CCC2)nc(=NCC23CCC(C2)C(C)(C)O3)[nH]c2c1COC2 Nc1cc(Cl)ccc1C(=O)NC1CS(=O)(=O)CC1NC(c1c[nH]cc1C1CC1)=O C(CC(=O)N(CC(O)CNC(c1cccc(CC(C)C)c1)=O)C)(C(C)C)OCC N1(CC(=O)NCC2CCCN(C(c3cncnc3)=O)C2)C(=O)C=CC1=O CCC(N=c1ccnc(NCC(C)CC2CCCCC2)[nH]1)C1CCOCC1 c1(C(N2CC(CCNC(C(C(C)C)O)=O)C2)=O)cc2ccnc(Cl)c2s1 C1(NCC)CN(C(C2C3CCC23OCC(=O)OC)=O)CC1CCO.C1(CO)CC1 c1(OC)cc(C(=O)NCCCc2ccccc2)cnc1NC1CC2(CO)CC1C2 CCCC(C(=O)NCCCC(CO)NC(=O)C(C)N1CC(C)C1)C(C)C C(=O)(CC1=CSC2=NCCN12)NCC1(O)CCN(C(C2CCCC(C)C2)=O)CC1 S(=O)(=O)(c1c(C)cccc1Cl)N1C2CN(C(CCCC=C)=O)CC21 N1(C(C2C3CN(C(c4nnn(C)c4C(F)F)=O)CC32)=O)CCn2cncc2C1 Cc1ccc(N2CCCC(NC(C3CC(C)(F)C3)=O)C2)c([N+](=O)[O-])c1 C1(CC(N2CC3(CC(NC(C4(OC(C)=O)CC4)=O)C3)C2)=O)C(=O)NCC(=O)N1C c1(C(=O)NCC2CCC(NC(CCC(=C)Cl)=O)C2)cc(OC)c(S(N)(=O)=O)s1 C1(C(N(C)CC2CCCCN2C(=O)Cc2ccnc(O)c2)=O)OC2CCC1CC2 Cc1cc(C(=O)N(C(C)C(=O)N(C2CC(C)(C)C2)C)C2CC2)cc(F)c1 CC(C)(C)C(C(=O)NCC1CNC(=O)CO1)NC(=O)CNC=O c1(C(=O)NCC2CCC(C)N(C(=O)COC3CCC3)C2)cc2ccccc2cn1 CC1CC23CCN(CC2)C(=O)C2(CCCC(=O)N1C3)CCC2.C1(C(N)=O)CC1CF C1(CC(=O)NCC2(n3ccnn3)CC2)CCCOC1.C12C=CC(C1)NC2=O c1(CCc2nnc(-c3ccccc3)o2)cccc(-c2cn[nH]c2)n1.CC(C)(C)O C1(O)(OCC)CC2CCC(C1)N2N1CCN(c2ccc3cccc(F)c3n2)CC1 N1(C(CCn2c(C)cc(C)n2)=O)CCN(C)C(CNC(C2CC(O)CN2C)=O)C1 C1(NC(=O)C(c2cccnc2)O)CN(C(c2cncc(F)c2)=O)CC2(CC2)C1 C(=O)(CCS(N)(=O)=O)N1CC(NC)C(SC2CC2)C1.c1(C(=O)N)ccc(C(N)=O)cc1 N1(C(c2cc(C)no2)=O)CCC2(CCCN2c2nc(C(C)C)ccc2C#N)CC1 CC1CCN(C(C2CSC2)=O)C(CNC(=O)CN(C)Cc2ccccc2Cl)C1 N1(C(c2ccns2)=O)CCC(C2CCN(C(c3cnc(C(F)(F)F)s3)=O)C2)CC1 N1(C(C(c2cn(C)nn2)NC(CCCSC)=O)=O)CCC(F)(F)C(C)C1 c1(C(N(CCC(C(C)C)NC(=O)CC(C)CF)C)=O)ccc2c(c1)CN(C)CC2 Cc1sc2ncnc(N3CCCC(C)(CNC(=O)C=Cc4cnc[nH]4)C3)c2c1C N1(C(C(c2nc(CC)sc2)N)=O)CCOC(C(=O)OC)C1 C(=O)(C1CCCc2c[nH]nc21)NC1(CC=C)CCN(C(c2cc(N)ccn2)=O)C1 Cc1ccc(CC(=O)NCCC2(CC=NC(=O)C(C)NS(C)(=O)=O)CCC2)o1 C12(C(=O)NCCCCNC(C=CCN(CC)CC)=O)CCCN1CC(O)C2 c1(C(CNC(c2c(Br)noc2C)c2n(C(CC)C)nnn2)(C)C)ccc(F)cc1 CCCC(C)(CCC)C(=O)NCC(CC(C)C)NC(c1cnn2c1OCC2)=O Cc1cc(C(N2CC=CC2C(=O)NCC2COC(=O)N2)=O)c(C)s1 C1(NC(C(C)OCC#C)=O)C2CC1CN(C(=O)C(N1CCC(C)C1)=O)C2 C1(NC(c2sc(CC)c(C)c2)=O)CN(C(c2ccc(F)cc2O)=O)CC12CC2 C1(C(=O)NC2(C(=O)OC)CCC2)(CNC(=O)C(C)Cc2ccco2)CCCC1 Cc1cnc(C(=O)NCC2(NC(c3csnc3C3CC3)=O)CCCCC2)nc1 C=CCCCCCN=c1ccn2ncc(S(=O)(=O)NC(C)CC(N)=O)c2[nH]1 C1(CC=C)(NC(c2nc(Cl)ccc2Cl)=O)CCN(C(C2(Br)CC2)=O)CC1 C(CO)(C(C)N)NC(=O)CN(C(c1cc(C(N)=O)[nH]n1)=O)CCC.C(CC(C)C)CC c1(C(=O)NCC(CCNC(C2C(=C)C2)=O)OC)cnn(C)c1Cl n1(CC(=O)N(CCN(CC(C)O)CCOC)C(C)C)cc2ccccc2n1 C1(C(N2CCC(OCCOC)C2)=O)CN(C(c2c[nH]cc(Cl)c2=O)=O)CCC1(F)F C(=O)(C1CSc2ccccc21)NC1C(NC(C=Cc2c(C)n(C)nc2)=O)COC1 C1(CC(=O)Nc2cc(I)ncn2)(CNCc2c(CC)nco2)CCCC(=O)N1 N1(C(CC(C=C)C)=O)CC(CNC(c2cncc(N(C)C)c2)=O)CC1(C)C C1(C(=O)NC(C#C)CC2CC2)CCc2nc(C#N)sc2C1 c1(C(=O)NC(C2(O)CN(C(c3nc(C)c(C)s3)=O)C2)C)ccc(Cl)nc1C CCCCC(CNC(C1CN(C(=O)CCC2CCOC2)CC1C)=O)CCC N1(CCNC(C(C)n2cccn2)=O)CCN(C(C2(C)C=CCCC2)=O)CC1 c1(OC)ccc(CCNC2CCC(=O)N(C)C2=O)c(F)c1 C1(NC(c2cccc(=O)o2)=O)CCC2(CC1)CC(NC(=O)C(O)CC1CC1)C2 c1(C(=O)NCCN(C(=O)C(C)OC2CC2)CC(C)O)cnc(C(C)(C)C)o1 c1(C(=O)NCC2(NC(C=CC(C)(C)SC)=O)CC2)cc(C)n(C)c1C c1(C(=O)NCC2(O)CCN(C(C(CC)(CO)OC)=O)C2)c(Cl)nc2ccccn12 c1(C(N(C2CC(C(=O)NCC(O)CC3CCCC3)C2)C)=O)ccn(C)n1 N1(C(C(Cn2cccn2)NC(c2nn(CC)c(O)c2)=O)=O)CCC2(CCSC2)C1 N=c1c(C(N2CCC(NC(=O)CC3CCOCC3)CC2)=O)c[nH]c2ccccc12 NC(=O)CC(O)C(=O)NC1CC2(C1)CC2C(=O)NCCOc1ncccn1 C1(C(N2CC(CNC(C3(CC#C)CCOCC3)=O)C2)=O)CC12CC(F)(F)C2 N1(C(C2CCC(NC(COC)=O)C2)=O)CCCSc2cc(C)ccc21 C1(O)(C(N(C)CCNC(C2CCC2C(C)(C)C)=O)=O)CCc2ccccc2C1 N1(C(C(C)=CCC)=O)CC(C(=O)NCc2cn(CC3CC3)nn2)CCC1(C)C c1(NC(=O)NC(CCOC)(C)C)c(N)cccc1Br Cc1c(O)ccc(CN2CC(CC(=O)O)CC(C)C2)c1C c1(C(C(=O)NCC(C2CCCCC2)NC(C2C(=C)C2)=O)C)ccccc1F c1(C(=O)NCC=CCNC(c2cn(CCC)nc2)=O)csc(=NC)[nH]1 CCC(C(=O)NCC(C)CN(C)C)N(C)C(c1ccc(C)s1)=O Cc1ccc(C(=O)N(C)CC2COCCN2C(=O)CCCc2nc(C)no2)cc1 CC(C(=O)N1CCC(NC(c2cc([N+](=O)[O-])n[nH]2)=O)C(O)C1)S(N)(=O)=O N1(C(Cn2c(C)ncc2)=O)CC(NC(c2cc(C(F)(F)F)cc(F)c2)=O)C(C#N)C1 C1(CCOC)(NC(=O)C(C)CS(C)=O)CCN(C(c2ccnc(CO)c2)=O)CC1 C(CCCCCNC(c1ccc(Cl)cn1)=O)NC(c1c(COC)ncs1)=O C(c1ccc(F)cc1)=CC(N1CCN(C(c2n[nH]cc2Br)=O)CC1)=O C1(CC(=O)NC(CC)C(=O)NC23CC(F)(C2)C3)CCOC1(C)C N1(C(C(CO)NC(CSCCC(C)C)=O)=O)CCNC(=O)C1 N1(C(C(C)c2cccs2)=O)CC(NC(c2c[nH]cc2-c2cnn(C)c2)=O)C(F)C1 CC(C(=O)NCC1CC(C(=O)NC2(CN(C)C)CC2)C1)N1CCCC1 Cc1c(NCC(F)(F)C(F)F)ncnc1N1CCC(CC2CCC2)CC1 N1(C(CC(c2ccc(CC)cc2)C)=O)CCN(C(=O)CCCOC)C2CSCC12 c1(SCC)ccc(CC(=O)NC(C)C(C)NC(=O)Cc2cnn(C(F)F)c2)cn1 C1(O)(C(C(=O)OC(C)(C)C)(F)F)CCCN(C(N2CCC=C(Br)C2)=O)C1 N1(C(CS(CCC)(=O)=O)=O)CCC2(CC1)NC(=O)N(C)C2=O C=C(C)CC(C(=O)NCC#CC(F)(F)F)NC(=O)CCn1cnnn1 c1(C(N2CC3(CC(NC(C(C)n4cccn4)=O)C3)C2)=O)cc2cccnc2[nH]1 c1(OCC(=O)Nc2cn(C)nc2)ccc2c(c1)OCCO2 C(=O)(C(C)CCC(C)(C)C)NC(C(=O)OC)C.N12CCC(C1C#N)NC2=O C1(NC(C(CC)SC)=O)CC1C1CCCN(C(c2cc(C)n(C(F)F)n2)=O)C1 C(=O)(C1=CS(=O)(=O)CCC1)N1CCC(C2CC2)(CNC(C2(OC)CC2)=O)C1 O=C(CC1=Cc2ccccc2C1)NCCC1CCCN(C(=O)C(O)CC2CC2)C1 CCCC(CC)C(=O)N1CCCC(N(C(C2CC2C2CCCC2)=O)CC)C1 c1(C(C)C)ncncc1C(=O)NC(C)CNC(c1ccc(SC(F)(F)F)s1)=O CN1CC(=O)NC1CC(=O)NC12CC(NC(C3CC34CC4)=O)(C1)C2 N#Cc1ccc(C(N2C(C(=O)NCC3COCCO3)CC3CC23)=O)c(O)c1 CC(CCC(=O)N1CCC(CN(C)C)C1)NC(=O)CCC1CCCOC1 C1(NC(c2c(CC)nns2)=O)CN(C(C2CC(F)C2)=O)C2(CCOC2)C1 c1(C(=O)NCC(CC=C)NC(c2cc(F)ccc2C)=O)c(F)ccc2[nH]ccc12 CC1(C)OCCC1CC(N1CCSCC1C(=O)NC1C=CC(CO)C1)=O c1(CC(=O)N(C2CC(NC(C3C(C=C)CC3)=O)C2)C)nc(C2CC2)nn1C C1(N(C(CNC(=O)OCC)=O)CCO)CCN(C(=O)C(Br)=C(C)C)CC1 C1(CC(=O)NC(C2CC(NC(C3(CC=C)CCCC3)=O)C2)C)CC(CC)=NO1 c1(CNC(C2CCN(C(=O)COCC3CCCCC3)CC2)=O)cc(F)cc(F)c1 C12(C(=O)NCCCCCNC(C(CC=C)CC)=O)CC(CO)(C1)OC2(C)C c1(N(C)CC)ccc(C(=O)N(CC(C)CNC(=O)C(C)(C)OC(C)=O)C)cc1 c1(NCC2(C)CC(F)(F)C2)ccc(S(=O)(=O)NCC2CSCCO2)cc1Cl c1(C(=O)NC(c2ccccc2)CNC(=O)CCc2nccs2)cc(Cl)nnc1O CC1CCCC(OCCNC(=O)CCC(=O)NCCSc2nccs2)C1 c1(C(=O)NCC23CC2CN(C(C2CC2C(F)F)=O)C3)ccc2oc(O)nc2c1 C1(NC(C(c2cncn2C)C)=O)CCC(C(=O)NCCn2ccnc2)C1 n1(CC)ccc(CC(=O)NC(C)(C)C(C)NC(=O)OC(C)(C)C)n1 C1(NC(C2(C)CC=CCO2)=O)CCN(C(c2scnc2Cl)=O)CC1O c1(C(C(=O)NC)N(C(CCO)c2cccs2)C)cccc2cncn12 N1(C(C2(CCCC)CC2)=O)CC2CCCC2(NC(c2onc(OC)c2Br)=O)C1 N1(C(CCS(=O)(=O)NC)=O)CC2ON=C(CNC(=O)COCC3CC3)C2C1 C1(C(F)(F)F)(C(=O)NCC(C)CNC(=O)C(F)=C2CCCC2)CCOCC1 c1(ON(C)C)cncc(C(=O)NCC2C3CC3CN2C(=O)C#CC(=O)CCC(C)C)c1.OC C1(C(=O)NCC2C(NC(c3ccc(-c4ccccn4)s3)=O)C2)CCC(F)CC1 CC(C)CCCCC(=O)NC1CN(C(=O)C(c2ccccn2)C)C(C)(C)C1 c1(C(=O)NCCCN(C(c2ccoc2C(C)C)=O)CC)nnc(O)nc1O N1(C(CC2(C#N)CC2)=O)CCC2CCC(NC(=O)C(O)Cc3cnc[nH]3)C1C2 C(=O)(C1=CNS(=O)(=O)N=C1C)NC1CC2CN(C(CCSCCC)=O)C1C2 CCCCC(CNC(c1cc(C)n(CCO)n1)=O)NC(C1CCCO1)=O CCC(C)(C)CC(=O)N1CC(NC(c2cc(N(C)C)nc(Cl)c2)=O)C1 c1(C(=O)NC(COCCOC)C(C)C)ccccc1NC(c1ccns1)=O C(=O)(C1CCCc2c(O)cccc21)NC1(COC)CN(C(=O)C(O)C(F)(F)F)C1 Cc1ncc2n1CCC(C(N1CCC(N(C)C(c3ccnc(O)c3)=O)C1)=O)C2 C(CCN=C(NCc1n[nH]c2c1CCCC2)NCc1ccns1)SC Cc1nn(C)cc1CC(=O)N(C1CN(C(c2nn[nH]c2C(F)(F)F)=O)C1)C CCC(CN(C)C)C(=O)N1CCC(C)(NC(c2ccoc2)=O)C1 CCC1=C(C(=O)NC2CCCC(NC(=O)CSCc3cccs3)C2)SCCO1 Cn1nc([N+](=O)[O-])cc1CNC(=O)NCC(=O)NCC1(C)CCC1 N1(C(CC(CC)(F)F)=O)CCOC2(C1)CN(C(=O)C(O)CN1CCOCC1)C2 N1(C(CCC(N)=O)=O)Cc2ccc(CNC(c3cn[nH]c3)=O)cc2C1 c1(C(=O)NC(CNC(CSCC#C)=O)C)ccc(NS(=O)(=O)CCCC)cc1 Cc1cc(C(=O)NCC2(C)CCCC2NC(c2cn(C)c(=O)cn2)=O)nnc1O N1(C(c2cccc(CNc3ncn(C)c(=O)c3)n2)=O)CCSC2CCCCC12 c1(OCC(=O)NC2(CN(C)C(c3cnn[nH]3)=O)CC2)ccc(F)cn1 c1(C(=O)NCC2CC(OCC)C2)sccc1S(=O)(=O)NC N1(C(c2c(C)csc2C)=O)CC(C(=O)NCCC(C)CO)C2(CC2)C1 C1(CC#C)(C(=O)N(C2CCC3CC23)C)CCN(C(C2CCOC2C)=O)C1 N1(C(c2c(C)cccn2)=O)CC(C(=O)NC2CC(O)C2N(C)C)C2(CC2)C1 N12CC(C(C)(C)C1)C2=O.c1(CCCNC(CC(C)C)=O)ccccc1C(F)(F)F C12(C(N(CCN(C(C)C)C(c3cccc[n+]3[O-])=O)C)=O)CC3CC(C(=O)N1)C2C3 CC1C(NC(c2cccc(S(C)=O)c2)=O)C(C)CCN1C(c1cnn[nH]1)=O N1(c2ccnc(C(CC)C)n2)CCC(NC(C2CCCCS2)=O)C2(CCC2)C1 CC1CN(C(=O)CCc2cscn2)C1C(=O)Nc1cccnc1 C1(Cn2cc(-c3ccco3)cn2)(CNC(=O)CSC(F)F)CC12CCC2.n1(C)ccnn1 N1(C(C2(C)CC(NC(CCCCN(C)C)=O)C2)=O)CC(C2CCCCC2)C1 N1(C(C2N(CC)CCCC2)=O)CC(NC(c2cc(OC)ccc2Cl)=O)C2(CC2)C1 N1(CC#C)CCOC2(CCCN(C(c3cc([N+](=O)[O-])cc(C)c3C)=O)C2)C1 CCC(CC(=O)N(C(C)C(=O)N(CC(C)(F)F)C)C(C)C)OC C1(C(=O)NCC(N2CC3CCC3C2)=O)CC2C(C1)C2(F)F C1(C(=O)NCC2N(C(C3CCC3)=O)CCCC2)CCc2nnc(C(F)(F)F)n2C1 c1(CC)cnn(CC(=O)N(CCC(=O)NC2CSCC2C)CCO)c1 c1(CCCNC(C(C)NC(=O)NC)=O)cn(CCC(C)C)nn1 C1(NC(c2n(C=C)nnc2)=O)CN(C(=O)CN2CCC(C)C2)C2(CCC2)C1 Cc1ncc(C(=O)NC(C)CCCNC(C2(C(C)(F)F)CC2)=O)[nH]1 N1CCS(=N)(=O)C(C)C1.Cc1c(-c2ccc(C(F)(F)F)cc2)n[nH]c1C=O N1(C(c2cc(C)[nH]n2)=O)CCC2(CC1)CN(c1ccnc(S(C)(=O)=O)n1)CCO2 N1(C(c2c(CC)cno2)=O)CCCC(N(C(=O)CC2CCOC(C)(C)C2)C)CC1 N1(C(CCN2CC2=O)=O)CCC2CCC12.C(C(C)C)N(CCOC)C c1(C(N2CC3CCN(C(=O)CCC(F)F)C3C2)=O)cc(Cl)c(F)cc1F CCC(C)C(C(=O)N1CCCOC(CNC(c2cc(C)c(C)[nH]2)=O)C1)OC N1(C(c2c(CC)n(C)nn2)=O)CC(NC(=O)CN2CCC(C)CC2)C(C2CC2)C1 c1(OC)cnc(Cl)cc1C(=O)NC(C1(CNC(=O)CCC(F)(F)F)CC1)C CC#CCCC(=O)NC1CCN(CCNC(C23CCOCC2C3)=O)CC1 CC(O)C(F)(F)C(=O)NCC(C)NC(=O)C(C)(O)CCc1ccccc1 CCC(C(=O)N1CCCC1CNC(=O)C(C)=C1CCC1)SC N1(C(COC(C)C)=O)CC2CC(NC(=O)CC(C)n3cccn3)CC1C2 c1(C(=O)NC2C(C)CCN(C(=O)Cc3cncnc3)C2)cc(F)c(O)c(F)c1 c1(C(=O)NC)ccc(C(=O)N(CC(O)CN(C)C(C2CC(=O)N(C)C2)=O)C)cn1 Cn1ccc2nc(N(C3CCCCNC3)C(c3cccc(Br)n3)=O)ncc12 C(=O)(CCCS(N)(=O)=O)NC1CC(NC(c2cnc(N)c(CO)c2)=O)CC1O n1(C(C)C)[nH]cnc1=NC(=O)C(=O)NC(C)CF N1(C(c2nc(C)n(C)n2)=O)CC2(CCN(C(C3(N=[N+]=[N-])CC3)=O)CC2)C1C(C)C C(=O)(C1=CS(=O)(=O)CCC1)N1C(C)CCC(NC(=O)C=Cc2ccc[nH]2)C1 C1(C(C)C)CC(CC(=O)N(CC(C)(C)CNC(=O)CC2(C#N)CC2)C)CCO1 N1(C(C2CCN(C(CC(C(CC)C)O)=O)C2(C)C)=O)C2CCC1CC(C)(O)C2 CCC(C)(CO)C(=O)N1CC2CC2(CNC(=O)COCc2nnc(C)s2)C1 N1(C(CC(C=C)(C)C)=O)CCCCCC(NC(c2occc2C)=O)C1 c1(CNC(C2CC(CC)C2)=O)cccc(NC(=O)C(C2CCCO2)OC)c1 N1(C(CNC(c2ccc(C)cc2)=O)=O)CC2=C(C1)CN(C(c1ccc(C#N)o1)=O)C2 c1(CN2CCN(CCC(=O)N(C)C)CC2)ccc(F)c(C(F)(F)F)c1 C1(NC(C2(CNC(C3CCC(=O)C3)=O)CCC2)=O)CCC2(CCC2)C1 CC1=C(C(=O)NC2CCN(C(c3ccncc3N)=O)C2)Cn2ncnc2N1C Cc1noc(C)c1C(=O)NCC1C=CCN1C(=O)COCC(F)(F)F C(=O)(C1CCCc2nc(C)[nH]c21)NCC1(C)N(C(c2cncc(C)c2)=O)CCC1 c1(C(N2CCC(C)(NC(=O)C(O)C3CC3)CC2)=O)cc([N+](=O)[O-])ccc1Br c1(CN)ccc(C(N2CCCC2CNC(c2ccc(C3(C)CC3)cc2)=O)=O)cn1 CN1C(=O)SCC1C(N1CCC1CNC(c1ncccc1OCCF)=O)=O C12(C(N(CC(C)NC(c3n(CC#C)ccc3)=O)CCOC)=O)CC1COC2(C)C C1(CNC(C2CCCN(C(C3(C(=O)NC)CC3)=O)C2)=O)C2CCC3C(C2)CC13 N1(C(c2c(C)cccc2Cl)=O)CCC2(CCC(NC(=O)CC34CCCC3C4)C2)C1 Cc1ccn(C(C)CC(=O)N2CC(CC(C)NC(c3cncnc3)=O)C2)n1 c1(S)ccc(CC=O)cc1.C1(NC(=O)CN2CCSCC2)CC(F)(F)C1 c1(N2CCCC(NC(c3ccc(CC#N)cc3)=O)CC2)ncc2nccnc2n1 Cc1cc(C(N2CCOC(C)(CNC(=O)COCCCF)C2)=O)c2n[nH]cc2c1 C1(NC(C2N(CC)CCCC2)=O)Cc2ccccc2C1NC(C1CC=CCO1)=O CC(=O)CCCC(C)C(=O)NC1CN(C(=O)C2=CCCC2)CC12CCOCC2 c1(CN(C(C=C)C)Cc2nccs2)cc(OC)c(OC)cc1C(F)(F)F C1(NC(c2cncnc2C2CC2)=O)CC(O)CN(C(c2cc(Cl)c(Cl)s2)=O)C1 N1(C(C(C2CCN(C(C(C)C(=O)OCC(C)C)=O)CC2)C)=O)CCC(C)(C2CC2)C1 C1(SCC(=O)NC2CCN(C(C3(c4ccncc4)CCC3)=O)C2)CCCC2CC12 c1(NC(C2C=CC2C2CCN(C(=O)OC(C)(C)C)CC2)=O)cc2scnc2[nH]1 c1(C(=O)NC(C#C)CC2CCC2)cccc(COCC(C)C)c1 C1(NC(C2(OCC)CCCC2)=O)CC(C(=O)NCC2(C#N)CCC2)C12CCC2 C(CCCC(=O)N1CC(CCCCNC(=O)C(C)CCN(C)C)C1)SC c1(C(=O)NCC(CNC(c2c(CCC)nco2)=O)O)cncc(OC(C)C)c1 N1(C(c2cccc(=S)n2O)=O)C2CCCC1CC(n1cc(C(=O)O)nn1)C2 c1(OC(CC)C)ccc(C(N2CCC(F)(CNC(=O)OC(C)(C)C)C2)=O)cn1 C(=O)(CC(=O)NCC)NCC(C)N(C)C(c1cnn(C2CC2)c1)=O C(=O)(C1=CCCCN1C(=O)OC(C)(C)C)N1CC(NC(COC(C)C)=O)C(C)C1 c1(NC(=NCc2ccc(C(C)(C)C)cc2)NC2CCCC2)ccc2occc2c1 C(C1=CCN(C(=O)C(c2ccccn2)O)CC1)NC(C=C(C)Cl)=O C(=O)(C(O)P(C)(C)=O)NC1CC2(C(NC(c3cc(OC)nn3C)=O)C2)C1 c1(C(C(=O)NCC(C)NC(CC2(C(=O)OCC)CCCC2)=O)C)ccc(C)cc1 N1(C(=O)CCc2cncnc2)CC2CC2(C(=O)Nc2cncc(C(F)F)c2)C1 C1(NC(C2CCCN(C(C(CO)OC)=O)C2)=O)CC12CCOCC2 C1(NC(CC)CC2CCN(S(C)(=O)=O)CC2)CCCC(C)(C)C1 C#CC1(CNC(C2CCN2C(=O)CN(C)C2CC2)=O)CCOCC1 CC(CNC(C12CC(F)(C1)C2)=O)C(F)C(=O)NC1CN2CCCC1C2 N1(C(CP(C)(C)=O)=O)CCOCC(CNC(=O)C(O)C2CCC2)C1 C1(C(N2CCCC(C)C2CCO)=O)(OC)CCN(C(=O)CCc2nccs2)CC1 Cc1cc(C(=O)N(C)CCN(C)C(c2nocc2C(C)(C)C)=O)sn1 C1(CCC)CC(C(N2CC3C(CNC(=O)COc4cc(C)on4)C3C2)=O)CCO1 c1(C(C(=O)NCCOCC)N(C(C)CCC(C)C)C)nn(C)nc1Br c1(CC(=O)NCCN2CCC(NC(C3CCOC3)=O)CC2)c(Cl)cccc1Cl C1(CNC(C2CCCN(CC)C2)=O)CC2(C1)CN(C(=O)COc1ccon1)C2 C12(C(N(CCN(C(C(CC)COC)=O)C)C)=O)CCC(C(F)F)(CC1)CC2 CCCC(CCC)C(=O)N1CCCC1C(C)NC(=O)COCc1nc(C)no1 C1(C(=O)NCC(CCNC(c2cc(OC)ncc2)=O)O)Cc2cc(Cl)ccc2O1 c1(OC(C)C)cccc(-c2ccccc2CNc2cnc(Cl)cc2I)c1 c1(CC)ccc(F)c(C(=O)NCC2(C)CCN(C(c3nc(C4CC4)cs3)=O)C2)c1 Cn1ncc(C#N)c1C(N1CCC2(NC(=O)Cc3cnc[nH]3)CC2C1)=O N1(C(CC2ON=C(CC)C2)=O)CCC2(CC(NC(=O)CCN(C)CCO)C2)C1 c1(C(N(CCCNC(c2ccsc2-n2cnnn2)=O)CC)=O)nc(Cl)ccc1F c1(NCC)cc(=NC(C)c2ccco2)[nH]c(NC(=O)OCC)n1 c1(C(=O)NCC(CNC(c2c(CC)nc(C)n2C)=O)C)cnc2n[nH]c(C)c2c1 N1(C(C2C(CNC(c3ccc(O)nc3)=O)CC2)=O)CCC2CCCC2CC1 N1(CC(=O)NC(CSCC)C(=O)N2CCC2c2ccc(O)cc2)C(=O)CCCC1=O CC1(C)CC(=O)N(CC(N2CC(NC(C3CCCC34CC4)=O)C3(CC3)C2)=O)O1 c1(C(N2CC(NC(CC3CCCC(OC)C3)=O)C2)=O)cc(Br)cnc1C c1(Oc2c(CNC(CC(C)c3ccncc3)=O)cccc2)ccc(Cl)cc1Br C12(CNC(C3(C)COC3)=O)CCC(CNC(=O)C#CC(C)(C)C)(CC1)CO2 C=CC(C)(O)CC(=O)N1CCOC(CNC(=O)CCc2ccc(C)c(C)c2)C1 C1(CNC(C(C)O)=O)COCCN1C(c1cc(C(F)(F)F)n[nH]1)=O C(CC(=O)NCC1(F)CCOCC1)(C(F)(F)F)NC(C(COC)C)=O C#Cc1ccccc1CC(=O)NC(C)(C)CCN(C(=O)CCCC#CC)C CC(C(=O)NCC1(NC(C2CSC2)=O)CCOC1)C(=O)N1CCOCC1 n1(CC(=O)NC2(C)CC(NC(CCCC(C)(C)C)=O)C2)nc(O)c2c1CCCC2 CC(O)C(C)(C)CNC(=O)CC1(C)CCN1C(C1CC2CCC2C1)=O Cc1ccc(Cl)cc1C(N1CC(CC(C)NC(C2CC(N3CCCC3)C2)=O)C1)=O C1(NC(c2csc(Cl)c2)=O)CCOCC1NC(C1CC(F)(F)C1)=O c1(CNC(C2C(C)CCCC2)=O)ccc(C#N)cc1F.C12CC(C)(C)CN1C2=O N1(C(c2ccc(NS(C)(=O)=O)nc2)=O)CC2ON=C(CNC(=O)COC(F)F)C2C1 c1(C(=O)NCC(CCNC(c2c(COC)cco2)=O)O)cc2nc(F)ccc2o1 C(=O)(C1c2ccccc2C2CC1C2)NCC1C(CNC(C2(CCC=C)CC2)=O)C1 C(=O)(C1=C(CF)N(c2cccc(F)c2)C(=S)NC1c1cccc(OC)c1)OC c1(C(=O)NCCN(C(C)C)C(c2cccc(N)c2F)=O)ccc(F)cc1F C1(NC(CSC(=N)N)=O)COC2(C1)CN(C(c1cc(C(F)(F)F)on1)=O)C2 C1(NC(C2(CO)CCN(C(c3c(C)csn3)=O)C2)=O)CC2C(C1)C2(F)F C1(=CC(=O)NC(CN(C(c2c(C)cccc2O)=O)C)C)C2CC3CC(C2)CC1C3 CC1CCN(C(C2CCSC2)=O)CCN1C(c1ccc(CO)c(F)c1)=O C1(NC(C=CCOC)=O)CC2C1CCN2C(c1nnn(C)c1N)=O Cc1cc(C(=O)NCC2CCN(C(=O)CCC3CC3(F)F)C(C)C2)cc(N)c1O N1(Cc2c(N)c(Br)ccc2)CCC2CN(Cc3ccccc3)CC12 CC1C2C(CCN2C(=O)C2=C(C)CC2)CN1C(=O)COc1ccc(CO)cc1 C1(NC(=O)C=CCF)CCC(CCNC(c2cc(CCO)on2)=O)C1 c1(C(=O)NCC(CNC(CCc2nc(C)sc2)=O)C)nccc2c1NCCC2 C(CC1=CCCCCC1)NC(C1N(C(CCCOC)=O)CCC(C)C1)=O C1(C(C)(C)NC(C2CC2(F)F)=O)CCN(C(=O)CCc2ccccc2)C1 c1(N(C(C2(CNC(c3[nH]nnc3CC)=O)CC(=C)C2)=O)C2CC2)ccc(F)cc1O C12CCCC3CN(CC13)C(=O)N2.CC(CCC1CCCO1)NC(=O)OC(C)(C)C c1(CCC(=O)NCCN(CC(C)O)C(=O)CN2CCCNC2=O)cncc(F)c1 c1(NC(CCC)CNC(C2CC23CCSCC3)=O)ncnc2onc(C)c12 CCC(C(=O)NC1CC(NC(c2c(Br)ccc(F)c2F)=O)C1)C(C)(F)F C(=O)(C(CC(C)(C)CC)NC(=O)OC(C)(C)C)NC1CCCN(CC=C)C1 N1(C(CC(=C=C)C)=O)CCCC(NC(c2csc(CC)c2)=O)CC1 c1(COC)cc(=NCC2CC(C)N(C(=O)CCc3ncccn3)C2)[nH]cn1 c1(CN2CC(=O)N(Cc3nnn(C)n3)C2=O)nc2cc(F)c(F)cc2[nH]1 Cc1ccccc1-n1cc(C2CN(C(C3CCC(C(C)(C)C)C3)=O)C2)nn1 Cc1nncc(CN(C(C23CC(C)(CN2C(C2CCC4(CCC4)C2)=O)C3)=O)CC)c1C C1(C(N2CCCN(C(c3c(C)ccs3)=O)C(C)C2)=O)CCC(=O)N2CCCCC12 C1(NC(C(CCC)NC(N)=O)=O)CN(C(=O)C(C)(C)SC)CCC1(F)F Cc1cc(-c2cn(CC3CCCN3C(=O)CCOC(C)C)nn2)sc1C N1(C(Cn2c(C)cc(C)n2)=O)CCC2(CCCN(C(C3CCCC34CC4)=O)C2)C1 Cc1nnn(C)c1C(=O)NCCC1CN(C(=O)C(c2cnn(C)c2)O)CCO1 CC1(C)CCC(=O)N(NC(=O)c2cncc(-n3cnnn3)c2)C1 c1(OCCC)ccccc1NCC(O)CNC(=O)C(C)(C)CNC(=O)C1CC1 c1(-n2c(C3(F)C(C)C3)nc(Cc3cccc(Br)c3)n2)cc(Cl)ccc1CO c1(C(=O)NC2(C)CCCN(C(Cc3cc(C)on3)=O)C2)cnc2[nH]nnc2c1 CC1=C(C(=O)NCCC2CCCN(C(=O)CCc3ccoc3)C2)CCCC1 c1(C(=O)NCCCC(C)NC(c2c(OC)n[nH]c2)=O)nn(C)nc1C C1(C(=O)NCC2CC3CCN2CC3)(CC)CNCCC1O C1(C(=O)Nc2cc(F)c(Cl)cn2)CCC2(CN(C(=O)CCN3CCOC(O)C3)C2)O1 c1(C(=O)NC2CCN(C(c3c(C)cc(C(F)(F)F)s3)=O)C2)c(C)cc[nH]c1=N CC(C)(C)C#CC(=O)N1CC(NC=O)C(N)C1.C1(NC(=O)OC(C)(C)C)CC(O)C1 C(=O)(C1=CC2C=CC(C1)C2)N1CC(CC(C)NC(C(C(CC)C)OC)=O)C1 Cc1ccc(C(c2nnnn2C2COC2)NC2CC(=O)N(O)C2)c(C)c1C N1(C(CC2CCC(C)O2)=O)CCCC12CCCN(C1CC1)C2=O Cc1cc(C#N)ccc1OC(c1cnn(-c2ccccn2)c1C)=O Nc1cc(C(=O)NC2CCCC(NC(c3sccc3Cl)=O)C2)c(F)cc1F c1(C(=O)NCC2CN(C(CC=CCC)=O)C(C)C2)cn(C)c2ncccc12 c1(C(N2CC(NC(C(CN(CC)CC)F)=O)(CO)C2)=O)cc2ncccc2o1 CC1(CCNC(=O)COc2ccccc2Cl)CCN(C(=O)C=C(Cl)Cl)CC1 C1(CC)C(NC(c2sc(C)nc2C)=O)CCN1C(=O)C(CO)NC(N)=O Cc1ccc(F)cc1-c1cn(Cc2ccccc2Br)nn1.N12CCN(CC1)CC2 c1(C(=O)NCCC2CC(CNC(C(C)N3CCC3)=O)C2)c[nH]nc1C(F)(F)F c1(C(N(C)CC2CCN(C(CN(C(COC)=O)C)=O)C2)=O)c(C)ncn1O c12ccccc1N(Cc1ccc(Cl)cc1)C2=O.C1(C(=O)OC)CC1C(=O)N(C)C N1(C(C2CCC(=C)CC2)=O)C2CCC1CC(CC=C)(NC(=O)CCS(C)=O)C2 C1(C(=O)NC(CNC(C(C)OC2COC2)=O)(C)C2CCC2)CCC(NC(N)=O)CC1 Cc1nc(-c2ccc(C(=O)NCCCN(C(=O)Cc3cc[nH]n3)C)s2)cs1 C1(C(N2CCC(CNC(=O)CC3OCCO3)C2)=O)(OC)CC(CF)C1 c1(Nc2c(C(C)C)nns2)nccc(=NC(C)C2CCN(C)CC2)[nH]1 c1(COC)cc(C(=O)NC(C)CCNC(C2(C)CCCO2)=O)no1 N1(C(CNc2nc(OCC)sn2)=O)CCC(NC(=O)CC2CC2C)CC1 C=CCC(CNC(c1ccc(OC)s1)=O)C(=O)N(CCC)CCC C1(C(N2CC(CNC(CNS(CC)(=O)=O)=O)(OC)C2)=O)COC2CCCCC12 C12(CNC(CC(CC=C)(C)C)=O)CCCCC1CN(C(=O)CN(C)CC)C2 C1(C(=O)Nc2c(CC)nn(C)c2)C(C)OCCN1C(=O)C(N1CCOC1=O)C c1(C(C)Nc2ccc(CN(C)C)nn2)ccnc(F)c1 c1(C(=O)NC(c2cccs2)C)coc(CNC(c2nc(Cl)cs2)=O)n1 C(=O)(C(F)C(C)(C)O)N1CC2C(CNC(c3c(C)oc(-c4cccs4)n3)=O)(C2)C1 c1(C(N2C(CNC(CCCNC(C)=O)=O)CCC2)=O)cccc2c1NCC(C)C2 Cc1nc(O)sc1C(=O)N(C1CN(C(=O)C(C)C(C)C)C1)C C(=O)(C1Cc2ccccc21)NC(C1(n2ccnc2)CC1)=O.C1(=O)C(O)CCN1 C1(C(N(CCOC)CC)=O)CCCCCN1C(c1cnncc1OC)=O C1(CNC(CC2(CC(=O)OC)CC2)=O)CCN(C(C2CC(OC)C2)=O)C1(C)C N1(C(C(C)(C)C2CCN(C(C3CCCC(=O)N3)=O)C2)=O)CCCC2(CC2)C1 c1(C(=O)NC(CSC)(C)C(=O)NCCOCC(C)(C)O)ccc(C)c(O)c1 C1(CNC(c2c(C#C)cn(C)n2)=O)CN(C(=O)C(C)(C)n2cccn2)CCC1(F)F C1(NC(=O)C=Cc2ncc[nH]2)CC2CCC(C1)N2C(c1ccc(F)c(Cl)c1)=O N1(C(C2CC3(CC(=C)C3)C2)=O)CCC(N=c2cc(C)[nH]c(C(=O)OC)n2)C(C)C1 C(=O)(Nn1ccccc1=O)C1(NC(C2CC(C)OC2C)=O)CCCC1 CC(O)CCC(=O)N1CC(C)CC1C(=O)Nc1cc(I)ncn1 c1(C(N2CC(N3CCN(C(C(C)C#N)=O)CC3)C2)=O)cc(N(C)C)c(C2CC2)nn1 N1(C(CSCC=C)=O)CCCC1CN(C)C(C1OCCCO1)=O N=c1[nH]cnc2c(C(N3CCC4(CC3)CC4CNC(c3cn[nH]c3)=O)=O)cnn12 c1(C(=O)NC2CCC(F)(CNC(C(CCCC)O)=O)C2)ccc2c(c1)CCC=C2 N1(C(c2c(NC(C)C)ccc(Cl)c2)=O)C2CCCC1CN(C(C1C(C)C1C)=O)C2 C1(NC(C2N(C(Cc3c(C)n[nH]c3)=O)CC=CC2)=O)COC2(CCCC2)C1 C(CCC(O)C(=O)NC1(CN(C)C)CCCC1)NC(CSCCCC)=O C(=O)(C(CO)C(C)(C)C)N1CCC(NC(COCCCCCC)=O)C1 C(C(CNC(=O)Cc1cc(F)cc(F)c1)C(F)(F)F)NC(C1N(CC)CCC1)=O C1(COC)(NC(c2cnc(OC)cn2)=O)CCCN(C(c2occc2C)=O)C1 CC1(C)CN(C(c2cccc(Br)c2F)=O)CC1NC(c1ccncc1N)=O C(=O)(C(C)(C)C(=O)NC1(CNC(c2cc(F)n[nH]2)=O)CCCCC1)OCC CC1(C)CN(C(C2CC3CCC3C2)=O)CC1CNC(c1cncc(OCF)c1)=O c1(C(N(CCCCNC(=O)COC2CC=CC2)C)=O)ncccc1N(C)C C1(OC)CCC(CC(=O)NCC(=O)NCC(N2CCC(F)(CF)C2)=O)CC1 c1(CCC(=O)NCC2CC(F)(CNC(=O)OC(C)(C)C)C2)ncccc1F c1(NC(C2C=CC(NCc3cnc[nH]3)C2)=O)ccc(Br)nc1CCC c1(NC(CN2C3CCC(CCCC=C)(C3)C2)=O)cccc2c1CCC2 CC(CC#N)(C(=O)N1CCC(O)(c2ccccc2)C1)Nc1ccc(F)cc1 N1(C(C(C2CC2)OCC)=O)CCC2CN(C(C3(CF)CC=CCC3)=O)CC2C1 N(C1CCCc2n[nH]cc21)C(CCC1(C)CN(C(=O)OC(C)(C)C)C1)=O N1(C(C(C(C)NC(c2n(COC)ncc2)=O)(C)C)=O)CC(=O)N2CCCC2C1 Cc1cc(NC(C2CCCCC2NC(=O)C(C)(F)C(C)(C)F)=O)c(O)c(C)n1 C1(O)(C(=O)NC(CC)CN2CCCC2)CCN(C(C2CC(=O)N(C)C2)=O)CC1 N1(C(CCc2scc(C)c2)=O)CC(C)N(C(=O)CCN2CCCS2(=O)=O)CC1C C1(CNC(CN(C)C2CC2)=O)CN(C(=O)CC2(O)CCCCC2)CCCO1 c1(CC)ccnc(C(=O)N(C)Cc2nocc2C(=O)NC2CCC(O)C2O)c1 N1(C(CC(=O)OCC)=O)CCN(C(c2cc3sc(C(C)=O)cc3s2)=O)CCC1C C1(CC(=O)NCC2(F)CC(NC(C(CC)OC(C)C)=O)C2)Cc2ccccc2C1 C#CCC(C(=O)NCc1cncs1)NC(=O)CC1CCCOC1 c1(C(N2CCN(C(C(n3c(C)ncc3)C)=O)CC2CO)=O)cc2ccccn2c1 c1(OC)ccc2c(c1C)N(C(=O)CCn1ncn(C)c1=O)CCC2 c1(C(=O)NCCCCN(C(=O)C(O)C(F)F)C)ccc2c(c1)CCCC(=O)NC2 c1(OC)ccc2ccccc2c1CN1CCC1C(=O)NC1CSC1 C(C1Cc2ccccc21)NC(=NCCC#C)NC(c1ccc(Br)cc1)C C(=O)(C(C)(Cc1ccc(Cl)cc1)NCC(c1cccc(C)c1)(F)F)OCC N1(C2CCCCC2)CCC(NC(=NCC2CC2)NCC2CC3(CC3)CO2)CC1 CCCCC(C)C(=O)NCC1CCCN(C(=O)CCN(c2ccccc2)C)C1 C(=O)(C1COc2ccccc21)N1CC(CCNC(=O)CNC2CCNC2=O)C1 Cc1[nH]nc2c(C(=O)NC3CC(F)(CNC(=O)CCn4cccn4)C3)cccc12 C1(CNC)CC(N=c2[nH]cnc3cnn(C)c23)C1.C1(CC)CCCOC1 C1(C(=O)NC(CC(C)C)COC)(NC(C=CCC)=O)CCC(C)(C)C1 N1(C(C2CCCC(NC(C3CCCN(CC)C3)=O)C2)=O)CC(C2CCCCC2)C1 c1nc(=NCCC2COCCO2)[nH]c2c1COC2.O=C1OCCN1C1CCC1 C=CCC(C)(C)CC(=O)NCC(CNC(=O)Cc1sc(C)nc1C)CO N1(C(c2c(C)scc2)=O)CCC(OCCCNC(C23CC(C)C2C3)=O)CC1 N1(CC2C(CC(=O)N(C)CC)CCC2)CCCC(C(N(CCF)CC)=O)C1 C(=O)(CC(C)CNC(C1(C)CC1(C)C)=O)NCCN1CC(OC)C1 N1(C(COCCOCC)=O)CC(N(C)C(C2CC3CCC2CC3)=O)C(C)(C)C1 C1(C(N2CC(CO)C2)=O)CC(C(C)=NO)C1(C)C.CCCCCCOC.C1C(=O)N1 C1(C)(CNC(c2c[nH]c(=NC)s2)=O)CN(C(C2CCC(F)(F)C2)=O)CC1C Cc1nc(Nc2cc(C)c(O)cn2)c2cccnc2n1 C1(NC(c2ccc(SC)s2)=O)(CO)CCN(C(c2nc(C)ccc2C)=O)CC1 c1(C2N(C(C3NC(=O)C4CCC34)=O)CCC2)ccccc1[N+](=O)[O-] c1(C(N2CC(NC(C(C)C)=O)C2)=O)nn(-c2ccccc2F)c2c1CCCC2 c1(C(N2CC(OC(=O)CC(C)CF)C(CNCC)C2)=O)cc(F)c(F)cc1Cl C1(NC(=O)Cc2cccnc2O)CCCCC12CCCNC2 N1(C(CN(C)C)=O)CCCC2(C1)CN(C(c1ccccc1Sc1cc[nH]c1)=O)C2 c1(C(=O)NC(CC=C)CNC(=O)C(COC)N(C)C)cc(Cl)c(OCC)c(Cl)n1 c1(C(N2CCC(N(C(=O)CCn3cnnn3)C)CC2)=O)cc(F)c(CO)c(F)c1 N1(C(c2ccsn2)=O)CC(NC(C2CC(c3cccc(Cl)c3)(O)C2)=O)C(O)C1 N1(C(C2(C(C)C)CCC2)=O)CC2CCN(C(c3cccc(C#N)c3)=O)C2C1 Cn1cc2c(n1)CCCC2C(=O)NCC1(C)CCN(C(=O)Cn2cnnc2O)C1 C(C(F)(C(=O)NC(C)(C)CCCO)C(C)C)NC(CCCOCCOCC)=O c1(C(N(CC(CO)(CO)NC(Cc2c(C)noc2)=O)C)=O)cccc2ncsc12 N1(C(CN(C2CCNC(=O)C2)C(C2C(C)(C)C(=O)C2)=O)=O)CCCCCCC1CO N1(C(c2c(OC)scc2)=O)CCCC(C2(NC(C3COC4COCC34)=O)CC2)C1 C1(CC)CCCCCCN1C(=O)C(C)NC(C1CC(=O)C12CCC2)=O N1(C(CC(C)C2CCCO2)=O)CCCOC(CNC(=O)CC2(CO)CC2)C1 N1(C(CCCOCCC)=O)CC(C(F)(F)F)CC1CNC(=O)C(CC)SC C1(C(N2CC(COC)(NC(C3CCN(S(C)(=O)=O)C3)=O)C2)=O)CCCS1(=O)=O C1(C(=O)N(C(C2(Cc3nc(OCC)sn3)CCCCC2)=O)C2CC2)CCCNS1(=O)=O CCC(C(C)C)NC(=O)C#CCNC(c1cnc(C)o1)=O C1(N(CCOC)C(C2C(C)(OC)C2)=O)CCNCC1 C1(C(=O)NC)CCCCN1C(=O)CNC1CCN(c2cccc(F)c2)C1=O C(=O)(C1=C(C)CCOC1)N(CCCN(C(CCC(=C)C)=O)C)C(C)C CCCCCC(C)(C)C(=O)NCCCN(C(c1cnn(C)c1N)=O)C1CC1 CCC(CC(=O)N(CC(O)CN(C(=O)CCn1ccnc1)C)C)C(C)(C)C c1(NC(C(C)NC(C(CNC(CC)=O)CC2CCCC2)=O)=O)ccnnc1O Cc1ccc(C(=O)N(CC(C)(C)CNC(C2CS(=O)(=O)C2)=O)C)cc1Cl C(CCCCNC(C1CN(CC(C)C)C1)=O)N(C(C(C)SC)=O)C c1(C(N2CCC(CCCNC(c3[nH]n(C)c(=O)n3)=O)CC2)=O)ccc(O)c(Cl)n1 N1(C(C2(COC)COC2)=O)CCC(C)C(NC(c2ccncc2C(F)F)=O)C1 C1(NC(C2CC2c2ccccn2)=O)(CO)CN(C(C2CC23CCC3)=O)C1 C12(C(C(F)(F)F)NC(=O)NC3C(CC)C3)CC3CC(CC(C3)C1)C2 c1(C2(C(=O)Nc3nccc(CN)c3)CCCC2)cccc(F)c1F Cc1cc(C(=O)NCC2(O)CCOCC2)ncc1-c1cnn(C(C)C)c1 N1(C(c2c(C#C)c[nH]n2)=O)CC2(CCCC2)C1C(=O)NCCCc1cnccn1 C1(COC)CC(=O)N(C2CCN(Cc3c(C)ccn3C)C2)C1 c1(C(=O)NC(CCOC)C(=O)NCCc2cnc(C)[nH]2)c(C)cccc1O N1(C(=O)NCCc2nc(-c3ccc(C)o3)sc2)CCOc2ncccc2C1 c1(C(N(CCOCC)CC)=O)cc(I)c(Cl)cc1OC(F)(F)F Cc1ccc(C)c(C(N2CC(CC(=O)NOCC(O)C(C)C)CC2C)=O)c1 C1(C(N2C(CNC(c3c(C)ocn3)=O)CCCC2)=O)CCC(=O)N(CC(F)(F)F)C1 C1(C(=O)NCCN(C)C(c2cc(N3CCCC3)ncn2)=O)CN(S(N)(=O)=O)C1 c1(OC)ccccc1C1C(O)CCN1C(C1CC1c1noc(C)n1)=O c1(CN(C)Cc2snc(C)n2)cccc(Cl)c1Cl c1(C(N2CCN(C(C34CCC(CF)(CC3)CC4)=O)CC2)=O)cc(Cl)cc(F)c1F c1(CC)c(C(=O)NC(C)C(CO)NC(=O)CC2CCNC(=O)C2)cnn1CC C(CCC(O)C(=O)NC1CCCN(CCO)C1)NC(c1cccn(C)c1=O)=O CC1OCCC1CC(=O)NCc1cc(C(N)=O)co1.c12c[nH]nc1C(=O)NC2 c1(C(C)C)ccc2ccccc2c1.c1(CC(C)C2CCC2)nnnn1C1CCC1 C1(NC2C(OCCOC)COCC2)CCC2(CC1)CC(C(=O)O)C2 N1(CC(Cc2ccccc2)OC)CC2CC1CN2C(=O)CC1CCOC(C)(C)C1 c1(C(C(=O)NCCCC(C)NC(c2cn(C)[nH]c2=N)=O)O)cc(Cl)cc(Cl)c1 N1(C(CCCNC(C)=O)=O)C2CCC1CN(C(C1COCC1C(N)=O)=O)C2 C1(CNC(CCCN(C(C(C)CC2CC2)=O)C)=O)CCCOC1(C)C n1(CC(=O)NCC(C)CN(C(=O)CCc2cc[nH]n2)C)cnc(Br)c1 C1(N(C(c2ccc(CSC)o2)=O)C)CC12CCN(C(=O)CSc1cccs1)CC2 n1(CC(N2CC(CCCCNC(CCOCCOC)=O)C2)=O)ccnc1C CCCC(C(=O)NCC1(O)CN(C(c2ncoc2-c2cccs2)=O)C1)NC(N)=O C=C1CCN(C(=O)CN2CCC(OC)C2)C(C(N2CCC2CO)=O)C1 C1(CNC(c2cccc(C(F)(F)F)c2F)=O)CCN(C(=O)C(F)F)CC1(F)F CC1(F)CCN(C(C2CC(CNC(C3CC34CCOCC4)=O)C2)=O)CC1 c1(NC(c2n(C(CC)(C)C)nnn2)C2CN(CC(F)F)C2)ccc2nccn2c1 n1(CC)cc(CCOCCO)nn1.n1(C)cc(C)cn1.C1(=O)CCOC2CC(C2)CN1 C1(NC(CNC(=O)OC)=O)CC2CN(C(=O)CCC3CCOCC3)CC12 O=C(C1=CCSC1)NCC1(CNC(=O)CCc2ccoc2)CC1(F)F c1(SCC(=O)NCC2(NC(=O)C=C(Cl)Cl)CCOC2)nccc2ccccc12 c1(NC(=O)Nc2c(F)cc(Cl)cc2F)cccc2c[nH]nc12 N1(C(C2C(CCC)C2)=O)CCCC(C(=O)NCC)C1CC CCCCC(O)C(=O)NC1C2CC1N(C(C1CN(C3CCOCC3)C1)=O)C2 c1(CC)cc(C(=O)NC2CC(O)(CNC(=O)CCOC)C2)on1 CCCC(O)C(CO)NC(=O)C=CCN(C(=O)CCc1cnc(C)o1)C CC1OC2(C(=O)NC3CN(C(=O)Cc4cnccn4)CC3C)CCC1CC2 C(CC(C)(C)CC(=O)NCCSc1[nH]nc(SC)c1C#N)OC c1(C(=O)NCCN(C(C2C(C)(CC3CC3)C2)=O)CC)ccc(OCC)c(OC)c1 CCCCCCC(CC)C(=O)NCC1CCCN1C(C12CCC(CC1)C(C)O2)=O C1(NC(c2cc[n+]([O-])cc2)=O)CCN(C(=O)CCC2CC(N3CCOCC3)CC2)CC1F C1(OC)CC2N(C1)C(=O)C1(CC1)NC(=O)NC2.c1(NC)cccc(Cl)c1 C1(NC(C(CO)OC)=O)CCN(C(c2cc(C)[nH]n2)=O)C12CCC2 c1(CNC(C2CSCN2C(=O)CC2CCCC2)=O)ccncc1Cl C=CCCCC(C)(C)C(=O)N1CC2=C(C1)CN(C(=O)CCn1nc(C)nc1C)C2 CC1=C(C(=O)NCC2CC(C)CN(C(=O)CCC3CCCO3)C2)CCC1 C1(CC=C)(C(=O)NCC(=O)NOC)CCCN1C(=O)CC1CCCC(=O)C1 c1(OCC)ccccc1C(=O)N(CCC(C)NC(=O)C(=O)NCCC(N)=O)C c1(C(=O)NC(CC)CNC(=O)C=C(C)C(F)F)cc(OC)c(Cl)cc1Cl CCC(C)(C)CC(=O)NC1CC(CNC(=O)CCN2CCP(C)(=O)CC2)C1 c1(NC(c2c(C)nn(C)c2N)=O)cccc2c1OCCC2O C1(NC(=O)CCCc2cccs2)CN(C(c2cnns2)=O)CCC1C(F)(F)F c1(CN2CC(NC(c3ccc(C#C)cn3)=O)C(C)C2)ccccc1S(=O)(=O)CC c1(OC)nc(C(N2CCC(OCC(=O)NCC(C3CCCC3)O)C2)=O)co1 CC1CC(C(=O)NCC2CCN(C(c3cnn(CCF)c3)=O)CC2O)CC(=O)N1 C1(CNC(C2SCCS2)=O)N(C(=O)COC2CC=CC2)CCCC1(C)C N1(C(CCC=C)=O)CCC(CNC(=O)Cc2ccnc(F)c2)C(C)(C)C1 c1(C(N2C(C)CSCCC2)=O)cc(S(=O)(=O)NC2CCCC(O)C2)ccc1C#N c1(C(=O)NCC(CNC(C2(CC#C)CCCO2)=O)OCC2CC2)cccc(OC)n1 C(CC)(CC(F)(F)F)NC(C1(C#C)CN(C(=O)CCCC2CCCO2)C1)=O N1(C(CC=C=C)=O)CC2CCN(C(c3scnc3C(C)C)=O)CCC2C1 N1(C(C2C(CC)N(C(c3ccc[n+]([O-])c3)=O)CC2)=O)CCC(F)C(O)C1 CC(C(=O)O)C(C)N=c1ccn2ncc(S(=O)(=O)NC3(C)CCC(C)(C)CC3)c2[nH]1 c1(C(N2CC(C(=O)Nc3cc(C)c(F)cc3)C2)=O)cc2cccnn2c1 N1(C(CCOC2CN(C(c3c(=O)cc(C)[nH]c3)=O)C2)=O)CCCCN(C)CC1 C(=O)(C1=CCCCC1)NC(C(=O)NCC1CN(CC)C(=O)O1)Cn1ccnn1 CCC(C)CC(=O)C(=O)N(C)CC=CC(N1CCCC(F)CC1)=O C#CC1CCN(C(=O)CC2C(NC(C3COCC(C)O3)=O)CC2O)C1 N1(C(CCOC)=O)CC(C(F)(F)F)OCC1CNC(c1cc(C)c[nH]1)=O C(=O)(CCC(C)=O)NC(C1C(C(N(CC(COC)(F)F)C)=O)OCC1)C1CC1 C#Cc1cnn(CC(N2CCC(C(=O)NC(C)Cc3cccs3)(C(C)C)C2)=O)c1 C(=O)(C(C)(C)C(=O)NCCC1CCN(C(=O)Cc2cnc[nH]2)C1)OC c1(C(=O)NCCCC(C)(C)NC(C2C(=C)CC2)=O)c(C)ccc(Br)c1N c1(OC)ccc(C2(COC(C3CC(O)C(F)C3)=O)CC2)cc1Br c1(C(=O)NC(CN(C(=O)C(C)(O)C2CCOCC2)CC)C)cnccc1Cl c1(C(=O)NCC2C(NC(c3cn(C4CC4)cn3)=O)C2)cccc2c1CCC2 c1(C(=O)NCC(c2csc(Cl)n2)=O)cc(CNC(=O)NCCOC)ccn1 c1(C(N2CC(NC(C3(OC)CC3)=O)C2)=O)ccnc(C)c1Cl C1(CCC)CCCN(C(=O)CCN(C(C2(Cl)CCC2)=O)C(C)C)CC1 c1(C(N(C2CC3CCC(C2)N3)Cc2ccc(C)o2)=O)cc(Br)c(C)c(Br)c1 NS(=O)(=O)c1ccc(C(O)CNC(c2cc(F)ccc2F)=O)cc1 N1(C(c2nn(CC)c(O)c2)=O)CCC2(CC1)CCN(C(C1CC3C=CC1C3)=O)C2 C(CCSC)(C(C)(C)C)NCC(C)(C(N)=O)OC.OC c1(CC(=O)NC2C(C)CN(CCc3ccc(F)cc3)CC2)cccc2nsnc12 c1(COC(C2(SCC)CC2)=O)n[nH]c2c1CN(C(=O)CCC1(C)N=N1)CC2 Cc1nc(C)c(F)c(=NCC2CN(C(=O)C(c3cccc(Cl)c3)O)CC2C)[nH]1 C1(C(N2CCC2CF)=O)CCOCCN1C(C1CC2C(C1)C2(F)F)=O C1(NC(CCCCCC)=O)(CNC(=O)CC(C)COC)CCC(F)(F)CC1 C(CO)(CCCCNC(=O)C=C1CC1)NC(CCOC(C)C)=O CN1CC=CCC1CC(N1CCCCC1CCCNC(c1ccccc1)=O)=O CCC(O)C(F)(F)C(=O)NC1CC2(C1)CC(C(=O)NC1CC(=O)NC(=O)C1)C2 C1(COC)(CNCCCCNC(=O)CCC2CCCCO2)CC(=O)C1 Cc1cncc(OCC(=O)NCC2C(C)CCN2C(C2OCCCO2)=O)n1 C#Cc1ccc(CN2CC(c3nc(C(N4CC5C(OC)C5C4)=O)nn3C)C2)cc1 C12(CNC(=O)Cc3csc(Cl)c3)CCC(CC1)N2C(=O)Cc1cn[nH]c1 N1(C(CSCCC(C)C)=O)CCCC1CN(C(C1CC1(F)F)=O)C1CC1 C1(CCC)(NC(c2ccnnc2O)=O)CCCN(C(C23CCC2C3)=O)C1 N1(C(C(Br)=C(C)C)=O)CCCC2(NC(c3cccn4nccc34)=O)CC2C1 c1(C(=O)OCCC(C)OC)c(Cl)nnc(Cl)c1N C(=O)(C1=NNC(=O)CC1)N(CCCNC(C1CC2(C)OCC1C2)=O)CCO Cc1ccc(-c2noc(C(=O)N(C)C)n2)cc1F.N12CC(CC1C(=O)O)C2 C(=O)(CC(C)CCC(=O)N1CC=C(CNC(c2cccc(Cl)c2Cl)=O)CC1)OC C#Cc1ccc(C)c(NC(C2CCC(C)CN2C(c2ccc(F)s2)=O)=O)c1 CC1CCCC(CNC(C2(NC(=O)C(C)c3ccco3)CC2)=O)CC1 C1(OC)CC(C(N2CC(C(C)NC(c3cccn3C(C)C)=O)C2)=O)N(C(C)C)C1 N1(C(CC#C)=O)CCCCC1CCN(C)C(c1cncc(Br)c1)=O c1(N2CC(C#N)OCC2)ncc(S(=O)(=O)NC2CCCOC2)cc1Cl N1(C(C(C)CNC(c2ccco2)=O)=O)CC2(CNC(C3(C#N)CC3)=O)CCC1C2 c1(C(=O)NC2CCN(C(c3ccn(C(C)C)n3)=O)C2)n[nH]c2c1CCOC2 C=CCC(CNC(c1cnc(=N)[nH]c1)=O)C(=O)N1CCOC(CF)C1 c1(C(=O)NCCN(C(=O)CC2COc3ccccc32)C)ccc2ccccc2c1 N1(C(Cc2n(C)ccn2)=O)CC(O)CC1C(=O)NC1CN(C(N)=O)C1 C1(NC(C2(CC=C)CCCCC2)=O)CC(NC(C2(OC)CCCC2)=O)C12CCC2 C1(CCNC(CNC(=O)NC)=O)CC(OC)CN1C(c1ccn(C)n1)=O c1(OC)c(C(=O)NCC(C)(C(C)C)NC(c2ncccc2F)=O)cc(Cl)cc1Cl N1(C(C2CC(OC)(OC)C2)=O)CCCC2(C1)CN(C(=O)C(C)N=[N+]=[N-])C2 C=CCC(C)(C(=O)NC1(CNC(c2cc(OC)cc(C)n2)=O)CC1)N(C)C N1(C(C2N(C(C)C)CCCC2)=O)CCC2CC1CN2C(c1cnn(C2CC2)c1)=O C12(C(=O)NCCCN(C(c3cc(C(C)C)nn3C)=O)C)CSCC1C2(F)F c1(C(N2CCC(C(C)NC(C(C=C)(F)F)=O)C2)=O)cncc2ccccc12 c1(C(=O)NC(C2CC(NCc3c(OC)c(C)ccc3)C2)=O)c(C)cc(O)cc1C Cn1cc(C(=O)NC2CCN(C(C3(C#N)CC3)=O)CC2)c(C(C)(C)C)n1 CCC(CCOC)C(=O)NC1CCC1NC(c1c[nH]cc1-c1cc(F)cc(F)c1)=O C1(C(N2CCN(C3CCN(C(c4c[nH]c(=N)s4)=O)C3)CC2)=O)CC1C1CCCC1 Cc1cccc(C2(NC3CCN(C(=O)C(F)F)CC3)CCC2)c1 c1(C(=O)NCC(CC=C)NC(=O)CSCC(C)(C)C)nn(C)c2c1C(O)CCC2 C1(NC(C=Cc2c(C)ncs2)=O)COCCN(C(C2CCC(C)C2)=O)C1 N1(C(c2cc(=O)n(CCF)[nH]2)=O)CCN(C(=O)C(c2ccccc2)F)C2CCC12 CCC(CC)C(C)C(=O)N1CC2CC2(CNC(C2CC(n3ccnn3)C2)=O)C1 c1(C=O)cc(O)nc(O)n1.N1(N(C2(CCCCO)CC2)C)CCC(OCC=O)C1 C12(CNC(C(CC)F)=O)CCCC1N(C(c1ccc(Br)c(O)n1)=O)CC2 C(=O)(C(CC(F)F)NC(c1nccnc1N)=O)NCP(OCC)(C)=O C(=O)(C(CC(=O)OC)N(C)C)NCC1(O)CC(NC(CCN(CCC)C)=O)C1 c1(OC)ccc(C(N2CC(C(O)C(=O)N(C)CCN(C)C3CC3)C2)=O)cn1 CC(F)(F)C(F)C(=O)N1CCCC1(C)CNC(=O)CCC1CC1(F)F CC(C)(C(=O)NC1CCCC1(C)COC)C1=CCS(=O)(=O)CC1 C(=O)(CCC1=CCCCC1)N(CCNC(C=C1CCC(C)C1)=O)CCOCCO C1(CN(C(c2cnc(C(C)C)[nH]2)=O)C)CCCN(C(=O)CC2CCNC2=O)C1 CCS(=O)CC(=O)NC1CCN(C(c2cccc(C(C)(F)F)c2)=O)C1C(C)(C)C N1(C(c2ccncc2Cl)=O)CCc2nc[nH]c2C1.c12nocc1C(=O)NC2C c1(C(N2C(C)CC(CNC(c3cc4scnc4[nH]3)=O)C2)=O)ccc2c[nH]nc2c1 N1(C(c2ccc(C(=O)OC)[nH]2)=O)CC2CCCN(C(=O)CN(C)C(C)=O)C2C1 c1(C(N2C(CC(F)F)CN(C(C3(C(F)F)CC3)=O)CC2)=O)ccc2occc2c1 c1(CC)nc(C(=O)N(C)CC2CCCCN2C(=O)C(C)C2CC2)c(N)s1 c1(C(N2CC3CC2(COC2CCN(c4n(C)ccn4)C2)C3)=O)cnc2n1CCC2 C1(CNC(C(CC)OCC)=O)(NC(=O)CCCSC(C)(C)C)CCCCC1C N1(C(c2c(C)nn[nH]2)=O)CCC(NC(=O)CCC2CCCC2)C(CO)CC1 C1(C(=O)OC)OCCNCC1N(C1CCCC1SC)C(c1cccc(F)c1)=O c1(C(=O)NCC2N(C(c3c(C)nc(Br)cc3)=O)CCCC2)cccn2ccnc12 C1(CC(=O)N(C2CCN(C(=O)CC3(O)CCCC3)C2)CC)CCCCN1C C(C(C)(C)C1=CCCC1)NC(C1(C)CCCN1C(=O)CC1=CCCC1)=O C(C)(CO)(C(=O)N(CC(O)CNC(C1CCC(F)(F)C1)=O)C)OC c1(CSCC)nc(Cc2c[nH]nc2-c2ccc(F)cc2)n(-c2ccc(Cl)nc2)n1 CC1CCC(=CC(N2CCC(C(C)NC(c3cc(O)n(C)n3)=O)CC2)=O)CC1 c1(N2C(CNC(c3cccc(F)c3F)=O)CCC2)ncnc2c1SCCC2 N#Cc1cn(-c2ccccn2)c(=O)n(C(=O)c2ccc(Cl)cc2)c1=O.O1NC1=O N1(C(c2ccc(I)c(C)c2)C(=O)NCC(=C)C)C2CCC1CN(C)C(=O)C2 C(=O)(CCC(C)S(C)(=O)=O)NCC(C)(C)NC(CC(COC)C)=O Cc1cccc(C)c1CC(=O)N(CCNC(=O)CC(O)CSCCN(C)C)CC1CC1 N#Cc1cc([N+](=O)[O-])ccc1N1CCC(C2(NC(=O)COC3CCCC3)CC2)C1 C12(NC(=O)CCSC(F)(F)F)CCCN(C(=O)Cc3cnoc3)CC1C2 CC1SCCC1(c1nnnn1CCC1CC1)NCc1cccs1 CC1CC(O)CCN(C(C2CCC(CNC(C3CC4(CCC4O)C3)=O)CC2)=O)C1 C1(CC(=O)NCc2ccc(C(=O)NC(CCC=C)C3CC3)s2)CCCC(O)C1 N1(C(C(CC)OC)=O)CCC(C2CCCCN2C(=O)COC2CCOCC2)CC1 CC(=O)CCCC(C)C(=O)NCCNC(C1CCOC(C)C1)=O C1(C)(C(=O)NCC2(CCNC(c3c(C)n(C)cn3)=O)CC2)CCC(F)(F)CC1 Cc1cc(C(N2CC(O)CC2(C)CO)=O)ccc1S(=O)(=O)C(C)C C1(C(=O)NC(CCCCC)C2CC2)CCCCCN1C(=O)CCC(C)=O C1(NC(CCSCCC)=O)CCN(C(c2ccccc2C)=O)C12CCC2 C(=O)(CC(O)CC(C)(C)C)N1CCN(C(CC(CC)CC)=O)CCC1c1cn[nH]c1 c1(OC)ccccc1C(c1ccoc1C)NC(C1CC2(CCC2)C1)=O c1(NC2CC(NC(Cc3cc(C)no3)=O)C2)nc2c(cc1C#N)CCOC2 CCC(C)C(O)C(=O)NCC1(c2ccccc2F)CCN(C(=O)C=CCF)CC1 N1(C(c2cccc(CC)c2N)=O)CCC2(C=C(C(=O)NC(C)(C)C)C2)C1 CCC(CCOC)C(=O)NCC1(O)CCN(C(=O)COc2cc(C)cc(C)c2)C1 CC1(C)CCC(NC(C2COCCC2NC(=O)Cc2cncs2)=O)C1 c1(C(=O)NC(C)C(c2cccc(Cl)c2)C)ccc2cc[nH]c2n1 C1(C(N2CCC(C)(NC(C(C)c3ccco3)=O)C2)=O)CCc2ncnn2C1 C1(CCOC)CN(C(=O)COC(F)(F)F)CCN1C(c1cc(Cl)c(Cl)s1)=O c1(N2C(=O)CCN(c3ccc(C)cc3C)C2=O)cc(C#N)ccc1OC(F)F C(C)(N=c1nc2sccc2c(NCc2ccc(F)nc2)[nH]1)c1ccc(C)cc1C c1(OC)nccc(C(=O)NCCN(C(=O)CCn2ccnc2)C(C)C)c1Br c1(CC(=O)NC2CCC(N3CCN(C(C(C)(C)C)=O)CC3)C2)c(F)cccc1Cl C(=O)(C(C)(C)S(C)(=O)=O)NCC(CN(C(C12CCC(CC1)O2)=O)CC)(C)C Cc1ccc(CNC(C2CCCN(C(=O)NC3CC3C(F)F)C2)=O)c(C)c1 c1(CC)cc(C(N2CCC(C(F)F)(CNC(C3CC(=O)N3)=O)C2)=O)nn1C c1(C(=O)NC2CC(C(=O)NC(CC)CC)CC2O)ccc(CO)c(F)c1 c1(CC(C(=O)NCC2C(CNC(C3CN(C)C3)=O)C2)O)ccccc1Cl CC#CCCC(=O)N(C)CCNC(=O)CC1CCN(CC(F)(F)F)C1 CN1C(=O)CCC1C(N1CC2CC1C2NC(C1CCC(O)CC1)=O)=O C1(COC)(NC(C2CC=CCC2)=O)CCC(C)C1 c1(CNC(C2CCCN(S(=O)(=O)CCCCl)CC2)=O)ccc(F)cc1Cl C1(N(C(CCC2N(C(c3c(CC)csc3)=O)CCC2)=O)C2CC2)CCCC2(CC1)CC2 CC1(C(=O)NCc2ncoc2CCNC(c2cc(C(N)=O)c[nH]2)=O)C=CCC1 C#CCCCC(C)C(=O)N1CCN(C(c2ccc(C(C)(C)C)cc2N)=O)C(C)C1 N1(C(C(C)OCCC(C)C)=O)CCCN(C(C2CC3CCC2O3)=O)CC1 N1(C(C(C)NC2CCCCC2)=O)CC2CCN(C(c3ccc(Cl)cn3)=O)C2C1 C(=O)(C(C#N)C(C)(C)C)NC1CC2(CC(NC(c3cc(CC)no3)=O)C2)C1 c1(C(=O)NC(C)CCCCNC(=O)CC(F)F)cccc(O)c1F C1(N(C)C)CCC(C(=O)NC2CCCC2CNC(c2ccn(C(F)F)n2)=O)CC1 c1ccc(C(N2CC(N3CC(O)C3)C2)=O)o1.C12(CC1)CCNC2=O.COC N1(C(C(C)(C)CF)=O)Cc2ccccc2C(CNC(=O)Cn2cccnc2=O)C1 n1(CC(=O)NCC2OCCN(C(C(CC)(C)OC)=O)C2)ccc(=O)n(C)c1=O Cc1nn(C(C)(C)C)cc1C(N1CCC(NC(=O)C=Cc2cc[nH]n2)C1C)=O C(=O)(CCC(=O)NCC1CC(C)N(C(c2cc(COC)oc2C)=O)C1)NCC C(=O)(C1=C2CCCN=C2NN1)NC1CCN(C(COC2CCCC(C)C2)=O)CC1 C(C)(C(C(=O)Nc1cnn(CC)c1)C(C)C)NC(CC=C)=O c1(NC(C2c3ccc(o3)N2C)=O)ccccc1OC.C1(CC=C)(SC)CC1.CC#N C1(N(C(=O)C(CC)N(C)CCC)CC#C)CCN(C(c2cnc(Cl)s2)=O)CC1 C12(NC(c3ncc(Br)cc3F)=O)CCN(C(=O)C=C3CCOCC3)CC1C2 CCCCC(CC(=O)NC1(C(C)O)CC1)NC(C1(CO)CCCC1)=O C(CC(F)F)(C(=O)NCC1(C)CCCC1)N(C)C(C1CC12CCCCC2)=O c1(-c2onc(-c3c(CC)cccc3)n2)ccc2ncn(C)c(=O)c2c1 C1(O)(CC(=O)NCCN(CCOCCCC)CCOC)CCCCC1 C1(CC(NOCCOC)=O)CCCCN1C(=O)CC1(OC)CCCC1 C1(Cn2cc(C3(N(C)C)CCCC3)nn2)COCCN1C(c1ccncc1N)=O c1(COC)nc(C)c(C(N2CCCC2(C)C(N2CCC(CN(C)C)C2)=O)=O)o1 O=C(C1=CS(=O)CCC1)NCC1CCC(Oc2ccncc2)C1.C12(O)CN(C1)C2=O C(CC(=O)N=c1ccn(CC(=O)OC)[nH]1)N(C(=O)C(C)NCC1CC1)CC=C C(C(CC(=O)NCC1CC(NC(c2ccc3nn[nH]c3n2)=O)C1)C(F)F)N(C)C C1(C(N2C(C(=O)NC3(C(=O)OC)CCOCC3)CCC2C)=O)CC2C(C1)C2(F)F C1(CC)CCCCC1C(=O)NCCOCCOCCNC(c1n[nH]c(C)n1)=O C1(C#N)(CN(C)C(c2cnn(CCNC(=O)OC(C)(C)C)c2)=O)CCC1 CC1C(NC(C2(C)CCCCC2)=O)CCN1C(C1CCC1C(F)F)=O C1(CNC(C(c2cccnc2)NC(CNC(N)=O)=O)=O)CC2(CCC2O)C1 N#CC1CCN(C(=O)COC2CCN(C(=O)CC3CCC(=O)N3)C2)C1 N1(C(C2CCC(=O)NC2)=O)CC2CC(CNC(=O)Cc3ccc(O)cn3)C2C1 NC(=O)C(F)(F)CNS(=O)(=O)CC1C2CN(C(=O)OCc3ccccc3)CC12 C(=O)(C(F)CCC(C)(C)C)NCC(=C)CCNC(c1noc2ccccc12)=O c1(C(N(C2CCN(C(c3coc(CO)c3)=O)C2)CC)=O)cc2c(SC)cccc2[nH]1 C1(NC(C(CC)N(C(C)C(=O)NC)C)=O)CC2CCC(C1)N2C(=O)CC(C)(C)OC C12(NC(C=C(C)C(C)(C)C)=O)COCCC1CN(C(c1ccoc1C)=O)C2 N1(C(CC2C(CC)C2)=O)CCCN(C(C2(CF)CC2)=O)CC1 c1(C(C)(C)C)cnc(CCC(=O)NCC2(NC(C3CSCCS3)=O)CCOC2)o1 c1(C(=O)NCC=CCNC(C(n2cc(Cl)cn2)C)=O)ccc(C(F)F)nc1 c1(C(=O)NCC2N(C(C3(CCOC)CCC3)=O)CC2)cn(C)c(=O)cc1C N1(C(C(c2c(OC)cccc2Br)C)=O)CCC=C(C(=O)Nc2c(C)cccc2C)C1 C1(CC=C)(NC(c2c(C(=O)OC)cnn2C)=O)CCN(C(c2ccns2)=O)CC1 C#CCCCC(C)C(=O)NCCCCCCN(C(=O)C=CC(C)(C)C)C C1(Cl)(C(N(CC(C)(C)NC(C=C(CCC)C)=O)C)=O)CC1(F)F Cc1cnc(Cl)[nH]c1=NC(=O)C1COCCN1C(=O)Cc1cnn(C)c1 c1(CC(=O)NC(C)CN(C(=O)C(CO)SC2CCCC2)C)n[nH]c2c1CCCC2 CCCCCS(=O)(=O)CC(=O)N1CCCN(C(c2ccc(Cl)c(C)c2)=O)CCC1 CCC(C)(C)CCCC(=O)NCCC(C)N(C(=O)Cc1cc(C)cs1)C Cn1ncc(C(N2CCOCC2CC(=O)NCC2=CCCC2)=O)c1Cl c1(C(N(C(C)CNC(C2CC2C#N)=O)CC)=O)c(C)cnn1-c1ccccc1 c1(C(=O)NC2C(C)(C)C2)c(Cl)cnc(Cl)c1Cl.C12CC3(C1)CC(C3)C(=O)N2 C(=O)(CCCn1ccnn1)NC(C1CN(C(c2ccc(C)o2)=O)C1)C CC1(C)CN(c2cc(NC3CC4(C)BOC4C3)ncn2)CCC1O CCC(C(=O)N1CCN(C(c2c[nH]nc2[N+](=O)[O-])=O)CC1C1CC1)C(C)(F)F C(=O)(CC(C)(C)C(F)F)N(CCOCCNC(c1cnc(SC)s1)=O)C CC(C)C(C)(CNC(=O)OC(C)(C)C)NC(c1ncc(Br)cn1)C S(=O)(=O)(c1cccnc1NCC(C(C)C)CC)N.C1(N)CCCCC1C(N)=O c1(C(=O)NC(C(C)(C)NC(c2n(CCOC)ncc2)=O)C)nccnc1C(=O)OC C(=O)(C(C(C)(C)O)NC(c1cnn(C)c1N)=O)NC1(CC=C)CCOC1 N1(C(C(C)(C)OC)=O)CCN(C(c2cccnc2-n2ccnn2)=O)C(C(F)F)C1 C=Cc1ccc(C(=O)NC(CCCC)C(=O)NCCOC)cc1.C1(CCF)CC1 S(=O)(=O)(c1ccc(=NCC(O)c2ccc(Cl)c(Cl)c2)[nH]c1)NCCCCOCC c1(C(=O)NCCNC(C2CC=CCC2)=O)ccnc2cc(F)cnc12 c1(OC)c(CCC(=O)NCC(O)CCOC)cccc1F c1(C(C)C(=O)NC(C(=O)NCc2ccon2)C2CCC2)ccnn1C Cc1cn(C)nc1NC(=O)C(N1CC(C)CC1C(N1CCC(N(C)C)CC1)=O)=O Cc1cc(NC(C2CC2c2cnn(C)c2)=O)ccc1NC(=O)COCP(C)(C)=O C1(C(C)C)CC(NC(=O)NCC(C(F)(F)F)N(C)C)CCO1 C1(C(=O)NCC(C)NC(C2(CCF)CC2)=O)CCc2nnc(C(F)(F)F)n2C1 CC(CCCc1ccccc1)C(=O)NCC(C)NC(=O)CC1CC2(CCC2)CO1 C(=O)(CCCCCCN=[N+]=[N-])NCC1N(C(C(CCC)N(C)C)=O)CCCC1 N12CCN(CC1)CC2=O.C(C)(C(=O)NCC(CO)c1cncs1)SCC C1(C)(CNC(c2c(CC)oc(C)c2)=O)CN(C(=O)CC2C=CS(=O)(=O)C2)CCO1 c1(C(C(=O)NCCNC(C2CC=CC2)=O)(F)F)cccc(Cl)c1 N1(C(C23C(CN(C(c4cccc(C)c4F)=O)C2)C3)=O)CCCCC(F)(F)C1 N1(C(CC(C)c2cccnc2)=O)CCCC(CNC(C2(CO)CCCO2)=O)CC1 C(=O)(C1=CCC(C)CC1)N1CCN(C(CNC(=O)OC)=O)C(CO)C1 c1(C(=O)NCCC(=O)NC(C(C)O)(C)C)cccc(OCC2CCOCC2)c1 C1(CNC(C(CC)SC)=O)(NC(=O)C=Cc2cnn(C)c2)CCCCC1 C(=O)(N=c1cc[nH]c(C)c1F)C1C(NCc2c(F)ccc(OC)c2Cl)CCC1 c1(N(C(=O)CCCCCO)C2CNCCC2(F)F)c(Cl)ncc2ccccc12 c1(OC)cnccc1OC(C)C.c12cc(n[nH]1)C(=O)N(C)C1CCN(C1)C2=O Cc1cccc(N)c1C(=O)NCCNC(c1cc(CC2CC2)on1)=O C1(N(C)C(C2CC(C(F)(F)F)C2)=O)CCCN(C(c2cnn(C)c2C(F)F)=O)CC1 c1(CC)cc(NC(C2(CNC(=O)CN3C(=O)CNC3=O)CC23CCC3)=O)ccc1F C1(OC)CC(CNC(c2c[nH]nc2C(C)C)=O)N(C(=O)C(F)C2CCCC2)C1 c1(C2CCN(c3ccnc(NCc4cnc(CC)s4)n3)CC2)cc(F)cc(Cl)c1 C(=O)(CS(=O)(=O)c1ccccc1C)N1C(CNC(CNC(=O)NC)=O)CC1 C1(C)(C(N(CC(CNC(c2cc(COC)on2)=O)O)C)=O)CCNC(=O)C1 CCCC(CC)N=c1cc(C)[nH]c(=NCc2cc(C)cs2)[nH]1 C12CCC(CC1)CNC(=O)CC1CC1C(C)(C)NC(=O)CN2C.C(N)(=O)NC.C1CC1 CCCCC(C)NC(C1CCN1C(c1cncnc1)=O)=O c1(C(=O)NCC23OCC(CNC(C(C(C)C)(C)O)=O)(C2)C3)sccc1S(C)(=O)=O C(=O)(C(O)CC(N)=O)NC(C1CCN(C(C2(COC)CC2)=O)C1)C Cc1ccc(C(O)C(=O)NCC2CC(NC(c3c(Br)noc3C)=O)C2)cc1 c1(CNC(C(C2CCCN2C(=O)CC2CCC3CC23)(C)C)=O)nnnn1C1CC1 c1(C(=O)NCC(CCCC)NC(C(CC=CC)C)=O)cc(C(C)C)n(C)c1C c1(C(=O)NC2C(C)CN(C(c3coc(Cl)c3)=O)C2)ccc(F)c(O)c1F CCC(C)CC(C)C(=O)N1CC(CNC(=O)C(c2ccc(Cl)cn2)(F)F)(OC)C1 c1(COc2cc(C)nnc2)cnn2cccc2c1 C1(OC)CCN(c2nnc(-c3oc(C4CC4)nc3C)n2CC2=CCCC2)C1(C)C CC1CN(C(=O)C(F)(F)C(O)C2CC2)CCC1CNC(=O)COCCF C#CCCCC(C)C(=O)N(C(CC)CC(=O)NC(CC)C1CCC1)C c1(OC)ccc(CCN2CCCC2)cc1-c1ccc(CN2CCOC(C)C2)cc1 c1(C(=O)NCC2CCC2NC(C2CCC(=O)N2C2CC2)=O)cccc2occc12 CC1(C(=O)NCCNC(=O)CC2CCCC(=O)N2)COC(=O)N1 N1(C(c2cc(CC)nn2C)=O)CC2CC(NC(=O)CC3CCC(O)C3)C2C1 N1(C(C(C(C)C)SC)=O)CC(CO)C2(C1)CN(C(c1csc3ccccc13)=O)C2 C1(C(C)(C)NC(COCC(=O)OC)=O)CCN(C(=O)Cc2cc[nH]n2)C1 C1(O)(CNC(C(CCNC(C(C)(C)CO)=O)O)=O)CC2CCC1O2 C=Cn1nccc1C(=O)N(C)CCC1CCCCN1C(c1ccc(C(C)=O)[nH]1)=O S(=O)(=O)(c1cccc(=NCC(F)(F)C2CC2)[nH]1)NCC1(COC)CCCOC1 C1(C(N2CC=CC(NC(CC(C)n3ccnc3)=O)C2)=O)CCCC(=O)CC1 C12(NC(C=CC)=O)CC(CNC(CNc3cccc(OC)c3)=O)(C1)OC2(C)C C(=O)(CCN=C(NCC1CC1(Cl)Cl)NC(C)CN1CCc2sccc2C1)NC C(=O)(C1=NOC2(CCC2)C1)N(C)CC1(O)CN(C(=O)CC2C=CCC2)C1 Cc1cc2n(n1)CCN(c1cc(N3CCOC(C)C3)nc(S(C)(=O)=O)n1)C2 N(C1c2ccccc2CC1NC(c1ccc(C2CC2)o1)=O)C(C1C(C)CCO1)=O N1(C(C(C)OC)=O)CCC2(CCN(C(c3cc(N)ccc3C(F)(F)F)=O)C2)C1 C1(CCC(=O)NCC(C)(C2CCC2)NC(CCSC)=O)C(=O)ON=C1C CCCCCCCCCCC(C)NC(=O)Nc1cc(Cl)cc(Br)c1F C1(NC(c2c(C)ccs2)=O)CC12CCN(C(c1c(F)ccc(O)c1F)=O)CC2 n1(CCOC)c(C)cc(C(=O)NC(CNC(=O)CC23CCC(CC2)C3)C(C)C)c1C C(c1ccncc1)=C(C)C(N1CCOC(CN(C)C(C2CC2C(F)(F)F)=O)C1)=O C1(NC(C(C)CC2CC2)=O)(CO)CCN(C(c2coc(CO)c2)=O)CC1 c1(C(CC)C(=O)N2CC(NC(c3ccc(COC)o3)=O)C2)ccc(F)cc1 C1(C(N2CCC(C)(CNC(c3c(CC)nn(C)c3)=O)C2)=O)CC12CCN(C)C2 N1(C(c2cc(Cl)ccc2C(F)(F)F)=O)CCn2ncc(C3=CCCC3)c2C1 c1(C(N2CCCC(NC(c3cc(O)ccc3Br)=O)CC2)=O)ccc2sccc2c1 N1(C(CCC2CCN(C)C2)=O)CCN(C(=O)CN(c2ccccc2)C)C2CCC12 C(=O)(CCCCC(N)=O)N(CC(C)(C)C(N1CC2(CCN2C)C1)=O)C N1(C(=O)NC(c2cccc(Cl)c2)C(C)C)CC(O)C2(CCCC2)C1 c1(C(N2CCN(C(c3ccc(C)c(O)c3)=O)C3C2C3)=O)[nH]nc2ncccc12 c1(C(=O)NCC2N(C(CC)=O)CC2)cc(C2(C)COC2)no1 c1(CC)cc(=NC(=O)CC(=O)N2CCC(O)CC2C(=O)N(C)CCO)[nH]n1C CC1CN(C(C2C(C)(C)C2(C)C)=O)CC(C)C1NC(c1cc(Cl)c(Cl)s1)=O C1(CC)CCCN1C(=O)C(CC1CCCC1)NC(=O)C(=O)NCC1CC1 N1(C(CC(CC)CN(C)C)=O)CC(C)N(C(c2cncc(C)c2)=O)CC1C c1(C(N2CCC(CCNC(C(C)CC(N)=O)=O)C2)=O)cnn2c1CCCC2 C(C(=O)N1CCC(O)(CCNC(c2ccc3c(c2)CC3)=O)C1)(C(C)(C)C)SC C1(C(=O)OC)CC(N2CC(n3cc(C4C5COCC45)nn3)C2)C1 N1(C(C(C(=O)OC)C)=O)CC(C2(NC(C3CCCNC3=O)=O)CC2)C1 c1(C(N(CCN(C(C)C)C(C2CC3CCC(C2)S3)=O)C)=O)cc2n(n1)CC(F)C2 N1(C(CCCC=C)=O)CC2CN(Cc3ccc(O)c(C)c3)C2C1 c1(C(=O)Nc2c(C)nc(F)cc2)n[nH]c2c1CN(Cc1sccc1C)C2 N1(C(CC(C=C)C)=O)CC2CC(C1)CN(C(=O)CC1NC(=O)CN(C)C1=O)C2 CCCCCC(C)(CC)C(=O)NCCCCCCn1cc(CC2CCCC2)nn1 N1(C(CC(CC)CC)=O)CC2(CCC2)CC1CNC(c1c(C)ccc(C)c1C)=O C=CC(C)(O)CC(=O)N1CCCC(c2n[nH]c(CNC(=O)CCOCC(F)F)n2)C1 C1(CC(=O)NC(C(=O)OCC)C)CC2(C1)CN(C(=O)CN(C)C(N)=O)C2 CC(C)(C(=O)NC(CNC(c1n[nH]cc1C1CCC1)=O)C1CC1)c1cc[nH]n1 C(=O)(N=c1cnn(C2CN(C(=O)Nc3ccccc3)C2)[nH]1)c1cc(CC)on1 C=C=CCCC(=O)NCCC(=C)CNC(c1occc1Br)=O c1(C(CSCC(=O)NC(CN(C(C(N2CCOCC2)C)=O)C)C)=O)ccccc1 C1(NC(c2cnc(C(C)C)nc2)=O)CC(C)CN(C(c2cc(Cl)ccc2N)=O)C1 C=CCCCCC(=O)NC1(C(=O)NCCCC(=O)NC)CC1(C)C C=C(C)CC(C(=O)NC(C)CCC(=O)NCCc1ncoc1C)OC Cc1ccc2c(c1)CC(C(=O)OCC1CCCN1)S2(=O)=O CC1=C(C)CC(C(=O)NC2CCC(Cn3cc(COCCO)nn3)CC2)CC1 C12(C(NNC(=O)Nc3ccnc(Cl)c3)=O)CCCC1C2(F)F c1(CC)nc(C)c(C(=O)NC(C2CCN(C(c3cccc(CCO)c3)=O)C2)C)s1 c1(C(N2CC(NC(C(C)OCCOCC)=O)C2)=O)cc2c(nc1O)CCOC2 N1(C(c2nc(C(C)C)oc2)=O)CC(C2CC2)(C(N2CC3(C=CC3)C2)=O)C1 N1(C(C=C(C)C(F)F)=O)CCOC2CN(C(c3cc4[nH]ccc4s3)=O)CC12 c1(-c2cnc(Cc3cccc(OCC)c3O)nc2)cccc2c1OCC2 C(=O)(C(O)C(F)(F)F)N(CCC(N1C(C(N(C)C)=O)CCC1)=O)C1CC1 c1(C(N2CC(CC)C(NC(C3CC(C)(C)C3)=O)CC2)=O)cncc2sccc12 N12CCCC(C1C)NC(=O)C(C)N(C1CC1)C(=O)CCC2=O.C(C)(C)SC N1(C(C=CSC)=O)CCN(C(c2nnccc2C)=O)C(C)C1C C1(NC(c2c(C)cn[nH]c2=N)=O)CC2CC(C1)N(C(=O)CC1CC3CC3C1)C2 S(=O)(=O)(c1cc(C(=O)O)cs1)NCC(=O)Nc1c(C)noc1-c1ccccc1 c1(CC(=O)NC(COC)CC(=O)NCCn2cc(CO)nn2)nc(Br)n(C)c1C C1(CC(=O)NCC2(NC(CCc3cc(C)[nH]n3)=O)CCCC2)CCCCC1(C)C c1(C(N2CCCC2CC(c2ccco2)O)=O)cccc(C2CC2)n1 C1(CC(N2CC(NCc3ccc(Cl)nc3)CC(F)C2)=O)CN2CCC1CC2 C(N=c1[nH]c(N2CCCC3(C=CCO3)C2)nc2cccnc12)c1nnc(C)o1 Cc1c(CCC(N2CC(NC(=O)C(C)C3CC3)C(O)C2)=O)cnn1C c1(NC(CC(CCC)NC(=O)OC(C)(C)C)=O)ccc2ccn(C)c2c1 CC1(C)CC(NC(=O)CC(CNC(=O)Cc2cncs2)C2CCC2)C12CC2 Cc1cc(C(=O)NCC(C)(C)OCCNC(c2c(C)nc(C)n2O)=O)cc(F)c1 c1(C(=O)NCCC(C)(C)NC(C(C2CCCOC2)OC)=O)cccn2nccc12 C(=O)(CCC(C)(C)C)NCCCCNC(C1(Cc2c(C)cccc2)CC1)=O N1(C(CC(CC)(F)F)=O)CCN(C(C2(C)CC(C)=NO2)=O)CC(C)C1 N1(Cc2c(C)nn[nH]2)CCC(C2CCCN(C(=O)C(C)NC(c3cccs3)=O)C2)C1 C(=O)(C1=C(C2CC2)N(C)C(=O)N(C)C1c1cnc2n1CCC2)OC Cn1c(NC(N2CCCC(CCC(F)(F)F)C2)=O)nc2c(F)cc(Br)cc12 C1(C)(CC)CC(NC(=O)CNC=O)CN1C(c1oc(C)nc1C)=O c1(C(=O)NC2C(NC(CC=C=C)=O)CC2)ccc(C#N)c(Cl)c1 c1(C(=O)NCCCCCCNC(=O)Cc2cc(Cl)cs2)cn2ncccc2n1 C1(c2nnnn2CC2CCCO2)(NC(CC(C)(C)C)C)CCC=CCC1 c1(-c2cn(CC=C)nc2)nc2ccc(C(=O)Nc3ccc(C#N)o3)cc2s1 CCCC(CCC)CC(=O)NCC(CO)NC(=O)COc1ccc(OC)cc1 CCCCCCCC(=O)NC1CC(C(=O)N(CC(=O)OC)C)=CC1O c1(C(N2CC3(C(C(=O)N(CC4CCN(CC)CC4)CC)C3)C2)=O)cc(F)cc(Br)c1F C1(C(=O)NC(CC)COC)CC2CCCC2N1C(C1CC(=O)N(C)C1)=O C1(NC(c2ncccc2F)c2n(CC)nnn2)CCCN(C)CC1 c1(C(N2CCN(C(=O)CSC3CC3)C3C2C3)=O)cc(Cl)cc2ccncc12 C12(NC(c3c(C)cc(Cl)cc3)=O)CCCC1N(C(=O)C=Cc1cncn1C)CC2 c1(CN(C(C(C)N(c2ccccc2)C)=O)CCNC(=O)CCF)ccccc1 c1(C(N(C(C(C)C)C)CCC#N)=O)cn(CCNC(=O)C(F)C2CCCC2)cn1 c1(C(=O)N(c2nnc(-c3ccccc3)s2)C2CCCC2)ccc(C2CC2)cc1 N1(CC(=O)NC2CCN(C(=O)Cc3cn[nH]c3)CC2F)CCCCC(O)C1=O c1(C(N(CCOC)CCNC(=O)Cn2cccn2)=O)c(F)cc(C)cc1F C12(C(=O)NC3C=CC(CC=C)C3)COC(C1)C(NC(c1c(C#N)ncn1C)=O)C2 c1(OC)oc(C)nc1C(N1CC(O)(CNC(=O)CCc2ncc(C(C)C)o2)C1)=O C12(c3cn(CC(=O)NC(CC(C)C(=O)Nc4ccco4)=O)nn3)COC(C1)C(O)C2 C1(C(=O)Nc2cnc(OC3CCSC3)s2)CC2(C1)CN(C(=O)CC1C(=C)C1)C2 C(=O)(C(CO)C(F)(F)F)NC1C(NC(c2c(CC)c(C(=O)OC)c(C)[nH]2)=O)C1 C(=O)(C(O)CSC)N(CC(=O)NCC(C)OC)CC1CC1 c1(C(=O)NCC2C(NC(c3cccc(C(C)C)c3F)=O)C2)ccc2c(c1)NCC2 C(=O)(CC(C(=O)N1CCN(C(=O)C(C)SCC)C(C)C1)N(C)C)OC.C1C(=O)N1 c1(C(=O)NCCC(C)N(C)C(c2cc(Cl)cnn2)=O)ccnn(C)c1=O c1(C(=O)NC2C(CNC(Cc3cn(C)nc3)=O)CCC2)cc2n(n1)CCCC2=O C1(CNC(C(C)Cc2ccncc2)=O)CN(C(=O)Cc2ncc(C(C)C)o2)CCO1 C1(C(=O)OCC)CCCN(S(=O)(=O)N=S(C)(=O)C)C1 CCS(=O)CC(=O)N1CCC(C)(CNC(=O)Cc2ccnn2C2CCCC2)C1 c1(CC)cc(=NCCCC(C)(C)NC(c2cnc3c(c2)CCCO3)=O)[nH]cn1 N1(C(c2cc(C(CC)C)no2)=O)CCC2CCN(C(=O)CC3=CCCC3)C2C1 C1(NC(C2C(C)CCO2)=O)CCCC(CC(=O)NCCc2cccn2C)C1 c1(-c2c(OC)cc(C#N)cc2)nc(C2COc3ccccc32)nn1C(COC)CO Cc1c[nH]cc(C(=O)NC2CC3(C(N4CCOC(C)C4C)=O)COC2C3)c1=O n1(CC(C)C)[nH]c(CC(=O)NCCCC(C)NC(C2CCCOC2)=O)cc1=O C1(C(N2CCC(O)(CN(C)C(C3CC4(CSC4)C3)=O)C2)=O)CN2CCN1CC2 C#CCCCCCCC(=O)N(CCC(C(C)C)NC(=O)C(C)(C)CCSC)C S(=O)(=O)(CC(=O)NCC1(CNC(=O)C(=O)C(C)C)CCC1)NCC N1(C(C2C(CC)CCC2)=O)CC2CC(C1)CN(C(c1cnc(S)nc1)=O)C2 C(=O)(C1CCc2c[nH]nc21)NC1(CNC(c2cc(C)c(F)cc2Cl)=O)CCOC1 CCC(C)(CNC(c1n[nH]cc1Cl)=O)NC(C1CC(=O)C1C(C)(C)C)=O c1(N(C)C)cnc(C(N2CCCC(CNC(c3cocc3C(N)=O)=O)C2)=O)cn1 c1(OC)cc(Cl)c(Br)cc1NC(C(CCC(C)C)N(C)Cc1ccc(C)cc1)=O C1(C(=O)NCC2(C(C)NC(C(C)OCC=C)=O)CC2)CCOCC=C1 N1(C(c2nocc2NC(=O)CN2CCCC2)C)CC2(CCCC2)CC1C Cc1c(C(N2CCC2CNC(C2(C)CC(C)OC(C)C2)=O)=O)cccc1[N+](=O)[O-] N1(C(c2c(C)nn(C3CC3)c2)=O)CC2(C)CC1C2NC(c1c[nH]ccc1=O)=O N1(C(C2CCN(CC)C2)=O)CCC(NC(c2sccc2SC)=O)C12CC2 C(=O)(C(C)S(N)(=O)=O)N1CC(C(=O)NC(c2ccncc2)C)C(C)C1 c1(C(=O)OC)ncc[nH]c1=NC(=O)c1ncoc1CSc1ccc(Cl)nc1 c1(C(C)C)ccc(C(=O)NC(C)CC(C)NC(c2ccc(COC)cc2)=O)cc1 N#CC1(N(S(=O)(=O)c2nccs2)C(=O)CCc2ccc(F)cc2Br)CCN(CCl)C1 n1(CCC(N2CC(OC)(CNC(=O)CCC3CC3C)C2)=O)cnccc1=O C1(CC#C)CCCCN1C(=O)CC(CC)NC(=O)CSCC c1(C(=O)NCCCCNC(c2cnc(C3CC3)nc2O)=O)cccc2nsnc12 c1(C(N2CCC(CNC(C3(C(F)F)CC(=C)C3)=O)C2)=O)cc2c([nH]1)CCC2 c1(CNc2c(CC(N3CCC(F)CC3)=O)cccc2)cccc2nccnc12 C(=O)(CCC(C)(C)F)NCCC1CCN(C(CC2CC(OC)C2)=O)CC1 C(=O)(C(C(C)(C)C)N(C)C)N1C(C(N2C(C=C)CC2)=O)CSCC1 C12(C(=O)NC(C)(C)CNC(=O)C3=CCSC3)C3C4C1C1C2C3C41C(F)F CCC(CNC(C1CCN(C(C)=O)C1)=O)(CC)NC(c1cc(C(N)=O)[nH]n1)=O C1(CNC(CC2(CSC)CC2)=O)(CO)CCCN(C(=O)C(O)C(F)(F)F)C1 C1(NC(C(n2cc(C)nc2)(C)C)=O)CCCN(C(C2CNC(=O)N2C)=O)CC1 N1(CC=C(C)C)CCC(C(=O)OC(C)C(N)=O)c2ccccc21 N(C(=NCC1CCOC1)N1CCc2c(F)cc(F)cc2C1)C(c1cncnc1)C C(=O)(CC(F)(F)CS(C)(=O)=O)NC(C(C)NC(C1(C2CCC2)CC1)=O)(C)C N1(C(C2N(C(C)=O)CC(O)C2)=O)C2CCC1CC(NC(c1ncccc1Cl)=O)C2 C1(CNC(C(C)SCC)=O)CCC2(CN(C(C3CCC4(CCC4)CC3)=O)C2)O1 C1(C(=O)NCC2(CCNC(C(F)=CC)=O)CC2)OCCC1(C)C Cc1sc(C(=O)NCCOCCNC(=O)Cn2[nH]cnc2=N)c(C)c1C Cc1cc(C(=O)NCC2COCC2NC(=O)CCC2=NNC(=O)C2)c(C)c(C)c1 N1(C(C(C)N(C(C2N(CCC)CCC2)=O)C2CC2)=O)CCC(C2CCCC2)C1 C1(C#CC(=O)N2CCC(NC(c3nc(C)ccc3C)=O)C2)(CC)COC1 Cc1cccc(C(C)C)c1OCC(=O)NC(CNC(c1ccncc1C)=O)CO C(CC(C)C)(C(=O)N1CCCC(C(C)(C)C(=O)NC(C)C)C1)NC(CSC)=O C12(NC(CC(n3ccc(C)n3)C)=O)CC(C1)N(C(=O)CCCc1cnn[nH]1)C2 c1(C(N(C2CN(C(C(C)=C(CC)C)=O)CC2F)C)=O)cc(F)c(F)cc1OC c1(C(N(C)CC2CN(C(c3ccncc3Cl)=O)CCO2)=O)cccc2c1COC2 C1(C(C)C)CN(C(c2cc(C(F)(F)F)c[nH]2)=O)CCN1C(c1cncc(Cl)c1)=O c1(OC)cccc(CNC(c2c[nH]nc2CNC(=O)C(C)OCOC)=O)n1 c1(OCCOCCOC)cccc(OC)c1NC(=O)NCCC(=O)OC c1(C(N2CC(CNC(c3n[nH]c(C)c3Cl)=O)C(O)C2)=O)cc(Cl)c(F)cc1F c1(C(N2CCC(C(=O)NC(COC)C(C)C)C2)=O)c(OC)cccc1C N1(CC(=O)N(CC(=O)N(C)CC2CCN(CC)C2)CCC)C(=O)CCC1=O S(=O)(=O)(c1cccc(-c2ccnn2C)c1)NC(c1noc(C(F)F)n1)C C1(NC(C(c2ccccc2)SC)=O)CN(C(C2CCC(=O)N2)=O)CC12CC2 N1(C(C2(C)CC=C(C)CC2)=O)C2CCC1CN(C(c1nn(C(F)F)cc1Cl)=O)C2 c1(C(=O)NCCC2OCCCN(C(C(C=C)O)=O)C2)cc2ccccc2c(=O)o1 CCS(=O)c1ccccc1NC(=O)NCCC(C)(O)C1CCCCC1 C1(NC(c2ccc(CCC)s2)=O)CC2CCC1C(NC(=O)C#CC(C)(C)C)C2 C1(C(CC)C)CCN(C(=O)C(F)C2CC(NC(=O)C=C3CCC3)C2)CC1 N1(C(c2c(C)nsc2)=O)CC(NC(c2n[nH]cc2C2CC2)=O)C(N=[N+]=[N-])C1 c1(NCCC=CC=C)[nH]c(=NCc2oc3ccccc3c2C)nc2ncn(C)c12 C1(C(=O)NC2C(OCC)CC2)CN(C(=O)CCCCNC(N)=O)CC1SC C1(NC(=O)NC2(c3cccc(F)c3F)CCCC2)C(CO)C2CCCCC12 c1(C(=O)NCC(C)(CO)NC(CNC(c2n(C)ncc2)=O)=O)nccc(F)c1Cl N1(CCC)CCN(C(=O)C(C(C)O)NC(C2CC(C)(F)C2)=O)CC1 c1(C(N2C(C(=O)NCC(CC)C(C)C)CC(OC)C2)=O)cc(C)nc(C)n1 N1(C(C)C)CCN(C(=O)CCc2c(F)cccc2Cl)CC1C CC1=C(c2ccncc2)CN(c2nc(N(CCC#N)C)c3c[nH]nc3n2)CC1 c1(N(C)C)ncnc(NCC2(C)CC(C(=O)Nc3cc(C4CC4)on3)C2)c1[N+](=O)[O-] C1(NC(c2ccc3nc(N4CCCCC4)sc3c2)=O)CCc2nnnn2CC1 N12C3CCCC1CC(C3)C2=O.CCCCCCC(c1ccccc1)NC(=O)CO C1(C)(CCNC2(c3n(C(C)(C)C)nnn3)CC(c3ccccc3)C2)CCCCC1 Cc1cc(C(=O)N(CC(=O)NOCC2CCOC2)C(C)C)ns1 c1(C(N(CCCNC(c2c[nH]c(=O)cn2)=O)C2CC2)=O)ccc(Cl)cn1 c1(C(N2CCC(O)(C(C)NC(COC(C)=O)=O)C2)=O)c(C)ncc2ccccc12 c1(NCC2CCC(C(F)(F)F)O2)nc(N2CCN3CCCC3C2)nc2ccsc12 CC1CCC(CNC(c2ccc(F)cc2)=O)N(C(c2cccc(CF)c2F)=O)C1 c1(C(=O)NCC2(C)CCC(NC(c3nc(CC)sc3)=O)C2)cnn2cnnc2c1 C(c1ccncc1)=C(C)C(=O)NC1CCC1NC(=O)C(C(C)C)N1CCCCC1 N1(C(c2cc(C)ncn2)=O)CCOCC(NC(=O)CC(O)C(C)C)C1 C1(C(=O)NCCCOCCN(C(C2(CC)CCCC2O)=O)C)CC12CCOCC2 Cc1cc(Cl)c(Cl)cc1NC(N1CCOC(CNC(=O)CC=CC(C)(C)C)C1)=O N1(CCCNC(C2C(=C)CC2)=O)CCN(C(C2(F)CCOC2)=O)CC1 C1(C(=O)NCC2CN(C(=O)C(c3ccccc3)F)C2)CCCOCC1 c1(C(C(=O)NC2C(OC)CN(C(=O)C3=C(C)OCC3)C2)=O)c[nH]c2ccccc12 C=CCC(CC(C)C)C(=O)NC1(C(=O)NC2CC2O)CCC1 c1(CN(C(C2CCC(C)C2)=O)C2CC2)ccc(CNC(c2n[nH]cc2Cl)=O)cc1 C1(CN(C(CN(C)C)=O)C)COCCN1C(=O)CC1CCC(O)C1 c1(C(N2C(C)(CNC(Cc3ncc(C)s3)=O)CCC2)=O)ncnc2c1CCCC2 CN1CC2(CCN(C(c3ccc(F)c(-c4ccc(C(=O)O)nc4)n3)=O)CC2)C1 C1(NC(c2cc(C(N)=O)[nH]c2)=O)C2CCC1N(C(c1cnc(C3CC3)s1)=O)C2 N1(C(c2c(OC)ccs2)=O)CCC(C)C(NC(=O)COc2cc(F)cc(F)c2)C1 c1(SC)cnc(Cl)[nH]c1=NC(CNc1ccc(C(F)(F)F)c(F)c1)COC C1(C(=O)NC(CNC(C(c2nc(C)sc2)=O)=O)C(C)C)CC2CCC1O2 Cn1nc(C(=O)NCC2CN(C(c3ccc(C(N)=O)cc3)=O)CC2O)ccc1=O CC(CCC(=O)N1CCC(O)(SCC(=O)Nc2cnns2)C1)N(C)C c1(C(N2C(C)(CNC(C(CCSC)N(C)C)=O)CCC2)=O)ncnc(O)c1Cl C#CCCCC(C(=O)NCc1cccs1)N1CC(CO)C2(CCC2)C1 N1(C(C(=O)NCC)=O)CCn2c(CNC(C3CC(=O)C3)=O)nnc2C1 N1(C(c2nn(C)cc2I)C(=O)NCCOC)CCCCCC1c1cccc(C)c1 N1(C(c2nnn(C)n2)=O)CC2CC(NC(=O)CCc3ccc(=N)[nH]c3)C1C2 CON1CCC(C(=O)NC2CC2NC(C2COCCC2(F)F)=O)CC1 C(=O)(C1=CCCSC1)N1CC(CC(COC)O)C1.C1(=O)C(O)CCN1 C1(NC(c2cncc(OC)c2)=O)CC2CC(NC(c3cc(C)n(C)c3)=O)CC2C1 c1(C(=O)NCC2N(C(CC3C(=O)NC(=N)S3)=O)CC2)coc2cc(F)ccc12 CCCCCCC(C)NC(C1(F)CCCN(C(c2cnc3n2CCC3)=O)C1)=O C1(C(C)(C)C)CCCCN1C(=O)CCNC(=O)CCc1ccccn1 C1(NC(c2nc(CC)oc2)=O)CN(C(c2ccc(COC)[nH]2)=O)CCC1C C1(C2CCCCC2)(C(N2CC(C(N(C)CC3(NC(N)=O)CC3)=O)OCC2)=O)CC1 CC1CCC(C(=O)NCC(c2cccs2)C)N(C(c2csc(Cl)n2)=O)C1 C(=O)(C1CCc2nccn21)NCCC(C)N(C)C(C1CN2CCN1C(C)C2)=O C=C(Cl)C(C)(C)C(=O)N1CCCC(CNC(=O)Cc2cccc(Cl)c2F)C1 CN=c1[nH]c(=NCc2cc3cc(Br)ccc3o2)[nH]c(=NCc2nccn2C)[nH]1 CCC(CN=c1cc[nH]cc1S(=O)(=O)NC12CCC(CC1)C2)N1CCCC1 c1(CCC(=O)NCC(CO)NC(C2(C(C)C)CCC2)=O)c[nH]c(=N)[nH]1 Cc1nnc2n1CCCC2C(=O)NCCOCCNC(=O)CN1C(=O)CCC1=O c1(C(N2CCN(C(C(CC#C)C)=O)CC2C)=O)cc(F)cc(C)c1O CC1(C(=O)NCc2cccc(O)n2)C=CCN1C(=O)Cn1cc(C#N)cn1 Nc1ccc(C(=O)NC2CC23CC(NC(c2ncc(Cl)cc2Cl)=O)C3)c(Cl)c1 O1NC(=O)C(C)(C)C(C)NC(=O)C1.C(=O)(C(C)C1CCC1)NC C12(NC(c3c(C)n(C)nc3)=O)CCC(CNC(c3nccc(Cl)c3F)=O)(C1)OC2 N1(C(c2c(C)nn(C)c2N)=O)CCC2(CC1)CN(C(c1occc1Cl)=O)C2 N1(C(CSS(C)(=O)=O)=O)CC2CC(C1)N2C(C1CNC(=O)C1)=O c1(C(=O)NCC2C(NC(C(C)OCCOCC)=O)C2)ccc(N)c(Cl)c1 CC1N(C(N2C(OC(C)(C)C)COC(C)C2)=O)CCCC1(C)C N1(S(CC)(=O)=O)CC2CCC1CN2Cc1cnc(Cl)cn1 C1(CNC(CN(C)CC)=O)CCCC1NC(c1cc(Cn2cc(Cl)cn2)cs1)=O C1(NC(=O)Nc2ccc(CC)nc2)CCN(CCOc2ccccc2F)CC1C C=C1CCC(C(=O)N(C2CCCN(C(=O)C(F)OC(F)(F)F)C2)CCO)CC1 C12(C(=O)NCC(CCOC)NC(c3nnc(C)s3)=O)CCC(CC1)CC2 C1(NC(C2(COC)CC2)=O)CC2(CCCCN2C(C2SC3C=CC2CC3)=O)C1 N1(C(CC2(NC(C)=O)CC2)=O)CCC2CCCN(C(=O)Cc3nc(=N)[nH][nH]3)C2C1 C1(C(=O)NCCN(C(C2C(OCC)C2)=O)C2CC2)CCC(O)CC1 c1(C(C)NC(C2CCCO2)=O)cc(NC(=O)NC(c2cn(C)nn2)CO)on1 c1(CCC(=O)NC2C(NC(CCC#CC)=O)CCCC2)c(Cl)cccc1[N+](=O)[O-] N1(C(C(C#C)(C)C)=O)CCC2(CC1)CN(C(=O)C(C)CCCCCC)C2 N1(C(c2cn(CC)nn2)=O)CCC(C(=O)N2CC(C)C2(C)C)=C(F)C1 N1(C(=O)Nc2ccc(OC)cc2)CCC(C)C(NC(C2C=CS(=O)(=O)C2)=O)C1 C(C(=O)OC)(C(C)C)NC(C(c1ccccc1)ONC(C1(CC)CCCC1)=O)=O C1(NC(c2cnc(C)n2C)=O)CN(C(C2Cc3nccn3C2)=O)C2CCCC12 c1(CC(N2CCC(N(C(c3c(N)non3)=O)CC3CC3)C2)=O)cccc(F)c1F N1(C(=O)CC2OCCC2(C)CC(N2CCC(CC)O2)=O)CC23CCC2(COC3)C1 C=CCC(C)C(=O)N(CCNC(c1ccc(C(C)C)cc1)=O)CC1CC1 C(N=C(NCC1(C)CC1(C)C)NC(CC)CC)C1C(=C)C1 Cc1nc(C)c(CC(=O)NC(C)CN(C)C(c2cc(N)ccc2O)=O)c(O)n1 N1(C(C(CCC)NC(c2ncn(C)n2)=O)=O)CCC(C)=C(F)C1 c1(C(=O)NCC(C2CCOC2)NC(c2cc(C(=O)OC)on2)=O)ncncc1Cl N1(C(COC2CC3CCC2CC3)=O)CCC(OC2(C#C)COC2)C(C)(C)C1 c1(C(C2CCCC(N(C)C)C2)Nc2nnnn2C)cc2ccccc2oc1=O c1(C(=O)NC2C(CNC(c3n(C(C)(C)OC)ccc3)=O)C2)cnn2cccnc12 c1(CC(C(=O)N(C(C)C)Cc2ccncc2)C)ccc(F)cc1 Cc1ccc(C(N2CC(O)(CN(C)C(c3c(C)coc3C3CC3)=O)C2)=O)c(C)c1 CC1CCCCN(C(=O)C(C(C)(C)O)NC(=O)COC(C)(C)C)C1 C1(CNC(CCC#CC)=O)CN(C(C2CC(=C3CCC3)C2)=O)CCC1(C)C C#CCCC(O)C(=O)NC(C1(O)CCN(C(c2ccn(CC)c2C)=O)CC1)C C(=O)(C(C)(C)CC(F)F)NC(CCOC)C(=O)OCc1ccc(CN(C)C)cc1 CCCC(CCCNC(C1CC12CCC2)=O)NC(c1ccc(OC)cc1Cl)=O N1(C(CN(CCC)C)=O)CCC(CO)(NC(=O)C(C(C)C)c2cccnc2)C1 C1(CC)CN(C(c2ccnn2CCC(F)(F)F)=O)CC(CC)O1 c1(C(=O)NCc2c(C(N3CCC(CCC)C3)=O)scc2)ccccc1Cl C1(n2ncc(C)c2)CCN(C(=NCC2CC2)NCc2cccc(Br)c2O)C1 N1(C(CC(C)C2CC2)=O)CC2CCCCC2(NC(=O)Cn2ncnn2)C1 c1(-c2cn(CCC(=O)NC(C)CCN3CCCC3)nn2)ccc(C(F)(F)F)cn1 CC(C)(C)CC(C)(C)C(=O)NCC1CCC(NC(=O)COCc2nc[nH]n2)CC1 Cc1cc(C)n(CC(N2CCNCCC2c2ccccc2)=O)c(=O)n1 CCCC(O)C(CO)NC(=O)CN(C(c1cc(C)nnc1C)=O)CC1CC1 N1(CC(C)(C)NC(=O)C=Cc2cccnc2)CCN(C(C2CCNC2=O)=O)CC1 C1(NC(C2(CC=C)CCOCC2)=O)CCN(C(C2(C#N)CC2)=O)CC1F S(=O)(=O)(c1ccccc1C#N)NCc1c(OC)ccc(F)c1Br.C12CC(C1)CO2 c1(C(=O)NCCc2cccnc2)cc(-c2c(CO)cccc2F)cc2[nH]ccc12 C1(NC(c2c(C)cc(F)nc2)=O)CCN(C(=O)CC2CCC3CC23)CC(O)C1 CC1(C)CCCCCC1NC(C1CCC(NC(c2cc[n+]([O-])cc2)=O)C1)=O Cc1cnccc1C(N1CC(CF)(NC(C2COC(=O)C2)=O)C1)=O C=CCC(CC)C(=O)N(C)CCOCCCN(C(=O)C(C)C)C.C1(=O)CN1C N1(C(COCCNC(COC2(C)CCC2)=O)=O)CC2CC(CO)CC(C2)C1 C1(c2cnc(NC(CC3CCCC(C)(C)C3)=O)s2)Cc2ccccc2C1 C(C(=O)NCc1nnn(C)c1C(=O)NC(CO)CCO)(C(C)C)NC(C)=O c1(C2C(C(=O)NC3C(NC(CCCN(C)C)=O)CC3)C2)ccccc1F c1(CC(=O)NC(CNC(C(C)OC)=O)C2CCC2)ccsc1Cl O(NC(=O)CN(C(=O)CC)CCN(C1CCCO1)C)CCC CN(CCCC(=O)N1CC(CC(N2CCOC(C)(C)C2)=O)C2(CC2)C1)N=O CC1CN(C(=O)CS(C)(=O)=O)CCC1N(C(=O)C(F)(F)C1(O)CCCC1)C c1(C(C(C)NC(c2c[nH]c(C(C)(C)C)c2)=O)C)ccc(C(F)(F)F)cc1 c1(C(NOC(=O)C=CCF)=O)ccc(NC(C(F)(F)F)C2CC2)nc1 C1(NC(c2c(C)ccc(=N)[nH]2)=O)CCCCC12CCN(C(C1CC(F)(CF)C1)=O)C2 C(=O)(CCCC(F)F)NCC(C)(C1CC1)NC(CC1C=NN(C)C1=O)=O CCCCCC(C)(C)C(=O)N(CCCN(C)C(C1CC(=O)N(OC)C1)=O)C CC1CN(C(=O)CCOc2ccccc2C#N)C(C)CN1C(=O)C(C)(F)F CCC(C(=O)N1CCC(C)(C)C(C(=O)N(C)Cc2cnc[nH]2)C1)C(F)(F)F N1(C(=O)C2=CCOC2)CCN(C(c2ccc(-c3cccs3)o2)=O)C(C(F)(F)F)C1 C1(C(C(=O)NCC(CNC(C2(CC#C)CCCO2)=O)(C)C)O)CCCCCC1 N1(C(C2(O)C(C)(C)C2)=O)CCC2(CCOCC2)C(NC(=O)Cc2cn[nH]c2)C1 N1(C(CCCOCC=C)=O)CCC(C(C)NC(C2CC(N(C)C)C2)=O)CC1 n1(CC)c(C)cc(C(=O)COC(=O)OC(C)Cn2cccnc2=O)c1C c1(CC(CN)N(C(C2CCCN2Cc2cccnc2)=O)C2CC2)ccc(F)cc1 Cc1cnc(C(=O)NC2CCCN(C(=O)CCc3nnc(C4CC4)o3)C2)c(F)c1 C1(NC(c2ccc(C)nn2)=O)CN(c2ccnc(N3CCOCC3)n2)CC1(C)C C1(NC(C=CCCC)=O)CC2CC(NC(c3n[nH]c(C4CC4)c3C)=O)C1C2 C1(CCC)(C(=O)N(C(C)C(=O)N(CCC(O)CO)C)C2CC2)CC(=O)C1 C1(C)(CSC)CCN1C(=O)C(F)CC1CN(C(=O)COc2cc(C)on2)C1 C1(N(C(=O)Cc2nc(Br)sc2C)C)CCCN(C(=O)C(=O)NC2CC3CCC2O3)C1 C1(CNC(Cc2ccc(C)s2)=O)CCN(C(c2nnn(C)c2N)=O)C1(C)C c1(NC(C2CC2NCc2ccc(F)s2)=O)ccc2sc(Cl)nc2c1 C(CC1=CCN(C(c2cc(Br)sn2)=O)CC1)NC(=O)CC1CCC2CC12 C1(CC)CN(C(=O)C(C2(C)CC2)NC(=O)COCCF)CC1O N1(C(c2cnc(C)[nH]2)=O)CC(=O)NC2CN(C(=O)C(C)(C)N(C)C)CCC12 N1(C(c2cncc(O)c2Cl)=O)CCCC(C2CN(C(=O)C(O)C(F)F)C2)C1 CCCC(C)(C)C(=O)NC1CC(F)CN(C(=O)CC2CCN(C)C2=O)C1 CCC1=NOC(C(=O)NC2CCOCC2C(=O)NCC2(C)CC(O)C2)C1 CCCC(C#N)C(=O)N1CCC(C)C1CNC(c1ccc(Cn2ccnn2)o1)=O C(=O)(CS(=O)(=O)CCO)N1CCN(C(c2cc(C)cc(C(F)F)c2)=O)CC1 C(=O)(C1=CC2(CCOCC2)C1)N1C(CCNC(=O)C(CSC)OC)CC(OC)C1 C1(NC(c2ccc(C)c(C)c2)=O)CN(c2ncc(Br)cn2)CC12CCOCC2 N1(C(C(CC)N(C)C)=O)CCC(C2CC2)(NC(c2csc3ccccc23)=O)C1 N1(C(Cc2nc(C)oc2)=O)CC2CC(NC(C3CCOC3(C)C)=O)CC1C2 n1(CC(=O)OC(C)(C)C)cc(C(C2(NCC(F)(F)Cl)CCC2)=O)nn1 Cc1cccc(F)c1C(=O)NC1C=CC(C(=O)NCc2nocc2C(C)C)C1 C#Cc1ccc(=NCCn2cc(Br)ccc2=O)[nH]c1OC c1(CCC(=O)OC(C(C)C2CCC2)=O)c(Cl)cccc1F Cc1cccc(CC(=O)NCc2cc(C(=O)NC3(CO)CCOC3)co2)c1 C1(C2N(C(Cn3ccc(C)n3)=O)CCC2)CCN(C(=O)CCc2nncs2)CC1 c1(C(=O)OC(C)C)cccc(CN2CC(NC(c3ccoc3)=O)C(O)C2)c1 C1(CNC(C2N(N=O)CCC2)=O)CC2CCC1N2c1cc(C2CC2)nc(Cl)n1 C(C(C)(COC)C(=O)N1CCCC(C)(C)C1C(=O)NC1CC(=O)NC(=O)C1)OC N1(C(Cc2ncc(C)s2)=O)CCC(O)(CCNC(=O)CCCCCF)CC1 CC1(C(N2CC(CCNC(C3CC3F)=O)C2)=O)Cc2ccccc2N1 C1(C(=O)NC(C2CCN(C(C3(C)CCCC3)=O)C2)(C)C)CCC1(C)C C1(NC(CCC(=O)NC)=O)CCCC12CN(C(C1CC3(C1)CC3F)=O)C2 N1(C(C2(CC(C)C)CC2)=O)CC(CCO)(NC(C2CC2(F)Cl)=O)C1 C12(NC(c3c(C)cc(C)o3)=O)CCCC1N(C(=O)Cc1ccc(Cl)cc1C)CC2 C12(C(=O)NC3C(c4n(C)ccn4)CN(C(=O)CSC(F)F)C3)CCC(CC1)CC2 CC1(C)CCCC(CC(N2CCC(O)(CCNC(=O)Cn3cnnc3O)C2)=O)C1 c1(CO)cc2c(N(C)CCN(CCOC)C)ncnc2s1.c12coc(c1)C2=O n1(CCC)cc(C(=O)NCC2(CN(C(=O)CC(C)OC)C)CC2)c(C)n1 c1(CN2C(CNC(=O)C=Cc3ccccc3Cl)CC(=C)C2)c(Cl)cccc1B(O)O Nc1cc(F)c(C2CC2N2CC(=O)N(CC(=O)Nc3ccc(F)cc3)C2=O)c(F)c1 N1(C(CCC=CCC=C)=O)CC(C(=O)N(CCCO)CCCO)CC1(C)C C=Cc1ccc(C(=O)NC2CCN(C(=O)C(C)C3CCC3)C(C)C2)cc1 C1(NC(CCCC)=O)CN(C(=O)C(C)NC(=O)OC(C)(C)C)C2CCCC12 CC(CC(=O)N1CC2C(NC(C3CCN(CC(F)(F)F)C3)=O)C2C1)C(F)(F)F CC1(O)CCN(CC(N2CCC(O)C2)=O)C1.C12CCCN(C1)C2 C(CC(N=c1cc[nH]c(-c2cccnc2)n1)C(C)C)N(c1cc(CC)no1)CC C(CCC(C)C)(C(=O)NCc1ccncc1F)NC(Cc1cc(C)n(C)n1)=O C1(NC(CC2(OC)CN(C(c3ccc([N+](=O)[O-])s3)=O)C2)=O)CCCCC1(C)C c1(C(N2C(C)CN(C(=O)CC3CCCNC(=O)C3)CC2)=O)nc2cccnc2s1 O=C(N=c1nn[nH]n1-c1ccccc1Cl)NC(c1nnc(CO)s1)C1CCC1 N1(C(C(CC)Oc2c(Cl)cccc2Cl)=O)CC2(CCOCC2)C1OC c1(OC(C)C)ccc(C2CCN(Cc3cccc(C#N)n3)C2)cc1OCC1CC1 C1(OCC)CCN(C)CC1.c1(C(N2CC(CCCCC(=O)O)C2)=O)conc1C(=O)N Cc1nn(CC(N2CCN(c3ncc(O)cn3)CC2)=O)c(=O)o1 c1(NC)ccc(F)cc1C(=O)NCCCN(CCO)C(c1coc(Cl)c1)=O C1(NC(c2c(C)cccn2)=O)C(CNC(c2cnoc2C)=O)CCC12CCC2 C1(NC(N(CCNC(C(C)OCC#C)=O)CC2CC2)=O)CCCCC(=O)C1 C1(NC(=O)CCCC(=O)N2CCC2)CN(C(=O)C=CC2CCC2)CC12CCOCC2 C1(C(=O)NCC2(F)CC(CNC(c3nnsc3C)=O)C2)(OC)CCCOC1 c1(CC(C)N(CC(O)CN(C)C(C2CC2C(F)F)=O)C)ccccc1 c1(C(C(F)(F)F)OC)ccccc1NC(c1nc(C)cn1C)c1ccccc1Cl c1(C(=O)NC2C(C)(CNC(c3csc(CO)n3)=O)CCC2)ccnc2[nH]cnc12 c1(C(N(CCN(C(c2ccc(CO)[nH]2)=O)CC)CC)=O)ccc(Cl)c(C)c1 N1(C(C(C2(O)CN(C(CC(C)n3ccnc3)=O)C2)F)=O)CCC(C2=NOCC2)C1 C=CCCN=C(NCc1cc(C)ccc1Br)NCC1C(C)C1C N1(C(c2cc(C)c(C)o2)=O)CC(C2CCN(C(C3(F)CCOC3C)=O)CC2)C1 C1(N(CC#C)C(C2CCOC2C2CC2)=O)CCN(C(c2ncoc2C)=O)CC1 c1(C(=O)NC(C)C(=O)N(CCCNC(C2C(Cl)(Cl)C23CC3)=O)C)ccccc1Cl N1(C(c2c(C)nsc2C)=O)CC(CNC(=O)CC2CCCN(C)C2)C(F)(CO)C1 CCCC(C(=O)NCC1CCN1C(C1CCOC(C)(CC)C1)=O)S(N)(=O)=O CC1CN(C(=O)CN2CCOCC2=O)CCC1CNC(c1csnc1Cl)=O Cn1ccc(-c2noc(C3(C4CCNCC4)CCC3)n2)n1 Nc1cnc(C(=O)NCC2CC(O)CN2C(=O)CCc2ccoc2)c(Cl)c1 c1(C(=O)NC(C)CCNC(=O)C(c2ccccc2F)O)cccc(P(C)(C)=O)c1 CC(=Cn1ccnn1)C(=O)NC1COCCC1NC(=O)CC1CCC(F)(F)CC1 C1(C(=O)NCCCOCCN(C(C(C)CC2CC2)=O)C)CCc2nn(C)cc2C1 N1(C(C2C(=C)C2)=O)CCC2CC12C(=O)NCCOCCO CC(C)C(CCN(C(=O)CCc1cc[nH]n1)C)NC(C1(O)CCCC1)=O C1(NC(c2n(CC#C)ccc2)=O)CC(NC(c2cnn(C)c2)=O)C12CCC2 C(=O)(C(O)C(F)(F)F)NC1CC(C)(CNC(c2ccc(F)c(Cl)c2)=O)C1 N1(C(c2c(CC)cccc2)=O)CC(NC(=O)CC2C(=O)N(C)N=C2C)CC(C)C1 C1(C(=O)NC(CNC(C2C(C(=O)OC)C=C2)=O)(C)C2CC2)CCCCN1C Cc1ccc(C(C)(C)C(=O)NCC2CN(C(=O)C3=CCC3)C3CC23)cc1 c1(CC(N2CCC(NC(C=CC)=O)C2CC)=O)c[nH]c2cnccc12 Cc1ccc(S(=O)(=O)NCC(N2CC3CC3C3CC23)=O)c(C)c1 c1(CCNC(C2CC2F)=O)ccc(CNC(C2CC(F)C2)=O)cc1 C(CCF)(C(=O)NCCCc1nccs1)NC(C1C(C)OCC1)=O c1(C(N(CC(CC)NC(c2cc(C(CC)CC)no2)=O)C)=O)nnc(O)cc1O C(=O)(C(=O)C(=O)SCCN)NCC(C)C.CCCN1CCC1CC c1(C(C)=O)ccc(CN(C)CC2(O)CN(C(c3cnns3)=O)C2)cc1 C1(C(N2CCC(COC)(CNC(=O)C(F)F)CC2)=O)CC(C(C)(C)C)=NO1 C1(C(=O)NCCc2nnc(C)s2)CC(C)CN(C(C2C=CC=CC=C2)=O)C1 C=CCN(OC)C(=O)C12C(NC(=O)CCc3csnn3)C3CC1C2C3 C12CC13CCN(CC3)C(=O)C(=O)NC2.C=C(C)CC(C)C(=O)NC(C)C c1(OC)ccnc(OC)c1C(=O)NC1CCN(C(C2COC(=O)O2)=O)C1 C1(C(=O)NCC2CCC(NC(CS(CC)(=O)=O)=O)CC2)COC2(CCC2)CO1 N1(C(c2c(C)cnn2C)=O)Cc2nccn2CC(NC(=O)CCc2ccoc2)C1 c1(CC=C)cccc(C(=O)NC2CN(C(=O)C(C)(O)CC)CC2CCOC)c1 S(=O)(=O)(c1cscc1F)N(C(=O)Cc1ccccc1C(F)(F)F)C C1(CN)CC2(CCO1)CC2.N1(COC)CC2CC1CS2 C1(CC(=O)NC(CCCC=C)C2CC2)CC2(CC2)CN1C(=O)C(F)=CCC c1(OCCC(=O)NCCNC(C(CC)COC)=O)ccc(Cl)cc1Cl C=CCCC(C(=O)OC)NC(=O)CC1CCCCN1C(=O)COCCCN(C)C C1(NC(C(C)NS(C)(=O)=O)=O)CN(C(c2cnc(N)cn2)=O)CC1S(C)(=O)=O C(=O)(CCC(F)F)NCC(CNC(=O)Cn1ccc(C(F)(F)F)n1)O [N-]=[N+]=NC1CC(C(=O)NC2CC3CCC2O3)N(C(c2ccc(C#N)cc2)=O)C1 Cc1ccc(-c2cc(C(=O)NCC3CC3CNC(=O)Cc3ccsn3)n[nH]2)s1 C1(OC)C(NC(=O)CC(C)(C)C2CCCCC2N)CC12CCC2 c1(CC(N2CCC(n3cc(CN(C)C)nn3)C(O)C2)=O)ccc2nc(O)[nH]c2c1 C(=O)(C1=Cc2ccccc2C1O)OC(C1(C)CC1)C C1(C(=O)NC2C(c3n(CC)cnn3)C2)CCN(C(C2CC(=O)N(C)C2)=O)C1(C)C c1(OCC)c(C(c2nnnn2C(C)(C)C)NC2CC2C(F)(F)F)cccc1Cl C1(NC(CN(c2ncccn2)C)=O)CC2CC(C1)N(C(=O)Cc1ccc(Cl)s1)C2 C1(C(=O)NCc2ccc(C)nn2)CCN(C(=O)CCCn2ccnc2)CC1C C#CCC(O)C(=O)N(C1CC(F)CN1C(=O)COC1CC(F)(F)C1)C N1(C(C(CC)=CC)=O)CC2CC2(NC(=O)CCc2cnc[nH]2)C1 C1(CC)CN(C(=O)C(c2ccccc2F)O)CCC1NC(C1CCOC1)=O C1(OC)CC(NC(=O)NCC2CCCC2OC)CC1OC(C)(C)C Cc1ccc(C(=O)NC2CCCC2NC(C2(C(F)(F)F)CC(C(F)F)C2)=O)c(Cl)c1 N1(C(C(CCOC)C)=O)CCN(C(c2cn(CC(F)(F)F)nn2)=O)C(C)C1 Cc1cc(C(c2nnnn2C)NC2CN(c3ccccc3)C2=O)sc1Br C1(C(=O)NC(C)CNC(=O)C=C2CCC(C)C2)(OCC)CCC(C)(C)CC1 c1(OC)ccc(Cl)c(C(=O)NCC2(F)CCCN(C(=O)CC=C(C)C)C2)c1 N1(C(c2ccnc(C(C)C)n2)=O)CCCC(NC(C2CSC2)=O)C(F)C1 c1(N(C)C)ncnc(N(C2CCN(C(=O)C3=CCC3)C2)C)c1[N+](=O)[O-] c1(C(N2CC(F)CC(NC(C(C=C=C)C)=O)C2)=O)ccc2cc(O)ccc2n1 CCCCCC(O)C(=O)N1CC2C(CNC(C3CCC(=O)NC3)=O)C2C1 C1(COC)(CNC(=O)Cc2cc(C)on2)CCN(C(c2ccc(SC)s2)=O)C1 N1(C(C(C)=CC)=O)CCC(C(C)C(=O)NCC2CN3CCC2C3)CC1 C=C=CC(C)C(=O)N(CCC(c1cccs1)NC(c1c(C(C)C)cnn1C)=O)C c1(C(=O)NC2CN(C(C(C(C)C)NC(C)=O)=O)CC(F)C2)c[nH]c2ccc(Br)cc12 C1(OC)CCN(C(C2CC(F)CN2C(=O)NCc2cc(C(=O)OC)nn2C)=O)CC1 C1(CCC)CC(C(=O)N(C)CCNC(c2nc(C)n(C)n2)=O)CCO1 N1(C(Cc2ccc(C#C)cc2)=O)CCC2(CC1)CN(C)C(=O)O2.CC(C)C C1(CNC(CCn2ncc(C)c2)=O)CCC(CNC(C2CC3C=CC2C3)=O)CC1 C1(NC(C(C2CCCC2)OCC)=O)CC2(C1)CC(NC(C1CNC(=O)N1C)=O)C2 C(=O)(C(CC(C)C)C(C)C)N1CC(CC)C(CNC(c2cnnc(C)c2)=O)CC1 c1(C(N2CC(=C(CNC(C(COCC)N=[N+]=[N-])=O)F)C2)=O)nc(C)c(C)[nH]c1=O N1(C(C(C)OCC2CC2)=O)CCCC1CC(C)(C)NC(=O)C(C)(C)C c1(C(N2CC(NC(c3cc(CCOC)on3)=O)(CO)C2)=O)cc(O)ccc1C S(=O)(=O)(c1cccc(Cl)c1)N1CC(CC(N2CCC(F)C2)=O)OCC1 C12(CNC(c3ncc(C)nc3)=O)CCCC1CN(C(=O)C(C)C1CC1)C2 C#Cc1ccc(C(=O)NC2CC(NC(=O)C(=O)NCC(F)F)C2)c(OC)c1 N1(C(CNC(c2cccs2)=O)=O)CC(NC(C2CC(OOC(F)(F)F)C2)=O)C(O)C1 c1(NCC2CN(C(C(CC)(C)OC)=O)CC2C(F)(F)F)ccc(F)cc1[N+](=O)[O-] C1(C(=O)NC(C(=O)NC)C)CCC2(CC2)N1C(C1CCOC1C(C)C)=O c1(CC)conc1CC(N1CCC(Cc2cn(CCCN3CCCC3)nn2)C1)=O N1(C(c2cccc(NC(C)=O)c2)=O)CC(C)N(C(c2cccc[n+]2[O-])=O)CC1C C12CN(CCC1(C)C)C(=O)C1(CC1)C(=O)OC2.Cc1cc(C(=O)NCC)on1 C(C(C)N=c1[nH]c(Cl)nc(C)c1F)NC(Cc1ccc(C)cc1Cl)=O c1(C(N(CCCCCn2cc(CC3CCCCO3)nn2)CC)=O)n[nH]nc1OC N1(C(c2cc(CC)c(C)s2)=O)CCCC1C1CCCCN1C(=O)CSC(C)(C)C C(CC#CC)(C(=O)N(C)Cc1cccnc1)NC(C(C=C)O)=O c1(CCC)ccc(C(=O)NCC2COCC2NC(=O)C(C)(O)CC)cc1[N+](=O)[O-] C1(CC)CC(C(=O)NCCS(=O)(=O)NC)CCN1C(=O)Cc1ccc(Cl)cc1Cl CCC(O)CC(=O)NC1CCN(C(c2nc(Cl)sc2C)=O)C1 C1(CC(N2C(CC(C)C)CC2)=O)CN(C(c2ccc([N+](=O)[O-])o2)=O)CC1(C)C N1(c2snc(C)n2)CC2CCC(C1)C2CNC(=O)Cc1cnn(C)c1C N1(C(CC(C=C)CCC)=O)CCCCC2(C1)CN(C(=O)CC(F)(F)F)C2 C1(C(=O)NCC(COC)NC(=O)C(O)C2CCC2)CCCCN1C c1(COC)cc(C(N2CC(O)(CNC(=O)CCCc3csc(C)n3)C2)=O)n[nH]1 Cc1cccc(OCC(=O)NC2C=CCN(C(c3cncn(C)c3=O)=O)C2)c1C c1(C(N2CC3CN(C(C4(n5cccn5)CC4)=O)CC3N2)=O)cc(Cl)c(F)cc1Cl N1(C(C2(C)CC(C)(C)C2)=O)CCC2(CCCN(C(c3ccc(F)c(O)c3)=O)C2)C1 c1(C(=O)NCCCCN(C(=O)C(C)(C)CN(C)C)C)c(F)ccc(F)c1O CCC(C)CCCCC(=O)NCC(C)N(C(c1cc(SC)n(C)n1)=O)CC c1(C(N(CC(C)CNC(=O)CC2COC(=O)C2)C)=O)ccnc2[nH]cnc12 c1(C(C)C(=O)NCCOC(C)(C)CNC(C2CC23CCC3)=O)ccccc1Br C(=O)(C(CO)NC(c1cc(C)cs1)=O)NC1CC(COC)C1 n1(C(c2nc[nH]n2)C)ccnc1-c1cc(C2CCOCC2)on1 C1(C(=O)NC2CCCC(NC(C(CC=C)(F)F)=O)C2)COc2ccc(F)cc2C1 c1(OC)cccc(C(=O)NC(c2noc(CC(C)(C)C)n2)CC2CCCCC2)c1 Cc1ccc(OCC(=O)NCC(O)CNC(C2(c3cnnn3C)CCC2)=O)cc1 CC1(C(=O)NCC(O)CNC(=O)C2=CCC2)COCCO1 c1(CC)cc(C(N2CCC(C)(C)C2CNC(C2CCCN2C=O)=O)=O)cc(O)n1 C(=O)(C1=CCCSC1)N1CCC(CCCCCNC(c2c(C)ocn2)=O)CC1 N1(C(CN(C)C(N)=O)=O)CC2CCCC(C1)N2C(C1CC12CCOCC2)=O c1(C(C2(C)CCCO2)NC(=O)C(=O)N(C2CC2)Cc2ccco2)ccccc1Cl C12(NC(CNC(=O)CC(F)(F)F)=O)CCCC1N(C(=O)Cc1cnco1)CC2 C1(NC(c2c(C(C)C)occ2)=O)CCC2(CCCN(C(=O)Cc3cncs3)C2)C1 c1(C(=O)NC(CN(C(=O)CCC2CCOC2)C)(C)C)nc2n(c1Br)CCC2 c1(OCC(C)C)ccc(C(N2CC(O)(C(C)NC(C3(C)CSC3)=O)C2)=O)cc1 C12(CCc3ccccc3C1)C(=O)N2.CC(C)(CCl)C(=O)Nc1c[nH]nc1C(N)=O C1(CC(=O)NC(CN(C(=O)CN2CCCCC2)CC)C)CCS(=O)(=O)C1 C(C=CC(=O)N(CCCNC(=O)CNS(N)(=O)=O)CCO)(CC)=CC C1(N(C(CC(C)O)=O)C2CC2)CCNCCC1C N1(C(CCC(=O)OCC)=O)CCC2(CC1)CC(C)N(C(c1cnsc1)=O)C2 C(CC(F)(F)Cn1cncn1)OC(CCCC=C)=O C1(CNC(C(C)NC(CC)=O)=O)CC2CN(C(=O)C=C(C)C(F)F)CC12 CC1CCC1N=c1ccnc(NC(CC2CC2)Cc2cccs2)[nH]1 Cc1n[nH]c2cnc(C(=O)NCC3CN(C(C4CC5CCCCC45)=O)C3)cc12 n1(C(C)C)ccnc1C(N1CC(O)(C(F)C(=O)NCC2CCOC2C)C1)=O S(=O)(=O)(c1ccc(Cl)cc1Cl)N(c1ccc(C=CC2CCC(=O)O2)cc1)CCO C1(c2cn(CC(=O)NCC3CC(CC4(O)CCC4)C3)nn2)(OC)CCOCC1 C(C)(C(O)C(=O)NC1CC(NC(c2cccc(N)n2)=O)C1)SC N1(C(CN(C)C(N)=O)=O)CCC(CNC(=O)C=Cc2cn(C)nn2)C1(C)C c1(NC)ccccc1C(=O)NCC(C)C(=O)Nc1ccccc1NC n1(CC=C)c(N2CCC(C)(OC(C)C)C2)nnc1C1CCC1 C1(C(=O)NC(C(=O)N(C2CCC2O)C)Cn2cccn2)CCCC(CF)C1 c1(C(CNC(C(C(C)NC(N)=O)(C)C)=O)(F)F)ccc2c(c1)OCCO2 C1(NC(C(CCC)OCC)=O)CCN(C(=O)Cc2c(C)n[nH]c2C)C12CCC2 C1(NC(C=CC)=O)CN(C(c2ccn3ccnc3n2)=O)CCC1(C)C C(=O)(C1=NN(C2CC2)C(=O)CC1)NCCN(C(c1nn(C)c(O)c1)=O)CC1CC1 Cc1onc(CC(=O)NC2CC(C)N(C(C3CCCOC3)=O)C2)c1C#N c1(C(=O)NC2(CC=C)CCN(C(c3cc(C)n(C)c3)=O)C2)cc(F)c(C)cc1F c1(NC(C)COc2cccnc2)nccc(=NCC2=CCCOC2)[nH]1 Cc1nc(-c2ccccc2)[nH]c1C(=O)NCCCC(C)NC(=O)C(C)O N1(C(c2nc(C)[nH]n2)=O)CCCC(C2CCCCN2C(=O)CC2CCN(C)C2)C1 c1(C(N2C(C(=O)NCCC(C)N(CCC)C)C(C)CC2)=O)cnc(O)c(C)c1 C(CCC(C)(C)C(=O)N1CC2CCC(CNC(=O)C(C3CC3)C3CC3)C2C1)OC C(=O)(C1=CC2CCC=CCCC12)NC12CC(CNC(C(N=S(C)(C)=O)=O)=O)(C1)C2 Cc1ccn(CC(=O)NCC2(CNC(c3cncc(Cl)c3Cl)=O)CC2)c(=O)c1 Cc1cn2c(C(=O)NCC(C)(O)CNC(C3CC3C)=O)cnc2s1 N1(C(CC2CC(NC(c3cncc(C)c3)=O)C2)=O)CC2COCC2C1 N1(C(c2ccc(-c3ccc(C)o3)s2)=O)CC=CC(NC(=O)C(F)F)C1 c1(-n2c(C3C(CC)C3)nc(-c3ccnn3C)n2)ccc2[nH]ncc2c1 N1(CC)CCCC2C1CCN2CC1CC2CCN(CC(C3CCCCC3)O)CC12 C=C(C)C1OCCC1C(N1CCC(C(F)F)C1)=O.N12CC(C1)CC=CC2=O c1(C(=O)NCC2CCN(C(Cc3c(C)nc[nH]3)=O)C2)cc2ncccc2o1 Cc1cccc2cc(C(=O)NC3C4CCN(C(=O)C(C)(C)O)C34)oc12 N1(C(c2cc(SC)oc2)=O)CCCC(CNC(=O)C(c2ccccc2)F)C1 c1(C(=O)NCC(C)(C)NC(C(n2ncc(C)c2)C)=O)c[nH]nc1[N+](=O)[O-] Cc1ccc(Cl)c(OCC(N2CC3CC3(CNC(C3(CF)COC3)=O)C2)=O)c1 C(=O)(CCC1=CCc2ccccc21)N1CCC(NC(C2C(C)CCC2)=O)C(F)C1 c1(CC(=O)NCc2csc(CNC(c3cc(C(N)=O)c[nH]3)=O)n2)ccc(Cl)cn1 c1(C(=O)NC2CN(CCC)C(=O)C2)cc(Cl)c(Cl)c(CC)c1 c1(C(N(C2CCCCC2)CC)=O)ccc(-c2cccnc2C(=O)NC)nc1 C1(CC(=O)NCC2(CC)CC2)CN(C(C2CCC(C)(O)CC2)=O)CC12CC2 Cc1cc(Br)cc(C(N2CCN(C(=O)C=Cc3cn[nH]c3)C(C)C2)=O)c1F Cc1cc(OC(C2CN(C(=O)Cn3nccn3)CC2O)=O)sc1C(=O)OC(C)C N1(C(CSCC)=O)CC2(CCC(NC(=O)CC3(O)CCOC3)CC2)C1 c1(C(C)OC)ncc(C(=O)NC(C)CNC(c2cccn2CC2CCCC2)=O)s1 c1(C(=O)NCC2(O)CCN(C(C(C=CCCC)O)=O)CC2)ccn2ccnc2n1 c1(CC(=O)NC(CCCC)CNC(c2cnc(C)[nH]2)=O)ncn2c1CCC2 C1(N(C(C(C2CCC2)OC)=O)C)CCCCN(C(c2ccc(C(N)=O)cn2)=O)C1 C1(C(N2CCCC(CN(C)C(c3nc(O)[nH]c(=O)n3)=O)C2)=O)CCCC2CC12 c1(NC(C2COCCN2Cc2cc(C(F)(F)F)cc(F)c2)=O)cc(Cl)c(O)c(Cl)c1 CC1CC(CNC(=O)CC2CC=CC2)CN1C(=O)Cc1cncnc1 c1(C(=O)NC2C(CC)CN(C(=O)CCN3CCC3)C2)cc(C)c(C)cc1C c1(C(=O)NCCCCNC(C(C)NC(CC)=O)=O)ccc(S(=O)(=O)NOC)cc1 C=CC(CC)CC(=O)N(CCCNC(=O)Cc1ccc(CC)c(F)c1)C c1(CNC(C2(C=C)CCC2)=O)cc(C(=O)N(CC(C2CCCC2)O)C)ccn1 C12(C(=O)NCCN3CCC(NC(=O)C4=COCC4)CC3)CCCC(C1)OC2 CC#CCCCC(=O)NCC(C)(C)C(=O)N(CC(=O)N(C)C)CC c1(C(N2CC(C3N(C(CC=C)=O)CCC3)(O)C2)=O)cc([N+](=O)[O-])nn1C C(=O)(CCCC(=O)N1CCC(=CCOC2CCN(C(=O)C(C)O)C2)CC1)OCC N1(C(c2scc(C)c2)=O)CC(NC(c2cc3ccsc3s2)=O)CC12CCOCC2 C1(CNC(CCOC)=O)CN(C(c2cccnc2OC(F)(F)F)=O)CC1C CC1=C(C)CC(C(=O)NCc2cc(C)c(C(=O)NCc3cccnc3C)o2)CC1 C(C1(O)CCc2cc(F)ccc21)NC(c1cc(C2CCOC2)[nH]n1)=O N1(C(c2c(C)c(F)ccc2)=O)CC(NC(c2ccnnc2S)=O)CC2(CCC2)C1 N1(C(C2C(C)(C)CO2)=O)CC2CC1CN2C(c1cnc(CCC(F)(F)F)s1)=O C12(C(=O)NC(C)CC3(O)CN(C(=O)CC4C=CCC4)C3)CC3CC(CC(C3)C1)C2 N1(C(c2ncc(C)cc2F)=O)CCCC(C)(C)C1CNC(C1(C)CC2CC2C1)=O CCCCCC(=O)NCCC(=O)N(CCNC(=O)CC1(C(F)F)CC1)C1CC1 c1(C(N2CCC(CCNC(c3c(C)scc3)=O)C2)=O)ccc2c(c1)CC2 CC1(C)CC2(C1)C(=O)NC2.C1(NC(C2CC3CC3C2)=O)CC2CCC1O2 C(=O)(CCC(C)O)NCC(CNC(COCCOC)=O)C c1(OC)ccc(CC(N2CC(NC(c3cnc(C)nc3)=O)C(C)C2)=O)c(C)c1 C1(NC(C(=O)NCC)CC)C=C(c2ccccc2)CC1 C1(C(N2C3CC(C(N4CCCC5(CC5)C4)=O)C2CC3)=O)C2Sc3ccccc3C12 N1(C(C(CC)SC)=O)CCC2(CCCN2C(=O)CCNC(=O)Cn2cnnn2)C1 N1(C(COCCC#C)=O)CCCCC(N=c2nc[nH]cc2C#N)C1 c1(C(=O)NCC2C(C(=O)NCCC3CCC4CC34)CCC2)ncccc1F C1(NC(c2n(CCCC)ncc2)=O)CC(O)CN(C(=O)CC2CCC=CCC2)C1 N1(C(C(CC)(F)F)=O)CCCC(F)(C(=O)NCCNC(=O)NCC)C1 N1(C(CC=C)=O)CC2(CCCN(C(c3nc(C)cnc3C)=O)C2)C1 c1(C(C)C)cc(C(=O)NCC(C2CC2)NC(c2sccc2OC(F)F)=O)n[nH]1 C1(NC(c2nc(C(C)C)oc2)=O)CC2CC(C1)N(C(C1(C)CC(O)CN1C)=O)C2 C1(NC(c2c[nH]c(C(F)(F)F)c2)=O)CC1C1CCCN(C(=O)Cc2ccno2)C1 N1(C(C=CC=CC)=O)CC(NC(C2C(c3ccccc3)C2(F)F)=O)C(O)C1 C1(CC)(Nc2ncnc(Cl)c2CO)CCN(C(c2cc(=O)n(C)cn2)=O)CC1 CCC(C)(CNC(=O)C(C)C(C)C)C(=O)NN1CCCC1C C12CCCC13CN(C3)C2=O.N12CCN(CC1)CCCC2=O.C(C)(C)(C)OC(C)=O N1(C(C2C(CCC)C2)=O)CCC(C)C(NC(=O)C=CCF)C1C Cc1cnc(CNC(C2CSCN2C(C2CCCCO2)=O)=O)[nH]1 N1(C(N2CC(C)C(C(=O)OC(C)(C)C)C2)=O)CC(C)C(F)(F)C1 C=CCC(CC(F)F)NC(C1CN(C(=O)CC2(OC)CCC2)CC1C)=O CC1(C)CN(C(c2sccc2Cl)=O)CCC1C(=O)NC(CO)CCC1CC1 N1(C(C(CO)OC)=O)CCOC(CNC(=O)C(N2CCC(O)CC2)C)C1 N1(C(Cc2cc(C)sc2)=O)CCN(C(C2CCOC2C(C)C)=O)CC(C)(F)C1 C1(NC(C2(CC#C)CCCC2)=O)CCC(C)N(C(=O)Cn2cc[n+](C)c2)C1 CC1CN(C(=O)C(C)(C)c2ccccn2)CC1NC(=O)C=Cc1cccs1 Cc1ccc2nnc(C(C#N)C(=O)N(C)C)n2n1.c12cc(cnc1O)C(=O)NNC2=O N1(C(c2cnccn2)C(=O)Nc2c(C)cccc2)CC23CCCC2(COC3)C1 C(=O)(C1CCc2ccccc21)N1C(CCNC(c2cnc(O)o2)=O)CSCC1 CC1(C)CC(C(=O)NCc2cccc(O)c2)CCN1C(C12CCCC1C2(F)F)=O Cc1[nH]cc(C(=O)NC2CN(C(=O)CC3CCCC3O)CC2(C)C)c(=O)c1Cl C1(C(N(C2CCN(C(c3c(C)con3)=O)C2)CCO)=O)CC12CC(O)C2 C#CC1(C(=O)NC(COC)C(C)C)CCN(C(=O)CCc2ccccn2)CC1 C(=O)(CCCCNC(C1CCCCN1C(c1ccc(F)s1)=O)=O)OCC N1(CC2CC(C(=O)OCC)C2)CCC2(CC1)CC(Cc1ccc(F)cc1)=NO2 C1(N(CCCOCC)C)CCCC1CNC(C1(O)CCC1)=O C1(CNC(C(C)CO)=O)CCC2(CN(C(=O)Cn3cc(Br)cn3)C2)O1 C1(SC)CN(C(C2CCCCC2O)=O)CC1NC(c1ccncn1)=O c1(C(=O)NC2CCN(C(C(C(CC)O)(F)F)=O)C2)sc2cccc(F)c2c1Cl C1(NC(c2cnc(S)[nH]2)=O)CC2CC(C1)N(C(c1ncsc1Br)=O)C2 Cc1nccc(CNC(=O)C=CCC(C)(C)NC(=O)Cc2cc[nH]n2)n1 C(=O)(CC1OCCc2sccc21)NCC(C)(CO)NC(C(CC#C)C)=O c1(C(N2C(C(C)(C)NC(C(C=CC)O)=O)CCC2)=O)cnc2cnn(C)c2c1 C1(C(=O)Nc2scc(C)n2)CC12CCN(c1ncnc(C)c1Br)C2 N1(C(CCC=C)=O)CCCC(C(=O)Nc2cccc(C(C)O)c2)CC1 C(=O)(C=C1SCC(=O)N1C)N1CC(NC(C(CC=CCC)C)=O)C(OC)C1 C12(C(=O)NC3C(C=C)OCC3)COCC1CN(C(=O)Cc1cccc(F)c1)C2 c1(NCCN(C(C)C)C(C2(C)CCC(=O)NC2)=O)ncc([N+](=O)[O-])cc1F CCCC(C)(C)C(=O)NCC1(O)CCCN(C(c2nccc(Cl)c2O)=O)C1 C1(C(=O)NCC2CCC(NC(COCC(C)C)=O)C2)CC2CCC(C1)C2(F)F C1(OC)CC(CNC(=O)Cn2nnc(-c3ccco3)n2)N(C(c2ccc(F)s2)=O)C1 n1(-c2cccc(C)c2)nc(C2CC=CCC2)nc1C1CCc2c[nH]nc21 c1(CC(=O)N(CC(C)N(C)C(C2CCC23CCC3)=O)C)c(F)cccc1F c1(CNC(c2c(C)scc2)c2nnnn2C2CCC2)ncc(Br)nn1 C1(C(=O)NCC2(OCC)CN(C(=O)C(Br)=C(C)C)C2)CC2C(C1)C2(C)C C1(NC(=O)CN2CCCC2)C2CN(C(c3csc(C(F)(F)F)n3)=O)CC12 C(=O)(CCCCC(C)(C)C)NC1CC(CCNC(C(C)NC(=O)C2CC2)=O)C1 C1(CCC(C)C)(NC(OCC#CC)=O)CN(C(c2cc(Cl)c(Br)s2)=O)CCC1O C(C1CCCC1)=C(C)C(=O)NC(C)C(=O)NC(C)Cc1nn[nH]n1 c1(CN(C(CN2CCC(CCCC)C2)=O)C)ccccc1Cl C1(NC(C(c2ccc(C)cc2)F)=O)CCN(C(c2cccc(Cl)c2)=O)C(C)C1 N1(C(CC(N2CCCC2C(=O)NC2CCN(CCO)CC2)=O)=O)CC2CCC1C2 N1C(=NCCCOCCS)NCC1.C1(C(C)NC2CCCC2)CCN(C)C1 N1(C(Cn2c(C)nnn2)=O)CC2CC1CN2C(c1sc(=N)[nH]c1C1CC1)=O Cc1nn(C2CCCCC2)cc1C(=O)NCC12CC(CN1C(=O)C=C(Cl)Cl)C2 C1(NC(c2c(C)c(Cl)ccc2)=O)CCN(C(=O)C2=CCCO2)CC1(C)C c1(C(=O)NCC2C(C)CN(C(c3cccnn3)=O)C2)cc(S(C)(=O)=O)ccc1Cl C1(Nc2cc(N3CCN(CC)CC3)ncn2)CCC(OC(F)F)CC1 CCC(C(=O)NC(C1CCN(C(c2[nH]nnc2C2CC2)=O)C1)(C)C)c1ccccc1 C1(CNC(c2c(C)nns2)=O)CN(C(=O)CCc2nncs2)CC1O C(=O)(C(N=[N+]=[N-])C(C)C)N1CCC(CC)CC1CC(=O)NOCCOC c1(C(N2CC(C3CN(C(C(CC)OCC)=O)C3)OCC2)=O)ccc(Cl)cc1N c1(C(=O)NCC2CN(C(c3cc(C)nc(C)n3)=O)C(C)C2)cnc2n1CCCC2 CC1(C)CCCC(C(N2CCCC2C(C)(C)CNC(C2CC3(CC3)CO2)=O)=O)C1 C1(C(N2C(CCNC(C(C3CCC(=O)N3)C)=O)CSCC2)=O)COC2COCC12 C(CC(=O)NCC(C)(CC(C)C)NC(c1cnn[nH]1)=O)(C(F)(F)F)OC Cc1nc(N(CCC(C)NC(C2(n3cncn3)CC2)=O)C)c(C)c(Cl)n1 c1(N2C(=O)CC(NC(CCC#C)(C)C)C2)ccc(Cl)c(Cl)c1 C1(C(N(C(C)C(N2CCOCC2)=O)CC)=O)CCOC12CCOCC2 c1(C(=O)NC(C)C(C)NC(C2CSC2)=O)cnn(-c2ccccc2)c1 C1(N(C)C)CCC(NC(C2CCN(C(=O)Cc3cncnc3)CC2)=O)CC1 Cc1cc(N)c(F)c(C(N2CC(NC(C34CCC(CC3)C4)=O)C(O)C2)=O)c1F CC1CN(C(c2csc([N+](=O)[O-])c2)=O)CC1(C)CNC(=O)C(c1ccccc1)F C1(N(C(c2ccc(CNC(c3ccc(C)nc3)=O)cn2)=O)C)CCCC(C)(C)C1 c1(C(=O)NC(CNC(C(C)SCc2nncn2C)=O)C2CC2)ccc(N)cc1Cl N1(C(C2C(=C)C2)=O)CC2CCC1CC2NC(=O)C(C)(C)CF CCCC(C(=O)N(C)Cc1ccc(C)cn1)NC(c1ccccc1)=O C1(C(=O)NC2(COC)CN(C(c3cc[nH]c3C)=O)C2)Cc2cc(F)ccc2O1 C(=O)(C(CC(C)C)CC(C)C)NC(CCNC(c1cc(C)c(Cl)cc1)=O)C Cn1nc2c(c1C(N1CC3C(CNC(c4ccccn4)=O)C3C1)=O)CSCC2 CC1(C#CC=O)COC1.C1(=C2CCC3(CC2)CC3)C2CC(O)C1NC2 c1(C(=O)NC2C(C)N(C(C3C4CCC(F)(F)C34)=O)CC2)cc(S(N)(=O)=O)oc1Cl CCCC(CC)CCC(=O)NC1CN(C(c2ccc(C#N)s2)=O)CC1O N1(C(C(CNC(CCCCC=C)=O)CC2CC2)=O)CCC(C2CCC2)CC1 C1(CNC(C2CCCS2(=O)=O)=O)CN(C(c2coc(CO)c2)=O)CCO1 C(=O)(CC1=NNC(=O)C1)NCC1(C)CCCN1C(c1cc(Cl)nc(=N)[nH]1)=O Cc1cc(F)c(C(=O)O)cc1NC(=O)C(=O)NCCCNC(=O)CCCC1CC1 C1(NC(=O)CO)CCN(C(c2c[nH]nc2OCCCCOCC(F)(F)F)=O)C1 C1(C(=O)NCc2ncc(C)s2)CC2(CCN(C(=O)C(N3CCNC3=O)C)C2)C1 c1(C(=O)NC2(CNC(c3ccc(OC)s3)=O)COC2)ccc2ccsc2c1 CC(=O)CCCC(=O)NC1CCOC1C(=O)NOC(C)C c12ccc(F)c(c1F)NC2=O.CC(CNC(=O)C(O)C1CCC1)CC1CCCC1 c1(C(=O)NC2C(OC)COC2)oc(CNC(C2(CO)CCCC2)=O)nc1C C#CCC(C(=O)NC(c1cnn(C)c1)C)NC(c1coc(C(C)C)n1)=O C1(F)(CNC(C(CC)SC(F)(F)F)=O)CCCN(C(=O)C(N)=O)C1 CC(O)CCCCCC(=O)N1CCOCC1.N1CNS(=O)(=O)CCOC1 C1(NC(C2(CCCC)CCC2)=O)CN(C(c2cccc(CF)c2)=O)CC1O c1(C(=O)NCC2CN(C(c3c(C)onc3CO)=O)CC2C)c[nH]c(=N)nc1C N1(C(CNC(=O)NC)=O)CCN(C(c2cc(O)nc(C)n2)=O)C(C(C)C)C1 CC(C)CCCC(C)C(=O)N(C)CCC1CCN(C(C2COC(=O)N2)=O)CC1 C1(NC(C(c2ccccc2Cl)C)=O)CCCC2CN(c3ccnc(C#N)n3)CC12 CCCC(C)C(=O)N1CCC(F)(C(=O)Nc2nccnc2C)C1 c1(NC(C2CCCN(c3cc(C)nc(C)n3)C2)=O)ccc(C(F)(F)F)c(F)c1C C1(NC(C(CCN(C)C)O)=O)(CO)CCCN(C(=O)Cc2cccc(O)c2)C1 N1(C(C(C(CC)CC)C)=O)CC(CNC(=O)C=Cc2ncc[nH]2)OC2COCC12 C1(C(=O)NCc2cc(C(N(CC)CC)=O)no2)CCOC(C)C1 CC1CCN(C(C2CC(NCc3cc(Br)c(F)cc3Cl)C2)=O)CC1(F)F C1(OC(C)C)CN(C(=O)C(C)NC(C2CCCO2)=O)C1 c1(OC)ccc(C(=O)NC(C2CCCN2C(C2CC(F)CN2C)=O)C)cc1F C1(NC(Cc2ccc(C)cc2)=O)C(C)CCN(C(=O)Cc2cnccn2)C1C C(C1=CCCN(C(C2(F)CCCCCC2)=O)C1)NC(c1ncccc1CO)=O C(CC(=O)NC1CCC(CC)CC1)(C(C)C)NC(c1c(CCC)cccc1)=O C1(C)(C(N(CCOC)CCNC(C23CCC(CC2)C3)=O)=O)CCCS1(=O)=O C1(C(=O)NC2CC(O)(CNC(C(C)CC3CCCC3)=O)C2)CC(=O)N(O)C1 C1(NC(=O)CCOCC(F)(F)F)CS(=O)(=O)CC1N=c1ccnc(CC2CC2)[nH]1 N1(C(c2cc(OC)n[nH]2)=O)CC(C)CCC1C(=O)NC(C#C)CC1CCCC1 C1(CNC(CC2(C=C)CC2)=O)CC(NC(c2cn(C3CC3)nn2)=O)C12CCC2 c1(C(=O)NC(C(C)C)C(=O)NC(C)CS(C)(=O)=O)cccc2ccoc12 N1(C(=O)NCC(CC(C)C)CN(C)C)CC(O)CC2(CCCC2)C1 C(c1ccc(C#N)cc1)=CC(=O)NC1CCC(C)N(C(c2cccc(=O)o2)=O)C1 N1(C(C=C(C)CCc2ccccc2)=O)CC2OCC(NC(=O)C3=CCCS3)C2C1 CCC(O)C(F)(F)C(=O)NCC1C2CN(C(c3ccc(N)cc3OC)=O)CC12 c1(OCC(N2CC(NC(C(C)C(F)F)=O)C2)=O)ccc(Cl)cc1F C1(NC(c2c(OCC)nccc2)=O)CC2CC1N(C(C13CC(F)C1C3)=O)C2 c1(C(N2C(CNC(c3c(CC)non3)=O)C(C)CC2)=O)cncc(S(N)(=O)=O)c1 N1(C(c2c(C)n(C)nc2)=O)CC(F)(F)CC1(C)CNC(=O)Cc1ccnnc1O C1(NC(C2CCOC2)=O)CCC(NC(=O)C(F)(F)COc2ccc(F)cc2)CC1 C12(C(N3C(CNC(c4ncsc4C4CC4)=O)CCCC3)=O)CCCN(CCC1)C2 c1(NC(C(N2CCC(C)(NCCN(C)C)CC2)=O)=O)ccccc1[N+](=O)[O-] C12(CNC(=O)Nc3c(C)c(Cl)ncn3)CCC(CC1)C(C)(C)O2 CC(CN=c1[nH]cncc1Cl)Oc1cccc(Cl)c1Br Cc1[nH]nc2c1CC(C(=O)NC1CC(CCNC(=O)CCC(=O)N(C)C)C1)CC2 CCCC(C)(O)CC(=O)NC(C(=O)NCC1(N(C)C)CCC1)C(C)C Cc1ccnc(C(N2CCOC(C(C)NC(C3CC(C)(C)C3)=O)C2)=O)n1 CC1CN(C(c2c(Cl)nsc2Cl)=O)CCCN1C(c1ccc(-n2cccn2)cc1)=O C1(CC(=O)N(C)CCO)CCCCN1C(C1C=CC=CC=C1)=O Cc1cc(C(=O)NC2COCCC2NC(C2CCC(C)(C)CO2)=O)cc(C)c1N CCC(CC)(CN=c1c(C#N)c[nH]c2c(C)cc(F)cc12)OC c1(C(N(C2CN(C(C(CC=CC)CC)=O)CC2(C)C)C)=O)[nH]cc2c1CCCC2 c1(C(N2CC(C)(NC(C(CC)C(C)C)=O)C2)=O)cc2c(o1)CCCNC2=O C12(C(=O)NC(c3cncs3)C)CCC(CC1)N(C(C1CCOC1(C)C)=O)C2 CCCCCCNC(=S)NC1CC=CC1 c1(C(=O)NCC(CC=C)NC(c2ccc(COC)o2)=O)ccc(Cl)nc1 Cc1ccc(C(=O)OCC(C)C(C)(C)CN(C)C)c(F)c1.N12CC3CC1(C3)C2=O c1(N(C)C)cc(C(=O)NC2CCC2NC(c2cnc(C(C)(F)F)s2)=O)ccn1 C(CC(C)C(F)(F)F)NC(=O)NCC1CC(C)SCC1 C1(NC(CCCC)=O)CCC2CN(C(=O)Cc3ccc(Br)c4nsnc34)CC2C1 c1(C(N2CCC(CN(C(Cc3ccc(C)s3)=O)C)C2)=O)cnn2c1CCCN2 C(=O)(C1=C(F)CN(C(C2CN(C(N)=O)C2)=O)CC1)NC1CCCC(C#C)C1 c1(C(=O)NC(C2(O)CN(C(C3CC(F)CN3C)=O)C2)C)c[nH]c2ccc(F)cc12 C(=O)(C1=Cc2ccccc2OC1)N1CCN(C(CCCCC)=O)C(C)CC1 Cc1ccn2ncc(C(=O)NC3CC(NC(c4cc(CO)[nH]n4)=O)C3)c2c1 C1(CNC(C2CCC(=O)C2)=O)CCN(C(C2CCN(CC(F)F)CC2)=O)C12CC2 C1(C(=O)NC23C(NC(C(C)=C4CC4)=O)CC(CC2)C3)CCn2nnnc2C1 C#CC(CC(C)(C)C)NC(=O)C(C)N(C(C1(C)CC(C)(C)C1)=O)CC N1(C(CCOC)=O)CCCC(N(C(=O)CCCc2sccc2C)C)C1 c1(-c2n(C)ccn2)ccncc1NC(=O)NC1CCCC1c1cccc(F)c1 N1(C(C(CC(=C)C)C)=O)CCC2CCN(C(c3c(C)[nH]c4ccccc34)=O)CC12 c1(N2CC3(C(NC(c4occ(C)c4)=O)CCC3)C2)cc2nncn2c(C)n1 Cc1nc(C2CC2)oc1C(=O)NCC(C)NC(=O)CC(C)CN(C)C Cc1ccnc2c1CC(C(=O)NCC1CCCC1NC(c1ccsc1Cl)=O)CC2 CCCC(CCC)C(=O)N1CCC(NC(c2c(F)ccnc2Cl)=O)CC(O)C1 C1(CNC(CCSCCN(CC)CC)=O)C(O)C(O)CN1C(=O)CCS(C)(=O)=O N1(C(CC2N(C)CCC2)=O)CC2CC2(CNC(c2cnc(Cl)s2)=O)C1 C=C(C)C1OCCC1C(=O)NC1C2CC1N(C(c1cnncc1C)=O)C2 C1(NC(C2C(C)OCC2)=O)CCN(C(C2CNC(=O)C2)=O)CC1(C)C C(=O)(CC(C(C)C)OCC)N1C(C(C)(C)CCNC(C=CCCC)=O)CCC1 C1(C(=O)NCC2CCN(C(=O)CN3CCCCC3)C2)CC(c2ccncc2)=NO1 C1(C(=O)NC(CN(C(C2CC3(CCCCC3)C2)=O)CC)C)CN2CCN1C(C)C2 N1(C(C=C(C)CCc2ccccc2)=O)CC(NC(=O)CC(C)C)CC(C)(C)C1 C1(C2CCCC2)(NC(C2CCCC2NC(C2CCC=CCC2)=O)=O)CC1 c1ncnc2c1ncn2C1CC1C.N12CCCC(C1)CC(=O)C(C)(C)C2=O.CS C=CC1CCCN1C(=O)C(C)(CSC)NC(C1COCC1C(N)=O)=O C(=O)(C(O)C(F)(F)F)N(C)CCN(C(=O)CCc1cc[nH]n1)C c1(C(N2CC(NC(C3CC3C3CCC3)=O)CC(C)C2)=O)ccc(S(C)(=O)=O)s1 CC1CN(C(C2OCCC2NC(=O)CC2CC(F)C2)=O)CCC1(F)F C1(N(C(C=CCC)=O)CCCCCC)CCN(C(=O)CC(=O)NCCCC)CC1 N1(C(COC(COC)(C)C)=O)CC(C)(C(=O)NCc2ccncc2F)CC1(C)C c1(C(=O)NC2CC(NC(C3(CC#C)CCCO3)=O)C2)sc(C(C)(C)C)nc1C C(=O)(C1=NOC(CNC(c2cc(C)c(C)[nH]2)=O)C1)NCC=CCOCC N1(C(C(=O)NC(C)C)=O)CC(C)C(NC(c2c[nH]c3ccccc23)=O)C(C)C1 C1(C2N(C(c3scnc3Cl)=O)CCC2)CCCN(C(c2cc(CO)[nH]n2)=O)C1 CCC(C)(CC)C(=O)NCC(C1CCN(C(=O)C(C)C2CC2)CC1)F N1(C(C=C(COC)C)=O)CCCC(C(C)(O)CNC(=O)CSCC(F)(F)F)C1 N1(C(C2CC(=O)NCC2)=O)CCCCC12CCCN(C(c1ccsc1Cl)=O)C2 N1(C(C2C3(CC(=O)NC2)CCC3)=O)CC2CCN(C(=O)COC(F)(F)F)CCC2C1 C(=O)(CC(C)(O)C(F)(F)F)NCC(C)CNC(c1cnoc1-c1ccc(Cl)s1)=O c1(CCNC(=O)Nc2cccc(COC)c2)ccc2[nH]ccc2c1 O=C(C1c2ccccc2CN1Cc1cnc(F)cc1C(F)(F)F)N1CCC(Br)C1 c1(OC)cc(C(=O)NCC#CCNC(=O)C(C)OCC(C)C)c(Cl)cn1 C(=O)(C1=CCC2CCC1N2C(c1nccnc1C)=O)N1CCC(C)(COC)CC1 c1(OCC(=O)NCCN(C)C(C2CC(N3CCCC3)C2)=O)cccnc1.C1(N)CC1 CCCCCCCCC(C)C(=O)N1CCCC(C2(NC(=O)CNS(C)(=O)=O)CC2)C1 C1(CNC(c2cc(SC)ncc2)=O)C(C)CCCN1C(c1occc1C)=O C(=O)(C(C)CCC(C)(C)C)N1CCC(O)(CN(C(c2c(C)nc[nH]2)=O)C)C1 c1(C(N2CCOCC2)=O)cn2c(n1)CN(C(=O)C(C)n1cncn1)CC2 N1(C(Cn2ccc(C)n2)=O)CCC2(CCCN(C(c3cc(C#N)[nH]c3C)=O)C2)C1 N12CCC(CC1C)C2.c1(CC(n2cc(-c3nc(C)sc3)nn2)C)cnc(S)n1C c1(C(N2CCC(C)(NC(C(CCCCC)O)=O)C2)=O)c(C)nn2c1CCCC2 Nc1c(C(=O)NCCNC(c2[nH]nnc2-c2ccccc2)=O)cccc1F C1(C(C(=O)N(C)CC2CCO2)NC(C)=O)CCCCC1 c1(CNC(=O)NCC2(C)CCC(C)(C)C2)cscc1S(C)(=O)=O C1(NC(C=C(C)C2CC2)=O)C(CNC(C2(n3ccnn3)CC2)=O)CCC12CCC2 c1(CNC(CC(=O)NCCCCCC)c2nn[nH]n2)cccc2oc(C)cc12 C(=O)(C(C)(O)C(C)C)NC1CCC(N(CCC(=O)NC)C(=O)OC)CC1 C1(NC(C2CC(C)(C)C2)=O)CCN(C(=O)CCCCNC(N)=O)CC1O C1(S(N)(=O)=O)(C(N(CCCN(C)C(c2coc(-c3cnn(C)c3)n2)=O)C)=O)CC1 N1(C(C(CCC)O)=O)CCN(C(C2CCC(=O)N(CCOC)C2)=O)CCC1C c1(-c2nc(-c3cc(N(C)C)ncc3)nn2Cc2ccc(Cl)cc2)cc2n(n1)CCO2 c1(Sc2c(C)n(C)nc2CN=c2ccnc(CC(C)C)[nH]2)nn(C)c2ccccc12 N1(C(C(CC=C)OC)=O)CC(CNC(c2ccc(CCC)[nH]2)=O)CCC1C C#CCC(C)(C(=O)N1CCC(O)C(C)C1)NC(c1cc(C)c(C)cn1)=O N1(C(c2n(C)ccn2)=O)CC2CCC1C1CN(C(=O)CCc3ccnn3C)CC21 c1(C(N2CC(CNC(c3c(C)csc3)=O)OCC2)=O)cc(Br)c(F)cc1F C1(C(=O)NCc2ccoc2C(=O)NC(C)CCO)(COC)CC=CC1 c1(OC(C)C)ccc(NC(c2c[nH]nc2COCC(F)(F)F)=O)cn1 C(CCCCC(=O)N(C(C)(C(=O)NCc1ccc(F)cc1C)C1CC1)C)OC NS(=O)(=O)c1cc(C(=O)NCCN(C(=O)C(F)(F)C(O)C2CC2)CC2CC2)co1 n1(C(C)C(=O)O)cc(CN(CCCO)CCF)nn1 N1(C(C2C(C)CCO2)=O)CCOC(C(=O)NC(C2CCOC2)CO)C1 N1(C(CC2CN(C)C(C(F)(F)F)CC2)=O)CCC23CCCCC2(C1)C3(F)F N1(C(C(C)NC(c2cnn[nH]2)=O)=O)CCC1(C)C c1(OC)nscc1C(=O)NCc1cc(C(=O)NCCCCCC2CC2)no1 c1(C(N2C(C(=O)Nc3ccc(N(C)CC)cc3)CCCC2)=O)ncnc(O)c1F C(CC(C(=O)NC(C)C(O)C(F)F)NC(=O)C(O)Cn1cncn1)OCC c1(C(=O)NCc2c(CNC(C3C(CC)CCO3)=O)nccc2)snc(Cl)c1Cl c1(CCNC)cccc2ccccc12.C1C(C)CNC(=O)N1CCCC c1(NC(C(C2CCCC2SC)N(C)CCNC(C)=O)=O)c(OC)cnnc1OC N1(C(C=Cc2scc(C)n2)=O)CC(NC(c2cnc(C)nc2C)=O)CC12CCC2 CC1(C)CCN(CCNC(c2ccc(CNC(C3CC3(F)Cl)=O)o2)=O)C1 c1(C(C)=O)ncc(C(N2CCC(C3CCCN3C(=O)CC3CC(C)(C)C3)C2)=O)s1 C1(c2nc(CCCN(C)C)on2)(CCc2ccon2)CCCCC1 c1(OC)ccc(C(=O)NC2CCN(C(c3cnc(F)c(C)c3)=O)CC2F)cc1Br CCCCCCCCC(=O)N1CCOCC1CN(C(=O)C(C)(CC)CO)C CC1(C)CCCC1CNC(c1[nH]ccc1-c1ccccc1)=O C=CCCCC(C(=O)NC(CC)C(C)(C)C)NC(=O)COCCF c1(NC(=O)NNC(=O)c2ccsc2)cc(F)c(F)c(F)c1 C(CC1CCCC1)(C(=O)NC(CC1CC1)C(=O)NC(C1(O)CCC1)C)OC c1(C(N2C(COC)CN(C(=O)C=CBr)CC2)=O)ccnc2ccccc12 C#CC12CC(CN1C(c1cn(CCNC(c3cc(Cl)n[nH]3)=O)cn1)=O)C2 C(CNC(=O)CCC1(OC)CCCC1)(CCOC)NC(CCOCCOC)=O C1(NCc2n(C)ccc2)CCCC2CN(C(=O)OC(C)(C)C)CC12 CC(C)S(=O)(=O)c1ccc(F)cc1CNCCCN(C1COC1)CCO N1(C(c2ncn(CC)c2)=O)CCC2(NC(c3ccn4ccnc4n3)=O)CCCC12 c1(CC(=O)NC2CCN(C(C3CC(C)N(C)C3)=O)CC2)c[nH]c2ccncc12 c1(SCCCC)cccc(C(=O)N(C)CCN(C(=O)C(C)CC2CCCO2)C)c1 N1(C(c2nc(C)n(C(F)F)c2)=O)CCCC2CN(C(=O)C(Cl)=CCl)CC12 C12(NC(=O)CN3CC=CC3)CCOCC1CN(C(c1cccc(CO)c1)=O)C2 c1(OC)ccc(-c2cc(C(=O)NC3C4CN(C(C)C)CC34)c[nH]2)cc1 CC(C(=O)NCCC1CN(C(c2cc(Cl)c(Br)cn2)=O)C1)C(C)(C)C CCC(C)C(O)C(=O)N1CCN(C(c2cccc(-n3ccnn3)c2)=O)CC1CO c1(C(=O)NC2C(NC(c3cn(CCC=C)nn3)=O)COC2)cncn(C)c1=O N1(C(CCOCCC)=O)CCCC(N2CCN(C(=O)C(C)c3cc[nH]n3)CC2)C1 C1(CNC(c2c(CCC)n[nH]c2)=O)CN(C(c2c(SC)noc2C)=O)C(C)(C)C1 C(=O)(C1=NOC(C)C1)NCC1CN(C(CCOc2c(CC)cccc2)=O)CC1C C1(C(N(C)Cc2c(CNC(C=CCCC)=O)cccc2)=O)CCc2nncn2C1 C1(Nc2ncc(C(=O)OC)cn2)CCN(C(=O)CCCC(C)(C)C)CC1(C)C Cn1cnc(CC(=O)NC(C2CCOC2)CNC(=O)CSC(C)(C)C)c1 c1(CN(c2ccnc3ccnn23)C(C2CCCNC2)C)ccc(F)c([N+](=O)[O-])c1 c1(C(=O)OC)ccccc1C(=O)NC(CNC(=O)CCC(C)OC)C1CC1 CC(C)CCC(=O)NCC(=O)NC1C=CCN(C(C2CCON2CCOC)=O)C1 n1(CC)c(CNC(=O)CN(C(=O)CC2CCOCC2)C2CC2)nnc1O C(=O)(C(CC(C)C)OC)NC1CC(NC(c2c(C)nc(CC)s2)=O)C1 c1(OC)ccc(CO)cc1C(=O)N(C1CCC(NC(c2cc(=O)cc[nH]2)=O)C1)C c1(C(=O)NC2C3CC(NC(C=CSC)=O)CC32)ccc(S(C)(=O)=O)s1 Cn1ncc(C(=O)NCC(c2ccccc2)NC(=O)Cc2sc(O)nc2O)c1Cl c1(C(C)C)ccc(CC(=O)NCC(C)(CO)NC(=O)C(C)C2CCCC2)cc1 C1(CC(=O)NCc2csc(CCC)n2)CCCN(C(=O)CSC2CCOC2=O)C1 CC1CCCCC1(CNC(=O)CN1CC(=O)NC1=O)NC(=O)CCCC(F)F c1(C(=O)NC2CCC(CNC(c3occ(C)c3C)=O)CC2)ccc2nccn2c1 c1(C(=O)NCC=CC(=O)NC2(C(C)O)CC2)cnco1 C1(CNC(C2N(C(C(C)N3CCCC3)=O)CC(=O)C2)=O)CC2CCC(C1)O2 C(C)(C(=O)Nc1nccc(Sc2ccc(C)nc2NC)n1)(C(C)C)OC C#CCC(C)(C)C(=O)N(C)CCOCCN(C(=O)C(CCSC)NC=O)C C1(CCC)CN(C(=O)COCCOC)CC1C(=O)Nc1cc(CO)on1 CC1(C)CCC(C(=O)NC2C3CN(C(=O)C(C4CC4)C4CC4)CC23)O1 c1(C(=O)NC(C)C(C)NC(C2(CCF)CCC2)=O)ccncc1C(F)F c1(C(=O)OC)cc(CC(c2sc(F)cc2Cl)=O)c(C)s1.C(CS)N C1(NC(CC2CCC(NC(COCC(=O)NCC)=O)C2)=O)CC(C)(C)C12CC2 C(CC(=O)NCCC(C)OC)(C(F)F)NC(C1(CC)CC(C)(C)C1)=O C1(C(CNC(C=CCC2(NC(Cc3c(C)con3)=O)CCC2)=O)O)CCC(C)CC1 c1(C(=O)NC2CCC(NC(C(N3C(=O)CCC3=O)CC)=O)C2)nccc(C)c1N c1(C(=O)OC)ncc(Cl)cc1O.c1(C2=C3CN(C3)C2=O)ccc(Br)c(F)c1 c1(C(=O)NCC2CCN(C(=O)CCc3ccc(Cl)cc3F)C2)ccc(Cl)c(Br)c1 c1(C(=O)NCC=CCNC(C2CCN(C)S2(=O)=O)=O)cc(F)c2ccccc2c1 N1(C(C(C=C)(C)C)=O)CC(CC(=O)NC2CN(C)CC2C)C2(CC2)C1 C1(SC)CCN(C(c2onc(-c3cc(Br)sc3Cl)n2)=O)C(C)C1 O=C(C1=CCCN(c2ccc(C3CC3)nn2)C1)Nc1ncncc1Br C(=O)(CCCCC(F)F)N1C(C(C)C)C(NC(=O)Cn2nccn2)CC1 C(=O)(CC(O)CC(C)(C)C)NC1C2N(C(C=COCC)=O)C(CC2)C1 C=C(C)CCN=c1cc[nH]cc1S(=O)(=O)NCC1(NC2CCC2)CC1 N1(C(c2cnn(C(C)CC)c2)C(=O)NCC=C)Cc2ccccc2C1CCO CCCCC(CC)CC(=O)NC(CCC)C(O)C(=O)NC1CN(CC)C1 N1(C(C2C(C)OC(C)C2C)=O)CCC(Nc2ncc(Br)c(O)n2)C2(CCC2)C1 C1(CNC(CCOC)=O)COCCN(C(C2CCCC(C(F)(F)F)C2)=O)C1 N1(C(C(CC)SC)=O)CC(=O)NCC1C(=O)NCC1CC1 C12(CNC(=O)CC3=CCCC3)CCCCC1N(C(c1ccc(CO)s1)=O)CC2 N1(C(C2CN(C(C)=O)C2)=O)CCC(O)C(NC(c2c[nH]nc2C2CC2)=O)C1 N1(C(c2n(CC)nc(C)c2)=O)CC(CNC(c2cnc(SC)s2)=O)CC1(C)C N1(C(C2CCC3(CC3)C2)=O)CCCCC2(C1)CN(C(C1CCCCO1)=O)C2 C1(NC(C(CSC)C)=O)CS(=O)(=O)C2CN(C(=O)C=C(C)Cl)CC12 Cc1cc(C(N2CCC(C(C)NC(=O)COCCCF)CC2)=O)c(C)nc1C c1(NCC(C)SC(F)(F)F)ccccc1NC(=O)C(=O)NC(C1CCC1)=O CCC(C)C(C(=O)N1CC(C)(CCC(=O)NC)C1)N(C)C(C1CN(CC)CCO1)=O c1(C(N2CCC(N(C(C=CC(CC)C)=O)C)CC2)=O)ccc(Cl)c(F)c1 C(=O)(CCCCC(F)F)N1C(C2CCN(C(C3C(OC)CN(C)C3)=O)C2)CCC1 C1(CN(C(C(C)NC(N)=O)=O)C)CCCN(C(C2CC2Br)=O)C1 C1(NC(C2CCC3(CC3)N2C(C2CC(F)(F)C2)=O)=O)CC2(CCCC2)C1 C(=O)(CCCS(N)(=O)=O)NC1CCC(NC(C(C)Cc2ccncc2)=O)CC1 C1(NC(C(C)CF)=O)COC2(C1)CN(c1ncnc3[nH]cnc13)C2 C12(C(=O)NCC(C)CN(C)C(c3cc(F)cnc3O)=O)CCCC1CC(=O)CC2 c1(CC(N2CCOCC(NC(CCC(=O)N(C)C)=O)C2)=O)nnc2n1CCCC2 c1(SC)ccsc1C(=O)NCC(O)CN(C(=O)CC1C=CCCC1)C C(C(N)=O)(C(F)(F)F)N(C(CCC)C(=O)NO)C1CC1 Cc1n[nH]c(C)c1C(C)C(=O)N(CC(C)N(C)C(c1ncccc1CO)=O)C C1(C(N2CC(N(C(C(C)(CC3CCC3)OC)=O)C)C2)=O)C(F)(F)C12CCC2 N1(C(c2cccc(N(C)C)c2)=O)CC2CC1CC2NC(c1cc(O)cc(Cl)c1)=O C1(NC(C2CC(=C)C2)=O)CC(C(F)(F)F)(NC(C2(N3CCCC3)CC2)=O)C1 C=C1CCC(C(N2CC3CC3(CNC(c3nc(C)oc3OC)=O)C2)=O)CC1 C1(C(=O)NCCCCN(S(C)(=O)=O)C)COC2(CCC2)CN1 c1(C(=O)NCC2OCCN(C(CSC)=O)C2)c(F)c(F)c(Cl)c(F)c1F C1(C(=O)NCC2CCN2C(=O)CN(C(=O)C(C)C2CCCC2)C)(SC)CCC1 C(=O)(C(=O)NOC)N1CCC(NC(CC2(C=C)CCC2)=O)C1 c1(CCNC(C(=O)NC(C)(C)CCC2CCCCC2)=O)ccncc1Cl N1(C(=O)NC(c2nncs2)C2CC2)CCC(n2cncn2)C1 C1(C(=O)OCC(=O)N(CC#N)C(c2cccc(Br)c2)=O)COC2(CCC2)C1 CCCC(C(=O)NC(C)(CNC(C1(F)CCCCC1)=O)CO)c1ccc(Cl)cc1 c1(-c2n(C(COC)C)nc(-c3ccc(N)cn3)n2)cnn2c(N(C)C)ccnc12 c1(CCC)cc(C(=O)N(c2ccccc2)CC2CCOC2C)cc(O)n1 CC1(C)CC(C)(C(=O)NCc2nncs2)CN1C(c1ccc2[nH]ccc2n1)=O Cc1cccc(C(=O)NC(C)(C)CCNC(=O)C(C)CSc2ccccc2)c1F C(C(C#C)NC(C1(NC(=O)C(C)OCOC)CSC1)=O)SCC#C C(=O)(C(C)CC(N)=O)Nc1c(C2N(C(Cc3cc(C)no3)=O)CCCC2)n[nH]c1 O(NC(=O)CCC(C(C)C)NC(=O)C(CSC)CC)CCOCCCCC c1(C(=O)NC(C)CCNC(=O)CN2CCOC2=O)cc(O)cnc1Cl Cc1c(C(=O)NC2CC2NC(=O)C(F)(F)C2(O)CCCC2)cncc1Cl c1(C(=O)NC2C(CNC(c3ccc(OCC#C)cc3)=O)CC2)cc(C)cnc1C c1(C(N2C(CC(=O)Nc3c(OCC(N)=O)cccc3)CC2)=O)ncc(F)cc1N Cc1nnc2n1CCC2(C)C(=O)NC(C)Cn1cc(CCO)nn1 c1(CC(C)NC(=O)CC2CCCN2C(c2cnc(C3CC3)o2)=O)cccnc1 O=C(NNc1ccc([N+](=O)[O-])c(F)c1)c1cncc(Sc2ccc(Cl)cc2)n1 N1(C(CS(C)(=O)=O)=O)CCCC2(C1)CN(C(C1CC3CC1C3)=O)CCO2 C(=O)(C(C)CCC(C)(C)C)NCC(CC(C)C)(C)NC(c1nccnc1N)=O n1(CC(=O)NC(C)CCCCNC(=O)C(C)N(C)C)cc2ccccc2n1 N1(CC)CC(C(=O)N(CCCNC(C2CCCN(C(=O)NC)C2)=O)C2CC2)NC1=O CC(CC(=O)NC(C)CN(C)C(c1ccnc(Cl)c1)=O)C(F)F CC(C)CCCC(=O)NC(CCN(C(=O)CC1CC1(C)C)C)C(C)C N1(C(C=NOC)=O)CCN(C(=O)Cc2nnc(O)s2)C(c2ccc(F)c(F)c2)C1 N1(C(C2CCCC(=O)N2)=O)CC(NC(=O)C=Cc2cncnc2O)CC2(CC2)C1 c1(C(C)NC(C(=O)N(CCC=CBr)C(C)C)C)cccc(F)c1 C(C(=O)N=c1cc(Cl)nc(Cl)[nH]1)OC(C=Cc1c2cc(C)[nH]c2ccc1)=O c1(C(=O)NCC2CCN(C(=O)C=C3CC3)C2)cc(=O)n2ccsc2n1 c1(OC)cc(C(=O)NC2CCN(C(=O)C(C)(C)CF)CC2CO)c(Cl)cc1Cl c1(CC)sc(=N)[nH]c1C(=O)N(C1CCN(C(=O)COc2ccsc2)CC1)CC N1(C(C(C(CC)CC)O)=O)CC(NC(c2ccc(=O)n(C)n2)=O)CC12CCCC2 C1(C(c2nnnn2C2CC2)NCCC2(C)CCOC2)(OC)CCCCCC1 C1(CNC(CS(=O)(=O)N(CC)CC)=O)(COC)CCN(C(C2(F)CC2C)=O)CC1 c1(C(N2CCC(NC(c3c(C)nn(C)c3)=O)C2)=O)ccc(=O)n(C(C)C)c1 c1(C(N2C(C)COCC2)=O)cc(O)nc2c1CN(C(C1CCCCS1)=O)CC2 Cc1ncnc(C)c1CC(=O)NCC1=CCN(CC2CCC(=O)N2C)CC1 N1(CCC)CCCC1C(N1CCC(C(=O)NC(c2cccs2)C)C1)=O C1(NC(c2c(C)n(C)cc2)=O)CC2(C1)CC(C(=O)NC1CCN(C(C)(C)C)C1)C2 C1(C(=O)Nc2cccc(COC)c2)N(C(=O)CCc2cccs2)CCC1(C)C C(=O)(C(CC)C(C)(C)CC)N1CCN(C(C2(C(F)F)CC(=C)C2)=O)CC1 C1(CNC(C(C)NS(C)(=O)=O)=O)CN(C(c2ccc(F)cn2)=O)CC(C)(C)O1 CC1(C)CN(CCC2CCN(CC(F)(F)F)CC2)C1C1CCCO1 CCCCCC(O)CC(=O)NCc1ocnc1C(N1CCCC1(C)COC)=O C1(CCC)CN(C(=O)CC2(N(C)C)CC2)CC1C(=O)NCc1noc(C)n1 CC1(NC(c2cccc(OCC3CCCO3)c2)=O)CCCN(C(=O)CCC#N)C1 N1(C(C(C2CCOCC2)OC)=O)CCOCC(NC(c2cccc(CO)c2C)=O)C1 Cc1ccc(CC(N2CCC(NC(c3cc(Cl)cn3C)=O)C(CO)C2)=O)cc1Cl CCCCCC(C)(CC)C(=O)NCCC1CN(C(=O)C(C(C)C)NC(=O)NC)C1 CC1CCC(NC(=O)CCCCC2CC2)CN1C(=O)CCOCC1CC1 C1(C(c2ccsc2)=O)CN(C(C2CCCN(CCCO)C2)=O)CCO1 N1(C(c2cnn(C)c2Cl)=O)CCC2(CCN(C(C3CC(C(F)F)C3)=O)C2)C1 CC(F)(F)CCC(=O)N1CCC(N2CCN(C(=O)Cc3ccsn3)CC2)CC1 c1(C(N2CCC(NC(C(C)C3CC3)=O)C2)=O)ccc2c(c1)OCCO2 C1(O)(C(C)NC(C2CC(=O)CN2C(=O)CC2OCCCO2)=O)CCCCC1 C(=O)(C1Cc2c(Cl)cccc21)N1CC(CNC(c2cncc(OC(C)C)c2)=O)C1 O=C1CCN2C(=O)C2N1.C1CCCN(C(c2ccc(-c3cccs3)o2)=O)C1.C1CC1 C1(C(=O)NCC2CN(C(Cc3c(C)ncs3)=O)C(C)C2)CCc2n[nH]cc2C1 C(CN=c1ccc([N+](=O)[O-])c(C)[nH]1)C1CCN(C(c2c(OC)cncc2)=O)C1 N1(C(c2c(C)nc(C(C)C)cc2)=O)C2CCCC1CN(C(C1CSCCS1)=O)C2 c1(N2C(C)(C(N3CCCCCC3)=O)CCC2)ncnc2c1SCCC2 Cc1ocnc1C(=O)NCC1CCN1C(c1cn(-c2cnn(C)c2)cn1)=O N1(C(CCCC)=O)C2CCC1C(F)CC2.C1(C=O)(CC)CCCC1 C1(C(N(CC(O)CNC(=O)Cc2ccon2)C)=O)CC(C)(C)SC(C)(C)C1 c1(NC(C2CN(C(C3(COC)C=CCC3)=O)C2)C)ncc(S(C)(=O)=O)cc1Cl C=CC(CCC)CC(=O)N1CC2(CCC2)CC1CNC(c1cc(F)cnc1O)=O n1(CC(=O)NCC=C)cc(CNC(=O)CC2CCCCO2)nn1 c1(C(N2CC(NC(CC(CC)SC)=O)C2)=O)ccc(OC(C)C)cc1N c1(C(=O)NCC2C(NC(C(CC)OC)=O)CC2)ccc2c(c1)nnn2C N1(C(Cn2ncc(C#C)c2)=O)CC(NC(=O)Cc2cc(C)cc(C)c2)C2(CC2)C1 c1(C(=O)OC(=O)CCCCOc2ccccc2)ccc(C(=O)C(F)F)cc1 C1(C(=O)NC(C2CCN(C(c3ccoc3)=O)C2)C)C2CCC3(COC(=O)C13)O2 N1(C(C2CC(C(=O)OCC)C2)=O)CCCC1c1cn(C(C)(C)C)nn1 N1(C(CNS(CC)(=O)=O)=O)CC2CC1CN(C(C1CCC(C(N)=O)CC1)=O)C2 N1(C(c2nc(NC(c3cc(F)ccc3I)=O)sc2)=O)CCCC(F)(F)C1 C(=O)(C(CCC)OCC)NCC#CCNC(C(C=C)c1ccccc1)=O C#Cc1cccc(C(=O)NCC2CN(C(=O)Cn3cc[n+](C)c3)CCC2C)c1 N1(C(C(CNC(CSCCSC)=O)C)=O)CC=CC12CCCC2 c1(C(=O)NCCOCCNC(=O)C(C2CCCCC2)O)cc(F)sc1Br C(CCC(=O)NC1(CN(C)C)CC1)=C(C)C.c12ccc(o1)C(=O)NC2 C(=O)(C#CC1CCCOC1)NCC(C)(CNC(=O)CCc1ccccn1)OC C1(C(N(CCCCN(C(Cc2c(C)n[nH]c2)=O)C)C)=O)CC(=O)N(C(C)(C)C)C1 N1(C(C(=O)C2CCC2)=O)CCC(NC(c2c(C(F)F)cccc2F)=O)C(F)(F)CC1 C12(C(=O)NC(C34CCC(CC3)C4)C)COC(C1)C(NC(=O)C#CC1CCC1)C2 C1(NC(CCC2C(C)C2)=O)CN(C(c2cc(Br)cn2C)=O)CC12CCOCC2 c1(C(N2CCC(F)(CNC(C3C(C=C)C3)=O)CC2)=O)ccc2c(c1)CC(C)(C)C2 c1(C(=O)NCC2C(NC(C(C)N(C)C)=O)C2)c2n(c(=O)n1C)CCCC2 Cc1ccc(C)c(C(=O)NCCC2CCN(C(c3nn(C)c(C)c3Cl)=O)C2)c1N N1(C(c2cn(C)nc2O)=O)CC(NC(C2CS(=O)(=O)C2)=O)CC2(CCC2)C1 c1(CC)cc(C(=O)N(C(C)CNC(c2cn(CCOC)nc2C)=O)C)ccc1C C1(NC(c2ncccn2)=O)COC2CN(C(c3ccnnc3)=O)CC12 C(=O)(CCC(C)(C)[N+](=O)[O-])NC1(C)CC(NC(c2ccc(CC)c(CC)c2)=O)C1 c1(CC)noc(CC)c1CC(=O)NC1CC(CNC(=O)C(C)(C)OC)C1 C1(O)(CNC(C2C(COC)C2)=O)CCN(C(c2cnc(C3CCOC3)s2)=O)CC1 c1(C(N2C(C)(CNC(c3ncnn3C3CCC3)=O)CCC2)=O)cc([N+](=O)[O-])n[nH]1 Cc1nn(-c2ccccc2)c(C)c1CC(=O)NC1CCN(C(C2(C)CCC2)=O)C1 C1(C(=O)N(C2C=CC(C(=O)NCC3(O)CCSC3)C2)C2CC2)CC12CCOCC2 C(=O)(CCCCC(C)(C)C)N1CC2C(NCc3nc(C(C)C)sc3)(CCC2)C1 N1(C(C2CC(OCC)C2)=O)CC2CCN(C(c3cccnc3OC)=O)CC2C1 c1(NC(C2C=CC(NC(c3cccc(Cl)c3Cl)=O)C2)=O)ccc(C(F)F)cc1F C(=O)(C(C)(C)c1cncnc1)N(CCC(=O)O)CCCC(c1ccccn1)CO CC1COCCC1C(=O)N(C)CCN(C)C(c1cc(-n2cccc2)ccn1)=O N1(C(CC(CC)(C)C(=O)OC)=O)CCC(C2CCN(C(=O)CNS(N)(=O)=O)C2)C1 N12CCCCC1C(C)(C)CCC2=O.CCCCCCN.c1(C2C(=O)N2)cnoc1 C(c1cncc(C(F)(F)F)c1)=CC(=O)NC(CNC(CN1C(C)CCC1)=O)(C)CO C1(CF)CCC2CCC1N2c1nc(-c2ccc(C(F)(F)F)cc2)ns1 c1(C(N(C)CC2CCN(C(=O)Cn3cnnc3)CC2)=O)cc([N+](=O)[O-])cnc1O CCC(F)C(=O)N1CCC(N(C(=O)C(C)=C(C)CC)CCO)C1 C1(C(=O)NCC(CC)NC(=O)COCC2(F)CC2)CCC(C(C)(C)C)CC1 c1(NC(C(C(CC)O)C)=O)ccc2nccn2c1.C12(COC)C=CCN1C2=O Cc1oc(C(C)C)nc1C(N1CCC(CF)(NC(c2cnccc2Cl)=O)C1)=O C(=O)(C(CC1CC1)CC)NC(C(=O)N(CC(CCC)O)C)C1CCCC1 N1(C(C2CC(=O)C2)=O)CCC2(CCCN(C(c3cc4ccnc(Cl)c4s3)=O)C2)C1 c1(C(N2CC3(CC(NC(=O)CC4CS(=O)(=O)C4)C3)C2)=O)noc2cc(Cl)ccc12 c1(OC)c(C(=O)NC(C)(CNC(C2CCCC(C)O2)=O)C2CC2)nc(O)nc1O N1(C(C(C(C)C)NC(C=CC(CC)C)=O)=O)CCC12CCCSC2 c1(CCNC(=O)NC2CCCC2n2cccn2)cccc(F)c1 c1(NC(=O)NC2(c3c(C)ccnc3)CC2)ccc(S(N)(=O)=O)c(C)c1 CC1(C)CCCC(C(=O)NC(CNC(c2cnc(=N)[nH]c2)=O)C2CC2)O1 c1(OC)ccc(F)c(C(N2CCCC2CCNC(c2cnc(S)[nH]2)=O)=O)c1 C(CC(=O)NOC1CCCCC1)CC(N1CC(CC2(NC(N)=O)CCC2)C1)=O Cc1cc(F)c(C(=O)NC(C2CCOC2)CNC(=O)CC(C)(C)C)cc1F C1(OC)CC(NC(=O)Cc2ccc(C(=O)CN(C)C)cc2)C1(C)C C#CC1(NC(C2CCC(CNC(=O)C=CCN3CCC3)C2)=O)CC(F)(F)C1 C1(O)(CCNC(CP(C)(C)=O)=O)CCCN(C(C2CCC(O)C2)=O)C1 c1(C(=O)NC2CN(C(C(CC=CC)C)=O)CCC2)c[nH]c(=O)c2ccnn12 CC(C)CC(O)C(=O)N1CCN(c2ccc(C(=O)N(C)CCO)cn2)CC1 n1(CC)c(N(C)C(c2ccc(F)cc2F)=O)cc2ccccc12 c1(N(C(CNC(C2CCN(C(C)=O)CC2)=O)C)C)cc(S(C)(=O)=O)ncn1 C(=O)(C(O)CCCNC(C1(C#N)CC1)=O)NC(C)(C)C(N)=O c1(OCC(=O)OC(=O)C(C)N(CC)CC)ccc(N(CC)CC)cc1C.CC N#Cc1ccncc1C(=O)NCC1OCCC1C(=O)NCC(N1CCCC1)Cl C(=O)(CS(=O)(=O)C(C)(C)C)NCC1(O)CCN(C(C2CC(OC)C2)=O)C1 N1(C(C(C)n2ccnc2)=O)CCOC(C(=O)Nc2ccc(F)cc2)CC1 C(=O)(CCN=C(NCc1cc(C(C)C)no1)NC1CCOC(C)(C)C1)NC N1(C(C(=O)NCCOC)=O)CCN(C(=O)CCc2cnco2)CC1C1CC1 C(=O)(C1=CCC(NC(c2cc[nH]c2)=O)C1)NCCC1C(C)CCO1 CC(C(=O)NN=c1ccn(CC#N)[nH]1)S(=O)(=O)c1ccccc1C(F)F N1(C(C(C)=C(C)C)=O)CCC2(CC(NC(C3(C(N4CCCC4)=O)CC3)=O)C2)C1 c1(COC)nc(-c2nc(-c3ccc(O)cc3)nn2C2CCOC2C)sc1C CCCCCC(=O)N1CC(C)(NC(=O)Cc2cn(CC3CC3)nn2)C1 c1(C(N2C(C(N3CCCC(C)C3CCO)=O)CC(=C)C2)=O)ncc2ccccn12 c1(SC)ccc(CCCC(=O)NC2C3CC2N(C(C2CCC(=O)O2)=O)C3)cc1 C1(C(C)NC(CN(C(=O)C(C)n2ccnn2)CCC)=O)(CO)CCC1 CC1(O)CN(C(C2(NC(=O)CCc3ccc[nH]3)CC(O)C2)=O)C1 c1(OC)cccc(CNCC2CC(C(=O)NCc3ccncc3Cl)C2)c1 C(CC(C(C)(C)C)NC(c1cccc(NC(=O)C(C)(C)C#N)c1)=O)N(C)CC#N CC(C)CC(C(=O)N1CC2CC2C2CC12)ONC(=O)CC1C=NN(C)C1=O c1(C(=O)NCC2(C(F)F)CCN(C(c3c(CC)c[nH]c3)=O)C2)c(C)cnnc1O c1(C(N2CCC(N(C(=O)C3=CC(C)(C)C3)CC)C2)=O)ccc(CO)c(F)c1 C1(C)(C(=O)NC(C)CC2(C(F)(F)F)CCC2)CC1(C)C c1(NC(CNC(c2c(C)nc(CC3CC3)o2)=O)C)cc(C#N)c(F)cc1[N+](=O)[O-] Cc1c(NC(c2nc(C3CCOC3)nn2C2CCS(=O)(=O)C2)=O)cnn1C1CC1 C1(C(N2CCC(O)(C(C)NC(CSC)=O)C2)=O)CCC(O)CN1C C(=O)(CC(C)(C)C#N)NC1CCCC(NC(=O)Cc2cccs2)C1 c1(NC(=O)NCCNC(C)=O)ncc(-c2csc(N(C)C)n2)cn1 N1(C(c2csc(Br)n2)=O)CCOC(c2cn(C3CCC3O)nn2)C1 c1(OC)cc(OC)cc(CC(N2CC(F)CC2C(=O)NC(C(F)(F)F)C2CC2)=O)c1 N1(C(C2(CC#C)CC2)=O)CCC2CCN(C(c3cc(O)nc(O)c3)=O)CC2C1 CC(C)C(=O)CCCN1CCN(C(C2(C)CCC(C)C2)=O)CC1 c1(CNC(C2C3CN(c4c(CC)cncc4)CC32)=O)cc2n(n1)CCC2 C(=O)(C#CC1CCC1)N1CCC(C(C)NC(c2ccn(CC)n2)=O)C1 C(=O)(N=c1[nH]nc(C(C)(O)CC)s1)NC(C1CC(F)C1)CC c1(C(N(CCCOCCNC(C2C(CCC)C2)=O)C)=O)ccnc(C)c1Cl c1(C(=O)OC)cc2c(c(S(=O)(=O)Nc3cccc(N4CCCC4=O)c3)c1)CCC2 CCC(C)C(C(=O)N(C(C)(C(=O)NC1CC1CC(C)C)C1CC1)C)OC c1(NC(C2CN(Cc3ccc(CN(C)C)cc3)C2)=O)ncc(Br)cc1F Cc1cncc(C(=O)NCCCCC2CN(C(C3(CN(C)C)CC3)=O)CCO2)n1 C1(C(=O)NC23CC(C)(C2)C3)CC12CCN(C(C13CC(CO)(C1)C3)=O)C2 C(=O)(CC1=CCCCC1)NC(CC=C)CNC(=O)CCn1cnnn1 c1(C(=O)NC2C(NC(=O)C3=CCCOC3)CCC2)ccc2c(c1)COCCN2 N1(C(CN2CC(OC)C2)=O)CC2CC(N(C)C(C3CC3C(C)(F)F)=O)C1C2 C1(C)(CNC(CCN(CC)CC)=O)CCN(C(c2ccnn2CC#N)=O)C1 C1(CCC)CN(C(c2cc(C(=O)OC)cs2)=O)CCN1C(c1cccnc1Cl)=O N1(C(CN(C)C(N)=O)=O)CCCC(O)(CNC(C2(C)CCC(F)(F)CC2)=O)CC1 c1(C(CNC(=O)NC2CC3(C2)CC3F)O)ccccc1F C(=O)(CCC(C)(C)NC(c1cn(C)c(=O)n1C)=O)NCc1c(C)nn(C)c1 CCC(CC(F)(F)F)C(=O)N1CCC(NC(c2cnc(-n3cccn3)cn2)=O)C1 C(Cc1cc(F)cc(F)c1)N=c1[nH]n2ccnc2s1.c1nn[nH]n1 Nc1cc([N+](=O)[O-])ccc1C(=O)NC1CC(CNC(c2nsnc2O)=O)C1 N1(C(=O)CC2CC3CCC2C3)CC2CN(C(C3(Br)CC3)=O)CC(C1)O2 C#Cc1ccc(C(=O)NC(C)(C)C(N2CCC(O)(CC(C)C)C2)=O)cn1 C(=O)(C1CCCc2ncccc21)NC12C(CN(C(c3c(C)nn(C)c3Cl)=O)C1)C2 c1(C(N2CC(NC(C=CC(CC)=CC)=O)C3C2C3)=O)ccc2nncn2c1 Cc1cccc(C(=O)N(C)CCn2cc(CN3CC4CC4C3)nn2)c1Br C(C(N=[N+]=[N-])C(=O)N1CCCC12C(=O)NOC2)OCC.C1(C)(CO)CCCC1 C1(N(C(=O)CC(n2nc(C)cc2C)C)CC)CCC(NC(=O)CO)CC1 S(=O)(=O)(c1ccc2c(c1)CN(C)C2=O)N1CCN(CC)C(C)(C)C1 Cc1nc(NCc2ccc(Cl)c(C)c2)cc(=NCc2cnn(CC(F)(F)F)c2)[nH]1 C12(C(N3CCCC(c4cncn4C)C3)C)CCC(Nc3ccccc3)(CC1)CC2 C(=O)(NNC(=O)NC1CC(Cc2ccccc2)C1)c1ccc(C)o1 N1(C(CCSCCC)=O)CC2CCC2(CCNC(c2nccnc2C(N)=O)=O)C1 C1(OCC)CCN(C(=O)C=CC(N2CC(OC)(NC(=O)C3CC3)C2)=O)CC1C c1(C(=O)NC(C(=O)NCc2c(C)nc(C)s2)CCF)ccc(C)c(O)c1 n1(CC)cc(Cl)cc1C(=O)NCC(C1CCCC1)NC(=O)CC1CSC1 c1(C(=O)NCC2CC(COC)CN2C(=O)CCCC2CCC2)cc(Cl)cc(Cl)n1 C1(C)(N)CCN(N(C(=O)CCCNC(c2ccccc2)=O)c2cscn2)CC1.CC c1(C(=O)NC2CN(C(c3c(CCC)occ3)=O)C2)ccc(OC(F)(F)F)c(C)c1 c1(C(=O)NC2CCC2NC(=O)C(F)CC2CCCCC2)cnc2[nH]nnc2c1 C1(C(=O)NCCn2c(C)ncc2)CC(O)CN1C(=O)CCC1CCCCC1 C=CCCCCCC(=O)NC1CCN(C(=O)CCN(CC(C)C(C)C)C)CC1F c1(C(N2C(C)C(C(F)(F)F)OCC2)=O)cc2cccc(Br)c2cn1 c1(C(=O)NC2CCCC(C(=O)Nc3cnoc3)C2)cc(F)cc([N+](=O)[O-])c1 c1(C(N2C(CO)CC(NC(c3c(CC)ocn3)=O)C2)=O)cc(C)nc2ncnn12 N1(C(CN(C(C)=O)C)=O)CCC2(NC(c3ccc(F)cc3Cl)=O)CCCCCC12 CCC(CC(=O)N1CC2C(CN(C)C(c3cncc4c[nH]nc34)=O)C2C1)C(C)C N1(C(C=C(C)C2CC2)=O)CCC(C)(C)C1CC(N1CCCC1)=O.C1(N)CCC1 N1(C(C=CCCC)=O)CCC2(CCC(C(F)(F)F)N2C(C2C=CCC2)=O)CC1 n1(CCC)cc(C(=O)NC(C2COCCO2)C)c(C)n1 C1(C(=O)NC2C(C(C)C)N(C(C3CC(=C4CCC4)C3)=O)CC2)CN(S(N)(=O)=O)C1 c1(CCNC(C(CN(C)C)NC(=O)CN2CCCC2=O)=O)cccnc1O N1(C(CC(CC#C)c2ccccc2)=O)C2CCC1CN(C(=O)C1=CCCCO1)CC2 c12cc(F)c(cc1F)S(=O)(=O)N1CC(CC1=O)C2=O.c1(C(=O)OC)cn(C)cn1 Cc1cc2c(cc1CNC(=O)N(CCO)CC1CC1)CCO2 N1(C(c2c(C)ccnn2)=O)CCCC(CO)(NC(c2cccs2)=O)C1 Cc1noc2ncc(C(=O)NC3CC(O)(CNC(=O)C(C)Cn4ccnc4)C3)cc12 C1(OC)CC(CNC(=O)Cc2cscn2)N(C(=O)CCc2cnn(C)c2C)C1 C1(n2cc(-c3n(C(C)(C)C)ncc3)nn2)CN(C(=O)CCP(C)(C)=O)CCC1O Cc1nnc(NC(c2cc(N(C)C)cnn2)c2nnnn2CCCF)n1C O=C(CCCCCn1cc(-c2ccccc2)nn1)NC1CCOC1c1nc[nH]n1 c1(NC(C)CN(C)C)ccc(S(=O)(=O)NC2CC2CF)cc1C#N N#CC1(C(N2CC(CCCCNC(C3CC34CCCCC4)=O)C2)=O)CCSCC1 c1(OC)ccc(C(=O)NCC2CN(C(C3(C4CC4)CC3)=O)CC2C)c(OC)c1Cl C(=O)(C(Cc1ccccc1)CC(C)C)N1C2CN(C(C(CC)CCOC)=O)C(C2)C1 C1(C(=O)NCC2C(C)C2)CCC2(CC1)CCN(C(=O)C(c1cc(F)ccn1)=O)C2 N1(C(c2c(CC)occ2)=O)CC(C2(NC(=O)CN(c3ccc(Cl)nn3)C)CC2)C1 CCC(COC)C(=O)N1CCC(CC(=O)NC(C)CC(C)O)CC1 Cc1cc(C(=O)NC2CCC2NC(c2csc(Cl)c2Cl)=O)ncn1 CC(C)C(CC(=O)N1CC2C(C(N)=O)C2C1)NC(=O)C(C1CCOCC1)O C1(CNC(C2CC(OC)C2(C)C)=O)CC(C)CN(C(=O)CC2(OC)CCC2)C1 CC1CCCCC1(CNC(=O)CC1=CCCC1)NC(=O)C1=COCC1 Cc1cc(O)nnc1C(=O)NCCC1CN(C(C2CCC(C)CC2)=O)CC1C c1(C(=O)N(CCNCC2(CC(F)F)CCOCC2)CC2CCCC2)cccc(O)n1 C12(C(=O)NCCc3ccc(CN4CC(C)OCC4)cc3)CCCCC1OCC2 N1(C(C2(C(=O)NC3C(C)C3)CC=CC2)=O)CCC12CCC(O)CC2.C1C(=O)N1C(C)C C1(C2CC2)(CNC(C2CC(OCC)C2)=O)CCN(C(C2COC(=O)C2)=O)C1 C1(NC(CN(C(Cc2n(C)ccn2)=O)CCNCCO)=O)CCCCC1C#N N(C1CC2(CCN(c3ccc(C#N)nc3)C2)Oc2ccccc21)C(C=C(C)Cl)=O C(=O)(C(C)CC(N)=O)NC1C(CNC(c2c(C(C)C)scn2)=O)CC1 C1(NC(C(C(C)O)NC(=O)OC)=O)CN(C(=O)Cc2n[nH]c(=N)s2)CCC1(C)C C1(NC(C(c2n(C)ccn2)(F)F)=O)(CNC(=O)CC2CCC(O)C2)CCOCC1 c1(C(=O)NC(CNC(C2=CC(C)(CC)C2)=O)(C)C2CC2)ncc2c(F)cccn12 C12C3C=CC(C3)C1C(=O)N2.c1(COCCC#N)ccccc1F N1(Cc2cccc(C)c2)CCCC(NC(=O)CNC(=O)CC(C)(C)C)CC1 C1(NC(c2nnn(CC)c2C)=O)CC(NC(c2occc2Br)=O)C12CCC2 N1(C(C(C)(N(C)C(c2cnco2)=O)C2CC2)=O)CCCC2(CCC2)C1 c1(N(C(C#C)C)C)nnc(C(C)OCC)n1CC(=C)C C1(CC(=O)NCC2N(C(C3=CN3C)=O)C3C(C2)C3)CN2CCN1CC2 N1(C(c2nnnn2CCC)(C)NC(C(=C)C)C2CC2)CCc2ccccc2C1=O c1(C(=O)NCC(=O)NCC(CNC(C2(SC)CC(O)C2)=O)O)ccccc1Cl C(=O)(C1CCCc2nncn21)N1CCC(O)(CN(C)C(c2ccc(F)cn2)=O)C1 N1(C(C(CC=CC)CC)=O)CCC2CN(C(=O)C=Cc3scnc3C)CC12 c1(N(C(=O)Cn2cc(CCC(=O)O)nn2)CC)c(I)cnn1C.C1C(C)S1 CC(CC(=O)N1CCCC1CC(=O)NCCC1(C)N=N1)C(C)(C)C c1(OCCC#C)ccc(C(N2CCC(C)C2CNC(=O)CCOC2CC2)=O)cc1 C(=O)(CCCCC#N)NCC1CCC(C(N(c2ccccc2)CC)=O)O1 C(=O)(CC(F)(F)C(C)(F)F)N1CCC2(CN(C(C3C(CC)C3)=O)C2)C1 C1(OC2CN(C(=O)NCCNC(=O)COC3CCOCC3)C2)Cc2ccccc2O1 Cc1cc(C)c(C(N2CC(CNC(C3CCCC3)=O)C(C(F)(F)F)C2)=O)c(=O)o1 Cc1cc(C)c(OCC(=O)NC2(F)CCN(C(C3CCCCS3)=O)C2)c(C)c1 N1(C(c2c(C)n(CCNc3ccc(F)cc3)nc2)C)CCC2(CC(C#N)C2)C1 C1(NC(CC(C)NC(C)=O)=O)C=CCN(C(=O)Cc2ccccc2OCC#N)C1 C1(NC(CC=CC)=O)CC12CCN(C(c1nn(C)c(Cl)c1Cl)=O)CC2 CC1Oc2c(F)cccc2C1NC(c1ccc(C#N)cc1Br)=O C1(C(=O)NCC2CCCC2O)(CC)CN(C(=O)CC2(O)CCCC2)C1 C1(NC(c2cccc(CN3CCOC3=O)c2)=O)CCN(C(=O)CC2CC2)CC1O C1(C(N2CCC(OC)(CNC(=O)C(C(C)C)NC(N)=O)C2)=O)CC2(CCCC2)C1 CCC1=C(C(=O)NC23CC4CCC(C2C3)N4C(c2c[nH]nc2C)=O)SCCO1 N1(C(C(CC)OC)=O)CC2C(CN(C(=O)CC3CC=CCC3)C)C2C1 C1(C(=O)NCCC2(O)CN(C(C3(C)C=CCCC3)=O)C2)Cc2nccn2C1 c1cc2c(cc1-c1cc(N3CCCCC3)ccn1)CCCCC2 c1(CN2CCC(C(C(=O)Nc3nc(C)sc3)C)CC2)cc(F)ccc1[N+](=O)[O-] N1(C(c2c(CC)csc2)=O)CCCC12CCN(C(c1cscc1OC)=O)C2 C1(CCC)CN(C(c2c(C)cnn2C)=O)CCN1C(C1CC1c1ccccc1)=O C1(C(=O)NCC2CN(C(c3ncn(C)n3)=O)CC2O)CCCCNC1=O C#CCC(C)(C)C(=O)NCC1(C)CCCN1C(c1nc(C)ncc1Br)=O C(=O)(CCCCN1CCCC1)N(C)C.C12(c3nnnn3C3CCC3)CC(C1)N2 C1(NC(=O)Cn2ccc([N+](=O)[O-])n2)CCN(c2ccnc(CO)n2)CCC1CO C(=O)(C(C)CC(C)(C)C)NCC1N(C(C2N(C(C)=O)CSC2)=O)CCCC1 c1(C(=O)NC(CN(C(c2c(CCC)n(CCO)nc2)=O)C)C)cccn(O)c1=O c1(SC)nc(C)cc(=NCC2(C)CC2)[nH]1.C1(CC=O)CC2(CC2)C1 N1(NC(=O)Cc2cccc(F)c2)CCC12CN(S(=O)(=O)CC1CC1)C2 C1(C(=O)NC(C)CCNC(=O)C(O)Cn2cncn2)COC2COCC2O1 C1(CN(C)C(C2CN(C3CCC3)C2)=O)CCCN(C(C2(CF)CCC2)=O)C1 c1(C(N)=O)ccccc1NC(C1CCN1C(C1CC2CCC1C2)=O)=O Cc1[nH]nc(C(=O)NCC2CCN(C(c3cc(-c4cnn(C)c4)on3)=O)C2)c1F C(=O)(C(C)(C)C(N)=O)NCC1(C(=O)NC2C3CN(CC)CC32)CCCO1 C(N=c1[nH]c2c(c(=NC3CCc4cccc(N(C)C)c43)[nH]1)COCC2)C1C(C)CC1 Cn1nc(I)cc1C(c1nnnn1CCC1CC1)NCCCC1CC1(Cl)Cl C1(C(=O)NCCCN(C(C2CC2C(F)(F)F)=O)CC)CC2CC2C1 c1(C(=O)NCC(CC)NC(=O)Cc2cc(F)ccc2F)cnn2cccc(Cl)c12 c1(CN=C(NCCOC)NC(C)Cn2ccnc2)ccc(F)c(O)c1 N1(C(C(CCC)N(C)C)=O)CC2(CCN2C(=O)CCC2CCC2)C1 N1(C(C2C3CC(C)(C3)OC2)=O)CCCC2(C1)OCC(O)C2O N1(CC(=O)NCCCC)CC(NC(c2cnsn2)=O)CCC1C CC1CC(CNC(=O)CS(C)(=O)=O)CCN1C(C1CC2CCC(C1)S2)=O CC1(C)CNC(=O)CN1NCn1c(C)cnn1.c1(C)ccccc1 Cc1cc(C(N2CCC(F)C(NC(C3CC(Cl)(Cl)C3)=O)C2)=O)ccc1Cl C=CC1OCCCC1C(=O)NCCC1CCN(C(C2(C3CC3)CCCO2)=O)C1 CCCCC(CC)CC(=O)N1CCC(C)(C)C(C(=O)NC2CC(O)(CO)C2)C1 CCCCCC=NCCCN(C(=O)CCF)C O=C(CCC(F)F)NCCC1CCCN(C(c2cccc(OC(F)F)n2)=O)C1 c1(C(C(=O)NC2CCC(F)(F)CC2)N(CCCCCO)C)cc(Br)c([N+](=O)[O-])s1 c1(C(N2CCC(C(N)=O)C(C)(C)C2)C(=O)NC)ccc2c(c1)CC(C)O2 Cc1cc(C#N)cc(C)c1C(N1CCCC1C(C)NC(=O)Cc1n[nH]c(=N)s1)=O c1(C(=O)NCC(CC=C)NC(=O)C(C)(C#N)CC)coc2c(F)c(Cl)ccc12 CCC(CCCC(=O)OC)NCC1(O)CC2CCCC12 C(c1cc(C)cc(C)c1)=CC(=O)NC(CCN(C(c1c(CC)n(C)nn1)=O)C)C C#Cc1ccc(Cl)c(C(N2CCCC(CNC(=O)C(C#N)CC)C2)=O)c1 n1(CCNC(c2cnn(CC(C)(F)F)c2C2CC2)=O)c(=O)oc2ccccc12 N1(C(c2c(COC)scc2)=O)CCC(C)(CCNC(=O)C(CO)N(C)C)CC1 N1(C(=O)OCC)CCC(CO)(NC(=O)CC2CC2OC2CC2)C1.C1C(=O)N1 N1(C(C(=O)NC(C)Cc2ccc(F)c(F)c2F)=O)CCCC1C1OCCO1 C1(CNC(C=C(C)C(F)F)=O)CCC(CNC(=O)C=C2CCCCC2)CC1 c1(C(N2CCCC2(C)Cc2cc(Cl)cc(Cl)c2)=O)nc(Cl)ccc1C(F)F N1(C(C(CO)NC(c2ccc(CC)cc2)=O)=O)CCOC2CCCC12 Cn1nc(C(=O)NC2CC(C(=O)NCCC(N)=O)C2(C)C)cc1O n1(CC(N2CC(N(C(C(F)OC)=O)C)C3(C2)CC3)=O)nnc2ccccc12 N1(C(c2cc(C)cc(Br)c2)C(=O)N(C(C)C(=O)NC)C)CCC(C2CCOC2)CC1 Cc1cc(NC(=O)CCC2CCCO2)cc(CNC(c2coc(CC3CC3)c2)=O)c1 C(=O)(CC(O)C(C)(C)C)NC(C)CN(C(=O)Cc1ccccc1)C C1(C)(CNC(C2CC(OC)C2)=O)CCCN(C(=O)CCc2c[nH]c(=N)[nH]2)C1 CC1C(NC(c2cn(C(F)F)cn2)=O)CCCN1C(=O)CCC1CC1 CC1C(NC(=O)C(C)(C)C2CCCCO2)CCN1C(=O)CC(F)F CCC(CC)CC(=O)N1CC(CC(N2Cc3c[nH]nc3C2)=O)(OC)C1 N1(C(c2ccno2)=O)CCC2CCCN(C(=O)CCC3CCCCCC3)C2C1 C1(C)(OC)CC(NC(C2CCC(NC(c3cnn4c3CC4)=O)CC2)=O)C1(C)C N1(C(Cc2ccc(C)c(Cl)c2)=O)CCC2CN(C(=O)Cn3cnnc3O)CC2C1 C1(CC(=O)NCC2C=CCC2)(OC)CN(C(=O)CC2CCCCO2)C1 C(=O)(C(O)C(C)(C)C)NC1CC(NC(C(c2c(OC)cccc2)C)=O)C1.N1(C)CCCC1 C1(C#N)(C(=O)Nc2cccc(CNC(C(CCC)OC)=O)c2)CC12CCCC2 C1(C(CC)Nc2cc(C)ccn2)CCC(C2CCCCO2)CC1 Cc1ccnc(C)c1NC(C1CCC(NC(=O)C(C)Cc2ccccn2)C1)=O CC(C)(C)CC(=O)N(CCCO)CCN.N12CCCC(C1)C(C)(C)C2=O C1(C(=O)NCC2C3CN(C(=O)C=CC=C(Cl)Cl)CC23)CCCCCS1(=O)=O Cc1ccc(C)c(C(=O)NCCNC(=O)COc2ccc(F)c(Cl)c2)c1 N(C(=NCCSC1CC1)NCC1(C(C)(F)F)CCC1)Cc1nnn(C(C)(C)C)n1 C1(c2cn(C3C(NC(CC4CCC(C)O4)=O)CCC3)nn2)CC2(CCC2)C1 CCC(C)C(C)C(=O)NCC1(NC(c2occ(C)c2C)=O)CCCCC1C C(=O)(C1NCCc2cc(OC)ccc21)CCCCCCCCCC C1(CNC(=O)CCC2CCCC2)CC2CCC1N2C(=O)CCOCC(F)(F)F N1(C(c2ccc(C)[nH]2)=O)CCCC(C2CC2NC(=O)CCCCCn2cnnn2)C1 C12(CNC(C3(CF)CCN(C(CSCC#C)=O)C3)=O)CCCC1CCC2 C(=O)(CCCCCCBr)N1C(C(=O)NC(c2ccc(C#N)s2)C)COCC1 C1(C(=O)NC(C2CCOC2)(C)C)COCCC1NC(c1cccc(CO)c1)=O c1(C(N2CCCC(CCCNC(=O)COC3CC3)C2)=O)occ2c1CCOC2 c1(C(=O)NC2CC(CNC(c3c(C#C)c[nH]n3)=O)C2(C)C)c[nH]c2cnccc12 N1(C(C2C(C#C)C2(C)C)=O)CCC2(CCC(CNC(=O)Cn3ncnn3)O2)CC1 N1(C(CNc2ccn(-c3ccc(C)cc3)n2)=O)CCC2(O)CCOCC2C1 CCC(C)(O)C(=O)N1CCOC(CN(C(=O)CN2CCCS2(=O)=O)C)C1 C(CCCCC(=O)NC1CC1C)NC(C1C(C)CC1)=O O=C(N=c1cc(Cc2ccc(F)cc2)[nH][nH]1)c1cccc2c1COC2 Cc1nc(Br)cnc1NC(C1(F)CCN(C(=O)C(=O)C(C)C)C1)=O Cc1c(NCCCc2ccsc2)ncnc1N1CCC(CSC(F)F)C1 C1(NC(C(C)CC2CCC2)=O)CCC2(CCCN2C(=O)CC(C)(C)C(F)F)CC1 C(C)(C)(CN(C(=O)C(C)N(C(C1CC(F)C1)=O)C1CC1)C)OC CCCCCCC(C)C(=O)NC1CC(C)(NC(c2cncc(Cl)c2)=O)C1 N1(C(C2C(C(C)O)C2)=O)CCCC(C2(NC(C3(O)CCCCC3)=O)CC2)C1 Cc1nccc(C(N2CCC2CNC(=O)Cc2ccc(Cl)c(F)c2)=O)c1C.C1(C(=O)O)CCCO1 C1(NS(CC)(=O)=O)CN(C(=O)OC(C)(C)C)C2(CCC2)C1.C1C(=O)N1 CCCC(C#N)C(=O)NC1CCCCN(C(c2ccc(C(F)(F)F)nc2Br)=O)C1 N1(C(c2c(C)ocn2)=O)CCN(CCN(C)C(C2(C)CC=CCO2)=O)CC1 N1(C(=O)Nc2c(C)cccc2)C2CC1CN(Cc1ccnc(F)c1)C2 c1(C2CC(C(=O)NCC3CCC(NC(c4sccc4Cl)=O)C3)C2)ccccc1 C1(NC(CCC=C)=O)CC2CC(NC(C3CCCC34CCC4)=O)C2C1 C1(C(N2CC(CCC)N(C(c3csnc3Cl)=O)CC2)=O)CCCN2CCCCC12 c1(C(N2C(C(=O)O)C3(C2)CCCC3)=O)ccc2nncn2c1 N1(C(=O)CCOC2CC2)CCCC2(CCN(C(=O)CC3CC4CC4C3)CC2)C1 C(=O)(C1=C(C)N(C)c2nnnn2C1)N1CC(CNC(=O)NC(C(=O)OC)C)OCC1 Cc1nc(O)[nH]c1C(=O)NCC(C)(C)CN(C)C(c1ccc(Cl)o1)=O c1(NCC(c2ccccc2OC(C)C)N(C(C)=O)C)ccc2nnnn2n1 Cc1cnc(N2CCOC(C(C)NC(c3cc(C4CC4)on3)=O)C2)nc1O c1(C(=O)NC(C)CNC(=O)CCC2CCC2)cc2sccc2[nH]1 C(=O)(CCCC(=O)NCC(=C1CCSCC1)F)N1CC(CNC(CCCSC)=O)C1 c1(C(N2CCC(CNC(=O)N)C2)=O)ccc(F)c(NC(CCC)=O)c1F c1(C(=O)NC(C2CCOC2)CNC(C2(CC=C)CC2)=O)c[nH]nc1C1CCOCC1 N1(C(c2[nH]cc(COC)c2)=O)CCC(C(C)NC(c2cccc(SC)n2)=O)CC1 CC1CN(c2ncccc2S(=O)(=O)N2CCCC3(CCC3)C2)CC(C)(C)C1 N1(S(C(C)(C)C)(=O)=O)CC2CC1CC2NS(=O)(=O)CC1CC1 C#CCCC(O)C(=O)N1CC(C2(NC(=O)CCC3CC(F)(F)C3)CC2)C1 c1(C(=O)NCC(CCC)NC(C2COCCO2)=O)cc(F)cc(F)c1 N1(C(C(C=CC)O)=O)CCN(C(c2nc(C)ncc2Br)=O)CC(O)C1 C#CC1COCCN1C(=O)CCC(CC)NC(=O)CC(C)N(C)C N1(C(c2c(C)cc(F)cn2)=O)CCC(N(C)C(C2C(C)C2(F)F)=O)C2(CC2)C1 C1(NC(C(Cn2ccnn2)NC(CCC(C)N(C)C)=O)=O)CCCN(C)C1=O C12(C(N3CCC(CC#C)CC3)=O)CCCC1CCN2C(c1sncc1CC)=O N1(C(Cc2cc[nH]n2)=O)CCC(C)(C)C1NC(c1c(C)nccc1)=O C1(C)(C(=O)NCC2(NC(CCC(C)(F)F)=O)CCOC2)Cc2ccccc2C1 c1(NCCNC(=O)NCC)ccccc1S(C)=O C1(C(N2CCC(O)(CNC(=O)CCc3cc(Cl)cs3)C2)=O)CC2C(C1)C2(F)F c1(OC)ccc(OC)c(C(=O)NC2CCC(CNC(c3ccnnc3O)=O)C2)c1 c1(OC)ncccc1C(N1CC=CC1C(N1CCOCC1C(F)(F)F)=O)=O C1(C(N2CC3CC(CNC(c4ccc[n+]([O-])c4)=O)C3C2)=O)CCc2ncsc2C1 N1(C(C2CCN(CC)CC2)=O)C2CCC1C(C(=O)NC1CC1(C)C)C2 C(C)(CC(=O)NC1CCN(CCOC)C1)NC(COCC(=C)C)=O c1(CNC(C(=O)OC)COC(C)(C)C)cn(C)c2ccccc2c1=O C(CCO)(C(=O)NCC1(NC(c2cc(C#N)no2)=O)CC1)N(C)C c1(CC(=O)NC(C2CCN(C(COC(CC)C)=O)C2)(C)C)ccc(F)cc1F Cc1ncncc1C(=O)NCC1COC(CNC(C2CCCN2C2CC2)=O)C1 c1(OC)c(F)ccc(F)c1C(=O)NCC1CC1NC(C1(P(C)(C)=O)CC1)=O CC(C(C)(C)C)=CC(=O)NC1CCC1NC(=O)C(C)(Cl)Cl Cc1cc(C)n(CC(=O)NC2CCCC2(C)NC(=O)CP(C)(C)=O)n1 CN(S(=O)(=O)N1CCCN(CC2(C(=O)O)CC3CCC2CC3)CC1)C1CC1 C1(C(=O)NCCCN(C)C(C2CCCC2C(F)(F)F)=O)CCN(CC(F)F)CC1 CCC(F)(F)CCN=c1nc2scnc2c(NCC2(OCC)CCOCC2)[nH]1 O=C(CCCC(F)(F)F)NC1CC2CC1N(C(c1ccc3sncc3c1)=O)C2 C(=O)(CCS(C)(=O)=O)NCC(c1ccc(OC)cc1)N(C)C.C12CC1CNC2=O c1(C(=O)NCC2CCN(C(c3nnc(C)s3)C)C2)n[nH]c2c1COCC2 c1(-n2c(C(C)NC(=O)OC(C)(C)C)nc(CC(C)=O)n2)ccc2nc(C)[nH]c2c1 n12ccc(n1)NC(=O)NC1CC1C2.C1(CC)CCOC1CC1CC1 C1(CCNC(c2cccc(C)c2C)=O)CN(Cc2nc(C(C)C)no2)CCS1(=O)=O N1(C(Cc2cn(CC)nc2)=O)CCCCC(NC(c2nn[nH]c2Cl)=O)C1 C1(C(=O)NC(C2CCCC2)CNC(C2(CC(C)C)CC2)=O)CC=CC1 c1(C(=O)NC2C(C)CCN(C(=O)Cn3cccn3)C2)cc(F)c2c(c1)nnn2C C1(NC(=O)C(F)=CC2CC2)CN(C(C2CCC3(CCC3)O2)=O)C2CCCCC12 C1(C(=O)NC2CN(C(c3ccc(C(N)=O)s3)=O)CC2CO)CCCCC1C1CC1 N1(S(CC(=O)OCC)(=O)=O)CCC(F)(F)C(NC(c2cnn(CC)c2)=O)C1 N1(C(CC2C=NN(C)C2=O)=O)CCC(C2CCCN(C(=O)CC3CCC4CC34)C2)C1 C1(C(=O)NC(CC(=O)N(CC#C)CC2CC2)C2CC2)CCC(C)=C(C)C1 CC1CN(C)CCC1NC(c1ncoc1CNC(C1CCC(=O)N1)=O)=O C(C(F)C(=O)NOCC=CCl)C1CN(C(c2c(C(=O)OC)scc2)=O)C1 N1(C(=O)Nc2nnn(CS(C)(=O)=O)n2)CCC2(O)CCOCC2C1 c1(C(=O)NCC(=O)NCC(=O)Nc2c(OCC)n[nH]c2)ccc(O)c(C)c1 n1(CCC)cc(Cl)c(C(N2CC(=C(F)CNC(=O)C(C)(C)OC)C2)=O)n1 n1(CCC)c(C)cc(C=CC(=O)N(C2CCCC(NC(=O)C(C)(C)F)C2)C)c1C N1(C(c2cc(Br)cs2)C(=O)NC(C(=O)OC)CC(C)C)CCC(C#N)CC12CC2 C1(C(=O)NCC(N)=O)CC2(CC2)CN1C(c1ccc(OC(F)F)c(F)c1)=O C(c1ccc2[nH]ccc2c1)=CC(=O)N(CC(C)NC(CCC(C)OC)=O)C Cc1ccc(C(=O)N(C(C)(C(=O)N(C)CC2CCCCO2)C2CC2)C)c(C)n1 Cn1cc(C=CC(=O)NCCCN(C(C2(CCF)CCC2)=O)C2CC2)cn1 Cc1cc(F)ccc1CC(N1CCCC(CNC(C2CC(C(C)C)=NO2)=O)C1)=O C1(CNC(C(C(C)C)(C)C)=O)CN(C(c2ccnc(SC)c2)=O)CCC1(C)C Cc1cccc(OC(F)F)c1C.C(C(C)(C)CN)N(C(=O)OC(C)(C)C)C(C)C1CC1 C(=O)(C(C)S(C)(=O)=O)N(C1CCN(C(C2CCCC(OC)C2)=O)C1)CC O=S1(=O)CC2CC(C1)NC(O)C2N=c1ccnc(NCc2ccc(F)c(F)c2)[nH]1 CC1CN(C(=O)CC2(O)CCCC2)CC1CC(=O)NC1CC(=C2CCC2)C1 N1(C(CS(=O)(=O)NC)=O)CCN(C(C23CC(C2)C(C)O3)=O)CC1C CCCCC(CC)CC(=O)NCC1(F)CC(CNC(=O)CC2CCCC23CC3)C1 c1(C(N2CC(COC)(CNC(=O)CN(C3CCC3)C)C2)=O)cnn2c1CCC2 N1(C(C(C=C)C)=O)CCCC(C)(C(=O)Nc2cccc(O)c2)C1 C1CCCCCC(=O)N(C2CCC2)C(C)C(C)(C)C(=O)N1.C(C)(C)(C)OC(C)=O c1(C(C(=O)NC(C2CCCCC2C(F)(F)F)C)(F)F)ccc(F)cc1F c1(C(C)C)ncncc1C(=O)NC(C)CN(C)C(C1CCSC1)=O C1(NC(C2(COC)CCOCC2)=O)CCN(C(C2CCOC2C)=O)CC(C)(C)C1 Cc1nc(O)ccc1C(=O)NC(C1CCN(C(c2cccc(C3CC3)c2)=O)C1)C N1(C(Cc2ccc(C)s2)=O)CCC2CCC12CNC(=O)CN(c1ncccn1)C CCC(C)CC(C(=O)NCCn1c(O)nnc1O)NC(=O)C(=O)C(C)CC C1(CCNC(=O)C=Cc2cocn2)CN(C(C2CC(n3ccnc3)C2)=O)CCO1 Cc1nccc(C(=O)NCC2CC(C)CN(C(C3CCN3C(C)(C)C)=O)C2)c1Cl c1(OCCC)ccc(-c2cscc2C(=O)N(C(C)C)CC2CCNC2)cc1 Cc1cccc(C(N2CCCC2CNC(=O)CC2OCCCO2)=O)c1F c1(OC)ncc(C(N2CCC(O)C2C(=O)Nc2ccc(I)cc2F)=O)cc1F N1(C(=O)NCCc2cc(N)c(F)c(F)c2)CC(=O)NC2CCCCC12 N1(c2cccc(CC)c2)CCN(C2CN3CCC2CC3)NC1=O Cn1cnc(C(=O)NC2C3CC2N(C(c2cc(F)cnc2O)=O)C3)cc1=O C1(C)(C(=O)OC)COCCN1C(=O)Cc1ccnc(CCN)n1 CN1CC(NC(c2cc(Cl)c([N+](=O)[O-])[nH]2)=O)CC12CCCC2 Cc1cc(O)cc(O)c1C(=O)NC1CC2(C1)CN(C(c1ccncn1)=O)C2 C#Cc1ccc(F)cc1C(=O)NC(CC)(CC)CCNC(C1(COC)CC1)=O N1(C(CCNC(=O)OCC)=O)CCN(C(=O)NOCC(O)CO)C(=O)C1 c1(C(N2CCN(C(CCC(=C)Br)=O)C(C)C2C)=O)ccc2nc(O)oc2c1 c1(C(C)C)ccc(C(c2nnnn2C2CC2)NCC2(CO)CCC2)cc1 c1(C(N2CCC(N(C(c3c(OC)cccn3)=O)C)C2)=O)ccnc2cc[nH]c12 c1(C(N(C(C)C(N2CCCC2CN(C)C)=O)CCC)=O)ccnc(OC)n1 C1(N(C(CC(=C=C)C)=O)C)CN(C(C2(C#N)CC(=O)C2)=O)CC12CC2 N1(C(CC2(OCC)CC2)=O)CCCC2C1CCN2C(C1CCCC1C)=O c1(C(=O)OCCC(C)n2cccn2)ccc([N+](=O)[O-])cc1 C1(C)(C(N2CCCC(NC(C(COC)(C)O)=O)C2)=O)CCC(F)(F)CC1 C1(C(=O)NC(C(=O)N(CCCC)C(C)CC)(C)C)COCCC1C c1(C(N2CCC(N(C(c3cnc(CC)s3)=O)CC)C2)=O)cccc(C(C)C)c1F c1(NC(C2CC(NC(c3ccc(Br)c(Cl)c3)=O)C2)=O)nc(Cl)ccc1O n1(CCCCC(=O)OCCCN2CCC2)c(=O)oc2ccccc12 C12(CNC(=NCCCSC)NC(C3COC(=O)N3)=O)CC3CC(CC(C3)C1)C2 C(=O)(C(C)CCCC(C)C)NCC1=CCN(C(CC(C)n2ccnc2)=O)CC1 C(=O)(C(C)CC(C)C(C)=O)NC(c1cccnc1)C(=O)NC1(C#C)CC(F)(F)C1 c1(C(=O)NC2CC(C)N(C(=O)CCSC(F)(F)F)C2)ccc2oncc2c1 N(C(=NCCc1ccc(F)cc1)N1CCC(O)(C(F)(F)F)C1)Cc1nnc(C)s1 c1(C(=O)NCC23CC(NC(CCCCSC)=O)(C2)C3)cnc2[nH]c(O)nc2c1 CC(C)C.c1(C(CSC)NC(CN(CC(C)C)C2CCC2)=O)ccco1 c1(OC)ccccc1NC(=O)C(c1ccc(C2CC2C)o1)N(C)CC1CCCC1 N1(C(c2c[nH]c(=NC)s2)=O)CCC(C)C(NS(=O)(=O)CCCF)C1 N1(C(C(C)O)=O)CCOCC(C(c2ccco2)NC(=O)CC(C)(C)C)C1 c1(C2(C(N3C(C(N)=O)CC(F)C3)=O)CC2)c(Cl)cccc1Cl C=C1CC2CCC(C1)N2C(C1CCN(C(=O)CC(CC)C(C)C)CC1OC)=O N1(C(c2cc(Br)c(C)s2)C(=O)NCCCCCC)CCC(O)C(F)C1 CCCCS(=O)(=O)N1CCCC1C(N1CCCC1CNC(c1cnnc(Cl)c1)=O)=O N1(C(CC(=O)NCC)=O)CCCC2(C1)CN(C(C1(C)CCNC1=O)=O)CCO2 C1(SC2CCCC2)CCN(C(=O)C(C)(C)Cl)CC1C.c12nscc1C(=O)N2CC c1(C(=O)NC2C(NC(=O)Cc3ccc(Cl)cc3F)C2)csc2ccccc12 c1(CC(=O)NC(C(C)(C)NC(C(F)OC)=O)C)ccc2c(c1)CCC(C)(C)O2 CC(C)(C(=O)NCC1(O)CN(C(C2CC2CF)=O)C1)C(O)c1cc(Cl)cc(Cl)c1 C(F)(F)(CN=c1ccc(C(=O)OC)n[nH]1)c1c(OCCCC)ccc(C(F)(F)F)c1 Cc1cc(C(=O)NCC2CCN2C(=O)CCSCC(C)C)nn1C(C)C c1(C(=O)OCC)cc2c(s1)CCN(S(=O)(=O)CCc1cccc(C#N)c1)C2C c1(C(N2C(CN(C)C(C3CC34CCC4)=O)CC(F)C2)=O)ccnc2c1CCC2 C1(C(=O)NCC2C3N(C(C4C(C)C4)=O)C(CC3)C2)CC2(C1)CC(C)(C)C2 N1(C(c2c(CC)c[nH]c2)=O)CC(NC(=O)C(CCNC(C)=O)OC)CC12CCC2 C(=O)(C1CC(=O)c2c(F)cccc21)NCC1CCN(C(c2cc(OC)ns2)=O)C1 C#Cc1ccc(F)cc1C(=O)NCC1CN(C(C2C3CCC2(C)C3(C)C)=O)C1 c1(C(=O)NCC(C)C(=O)N(C)CC2(C)CCCO2)cc([N+](=O)[O-])n[nH]1 N1(C(c2cc(C)c(C)[nH]2)=O)CC2CC3CC2C1C3NC(=O)C(C)SC(F)(F)F C(=O)(C1CCc2ccccc21)NC1CC(C)N(C(=O)C(C)Cc2ccccc2)C1 N1(C(CC2C(C)CCN(C(=O)COCC3CC3)C2)=O)CC2CC(C1)C2(C)C N1(C(C(C(CC)C)NC(c2cc(CO)on2)=O)=O)CCC2(CCOC2)C1 c1(C(N2CC(CC(=O)Nc3cc(OC)ncc3)OCC2)=O)cc(O)cc(Cl)c1 N1(C(C2N(C(C(C)NCc3cc[nH]n3)=O)CC(C)C2)=O)CCC2(CCOC2)CC1 c1(C(=O)NCc2c(C)occ2)ccc2c(n1)CN(C(C1CC(C)N(C)C1)=O)CC2 Cc1cnc2c(C(=O)N(C3CN(C(c4cc(C#N)cs4)=O)CC3O)C)cnn2c1 N1(C(c2c(OC(C)C)nccc2)=O)CC2CCN(C(=O)Cc3nc[nH]n3)C(C2)C1 C1(CNC(c2ccc(Br)cn2)=O)COCCN1C(=O)CC1C=CCC1 N12CC(C)CC1c1ccc(cc1)-c1cscc1C2=O.COC N1(C(CCCCC)=O)CCCC2(C1)C(NC(c1ccc(C)cc1)=O)CCN2C c1(CC(=O)NCCOC2CCN(C(C(CC)n3cncn3)=O)C2)c(C)noc1Cl C1(F)(C(=O)NCC2CCC(=O)NC2)CCN(C(c2cc(F)ccc2I)=O)CC1 C1(NC(c2c(C)cccc2N)=O)CC2(CCCCN2C(C2CCCC(O)C2)=O)C1 c1(C(=O)OCC)noc(CC)c1Sc1cncc(C(F)(F)F)n1 O=C(C1CCCn2cnnc21)NCC1C=CCN1C(c1nc(Cl)ccc1F)=O Cc1cnc(COCC(=O)NCC2CC2CNC(c2[nH]cnc2C(C)C)=O)o1 N1(C(C(c2ccc(CC)cc2)(C)C)=O)CCCC2(NC(=O)C(N)=O)CCCC12 C1(CNC(CC(CC)(C)C)=O)CC2(CCOCC2)CN1C(c1cnc(O)o1)=O c1(C(=O)NC2C(SC)CN(C(c3cc([N+](=O)[O-])c[nH]3)=O)C2)ccc(F)c(C#N)c1 C=Cc1ccc(NC(N2CCC(C(=O)OC(C)(C)C)C(C)C2)=O)nc1F C1(CCNC(C=Cc2ncc(C)[nH]2)=O)CN(C(c2cscn2)=O)CCCO1 C(=O)(C(F)(F)CNC(c1cc(CNC(=O)CC2CC=CCC2)[nH]n1)=O)OC CC1=C(C)CN(C(c2sccc2CNC(c2ccn(C(F)F)n2)=O)=O)C1 c1(C(N(C(C)C)CCN(C)C(C2(O)CCCN(C)C2)=O)=O)c[nH]c2cccnc12 C=C(Cl)CCC(=O)N1CC2C(CN(C)C(c3cnoc3C3CCC3)=O)C2C1 c1(C(N2CC3(CC(NC(C(C#C)(C)C)=O)C3)C2)=O)cc(Br)c2[nH]c(C)nc2c1 c1(CN=C(NCC2(F)CCC2)NCc2ccco2)nnc2cccnn12 C(=O)(C1=CC2CCC(C1)C2)N1C(C(N(C)CCc2nccs2)=O)CCCC1 CCCCS(=O)(=O)NCC(=O)Nc1cc(NC(c2ccccc2OC)C)n(C)c1 C=C(C)CC(C(=O)NCc1cc[nH]c1C(N1CCC(C)(OC(C)=O)C1)=O)OC N1(C(CC(C)(C)OC)=O)CC(NC(=O)C=CC2CCOC2)CC(C)C1 C1(C(=O)NC(CC)CO)CN(C(=O)CS(=O)(=O)Cc2ccc(Cl)s2)CCC1O N1(C(c2c(C)ccnc2)=O)CCC2CCN(C(=O)C3=CCCCC3)CC2C1 C12(CNC(C(n3c(C)ncc3)C)=O)CCCC1N(C(c1cscn1)=O)CC2 CCCC(C(=O)NCC#CCNC(C1(n2cccn2)CCC1)=O)S(N)(=O)=O C(CN=c1[nH]c(=NCCCn2cnnn2)[nH]c2c1CCC2)OCC(=C)C Cn1ncc2c(=O)n(CCC(=O)N3CC(CCNC(=O)C(C)(F)F)C3)cnc12 N1(C(C(CC)C)=O)CC(CO)C2(CCN(C(=O)Cc3c[nH]nc3O)CC2)C1 c1(C(N2CCC(NC(C(C=C)O)=O)C2)=O)ccc(-c2ccc(F)cc2)n1C C1(CNC(C2N(C(CCSCCC)=O)CCC2C)=O)CCCC(C)CC1 c1(NC2CCC3(CC(OC)C3)CC2)nc(=NC2CC(F)(CO)C2)[nH]c2c1CCC2 c1(C(=O)NCCC(=O)NC(C)C)cc(Br)cc2nn(C)cc12 N1(C(CCc2ccn(C)n2)=O)CCCN(C(=O)CCC2CCC(=O)N2)CCC1 C(c1cc2ccccc2o1)=CC(=O)NC1CCCC(NC(C(C)(C)C(N)=O)=O)C1 c1(C(=O)NCC2CC(C)N(C(C3CCC3)=O)C2)nc2n(c1Cl)CCCC2 n1(CC(=C)C)nnnc1C(c1cccs1)Nc1cnn(Cc2nccs2)c1 c1(CC)[nH]c(C(=O)OC)c(C)c1C(=O)N.C1(C(=O)OC)CCC2(CC2)CO1 CCCCCC(C)(CC)C(=O)N1CC=CC(NC(=O)CSC(C)(C)C)C1 C(=O)(CC(P(C)(C)=O)C(F)(F)F)NCCC1N(C(C(C)O)=O)CCC1 Cc1ccc2c(C(=O)NCC(C(C)C)NC(C34COCC3C4)=O)coc2c1 C(=O)(C1=CCCOCC1)N(CC(CN(C(=O)C(C)Sc1nncn1C)C)O)C Cn1cc2c(CN3CCC(O)C(C(=O)Nc4cccc(Cl)c4F)C3)cccc2n1 Cc1cc(C(=O)N(CCCn2cc(-c3nc(C4CC4)cs3)nn2)CCO)sn1 O=C(CN=c1cc[nH]cc1)NC1CCCC(NC(=O)C(F)(F)C2(O)CCC2)CC1 Cc1c(C(=O)NC(C2CCCN2C(=O)C(C)SC2CC2)(C)C)cnn1CCO C=C(C)C(C)(O)C(=O)NC1CC(C)N(C(C2CCCCNC2=O)=O)C1 c1(NC(c2cc(-c3ccccn3)c[nH]2)=O)cccc(C(F)(F)F)c1 Cc1cc(C(=O)N(C)CC2(O)CN(C(=O)CC3CCCC(C)C3)C2)oc1C(=O)O N1(Cc2ccc(C)cc2Br)CCC2(CC1)CC(NC(=O)Cc1c(Cl)cccc1Cl)C2 c1(C(=O)NC2C(OC)CN(C(=O)C(C)c3cncs3)C2)nn2c(c1C)OCCC2 c1(OC)cc(C(N2CC3CC2C3NC(=O)C=Cc2ccco2)=O)ccc1O C1(C(=O)NCCNC(=O)NC)CCCN(C(c2ns[nH]c2=O)=O)C1 c1(CC(=O)NCCCN(C(c2nnn(C)c2N)=O)CC)cc(F)ccc1OC CCCC(CCC)CC(=O)N1CCC2CCC(C1)S2 C1(C(NOCCCC#C)=O)CC2(CC2)CN1C(c1ccc(=N)[nH]c1)=O N1(C(c2ccc(Cl)c(I)c2)=O)CCC12CCN(C(C1(O)CCCCCC1)=O)CC2 C1(C(=O)NC(c2ccnn2C)CC)CC(=O)CN1C(c1csnc1Cl)=O c1(C(N2CCC(O)CC23CC3)=O)[nH]cnc2nc(-c3ccccc3)cc1-2 C1(CNC(c2nn(CC)nc2C)=O)CC(F)(F)CN1C(c1csc(C(=O)OC)n1)=O c1(CC(=O)NCCC2(NC(=O)C(O)CN3CCCC3)CCCC2)cccc(O)c1 C(=O)(CCN(OC)C(=O)C(C)CN(C)CC1CC1)N1CCC(SC)C1 N1(CCNC(C(=O)N(CCCOc2cccc(F)c2)C)=O)CCC(O)CC1 C(=O)(C(C)C1=CCCC1)N(C1CCCN(C(Cn2ncc(C#C)c2)=O)CC1)C C(=O)(C1=C(C#N)CCC1)NC(C1CN(C(=O)Cc2ccc3scnc3c2)C1)C C(C)(C)(CC(=O)NCCC1CN(C(C2(O)CCC2)=O)CCO1)OC c1(C(N2CCCC(CN(C(c3c(C)scc3)=O)C)C2)=O)ccc2c(c1)C(C)CO2 C(=O)(C1=CCCCO1)NCC(CC(=O)N1C(CNC(C)=O)CCC1)O C(C(C)(C(=O)NC(C1NC(=O)NC1=O)C)NC(c1cc(C)co1)=O)SC C1(CC(=O)NCC(C2(O)CN(C(c3cc(C)[nH]n3)=O)C2)(C)C)SC(=N)NC1=O Cc1ncnc(C)c1C(=O)NC1CCC(C(=O)NC2CCCC3(C2)N=N3)C1 CC1CCC(CO)N1N1CCN(c2cnccn2)CC1 N1(C(c2c(C(C)C)n[nH]c2)=O)CC2CCCC(NC(C3OCC3(C)C)=O)C2C1 Cc1nc[nH]c1CC(O)C(=O)NCC1C=CCN1C(=O)C=CC(C)(C)C C(=O)(CCCCCCCCCO)N1CCC(NC(CC=CC(C)(C)C)=O)C1 C1(NC(COCCN(C)C)=O)CC2(C1)CC2NC(=O)C(C)(C)c1cccnc1 C1(CCOC)CN(C(C(=O)NCCCC2CC2)C(C)c2cccc(Cl)c2)CCN1C c1(C(=O)OC)cccc(C(N2CCC(CF)(NC(=O)CC3CCC3)C2)=O)n1 C1(N(C)C)CN(C(=O)C=CCC(=O)CC2(O)CCC2)C1 CC(C)C(C(=O)N1C(CO)CCCC1C)C(C)NC(c1cncc2[nH]ccc12)=O C1(OC)CN(C(c2ccco2)=O)CC1NC(C1CCC(C(C)C)CC1)=O C#Cc1ccccc1CC(=O)NCC(CCC)C(=O)NCC1COC(C)(C)C1 N(C1CCOc2ccc(Br)cc21)S(=O)(=O)c1ccc(Br)cc1F C12(C(=O)NCCC3(NC(c4cnn(CC5CC5)c4)=O)CCC3)CCC(CC1)CC2 C1(C(=O)N(C(CO)C(C)C)C)(CC)CCCN(C(=O)CN2CCNC(=O)C2)C1 Cc1nc(O)ccc1C(=O)N(CC(C)CNC(c1cccc(O)n1)=O)C C(CCC(C)(C)C(=O)NC1CC(C(N)=O)C1(C)C)NC(C1N(C)CCCCC1)=O C(C(=O)NC1CC(C)(NC(=O)C(C)CSC(F)(F)F)C1)(C(C)C)NC(=O)OC c1(C(N2CC(CC)N(C(C3CCC3CF)=O)CC2)=O)cc2c(s1)CCOC2 Cc1c(CNC(C2(C)CCCC2)C(C)C)cnn1-c1cccc(Cl)c1 Cn1[nH]c(=NC(=O)C(Cc2cncs2)Sc2ccccc2Cl)cc1Cl CC1CCCCC1(C)C(=O)NCC1CC(CNC(=O)Cc2c[nH]nc2O)C1 C1(NC(CC2(C=C)CN(C(C3CCC3(F)F)=O)C2)=O)CCN(C)CC1C#N N1(C(C=C(NC(C)=O)C)=O)CC2CC1CCC2NC(c1ccc(SCC)cc1)=O c1(C(=O)NCC2N(C(c3n(C)ccc(=O)c3)=O)CC=C2)[nH]nc2c(Cl)cccc12 C=C(C(=O)N1CC2CC2(C(=O)NCCC(C)(C)O)C1)C(F)(F)F C1(CCNC(=O)Cc2cncn2C2CC2)CCCN(C(c2c[nH]nc2C(=O)O)=O)C1 CC(C)(CC(=O)NCC1COC(C)(C)CN1C(c1ccc(N)cn1)=O)CC(F)F CC1C(O)CCN1C(=O)CC1CCCCN1C(c1ccc(CO)cn1)=O C1(NC(C2(C)CN(C(C(C)NC(C)=O)=O)C2)=O)CN(C(C)C)CC1C c1(C(=O)NC(C2CCN(C(C34CCC(C)(C3)OC4)=O)C2)C)cc2c([nH]1)CCCC2 Cc1ccc(C(=O)NC(C)(C)CCNC(C2(c3cccs3)CCCC2)=O)c(C)c1 C(=O)(C(Cc1ccco1)NC(=O)CCN(C)C)N(CCCCO)CC Cc1nn(C)cc1CCC(=O)NC(CNC(=O)CN1CC2CC2C1)C(C)C C(=O)(C(C(C)C)NC(C)=O)NCC(CC)NC(=O)CC(CC)c1ccc(Cl)cc1 c1(C(N2CCN(C(c3c(CC)scn3)=O)C(C)C2)=O)cncc2nc(C)[nH]c12 Cc1cc(N)cc(C(N2CC(C(C)NC(=O)CCc3cccnc3)C2)=O)c1F C(C)(CC(=O)NC1C=CC(CC(=O)NC(C)C(C)n2cccn2)C1)OC N1(C(C2C3CC4C(C3)C24)=O)CCC2CN(Nc3cc(CC)nc(C)n3)CC12 C1(C(=O)NC(CCC)(C)CO)CN(C(=O)C(=O)N(C)C)CC(C)(C)C1 c1(CC2(C(=O)NCC(C)(C)CNC(C3CCC4CC34)=O)CC2)cccc(Cl)c1 c1(C2(NC(C3C(=C)C3)=O)CC2)nccc2ccccc12 Cc1nn(C)c(C(=O)NC(C)CNC(=O)C(c2ccc(F)cn2)(F)F)c1[N+](=O)[O-] Cc1cc(CC(=O)NC23CC(NC(=O)Cc4cc(C)on4)(C2)C3)cc(F)c1 C1(C(N(CC(=C)C)CC)=O)CC2CC1CC2NC(=O)CNC(=O)OC C1(C(N(C2(C#C)CCC2)C)=O)CC(C)(C)CCN1C(=O)C(O)CCNC(=O)C1CC1 C1(C(N2CC(C)C(N(C)C)C2)=O)CC2CN(C(=O)CSC(F)F)CC2C1 N1(C(c2ccc(N(CC)CC)cc2)=O)CC2CCC2(NC(C2CC(O)C2)=O)C1 C1(CNC(C2OCCN(C)C2)=O)COCCN(C(c2cc(Br)oc2Cl)=O)C1 C1(NC(C(n2cc(CC(C)(C)NC(C(C)N(C)C)=O)nn2)C)=O)CCCC(F)C1 C(c1cc[nH]n1)=CC(=O)NC(C(N1CCC(n2ccnc2)C1)=O)c1ccoc1 O=C(C1=C(Cl)CC1)NC(CO)C(=O)NCc1ccc(CO)cc1 C=CC1(CC(=O)NCC2CC2C(=O)OC)CN(C(=O)CC2CCCN2C)C1 c1(C(=O)NCCCN(C(C2CC2CF)=O)CC)cc2n(c1)CCCC2 C1(NC(c2c(SC)cnn2C)=O)CCCC(NC(c2cc(C(F)F)no2)=O)CC1 c1(C(N2CCC(C(c3ccccc3)O)CC2)=O)cc(Br)ccc1Cl CC(C(O)C(F)F)NC(=O)CC1CCCC1NC(c1cc[nH]n1)=O CC1CC(NC(C2CCC(CS(=O)(=O)N(C3CCCCC3)C)C2)=O)CC(C)O1 C(=O)(CC1=NN(C)C(=O)C1)NC(CCC(=O)N(CCCCO)CC)C(C)C c1(COC)cccc(CC(=O)NC2CC(NC(=O)C(C)CC3CCC3)C2)c1 CCC(C)CC(C(=O)NC1CC(CO)C1)NC(c1cocc1C)=O C(CCN(C)C(c1ccnc(C(C)(C)O)c1)=O)(C(C)(C)C)NC(CCC#C)=O c1(C(N2C(C)CC(CNC(=O)C=Cc3cscn3)C2)=O)cc(=N)[nH]c(=N)[nH]1 C12(CNC(c3cc(C)ns3)=O)CCC1CN(C(c1cc(C)n(C(C)C)c1C)=O)C2 C1(C(=O)NC2(CC=C)CCN(C(=O)C=CC(=O)N(C)C)C2)CCC2CC2CC1 C1(C)(C(=O)NCC23CC(NC(C=Cc4ccc(C)o4)=O)(C2)C3)CCS(=O)(=O)CC1 c1(C(=O)OC)ncc(NC(CC2(C3CC3)CC2)=O)cc1F.C12(O)CC(C1)NC2 C#CCCCC(=O)N(c1ccccc1C(=O)OC)CCNC(=O)C(CC)OC CCCCC(C)(F)C(=O)NC(C)C(=O)NC(c1cnc[nH]1)C c1(-c2nc(C(C(C)C)O)nn2C(C)C2CC2)c(C(F)(F)F)cccc1Cl c1(C(=O)NC(C(C)NC(C2C(COC)C2)=O)(C)C)oc2ccc(Cl)cc2c1C N=c1[nH]c(Cl)c(Cl)cc1C(N1CCCC(CNC(=O)CC2C=CCC2)C1)=O C1(OC)CN(C(=O)CC(C)(C)OC)C(C)(CNC(=O)CCn2cnccc2=O)C1 Cn1c(C(N2CC=CC(CNC(=O)C=C(Cl)Cl)C2)=O)cc(Cl)c1Cl N1(C(CP(C)(C)=O)=O)CC(C2CN(C(=O)CC3CCC34CCC4)C2)C1 c1(CC)cc(C(N2CCCC(C)(NC(=O)C(C)n3cccn3)C2)=O)ccc1OC C1(CCOC)(SC(C)C)NC(=O)N(CC(c2ccc(F)cc2)=O)C1=O c1(C(=O)NC2CCC(NCc3cncc(C#N)c3)C2)ccnc2c1OCO2 N1(C(C2N(C(C)=O)CCCC2)=O)CCN(C(=O)CCN2CCN(C)CC2)CC1C c1(C(N2C(C(C)(C)NC(C3C4COCC34)=O)CCC2)=O)cc(Cl)c(F)cc1O N1(C(N2CCCC(C)(C(F)(F)F)C2)=O)CCc2sccc2C1 CC(CCCCNC(=O)C(C1(O)CCOCC1)(F)F)NC(=O)Cc1cnns1 Cc1cc([N+](=O)[O-])ccc1N(CCCN(C(=O)CCCCO)C)C C12CCCN(C1)C(=O)Nc1csc2n1.c1(C(COC)=O)nncs1 N1(C(C2(NC(N)=O)CC2)=O)CCN(C(C2CC2C2CCCC2)=O)C2(CCC2)C1 C1(NC(c2cccc(C(N)=O)c2)=O)CC2CC(NC(C3(F)CCCC3)=O)C2C1 c1(C(=O)NC2CN(C(C(C=C)(C)O)=O)CC2O)cnn2ccncc12 N1(C(C(CCC)O)=O)CCCN(C(c2cccc(Cl)c2OCC)=O)CC1C c1(C(=O)NCC=C2CCN(C(c3c(C(=O)OC)csc3)=O)CC2)cc(Cl)cc(Cl)n1 c1(C(N2CCC(NC(C3CC(F)C3)=O)C2)=O)cncc(C2CC2)c1 CC1(CNC(=O)CSCC(c2ccccc2)=O)CCN(C(=O)C(F)CC2CC2)C1 N1(C(CC2CCN(C(c3c(CC)cco3)=O)C2)=O)CCC(F)(CC)C1 C(=O)(CCCC(F)(F)F)NC1CC(C)N(C(c2cc3occc3s2)=O)C1 C1(CNC(Cc2cc(C)sc2)=O)CN(C(=O)CN2CCCC(CO)C2)CCN1C CC(C)CCC(C)NC(=O)C(=O)NCC1CCN(S(C)(=O)=O)C1 C(=O)(C(F)(F)CCn1ccnn1)NC(C(C(C)C)NC(c1ccn(C)c1)=O)C c1(CC(=O)NCC(CC)(C)NC(C2CC23CC(F)(F)C3)=O)c(C)nc(O)nc1O c1(C(=O)NC(C2(O)CCN(c3nc(C4CC4)ns3)C2)C)cn2ccsc2n1 N1(C(C(C(=C)Cl)(C)C)=O)CCC2CCN(C(c3ccn4c(C)cnc4c3)=O)C2C1 c1(C(=O)OC)cc(C(=O)NC2CCC(N(C(=O)C(C)N3CCC3)C)CC2)c(C)[nH]1 c1(NC(=O)NC2C(C#N)CCC2)c(-c2cccc(Cl)c2)cccc1F c1(OC)ccc(NC(C2(C3CCCN3C(=O)CNCCCN=[N+]=[N-])CC2)=O)cc1 CC(C1=CCN(C)CC1)NC(C1CC2CN(C(=O)C#CC(C)(C)C)CC2C1)=O CCCCC(C(=O)N(C1CCCCCC1)CCNC(C1CC=CCO1)=O)C(C)C C(=O)(C1CCCn2ccnc21)N1CCC(OC)(CNC(=O)CNC=O)C1 N1(C(CC(C)F)=O)CCOC(C(=O)N(C2CCCCC2O)C)CC1 C1(Cc2c(C)noc2C)CN(C(C2CC3CCC2C3)C(=O)NC2CC2)C(C)CO1 S(=O)(=O)(c1ccc2[nH]c(=NCC(F)F)sc2c1)N(CCC(C)O)C Cc1cccc(C2=CCN(C(C3CC4CC4N3C(=O)COC(C)(C)C)=O)CC2)c1 C1(CNC(c2c(CC)noc2C)=O)CCCCCN1C(C1CCCOC1)=O C(C(=O)NC(CC(C)C)C(=O)NCC1CCCCCC1)(C(C)(C)C)OC CC(C)CC(C)(C)C(=O)NC(C)C(C)NC(c1ccc2nn[nH]c2n1)=O C1(F)(CNC(C(=Cc2ccco2)C)=O)CCN(C(=O)Cn2ncn(C)c2=O)CC1 N1(C(=O)CO)CCC2(C=CCO2)CC1.n1(CC=O)ccc(C2CC2)n1 C1(O)(C(=O)NCc2ccsc2)CCN(C(C2CCC(F)(F)C2)=O)C1 c1(NC(C(N2CC(OC)C(c3ccncc3)C2)=O)=O)cc(F)ccc1C C1(C(=O)NCc2nnc(CO)s2)CCN(C(=O)CCCCn2cc(CO)nn2)CC1 c1(CCC(=O)NCCC2CCCN(C(C3C(C=C)C3)=O)C2)c(C)ncnc1O c1(C(=O)NCC(C)CNC(C2(O)CCC2)=O)cccc(C2CC(F)(F)C2)c1 CC1CCC(C(N2CCC(N(CCO)C(C3CNC(=O)N3C)=O)CC2)=O)C(=O)N1 C1(C(C)C)CCCN(C(=O)Nc2cn(CC(N)=O)nn2)CC1 Cn1nc(C(=O)NCCC2(O)CN(C(=O)CC3CCC4CC34)C2)cc1Cl C12(C(=O)NCCOCCN(C(=O)C(C)(C)C3CC3)C)CCC(C)(CO1)C2 c1(C(N2C(C)C(NC(=O)C(O)Cn3cncn3)CCC2)=O)ncnc2c1CCC2 C1(C(N2CC(C=C)(CC(=O)NCCC(O)C(F)F)C2)=O)CCCCCN1C C#CC1(C(N2CCCC(CC)CC2)=O)CCN(C(c2ccsc2)=O)C1 C(CCCC(=O)N1CC(C(=O)N(CCCO)C(C)C)C1)OC c1(C(=O)NCC(C)N(CC(N)=O)C)ccc(C(F)(F)F)o1 N1(C(c2c(C)n(C)nc2)=O)CCCC(C)C1CCNC(=O)C=C1CCN(C)C1 N1(C(c2ccn(C(F)(F)F)n2)=O)CCC(n2cncn2)C1 C1(C(=O)OC)CC12CCN(N1CCN(Cc3ccccn3)CC1CO)CC(C)(C)O2 C12(C(N3CC(CCCCNC(=O)CCCC4CCOCC4)C3)=O)CC1CCC2(F)F c1(C(N2CC(O)(CN(C(C(=O)OC)=O)C)C2)=O)cc(F)ccc1OCCN(C)C CCC(C)(C)C(=O)C(=O)NCC1(C(=O)NCC(O)C(C)O)CCCC1 c1(CCC(=O)NCC2CC(O)CN2C(C2CC3CC2C3)=O)c(Cl)cccc1Cl c1(C(=O)NC2CC(NC(C(CCC)CC)=O)C(O)C2)cc2[nH]nnc2cc1OC N1(C(C(C=C)O)=O)C2COCC1CC(NC(=O)CC1CC(SC)C1)C2 N1(CC(N2CCN(C(c3c(C)nncc3)=O)CC2)=O)CC(=O)N(C)C1=O Cc1noc(C)c1NC(C1C2CC1N(C(c1cccc(CO)c1)=O)C2)=O c1(OCC)ccc(C(=O)NCCCCCCNc2ncnc(O)c2Br)cc1C CC1(C)CCOC1C(=O)NCCC1CC(NC(C2CCCC2(F)F)=O)C1 c1(C(=O)NC2CCN(C(C(=O)NCC)=O)C2)ccc(F)c(Cl)c1N N1(C(C2C3(CCN(Cc4c(Cl)ccc(C#N)c4)C3)C2)=O)CC2OCCOC2C1 C(C(C)(C)CCl)(c1nnnn1C(c1cccc(F)c1)C)NCC(CC)(CC)SC C1(C(=O)NCC(c2ccc(Cl)cc2)C)CC2CC2N1C(C1CCC(F)C1)=O CC1C(C)N(C(c2nn(C)cc2N)=O)CCN1C(C1CC2(CSC2)C1)=O CC(C)CCC(C(=O)NCCc1ncccn1)NC(c1cc(F)cc(F)c1)=O C12(NC(c3ccc(C)nn3)=O)CCOC(CNC(c3csc(C(C)C)n3)=O)(C1)C2 C(=O)(C(CO)C(F)(F)F)CCC.N1(C(CNC2CC2)=O)CC(=O)NC(C2CC2)C1 CC(C)C(CC(=O)NC(C)(CO)C1CCCC1)NC(=O)Cc1cc[nH]c1 N1(C(C(C)NC(=O)NC)=O)CC(C)(C)CC1CNC(c1ccc(CO)c(F)c1)=O Cc1ccc(COC(F)F)nc1Br.c1(OCC(CS)O)ccc(C(C)C)cc1 C12(CNC(c3cccc(Cl)c3)C)CC(C)(C1)OC2C(=O)O c1(C(N(C2CC(CC(F)(F)F)C2)CCNC(C2(SC)CC2)=O)=O)ccnc(S)c1 N1(C(CCCC(C)N(C)C)=O)CCC2CN(C(=O)CC3CCCS(=O)(=O)C3)CC12 C12(NC(c3c(Cl)nc(OC)s3)=O)CCN(C(=O)Cn3ccc(O)nc3=O)CC1C2 S(=O)(=O)(c1ccc(-c2nnc(C(F)F)o2)cc1)NC1CCC(C)CC1 c1(N2CCCC3(NC(C(C(CC)C)C)=O)C(C2)C3)ccc2c(n1)CCCC2=O c1(C(C)C)n[nH]cc1C(=O)NCc1n[nH]cc1C(N1CCC(CN(C)C)C1)=O N1(C(C(=O)N(C2CCN(C(=O)OC(C)(C)C)C2)C)C)CC=CCC1 CC(C)C(C(=O)N(C1CC1)C1CC1)NC(=O)OC(C)(C)C.C12CCCN1C2=O N1(C(C(COCC)N=[N+]=[N-])=O)CCC2(CC1)CC2C(=O)NCc1ccncc1F N1(C(c2c(CC)ncnc2)=O)CC2CCC(CNC(=O)C(C(C)C)N(C)C)(C2)C1 c1(OC)ccc2cc(-c3nn[nH]n3)oc2c1.n12nc(c(C)n1)CNC(=O)C2 C1(NC(C2CC=C(C)CC2)c2nnnn2C2CC2)CC2CCC(C1)C2 C1(C(N(C(C)CNC(c2cc(C3CCC3)no2)=O)C)=O)COCCN1CC(F)F N(C)(C(=NCC1=C(C)OCCS1(=O)=O)NC(C)C)CCc1cc(OC)c(C)cc1 C(C(=O)NNC(=O)C1CC2(CCN2C(C)=O)C1)(C1CC1)OCC CC1CCCC(CC(=O)NC2CC3(C2)CC3C(N2CCCCC2C(=O)NC)=O)O1 C1(NC(C(N2CC(C)(C)C2)C)=O)CC(C(=O)NCC2CC3(CCO2)CC3)=CC1O N1(C(C(CC=CC)C)=O)CC2(C(=O)N(C)Cc3ccccc3F)CCC1CC2 c1(C(=O)NC(CCOC)CNC(=O)C(O)CC(C)C)ccc2cc(Cl)ccc2c1 C1(NC(C(=O)N(C)C)=O)CC(CNC(C23CC(CO2)C3)=O)C1(C)C N1(CCC(C)NC)CC(C(=O)OC)C2(CCCC2)C1 C1(NC(=O)CN2CCCCC2)CCCN(Cc2ccc(-n3cccn3)nc2)C1 C1(NC(C2C(CNC(CN(C)C(N)=O)=O)C2(C)C)=O)CCCCCC1O CC1CC(C(=O)NC(C2CCN(C(=O)COCC3CC3)C2)C)CC(C)(C)C1 c1(CC)ncc(C(=O)NC(CCNC(=O)C(c2ccc(Cl)s2)C)C(C)C)cn1 N1(C(c2c(C)nns2)=O)CCCCC1C(C)NC(=O)Cc1ccn(C)n1 C#CCCC(O)C(=O)N1CC(OC)C(NC(c2c(Cl)cnn2C2CC2)=O)C1 N1(C(C)C)C(=O)COCC1C(=O)NCC1C2CC1N(C(=O)Cn1cncn1)C2 C1(C(C)C)CN(C(=NCCSc2ccccc2)NCC2CCCCO2)CCO1 C1(N(C(=O)CSC(F)F)C)CCCC(NC(=O)CCC2CCCO2)C1 Cc1cnnc(O)c1C(=O)NCCC1CSCCN1C(c1cn(C)nc1C)=O C#Cc1cccc(CC(N2CCOCC2C(=O)NCc2ccc(F)cc2C)=O)c1 C(CCO)(C(F)(F)F)NCCCCNC1CCC(=O)CC1 N1(C(CCC)=O)CC(c2cn(Cc3cnn(C)c3Br)nn2)C(O)C1 C(=O)(C1=CNC2=NCCCN12)NC1(CO)CCCN(C(C(=O)N(C)C)=O)C1 c1(C(=O)NCCCN(C(CC(=O)OC)=O)C)ccc(-c2ccncc2)c(C)c1 C1(C(N(CCOC)CCNC(C2SCCCS2)=O)=O)CCC2(CC1)CC2 c1(CC)ncncc1C(=O)NC1CC(CCNC(=O)CSCc2ccccc2)C1 CC(CNC(c1nocc1Cl)=O)CC(=O)N(C)CCc1nccs1 C(=O)(C1CCC(=O)c2ccccc21)N1CCN(C(CNC(CC)=O)=O)CC(O)C1 CN1CC(CN2C3C(C(=O)ON)CC(CC3)C2)N(C(C2CCC(=O)O2)=O)C(=O)C1 Cc1cc(C(=O)NCCN2CCS(=O)(=O)CC2C)c2nccc(C)c2c1 c1(NC(C2CC(F)CN2Cc2ccc(Cl)nn2)=O)ncc(Br)nc1Br C(=O)(C(C)(CO)OC)NC.C=C(C)CC(=O)NCC1(C(=O)OC(C)(C)C)CCCC1 C12(NC(c3c(CC)c[nH]c3)=O)CC3CCC(C1C2)N3C(=O)CCOC1CCC1 n1(CC(=O)NCC(CNC(CCCc2nc(C)sc2)=O)(C)C)cc(F)ccc1=O C#CC1CCCC(NC(=O)C(COCC)NC(=O)CC(C)N(C)C)C1 CCC(C)CC(C)C(=O)N1CCC(CNC(c2cccc(OC(C)C)c2)=O)C1 C(=O)(CC(C)(C)C=C)N(CC1(CC=C)CN(C(=O)CCC2CCCN2C)C1)CC CC1(C)COC(C(=O)NCC(C)(CO)NC(=O)CC2COCC2(C)C)CO1 C1(CNC(C2(COC)CC2(F)F)=O)CN(C)CCN1C(c1cc(O)ccc1F)=O N1(C(c2ccncc2)=O)CC2CCC(C1)N(C(c1cc(Br)c(F)c(F)c1F)=O)C2 C(CCC(=O)NC(CNC(=O)CCCC1CCOCC1)CO)=CCC=C C1(C(=O)NCC2(O)CN(C(C3C(C)(C)C3C(F)F)=O)C2)CCC2(C1)N=N2 CC(F)(F)CC(=O)N1CCCCC1C(NCP(C)(C)=O)=O.N1(CC)CCOC1=O N1(C(C)=O)CC(C2CCCN(C(C3(c4cnccc4Cl)CCC3)=O)C2)C1 C=CCCCCCC(=O)N1CC(O)(C(C)(C)CNC(=O)C(C)(C)c2ccsc2)C1 C1(C(N2C(C(=O)N(CCOCCO)CC3CC3)CSC2)=O)CCOCC1 C=CCC(CC(C)C)C(=O)NCC1(NC(c2ncccc2C)=O)CCC1 c1(C(N2CC3CC3(C(=O)Nc3cncc(F)c3)C2)=O)c(C(F)(F)F)cccc1Cl Cc1c(CC(N2CC(NC(=O)CC3OCCO3)C3(CC3)C2)=O)ccc(Cl)c1Cl c1(CNC(C2CCCN(C(CC(=O)OCC)=O)C2)=O)c(Br)cc(Br)c(O)c1Br C12(C(N3C(CNC(C4N(C(C)=O)CCCC4)=O)CC3)=O)CCC(C)(C(=O)O1)C2(C)C c1(C(N2CCCC(C(=O)NCCC#C)C2)=O)cccc(Br)c1O c1(CC(=O)NCC2CCN(C)C2)c[nH]c2cnccc12.C1(OC)CC2N(C1)C2=O C12(CC)CN(C(=O)CCCn3cncn3)C(CNC(=O)CSCC(C)C)(C1)C2 N1(C(N(C)C)=O)CCC(C(N2CC(N(C)C(C3CC4CC4C3)=O)C(F)C2)=O)CC1 N(C1CCC(Nc2ncccn2)c2ccccc21)C(=O)C(c1ccc(F)cc1)F C(=O)(CC(C(F)F)NC(=O)C(c1ccccc1)C)Nc1cnc(C)nc1 C1(NC(CN(CCOC)C)=O)CCC(O)CN(C(=O)C(N2CCNC2=O)C)C1 c1(C(=O)NCC(CC)NC(C2C3CCOCC23)=O)cn(C)nc1C1CCCC1 c1(C(=O)NC2(C(=O)NC(c3nccs3)CC)CCC2)cc(CO)cs1 C1(CNC(CN(C(=O)CC2CCCC2C)CCC)=O)CC(F)(F)C1(C)C C1(C(N2CCC(C3CCCO3)C2)=O)(NC(=O)C(C2CC2)C2CC2)CC(F)(F)C1 CCCCCC(C)(CC)C(=O)NCC1CCN(C(=O)C=CI)C1 C1(O)(CN(C)C)CCN(C(c2ccnc(CNC(C3(C)CCCS3)=O)c2)=O)C1 CC1(C)C2CN(C(c3ccc(OC(C)(C)C)cc3I)=O)CC12.c12ccc(cn1)[nH]2 c1(NC(C2(CNC(CC3C(C)(C)CCC3)=O)CCC2)=O)nc2ccccn2c1F c1(CN2CC3N(C(=O)Cc4cnccn4)C3C2)ccccc1[N+](=O)[O-] C(F)(C(=O)NCCC1CC(NC(=O)C(C)n2cnnn2)C1)OC C1(NC(CSCC(=O)OC)=O)CC2(CCN(C(c3ccns3)=O)C2)C1 C1(C(N(C)Cc2cn[nH]c2)=O)CC12CCN(C(c1cnc(S)nc1)=O)C2 c1(CC)oc(C(N2CC(OCC(=O)NC3CCC=CCC3)(CC)C2)=O)cc1C CCCCC(C)(F)C(=O)N1CC(CNC(=O)C(C(C)(C)C)NC(=O)NC)(OC)C1 C12(C(N)=O)CCCC1(C(N1CC(CO)(NC(C3CC3F)=O)C1)=O)C2 N1(C(C(c2cccs2)NC(c2c(C)n(C)cc2)=O)=O)CC2CC3CC2C1C3 S1(=O)(=O)c2ccccc2N1C(=O)NCCC.C1(NCC)CCCN1C C(=O)(CC1=NNC(=O)C1)N1C(CCNC(C(CN(C(=O)OC)CC)F)=O)COCC1 C1(C)(NC(CC2(OC)CN(C(=O)C(F)C(C)(F)F)C2)=O)C(C)(C)C1(C)C C(N=c1ccn(CC(=O)N(C(C#N)C(N)=O)CC(C)C)c(O)n1)c1cccc(C)c1 C=Cn1nccc1C(=O)NC1(CNC(C2ON=C(C)C2C)=O)CC1 C(CC(F)F)(C(=O)NCCC1(OC)CCCC1)NC(C1C(OC)CC1)=O CC1CC(=O)NC(C(N2CC(=O)NCC2C(=O)NC2CCC=CCC2)=O)C1 C1(NC(c2scc(C)c2)=O)CC(C)N(C(C2CCC(N(C)C)CC2)=O)C1 c1(C(=O)NCCC2CC(C(N3C(C(C)(C)C)CCCC3)=O)C2)ccc(F)c(F)c1 C1(CCNOC(CCC2(C)N=N2)=O)CCCCN1C(=O)CCCC1CCCC1 C1(C(=O)NCC=CCNC(c2nccc(C)c2)=O)CC2CCCC(C1)C2(F)F N1(C(c2ccn(CC)n2)=O)CCCCC(CNC(=O)Cc2conc2C)C1 CCCCCC(C)(CC)C(=O)N1CCCC1Cn1cc(CNC(=O)OC)nn1 N1(C(C2(NC(=O)C=CCCC=CCC)CC(=C)C2)=O)CCC(C)(C)C(CO)C1 C1(CC(=O)NC2(C=C)CCC2)CCN(C(=O)C(C)CN(C)C)C1(C)C C1(C(N2C(C3(C(N4CC=C(C)C4)=O)CC3)CCC2)=O)C2CCCC(=O)C12 C1(C(=O)NC2CC(C)(CNC(C3CC(O)C3)=O)C2)CCCC(C)(C)CC1 C=CCC(CC(C)C)C(=O)N(C)CCc1cn(C2CCCC(O)C2)nn1 C1(NC(c2cnc(Cl)s2)=O)CC12CCN(C(=O)CN1CC=CC1)CC2 S(=O)(=O)(c1ccc(Br)cc1)N1CCC(C(N(CCC(=O)OC(C)(C)C)CC#C)=O)C1 c1(C(=O)OC)ccc(F)c2c1CN(C(c1cccc3sc(O)nc13)=O)CC2 N1(C(C(CC#C)C)=O)CCCC2CN(C(C3CC(SC)C3)=O)CCC12 C1(SC)CN(C(c2ccc[nH]2)=O)CC1NC(c1nn(C(C)C)nc1Br)=O N1(C(C2CC2CF)=O)CC(NC(C2(N3CCOCC3=O)CC2)=O)CC12CCCC2 N1(C(c2ccc(OC)s2)=O)CC(CNC(c2sccc2OC(F)F)=O)CCC1C C1(CNC(C(CC=C)(C)C)=O)CN(C(c2ccc(CCF)cc2)=O)CCC1(F)F CCC(CC(F)(F)F)C(=O)NC(C1(C)CCCC1)Cc1ccncc1Br N(C1CN(C(=O)CN=S(C)(C)=O)Cc2ccccc21)C(C(C)OC)=O CC1(C)CC(C(=O)NC2COCC2C(=O)NCCOc2ccncc2)CCO1 C(=O)(C(C)C(C)n1cccn1)Nc1c(C(N(CC(=O)NC)C)=O)nns1 C=CCC(C)(C)C(=O)NC1CCN(C(=O)C=Cc2ncc[nH]2)C(C)C1 c1(C(C)=O)ccc(C(=O)NCC2CN(C)CCN2C(=O)C2=CCSC2)cc1C C(C1c2ccsc2CCN1C(c1sccc1S(C)(=O)=O)=O)NC(CSCC)=O N1(C(CN(C(=O)OCC)C)=O)CCCC1CNC(C1COCCO1)=O C1(CN(C(=O)C(C2(N(C)C)CCCCC2)(F)F)C)CN(C(=O)C(F)F)CCCO1 N1(C(C2CC(CF)C2)=O)CCC12CN(C(C1CC(=O)N(C3CC3)C1)=O)C2 CCCCC(C(=O)NCc1cc(CC)ccn1)NC(=O)C(C(C)C)OCC C(C(=O)N=S(C)(C)=O)NC(c1ccncc1C)c1n(CCCSC)nnn1 C=CC1CCCN(c2ncnc(NCc3ncc(Cl)n3C)c2C)C1 CC(C)(C)C(O)C(=O)NCC1(C(=O)NCC2(CC3CCC3)CC2)CC1 C1(C(N2CC3C(CNC(C=C(CCC)C)=O)(C3)C2)=O)(CF)CC2(CCC2)C1 c1(SC)cccc(C(=O)NCC2COC(CNC(c3coc(C(C)=O)c3)=O)C2)c1 CC1(C)COCCC1C(N1CCC(CNC(=O)Cc2csc(C(F)F)n2)CC1)=O CC(C)(C)C1CCNc2c(C(=O)NCCNC(c3ccc(Cl)cc3)=O)cnn21 N1(C(c2c(OCC)ccs2)=O)CCC(NC(=O)CCC2CCCCN2C)C1C1CC1 C12(NC(C(C=C)O)=O)CCC(CNC(C3(OCC)CCC3)=O)(C1)OC2 C1(CCC)CN(C(=O)C(C)CBr)CCN1Cc1cc(C(F)(F)F)cc(Br)c1 C1(C)(CNC(CCC2(C)CC2)=O)CC(F)(F)CN1C(c1cccc(Cl)c1O)=O C1(CC)CN(C(C2COCC2NC(C2CCC3CC2CO3)=O)=O)CCCO1 C1(CC)CCCN(C(=O)Cn2ccnc2)C1C(N1CCN(C)C(COC)C1)=O c1(C(N2CC(C)(NC(=O)Cn3nnc(C(F)(F)F)n3)C2)=O)cn2cccnc2n1 C(=O)(CC(CC)NC(C1(CCC)CCCN1)=O)NCCC N1(C(CCN(C(C)=O)C)=O)CCCCC1CNC(C1CC(CC2CC2)C1)=O C1(N(c2cc(OC)ncn2)CC(N)=O)CC(C)(C)C12CC2 C1(OC)C2CCN(C(=O)NC3CCCCC3c3nc(S)n[nH]3)C2C1(C)C c1(C(=O)NCC(N(C)C(C2CCC2C(C)(C)C)=O)C2CC2)cc(Cl)c(Cl)n1C C1(NC(C(C)(C)CC#N)=O)CCC2(CC1)CCN(C(c1conc1C1CC1)=O)C2 c1(CNC(c2c(C)n[nH]c2)=O)ccc2c(c1)CCC2NC(=O)C(F)(F)C(O)C1CC1 CCCC(C(N)=O)NC(=O)CCn1cc(C2(C(=O)OCC)CCCC2)nn1 C(=O)(CC(C)C(=O)OC)NCCC1CCN(C(C(CC)CC)=O)C1 C=C=CCCC(=O)NCC1CCC1NC(=O)C(N1CCOCC1)C1CC1 c1(C(=O)NCc2nc(C(CC)NC(=O)CC3C=CCC3)sc2)[nH]cc(C)c1C c1(OC)c(F)cc(C(=O)N(CCNC(=O)C(c2ccc(C)s2)C)C2CC2)cc1Cl c1(C2C(C(=O)OC)C2)noc(C)n1.C1CCN1 Cc1csc(=NCC(=O)NCC2CN(C(C3CCCC3S(C)(=O)=O)=O)C2)[nH]1 c1(C(=O)NC(C)CCNC(=O)C=C2CC2)cc(O)cc(=O)o1 N1(C(C2CN(C)C(=O)N2)=O)CC2CCC1(CNC(=O)CCCS(N)(=O)=O)CC2 N1(C(C(C=C)O)=O)C2CCCC1CC(NC(=O)Cc1ccccc1S(C)(=O)=O)C2 c1(C(N2CCC(c3ccccn3)C2)C(=O)NCC(=C)C)ccccc1C CCC(C)C(O)CC(=O)NCC1C=CC(NC(=O)C2=C(C#N)CCC2)C1 CC(C(C)C(=O)NCC1CCC(CNc2ncccc2[N+](=O)[O-])CC1)S(C)(=O)=O N1(C(C)=O)CC(CC(=O)NCC2(NC(=O)CO)CCC2)C1 c1(C(=O)NCC(C(=O)NCc2ccnn2C(C)C)OC)cccc(Cl)c1 N1(C(C(N2CCC(C)C2)=O)=O)CCCC(O)(CN2CCCC2)CC1.C(=O)(CS)NC C1(C(N(CCCNC(C2CC(C)(C(=O)OC)C2)=O)C)=O)CCC(N(C)C)CC1 c1(C(N(CCNC(C2C(SC)CCC2)=O)C(C)C)=O)ccncc1Br N1(C(C(C2CCCC2)NC(=O)Cc2ncccc2F)=O)CC2CCC(O)C2C1 c1(NC(C)C(C2CCCCC2)NC(C2CCOC2)=O)ncc(C#N)cc1Br N1(C(CC(CC)O)=O)CCC(NC(c2c(C)coc2C(C)(C)C)=O)C(CC)C1 C(=O)(C(CNC(=O)CCCn1cncn1)OCC(=O)NC1CC(N)C1)NC.C1CCC1 C1(F)(NC(=O)NCC2C(C(NOC(C)(C)C)=O)CCO2)CCOCC1 Cc1c(NC(=O)C(CCC2CC2)NC(c2csc(CO)n2)=O)cnn1C N1(C(CCSC)=O)CCC(CNC(c2n[nH]cc2-c2ccccc2)=O)C(C)C1 c1(C(N2C(CN(C(C3CC=C(C)CC3)=O)C)CCC2)=O)cccc(Br)c1N N1(CC)CC(C(=O)NC(C)CNC(c2nccnc2OC)=O)CC1=O C12(NC(CC(C)C)=O)CC1CN(C(c1noc(-c3ncccc3F)n1)=O)C2 C1(CNC(C2(CSC)CCOCC2)=O)CN(C(c2ncc[nH]c2=O)=O)C(C)(C)C1 C1(C(=O)Nc2c(C)nsc2)(NC(c2cc[n+]([O-])cc2)=O)CCCC1C NC1COC2(NC(N3CCCC(Cc4cc[nH]n4)C3)=O)CC1C2 C(=O)(C1=CC2CCC(C1)C2)NCC1(CNC(C(CC#C)(C)C)=O)CC12CCC2 c1(OCc2cn(CCCOC)nn2)cc(N2CC(SCl)C2)ccc1[N+](=O)[O-] C=C(C)CC(C(=O)N(C)Cc1ncoc1CC)OC.C1(C)C(=O)N1 C1(CN(C(=O)C#CC2CC2)C)CN(C(=O)CC2CCCC2O)CC12CC2 C1(C(=O)NCCC2CCCC2(F)F)(CNC(=O)OC(C)(C)C)CCOCC1 c1(N2C3CC(CC)CC2CC3)nc(=NCc2cnn(C)c2C)[nH]c2c1CCCC2 C(=O)(C1=CCCCCC1)NCC(C)(C)OCCO.C(C=O)N(CC(=O)NC)C c1(C(N(C)Cc2cc(Cl)ccc2Cl)=O)cc2c(ncc3ccccc23)s1 C(N=c1[nH]c(=NCCCN2CCCC2)c2ncccc2[nH]1)CCN1C(=O)OCC1 c1(CNC2C(C(=O)Nc3c(C)ncnc3)C2)c(F)cc(C#N)cc1F N1(C(CCCOC)=O)CCC2(CC1)CN(C(c1ccc(F)c(C)c1)=O)CC2(F)F C1(C(C)NC(CN(C(=O)CN(CC(F)(F)F)C)CCOC)=O)CC1(C)C C1(NC(=O)CCc2cnc[nH]2)CC(NC(C2CCC3(CC3)C2)=O)C12CCOCC2 c1(-n2ncc(C(N(CC(CNC(C(CC)(C)C)=O)O)C)=O)c2)ccc(F)cc1F N#Cc1ccc(C(=O)NC2(CF)CCN(c3ncc(Br)cn3)C2)cc1F C1(C(=O)OC)CCC(NC(=O)CCC(N)=O)CC1.c12nnsc1CNC2=O C1(C(=O)OC)CC=CCC1OC(=O)CC1(CNC(=O)OC(C)(C)C)CCC1 c1(C(=O)NCC2(F)CC(NC(c3cnc(OC)s3)=O)C2)cc2c(cc1N)CCC2 c1(NCc2c(C(=O)OC)ocn2)ccc(CCNC(c2ccccn2)C)cc1 C(C(CC(F)(F)F)NC(C1CC(=O)NC1(C)C)=O)NC(C(C=C)CC)=O N1(C(CCCC)=O)CC(C(=O)NC23CC(F)(C2)C3)C(F)(F)C1 O=S(=O)(c1cccc(N2CCOC(C3CC3)CC2)n1)NCCCN1CCCC1 N1(C(C(C2CCN(C(CCCSC)=O)C2)(C)C)=O)CC2(CCN(C)CC2)C1 C1(C(=O)NCCCn2ccnc2)CC(O)CCN1C(c1cc(F)cnc1O)=O C=C1CC(C(=O)N(CC(C)C#N)C)(CN(C(N)=O)CC2CC2)C1 c1(C(N2CCC(C(C)C#N)CC2)C(=O)NC)ccc(OCC(C)C)nc1C C1(C(=O)OCC(=O)N(CCSCCC(C)C)CC)CN(C(C)=O)C1 C1(NC(NCC(COC)C(C)C)=NCC2CC2)CCn2c(C(F)(F)F)nnc2C1 c1(CNC(C(C(C)OC)NC(=O)CC2CNC(=O)O2)=O)nn(C)c(=O)n1C CN1CCC(CC(=O)NCCCNC(C2CCC(=O)NC2)=O)C1=O C(=O)(CC(C(F)(F)F)c1ccon1)NC(CCNC(C(C)NC(N)=O)=O)C N1(C(c2c(C)cccn2)=O)CCC(NC(C2CCC(=O)N2)=O)C(CO)CC1 c1(OCC)ccc(-c2cccc(C(=O)NCc3ccnc(CO)c3)n2)cn1 c1(N(C)C(c2cnn(-c3ccc(O)cc3)c2C(F)(F)F)=O)nc2ccccc2o1 Cc1ccc(C(=O)N(CC(C)N(C(=O)CCn2cncn2)C)C)c2cccnc12 c1(OC(C)C(=O)NCC(CO)NC(c2cnc[nH]2)=O)ccc(F)cc1 C(=O)(C1CCC(=O)c2cccn21)N(CCNC(C=C(CCC)CCC)=O)CCC c1(CCC)onc(C)c1C(N1CC(N(C)C(C2CC2N2CCOC2=O)=O)C1)=O C(=O)(C1=CCC(F)(F)CC1)NCCCOCCNC(C1CCCC(=O)N1)=O C(C(C(=O)N(CCCOCCNC(C1CC1C)=O)C)C(F)(F)F)OC c1(C(=O)NCC2C(CNC(c3c(CC)nns3)=O)C2)cc2c(F)cc(Cl)cc2[nH]1 CC(N=c1nc2c(cnn2C)c(NCc2ccc(CO)o2)[nH]1)C1CC1 N1(CC)N=C(C(=O)N2CC=CC2CNC(c2cnc(C(C)(C)C)s2)=O)CCC1=O Cc1nccc(C(=O)NCC2CCCN(C(C34CC5CC3C4C5)=O)C2)c1Cl CC(C)CS(=O)(=O)CC(=O)N1CCOCC(CNC(=O)C(F)C2CCOC2)C1 C1(NC(C(CC)C)=O)CCN(C(=O)Cc2cccc(N)c2N)CC12CCC2 CC12CCC(C(=O)NCc3cccc(NC(=O)C(=O)c4cccs4)c3)(CO1)C2 C1(NC(C2OCC(C)C2)=O)CC2CC(C1)N(C(=O)C=Cc1ccccn1)C2 C1(C(CNC(c2cc(C)co2)=O)NC(CCCOCC=C)=O)CCCCCC1 Cc1ccccc1CC(=O)NC(C)(C)CC(=O)NC(CC1CC1)C1CC1 C1(CNC(C(C2CC2)OC)=O)CN(C(=O)C(F)=C(C)C)C2(CCC2)C1 c1(C(=O)NC2CC(CO)NC2=O)cccc2ccc(Br)nc12 Cc1c(CNC(=O)NCCN2CCOCC2)cnc2cc(Cl)ccc12 C1(NC(c2cn(C)nn2)=O)CC2(CCCN(C(=O)CC34CCC(CC3)CC4)C2)C1 Cc1ccc(F)c(CS(=O)C(C)C(=O)NC(C)C(=O)Nc2ccnn2C(C)C)c1 N1(C(c2c(C)nn[nH]2)=O)CCCC(NC(c2cn3c(n2)CCC3)=O)C1C CC(=O)C(C)(C)CC(=O)N1CC(C(N)=O)(NC(=O)C2=CCCSC2)C1 N1(C(c2c(C)[nH]c(=N)[nH]2)=O)CCC2OCCC2C1 N1(C(CN(C)CCO)=O)C2CCCC1CN(C(=O)CC1Cc3ccccc3C1)CC2 c1(CC(=O)NCC2OCC(CNC(C=CCOC)=O)C2)cccc(F)c1O N(C(=NCCCOC)NC(C)COC(C)C)CC1CN(C(=O)OC)C1 C1(CNC(c2c(OC)cc(C)cc2)=O)CC2CCC1N(C(=O)CC13CC(C1)C3)C2 c1(CC(=O)NC(CC=CC(=O)NC(c2ccn(C)n2)CC)(C)C)c(C)noc1C C12(C(=O)NC3(CN(C)C(c4cc(F)cc(N)c4F)=O)CC3)CCCCN1CCC2 C1(CC(=O)NC(C(=O)N(C(C(=O)OC)C)C)c2ccoc2)CC(F)(F)C1 C(c1c[nH]nc1C)=CC(=O)NC(CC)CN(C(=O)C(CSC)OC)C C#CC1CCCN1C(=O)C(C)(C1CC1)N(C(=O)CCc1cc(C)no1)C c1(OC)ncnc(NCC2CCCCN2C(C23COCC2C3)=O)c1OC N1(C(c2c(C)cc(N)c(Br)c2)=O)CCC2CCN(C(=O)CC(C)C(F)F)C2C1 c1(CC(=O)NC2(OC)CCN(C(=O)COC(F)F)CC2)ccc2cnccc2c1 Cc1[nH]nc2ccc(C(=O)N(C(C)CN(C)C(C3CCCCCC3)=O)C)cc12 C1(C(F)(F)C(=O)N2CCC(N(C)C(c3ccncc3Cl)=O)C2)(OC)CCCCC1 N1(CCC(=O)NCC(CN(C)C(C2CC=CCO2)=O)O)CCCCC1 C(=O)(C#CC1CCCOC1)N(C)CC1CCN(C(=O)C#CC2CCCCC2)C1 C1(CC)(NC(C2CCN(CC)CC2)=O)CCN(C(c2ccc(=O)n(C)c2)=O)CC1 C1(CCOC)CCC(C(=O)Nc2ccc(-c3nn[nH]n3)nc2)CC1 C(=O)(C1=CS(=O)(=O)CCC1)N1CC2(CC(NC(c3cc(Cl)n[nH]3)=O)C2)C1 CCCC(C(=O)N(CC(F)(F)COC)C)NC(C1(OC)CCOCC1)=O C12(NC(C=Cc3c(C)ncs3)=O)CCC(CNC(=O)C3=CCCC3)(CC1)OC2 N1(C(c2c(F)ccc(OC)c2)=O)CCN(C(=O)CNC(N)=O)CC(C)C1 Cc1cc(Cl)cc(N)c1C(N1CC=CC(NC(=O)C=CCCC(C)C)C1)=O CC1(C)CC(NC(C2CCCC2)=O)CN(C(=O)C(C)CNC(=O)C2=C(Cl)CCC2)C1 C=CCC(Cc1ccccc1)C(=O)NCc1c(C)ccn1C C1(NC(CC2N(C(Cc3ccc(C)o3)=O)CC2)=O)CC12CCCC2 N1(C(c2ccc(OC)cc2)=O)C2CCC1CC(NC(=O)C(C)N=[N+]=[N-])C2 C1(CNC(CC=CC=C)=O)CC(C(=O)NC(CO)(CO)CO)=NO1 C1(C(N(C2CN(C(c3cnc(CC)o3)=O)CC2O)C)=O)CCc2nnc(C)n2C1 c1(C(=O)NCC(CNC(C2(CC(=O)OCC)CCCC2)=O)O)ccc(=O)n(C)c1 CC(CNC(c1cccc(=O)o1)=O)C(F)C(=O)NCC(C)(C)C(C)(F)F n1(CC)ncc(Cl)c1C(=O)NCC(C)N(C(=O)CC(C)C1CC1)C C(c1cccc(Cl)c1)=C(C(=O)NCC1CCN(C(c2c(C)nc(OC)s2)=O)C1)C c1(C(=O)NCCN(C(=O)CCCCCF)CCOC)cc[nH]c(=NC)c1 N1(C(c2cc(C)nc(C)c2)=O)CCC2(CCCN2C(C2CCOC2(C)C)=O)C1 c1(C(N(CCNC(C2C(CC)C=C2)=O)CCOC)=O)nccn2nccc12 C12(CNC(C(C3CCOCC3)C)=O)CCC(CC1)CN2C(C1(CCO)CC1)=O C(C(O)C(F)(F)F)N(C)Cc1cn(Cc2cccc(Cl)c2)nn1 C1(C(N(CC)Cc2nccs2)=O)(C(C)C)CCN(C(c2nc(C)sc2C)=O)C1 Cc1nc(=NCCc2ccnn2C)[nH]c(=NCc2cc3c(s2)CCOC3)[nH]1 c1(C(=O)NC2CCCN(C(C(C)OCC=C)=O)C2)ccn2ccnc2n1 CN1CCCC(C)(C(=O)NC(CC(=O)NCC2CCCNC2=O)C2CC2)C1 O=S(=O)(c1cccnc1N1CCC2(CCCNC2=O)C1)NCC(O)CF C(c1cccnc1)=CC(=O)NCCOCCNC(c1cn(CCCC#N)nn1)=O C(CC(C)C)(c1ccc[nH]1)NC(=O)NC(c1nccs1)CC C(C(C)(C)C(=O)O)C(N(C1(c2cn(-c3cccnc3Br)nn2)CC(=O)C1)C)=O c1(-c2cn(C3(C(N(C(c4n(C)nnc4)=O)C4CC4)=O)CC3)nn2)cccc(Cl)c1 C(=O)(CCCS(C)(=O)=O)N(C1CCN(C(C2CCOC2=O)=O)CC1)C C1(NC(c2c[nH]c3ccccc23)=O)COC2(C1)CN(C(=O)CC1CCCCC1)C2 c1(CC(=O)NCC(=O)NCC(CNC(=O)C2CC2)OC)n[nH]c2c1CCCC2 c1(COC)cc(F)c(Cl)cc1Cl.C1C#CC(=O)N1 C1(NC(CCSCCC)=O)CCC12CN(C(c1cn(C)nc1O)=O)C2 O=C(N=c1[nH][nH]c2c1COCC2)C1CCN(C(=O)C(F)(F)F)C1 CCCCCC(O)CC(=O)Nc1sc(C)cc1Cl.C123COC(C1)(C2)CNC3=O C#CCCCC(C)C(=O)NCC(C)(C)CN(C)C(C1CCc2n[nH]cc2C1)=O N1(C(c2sc(CC)c(C)c2)=O)CCCN(CCNC(c2c[nH]c(C#N)c2)=O)CC1 c1(SCC#C)cccc(C(=O)NCC2CCCN2C(c2ccnc(C)c2)=O)c1 N1(C(CSCCCC)=O)CCC(C(F)F)(CNC(c2nn(C)cc2C)=O)C1 C1(OC)CC(NC(C2CC=CC2)=O)CN(C(C2(N3CCOCC3)CCC2)=O)C1 N1(C(c2onc(COC)n2)=O)CCCCC(N(C)C(C2(C)CCN(C)C2=O)=O)C1 CC(C)CCCC(=O)N1CCC(C(C)CNC(=O)CC(O)CN(C)C)CC1 N1(CC(=O)NC(C(C)=O)(C)C)CC2CCC1CNC2=O N1(C(C(C)C(C)O)=O)CCOCC(CNC(c2scnc2Cl)=O)C1 N1(C(C(CCCCC)O)=O)CCC2CN(C(=O)CCC3C(=O)NN=C3C)CC2C1 c1(CNC(CC2CCC(C)C2)=O)nc(CNC(=O)CS(C)(=O)=O)cc(O)n1 CCC(C)(CNC(=O)CC1CN(C(=O)CC2CSCCO2)CCO1)CO C(CC(N)=O)(C(=O)N1CCC(C)CC1)NC(c1nccc(OC)c1)=O c1(OC)cc2[nH]cnc2cc1C(N1CCCC(C)(CO)C1)=O C12(CCCCCC1)C(=O)N2CC.C(=O)(CC(C)(C)C#N)N1CCC(F)(COCC)C1 c1(C(C)(C)C)ccc(C(N2CCC(NC(C3CC(C)(CN)C3)=O)CC2)=O)c(N)c1 C1(CN(C(=O)CC2(N3CCCCC3)CCCC2)C)CCCN1C(C1(C)CCC1)=O Cn1[nH]c(C(=O)NC2(Cn3cc(COC4CCOCC4)nn3)CCC2)nc1=O Cc1ccc(-n2cc(C3CCN(C(C4CC5CC(=O)C4O5)=O)CC3)nn2)c(O)n1 c1(C(=O)NCCCN(c2nnc(C3CC3)o2)C2CC2)ccc(-c2ccco2)[nH]1 Cc1cccc(C)c1CO.N12CCOC(C)(C1)COCC2C(=O)NC(C)(C)C N1(C(C(CC)O)=O)CCC=C(C(=O)Nc2ccsc2)C1 CCCCC(O)C(=O)NC1CCN(C(=O)C(C)C(O)C(C)C)C12CC2 C1(CN(c2cn(C)nc2)CCO)CCC(N2CCOCC2)CC1 c1(CNC(C(Cn2cncn2)NC(C2COCC(C)O2)=O)=O)cccc2ccnn12 c1(C(=O)NCC2(C)CCC(NC(c3c(C)c[nH]c3)=O)C2)ccc(O)c(Cl)n1 Cc1cc(-c2cnc(CNC(c3ccc(C(F)(F)F)nc3C)=O)nc2)cc(C)c1 N1CC2CCC(C1)N2C1CCN(C(=O)C(C)O)CC1.CCCCCCCO c1(OC)ccc(S(=O)(=O)N2CC3CN(Cc4nc5ccccn5c4C)C3C2)cn1 N#Cc1cc(C(=O)NC2(C(=O)NCC3CCCCCC3)CCSC2)c[nH]1 Cc1cc(CC(N2CC(CO)(NC(=O)COc3ccsc3)C2)=O)no1 c1(Nc2ncc(Br)cn2)ccc(C(=O)NCC2C=CCN2CC2N(C)CCC2)cc1 Cc1onc(C(=O)NC(C)C(C)NC(c2ncc(F)cn2)=O)c1[N+](=O)[O-] N1(C(C=C(CCC)C)=O)CC(NC(=O)CC(C)(C)CC)CC2(CC2)C1 c1(C(N(CC(=O)OCC2CC2CNC(C2CC2)=O)C)=O)csc(C#N)c1 c1(C(=O)NC(C(=O)N(CC(COCC)O)C)CCC2CCC2)cc(C)cc(F)c1 CC1=NNC(=O)C1CC(=O)NCC1(F)CCC(NC(c2csc(C)c2C)=O)C1 c12ccc(F)c(c1)CNC2=O.C1(C(=O)N)C2COCC12.C12CC1CNC2=O.CO C1(CC)C(C(=O)NC2CC(CO)C3CC23)CCCN1C(=O)CC1CCOCC1 c1(CSC)cc(C(=O)N(CCCNC(C2CC2(C)Br)=O)CCO)sc1C C(=O)(C1=C(Cl)CCC1)N1CC(C(N(CC(=C)C)C)=O)C(C)C1 C(C(CC(C)(C)C)NCCSc1nccs1)OC CCC(C)C(C(=O)NCC1CN(C(=O)C2=NOCC2)C1)NC(N)=O C(C(=O)N(CC)CC1CCCN(C(=O)C=CCCC(C)C)C1)(C(C)C)OCC C1(OC)(CO)CCN(C(C2CC(=O)N(c3ccc(Cl)cc3)C2)=O)CC1 N#Cc1ccc(CN2CCOC(CC(=O)NC3CC(O)C3)C2)c(Cl)c1 N1(C(=O)OC(C)(C)C)CCC(NC(CCc2cn(C(C)(C)C)nn2)=O)CC1 c1(CNC2CCN(C(c3ccn(C)n3)=O)CC2F)cc(F)c(C#N)c(F)c1 c1(C(C2CN(CC3CCN(c4ccccn4)CC3)CC2F)=O)cccc(Cl)c1F CCC(C)C(O)C(=O)NCC1(NC(=O)C#CC2(C(F)(F)F)CC2)CCCCC1C C(=O)(C1=C2CCCN=C2NN1)N1C2C(NC(c3ccc([N+](=O)[O-])[nH]3)=O)C(CC2)C1 CC(N=[N+]=[N-])C(=O)NCC(C)NC(C1(c2cc[nH]n2)CC1)=O Cc1cnc(C(=O)NC(CNC(c2ccc(F)s2)=O)C(C)C(C)C)c(F)c1 c1(C(N2CCC(N(C(c3cccc(C)c3Cl)=O)C)C2)=O)ccc2c(c1)COCC2 c1(C(N2CCCN(C(C(C)C)=O)CC2C(C)C)=O)cc2cc(F)cc(F)c2o1 N1(C(C2N(C)CCC2)=O)CC(CNC(=O)C=Cc2ccco2)OC2(CCC2)C1 C(=O)(CCP(C)(C)=O)N(C(C)CN1CCC1)C.c12nc(no1)NC(=O)CC2 N1(C(c2ncc(C)o2)C(=O)NC2CCC2)CCC(C2CCCC2(C)C)C1 C1(C)(C(C)=O)CC[n+]2c(C)nn(C)c21.c1csc(C#N)c1 N1(C(COC)=O)CCC2(CC1)CN(C(c1ccc(SC)o1)=O)Cc1ccccc12 N1(C(C=C(C)Cl)=O)CCN(C(=O)Cc2nc3ccccc3o2)CC(O)C1 C1(CNC(Cn2ccc(C)n2)=O)(NC(c2cnc(C(C)C)s2)=O)CCCCC1 C1(F)(C(=O)NCC=CCNC(c2cccc(OC(C)C#N)c2)=O)CCS(=O)(=O)C1 O=C1C(C(F)(F)F)CCCN1Cc1nnc(N2CCCC2)s1 C12(NC(C=CC=CCC)=O)CCCC1CN(C(=O)Cc1cscc1C)C2 Cc1ccc(=NCCC(=O)NCC2CCCCN2C(=O)Cc2ncc(C)[nH]2)[nH]c1 N1(C(C2(SC)CCC2)=O)CCC(C)C(CC(=O)NCc2cc(C)on2)C1 O=C(C1=CCN(C(C2CN3CCC2CC3)=O)C1)NCc1ccccc1Cl C1(C(=O)N(C2CC2)Cc2ccnc(F)c2)(NC(Cc2c(C)ncs2)=O)CCOCC1 C(CCC(C)C)=C(C)Cc1nccs1 [N-]=[N+]=NC1CC(C(=O)NC2CC(CNC(=O)Cc3ccnn3CC(F)(F)F)C2)C1 C(=O)(CCS(N)(=O)=O)NCC(N(C)C(C1CN(S(C)(=O)=O)C1)=O)C1CC1 CCC(C)(C)CCCC(=O)NC(C)C(C)C(=O)N(C1CN(C)C1)C C1(NC(c2ccncc2O)=O)CC2(C1)CC(C(=O)NCc1ccc(F)cc1O)C2 N1(C(CNC(=O)OCC)=O)CCCC(CO)(NC(c2c[nH]c(C)cc2=O)=O)C1 C(=O)(C#CC1CCOCC1)NCCOC1CCN(C(C(CC)SC)=O)CC1 c1(NC)ccc([N+](=O)[O-])cc1C(N1CCC(C)C(NC(=O)CCCCSC)C1)=O c1(SC)ccc(-c2nc(C3CCC(C)C3C)n(-c3cnnn3C)n2)nc1 C1(C(N2C(CN(C(C3CC=C(C)CC3)=O)C)CCC2)=O)CCCCCN1C C1(CCNC(C2C(C)C2)=O)(NC(=O)CSC2CCCC2)CCCC1 N1(C(CC(CC)(F)F)=O)CC2(CCN(C(c3cc(Br)n[nH]3)=O)CC2)CC1C c1(OC)ncc(NC(C2(C)CC(O)CN2C(=O)Cc2ccccn2)=O)cc1F C1(NC(=O)NC)C2CC3CC(C2)CC1(C)C3.c1(CN)ccc(C(F)(F)F)cc1 C1(C2CC2)(CC)CCCCN1C(c1cc(F)ccc1C)C(=O)NC1CCCC1 N1(C(C2CC(=C)C2)=O)CCOC2(CCC(N=c3[nH]c(O)ncc3C)CC2)C1 C#Cc1ccc(C(=O)NCC2CC(NC(C3CC4(CC4)C3)=O)C(O)C2)nc1 c1(NC(C)=O)ccc(Cl)c(C(=O)NC(C)Cn2ccnn2)c1 C=CCCCC(=O)NC1CCCC(CC(=O)N(CCOC)CC2CC2)C1 C=CC(CCC)CC(=O)NC(CCSC)C(=O)NC1CC(=O)N(O)C1 N1(CCC)CCCCC1C(=O)NC1CC(CO)N(C(c2cc(C3CC3)cs2)=O)C1 N1(C(c2cc(Br)ccc2F)=O)CCCC2C1CCN2Cc1ccc(F)c(F)c1F c1(OC)ccc(NC(=O)C(C2(O)CN(C(=O)C(C)C(C)(C)C)C2)F)cc1C S(=O)(=O)(c1cccc2cccnc12)N1CCN(C(C(C(C)C)S)=O)C2(C1)CCC2 C(=O)(CCCCC(C)C)N1CCCC(N(C(C(C=CC)O)=O)CCF)C1 N1(C(C(C)OC2CCCC2)=O)CCC(C)(CC(=O)N(C2CC3(CCC3)C2)C)C1 c1(C(=O)NC2C(NC(c3cnnc(O)c3)=O)COC2)n[nH]c2c1COCC2 c1(C(N2CC(O)(CNC(c3ccc(C(C)C)cc3)=O)C2)=O)[nH]nc([N+](=O)[O-])c1Cl N(C(=NCCOC)N1CCN(C(C)C)C(=O)C1)C(C#C)C(C)(C)C N1(C(c2c(C)c[nH]n2)=O)CCN(C(=O)Cc2ccccc2[N+](=O)[O-])CC(C)(C)C1 C1(C(=O)NC2C(NC(c3ccc(C(N)=O)s3)=O)COCC2)CC2CCC1CC2 N1(C(C=Cc2c(C)nsc2)=O)C2CC1CN(C(c1ccc(CO)o1)=O)C2 C12(C(N3CC(N(C(C(CCC)C)=O)C)C(C)(C)C3)=O)CCC(O)(CC1)CC2 C=C1CCN(C(=O)C(C)C(F)(F)F)C(n2cc(CN3CC[Si](C)(C)C3)nn2)C1 O=[N+]([O-])c1cnc2c(F)ccc(Br)c2c1CNS(=O)(=O)CC1CCCC(F)(F)C1 c1(OC)ccc(C(F)(F)F)c(Cc2cn(CC3COC(=O)O3)nn2)c1 N#Cc1cc(F)c(C(=O)NCCCNC(C2CCc3nncn3CC2)=O)c(F)c1 C(CC(=O)NCCC1CCN(C(c2cccc(N)c2C)=O)C1)(C(F)(F)F)OC CCS(=O)(=O)NNC(=O)c1c(F)cncc1Br C(CN=c1[nH]c(N2CCC(C3CCC3)C2)nc2c1COCC2)OC1CN(C)C(=O)CC1 CC1CNCC(C)N(C(=O)C(N2CCC(O)CC2)=O)C1.c1(C)csc(=N)[nH]1 C=CCC(C)(CC)C(=O)NC(C1CN(C(c2nccc(C)c2N)=O)C1)C C1(C(=O)OC)CCN(C(=O)C(CNC(c2cc(C)sn2)=O)N(C)C)O1 c1(CC(=O)NC(C(C)C)CNC(=O)C2=COCC2)ccc2nsnc2c1 C1(CN(C)C(C2CC2C#N)=O)CCN(C(C2CCCN(c3cnccn3)C2)=O)CC1 C(C(O)C(=O)NC(C)(C)C(=O)NCCc1ncn(C)n1)OC C(C(C)(C)C(C)(C)C)NC(CC1(NC(C=CC=CCC)=O)CCC1)=O O=C(C#CC1CCCC1)NC(CNC(c1sccc1-c1ccccc1)=O)C1CC1 C1(NC(C(C)OCC(C)C)=O)CCCC1(C)CN(C)C(C1CC2(CC2)C1)=O C(=O)(CCCCCC(C)C)N(CCC(N1CCCC(OCCOC)C1)=O)CC=C CC(Cl)C(=O)NCCC(C)NC(C1CSC1)=O C=CCCC(C)(C)C(=O)N1CCCC(C)(NC(c2cnn(CC=C)c2)=O)C1 CN1CCS(=N)(=O)CC1C(=O)NCC1CCCN1C(C1CC1F)=O c1(C(N=c2cc(C)o[nH]2)=O)ccc2c(-c3ccc([N+](=O)[O-])cc3)nn(C)c2c1 N1(C(C23CCN(C(c4ccc(Cl)cc4)=O)C2CCC3)=O)CCCC(C2CCC2)C1 CC1CC2CN(C(C3(NC(=O)CCC4CC(C)C4)CC(CO)C3)=O)CCN2C1 C1(C(=O)NC2CCC2)CC(O)CN1C(c1ccc(Cn2ccnc2)cc1)=O c1(OC)nccc(C(N2CCC(O)C(C(=O)Nc3ncc(F)c(Cl)n3)C2)=O)c1Cl C1(C)(C(=O)NC(CCOC)C(C)C)CC(O)CN1C(c1ccc(F)c(O)c1)=O N1(C(c2c(OC)cnc(Br)c2)=O)CCC2(CC1)CC(C(=O)NC(C)C#N)CO2 N1(C(CSc2n(C)cnn2)=O)CCCC(C)(C)C1CNC(C1(C)CCNC1=O)=O CC1=C(C(=O)NC2CC=C(C(=O)NC3(c4ccno4)CC3)C2)CCCO1 C1(CN(C)C(C2(CCF)CC2)=O)CCCN(C(C2(C(C)(F)F)CC2)=O)C1 C(=O)(CC(C)(O)COC)NCC(CC)NC(c1sccc1C(C)=O)=O N1(C(C2C(C)CCCC2)=O)CCC(CO)(CNC(c2c(N)cccc2Cl)=O)CC1 C1(C(N(C)CC2(NC(=O)CSC(F)(F)F)CC2)=O)CCOC1=O CCCCC(C(=O)N1CCC(C(C)CNC(=O)C=Cc2ccoc2)CC1)C(C)C N1(C(c2n(C)ccc2)=O)CC2(C1)SCCC2NC(c1sc([N+](=O)[O-])cc1Cl)=O N1(C(C(n2cc(C(c3cnn(C)c3C#N)NC)nn2)C)=O)CCc2ccc(Br)cc2C1 c1(C(N2C3(CNC(C(C(C)C)NC=O)=O)CC(C2)C3)=O)cccc(C(N)=O)c1F c1(CCNC(C(=O)N(CCOCCO)CC)=O)ccc(NC(CC)=O)cc1 c1(C(N2CC(NC(c3ccc(C)cc3)=O)C(F)C2)=O)n[nH]c2c1COC2 N1(C(COCCSC)=O)CCC(NC(c2cccc(C(F)F)n2)=O)C2(CCC2)C1 C1(C(=O)NC(C#C)(C)CC)CC2CC2N1C(=O)C(N1CCCCC1)C N1(C(C2(CC)CCNC2=O)=O)CCC2CN(C(=O)C=CBr)CC2C1 c1(C(N2CCNC(C3CC3(F)F)C2)=O)coc2c1COC2 N1(C(COCC)=O)CCN(C)C(CNC(=O)CCc2nncn2C)C1 C(C(C)(C)CNC(c1cnc[nH]1)=O)N(C(=O)C(F)(F)c1ccnn1C)C c1(C(=O)NC2(C)CCN(C(c3c(Br)cc(C)s3)=O)C2)cccn2nncc12 C1(C(=O)NC2C3(CC(OC)C3)C2)CCC2(CCCO2)CC1 Cc1ccc(OCC(C)C)cc1-c1ccc(NCc2ccco2)nc1 N1(C(C2C(C)(CC)C2)=O)CC=C(C(=O)NCCn2cnc(C)c2C)CC1 N1(C(CC(CNC(COC2(C#C)COC2)=O)O)=O)C2CCCC1CC2 N1(C(C2C(C(C)C)OCCC2)=O)CCCN(C(=O)C(C)(C)CN(C)C)CC1 C1(CN(C)C)CCN(Cc2n[nH]cc2I)CC1 C1(O)(CNC(CC2C(CC)C2(F)F)=O)CCN(C(c2nn(C)cc2N)=O)C1 c1(C(=O)OC)ccc(CC(=O)N(C)Cc2ccc(Br)cc2)cc1.C1(C)C(=O)N1 N1(C(C2(CF)CC2)=O)C2CCC1CC(NC(C1(CO)CC(F)(F)C1)=O)C2 Cc1[nH]nc(C(=O)N(CC(=O)NC2C(=O)OCC2CO)C)c1C CC1CCn2ncc(CNCc3c(Cl)nc4ccccn34)c2C1 N1(C(C=Cc2cnc(C)s2)=O)CCCC(C2CC2NC(=O)CNC(=O)C2CC2)C1 C1(NC(=O)C=CCOCc2ccccc2)COCCN(C(=O)CC2(O)CC2)C1 c12cccc(c1F)NC(=O)CC2.n12cc(nn1)C2.N12CC(C1)OCC2=O.CC Cc1cnc(F)c(CNC(C2CC23CC(NC(C2CC2Cl)=O)C3)=O)c1 c1(C(C2(C(=O)O)CCOC2)N(CCO)CC2COCO2)ccccc1 c1(C(=O)NCCCCCCNC(C2C(C=C)(C(F)(F)F)C2)=O)c(C)nc(C)n1O CC1(C)CCC(CNC(=O)CS(=O)(=O)CCO)N(C(C2CCC(C(N)=O)O2)=O)C1 c1(-n2c(C(C)(C)C)nc(C(CC)O)n2)ccc(Cl)c(C)c1 C1(NC(=O)Cc2ccccc2O)COCCN(CC(=O)NCCO)C1 C=CCC(CC=C)C(=O)NC(C1CCCN1C(=O)C=Cc1ccc(F)c(Cl)c1)(C)C c1(C(c2n(C(CC)C)nnn2)NCCc2ccc(OC)cn2)cccc(N(C)C)c1 C(=O)(C1=CCC(F)(F)CC1)N1C2C(CNC(c3c(C)nc(C)[nH]3)=O)CC(CC2)C1 c1(C(=O)NC(C)(Cc2ccc(F)c(Br)c2)C(C)C)nncc2c1CCCC2 c1(N2CCC(C(=O)NC)C2)ccc(NC(=O)Cn2nc(C)cc2C)c(C)n1 C1(NC(COCCC#C)=O)CC(O)CN(C(=O)CCc2nnc(S)n2C)C1 CCC(C)(C)C(=O)C(=O)N(CCC(CCCC)NCC(C)C(C)O)OC C(C(=O)N1CCCC1C(C)NC(=O)CSCc1nc(C)no1)(C(C)C)SC n1(CC(=O)NCC(CNC(c2c(C)cns2)=O)C(F)(F)F)cc(S(C)(=O)=O)cn1 N1(C(C2CC(C#C)(O)C2)=O)CC(NC(=O)C(F)n2cccn2)CC2(CC2)C1 C(=O)(CCP(C)(C)=O)N1CCCC(CCC(=O)N(C)Cc2cnc[nH]2)C1 Cc1cc2c(cc(C(=O)NC3C(O)CC3O)n2CC(F)(F)F)s1 Cc1cc(C)c(C(=O)NCC(C(C)C)NC(c2[nH]c(=N)ccc2C)=O)c(C)n1 C1(CC)CN(C(=O)COc2ccsc2)CC1NC(c1cc(C)nn1CC(F)F)=O CC(C(=O)NC(Cn1cccn1)C(=O)Nc1cc(Cl)cnc1O)C(F)(F)F Cc1nc2ccc(COC(=O)C3=CCC(C)CC3)cc2o1 C1(C(N2CCCC2CNC(C2CCOC2)=O)=O)CCCC2CCCCC12 c1(C(=O)NC(CN(C(c2cn[nH]c2)=O)CC)C)ccc(OC2CC2)cc1 C1(C(=O)NCCCN(CCCNC(C(C)SCC)=O)C)CC2CCCC12 O=C(C1=COCC1)NCCOC1CCCC(O)C1.C1COCCO1.C1CO1.C1CO1 C(=O)(C(F)C(F)(F)F)NCC(C)(C)C1(CCNC(=O)C(N)=O)CC1 c1(OC)ccc(SCC(=O)N(CCCNC(=O)C(C)(C)O)CCO)cc1 c1(C(=O)NC2CN(C(C3(CC)CCCC3O)=O)CC2O)cc(F)cc2nn[nH]c12 c1(C(=O)NC(CNC(COCCC#C)=O)(C)C2CCC2)nn(C)nc1Br C1(CC)CN(C(c2ccc(SC)o2)=O)CCC1NC(=O)CC1CCCCC1(F)F c1(C(N2CCC(C(C)NC(c3cc(Cl)ccc3N)=O)C2)=O)nc2ncccn2n1 C1(C)(CCNC(C2(C)C(C)(C)C2)=O)CCN(C(c2ccc(C(N)=O)[nH]2)=O)C1 Cc1cc(C(N2CCCC(c3nc(C)cs3)C2)C(=O)NC(C)C)cc(F)c1 CC1CN(CCCCCNC(c2cc(-c3ccc(F)cc3F)co2)=O)CC(C)O1 C1(NC(c2ccccc2F)=O)CC(O)CN(C(=O)C=C2CCCC2)C1 c1(OC)ncc(C)c(NC(=O)C(N2CCC(C)CC2)=O)c1Cl.C12(CC1)CCC2 c12cncc(c1)OC2=O.CCC(CN(C(=O)C(=O)NCC1CC1)C)NCC(F)F C=CC(C)(O)C(=O)NC1CC(NC(=O)C=CC=CC=CC=CCC)C1 C(CC(C)(C)CC(=O)N1CCCN(C(C2(Nc3ccccc3)CC2)=O)CC1)OC CCCC(CNC(C12CN(C(=O)C(C)(C)C)CC1(c1ccccc1)C2)=O)CCO C1(C(=O)NCc2c(C(=O)NC3CCC(C(C)(C)C)C3)n[nH]c2)C2CCC(F)(F)C12 C(=O)(CCCCCCNC(c1coc(N(C)C)n1)=O)N1C(CCCC)CCC1 C1(C(=O)N(C)CC2CCCC2NC(C2SCCCS2)=O)(COC)CC1(F)F CC1CN(C2CCN(C(=O)C3CC3)C2=O)CC1C(N)=O Cc1ccc(F)c(C(N2CSCC2C(=O)NCCCOCC(F)F)=O)c1 N1(C(CS(CC)=O)=O)CC(NC(c2conc2C2(C)COC2)=O)CC1(C)C c1(C(=O)NC2CC2NC(C2(N(C(C)C)CCO)CC2)=O)ccc2c(c1)C(=O)CCC2 C(=O)(C(C)(F)C(C)(C)F)NCCCC1OCCN(C(c2cnn(CC)c2C)=O)C1 N1(C(C(CC(=O)OC)(C)C)=O)CCCC(C2CN(C(=O)Cc3ccsc3C)C2)C1 N1(C(C(CC)n2ccnc2)=O)CCC(CN(C(=O)CC2(N(C)C)COC2)C)CC1 N1(C(c2occ(C)c2)=O)CC2(CCC2)CCC1CNC(=O)Cc1ccc(Cl)cn1 C#Cc1ccc(C(=O)NC(C)(CNC(=O)C=CBr)CO)cn1 N1(C(c2ccc(OC)nc2)=O)CC2(CC2)CC1CNC(C1CCOCC1CF)=O C(=O)(C(CC(F)F)N(C(=O)CC1CCCCN1C)C)NC(COC)C(=O)OC N1(C(C2CCN(C(C3(CCCC)CC3)=O)CC2C)=O)CCCC2(CC1)CC2 N1(C(C(Cc2ccc(C)cc2)O)=O)CC2(CC(NC(C3CC(N(C)C)C3)=O)C2)C1 c1(C(N2CCCC3(CNC(C(C)(C)CO)=O)C2C3)=O)ccc2ccncc2c1 N1(C(C(C2(C(F)F)CC2)N(C(=O)OC(C)(C)C)CCl)=O)CCOCC12CCS(=O)(=O)C2 C1(CCNC(CNC(=O)NC)=O)CSCCN1C(=O)Cc1nnc(C)o1 N1(C(C2=CCC(NC(C(COC)(C)C)=O)C2)=O)CCC2(CC1)CC2OC c1(NC(C2CC(NCc3c(C)nc[nH]3)C2)=O)cc(Cl)c(Br)cc1Cl C(=O)(N1OC2C=CC1CC2)C1C(CCC)CN(C2(C(=O)O)CC2)C1 N1(C(C(C)SC)=O)CC2CCC(C1)N2C(C1C=CCCC1)=O C=CCCC(C(=O)N1CCCC(C)(O)C1)NC(=O)Cc1c[nH]nc1C Cn1cccc1C(=O)NCC(C1CCCC1)NC(c1ncoc1C(C)(C)C)=O c1(C(N2CCC(C3CCCN3CC3N(S(CC)(=O)=O)CCC3)C2)=O)ncccc1C c1(C(=O)NC(C)CCNC(c2ccoc2C(F)(F)F)=O)cc2cccn2cn1 c1(C(=O)NC(CNC(C(COC(C)=O)O)=O)CO)cn(C2CC2)nc1C(F)(F)F Cc1ccc(C(N2CCCC(C)(NC(c3cc(Cl)c(Cl)[nH]3)=O)C2)=O)c(C)n1 c1(CN2CC(CC(N3CC(C)CC(COC)C3)=O)C2)cccc(Cl)c1[N+](=O)[O-] CC1CN(C(=O)CCn2ccccc2=O)CC1CNC(c1n[nH]cc1Cl)=O N#CC(C(=O)NCCC1CCCN1C(c1cnc(Cl)s1)=O)C1CC1 n1(CC)ncc(C(=O)NCC2C3CN(C(c4ccnc(C)c4)=O)CC23)c1C1CC1 n1(CC(=O)NC(CCN(C(=O)CCc2ncc[nH]2)CCCN(C)C)=O)cnnc1O CCCC(CC=O)C(=O)NCC(C)NC(c1cn(C)nc1-c1cccc(Cl)c1)=O C1(C(C)(C)CNC(=O)Cn2nnc(C(C)(C)C)n2)CCCCN1C(=O)CC1CCC1 CCCCCCC(CC)C(=O)N1CC(OC)C(NC(=O)C(CC)C(F)(F)F)C1 c1(CC)nc(C(=O)N(C)CC2CCN(C(c3cnc(O)n3CC)=O)CC2)c(C)o1 c1(OC)ccc(C)cc1C(N1CCC(C)(C)C1CNC(C12CCC(C1)C2)=O)=O C1(CN(C)C(c2cncc(OCF)c2)=O)CCCN(C(=O)CNS(=O)(=O)N(C)C)C1 c1(C(=O)NCC(C(=O)NC2CCOC(C3CC3)C2)OC)cccc[n+]1[O-] N1(C(C=Cc2ccc(CC)o2)=O)CCN(C(C2CCCCS2)=O)CC1C(F)F C=CC1(C(=O)NCCc2ccccc2C)CCN(C(=O)C(O)Cn2cncn2)C1 C(=O)(CC(O)CNC(=O)CCc1cc(C)no1)NC1(C(N(OC)C)=O)CC1 c1(C(=O)NCC(C)(C)C2CCCO2)cc(C(N)=O)no1 C#CCCC(O)C(=O)N1CC(OC)CC1CCNC(=O)CC1COC(=O)C1 C1(O)(CCOC)CC2(CCCN(C(=O)NC3CS(=O)(=O)C3(C)C)C2)C1 C(=O)(C(CC(C)(C)C)OCC(C)(C)OCC(=O)OC)Nc1ccc(OC)cc1 C(CN=c1[nH]c(=NCC2CCCCC2OC(N)=O)c2cc(Cl)ccc2[nH]1)CC N#CC1(C(=O)NCCCCCC(=O)N2CCN(C3CC3)CC2)CCCOC1 C1(O)(C(N(CCNC(C2C(C(=O)OCC)CC2)=O)CC2CC2)=O)CC(F)(F)C1 c1(C2CC2)cccc(C(N2CC(CNC(C3(CC)CC3)=O)C3CC23)=O)c1 C#CCCCCN(C(C1CCOCC1)C(=O)Nc1ccccc1)C N1(C(C2CCC(=C)CC2)=O)CC2CCN(C(C3CC3C3CC3)=O)CC(C2)C1 N1(C(CC2CC(CC)OCC2)=O)CCCC(NC(c2cc(O)ccc2F)=O)C1C c1(N2CCC(C(=O)NC(C(C(C)(F)F)Cl)=O)C2(C)C)ccc2ccccc2c1 C(=O)(C(C)(C)COCC(F)F)NCC(C)N(C(=O)CCC1CCN(C)C1)C C12(CNC(c3c(C)nsc3)c3nnnn3C3CCCCC3)CC(CO)(CO1)C2 C1(C(C)C)CCCN(C(c2sccc2Br)C(=O)NCc2csc(Br)c2)C1 C1(NC(C(c2ccn(C)n2)(F)F)=O)CS(=O)(=O)N(C)C1(C)C c1(C(N2C3CN(Cc4scc(COC)n4)CC32)=O)ccc(C#N)cc1C N1(C(C2(CC)CC2(F)F)=O)CCC2(CCCC2NC(=O)CC2CC=CC2)CC1 C1(CCC(C)C)CCN(C(C2CCC(=O)O2)C(=O)NCc2ccccc2)CC1 C1(CNC(=O)C(O)C(F)F)CCCN(C(C2CCCCCCC2)=O)CC1 c1(C(N(C(=O)Nc2ccc(OCCOC)nc2)C)C)nc2ccc(Cl)cc2[nH]1 C#CCC(O)C(=O)NCC1CCN1C(c1ccc(C(F)(F)F)[nH]1)=O C1(Cl)(C(N(C2(CCNC(C3CCCS3)=O)CCC2)CC)=O)CC1(F)F c1(C(N(C2CCN(C(=O)CC3COCCO3)C2)CC)=O)ccc(C)c(F)n1 c1(C(=O)NCC2C3CN(C(=O)CSC45CC(F)(C4)C5)CC32)ccccc1Br c1(C(C(=O)N(CCCNC(=O)C=CCO)C(C)C)O)cccc(Cl)c1 C12(CN(C)C(c3cnn(C)n3)=O)CC(CO1)N(c1nc(-c3ccccc3)ns1)C2 c1(C(N(CC(C(=O)NC2CCCC(OC)C2)C)C)=O)cc(C)ccc1F c1(OC)ccc(C(N2CC(OC)C(NC(C3(N=[N+]=[N-])CC3)=O)C2)=O)c(Cl)c1 C(=O)(CC(C)C(=O)NC(C(N1CC(C)(N(C)C)C1)=O)C1CCOC1)OC CC(C)(C)C(C)(C)C(=O)NCCN1CCN(C(=O)C#CC2CCCC2)CC1 C12(NC(C3CCC4CC4C3)=O)CCCC1N(C(c1cnc3n1CCC3)=O)CCC2 N1(C(=O)OCCCC)CC(F)CC1C(=O)NC1CCCN(c2ccccc2)C1 c1(C(=O)NC2CCCC(C(=O)NC3CCCCO3)C2)c(O)cccc1F N1(C(CC=C=C)=O)CC2CC2(NC(c2cnc(S)nc2)=O)C1 Cc1cccc(CC(N2CCC(N(C)C(C3(C)CCN(C)C3)=O)C2)=O)c1C C(=O)(C(C(=O)N1CC(CNC(=O)C(=O)NC2CC2)CC1(C)C)OCC1CC1)OC C=CCC(C)(C)C(=O)N1CCC(NC(=O)Cn2cc(Br)c(C)n2)C(C(N)=O)C1 c1(OC)c(NC(N2CCC(OC)CC2C)=O)cc(Cl)cc1C C(=O)(C(F)(F)Cc1ccc(F)cc1)NC1CC(CCNC(COCCC=C)=O)C1 C(=O)(C(O)CC(C)(C)C)NCCC1CC(C)N(C(=O)CC2CCCCCC2)CC1 Cc1nc(CC(C)C)sc1C(=O)NC1CC1CNC(=O)CCOCCC(C)C CC#CCC(C(=O)N1CC=CCC1CO)NC(C1CCC(C)CC1)=O C1(C(N(CC(CN(C)C)O)C)=O)CC2CCC(C1)N2C(C1CCCC1(C)C)=O C1(CC#C)(C(=O)N(C2CC(C(=O)N(CC(CC)OC)C)C2)C)CCC1 C1(C(N2CC(C)(CF)C2)=O)CCN(C(=O)C2CCC3(CCC3)O2)O1 c1(C(=O)NC)c(C)cc(NC2CC3CC(NC(C=CC(CC)C)=O)C3C2)cc1C Cn1[nH]c(=NC(=O)NC(C(C)(C)C)c2cnn(C)c2)c(=O)n(C)c1=O C1(C(=O)NCC2C(C(=O)NC(C3CCCCC3)CO)CCC2)CC2CCC2C1 c1(CC(C)C)cc(-c2nc(-c3cncnc3)nn2C(C2CCCCC2)C)n(C)n1 O=C(C#CC1CCCOC1)NCC1CCCCN1C(=O)CCc1ccc(Cl)cc1 c1(C(=O)NCC(C)CNC(=O)C(C)(C)CN(C)C)cnn2c1N(C)CC2 c1(CN2CCC(N(C(CCCC(C)=O)=O)C)C2)ccccc1S(C)(=O)=O O=C(C1=Cc2ccccc2OC1)NC1CCCC1NC(c1cc(F)cc(F)c1)=O CCC(C)(C)C(=O)N1CC(CNC(c2cncnc2-c2ccccc2)=O)C(O)C1 CC(C)C(C(=O)N1CCCC(C(=O)NC(C)C(N2CCCCC2)=O)C1)C1CCC1 c1(CC)ccc(O)c(NC(=O)CC(CC)NC(c2cc(C(N)=O)[nH]n2)=O)c1 C1(C(N2CC(OCC(=O)NCC#C)C2)=O)CCCN1C(=O)C1CC1 CCC(O)C(F)(F)C(=O)NC(C1CN(C(=O)CC2CCC3CC23)C1)C C1(C(=O)NC2CCC(NC(c3ocnc3C(F)(F)F)=O)CC2)CC2COCC2C1 CCCC(C)(C)COC(=O)Cc1ccc(CN(C)C)cc1 c1(CC(=O)NCC2(F)CC(CNC(C3CC3F)=O)C2)ccc(Cl)c(F)c1 C(CCCCCC(=O)N(C1CCCC1)CC1CC1)NC(c1c(CC)nco1)=O C(=O)(C(O)(C(F)(F)F)c1ccccc1)NC1C(CNC(c2ccoc2)=O)CCC1 n1(CC(N2CCCCC(N(C(=O)C3=CCOCC3)C)C2)=O)ncn2nccc2c1=O C(c1cccc(F)c1Cl)=CC(=O)NC1C(NC(C=CC=CC)=O)CCOC1 CC1(NC(=O)CC23CC(C2)C3)CCN(C(C2CC3(C2)CC3F)=O)CC1 n1(CC)nc(C(=O)NCC(CC2CCCC2)C(=O)NC(C)C(F)F)cc1C C(=O)(C1CCc2c[nH]nc21)N.c12ccc(cc1)CNC(=O)N1C(CCC1)C2(C)C.CO C1(C(=O)Nc2cn(CCC)nc2)CC(NC(c2cnccc2C)=O)C12CCC2 c1(C(N)=O)ccccc1Cl.C12CCN(CC1)C(c1ccc(C(F)(F)F)cc1)C(=O)N2 c1(C(=O)NC(CNC(CCC(C)(C)O)=O)C(C)(C)C)cc(Cl)c([N+](=O)[O-])[nH]1 c1(CC(=O)NC(C)CCNC(C2CN3CCN2CC3)=O)c(F)cccc1C#N n1(CCC)cc(Cl)c(C(=O)NC2CCN(C(=O)CC3OCCC3C)C2)n1 Cc1cc(=O)n(C)nc1C(=O)NCCNC(c1cccc(Br)c1F)=O c1(N2CCCC(CC)CC2)nc(NCC(C)(C)C(F)F)c2cnn(C)c2n1 C(=O)(CCC(C)(C)C(=O)c1ccc(C(=O)N(c2cccc(C)c2)C)c(F)c1)OC C1(NC(C(CC)OCC)=O)CC2CC(NC(c3cccnn3)=O)CC12 C=C1CCN(C(c2cnn(CCNC(c3ncoc3C)=O)c2)=O)C1 C(=O)(N1OC2CCC1C2)C1CC(NC(CCc2c(C)ccnc2)=O)C1 Cc1ncc(CCC(N2CC(O)(C(C)NC(=O)CNc3ccccn3)C2)=O)s1 c1(CC)ncccc1C(N1CCC(OCCNC(=O)CCc2ccc(C)o2)C1)=O N1(C(c2c(C)cc(CC)o2)=O)CCCC(C)(C(=O)NC2(C(=O)NC)CCC2)C1 c1(C(=O)NC2C(C)(C)CN(C(=O)CCCC3CCC3)C2)nc2ccc(Cl)nn2n1 c1(CC)cc(NC(c2cn(C3CN(C(=O)CCC(C)(F)F)C3)nn2)=O)cc(O)c1 c1(N2CC(C)(CNc3ccc(OC(F)(F)F)c(Cl)c3)C2)nccc(S(C)(=O)=O)n1 C1(C)(CNC(C2N(C)CCC2)=O)CCN(C(C2CNC(=O)N2C)=O)CC1 c1(OC)cccc(C(=O)NC2CCC(CNC(=O)Cc3cccc(C)n3)C2)c1O c1(C(=O)NC(CNC(COCCOCCOC)=O)CO)ccc(C)c(C)c1Cl C1(CC(=O)NCCOCC(N)=O)CCCN(C(=O)C(c2ccccc2)O)C1 C1(C(=O)NC2(C)CN(C(C3(C#N)CC3)=O)C2)CC2(C1)OCCO2 c1(C(=O)NCC2C(NC(Cc3ccc(C)cc3Br)=O)C2)cc2ncccc2o1 C1(CNC(C(C)(C)OC(C)C)=O)C(C)CCN1C(=O)CCC1OCCO1 C(=O)(C(CN(C(=O)Cn1cnc(=N)[nH]1)CC)C(C)(C)C)N1CC(C(CC)CC)C1 C1(CNC(c2cn(C)nc2)=O)CN(C(=O)COCC2CCC2)C2(CCC2)C1 CC1CC(NC(C2CC(O)C2)=O)CCN1C(c1cccc(C(F)F)c1Cl)=O c1(C(=O)CN2CCCC2Cc2ccccc2)ncc(C2CCCCO2)s1 C(=O)(CCCCC(C)C)NC(CC=C)CC(=O)NCCc1cnco1 C1(NC(c2n(CC)ncc2)=O)CC(C(=O)N(CCO)C(C)C)C(C)C1 C=CCCC(CCC=C)(c1nnnn1CC(F)F)NCCN1CCOCC1 C1(C(=O)NCC2(F)CC(NC(C3C(C)C3C)=O)C2)CCCCCC1 N1(C(c2cnc(OC)s2)=O)CCC(NC(c2cc(C(C)(C)C)c[nH]2)=O)C12CC2 c1(C(=O)OC)ccc(NC(=O)CCc2cc(C)ccc2C)cc1OC1CC1 c1(CC(=O)NC2C(CNC(C(C)C3CCC3)=O)C2)sc(O)nc1O C1(CC=C)(NC(C2COCC(C)(C)O2)=O)CCCN(C(=O)CCC2CC2)C1 N#Cc1ccccc1C(=O)NCC(O)C(=O)N1CCCC1C(N)=O CCC(C)CCCCC(=O)NC1CC1CNC(=O)CCOCCOC C1(O)(CNC(C(F)=CC)=O)CC(NC(=O)C(O)c2ccco2)C1 c1(OC)cc(C)c(C(N2CCC(N(C)C(C3CCC4(CCC4)O3)=O)C2)=O)cn1 c1(C(C(N2CC(N(C(c3c(C)n[nH]c3)=O)C)C2)=O)C)cc(Br)ccc1F C1(C)(CSC)CN(C(=O)C(C)(C)C2CCN(C(=O)CCCOC(C)C)C2)C1 C1(C(N2CC(COC)(CNC(=O)CCN3CCCC3=O)C2)=O)CCCC(=O)C1 c1(OCCC(=O)NC(C)CNC(C2CC3CC2C3)=O)ccc(S(C)(=O)=O)cc1 C(=O)(C(C)C(C)COC)N(CCC)CCNC(c1cccnc1OC)=O N1(C(C2(OC)CCCC2)=O)CCC(NC(=O)Cn2cncn2)CC(C)(C)C1 C1(NCc2cnc(C(=O)OCC)s2)CCCCC1Cn1cc(CCCO)nn1 c1(C(N2C(CCNC(c3ccc(C(N)=O)o3)=O)CCC2)=O)cc2ccccc2[nH]1 n1(CC(=O)NC2CC(C)(NC(c3ncnc(C)c3C)=O)C2)cc2ncccc2n1 c12ncnc(c1C)N2.c1(CN(CC(c2ccccc2)OC)CC)cccc(Cl)c1 c1(CC)nc(C)c(C(=O)NCC2(F)CCC(CNC(c3n[nH]cc3CC)=O)C2)s1 C(CCCC(=O)NCC1C=CCN1C(=O)CC1CC1c1ccccc1)OCC Cc1ccccc1SCC(=O)NCC1CC2CC2N1C(=O)Cc1sc(O)nc1O c1(C(N(CCOC)CCNC(=O)CCC2(C(=O)C3CC3)CC2)=O)cscn1 CCCC(CCCNC(c1sccc1C(C)C)=O)NC(=O)C(C)C(F)F N1(C(CCCSC)=O)CCC(C(C)NC(=O)CC2CCC=CCC2)CC1 c1(C(=O)OC)cccc2c1OC(F)(F)O2.C(=O)N(CC)CC1CC1 Cc1nnc2n1CCCC2C(=O)NC1CCN(C(=O)CN2CSCC2=O)C12CC2 N1(C(c2ccoc2Cl)=O)CCC2CCCN(C(=O)COCC(F)(F)F)C2C1 N1(C(=O)CC2CCOC2)CC2C3CCC(C2C1)N(C(=O)CC(=O)NC1CC1)C3 c1(C(=O)NC2CC(CC(=O)NC3C(C)CC3)C2)ccc(N2CCOCC2)cc1 C=CC1(C(=O)NCC[Si](C)(C)C)CCN(C(c2ccn(CCC)n2)=O)C1 N1(C(CCC=C)=O)CC(NC(=O)C(C)(O)Cc2ccccc2)CC2(CC2)C1 c1(CCCC(=O)N(C(CNC(CC(CC)C)=O)C2CC2)C)nc2ccccc2o1 C1(C(=O)NCc2ncnn2C(C)C)(COC)CN(C(c2cccn2C)=O)C1 C#Cc1ccc(OC)c(C(N2CCC(CNC(=O)Cn3cnc(=N)[nH]3)C2)=O)c1 C(C(C)C)(C(O)C(=O)NCCC1CCN(C(C2CC3(CCC3O)C2)=O)C1)OC C1(C(=O)NC)Cc2c(O)cccc2N1CC1(C(=O)NC2CCC(C)(C)CC2)CC1 Cc1cc2c(cc1Cl)C(NC(=O)CCOCC1CCCC1)CO2 C(=O)(CCC(C)(C)F)N(C(CC1CCC1)C(N1CCCCC1C1CCC1)=O)C c1(OC)cccc(C#N)c1C(N1C(CNC(c2ccc(OC)cc2)=O)CCC1C)=O N(C1CCCc2nn(C)cc21)OC.C1(OC)CC(CNC(=O)N)CC1OC C12(NC(C3CC34CCC4)=O)CCCC1(F)CN(C(=O)C(F)(F)C(F)F)C2 c1(C(=O)NCC(CC)NC(=O)CCOC2CC2)cncc(C(F)(F)F)c1 Cn1cnc(C(N2CC(C(N)=O)(CNC(C3(n4cc(Cl)cn4)CC3)=O)C2)=O)cc1=O C1(NC(CSCC#C)=O)(CNC(C2CCCC(O)C2)=O)CCCCC1 C1(NC(=O)Cc2sc(O)nc2O)CS(=O)(=O)CC1NC(c1ccnn1C(F)F)=O C1(C(C)=O)CC(=O)N(CC(=O)Oc2nc(C)c(-c3ncoc3C(F)(F)F)s2)C1 C1(NCCNC(c2c(C)nn(C3CCC3)c2)=O)CC(N=c2ccc(C#N)c[nH]2)C1 N1(C(CCCNC(C2=C(C)OCCC2)=O)=O)CC2CN(C)CC2(C)C1 C(=O)(C1CCc2ccccc21)NC(CNC(=O)CC(=O)COC1CCCOC1)CO Cc1cc(C(N2CC3CC3(CNC(C34CC(C#N)(C3)C4)=O)C2)=O)cc(C)c1Cl c1(C(N(CCC(=O)N(CC(C)C)C)C)=O)ccc2occc2c1 C(=O)(C1CCCc2nncn21)NC1CC(N(C(C=Cc2c(C)coc2C)=O)C)C1 c1(NC2CN(C(COc3c(F)ccc(C)c3)=O)CC2C)cnc2[nH]nnc2c1 C1(C(N2CC(C(N)=O)C2)=O)COCCN1C(=O)CCc1cncnc1 c1(CN(C)C(C2CNCCOC2)=O)cc(Br)cc(F)c1O C(=O)(CCCC(C)(C)C)NCC(CC)N(C(=O)CCc1cccc(O)c1)C C(C1=CCCN(C(=O)C=CCF)C1)NC(C(CCC)OC)=O C1(CCCC)CCN(C(=NCC(O)c2c(C)oc3ccccc23)NC2CC2)CC1 c1(OC)nc(C)cc(=NC(=O)C2CN(C(=O)CCc3ccoc3)CCS2)[nH]1 C1(NC(c2c(C)cc(F)cc2)=O)C2COCC1CN(C(c1ccc(C#N)[nH]1)=O)C2 CC1(C)CCN(C(=O)CC2CCC2)C(C(=O)NC2(C)CCC(=O)NC2=O)C1 c1(C(C)C)nc(NCC(C)C(F)F)cc(=NCc2cncc(C(F)(F)F)c2)[nH]1 c1(NC(CCC=C)C)nccc(=NCCc2ccc(C#N)cc2)[nH]1 N1(C(C2CC(OCC)C2)=O)CCC(C(C)(C)NC(=O)C=CC2CCCN2C)CC1 N1(C(CNC(c2cccs2)=O)=O)CC(CNC(C2CC3CCC2O3)=O)C(O)C1 c1(CCC(=O)NCC2(F)CC(NC(=O)CC3CCCO3)C2)ccc(O)cc1 c1(CC)ccc(C(N2CCOCC2CNC(=O)CC2COCCN2C)=O)cc1N C12(NC(C(C)c3cccs3)=O)CCCC1N(c1ncnn3cccc13)CC2 C1(CNC(c2cc(C)cc(Cl)n2)=O)CC2COCC2N1C(C1CCCSS1)=O C(CC1CC1)(CC(=O)N=c1ccn(C2CCC2)[nH]1)N(C)C(c1ccncn1)=O C=Cc1cncc(C(=O)NC2C3CCC2N(C(c2cnc(C(C)C)o2)=O)C3)c1 c1(C(N(CC=CC(=O)NCC(C)Cn2cccn2)C)=O)csc2cc(Cl)cnc12 c1(CC)ccc(CNC(=O)C(Cn2cncn2)NC(=O)OC(C)(C)C)o1 N1(C(C2CCCN(CC)C2)=O)CCC(C)N(C(c2ccc[nH]2)=O)CC1 N1(C(c2c(OCC)cccc2)=O)CCN(C(c2[nH]cnc2CC)=O)CC2(CC2)C1 Cc1nn(C(C(CO)C)C)c(C)c1C1CC1.c1(C(C)N)nc(S)no1.CCCCF c1(C(=O)OC)cc(C(=O)OC(=O)CC2CCC(=O)NC2)ccc1OC CC(C)(CC(=O)NC1CCCN(C(=O)CSCc2ncc[nH]2)CC1F)CC(F)F c1(N2CC(C)(NC(C(C)NC(=O)NC)=O)C2)c(C(N)=O)cccc1[N+](=O)[O-] C12(C(=O)O)CN(Cc3c(O)sc4ccccc34)CC1CCCO2 Cc1c(C(N2CC(NC(=O)C(C#N)=CC3CC3)C(C)C2)=O)ccn1C(C)(C)C C(=O)(CC1=CCCCC1)N1CCCC(NC(C2CC(=O)N(c3cccnc3)C2)=O)C1 C12(C(N3CC(NC(C4(CCOC)CCCCC4)=O)C3)=O)CC3CC(C(=O)N1)C2C3 C(=O)(CC1COc2cc(O)ccc21)N1CCC(N(C(c2[nH]cnc2C)=O)CC)C1 C#CCC(C)(C)C(=O)NCC(CO)NC(=O)Cc1cccn1C Cc1nc2ccc(C(=O)Nc3cc(-c4cccc5[nH]ncc45)ccn3)cc2[nH]1 c1(CC(=O)NCC(O)CNC(=O)CC(O)C2CCC2)cnc(C2CCCC2)o1 Cc1ncc2n1CCC(C(=O)NCC(O)CCNC(=O)CC(C)(C)C(F)(F)F)C2 c1(C(=O)NCC2C=CCN2C(=O)C=Cc2ccccc2Cl)ccc(C#N)c(O)c1 C(N=c1cc[nH]cc1[N+](=O)[O-])c1c(OC)cc(OC)cc1 C1(CCC(=O)O)CON(C(=O)COc2cn(-c3ccc(F)cc3F)nn2)C1 c1(C(N2CCC(O)(Cc3ccsc3)C2)C(=O)NCC)nn(CC(F)(F)F)cc1C C(=O)(C(C)P(C)(C)=O)N1CC2C(CNC(CC(c3ccc(C)cc3)C)=O)C2C1 C(c1c(Cl)nc2sccn12)=CC(=O)NC1CN(C(c2cc[nH]c2)=O)CCC1CO N1(C(C2C(C)(CC)C2)=O)CC2=C(C1)CN(C(=O)CC1(OC)CCOCC1)C2 Cc1cnc(F)cc1C(=O)NCCOC1CCN(C(=O)CC2(C#N)CCC2)CC1 C(=O)(CCCCC(F)F)NCC1(O)CN(C(C=Cc2nnn(C)n2)=O)C1 C1(C(=O)NC(CC)(C)CNC(=O)C(Cl)=CCl)CCn2nnnc2C1 C1(CC=C)(C(=O)N(C)CCn2cncn2)CCCN1C(=O)CC1CCCOC1 C1(C(=O)NC23CC(NC(C45CC(CO4)C5)=O)(C2)C3)CCc2nn[nH]c2C1 C1(C(N(C)CC2(NC(c3nncn3C3CC3)=O)CC2)=O)CC2(CCCC2)C1 C1(C(=O)NC(CNC(c2cc(C(=O)OC)ncc2)=O)C2CC2)CC2CCC(C1)C2 c1(OC)ncc(C(=O)N(CCCNC(=O)CCSc2ccc(Cl)cc2)C)c(C)n1 CCC(CC(F)F)C(=O)N1CC(NC(c2cc(C(N)=O)cc(C)c2)=O)CC1C C1(NC(c2c(CCC)occ2)=O)CN(C(=O)C(c2ccccc2)N(C)C)CC1O c1(OCC#C)ccc(C(=O)NC(C)CN(C)Cc2ccoc2CCC=C)cc1 c1(C)cc2c(s1)CCC(C)C2.N1(C(C(C)=CC)=O)CC2C(C1)c1cn(nn1)N2 C1(CC)CCOCC1Nc1ccc(-c2cncc(OC)n2)nc1 C1(C)(C(N(C)C2CC2)=O)CCCN(CC(N2CCCCC2c2cc(F)cc(Cl)c2)=O)C1 c1(OC)ccc2cc(C(=O)NCC3CCN3C(=O)Cc3ccc(C)cn3)sc2c1 C12(C(N3CCC(NC(CCc4onc(CCC)n4)=O)CC3)=O)CCCC(C1)OC2 C1(C(=O)NC(CCNC(C(C2CC2)OCC)=O)C)CCCC2(CCC2)O1 C1(C)(NC(C(=O)NCCN(C)C2CC2)=O)CN(C2CC2)C(=O)O1 c1(C(=O)NCC(CC)NC(=O)CCCC(C)=O)nc(Cl)ccc1OC(C)C N1(CC(N2C(CN(C(=O)C=Cc3ccco3)CC)CCC2)=O)CCC(C)CC1 C1(OC(C)(C)C)CCN(c2ccc(NC(=O)NCC34CCC(CC3)O4)cn2)CC1 C12(CNC(C(C)=C3CCCC3)=O)CC1CN(C(=O)Cc1sccc1Cl)C2 C12(NC(CCC(C)OC)=O)CCC(C1)N(C(C1(c3ccccc3)CCCC1)=O)C2 CC1CCN(C(=O)COCCNC(=O)CC2(CO)CCC2)C1 C(N=c1[nH]c2c(c(=NC3CC4CC5C(C4)C35)[nH]1)CSC2)C12C=CCC1C2 C(=O)(C(C)(C)COCC(F)F)NC(C)C(C)NC(c1ccncc1F)=O N1(C(C(C)N(C)C)=O)CCC(C2CN(C(C3(c4ccc(C)cc4)CC3)=O)C2)CC1 N1(C(CC(CC)c2ccccc2)=O)CCN(C(c2ccc(C)nc2C)=O)C(CO)C1 c1(C(N(C2CCN(C(c3ccc[n+]([O-])c3)=O)C2)C)=O)ccc2c(C#N)c[nH]c2c1 C1(C(N(C2C3CN(C(c4ccn(CC)n4)=O)CC32)C)=O)CCc2c(cnn2C)C1 N1(C(C2(NC(c3nccc(C#C)c3)=O)CC(O)C2)=O)CC2CCC(O)CC2C1 C1(COC)CCOC2(CCCC2)C1.N12CCN(CC(O)C1)C(=O)c1ccc2nc1 C1(C(N(CC2CCN(C(CSCCCC)=O)C2)CC)=O)CCC(C(N)=O)N1C C(=O)(C(O)C(F)(F)F)N1CC(NC(=O)CCCCc2ccc(Br)cc2)C1 N1(C(CC2C(C)=NNC2=O)=O)CC2CCN(C(=O)CCC3OCCO3)C2C1 Cc1cc(C(F)(F)F)cc(C(=O)NC(C)CC(C)NC(=O)C=CC2CCCC2)n1 C1(CC(=O)NCC2CCCN(C(=O)COc3cnn(C)c3)C2)(OC)CCCCC1 C(=O)(C(CC(N)=O)NC(=O)CC1CC(=O)C1)NC1CCN(C(C)=O)CC1 c1(C(=O)NCC(C)C(F)C(=O)NCC(c2ccncc2)C)cncc2[nH]ccc12 c1(C(=O)NC(C)CCNC(c2ccc3c(c2)COC3)=O)ccc2c(c1)C(C)CO2 N1(C(c2cnc(OC)c(Cl)c2)=O)CC2CC1CCC2NC(c1cc(Cl)c(Cl)s1)=O N1(C(c2c(C)cccc2O)=O)CCCC(C2CN(c3ccncn3)C2)C1 CC1=CCC(N=c2ccc(Br)c(S(=O)(=O)NCCn3ncccc3=O)[nH]2)CC1 c1(CC)cccnc1C(N1CC(OC)C(NC(C2CC2C(C)C)=O)C1)=O C=C(C)C1OCCC1CNC(=O)CC1COC(CNC(=O)CC(C2CC2)C2CC2)C1 c1(CSCCn2cc(C(=O)OCCOC)nc2)nc(C)c(OC)n1C c1(C(N2CCN(C(CC(C)C(F)F)=O)CC2CC2CC2)=O)c[nH]c2ncccc12 C1(C)(COC)CCC(NC(C(OCC)NC(N)=O)=O)CC1.C1(=O)CCN1 CCCC(O)(CCC)CC(=O)NC(C)C(CO)NC(c1cnn(C)c1SC)=O C(=O)(C(C)C(O)C(C)CC)N(C(C)CNC(c1ccccc1)=O)CC c1(CCC(=O)N(CC(CC)NC(C2CCC(=O)O2)=O)C)cncc(F)c1 CCCCCC(O)CC(=O)NC12CC(NC(C3CC(N4CCCC4)C3)=O)(C1)C2 c1(C(c2nnnn2C2COC2)NCc2cn(CC)nc2C)cccc2cccnc12 C(=O)(C1=C(C)N(C)c2ncnn2C1)OC1CCN(C(c2c(OCC)c(C)cs2)=O)C1 N1(C(=O)NC2CCN(C3CCC34CCCC4)C2)CCC(C2=NOCC2)C1 C(C(CCCC)NC(=O)Cn1ncnn1)NC(C(F)=CCC)=O C(CCO)(C(=O)N1CCOC(CNC(=O)C=Cc2ncc(C)[nH]2)C1)N(C)C C1(C(=O)NCCN(CCOC)C(C2(C)CCCCC2)=O)COCCC1(F)F Cc1nc2ccccc2cc1C(=O)NC1COCCN(C(C2(C(N)=O)CC2)=O)C1 N1(C(C2C(=C)CC2)=O)CCCC(C(=O)NCC2CCN(c3nnc(C)s3)CC2)C1 C(=O)(C1CCCn2nccc21)NC(CCCNC(C1N(CC)C(=O)CC1)=O)(C)C N1(C(CSCC=C)=O)CCC2(C1)OCc1ccccc12 C1(CNC(Cc2c(C)ccs2)=O)CC(C)(C)CN1C(C1CC12CCOC2)=O CCCC(CNC(=O)Cn1nc(C)cc1C)C(=O)NCC1(C2CC2)CCC1 C1(C(N(C)CC2CCCN2C(=O)CC2CCC(=O)C2)=O)CC12CCOC2 N1(C(C(F)=CCC)=O)CCC(C(N2CCC(CC)(COC)C2)=O)C12CC2 C(C)(CC(C)NC(c1nnn(C)c1COC)=O)NC(CNC(=O)OCC)=O c1(CC)nc(C)c(C(=O)NCC(C(C)(C)C)NC(=O)CCC(C)N(C)C)o1 c1(NC(C(c2cccs2)NC(C2CC=CCO2)=O)=O)ccc2nccn2c1 CC(C)C(F)(CNC(=O)CSCC1CCC2(CCC2)CO1)C(=O)NCC(N)=O c1(-c2cc(C(=O)NC3CC(N(C(CCC=C=C)=O)C)C3)on2)cccc(C#N)c1 C1(CN(C)C(c2cccnc2I)=O)CCN(C(=O)CS(=O)(=O)N2CCCC2)CC1 C1(NC(CC(CC)(F)F)=O)CCN(C(c2nocc2Cl)=O)C12CCC2 Cc1cc(N)n(CC(N2CC(CNC(c3sccc3C)=O)C(C)C2)=O)n1 C1(CC(=O)NC(CCNC(C2(C(=O)NC)CCC2)=O)C(C)C)CCCC(C)(C)C1 C1(C(N2CCC(N(C)C(C3COCCO3)=O)CC2)=O)(COC)CC=CCC1 N1(C(CC=CCC)=O)CCC(C)CC1CNC(=O)Cn1ccc(C)cc1=O C(c1ccccc1F)=CCC(=O)NC1CC(CNC(C(CC)(C)C)=O)C1 c1(NC(=O)NC)cccc(C(N2CC(NC(C3SCCC3C)=O)C2)=O)c1 N1(C(C(c2ccc(C)s2)C)=O)CCC2(CCC(NC(=O)CCC3CCC3)C2)CC1 C1(C(=O)Nc2cn(CC(C)(F)F)nc2)CCCCC(F)(F)C1 C(=O)(C(F)=C(C)C1CC1)NCC(C)NC(C=CCCC)=O C1(NC(c2ccc(-c3ccc(Br)cn3)cc2)=O)CN(S(=O)(=O)C(Cl)(Cl)Cl)CC1F CP(C)(=O)c1cnc(C(N2CCC2CNC(c2sc(C#N)cc2Cl)=O)=O)nc1 CC12CN(N3CCC3CN(CC3(C)CCOC3)CCO)CC1(CCCOC)CC2 C#Cc1cnc(NC(C2CCC(NC(c3c(C)cccc3C)=O)C2)=O)cn1 C12(CNC(c3nccc(C)c3)=O)CCCC1N(c1nn3cc(C)nc3s1)CCC2 C(c1ccc(C)cn1)=CC(=O)NC1C(NC(C(CCC)C)=O)CCC1 C1(C2(O)CN(C(c3ccc([N+](=O)[O-])o3)=O)C2)(CNC(C=NOC)=O)CC1 C1(C(N2C(C(=O)NCC3CCCCO3)CSCC2)=O)CC2C(C1)C2(F)F c1(C(=O)N(C(C)CCNC(=O)CC2CC(NC)C2)C)cccc(C(N)=O)n1.CO C1(NC(c2c(COC)noc2)=O)CCCN(C(c2cnc(N(C)C)cn2)=O)C1C C1(CNC(=O)CSCC2CCCO2)CN(C(c2cnccc2Cl)=O)CCCO1 c1(C(=O)[NH+](Cc2c(C(=O)NC3(C)CCC(C)C3)n(C)nc2)[O-])n[nH]c2c1CCC2 c1(C(C(=O)NCCCOC)N(C(CC)CC)C)c(C)noc1C c1(C(=O)NC(C(C)C)C(C)NC(C2(O)CCCCCC2)=O)ccsc1S(C)(=O)=O c1(NC(c2cc(-c3nc[nH]n3)ccc2F)=O)c(F)cc(F)cc1Br C1(CC)CCN(C(C2CC2CC)=O)C1CNC(=O)CC1(F)CC1 c1(NC(C2(NC(CC3CN(C)C3)=O)CCOC2)=O)cn(C)c(=O)nc1O c1(NC(C(C)C)CCO)ccc(S(=O)(=O)N2C3CCCC2CC3)c2ccncc12 C1(C(N(C(CC)C)CCOC)=O)C2CN(Cc3ccc(O)nc3)CC12 c1(NC(C2NCCN(C(c3n(C)ccc3)=O)C2)=O)cccc2c[nH]nc12 c1(C(N2C(C(C)NC(C(CC(C)C)C)=O)CCC2)=O)cccc2c1NCC2 C(=O)(C=CS(C)(=O)=O)NC(C)CCNC(=O)CCC1NC(=O)NC1=O Cc1ccc2c(CC(N3CC(CNC(C4C=CCCC4)=O)C(C)C3)=O)c[nH]c2c1 C(c1ccccc1F)=CCC(=O)NCCC1CCCN1C(=O)CCc1nncs1 N1(C(C2(CCOC)CC2)=O)CC(NC(=O)CN2C(=O)CN(C)C2=O)CC(O)C1 N1(C(=O)Cc2ccc(F)c(F)c2)CCC2(CC(NC(=O)C(F)(F)C(F)F)CO2)C1 N1(C(C2N(C(C3C(C)(C)C(F)(F)C3)=O)CC=CC2)=O)CCC12CC(C)(CO)C2 C1(C(=O)NC(C2N(C(Cn3ncc(CC)c3)=O)CCC2)C)C2CCCCCCC12 C12(C(=O)NC3CCC(NC(CN(CC)CC)=O)CC3)CCCCC1CS(=O)(=O)C2 c1(C(N(C(C)C)C(C2CCCCO2)Cc2nc(C(=O)O)n[nH]2)=O)ccc(Cl)cn1 C(=O)(C(C)(O)C(F)(F)F)NCCCCNC(Cn1ncc(C)c1)=O c1(C(=O)NCC2N(C(CC3(C)CCCO3)=O)CC=C2)ccn2nnnc2c1 Cc1cc2ccc1c(=O)[nH]2.n12cnnc1C2.C1(C(N)=O)CCOCC1 CC(C)C(C(=O)N(C1CCCCC1O)C)NC(=O)COc1cccnc1 CS(=O)C1CN(C(c2cc(CNC(=O)Cn3cc(CO)nn3)no2)=O)C1 CC(=O)CCCC(=O)N1CCN(C(c2csc(C)c2N)=O)C(c2cn[nH]c2)C1 CC1C(C)N(C)CCN1C(=O)C(CCF)NC(C12CC(CO)(C1)C2)=O c1(CN(C(=O)C(=O)N(C)CC2CC3CCC2C3)CC=C)ccc(F)cc1 c1(C(N(CC(C)CNC(C2CC23CC(F)(F)C3)=O)C)=O)cccc2[nH]ncc12 C1(C(=O)NCCC(=O)NCC)CCCC(CNC(=O)COc2ccncc2)C1 N1(C(=O)C=CC2CCCC2)CC2(C1)CN(C(=O)CC(O)c1ccccc1)CC2CO N1(C(C(C)NC(N)=O)=O)CCCC12CCN(C(=O)Cn1cnc([N+](=O)[O-])n1)C2 CC1COC(C(=O)NC(C)(C)CN(C)C(c2csc(C(F)F)n2)=O)C1 Cc1nn2ncccc2c1C(=O)NC1CC2CC1CN2C(C1(NC(C)C)CC1)=O Cc1ncc(CCC(=O)NCC23CC(NC(=O)CCc4cn[nH]c4)(C2)C3)o1 c1(C(F)(F)F)cn2ncnc(NC3CCNc4sccc43)c2n1 c1(C(=O)NCC(C)CN(C)C(c2nn(C)cc2C(C)=O)=O)nc2ccccc2[nH]1 C12(C(=O)NCc3cc(CC)[nH]n3)CC(CN1C(=O)C(CN(C)C)N(C)C)C2 N1(C(c2c(C)nc(CO)nc2)=O)CCN(C(=O)CC2CNC(=O)C2)CC12CCC2 C(CCCCCCCO)=CC(=O)NC12C(NC(C=C(C)C(F)F)=O)CC(CC1)C2 N1(C(CCCOc2c(C)cccc2)=O)C2CC1CN(C(=O)CCC(C)(C)F)C2 c1(C(=O)NC2(CO)CCCN(C(C(C)OC)=O)C2)cc2cccc(C)n2n1 c1(C(=O)NCC(CO)NC(C#CC(C)(C)C)=O)c[nH]ccc1=Nc1ccccc1 Cc1cc(Cl)c(C(N2CCC(NC(=O)CN3CCCCCC3)C(C)C2)=O)cc1F CC(C(=O)N1CC(NC(C2(C(F)F)CCCC2)=O)C(F)C1)C(C)(F)F N1(C(c2c(OC)csc2)=O)CCN(C(=O)Cc2cc(Cl)n(C)n2)CC1CC(F)F C(C(F)(F)F)(C(F)(F)F)CCn1nccc1-c1cnc(C2C(n3ncc(C)c3)C2)nc1.OC C1(C(N2CCCC(C(F)F)C2)=O)CC(F)(F)CN1C(C1CCOC1)=O C1(CNC(CN(C)CC)=O)C=CC(NC(=O)CCCSC(C)(C)C)C1 CCCCCCC(F)C(=O)NCC(O)CCNC(c1cn(C)[nH]c1=N)=O N1(C(C2(c3cccc(Cl)n3)C(NC(=O)OC(C)C)C2)=O)CCOC2CC12 N1(C(c2cnc(OC)s2)=O)CCC(CO)(CNC(=O)C(N2CCN(C)CC2)C)C1 c1(NC(C2CC(CC#N)C2)=O)cc(=NCc2cnc(C(F)(F)F)s2)[nH]cn1 c1(C(N(CC(CC)NC(C(CCC#C)O)=O)C)=O)c(C)c(C)cc(C)c1C N1(C(c2c(C)nc(C(F)(F)F)s2)=O)CC(C)N(C(c2ccc(C#N)o2)=O)CC1C n1(CC(=O)NCC2(F)CC(NC(CC3C(=O)NC(=N)S3)=O)C2)ccc([N+](=O)[O-])n1 c1(OC)ccc(NC(C2CN(C(C34CC(F)(C3)C4)=O)C2)=O)c(Br)c1 C12(CC(=O)N(C(C(=O)NCC3(O)CC(CO)C3)C3CC3)C)CCCC1C2 C1(C(=O)NC(C(C)C)CCNC(c2ccc(=O)n(C)c2)=O)CCCC1S(C)(=O)=O Cc1ccc(C(N2CC(NC(C3Cc4nncn4C3)=O)CC2(C)C)=O)c(O)c1 C1(S(C)(=O)=O)(C(=O)NCC2CN(C(C3=C(C)OCC3)=O)C(C)C2)CCOCC1 c1(C(C)(C)C)ncc(C(=O)NCC2CCN2C(C2CN(c3nncs3)C2)=O)s1 C1(C(NOCC=C)=O)COC(C)C1.c1(C(=O)SC(C)CN)c[nH]c(C(N)=O)c1 C12(C(=O)NCCC3CN(C(C(C4CC4)OC)=O)C3)C=CC(CC1)C2 c1(CCC(=O)N(C2CCN(c3cnc(F)cn3)C2)CC)cccc(F)c1F CC(C)C(O)C(F)(F)C(=O)N1CCC2CN(C(c3cccc(F)c3O)=O)C(C)C12 Nc1cc(Br)cnc1C(=O)NC1CCCN(C(C2(C(F)(F)F)CCC2)=O)CC1 CC1=NN(C)C(=O)C1CC(=O)NC1COCCN(C(C2CCOC(C)(C)C2)=O)C1 N1(C(C2(OC)CCSC2)=O)CCN(CCCNC(C2(C)CCNC2=O)=O)CC1 C(=O)(C(Cc1ccccc1)NC(C1CCCN1C(=O)Cc1ccco1)=O)OC c1(CN2CCC(NC(Cc3c(C)noc3C)=O)C(O)C2)cc(Cl)cc(Cl)c1O Cc1cc2nc[nH]c(=NCC3CC(CNC(c4cc(CF)on4)=O)CO3)c2[nH]1 Cc1ocnc1C(=O)NC(C1(O)CN(C(c2sccc2C(F)F)=O)C1)C CCC(F)(C(=O)OC)C(=O)N1CC2CC1C2CNC(=O)C(c1cccc(C)c1)O C=CC(C)(C)CC(=O)N(C)CC1CCC(CNC(C23CCCC2C3)=O)CC1 N1(C(c2c(SCC)cccc2)=O)CCCC(COC)(NC(=O)C#CC(C)(C)C)C1 Cc1cc(NC(=O)CC2CCCCC(=O)N2)ccc1NC(=O)CS(N)(=O)=O C1(C(N(CCCNC(C=C2CCC(C)CC2)=O)C)=O)CCC2C(CC1)C2(F)F N1(C(C(CC(C)C)NC(=O)CC2CCC(=O)CC2)=O)CCCC(C)(C)C1C c1(CCC(=O)N(CCCNC(c2csc(O)n2)=O)C)cc(F)cc(F)c1 N1(C(CC2(OC)CCC2)=O)CC(CNC(=O)CC2(C#C)CCC2)C(O)C1 c1(C(N(CC(C)(C)CNC(=O)CN(CC(C)(C)C)C)C)=O)cn(C)ccc1=O c1(Nc2c(SCCC(=O)OC)cccc2)ncc2[nH]ncc2n1 C(C(C)(C(N)=O)NC(c1cc(CN(C)C)c[nH]1)=O)NC(C1(CC)CCCCC1)=O C(=O)(CC(C)CC(C)(C)C)N(C)CC1N(C(Cc2cn(CC)nc2)=O)CCCC1 C1(N(C(=O)CN(C)C(N)=O)CC)CCCN(C(=O)CC2C=CCCC2)C1 C1(N(CCC)C(C2CC(OCC3CC3)C2)=O)CCN(C(=O)CCSC)C1 Cc1ccc(OCC(=O)NCCC2CCCN2C(=O)Cc2ccc(F)nc2)cc1 C1(NC(CN(C2CCC2)C(C2(CC=O)CC2)=O)=O)CC2(CCCC2)C1.COC C1(C(=O)NCCCCN(CC(C)C)CC)CCC(C)(C)N(C(c2ccoc2)=O)C1 C1(c2cnn[nH]2)(C(=O)NC(CC)CNC(=O)C=C(C)C(F)F)CCCCO1 C(=O)(C1=NOC(c2ccccc2)C1)NCCCNC(C(c1cnccn1)C)=O CC1CN(C(c2cnn(C)c2N)=O)CCCN1C(C1C2(CC2)C12CC2)=O CS(=O)(=O)c1ccc(Cl)c(C(N2CCN(C(=O)CCOC3CC3)C(CO)C2)=O)c1 c1(C(=O)NCC(CO)NC(c2cccc(OC(C)C)c2)=O)n[nH]c2c1COC2 C1(C(C)C)CNC(=O)CN1C(=O)CCCC(=O)c1cccc(Br)c1 C12(NC(C#CC(C)C)=O)CCCC1N(C(=O)CSCc1csc(=N)[nH]1)CC2 N1(CC)OCC(NC2CCOC(c3ccncc3)C2)C1=O CC1CC(CC(N2CCC2CC2CC2)=O)CN1C(=O)Cn1cccc1 c1(CC(CC)NC(=O)C(c2cccc(F)c2)C)ccc(O)cc1 c1(C(N2CCC(C(C)NC(c3c(C)coc3)=O)C2)=O)cc(C(N)=O)ccn1 C1(C(=O)NC(c2ncccn2)C2CCCN2)Cc2ccccc2O1 N1(C(Cc2c(C)noc2)=O)CC2(CC2)CC1CNC(=O)C(C)Cc1ccco1 C1(Nc2ncc(C#C)cn2)CC2CC(C1)N(C(C1CCCCC1C(F)(F)F)=O)C2 C1(C(N2CC(C(C)NC(=O)CCCn3ccnc3)C2)=O)C(C)(C)C1(F)F N1(C(c2cn(CC)nc2C)C(=O)NC(C)C)CCS(=O)C(C)C1C C(=O)(CC(C)C(F)(F)F)NCC(=C)CCNC(=O)Cc1cccc(C2CC2)c1 CC(CC(=O)NC1CN(C2CCC2)C1)NC(=O)CCC1CC1(F)F n1(CCC)ncc(CCCCCCOCC)c1C.C(C(C)(C)C1CC1)(c1nnnn1C1CC1)N c1(CCC(=O)NCCN(C(c2c(NC)c(F)ccc2)=O)C)cccc([N+](=O)[O-])c1 c1(C(=O)OC)ccc(C=CC(=O)NC2CCC(NC(=O)CC3(C)CCC3)C2)cc1 n1(CC)cnc2c(NC(C)CC(N)=O)[nH]c(=NC(C)c3ccccc3)nc12 N1(C(c2c(C)n(C)nc2)=O)CC(O)(C2CCN(C(=O)CC3CC3(Cl)Cl)CC2)C1 C#Cc1cccc(CC(=O)NC(C)(CO)C(=O)NCC=CBr)c1 c1(C(N(C)CCO)=O)cc(Br)c([N+](=O)[O-])[nH]1.n1(CCN(C(=O)O)CC)cc(C)nn1 c1(C(C)C)ncc(C(=O)NCC(C)N(C(=O)C=CCO)C)n1C c1(NC(C2CCN2CC(N2CCSCC2)=O)=O)cc(O)cc(Cl)c1 c1(C(CC)C)nc(N(C)CC2CN(C(C3C=CCC3)=O)CCO2)cc(C)n1 C(=O)(CCCCCn1cc(CN2CCCC2C)nn1)NC(c1ncccn1)CC Cc1nc(C(N2CCCC2CNC(c2ncc3ccccn23)=O)=O)c(=O)[nH]c1C c1(C(=O)NC(C)(CNC(c2nc(C3CC3)cs2)=O)Cn2cccn2)cccc(Cl)c1 CC(CCNC(=O)Cn1ccc(C(F)F)n1)CCNC(c1cc[nH]n1)=O c1(NC(=O)NC(C2CC(F)(F)C2)CO)cccc(NS(=O)(=O)C(F)(F)F)c1 C1(NC(c2ccc(C)o2)=O)C(C)CCN(C(c2ccc(Cl)nc2Cl)=O)C1C N1(C(c2cc(C)c(O)nc2)=O)CC2CN(C(c3cc(O)nc(O)n3)=O)CC2(C)C1 c1(C(C(=O)NCCOCC)N(C(C)C(C)C)CC2CCCO2)ncc(Cl)cc1Cl N1(C(c2cn(CCC)nc2)=O)CCC2(CC2NC(=O)CC2CCCC23CC3)C1 C1(C(N(CCC)C)=O)CCCN(Cc2cccn(CC(C)OC)c2=O)CC1 c1(C(=O)NCC2C(NC(C(COCCOC)(C)C)=O)C2)cc2[nH]ccc2s1 CC1(C)CC(C(=O)NOCCCN=[N+]=[N-])(CNC(C2CC(=C3CC3)C2)=O)C1 N1(C(C(C)N(C(c2c(C(C)C)noc2)=O)C)=O)CC2(CCCC2)C1 N1(c2snc(C)n2)CCCCC(NC(=O)Cc2ccccc2OC(C)C)C1 C1(CC(=O)N(CCCC(=O)NCC2(OC)CC2)C)CC2(CCC2)C1 C=CC1(C(N2CCCC3(C2)N=N3)=O)CCN(C(=O)C(C)n2cccn2)C1 CN1CCN(C2CC(C(=O)NCc3c[nH]c(=N)o3)C2)CC1.C12CCN(CC1)C2=O C(CCC(=O)NCC1CCC1NC(c1ccnn1CCC)=O)NC(=O)NCC#C c1(C(N2CCN(C(c3c(C)cc(C)o3)=O)CC2)=O)cccc2ncnc(O)c12 C(=O)(C(C)(C)C(=O)N(C)C)N(CCC(C)NC(C)C)C.c1cc(Cl)sc1Cl O=C1CC(C(=O)NC2CN(C(c3cnsc3)=O)CCC2CO)CC(=O)N1 CCCC(F)C(=O)N1CCCC1CCNC(=O)CCC1CC(F)(F)C1 C(C1=CCN(C(c2ccn(C(F)F)n2)=O)CC1)NC(C(C)(C)c1ccncc1)=O C(C)(C)(CC(F)C(=O)N1CC(CC2CC2)C1)NC(C(Br)=C(C)C)=O C(=O)(C1=COCC1)N1CCC(N(C(=O)C(O)C2CCC2)CC#C)C1 CCCCCC(C)(CC)C(=O)N1CC(CCCCNC(=O)CC(=O)NCC)C1 C1(OC)CC2N(C1)C(=O)C=CCC(=O)NCC2.C1(=O)CN1.C(CCF)OC C1(NC(CCn2c(C)cc(C)n2)=O)CCN(C(=O)Cn2ncnn2)CC1C C(=O)(CCCC(C)(C)C)N1C(C)CC(CC(=O)NCC2(C)CC2)C1 c1(OC)ccc(C(C)NNC2COc3ccccc32)cc1S(N)(=O)=O c1(N2CCCC(NC(c3scc(C)c3)=O)C2C)ncnc2sc(C(C)(C)C)cc12 N1(C(C)C#N)CCN(C(=O)CCC2CCN(C(=O)Cc3nccn3C)C2)CC1 N1(C(CCC(=O)NC)=O)CCCC(C)(CNC(=O)CC2(OC)CC2)C1 C1(NC(C=CCCCCC)=O)CCC(C)N(C(c2cccc(C(N)=O)n2)=O)C1 c1(C(=O)NCCCCNC(C(CC(C)C)OC)=O)cc2cn[nH]c2cn1 CCCC(C(O)C(=O)NC(C(C)(C)O)C1CC1)NC(=O)CN=[N+]=[N-] CCCCCC(C(=O)N1CC2(CCC(CNC(c3cc(OC)no3)=O)O2)C1)C(C)C N1(C(c2cc(C)ncc2C)=O)CC2(CCCC2)C1C(=O)NCCC(C)N1CCC1 c1(CNC(C(C)=CCC)=O)cccc(C(=O)NC2(C)CC=CC2)c1 c1(CC)cc(C(N2CCN(C(C3CC3C)=O)C(C(C)C)C2)=O)c(C)nn1 n1(CC=C)nnnc1C(c1csnn1)NC1(c2ccccn2)CC1 C=CCCCC(=O)NCC(C)(C1CC1)NC(c1snnc1C1CC1)=O c1(NC(=O)OC(C)(C)C)cc(NC(=O)C(c2cccc(Br)n2)(F)F)cc(Cl)c1 C(=O)(CC1=CCCC1)N1C(CNC(C(c2cc(F)ccc2Br)C)=O)COCC1 N1(C(C(CC=C)NC(C)=O)=O)CCCCCCC1C(=O)NC1(CO)CC(F)C1 c1(C(=O)NCCC2N(C(CC(=O)NCC#C)=O)CC(OC)C2)cn2c(n1)SCC2 C#CC1(C(=O)NC2(c3cc[nH]n3)CC2)CCN(C(c2ccncc2N)=O)C1 C1(NC(c2c(C(C)NC(C(CC)=CC)=O)noc2)=O)(CO)CCC(C)C1 N1(CCNC(CS(C)(=O)=O)=O)CCCCN(C(=O)CS)CC1.C1(SC)CCCC(F)C1 c1(C(=O)NC(C2CCCN(C(=O)CCc3cnn(C)c3)C2)C)ccnnc1O n1(COC)nc(S)ccc1=O.C1CCCC1 C1(NC(c2cnc(CCC)s2)=O)CCN(C(=O)C2CC2)C12CCCC2 Cc1oc(CO)cc1C(N1CCC(CNC(=O)C(C)Sc2ccccc2Cl)C1)=O C1(C)(CNC(c2n(CC)nnn2)c2cn(C3CC3)nn2)CCC(=O)NC1 c1(C(=O)CCN(C(c2nc(C)no2)CC)C(C)(C)C)cc(-c2cccs2)[nH]n1.OC c1(OC)cc(C(=O)NC2CC(O)CN(C(=O)Cc3cnns3)C2)ccc1O C1(C)(CNC(CNC(c2n(C(C)C)ccc2)=O)=O)CCCCC1O C(CCC(C)(C)C)(c1n(CCCC)nnn1)NCc1cc2c(s1)CCC2 CN1CC(O)CCC1CNC(C1CCN(C(=O)C=CC(=O)N(C)C)C1C1CC1)=O c1(C(N2CC(c3ccccc3)(N(c3ccn(C)c3C)C(C)=O)C2)=O)cnc(O)cc1C c1(CC(N)=O)ccc(NC(=O)CC2CN(C(c3cc(Cl)ncn3)=O)CCO2)cc1 CN1C(=O)C(=O)N(CC(=O)NCC2(C)CCCN2C(c2ccno2)=O)C1=O C1(CC(=O)OCC(=O)NC2CC2NC(C2CCCCC2)=O)CCCOC1 Cc1nnc(CCC(=O)NC2(C(=O)NC3CCCC3F)CC(F)C2)n1C c1(NS(C)(=O)=O)ccc(O)c(F)c1.C1CCCN1C.CCOC N1(CC)CCC(NC(c2cc(CNC(=O)C(C)N3CCCC3)[nH]n2)=O)C1=O c1(-c2cc(C(=O)NCC3C(NC(=O)CC4CSCCS4)C3)on2)ccc(F)cc1 Cc1c(C(=O)NC2CN(C(C3CC3C)=O)C2)oc2ccccc12 Cc1nc(N2CCC(=CCNC(=O)C(C)CCN(C)C)CC2)c2ccsc2n1 N1(C(CC)=O)CCN(C(c2ccc(SC(F)(F)F)o2)=O)CC(C)(F)C1 N1(C(c2c(OC)nsc2OC)=O)CCCC2CN(C(c3n[nH]c(C)n3)=O)CCC12 c1(C(=O)NC2C3CN(C(C(C)OCCOC)=O)C2CC3)nccc2occc12 C(=O)(C(CO)C(C)(C)C)N1CC(C=CC)C(C(=O)NCc2cnccc2NC)C1 c1(C(=O)OC)cc(CNC(=O)CN2CCC(=O)C2C)n(C)n1 N1(C(Cc2cc(C)on2)=O)CCC2(CCN(C(=O)C(O)CC3CC3)CC2)C1 c1(-c2ccc(N)cc2)ccc2ccncc2c1[N+](=O)[O-] c1(C(N2C3C(C(=O)NC4CCC(C)CC4)C(C3)C2)=O)cccc2cccnc12 c1(C(N(CCC(C)NC(=O)CC2CC2)C)=O)ncc(-c2ccncc2)s1 C(C(C(F)(F)F)N1CCN(C(c2cc(Br)n[nH]2)=O)CC1)NC(C(C)=CC1CC1)=O C1(C(NCP(C)(C)=O)=O)CCCC(NC(C2(C(C)(C)OC)CC2)=O)C1 C1(NC(c2cc(C(N)=O)no2)=O)CCSC12CN(C(=O)CC1CCOC1=O)C2 c1(C(=O)NCCC2CCN(C(Cc3n[nH]c(=N)s3)=O)C2)ccc2cnoc2c1 C1(C(N(C2(COC)CC2)C)=O)CCN(C(=O)CSC(F)(F)F)O1 c1(C(=O)NCCN(C)CCOC(=O)CC2CCC(O)C2O)ccc(F)c(F)c1 CC(Cc1cnc[nH]1)C(=O)N(CC(C)CNC(=O)C(C)OC1CCCC1)C C1(NC(C(CC#C)C)=O)CCN(C(c2cc(OC)c(Br)cc2F)=O)CC1(C)C S(=O)(=O)(CCCCCCCC(=O)O)N(C(C1CCCCC1)C#C)C CCCC(=O)N(CC(=O)NCCc1ncc[nH]1)CC(C)C O(NC(=O)C(CC)NC(c1ncoc1CC)=O)CCCC#C Cn1nccc1C(F)=CC(=O)NC1CC1CNC(c1cc(Cl)sc1Cl)=O C1(S(C)(=O)=O)(C(=O)NC(C(C(C)C)NC(c2cc(=O)cc[nH]2)=O)C)CC(O)C1 C(CCO)(C(=O)NC1CCCCC1NC(c1csc(-c2cn[nH]c2)c1)=O)N(C)C C(C(N=c1c(C#N)c[nH]c2ccccc12)C(C)C)NC(Cc1nc(C)sc1C)=O C1(CC(=O)OC(=O)Cn2ccc(CO)n2)(CC#C)CCCCC1 N1(CCNC(COCC(=C)C)=O)CCC(NC(=O)C(C)C2CCCO2)CC1 c1(C(=O)NCC(N(C(CC(C)O)=O)C)C2CC2)cnc(O)c2ncccc12 c1(COCC(=O)NCCCCNC(C(C)n2cncn2)=O)cccc(Cl)c1 C1(C(=O)NC2CCCN(C(CN(C)CC)=O)CC2)CC12CCC(C)(C)CC2 c1(C(N(C2CN(C(=O)CCc3nccn3C)C2)C)=O)cc(C(F)(F)F)cnc1N c1(C(N(C(CNC(C(C)=CC)=O)C)C)=O)ccc(-c2ccccc2Cl)nc1O C1(C)(C(=O)OCC)CC2CN1C(=O)C1CC1C(=O)O2.c1(COC)cccnc1O c1(C(N2CC(CNC(C3CC34CCCCC4)=O)C2)=O)csc2c1CCCC2 c1(C(=O)OC)cc(F)c(ON(C2CCOCC2)C2CC2)c(Br)c1 C(=O)(CCS(=O)(=O)C(F)(F)F)N1CC(NC(CC(CC)(C)C)=O)C(O)C1 C1(NC(c2c(C)nccn2)=O)CN(C(C2CCC(O)CN2C)=O)CCC12CCC2 c1(CCNC(N2CC(n3ncc(COCC)c3)C2)=O)ccc2oc(C)c(C)c2c1 C1(O)(C(=O)NCCCN(c2ccccc2)C(C2(C)C(C)C2)=O)CCOC1 c1(C(=O)NC(CC)CNC(=O)CC2(C)CCOCC2)ncnc(C)c1OC N1(C(c2ccc(C)s2)=O)CC(C)OC2(CCN(C(C3CCCSC3)=O)C2)C1 Nc1c(C(N2CC(O)(CCNC(C3CCCS3)=O)C2)=O)cc(F)c(F)c1F N12CC3(CC3)CC1NCCC2.C(=O)(CCC(F)F)NCc1ccc(COC)s1 n1(CC)cnc2c(NCCCC3(C)CCC3)[nH]c(=NCC=C(C)C)nc12 C12(NC(CCCCSC)=O)CC(CNC(=O)C(O)CN(C)C)(C1)OC21CCC1 c1(COC)cc(C(=O)NCC(F)(F)Cn2cc(CO)nn2)cs1 CCCCC(CC)CCC(=O)N1CC(C)(NS(=O)(=O)c2ccc(C(=O)NC)cc2)C1 c1(C(N2C(CNC(C3CC(O)(CC#C)C3)=O)CCC2)=O)cc2cc(C)ccc2o1 CC1=C(C)CC(C(=O)N(C(CNC(=O)CS(N)(=O)=O)C2CC2)C)CC1 N1(C(COCCCOC)=O)CCN(C(=O)CCS(=O)(=O)N(C)C)CC(C)(F)C1 N1(C(CN2CCN(C(C(c3cccnc3)C)=O)CC2)=O)CCC2(CC1)CC2 c1(CC)ccc(NC(c2nnnn2C2CCOC2)C2(SC)CC2)c(C(C)C)c1 C(=O)(C=CS(C)=O)NCCC1CCN(C(C2(COC)CCC2)=O)C1 C1(C(=O)NCC2CC2C2CCCO2)CN(C(=O)CC2(O)CCC2)CCO1 CC1=C(C)CC(C(=O)NC2CN(C(C3CC(F)CN3C)=O)CC2C(F)(F)F)CC1 c1(C(=O)NC2CN(C(C3C(C(C)C)(CC)C3)=O)C2)nccc2ncccc12 N1(C(C(C)NC(C(C)=NOCC#N)=O)=O)CCCC2(CCOC2)C1 c1(C(N(C(C)CNC(c2ccc(F)c(O)c2)=O)CC)=O)cc2c(nn1)CCCO2 CC1(C)CC(=O)NC1CNC(=O)C(C(C)(C)C)NC(c1ccc(F)cc1F)=O C(=O)(C(C(C)C)NC(C)=O)NC1CC(=CCC(=O)NCC(CSC)OC)C1 N1(C(c2nc(OCC)oc2)=O)C2CCC1C1CC1(NC(=O)C(CC)n1cncn1)C2 C1(CNC(C2CN3CCCC2C3)=O)CN(C(=O)C2CC2)CCC1(F)F N1(C(C(CC#C)O)=O)CC(C(=O)NC(C)(COC)CC)C2(CC2)C1 C(=O)(C(CC(C)C)NC(C)=O)NCC(CNC(CC1(C=C)CC1)=O)OC N1(C(CC(C)C)=O)CC2CCN(C(c3cc[nH]c3)=O)CC2C1 c1(N2CC(C(=O)NCc3cccc(OCCO)c3)C3(C2)CC3)nc2ccccc2s1 C1(CC#C)(C(=O)NCC(C)C2CCC2)CCN(C(=O)CCCC#N)C1 C1(C(N(C(C)CC2CC2)C)=O)CC(C)(NC(=O)COCCCN(C)C)C1 CC1C(NC(=O)CC2(C)CCC2)CCCN1C(c1csc(C(F)(F)F)n1)=O C1(C)(Cn2cc(C(CC)O)nn2)CCN(C(c2ccncc2C(F)F)=O)C1 c1(OC)cc(C(N2CCCC(NC(=O)C(=O)O)C2)=O)cc([N+](=O)[O-])c1 C1(C)(C(=O)NC(C2CCN(C(C34CC3CNC4=O)=O)CC2)C)COC(=O)C1 C1(C(N(CC(=O)N(C(C)C(C)CC)C)CCOC)=O)CC(C)CC(=O)N1 C(=O)(CCCCCO)N1CCC(N(C(C)(C)C)C(C2CC2C2CC2)=O)CC1 C1(C(=O)NCc2cn(CC3CC3)nn2)CCN(C(=O)C(F)=CC2CC2)C12CCC2 Cc1cccc(COCC(=O)NC(C2CCN(C(C3CCCC(=O)O3)=O)C2)C)c1 Cc1ccn2c(C(=O)NC3CN(C(=O)CC4CCCOCC4)CC3C)cnc2c1 N1(C(C(C)(O)C2CC2)=O)CCN(C2CCCN(Cc3ccccc3CO)C2)CC1 CCC(C)(CCNC(c1cnc(-c2cccs2)o1)=O)NC(=O)CCc1cncs1 C1(C(N2CC(OC(C)=O)C2)=O)CCN(C(=O)c2cc(C)cc(O)n2)O1 CCCC(C)(C)CC(=O)N1CCN(C(c2cc(C#N)ccc2Cl)=O)C(C2CC2)C1 C1(NC(CCOCCCOC)=O)CCC2(CC1)CC2NC(=O)C(C)C(C)(C)C C1(C)C(=O)N1CCNC(CNC(=O)OCCCC)=O.C1(CSC)CC1 N#Cc1cccc(CCC(=O)NCCC2CN(C(C3CCS(=O)S3)=O)CCO2)c1 c1(C(N2CCCCC2C(C)CO)C(=O)NCCOC)cc(C)ccn1 c1(C(=O)NCCOC2CCN(C(C(CC)C(C)C)=O)C2)ccc2nnnn2c1 n1(CC(=O)N(CC(O)CNC(=O)CC2(O)CCCCC2)C)ccc2ccccc12 CC1=NOC(=O)C1CC(=O)NC12CC(CNC(=O)CCCCN(C)C)(C1)C2 C1(CCCC)CN(C(c2[nH]ccc(=O)c2C)=O)CCN1C(c1cnc(SC)s1)=O CCC(O)C(C)C(=O)NCC(C(=O)Nc1cncnc1OC)OC N1(C(CN2CC(CC)C2)=O)CCCC(C2(NC(C3(C(F)F)CC3)=O)CC2)C1 N1(C(C(CCC)OC)=O)CC(NC(=O)CCc2ccc(Cl)cc2)CC(F)C1 c1(OC)c(F)ccc(F)c1CN1CC(NC(c2cn(C)cn2)=O)C(F)(F)C1 C(=O)(C1CCCc2ncnn21)N(CCC)CCNC(c1ncccc1CC)=O c1(C(N2C3C(C(N4CCCC(CC)(CO)C4)=O)C(C3)C2)=O)cc(C)cc(C#N)c1 C(CCC(C)C(=O)NC(C1CCN(C(=O)C=C2CCOCC2)CC1)CO)OC c1(OCC(N2C3CCC2C(NC(=O)C(F)(F)CO)C3)=O)ccc2c(c1)CCC2 n1(CC(=O)N(C)CC2CCCN2C(c2ccnn2C)=O)sc(=N)[nH]c1=O C1(C(=O)NC(CC(=O)NCC(C)C)C2CC2)CC2(CC2)CO1 C1(F)(CNC(c2n(C)nc(C(F)F)c2)=O)CCN(C(C2(C)CC(F)C2)=O)CC1 CC1(C(=O)N(CC(N2CCOC(CC(N)=O)C2)=O)CC2CC2)CC(C#N)C1 N1(C(C(C)OC)=O)CC(C2(NC(=O)C(=Cc3cccc(F)c3)F)CC2)C1 c1(CNC2(c3n(CC)nnn3)CCC(C)C2)cccc(C(F)F)c1F N1(C(c2c(C)nc(C)[nH]2)=O)CC(CCNC(=O)CC2CC3CCC2O3)OC(C)C1 Cc1ccc(C(=O)N(C2CCN(C(c3cc(N)ccc3F)=O)CC2C)C)c(O)n1 N1(C(c2cnn(C3CCOC3)n2)C(=O)NC2(C)CC2)CCN(C)C2(CCOC2)C1 C1(COC)(NC(=O)COCC(C)C)CCCN(C(=O)C(C)C(C)(C)C)C1 N1(C(C=C(CCC)C)=O)CCCC(CCNC(=O)CCn2cc(C)cn2)CC1 CC1(C)C=CC(N)CC1.C1(OC(=N)O)CC(OCC(=O)NC2CCCC2)C1 C(=O)(CC(C(C)C)NC(C1CC(C)(C)CCO1)=O)NC(CC#C)C Cc1[nH]nc2cc(NC(c3c(-c4cnc(O)c(CO)c4)cncc3F)=O)ccc12 C1(NC(C(C2CCC2)OC)=O)CN(C(=O)C(C)(C)C#N)CC1c1ccccc1F C1(NC(COCc2cc(C)on2)=O)CC12CCN(C(=O)CCC1OCCO1)C2 CCC(O)CC(=O)NCCOCC(=O)NCC1CCC(=O)NC1 c1(C(N2CCC(C)(CCNC(CCCOCC=C)=O)C2)=O)cc(C)ccc1N c1(C(N(CC(C)NC(=O)COCC(c2ccccc2)=O)C)=O)ccn2ccsc12 O=C1CC(=O)c2cc(OC(=O)CC=C(Cl)Cl)ccc21 c1(CN(CC(C)(C)C)CC2CC3C=CC2C3)ccc(C2CC2)cc1 C1(NC(c2c[nH]nc2CCNC(C2(F)CCOC2)=O)=O)CC(O)C(O)C1 C1(NC(c2c(C)ncnc2C)=O)CCC2CCN(C(=O)C(C)n3ccnc3)C12 C1(C(=O)NCC(CC=C)(C)C)CC(F)CCN1c1c(NC)cccc1 c1(C(=O)NC2C3OCC(NC(c4c(C)occ4)=O)(C3)C2)cn2cc(Cl)cnc2n1 C(=O)(CCCCC(F)F)NC1CN(C(c2ccc(N(C)C)cc2)=O)C2C1C2 C1(OC)CN(C(=O)OC(C)(C)C)CC1C(=O)Nc1cc(-c2ccccc2)ns1 c1(C2C(C(=O)NCC(CN(C(=O)Cn3[nH]cnc3=N)C)O)C2)cnn(C)c1 C(N(C)N1CC2(C)C1C2)SC(C)C.C(C)(C)(C)OC(=O)N.C(=O)(C1CC1)NC C1(C(=O)NCC(CC)NC(CSCCCC)=O)(C(=O)NCC)CCOCC1 N1(CCC)CCCC(C(=O)N(C(C)CCNC(=O)CCc2cc(Cl)cs2)C)C1 C1(CC)(NC(=O)CC2CCCC2)CCN(C(c2c(OC)noc2C)=O)CC1 C1(NC(c2nc(C(C)NC(CN(C(=O)OC)C)=O)oc2)=O)CC(=O)N(O)C1 C1(CNC(C(C(=O)OC)(C)F)=O)CC2CCC(C1)N2C(C1CCCN(C)C1)=O Cc1ccc(C)n1CC(N1CC(O)(C(C)(C)CNC(C2CCCCN2C)=O)C1)=O N1(C(=O)Cc2cn[nH]c2)CCC(C2CCO2)CC1 CCCC(C(=O)NC(C)(C)CCNC(=O)CC1CCC(F)(F)C1)OCC C1(NC(C=C(CCC)C)=O)CS(=O)(=O)C2CN(C(c3nscc3C)=O)CC12 c1(C(N2CC(NC(c3cc(-c4ccncc4)no3)=O)C2)=O)cc(Cl)cc(Cl)c1Cl N1(C(c2cc(COCC)ncn2)=O)CCN(c2cccc(Br)c2)C(=O)C1 c1(C(N2CC(N(C(c3c(C)noc3)=O)C)C(F)C2)=O)cccc(C(F)(F)F)c1Cl Nc1c(C(=O)NCCC(F)Cn2cc(C3CCCC3)nn2)cc(F)cc1Br c1(C(=O)NCC2CC(NC(c3cc(C)sc3C)=O)CC2O)ccsc1S(C)(=O)=O N1(C(C2N(C(=O)COc3ccsc3)CCC2O)=O)CCOCC(C2CC2)C1 C1(C(=O)NC(CC)CCCO)C(C)OCCN1C(C1CCCC1O)=O C1(N(C)C(=O)Nc2ncoc2C2CCCC2)CCC(C)(C)CC1 c1(NC(C2CC(F)CN2Cc2cncs2)=O)cccc(OC(F)(F)F)c1Cl CC1CN(C(=O)Cc2ccccc2)CC1C(N1CCCC1CCO)=O c1(C(=O)NCC(CC)NC(c2ccccc2OC)=O)cnc(C)nc1OC C12(C(=O)NN3CC(F)(C(=O)OC)C3)CCC(N(C)C)(CC1)CC2 c1(OCC)cncc(C(N2CCC(OCCNC(c3ccnnc3C)=O)C2)=O)c1 N1(C(C=Cc2occ(C)n2)=O)CCC2C(NC(c3ncccc3Br)=O)CC12 CC12CC(C(=O)NC3(O)CCCN(C(C4CC(OC5CC5)C4)=O)C3)(C1)C(C)(C)O2 c1(C(=O)NC2CC(CNC(c3c(C#N)csc3)=O)C2)cnc2[nH]c(O)nc2c1 Cc1csc(C(=O)N(C)CC2CCCC2NC(c2ccnn2CCF)=O)c1C CC1(NC(=O)C(=O)NCCNC(=O)C(c2ccccc2)=O)CC2C=CC1C2 c1(NC(C2(C)CN(C(c3cc(C)cc(C)c3)=O)C2)=O)ncc([N+](=O)[O-])cc1Cl Cc1c(C(N2CCC(NC(C3(SC)CC3(C)C)=O)CC2)=O)ccn1C(C)C C1(c2n(CCC)nnn2)(NCCCc2nnc(C(C)(C)C)s2)CCS(=O)(=O)CC1 CCC(CC)C(C)C(=O)NCC1CCN(C(c2cc(C)ccc2N)=O)C1(C)C N1(C(CC2(C(CC)O)CC2)=O)CCCOC(CCNC(=O)C=C(C)C(F)F)C1 N1(C(=O)Cn2cnc(Br)c2)CCCN(C(c2nc(Cl)ccc2F)=O)CCC1 C1(NC(c2c(C)cc(CC)o2)=O)CCN(C(c2sc(C(C)C)nc2C)=O)CC1O Cc1snnc1C(=O)NCC1(N2CCCC2)CCC1.C1(C2C3CC3CN2)CCCC1 c1(C(N(C2C(C)CCN(C(CCC=CC)=O)C2)C)=O)cccc2c(C)ccnc12 Cc1ccc(F)cc1CN=c1[nH]c(CC(N2CCCC(C#N)C2)=O)cs1 C=CC1(C(=O)NCC2(C)CCC(=O)N2)CCN(C(c2ccnc(C)c2)=O)C1 CN1CCCC(CNC(C2C=CCN(C(=O)C=Cc3ccncc3)C2)=O)C1 Nc1cccc(C(=O)NC2CCC(NC(c3coc(C(F)(F)F)c3)=O)CC2)c1N c1(NC(=O)NC(C#C)C2CCC2)noc(-c2ccccc2)c1Br N1(C(CCCC(C)C)=O)C2CCC1CC(N(c1ncccn1)C)C2 C(=O)(C(CC(C)C)CC(C)C)NC1C(CNC(C(C=C)(C)C)=O)CCC1 C12(C(=O)NC3CC(N(C(c4c(C)nc(C5CC5)[nH]4)=O)C)C3)CCCN1CCC2 CC1COCC(CC(=O)NN2CCCC2CCO)O1.c12cc(on1)C(=O)NCC2 C1(Nc2nc(C(F)(F)F)nc(N3CC4C(C3)C4(F)F)c2)CCc2nnnn2CC1 c1(C2(n3cc(C4CN(C(C(CC)C)=O)C4)nn3)CCC2)cccc(Cl)c1 C12(C(=O)NC3CCCC(C(=O)OC)C3)C=CC(CC1)C2.C12(CC1)C(=O)N2 N1(C(C(C)C2CC2)=O)CC(NC(C2(CO)CCOCC2)=O)CC(C)C1 N1(C(C2N(CCC)CCC2)=O)CC(NC(=O)C(C)OCCN(C)C)C2(CCC2)C1 c1(C(N(C(CNC(c2ccc(OC)cn2)=O)C)C)=O)ccc2ocnc2n1 c1(CN(C(c2c(C)cco2)=O)C(C)C)ccc(Oc2cccc(F)c2)nc1 C(=O)(C1=NOC(C)(C)C1)NC(C)C(=O)NC(C)Cc1ccnn1C N1(C(CC2CC(CC)OCC2)=O)CCCC2(NC(=O)C(C)C3CCCC3)CC2C1 C1(C(N2CC(C(C(C)C)O)C2)=O)CCN(C(C2CC3CCC3C2)=O)CC1C c1(NC(C2CCCN(Cc3c(Cl)ccnc3Cl)CC2)=O)cc(CO)cc(F)c1 c1(C(N2C(CNC(CC=C(C)C)=O)CCCC2)=O)cnc2ccnn2c1C c1(COC)ccc(C)c(C#N)c1.C12CSCN1C(=O)C(O)Cc1cn(nn1)C2 N1(C(CCN(C(c2c(CC)nn[nH]2)=O)CC)=O)CCC(C)C(CC(=O)OC)C1 N1(C(CCNC(COC)=O)=O)CC2(COC(CNC(=O)Cc3cnsc3)C2)C1 Cc1ccc(C(=O)NCC2CN(C(=O)Cn3cnc(Br)c3)C2)s1 C1(C(=O)NCC(=O)NC2CC2)(CC)CCCN(C(C2CCCC(C)(C)C2)=O)C1 n1(CC(=O)N(C(CNC(CCC#C)=O)C)C)[nH]cc2c(=O)ncnc1-2 C1(NC(c2ncccc2O)=O)CN(C(c2cnn(C3CC3)c2)=O)CC12CC2 CC1(NC(C2CCC(=O)N2)=O)CCN(c2nnns2)CC1 CC1(C)C2CC1CC(=O)N2.c1(C(N2CCC2(COC)CO)=O)ccc(=N)[nH]c1 C1(NC(C(CC)C(C)O)=O)CC2(CCN(C(=O)C#CC3CCCO3)CC2)C1 c1(CC(=O)NCC(C)NC(c2cccc(OCCOC)c2)=O)ccc(C#N)cc1 C=CC(C)(CC)C(=O)NC1CCN(C(C23CC(C)(C2)OC3C)=O)CC1C N1(C(c2[nH]cc(C)c2)=O)CCN(Cc2cnn(-c3cccc(C#N)c3)c2)C2CC12 N1(c2c(C)c(NC3CCCN(CC4CC4)C3)ncn2)CCCC1C1CCCO1 C(=O)(C1=CCC(NC(=O)CCCCC#N)C1)NCC(COC(C)C)O CC1C(C)N(C(C2CCC3CC2CO3)=O)CCN1C(c1cc(C(F)(F)F)n[nH]1)=O c1(C(N2CC3C(NC(c4nc(CC)oc4)=O)C(C3)C2)=O)cccc2nnn(C)c12 c1(C(=O)NC(C)CN2CCN(C(=O)C=C(Cl)Cl)CC2)cnc2[nH]cncc1-2 c1(OC)c(CC(N2CCC(C(C)NC(=O)CC(=O)NC3CC3)C2)=O)cccc1F CCCCS(=O)(=O)N1CCCC(C(=O)CN(S(C)(=O)=O)C(C)C)C1 c1(CNC(c2c(C)noc2C)=O)sc(=NCc2c(O)cccc2F)[nH]c1C C1(C(=O)NCCCNC(C2(C(=O)OC)C(=C)CC2)=O)COCCC1C c1(C(=O)NCC2C(NC(=O)CCc3ccon3)C2)ccc2nsnc2c1 C(C(=O)NN1CCCCC1C)NCCN(C(=O)C(F)OC(F)(F)F)CCOC C(=O)(CCCCCCCCC1CC1)NC1C(NC(C(C)(C)OCC)=O)C1 c1(-n2c(SC(C)CCc3nnn(-c4ccccc4)c3C)ncc2)ccc(OC)cc1 N1(C(C2(C)CC(=C)C2)=O)CCC(NC(=O)CC2(C#N)CCC2)C(C)C1 C#CC1(C(=O)NCc2cc(F)ccc2C)CCN(C(=O)CC2CC3CCC2O3)C1 c1(OC(C)C)cccc(CCC(=O)N(CC(C)CNC(=O)C(C)CN(C)C)C)c1 C1(CC)CN(N2CC(NCCN)CC2C)CC2(CCC2)C1.C1C(=O)O1 O=C1CCCCC(C(N2CCCN(C(C3CCC(F)(F)C3)=O)CC2)=O)N1 C1(C(N2CCC(C(=O)NC3C(CN(C)C)C3)CC2)=O)CCC2(CC1)CC2 CC1(C)CC(C(=O)O)CCN1C(=O)CC(O)CNC(c1cccnc1)=O CS(=O)C=CC(=O)N1CC(NC(C2(CF)CC(F)(F)C2)=O)C(CC2CC2)C1 c1(CCN(C(C2CC3CCC2C3)C(=O)NCCOC)CC2CC2)cccc(Cl)c1 C(=O)(CC1CCOc2ccccc21)NCCCC1(NC(C2CC(O)C2)=O)CC1 C(=O)(CC(O)CC)N(C1CCN(C(C2CC2F)=O)CC1)CCC N1(C(CCc2onc(CCC)n2)=O)CCC(NC(=O)C(O)CC(N)=O)CC1C c1(N(C)Cc2c(OC)nccc2)[nH]c(=NC2CC3CC3C2)nc2sccc12 N1(C(C(C)OC)=O)CCC2(CC1)COC(CNC(=O)C(C)(C)n1cnnn1)C2 CCCC(C#N)C(=O)N(CC(CO)(CO)NC(c1ccnc(N(C)C)c1)=O)C N1(C(c2n(CC)nc(C)c2)=O)CC2CCC2(NC(c2ccoc2Cl)=O)C1 C(=O)(C(CC(C)C)N1CCCCC1=O)NC(CNC(CC1CC(OCC)C1)=O)C c1(CNC(c2cc(Cl)ccc2Cl)C(=O)OCC)cc(F)cc(F)c1F c1(CC(=O)NC2CCN(C(CN(C(C)C)C)=O)CC2CO)ccc2nn[nH]c2c1 N1(C(C2CC(OC)(OC)C2)=O)CCN(C(=O)CC2CCCC(C)(C)C2)CC1C C(=O)(CC(C)(C)C)NC(C(C)C)c1nc[nH]n1.C1(C(C=O)C)CCN(C)CC1 CC(C)C(CNC(c1ccn(C)c1)=O)C(=O)N1CC(C)C(C)(CO)C1 c1(CC(=O)NC2(C)CCN(c3nnc(-c4ccccc4)s3)C2)ccc(Cl)c(Cl)c1 C1(C(CNC(c2ccno2)=O)F)CCN(C(c2ccc(OCCO)cc2)=O)CC1 C(=O)(C(CCCC=C)NC(=O)COC1CC1)N.C#CCC(C)(CCC(=O)O)CO c1(C(=O)NCC2N(c3ccnc(C(C)(C)C)n3)CCCC2)c(F)cc(Cl)cc1Cl C1(CC)CN(C(c2ccc(CF)cc2)=O)CC1NC(c1cc(C#N)c[nH]1)=O N1(C(CN2C(C)CCCC2)=O)CC2(CC(NC(=O)C(C)C(F)F)C2)C1 C1(C(=O)NC(COCC)C(C)C)CCCCN(C(=O)C(C)CC)C1 C=CCC(CC(=O)N(C1CCOC(C)(C)C1)C)NC(=O)C1=C(C)CC1 c1(CC(=O)NCC(CNC(C=CC=CC)=O)C)ccc2c(c1)CCN2C c1(C(N(C2CN(C(=O)Cc3ccc(Cl)nc3)CC23CC3)C)=O)n[nH]c2c1CCC2 C(=O)(C1=CC2(CN(C(=O)C(C)C3CCOC3)C2)OC1)Nc1cncc(COC)c1 N1(C(CCOCC#C)=O)CC2C(CNC(C3(COC)CCC3)=O)C2C1 C1(OCC)COCC1N=c1[nH]c(=NC(C)Cc2ccc(Cl)cc2)[nH]c2c1CSC2 CCN=c1cc(C(=O)NCCCN(C(=O)CN2CCCCC2)C)cc[nH]1 CC(C)C(C(=O)NCC(CNC(C12CCCC1(C(N)=O)C2)=O)C(F)(F)F)C(C)C C1(CNC(C(CCC)C)=O)CCCC2(CN(C(=O)CSC3CCCCO3)C2)O1 C=CCCC(C(=O)N1CCOCC1CC)NC(=O)C=CCN1CCC1 C(=O)(NNC(=O)c1cc(COC(C)C)on1)NC(CC)C CC1CC(N=c2c([N+](=O)[O-])c[nH]c3cc(Cl)ccc23)CCN1C(c1ccno1)=O c1(-n2cc(C(CCC)NC(c3ccccc3CC)=O)nn2)cc(F)ccc1C C1(C(=O)NCc2c(C(N(C3CCCC3O)C)=O)n[nH]c2)CC2CC(=O)C1O2 Cc1cc(C(=O)NCC(=O)NC(C)C(C)NC(c2cc(C#N)c[nH]2)=O)n(C)n1 N1(C(C(COC)C)=O)CC2CCC2(CNC(=O)CNC(=O)CC2CCCC2)C1 N1(C(C(CSC)C)=O)CCN(C2CCN(C(=O)CSCc3ncc[nH]3)CC2)CC1 N1(C(CC(C=C)C)=O)CCC(NC(=O)C2=CCCO2)C1(C)C C1(C(=O)OC)CC(C)N(c2nnc(C(C)C)n2Cc2cscn2)C1 CC(F)(C(=O)NCC1CN(C(=O)CCCc2nncn2C)C1)C(F)(F)F c1(C(=O)NCC(CCCC)NC(c2cc3scnc3[nH]2)=O)n[nH]c2c1CC1CC21 C1(C(=O)NC2CN(C(C(c3scc(CC)n3)(F)F)=O)C2)CCS(=O)(=O)C(C)C1 C(=O)(C(CNC(=O)C(C)C1(O)CCC1)C(C)C)NCC(COCC)(C)C N1(C(c2cn(CCCC)nn2)=O)CC(CNC(c2ccoc2Cl)=O)C(F)(CO)C1 Cc1csc(C(=O)NC2CCC2NC(C23C=CC(CC2)C3)=O)c1Cl CC1CN(C(C2CCCC(F)(F)C2)=O)CCN1C(=O)CN1C(=O)CN(C)C1=O CC1(C)OC(=O)C(CC(=O)NC2CC(N(C(=O)COC(F)(F)F)C)C2)O1 C12(OC)CCCCC(C(=O)NCCN(C(=O)C3=CCCS3)C)(C1)C2 c1(C(=O)NC(C)CNC(c2ccc(C(F)(F)F)o2)=O)cc(Br)cnc1O c1(SCC)nc(C)c(CC(=O)NC(C)C(=O)OCC2CCS2(=O)=O)s1 c1(C(=O)NC(CC)CNC(c2cccnn2)=O)ccc2nc[nH]c2c1F N1(C(C(C)(C)SC)=O)CC2CC2(CNC(C2(C(C)C)CCC2)=O)C1 N12CCN(CC1)c1ncc(cn1)C(=O)NC(C)C2.N(CCO)(CC)CC N1(CC(C)C)CCCC(C(=O)NC2CCN(C(=O)Cc3cnoc3)C2C(C)C)C1 C(=O)(C1=COCCO1)N1CCC(C(C)NC(=O)C(F)(F)c2ccsc2Cl)C1 c1(C(=O)OC)cccc(-n2ncc(C3OCCC3C(C)C)c2Br)c1 N1(C(c2csc(Cl)n2)=O)CCOC(C2CN(C(=O)C=CC=C(Cl)Cl)C2)C1 C1(C(=O)NCC2=CCN(C(C3C(C)(CC)C3)=O)CC2)CC(c2cccnc2)=NO1 C=CCCCCC(=O)N1CCCC(NC(C2CCCC2F)=O)CC1 C1(NC(c2ccc(C3CC3)o2)=O)CN(C(C2CC3CCC2O3)=O)CC2(CC2)C1 C(=O)(CC(C)C(F)F)NCC(CNC(CCc1c(OCC)cccc1)=O)CO C(C(CN(C)C)C(=O)NC1CC1CC(C)(C)C)NC(CC(C)F)=O C(=O)(N=c1cccn[nH]1)C1CC2CN(C(c3ccc(SC)cc3)=O)C1C2 Cc1cccc(CC(N2CCC(NC(=O)CC3CCCCC3F)CC2)=O)c1F C12(C(=O)NCC3C(NC(C(C)(C)C)=O)C3)CCC(C(F)F)(CC1)C2 C1(O)(CC#C)CCN(C(C2C3CC2N(C(C2CCC(CC)C2)=O)C3)=O)CC1 C1(C#N)(NC(c2cn(CCNC(C(C)NC(=O)C3CC3)=O)nn2)=O)CCOCC1 C(Cc1ccco1)(C(=O)NOCCC(F)F)NC(=O)COC1CC=CC1 C(=O)(C(CC1CC1)CC1CC1)NCNC(C(c1[nH]c(=N)sc1)=O)=O CC(C(CO)NC(C1(C2CCCO2)CC1)=O)NC(=O)CC(C)c1ccncc1 C12(CNC(CCn3nc(C)c(C)c3C)=O)CCC1CCN2C(=O)COC(C)(C)C c1(C(=O)OCC)sc(C(=O)NCCC(O)CNC(C2CC2F)=O)c2c1CCCC2 C1(NC(c2scc(C)c2C)=O)CN(C(=O)CC23COCC(C2)C3)CC1(C)C c1(C(=O)NC2C(NC(C3C(C)CCC3)=O)C2)cccnc1Oc1ccccc1 n1(C(C)C)ncc(C(=O)NCC2C3CC2N(C(C2CCC(F)CC2)=O)C3)c1N c1(OC)c(F)cc(F)c(NCCNC(=O)CN2CCS(=O)(=O)CC2)c1[N+](=O)[O-] C(N=c1cc(-c2ccccn2)nc[nH]1)C1N(CC2S(=O)(=O)CCC2)CCC1 C1(NC(CCCOCCOC)=O)CN(C(c2n[nH]cc2Cl)=O)CC1n1cccn1 C12(C(=O)NCC3(OC)CCC3)CCC1CN(C(c1cc(Br)co1)=O)C2 c1(C(=O)NCCN(CCC)C(c2cc[nH]c2)=O)ccnc(OC(C)CC)c1 C1(CNC(C2(CCC)CCC2)=O)CCN(C(=O)CCC=CBr)CC1C CS(=O)(=O)C1(C(N2CCN(C3CN(C(=O)CC=C(Cl)Cl)C3)CC2)=O)CCC1 c1(CC(=O)NC(CN(C(CCCc2nc(C)sc2)=O)C)(C)C)cc(C)cn1C c1(CC(N2CC(CN(C(C3CC(=C)C3)=O)CC)C2)=O)nnc(O)s1 N1(C(c2c(C#C)c[nH]n2)=O)CCC(C=C)(C(N2CCCC(C(=O)NC)C2)=O)CC1 C=CC(CC)CC(=O)NC1CCN(C(=O)CNC(c2c(F)cccc2Cl)=O)C1 C(=O)(CCCN=[N+]=[N-])NC(C(=O)NCC(C)C(F)(F)F)(C)C1CCC1 N12CCC(C(O)C1)CNC2=O.c1(OCC2CCC(=O)N2)ccc(F)cc1 c1(NC2CCN(C(C(=O)NCC(COC)C(C)C)=O)CC2)ccc(S(C)(=O)=O)cc1 CCCCC(CC)CC(C(=O)NC1CCCC1)N1CC=CC(O)C1 c1(-c2ccc(C)c(O)c2)ccn2cnnc2c1.O=C1CC(C)CCN1 N1(S(c2ccc(SC)s2)(=O)=O)CC(C)(C)OC2(CNC2)C1 N1(C(CC(CNC(C2CC=CC2)=O)OC)=O)CC2(CCC(=O)NC2)C1 c1(CNC2CCC(N(c3ccccc3)C(=O)CC3CC34CC4)C2)cccc(F)c1 Cc1cccc(Cl)c1CC(N1CCC(O)(CCNC(C2(C#N)CCC2)=O)C1)=O C=C=CCC(=O)NC(C1CCCN1C(C1CCOC1)=O)C C#CC1(C(=O)OCC)CCN(C(C(=O)NCCc2cc(C)no2)c2ccsc2)C1 O=C(CCCCCl)NCC1CC1(F)F C=CCCCCCCC(=O)N1CCCC(NC(=O)C(C)NC(C)=O)C1 c1(NC(N2CC(F)(C(=O)Nc3c(C(=O)OC)ccs3)C2)=O)cccc(Cl)c1Cl N1(C(c2cc(=N)[nH]cc2)=O)CC2CCN(C(=O)CCc3cnoc3)CCC2C1 C(C(CC(C)C)NC(c1csnc1Br)=O)NC(C1(COCC)CC1)=O C(=O)(CC(CNC(=O)C(C)(C)N1CCCC1)C1CCC1)NCC(C1CCC1)OCC C1(CC=C)(NC(C2CC2C)=O)CCN(C(=O)Cn2cccn2)CC1 CC(C)CCC(O)C(=O)N1CCN(C(C2(CC(C)C)CCCC2)=O)CC1C(C)C c1(-c2n(OC)ccn2)c(C)nn(C2(c3ccc(-c4nc(=O)o[nH]4)cc3)CC2)c1C C(Cc1ccccc1)(CCNC(=O)C(C)Nc1cncnc1)NC(CCC)=O Cc1nc(N2CCOCC(CNC(=O)CC(O)C(C)C)C2)cc(Cl)n1 C1(COC)(CNC(C2CCN2C)=O)CCCN1c1nnc(-c2ccon2)s1 Cc1ccccc1-c1cn(C(C)CN(C(=O)CCN2CCCC2)C2CC2)nn1 CC(CCC(C)(C)C)C(=O)NC1(C(=O)NC2CCn3cncc3C2)CC(F)C1 N1(C(CCN(C)CCO)=O)CCCC(C2CCN(C(=O)C(C)(C)CN(C)C)C2)C1 Cn1nc(Br)c2ccc(C(N3CC(F)CC3C(=O)NC3CC3)=O)cc12 N1(C(c2c(C)c(Cl)cnc2)=O)CC2CN(C(=O)CSC(F)F)CC2(C)C1 Cn1ccc2ccc(NC(C3(F)CN(Cc4cncc(Br)c4)C3)=O)cc12 C1(C(=O)NC2CCN(C(CCC=C)=O)C(C)C2)CCc2nc(C3CC3)ncc2C1 CCC(COC)C(=O)NCc1ccc(C(N2CCC2(C)C)=O)nc1 C(=O)(CCCCCO)NCC(C)(CNC(=O)C(C)=C(C)C)OC c1(CNC(C2N(C(C)=O)CCC2)=O)ccc(CNC(C2CCCS2)=O)c(F)c1 C#CC1CN(C(=O)C(CNC(=O)CNC(=O)C(C)(C)C)N(C)C)CCN1C C1(NC(C(CC)C)=O)CCCN(C(=O)C=Cc2ccc(SC(F)F)cc2)CCC1 C(CCCC(C)(C)C(=O)NNC(=O)c1ccncc1Br)NC(C(C)C(C)(C)C)=O c1(C(=O)NC(CN(C(c2c[nH]nc2C2CCCO2)=O)CC)C)cnc(OC)cn1 C1(NC(C2CCN(C(=O)CC)C2)=O)CC(F)(F)CC1NC(C(CC)(C)C)=O C1(NC2(c3nnnn3CCSC)CC(COC)C2)CC(O)C(O)C1 N1(C(CCCCCC)=O)CC2CC(C1)N(C(c1nn(CC)c(=O)cc1O)=O)C2 N1(C(C(C)=CC)=O)CCN(C(=O)CC(C)(C)C2CC2)CC1CF c1(CC)cc(C(=O)N(CC(N2CCN(C(=O)C(CO)N(C)C)CC2)=O)C)ncn1 O=S1(=O)CCCC1Cn1cc(Nc2ccc(CC3(CCCCO)CC3)cn2)nn1 c1(OC)cccc(O)c1C(N1CCN(C(c2ccco2)=O)C(CC(F)F)C1)=O Cc1cc(O)cc(Cl)c1C(N1CCC(O)(C(=O)Nc2ccc(CO)c(F)c2)C1)=O N1(C(CCOCC)=O)CC(NC(c2cnc(N(C)C)s2)=O)CC(C)C1 c1(CN2CCN(CCC=C)CC2)cc(F)ccc1N1CCCCC1 C(=O)(C(F)CC(C)(C)C)NC1CC(CCNC(c2c(C)n(C)nn2)=O)C1 Cc1nnc2ccc(C(N3CC(NC(C4CC5(CC5)CO4)=O)C(C)C3)=O)cn12 CC1CNCC(NC(C2CCN2C(=O)CC(c2ccc(Cl)cc2)O)=O)O1 CCCCCC(C)(CC)C(=O)N1CC2CCCN(C(c3sccc3Cl)=O)C2C1 C1(NC(C2N(C(c3[nH]cc(C(C)=O)c3)=O)CC2)=O)C2CC3C(C2)C13 C1(NC(c2nccc(OC)c2OC)=O)C(C)CN(C(C2(C(F)F)CC2)=O)CC1C C1(NC(C(c2ccc(C)cc2)O)C)CC(C)(C)OC(C)(C)C1 N1(C(C2=C(C)CC2)=O)CC(NC(c2ccc(Cl)c(O)c2)=O)CC12CCC2 c1(CC(=O)NCC(N(C(C(F)=CC)=O)C)C2CC2)ccc(C)c([N+](=O)[O-])c1 c1(CN2CCC(CNC(CCC3(C)CC3)=O)C2)ccc(C(F)F)cn1 c1(COC)nc(=NC(=O)c2ccc(C(C)(C)S(C)(=O)=O)cc2)o[nH]1 C(=O)(C1c2ccccc2C1)N(CC(C)NC(C1CCCN1C(=O)C(C)(C)C)=O)C C1(NC(CCn2c(=O)cc(C)nc2)=O)C(C)(C)CN(C(=O)C(C)(F)F)CC1(C)C n1(CC(N2C(CNC(C(CC#C)C)=O)CCCC2)=O)nc2c(n1)CCCC2 N1(C(CC(C)F)=O)CCc2c(c(CNC(C3CCCC3CF)=O)nn2C)C1 C1(C(=O)NCCC2(O)CCN(C(CNC(C)=O)=O)C2)CCc2nnc(O)n2C1 c1(C(N2CCN(C(c3nc(C)oc3)=O)C3C2C3)=O)ccc2occc2c1O c1(C(=O)NC(C2CN(C(C3CC(C(F)F)C3)=O)C2)C)cccn2nncc12 C(=O)(CC1CC(C(C)C)c2ccccc21)NCC1C(NC(COC(C)=O)=O)C1 c1(C(=O)OC)ccc2nc(NC(c3ccc(Cl)cc3Cl)=O)[nH]c2c1 Nc1ccc2nc(N3CCCC(C4CC4)(NC(=O)C=CC(F)(F)F)C3)sc2c1 c1(C(=O)NC2CCN(C(C3(COCC)CC(F)(F)C3)=O)C2)cc(S(N)(=O)=O)c[nH]1 N1(C(CC(C(F)(F)F)OC)=O)CCC(NC(=O)CCOC(C)=O)C2(CCC2)C1 C(=O)(C(C)CC(F)F)NC(c1ccc(C)cc1)CNC(=O)C(C)n1cccc1 N(C1c2cc(F)ccc2CC1(C)C)CC(C1(C)CCC(=O)N1)(C)C c1(OC)ccc(C(=O)NC2CN(C(C3(C#N)CC(F)(F)C3)=O)CCC2C)c(C)c1 N1(C(C(CC)(C)O)=O)CCC(O)(CCCNC(C2CN(C(C)=O)CCO2)=O)CC1 N1(C(c2c(NC)cnnc2)=O)C2CCC1C(NC(=O)COC1(C)CCCC1)C2 CC(=O)CCCC(=O)NCC1CN(C(c2cc(CN(C)C)on2)=O)CCC1C c1(C(=O)NC2C(CNC(C(C)(C)c3ccccn3)=O)COC2)cnc2n1CCS2 N1(C(C2(CC)CCN(C(=O)CC3CCC(=O)C3)C2)=O)CCC2(CC1)CC2C#N C1(NC(CCCCN(C(=O)CSc2nc[nH]n2)C)=O)COCC1C1CC1 CC(C)(CC(=O)N1CC(C2(NC(=O)CCc3ccc(F)nc3)CC2)C1)C(F)F c1(C(=O)NC2CCN(C(C3(C)COC3)=O)C2)cnc2n1CCS2 c1(C(N2CC(NC(c3cnn(CCF)c3)=O)C3(C2)CC3)=O)cnn2ccccc12 C12(NC(COCCCOCC=C)=O)CCC(CC1)N(C(=O)CC(C)C1CC1)C2 Cc1cc(NC(=O)C(C)N(C)C(c2ccnc3cc[nH]c23)=O)c(O)cc1F S(=O)(=O)(c1ccc(NCCC(C)(C)CO)cc1Cl)NCC1(COC)CCC1 c1(CNC(C(CCOCCO)NC(CC(CC)C)=O)=O)cc(C)nc(C)c1 CN1CC(CNC(C2(C)CCN(C(C3CCN3C)=O)C2)=O)CC1=O C1(NC(c2c(CC)ccs2)=O)CN(C(=O)C(O)CC(F)F)Cc2ccnn2C1 N1(C(C2CC(CC)C2)=O)CC(C)(C)OCC1CNC(=O)CS(=O)(=O)NC c1(NC(=O)CSc2cccc(CO)n2)ccc([N+](=O)[O-])cc1 CC(CCC(=O)N1CC2C(C)C2C1)NC(=O)C(C)(F)F c1(Cc2c(C)non2)nc(-c2ccn(C)n2)nn1-c1cnn(C)c1 Cc1c(Br)c(C(=O)NCC2(O)CN(C(=O)C3=CC(C)(C)C3)C2)nn1C C(=O)(C1CCCc2ncc(C)n21)NC(C1CCCC1)CNC(CNC(C)=O)=O c1(C(=O)NCCCN(C(c2ccsc2Br)=O)CC)c[nH]c(=O)cn1 c1(C(=O)NCCC(C)(C)NC(CCCOC)=O)cnc2c(c1)CCCO2 c1(C(N2CCC(N(C(c3cnc(CC)[nH]3)=O)C)C2)=O)ccc(=O)n2c1CCCC2 N1(C(C#CC(C)C)=O)CCC(O)(CN(C)C(c2ccccc2CCN(C)C)=O)CC1 C1(C)CC2(CCN(CC(=O)N(CC(C)(C)C)NC(C(C)(C)SCC)=O)C2)CO1.CC C1(C(=O)NC(C(C)C)CCNC(c2cnc(N)c(O)c2)=O)Cc2ccccc2O1 Cc1ccc(F)c(C(N2CC(F)CC2C(=O)NC2CC(c3ncc[nH]3)C2)=O)n1 N1(C(Cc2cn(C)nn2)=O)C2CCC1CC(C(=O)NCCCC(=O)NC1CC1)C2 c1(OC)c(C(=O)N(C)CC2CCCN(C(C3(Cl)CC3(C)C)=O)C2)nc(O)nc1O C(=O)(C(C)(C)C1=CCSCC1)N(C)CCNC(C1CCOC(=O)CC1)=O c1(C(=O)OC)ccc(CCCCNC(=O)C(C)COc2ccccc2)cc1 C1(OC)CN(C(C2CC(C(N3CC(O)CC3CO)=O)C2)=O)CC1NC(C)=O C(=O)(C(C)C(=O)N1CCCC1CN(C)C(c1csc(-c2cnccn2)n1)=O)OC C(C)(CCCN=c1[nH]cc(C#N)cc1C)NC(C(C)OCC)=O Cc1cc(O)cc(C)c1C(=O)NC1CCN(Cc2csc(Br)n2)C1 N1(C(C(C)S(C)(=O)=O)=O)CCC2C(CCCN2C(=O)CCCC(N)=O)C1 C1(CC(N2CCC(OCC)C2)=O)CCN(C(c2c[nH]ccc2=O)=O)CC1 C1(COC)CC(CNC(=O)Cn2nccn2)N(C(c2cccc(C(F)F)c2)=O)C1 N1(C(C=CCC(C)(C)NC(C(C(C)C)N(C)C)=O)=O)CC(O)CCC1C c1(C(=O)NCCC2CCC(NC(=O)CCC3CCC3)C2)cccc2c1CCC2 C(=O)(C(C)(C)C(F)F)NC(C(C(=O)NC1CC(C(C(=O)OC)F)C1)C)C C1(C#N)(C(=O)NC2(C(N(C)CCC3CCCO3)=O)CCC2)CCC1 C(=O)(C1=Cc2ccccc2OC1)N1C2(CO)CCC(C(=O)OC)(CC2)C1 C(CC(=O)NCCn1ccnc1)(C(F)F)N(C)C(c1cc[n+]([O-])cc1)=O C1(CC)CCCCC1NC(c1c(CNC(=O)C=Cc2ncc[nH]2)cnn1C)=O C(=O)(C1=CCC(C)(C)CC1)NC1CCCN(C(Cc2cnc(C)s2)=O)C1 n1(CCCC)nnnc1C(c1cn(C(C)C)nn1)NCC(c1ccccc1)C C1(NC(C2(C#C)CN(C(=O)CCC(=O)C3CC3)C2)=O)CCC12CCCC2 Cn1cc(Br)c(CNC(=O)NC2CCC(c3ccccc3)C2)n1 C1(C(=O)NCCN2C(=O)CCC2=O)CCN(C(c2n[nH]cc2Cl)=O)CCO1 N1(C(C2(C)CC(=C)C2)=O)CCC2CCCC(C1)N2C(c1ccncc1)=O C1(C(C)(O)CNC(C2SCCCS2)=O)CCN(C(c2cn(CCO)nn2)=O)CC1 C1(C(=O)NCCc2nc(C)sc2)C2CCN(C(c3cc4n(n3)CCO4)=O)CC12 C1(C(=O)NCCCCCC)C(O)CCN1C(=O)C(C)Oc1ccccc1 C1(C(C(=O)NCC2CCC2NC(=O)CNc2cccnc2)OC)CCCCCC1 c1(C(=O)NC2CC(C)(NC(c3cnc(C4CC4)s3)=O)C2)cncc2cccnc12 C1(C(=O)NCC#CC)CCN(C(c2csnc2C)=O)C1C C1(C(N(C2CCCNC2)C(c2ccncn2)=O)=O)CCC(F)CC1 Cc1nc(C)c(C(=O)N(C)CC2(O)CCN(C(c3csc(C(F)F)n3)=O)C2)o1 C(C)(CCCCCO)NC(C1N(C(Cn2ncc(C)c2)=O)CSC1)=O N1(C(C(C2CCC2)NC(c2ccc(C#C)cn2)=O)=O)CCCC[Si](C)(C)C1 N1(C(C2COCCN2C(C2C=CCCC2)=O)=O)CCn2nccc2C1 CC1CN(C(C2CCN3CCC2C3)=O)CCCN1C(c1ccc(F)c(F)c1)=O CC(C)(CNC(=O)CO)CNC(=O)CCNC(C1CCCC1)=O C1(C(N2CCC(CC=C)(NC(c3csc(=N)[nH]3)=O)C2)=O)CC2(C1)CC(C)(C)C2 O=C(CS(=O)(=O)c1ccc(C)cc1)NCC1=CCN(C(c2ccccc2)=O)CC1 N1(C(CCNC(=O)OCC)=O)CCCC(C(C)(O)CNC(=O)CCCF)C1 C(CC1CCC1)(C(=O)N(CCC(=O)NC1CC2CC2C1)CCC#N)OC N1(C(c2cc(C)n(C)n2)=O)CC2CC1CN2c1nccc(N2CCOCC2)n1 CCCC(O)(CCC)CC(=O)N(C1CCCCC1N(C)C(C1CC=CCC1)=O)C C(=O)(C=C1SCC(=O)N1C)NCC1CCCN(C(C2CC(C(=O)OC)C2)=O)C1 N1(C(C(CC=C)CC)=O)CCC2(C=C(C(=O)NOC3(CO)CC3(F)F)C2)C1 C1(NC(C2N(C(C)=O)CC(O)C2)=O)CN(C(c2[nH]nnc2C)=O)CC1C1CC1 C1(COCC=C)CCN(N2CCCC2CSc2ccccc2)CC1 c1(C(C)(C)C)ncc(C(=O)NC2CC3(C2)CC3NC(C2CC2F)=O)cn1 c1(C(=O)OC)cnc2nc(NC(c3cccc(O)c3OC(F)F)=O)ccc2c1 c1(N(c2ccc(Br)cc2)C)nc(O)c([N+](=O)[O-])c(O)n1.C12CCCN1C(=O)NC2 C(=O)(C1=C(Cl)CCOC1)N1CC(CC(=O)NCC2(c3nn[nH]n3)CC2)C2(C1)CC2 C1(NC(Cc2nc(C)[nH]n2)=O)CN(C(=O)CC2CCCC(=O)N2)CC1C C=CCCCC(=O)N1CCCC(N(C(=O)Cc2csc(C(=O)OC)c2)C)C1 c1(C(N2CCCCC2CCN(C)C(c2cnn(CC)n2)=O)=O)cccc(C)c1C N(S(=O)(=O)N1CCNCC12CCNCC2)C(C)C(F)(F)F c1(C(N2CCC(C(NC)=O)C2)=O)ccc(F)cc1.C(CCC)=CCC CC1OC2(C(=O)NCCCCCCNC(=O)COC3CCCCC3)CC1C2 C1(c2n(-c3c(OC)c(Br)ccc3)nc(-c3cscn3)n2)CCc2nccn2CC1 N1(C(c2n(CC)nnc2)=O)Cc2[nH]nc(C(=O)NCCN(C)C)c2C1 N1(C(c2c(C)nc(O)cc2)=O)CC(N=c2[nH]c(Cl)ncc2C(N)=O)CC1C c1(C(C)C(=O)NC2(CN(C(=O)CCS(C)(=O)=O)C)CC2)cc2ccccc2s1 C(=O)(CC1=CCCCC1)NC1C(C)CCN(C(c2c(C)oc(C)c2Br)=O)C1 C1(CNC(=O)Nc2c(OCC)c(F)ccc2)CCN(c2ccncn2)CC1(F)F C(=O)(C1=NN(CCO)C(=O)CC1)N1C2CN(C(c3ccc(C)c(N)c3)=O)CC1CC2 C1(CC)(CC)CCCN1C(=O)CC1CCN(C(=O)CCCCC2CC2)CC1 C12(C(N(CCC(C)NC(C3(CC#C)CC3)=O)C)=O)C3CCC(CC13)C2(F)F c1(OC)cc(C)cnc1C(=O)NC1CCC(CCNC(=O)C2=CCC2)C1 C(=O)(CCCCO)NCC(C1CCCC1)NC(C(c1cn(C)nc1)O)=O C1(C(=O)NC(CC(C)NC(C#CC(C)C)=O)C)CCCCC1(F)F N1(CC(N2CCCN(C(C3CC(F)C3)=O)CCC2)=O)CCCCCCC1=O C(C(C)(C)NC(=O)NC1(NCC(F)F)CC1)OC C1(C(N2CC(CCNC(c3ccc(C(N)=O)nc3)=O)C2)=O)CCc2n[nH]cc2C1 N1(C(C(CC[SH](C)C(N)=O)O)=O)C2CCC(C2)C1CNC(=O)Cc1cccc(Cl)c1 c1(NC(C=C(C)CNC(=O)CCc2nc(O)n[nH]2)=O)ccsc1C c1(C(=O)NC2CCCC2NC(C2(C(F)(F)F)CCC2)=O)cccc(=S)n1O C1(CNC(C2OCCN(C)C2)=O)CCC12CCN(C(=O)CCC#N)CC2 C1(C)(C(N(CCCNC(C2CN(C(C)=O)C2)=O)C(C)C)=O)CC(C#N)C1 N1(C(C(CC#C)C2CC2)=O)CCC(C(=O)NOCC(C)(C)C)C1(C)C Cc1cc(C(=O)N(CCCNC(C2(F)CCOC2C)=O)C)cc(C(F)F)c1 c1(C(=O)NCCCC2(NC(C(c3ccc(Cl)cc3)C)=O)CC2)ccc(Cl)cc1Cl C(=O)(C1Cc2ccc(F)cc21)NC1C(NC(c2cnc(O)cc2O)=O)CCC1 N1(C(C2N(C(=O)C(=O)N(C)C)CCN(C)C2)=O)Cc2ccncc2C1 C(=O)(C(C(C)C)C(C)C)NC1CCCC(NC(c2c(C(C)C)cccc2Cl)=O)C1 N1(C(CC2CCC(NC(C3CC(C)(O)C3)=O)C2)=O)CC(CO)C(O)C1 c1(C(N=c2nnn(C(C)(C)C)[nH]2)=O)cc2cnccc2[nH]1 C1(OC)CN(C(c2cccc(OC)c2C)=O)CCC1NC(=O)C=CCC1CC1 C(c1nc2ccccc2[nH]1)=CC(=O)NC1C(CC)N(C(c2cnc(O)o2)=O)CC1 c1(SC)ccc(NS(C)(=O)=O)cc1.N12CCCC(C1)N(C1CC(C)OC1C)C(=O)C2=O c1(C(N2CC(CNC(c3csnn3)=O)C(O)C2)=O)cc(F)cc2cnccc12 C1(N(C(C(=O)NC(C)C(C)n2cccn2)=O)C)CCC(C)(C)C1 N1(C(C(CC=C)CC)=O)CCCC(C)(C)C1CCNC(c1ncoc1CC)=O c1(C(=O)NCCc2occ(CC(=O)NCC(C)=CC)n2)ccccc1CC c1(C(=O)NCC(CC)N(C)C(c2c[nH]c(C(N)=O)c2)=O)ncc(C)s1 c1(C(N(C(CNC(C(C(C)C)c2cnc(C)s2)=O)C)CC)=O)nccn2nccc12 C1(C(=O)NCc2ccc(C)o2)CC=CCN1C(=O)CCc1ccccc1 CCCC(C(=O)OC)C(=O)NCC1CC(F)CN1C(=O)CC1CCC(=O)NC1=O Cc1conc1C(c1nnnn1C(C)(C)C)NC(Cc1nc(C)on1)=O.C(C)C C(C1CCOCC1)=CC(=O)N(C(C(=O)N(C1CCN(CC)C1)C)C)C1CC1 CCC(COC)C(=O)N1CC(NC(c2sc(Cl)cc2Br)=O)CC1C CCC(C(=O)NCCc1ccc(C(F)(F)C(F)(F)F)s1)C(C)O C(=O)(C1Cc2ccc(F)cc21)N1CCC(C)(CNC(C2CCCCN2N=O)=O)C1 CC1CCC(NC(=O)CCCCC2CC2)CN1C(c1ccc(Cl)c(F)c1)=O C1(C(=O)NC(CC)CNC(C2CCC(C)(C)CO2)=O)CCC2(CCCC2)CC1 C(C(C(F)(F)F)N1CCN(C(c2ncncc2Cl)=O)CC1)NC(C(CC)C)=O C(=O)(C(C)(C)CC(F)F)NC1CCC(NC(C2CCC(C)S2)=O)CC1 C1(C(C(=O)NCCC#N)N(CCOC)C(C)C2CC2)CCC(C)C1 N1(C(C(CC=C)(C)C)=O)Cc2occ(C(N3CC(=O)NC(CC)C3)=O)c2C1 c1(C(=O)NC(c2ccc(OCCBr)cc2)CNC(=O)C2CC2)ccccc1Cl c1(C(N2CCCC(C3CCCCN3C(=O)C(F)F)C2)=O)sc(NC2CC2)nc1C N1(C(C=Cc2c(C)noc2C)=O)CCC2(CCCN(C(=O)C3=NOCC3)C2)CC1 C1(C(N2CCC(C(=O)OC)(CO)C2)C(=O)NCC(=C)C)CCCOCC1 c12c(cc(F)cc1F)C(=O)N(CCN)C2=O.C(=O)(CNCC=CCSC)C1CC1.CC c1(NC(=O)NC2C(C)(C)CC2)nc2ccc(F)cc2s1 c1(OC)ccnc(O)c1C(=O)NC1CCC(NC(c2ncc(Cl)s2)=O)C1 C1(CNC(c2oc(-c3ccco3)nc2C(F)F)=O)CCCCN(C(C2CCO2)=O)C1 c1(N2CCC(N(C(CCC)=O)C)CC2)nn2cc(C)nc2s1 c1(CNc2c(C(=O)Nc3ccc(O)c(Br)c3)n[nH]c2)cc([N+](=O)[O-])ccc1Cl C1(NC(c2c(C)n(C)cc2)=O)CCN(C(c2cnc(C3CC3)nc2O)=O)CC1C C1(CC(=O)NC2CC(C(C)O)C2)CC(O)CN1C(=O)CCc1cnn(C)c1 N1(C(CSS(C)(=O)=O)=O)CCCC(O)(CCNC(c2cc(C(F)F)n(C)n2)=O)C1 c1(C(=O)NCC2CC3CCC(C2)N3C(C2CC2F)=O)cc2cc(F)ccc2o1 C1(C(=O)NCC(CC)NC(c2ccccc2F)=O)CCCC(N(C)C)C1 CC1CCC(CC(=O)NC2CCCCC2Nc2ncccc2CSC)CC1C c1(C(=O)NCCN(C(c2ccn3ccsc23)=O)CC)ccc(C)c(C)c1 N1(C(C2C(C)C2)=O)CCCC2(CCCN2C(=O)C(c2ccc(Cl)cc2)O)C1 N1(C(C)C(F)(F)F)CCC(C)(NC(=O)CC(C)C2CCCO2)C1 N1(CCOCC)CCc2sc(S(N)(=O)=O)cc2C1.C1(=O)C(c2cscn2)N1 C(=O)(C1=CC2(CCN(C(=O)C(CO)C(F)(F)F)C2)C1)N(C1CCCC1)CC=C N1(C(=O)Nc2cccc(-c3cncnc3)c2)CCC(C2(c3ccccc3)CC2)CC1 N1(C(C(C)OCCC=C)=O)CCN(C(C2(CC(F)F)CCC2)=O)C2CCCC12 CC(C)CCC(=O)C(=O)N1CCC2CC12C(=O)N(C(C)CN(C)C)C c1(CN2CC(NC(Cc3cccc(C)c3)=O)C(C#N)C2)ccccc1S(C)(=O)=O c1(C(N2C3C(NC(CS(CC)=O)=O)CC(C3)C2)=O)cc(N)cnc1C c1(C(=O)OC)cnn(C)c1C(=O)NCC(CO)NC(c1cc(C)cs1)=O.C12CC1C2 C1(CNC(CN(C(=O)OCC)C)=O)(NC(C2C(C)C2(F)F)=O)CC(F)(F)C1 c1(N2CCC(N(C)C(c3ccc([N+](=O)[O-])s3)=O)C2)nc(Cl)nc2nc(Cl)n(C)c12 C(=O)(CC(C(F)(F)F)OC)NC1CC(F)(CNC(C(c2ccc(OC)cc2)C)=O)C1 N1(C(COS(C)(=O)=O)=O)CC(CNC(=O)COCC(F)(F)F)N2CCC1C2 C1(F)(C(=O)NCCN(CCOC)C(C2OCC2(C)C)=O)CCS(=O)(=O)C1 C1(C(=O)NC2(COC)CN(C(=O)Cc3cc(C)n(C)n3)C2)CC1C1CC1C c1(C2(O)CN(CCCNN3CCC(C(=O)NCC)CC3)C2)ccc(F)c(OC)c1 N1(C(C(c2cccc(Cl)c2)C)=O)CCCN(C(=O)CCc2nccn2C)CCC1 c1(CC(=O)N(C(C)CCNC(C2CC3(CCC3)C2)=O)C)cccc2ccsc12 n1(CCOC)cc(NC(=O)CC2(C)CCN2C(=O)C(C)c2cc[nH]n2)nn1 C1(C(c2nnnn2C2CCOC2)NCCOC)(OC)CCCCCC1 C1(C(NOCCN(C)C)=O)C(C2CC2)CCN1C(C12CCC(CC1)CC2)=O C1(CC(=O)NC(CCOC)CNC(=O)CN2CSCC2=O)CCCCC1F C12CCC(C1)C(=O)N2.c1(C(=O)NCC2N(C(COC)=O)CC2)cccnc1 c1(C(N2CCCC(n3cc(C(C)=O)nn3)CC2)=O)nc2ccccc2nc1C c1(C(N2CCC(C3N(C(CC(C)C4CC4)=O)CCC3)C2)=O)cc(Br)n(C)c1 C1(CNC(c2ccc(-c3ncon3)cc2)=O)CCCN(C(C2CCCOC2)=O)C1 c1(C(N2CC(NC(c3c(C)c[nH]n3)=O)C(CO)CC2)=O)cc(C)c(Cl)c(C)c1 c1(C(N2CC(O)(CNC(C3C(CC)CCC3)=O)C2)=O)c(C)nc2sc(C)cn12 C1(NC(c2nc(Br)c[nH]2)=O)CCN(C(c2cccnc2C2CC2)=O)CC1F c1(CC)cc(N)ccc1C(=O)NC1CC(NC(=O)Cc2cn(C)nn2)C1 N1(C(CCCCCN(C(=O)CCC2CC2)C)=O)CCC2(CNC(=O)N2)C1 C1(CN(CCNC2CC2)CC)Cc2ccccc2O1 C(=O)(C1=NOCC1)NC1CC(CNC(CC(C)c2ccncc2)=O)C1 Cc1nc2ccccc2n(CCNS(=O)(=O)C(C)CN(C)C)c1=O C(CC(C)(C)C)(C(=O)N(CCC(C)NC(=O)C(c1cn(C)nc1C)O)C)OC C12(NC(C(C3CCC3)OC)=O)CC3CC(C1)CC(NC(=O)CCC(C)(C)F)(C3)C2 C1(CC)CN(C(=O)COCc2cc(C)no2)CCC1NC(=O)CCCn1cncn1 Cc1[nH]c(C#N)cc1C(=O)NCC1C2CN(C(c3ccsc3C3CC3)=O)CC12 N1(C(C2N(C(c3c(CC)[nH]cc3)=O)CCCCCC2)=O)CC(CO)C(C2CC2)C1 Cc1ccnnc1C(N1CCC(C(C)(C)NC(c2c[nH]c(C(N)=O)c2)=O)C1)=O Cc1cccc2c(CNC(=O)N(C(c3ccc(F)cc3)C(C)C)C)cccc12 N1(C(C2CCC(CC)C2)=O)CCC(CN(C)C(C2(O)CCCC2)=O)CC1 c1(C(N(CCCNC(C(CCC#C)O)=O)C)=O)coc2c1CS(=O)(=O)C2 N1(C(c2cn(C(C)(C)C)nn2)=O)CCN(C(C2CCC(C)CC2)=O)C2CC12 CC(C(=O)NC1CCCC1NC(=O)C(F)(F)C1(O)CCC1)S(N)(=O)=O Cc1cc(C)c(C=CC(=O)NC(C)CCNC(=O)CN2CCC(O)CC2)cc1C N1(C(CC)=O)CCCN(C(C2CCCC2CNC(=O)CCCSC)=O)CC1 c1(NC(c2ccc(Br)cc2)C=C)nc2c(c(=NC(C)c3nc[nH]n3)[nH]1)SCC2 C(=O)(C(CCS(C)=O)N(C)C)NCCC(C(C)C)NC(c1c(C)nc(C)[nH]1)=O C(=O)(CC(C)CC(C)C)N1CCN(CCNC(C=Cc2c(C)cncc2)=O)CC1 C1(NC=O)CC12CCC(NC(=O)C=CCO)CC2.N12CCN(C1=O)NC(=O)C2 c1(CC(=O)NCC(C)NC(=O)C(F)(F)c2nccs2)ccc(O)c(F)c1 C1(OCC)C(N=c2[nH]c3c(c(=NCC4CCCCN4C)[nH]2)COCC3)CC12CCC2 CCCCC(CC(=O)NCCCCCF)NC(c1ncccc1F)=O c1(OCC)ncccc1C(N1CCOCC1CNC(=O)C1=C(C)CC1)=O c1(C(=O)NCCCCCNC(c2c(C(C)C)cccc2)=O)ccc2c(c1)OCO2 N1(C(C(c2n(C)ccc2)O)=O)CC=C(CC(=O)N2CC3CC2(CO)C3)CC1 N1(C(C=CC(=O)OCC(C)C)=O)CCN(C(=O)CCC2CCCCO2)CC1C C(=O)(CCCC(=O)OC)NCCCCC(C)NC(c1cn(C)nc1C(F)F)=O c1(C(=O)NCC(C)CNC(c2ccncc2N=[N+]=[N-])=O)nc2n(c1Cl)CCCC2 c1(C(=O)NC(CC(C)C)CNC(=O)C(C)(C)c2ccnn2C)cc2[nH]ncc2s1 C1(OC)CCC2(C(=O)NCC34CC(CN3C(c3csnc3C3CC3)=O)C4)CC12 C1(NC(c2cc(C3CC3)no2)=O)COCCC1C(=O)N(C1CC1)Cc1ccsc1 c1(C(=O)NC2CCC(N(C(=O)CCc3ccccc3O)C)C2)ccc(Cl)c(Cl)c1 c1(C(N(C)CC2(NC(C=C(C)C(C)C)=O)CC2)=O)cn(CC2CCCO2)nn1 c1(C(C)=O)ccc(Br)cc1C(=O)OC(CC1CC1)C(=O)O C1(NC(c2ccc(SC)s2)=O)CN(C(c2cnc(C(F)(F)F)s2)=O)CCC1C C=CCC(C)C(=O)NC(CCOC)C(=O)NCCCCCSC C1(CC#C)(C(=O)N(CC(C)N(C)C(c2ccn(CC)n2)=O)C)CCOC1 c1(Cn2ccc(C(=O)NC(C3CCCCCC3)C#C)n2)ccccc1F c1(C(N2CC(CC)C(C(=O)Nn3cnnc3C)C2)=O)cc(C)cc(O)c1 C1(C)(C(N(CC(C)CNC(=O)C#CCc2ccccc2)C)=O)CC(O)CN1C C1(C(=O)N(c2ccc(NC3CC3)cc2)C(=O)CCC)C2Cc3ccccc3C12 C1(CC(=O)NCCCCN(C)C(C2CC2CF)=O)COCC(C)(C)O1 N1(C(c2cc(=N)[nH]cc2)=O)CC(NC(=O)Cc2cnns2)CC2(CCC2)C1 c1(CC(=O)NCC#CCNC(c2ccc(C)cc2)=O)cccc(Br)c1Cl CCCC(C)(C)CC(=O)NC(C)CC1CN(C(=O)Cc2ccccn2)C1 N1(OC(=O)CCc2ccc[nH]2)CCCC(CC(=O)NCC2COC(=O)N2)C1 C1(CN(C(C2CCC2OC)=O)CC)CCCN(C(=O)C(c2cnn(C)c2)O)C1 c1(C(=O)NC2CCCC2NC(C2CCC2(F)F)=O)cnc2c(F)cccc2c1 C(C(C(=O)NCCCNC(N)=O)NC(c1cc(C)c[nH]1)=O)OCC C1(NC(c2onc(CC)n2)=O)CN(C(=O)C=CSC)C2CC12 CC1CN(C(=O)CC2(C)CCCO2)CC1CNC(=O)CC1(CO)CCC1 c1(C(=O)NC2(CF)CCN(C(CCc3n(C)cnc3)=O)C2)ncnc2c1CCC2 c1(C(N(C(CNC(c2c(CC)cccc2)=O)C2CC2)C)=O)cn2c(n1)CCCC2 Nc1cc(C(=O)NCC2CCC(NC(c3ccc(Cl)cc3Cl)=O)CC2)ncc1Cl C12(NC(c3cc4c(s3)COCC4)=O)CCCC1CN(C(=O)Cc1cnns1)C2 C(C1=NOC2CCCC12)NC(C(CC(c1ccccc1)SCC(=O)NC1CC1)N)=O C(=O)(CCCC(=O)N(C)C)NC(C(C)NC(c1cccc(N)n1)=O)C C(C(COC)CC(=O)NCC1CN(C(c2n[nH]c(C)c2C)=O)C1)OC C1(C(=O)NCC2(CC)CC2)(C(C)C)CCCN1C(=O)C(C)(C)N(C)C(=O)OC c1(C(N(CCC(C(C)C)NC(c2c(CC)cno2)=O)C)=O)ccnc2[nH]nnc12 C1(C(=O)NCCN(C(=O)CC(C(F)F)c2ccccc2F)C)Cc2nncn2C1 C1(NC(CN(CCC(C)C)C(=O)CSC(F)F)=O)CC2CC1C(O)C2O N1(c2[nH]c(=NCCN3C(C)CCC3)[nH]c(=N)n2)CC2(CCCC2)c2ccccc21 N1(C(C=C(CC)C)=O)CCC(C2(NC(c3ncn4c3CCCC4)=O)CC2)CC1 C1(C(=O)NCC2(C(=O)NC(c3cn(C)cn3)C)CC2)CC2(CSC2)C1 N1(C(C)=O)CCCCC1C1(CC(=O)NCCc2ccc(Br)s2)CCCC1 N#Cc1cc(F)c(F)cc1C(N1CC2CN(c3cnccn3)C2C1)=O Cc1nc(Cl)sc1C(N1CCN(c2cccc(Cl)n2)CC1)C(=O)NCC1(C)CC1 C(C(O)C(C)(C)C)C(N1C(Cn2cc(-c3cn(C(CC)C)nc3)nn2)CCC1)=O CC(C)CC(N)CC(=O)N1CC2CCCC1C2C(C)O C1(NC(C2CS(=O)(=O)CC23CC3)=O)CCCC12CN(C(c1ccc[n+]([O-])c1)=O)C2 c1(C(=O)NCC2CCC(NC(CC(C)C3CCCO3)=O)C2)cn2cc[nH]c(=O)c2n1 N1(C(CC=C)=O)CCC2CCC(NC(c3cc4n(n3)CCCN4)=O)C12 Cc1cc(F)c(C(=O)N(C2CCN(C(C3CCCCN3C)=O)C2)C)c(F)c1 c1(CC(=O)N(CC)CC2CN(C(=O)NC3CCCCC3)CCO2)nnc(C)n1C C1(NC(C(C)N(C)Cc2ccco2)=O)CCCCC1C C1(F)(C(=O)NC(CC)CN(C)C(C2CC(C)(CC)C2)=O)C(C)(C)C1(C)C C1(NC(=O)Nc2ccc(C3CCOC3)s2)CC(CO)C12CCC2 C1(C(=O)NC2CCC(NC(c3cccc(OC)n3)=O)CC2)CCOC(=O)CC1 C1(CNC(C2C(CC)C2)=O)CCCC2(CN(C(c3cccc(C)c3O)=O)C2)O1 c1(COC)cc(C(=O)NC2(CCCNC(C3CCCN3C3CC3)=O)CC2)on1 C1(C(N2CC(NC(C34CC3CCC4(F)F)=O)CC(C)C2)=O)CCN(S(N)(=O)=O)CC1 N1(C(Cn2ccc(C)n2)=O)CC2(C1)SCCC2NC(=O)Cc1ccnn1C c1(C(=O)NC2CCN(C(C34CCCCC3OCC4)=O)CC2)ccc(F)c(F)c1F c1(C(=O)NCCC(CC)(CC)NC(=O)C(O)CN(C)C)n[nH]c2c1CSCC2 C1(C2CCOCC2)(C(=O)OCc2cn(C3CCCC3)cn2)CCOCC1 CC1CCCC1(C(N1CCC=C(Cl)C1)=O)NC(=O)CC1C(C)(C)C1(C)C c1(C(=O)NCCC2(C)CCN(C(=O)CC3OCCC3(C)C)C2)cccc(F)c1N C1(O)(CC(=O)NCC2OCCC2C(=O)NCCc2ccoc2)CCCCC1 N1(C(C=CC)=O)CCC2(NC(c3cc(Br)co3)=O)CCCC12 C12(C(=O)NC(C3CCCN3C(=O)Cc3ccc(O)nc3)C)CC1COC2(C)C C1(NC(c2nn(-c3cccc(C)c3)c(C)c2)=O)CCN(C(C2CC2C)=O)C(C)C1 C(c1ccc(Br)o1)=CC(=O)NCC1CCC(NC(C2CCN2C2CCCC2)=O)C1 N1(C(C(CCC)(C)C)=O)CCOC2(CCCN(C(=O)C(C)(COC)OC)C2)C1 C1(C(=O)NC(C(C)C)CCNC(=O)CCN2CCN(C)CC2)CN(C)CC(C)O1 Cc1cc(C(=O)NC(C2CN(C(=O)Cc3ccc(C)s3)CCO2)C)ncc1C(F)F C12(CNC(C(CC)N(C)C)=O)CCC(CC1)CN2C(=O)CCNC(=O)CO CC1CCCC1(C(=O)NOCC1(CF)CC1)NC(=O)CC1CCCC1O CCC(C)C(C)(c1nnnn1-c1ccccc1C)S(C)(=O)=O.c1(N)cnn(CC)c1C c1(OC)cc(F)c(C(=O)NC(C)(C)CNC(c2ccc3sccc3c2)=O)c(F)c1 Cc1cc(C(N2CC3CCN(C(=O)CS(C)(=O)=O)CC3C2)=O)ccc1[N+](=O)[O-] CC1(C)CCOC1C(=O)NC1CN(C(c2ccnnc2)=O)C1 C12(C(=O)NC3(CNC(=O)CCC4CCCCC4)CCCO3)CC3CC1C2C3O c1(NC(N2C(c3nc(C)c(C)[nH]3)CCC2)=O)ccccc1S(=O)(=O)C(F)F CC1CN(C(C2(C)CCCN2C(c2ccc(O)c(F)c2)=O)=O)C(C)CO1 N1(C(c2c(CC)ncs2)=O)CCC2CN(C(C3CC=CC3)=O)CCC2C1 c1cc(N(C2(C(F)(F)F)CCNCC2)C2CC2)c2ccncc2c1 C(=O)(C(O)CCCNC(C1CCC(OC)C1)=O)NCc1c(OC)cccc1 Cc1ccc(C)c(OCC(=O)NC2C3CC2N(C(c2cc(C(N)=O)c[nH]2)=O)C3)c1 c1(C(=O)NC2CN(C(C(COC)COC)=O)CC(F)C2)cc(Cl)cc(C)c1OC C1(CC)CCCN1C(=O)C(=O)Nc1cc(CNC(=O)COCP(C)(C)=O)on1 C#Cc1ncccc1NC(C1CN(C(=O)NCCC)C1)=O C1(CCC(C)C)CCN(Cc2cnc(C(C)(C)C)o2)CC1 c1(N2CCCC(NC(c3cccnc3C3CC3)=O)C2)cccc(F)c1[N+](=O)[O-] N1(c2c(C#N)cc(C)c(C#N)n2)CC23CCCC2(CN(S(C)(=O)=O)C3)C1 c1(C(N2CC3CC(NC(C(C(C)C)N(C)C)=O)C3C2)=O)c[nH]c2cc(N)ccc12 C(=O)(C1=CC2C=CC(C1)C2)NC1CCC(CC(=O)NC(COC)C)C1 N1(C(C2(NC(=O)NCC)CCCC2)=O)CC(CNC(=O)C(C)=C(C)C)CC1C C(=O)(C(F)(F)C1=CCOCC1)NCC1(C(C)NC(=O)CCc2ccco2)CC1 C1(C(=O)NC(C2CCN(C(c3cn(C)nn3)=O)C2)C)Cc2cc(Cl)ccc2C(=O)O1 Cn1nc2c(c1C(=O)NCCN1CCN(C(C3CCNC3=O)=O)CC1)CCCC2 C1(N(C(CCc2c(C)ncs2)=O)C)CCCN(CCCCCF)CC1 C12CN(CCO1)C(=O)C2.n1(CC(c2nc[nH]n2)C)cc(C2(C)CCCO2)nn1 c1(CC)ccnc(C(N2CCC(C(=O)NC3CC3C3CC3C)(C(C)C)C2)=O)c1 N1(C(C=COCC)=O)CCC(NC(c2ccco2)=O)C(F)C1 c1(C(=O)NC2CCCC3CCCCC23)cccc2c(Br)[nH]nc12 N1(C(c2cn(CCN(C)C)nn2)=O)CCCC(CNC(c2nnn(C)c2N)=O)C1 C123CCC(CC1)(C2)C(=O)N3.C(=O)(C(O)C(C)C)NCCCNC1CC1.CSC N1(C(CONC(C(CSC)C)=O)=O)CC2(CCCCCC2)C1 C1(NC(C2(CC)CCN(C(C3CCC4CC34)=O)CC2)=O)CCC2(CCC2)CC1 C1(NC(C(C)(C)OC(C)=O)=O)CC12CC(NC(c1cc(C3CC3)ccn1)=O)C2 c1(C(N(CC(C)N(C(C2C(CCOC)C2)=O)C)C)=O)ccc(O)nn1 C12(CNC(C(C)OCC)=O)CC3CC(CC(NC(=O)C=CC4CCOC4)(C3)C1)C2 C1(F)(C(=O)NCCCCN(C(C)C)C)CCCN(C(C2CC(=C3CC3)C2)=O)C1 C1(CC#C)(C(=O)OC(C)C)CCCCN1CCC(=O)NC1CCCCCC1 C1(OC)(CNC(=O)C(C)OC)CN(C(c2occc2Cl)=O)C1 Cc1cccc(O)c1C(=O)NC1CCCC(NC(C2(C)COCCO2)=O)C1 C(C(C)(CO)OC)NC(CN(CC#C)C(C1CCCC1CCC)=O)=O c1(C(=O)NCC(CNC(C=C(CC)CC)=O)(C)O)ccc2c(c1)CNC(=O)N2 C1(C(=O)NCCOCCN(C(COCCC#C)=O)C)CCCOC1c1ccccc1 C1(NC(C(c2c(F)cccc2F)C)=O)C2CC1CN(C(c1cc[nH]n1)=O)C2 c1(C2C(C(=O)NC(C3CN(C(c4cc(O)no4)=O)C3)C)C2)cncn1C CCC(C(=O)N(C)CC1CCOCC1)N(C)C(c1ccc(COC)o1)=O CC1(C)CC(NC(c2cscn2)=O)CN(C(c2ccc(-c3nc[nH]n3)cc2)=O)C1 C(C(C)(CC)C(=O)NC(CC)C(C)(C)C)NC(C(C1CCC1)OCC)=O NC1(C(=O)NC2CCCC2Cc2ccc(F)cc2)CC12CCC2 Cc1nccc(C(=O)NCC(C)(C)C(=O)NCCCC2CC2C)c1N c1(C(N2C(CN(C(=O)C(=O)C(C)(C)C)CC)CCC2)=O)ccc(OC)c(Cl)c1 N1(C(CC2(OC)CN(C(C(C)OCCC=C)=O)C2)=O)CC(CO)C(C2CC2)C1 C1(C)(C(CNC(C2C(OC)CC2)=O)(C)C)CCCN1C(c1cc[nH]c1)=O n1(CC(C)C)c(N(C)CC2CCCC2O)nnc1C1CCC(C(F)(F)F)O1 c1(OC)noc(C)c1C(=O)NCCC1(O)CN(C(c2cncc(O)c2)=O)C1 C12(NC(COc3c(C)cc(Cl)cc3)=O)CCCCCC1N(C(=O)C(F)F)CC2 CC(=O)CCCC(=O)N1CCC(N(C)C(c2ccc(-c3cscn3)nc2)=O)C1 c1(NC(C2C(NC(CCC)=O)CCC2)=O)ccc(C)nc1 C(CCCC(=O)NCC1CCOC1C(=O)NCC(C)C1CC1)NC(C)=O CC1CCN(CC(=O)N(C(C)CN(C)C(c2ccn(CCF)n2)=O)C)CC1 c1(CC)ccncc1NC(=O)C(C1CN(C(C2CC(C)CCS2)=O)C1)OC c1(NC(C23C(CN(C(C4C(C)(C)COCC4)=O)C2)C3)=O)cccc2c1CCC2 C1(C(=O)NCC(C(=O)NCC(CC)OC)N(C)C)CCC(=O)N1CC C(CC(F)F)(C(=O)NCCOc1ccncc1)N(C)C(C1NC(=O)NC1=O)=O c1(C(=O)NCC2CCN(C(=O)CCOc3ccc(Cl)cc3)C2)ccc(CO)nc1 C1(N(C(=O)Cc2cnccn2)C)CN(C(c2cn(C)c(C(F)F)n2)=O)CC12CC2 CCC(C)CCC(=O)N1CCC(Cn2cc(-c3cccc(OC)c3)nn2)C1 C(=O)(C(O)C1=CCCCC1)N(C1CC(NC(=O)Cn2ncc3ncccc23)C1)C c1(OC)cc(NC(N2CCC(C)(C(=O)NCc3cccc(Cl)c3)C2)=O)cc(F)c1 c1(OC)cc(OC)c(C(=O)NC(CNC(=O)C(C)C(C)(C)C)C2CC2)cc1OC c1(NCC(CN(CCC)C(C)C)(C)C)ccc(OC)c(C(C)C)c1 C1(CC)CN(C(=O)Cn2cnc(C(=O)OC)n2)CCC1CNC(=O)Cc1ncc[nH]1 c1(C(=O)NCC2CCCC(NC(C3(OC)CCOCC3)=O)C2)ncc(Cl)nc1Cl C1(CNC(CC2(OC)CCCC2)=O)CC(C)(C)CN1C(c1cn(C)nc1C(C)C)=O N1(C(CC(=O)NCCC(F)(F)CO)=O)CCCC(C(=O)Nc2nccs2)C1 c1(C(N2CCOCC2C2CCC2)C(=O)NCCCF)cc2nc(F)ccc2o1 N1(C(C2(SCC)CC2)=O)CCN(C(=O)C(C(C)C)N2CCCCC2)C(CO)C1 C1(CC)CCN(C(=O)CS(C)(=O)=O)C1C(=O)NC(C)CC1CC1 CCC(C)C(O)C(=O)N1CC(CCNC(c2csc(-c3cnn(C)c3)n2)=O)C1 C1(C(N2C(CNC(C(CC#C)C)=O)CC(F)(F)C2)=O)CC2(C1)CC(C#N)C2 Cc1ccc(-c2ocnc2C(=O)NCC2CC2NC(C2(C)CC2(F)F)=O)s1 C=C(CNC(C1CC1(F)F)=O)CCNC(=O)C(O)Cn1cncn1 C1(C(N2C(C=CC(N3C(CN(C)C)C=CC3)=O)CCC2)=O)CC(=O)CC(=O)N1 c1(C(=O)NC2(CO)CCN(C(C(CC)OC)=O)C2)cnn2ccc(C)nc12 c1(C2CCN(C(=O)NCc3cc(CCC)n[nH]3)C2)ccc(Br)cc1 Cc1cc(-c2nc(-c3ccc(CCF)cc3)n(C(C3(C)CC3)C)n2)c(C)o1 N1(C(C(CC2CC2)NC(c2cc(C(C)C)[nH]n2)=O)=O)CCC2(CSC2)C1 CP(C)(=O)C1CCCCC1C(N1CC(NC(=O)CC2C=CCCC2)C1)=O N1(C(CCCCCOC)=O)CC2CC(C1)CN(C(=O)CC1CC3(CCC3)CO1)C2 N1(C(CC(C(C)OC)NC(=O)CC(O)C2CCCC2)=O)CCCC2(CCC2)C1 N12CCC(C)C(C1C)NC(=O)C=CCCC2=O.C1(O)(OOCCCCC)CCCC1.C.OOC c1(C(=O)NC2CC(NC(C3C(C=C)OCC3)=O)C2)cc(C)c(F)cc1Br c1(CC(=O)NCCN(C(C(COCC)C)=O)C2CC2)coc2cc(CC)ccc12 N1(C(CCCCC)=O)CCC(C(F)(F)F)C(N(CC(C(=O)NCC)F)CC)C1.CC S(=O)(=O)(c1c(Cl)cc(Cl)cc1Cl)NCc1cccc(NC2CCCC(C)CC2)c1 c1(OCCC)cncc(C(N2CC(CNC(=O)C(=O)NC3CC3)(OC)C2)=O)c1 S(=O)(=O)(c1ccccc1NC(=O)C(C)(CC)CO)N(CC)CC.C(CSC)N C(CCCCCC(=O)NC12CC1CN(C(=O)CN(c1ccccc1)C)C2)OC S(=O)(=O)(c1cnc(N2CCC(CCC)C2)cc1C)NC(CCC=C)(C)C c1(C23OCC(NC(=O)Nc4cccc(OCCF)c4)C(C2)C3)c(F)cccc1F CC1(C)Cc2ccc(C(N3CC(O)CC3CNC(=O)CC#N)=O)cc2O1 C1(C(=O)NC(C)C=CC(=O)NC2CC3CCC2C3)COCCC1(F)F N1(C(c2n(C)c(=O)ccc2)=O)CCC2(CCCC2NS(=O)(=O)CCCCl)C1 C(=O)(C(C(C)(C)C)C1CCC1)NC1(CO)CN(c2cc(COC)ncn2)C1 C1(C(=O)NCCC2CCOC2)CCCCN1C(=O)CCC(=O)NC c1(C(=O)NC2CN(C(=O)CCC3CCC3)CC2O)ccc(Cl)c(C(F)(F)F)c1 C1(C(=O)NCC2(CNC(C3N(C(=O)OCC)CCC3)=O)CCC2)CC(=O)N(C)C1 N1(C(c2c(CC)[nH]nc2Cl)=O)CCCC(NC(c2ncc(Cl)cc2Cl)=O)C1C c1(OC)ccc(NC(=O)NCC(N2CCN(C(=O)CC(F)(F)CC)CC2)=O)nc1 C1(C(N2C(CNC(C3COCCO3)=O)CC(C)(C)C2)=O)CCc2nc[nH]c2C1 C(CCCCC(=O)N1CCCCC1CF)NC(C1CCN(C(C)C)C1)=O c1(C(N(CC(C)NC(C(CCC)N(C)C)=O)CC)=O)cccc2nc(N(C)C)oc12 CCC(C)C(O)C(=O)NCCN1CCC(NC(=O)CCCn2cccn2)CC1 Cc1cc(C(N2CCC(CNC(=O)C(F)(F)c3cncs3)C(C)C2)=O)cnc1O c1(C(=O)NCC2(NC(C(C(C)C)OC)=O)CCCCC2C)cncc2ccsc12 c1(OCCNC(CC2CCN(C(c3c(C)n[nH]c3)=O)C2)=O)c(C)ncnc1C CC1CCN(C)CCN1C(N1CCC(CC(C)(F)F)CC1)=O CCC(C)C(C(=O)NCC(C)(C)CNC(=O)CCCC1CCC1)NC(=O)C(C)C Cc1cn2cc(C(=O)NCC34CC(CN3C(C3CCC(F)C3)=O)C4)nc2s1 N1(C(c2c(C(C)C)nns2)=O)CC2CC(C1)C(CO)C2NC(c1nonc1N)=O N1(C(CCN(CC=C)C(c2n[nH]c(C)c2O)=O)=O)Cc2cncnc2C1 c1(CC(=O)NCC(CNC(c2c(CC)occ2C)=O)C)cccc2cccnc12 c1(OC)ccc(NC(c2cnnc(O)c2S(=O)(=O)N(C)C)=O)c(Cl)c1 N1(C(CCOC)=O)CCC(CO)(NC(=O)C(C)OCc2ccccn2)C1 c1(C(N2CC(CC)N(C(c3oncc3C)=O)CC2)=O)c(C)ccc(Br)c1F n1(CC(=O)NC(C)CN(C)C(C2(C(F)F)CC2)=O)c(C2CC2)nc2ccccc12 CC(C(=O)NCC1(NC(c2cc(C(C)C)cc(Br)c2)=O)CC1)P(C)(C)=O c1(C(N2CCN(C(c3ccnc(Cl)c3)=O)C3CC23)=O)cccc([N+](=O)[O-])c1Cl C=CCCCC(C(=O)NC(C)(CO)C(F)(F)F)NC(=O)COCC(F)F C1(CCC(=O)NCC(N(C)C(C2(C)CC2(F)Cl)=O)C2CC2)CCCCN1C C(CNC(C1CCCC1OC)=O)(CCNC(C1(O)CC(C)C1)=O)OC C1(CNC(C=CS(C)=O)=O)CN(C(=O)CCOC2CCCC2)CCCO1 c1(C(CCCCCC)C2CC2)cc(=NCc2cc(C)cc(C)c2)[nH]c2ccc(Cl)cc12 C1(CNC(C2C(CC)C2)=O)C=CC(NC(=O)CC2(C(=O)NC)CC2)C1 C(CCC(N)=O)(C(=O)N(C)CC1(O)CN(C(C2(C)CCN(C)C2)=O)C1)NC(C)=O C1(NCc2nc(C)nn2-c2ccc(F)c(Cl)c2)CCCC2(CCC2)O1 C=CCC(CNC(c1ccc(C2CC2)o1)=O)C(=O)N1C(CO)CC1CO C12(N(C)C)CCC(C(N3CC4CC4(CNC(c4cnns4)=O)C3)=O)(CC1)C2 Cn1ccc2[nH]c(C(=O)NC3CCCC(NC(=O)Cc4c[nH]nc4O)C3)cc12 C(=O)(C(C)CC(=O)OOC(F)F)NCC1(O)CC(NC(CSCCOC)=O)C1 C1(NC(C2(C3CC3)CC2)=O)CS(=O)(=O)CC1N=c1[nH]ncs1 c1(CC(=O)NCC(CNC(CC(CC)(F)F)=O)F)cccc([N+](=O)[O-])c1C C(=O)(C1=CC2CCCC12)NCC1CCC(NC(CC2(C(=C)F)CCC2)=O)C1 CC1OCCCC1C(=O)NC12CC(C1)N(C(=O)Cn1ncnn1)C2 c1(C(N(CC(C)CNC(C2CC(F)(F)C2)=O)C)=O)cccc2c1CC(C)(C)C2 C1(CC=C)(NC(C2(C(C)C)COC2)=O)CCN(C(c2ccc(SCC)cc2)=O)C1 c1(CC)cc(C(=O)NCC2(O)CCN(C(C3(C)CCCC3(F)F)=O)C2)cc(O)n1 C=CCC(CC=C)C(=O)N1CC(C)CC1C(=O)Nc1cc(C2CC2)ns1 C1(NC(c2ccc(C3CC3)cn2)=O)C2CC1N(C(C1(O)CC(CF)C1)=O)C2 C(=O)(CS(=O)(=O)CC(=O)NCC(CO)NC(=O)CC1C=CS(=O)(=O)C1)OC c1(C(=O)NC2CCN(C(Cn3c(C)nc(C)n3)=O)C(C)C2)cc(N)cc(O)c1C c1(C(=O)NCC(C)N(C(CC2(C=C)CCC2)=O)C)cccn2cncc12 C1(N(C)C)CN(C(=O)C=CCC(C)(C)NC(=O)CCc2ccc[nH]2)CC1O N12CC3CC(CC3C1)C(=O)N(CC1CC1)CC2=O.C1(C=O)CCC1.C1(C)CC1 C(=O)(C(CO)C(N(CC)CC1CCCN1C(=O)COCC1CCCC1)=O)N.C1CC1 C=C=C(C)CC(=O)NCCCC(=O)NCc1cccc(OC)n1 C1(C(N(CCc2ccsc2)N(C(=O)CSC)CC)=O)CCC1(C)C C=C(C)C(C)(O)C(=O)NCC(C(C)C)NC(c1cncc(N2CCCC2)n1)=O O(NC(=O)C(C1CCOC1)NC(=O)C=Cc1ccccc1)C(c1ccco1)C N(C)(C1CN(C(=O)C(=O)NC)CCc2ccccc21)C(CC(CC)C1CC1)=O c1(C(N(C(CCNC(COCCC=C)=O)C)C)=O)cccc(C2OCCO2)c1 N1(C(C2(SC)CC(=O)C2)=O)CC(C(=O)NC2CC3(C2)CC(C)(C)C3)CC(C)(C)C1 C=CCC(C(=O)N1CCCC1(C)C(=O)NCC(C)(C)OCCO)NC(C)=O CCN(C(C)c1cncs1)N(C)C1CCc2c(F)cccc21 CC1(C)C(c2cccc(Cl)c2)CCN1C(=O)NCCCC[N+](=O)[O-] Cc1cc(C(F)(F)F)ccc1C(=O)NC1CCN(Cc2cnccc2Cl)C1 c1(C(=O)NCC2(C(F)F)CCN(C(C3CC=CCO3)=O)C2)ccn2c1CCCC2 S(=O)(=O)(C1CCC(=O)CC1)N1CCN(Cc2cccc(C(=O)NC)c2)C2(C1)CC2 C(=O)(C(C)CC)N(CC(=O)NCCSC1CC(C(=O)N(C)C)C1)CC CS(=O)(=O)c1cc([N+](=O)[O-])ccc1NC1CC(C2CCCNC2)C1 CCC(C(=O)OC)C(=O)N1CC=CCC1C(N1CC(CO)C1(C)C)=O c1(CC(=O)OC)c(C)nn2c1CN(C(=O)NCCSC)CC2 C1(C(=O)NC2(CO)CN(C(C3(c4ccno4)CC3)=O)C2)C2CCC(=O)C12 c1(C(=O)NCc2cc(O)ns2)ccc(CNC(c2csnc2Cl)=O)cc1 C1(NC(c2cncn2-c2ccccc2)=O)(CO)CN(C(=O)CCc2ccoc2)C1 N(C1CN(C(=O)C=CS(C)=O)CCc2ccccc21)C(c1cc(OC)nn1C)=O CC1CCn2ncnc2N1C(=O)NC1(C)CCCC1N1CCCC1 c1(CCC(=O)NCCNC(C2(Cl)C(C)(C)C2)=O)ccc(N)cn1 C(=O)(C(CO)NC(=O)CN1CC2CC2C1)N(C(CC1CCCC1)CO)C C(=O)(C(CN=[N+]=[N-])NC(c1occc1C)=O)N(C)Cc1n(CC)cnn1 c1(C(=O)NCC(CO)NC(C2CCC(F)(CN)C2)=O)cn(CCO)c(=O)nc1O CCCCC(=O)NCC(C)CNC(C1(CCOCC)CCCC1)=O N1(C(C2C(C=CC)CC2)=O)CC(NC(=O)C(C)(C)CC#N)C(C)(C)C1 c1(CCC)cc(C(=O)NC(CC2CCCC2)C(=O)NC2CC=CCC2)n[nH]1 c1(CC(=O)N(C)CCN(C(=O)CC2CC=CC2)C)ccc2nsnc2c1 c1(C(=O)NCCCC(=O)N2CC(OCC(=O)NC)C2)cc(C#N)ccc1N c1(CC(=O)NC(CCCNC(c2cnc(SC)s2)=O)C)c(C)n[nH]c1C c1(-n2ncc(C(=O)Nc3nc(OCC)oc3)c2)nn(C)c2c(=O)[nH]cnc12 C1(C(=O)NCC(C)C(=O)NCCC2(C)CCC2)CCC2(CCC2)O1 c1(C(N(C2CC(NC(C34CCC3C4)=O)C2)C)=O)csc(C2CC2)n1 C1(C(=O)NCc2scnc2Cl)CCOCCN1C(=O)CC1C=CCC1 N1(C(=O)C=Cc2ccoc2)CCC2(C1)CN(C(C1CC(CCO)C1)=O)C2 c1(C(N2C(CC)CC(C(=O)OC)CC2)=O)cc(C#N)ccc1Cl c1(OC)ccc(C(N2CCC(CCF)CC2)C(=O)NC2(C)CC2)cc1C1CC1 C1(C(N2C(C#C)CC2)=O)(OC)CCN(C(c2ccc(CC)o2)=O)C1 c1(C(=O)NCC2CCN(c3ccnc(CC4CC4)n3)CC2)cccc2c1CCC2 C(=O)(C(F)(F)c1csc(=N)[nH]1)NCC(CN(C)C(C1(N(C)C)CCC1)=O)O O=C(CCCC1CCCC1)NCCN1CCOCC1.C1(=O)CCCN1.C1C(=O)N1 c1(C(=O)NC(CCNC(C2(CCCC)CC2)=O)C)cncc2c1CCCC2 C1(CC(=O)NCC2(F)CN(C(C(C(C)C)C3CCC3)=O)C2)CCCCC1(F)F N1(C(C(CCC)C)=O)CC=C(CNC(C2CCCC(O)C2)=O)CC1 Cc1[nH]nc2ccc(C(N3CC4(CC4)CC3CNC(=O)CC3(C)CC3)=O)cc12 c1(C(=O)NCCCC(c2ccccc2)NC(CCC#C)=O)cc(Cl)c(Cl)s1 C1(C(=O)NCCN(CCC)C(c2cn(CCN(C)C)nn2)=O)CC2COCC(C1)C2 Cc1ccnc(C(=O)N(CC(C)(C)NC(c2ccncc2)=O)C)c1Br c1(C(=O)NC(CCCNC(c2n(CC)ncc2)=O)C)nc(O)nc(O)c1N C1(O)(CNC(c2ccc(CO)cc2)=O)CCCN(C(=O)C(F)C2CC2)C1 c1(CN(CC(C(C)C)OC)C=O)ccccc1-n1nc(C)cc1C CC1C2CC(C2NC(C2CCN(C)CC2)=O)N1C(=O)C1=CCCOC1 C1(C(NOCCN(C)C)=O)(CF)CCN(C(c2cnsn2)=O)C1 C(CNC(=O)C(C)n1ccnc1)(CNC(=O)CC1(NC(C)=O)CC1)OC c1(CC)nc(C#N)cc(=NC(C)CNC(=O)Cc2ccco2)[nH]1 c1(CC(N2C(CNC(C3CCOC3)=O)CC(O)C2)=O)ccc([N+](=O)[O-])cc1 N1(C(CCCOCC)=O)CCCCC12CC(NC(=O)Cc1ccc(CC)cc1)C2 CC1CC2CCC(C(=O)N(c3nnc(C4CC4)o3)C)CN2C1 C(=O)(C(C)(O)C(F)(F)F)Nc1cc(C)c(NC(=O)C(C(C)C)n2cccc2)cc1 C1(C(N(C(CNC(c2ccc(C#C)o2)=O)C2CC2)C)=O)CC2(C1)CC2(F)F CC(C)(C(=O)NC1CNC(=O)OC1)C1=CCN(C(C2CC2c2ccccn2)=O)C1 C(=O)(C1=C2CCN=C2NC=C1)N1CC(CNC(CCc2cc(C)cc(C)c2)=O)C1 C1(C(=O)NCCN(C(=O)C2CC2)C(n2cccn2)C2CC2)CCCC1O C1(NC(CCc2cnc(C)s2)=O)C(CNC(=O)C(C)(C)CC#N)CCC12CCC2 C12(c3onc(CC(C)(C)CCO)n3)CC(N=[N+]=[N-])C1C2 N(C(=NCCC1CCC1)NCC1CCCO1)CC1CCC(C(F)(F)F)CC1 C=CCC(C(=O)N1C(C(N2CC(C#N)C2)=O)CC2CC12)OC c1(NC(C2N(C(C(C)(C)O)=O)CCC2)=O)ccccc1C(=O)N.c1(CC#N)ccccc1 C(=O)(C(O)P(C)(C)=O)N(C1CC1)CC1CCN(C(C2N(C)CCC2)=O)CC1 c1(C(=O)NCCOCCN(C)C(C2(Cl)CC2(F)F)=O)ncccc1F C1(C(=O)NCC(C2CCN(C(C(C)C)=O)CC2)(C)O)CC(=O)N(C)C(=O)N1 N1(C(CC(C)n2cccc2)=O)CCC(O)C(NC(C2CCCN2N=O)=O)C1 c1(N(C)C(=O)OC(C)(C)C)cc(NC(C2CC2Cl)=O)ccc1[N+](=O)[O-] C1(CNC(C=C(CC)C)=O)CN(C(c2ccnn2C)=O)CCC1C(F)(F)F C(c1nc2ccccc2[nH]1)=CC(=O)NCC=CCNC(=O)C#CC1CCOC1 C(=O)(CC(C)(CN(C)C)C(F)(F)F)N1CCC(C)(NC(c2n(CC)ccc2)=O)C1 c1(OCCC)ccc(C(=O)NCC2CC2NC(=O)C(C)(C)F)cc1OCC C1(O)(CN(C(C(CCC)OC)=O)C)CCCN(C(C2(c3cccnc3)CC2)=O)C1 C=CCC(C)(C)C(=O)NCC1CN(C(c2cnco2)=O)CCC1C N1(C(C(C2CCN(C(c3nn(C)c(Cl)c3)=O)C2)F)=O)CC2OCCOC2C1 C(Cc1ccccc1)(C(=O)N(C)CCOCCN(C(=O)CC(C)F)C)NC(=O)NC C(=O)(CC1=NNC(=O)C1)N(C1CCN(C(c2c(C)cc(N)cc2)=O)C1)CCO c1(COC)ccc(-n2ccnc2-c2cn(C)nc2-c2cscn2)c(F)c1 c1(CN(C=O)CCNC(=O)CNC(c2ccco2)=O)ccco1.C1(=O)CN1 N1(C(CNC(=O)OCC=C)=O)CC2CC(C1)C2NC(=O)C(O)C(C)CC N1(C(CCC)=O)CC2CCC2(CCNC(C2CC3(CCCC3)C2)=O)C1 C(=O)(C(C)C(C)C)N(CC(C)N(C(=O)COc1ccsc1)C)C Cc1nc(C)c(C(N2CCC(NC(=O)C(c3ccnc(C4CC4)c3)(F)F)C2)=O)[nH]1 CN1CCN(C(=O)CC2(N(C)C)CCC2)C(CNC(c2cc(C3CC3)ns2)=O)C1 C1(NC(Cn2c(C)nc(C)n2)=O)CC(NC(=O)CN(C)C)C12CCOCC2 Cc1[nH]nc2ncc(C(N3CCC(CO)(NC(=O)C(C)c4ccco4)C3)=O)cc12 C1(CC)CN(C(=O)CCCCCSCCCOC)CCC1NC(c1ccc(F)o1)=O Cn1cc(C(=O)NCC2(NC(c3ccc[n+]([O-])c3)=O)CC2)c(-c2cccnc2)n1 c1(C(=O)NCCC2N(C(c3n[nH]c(=N)[nH]3)=O)CCSC2)ccc2c(n1)CCC2 CCC(CC(C)C)C(=O)NC(C(N1CC(=O)NC(=O)C1)=O)C1CCCC1 N1(C(C(CC)F)=O)CCC2(C1)CN(C(c1cc(C)ccc1F)=O)CCO2 N1(C(C2CC3C=CC2C3)=O)CCCC2(C1)CN(c1ncc(F)cn1)CCO2 N1(C(c2nc(CC)sc2N)=O)CCC(C)N(C(=O)CCc2ccccn2)CC1 C1(CC(=O)NCC2C(C(=O)NCCCSC)C2)CCC(C)(C)C1 c1(C(=O)NC2(CC)CCCN(C(C3C(C=C)CC3)=O)C2)cc2nnn(C)c2s1 C12(F)CCCN(CC1)C(=O)NC2.Cc1ccc(-c2noc(C(F)F)n2)n1C C1(N(C)C)CCCN(CCC(=O)NCC2(O)CN(C(=O)CC3CCCOC3)C2)C1 c1(CNC(C(CO)NC(C2C3CC(=O)CC32)=O)=O)ccc(F)c(F)c1 C1(CC(=O)NCCCOCCC(=O)NC23CC(CO)(C2)C3)CC2(CCC2)C1 CC(C)C(CCC(=O)NCCCCS(C)=O)NC(=O)C=Cc1ccsc1 N#Cc1ccc(N2CCC(C(=O)NCC3CC(NC(C4CCC4)=O)C3)C2=O)cc1 c1(CC(C)NN2CCCC(C3CCCCN3C)C2)ccc(OCC(F)F)cc1 c1(OC)c(C)nc(C(C)(C)C)[nH]c1=NCC1(F)CCN(C(c2ccncn2)=O)CC1 c1(CC(=O)NCCN(C(=O)CC(C)CN(C)C)CC)ccc(F)cc1 C=CCCC(F)(F)C(=O)N1CC(CC(F)C(=O)NCC2CNC(=O)C2)C1 C=CCC(C)(C)CC(=O)N1CCN(C(c2c[nH]nc2F)=O)CC(CO)C1 N1(C(c2c(C)cco2)=O)CCCOC(CNC(c2ncccc2C(F)(F)F)=O)C1 C(=O)(CC1=CCCCC1)N1CC(OC)C(NC(c2cnc(Br)s2)=O)C1 c1(CC)ccccc1C(=O)N(C)CCNC(=O)C=Cc1sccc1C c1(C(N2C3CC(NC(c4cn(C)nc4C(F)F)=O)(C3)C2)=O)ccc2ccnn2c1 C12(CNC(c3[nH]cc(C)c3)=O)CCCC1CN(C(=O)CCc1nncs1)C2 C1(N(C)CCn2cnnc2)CN(C(c2ccc(C3(C(=O)O)CC3)nn2)=O)CCO1 CC#CCCCC(=O)N(CC(=O)N(CCCCO)C)CCOC c1(OC)cc(N)c(Cl)cc1C(N1CC(NC(=O)C(C)(C)CF)CC(O)C1)=O Cn1cc(C(=O)NC2CCC(NC(c3occc3Br)=O)C2)c(-c2cccs2)n1 C1(CC(=O)N(C2CCCN(C(c3ccc(CSC)o3)=O)C2)C)CC(C)(C)CCO1 Cc1cccc2c(C(N3CCCC(NC(c4snc(Cl)c4Cl)=O)C3)=O)coc12 C(=O)(C(C)C(F)(F)F)N1CCC(CC(C)NC(c2cnc(Cl)n2C)=O)CC1 N1(C(C(CSC)OC)=O)CCC2CN(C(C3CC(OC4CCC4)C3)=O)CC12 c1(NC(C2CN(C(C(C3CC3)OC)=O)CC2C)=O)nccc(C)c1C(C)=O N1(C(c2cnc(C(C)OCC)s2)=O)CCN(C(C2CCC(=O)O2)=O)CC2(CC2)C1 C1(C(=O)NC(C2(O)CN(C(=O)CS(C)(=O)=O)C2)C)CCC2(CCC2)O1 Cc1nc(NC(C)C(C)(C)CO)cc(NCCCCC(F)(F)F)n1 c1(C(C)(C)C)ncc(C(=O)NCC2CC2NC(=O)CSCC#N)[nH]1 C1(C)(CC)CC(NC(c2[nH]cnc2COC)=O)CN1C(=O)CCNC(=O)C=CCl N1(C(N2CCN(CC(=O)Nc3cn(CC)nn3)CC2)=O)C2CCC1CC1(C2)N=N1 C(=O)(CC(C)(C)C(F)(F)F)N1CC(C)N(C(=O)CCn2ncn(C)c2=O)CC1 N1(C(c2ccc(CC)nc2)=O)CC2CCC1C(NC(=O)C(C)C(C)(C)O)C2 C(CCN=c1nc(O)c2cccc(Br)c2[nH]1)NS(c1cccc2c1CNC2=O)(=O)=O C#Cc1ccc(C(N2CC(C(=O)NC(C3CCCCO3)CC)(CC)C2)=O)o1 c1(C(=O)NC2CC(CCNC(C(C3CCC(=O)N3)C)=O)C2)c[nH]nc1F Cc1ccccc1C(N(c1nnc(C2CCCN2C)s1)Cc1cccnc1)=O C1(C2CC2)(C(N2CC(N3CCCC3=O)C2)=O)CN(C(C2C3CCCOC23)=O)C1 c1(C(N2C(CN(C(CSCCC)=O)C)CCC2)=O)cc2cccc(OC)c2[nH]1 CCCCCC(O)C(=O)NC(CC(N)=O)C(=O)NCC(C)=CCCC CC1CC(N(C(=O)C(F)(F)C2CC2(C)C)C)CCO1 C=C1CC(C(=O)N(C(C)C(=O)O)Cc2ccccc2)N(S(=O)(=O)CC2CC2)C1 S(=O)(=O)(C1CCCCC1)N1CCC(NC(c2cccs2)=O)CC1 c1(CNC(C2N(C(c3cc(C)oc3C)=O)CCC2O)=O)ccc(O)c(C)c1 C12(C(=O)NC(c3onc(C)n3)C)CC(CO)(CN1C(C1(C)CCCO1)=O)C2 c1(C(=O)OCC)cncc(=NC(=O)C(F)CC2CN(CC3CCC3)C2)[nH]1 CCC(CC)C(O)C(=O)N(CC(C)(C)C(=O)NCC(C)CCO)C c1(CC)cncc(C(=O)NC2(C)CCN(C(=O)C(C)(O)Cc3ccccc3)C2)c1 N1(Cc2nc(C(C)(C)C)on2)CCN(CC2CCC(F)(F)C2)CC1 N1(C(CC)=O)CCN(C(C2CCC23CCC3)=O)CC1c1cccc(Cl)c1 C1(C(N2CC3C(NC(c4c(CC)ncnc4)=O)C3C2)=O)CCC2CC(C)CN2C1 C=CCC(CC)C(=O)NC1C=CCCC1C(=O)NCC Cc1c(C=CC(=O)NCC2CC(O)CN2C(C2CCOC(C)C2)=O)cnn1C c1(C(=O)NCC2C(C(N(C)Cc3ccc(C)s3)=O)CCC2)ncccc1F c1(C(N(C)CCc2ccccc2)=O)ccc(F)cc1Cl.C(=O)(CCO)OC1CCC1 CC(N(C)N1CCC2NC(=O)CCC2C1)C1CC2(CCOCC2)C1 C1(C(N2CC(COC)(CNC(C3CC3C(N)=O)=O)C2)=O)CC(O)CN1C(C)=O N1(C(Cn2c(C)ccn2)=O)CC2CCCC(C1)N2C(c1cnc(CO)nc1O)=O c1(C(=O)NCC23N(C(C4C(C)C4)=O)C(CC2)CC3)cc2c(nn1)CCCC2 N1(C(c2c(C)nsc2)=O)C2CCC1CN(CCOCCN(C)C)CC2 c1(C(=O)Oc2c(C)ccc(C(F)F)c2)cc(C)nc2[nH]cnc12 Cc1ccc(F)c(N)c1C(N1CC2C(CNC(C3(n4cncn4)CC3)=O)C2C1)=O N1(C(C(c2ccccc2)OC)=O)CCC(CNC(C23CC(C(C)(F)F)(C2)C3)=O)C1 c1(NC(=O)NCC2(OC(C3CC(N(C)C)C3)=O)CCOCC2)ccc(C#N)cc1 N1(C(Cc2c(C#C)cccc2)=O)CCC2CCN(C(=O)CC(C)(C)OC)CC2C1 C1(CNC(Cc2nc(C)[nH]n2)=O)CN(C(=O)CC2CCCC(=O)N2)C2(CCC2)C1 c1(C(=O)NC2(C)CC(NC(c3c(C#C)c[nH]n3)=O)C2)nc(OC)cc(OC)n1 CC(CC(N)=O)C(=O)N1CCCC(N(C(=O)CCN2CCCCC2=O)CCO)C1 CC(C)(C)C(C(=O)NC1CCCCC1(C)O)NC(c1cccc(F)c1F)=O Cc1nc(C(N2CCN(C(=O)Cc3csc(C)n3)C(CF)C2)=O)ccc1[N+](=O)[O-] C1(NC(C(C)SCC2CCCO2)=O)C2CN(C(c3ccc(F)s3)=O)CC12 C1(NC(C2(CC=C)CC2)=O)CN(C(c2cn(C)cc2C)=O)CC12CC2 N1(C(c2cn3cccnc3n2)=O)CCC2(CCCN(C(c3occc3Br)=O)C2)C1 N1(C(c2ccc(CNC(CS(CC)=O)=O)o2)=O)CCC2CCN(C)CC12 C1(C)(C(=O)NC(COC(C)=O)CO)CN(C(C2COCC2C(N)=O)=O)C(C)(C)C1 C1(CC(=O)NC2CC(NC(COCCOCC)=O)C2)COCCOC1 C12(C(N3CC(N(C)C)C3)=O)CC(CN(C(c3cc(F)ccc3F)=O)C1)C2 N1(C(c2cn(CC)nn2)=O)CCC(C)(C)C(NC(=O)CC(C)c2cccnc2)C1 Nc1ccc(CCC(=O)NC(C(=O)NCc2cc(Cl)ccn2)C2CCCC2)nc1 N1(C(c2c(OC)nc(C)s2)=O)CC2CCCC(C1)N2C(=O)C(C)CN(C)C c1(C)cc2occc2s1.c1(C(N(C)CCN2CCC2)C2CC2)cccs1.S c1(C(=O)NC2CN(C(CC=C(C)C)=O)C(C)C2)coc(S(=O)(=O)N(C)C)c1 CC(C(=O)N1CC2CC(NC(=O)CCc3cccs3)CC2C1)C(C)C(C)(C)C Cc1noc(C)c1C(C)C(=O)NC(C)(CNC(=O)CSS(C)(=O)=O)C(C)C C(=O)(C(CC(C)C)NC(c1ccc(O)nc1)=O)N1CCC(COC(C)=O)C1 N1(CC)C(=O)CCC1CC(N1CC(F)(CNC(C2(CSC)CC2)=O)C1)=O N1(C(C(C)(C)SC)=O)CCC2C(C1)NC(=O)CN2C(=O)CC1CC(F)C1 S(=O)(=O)(c1cccc(=NCc2cc3c(s2)CCCC3)[nH]1)N(C(C1CCCO1)C)C c1(C(NC(=NC)NCc2cc(C(F)(F)F)co2)C)cccc(C)n1 C1(n2cc(CC(N)=O)nn2)CC2CCC1(NC(=O)CSCC(=O)O)C2 N1(C(CCc2cnc(C)s2)=O)CCC(NC(C2(C(N)=O)CC2)=O)C(O)C1 CC1(C)CN(C(C2CCC3CC3C2)=O)CC2(CN(C(C3CC34CC4)=O)C2)O1 CC1CCC(CNC(=O)CSc2ccc(C#N)cc2)CN1C(=O)Cc1ccon1 c1(NC(CC)C(=O)NCCNC(c2ccc(N(C)C)cc2)=O)ccc(C#N)cc1 c1(C(N(C(C)CN(C(=O)C(C)(C)S(C)(=O)=O)C)C)=O)c(F)ccc2n[nH]cc12 N1(C(C=C(COC)C)=O)CC(C(=O)NCC(c2nccs2)C)C(C2CC2)C1 c1(NCCc2ccc(SC)cc2)ccc(S(=O)(=O)N2CCOCC3CC23)cc1Cl c1(OCC(=O)NC2C(CNC(c3cnc(C(C)(C)C)[nH]3)=O)CC2)ccc(Cl)cc1F C=CC1(C(=O)NC(C2CN(C(=O)C(C)C(C)O)C2)C)CCOCC1 C(CCN=C(NCC1(O)CCN=C2CCCC12)N1CCC(F)C1)OC(C)C CC(C)C(C)(CNC(c1cccc(Br)n1)=O)NC(C1CCC2CC12)=O C1(C(=O)NCC(CNC(=O)CCCOC)OC)COC(C)C1.c1ccccc1 C1(C)(C(N(C2CCC(=O)N2)CC)=O)CCN(C(=O)C(C)C2CCC2)CC1 N1(C(CC(CNC(c2cccc3nccn23)=O)O)=O)CCCC12CCCC2 c1(C(N(C2CCN(C(=O)CC3CCOC3=O)C2)C)=O)ncc(Cl)n1C CN1C(=O)CSC1=CC(=O)NCC(C1CCN(C(C2CCC2C(N)=O)=O)CC1)(C)C CCC1=NOC(NC(C(N2CCC(CN(C)Cc3cccnc3)C2)=O)=O)C1 c1(OC)ccc(CCCCC(=O)NCCCCN(C)C(c2csnn2)=O)cc1 C12(NC(=O)CCC3CCCOC3)CCCN(C(c3cc(F)ccc3F)=O)CC1C2 c1(C(=O)NCC(c2cccc(C)c2)NC(CCCOC)=O)scc(C)c1C C1(C(=O)NCC(C)N(C)C(c2cc(C3CC3)[nH]n2)=O)CC12CCC(C)(C)CC2 C(=O)(C1CCCc2sccc21)NC1N(C(=O)OC(C)(C)C)CC12CCNC2=O Cc1ccnn1CC(=O)NCCCNC(c1n[nH]cc1C(C)C)=O C1(OC)CC(NC(=O)C=Cc2cccc(F)c2)CN(C(=O)CC2CC3CC3C2)C1 Cc1nc2cc(C(=O)NCC3CCCCN(C(C4CC4C#N)=O)C3)ccc2s1 c1(C(=O)NCC2CC2NC(c2csc(CO)n2)=O)ccc(OCCF)cc1 c1(CN2CCC(F)(C(=O)Nc3ccc(Cl)nc3)CC2)c[nH]c2cccc(Cl)c12 C1(OC)CCC(N(C(=O)C(C2CC2)C2CC2)C)CC1.C1CNC(=O)N1 CC1(C)NC(=O)OC1C1(NC(C(N2CCC(C)(CCN)C2)=O)=O)CC1 CN1CCN(C(=O)C(c2ccccc2F)O)CC1CNC(c1cccnc1Cl)=O N1(C(C(C(C)C)NC(C)=O)=O)CCCC(NC(c2cc(F)ccc2F)=O)CC1 C1(C(=O)NCCOCCC(=O)NCC(COC)(C)C)CCC2(CC2)C1 CS(=O)(=O)CCC(=O)N1CC2C(CNC(c3ccc(C(N)=O)nc3)=O)C2C1 c1(C(C)C)ccc(C(=O)N(C)CCN(C)C(c2cc(-c3ccoc3)[nH]n2)=O)o1 C1(CNC(C(C2CCOC2)NC(C(C2CC2)OC)=O)=O)CCN(C)CC1 N1(C(C(CCC)C)=O)CC2CN(C(c3c(C)ncnc3C)=O)CCC12 c1(OCC(=O)N)noc(C)c1C(=O)NCC.C1(C)CC2(CNC(=O)OC)CC1C2 c1(OC)nccc(C(=O)NCCC2CCCN2C(C2CCCC(OC)C2)=O)n1 c1(C(=O)NC(C(=O)NCC)CSC)ccncc1OCCN(C)C c1(NCC(CC)C)ccc(S(=O)(=O)NCC(c2ccccn2)O)c(Cl)c1 N1(C(C2(COC)CCC2)=O)CC(NC(C2NC(=O)OC2(C)C)=O)CC2(CC2)C1 C1(N(CCCC)C(C2CC=CC2)=O)CCN(C(C2(C)CC(C)(C)C2)=O)CC1 C(=O)(C(C)C(C)(F)F)N(C)CC1N(C(C(CC=C)NC(C)=O)=O)CCCC1 C#CC1(C(=O)NCc2n[nH]c(C)c2C)CN(C(C2CCN(C)C2C)=O)C1 C(C(COC)C(=O)N1CCC(C(C)NC(=O)CC2CCCCN2C)CC1)OC C1(O)(CCCN(CCOCC)C(C)=O)CCS(=O)(=O)CC1 C1(C(=O)NCC2CCCN(C)C2)CC(O)CCN1C(=O)CCC1OCCO1 c1(CC)sc(C(N2CCC(n3cc(C4(CC)CCCC4)nn3)C2)=O)cc1Br Cc1ccc(NCc2ccco2)c(NC(C23CCC(CC2N2CCCC2)C3)=O)c1 c1(CC(N2C(C(=O)OCC)CC2C)=O)ccc(O)cc1Br C(=O)(CCCCSC)NCC1(O)CC(CNC(COCCC)=O)C1 c1(C(N(C2CCN(C(=O)CC3CNC(=O)C3)C2)C)=O)ccccc1-c1ccccc1 C=CC(C)(O)C(=O)NC1CC(C)(C(=O)NCCc2cncc(C)n2)C1 C(=O)(C(C#N)(CC)SC)N(CCNC(c1n(CCC)ccn1)=O)CCOC(C)(C)C C12(CNC(CCOCC(N)=O)=O)CCCC1N(C(=O)CCBr)CCC2 C(C)(CCCCNC(=O)C(C(C)C)n1cnnc1)NC(C(CC)SC)=O C1(CNC(C(COC)N(C)C)=O)CC2CCC1N2C(=O)C=C(C)Cl C1(C(N(CCNC(C(CC)OC)=O)CC2CC2)=O)CCc2cncn2C1 c1(C(=O)NCCCCNC(c2n(CC)c(O)nc2)=O)cnc2c(c1)nnn2C C1(CC)CN(C(c2ncnn2C(C)C)=O)CCC1NC(c1cc(C(C)C)no1)=O N1(C(C2OCCN(CC)C2)=O)CCOCC(C(=O)NC(C)(CC)CC)C1 c1(C(CCC(=O)OC(CNC(C)C2CC2)=O)=O)csc2ccccc12.C1CCCCN1 N1(C(c2c(C)cnn2C)=O)CCCC(C)(CNC(c2ccsc2C)=O)C1 Cc1cc(Cl)ncc1CCN(C1CCC(OC(F)(F)F)C1)C(=O)NN1CCCCC1 CC(C)CC(CNC(c1csc(O)n1)=O)NC(=O)C(O)C1CC1 C1(C(=O)NC(C2CCCC2)CO)COC2(C1)CN(C(=O)Cc1cnns1)C2 N1(C(C2CCC(CC)O2)=O)CC=CC(NC(=O)Cc2nnc(O)s2)C1 c1(OC)cc(C=CC(N2CCCC2CN(C)C(c2cc[nH]c2C)=O)=O)ccc1F C(=O)(CCS(C)(=O)=O)N1CC(OC)C(C(N2CCCC(F)C2)=O)C1 CC1CN(C(C2CSCCN2C(=O)CCc2ccn(C)c2)=O)Cc2nncn21 CC(C)CC(O)C(=O)NC1CCC(C)(CNC(c2cnc(C3CCC3)o2)=O)CC1 N1(C(CCSCCCC)=O)CCN(C(=O)C2=CCOCC2)CC12CC2 Cc1ccc(O)c(C(N2CC(C3CN(C(C4OCCC4(C)C)=O)CCO3)C2)=O)c1 c1(CC(N)=O)ccccc1CCNC(=O)NC1CC(CO)C(O)C1 C1(NC(c2n[nH]c(CC)c2Cl)=O)CCC2CCN(C(C3CCCC34CC4)=O)C12 N1(C(C(C)=C2CC2)=O)CCCC1CNC(c1ccc(CN(C)C)s1)=O C(CS(=O)(=O)CC(=O)NC1CCN(C(c2cc(OC(F)F)n(C)n2)=O)CC1)OC Cc1nnc2n1CCN(C(C1C3CN(C(C4(C)CCCN4)=O)CC13)=O)C2C c1(C(=O)NCC(C)NC(C(CC)OC2CCCC2)=O)c(F)ccc2ccncc12 C1(CN(C(=O)C(C)(F)F)C)CC2(CCN(c3nnc(-c4ccon4)s3)CC2)CO1 C1(CC=C)COCC1NC(C1(NC(=O)C(C)(C)c2ccno2)CC1C)=O Cc1cc(C(F)(F)F)ccc1C(=O)N(CCCCNC(c1cncn1C)=O)C1CC1 CC(C)C(C(=O)NCC=CC(C)(C)C)C(C)NC(=O)C(C)N=[N+]=[N-] C1(CNC(C)=O)CN(C(c2cc(C(F)(F)F)cc(I)c2)=O)CC12CCOCC2 C1(CC(=O)NCC2(NC(C3(SCC)CC3)=O)CC2)OC(C)(C)OC1=O C#CC1(O)CCCN(C(=O)CC2CCN2C(=O)C(=O)NC2CC2)C1 c1(C(N2CCN(C)C(c3ccc(F)cc3)C2)=O)ccc2c(c1)C(N)CC2 C1(N(CCCn2cc(CC(C(C)C)(C)O)nn2)C(=O)C2CC2)CCOC2(CCC2)C1 c12ccc(C(F)(F)F)nc1[nH][nH]c2=O.C1(N(CCC)CC)CC1C(N)=O C1(C(=O)NCC(C)NC(C2CCCN2C=O)=O)CN2CCCC1C2 Cc1c(C(=O)NC2(CO)CCN(C(C3C=CCCC3)=O)C2)cnn1CC(F)F CS(=O)(=O)c1ccc(C(F)F)cc1F.C1(=O)CC(c2ccc(Br)cc2)C(=O)N1 Cc1nc(C(=O)NC2CCN(CCNC(C3CCC3C)=O)CC2)c(C)s1 N1(C(CSC(C)C)=O)CC(CO)C2(C1)CN(C(=O)CC1CCCC1)C2 c1(OC)cc(N)c(F)cc1C(N1CCCC(NC(C2CCCC2F)=O)C1)=O N1(CC(=O)NC2C=CC(CC(=O)NCCC3N(C)CCC3)C2)CC(=O)NC1=O C(c1ccc(Cl)c(C(F)(F)F)c1)=CC(=O)NCC(CC)NC(C12CC(C)C1C2)=O C1(CCC(=O)NCC(C)(C)NC(CCN(CCCCC)C)=O)CCC(=O)C1 C=CCC(C)(CC=C)NC(=O)C(C(C)O)NC(=O)CCN1CCCC1=O C1(C(=O)NC2C3CN(C(C(C)NC(N)=O)=O)CC2C3)CC2CC(O)CC(C1)C2 c1(C(N2C(C(N3CCCC4CCCCC34)=O)CCCC2)=O)c[nH]c2ccc(I)cc12 C1(C(=O)NCCCN(C(c2c(NC)snc2C)=O)C)CCOC2(CCCCC2)C1 C1(C(=O)NC2CCC(CC(=O)NCCc3cc[nH]n3)CC2)CC2CC(=O)C1O2 N1(C(COCCCC#C)=O)CC(NC(c2c(C)noc2CC)=O)C(C(F)(F)F)C1 N1(C(CC(C)OC(C)(C)C)=O)CCOCC1C CC(C)CS(=O)(=O)CC(=O)NCCC1(N(C2CCCC2)C(C2CN(C)C2)=O)CC1 c1(OC)cc(-n2nc(C3CCCC3)nc2C(C)C(C)C2CCC2)cc(F)c1F C1(C(=O)NCC(C(C)O)C)CCOCCN1C(=O)CC(C)(C)O N1(C(C2C(C)C2C)=O)Cc2cccc(CNC(=O)CCc3cnn(C)c3)c2C1 CCCCC(CO)NC(=O)CC(CC)NC(c1sccc1CO)=O CC1OCCOC1C(=O)NCC1(CO)CCN(C(C2C=CCC2)=O)C1 c1(N(CC(C)(C)CNC(C2CC3(CC3)C2)=O)C)c(Br)cncc1[N+](=O)[O-] CCC(C)CCC(=O)N1CC=CC1CNC(=O)CCNC(c1ccccc1Cl)=O C(=O)(CCCCN(C)C(C1CCCC1)=O)N(C(C=C)C1CC1)C C12(C(=O)NCCC(COC)OC)CC(CN(C(=O)CCCC(C)C)C1)C2 N1(C(c2ccn(CC)n2)=O)CCOCC1CC(=O)NCC(C)(O)C1CC1 C1(CC(=O)NC23C(CN(C(C4C5(CC(OCC)C5)C4)=O)C2)C3)CCC(C)(O)CC1 CC(CCN=c1[nH]c(N(C)Cc2cccnc2)nc2ccsc12)C(F)F C1(CNC(CNC(N)=O)=O)CN(C(c2cc(C3CC3)cs2)=O)CC1(F)F C(=O)(CCCCCF)NCC1(CN(C(c2ccc(OCC)nc2)=O)C)CC1 c1(CCCC)ccc(C(=O)N(C2CC(NC(c3c(C)csc3Cl)=O)C2)C)c(C)n1 N1(C(C(CSC)C)=O)Cc2nccn2CC(NC(C2(CC3CC3)CCCO2)=O)C1 N1(C(C(SC)SC)=O)C2CCCC1CN(C(c1cc(C#N)c[nH]1)=O)C2 C(C(CC(C)C)NC(C1CCCN1S(C)(=O)=O)=O)NC(C=C(C)C)=O N1(C(CC(C)(C)C)=O)CC2(CNC(c3ccc(Cl)cc3)=O)CC1CO2 C(C(C)(C)C(=O)NCC(C(C)C)NC(=O)C(C)CN1CCOCC1)NC(C)=O c1(C(=O)NCC(C)(C(C)C)NC(c2c(C)oc(CO)c2)=O)ccc2ccsc2c1 C1(C)(CCNC(C(C)(C)OCC)=O)CCN(C(=O)Cc2nocc2C)C1 c1(C(=O)NC2CCCCC2NC(c2cccnc2O)=O)cc2c(nn1)OCCS2 c1(C(N2CC(C)N(C(c3cccc(Cl)c3O)=O)CC2)=O)cc2cnccc2o1 N1(C(c2n(CC)nnc2C)=O)CC2CCC1CN2c1nnc(C(F)F)o1 C(=O)(CC1=CCN(C)CC1)N(C)CC1CCN(C(C(Br)=C(C)C)=O)C1 N1(C(c2cnc(C)s2)=O)CCC(NC(C2(F)CCS(=O)(=O)C2)=O)CC1C c1(C(N(CCCNC(COCCC)=O)C2CC2)=O)cccc2[nH]c(C)cc12 c1(C(=O)NC(CNC(COC(C)=O)=O)C(C)(C)C)cccn(CC(C)(C)C)c1=O c1(C(N2CC(CCNC(c3ccn(S)n3)=O)C2)=O)cc2nn[nH]c2cc1F N(C1CCCc2c1cnn2CCO)CC1N(C(Cc2n(C(C)C)ncc2)=O)CCC1 Cn1[nH]c(=NC(=O)c2cccc3ccc(C4CC4)cc23)cc1Cl CCCC(CNC(=O)C(C)C)C(=O)N1CCCC1C(c1ccccc1)C1CCC1 c1(NC(CCC(=O)OCC)=O)cnc(F)cc1C(=O)Nc1c(C)cccc1Br C(=O)(C1CCc2ccccc21)N1CC(NC(CCc2c(C)noc2Cl)=O)(CO)C1 C1(CNC(c2c(CC)cccn2)=O)C(OC)C(OC)CN1C(=O)C(O)CC(N)=O c1(C(N2CC(CCCCNC(=O)CSC3CC3)C2)=O)cc2ccc(F)cc2o1 N1(C(C(C(C)C)=O)=O)CC(C(N2CC(O)CC2(C)C)=O)CC(F)(F)C1 c1(C(N2CC(CNC(c3coc(CO)c3)=O)OCC2)=O)cn2cccc(F)c2n1 N1(C(C(CC)CC)=O)CCN(C(c2ccc(Cn3cc(Br)cn3)o2)=O)C2CC12 c1(C(=O)NC2C(NC(Cn3c(CCC)nnc3S)=O)C2)[nH]c2ccccc2c1C Cc1ccc(N)c(C(=O)NCC23CC(NC(=O)CCC4CCC4)(C2)C(C)O3)c1F c1(C(N2CCC(OC)(CNC(=O)C=C3CCOCC3)C2)=O)cnc2ncccn12 CN1CCN2CC1CNC(=O)c1c(ccs1)C2=O.C12(NS(C)(=O)=O)CC(O)C1C2 C(C(CC(=O)NC1(C(N)=O)CC=CC1)NC(c1nonc1N)=O)OC C1(NC(CC2CN(C)CC2O)=O)CCCCCN(C(=O)Cc2cncc(F)c2)C1 C(C(=O)N1CC(CCNC(C2CCN(C(=O)N(C)C)CC2)=O)C1)(C(C)(C)C)SC c1(NC(C2N(CCN)CCOC2)=O)ccc(F)c(I)c1 N1(C(c2cnc(OC)s2)=O)CCOC(CNC(=O)CC2CC3CCC2C3)C1 CC(CC(C)(C)C)C(=O)NC1CCCCC1NC(=O)Cc1ncn2c1CCCC2 C1(S(N)(=O)=O)(C(=O)NC(CCNC(c2cc(C)oc2C)=O)C)CCCC1 c1(CC(=O)N(CCN(CC)CC)CC)cc(CSC)no1.C1C(C)C(=O)N1 c1(OC)cccc(C(O)C(=O)NCC2(F)CC(NC(=O)C=C(C)C)C2)c1 C1(NC(=O)Cn2cnc(Br)n2)CCN(C(=O)CCn2cncn2)CC1O c1(C(N(CCCN(C)C(c2cc(C3CC3)cs2)=O)C)=O)cc2n(n1)CCNC2=O c1(C2(CC(N3CC(C)C(NC(c4cccnc4)=O)C3)=O)CC2)cccc(C#N)c1 c1(CCCC(=O)NCCCN(CC(C)O)C)cc(Br)no1 N1(C(c2cc(OC)ns2)=O)CC(C2CCCCN(C(c3csnn3)=O)C2)C1 N1(c2ccnc(SC)n2)CCC(NC(c2[nH]nc([N+](=O)[O-])c2Cl)=O)C(C)(C)C1 Cc1nc(-c2ccc(Cl)s2)sc1C(=O)NC(C1CCCC1)C#N N1(CC(=O)NCC(Cc2ccccc2)NC(c2c(C)non2)=O)CCOCC1=O C=CCCC(C)(c1nnnn1CC1CCOCC1)NC1(c2ccccc2Cl)CC1 Cc1nc(N2CCC(NC(=O)CC3CCCC(C)C3)C2)ncc1Br CC1(C(=O)NC2CC(C(F)C(=O)NCc3ccc(F)c(F)c3)C2)CC2CCC1O2 C1(CCC(=O)CC(C)C)CCC(C(=O)ON2CCC2=O)O1.C(CCCC)(NC)CC c1(NCCC2N(C(c3cnccn3)=O)CCCC2)nc(Cl)nc2[nH]c(O)nc12 c1(C(=O)NCCCC2(NC(c3n[nH]c4c3CCC4)=O)CC2)cccc2c1COCC2 C(CC(C)C)(C(N)=O)NC(CC)C(=O)NCCC(C(C)CC)OC C1(NC(c2cncnc2)=O)CN(C(=O)CC2CCC23CCC3)C2CCCCC12 Cc1cc(C)n2nc(C(=O)NC(C)(C)CNC(c3ncncc3C#N)=O)cc2n1 N(C)(C1CN(C(c2cc(C)n(C)c2)=O)CCc2ccccc21)C(CC=CC=C)=O C1(C(=O)OC)CN(C(=O)NCC(C2CCOC2)O)c2ccccc2O1 c1(C(N2CCC(NC(c3cncc(Cl)c3)=O)(CO)C2)=O)cnc2ccccc2n1 C1(C(N2CC(C(C)NC(=O)C(=O)N=S(C)(C)=O)C2)=O)CCCC1S(C)(=O)=O CC(Cc1cccs1)CN=c1nc(N2CCC3(C=CCO3)CC2)c2cc[nH]c2[nH]1 N1(C(C(CC=C)(C)C)=O)CCC2CN(C(=O)Cc3nn(C)cc3[N+](=O)[O-])CC2C1 N1(C(C(C(=O)OC)OC)=O)CC2CN(C(C34CCC3CC4)=O)CC2C1 Cn1cc([N+](=O)[O-])cc1C(N1CCCC1C1(O)CN(C(C2C=CCCC2)=O)C1)=O N1(C(C(CCSC)OC)=O)CCC(C(=O)N(C)OC)C(C)(C)C1 Cc1ccc(CNC(C23CC2CN(S(=O)(=O)CC#N)C3)=O)c(I)c1 CCCCC(CNC(c1coc(C(N)=O)c1)=O)NC(=O)Cc1cnc(C)s1 c1(C(=O)NCC(C)NC(CCCOC(C)=O)=O)cc(C)cc(O)c1 C1(CNC(c2cc(C)n(C)n2)=O)CN(C(C2CCC3(CCC3)C2)=O)CC1(C)C Cc1cncc(C(N2CCOC(CCNC(=O)Cc3ccc(C)s3)C2)=O)n1 c1(C(=O)NCC2(CF)CCC2)cncc(-n2cccn2)n1 c1(NC(CC(=O)O)CNC(c2cccc(F)c2I)=O)nccn2cnnc12 C(=O)(CCC1=NNC(=O)CC1)N1C(CNC(C2(CO)CCC2)=O)CCC(C)(C)C1 c1(C(=O)NC(C)CN(C)C(c2coc(O)n2)=O)c(F)ccc2c1OCC2 CC(C)(O)CC(=O)NCc1ccnc(N(C(=O)Cc2ccsc2)CC2CC2)c1 N1(C(C2COCC(C)O2)=O)C2CCC1CC(C(N1CCC3(CCCO3)C1)=O)C2 C1(C(=O)NC2CN(C(C3CC(SC)C3)=O)C2)CCCOCC1 N1(C(=O)NC2CC(Cl)(Cl)C2)CC(O)CC1CCn1cc(CO)nn1 C#CCC(C)(C(=O)N1CCC(O)C(CO)C1)NC(C1C=CCC1)=O C=CC1(CC(=O)NCC(C)OC(F)F)CN(C(c2coc(C(F)F)c2)=O)C1 c1(NC(C2CCCC(NCc3ccc(C#N)cc3)C2)=O)c(F)c(F)nc(F)c1F c1(C(=O)NC2N(C(C)=O)CCCC2)cc(Br)c(F)cc1Cl.N12CCC1C2=O c1(C(N2CC(F)CC(C(=O)NCC3(CO)CC3)C2)=O)ccc2c(Cl)ccnc2c1 N1(C(Cc2nc(C)[nH]n2)=O)CC2CC(NC(C3CCCC34CC4)=O)C2C1 c1(N(C(c2cnon2)=O)CC2(O)CCNCC2)ncc2c(Cl)cccc2n1 C(CC(=O)N(C1CCN(C(=O)CC2(O)CCC2)C1)CC)(C(C)C)OCC c1(CC(=O)NC(C)C(C)NC(=O)CCF)cnn(-c2ccccc2)c1 c1(CN2CC3(C(C(N4CC(=O)NC4)=O)C3)C2)cc(Cl)cnc1Cl n1(CC(=O)NCCCN(C(CC(CC)C)=O)CC2CCCC2)nc(C)ccc1=O C1(C(=O)NCc2ccc(NC(C)=O)o2)CC12CCN(C(c1ccc(Cl)cc1Br)=O)C2 C(c1cnc(C)s1)=CC(=O)NCCCCN(C(c1cc(COC)no1)=O)C c1(C(=O)NC(C)CC2CN(C(C3OCCO3)=O)C2)ccnc2ccccc12 c1(SCC)nnc2ccc(-c3ccc(OC)nc3)cn12.C12CN(CCO1)C2=O CCC(C#N)C(=O)NC1(C(=O)NC2C=C(C)CCC2)CCOCC1 N1(C(c2c(C)csc2C)=O)CCN(C(=O)NCC2CCC3CCCC23)CC1C#N c1(C(=O)NC2CCOCC2NC(C2CSCCS2)=O)ccc2nn[nH]c2c1 CC1CN(C(C2CN(S(=O)(=O)C(F)F)C2)=O)CCC1N(C(=O)Cc1nc[nH]n1)C Cn1c(-c2nc(Cc3cccs3)nn2CCC(C)(C)C)cc2ccsc12 Cc1ncc(NC(C2CCC3(CN(C(C4CCC(C(N)=O)O4)=O)C3)O2)=O)c(O)n1 Cc1cc(C(=O)NCC2CCCN2C(c2ccc(I)cc2F)=O)cc(O)c1 C1(C(N2CCCN(C(C(CC)(C)OC)=O)CC2)=O)CC2(C1)C(C(=O)O)C21CCC1 CCCC(O)C(=O)NCC(CC)N(C(=O)CC1(C(F)(F)F)CC1)C N1(C(CN(C2CC2)CC)=O)CC(NC(=O)CCC2(C)CC2(F)F)CCC(O)C1 c1(Cc2nc(=NCC3(C)CCC(NC(=O)OC(C)(C)C)C3)s[nH]2)ccc(Cl)cc1 N1(C(C2=C(C)OCCS2)=O)CCC2(CC1)CC(NC(=O)CC1COC3CC1C3)C2 CC1(C)CCC(C(=O)NC2CC(C)(NC(=O)CCCc3ccc(O)cc3)C2)CC1 N1(C(C(C)SC)=O)CC(O)(C2(CNC(c3ncc(Br)cc3OC)=O)CC2)C1 CC1(C)CCC(C(=O)NC2CC(C)(O)C2)(NC(=O)COC2CCC2)C1 N1(C(C(Cn2ccc(C)n2)C)=O)CCC(C)N(C(=O)Cc2cncn2C)CC1 c1(C(=O)NCC(CC)NC(=O)C(N2CCCCCC2)C)cnc2n1CCCCC2 CC(C)C(C#N)C(=O)NC1CC(C)(C(N2CCCC(CN=[N+]=[N-])C2)=O)C1 Cc1cc(Br)c2ncnc(C(=O)NC(c3sccc3C)C(C)C)c2c1 c1(C(=O)NC2(C)CN(C(C(CC)SC)=O)C2)nc(-c2ccco2)sc1C C1(COC)CC(CNC(=O)C(c2ccc(Cl)cc2)=O)N(C(=O)Cc2cnns2)C1 c1(OC)ccc(C(=O)NC2CCCN(C(C3CC3C(C)C)=O)CC2)cc1O CC1CCN(C(=O)CCOC2CCC2)C(CNC(C2CC3CC(=O)C2O3)=O)C1 Cc1nc(Cl)c(NC(C2CC(F)CN(C(=O)C3CC3)C2)=O)c(Cl)n1 N1(C(C2CCN(CC)C2)=O)CCC(C(N2CCC3(CCCO3)C2)=O)CC1(C)C c1(C(=O)NCC2CCC(NC(C(C)Cn3ccnc3)=O)C2)cc2n(c1)CCOC2 c1(N2CCC(NC(c3ccc4cncn4c3)=O)C(F)C2)ncnc2cccnc12 c1(OC)nsc(OC)c1C(=O)NC(C)CCN(C(=O)Cn1cnnn1)C N1(C(CCSCC)=O)CCC2CCN(C(c3nn(C)c(N)c3CC)=O)CC2C1 C1(CNC(C=CC(=O)N(C)C)=O)Cc2ccccc2CN1C(=O)CC(C)C(F)F C1(Cc2ccccn2)CN(c2nnc(CC3CCSC3)n2CC2CC2)CC(C)O1 C(=O)(C1=CC2(CN(C(C3C=CCS3)=O)C2)OC1)Nc1c(C)nsc1 C(=O)(C(=O)C(F)(F)F)NC1C(NC(C(C2CCC(=O)N2)C)=O)CCCC1 C1(NC(c2nc(OC)c(C)s2)=O)CCN(C(c2cc(C#N)c[nH]2)=O)C(C)C1 c1(C2c3n(nnn3)CCOCCCN2)c(Cl)cnn1C.Cn1cccn1.C1(O)CC1 CC1CN(C(C2(C)CCN2Cc2ncccc2Br)=O)CC(=O)N1 CCCCC(CC(=O)NCC1CCCSC1(C)C)N(C(=O)OC(C)(C)C)C(C)C CC1CN(C(=O)CC(C)N2CCOCC2)CCC12CCN(C(C1CC1F)=O)CC2 C(=O)(CC1CCc2ccccc21)N1C(C)(C)CC(NC(=O)CCCC2CCC2)C1 C#Cc1cnn(CC(=O)NC(CNC(=O)COCC2CCCO2)(CC)CC)c1 C1(n2c(C(CCCC)(C)NCc3cccc(C)c3)nnn2)(CSC)CCC(F)(F)CC1 N1(C(C(COC)C)=O)CCC(C)(C)C(C(=O)NCc2ncccc2C)C1 C1(C)(NC(c2cc(C(C)(C)C)n[nH]2)=O)CCCN(C(c2cnn3c2OCC3)=O)C1 c1(N2CCC(C(C)C#N)CC2)nc(=NCC2CCC3CCC23)[nH]c2c1COCC2 C1(N(C(c2c(-c3cncc(C)c3)nccc2)=O)C)CCCCN(CCO)C1 C(CC)(CCCC(=O)NCC[Si](C)(C)C)NC(C1C(CC)C1)=O CCC(C)CC(=O)N1CCC(C(C)(C)CNC(C2(C)CCCOC2)=O)CC1 C12(C(N3CC4C(CNC(CCC(=O)NCCC)=O)C4C3)=O)CCCN(CC1)C2 N1(C(COCCNC(c2cc(CCC)on2)=O)=O)CCn2nccc21 N1(C(C(C)OCC)=O)CCC(O)(CNC(c2ccnn2CCC2CCC2)=O)C1 c1(C(=O)NCCC2OCCN(C(C(C3CC3)SC)=O)C2)c[nH]c2c(C)cccc12 C1(C(=O)NC2(CCNC(c3cccc(C)c3)=O)CC2)CN2CCN1C(C)C2 N1(C(c2cc(C(=O)OC)on2)=O)CCC2(CCC2)C(CNC(=O)CCC2CC2)C1 c1(C2C(C(N3CC4C(NC(COCC(=O)NC)=O)(C4)C3)=O)C2)ccc(C)cc1C Cn1cc2ccc(NC(C3CN(Cc4csc(Br)n4)CCC3(F)F)=O)cc2n1 CC1(C)CC(NC(c2ncoc2C(C)(C)C)=O)CN(C(=O)C=C2CCCC2)C1 C(N=c1[nH]c(N2CCN(CC(OC)OC)CC2)nc(=N)[nH]1)c1n(C)nc(CC)c1Cl N1(C(C(C(C)O)N(C)C)=O)CC2(C1)SCCC2NC(c1cc2cnccc2o1)=O N1(C(C(CC)C#N)=O)CC(C2CCCN(C(=O)Cc3ccco3)C2)C1 N1(C(CSCC(C)C)=O)CCC(CF)(NC(=O)C(C)Cc2ccccc2F)C1 CCCCC(C(=O)N1CC(C(C)OC)C1)NC(=O)Cc1cccnc1F C1(C)(SCCCOc2c(C)cccc2)Oc2ccccc2O1 C12C=CC(C1)CC(=O)N2.c1(C2(NC(C3CC(C(N)=O)C3)=O)CC2)cc[nH]n1 c1(C(=O)NC2C(C(=O)Nc3ncc(C#N)nc3)CCC2)ccc(I)c(F)c1F c1(C(=O)NCCOCCCNC(=O)CCC2CCCO2)nccc2n[nH]cc12 Cc1sc(C)c(C(=O)NCC2(O)CN(C(=O)CCCC3CCC3)C2)c1C#N N1(Cc2cc(F)c(OC)c(F)c2)CCC2(CC1)CCN(C)C2 c1(C(=O)NC2CCN(C(CCC=C=C)=O)C2)cc(C(=O)OCC)cc(F)c1F C1(C(=O)NCC(CC)NC(c2cn(C)cc2C)=O)CCNC(=O)C1 C(=O)(C1=CSCS1)NC(C)CCNC(c1cc(-c2cnn(C)c2)no1)=O N1(C(C2C(OCC)C2)=O)CC2C(N(C(=O)CCc3ccsc3Cl)C)C2C1 N1(C(c2cn(CC)nn2)=O)CCCC1C1CCCN1C(c1nc(=N)cc[nH]1)=O N1(CC(C2CC2)OCC)CC2CC(O)CC1C2.N12CC(C1)C2=O c1(OC)cc(C(N2CCCC2c2cn(-c3ccccn3)nn2)=O)sn1 C#CC(CC(C)(C)C)NC(=O)C(CCOCCO)NC(c1cccc(CO)c1)=O Cc1cc(C(=O)N(CCC(C)NC(C2CCC(=O)N2C(C)C)=O)C)oc1C N1(C(C(O)(F)F)(F)F)CCN(N2CCOC3(CCSCC3)C2)CC1 Cc1nc(O)sc1C(=O)NC1CCCCC1CNC(c1cc(C(N)=O)c[nH]1)=O CCC(F)(F)CC(=O)NC(C)C(C1CCCCC1)NC(C1CS(=O)(=O)C1)=O C(=O)(C(O)C1=CCCCC1)NCC(C)(CO)NC(C1CC(CC(F)(F)F)C1)=O S(=O)(=O)(c1cccc(C#N)c1)NC(c1c(C)n(CCO)nc1)=O c1(C(N2C(CNC(CS(CC)(=O)=O)=O)CC(F)C2)=O)cc2cccn2cn1 Cc1ccc2c(=NC(C)c3cc[nH]n3)[nH]c(=NCCC3(C)CC3)[nH]c2c1 S(=O)(=O)(c1cccnc1N1CC=CCC1)NC(c1c(C)cccc1)CC(C)C CC12CCC(C(=O)NCC3CN(C(c4csc(-c5ccncc5)n4)=O)C3)(C1)OC2 CC(C)(CCCNC(c1cc(Cl)n[nH]1)=O)C(=O)N1CC(O)CC1C1CC1 N1(C(C(COC(C)=O)C)=O)CCC(C(N2CC(CS(C)=O)C2)=O)CC1 C(C)(C(=O)NCCC1CC1)N(CCC)C(C1(C#N)CC1)=O C1(CN(C)C)(NC(C2CC(CNC(=O)CSCCC#N)C2)=O)CCCCC1 c1(OC)ccc(CO)cc1-c1cc(F)ccc1C(=O)NCCN1CCC(C)CC1 C1(NC(C2CC23CCC3)=O)CCN(C(=O)CCC2CCOCC2)C(C2CC2)C1 c1(Cc2n(C(C=C)C)nc(-c3cccc(OC(C)C)n3)n2)noc2c1CCCC2 c1(N2CCCC(CC=C)C2)nc(N2CCC3(CC2)CC3C#N)nc2c1CSC2 c1(NCC(CCC)C)ncccc1S(=O)(=O)NC(Cc1nccs1)CO c1(-c2cc(C)c(O)cc2)ccc2ccnc(NCc3cn[nH]c3)c2c1 C1(N(C(=O)C=Cc2cn(C)nn2)C)CN(C(c2cncn2C)=O)CC1(C)C CC1C(NC(=O)CC2OCCOC2(C)C)CCCN1C(c1nn(C)cc1Cl)=O CCCCN=C(NN)NCC1CCC2(CC1)CC2.c1(C)ncccn1 C(C(C)(C)CNC(=O)C(c1ccco1)NC(C1CCCC1F)=O)SC N1(C(CCCN(C(C)=O)C)=O)CCOC2CCN(C(C3CCCN(C)C3)=O)CC12 c1(C(N2CCCC(CN(C(=O)Cc3c[nH]ccc3=O)C)C2)=O)cc(O)ncc1Br C(=O)(C1=COCC1)N(C)CC1CCC(NCc2ccsc2C(=O)O)CC1 C1(NC(=O)C=C2CCOCC2)CN(C(=O)C=CC2CCC2)C2CCCCC12 N(C(=NCCC(C)O)N1CCSC(CCN(C)C)C1)CC(=C)C c1(C(N2CCN(C)C(CNC(C3CC4(CCC4)C3)=O)C2)=O)[nH]cc2c1CCCC2 N1(C(C2C(C(C)O)C2)=O)CCC(NC(c2cncc(Cl)c2Cl)=O)C2(CCC2)C1 c1(C(=O)NCC(C(C)C)NC(C2C(C=C)C2)=O)cnc(C)nc1C CCCC(C)(O)C(=O)N1CCC(C2CCCN2C(=O)Cn2cc[n+](C)c2)CC1 c1(CNC(Cc2c(CC)cccc2)=O)ccc(O)nc1C.C123CC(C1)(C2)NC3=O N1(C(C2C(C=C)C2)=O)CCC(C2N(C(=O)CCOC3CCC3)CC2(C)C)CC1 N1(CC(CC)C)CCC2CCC(C1)N2C(c1cncc2[nH]ccc12)=O c1(C(=O)NC2CCN(C(c3cccnn3)=O)C2)ccc(C(F)(F)F)nc1O c1(OC)ccc2sc(C(=O)N(C3CN(C(=O)C(C)=C4CCCC4)C3)C)c(C)c2c1 C(C)(C)(CCC(=O)N1CCCC1C(Cc1ccccc1)NC(=O)C(F)OC)OC c1(C(=O)NCC2(O)CCN(C(C=CCCC)=O)C2)ccc2ccc(Br)cc2n1 C1(NC(CCc2ccc(C(=O)NC(CCC)CCO)[nH]2)=O)CCC(F)(F)CC1 CC(CC(=O)N1CCCC(NC(=O)CCC2OCCO2)C1)CC(F)(F)F CCCCCCC(C(=O)NCC(O)CNC(c1cncc(NC)c1)=O)NC(C)=O c1(C(=O)NC2CC2)cc(C(=O)NCC2CC(C)C2)no1.C(C)(C)(C)NC(=O)O.CS Cc1cc(C(=O)NC23CCC(NC(C45CC(CO4)C5)=O)(CC2)C3)ccc1F C#CC1(C)CCCN(C(=O)CC2(CNC(C3CC34CCOC4)=O)CC2)C1 CCCC(C(=O)N1CCC(C(C)NC(=O)Cc2nocc2C)C1)S(N)(=O)=O c1(C(=O)NCC(CCC=C)O)cc(C#N)cc(C#N)c1 c1(CNC(c2c(CC)cncc2)=O)cccc(NC(C2(COC)CCC2)=O)c1F C(CCN=c1nc2scnc2c(NCCCC(C)O)[nH]1)N1C(C)CCC1 Cc1cncnc1C(N1CCC(CC(=O)NCCCNC(N)=O)C1)=O N1(C(CNC(=O)OC)=O)CCCC2C1CCCN2C(=O)C=Cc1ccc(F)cc1 c1(OC(C(CO)OCC(C)(C)O)=O)cccc2c(C#N)c[nH]c12.C1(=O)CO1 C12(NC(C(CCN(C)C)O)=O)CN(C(c3ccc4c(c3)OCC4)=O)CC(F)(C1)C2 C1(C(=O)NCC(C)(C(C)C)NC(Cc2c(C)cccc2)=O)CC2C(C1)C2(C)C C1(NC(C=C(COC)C)=O)CCOCC1NC(=O)CCN1CCC(C)CC1 C1(C(=O)OC2CC(NC(C(CCCOC)C)=O)CC2OC)Cc2cccnc2C1 N1(C(C(C)NC(=O)NC)=O)CCC(CNC(c2ccnn2C2CC2)=O)C1 c1(NC(C2(C)CCN(C(c3c(Cl)cccc3Cl)=O)C2)=O)c(O)ncnc1O O=C1CC(C(=O)NCC2(O)CC(C(N3CCC(c4cc[nH]n4)C3)=O)C2)C2(CCC2)C1 CCC(CC)C(C(=O)N1CCCC(NC(c2cnoc2C(C)C)=O)C1)OC c1(C(N2C(C3(NC(C(CC)NC(N)=O)=O)CC3)CCC2)=O)c(Cl)nn(C)c1Cl Cc1ccc(C(=O)NC2CN(C(c3cc(-c4ccccn4)c[nH]3)=O)CC2C)nn1 c1(N2CCCC(C)(CC)CC2)cc(Br)ccc1S(=O)(=O)NCC1CCCS1 c1(C(=O)NCC2CN(C(C3C(C(=O)OCC)CC3)=O)C2)cn2ccc(F)cc2n1 C1(C(=O)OC)C(F)(F)C12CC(C(=O)NCC1CCC3COCC3O1)C2 N1(C(=O)Cn2nnnc2C2CC2)CC2CCC(C1)N2C(C1CC(O)C(F)C1)=O C1(NC(CN(C2CCC2)C)=O)CCN(C(c2ccn3cncc3c2)=O)C12CCC2 c1(CC(N2C(CNC(C3(C)ON=C(C)C3)=O)C(C)CC2)=O)c(O)nc(=N)[nH]c1C N1(C(C2N(CC)CCC2)=O)CCOC(C(N2CCC(F)CC2)=O)C1 c1(OC)cc(CN2CC(CNC(c3cncc(Cl)c3C)=O)C2)cc(Br)c1O C1(C(=O)NCCN(C(=O)CN2CCCS2(=O)=O)C(C)C)Cc2ccccc2CO1 CCC(CNC(c1cncc(O)c1)=O)(CC)C(=O)NCC(C)(C)C(C)(C)O C1(CC(=O)N(C2CCN(C(=O)CCCSC)CC2)CC#C)CCCCC1(F)F CC1(CNC(=O)Cn2cnnn2)CCCN1C(c1ccc(C(F)(F)F)s1)=O C1(CNC(c2cccc(CC)n2)=O)CCCN(C(=O)CC2CCCCS2)CC1 C1(C(N2CCC(C(C)NC(C(CC)F)=O)C2)=O)CCc2ccccc2O1 c1(C(C(=O)NCC)N(C2CCCN(C(CC)CC)C2)C)nc2ccccc2nc1C C(=O)(C(CC)C(C)(C)CC)NCC(CCCC)NC(c1ccn2cnnc2c1)=O c1(C(N(C2CCC(NC(=O)C=CC(C)(C)C)C2)C)=O)ccc(P(C)(C)=O)s1 C1(NC(C2CC(=C)CN2C(c2nc[nH]n2)=O)=O)CC(C)OC(C)C1 Cc1ccc(Cl)c(OCC(=O)NC2CC(NC(=O)CC3CCC3C3CC3)C2)c1 c1(C(N(C)CC2COCCN2C(=O)CCCC#N)=O)cn2c(n1)CCCC2 N1(C(C(C)CO)=O)CC23CCCCC2(C1)CN(C(c1cscn1)=O)C3 c1(OC)cc(N)ccc1C(=O)NC1CCCC1NC(c1cc(C)on1)=O c1(C(=O)NCCN(C)C(C23CCC(CC2)CO3)=O)cc([N+](=O)[O-])ccn1 N#Cc1ccc(C(=O)Nc2cccc(N3CC(O)C3)c2)c(OCC(F)F)c1 c1(-n2ccc(C(=O)NCCNC(C34CCCCC3C4)=O)n2)ccccc1F N1(C(C=C(C)C)=O)CCC2C(C(=O)NC(C)C(O)C(F)F)C2C1 N1(C(c2cnn(CC)n2)C(=O)NC2CCC2)CCOc2c(Br)cccc2C1 C1(C(C)C(=O)NC(C)C(F)F)CCN(C(=O)COc2cccc(F)c2)CC1 Cn1c(C(=O)NCC2(C(C)(C)C)CCN(C(c3csc(O)n3)=O)C2)cnc1Cl c1(C(=O)NCn2cc(C(=O)NCC3(F)CCCCC3)nn2)cncc2[nH]ccc12 c1(C(=O)NCC2CCN(C(c3cn(C(C)(C)C)nc3)=O)C2)cc2ccsc2[nH]1 C(CCCCCNC(=O)CCc1nc(N(C)C)no1)NC(CC=C)=O N1(C(C2CC(OC)(OC)C2)=O)CC2CCCC2(C(=O)N(C)CC2CCCO2)C1 CC1C(=O)NC(=O)CN1C(=O)C(CO)NC(c1ccoc1Br)=O C1(C(N2CC(C(=O)NC(C)CCc3cn[nH]c3)C(F)C2)=O)CC(C)(C)CN1C c1(C(=O)NC2CCC(C(=O)NCC(F)(F)F)C2)ccc(I)cc1[N+](=O)[O-] C(CC(C)C)(C(=O)NCC1CN(C(=O)CCCC(C)O)CC1C)NC(=O)OC Cc1cnc2ccccc2c1C(=O)NCC1(O)CC(NC(=O)CNC=O)C1 C1(C(N(CCCOC(C)C)C)=O)CC(C)(C)CN1C(=O)CC1COCCO1 N1(C(Cc2ccc(C)cc2)=O)C2CCCC1CN(C(C1(C)CC1)=O)CC2 C1(C(=O)NCCC2N(C)CCC2)C2CCCC1CN(Cc1cncc(Br)c1)C2 C1(NC(c2c(C)occ2)=O)(CO)CCCN(C(C2CC2C(C)(F)F)=O)C1 c1(C(N(C)C)=O)ncccc1C=O.c1(C(=O)NC(CN)C2CC2)sc(N(C)C)nc1Cl.C(CC)C.C c1(-n2c(C3CC3)nc(C(C3CC3)OC)n2)cccc([N+](=O)[O-])c1.c1(C)ccncc1 n1(CC(=O)NC(CC)CN(C(=O)CC2SC(=N)NC2=O)C)c(C)nc2ccccc12 c1(CC)cnccc1C(=O)NCC(C)(C)CNC(=O)C(C)n1ccnc1 N1(C(CC(=O)OC)=O)CCN(C(C2CCN(S(C)(=O)=O)C2)=O)C(C2CCC2)C1 C1(F)(C(=O)OCC)CN(C(C2CC23CCC3)=O)C1.C1(=O)C(C2(O)CCC2)N1 c1(-n2ccc(C(=O)NC3(C)CCCC3(F)F)n2)cccc(C#N)c1.CC1(C)CO1 Cc1cc(Cl)c(Cl)cc1NC(C1CC2(CC(NC(c3ccccc3I)=O)C2)C1)=O CC(C)C(C(=O)NCCc1cncs1)C(C)NC(c1ccsn1)=O c1(NC23CCC(NC(C=CC)=O)(CC2)C3)ncnc2c1nc(O)n2C N1(C(CN(CCOC)C)=O)CCC2CCC12CNC(=O)CSc1cccs1 C1(CNC(C(C)=C(CC)C)=O)CCCC2CN(C(c3ncc[nH]3)=O)CC12 C=C(Cl)CCC(=O)NCc1cccc(NC(=O)CC2CCCN2CC)c1 c1(C(N2CCCC(CN(c3scnc3Cl)CC)C2)=O)cc[nH]c(=NC)c1N C1(C(N2CC(C(C)(C)O)(C(F)(F)F)C2)=O)CCCN(c2ccc(CO)cc2)C1 C1(O)(CS(N)(=O)=O)CCCN1C(=O)C(N1CCSCC1)=O.c1ccccc1Cl C(C(=O)N(C1(CC(=O)NC(C)(CO)C(C)C)CC1)C(C)C)(C(C)C)OCC N1(C(C2(C)C(C)C2)=O)CCCC1(C)CNC(c1cc(Br)ccn1)=O C1(Nc2ncc(C(=O)OCC)c(C)n2)CC2(CCN(C(=O)C(S)C(C)C)CC2)C1 C(=O)(C1=CC2(CCOC2)C1)NC(N1CCCC1c1c(N)cc(Br)cn1)=O c1(OC)ccc(Br)c(CCC(=O)N(C2CCOC2)C2CNC2)c1 C(=O)(CC(C)(C)CNC(C1CC(C)(C)C1)=O)NC(c1ccno1)C C1(NC(CN2CCN(C)CC2)=O)CN(C(c2ccc(O)nc2)=O)CC1N=[N+]=[N-] Brc1cccc(-c2n[nH]c(CSc3cc(C4CCC4)on3)n2)c1 C1(O)(C(=O)NCC2(C)CCCN(C(CC(=O)NCC)=O)C2)CCCC(C)(C)CC1 C1(C(=O)NCC2(F)CN(C(c3n(CC#C)ccc3)=O)C2)CCCCC1(F)F N1(CCN(C(CCC2C(=O)NCC2)=O)CCO)CCCC(CC2CCC(F)C2)C1 C12(C(=O)NC3CC(NC(c4c(NC)nccc4)=O)CC3O)CCCN(CCC1)C2 Cc1cccc(C(CNC(c2ccc(C)cc2)=O)NC(C2(C)CC2C)=O)c1 C1(NC(CCC=C)=O)COC2(CCN(Cc3cccc4cccnc34)CC2)C1 c1(C(=O)NC2C(C)N(C(c3ccc(=N)[nH]c3Cl)=O)CCC2)ccn2ccccc12 C1(NC(C2(CNC(CCCC3(CC)CCCC3)=O)CCC2)=O)(CO)CCC(C)C1 C(=O)(CC1=CCN(C(=O)CCC2CCC(=O)C2)CC1)N(C1C(C)CCCC1C)C CC1=C(C)CC(C(=O)N(CCCNC(c2cc(O)cnc2Cl)=O)C)CC1 CC(C)C(C)(O)C(=O)N(C1CCN(C(=O)CC(c2ccon2)C2CC2)CC1)CCO n1(CC(=O)NC2CC(NC(C=C(CCC)C)=O)C2)c(C2CC2)nc2ccccc12 C(=O)(N1CC(O)CCO1)C1C(NC(CC2CCCC(C#N)C2)=O)CCOC1 c1(C(N(C)CCNC(C2COC3(CCC3)C2)=O)=O)cnc2c(c1)NC(=O)CS2 N1(C(c2cccc(C)c2F)=O)CCCCCC(NC(c2onc(C)c2C)=O)C1 C12(NC(C(=O)NCCCOC3(C)CCC3)=O)CCC(CO)(CC1)CC2 c1(COC)ccccc1C(N1CCC(N(C)C(C2CCCS2(=O)=O)=O)CC1)=O C1(NC(c2c(C)noc2-c2ccccc2)=O)CC2CCC1N(C(=O)C(C)O)C2 N1(C(c2ccsc2I)=O)CCOCCC1c1ccccc1 c1(C(N2CCC(C(C)NC(=O)CC(C)CF)C2)=O)cc2cccc([N+](=O)[O-])c2[nH]1 N1(Cc2cn(CC3N(C(=O)CNC4CCCCC4)CCC3)nn2)CCCS1(=O)=O CN1CCCC12CCN(C(=O)CN(C1CCC1)C(c1cn3ccccc3n1)=O)C2 c1(C(=O)NC2CCC(NC(=O)Cc3ccccc3Cl)C2)cc(Br)cnc1F C(=O)(CC(C(F)F)NC(C1(CC)CCC1)=O)N1CCC(CCCC)C1 N1(C(C2(N(C)C)CCC2)=O)CC2CC(NC(=O)CCCCC(N)=O)C(C2)C1 N1(C(c2c(N)cccc2F)=O)CCC2C(C1)CN2C(c1cnc(C2CC2)nc1)=O Cc1cc(Br)cc(C(N2CC(F)(F)CC2CCNC(C2CC2CF)=O)=O)c1N c1(C(=O)NCCC2CN(C(C(C(C)C)F)=O)CC2C)nc2c(s1)COCC2 c1(CC)cc(NC(C2CC3CCC2N3C(C2(C3CCCO3)CC2)=O)=O)cc(F)c1 C1(CNC(C(COC)COC)=O)CN(C(c2cc(CO)cs2)=O)C(C)(C)C1 CCC(C)C(C(=O)N1CC=C(C(=O)NCC2=CCCC2)C1)N(C)C S(=O)(=O)(c1ccc(=NCC2CC2(Cl)Cl)[nH]c1)NCc1ccc(N(C)C)c(F)c1 N1(C(C2CC(O)(CNC(c3cc(C)sn3)=O)C2)=O)CCC(C2CCC2)CC1 CCCC(C)(O)CC(=O)N1CCN(Cc2ccc(OC)c(F)c2)CC1C#N C(=O)(CCP(C)(C)=O)NC(CNC(C(c1ccc(Cl)cc1)C)=O)CO C1(NC(c2cc(CC)nn2C)=O)CC12CCN(C(c1occc1C)=O)CC2 c1(C(=O)NC(CC)CNC(c2nn(C)nc2Br)=O)ccc(C#N)nc1O C1(CCC)CN(C(=O)N(C(C)C(=O)OC)C)CC1C(=O)N(CCC)CC CC1CN2CCN1C(C(=O)NCC(C)CNc1ccc([N+](=O)[O-])cc1)C2 C1(C(=O)NC2C(NC(CCNC(N)=O)=O)CCCC2)Cc2cncn2C(=O)N1 C(=O)(CCC(C)(C)C(=O)OC)NC(c1ccc(OC)c(OC(F)F)c1)=O N1(C(CN(C(=O)CN2CCCC2C)CCC)=O)CCN(c2nc(CCC)ns2)CC1 C1CCC(O)C(=O)OCCC2CC2C(=O)N1.c1(CCNCC)nncs1 C1(CNC(c2nc(C3CC3)cs2)=O)COCCN(C(c2cc(O)cc(Cl)c2)=O)C1 C#Cc1ccc(C(=O)NC(C)(C)CCCNC(c2coc(C(F)F)c2)=O)cc1F c1(C(C(=O)NCCC2N(CC(=O)NC3CC3)CCC2)=O)cc(Cl)cc(Cl)c1 N1(c2nccc(OCC)n2)CCC(NC(=O)COC2CC2)C(C)(C)C1 N1(C(CCC(=O)c2cccnc2)=O)CCOC2(C1)CN(C(=O)Cc1csnn1)C2 c1(CC(=O)NCC(C)N(C(c2cc(C)sc2C)=O)C)cccc(S(C)(=O)=O)c1 N1(C(C(CN(C(C)=O)Cc2ccccc2F)(C)C)=O)C2CCC1C(N)C2 C1(NC(CSCCOC)=O)CCN(C(=O)CCc2cccc(OC)c2F)C1(C)C c1(C(=O)NC(C)CCCNC(C2CC(O)C2)=O)ccc(S(C)(=O)=O)c([N+](=O)[O-])c1 C(C(C(=O)NC1CCC(NC(C2CC2CC(C)(C)C)=O)C1)OC)OC c1(C(=O)NCC(c2ccccc2)CNC(=O)CC2CCC2(F)F)ccc(O)nc1Cl CCC(C(=O)N1CCSCC1C(N1CCC(C(N)=O)CC1)=O)C(C)C C#CC(CC1CC1)NC(=O)C(C)NC(C1(C)CCC1)=O N1(c2nccc(C)n2)CCC(NC(c2cc(C(F)(F)F)nn2C(C)C)=O)CC1C C(=O)(C(O)P(C)(C)=O)N(CCN(C(C(CC#C)O)=O)C)C c1(CN(CCCC)C(C2CCN(Cc3cncc(F)c3)CC2)=O)ccc(O)cn1 C1(NC(C=CC(C)C)=O)C2CC1N(C(C1(C(C)C)CC1)=O)C2 C1(C(=O)NCCCN(CCCCNC(C2CC=CCO2)=O)C)CC(F)C(=O)N1 c1(C(N2CCC(CSC)C2)C(=O)NC(CC)C)nnc(-c2ccccc2)s1 c1(CN2C(C(=O)NCC3(C)OCCO3)CCCC2)cccc2nonc12 CCCCC(C)CCC(=O)N1CCC(CNC(=O)CCc2cncc(F)c2)C1 C(=O)(C(CC(C)C)C(C)C)NC(CC(=O)N(CC(CSC)(C)C)C)C(F)F C1(C(=O)NC2C=CCN(C(=O)C(Cl)=CCl)C2)Cc2nccn2C1 Cc1cc(CCCC(=O)N(C(CNC(=O)C2=CCC2)CC(C)C)CC)c(C)s1 C1(NC(CC(CC)(F)F)=O)COC2CN(C(=O)C(C(C)C)NC(C)=O)CC12 C(=O)(CC1=CCCCC1)N1CCC(C=C)(C(=O)NCC(F)(F)COC)C1 c1(OC)ccc(C(=O)NC(C2CCCN2C(C2CCC=CCC2)=O)C)c(OC)c1 C1(NC(C2CCCC(C)(C)C2)=O)CC2CCC(C1)N2C(=O)COCCCF c1(NCCOCCOCC)cc(S(=O)(=O)N2CCC(O)C(C)C2)ccc1C#N O=C1CC(C(=O)NC2CCCCC2C(=O)NC2(c3nccs3)CC2)=NN1 c1(C(C(=O)NCC(CN(C(c2[nH]cc(C)c2)=O)C)O)=O)ccc2c(c1)CCCC2 N1(C(c2cc(C(N)=O)no2)=O)C2CCCC1CN(C(=O)Cc1ccc(Cl)s1)CC2 C=CC1(C(N2CC(OC)C(C)C2)=O)CCN(C(=O)CC(=O)OCC)CC1 C(=O)(C1c2c[nH]nc2CN1C(=O)CC1(OC)CCC1)N1CCCN(CC=C)CC1 Cc1csc(CCC(=O)N(C)CCOCCN(C(=O)CC2CCCC2O)C)n1 Cc1ccc(OCCCOC(C2CC(=O)N(c3ccccc3Cl)C2)=O)cc1 N1(CC(N2C(CNC(C(c3cccc(Cl)c3)OC)=O)CC2)=O)CCCCCC1 C1(C(=O)NCCC2N(C(c3c(C)ocn3)=O)CCCC2)CCn2c(C)cnc2C1 C1(CC(=O)NC(C(=O)N(CCCO)C)C2(C)CC2)NC(=O)NC1=O Cc1cc(C(N2CCC(C(C)NC(=O)CN3CCS(=O)CC3)C2)=O)cc(Cl)n1 C1(C2CCOCC2)(C(N(CCCNC(=O)Cc2cc(Cl)no2)C)=O)CC1(F)F c1(C(=O)NCCC(C)(C)CNC(=O)CCNS(C)(=O)=O)ccc([N+](=O)[O-])o1 C=CCC(C(=O)N1CC(C)(C)C1C1CC1)NC(C1CC(CC)(CC)C1)=O C(CN=C(NCc1ccc(F)cc1)NCC(F)(F)C1CC1)NC(c1ncn(C)c1)=O CCCC(C)(C)CC(=O)N(C(C)CNC(=O)CC(C(C)C)c1ccccc1)CC C1(C(N2C(C(NOC(CC)CC)=O)C=CCC2)=O)CC2CCC(C1)O2 C(=O)(C1=CCCOCC1)N1C(C(=O)NCC2=CCN(C)CC2)CC1 c1(OC)cc(N)ccc1C(=O)NCCCCOC(=N)O.C12(CC1)C(=O)N2 c1(C(=O)NC(CC(=O)NCC(F)CO)CC2CC2)cc(F)ccc1F C=CCC(CNC(C1CCC(O)C1)=O)NC(C1CC(C)(C)C1)=O C(=O)(C#CC(C)(C)O)NC1CC(C(=O)NC(c2ccc(O)nn2)C)CC1O C12(NC(CCCSC)=O)CCC(CC1n1cc(-c3nc(C)cs3)nn1)C2 c1(C(=O)NCCCC(C)NC(c2ccc(CC)[nH]2)=O)c(F)ccc(C)c1Br N1(C(C2CCC(CC)CC2)=O)CCCN(C(=O)C2=COCCC2)CC1 N1(C(C(C=C)O)=O)CC(OC)CC1C(=O)OC(C)(C)C.c12ccc(cc1)CNC2=O Cn1cnc2c1CCCC2C(=O)NCC1(NC(=O)CC2COCCO2)CCC1 Cc1cc(S(N)(=O)=O)oc1C(N1CC2CC1CN2C(c1cnc(O)o1)=O)=O CC(C)(F)CC(=O)NCC1CC1CC(=O)NCCCCCC1CC1 N1(C(=O)OCC)CC(NC(=O)N(N2CCCCC2)C)CC1(C)CC c1(CC)nc(C(=O)NCCC2(CNC(c3cnncc3O)=O)CC2)c(N)s1 N1(C(Cc2cc(C)[nH]n2)=O)CC2(CCN(C(c3cnn(C(C)C)c3F)=O)C2)C1 C1(C(=O)NC(C(=O)NC2(CCCN(CCOCCO)CC)CC2)C)CC(C)(C)C1 C(CC(C)C)(C(C(=O)NC1CC(F)(F)C1)OC)N1CCC(O)(c2cnccn2)CC1 CC1(C)OCCC1CC(=O)NC1CCC(CC(=O)NCC2CC3C=CC2C3)C1 CC(CN1CCOCC1)C(=O)N1CC(OCCNC(C2(CCC#N)COC2)=O)C1 c1(C(=O)O)nn(CC(F)(F)F)cc1NCC1CCCC(N2CC(O)C2)C1 c1(C(=O)NC2CC(NC(c3ncc(OC)cn3)=O)C2)cc2occ(Br)c2[nH]1 CCC(C)C(CC(=O)N1CC(CC)CC(CC)C1)NC(=O)CNC(=O)C1CC1 c1(CC(=O)NCC(C2CCC2)NC(C=CC(=O)OCC)=O)cccc(F)c1Cl Cc1c(C(=O)NC2CCC(CCNC(C3CCCCCC3)=O)C2)noc1C1CC1 C1(CNC(CCn2ncc(C)c2)=O)CCC(C)CN1C(=O)C=Cc1ncc[nH]1 C1(N(C(C(C)n2cncn2)=O)C)CN(C(C2COC2)=O)CCC1C Cc1ccc2c(C(N3CCC(NC(=O)C4=C(Cl)CC4)C(C)C3)=O)coc2c1 N1(C(CNC(CC)=O)=O)CC2CC(C(N3CC4(COC(C)C4)C3)=O)C(C2)C1 Cn1c(I)cc2c(NC(C3CC3NS(=O)(=O)CCCCCl)=O)ncnc12 c1(NC(c2ccc(-c3ccc(O)cc3O)nn2)=O)ncc(F)cc1Br C12(C(=O)NC3(CO)CCN(C(=O)Cc4ccc(Cl)c(F)c4)C3)CCCC1CCC2 N1(c2cc(C)nc(C)n2)CC(NC(c2c[nH]c(=O)cn2)=O)CC2(CC2)C1 CCCCC(CCCC)C(=O)NC1CC2CC(NC(c3cccc(C)c3)=O)C1C2 c1(C(=O)NC2(CC(N)=O)CCN(C(C(C)OCC)=O)C2)csc([N+](=O)[O-])c1 C(=O)(C(O)C(F)(F)C(F)(F)F)NCCC1OCCN(C(c2c(CC)cno2)=O)C1 N1(C(c2cc(C)oc2C)=O)CC=C(CCNC(c2[nH]cc3c2CCCC3)=O)CC1 N1(C(c2cncc(OC)c2)=O)CCN(C(c2cnc(O)cc2C)=O)C2CC12 Cc1c(NC2CCN(C3CCC(N)CC3)CC2)ncnc1N1CCSCC1.OC(F)F C(=O)(C1=CCC2(COC2)OC1)N1CC(NC(C(CC(=C)C)C)=O)C2(CC1)CCC2 C1(C)(CNC(C(C)=C(CC)C)=O)CCC(NC(c2occc2C2CC2)=O)C1 CCC(C(=O)NCCc1cc(C(=O)NCC2(CO)CCOC2)no1)SC C1(NC(C2C(NC(CC3CC(CC)C3)=O)CCO2)=O)CCOCCC1C c1(C(=O)NC2(CNC(COCCOC)=O)CCOC2)cnn(CCO)c1C Cn1c(=N)[nH]c2cc(C(=O)NCC3(NC(=O)C=CBr)CCC3)ccc12 N1(C(CC(C(=C)C)OCC)=O)CC2(CCC2)CC1C(=O)NC12CCC(CC1)C2 C1(CCOCC(=O)NCC2CC2)CCCCC1.C(CCO)N(C1CC1)C(N)=O N=c1nc(CCC(N2CCC(C(=O)NCCS(N)(=O)=O)C2)=O)[nH][nH]1 C(CC(=O)N=c1ccn(-c2nc(C)cs2)[nH]1)(C(F)F)NC(C(CC#C)C1CC1)=O N1(C(C(C2CCCOC2)OC)=O)CCC(N(C(=O)C2=CCOC2)CCO)CC1 CC1C=C(C(=O)N2CCC(N(C(=O)CCCC3CC3)C)CC2)CC1 C#CC1CCCC(NC(=O)CCCCCN(C)C(C2(C#N)CC2(C)C)=O)C1 c1(CC(=O)NCC2C(NC(C(CC)c3cccnc3)=O)CCC2)ccccc1C Cc1ncnc(C(=O)NC(C)C(C)(C)C(=O)NC2CC(CCO)C2)c1C C(=O)(N=c1c(Cl)c[nH]cc1Br)N1CC2CN(c3nc(C)nc4c3ccs4)CC2C1 c1(CC)ccc(C(N2CC(CCNC(=O)C3=COCCO3)(OC)C2)=O)c(C)c1 C#Cc1cc(C(N2CC3(C2)CN(C(C2(C)COC2)=O)C3)=O)cc(N)c1 c1(OC)cc(C(=O)CNC(c2cc(C(F)F)nc(C(F)(F)F)c2)=O)ccc1C Cc1cc(C(N2CCC(NC(=O)Cc3cn[nH]c3)CC2C)=O)ccc1Cl CC(C)CC(C)CC(=O)NC1(C)CCCN(C(C2CCCOCC2)=O)C1 N1(C(C(C)CC2CCCC2)=O)CCC2(CCCCC2NC(=O)C=CC(C)(C)C)C1 C1(CN(C)C(C2CC2F)=O)CN(C(C2CCCN2C=O)=O)CCO1 C(=O)(CC(C)CNC(c1nnnn1CCn1cnnn1)Cc1ccco1)OC N1(C(=O)COCc2ccncc2)CC2CC(C1)N(C(c1cc(Cl)sc1Cl)=O)C2 N1(C(C(C=CC)O)=O)CC(NC(c2ncccc2SCC)=O)C2CC2C1 N1(C(C(c2ccc(O)cc2)C)=O)CCC2CN(c3ncc4[nH]ccc4n3)CCC12 c1(CC(=O)NC2C=CCN(C(=O)Cc3cnccc3Cl)C2)ccc(F)cc1F c1(CC(=O)NC2CC(CNC(C3C(C)(C(C)C)C3)=O)C2)c(Cl)cccc1Cl CC(C)CC(CNC(C1CCN(C(C2CC(O)C2)=O)CCO1)=O)CO C(c1csc2ccccc12)=CC(=O)NC1CCC(C)N(C(c2cc(Cl)ns2)=O)C1 c1(C(C)C)nocc1C(=O)NCC1(F)CC(NC(C23CCCC2C3)=O)C1 C1(C2CN(C(=O)C(O)Cc3ccccn3)C2)(NC(C2CCC(OC)C2)=O)CC1 CCC(C)(C)CC(=O)N1CCC1(C)CC(=O)N(C(CO)C(C)C)C c1(CC(=O)N(C2CCCC(NC(C3CCOC3)=O)C2)C)nc2ncccn2n1 c1(CNC(C2C(C)=CCS2)=O)nnn(C)c1C(=O)NC1CCC2CCC12 C1(COCC#C)CCCN1C(=O)C(CNC(c1ncn(C(C)C)n1)=O)OC C1(C)(CNC(C(=O)NCCOC)=O)CN(C(C2(Cl)CC2(F)F)=O)CCO1 C1(NC(C(C)CF)=O)CCC(C)(C)CC1Nc1cc(O)nc(C2CC2)n1 N1(Cc2n(C)ccc2)CC(NC(c2cnc(-c3ccccc3)s2)=O)C(O)C1 C1(CNC(COCC)=O)CC2COCC2N1C(C1CCCN1c1ncccn1)=O CCC(C#N)C(=O)N1CCC(OCCNC(c2cccc(SC(F)(F)F)c2)=O)C1 C1(CNC(C(C)c2cccs2)=O)CN(C(=O)C2=NOC(C)(C)C2)CCC1(C)C C(=O)(C1CCCn2cnnc21)NCC(CN(C(c1cnc(SC)s1)=O)C)(C)C c1(NC(C(=O)NC(CNC(C=CCC)=O)(C)C2CCC2)=O)ccc(Cl)cc1 C1(C)(NC(C(C)OCC#C)=O)CCCN(C(C2CCOC2)=O)C1 CCCC(C)(O)CC(=O)N1CCCC1CCNC(=O)C(C)=C1CC1 c1(OCC)cc(CC(=O)NC2CC2CNC(c2cnn(CC)c2C)=O)ccn1 N1(C(c2c(C)cns2)=O)CCCN(C(=O)Nc2ccccc2Cl)CC1 N1(C(C2(CCC=C)CN(C(c3sccc3CC)=O)C2)=O)CCC(C)C(O)C1 CCS(=O)(=O)CC(=O)N1CCC(C(=O)NC(C)CC(F)(F)F)C12CC2 C(c1cccs1)=CC(N1CCCC1C1CCN(C(C2(CO)CCCO2)=O)C1)=O c1(C(C(=O)NCCN(C(C(C=CC)O)=O)CCOC)CC)cc(C)ccn1 c1(OC(C)C(C)NC(=O)C(CC2CCC2)NC(=O)OCCO)ccccc1 c1(-c2n(CCN(CC)Cc3ccncc3)ccn2)cccc(-c2cnn(C)c2)c1 C1(C(N(C2CCC2)C(C)N)=O)C(NC(=O)C(F)CC2CCC2)C1(C)C C1(CC=C)(NC(C2CCC3CC23)=O)CCN(C(=O)C=Cc2cnc[nH]2)C1 c1(C(=O)NCCN(C(CC2C(C)C2)=O)C2CC2)cc([N+](=O)[O-])ccc1Br Cc1c(C(=O)N(CCC(=O)NC(C2CCCC2)C)CCCO)cccc1O Cc1cc(CCC(N2C(C(=O)NC3CC(OC(C)C)C3)CC2C)=O)on1 n1(CCCC)nccc1C(=O)NCCC(C)N(C(=O)C=CC(C)CC)C CCCCCC(=O)NC(C1CC(NC(c2cnn(C)c2CC)=O)C1)C c1(CN2CCN(C(=O)NCCCn3ccnc3)CC2)ccc2cc[nH]c2c1 c1(CC(CCCCNC(=O)CC(C)c2ccco2)C)cnccn1.C(=O)(CC1CC1)N C12(CC(=O)OC)CCC(C1)N(C(C)=O)C2.C12(CCCSC1)C(=O)N2 c1(C(=O)NC2CC(O)CN(C(=O)C3=CCCS3)C2)cc2scc(Cl)c2[nH]1 N1(C(CC#N)=O)CCCC2CN(C(c3cnncc3O)=O)CCC12 c1(C(N(C(C)C(=O)NCC2(C(=O)OC)CCC2)CC)=O)cnc[nH]1 c1(C(c2ccccc2Cl)NC(C(C)Sc2ccc(C)cc2)=O)cnc(Cl)c(C)c1 c1(OCC)ccc2cc(C(=O)N(C(C)CNC(C3CCCN3C=O)=O)C)[nH]c2c1 N1(C(C(COC)OC)=O)CCC(NC(C2(CC(C)=O)CC2)=O)C(C)(C)C1 N1(c2nc(-c3c(-c4scc(CCCCCC)c4)scn3)on2)CC2C(C)C2C1 c12cc(ccc1C)C(=O)N2.N1(C(CC)=O)CCN(c2ccccc2OC)CC1=O C1(C#N)(CC(C)C)CCN(C(=O)NCc2cccc(Cl)c2Cl)CC1 C1(NC(CCNC(COCC)=O)=O)CC(O)CN(C(=O)C(C)(C)NS(C)(=O)=O)C1 C(=O)(C(C)(C(C)C)N)NCC1(OCC)CCCC1.C1(C(=O)OC)CCCS1 C1(NC(CC(C2CC2)NC(=O)Cn2ccccc2=O)=O)CCCC(O)C1O c1(C(=O)NC(Cc2cccs2)CC(=O)Nc2cnc[nH]2)cc2ccoc2s1 CCS(=O)CC(=O)NCC(O)CNC(=O)CCc1nnc(S)n1C c1(NCCc2ccc(N)c(F)c2)cc(=NCCCc2n[nH]c(=N)o2)[nH]cn1 CC(CN1CCCC1)N=c1[nH]c2c(c(=NCc3cnsc3)[nH]1)CSC2 c1(C(C)=O)cc(C(N2CCCC2CN(C(=O)CS(=O)(=O)N(C)C)C)=O)cc(C)c1 N1(C(c2ccc(OC)c(OC)c2)=O)CCN(C(=O)CS(C)(=O)=O)C2CS(=O)(=O)CC12 c1(C(N2CC(NC(C(CC)NC(N)=O)=O)C(C)(C)C2)=O)c[nH]c(=N)c2[nH]ccc12 N1(C(CN(C(=O)CC2COC(=O)C2)C)=O)CC2C(C1)C2(F)F CCC1=C(C(=O)N2CCN3CC2=CCC(CC)C3=O)CCCO1.O(C(F)F)CC N1(C(c2cc(CC(C)C)nn2C)=O)CC2CC1CN2C(=O)C(C)n1ccnc1 C(=O)(C1=NOC2COCC12)NC1CCC(NC(C=Cc2c(C)ccs2)=O)C1 c1(C2(C(N3CCC(c4scc(C)n4)CC3)=O)CCCC2)ccc(F)cc1Br CCCC(C(=O)N(C)CC1CCCCN1C(=O)Cc1ccc(OC)cc1)OCC c1(C(=O)NC(c2c(OC)cccc2)c2ccccc2Cl)cc(F)cc(F)c1Br c1(C(=O)NCC=CC)nc(C(F)(F)F)n2ccccc12.C12(C)CCCN1C(=O)C2 CC1(C)NC(=O)N(CC(N2CC3CC2CCN3C(C2CCCSC2)=O)=O)C1=O C1(N(C(COC)=O)C)CCC(NC(C2(n3cccn3)CCC2)=O)C1 c1(CC(=O)N(CC(CC)NC(=O)C(C)O)C)ccn(C(C)C)n1 c1(N(C2CCNCC2)C(C(C)NC(=O)Cc2ccc(Br)cc2)=O)nccc(C#N)n1 C1(O)(CCNC(Cc2cc(C)ns2)=O)CCCN(C(C2CS(=O)(=O)C2)=O)C1 N1(C(=O)NC2CCCC2c2ccccc2Cl)CCSCC1NCc1ccn(C)n1 C1(C(=O)NC(C)(C)CC2(O)CCN(C(=O)CO)CC2)C2CCC3C(C2)CC13 C=CCC(C(=O)N(C(C)CN(C)C(C1CCC([N+](=O)[O-])CC1)=O)C)C(C)C c1(C(N(C2CN(C(C3(Br)CC3)=O)CC2O)C)=O)c(Cl)cccc1Cl N1(C(C(c2n(C)nnc2)=O)=O)CCC2CC2(NC(C23CC(CC4CC4)(C2)C3)=O)CC1 c1(C(=O)N)csc(C)c1.c1(C(CNC(COCC(=O)OCC)=O)NC)ccccc1 C=CC1(C(N2CCOC(C3CC3)C2)=O)CCN(C(C2CC(=C3CC3)C2)=O)C1 c1(C(N(C2CN(C(C3CCNC(=O)C3)=O)C2)C)=O)nc2ncc(CCO)cn2n1 N1(C(C(c2cccc(C)c2)C)=O)CC(NC(c2cnc(Cl)n2C)=O)CC12CCC2 c1(C(=O)NC2(C)CC(NC(=O)CC(F)F)C2)cc2nc[nH]c2cn1 C(=O)(C1CCc2ccccc21)NC(C)(C)CCC(=O)NC1CCN(C(N)=O)C1 CC(CCCC(=O)N1CCC(F)(F)C1)NC(=O)CN1CCC(F)CC1 C(c1ccccc1)=CC(N1CC(CCNC(C(CC)OC)=O)C1)=O CC1(C(N2CC3CC3(NC(c3ncc(C#N)cc3Cl)=O)C2)=O)CC2CCC(C1)S2 CC(C)(C(=O)N1CCCC(CN(C(C2(F)CCOC2)=O)C2CC2)C1)S(C)(=O)=O N1(C(C2(C)CN(C(c3ccc(CC)s3)=O)C2)=O)CC2C(CN(C)C)C2C1 C1(NC(c2n(CCCSC)nnn2)C2CC2)CCC(F)(Cn2nc(C)cc2C)C1 CC(CF)CC(=O)NC1(CNC(c2ccc[nH]2)=O)CCOC1 Cc1c(O)nc2ccccc2c1C(=O)NC1CN(C(=O)CCCCN=[N+]=[N-])C1 c1(C(=O)NC2CCC(CNC(CCCN=[N+]=[N-])=O)CC2)ccn2ccnc2c1 C1(NC(C(F)=C(C)C)=O)CCN(C(=O)C(=O)Nc2ccc(Cl)cc2)CC1O N1(C(Cc2c(C(=O)OC)cccc2)=O)CCCN(C(=O)C=CC=C(Cl)Cl)CC1CO N1(C(CC=C=C)=O)CCN(C(=O)CC2CCN(C(C(C)(C)C)=O)CC2)CC1CF c1(C(N(C)CC2(O)CN(C(C3(CCOC)CCCC3)=O)C2)=O)cc(O)ccc1F C(CC(O)C(F)(F)F)NC(C1(NC(Cn2ncc(CC)c2)=O)CC(F)C1)=O c1(C2C(C3N(C(C(CCC)C)=O)CCCC3)C2)cc(C)c([N+](=O)[O-])cc1[N+](=O)[O-] Cc1ccc(F)c(CC(=O)NC(Cc2ccccc2)CN)c1 c1(C(=O)NC2(CNC(C=CC(C)C)=O)CCOC2)ccc(S(N)(=O)=O)cc1F N1(C(C(C(C)C)F)=O)CCCC(C)(C)C1C(=O)N(C)Cc1ccns1 N1(C(CCCCCOC)=O)CCC(C(=O)NCC(C)(C)C(C)C)=C(F)C1 C1(C)(CCNC(C(C)CO)=O)CCN(C(=O)CCc2ccc(F)nc2)CC1 Cc1c(Br)ccc(CNC2CC2C(N2CCOC3CC23)=O)c1F C1(NC(=O)CCC2CCCC2)CC(NC(=O)C(=C2CCOCC2)F)C(O)C1 c1(CNC(=O)COc2ccon2)cnn2c1CN(C(C1(CC(F)F)CC1)=O)CC2 O=C1NCC2(CC(N=C3NC(N4CCC(F)CC4)=NC4=CC=C(C4=O)N3)C2)C1 N1(CC(F)F)CC2CCC(N(CC(F)(F)F)CC(=O)Nc3ncc(Br)cn3)C2C1 N1(C(c2nccc(CC)c2)=O)CC2CC(NC(c3ccc(F)nc3)=O)CC2C1 N1(C(c2c(OC)ccc(OC)n2)=O)CC2(C1)CN(C(=O)C(C)C1CCC1)CCO2 C(=O)(CC(C)(C)C)NC(C1(O)CN(C(=O)CNC(C2CCCCC2O)=O)C1)C N1(C(c2c(CCC)onc2C)=O)CCN(C(c2cc(Cl)no2)=O)C(COC)C1 C(c1ccccc1C(N1CCC(C2CCCN2C(c2cn(C)nc2Cl)=O)C1)=O)OC N1(C(CCCc2ccc(OC)cc2)=O)CC(NC(c2csc(O)n2)=O)CC1(C)C C1(c2n(CC)nnn2)(Nc2cccc(C(F)F)c2C)CCOCCC1C N1(C(C(CCC)N(C(=O)C=CC(=O)OCC)CC)=O)CCCC2(C1)N=N2 N1(C(CCC(CC)OC)=O)CC2CCCC(C1)N2C(C1CC(CC)=NO1)=O C(=O)(C(C)(Cl)Cl)NCC(C)(C1CC1)NC(CN(c1ccccc1)CCOC)=O c1(C(=O)NC2CCC(CCNC(C3(CC)CCCC3)=O)C2)ncc(N)nc1C O=C1CC(=O)CC(C(N2CCC2CC(=O)NCCOCC(F)(F)F)=O)C1 C1(C(N2CCC(O)(CNC(c3cnc(S)[nH]3)=O)CC2)=O)CC2CC1CC2(F)F O=C(N=c1c(Br)c[nH]cc1Br)C1CCCN1C(c1ccc([N+](=O)[O-])o1)C(=O)NC c1(OC)cc(Cl)ccc1C(N1CCCC(CCNC(c2cnsc2)=O)C1)=O c1(CCC)cc(C(=O)NCC(O)CNC(=O)C(C)C(F)F)c(C)o1 c1(C(=O)NC(C2CCCC2)CNC(C(C)SC(C)C)=O)cccn2c(C)nnc12 C12(NC(CCC#C)=O)CCCN(C(c3ccnc(C)n3)=O)CC1C2 C1(NC(=NCC2C(C)C2)NCc2ccco2)CCc2cnnc(O)c2C1 C(CCN(C)C(C1CCC12CCC2)=O)(C(C)C)NC(Cc1c(C)ncs1)=O N1(C(C2(C)CC(C)OCC2)=O)CCCC2(C1)CN(C(=O)CN1CCCS1(=O)=O)C2 CCCCC(C)(F)C(=O)NCC(C1CN(C(=O)CC2CC(SC)C2)C1)O CC1(C)CCC(NC(=O)C=Cc2cc[nH]n2)C(CNC(C2(C#N)CC2)=O)C1 c1(C(=O)NCC2(F)CN(C(COCC#C)=O)C2)cncc2ncccc12 c1(CNC(C=CCC)=O)cnn2c1CN(CC(c1ccc(OCC)cc1)C)CC2 Cc1cc(F)ccc1CNC(=O)C(N1CCCC(C(C)N)C1)=O N1(C(C(C)OCC=C)=O)CC(CNC(=O)CC2(C)CCC2)C2(CCC2)C1 c1(C(N2CCN(C(C3CC4CCC3C4)=O)CC2)=O)c(F)ccc2nc[nH]c12 O=C(NNc1ncc(F)cc1F)c1nc2ccc(Cl)cc2[nH]1 N1(Cc2cccc(C(=O)OC)c2C)CCn2ncc(OC)c2C1C N1(C(C2N(C)CC(C)(C)C2)=O)CCC2OCCN(C(=O)C#CC3CC3)C2C1 c1(C(c2nnnn2C2(C)CC2)NCCC=C=C)cnc(OC)c(C)c1 c1(C(=O)NC(C)CNC(=O)CC(C)(F)F)cc(S(N)(=O)=O)cc(Cl)c1F N1(C(c2c(C)coc2C(C)C)=O)C(C)CC2CN(C(=O)CNC(N)=O)CC12 C1(C(=O)NC2(C(=O)NC3C(C)(C(F)F)C3)CC(CO)C2)C2CCCC1CC2 C(=O)(C(C(C)O)NC(c1conc1C(C)NC(=O)C(O)CC1CCCC1)=O)OC CN1CC(C)(C)CC1C(=O)NC(CC(=O)NCC(F)CO)C1CC1 CCC(CC)CCC(=O)NC(CNC(=O)CC(C)(C)C#N)C1CC1 C=C(Cl)CC(C(=O)N(C1CC2CC2C1)C)NC(c1ncc(C)cc1F)=O N1(C(c2ccn(C(C)C)n2)=O)CCCCC(C(N2CC3CCC3(C)C2)=O)C1 Cc1ccc(C(=O)NCCCCCNC(c2cc3occc3s2)=O)c2c1CCC2 C1(C(N2C(C(N3CCCCC3)=O)COCC2)=O)COc2ccccc2C1 C#Cc1cncc(NC(=O)C(O)CCCNC(=O)C(C(C)O)N(C)C)c1 CC1CCN(C(c2cnn(C3CCC3)c2)=O)CCN1C(=O)CN1CCC(O)CC1 c1(C(N2CCN(C(c3c(CC)cc(Cl)cc3)=O)C(C)C2)=O)cc(F)c(F)cc1F C12(C(N3CCC(CNC(C(C)OCCOC)=O)C3)=O)CC(CCO1)C2 c1(C(C)C)cccc(CC(=O)NCCOCCCNC(c2ccon2)=O)c1 C1(C(=O)NC2C(NC(c3cc(CC)sn3)=O)CCC2)CCC(CC)CC1 c1(OCC(=O)N(C2CC(NC(c3nccnc3N)=O)C2)C)cc(F)ccc1F C1(CNC(C2C(Cl)(Cl)C23CC3)=O)CN(C(=O)Cc2cnccn2)CC1C(F)(F)F Cc1n[nH]c(C)c1SCC(=O)NCC1(CNC(=O)CCF)CCOC1 C1(S(N)(=O)=O)(C(N2CC3C(NC(C4N(C)CC(O)C4)=O)(C3)C2)=O)CCCC1 c1(C(N2CC3CC(C2)N3C(c2c[nH]c3cnccc23)=O)=O)c[nH]c2ncccc12 CC1CC(C)(C(=O)NCC2(CCNC(c3ccccc3C3CC3)=O)CC2)CCO1 c1(N2CC(CC=C)(NC(=O)CCc3ccccc3F)C2)cc(C(N)=O)nc(Cl)n1 c1(N(CC(=O)NC(C)CC2CN(C(=O)C(C)(C)F)C2)C)nn2cccnc2c1Cl N1(C(CC(C)NC(C2CC2)=O)=O)CCN(C(=O)C(F)(F)c2cccnc2)CC1C S(=O)(=O)(c1c[nH]c(C(=O)NCC2(F)CCCN(C(=O)C(C)SC)C2)c1)NC C#CC(CNC(=O)CC(C)NC(=O)C=CC(C)CC)C(C)C Cc1cc(Cl)ccc1C(=O)N(C1CCCN(C(=O)Cn2cnc(C#N)n2)C1)C c1(OCC(CC2CC(CC(=O)Nc3cccs3)C2)O)ccccc1 c1(NC(=O)NC(C(C)(C)C)C(N)=O)cccc(P(C)(C)=O)c1 N1(C(C)C)CCCC(N=c2ccnc(NC(C)Cc3cnn(C)c3)[nH]2)C1 CC1CN(C(=O)C(O)(C2CC2)C2CC2)CCN1C(c1coc(Cl)n1)=O c1(CC)cc(C)ccc1C(N1CCCC(N(C)C(c2ccn(C)c2CC)=O)C1)=O C1(NC(c2ncc(OCC)nc2)=O)C(C)CN(C(=O)Cc2scnc2C)CC1C Cc1cc2sc(C(=O)NC3CCN(C(=O)Cn4ccnn4)C3(C)C)cc2s1 C1(CC=C)(C(N2CC(CNC(=O)CC(C)C3CC3)(OC)C2)=O)CCOCC1 C1(C(=O)NC(CN(C(CCSCCC)=O)CC)C)CCC(=O)N1CC S(=O)(=O)(c1ccc(NCc2nn(C)cc2Cl)cc1Cl)NC(CCOC)C(C)(C)C N1(C(COC2(C)CCCC2)=O)CCC(C(=O)NC2CCC3CC23)=C(F)C1 N1(C(C(=O)NCC)=O)CC(C)C(NC(c2ccc(C3CC3)cn2)=O)C(C)C1 C1(C(N(C(C(=O)OC)C)C2CC2)=O)CCC(c2ccc(C)cc2)CC1 c1(CC)c[nH]nc1C(=O)NCCCCSC(C)C.C12(CC1(C)C)C(=O)N2 N1(C(C(C(C)C)CN(C)C)=O)CC(NC(=O)CC=C(Cl)Cl)C2CCCC12 c1(C(C)C)cnc(O)c(C(=O)NCC(CO)NC(C2CCC2(C)CF)=O)c1 C1(C(=O)NCCCC(C)NC(CCN(C)CC)=O)CCOC(C)(C)C1 N1(C(c2ncsc2OC)C(=O)NC)CC(O)C(O)C12CCC2 N1(C(CCC2CCC(NC(C3CSCCO3)=O)C2)=O)CC2CC(F)CC2C1 CC1CN(C(c2ccc(Cl)cc2F)=O)CCC1NC(=O)Cc1ccc(O)nc1 N(C1CC2(CCN(C(c3ncc(F)cc3C)=O)C2)O1)C(C=CC(CC)=CC)=O c1(C(=O)NCCC(C)NC(c2coc(C(N)=O)c2)=O)cnn(C)c1S(C)(=O)=O C1(NC(c2cc(-n3cccn3)ccn2)=O)C=CCN(CCNC(=O)C(F)(F)F)C1 c1(SC)cncc(C(=O)NC(C)(CNC(c2ncccc2Cl)=O)C(C)C)c1 C1(F)(CNC(C2N(N=O)CCC2)=O)CC2CCC(C1)N2C(C1CC2(CC2)CO1)=O c1(C(=O)NC(C2CN(C(C3C(C(C)C)C3)=O)C2)C)cc(F)cc2cccnc12 C(=O)(C(O)N1C(=O)CCc2ccccc21)NC(CC=C)CC Cc1ccc(C(N2CCC(NC(C3CCCN(C)C3)=O)C(F)C2)=O)cc1Br C1(CC(=O)NC2CN(C(C(C)(C)N(C)C)=O)CC2F)CC(c2ccccc2)=NO1 C=CCC(F)(F)C(=O)N1CCC(C(=O)NC2CC(O)C2O)(CF)C1 C1(NC(=O)C=CCO)COCCN(C(=O)C(O)Cc2ccc(C(F)(F)F)cc2)C1 CC1=C(C)CC(C(=O)NC2COCC2C(=O)NCC2(C#N)CC2)CC1 CC1CN(C(=O)OC(C)(C)C)CC(C)N(C(N2CCc3ccccc32)=O)C1 c1(NC(C(=O)Nc2ccc(OCCCSC)cc2)=O)ccc(S(C)(=O)=O)o1 C(=O)(CC(O)C(C)(C)C)N(CC(C)NC(c1ccc(OCC)cc1)=O)C CC1CN(C(C2CC(=O)NC2(C)C)=O)CCN1C(c1cc(Br)cs1)=O C1(C2CCCN(C(=O)CC3CC3)C2)(NC(=O)CCc2cc(Cl)sc2Cl)CC1 N1(C(c2cc(C)oc2C)=O)CC(NC(C2C3CCCC23)=O)CC2(CC2)C1 c1(C(=O)OC)ccc(OC)cc1C(=O)NC1CCCCN(CCCN=[N+]=[N-])C1 c1(-c2sc(SCC)c(C)n2)cc(CC(=O)NC23CCCN(CC)C2C3)ccc1O C(=O)(CCCCC(F)F)N1CC(CNC(CCNC(CCS(C)=O)=O)=O)N(C)CC1 CCCCC(F)C(=O)NCC=CC(=O)NCC(CO)C(F)(F)F C(CCC(C)C(=O)N1CCN(C(C2CCS(=O)(=O)N2C)=O)CC1)OC CC1CC=CCC1C(=O)N(C1CCN(C(c2cc(Cl)c[nH]2)=O)CC1)CCN(C)C c1(C(N2CC(NC(c3cc(SC)oc3)=O)C(OC)C2)=O)cnc2n1CCC(C)C2 c1(C2(CNC(=O)NC(c3c(OC)cccc3)C)CC2)ccc(C)cc1C C1(C(N(C)CC2CCN(C(CCC=CC)=O)C2)=O)CC2(CCC2OC)C1 C1(NC(C(CSC)(C)O)=O)(CO)CCCN(c2ccnc(Cl)n2)C1 C(C(O)C(=O)NC(c1cnn(C)c1)C(=O)N(C1CCOC1)C)=CCCC C(=O)(C(C)C(F)(F)C(F)F)N1CCC(N(C(C2(C)CCNC(=O)C2)=O)CC)CC1 C1(C(=O)NCC2(COCCNC(C3C(C(C)C)C3)=O)CC2)Cc2ccccc2C1 c1(C(N(CCCCNC(C(CC)C(C)O)=O)C)=O)ccc2c(c1)NC(=O)CS2 CC1OCCCC1C(=O)NC1(C(=O)NCCOc2ncccn2)CCC1 c1(C(C)C)ncc(Cl)c(C(=O)NC2CC23CC(NC(C2CCOC2C)=O)C3)n1 C1(C(=O)NC(C(C)C)CO)CN(C(C2COCCO2)=O)CC1(C)C N(C1CC2(CCC2)Oc2ccccc21)C(c1n(CC)nnn1)c1ncc(SC)s1 c1(C(N(C2C3CN(C(C(C)C(F)F)=O)CC32)C)=O)cc(F)cc(Cl)c1 Cc1[nH]c(C(N2CCCC(C)CC2)=O)c(C)c1C(=O)NCc1csc(C#N)c1 C#Cc1cnc(N2CC(=C(F)CNC(=O)CCc3ccccc3C(N)=O)C2)nc1 C1(O)(C(=O)NC2CC(N(C(C=CCN(C)CC)=O)C)C2)CCc2ccccc2C1 N1(C(c2c(SC)snn2)=O)CCC12CN(C(C1CCC(C(N)=O)C1)=O)C2 C1(C(=O)NCC(C2CCCCC2)NC(C(CC)F)=O)CCN(CCO)C(=O)C1 C1(c2ccc(NC(C3C(NC(=O)Cc4nn[nH]n4)C3)=O)cc2)CCCCC(=O)N1 C(=O)(C(C)C(C)S(C)(=O)=O)NC1(CC)CCN(C(=O)C#CC(C)(C)C)CC1 C(=O)(CN1C(=O)COc2ccccc21)N(C)CC1(CNC(C2(C)CC2F)=O)CC1 c1(C(N2CCC(=O)CC2C2CC2)=O)ccc(-c2nn[nH]n2)c(Cl)n1 c1(C(=O)NC2CN(C(C3CCC(C)O3)=O)CC2O)ccc2nccnc2n1 N1(C(c2sncc2Br)C(=O)NCCOC)CCc2c(c(C3CCC3)nn2C)C1 N1(C(CC=C)=O)CCC(NC(c2cc(O)n(CC)n2)=O)CC1 c1(CNCC2CCCN(C(Cc3cn(C(C)C)nc3)=O)C2)noc2ccccc12 N12CC3OCC(C3C1)C2=O.Cc1nc(C)c(NC(=O)CCOCC(F)F)s1 c1(C(N2CCC(Cn3cc(C(C(C)(C)C)O)nn3)C2)=O)nsc2ccccc12 Cc1cc2cc(C(=O)NCC3CC(C)(C)CN3C(=O)CCC(F)F)oc2cc1C c1(C(=O)NC(CCC)CNC(C2CC2C(C)C)=O)c(N)cccc1F C1(C(=O)OC)(CC)CN(C(C2(c3ccccc3)CC2)=O)C1.C1(S)CCCC1C c12cnc(Cl)cc1C(=O)N2.c1(NC)cccnc1C(=O)Nc1sccc1C(C)=O c1(CC)onc(C(=O)NCC2CC2C(N2CCOC(CC(N)=O)C2)=O)c1C O(C1CCCc2ccccc21)CC(=O)Cc1cccc(F)c1Br N1(C(COc2cccc(C)c2)=O)CCC(C)C(NC(=O)C=CCCCCO)C1C CC1CC(NC(=O)CCCn2cncn2)CN1C(=O)C=CCF C1(CCNC(c2cc(O)ncn2)=O)CN(C(C2CC2c2ccccn2)=O)CCO1 c1(C(N2C(CC(N3C(C)(CC)CC3)=O)CC(C)(C)C2)=O)cc2n(n1)CCC2 Nc1ncc(C(N2CCN(C(=O)CCCC(F)F)C3CC23)=O)cc1Cl C1(C(N2CCC(CN(C)C)CC2)=O)CNC(=O)CN1C(c1cnc2n1CCC2)=O CC(C(=O)NCCC1(O)CCN(C(C2(c3ccc(F)nc3)CC2)=O)C1)C(F)(F)F C1(OC)(CNC(c2ccc(C)c(Cl)c2)=O)CCN(C(c2c[nH]c(Br)c2)=O)CC1 c1(NC(C2CCC(C)(C)O2)c2nnnn2Cc2c(C)cnn2C)ccc(C)c(Br)c1 C12(C(=O)NCCC3N(C(C(C)O)=O)CCOC3)CC3CC(C(=O)N1)C2C3 C=CC(C)(O)CC(=O)N(C1CCN(C(=O)COCCCC)C1)CCC c1(C(=O)NC(CCCNC(CCN(CCC)C)=O)C)ncnc(C)c1OC C(N=c1[nH]c(Cl)ncc1F)C1C(CNC(c2c(C)nsc2C)=O)CCCC1 CC(CSC(F)(F)F)C(=O)NC1CC(C)(NC(=O)C(Cl)=CCl)C1 CC1(C)CC(CC(N2CCCC(CCO)C2)=O)N(C(c2csc(CO)n2)=O)C1 c1(C(N2CC3C(CNC(=O)CCC4CCCCO4)(C3)C2)=O)cc(O)nc(C(F)F)n1 C1(OCC)CC2(C1)CC2CN(Cc1ccco1)Cc1ccc(C)cn1 N1(C(CCC2(C)N(C(CC(CC)CC)=O)CCC2)=O)CCCN2CCCC2C1 C1(NC(CCc2nc(C)sc2)=O)CCC(N(C(=O)Cc2cccnc2Cl)C)CC1 C1(OC)CCCN(C(C2C3CC2N(C(=O)C(F)F)C3)=O)CC1 Cc1cc(Br)cc2[nH]c(C(N3CC(O)(CN(C(=O)C=C4CCC4)C)C3)=O)cc12 C(c1cccnc1C)=CC(=O)NC1CCN(C(CN(C)CC)=O)C1C1CC1 Cc1ncc(C(=O)NCC2(C)CC(NC(C3(COC(C)C)CC3)=O)C2)s1 CC1(C)CCC1C(=O)NC1COCC1NC(c1nscc1Br)=O N1(C(CCCOC(C)=O)=O)CCCN(C(c2cc3n(n2)CCOC3)=O)C(C)C1 C=CCC(CO)NC(=O)CCC1(C)CN(C(=O)CCSC)C1 c1(C(N2CCC(c3nc(C)on3)C2)C(=O)NCCCF)ccc(Cl)cc1O CN(C[Si](C)(C)C)C(C1CCCC(CC#N)C1)=O.n12cc(nn1)COCCCC2 C(=O)(C1=NOC(c2ccccc2)C1)N1C(C(=O)N(CCc2cc[nH]n2)CCO)CCC1 CC(C)CC(CNC(=O)CCOC1COC1)NC(=O)C(O)c1ccsc1 Cc1oc(C#N)cc1C(=O)NCC1(CNC(=O)CC(C)c2ccco2)CC1 C1(C)(C(=O)NCC2(CNC(c3cn(CCC)nc3)=O)CC2(F)F)CCCC1O C1(NC(c2csc(C)c2C2CC2)=O)COC2C(NC(=O)C(C)(C)N(C)C)COC12 c1(OCC)nc(C(N2CC(C(n3cc(C4(C)CCCO4)nn3)C3CCC3)C2)=O)cs1 CC1CCCCC1OCC(=O)N(C)CC1CN(C(=O)Cc2cnc(C3CC3)[nH]2)C1 c1(C(N2C(C)(COC)CC(NC(=O)CNC3CCC3)C2)=O)ccn2cccc2c1 C1(C(N(CCCNC(C2COC(=O)O2)=O)C(C)C)=O)CC12CCOCC2 N1(C(CCN(C)CC)=O)CCC(C(N2CCCC2C(C)O)=O)C1 C1(NC(C(COC)Oc2cccc(F)c2)=O)CC(C)N(C(=O)C)C1.c1(C=O)cnnn1C C(CC(C(=O)NCC1=CCCC1)NC(=O)C(C)N1CC(C)C1)SC c1(CC(=O)Nc2cc(COC)nn2C)cnc2n1CCCC2C C1(CC(=O)NCCN(C(CCN(C)CC)=O)C2CCCC2)CCCC(OC)C1 C1(C)(C(=O)NC(C2(CO)CC2)C)CCCN(C(c2ccc(=N)[nH]n2)=O)C1 c1(C(N2CCC(N(C(c3ccncn3)=O)CC)C2)=O)cc2nc(C)[nH]c2cc1F N1(C(CC2C(C)CCN(C(CCCOC(C)=O)=O)C2)=O)CC(C)(C)OCC1C C1(NC(=O)COCCCF)CN(C(C2CC3(CCC3=O)C2)=O)CC12CCC2 c1(C(=O)NCC2CN(C(=O)C3=CCCCO3)CC2O)cc(Cl)cc(Cl)c1Cl N1(C(C(C(CC)O)C)=O)CC2CCOC2(CNC(=O)CCc2cc(OC)no2)C1 Cn1nnc(C(=O)NC(C2CCN(C(=O)C(=O)C=Cc3cccs3)C2)(C)C)n1 C1(NC(C(CC)SC)=O)(CNC(=O)CCCCCNC(N)=O)CCCCCC1 c1(C(C(=O)OC)NCCCNC(=O)C(C)(F)C(=O)OC)cc(C)cc(C)c1 N1(C(=O)C(Cl)=CCl)CCOCC(NC(c2cnc(-n3cccn3)cn2)=O)C1 C1(C(=O)NCc2occ(C(=O)NCC3(CO)CCN(C)C3)c2)CCC(O)CN1C C(=O)(C1=CCC(F)(F)CC1)N(C(C)CNC(=O)C(Br)=C(C)C)CC CCC(C)(C)C(C(=O)N1CC2CCN(C(c3sc(C(C)C)nc3C)=O)C2C1)OC c1(CCN(C(=O)OC(C)(C)C)C2CC2)noc(-c2ccccc2)n1 n1(CC(=O)N(C(C)CC2CN(C(=O)C(F)OC(F)(F)F)C2)C2CC2)cnccc1=O CC(C)(CC(=O)NCC1(C)CCCC1NC(=O)C=Cc1cocn1)C(F)F c1(C(N(C(C)(C)CNC(c2ccsc2)=O)C)=O)cc[nH]c(=N)c1 C1(NC(c2sc(C)c(O)n2)=O)C(C)CCN(C(c2ccc(C)n2C)=O)C1C C1(C(C)NC(CCCN(C(C)=O)C)=O)CCN(C(=O)CC2(CO)CCC2)CC1 C(CC(C)(C)C)(C(=O)NC(C1CCCC1)CNC(=O)CCc1ccc(C)s1)OC c1(C(N(C(CCNC(CO)=O)C)C)=O)ccc(=O)n(CCCCCC=C)n1 c1(C(=O)NCC(CC2CCCC2)C(=O)NCCCCCC2CC2)ccc(F)cc1O C1(CCOC)(C(N2CCC(O)C(CO)C2)=O)CCN(C(c2cnccn2)=O)CC1 c1(OC)cnc(C(=O)NCC23CC2CN(C(=O)C2=CCCCC2)C3)c(OC)n1 Cc1ccc2c(CN3CCC(NC(c4ccc(Cl)c(C)c4)=O)C(F)C3)c[nH]c2c1 C12(NC(c3coc4c3CCCC4)=O)CCC(CN(C(=O)C(F)C3CCC3)C1)C2 C1(C(=O)NCCN(CC(C)O)C(=O)Cc2ccco2)CC(N(C)C)C(O)C1 n1(CC=C)c(N(C)Cc2ccc(NC(C)=O)cc2)nnc1C1CCCCO1 C1(C(N2C(CC(=O)OC)CCC2)=O)CN(C)CCN1C(C1CC(=O)CS1)=O C1(CCNC(c2n(CC)ccn2)=O)CSCCN1C(c1cn(C2CCCC2)nn1)=O CC(CC1=CCCCC1)NC(N1CCCCC1c1noc(-c2ccccc2)n1)=O C#CCC(C(=O)NC(c1ccccc1)C(=O)NCc1ccccc1F)C1CC1 c1(C(c2c(C)csc2)NCc2occ3c2CCCC3)c(C)ccc(C)c1C C1(NC(C(C(C)O)(C)C)=O)CCN(C(=O)OC(C)(C)C)CCC1(F)F N1(C(c2ccc(C#C)cn2)=O)CCC2C(C1)CN2C(=O)CN(C)C c1(CN2CC(F)(C(N3C(c4onc(C)n4)CCC3)=O)C2)cc(Br)cc(C#N)c1 N(C(=NCCN1CCCC1C)Nc1ccccc1)Cc1cc(C)no1 Cc1nc(C2C(C(=O)N(C)CC3(NC(C4CC4C#N)=O)CC3)C2(C)C)n[nH]1 N1(C(c2ccc(C(C)O)cc2)=O)CC2(CC(C(N3CCC(C)(C)CC3)=O)CO2)C1 CC(C)(C)C(C(=O)NC1(C)CCN(C(=O)C(N)=O)C1)C1CCC1 C1(CCC)CN(C(C2CC2Cl)=O)CC1C(=O)NCC1([Si](C)(C)C)CC1 c1(C(=O)NC2CN(C(C(CSC)C)=O)CC(O)C2)ccc2nc(O)sc2c1 C1(F)(CNC(C2CC(F)C2)=O)CCN(C(c2ccoc2Br)=O)CC1 C1(NC(CC(C)(F)F)=O)COC2C(NC(=O)CC3(C)CC(F)(F)C3)COC12 Cc1cc(-c2cn(CC3C(CNC(C4CCCO4)=O)C3(F)F)nn2)ccc1F Cc1[nH]nc(C(N2CCC(C(C)C(=O)N(CC(C)O)C3CC3)CC2)=O)c1O c1(C(N(CC(=O)N(C2CC2C)C)CCOC)=O)cn(C2CC2)cn1 C(=O)(CC1=NNC(=O)C1)NCC=C1CCN(C(Cc2c(C)nc(S)s2)=O)CC1 c1(Cn2ncc(C(=O)NC(CC)CNC(=O)CCCF)c2)ccccc1F c1(C(=O)NCC2N(C(CCSCC(C)C)=O)CC2)cccc(Cl)c1C Cc1nn(CC(N2CC3CC3(CNC(=O)C(C)CN(C)C)C2)=O)c(C)c1Br N(C(=NCCc1ccc(Cl)nc1)NCc1ncnn1C(C)C)CC(C)C C1(NC(Cn2nc(C)c(Cl)c2C)=O)C2CC3CN(C(C4CS(=O)(=O)C4)=O)C1C3C2 C(C(C)(C)CC(=O)NC12CCN(C(=O)CN3CCC(O)CC3)CC1C2)OC c1(C(=O)NCC2C(NC(c3c(COC)ncs3)=O)C2)cccc2ccccc12 C1(C(=O)NC23CCN(C(C(C)(C)SC)=O)C2CCC3)CCc2nc(=N)[nH]cc2C1 c1(C(=O)NCC(=O)NCCNC(C2C(C(=O)OC)CC2)=O)ncn(C)n1 C1(C(=O)NC(CC)COC)CCOC1CNC(c1c[nH]cc1C1CC1)=O c1(C(N2CCN(C(C=NOC)=O)C(CS(C)(=O)=O)C2)=O)cnc2[nH]cnc2c1 c1(CNC(CC(=O)NC2(CCCOCC#C)CC2)=O)coc2cc(F)ccc12 C1(C2CCN(c3cc(=O)n(C(C)C)c(O)n3)CC2)(NC(C2CC(=C)C2)=O)CC1 c1(CNC2(c3n(CCC)nnn3)CCC(CC)C2)cc(F)ccc1N1CCCC1 c1(C(=O)NCCN(C(c2ccc(CO)cc2)=O)CC)ccc(C)c(S(N)(=O)=O)c1 c1(SC)ccc2cc(C(=O)NC3CC3NC(C3OCC4CCCC34)=O)[nH]c2c1 c1(C(=O)NCCCN(C(C)C)C(C2CC3CCC3C2)=O)nc(C2CC2)ncc1Br C12(C(=O)NCC3C(C(C)C)C3)C(NC(c3ccc[n+]([O-])c3)=O)C3CC1C2C3 c1ccc([N+](=O)[O-])n1C.CC(C)CC(C)(C)ONC.C123CC(C1)(C2)c1cn3nn1 C1(C)(NC(N(CCCCCCN(C)C)C2CCS(=O)(=O)C2)=O)CCOC(C)C1 c1(CC(=O)NCCC2N(C(C(C3CCCC3)OC)=O)CCC2)ccnc(F)c1 c1(C(=O)NCCC2CC(NC(C3(F)CC3)=O)C2)ccc2c(c1)CC2 N1(C(c2ccc(OC)cn2)=O)CCC(C2(NC(=O)Cn3cccnc3=O)CC2)C1 C1(C(=O)OC(C)(C)C)(CO)CCCN1C(=O)CC(=O)NCCF.CC1C(=O)N1 C1(CNC(c2cc(Cl)ccn2)=O)CC2(CC2)CN1C(c1csc(CO)n1)=O C(C)(CC(=O)N(CCNC(C1(F)CCOC1)=O)C(C)C)SC C(N=c1[nH]c(=NCCOCCCF)c2c(F)cccc2[nH]1)c1c(C)cc(Br)nc1 Cc1cc(C(N2C3CN(Cc4ccc(-c5cccc(F)c5)cc4)CC23)=O)c(C)[nH]1 N1(C(C(=O)N(c2ccnn2C)C)=O)CCCC(C2CCCC(=O)N2)C1 Cn1cc(C(N2CCC(CO)C(NC(=O)CC3(O)CCC3)C2)=O)c(O)nc1=O c1(CNC(C2CCCN(c3ccc(C)nc3)C2)=O)noc2c1CC(C)(C)C2 c1(OC)ccc(CCNC(c2cc(Cl)ccc2C)=O)cc1OCCC#N Cc1sc(=O)n(CCC(N2CC(N(C)C(c3cc(C)ns3)=O)C3(CC3)C2)=O)c1C c1(C(=O)NC(CCN(C(c2cccc(C(C)=O)c2)=O)C)C)ccc(N=[N+]=[N-])cc1 N1(C(CS(N)(=O)=O)=O)Cc2ccccc2C(CCN(C)C(C23CCC2C3)=O)C1 C1(CC(N2C(C(C)NC(C3CC(F)(CO)C3)=O)CCC2)=O)CCC(F)(F)CC1 N1(C(C(C)C(NC)=O)=O)CCC(O)(CCNC(c2cc(C)ns2)=O)C1 C(=O)(C1=NOC(C)C1C)NC1(CNC(C(C(C)C)SCC)=O)CCCC1 c1(CNC(c2cc(C3CC3)[nH]n2)=O)cc(C(=O)NOCc2nc[nH]n2)n[nH]1 N1(C(C=CCOCCOC)=O)CC(NC(c2cc3sccc3[nH]2)=O)CCC1C c1(C(C)CC(=O)NCC(C)(C)CNC(=O)Cc2cncn2C)ccc(F)c(F)c1 CCCC(C)(C)C(=O)N1CCCC(CCNC(=O)CCCOCC)C1 c1(C(N2CCC(N(C)C(c3snc(O)c3Cl)=O)C2)=O)nnn2c1C(=O)NCC2 C(=O)(C1CCC(=O)c2cccn21)NCC1N(C(c2cn(C)nc2)=O)CCCC1 c1(C(C)NC(=O)NCCCC(O)CO)ccc(OCC(F)(F)F)cc1F C1(NC(=O)NCc2ccc(=N)[nH]c2Cl)CC2CCC(C1)N2c1nnc(Cl)cc1N C1(F)(CNC(c2cn(CC=C)nn2)=O)CCCN(C(C2(C)CCCS2(=O)=O)=O)C1 N1(C(c2cc(C)ncn2)=O)CCOCC(NC(c2c(C)nn(C(C)C)c2Cl)=O)C1 C1(NC(=O)C=CCCc2ccccc2)CN(C(=O)CN2CCCNC2=O)C2CC12 N1(C(C(C)=C(CC)C)=O)CCOC(CCCNC(=O)CCc2ccncn2)C1 N1(C(C2CCCN(C(CSCC=C)=O)CC2)=O)CCCN(C)CC1C N1(CC(C(C2CC2)OC)(F)F)Cc2ccc(-c3ccc(CO)cc3)cc2C1 Cc1ccsc1CN(C(=O)C(CO)NC(=O)CN1CC2CC2C1)C c1(C(=O)NCCCCN(C(C2C(=C)C2)=O)C)ccc(F)c(C(F)F)c1 CCCCCC(C)CC(=O)N1CC2(CC(CC(=O)NCCC(C)SC)C2)C1 c1(NC(=O)NCc2cccc(C(F)F)c2)cc2ccccc2c(=O)o1 C1(C)(C(=O)NCC(C)CC2CC2)CC(O)CN1C(c1ccn(CCF)n1)=O c1(C(=O)NC2C(N(CCC(=O)NCc3ccccc3)C)C2)cc2ccccc2o1 c1(OC)ccccc1C(C)C(=O)NCC1CCN(C(=O)C(c2ccnn2C)C)C1 c1(C(=O)NCCCC2CCCCN2C(C2CCCC2CF)=O)cnn2c1CCC2 C1(NC(CCCC=C)=O)CC2(C1)CN(C(=O)C(C)S(N)(=O)=O)C2 c1(C(=O)OCCC(CCC(=O)OC)C)cn2c(n1)CCCC2C C1(CNC(c2cc(C)ns2)=O)CN(C(c2cc3ccsc3s2)=O)C2(CCC2)C1 N(C(=NCc1cc(CC(F)(F)F)nn1C)N1CCC(C2(C)OCCO2)C1)C(CC)C CCCC(C)(O)C(=O)N1CC(NC(c2cc(OC)ns2)=O)C(SC)C1 c1(CNC2CC2(Cl)Cl)c(CSC)oc2ccccc12 N(C(=NCC(Cl)C(F)(F)F)NCc1ccnc(NC2CC2)c1)C(COC)C C1(C)(C(N2C(CN(C(=O)CC3(COC)CC3)CC)CCC2)=O)CCC(F)(F)C1 Cc1ccc2c(C(N3CCC(S(=O)(=O)N4CCCC4)C3)=O)ccnc2c1Cl N1(C(C(C=C=C)C)=O)CCC(C=C)(C(=O)NCC=Cc2ccccc2)CC1 c1(C(C)(C)C)cnc2[nH]cnc(N3CC4C(NC(=O)CN(C)S(N)(=O)=O)C4C3)c1-2 N1(C(=O)C2CC2)CCC(C(N2CC(F)(CNC(=O)CCc3cn[nH]c3)C2)=O)CC1 C1(C)(C(C)=O)CN(C(c2ccc(-n3cc(-c4cncs4)nn3)cc2)=O)C(C)(C)C1 C=CC(C)(CC)C(=O)N(C)CCC1CCN(C(=O)C(c2ccccc2C)C)CC1 N1(C(c2cc(C)nnc2C)=O)CC(NC(=O)Cc2cn[nH]c2)CC12CCOCC2 O=C(C1=CN2CCS(=O)(=O)N=C2C=C1)NCC1CC1NC(=O)C(F)C1CC1 C=CC1(c2cn(CCCOC)nn2)COCCN1CC1(C(C)C)C(C(=O)OC)C1 C1(NC(CN(C(C(C)OCOC)=O)C)=O)CCn2nnnc2C1 N1(C(c2cnn(C3CC3(F)F)c2)C(=O)NC(C)C)CC(C)(C)C1C1CCCO1 N1(CCOC)CCC(N=c2nc3scnc3c(NCCn3c(CO)nnc3)[nH]2)C1 N1(C(c2cccc(CC)n2)=O)CC2CC(NC(c3ncc(Cl)s3)=O)CC1C2 c1(C(=O)NCC=CCNC(=O)Cc2cccnc2)cnc(Cl)c(Cl)c1 C1(C(N(CC)Cc2ccccc2)=O)CC2OCCC2N(C(=O)Cc2n[nH]cc2Cl)C1 c1(C(=O)NC2CC(N(C(CSC)=O)C)C2)cn(CC2CCCO2)nn1 C=Cc1cnn(C)c1C(=O)NCC1CCCCC1NC(=O)CCCC(=O)N(C)C CCC(CC)CCCC(=O)N1CC2OCCN(C(c3nccc(F)c3Cl)=O)C2C1 c1(C(N2CCC(NCC(C)=CC(C)C)C2C(C)(C)C)=O)cc2c(s1)CCSC2 C#Cc1cc(C(N2CC(NC(c3ccnn3C=C)=O)CC2C)=O)cc(Br)c1 C(=O)(CCC(C)(C)C#N)N1CCC(C)C1CNC(=O)C1CC1.c12cc(on1)C2 C1(=O)CC(=O)NCC2CC(C2)CCN1.C(C(C)(C)C)NC(COC(CC)C)=O Cc1ncc2n1CCN(C(=O)C(CNC(=O)CC1CC(=O)NC1=O)CC(C)C)C2 C(CCC(C)(C)C(=O)NCCCSC)NC(c1c(CC)cccc1)=O c1(C(N(CCNC(C2C3CCCC23)=O)CC)=O)cc(OC(F)(F)F)cc(Cl)c1O N1(C(c2c(N(C)C)cccn2)=O)CCN(C(=O)Cc2ccccc2Cl)C(CF)C1 N1(C(c2c(CNC(c3cnn(C4CC4)c3)=O)ccs2)=O)CCOC(CN=[N+]=[N-])C1 C1(c2onc(CC(CCCCC)C)n2)Oc2cc(F)ccc2S(=O)(=O)N1C c1(OC)cccc2sc(NC(N3CCN(C)C4CC34)=O)nc12 Cc1ccn2cnc(C(N3CC4C(CNC(=O)C(C)CC(N)=O)C4C3)=O)c2c1 c12ccccc1-n1nnnc1C2NCC(COC)C(C)C.C1(CSC)CCCS1 C1(N(C)C(C2CC(C#N)C2)=O)CC12CCN(C(c1ccc(F)c(O)c1F)=O)CC2 C1(CC)(CNC(C2CCCC2NC(c2cc(Cl)n(C)n2)=O)=O)CCC(=O)N1 CCCC(CCCNC(=O)CCC(CC)OC)NC(=O)CCC1(C(=O)OC)CCC1 Cc1ccc(C(=O)N(C2(CC(=O)N(C)CC3CC3(F)F)CC2)C)cc1O C(=O)(C(F)CCC(C)(C)C)NC1C(C(N2C3CC(OC)CC2CC3)=O)C1(C)C N1(C(C2CCN(C)C2)=O)CCC2(CCC(CNC(=O)CC(C)(C)C)CC2)CC1 N1(C(C(C)=C2CCC2)=O)CCCC(CC(=O)NCCC2(C)N=N2)CC1 C1(NC(C2(SC)CC2)=O)CCCC(N(C)C(c2ccc(C(C)(C)C)[nH]2)=O)C1 O(NC(=O)C(c1cnn(C)c1)NC(c1cncc(O)c1)=O)CC=C(C)C C(=O)(C#CC1CCOC1)NC(C(=O)NCC1(OC)CCCC1)(C)CO N1(C(C(CC)N(C(=O)CC2(OC)CCC2)C)=O)CCOC(C)(CC)C1 Cc1ccc(F)cc1C(=O)NCCC(C)N(C(=O)Cc1ccn(C(F)F)n1)C c1(C(N2CC(OC)(CNC(c3cc4ccsc4s3)=O)C2)=O)cccn2cnnc12 Cc1nn2cc(C(=O)NC3(C4CCN(C(=O)C(O)C5CC5)C4)CC3)nc2s1 c1(C(N(C2CCC(NC(Cc3cc(C)sc3)=O)C2)C)=O)ccc(F)c2ccsc12 c1(C(=O)NC(C=C)CO)ccc(CNC(=O)C=CC2(C)COC2)cn1 C(=O)(C(CN=[N+]=[N-])NC(=O)Cc1ccns1)NCCC1CCC(C)(C)C1 C1(COC)CCC(C(=O)NC2CC(NC(=O)C(C)c3ccsc3)C2)CC1 N1(C(CC)=O)CCC(F)(C(=O)NCC(C)(CO)OC)CC1 CCCCCC(C)(C)C(=O)NCC1CCCN1S(C)(=O)=O N1(C(C2CN(OC)C(=O)C2)=O)CC2CN(C(c3cc4cccnc4[nH]3)=O)CCC12 c1(CCOC(CCOC(C)C)=O)cccc[n+]1[O-] CC1CN(C(=O)COc2ccc(F)nc2)CCC1C(=O)NC(C1CCCC1)(C)C Cc1cc(Br)cc(C)c1C(=O)NCC1CC(NC(C2CC23CC(O)C3)=O)C1 C(=O)(C(C)(F)C(C)(C)F)N1C(C(=O)NCC2CC(OC)C2)CC(=O)C1 c1(C(C(=O)NC(C)(C)C)N(CC(C)(C)OC)C)ccc(C(C)(C)C)cc1 c1(OC)cc(C(=O)NCC=CCNC(C2CCOC2c2ncc[nH]2)=O)sc1Cl CC#CCC(C(=O)N(CC(O)CO)C)NC(C1CCCS1)=O C(=O)(CCCC(=O)N1CC(CC(C)NC(C2(C)CC2(Cl)Cl)=O)C1)NC(C)C c1(C(=O)NC(CNC(c2ncc(CC)s2)=O)CC)cn2ccncc2n1 c1(C(N2C(CC)CN(C(C3CCC(=O)N3)=O)CC2)=O)cc2cc(C)ccc2o1 c1(CC)cc(C(N2CCOC(CCNC(=O)COc3ccon3)C2)=O)cc(N)c1 c1(C(N2CC(O)(C(C)NC(CC(=O)NCC)=O)C2)=O)c(C(F)(F)F)n[nH]c1C C(C(=O)N1CC(N(C(=O)COc2cc(C)on2)C)C(C)(C)C1)(C(C)(C)C)SC N1(C(C=C(CCC)C(C)C)=O)CC2(CCN2C(c2cnc(C)c(C)c2)=O)C1 c1(C(CNC(CC2N(C)CCOC2)=O)NC(=O)C(O)C2CC2)cc(F)cc(Cl)c1 c1(CC)cc(C(N2CCCC2CN(C(=O)C=C2CCSCC2)C)=O)no1 CCC1c2ccccc2CN1N1CC23CCC2(CC)CC3C1 CC1(C(N2CCCC2CNC(c2ccc(CN3CCCC3)o2)=O)=O)CCCCCC1 c1(C(N(C)CCNC(=O)C2CC2)=O)ccc(I)cn1 C1(CNC(c2c(CC)onc2)=O)CN(C(C2(Cl)CC23CCC3)=O)CCO1 C(=O)(C1=CCCCCC1)N1CC(NC(=O)COc2cncc(Br)c2)C(O)C1 CCC(C(=O)OC)C(=O)N(CC(N1CCCC(C(C)OC)C1)=O)C1CC1 N1(C(C(=O)NC(C)C)=O)CCCC(C(C)Nc2cc(C(C)(C)C)on2)C1 C1(CC(N2CCOC3CC23)C(=O)NC2COC2)CCCCCC1 c1(C(=O)NC)ccc(C(N2CCC(N(C(=O)COCCOC)CCO)C2)=O)cn1 c1(C(N2CCCN(C(Cc3cc(C)on3)=O)C(C)C2)=O)cc2ccc(Cl)cc2s1 C1(NC(=O)CSc2nnnn2C2CC2)CC1C1CCCN(C(=O)CSCCF)C1 c1(C(=O)NC(c2ccc(C(F)(F)F)cc2)(C)C(N)=O)ccc(Cl)c(C(F)(F)F)c1Cl N1(C(c2c(CC)ocn2)=O)CC2CCC2(CC(=O)NC2(C(C)(C)C)CCC2)C1 c1(NC(C2CC2CN)=O)ccc(S(=O)(=O)Nc2ccccc2)cc1.CC Cc1nn2c(c1CNC(c1cnnn1C)=O)CN(C(=O)C(c1cncn1C)O)CC2 c1(C(N2CC(OCCNC(CC(C)OC)=O)C2)=O)c[nH]cc(Cl)c1=O CC1=NOC(=O)C1CC(=O)NC(C1(O)CN(C(c2cncc(F)c2)=O)C1)C N1(C(C2(COC)CCCO2)=O)C(C(=O)NCCC(C)(C)C2CC2)CCC12CC2 Cc1ccc2[nH]nc(C(=O)NC3CN(C(C4CC(C)CO4)=O)CCC3C)c2c1 Cc1noc2nc(C(=O)N(CCC(C)NC(=O)COC(C)C)C)ccc12 CC(C)CS(=O)(=O)NCC1CCCC(NC(C2(F)CCCCC2)=O)C1 n1(C(C)CC2CN(C(=O)C(N)=O)C2)cc(Br)cc1C(=O)NCC1C(C)CC1C C1(CN(C)C(C2(Br)CC2)=O)CCCN(C(c2occc2F)=O)C1 CC(C)CC(CN(C)C)CC(=O)NC1CC(CNC(C2CCC(=O)C2)=O)C1 N1(C(C(C)CSc2ccccc2)=O)CC(=O)NC(=O)C1 c1(C(=O)NCC2(F)CN(C(C(C(C)C)C)=O)C2)cc(C(C)C)ccc1F C1(C(=O)NC2(CC=C)CCN(C(C3CCC(=O)N3)=O)C2)CCC2CCCCN12 CC#CCCCC(=O)N1CC2CC(NC(=O)CC(c3ccccc3C)C)C2C1 c1(OCC)ncccc1CNC(C1CCCN1C(=O)C(C(C)C)SCC)=O C1(C)(CC)C=C(C(=O)NCC2CC(NC(=O)COC3CCC3)CC2O)C1 C(=O)(CS(=O)(=O)C1CC1)NC1C(NC(CCN(c2ccccc2)C(C)=O)=O)C1 Cc1cc(C(N2CCCC2CC(=O)NCCC2CCCCO2)=O)ns1 c1(CN(C(=O)NC(C)(CC(F)(F)F)C(F)F)CCO)cc(O)n2nccc2n1 c1(C(c2n(CC(=C)C)nnn2)NCc2c(Br)cnn2C)cccc2ccncc12 N1(C(C(C(CC)O)(F)F)=O)CCN2CCN(C(=O)Cc3cncc(F)c3)CC2C1 c1(CC(N2CC(C)C(CNC(=O)Cc3ccns3)CC2)=O)ccc2nn[nH]c2c1 CC(C)(O)C(C(=O)N)NC(=O)C(=O)NC1CCNCCC1(F)F c1(CNC(C2(CC)CCOCC2)=O)nc(=NCC(C)COC)s[nH]1 N1(C(C(c2ccccc2)OCC)=O)CCOC(CNC(c2c(Cl)n[nH]c2C)=O)C1 CCC(C)(COC)C(=O)NCCCN(C(=O)Cc1coc(-c2cccs2)n1)C(=O)NC c1(C(N(C2CCCC(NC(C34CC(C3)C(C)O4)=O)C2)C)=O)cnc2c(c1)CCCO2 c1(NC(c2ccc(N3CC(C)OCC3)cc2)=O)cc(Cl)c(Cl)cc1O N#CCC(C(=O)N1CCOCC1CNC(c1cc(C2CC2)on1)=O)c1ccccc1 CCC(O)C(C)C(=O)N(CCCCNC(c1ccc(-c2cccs2)cc1F)=O)C C1(C(N(CCN(C(C2CCC2OC)=O)CC)CC)=O)CCC(N(C)C)CC1 c1(OCC)ccc(Br)c(NC(C2CC2NC(C2CNC(=O)CO2)=O)=O)c1 C12(C(=O)NCCC(C)(C)NC(C=CC(CC)=CC)=O)CCOC1CC(=O)NC2 c1(C(=O)NCC2OCCN(C(C(CC)C#N)=O)C2)cnc(C(F)(F)F)c(F)c1 N1(C(C=Cc2cn(C)nc2)=O)CCCC2C(NC(C3SCCS3)=O)C(C)(C)C12 c1(-c2ccc(CNC(c3n4c(nn3)SC(=C)C4)=O)cc2)ccc(O)c([N+](=O)[O-])c1 N1(C(c2ncoc2C(F)(F)F)=O)CC2(CCCN(C(c3ccnnc3)=O)C2)C1 C(=O)(C1CCCn2ccnc21)N(C)CC1(NC(=O)CCS(C)=O)CC1 Cc1nc2c(N3CCC(C(C)NC(=O)C(F)n4cccn4)CC3)ncnc2s1 CC(C)CC(O)C(C)C(=O)N1CCC=CC1C(=O)NC(C)C(C)n1cccn1 N1(C(c2ccn(COC)n2)=O)CC2CCCC(C1)N2C(C1OCCC1C(C)C)=O c1(C(N(CC)C)=O)ccccc1CN1CC=CC1.C(=O)(C=CCCOCCOC)C1CC1 CCC(O)C(C)C(=O)N1CCCCC(C(=O)NC2(C)CSC2)C1 c1(C(N(C(C(=O)N(CCOC)C)C2CC2)C)=O)csc(C)n1 c1(C(=O)NCc2cccc(NC(c3c(C)n(C)nc3)=O)c2)ncnc2c1CCC2 c1(CC(=O)NC2C(CNC(CCS(C)=O)=O)CC2)ccc(Cl)cc1F CC(C(=O)NCCOC1CN(C(C2CCN(c3ccccc3)C2)=O)C1)S(C)(=O)=O c1(CSC)ccccc1C(=O)NCC(C1CCC1)NC(c1ccn(C2CC2)n1)=O c1(C(=O)NC(C2CC=CCC2)C(=O)NC2C(=O)OCC2CO)cccc(F)c1F N1(C(C2(F)CN(C(C(CC)C(C)C)=O)C2)=O)CC(C)(C)CCC1C c1(C(=O)OC)ccc(C(=O)NCC2CC2CNC(c2cc(C)n(C)n2)=O)cc1F c1(CC(=O)NCCN(C(C2CCN(C)C2)=O)C2CC2)cnc(O)nc1O CC(C)CCC(=O)NCC1CCC(C(N(C)CC2(N3CCCC3)CC2)=O)CC1 C(=O)(C1CCc2cccnc21)NC(C(C)NC(c1cnn2c1CCC2)=O)(C)C c1(OC)cncc(C(N2CCC=CC2C(=O)N(CCCF)CCO)=O)c1 Cc1cc(C(F)F)ncc1C(=O)NC1CCN(C(C2(CO)CCCC2)=O)CC1F CCC(F)(F)CCN=c1[nH]c(COC)nc(=NCC(F)=Cc2ccccc2)[nH]1 C#CC1(O)CC(C(=O)OC2CCCN(CC(F)F)C2)C1 CC1CCCC(C(=O)NC(C)(CNC(=O)CCC(=O)c2cccs2)C2CC2)C1 C1(NC(c2c(OC)n[nH]c2)=O)CCN(C(C2CC(CN(C)C)C2)=O)CC1C n1(CCC(=O)NCC2(O)CC(CNC(CC(C)F)=O)C2)ccc2cccnc12 Cc1cc(C)c(C(=O)N(C)CC2COCCN2C(C2(CN(C)C)CC2)=O)s1 Cc1oc(CN2CCN(C(=O)CC(C)CC(F)(F)F)CC2)cc1S(N)(=O)=O.CC N1(C(c2ccc(C3(C)CC3)s2)=O)CCCN(C(C2COCCOC2)=O)CC1 C=CCC(C)(CC)C(=O)NCCC1(CNC(=O)CC2(C)CCCO2)CC1 CCC(C)C(O)C(C)C(=O)NCC(C)(C)CCC(=O)NC1COCC1N=[N+]=[N-] C(=O)(CC(CC(N)=O)CC(C)C)NCC1N(C(CSCC=C)=O)CC2(CCC2)C1 N1(C(COC(CC)(C)C)=O)CCC(C)C(CNC(C2(CC)CCOCC2)=O)C1 N(C(=NCCc1cc(C(=O)NC(C)C)ccn1)NCCn1cncn1)C(C=C)C.OC N1(C(C(CC#C)(C)NC(c2cnc(Cl)s2)=O)=O)CCCC2(CCC2)C1 C1(CNC(C2CCCC2CNC(C2CCC(C(F)(F)F)O2)=O)=O)CCCCO1 N1(C(c2cnc(C(C)O)s2)=O)CC2C(C(=O)NCC(N3CCOCC3)=O)C2C1 C1(CC)CC(C(=O)NCCCOC2CC23CCOCC3)CCN1C(=O)COC c1(C2CC(=O)C2)nc(-c2ccc(C(F)(F)F)cc2)nn1Cc1cccnc1 N1(C(C=COCC)=O)CCCC1(C)CNC(=O)Cn1cc(F)ccc1=O C(=O)(C1=CCC(C)(C)CC1)NC1C(NC(C(C)CSc2cn[nH]c2)=O)CCCC1 c1(CN2CCCC2)ccc(O)c(C(=O)NC2(C(C)(C)C)CS(=O)(=O)C2)c1 C1(CC(=O)NC2CC(NC(C(C)OCc3cccnc3)=O)C2)C=CS(=O)(=O)C1 C1(C(N2C(Cn3cc(C(C(=O)N(C4CC4)CC)=O)nc3)CCC2)=O)CC2C=CC1O2 N1(C(c2nc(C(C)C)sc2)=O)CCC(OCCNC(=O)C(F)CC2CC2)CC1 CC1CC=C(C(=O)N2CCC(NC(c3cncc(C4CC4)c3)=O)C(C)C2)CC1 N1(C(=O)NC(c2n(C)ccn2)c2ccccc2)CC(O)CC(O)C1 N1(C(C2(OCC)CCOCC2)=O)CC2CN(C(=O)C=Cc3csc(=N)[nH]3)CCC12 N1(C(c2ccc(C)nn2)=O)CC2CN(C(C34CCC(C)(CC3)CO4)=O)CC2C1 c1(C(N(CCN(C(CC(CCC)C)=O)C)C)=O)ccc2c(c1)NCC2 N1(C(CS(=O)(=O)NC)=O)CC2COCCC2(NC(=O)CCCC(C)(F)F)C1 C1(NC(CN2C(C)CCC2)=O)CC2CC1CN2C(c1ccc(C#N)cn1)=O CCCCC(CCCC)NC(C1CN(C(=O)CC(C)F)CC1(C)C)=O N1(C(C(Cc2ccc(Cl)cc2Cl)NC(=O)OC(C)(C)C)=O)CCCC(F)(F)CC1 n1(C(CCCC)C)c(-c2ccc(Cl)cc2)csc1=Nc1ccc(C#N)cc1 N1(C(c2c(COC)noc2)C(=O)NCCC2(C)CC2)CC2CC2C(OC)C1 N1(C(CC(=C)C)=O)CCCC(n2cc(NC(C3(CN(C)C)CC3)=O)nn2)C1 C1(CC)CCN(C(c2scc(N(C(=O)C(F)C3CCCC3)C3CC3)c2)=O)C1C CC1C(NC(=O)CCCCC2CC2)CC2CCC1N2C(c1cc(CF)on1)=O C(=O)(C(CC(F)F)NC(c1cnccn1)C(C)C)OC Cc1cn2ccc(C(=O)NC(C)C(C)NC(C3(C)CC(F)(F)C3)=O)cc2n1 c1(C(N2CCC(C)(CCNC(C3ON=C(CC)C3)=O)C2)=O)cccc2nncn12 C1(N(C)C)(C(N(CCCN(C(C2CCC(C)S2)=O)C(C)C)CC)=O)CCCSC1 C1(NC(CC(CN(C)C)O)=O)CN(C(c2nncn2C)=O)CC2(CC2)C1 c1(NCN)ccc(Cl)c(C(=O)NCC2(NC=O)CC2)c1.c1(C(=O)N)ncnc(O)c1Cl C1(C(=O)NCC(=O)Nc2c(F)cccc2F)CCc2ccccc2C1 c1(CC(=O)NCC(O)CNC(c2cc(F)c[nH]2)=O)ccc2c(c1)OCCCO2 Cc1cc(N(C)Cc2ccc(Br)cc2)nc(NC(C)C(c2ccccc2)O)n1 C1(NC(C(C)C)=O)CCN(C(=O)C(O)CC2CCOCC2)C12CC2 c1(C(N2CC3N(C(C(C(=O)OC)C)=O)CC(C3)C2)=O)cc(Cl)cc2ccncc12 c1(CC(=O)NC2CCC2CNC(c2cccc(=O)o2)=O)cnc2ccccc2c1 c1(C(=O)NCC2C(NC(c3cnc(OCC)nc3)=O)CCCC2)cc(C)n(C)c1C c1(OC)cc(C)nc(N2CCC(C)C(NC(=O)C=Cc3cncc(C)c3)C2)n1 CC1CCCC(CC(N2CC(CNC(=O)CCCCNC(N)=O)CC2C)=O)C1 c1(C(N(C)C2CC2)=O)nn(C)c2c(=O)[nH]ccc12 CC(CCC(C)(C)C)C(=O)N1CC2CC1C2C(=O)NC1CC12CCOCC2 N1(C(c2ccc(N)cc2Cl)=O)CCC2CC2(NC(C2(C(=O)C3CC3)CC2)=O)CC1 C1(NC(C(CC)(C)C)=O)CN(C(C2CCC=CCC2)=O)CCC1C C1(NC(C(C)NC(c2cccs2)=O)=O)CCN(C(=O)C(C)C2CC2)CCC1(F)F Cn1nccc1C(=O)N(CCNC(C1CC2CC2C1)=O)CCOC.c1(C)ccccc1 N1(CC(=O)NCC(C)(CO)NC(C2CC(n3cccn3)C2)=O)CCC(=O)NC1=O N1(CCC=C)CCC2(CN(C(c3cccc(Cl)c3C)=O)CC(C)O2)C1 c1(C(c2n(CC)nnn2)NCCC(C)COC)ccc(F)cc1 N1(C(CCCOC)=O)CCCC1(C)CCC(=O)NCC1(C(C)(F)F)CC1 Cc1cc(=O)ccn1CC(=O)NCC(C)NC(=O)CC1(O)CCOCC1 C1(C(=O)NC(C(=O)N(C2C(C)CCC2)C)Cc2cnc[nH]2)CC12CCCCC2 c1(C(=O)NCC(F)F)ncn2ccccc12.c12ccc(cc1)[nH]2 C1(NC(=O)COCCCF)CC2CC(NC(c3cc([N+](=O)[O-])c[nH]3)=O)CC12 c1(NC(CC)CC(C)CO)nccc(=NC(C)c2snnc2C)[nH]1 N1(C(CNC(C)=O)=O)CCCC(N(CCO)C(c2ncnn2C2CCOCC2)=O)C1 C(=O)(C(C)(C)C(F)F)NC1C(CNC(c2c(C)n(CC(F)F)nc2)=O)CCCC1 Cc1ccc(C(=O)NCCC2CCC(NC(=O)C3=COCCC3)C2)c(C)c1 C1(N(C(C2COCCO2)=O)CC)CCN(C(=O)Cc2cncnc2)CC1 N1(C(c2cc(CC)nn2C)=O)CCOCC(F)(CNC(C2CC2C(C)C)=O)C1 c1(C(=O)OCc2cc(F)cc(F)c2Br)n[nH]c2c1COCC2 c1(CNC2(c3n(CCCOC)nnn3)CN(CO)CC2C)ccc2sccc2c1 c1(OC)ccc(Cl)c(CN2CC3CC(C2)N3C(c2cc(OC)n(C)n2)=O)c1F O=S(=O)(c1ccc(Br)cc1F)NC1CCC(Nc2ncnc3sccc23)C1 c1(C(=O)NCC(CCCC)NC(C2CCC(=C)CC2)=O)cc(F)cc(F)c1O CC1(C)CCCCC(NC(C2(C)CCOC23CC3(F)F)=O)C1 C1(C(N2CC(CO)C2)=O)CC(C(=O)N2CCCC(SC(F)F)C2)=NO1 CC(C)CCCC(C)C(=O)N(CCC(=O)N(CCCCCO)C)CCO C1(NC(c2n(CCC)nc(C)c2)=O)CC2CN(C(C3CC(=C4CC4)C3)=O)CC12 N1(C(C(C=C)(C)C)=O)CC2CCN(C(=O)CC3CCC(C)(C)CO3)C2C1 C1(CCC)CN(C(c2ccnn2C(C)CC)=O)CCN1C(c1sncc1C)=O N1(C(C(C)OCCCCCC)=O)CCC(NC(C2(COC)CCCC2)=O)C(F)C1 c1(NC(C(c2cccc(Br)c2)(C)N)=O)ccc(S(F)(F)(F)(F)F)cc1 C=CCC(CNC(=O)CC1(CSC)CC1)NC(C1CCCN1C(C)C)=O C1(C(=O)NCC2(F)CN(C(C(C)Oc3cccnc3)=O)C2)CCC2(CCC2)OC1 c1(CC(=O)NC2C(C)N(C(=O)C(C)O)CCC2)cc(F)c(F)cc1F c1(C(=O)NCCCN(C(=O)Cc2cnc(C)s2)CC)c(F)ccc2[nH]ccc12 CCC(C)C(C)C(=O)NCc1ccc(C(=O)NCC(C)(C)C2CCC2)o1 N1(C(c2ccnc(C)c2N)=O)CC2CCC1CC2NC(=O)CC1COCC(C)O1 N1(C(C(C)N2CCCC2)=O)CCCCC1c1ncon1.N1CCCC2(CC2)C1 c1(C(=O)NC(C2CCN(C(C(CC)OC)=O)CC2)C)cc(N)cc(O)c1C c1(C(N2CCCN(C(C=CC(CC)=CC)=O)CCC2)=O)cc(O)c(OC)c(C#N)c1 C1(NC(C(C)CNC(C2(CO)CC2)=O)=O)CC(C)(C)OC1(C)C n1(CC)cccc1C(=O)NCCC(C)NC(c1ccncn1)=O N1(C(CNS(CC)(=O)=O)=O)CC(OC)CC(NC(=O)CCCN(C)C(C)C)C1 N1(C(C(Cc2ccccc2)N(C)C)=O)CC2CCCC2(NC(C2CCC2)=O)C1 CC(C)(CC(=O)NC1CN(C(=O)CCn2cc[nH]c(=O)c2=O)C1)C(F)F C1(C(=O)NC2(CC=C)CCCC2)CCCN1NC(=O)c1ccc(SC)s1 C=CCC(CNC(c1cnoc1-c1ccccc1)=O)NC(C1(C)CC1)=O Cc1ccc2[nH]cc(C3CCCCC3)c2c1.C12CCCCCC1N2 C1(CC)CCCC1N=c1[nH]c(N2C3CCC2CC(=O)NC3)nc2ncn(CC)c12 c1(SC)cc(C(N2CC(C(C)NC(c3csc(Cl)c3Cl)=O)C2)=O)c(C)o1 C12(C(=O)NCC(CC)NC(=O)CCc3nc(=N)[nH][nH]3)CC(CC(C)O1)C2 CC1CC(CNC(C2CCN(C(=O)CSC(=N)N)CC2)=O)CCO1 N1(C(C(CCOC)O)=O)CCC(CC(F)F)(CO)CC1 N1(C(CCCCCN(C)C)=O)CCC2(CC1)CC2C(=O)NCC1(C)CCCN(C)C1 C(=O)(C(F)(F)C(O)CCCC)NC(C)CC(C)C(F)F CC1(C)CN(C(=O)CCc2ccoc2)CC1CNC(=O)C=CC(F)(F)F N1(C(C(C)CN(C)C)=O)CCCC2CN(C(C3CCCN3C)=O)CC12 c1(NC(C2CCCN(Cc3cccc(OCC)c3O)C2)=O)c(C)cc(O)cc1O N1(C(C=CCOC)=O)CC(CNC(=O)CCSCC(C)C)OC2(CCC2)C1 CN1C2CCCC1CC(N=c1[nH]c3c(c(=NCCC4SCCS4)[nH]1)SCC3)C2 C(=O)(CC(C(F)(F)F)SC)NCC1(COC)CCCN1C(=O)CN1CCC(C)C1 C(CCNC(=O)CSc1cccs1)(C(C)C)NC(C(CC)C1CCOCC1)=O C1(C(N2CC(C)OCCC2)=O)CC2CCCC2N1C(=O)CCC1(C)CC1 c1(CCC(=O)NC(CC(=O)OCC)Cc2cccc(F)c2)cccc([N+](=O)[O-])c1 c1(CN(C(C2(C(=O)NC3(CC)CC3)CCC2)=O)C)ccc(OC)c(Br)c1 c1(-n2cc(CNC(C3C(C(=O)OC)C3)=O)nn2)cc(F)cc(F)c1 c1(COCCC(=O)O)c(Cl)cc(Cl)cc1Cl.C1(SC)CC(O)C(F)C1 C(CN=c1ccc(-c2ccccc2C#N)c[nH]1)NCc1cc(OC)ncc1 N1(C(c2cc(C)sc2)=O)CCCC2(CCCN2C(C2CCc3nnnn3C2)=O)C1 Cc1ccc(-c2cn(CC3CN(C(c4ccc(C)cc4C)=O)C3)nn2)c(C)c1 C1(CC)C(C(=O)NCC2CCC2C)CCCN1C(=O)CCC1CC1(F)F c1(C(N2CC(CNC(CC(C)OC)=O)C3(C2)CC3)=O)cc2ccccc2o1 Cc1nc(CCC(=O)NC(C2CN(C(C3(C)CC3(F)F)=O)C2)C)oc1C c1(C(C)N(C)C(C2CC2C(=O)N(C)C)=O)ncon1.C1(=O)CN1 Nc1cc(F)cc(Cl)c1C(=O)NC1CCC2CCN(C(=O)CC3CCCCC3)C12 N1(c2nccc(NC)n2)CCC2(CC2C(=O)Nc2cc(OC(F)F)ccc2F)C1 C(=O)(C(C)CC(C)(C)C)N(CCOCCC(=O)NCc1c(C)cn(C)n1)C C1(C(=O)NC2(CC=C)CCCC2)CN(C(=O)CC2CC3C=CC2C3)CCN1C C1(C(=O)NCCCCOC2CC2)CCN(C(C2(C)CNC(=O)C2)=O)CCO1 n1(CC)cc(NC(C2CCC(CNC(c3coc(C)n3)=O)C2)=O)c(C)n1 C1(C)(C(=O)OC)CNC(=O)C1.c12cn(nn1)CC1C=CCN1CCN(C)C2 C(=O)(C(C)Cc1cnco1)NC(c1cn(CC(=O)OC)nn1)(C)C C1(NC(C(C)N(C(C)=O)C)=O)CC(F)CN(C(=O)C(C)(C)c2nccs2)C1 CC(C(=O)N1CCN(C(c2ccc(-n3cncn3)nc2)=O)CC1C)C(C)(F)F CCC(C)CC(C)C(=O)N(C1CCN(C(C2CC23CCCC3)=O)CC1)CC1CC1 Cc1cn2c(n1)C(C)CC(C(=O)NCC(C(C)(C)C)NC(c1ncn(C)n1)=O)C2 Cc1cc2[nH]c(C(N3CC4(C3)CN(C(C3(c5ccccc5)CC3)=O)C4)=O)cc2s1 C=CC(C)(O)CC(=O)NCCC1(O)CCN(C(=O)CC2CC(C(F)F)C2)CC1 c1(CONC(c2cccc(C3CC3)c2)=O)c(Cl)cccc1[N+](=O)[O-] c1(C(N2CCC(O)(CNC(C34CCC(C3)C4)=O)C2)=O)ccc(Cl)cc1Cl C#Cc1c[nH]nc1C(=O)NCC1CC(NC(=O)C(C)CC=C)C1 c1(C(N(CC(=O)N(CCC)CCN(C)C)CC2CC2)=O)cc[nH]c2nccc1-2 C12(C(N3CCC(CNC(C4CCC(=O)NC4)=O)CC3)=O)CSCC1C2(F)F Cn1cc(C(N2CCCC2CN(C(=O)CN2CC3CC3C2)C2CC2)=O)c(O)nc1=O C1(CNC(C(CC)O)=O)(NC(c2ccc(C(N)=O)nc2)=O)CCOCC1 C1(OC)CC(CCNC(c2cccc(F)c2)=O)N(C(=O)C(C)CC2CCC2)C1 N1(C(CC2COCC(C)O2)=O)CCC(C)(NC(c2cc(C(F)F)nn2C)=O)CC1 N1(C(C(CCCC)=O)=O)CCC2CCC(C1)N2C(=O)C(N1CCC(C)C1)=O c1(-c2cn(C(C)COC(C)CCCCSc3nncs3)nn2)c(F)cncc1F C1(C(N(CC(C)N(C(CC2(CC)CC2)=O)C)C)=O)CC2CCCC2C1 N1(C(c2c(C)ccc(F)c2)=O)CCC2CC2(C(N2CC(N3CCCCC3)C2)=O)CC1 N1(C(C(C)N(CCC)C(c2cn3c(n2)CCC3)=O)=O)CCCCCCC1C N1(CCNC(COCCOCC)=O)CCC(C)(NC(=O)Cn2cncn2)CC1 CCCCCCn1nnnc1C(C1CCCCO1)(C)NCC1(CF)CCC1 C(=O)(CCCCC(=O)NCC1CCCN1C(=O)CN(C1CCCC1)C)OC C(=O)(C1(C)Cc2cccc(Br)c21)Nc1cccc(C2CCN(C)CC2)c1 CCC(C)C(O)CC(=O)N(CCC(=O)Nc1cnc2[nH]cnc2c1)CCO C=Cc1cnn(C)c1NC(C1C(C(=O)OCC)C1)=O.c12cccc(c1)NC(=O)C2 C1(NC(C2CC(SC)C2)=O)CCCCN(C(c2ccc(SC)cc2Cl)=O)C1 c1(C(=O)NC(CN(C(c2cccc(O)c2F)=O)CC)C)cnc(O)cc1C C12(NC(c3cccnn3)=O)CCCC1N(C(c1cncc(O)c1)=O)CC2 N1(C(C(C)=C(CC)C)=O)CCN(CC(C)NC(=O)C(C)(C)N2CCCC2)CC1 c1(OC)ccc(CN2CC3C(C2)N3C(c2ccccc2SC)=O)cc1 C(=O)(C1CCc2cccnc21)N1C(CNC(C(CCC)NC(C)=O)=O)CCCC1 C1(NC(C(c2ccc(C(F)(F)F)s2)N(C(C)COC(C)C)CC)=O)CC(F)(F)C1 N1(C(CC(CC)C2CCC2)=O)CC2CN(C(C3(NC(N)=O)CC3)=O)CC(C1)O2 C1(C(N2CC(C)C2C(=O)NCC(=O)N(C)C)=O)CCC(C2CC2)C1 C(=O)(C(O)CCC(C)C)NC1CN(C(C2(OC)CCSC2)=O)CC1F N1(C(c2cnn(C=C)c2N)=O)CC2C=CC1C(C(=O)NCC(F)F)C2 N1(Cc2sc(C)c(-c3ccc(F)cc3)n2)CC(N)CCc2ccccc21 c1(C(=O)NCCN(C(C2CC2(c2ccc(Br)cc2)F)=O)CC)ccc(Cl)cc1Cl O=C(C1CC(O)c2ccccc21)NCC1(F)CN(C(C2CCCC2C(F)F)=O)C1 c1(CCNc2ccnc(C(CC)C)n2)cccc(P(C)(C)=O)c1 c1(C(=O)NC23CC(NC(c4nc(CC)sc4)=O)(C2)C3)ccc2c(c1)OCCCO2 c1(C(N2CC=C(CNC(=O)C(F)C3CCOC3)CC2)=O)c(O)nnc2c1CCC2 N1(C(C2CC2CC(C)C)=O)CC(CNC(CN(CCOC)C)=O)C1 C1(CNC(CCOCC#C)=O)(CNC(=O)COC2CCCOC2)CC1(F)F CCC(CCC(=O)N1CC(C(=O)OC)(Cc2cc[nH]n2)C1)OC c1(OC)ncc(C(N2CCC(N(C)C(c3cn(C)nc3SC)=O)C2)=O)cc1Cl N1(C(C(C2CCCC2)OC)=O)CCCCC1C1CCCN(CCNS(C)(=O)=O)C1 CCC(C)CC(=O)N(C1CC1)CC1COCCC1NC(=O)C(=O)Nc1ccccc1 CCC(C)(C)C(=O)NC1CCCC1NC(c1c(Cl)csc1Cl)=O C(CC(C(=O)N(C)Cc1cccs1)NC(c1ccc(CO)nc1)=O)SC C1(CC=C)(CNC(C2CCSCC2)=O)CCN(C(=O)CSCCC(C)C)C1 C1(NC(C2(C)CCCC2)=O)CC=C(C(=O)N2CCCC2CCN(C)C)C1 c1(COC)ccc(C(=O)NC2(CCCNC(=O)C(n3ccc(C)n3)C)CC2)s1 C(=O)(C1=CNC2=NCCCC2=C1)NC1CCCN(C(c2cc(C)c(F)cc2)=O)C1 C1(CNC(C2(C3N(C(=O)OC(C)(C)C)CCC3)CC2)=O)CCc2nncn2C1 c1(C(N2CCC(C(C(=O)NCc3cccc(F)c3O)F)C2)=O)cc(O)ncc1F C1(C(=O)NCCOC(=N)O)CN(C(C2CCCC2C2CC2)=O)CC1(F)F CC1(C)OC2(C(=O)NC3COC4CN(C(C5(C)C=CCC5)=O)CC34)CCC1CC2 CCC(C)CCCCC(=O)NCCC1CCCN(C(c2cnc(COC)s2)=O)C1 c1(C(=O)NC2C(SC)CN(C(=O)C(C3CC3)C3CC3)C2)nccc2ncccc12 C(CC(C)C)(C(=O)N1CCN(C(c2ccc(F)cc2SC)=O)CC1C(C)C)OC c1(CC(=O)NCC(C)CNC(=O)CC2CSC2)cncn1C C1(NC(=O)CCc2ncc[nH]2)CCCC12CN(C(C13CCCC1CCC3)=O)C2 C1(CNC(C(n2cc(CCC=CCCCCC)nn2)C)=O)CCNC(=O)C1 O=C(N=c1[nH][nH]c2ccc(F)cc12)c1cc(F)c(F)cc1.C(F)(F)C(F)(F)F N1(C(c2sc(C)c(C)c2C)=O)CC=C(C(=O)NCCN2CCOCC2)CC1 N1(C(c2c(C)nccc2Cl)=O)CCCN(C(=O)CCC2OCCO2)C(C)C1 Cc1ncnc(C)c1OCC(=O)NCC(C)(C)NC(c1ccsc1C#N)=O C1(c2cn(C(CC)C)nn2)CCCCN(C(=O)CCOC2CCCOC2)C1 c1(SC)n[nH]c(=NCC(C)(C2CCCCC2)NC(c2ncoc2C(C)C)=O)s1 C12(C(=O)OC)CCCC1(C(=O)NC(C)(CSC1CC1)C1CC1)C2 C1(C(=O)NCC(Cn2cc(-c3cncn3C)nn2)OC)CC(C)N(C)C1 C(=O)(CCC(C)(C)C)NCC1C2CN(C(c3c(CC)nccc3)=O)CC21 N1(C(CC)=O)CCN(CNC(=O)CC(c2cccs2)NC(=O)CNC(=O)OC)CC1 CC(C)C(O)C(C)C(=O)NC1CC2(C1)CC(C(=O)NCc1ccoc1)C2 N1(C(CC)=O)CCC2(CC1)CC2C(=O)Nc1cc(O)ccc1Cl N1(C(CCCN(C(C)=O)C)=O)CCC2(CC2)CC1C(N1CC(CO)C2(CC2)C1)=O C1(C(=O)NC(C2CN(C(C34CCCC3CCC4)=O)C2)C)(OC)CCC(F)(F)CC1 CC(C)(O)C(F)(F)C(=O)N1CC2CC1(C(N1CC(c3cc[nH]n3)C1)=O)C2 C1(C(=O)NCCCCNC(C(COC)NC(C)=O)=O)COc2ccc(F)cc2C1 c1(-c2nnc(N3C(CCC)CCC3)n2CC2CCCS2)cc(F)cc(F)c1 c1(C(=O)NCCCN(CC)Cc2ccccc2Cl)ccc(C)cc1Cl Cc1ccc(C)c(C(=O)NC(C)(C)C=CC(=O)NC2CCN(C)CC2C)n1 Cc1ccccc1C(C)N(C)CC1CCCN1C(=O)CCc1cnc(C)o1 c1(CCC(=O)N2N(CC)C(CC)C(=O)N3CC(O)(C3)C2)ccc(C)cc1.OC C(=O)(C(C)(CC)CCC)N(C1CC(C(N(CCCC)CC)=O)C1)C N1(C(c2ccc(OC)cc2F)=O)CCC2CN(C(=O)C(C)(F)C(C)(C)F)CC2C1 N1(C(=O)Nc2cccc(SCC#C)c2)CCC(C)OC(C)C1 N1(C(CCC)=O)CCCCC1C(=O)NCC(C)N(C(c1c(O)noc1C)=O)CC C1(CNC(C=C(C)C(F)F)=O)CCCC1C(=O)N(C)CC1CCC1 CC1(C)C(NC(c2nsnc2O)=O)CC1CC(=O)NC1(CO)CCCCC1 CC1(O)CC2CCC1N2c1cccc(S(=O)(=O)N2CCc3noc(N)c3C2)n1 C#CCC(CC(=O)NCC12CCC(CC1)C2)NC(c1c[nH]nc1[N+](=O)[O-])=O C1(C(=O)NN2CCC(CNC(c3cc(C)n(C)n3)=O)C2)(CO)CC2(CC2)C1.CC O=S(=O)(c1ccc(NCC2CSCCO2)c(F)c1)NCC1CC2(C1)CC(O)C2 c1(C(=O)NC(CNC(CCC=CCC=C)=O)CC(C)C)cc(C)ccc1O N1(C(CCCC#C)=O)CC2CN(C(c3ccnc(OC)n3)=O)CCC2(CO)C1 C1(C(=O)NCC2N(C(CC(CC)CC)=O)CC3(CC3)C2)CCc2nnn(C)c2C1 N1(C(C(COCC)NC(=O)CC(C)(O)COC)=O)CCC12CCCSC2 N1(C(CC2(CS(N)(=O)=O)CC2)=O)CCC(F)(C(=O)NCCCF)CC1 C1(C(N2CC(C3CCCO3)C2)=O)(NC(C2(CF)CC(O)C2)=O)CCCC1 n1(CC(=O)NC2C3CN(C(C(CCC(C)C)O)=O)C2C3)nc2ccccn2c1=O C1(NC(=O)C(N2CCCC2c2ccon2)=O)CCCC1(F)F c1(C(N(CCN(C(c2ccc(Cl)s2)=O)CC)CC)=O)cnc(O)c(OC)c1 C1(NC(CN(C(COCCC(C)C)=O)CCO)=O)CCN(C)C1(C)C c1(-c2ccc(CC(=O)NC)cc2)n[nH]c2c1CN(C(c1c[nH]c(=O)cn1)=O)C2 Cc1cnc(CC)cn1.n1(CCn2cncn2)cc(CN)nn1 Cc1nc(CNC(=O)C(C)N(C(=O)C(CO)N2CCCC2)C)c(C)s1 CC1CC(NC(=O)CCC(N)=O)CN1C(=O)CCCc1ccsc1 c1(NC(C2(C)CCN2C(C2CC2c2ccccc2)=O)=O)cnn2ccccc12 CC(C)C(O)C(=O)NCC(C)CN(C(=O)CC1CC=CCN1C)C N1(C(C(C(C)C)NC(C)=O)=O)CCC2(CC2NC(C2CC2C2CC2)=O)C1 C1(NC(C=C(CCC)C)=O)CCS(=O)(=O)C12CN(C(c1c[nH]nc1F)=O)C2 c1(C(C)C)ccc(C(N2CC(CC(C)NC(=O)CC3OCCC3C)C2)=O)c(F)c1 CC1CCC=C1C(=O)N1CCCCC1C(=O)NCCCS(N)(=O)=O C1(CNC(C=CCOC)=O)CC(OC)CN1C(c1cncc(N)c1)=O CC(Cc1ccccc1)C(C)(O)OCCN(CC1CCCO1)Cc1cc[nH]n1 C(=O)(C1CCc2cccc(=O)n21)NC(c1ccc(OC(CC)(C)C)cc1)=O N1(C(C(C=C)(C)C)=O)CCC2CN(C(c3n[nH]cc3-c3ccccc3)=O)CC2C1 N1(C(CCN(CC)CC)=O)CC(CC(=O)NCc2ncccn2)CC1C c1(C(C)=O)cccc(CNCC2CCN(C(C3CC4(CC4)C3)=O)C2)c1 c1(C(=O)NC2CN(C(c3ccc(C#C)cc3)=O)CC(C)C2)cc(F)cc(F)c1O C(C(=O)N=c1ccn(CCO)[nH]1)(N(C(=O)C=Cc1cncs1)C)C1CC1 S(=O)(=O)(c1ccccc1-c1cncnc1)N1CC(C(=O)OC)C2(C1)CCC2 C1(C(=O)OC(c2cc(-c3ccccc3)co2)C)CC(F)(CN(C)C)C1 C=CC(C)(O)CC(=O)NCC1(C)CCN(C(c2ccncc2NC)=O)CC1 N1(C(c2ccccn2)=O)CCC2OCCCN(C(c3cscc3C(F)F)=O)C2C1 C(=O)(CCCC(=O)NC1CC(F)(CNC(c2csnc2OC)=O)C1)NCCC CC1(C)OC2CN(C(=O)C(N3CC(CO)OC(C4CC4)C3)=O)CC2O1 C(=O)(C(C)(C)CCF)N1C(C)CC(CC(=O)N(C)Cc2c(C)n(C)nc2)C1 C1(C(=O)NC(CNC(CC=C)=O)CC)CC(F)CN1C C1(CNC(CCC(C)O)=O)CN(C(=O)Cc2ccc(O)nc2)CC1(C)C c1(CNC(Cn2cc(C(=O)OC)nn2)=O)c(-n2cccn2)cccc1F c1(CC)onc(C)c1C(N1CCC(OCCNC(=O)CC2CSCCS2)CC1)=O Cc1cc(C(N2CCCC(CN(C(=O)CC3CCOC3)C)C2)=O)nc(C)n1 CC1(F)CN(C(=O)C=CC2CCOCC2)CCN(C(c2cccc(Br)c2)=O)C1 C1(C)(CC)C=C(C(=O)N(C2CN(C(c3cnn4cc[nH]c34)=O)C2)C)C1 CCC(CC(C)C)C(=O)NC1CCN(CCCNC(c2csc(C)c2C)=O)C1 c1(OC)ccc2c(=NCC3CCSC3)[nH]c(=NCC3CC4CC3CC4O)[nH]c2c1 CN1CC=C(CC(=O)N2CCC(C(NCP(C)(C)=O)=O)(C(F)F)C2)CC1 C12=CC(OCC)=C(C=C1F)C2.C12(CCC1)CN(C)C2.C(C(C)C)OCC c1(C(N2CCC3C(NC(C4CC(SC)C4)=O)C32)=O)ccc([N+](=O)[O-])cc1 C1(C)(C(N(CC(CN(C(=O)CSc2nnc(S)s2)C)O)C)=O)CCC2(CC1)CC2 Cc1cc(CNC(=O)C=CC2CCCN2C)oc1C(=O)NCC1(N(C)C)CCC1 C1(NC(CCC(C)=O)=O)COC2(CCN(Cc3cccc(O)c3)CC2)C1 c1(C(N2CCC(CCNC(=O)Cc3ccns3)CC2)=O)n[nH]c2c1CCC2 C1(NC(C2(NC(C)=O)CCCCC2)=O)CN(C(=O)C(C)C)CCC1C C1(C(=O)NC(CCCCNC(c2ncc(OC)cn2)=O)C)CNC(=O)CC1(C)C C(=O)(C(C)(O)CC(F)(F)F)N1CCCCC(CN(C(=O)CCC(N)=O)C)C1 C12(NC(C3C(=C)C3)=O)CCC(C(=O)N(C)CC3(C)CC3)(CC1)C2 C12(OC)CCC1CN(C(=O)C(F)CC1CN(C(=O)CNC=O)C1)C2 C1(CCC)CN(C(C2C3C4CCC(C4)C23)=O)CCN1C(c1cncc(N)n1)=O C12(CC(=O)N(C3(C(N(C4CCCCC4)C)=O)CCC3)C3CC3)CCCC1C2 C1(CNC(CC2(OC)CCC2)=O)CN(C(=O)CCN2CCOCC2)CCC1(F)F C12(CNC(C3N(C(CCC)=O)CSC3)=O)CC(NC(=O)C=CC3CC3)(CCO1)C2 c1(C(=O)NC2(C)CCN(C(C3(C)CCC(=O)N3)=O)CC2)nc2ncccn2n1 C12(c3nc(-n4cc(SC)cn4)no3)C(C(=O)C3CC3)C3CC1C2C3 c1(C(N(C)CC=CC(=O)NCCC2NC(=O)NC2=O)=O)cc(C)nc(C)n1 C1(F)(CNC(C(CC)n2ccnc2)=O)CCCN(C(=O)Cc2cccc(F)c2)C1 C(=O)(CC(C(F)(F)F)NC(=O)CCOCC1CCC1)N(C1CCOCC1)C c1(C(N2CC3C(NC(C(c4ccc(F)cc4)C)=O)C3C2)=O)c(O)ccc(Cl)c1F CCCCCCCCCC(=O)NCCCOCCCNC(c1cn(CC)nn1)=O C#Cc1ccc(C(=O)NCC2CCC(NC(c3cnnn3C(C)C)=O)C2)cn1 N#CC1=C(C(=O)N2CCOC(CC(N3CCC(OCCF)C3)=O)C2)CCC1 C(CCCCC(=O)NC1(C(=O)NCC2CC2)CCCCC1)OC(C)=O CCCC(C(=O)N1CCCC1=O)C(C)C N1(C(=O)NC2CCCN(c3ccc(Cl)nn3)C2)CCC(O)C12CCC2 N1(C(C2C(NC(c3cc(OC)c(F)cc3)=O)CCO2)=O)CC2CCC(CO)(C2)C1 N1(C(CC(C)Oc2ccccc2)=O)CCCC2CCN(C(c3ccco3)=O)CC12 C(=O)(CCCCNC(N)=O)N1C(CN(C)Cc2nn(C)c(=O)o2)CCC1 c1(CNC(C(=O)NCC2(NC)CC2)=O)ccc(Br)c(C)n1 c1(OC(C(CC)C2CCOCC2)=O)cn(C)nc1I c1(CN2CCC(O)(C(C(N)=O)(F)F)C2)n[nH]c2ccc(OCC(F)(F)F)cc12 CC(C)(CNC(=O)CNC(c1cnn(C2CC2)c1)=O)CO c1(C(=O)NC2CC(NC(c3c(C)nn(C)c3)=O)C(O)C2)cccc(F)c1F CC1CCCC(CCNC(=O)CCCNC(=O)COC2CCCC2)C1 c1(CS(=O)(=O)NC(C2CCC(NCC3(CC)COC3)C2)=O)ccc(F)cc1 N1(C(C2(C)CCCC2)=O)CCCC2(CCC(NC(=O)C=CC3CCCCC3)C2)C1 N1(C(c2cc(C)c(C)[nH]2)=O)CCCCCC1CNC(C12CC=CC(C1)OC2)=O C1(C(=O)NCC(C(C)C)NC(=O)C2=NNC(=O)C2)CCC(S(N)(=O)=O)CC1 c1(CC(=O)N(CCCN(C(=O)CC2CCC(=O)N2)CC)CC)ccnc(OC)c1 C1(C(=O)NCCN(C(=O)C(F)(F)CC2CCCO2)CCC)CCCCC(C)(C)C1 N1(CCc2c(C)nc[nH]2)CC2(C1)CN(C(C1(C=O)CC1)=O)C2.c1(S)ccccc1 c1(C(=O)NCC(C(C)C(C)C)NC(C(C)(C)SC)=O)ccc2cncn2c1C c1(C(=O)NC2(C)CC(NC(C(c3cccc(C)c3)O)=O)C2)ccc(F)c(Cl)c1 C12(C(=O)NC3(C)CCCC3)CC3CC(C1)CC(F)(C3)C2.C12C3CN(CC13)C(=O)N2 c1(C(N2C(CN(C(CCC(C)N(C)C)=O)C)CCCC2)=O)ccc(F)cc1O N1(C(=O)C(c2cccc(F)c2)F)CCN(C(=O)C2=CCSC2)C(CC2CC2)C1 Cc1ncc(C(=O)NC2CN(C(=O)CCCn3ccnc3)C3CC23)cn1 N1(C(=O)NCCCC(F)(F)F)CCN(C2CCC(C(=O)O)O2)CC1 C=CCCCCCC(=O)NC1CCN(C(c2nc(C)c(C)nc2C)=O)CC1(C)C c12c[nH]nc1C(=O)N2.C1(C(C(=O)OC)OC(=O)C=CC(=O)N(C)C)CCCOC1 c1(C(=O)NC(CNC(C2(NC(C)=O)CCCC2)=O)C)[nH]nc2ncccc12 CC(C)C(C(=O)NCCC(O)C1CCCC1)C(C)NC(=O)CC1(O)CCC1 C12(NC(Cc3ccc(CCC)cc3)=O)CCN(C(c3nc(O)c(C)s3)=O)CC1C2 O=C1NC(=O)C(C(C2N(C(=O)O)CC(O)C2)c2ccccc2)N1.O(C(F)F)CC Cc1noc(Cl)c1CC(=O)NCC1CC(CNC(=O)CNS(=O)(=O)N(C)C)C1 c1(C(=O)NC2(CO)CN(C(C3(C(N)=O)CC3)=O)C2)nc2cc(F)ccn2n1 C1(NC(c2c(CC)onc2)=O)CCN(C(=O)CSc2nnnn2C)C12CCC2 C=CC(C)C(=O)N(C1CCN(C(C2CCC2)=O)C1)C C1(NC(C2CCCCO2)=O)C2CCN(C(C3C4CC(F)(F)CC34)=O)CC12 c1(CC(=O)NCC2(OC)CN(C(c3cnc(C)s3)=O)C2)ccc(Br)cc1I C1(NC(C2(C)C=CCN2C(=O)CN2C(=O)CCC2=O)=O)CN2CCC1(F)CC2 C12(NC(C(O)NC(=O)OCC)=O)CCCC1CN(C(c1ccc(C)c(F)c1)=O)C2 CC1CC(=O)NCC1C(=O)NCCCC(=O)NCC(N1CCCC1)C N1(C(CCCC(C)NC(c2cc(=N)[nH][nH]2)=O)=O)CCC2(CCOC2=O)C1 N#CC1(NC(C2CCC2)=O)CCN(C(=O)CCN2C(=O)C=CC2=O)C1 c1(CNC(c2c(C)oc(Cl)n2)=O)cnc2c(c1)CNC2=O N1(C(c2cccc(C#C)c2C)=O)CCC2(CCN(C(c3cnnnc3C)=O)C2)C1 N1(C(C(C)OC(C)(C)C)=O)CCC(N=[N+]=[N-])(C(=O)NCCCN=[N+]=[N-])C1 C1(F)(CNC(c2nc(C)[nH]n2)=O)CCCN(C(C2CN(C3CCOC3)C2)=O)C1 N1(c2cc(COC)ncn2)CC2CC1CN(C(C1(C)CCCCCC1)=O)C2 N1(C(c2c(C)cc(Br)cc2)=O)CCC2CCN(C(C34CCCC3C4)=O)CC12 C(CCCl)(CCCl)(c1n(C(C)C(C)C)nnn1)NCc1cnn(C)c1 CCC(CCC(=O)NCC1OCCC1C)NC(=O)CN(C(=O)C(C)C)C c1(OC)c(C)cc(C)cc1C.c1(C(N2c3ccc(s3)C2)C)ccccc1C C(C)(CCC(=O)N(C1CCN(C(C2OCCO2)=O)C1)CC1CC1)OC N1(C(c2cc(C)no2)=O)CC2CC1C2NC(C12CCCC1(C(N)=O)C2)=O C1(C2(O)CCOCC2)(C(N2C(CN(C)C(C3CCCSS3)=O)CCC2)=O)CC1 C(=O)(CC1=CCN(C)CC1)N1CCC(O)(N(CC(N2CCC(C)CC2)=O)C)CC1 c1(C(=O)NCC)cc2[nH]nc(CN3CCN(C(C)COC)C(C)C3)c2cc1COC C12CCN(CC1(F)F)CC2.CCC(C(=O)NC)C(C)C.C(C)=CC=C C123CCC(CC1)(C2)NC(=O)C(C(C)(C)C)OC1CC(C1)C(=O)N3.N1(C(C)=O)CCCC1 C12CN(CCCC1(F)F)c1cc(ncn1)N2.Cc1cnc2ccccn12 C1(Nc2cc(SC)c(C)o2)COC2(CCC2)C1.c12cn(nn1)CCC(=O)N1CCC21 C1(C(=O)OC2OCCN(CC)C2)C2CCN(C(=O)CN(C(C)(C)CC)C(C)C)CC12 Cc1oc([N+](=O)[O-])cc1C(N1CCN(C(c2ccn(C)n2)=O)CC1CC(F)F)=O c1(C(C(=O)NCC2CC2)N(C(COCC)C)C)ccc2c(c1)CCCC2 Cc1cc(C(N2CCCC2c2ncc(C(=O)O)[nH]2)=O)n2nc(C(F)(F)F)cc2n1 c1(C(=O)NC2C(NC(=O)CCc3nc(O)n[nH]3)CCC2)cccc2c1CCO2 c1(C(=O)NC(C2CCOC2)CNC(CCNC(=O)C2CC2)=O)cccnn1 C(=O)(C(C)(O)C(C)C)N1CCC(CC(C)NC(C(C)OCCC(C)C)=O)CC1 c1(C(=O)NCCC2CN(C(c3c(C)cncc3C)=O)C2)nccc2c1NCCC2 CC(C(=O)N1CC(CNc2ccc(C(N(C)N(C)C)=O)[nH]2)C2(CC2)C1)C(C)(C)C c1(CC(=O)NC(C2(O)CN(C(c3c(C)csc3)=O)C2)C)ccc(Cl)cc1F C1(C(=O)NCC(C)N(C(=O)C(C2CCOCC2)C)C)COC2(CO)CC1C2 N1(C(c2cncc(C)n2)=O)CCC(F)(C(=O)NCc2ccn(C)n2)CC1 N(C(=NCCc1c(F)cccc1F)N1CCC2(C1)CC2(F)F)C(CC)C c1(C(N2CC(N(S(C3(CC)CC3)(=O)=O)C)C2)=O)ccc(O)c(C)c1O c1(C(C)NC2CCC(C)NC2)cc(Br)ccc1F c1(CC(=O)N(C)CCNC(C2CCC(C)(C)CO2)=O)ccc(O)c2ccccc12 C1(O)(CNC(c2cncc(C(C)C)c2)=O)CCCN(C(C2(C)CCCS2)=O)CC1 CC1CN(C(c2ccc(N(C)C)cc2)C(=O)Nc2ccccc2Cl)CC1N(C)C C1(C(=O)NCC(N2CCOCC2)=O)(NC(C(F)=C(C)C)=O)CC(O)C1 C1(NC(C(C(Cl)SC)(C)C)=O)C(NC(C2CN3CCN2C(C)C3)=O)CCC12CCC2 C(CCC(C)(C)NC(c1cn[nH]c1)=O)NC(C1(C=C)CCC1)=O C1(C)(OC)C=CCN1Cc1cn(CCCc2cccc(N)c2)nn1 C1(C(N)=O)CCCCC1C(=O)NC1CCCC(NC(C23CC(CC(F)F)(C2)C3)=O)C1 c1(OCC)cccc(F)c1C(N1CC(CNC(=O)Cn2nccc2C)C1)=O N1(C(C2(CC)CCCN2C(c2csc(CO)n2)=O)=O)CCCC(F)CC1 C12(C(=O)NC3CN(C(C=CCC)=O)CC3F)CC1Cc1c[nH]nc12 CCC(C(=O)N(C1CCN(CC(=O)NC(c2ccccc2)C)C1)C(C)C)C(C)C n1(CCOC)nccc1C(=O)NCC(C)CN(c1ccncc1)C.C(=O)(CNC)N c1(C(N(CCCNC(=O)CSCC2CCCO2)C)=O)ccc(F)c(O)c1 C(=O)(C(Cn1cncn1)NC(=O)CCc1cc(C)[nH]n1)NCC1(C(CC)O)CC1 c1(C(N2CC(CNC(C3ON=C(C)C3)=O)N(C)CC2)=O)ccc2nc(C)cn2c1 C1(NCc2sccc2)CN(Cc2cn[nH]c2)CC1F CC1CC(=O)Nc2ccc(C(=O)NC3(CO)CN(C(c4ccoc4)=O)C3)cc2N1 S(=O)(=O)(c1ccc(C)cc1F)N1C(C=C)CC(c2ccccc2)C1 CCC(C)C(CC(=O)NOCc1ccc(O)cc1)NC(=O)Cc1cccnc1 c1(C(=O)NCC(C)NC(=O)C2=COCCC2)cc2c(s1)CCC(C)(C)C2 C(=O)(C1CCc2cccnc21)NC1(CNC(=O)COc2ccccc2F)CCC1 CCCC(C)(CCC)C(=O)NCC(O)CN(C)C(C1CCCOCC1)=O c1(C(N2CCS(=O)CC2)C(=O)NCCCSCC)ccc(F)c(OC(C)C)c1 N=c1cc(C(N2CCC(CCCNC(c3cc(Cl)cnn3)=O)CC2)=O)cc[nH]1 N1(C(c2n(CC)ccc2)=O)CCC2(CCCN2C(C2(C)COC(C)(C)CO2)=O)C1 C(=O)(C1COc2ccc(Cl)cc21)N1CCC(N(C(C(=O)NCC=C)C)CCO)C1 c1(CC(=O)NCCC2OCCN(C(c3[nH]cc(C)c3)=O)C2)c(C)nn(C)c1Cl C1(CC#C)(C(=O)NCC(C)(O)CNC(c2ccc(CCC)[nH]2)=O)CCCC1 C1(NC(C2CN(CCC)C(=O)C2)=O)CC2CC(NC(=O)C=CC3(C)COC3)C2C1 Cc1ccc(O)c(C(N2CCCC2C(C)NC(=O)COCc2nnc(C)s2)=O)n1 O=C(C#CC1CCCOC1)NC1CC(NC(C23CCC(CC2)OC3)=O)C1 Cc1nnc(CN(C)C(C2CC=CCC2NC(=O)CC(F)(F)Cl)=O)n1C C1(C(=O)OCC)Cc2cc(Br)ccc2N1C(c1cccc(Cl)c1Cl)=O C(=O)(C(C)(C1CCC1)NC(C1CCNC1=O)=O)N(CC#C)CCF c1(C(=O)NC(CC(C)NC(C2CCCO2)=O)C)cccnc1O c1(C(N2CCC(C)C2CNC(=O)C=Cc2ccoc2)=O)nnc(O)nc1O c1(C(=O)NC2CCC(CNC(COCC=C)=O)C2)ccc(Br)cc1 c1(NC(C2CC3CC3N2Cc2cc(Br)c(Br)s2)=O)ccc(Cl)nc1Cl C1(C(N(CCCNC(c2ccc(SC)s2)=O)C(C)C)=O)CC2CCCCCC12 CCC(C)C(O)C(=O)NCCN(CCOCCO)C(c1ccnc(OC)c1)=O C1(NC(C(CC)C#N)=O)CCN(C(C23CCCN2CCC3)=O)CC(C)(C)C1 Cc1ccc(C(=O)NCC2(F)CC(NC(c3nncs3)=O)C2)cc1 N1(C(COC)=O)CCC(C(=O)NCC(F)(F)C(C)C)(OC)C1.C(C=O)NC C=CCC(C)C(=O)N(C1CC(NC(c2cn(C)c(O)n2)=O)C1)C N1(C(c2ccc(COC)s2)=O)CCN(C)CC1CNC(C1(O)CCOC1)=O C1(NC(CCSC)=O)CC(C(=O)NCc2cnco2)C(O)C1 c1(OC)nc(Cl)ccc1S(=O)(=O)NC(c1nnc(C2CCCCC2N=[N+]=[N-])o1)=O N1(C(CC(COC)C)=O)CCC(C(F)(F)F)n2nccc21 CC1(C)CCC1NC(=O)CC1CCN(C(=O)CCc2cnco2)C1 C1(NC(CC=C)=O)CCN(C(=O)CCC23CCC(CC2)C3)CC(O)C1 c1(C(=O)NCCC2COCCN2C(c2ccc(F)cn2)=O)ccc([N+](=O)[O-])nc1 c1(C(N(C2CCN(C(c3ccncc3)=O)C2)CC)=O)cc2ccsc2s1 C(CCO)(C(F)(F)F)NC(C1CC=CCC1NC(C1CC2(CC2)C1)=O)=O C(=O)(CC1=NN(C)C(=O)C1)NC1CN(C(C2(OC)CCOCC2)=O)C(C)C1 C#CC1CN(C(C2CCCCN(CC)C2)=O)CC1NC(C1CCCC1F)=O O(Nc1ncnc2c1CCC2)SC1=NOC(C)(C)C1 c1(C(=O)NCC2CN(Cc3ncccc3F)CCO2)ccc(Br)cc1 Cc1c(C(=O)NCC2(NC(=O)CCCC(N)=O)CCC2)sc2cccc(F)c12 Cc1cc(CCC(N2CCC(O)(CNC(c3sccc3CO)=O)C2)=O)cc(C)n1 C1(C(C)(C)C)CC(C(=O)NCCCCCNC(C23COCC(C2)OC3)=O)=NO1 C(CC(=O)N1CC(CC2CC2)C1)(C(F)(F)F)NC(c1nc(N(C)C)oc1)=O C1(NC(C2(C=C)CCC2)=O)CC2CN(C(c3ccc(CO)nc3)=O)CCN2C1=O C1(c2c(C)n[nH]c2)CCCN(C2CCN(CC(=O)NC3CC(=O)N(C)C3)CC2)C1 Cc1nc(CC(C)C)oc1C(=O)N(CC(C)(C)CNC(=O)CC(C)(O)C1CC1)C c1(C(=O)NCC(C2CCOCC2)C)ccc([N+](=O)[O-])c(O)c1 C1(CCNC(=O)CCc2cnco2)CCC(NC(c2ccoc2Br)=O)C1 Cc1cnc(NCC2CN(C(c3csc(Cl)c3C(F)F)=O)CC2C)nc1O C#Cc1cncc(C(=O)NC(C)C(C)NC(c2c(C)ccn2C)=O)c1 c1(C(C)NC(C23C(CN(S(C(C)C)(=O)=O)C2)C3)=O)cc2ccccc2cn1 C1C(=O)N=C2C=CN(N2)C2CN1C2.N1(CC(=O)OCCC(C)C)CCc2sccc2C1 N1(C(C(C)(C)C)=O)CCC12CN(C(c1ccc(C3CCCC3)cc1)=O)C2 C1(C(=O)OCC(C)C)COCCN1C(CCCOc1cc(C)on1)=O C(C(CC)(CC)NC(=O)C(CC)n1ccc(C2CC2)n1)NC(C(CC)NC(C)=O)=O N1(C(CC2CCN(C(C)C)CC2)=O)CC(NC(=O)CSC(C)(C)C)C(C2CC2)C1 Cc1ccc2c(c1)CC(C(=O)NCCCCNC(=O)C=Cc1ccsc1)S2 CC(Cn1cccn1)C(=O)NCC1(C(=O)NCC2CC2Cl)CC1 Cc1c(Br)c(C(=O)NC(CNC(C2COC(=O)N2)=O)C(C)C)nn1C c1(CC)ccc(C(=O)NC2CN(C(c3ccccc3NC)=O)CC23CC3)c(C)n1 c1(C(=O)NCC(CNC(CCN(C(C)=O)C)=O)C)cnn2c1CCCC2C c1(C(=O)NCC(C)NC(c2c(F)cc(F)c(F)c2F)=O)cc2cc(F)ccc2s1 C1(NC(c2cnn3cc[nH]c(=O)c23)=O)CCN(C(C2CC23CC3)=O)CC12CCC2 C1(C(=O)NC(CCCNC(C=CCC)=O)C)CCC(C)(O)CC1 c1(C(=O)NCC(CNC(C2(CCOC)CCC2)=O)C)csc(=N)[nH]1 C(=O)(C1=NNC(=O)CC1)N1CCCC(CC(=O)N(C)CCN2CCCC2=O)C1 C1(O)(C(C(=O)N(C2(C(=O)OC)CC2)C)F)CN(C(C2CS(=O)(=O)C2)=O)C1 CC1CC(NC(=O)C(C2CCCCC2)=O)CCN1C(C1CSCC(=O)N1)=O c1(C(N(C)CC2CCCN2C(C2CCNC2=O)=O)=O)cc2c(O)ncnc2cn1 C1(C(=O)NC2CCN(C(c3cccc(C(C)=O)c3F)=O)C2)CCc2nn[nH]c2C1 Cc1oc(C)c(C(=O)N(C)CCN(C(c2c[nH]c(C#N)c2)=O)C(C)C)c1Br c1(CC)c(C)nc2ncnn2c1NC(C)CC(C)NC(=O)CCCC(C)(F)F C1(CNC(CNC(CCC)=O)=O)CN(C(c2cccnc2C2CC2)=O)C2CC12 c1(C(=O)NCC2(NC(CC3CCCC(C)O3)=O)CCC2)ncn2c1CCCCC2 C12(NC(c3nc(COC)sc3)=O)CCCN(C(c3ccc(F)o3)=O)CC1C2 N1(CCC2CC(OCC)C2)C(=O)CN(CC(C)(C)Oc2cccc(C#N)c2)C1=O N1(C(C2C(CNC(CC)=O)C2(C)C)=O)CCC(F)(F)CC1 N1(CC(C(C)C)OC)CCC2CN(C(=O)CN3CCOCC3)C2C1 c1(OC)cc(OC)nc(N2CCCC2CNC(c2cc(F)cnc2Cl)=O)n1 CC(C)CC(F)C(=O)NCCOCCN(C(=O)CC1CCCCC12CC2)C C(=O)(CCC(C)(C)C#N)N(CC(=O)Nc1nc(C)c(C(C)C)s1)CCOC N1(C(C(CSC)O)=O)CCCC2(CCN(C(C3(CC(C)C)CC3)=O)C2)C1 N1(C(CCc2onc(C(C)C)n2)=O)CC2(CCN(C(C3CNC(=O)N3)=O)CC2)C1 c1(OC)c(C(=O)NC2CCN(C(=O)C=Cc3cnn(C)c3)CC2C)ncnc1C C(CC(=O)Nc1cccnc1F)(C(F)(F)F)NC(c1nn(C)c(F)c1)=O CC(CCC(=O)N1CC=CC1Cn1cc(-c2nccn2C)nn1)N(C)C C1(NC(c2ccc(N3CCN(C(C)=O)CC3)cc2)=O)CCCCC2(CC2)C1 c1(C(=O)NC(CN(C(C(CC)OC2CCCC2)=O)C)C)cccc2cnsc12 C1(NC(COCCCOC)=O)C=CCCC1C(=O)NCCCCSC CC(C)CC(C(=O)NCC1CCC(C)(C)OC1)n1cc(C2(C)CCC(=O)N2)nn1 N1(C(C2(C(C)(C)C)CCCC2)=O)CC(NC(=O)C=Cc2cc[nH]n2)CC(F)C1 CC(C)(C)C(CCC(=O)NC1CCCC1(C)CO)NC(=O)CCCC1OCCO1 C1(NC(c2ccc(C(C)C)s2)=O)CCN(C(=O)COCCCF)C1(C)C C1(C(N(CCC#N)CC)=O)CCCN1.C(C)(C(OC)OC)N C(C1c2ccccc2CN1C)NC(c1n(CC)nnn1)C(C)(C)C1CC1 CC(C)(C)CC(C(=O)N(CCCC1CC(C)(C)C1)C1CC1)NC(=O)OC(C)(C)C C(=O)(C(CCC)S(N)(=O)=O)NCC(CC=C)NC(C1CC(n2ccnn2)C1)=O C(=O)(CC1OCCc2sccc21)NCCN(C(c1c(C)c(Cl)cnc1)=O)C(C)C N1(C(C(C)OCC)=O)CCN(C(=O)CN(C(=O)CC2CC2(C)C)C)CC1 C1(C(=O)NC(C=C)CO)CN(C)CCN1C(c1cnncc1OC)=O CC1(C)C(=O)Nc2ccc(C(N3CC(NC(C4CSC4)=O)CC(F)(F)C3)=O)cc21 C(c1ccco1)=CC(=O)NCC=CCNC(C(n1ccc(C(F)F)n1)C)=O C(=O)(CC(C)F)N(C(C)C(=O)NCC1CC(C2CC2)C1)CC Cn1cccc1CC(=O)NCC1CC1CNC(=O)CNC(C1CCC1)=O N1(C(C2C(CCC)C2)=O)CC2CN(C(c3cc(CC)ccc3F)=O)CC2C1 N1(C(CSCC=C)=O)CCC(C(=O)NCC(Cl)C(C)(F)F)C(O)C1 c1(OC)ccc(C=CC(=O)NCCC2CN(C(c3ncccn3)=O)C2)cc1OC N1(C(C(C)CC2CC2)=O)CCC2(C1)CN(C(=O)CN(c1cnccn1)C)CCO2 CC1(C)CN(C(=O)CC2C=CCCC2)CC1CNCc1[nH]ccc(=O)c1O O=C(N=c1[nH][nH]c2cccnc12)C(=O)Nc1cnn2ccc(C3CC3)cc12 N1(C(=O)NCCOCCOCCOCCOC)CCC2(CC1)CN(C)C(=O)O2 C1(C(N(C(C)CNC(=O)CCc2cccs2)C)=O)CCC2(CC1)CC2 CCC(CC)C(F)C(=O)NC1CC(C)(CNC(=O)COCCc2cccs2)C1 CCCC(C)CC(=O)N1CCC(NC(c2cnn(-c3ccccn3)c2)=O)C1 C(=O)(C1=CNS(=O)(=O)N=C1C)N1CCCN(C(C(C=CCCC)O)=O)CC1C C1(NC(C(CC)(CO)OC)=O)CC12CCN(C(=O)CCn1ccc(C)n1)CC2 C1(NC(=O)Cn2ccnn2)CN(C(C2CCCOCC2)=O)CC1n1cccn1 CC1(C)CCCC(C)(NC(=O)C(CCF)NC(=O)CC(C)(C)CC2CC2)C1 CC(C)(C(=O)NCC=CCNC(=O)CCC1CCCO1)C1CCCO1 C1(C(=O)NC2C(C(=O)NC3CC(C(C)O)C3)CC2)CC(C)(C)CO1 c1(C(=O)NC2CC(C)(CC3CCC3)C2)cn2ccccc2n1.C1(=O)CN1 C(c1ccc(O)cc1)=CC(=O)NCC1CC(C)N(C(C2CC3C=CC2C3)=O)CC1 C1(CNC(c2c(C)c[nH]n2)=O)CN(C(C2CC3CCC(C2)S3)=O)CC1(C)C c1(OC)cncc(C(=O)NCC2CCCN2C(C2(C(N)=O)CC2)=O)c1C O=[N+]([O-])c1cccnc1N1CCOCC(n2cc(N3CCC(N)C3)nn2)C1 c1(COC(Cc2cc(OC)c(F)cc2)=O)cc(O)c2ccoc2c1 N1(C(C2(c3ccc(Br)cc3)CCC2)=O)CC2CC2C1C#N.Cc1cnncc1CN C1(COC)(NC(=O)C(C)N(C)C)CCN(C(=O)CC2C=CCCC2)C1 CCCC(C)C(=O)NC1(c2cn(CC(N3CCOCC3C3CCC3)=O)nn2)CC1 C1(CCC(=O)N(C)CC2CC=CCC2)CCN(C(=O)C(N2CCCCCC2)=O)CC1 c1(C(COCC(N2CC(CCCCNC(C=C(C)C)=O)C2)=O)C)cccc(F)c1 c1(CCC(c2n(CCC)nnn2)(C)NC2CCC2C(=O)OC)cccc(Br)c1 C(=O)(C(F)CCC(C)C)N1CCN(C(C=CSC)=O)CC1c1cn[nH]c1 C1(NC(=O)C2=CCSC2)CCN(C(c2csc(Cl)n2)=O)C(c2ccccc2)C1 N1(C(C2CCN(CCCCC)CC2)=O)CCCC(S(=O)(=O)NC2CC2)C1 c1(N(C(=O)CONC(=O)OC(C)(C)C)CC)ccc(C#N)cc1OC N1(C(c2cccnc2S)=O)CCC2(COC(CNC(C3CC(O)C3)=O)C2)C1 c1(-n2cc(NC(C(C)C#N)Nc3ccco3)nn2)cc(Cl)ccc1CSCC1CC1 C1(CC(=O)NC(CC#C)CC)C2CCCC2N1C(=O)CC1(C#N)CCOCC1 CP1(=O)CCN(CC(=O)NCC2CCN2C(=O)Cc2ccc(F)c(CO)c2)CC1 C1(NC(C(C2CC2)OCC)=O)CN(C(=O)C(=O)NOC)CCC1CO Cc1ccc2[nH]c(C(=O)NC(C)Cc3ccc(C#N)cc3)cc2c1C Cc1ccc(C(=O)NCCOC2CCN(C(C3CCCC34CCC4)=O)C2)nc1O CC1(O)CCC(CC(=O)NCCN2CCCN(C(=O)CCCN(C)C)CC2)CC1 N1(C(c2cc(C)nn2C)=O)CCC(NC(=O)C(c2ccccc2)O)C(F)C1 CC1OC2(C(=O)NC(Cc3cccc(Br)c3)C3CC3)CCC1CC2 c1(C(=O)Nc2c(C)ccc(CS)c2)nnc2c(Cl)cc(C(F)(F)F)cn12.C1(N)CC1 CCC(CNC(c1ccc(-c2ccsc2)nc1)=O)CC(F)F N1(C(C(C(C)O)N(C)C)=O)CC(NC(=O)CCOC2CCCC2)C(C)(C)C1 C1(C(=O)NC2COCCN(C)C2)CC(C)(C)CCN1C(c1ccc(C#N)[nH]1)=O n1(CC)cc2c(n1)CCCC2C(=O)NCC1CCN1C(=O)CCN1CCCC1=O CC1(C)CN(C(C23CCC(CC2)C3)=O)CC(C)(C)C1NC(=O)CCC1CC1C C(c1ccc2ncccc2c1)=CC(=O)NC(C)CCNC(=O)Cc1ccccn1 CC1(C)CCc2nc(O)c(C(=O)NCC3CN(C(C4C=CCCC4)=O)C3)cc2C1 N1(C(CNC(CCC)=O)=O)CCC2(CCN(C(c3ccc4ccccc4c3)=O)C2)C1 c1(N2C3CC(NC(C4(CC)CCC(O)CC4)=O)C2CC3)ncnc2[nH]ccc12 N1(CC(=O)NCC(O)CCNC(=O)Cc2cncc(Br)c2)CC2CCC1C2 C1(C(=O)NC2CC(NC(c3cc(C(C)=O)on3)=O)C2)CCn2cncc2C1 C1(CCC)(CO)CCN(C(=O)C(C)NC(=O)C(CC2CCC2)OC)C1 C(=O)(C1=COCCO1)N1CCC(N(CCC)C(C2CCC2C#N)=O)CC1 Cc1nc(N(C)C)sc1C(N1CCC(CN(C(=O)C=Cc2ccncc2)C)C1)=O C1(CNC(C2(CC)CCCCO2)=O)CC(C)CN(C(=O)CC(O)CN(C)C)C1 CC1CCCC(CC(N2CCC(CCNC(=O)Cn3cnnc3O)CC2)=O)C1 N1(C(Cc2c(C)nccc2)=O)CC(NC(c2cncc(CO)c2)=O)CC2(CC2)C1 CCC(C(=O)N(CC(C)NC(c1cc(C(C)(F)F)ccc1C)=O)C)C(C)(C)CC C(=O)(C(C(F)(F)F)Oc1ccccc1)NC1(NC(C(C)N2CCCC2)=O)CC1 Cc1cccc2c(C(N3CC(NC(C4COC(=O)C4)=O)CC3C)=O)n[nH]c12 CC(C)(O)C(F)(F)C(=O)N1CCN(C(C23CC(CC(F)F)(C2)C3)=O)CC(CO)C1 C(CC(C)(C)C)(C(=O)NCC1CCN1C(C1(C#N)CC2(CC2)C1)=O)OC c1(C(=O)NC2C(NC(c3cc(C)sc3)=O)CC2)c(C)noc1C(C)C CC1(CNC(C2(c3ccccc3)CC2)=O)CCCN(C(C2(C)C=CCCC2)=O)C1 Cc1ccc2nc(C)c(C(=O)NC3CC(CNC(C45COCC4C5)=O)C3)cc2c1 C(C(C)C(=O)NCCOC1CCN(C(=O)C(CO)N(C)C)C1)SC c1(CCC)nc(C(O)Cc2ccccc2F)n(-c2ccc(C3CC3)cc2)n1 C12(CC)CN(C(=O)C(F)C(F)(F)F)C(CNC(=O)CN(C)CC(N)=O)(C1)C2 c1(OC)ccc(C(=O)N(CC(C)CNC(=O)Cn2c(C)c(C)sc2=O)C)c(F)n1 c1(C(=O)OC2CCC2)ccc(OC(C(C)=C2CCCC2)=O)c(C)c1.C1C(O)CN1C C1(C(N2C3CC(NC(C4C(C)CCCC4)=O)C3CC2)=O)CN2CCCN1CC2 N1(C(C(C)C2CCCO2)=O)CCCC(CO)(NC(=O)Cc2ccn(C)n2)C1 Cc1nccc(C(N2CCCC(CN(C(=O)CSc3n[nH]c(O)n3)C)C2)=O)n1 Cc1cc(C(N2CCOC(CN(C)C(C3CC4(C3)CC(C)C4)=O)C2)=O)cc(C)n1 C12(C)CN(C(C)(C)C1)C2=O.C(C(C)(C)C(C)(F)F)NC(C)=O C1(C(N2C(C)CC(CNC(c3cc(OC)nc(C)c3)=O)C2)=O)CCn2nncc2C1 N1(C(C(C)CCCc2ccccc2)=O)CC2(C1)CN(C(C1CC1CF)=O)CCO2 c1(N2C(=O)CC(C(=O)NC(c3nc(CN(C)C)n[nH]3)C)C2)ccc2[nH]ccc2c1 Cc1nc(C(F)(F)F)oc1C(=O)NCC1CCCN(C(c2ccc(Cl)s2)=O)C1 C1(OC)CC(CNC(c2ccc(O)cn2)=O)N(C(c2ccc(C(C)C)cc2)=O)C1 c1(C(C)C)nccc(C(=O)NC2CN(C(c3cc(C(=O)N(C)C)ccn3)=O)C2)n1 CC1CCc2n[nH]cc2C1C(=O)NCCN(C(c1cc(CO)on1)=O)C1CC1 c1(C(N2CCC(Nc3nccc(OC)n3)C2)=O)cnn2cccnc12 C(=O)(CC(C(C)(C)C)NC(c1cncc(C2CCC2)c1)=O)OC Cc1cncc(C(N2CCCC2C(C)(C)C(=O)NC2C=CCC2)=O)c1 c1(C(=O)NCC(CC(C)C)NC(CCC(C)=O)=O)c(F)ccc(C)c1Cl C1(NC(c2cc(C(C)(F)F)n[nH]2)=O)CN(C(=O)C(C)(C)C(F)F)CCC1CO Cc1nc(NC(C)=O)sc1C(N1CC(F)C(NC(=O)Cn2cnnn2)C1)=O C(=O)(C#CC1CCCCC1)N1CCC(CC)(CC)CC1.C1(=O)CCC(C)(C)CN1 N1(C(C(CC#C)O)=O)CCC2CCC(C1)N2C(c1c(F)cc(C#N)cc1F)=O c1(C(N(CC(C)NC(c2ccn(C)c2)=O)C)=O)c(Cl)ccc(Cl)c1N c1(N2CCCN(C(c3c(OC)c[nH]n3)=O)CC2)ncnc2ccc(O)cc12 C(=O)(C(F)C(C)CNC(=O)C(COc1ccccc1)COC)OC C1(CC(=O)NC2CCC(CNC(C34COCC3C4)=O)C2)(OC)CCCCC1 C1(NC(CCC2(C)N=N2)=O)CC(=O)N(CC(c2cccc(Br)c2)=O)C1 CC1CCCCC1(CNC(=O)CN(c1ccncc1)C)NC(=O)C#CC1CC1 Cc1c(C(=O)NCC(C2CCOC2)NC(=O)C(F)=CCCF)cnc2ncnn12 C(=O)(N(CC)OC)CC1(CO)CC12CCC2.CCC1CC(=O)Nc2n1ncc2 N1(C(c2sccc2C(F)F)=O)CCC2CN(C(=O)CCc3nncs3)CC2C1 c1(C(N2C(C#C)CC2)=O)n[nH]c2c1CN(C(c1cnncc1NC)=O)C2 C(=O)(CCCCC#N)N1CCCN(C(c2ccc(C(C)O)cc2)=O)C1 CCS(=O)CC(=O)N1CC(C)(CCC(=O)NCC(C)(C)OCCO)C1 n1(CC)nc(C)c(C(=O)NC2C3CC(NC(C4COCC(C)O4)=O)CC23)c1Cl c1(C(=O)NCC(CO)NC(COCCSC)=O)sccc1-n1ccnn1 S(=O)(=O)(c1cccc(CN)c1)Nc1c(=O)cc(C(=O)OC)n(C)c1 C12(C(N(C3(C(=O)OC)CCC3)C3CC3)=O)CC(C)(CN1C(=O)C(F)C(F)(F)F)C2 C1(CNC(C=C(COC)C)=O)C(C)CCCN1C(c1ccnc(OC)c1F)=O C#CCCCC(c1nnnn1CCC(=O)OCC)NCC(CO)SC c1(C(=O)NC(C)C(C)NC(c2csc3c2CCCC3)=O)cccn2ccnc12 C12(C(N3CCC(NC(C4OCC5CCCC45)=O)(CF)C3)=O)CC3CC1C2C3O N1(C(Cc2ccc(C)s2)=O)CCC2CCN(C(c3cc(C(F)F)nn3C)=O)C2C1 N1(C(C=CC(C)(C)SC)=O)CC(CNC(c2ccc(O)nn2)=O)CC12CCC2 C1(CNC(CCC2C(C)(C)C2)=O)N(C(=O)CC2C(C)(C)C2(C)C)CCCC1(C)C C1(NC(CC)=O)CCC(C(=O)N(CCNC(c2csc(O)n2)=O)C(C)C)CC1 c1(N(C)CC2N(C(C3=NOC(CC)C3)=O)CCCC2)nc2cc(C)cc(C)c2s1 C(=O)(C1=C2CCN=C2NC=C1)N1C2CC(CN(C(C3(C)CC3Br)=O)C2)C1 CC1C(NC(=O)C(Cl)=CCl)CCCN1C(C1CC1c1ccsc1)=O C1(c2cn(CC(N3CC(C(C(=O)N(CC)CC)C)C3)=O)nn2)CC(F)(F)C1(F)F c1(C2(C(=O)NC3CN(C(c4cc(=O)cc[nH]4)=O)CC3F)CC2)ccc(Cl)c(Cl)c1 C1(NC(COCC(=O)NC(c2cccs2)=O)=O)C=CC(CNC(CN(C(C)C)C)=O)C1 c1(C(N2CC(C(N3C(O)(CC)CCC3)=O)NC(=O)C2)=O)cc(Br)cc2[nH]ncc12 C(=O)(C1CCCc2cccnc21)N1CC(OC)(CNC(C2CC(=O)CO2)=O)C1 C(=O)(C1=NOC(CC2CC2)C1)N1CCCC(C(C)(C)C)C1.C12(CC1)C(=O)O2.C(C)(C)(C)O CCC(O)CC(=O)NCCC(C(=O)NCC(C)C(=O)OC)OC C(=O)(CC(C)(C)C(F)F)NC1CC(NC(c2c(C(=O)OC)c(C)[nH]n2)=O)C1 N1(C(C2(CO)CCN(C(c3c(C)csc3)=O)C2)=O)CCC2(CCN(C)C2)C1 c1(C(N2CCC(CC)(NC(C3CC(SC)C3)=O)CC2)=O)ccc(F)c(OC)c1F N1(C(c2ccc(C)c(O)c2)=O)CCC(C2CC2)C1CNC(=O)CCCCC(F)F O=C(CCCn1ccnc1)NC(Cc1cnc[nH]1)C(=O)NC(CCO)C1CC1 C1(C(=O)NC2C(CCC)C2)C=CCN1C(=O)CC1CC(C)=NO1 C(=O)(CCCC(F)(F)F)NCCN1CCC(NC(c2ncc(N(C)C)nc2)=O)CC1 C1(NC(COCCOCC)=O)CC(F)(F)CC1C(N1CCC(O)(C(C)C#N)C1)=O C(C(C)C)(C(O)C(=O)NCCC(=O)NC(c1snnc1C)C)OC C(c1ccc(F)cc1)=CC(=O)NC1C(CNC(C(CC)C2CCC(=O)N2)=O)CC1 C(=O)(CC(C)C1CCCCC1)NCC(CC)NC(C1CCCCO1)=O C1(NC(C(=O)NCCN(C)C)=O)CCN(C(=O)CCN2CCC(O)CC2)CC1O C1(c2cc(C)on2)CC(CNC(=O)CCC2(C)CC2)(NC(C2CCC(F)C2)=O)C1.CO CCC(CC)(CCNC(C1CCN(c2ccccc2)CC1C)=O)NC(=O)C(C)C C(=O)(C(C)(C)C1=CCSCC1)NCC1CN(C(C=C(C)C(C)(C)C)=O)C(C)CC1 c1(C(N2CC(O)(CNC(C3C(C(=O)NCC#C)C3)=O)C2)=O)cccc(Cl)c1F C1(C(=O)NC(C2CCC2)C)COC2(C1)CN(C(=O)C(C)(C)F)C2 Cc1nc(CC(C)C)sc1C(N1CC(CNC(c2csc(CO)n2)=O)CC1C)=O CCCS(=O)(=O)CC(=O)NC1COCCN(C(=O)COCC(=O)OC)C1 C12(CNC(C(F)=CC)=O)CCCCC1N(C(=O)COCP(C)(C)=O)CC2 C(=O)(CC(C)(C)CCC)NC(CC=C)CNC(=O)C(C)S(C)(=O)=O c1(C(=O)NC2CN(C(C3=C(C)OCC3)=O)C(C)(C)C2)sc(S(N)(=O)=O)cc1C N1(C(c2ccc(COC)o2)=O)CC(NC(=O)C2=C(C)OCCS2)CC(F)(F)C1 CC1=C(C(=O)N2CC(NC(c3csc4nccn34)=O)CC2(C)C)COCC1 c1(C(=O)NCC2CCN(C3CC4C=CCC34)CC2)cc(Br)c2ccccc2n1 c1(C(=O)NCC(CNC(C(CCO)N(C)C)=O)CO)ccc(Cl)c(N)c1 Cc1cnnc(O)c1C(N1CC(C(=O)NCC2CCC2C)CC(C)C1)=O c1(C(=O)OC)cccnc1C(=O)NCC1(CCNC(=O)CCN2CCCCC2)CC1 c1(C(N2C3C(C(=O)Nc4nc(C)c(C)s4)C(C3)C2)=O)cc(Br)c(F)cc1C CC1(C)CC(CNC(=O)C=Cc2ccco2)N(C(C2CC=CCC2)=O)C1 N1(C(c2cnc(Cl)[nH]2)=O)CC2(C1)CN(C(c1c(Cl)csc1Cl)=O)CCO2 c1(OCC=C)c(C(N2CCOC(CCNC(=O)C(C)C3CCC3)C2)=O)cccc1C Cc1ccc(C(C(C)C)NC(N2CCC(Nc3ncccn3)C2)=O)s1 c1(C(=O)NCC(NC(CCn2ccc(C)n2)=O)CC2CC2)ccnc(OC)c1 Cc1cocc1C(N1CCC1C(=O)N(C)CCc1ccccc1)=O Cc1cc(F)ncc1NC(=O)C(c1ccoc1)NC(=O)C=CC1CCOCC1 C1(=CC(=O)NCC2C(CC(=O)NCCCCOCC)C2)CCCCC1 N1(C(c2ncn3c2CCC3)=O)CCCC2CN(C(=O)C(F)(F)c3cncs3)CC12 C1(NC(CCCC(C)c2ccccc2)=O)CC2(CCN(C(=O)C#CC(C)(C)C)C2)C1 C(CC)(CC(F)F)NC(CN(CCOC)C(c1ccc(C)cc1)=O)=O C(C(C)(C)CNC(=O)CC1CCC2CC12)NC(C=CC(=O)OCC)=O N1(C(C(C)CC2CC2)=O)CCCC2C1CCN2C(C12COC(CF)(C1)C2)=O c1(C(C)NC(=O)C(N)=O)ccc([N+](=O)[O-])cc1.C1(CC)CCCN(CC)C1 C(CCC(C)(C)C(=O)NCC1=NOC(C)C1)NC(C(n1ncc(C)c1)C)=O C1(N(C(c2cnc(CC)s2)=O)C)CCCN(C(=O)CC(c2cccc(F)c2)C)C1 c1(NC(C(=O)NCC2C3CN(C(C(CCC)O)=O)C2C3)=O)c(Cl)cccc1Cl c1(C2C(C(=O)Sc3ccc(C(=O)NC(C)C(C)n4cccn4)o3)C2)ccncc1F C1(C(=O)NC2(C)CN(C(c3cnc(COC)s3)=O)C2)C(C(=O)OC)CC(=O)N1C c1(C(=O)NCC2CN(C(Cc3c(C)noc3Cl)=O)C3C2C3)cnn2c1CCC2 Cc1cc(CNC(c2ccnn2C(C)C)=O)oc1C(=O)N(C1(CO)CC1)C c1(C(=O)NC(C)(C)CCCNC(c2cn(C3CCC3)nn2)=O)ccc(Cl)cc1Cl Cc1ccc(CCC(=O)NCCCCC(C)NC(c2cn(C(F)F)cn2)=O)c(C)c1 C1(=O)CC(C(F)F)NC(=O)C(CC)N1C.C(CCN=[N+]=[N-])SC C(C)(C)(CN=c1nc(CC2CC2)[nH]s1)C1CCN(C(C(C)CN(C)C)=O)CC1 CC1CN(C(C2C3CCC(C3)N2C(C2CC(F)CN2C)=O)=O)Cc2nncn21 c1(C(N(CCC(C)NC(C2(CC(C)C)CCC2)=O)C)=O)nnn2c1C(=O)NCC2 C(CC)(C(F)F)N(C(=O)NC(C1CCOCC1)C#C)C c1(CC(=O)NC(COC)C(=O)NCc2cocn2)cncnc1O C1(C(N2C(CCC)CCC2)=O)CCCC(NC(=O)C2CC2)CC1 c1(C(=O)NC(CCSC)C(=O)N(C)Cc2cc(C)cs2)cncc(F)c1C C1(SC)CN(C(C2(n3cncn3)CC2)=O)CC1NC(=O)CC(C)(C)O.C1CC1 N1(C(c2cc(C)ns2)=O)CC2CC(C)N(C(C3CC(O)(C(F)(F)F)C3)=O)C2C1 C1(N(C(Cc2ccc(C)nc2)=O)C(c2ccccn2)C)CCNCCC1C CCN=C(NCc1cc2ccccc2s1)N1CCCC(CSC)C1 c1(CC(=O)NCC(C)(C)Nc2cc(COC)ncn2)nc2c([nH]1)CCCC2 c1(C(N(CCCNC(c2coc(Br)n2)=O)C2CC2)=O)cc2ccccc2cn1 c1(C(CNC(C2(C(F)(F)F)CC2)=O)N(C(=O)C(F)n2ccnc2)C)cnn(C)c1 C(=O)(CCCCC(=O)NC)NC(CN(C(=O)CC1CCC2(CCC2)CO1)CC)C c1(C(=O)NC(CNC(Cc2c(C)n(C)nc2)=O)C(C)C)coc2c1COC2 C1(NCC)CCN(C(=O)NC2(CO)CCC2C(C)C)C1 Cc1cc(C)n(Cc2nc(-c3ccc(C)o3)nn2CCC2(C)CC2)c(=O)n1 N1(C(C=C(CCC)C)=O)CCCC(CC)(NC(c2cccc(C(=O)N(C)C)c2)=O)C1 N1(C(C2(C(C)C)CC2)=O)CCCN(C(c2nocc2C2CC2)=O)CC1C(C)C N1(C(C(COC)O)=O)CC2(C(N3CCC3C(C)O)=O)CCC1CC2 c1(C(=O)OC)ccc(F)cc1S(=O)(=O)NCCC1C=CCC1 c1(C(=O)NCC2COCCN(c3c(C#N)cncn3)C2)ccc2cncn2c1 C(C(=O)NCC(C)(C)NC(c1occc1Cl)=O)(C(C)C)c1ccc(C)s1 CN1CCC(CCNC(=O)C(O)CCNC(C2CSC2)=O)C1=O C(=O)(C(C)(C)CC(C)(C)C)NC1CCN(C(CN(CC)CC)=O)CCC1CO Cn1nc(C(=O)NCc2csc(C(=O)NCCCc3cccnc3)c2)cc1O c1(OC)ccccc1C(C)CC(=O)NC1CCC(NC(c2c[nH]c(=N)s2)=O)C1 C1(NC(CN(CC(C)(C)C)C)=O)CN(C(=O)Cn2nccc2N)C2CCCCC12 CC1(CC2CCCC2)CCCN1C(C1CN(C(=O)CC2NC(=O)NC2=O)C1)=O CN1CCC(C)(C(N2CCC(NC(=O)Cn3ccc(Br)n3)C(O)C2)=O)CC1 C1(NC(c2cnc(C)[nH]2)=O)CC2(C1)CN(C(C1CC3(C1)CC(C)C3)=O)C2 N1(c2cc(NCC(O)CSc3ccccc3)ncn2)CC(C(F)(F)F)C2(CC2)C1 c1(C(=O)NC(CCC)CNC(c2cc(C)sn2)=O)cnc2cccc(C)n12 C1(O)(CNC(CCCN(C)C)=O)CCN(C(c2ccc(CCF)cc2)=O)C1 C1(CC(=O)Oc2ccc(F)cc2)CCCN(N2CCC(CCOC)C2)C1 CN1CCN(C(C2CCC(=O)N(C)C2)=O)C(C(N2CCC2C2CCCCC2)=O)C1 N1(C(c2n(CCOC)ncc2)=O)CCCCC(CNC(=O)C(C)n2ccnc2)C1 c1(N(C(=O)COC2CCN(C(=O)C=CC(C)(C)SC)C2)CC)cc[nH]c(=N)c1 CN1C(=O)CCC1C(=O)NCCC1CC(NC(c2ncoc2Br)=O)C1 c1(CCC(=O)NC2C(NC(c3c(C)ncn3C)=O)CC2)ccc(F)c(F)c1F c1(SCC)cc(C(N2CCCC2CN(C(c2csc(Cl)c2)=O)C2CC2)=O)ccn1 C(=O)(CCS(N)(=O)=O)NC(C(C)(C)c1csc(-c2ccccc2F)n1)=O N1(C(CC2C(C)C2(F)F)=O)CCCN(C(=O)C=CC(=O)N(C)C)CC1 c1(NC(c2c(-n3cccn3)cccc2F)=O)cccn2nccc12 N1(C(c2c(C)nc(C3CCCN(C(=O)CN)C3)[nH]2)=O)CCC2CN(C3CC3)C2C1 C1(NC(c2n[nH]c(CC)c2C)=O)CCCC(C(=O)N(C)Cc2n[nH]c(C)n2)CC1 C(C)(C)(CCCCC(=O)N1CCCC(CN(C)C(c2cccc(O)n2)=O)C1)OC CC12CCC(C(N3CC4CCCC3(CNC(c3cccnc3)=O)C4)=O)(CC1)CO2 C(=O)(C(CNC(C1(C)CCCC1O)=O)CC1CC1)NCC1(C)CCC1 C(=O)(CC(C)C(=O)OC(C)(C)C)NCCC(=C)CNC(C1(CO)CCC1)=O c1(-c2cc(N(C(CNC(C3N(C(C)=O)CCC3)=O)C)C)on2)cc(C)cc(F)c1 c1(C(=O)NC(CC)CN(C(=O)CSCC(F)(F)F)CC)cc([N+](=O)[O-])cnc1N C#CC1CC2CCC1N(C(C1(CC=C)CCCN1C(=O)CCN=[N+]=[N-])=O)C2 Cc1coc(C(c2nnnn2C(C)C)NCCC2CCCCO2)c1 c1(N2CC(NC(c3ccc(COC)[nH]3)=O)C(C)CC2)ncc([N+](=O)[O-])cc1Br c1(OC)nc(C)ccc1C(=O)N(CC(C)O)CCNC(=O)CCc1nccs1 c12ccc(c([N+](=O)[O-])c1)NC2.C1(C)(SCC)CCC(NC(C2C3CCC23)=O)CC1 O=C(CC=C(Cl)Cl)NN1CCCC1C(=O)NC1CCCC(O)C1O C1(C(c2n(CCOC)nnn2)NC2(CSC)CCC2)CC2(C1)CC(C)C2 C(CCS(N)(=O)=O)c1cn(C2C([SH](C)CCO)CCC2)nn1.N12CC(C1)C2=O N1(C(c2cc(C)on2)=O)CCC(CC(=O)NCc2nnc(O)n2C)C1(C)C N1(CCNC(C2(NC(CNC(=O)OC)=O)CCCC2)=O)CCS(=O)CC1 N1(C(C(=O)NC(c2cccs2)CNC(=O)C(F)(F)F)=O)CCCC1C1OCCO1 c1(C(=O)NCC2(F)CC(NC(=O)CC3CC3(Cl)Cl)C2)cccc2ccncc12 c1(C(=O)NC2(CCNC(C=C(C)C3CC3)=O)CC2)csc2c1CCC(C)C2 N1(C(CNC(CCCCC)=O)=O)CC(NC(c2ncn(C(C)C)n2)=O)CCC1C Cc1oc(Br)cc1C(=O)NC1CCN(C(C23COC(CF)(C2)C3)=O)C1C1CC1 CCCN=C(NCc1cn(C)nc1-c1ccccc1)NC1CSC1(C)C C1(CNC(c2ccc(C#C)cn2)=O)CN(C(=O)C=C2CCCCC2)CCS1(=O)=O N1(C(c2ccc(=N)[nH]c2Cl)=O)CC23CCCCC2(C1)CN(C(=O)CCF)C3 CCC(C(=O)N1CC(CC(=O)NC(C)C(C)(C)C)(OC)C1)SC C(c1ccco1)=C(C)C(=O)N1CC(C(O)C(=O)N2CCC2C(=O)NCCO)C1 N1(C(c2c(CCC)nco2)=O)CCCCC(N(C(=O)CCCC(C)=O)C)C1 c1(C(=O)NCC2(OC)CCN(C(C(C(=O)OCC)OC)=O)C2)cccn2nccc12 C(CC(=O)NCC1CC1NC(=O)CC1(CO)CC1)(C(C)C)OCC c1(OC)ccc(F)cc1C(F)(F)C(=O)NC(CNC(=O)C(O)C1CC1)CC(C)C CCC(C(C)CN(C)C)NC(C1N(C(=O)COCC2CCC2)CC(F)C1)=O c1(CC)nnc2cc(NC3CC(NC(=O)CC4CC(OC)C4(C)C)C3)ncn12 C1(C(=O)NC2(C)CC=CC2)CCN(C(=O)C(O)C(F)(F)F)C(C)(C)C1 C1(C(N(C)CC2N(C(C3(Cl)C(C(C)=O)C3)=O)CCC2)=O)CC2C=CC1O2 C(CC(=O)N1CC(C)(C(=O)OC)CC1(C)C)(C(C)(C)C)NC.N1CC(OC)C(OC)C1 CN(Cc1c[nH]c2c(F)cccc12)N1CCc2c(cc(Br)cc2Cl)C1 c1(NC(COC)C2CC2)cc(N(CC(n2cccn2)C)C)nc(C(F)(F)F)n1 C1(OC)C2CC3CC1CC(C(=O)NCC(C(C)(C)C)NC(=O)CP(C)(C)=O)(C3)C2 C(CN=c1[nH]cncc1I)C1CN(C(c2c(C)noc2C(C)C)=O)C1 C1(C=C)(C(N(C(C#C)C)C)=O)CCN(C(c2cc(Cl)c[nH]2)=O)C1 c1(NC(=O)NC2CCC(CC)C2)cnc2c(c1)c(=O)n(C)c(=O)n2C N1(C(C(C)SC(F)(F)F)=O)CCN(C(=O)C2=COCC2)CC1c1ccccc1Cl Cc1cc(C(=O)N(C(C)C(C)CC)C2CC2)c(C)o1.C1C(=O)N1 C1(CC)COCCN1C(=O)C(CC1CCOCC1)NC(c1ccnc(CO)c1)=O CCCCCC(C)(C)C(=O)N1CC(NC(c2ccc(CO)o2)=O)CC2(CCC2)C1 C(=O)(C(F)C(C)CNC(=O)OC(C)(C)C)N1C(C#C)CCC1 N1(C(C(CC(C)C)F)=O)C2CCC1CN(C(C1CCS(=O)(=O)CC1)=O)C2 C(=O)(CC(C)(C)CCOC)N1CCC(N2CCN(C(CCCCOC)=O)CC2)C1 c1(OC)ccc(C(CNC(=O)NCCC(C2CCOCC2)O)C(=O)O)cc1OC CS(C)(=O)=NCC(=O)N1CCC(CNC(C2CC(=O)N(CC(F)(F)F)C2)=O)C1 c1(C(=O)NC(CC(C)NC(=O)C(c2ccccc2)N(C)C)C)nnc(O)cc1O c1(NCCC(=O)OCC)ccc(S(=O)(=O)NC2=Nc3ccc(Br)cc3SC2)cc1 c1(C(=O)NCC(C)OC(F)F)csc(N=S(C)(C)=O)n1.c12ccc(cc1)OC(=O)C2 C1(CNC(c2ccc(C)cc2N)=O)CCCCN(C(=O)C(O)c2ccsc2)CC1 CCC(CC(=O)N(CC(=O)NC1CC2CCC(C1)C2O)C)C(C)C n1(CCNC(c2cn[nH]c2)=O)cc(C(=O)NC2(CO)CC(F)C2)nn1 C(=O)(C1=CCCN(C(=O)C(C2CCC2)N(C)C(C)=O)C1)NC(CCSCC)C N1(C(c2c(C)noc2-c2cnccn2)=O)CCC(C)(C)C(NC(=O)CC(F)F)C1 c1(NC(C(CNC(C(C2CCOC2)OC)=O)(C)C)=O)c(OC)cccc1O Cc1cc(F)c(CC(N2CC(O)(CNC(c3n[nH]cc3C)=O)C2)=O)c(Br)c1 C(=O)(C(CO)C(C)(C)C)NCC(C)NC(c1c(C)nsc1)=O N1(C(C(CC)C)=O)CC(NC(c2cnn(CC(F)(F)F)c2)=O)CC12CCC2 c1(C(=O)NC23C(CC(=O)OCC)CC(CC2)C3)c(C)cc(C)nc1OC C(=O)(CS(=O)(=O)C1CC1)N1C2C(NC(c3c(C)ncn(C)c3=O)=O)CC(CC2)C1 C(=O)(C(F)(F)C1CCOCC1)NCC1C(NC(=O)CCC2CCOC2)C1 c1(-c2cc(C(=O)NCCC3CCN(C(C(F)OC)=O)C3)on2)cccc(F)c1 CC(=O)CCN=C(NCc1nnc2n1CCCCC2)N1CCC(c2nncs2)C1 C#CC1CN(C(c2cnc(O)n2C)=O)CCN1C(c1ccc(C)c(C)c1)=O C12(CNC(Cc3cc(C)no3)=O)CC(NC(c3csc(C(C)C)n3)=O)(C1)C(C)O2 c1(C(=O)NC2(CN(C(c3cnc(C)n3C(F)F)=O)C)CC2)cn2cnnc2cn1 C=C(C)C1OCCC1C(=O)NC1CC2(C(N3CCN(CC)C(C)C3)=O)COC1C2 C(=O)(C(C)C(F)(F)F)NCc1n(CC(N2CCC(CC)C2)=O)cc(Cl)c1 N1(C(C(CCC)C(=O)OC)=O)CC(NC(C2CC(C)(C)C2)=O)CC12CCOC2 Cc1ccc(C(=O)NCC(=O)NC2CC(NC(=O)CCCC3CCCCC3)C2)s1 Cc1cc(C(=O)N(C(CNC(=O)CN(C)S(N)(=O)=O)C2CC2)C)ccc1[N+](=O)[O-] C1(OC)CN(C(c2ccc(Cl)c(C)c2)=O)CCC1NC(c1cc(C)cc(C)c1)=O N1(C(C2C3CC(=O)CC32)=O)CC2CCCC1CN(C(c1csc3nnsc13)=O)C2 c1(C(N2CCCC(NC(CC3(C)CCCCC3)=O)CC2)=O)cnc2n1CCCC2 c1(CC)cccc(C(N2CC(OC)C2)=O)c1N.C12CCC(CC1)CC(=O)N2C C1(F)(C(=O)NCC(N(OCC)C)=O)CCCN(C(=O)CN2CCSCC2)C1 C(=O)(CC(O)C(C)CC)N1CCC(C#C)(C(N2CC(N(C)CC)C2)=O)C1 c1(C(=O)NCCCC(C)NC(c2scnc2Cl)=O)ccc(=O)n(O)c1 c1(N2CCNC(=O)C2Cc2ccccc2)nc2c(F)c(Br)cnc2s1 C(c1cccc(Cl)c1)=CC(N1CC(NC(c2c(C)nc(COC)s2)=O)(CO)C1)=O N1(C(c2ccc(COC)o2)=O)CC(NC(c2ncnc(O)c2F)=O)CC1(C)C C1(NC(c2c(C)nc(Cl)s2)=O)CN(C(=O)CCc2c(F)cncc2F)CC(F)(F)C1 C1(C(=O)NCCC(Cc2ccccc2)NC(=O)Cc2ccoc2)CCC(F)(F)C1 c1(OC)ccc(CNC(C2C=CC(NCc3cncc(C)c3)C2)=O)c(F)c1 N1(C(c2c(OC)cc(N)cc2)=O)CCCC2CN(C(=O)COCCO)CC12 c1(C(N(CCCN(C(=O)C(C2CCOCC2)O)C)C)=O)nn(C)cc1Cl N1(C(c2cncc(NCC)c2)=O)CCCC12CCN(C(c1nccnc1Cl)=O)C2 C(CC(C(=O)N(C)CC1(OC)CCC1)NC(=O)Cc1cccc(O)c1)=CC N1(C(Cc2c(C)ncnc2O)=O)CCCC(O)(CNC(=O)C(F)OC(F)(F)F)CC1 CCCC(CC(C)C)C(=O)N1CC(CCNC(=O)C=CCF)C(C)C1 N1(C(C(CC)CC)=O)CCCC1C1CCCN1C(=O)COc1ccc(C)cc1 C1(CNC(C2CCC(NC(COC(C)=O)=O)CC2)=O)CN(C)CCN(C)C1 c1(CNC(C2CCC(C)C2)=O)ccc2c(Br)nn(C)c2c1 N1(C(COC(CC)(C)C)=O)CCC(C(=O)NCC(C)(C)F)CC1C C1(C2CCN(C(=O)CCc3cccnc3)C2)(NC(=O)CC2NC(=O)NC2=O)CC1 c1(C(=O)NC2(C)CCN(C(c3sccc3C#N)=O)C2)cc2ccc(F)cc2s1 Cc1csc(Cl)c1C(=O)NCc1cccc(NC(=O)COCCF)c1 N1(C(CC(=O)N(C)C)=O)C2CCC1C(C(=O)NC1CC3CCC(C1)O3)C2 C(=O)(C1=C(Cl)CCC1)N1C(CNC(=O)CSCCc2ccccc2)CC1 CC(C)CCCC(=O)NC(CC1CC1)C(=O)NCC(C)(C)C(F)F C(=O)(C(C)(C)C(=O)NCCn1ccc(C(=O)NCCOc2cnn(C)c2)c1)NC C1(C(=O)NCCC(CCC)C)CCCCC1(C)NC(c1nccc(C)c1F)=O N1(C(c2c(C)nsc2N)=O)CCC(C)C(N(C(=O)C(C2CCCCCC2)O)C)C1 C1(NC(C=C(C)C)=O)CC(CO)N(C(=O)CCC=CBr)C1 N1(CCC(=O)N(C(C)CN(C)C(C2CCCSC2)=O)C)CCNC(=O)C1 C1(NC(c2cc(=O)cc[nH]2)=O)CC2C1CCN2C(c1cc(C(F)(F)F)no1)=O c1(C(=O)OCc2onc(C(C)C)n2)cc(Br)ccc1OCC1CCOCC1 C1(CC(=O)NCCN(CCCN(C)C)C(C2CCCCO2)=O)COC2(CCC2)CO1 CC1CCN(C(=O)CC2CCCN(C(=O)CCN)C2)CC1 N1(C(C(c2cncnc2)C)=O)CCN(C(=O)CC2CC2)CC1Cc1cccc(F)c1 C1(C(N2CCC(CN(C(c3cc(C)sc3C)=O)C)C2)=O)CCCNS1(=O)=O CCC(O)CC(=O)NC(CC1CC1)C(=O)N(CCC(=O)OC)CC N1(C(c2n(C(C)C)ncc2)=O)CCC(C)(NC(c2ccc(CS(C)(=O)=O)cc2)=O)C1 C(=O)(C(CC)C(=O)NCCCC(C)NC(C1CN(C(N)=O)C1)=O)OCC c1(OC)cc(OC)cc(C=CC(N2CCN(C(=O)CC3(C)CC3)CC2CF)=O)c1 C1(C(=O)NCCOC2CCN(C(=O)C=CC=C(Cl)Cl)C2)CCS(=O)(=O)N1 N1(C(c2ccnc(CC(C)C)n2)=O)CC(NC(=O)Cc2ccoc2)CC2(CC2)C1 N1(C(c2ccc(O)nn2)=O)CCCC2(C1)CN(C(C1(n3nccn3)CC1)=O)C2 C1(CCC(=O)NCc2c(CC)nco2)CCCN(C(=O)C(C)c2ccsc2)C1 Cc1cccc(O)c1C(=O)NC(C1CCN(C(C2CCCCC2O)=O)C1)C c1(C(=O)NCC(C(C)(C)C)NC(c2cnc(CC)[nH]2)=O)cc(C)c(Cl)cc1F C(=O)(CC(C(F)(F)F)NC(C1CCC(=O)N1)=O)NCCc1c(C)nn(C)c1 CC1=C(CNC(=O)C(C)(C)CN(C(=O)Cn2ccc(C)n2)C)CCC1 N1(C(CC(CC)C(C)C)=O)CC2CCCC(C1)N2C(c1ccnc(F)c1)=O c1(OC)cc(S(=O)(=O)NNC(=O)C(N)CO)ccc1NC(=O)N(C)C C1(CC(N2CC(N(C)CC)C2)=O)CN(C(c2cc[nH]c2C)=O)CCC1C N1(C(C=COCC)=O)CCC(O)(C(C)NC(C2CC3CC3C2)=O)C1 N1(C(C(=O)NCC)=O)CCN(C(=O)CCc2ccnn2C)CC1C1CCC1 C1(C)(CCC)CCN(C(=NCCOCC)NCc2cnccn2)C1 c1(CC(=O)N(C(CCNC(CC(C=C)C)=O)C)C)cn2ccsc2n1 C1(NC(C(c2ccccc2)SC)=O)CC2(C1)CC2NC(=O)C=Cc1cnc[nH]1 CCCCCCC(C)C(=O)N1CCC(OCCNC(=O)C(C)(C2CC2)OC)C1 c1(Sc2scc(CC3CN(C(C(C)(C)N4CCCC4)=O)C3)n2)ccccc1Cl C1(CC(N2CC(CC(CN(C(c3c(C)cns3)=O)CC)(C)C)C2)=O)CCCCC1O Cc1cc(CN2CCC(CC(=O)Nc3nc(O)cs3)C2)c(O)c(Br)c1 N1(C(CSc2n(C)nnn2)=O)CC2(C1)CN(C(C1CCCCCC1)=O)C2 c1(C(N2C(c3ccccc3)(CC)CC2)=O)cc(O)c(Br)cc1C C1(O)(C(=O)OC)CN(C(=O)CCN(C(=O)C(c2cnn(C)c2)C)C2CC2)C1 C(CCCCC(=O)OC(C(=O)N(CCC(C)C)CC1OCC2CCC1C2)C)OC N1(C(c2c(OC)nsc2)=O)CCCN(C(=O)CC2CCCNC(=O)C2)CCC1 C12(NC(=O)CO)CCOCC1CN(C(c1cc(F)ccc1C(F)F)=O)C2 O=C1CCCC(CC(=O)NC2CCCN(C(=O)C(O)Cc3ccccc3)C2)N1 C(=O)(C(F)(CNC(=O)C(C)N1CCCC1)C(C)C)NCc1ccc(SC)s1 CCC(C)(C(=O)N1CCC(O)(CCNC(c2ccc(Cl)c(C)c2O)=O)C1)C(N)=O C1(COCC(N2C(CC(C)O)CCC2)=O)CCC(C(F)(F)F)OC1 CCCCCC(O)C(=O)N1CCCCC1C(C)NC(c1cnc(N(C)C)s1)=O N(C1CC2(CN(C(c3ccn(C(F)F)n3)=O)C2)n2ccnc21)C(=O)C(O)C1CC1 N1(C(c2c(C)onc2Br)=O)C2CCC1CC(NC(C1(F)CC1)=O)C2 N1(C(c2n[nH]c(C)c2N)=O)CC2CC(NC(C3CCCCC3O)=O)CC2C1 n1(CC)ccc(C(N2CC(N(C(=O)CN3CSCCSC3)C)C(O)C2)=O)cc1=O Cc1c(C(=O)N(C)CC2CCCN(c3ncns3)C2)cnn1C(C)(C)C N1(C(C2C(C(=O)OC)C2)=O)CC2(C1)CN(C(=O)CCc1ccc(C)o1)CCO2 C1(C(Cn2cc(CSCC(=O)NC34CCC(C3)OC4)nn2)=O)CCS(=O)(=O)C1 N1(C(C(C)Sc2ccc(OC)cc2)=O)CC(NC(=O)CC(C)(C)C)CC(F)C1 C1(C(=O)NC(CCNC(C2(CC=C)CCCC2)=O)C)CC2CCC2C1 C12CC3CCC(C1)N3C(=O)C1(c3cn2nn3)CCC1.C1(SCC)CCS(=O)(=O)C1 C(=O)(C1=CCCCO1)N1CC(CNC(COCCCC)=O)C1 c1(N)ncc(F)cc1CC.c1(CCC)ncc(OC=O)cn1 c1(C(N2CC(CNC(C3C(C)OC(=O)N3)=O)C(C)C2)=O)cc2cc(Cl)ncc2[nH]1 N1(C(c2cc(OCC)n[nH]2)=O)CCC2(CCN(C(c3csc4nnsc34)=O)C2)C1 c1(C(N2CCC(C)(NC(C(C(C)C)OCC)=O)C2)=O)onc2cc(C)ccc12 c1(C(=O)NCC(C)C)cccc(CNc2ncoc2C(F)(F)F)c1 C(=O)(C1=CC2C=CC(C1)C2)N1C(C(=O)NCCCOCC)CCCC1 C1(C2CCCN(C(C3(C#N)CCCOC3)=O)C2)(NC(C(CC)C(C)C)=O)CC1 O=S(=O)(c1ccc(OC(F)F)c(F)c1)NC(CC(F)(F)F)CCCO C(C(C)(C)CC(=O)NCCC(C)N(C)C(c1ccc(N)c(N)n1)=O)OC(C)=O C1(NC(CCCCC#C)=O)CCN(C(c2cncc(N)c2)=O)CCC1CO c1(C(=O)OC)ccc(C(C)(CO)NC(c2nc(C)no2)=O)c(OC)c1 C1(C)(C(=O)NCc2scc(CNC(CS(CC)=O)=O)n2)CCC(C(C)=O)C1(C)C C1(CC(COC)NC(=O)COC2CCCC2)CCN(C(=O)C(F)C2CCC2)CC1 CCC(CC)C(C(=O)N1CC(F)(F)CC1C(=O)NC1CC(C)(CO)C1)OC C1(C(=O)NC(CC)(C)CCNC(=O)C(O)C2CCCC2)CC(=O)N(OC)C1 c1(OCC)cc(C(=O)NC(C(N2CCCC2C(N)=O)=O)C2(O)CCC2)on1 C(=O)(CCC(C)(C)C)NCCC1(O)CN(C(c2cc(C)c(C)[nH]2)=O)C1 N1(C(CCCCOC)=O)CCCC(CCNC(C23CCCN2CCC3)=O)CC1 O=C(C1=CC2CCCC12)NC1CC2(C1)CN(C(c1nccn3ccnc13)=O)C2 N1(C(c2c(C)nn(CCC)c2C)=O)CCC(C)N(C(c2cnc(N)cn2)=O)CC1 c1(C(C(=O)NCC2(CNC(C(c3ccn(C)c3)C)=O)CCC2)O)cccnc1 C(C)(CCC(C)C)N(c1cccc(C(=O)NCC2(OC)CN(C(C)=O)C2)c1)C1CC1 N1(C(C(Cc2cn[nH]c2)NC(c2cccc(C)n2)=O)=O)Cc2cncnc2C1 C12(NC(=O)C3=CSCS3)CCC1CN(C(c1cnc(O)c(Cl)c1)=O)C2 C1(NC(CN(C)C)=O)CC(CCC(=O)NCC(N2CCC2CC2CCCC2)=O)C1 C(c1ccc(Cl)cc1F)=CC(N1CCN(C(C(C)NC(=O)NC)=O)C(C)C1)=O c1(NC(C2CCCN(C(C3CCCCCC3)=O)C2)=O)cccc2scnc12 c1(C(=O)NC(CNC(C2C(CN(C)C)C2)=O)(C)C)ccn2cncc2c1 Cc1nc(N2CCCC(C)(CNC(c3coc(C(N)=O)c3)=O)C2)cc(C#N)n1 N1(C(c2[nH]c(=N)sc2)=O)CC2CCCC(NC(c3[nH]nc([N+](=O)[O-])c3Cl)=O)C2C1 c1(C(=O)NC2COC3(C2)CN(C(=O)CCn2ccnn2)C3)ccc2c(c1)COC2 c1(N2CCC(NC(COCC)=O)C(C)C2)ncnc2scc(C)c12 N1(C(C(C=C)O)=O)CCN(CC2(NC(=O)C(=Cc3ccco3)C)CC2)CC1 CC(C)C(O)C(F)(F)C(=O)NCC1CCCN1C(=O)CN(C)C(c1ccoc1)=O N1(C(CN(c2ccncc2)C)=O)CCN(Cc2sccc2Cl)C2CC12 c1(OC)c(C(=O)NC2(C)CN(C(=O)C(C)C(F)F)C2)ccc2c1CCC2 c1(CNC(=O)C(N2CCCCC2CCCc2ccc(Cl)cc2)=O)cccc(Br)c1 c1(CC)ccc(C(C(=O)NCC)N(CCOC)CCOC)s1 CCCCC(CNC(c1ccc(COC)[nH]1)=O)NC(c1cc(Cl)ccn1)=O c1(CC(C)C)ccc(C(=O)NCC2CC2NC(C2COCCO2)=O)cc1 N1(C(CC(C=C)CC)=O)CCOC2(C1)CN(C(c1[nH]c(=N)sc1C(F)(F)F)=O)C2 Cc1ccc(CC(=O)NCC2COCC2NC(=O)CC2=CCCC2)c(Cl)n1 S(=O)(=O)(c1cccc(N2CCOC(C)(CCO)C2)n1)N1C(C)CCCC1 Cc1c[nH]cc1C(=O)NC1(C(=O)NCCc2ccns2)CC1(C)C C1(C)(NC(Cc2ccc(CCC)cc2)=O)CCCN(C(=O)Cc2ccccn2)C1 c1(CCCC(=O)NCC2(CNC(C=CC)=O)CC2)ccccc1F c1(N(CCC(=O)NC(c2ccccc2)C)C)c2c(nn1C)CCCC2 c1(C(=O)NC(CN(C(C(C)NC(C)(C)C)=O)C)C)cc(O)nn1C C1(CC(=O)N(CC(C)CNC(c2ccn(C3CC3)n2)=O)C)COCCN1C c1(C(N(CCCNC(=O)C(C)O)CC)=O)cnc(OC)c[n+]1[O-] C1(C(=O)NC2C(NC(CC3(OC)CCOCC3)=O)C2)CCc2nc(C)ncc2C1 C(CN=c1cc(Cl)nc(C2(C)CC2)[nH]1)C1CC(NC(CC(C)NC(N)=O)=O)C1 c1(-c2nnc(CC(=O)CN3CCOCC3)o2)ccc(Cl)cc1Cl C1(NC(Cn2c(CCC)ncc2)=O)CC(C)CN(C(=O)CCCC(N)=O)C1 CC1(C)CCC(CNC(=O)NC2CC(CC(F)(F)F)C2)OC1 C(=O)(C1=CC2CCCC12)N1CCC(C(C)NC(c2c(CC)noc2)=O)CC1 N1(C(c2cnn(C(C)C)c2C)C(=O)NC)CCSC2CCCCC12 N1(C(c2c(C3(C)COC3)noc2)=O)CC(CNC(C2CC3CC3C2)=O)CC1(C)C N1(C(C2CCCN(C)C2)=O)CC23CCCCC2(C1)CN(C(C1COC(=O)C1)=O)C3 C12(CNC(=O)C(c3cccc(F)c3Br)O)CC3CC(CC(C3)O1)C2 c1(C(CN(C(C(=O)N(CC(C)OC)C)=O)C)(C)C)ccc(Br)cc1 C(=O)(C1c2c[nH]nc2CCC1C)N(CCCNC(c1n(CCC)ncc1)=O)CC Cc1cc(Cl)c(C(c2cc(Br)c(Br)o2)NCc2nnnn2C2COC2)cc1C C1(O)(n2cc(C(C)NC(=O)NC3(C(=O)OC)CCCO3)nn2)CCCNC1 N1(C(C2(CC(=O)OCC)CC2)=O)CC(NC(=O)COC(C)C)C(C)(C)C1 N1(C(c2ccn(CC)c(=O)c2)=O)CC(C2CN(C(=O)C(C)Cc3ccco3)C2)C1 N1(C(C(C)N2CCCC2)=O)CCN(C)C(CNC(C2(C)CCCC2)=O)C1 C1(OCCNC(C23CCC2C3)=O)CCN(C(=O)C(c2ccc(Cl)cc2)(F)F)CC1 C1(CC)CN(C(c2cccn2C(C)C)=O)CCN1C(c1cc(OC)cc(C)c1)=O C1(CNC(=O)CN2CCOC2=O)C(C2CC2)CCN1C(=O)CC1CN2CCC1CC2 C(CCCCC(=O)N1CCOCC(CNC(=O)C(C)(C)c2ccnn2C)C1)OC c1(C(N2CCC(COCC#C)C2)C(=O)NC)nc(F)ccc1Br c1(C(=O)NC2CC(C)CN(C(=O)CO)C2)cccc2nc(O)oc12 O=C(CS(=O)C(F)(F)F)NC1CC(CCNC(c2ccc(C3CC3)nc2O)=O)C1 C=C(Cl)C(C)(C)C(=O)N1CC2CC(C1)C2NC(c1[nH]c(C2CC2)nc1C)=O C(=O)(CCC(=O)NN(C)C)N(CC(N1CC(C=C)C(SC)C1)=O)CC1CC1 c1(C(N2CC(CCNC(=O)C(C)SC)(OC)C2)=O)ccc2c(c1)CCN2 Cc1nc2sc1c(=O)[nH]2.c1(C(=O)NCC23CC(N)(C2)C3)ccc(O)nc1.C1CC1 CC(CC(N)=O)C(=O)N(C(C)(C)CC(=O)N1CC(O)C(F)C1)C O=C(C1=CC2(CCOCC2)C1)NC1CC(O)CN(C(c2cccc(=O)o2)=O)C1 N1(C(c2c(CC)onc2)=O)CCC(c2cn(C3CC(CO)C3)nn2)CC1C C1(OC)CN(C(=O)CCc2cncc(F)c2)C(C)(CNC(=O)Cn2cccn2)C1 c1(NC(C2N(Cc3ccc(NC)cn3)CCC2O)=O)cc(OC(F)F)cc(F)c1 Cc1ccc(C(N2CCC(C(C)NC(c3nc(Cl)c(Cl)s3)=O)C2)=O)n2nccc12 c1(C(N(C2CCN(C(=O)C(C)(F)F)C2)CC)=O)cc(F)c(OC)c(Cl)c1 N1(CC)CCN(CC(=O)N(CCC(C)NC(C2CCCC2SC)=O)C)CC1 C(=O)(CC(C)(C)C(F)F)Nc1c(C(=O)NCC2N(C)CCN(C)C2)con1 N1(C(C23CCC(C(N)=O)(C2)C3)=O)CCCCC(NC(C2(C)CC=CCO2)=O)C1 C1(NC(C(C)N(C)C(c2cc[nH]c(=N)n2)=O)=O)CCC(O)C(O)C1 C1(C(=O)NCCCN(C)C(C2(C)CCOC2)=O)CC(=O)N(C(C)(C)C)C1 C(=O)(CCCC(=O)OC(C)(C)C)NCC(c1ccccc1)NC(C(C)c1ccco1)=O Cc1ncc(S(N)(=O)=O)c(C(=O)NC(C(F)F)c2cccs2)c1C N1(C(c2c(CC)ncs2)=O)CCC(C)C1CNC(=O)CSCc1cscn1 N1(C(CCC(=O)N(CCCc2ccccc2)C)=O)CCOC2(C1)CN(CCO)C2 c1(NC(C(=O)NCC(C)OCC#C)=O)ccc(C(F)(F)F)s1 Cc1n[nH]c(=NC2CC3CC(C2)N(C(c2cnc(C)n2C)=O)C3)s1 c1(CC)ccccc1C(N1CCC(CCNC(=O)CCc2cncn2C)CC1)=O c1(C(N(CCCCNC(CCN(C)CCO)=O)C2CC2)=O)ccc2cnoc2c1 N1(C(c2c(C)nc(COC)s2)=O)CCCCC(CNC(=O)C2=COCCO2)CC1 C(C(C)(CO)NC(=O)C(Cc1cn[nH]c1)NC(=O)CC1CC=CCC1)OC CCC(COC)C(=O)NCC1CC(NC(C2(C)CCCCO2)=O)C1 C1(C(=O)NC(C)CNC(=O)CC2CCCS2)CC(=O)N(c2ccc(Cl)cc2)C1 C1(CNC(c2cnn[nH]2)=O)CCN(C(=O)CC2CCC2)C1 CCCC(C)C(=O)NC(C1(CNC(C2CCCC2)=O)CC1)C C#CC1(C(=O)NCC(n2ccnn2)C)CCN(C(c2ocnc2C)=O)C1 N1(C(CCSCCN(C)C)=O)CC2(CCC2)CC1CNC(C1CCC1)=O c1(-c2nnc(COC(C(C3CN(CCOC(F)(F)F)C3)OC)=O)o2)ccccc1Cl C1(C(c2nnnn2C)NC(C(CC)CCOC)C)Cc2ccccc2C1 c1(CNc2ccc(-c3ccc(C)nc3)cc2)ccc(F)c2occc12 N1(C(c2c(C)nco2)=O)CC(O)(C2(CNC(C3OC4CCC3C4)=O)CC2)C1 Cc1coc(C(=O)N(C(C)CCNC(c2cn(CCO)nn2)=O)C)c1C CC1CN(C(=O)COC(F)(F)C(F)(F)F)CCC1CNC(c1cc(Cl)cs1)=O C(=O)(C(F)C(=O)N1CC(CCC(N2CC(OC3(CO)CCC3)C(O)C2)=O)C1)OC c1(CC)c(CSC)cccc1F.c12ccc(nn1)C(c1nnnn1C(C)C)N2 C1(C#N)(CC(=O)NC2CC(C)N(C(=O)CSc3cccc[n+]3[O-])C2)CCOCC1 C1(NC(CCC(C)OCC)=O)CCCCCC1NC(c1n[nH]cc1[N+](=O)[O-])=O c1(C(=O)NC(C2CCOC2)CO)nc(Cl)sc1Cl C1(c2n(CCCC)nnn2)(NCC2CC3(CC3)C2)COCC1n1cncn1 c1(CNC(C(C)OC(CC)(C)C)=O)cc(C(=O)NCC(C)(O)CSC)on1 CCC(C(=O)NCC1(NC(C2CC2COC)=O)CCC1)c1ccccc1 C1(NC(C(C)(C)NC(=O)NCCC)=O)C2CN(C(c3csc(CSC)c3)=O)CC12 c1(C2(OC)CN(C(c3sccc3C3CC3)=O)C2)ccccc1F Cc1c(NC2CCSC(C)(C)C2)ncnc1N(CCCCCO)C C12(C(=O)NCCCOC(=O)NC)CC(CO1)N(C(C1CC3CCCC3C1)=O)C2 C(N=c1[nH]c2c(c(=NC3CCCc4[nH]ccc43)[nH]1)CSC2)C1CC(C)(C)OC1(C)C CC1NC(=O)OC12CN(C(=O)C(c1ccccc1)NC(=O)C(=O)NC1CC1)C2 Nc1cnnc(NNC(=O)NC2CCCSC2)c1Cl c1(C(=O)NCCC(C)N(CCC)C)cc(CNC(C2CC2Cl)=O)on1 N1(C(Cc2c(C)cnn2C)=O)CC2(CC(NC(C3C=CCC3)=O)CO2)C1 C1(OCCN(C(C)C(c2ccccn2)=O)C)CCCCCC1.C(=O)O C1(C(=O)OC)CN(c2nnc(-c3ccccn3)n2CCC#N)C1(C)C Cc1cccc(C(=O)NCC2COCCN2C(=O)Cc2cc(F)cc(F)c2)c1Cl C1(C(=O)Nc2cnc(C)c(Cl)c2)CC2(CCC2)CN1C(C1COCC(C)O1)=O c1(CN2CC(NC(CCCC(C)C)=O)C(C)(C)C2)cccc2c1CCCC2 c1(NC(C2CC(F)CN2C(c2cncs2)=O)=O)cccc(-n2cccc2)c1 c1(NC(C2(C=C)CCC2)=O)ccc(NC(C2CC2C2CC2)=O)c(C)c1 C(CCCCCC(C)C)NC(C(CCOCC)NC(C1CCCC1C1CC1)=O)=O N1(C(Cn2cc(-c3cc(C)c(C)c(C)c3)nn2)=O)CCOC2(CCCCC2)C1 C1(C(=O)NC2(CCO)CCSC2)COc2cc(F)ccc2C1 C1(N(C)C(c2ccc(CC3CC3)o2)=O)CCN(C(N2CCCC2CO)=O)CC1 C1(COC)(NC(c2cnn[nH]2)=O)CCCN(C(=O)CC2CCC2C2CC2)C1 CC(C(O)C(F)F)NC(=O)CC1(CNC(=O)C=CCN2CCC2)CC1 c1(NCC(=O)OCC)nc(C)cc(=NCC(C)c2ccc(F)cc2)[nH]1 C(CC)(c1nccs1)(c1nn[nH]n1)NC(C1CCCO1)C c1(C(C)(C)C)cccc2c1OCC2C(=O)NCc1sccc1S(C)(=O)=O C1(O)(CCNC(C(CCO)N(C)C)=O)CCCN(C(c2cscc2C#N)=O)C1 CC(=O)C(C)(C)CC(=O)NC1CN(C(C2CC3C=CC2C3)=O)CC1CC1CC1 C1(c2n(CC)nnn2)(NCCc2cccc(Cl)c2Cl)CCCN(CCSC)C1 C=C=CCCC(=O)N1CCCC(CNC(N2CCCC2COC(C)(C)C)=O)C1 c1(C(=O)NC2CCCN(C(Cn3nc(C)c(Cl)c3)=O)C2)ccc(F)cc1F O=S(=O)(c1ccc(N2CCC(Cc3ccccc3F)C2)cc1Cl)NCC(O)SC C(CC1CCC1)(C(=O)N(C)CCN1CCCCC1)NC(C(C)N(CC)CC)=O C1(C)(CNC(CCSC)=O)CCCN1C(c1cccc(N2CCCCC2C)n1)=O C1(CNC(COCCC(C)C)=O)(NC(=O)CC2CCCSC2)CC(F)(F)C1 C(=O)(C1=CC(O)CCC1)NCC(CC(F)(F)F)NC(CCc1cccc(OC)c1)=O C1(N(C(C(CC)(C)C)=O)C)CCN(C(=O)CNC(c2cccc(C)c2)=O)CC1C c1(OC)ccc(NC(c2coc(C(C)NC(C3(F)CCCC3)=O)n2)=O)cn1 Cc1[nH]nc2cc(-c3ccn4ncc(C(=O)NC5C=CCCC5)c4c3)ccc12 c1(CC)ncsc1C(=O)NC1CCCC1CNC(c1cc(C2(C)CC2)on1)=O N1(C(c2c(C)nc(C(C)C)s2)=O)CCC(CO)C(NC(c2nn(C)cc2Cl)=O)C1 C1(NC(C(C)C)=O)CCCN(C(=O)C(C)(C)NC(c2cccs2)=O)C1C C(=O)(C(C)(C)C(N)=O)NC(CCNC(C(N1CC(C)C1)C)=O)C(C)C c1(CC(=O)NC2CN(C(CC(C=C)C)=O)C2)ccc([N+](=O)[O-])cc1 c1(NCC(=O)N(c2ccccc2)CCNC(C=CSC)=O)cc(F)cc(Cl)c1 c1(OC)ccccc1CC(C)N(C)C(c1cccc(N2CCOC2=O)c1)=O CCCCC(C)(F)C(=O)N1CCC(NC(C2CCC(C)(C)O2)=O)C(F)C1 C(CCCCN=[N+]=[N-])NC(C1C(NC(C2(CC=C)CCCC2)=O)COC1)=O N1(Cc2c(C)n(C)nc2)CC2(CCCCC2)C1C(C)C C(=O)(C(C(F)(F)F)C(F)(F)F)NCC1OCCN(C(CNC(CNC(C)=O)=O)=O)C1 N1(C(CC(CC)(C)C)=O)C2CCC1CN(C(C13CCC1C3)=O)C2 n1(CCC(=O)NC2CC(CNC(C3C(CC)OCC3)=O)C2)c(C)cc(O)cc1=O N1(c2c(=O)n(CCc3ccccc3)ccn2)CCOC2(CCC2)CC1 CN1CCN(C(c2ccc(=O)oc2)=O)C(CNC(c2cc(C(F)F)cn2C)=O)C1 c1(C(N2CCC(CCOC)(NC(CCC(=O)NC)=O)C2)=O)ccsc1S(C)(=O)=O c1(CC)cnccc1C(N1CCC1(C)C(=O)NC(CC(F)F)c1ccccc1)=O c1(NC(c2ccc(N3CCOCC3)c(F)c2)C)nc2ccccc2c(Cl)c1Br C(=O)(C1CCCc2ccccc21)N1CCC2CCC(NC(c3c(C)coc3)=O)C1C2 c1(C(N)=O)ccc(C(=O)NCCCN(C(=O)COC2CCOC2)C2CC2)cc1Cl c1(C(N2CCCC(C)(NC(c3cnc(C)n3C)=O)C2)=O)cccc(S(C)(=O)=O)c1 c1(N2CC(N(C)C)OCC2)[nH]c(=NC2CCOCC(C(N)=O)C2)nc2sccc12 CCCC(C(=O)N1CCCC1C1CCN(C(c2cnn(C(F)F)c2)=O)C1)OCC CP(C)(=O)C(O)C(=O)NCCN1CCC(NC(=O)CC2CC(F)(F)C2)CC1 c1(C(C)NC(=O)C(C)(N)C2CCCO2)ccc(Cl)cn1 c1(C(=O)NC(CC)(CNC(=O)CC2CCCCCCC2)CC)cnc2[nH]cnc2c1 C1(C(N2CC(CC)SCC2)=O)CN(C)CCN1C(=O)C(N1CCCCC1)C c1(C(N2CC(CC(N3CC(OCC(C(=O)NC)F)C3)=O)C2)=O)cccn(C)c1=O Cc1cc(C(=O)NCCNC(C2CC2C)=O)c(C)n1C1CCCCC1 N1(Cc2ccc(S(N)(=O)=O)nc2)C(=O)C2Cc3ccc(F)cc3N2C1=O c1(C(=O)OC)cccc(CCNc2ccncc2-c2cccc(OC)c2)n1 N1(C(CSCCOC)=O)CC2CC1(C(N1CCC(n3cnnn3)C1)=O)C2 c1(CC(=O)NCC2(CCNC(CSC)=O)CC2)cnc2n1CCOC2 c1(C(N2C(C)CN(C(CC3(CSC)CC3)=O)C(C)C2)=O)cccc(P(C)(C)=O)c1 C1(COC)(NC(=O)CC(C)(C)F)CCCN(C(c2coc(C)c2)=O)C1 N1(C(CCCCCSC)=O)CCC2(NC(C3CC4(CCOC4)C3)=O)CCCCC12 N1(C(=O)OC(C)(C)C)CC2CC2(NCc2snnc2C2CC2)C1 c1(C(N2CC(C(=O)Nc3ncc(Br)cc3CO)C2)=O)ccc2sccc2c1O Cn1cc(NC(C2CC(C)(NC(=O)CSC(F)F)C2)=O)n(C)c1=O C1(C(=O)NC2CC(C(=O)Nc3csc(Cl)n3)C2)CCc2ncnn2C1 C(CC(=O)NC1CC2CC(NC(=O)CCSC3CCCC3)C1C2)(C(C)C)OCC C1(C)(CC)CC(NC(=O)CCC(C)C)CN1C(=O)CNS(=O)(=O)N(C)C N1(C(c2cccc(I)c2)=O)CC2CCC(C1)N2Cc1cccc(Br)c1F N1(C(c2c(C)csc2)=O)CCCCCC1C(=O)N(C)CC1CCOC1 C1(C(N2CC(N(C(C(CC)C#N)=O)C)C2)=O)CS(=O)(=O)CC12CC2 C1(CC(=O)N(CCCNC(c2ccccc2O)=O)C2CC2)CCCCC12CC2 Cc1ccc(Cl)c(N)c1C(N1CCC(NC(=O)C(C)NC=O)C(O)C1)=O CC(O)C(C)(C)C(=O)NC(C1(O)CCCCC1)C(N1CC2CCC(C1)O2)=O N1(C(Cc2snc(C)n2)=O)CCOC(C)(CNC(c2ccc(CN(C)C)[nH]2)=O)C1 N1(C(C(C)(C)Br)=O)CCC(C(=O)Nc2cncc(Cl)c2)C2CC12 C(=O)(C1=COCCC1)NCC1(CCOC)CCN(C(=O)CC2(CO)CC2)C1 C12(CNC(CN3C(C)CCCC3C)=O)CCC(NC(C3CC3F)=O)(CC1)CO2 Cc1nn(C(C)C)c(C)c1C(N1CCN(CCF)CC1)=O c1(C(=O)NC(C)CN2CCN(C(=O)CC3CC=CC3)CC2)ccn2ccnc2c1 S(=O)(=O)(c1csnc1C(F)(F)F)NC(CCNc1c(C)cccc1)=O C(CC1CC1)(C(=O)NCCCN(C(=O)Cc1cnc(C)s1)CC1CCCC1)OC c1(C(N2C(CNC(C3CCC4CCC3O4)=O)COCC2)=O)ccc2sccc2c1 N1(C(CS(CC)=O)=O)CCCC(C)(NC2c3cnn4c3C(CC)CCC42)C1 Cc1cc(F)c(CC(N2CCC3CC3(NC(=O)CN(C)C3CC3)CC2)=O)cc1F Cc1ncc(C(=O)NCC(C)NC(=O)C(c2ccc(F)cc2F)C)cc1N Cc1ccc(C(N2CCC(C(=O)N(C)CC3CCCC3(C)C)(C(C)C)C2)=O)nc1 C(C(C)(C(=O)N(C1CCCCC1)C)NC(=O)CC1CCCO1)SC Cc1ccc(C(N2CCCC(NC(c3c[nH]nc3[N+](=O)[O-])=O)C2)=O)c(N)c1 C(=O)(C1Cc2c(Cl)cccc21)NCC1CCCC(NC(CCCCOC)=O)C1 C(=O)(CC(C)N(C(c1cc(Br)cs1)=O)C1CC1)NCCCOC c1(OC)c(NC(=O)N(c2cccc(OC3CCCC3)c2)C2CCC2)cccc1Cl N1(Cc2c(OC)ccc(OC)n2)CCC2(CCCCN(C(=O)C(C)C3CC3)C2)C1 c1(CC)nc2ccc(Cl)cn2c1C(=O)NCC1(CNC(=O)C2=CCCCC2)CC1 c1(C(N2CC3N(C(C(COC)C)=O)C(CC3)C2)=O)ccc(C)cc1[N+](=O)[O-] C=CCC(C)(C)C(=O)N(CCCNC(c1c[nH]c(C(N)=O)c1)=O)CCC c1(COCC)ccc(C(=O)NC2CC2C)cc1.N12CC3CC1C3C2=O CCC(=O)CCC(=O)NC(CC1CCC1)C(=O)NC1CN(C)CCC1O C1(NC(C(C2CCCC2)OC)=O)CN(C(=O)CCS(C)=O)CC1(C)C Cc1cc(C)cc(C=CC(=O)NCC(=O)NC2C(NC(C3CCC3C)=O)C2)c1 C1(CCNC(c2ccc(C(C)=O)nc2)=O)CCN(C(=O)C(F)=CC2CC2)C(C)C1 c12ccc(cc1)NC(=O)C(=O)N(C)Cc1csc-2n1.c1(C(=O)O)ccccc1 c1(C(N2CC(N(C(c3c(CC)c[nH]c3)=O)C)C2)=O)cc(O)c2ccccc2c1 Cc1nccn1CCNC(=O)CNC(C1CCC(C)O1)=O CCC(CC)CCCN(C(=O)C(Cc1ccoc1)NC(c1ccc(SC)o1)=O)C C1(OC)CCC(C(=O)NC(C)(CO)c2cccs2)CC1 c1(OC)ccccc1C(=O)NCC(O)CC(=O)N(CC(C)(C)CO)C c12c([nH]c(C)c1CC)C(=O)NC1CC2C1(C)C.C(CO)(C1CCC1)OCC N1(C(CC(CC=C)NC(c2nccs2)=O)=O)C2CCC1CC(CCF)C2 c1(CC)cccc(C(=O)CNC(C2CC2F)=O)c1.c12ccc(s1)CS2 Cc1ccc(C=CC(=O)NCC2(CCNC(=O)CCCC#N)CC2)s1 N1(C(C(CC)C(C)O)=O)CCc2nc(CNC(=O)COCCCOC)sc2C1 N1(CC(=O)N(CC(C)(C)CNC(c2cn(CC)nn2)=O)CC)CCS(=O)(=O)CC1 C1(C(N2CCC(CCNC(C(c3ccnn3C)C)=O)C2)=O)C2CCC(=O)C12 C#Cc1ccc(CC(=O)NCC2CN(C(=O)CC3CCCC34CC4)CCO2)cc1 N1(C(CCCOCCC)=O)CCOCC(NC(c2ccc(CO)cc2)=O)C1 C=C(C)C1CN(C(C23CC2CCN3C(c2occc2COC)=O)=O)CCO1 C1(CNC(=O)NCCC(=O)OCCCC)CC(c2cccs2)(OC(C)(C)C)C1 C=CC1(C(=O)N(C2CCCOC2)CC)CCN(C(=O)CC2CCCNC2=O)C1 C1(OC)CN(C(c2c(Br)noc2C2CC2)=O)CC1NC(c1ccoc1)=O CN1CC=C(C(=O)N2CCCC(Cn3cc(CN4CCC(=O)NC4=O)nn3)C2)C1 c1(-n2ncc(C(N(CC(C)NC(C3C(C)C3C)=O)C)=O)n2)ccc(F)cc1 O=S(=O)(c1cc(Cl)cc(Cl)c1)N1CC2CN(Cc3cc(Br)ccc3Br)C2C1 c1(C(=O)NCCCCC2CN(C(CC)=O)C2)cnc(N(C)C)nc1 c1(CC(=O)N(CCCNC(=O)COc2ccc(Cl)cc2)C)ccc(F)c(Cl)c1 N1(c2nccc(N(C)CC)n2)CCc2ccc(C#N)cc2C1 CCS(=O)CC(=O)N1CCC(C(C)(C)NC(c2cncc(C(C)C)c2)=O)C1 c1(OC)cc(C)ccc1C1(C(=O)NC(C)(CNc2cn[nH]c2)C(C)C)CC1 N1(C(c2nn(CC)c(C)c2)=O)CCC(CNC(c2cc(C)c(C)o2)=O)C12CC2 c1(C(=O)NC(CC)CN(C(=O)CCc2csc(=N)[nH]2)C)cn2ccsc2n1 CN1CC(O)CCC1C(N1CCN(C(C23CCC(CC2)CC3)=O)CC1CF)=O C(c1ccccc1Cl)=C(C(=O)NC1CCN(C(C2(CC)CCOCC2)=O)CC1)C C1(C)(NC(C2OCC(C)C2)=O)CCCN(c2ccncn2)C1 c1(C(=O)NCC(=O)NC(CC)(C)CNC(=O)CC2CC2)cncc(N)c1 c1(C(=O)NCCNC(=O)C=CC2CC2)c(-n2cccc2)sc2c1CSC2 N#Cc1cc2c(C(=O)OCc3cnn(C4CCCCO4)n3)nccc2o1 c1(OC)cccc(CC(=O)NCCn2cc(CNC(=O)C3CC3)nn2)c1 n1(C(C(=O)Nc2c(C)ccc(C(N)=O)c2)C)cnc2ccccc12 C1(CC(=O)NC(C2(N(C)C)CC2)C)N(C(c2cccs2)=O)CCC1(C)C N1(C(c2ccn(C)n2)=O)CC(=O)NCC1C(N1CC(=CCO)C1)=O c1(CC)ccc(C(N2CCC(F)(CNC(C3OCCOC3C)=O)CC2)=O)c(F)c1 Cc1ccc(CC(=O)NC2(CCNC(=O)CNC(C3CCCC3)=O)CCC2)cn1 C1(CNC(C(c2ccc(F)cc2)CC)=O)C2CN(C(=O)C(C)(C)CF)CC12 C1(NC(CC(=O)NCC#C)=O)C2CC3C1C3C2C(=O)NOc1cccc(C)c1 c1(SC)ccc(N)cc1C(N1CC2CC(NC(C3(C)CCC(C)(C)C3)=O)C1C2)=O C1(C)(C(=O)NCCC2CCN(C)C2)C=CCN1C(=O)Cc1cccnc1O C12(CCC1)C(=O)N2.C(CC(C)C)OCC(=O)N(C1(CCC)CC1)C c1(C(=O)NC(C)(CNC(CSCC#C)=O)CC)ccc(C)nc1NC C1(C(=O)NC(C2CCCCN2C(=O)COc2cc(C)on2)C)CC2CC1C1CC21 N1(C(C(C=C)O)=O)CCOCC12COCCN(C(C1Cc3nncn3C1)=O)C2 CC(C)CCCCC(c1nnnn1C(C)(C)C)NC1CC(F)C1 c1(C(=O)NCC2(F)CCC(NC(C3CC(C#C)(O)C3)=O)C2)nccc(Cl)c1C N1(C(C2CC(CNC(C3(O)CCOC3)=O)C2)=O)CCCC2(CCC2)C1 N1(C(c2cc[nH]n2)=O)CC2(CCOCC2)CC1CNC(C1CC(CC2CC2)C1)=O c1(CC(=O)N(C(CCNC(C(=O)NCCOC)=O)C)C)ccc(C)cc1Br C=C(CC(=O)N1CCC(N2CCN(C(=O)CCC3CC3)CC2)CC1)C(=O)NC C1(CNC(c2ncn(CCCC)c2)=O)CCCCC1NC(=O)C(c1csc(C)n1)=O N1(C(=O)NC(CC)COC)CC2CC(F)(F)CC2C1 CCC(CSC)(c1nnnn1CC=Cc1ncc[nH]1)NC.C1CCOC1 c1(C(=O)NC(CNC(Cn2ncc(C)c2)=O)CO)noc2c1CC(C)(C)CC2 c1(C(=O)NCC2C=CC(NC(C(C)OCC3CC3)=O)C2)c(C(F)(F)F)ncn1O n1(CCC)cc(Cl)c(C(N2CCCC2CNC(=O)C(C2CC(F)(F)C2)OC)=O)n1 c1(C(N2CCCC(NC(CC3(C)CCC3)=O)C2)=O)ccc2c(c1)COC2(C)C C1(N(CC)CC)CCN(S(=O)(=O)C(C)C)CC1.C1(=O)C(C)O1 C(=O)(C1=CCC(NC(c2c(Cl)cnn2C)=O)C1)NC(CC)C1CC1 N1(C(c2cn(CCC)nn2)=O)CCCC(C(C)NC(=O)CC2SC(=N)NC2=O)C1 C1(NC(c2cccc(C3CC3)c2)=O)CCCCC1NC(C1(F)CC2(CC2)C1)=O N1(C(=O)C2=CCC2)CCCC2(C1)CN(C(=O)C1SCCc3ccccc31)CCO2 CC1CCC(CC(=O)NCCOC2CN(C(=O)CSc3cccs3)C2)CC1C CC(C)(C)C(CC(=O)N1CCOC(CNC(C2(F)CCCCC2)=O)C1)C(F)F C1(C(N2C(CCNC(CC3CCC(C)(C)O3)=O)CCCC2)=O)CC2CCC1CC2 C=CC1CN(C(=O)Cc2cn(C)nn2)CC1NC(c1cc(F)ccc1N)=O c1(C(N2CCS(=O)(=O)C(C)C2)C(=O)NC(CC)C)cc2ncccc2s1 c1(CC(=O)NC2CCCC(N(C(C=C(C)C)=O)C)C2)c[nH]c2cccc(C)c12 c1(C(C(=O)NCCCC2CC2)N(CC=C)C2CC2)cc(Br)ccc1F c1(SCC(=O)NCC(CNC(c2cnc(C)s2)=O)F)ccc(F)cc1 C=CCC(CNC(C1(CC(=O)OC)CC1)=O)NC(=O)CC(C)n1cccn1 C1(CC(N2CC(C(C)NC(C3CC34CCCC4)=O)C2)=O)NC(=O)NC1=O C1(NC(C2CN(C)C2)=O)CCC(CCC(=O)N(CCCN=[N+]=[N-])CCO)C1 C(CCC(O)C(=O)NCc1ccc(CO)cc1)NC(C1(C)CCN(C)C1)=O C(=O)(CC(C)(C)C(F)F)NCCC1CN(C(C2CC3(CC(OC)C3)C2)=O)C1 C=CC1CN(C(C2CC3CC2C3)=O)CCN1C(=O)CCc1ccc(N(C)C)cc1 c1(C(N2C(C)CN(C(C34CCCC3C4)=O)CC2)=O)ccc2nc(CO)[nH]c2c1 C1(NC(c2n(CC)ncc2)=O)CN(C(=O)Cc2nc(C)sc2C)CC(C)(C)C1 N1(C(COC)=O)CCc2ccccc2C(NC(=O)C=Cc2cccc(Cl)c2)C1 c1(C(N2C(C)CC(CC(=O)NCCCN(C)C3CC3)C2)=O)ccc2ccoc2c1 C12(NCCCNC(CN(C)C)=O)CCN(C(=O)CC3CCC3C)CCC1C2 c1(OCCC(N2CCC(C)(NC(CC3ON=C(C)C3)=O)C2)=O)cc(C)cc(C)c1 c1(-c2ccc(CC)cc2)csc(=Nc2cccc(Cl)n2)n1CCc1ccccc1 c1(C(N(CC(O)CNC(C2C(C)C2(F)F)=O)C)=O)cccc2nc(O)n(C)c12 C1(C(=O)NCCN(C)C(C2CCCN2CCCO)=O)CC(C#N)(c2ccccc2)C1 C1(NC(CC2CC(C)N(C(c3cnsn3)=O)C2)=O)CCC([N+](=O)[O-])CC1 Cc1cn2c(C(=O)NCC(C)NC(C3(C#N)CCOCC3)=O)c(Cl)nc2s1 C1(C(=O)NC2CC(NC(=O)C(C3CCOCC3)O)C2)CCCCC(F)(F)C1 C1(COC(c2cc(C)nn2C(C)C)=O)CC2CCCCC12 C1(N(C(C(CC)F)=O)CCO)CCN(C(=O)Cc2ccsc2C)CC1 C1(C(=O)NC(CNC(C2(C(=O)OCC)CCCC2)=O)(C)CO)CCCS(=O)(=O)N1 c1(C(=O)NCCC(C)N(C)C(c2ccc([N+](=O)[O-])[nH]2)=O)c[nH]nc1S(N)(=O)=O Cc1cc(N(C)C(c2ccccc2F)C)ccc1OC(C)C N1(C(CCC2CCCN(C(C3CN(C)C(=O)CC3)=O)C2)=O)CCOCC(F)(F)C1 C(=O)(C(CC(C)SC)N1CCN(Cc2nc(CC)no2)CC1)NCCCC CCC(CN(C)C)C(=O)N1CCC(C)C1C(=O)NCCOCC1CC1 NC1CCCN(C(=O)NCCCNC(C2CCCCC2)=O)C1 C1(n2c(C3(C)CCN(c4ccccc4)C3)nc(C(CC)O)n2)CCC(F)(F)CC1 c1(OC)c(CC(N2CC(c3cc(C)ccc3OCC)C2)=O)cccc1F Cc1sncc1C(=O)NC(C)C(C)NC(c1cnc(S)nc1)=O C1(NC(CCOCC(C)(C)C)=O)C=CCN(C(=O)Cc2cccc(Cl)c2)C1 N1(C(CC(C)OC)=O)CCN(C(=O)C(=Cc2cccn2C)F)CC1C1CCCC1 N1(C(C2C(NC(C3(C)CC4CC4C3)=O)CCCC2)=O)CC(CO)C(O)C1 Cc1cc(C(N2CCN(C3CN(C(=O)C4=COCCC4)C3)CC2)=O)cc(N)c1Cl CC1(C)CCOC(C(=O)NC2C(C(=O)NOCC3(C)CCCCC3)C2(C)C)C1 C1(NC(c2cc3occc3s2)=O)CCN(C(=O)CCCC2CCC2)CC1F N1(C(c2ncc(CC)cn2)=O)CCCC2CN(C(=O)CC(C)C(C)(C)C)CCC12 C=Cc1ccc(C(=O)N(C2CN(C(C3(C#N)CCOC3)=O)CC23CC3)C)cc1 C1(C(=O)NCC(C2CC2)NC(c2cnn(CC(F)F)n2)=O)CCCCS1(=O)=O c1(N2CC(C)N(Cc3cccn3C)CC2)ncnc2c1CCC2 C12CC(F)(F)CN1C(c1c(Br)ncn1C)C(=O)N2.CN1CCC(N(C)C)C1=O C(=O)(C1=CCCC1C)N1CCC(N2CCC(NC(C=C(C)C(C)C)=O)CC2)C1 N1(C(C2(C(=O)OC)C(=C)CC2)=O)CCCN(C(=O)CCCSC)CC1 C(=O)(C1CCCc2nncn21)N(CCC(C(C)C)NC(=O)C=CCF)C C12(C(=O)NCCC(C)(C)OCC)CC(CN1C(C1CCCCN1CC)=O)C2 S(=O)(=O)(c1cc(C(N2CC3CC2CCC3C(=O)N(C)C)=O)n(C)c1)NC C(=O)(C1SCc2cccnc21)NC(C)CNC(c1cc(CO)ccc1Cl)=O C1(CC=C)(C(=O)NCCN(C(C)C)C(C)C)CCCN1C(C1C=CCC1)=O C1(CNC(c2n(CC)cc(Cl)c2)=O)CCCC2CN(C(=O)C#CC(C)(C)O)CC12 C#Cc1ccc(C(=O)NC2CC3CC(NC(C4(C)CCCO4)=O)CC3C2)c(C)c1 c1(C(N2CCC3C(O)CC23)C(=O)NCCSC)ccc2c(c1Cl)OCCO2 n1(CC)c(=O)c2ccccc2n2c(Sc3cc(C(F)(F)F)n(C)n3)nnc12 CCC(C(=O)NCC(C)(C1CC1)NC(=O)CC(O)C1CCCC1)C(C)(C)CC C12(CC(=O)N(CC(C)C)C)COC(C(F)(F)F)(C1)C2.c1(C=O)ccc[nH]1 c1(C(=O)NCc2c(OC)cco2)ccc2c(=O)c3ccc(Cl)cc3[nH]c2n1 C1(C(C)(C)C)Cc2occ(C(=O)NCC34CC(C3)C(C(F)(F)F)O4)c2C1 N1(CCN(C)C)CCN(C(=O)C(=O)NCc2cccc(Cl)c2)CC1 c1(C(=O)NCC(N(C(=O)CCc2ccncn2)C)C2CC2)coc2c1C(O)CCC2 c1(OCC)cc(C=CC(=O)NC2CCCCC2NC(=O)CC2CC2)ccc1O C(C(C(C)C(C)C)NC(=O)CN1CCCC1=O)NC(c1c(SC)n(C)nc1)=O C1(CNC(C(CCC)(C)O)=O)CC2CCC(C1)N2C(C1CCCCC1O)=O Cc1cccc(CCNC(C2(C)CN(C(c3ncccc3N)=O)C2)=O)n1 c1(NC(=O)C(=O)N(c2cnn(C)c2C)CCCC)ccc(N(C)C)cc1F N1(C(Cn2cc(C(C)O)nn2)=O)CCCC(CCNC(c2cc(Cl)cnn2)=O)C1 CCS(=O)(=O)c1ccc(CN2CC(O)(CNC(=O)C(C)NC(=O)OC)C2)cc1 CCC(C)C(O)C(C)C(=O)NCC(F)(C(=O)NCc1nncn1C1CC1)C(C)C C(C(C)(C)CCS(C)(=O)=O)NC(c1n(CCCCCC)nnn1)c1cccnn1 C(=O)(C(C)S(=O)(=O)CCC)NC(CC1CCN(C(C=CC=CCC)=O)CC1)C N1(C(C(C)NC(=O)CCCCC2CC2)=O)CCCC12CCCOC2 C1(C(N(C(C)C(=O)N(CC(O)C2CCC2)C)C2CC2)=O)CCCCNC1=O N1(C(C(c2cnc[nH]2)N(CCC)CCC)=O)CCC(N(C2CCC2)C)C1 C(C(C)(C)C(=O)NCCC1CCCCN1C(=O)CC1(C#N)CC1)OC C(CCCCCC(=O)N(C1CCN(C)C1=O)C)NC(C1(C)CC(C)C1)=O C(=O)(C(=O)CC(C)CC)N(CC(=O)N(CC)Cc1cccc(Cl)c1)CC#C c1(C(=O)NCC2C(NC(c3cnc(CC)o3)=O)CCC2)cnc(OC(F)F)c(F)c1 C1(C(=O)NC(c2ccc(Br)c(Cl)c2)(C)C)NC(=O)C2CCC12 CC1(C)CN(C(=O)C=Cc2cncs2)CCC1NC(=O)CC1CC2CC2C1 Nc1c(C(=O)NCCC2CCCN2C(=O)Cc2ccsn2)cc(F)cc1[N+](=O)[O-] Cc1ccc(Cl)c(C(=O)NCC2CCC2NC(c2cc(C3CCC3)nn2C)=O)c1 Nc1c(Cl)cc(C(N2CCCC2CN(C(C2CCCCO2)=O)C2CC2)=O)cc1Cl N1(C(C2(OC)CCC2)=O)CCC(C(=O)NC2C(C)CCC2C)CC1(C)C C1(C)(NC(c2ccc(C)n2C)=O)CCCN(C(C2CCCCN2C)=O)C1 c1(C(=O)NCCN(C(C2(C)CCCS2)=O)C2CC2)cccc(OCC(F)F)c1 N1(C(C2(C#N)CCCOC2)=O)CCC(C2(NC(C3CCC4CC4C3)=O)CC2)CC1 C1(NC(=O)CSc2cccc(F)c2)CC2CCC1N2C(=O)CC1CCC=CCC1 CC1(C(N)=O)CCCN(N2CC(Cc3ccc(C(F)(F)F)cc3)C2)C1 CCC(CNC(c1cc(C2CC2)no1)=O)(CC)C(=O)N1CCC(C)(C)CC1 Cc1cc(N)c(C(=O)NCCCNC(=O)Cc2occc2C)cc1C C1(CNC(c2cc(C(C)=O)on2)=O)CN(C(C2CC3(CCC3)CO2)=O)C(C)(C)C1 c1(C(=O)NCCCN(C(c2cc(-c3ccco3)on2)=O)CC)cc2n(n1)CCC2 C1(C(=O)NC(C)Cc2ccncc2)CC=CCN1C(c1scnc1Cl)=O N1(C(CC2(N(C(C(CC3CC3)OC)=O)C)CC2)=O)CC(=O)NC(C)C1 c1(CNC(C(C)OCC2CC2)=O)cccc2c1CCN(C(c1sccc1F)=O)C2 C1(O)(C(C)NC(C(C)OCCCC)=O)CCN(C(=O)C(C)=C2CCC2)CC1 c1(CN(C(C)C)CC2(C)CC2)cn(CCCO)nn1 N1(CC(=O)NCC(C)NC(C(CC2CCCC2)OC)=O)C(=O)CCC1=O N1(C(CSCCCC)=O)CCCC1CCNC(=O)CC1CC(F)C1 c1(SC)cc(C(=O)N(CCCCNC(c2[nH]cnc2C#N)=O)C)oc1C C(=O)(C(C)CC(C)(C)C)NCCC1N(C(c2sc(C)c(O)n2)=O)CCCC1 c1(N2C(=O)CC(NC(N(c3cccc(C(F)(F)F)c3)CC)=O)C2)cnccc1C#N CC1CCN(CC(=O)NCC2CCC(C(=O)NC(c3ccoc3)C)C2)C1 C1(C)(NC(c2cc(CNC(c3c(C)cn(C)c3)=O)sc2)=O)CC(C)(C)OC1=O c1(NC(CSCC(=O)NCC(C)NC(C2CCC(C)(C)O2)=O)=O)ccc(F)cc1 c1(OC)ccnc(F)c1C(=O)NCC1CC(NC(C2CC(C)OC2=O)=O)C1 C(CC(=O)N(CC(C)(C)C)CC1CC1)N(C(=O)CC1CC1(C)C)C c1(C(C)C)ccc(C(N2CC(NC(C3(C4CCCO4)CC3)=O)C(C)C2)=O)c(O)n1 C(CC(CNC(c1snnc1C(C)C)=O)NC(=O)CCc1cscn1)OC CC1CCC2(CO1)CN(C(C1(CNC(=O)CC3CCCC3)CC=CC1)=O)C2 N1(C(c2cc(OC)nn2C)C(=O)NC2CC2)CCC2(CCN(C)C2=O)C1 c1(C(N2C(COC(CC=C)C(=O)NCC)CCCC2)=O)c(Cl)ccc(OC)c1N Cc1ccc(C(C)(C)CC(=O)N2CCCC(C(N3CC(O)C3)=O)C2)cc1 N1(C(c2onc(C)c2C)=O)CCc2sccc2C1CNC(C1CCC(O)CC1)=O c1(C(=O)NCC2CCN(C(c3ccc(OC)s3)=O)C2)cc2c(Cl)cncc2s1 Cc1cc(C(=O)NC2CCC(NC(=O)C=CCO)C2)c(C)n1NC(N)=O c1(CNc2nccc(N3C4C(CO)C(CCC4)C3)n2)cnc2ccnn2c1 C1(NC(C2(CC(C)=O)CC2)=O)COCC1NC(c1cc(-c2ccccc2)[nH]n1)=O c1(C(=O)NC2CCCN(C(C(CC)CC)=O)CC2)ccccc1S(C)=O C1(NC(C(CC)CC)=O)CN(C(=O)C(F)(F)C(O)CC)CCC1(C)C Cc1ncc(Br)cc1C(=O)NCC1CC1NC(=O)Cc1ccc(C(F)F)o1 C(=O)(CC(C)C(C)C)NC(C1OCCN(C(c2c(C)cn(C)c2)=O)C1)C c1(NC(=O)NCC2C(C(=O)OCC)OCC2)cnn2cccnc12 Cc1cncc(C(=O)NCC2CC2NC(c2cn(CC(F)(F)F)nc2C)=O)c1 c1(C(=O)NC2CCCC2)nnn2c1CCCC2.C123CC(C1)(C2)NC(=O)CN(C)C3=O c1(C(=O)NCCOC(C)(C)CNC(C2(F)CC=CCC2)=O)cccc2occc12 CC(C(O)C(F)F)NC(=O)COC1CN(C(C2(C)COC(=O)N2)=O)C1 C1(C(N(C(C)C(=O)OC)CC#C)=O)CCN(C(=O)CC)CC1.C(C)(=O)O CCCCN(CCCNC(=O)N(C1(CC(C)C)CC1)C)CCC CC1(C(=O)NC2(CCO)CCC2)CCN(C(=O)C(CO)NC2CC2)CC1 c1(SCC)cccc(C(N2CC(C(N)=O)(CNC(c3ccccc3C)=O)C2)=O)c1 C1(F)(CNC(CC(C=C)C)=O)CCN(C(=O)Cn2cc(C(=O)NC)nn2)C1 Nc1c(Cl)cc(C(N2CCC(Oc3cc(Cl)ccn3)CC2)=O)cc1Cl C(=O)(CC1NC(=O)c2ccccc21)NC(C)CC1CN(C(c2cc(F)c[nH]2)=O)C1 C1(F)(CNC(C(C2CC2)OC)=O)CCCN(C(=O)CC2CCC(C)O2)C1 c1(C(C)C(=O)N(C(C)CCNC(C2C=CCCC2)=O)C)ccccc1F c1(N2C(=O)CC(C(=O)NCCNC(C3(C)CC=CCC3)=O)C2)ccc(F)c(F)c1 Cc1[nH]c(C#N)cc1C(=O)N(C1CC1C(=O)NCCOCCO)C1CC1 CCC(C)C(C(=O)NCc1cc[nH]c1C(N1CCCCC1CC(N)=O)=O)N(C)C C(C(CC(C)C)C(=O)N1CCOC(C(C)C)C1)NC(c1cccc(C)c1N)=O c1(C(=O)NC2CN(C(C3CCC(CC)O3)=O)CC23CC3)c(F)cc(Cl)cc1F CC1OCCC1CC(=O)NCC(C)(C)CN(C(=O)Cc1nccn1C)C1CC1 c1(C2C(C(N(CCN(C(=O)CCC=CBr)C(C)C)C)=O)C2)ccc(F)cc1 N1(C(=O)Oc2onc(CNC(=O)OC(C)(C)C)n2)CC2(CC=CC2)C1C(F)(F)F N1(C(C=CC(C)C)=O)CC(C(=O)N(C2CC(C)CC(C)C2)C)C(C2CC2)C1 CCCCC(CNC(C1CCCN1CCOC)=O)NC(c1cc(Cl)cn1C)=O c1(C(=O)NC2CCN(C(CC(C)(F)F)=O)C2)cnc2ccc(Cl)cn2c1=O CC(CC(F)F)C(=O)NCC1CN(CC(=O)NCc2ccc(SC(F)(F)F)o2)C1 C1(C(=O)NCc2cccc(NC(C(=O)NC3CC3)=O)c2)CCCCC12CC2(F)F c1(C(=O)NC2CCC(NC(CC(C)CF)=O)C2)cnc2c(c1)CCCO2 Cn1nc2cccc(S(=O)(=O)OC(F)F)c2n1.c12ccc(cc1)CC(=O)OC2 C1(COC)(CNC(=O)C=CCO)CCCN1C(=O)CCc1cnn(C)n1 c1(OC)cc(=NC(=O)C2(NC(c3cccc(F)c3N)=O)CCC(C)(C)C2)[nH]n1C c1(C(=O)NCC#CCNC(=O)C=CC2CCOCC2)c(Cl)ccc2c1OCO2 c1(C(=O)NCC23CCC(CC2)N3C(C2(O)CCSC2)=O)cccc(F)c1F N1(C(CC2C(C)=NNC2=O)=O)CCC(N=[N+]=[N-])(C(=O)NC(c2cnsc2)C)C1 C(C(=O)N(CCNC(C1(C(F)(F)F)CCCCO1)=O)CC)(C(C)C)SCC CC1(CNC(C2CSCN2C(c2cnncc2O)=O)=O)CCOCC1 CC1(C)CCOC1CC(=O)NC1CCCCC1CC(c1ccccc1)=O Cc1nn2cc(C(=O)NCCC3CCCN3c3nnc(C(C)C)o3)nc2s1 C(=O)(C(C)(C)Cc1ccccc1)NC1CCC(n2cc(CCN(C)C)nn2)CC1 c1(CCC(=O)NC(CC)CNC(=O)CCCNC(=O)C2CC2)ccc(C)c(Cl)c1 C1(C2CCC2)(C(=O)NCC2(O)CN(C(CSCC(C)C)=O)C2)CC1(F)F Cc1c[nH]nc1CNC(=O)C(F)C1CC(NC(=O)CC2CC(N(C)C)C2)C1 Cc1cc(C(=O)NC(C)C(=O)NCC(C)NC(c2cc(Cl)ccc2F)=O)cc(C)c1 C(=O)(CC(C)(C)C(F)F)NCCCC1(NC(CCN(C(CCC)C)C)=O)CC1 C1(CCCNC(c2cc[nH]n2)=O)CCCN(C(=O)C(c2ccc(Cl)cc2)O)C1 CCN=C(NCCC(C)(C)C1CC1)N(C)CCN(C)C c1(C(=O)NC2CC(C)CN(C(c3c[nH]nc3C3CC3)=O)C2)cc2cnccc2[nH]1 c1(OCC(=O)NCCC(C)NC(C2CCOC2)=O)ccc(F)cc1Br c1(C(N(C2CCC(NC(=O)CCN3CCCC3=O)C2)C)=O)cnc2[nH]ccc2n1 c1(C(N(CCN(CC(C)C)C(C2CC2CC(C)(C)C)=O)C)=O)cc2sccc2s1 CC1OC2(C(=O)NCc3ccc(CN(C)C(C4CCCC4)=O)cc3)CCC1CC2 CC(C)CC(F)C(=O)NC(C)CN(C)C(c1cc(OC(F)(F)F)cc(F)c1)=O c1(N(C)Cc2ccccc2Cl)[nH]c(=NCC(C)CN2CCCC2)nc2sccc12 N1(c2ccc(C(N3CCN(C(CCS(C)=O)=O)CC3)=O)cc2)CCS(=O)(=O)CC1 c1(OC)cc(C(N2CC(C(=O)NCc3ccc(Cl)nc3)C2)=O)cc(C(F)(F)F)c1 CC(CCC(=O)Nc1ccc(C(=O)CNC(N)=O)cc1)c1ccc(Br)cc1 c1(N(C)Cc2ccc(C)o2)nc(=NC2CSC(C)C2)[nH]c2c1CCC2 C1(NC(=O)CC2CC2)CCC(C(=O)Nc2c[nH]nc2C(N)=O)OC1 N1(C(c2c(SC)nccn2)=O)CCC(C)(C)C(CNC(c2ccccc2)=O)C1 C1(NC(c2cc(C)ns2)=O)C=CCC(C(=O)NC(c2cncnc2)C)C1 C1(C(C)NC(C2(CC#C)CCC2)=O)CCN(C(=O)CO)CC1 C1(NC(C#C)=O)CCCN(C(CCC)C(=O)N2CCOCC2)C1=O CC(C)CS(=O)(=O)NC(=O)CCc1cc(CO)on1 Cc1cncc(-c2cn(CC3CCCN(C(C4CCC4)=O)C3)nn2)c1 C1(NC(CC2CC(OC)C2)=O)CCN(C(c2ccoc2C(C)C)=O)C(C)C1 CC1C(C(=O)NCCCC2CCC2)CCN1C(=O)CCc1ncccn1 C1(=CC(=O)N(C(C)CNC(=O)C(O)P(C)(C)=O)CC)CN2CCC1CC2 C(=O)(C#CC1CCCC1)N(CCNC(c1nn(-c2ccccc2)cc1O)=O)CC C1(CC(=O)NCc2csc(Br)c2)CCCCN1C(=O)C=Cc1cn[nH]c1 c1(C(C)(F)F)ccc(F)c(CN2CCCC(CN)C2)c1 C1(CCC)CN(C(c2c(SC)cnn2C)=O)CCN1C(=O)Cc1csc(Cl)n1 CC1(C)CCc2onc(C(=O)NCC(C3CC3)NC(=O)C(F)CC3CC3)c2C1 c1(C(=O)NC2CC(F)(CNC(C(CC)N(C)C)=O)C2)c[nH]c2nccc-2c1 c1(C(=O)NCC(CC)NC(=O)CC2CC2C2CC2)ccc(-n2cnnn2)cc1 C1(C(=O)NC(C)(C)CNC(C2(Cl)CC2(F)F)=O)C2CN(C(=O)OC(C)(C)C)CC12 S(=O)(=O)(c1csc(C(=O)NCC2CCN2C(c2ccc(F)cc2N)=O)c1)NC C(=O)(C1CCCc2ccccc21)N1C(CNC(=O)C(c2ccc(F)cc2)O)CC1 N1(c2n(CC(C)C)c(Cc3cnc4n3CCC4)nn2)CCC2(CC1)CCS2(=O)=O c1(OCC)ccc(CCCC(=O)NC(C)CN(C)C(c2ocnc2CC)=O)cc1 c1(CNC(C2C3CCC(F)(F)C32)c2nc(C3CC3)no2)cnc2cc[nH]c2c1 N1(C(c2ccncc2O)=O)CC(C2CN(C(C3(Cl)CC3)=O)C2)C1 N1(C(CC(C)F)=O)CCC(C)(NC(=O)COCC(C)(C)C)C1 N1(C(=O)CSc2nc[nH]n2)CC2(C1)CN(C(C13CCC(F)(CC1)CC3)=O)CCO2 N1(C(CCc2ccc(C)nc2)=O)CC2CCC2(CC(=O)NCCCCN(C)C)C1 c1(CN(CC(=O)NC2CCC(CNC(C3C=C(C)CS3)=O)C2)C)cccc(Cl)c1 c1(C(N2CCC(CCNC(=O)C(F)C(F)(F)F)C2)=O)nnn2c1CCCCC2 c1(C(=O)NC(CNC(c2n(CC)ccn2)=O)C(C)C)ccc2c(c1)COCCN2 Cn1cnc(C#N)c1C(N1CCN(CCc2cn(C3CCOC3)nn2)CC1)=O CC(C)CCC(=O)Nc1ccc(-c2nccc(COCC3CCCO3)c2)cc1 CCC(C)(F)C(=O)N1CCC(C(C)(C)C)(CNC(=O)Cn2ccnc2C(C)C)C1 c1(C(N2CC3C(NC(c4scnc4Cl)=O)C3C2)=O)nnn2c1CCCC2 C1(NC(c2[nH]cc(C)c2)=O)C(C)CN(C(=O)CNC(=O)CN(C)C)CC1C c1(C(=O)NC2CC(CNC(C(C)SCCCC)=O)C2)cnn(CC(F)(F)F)c1 CC1CCN(C(C2COCCN2C=O)=O)CC1CNC(=O)CSc1nc[nH]n1 c1(C(=O)NC2CC(C)(CNC(C3CC34CCCC4)=O)C2)cc(C#N)cn1C C1(CNC(C=C(COC)C)=O)COC(CNC(c2c[nH]nc2Br)=O)C1 CCCCC(CC)(c1nnnn1C(C)(C)C)NCC(C)Oc1ccc(C)cc1 c1(CC)nnc2n1CCCC2C(=O)N1CCC(N(C(=O)COC2CCC2)CC)C1 N1(C(C2(C#C)CCN(C(c3cc(CO)ccn3)=O)C2)=O)CC(C)(C)C12CCC2 C(C(N=c1nc(C2CCOCC2)[nH]s1)C1CC1)NC(c1ccn2ccnc2n1)=O c1(CN(CCNC(=O)NC2CCCN2C)CC)ccccc1C C1(C)(C(=O)NCCC2CC(NC(C3N(CC)CC3)=O)C2)CCN(C)C1 Cc1c(Br)noc1C(=O)NCC1C=CCN1C(C1CC1c1ccccn1)=O CC12CCC(CC(C)(C)O1)C(NCC1CCCC(C(=O)OC(C)(C)C)C1(C)C)C2 c1(CNC(N(C)Cc2noc(C(F)F)n2)=O)cnn2cc(F)cc(F)c12 c1(C(N2CC(NC(CC3CC(OC)C3)=O)C(O)C2)=O)sc(Cl)c(Cl)c1C O=C1COc2c(C(N3CCSC4CCCCC34)=O)cccc2N1 C(c1c(C)coc1C)=CC(=O)NCC(CCOC)NC(=O)COCC(C)CC c1(C(=O)Nc2cccc(F)c2C(=O)NCc2ccco2)cnc2n1CCCC2 C1(=O)C#CC2(CC2)NCCN1.c1(C(=O)NCCC(=O)NC2CCC2)ccc(O)cc1 C1(CC)CN(C(N2CCN(CCC(=O)Nc3cnccc3Cl)CC2)=O)CCN1C c1(C(N(CCCOC(CCN(C)C)C)C)=O)ccnc(OC(F)(F)F)c1 N1(CCC)CCCC1C(=O)N(C1CCN(C(c2scnc2C(F)F)=O)C1)CC N1(C(c2cccc(C(C)=O)c2)=O)CCCC2CN(C(=O)CC=C(Cl)Cl)CCC12 C12(CNC(CC=C)=O)CC(NC(C3CCC3C)=O)(CO1)C2 O=C(C1=NOC2(CCN(Cc3ccc(F)nc3)C2)C1)NCc1cc(O)ccc1Br c1(C(=O)NCCCCC2CN(C(C=C(C)C)=O)C2)cnc2c(c1)OCC(=O)N2 CC1(NC(=O)COC(F)F)CCN(C(C2CC2c2cccc(OC(F)F)c2)=O)C1 c1(C(N2CC(NC(Cc3cc(C)[nH]n3)=O)C3C2C3)=O)cnc2cc[nH]c2c1 N1(C(C2(COC)CC2)=O)CC(C2CCCN(C(c3cccc4c3CCN4)=O)C2)C1 N1(C(CCOCC=CC(=O)NCCOC)=O)CC(NC(CC)=O)CC1(C)CC C12(C(N3CCC4(NC(CN(C(C)=O)C)=O)C(C3)C4)=O)C3CCC(CC13)C2(F)F Cc1cc(C(=O)N(C2CCN(C(C3NC(=O)CC3C)=O)CC2)CC2CC2)ccn1 C#Cc1cccc(C(=O)NCCCC(C)NC(C2OCCC2(C)C)=O)c1F c1(CC)ccccc1C(=O)NC1C(C(N2CCCC(c3cn[nH]c3)C2)=O)CC1 C(=O)(C1Cc2ccccc21)N1CCC(CNC(C(C)CF)=O)C12CCC2 C1(C(=O)NC2CN(C(C3(CC(C)C)COC3)=O)CC(C)C2)CCc2nccn2C1 Cc1c(C(=O)NC(C)CN(C(=O)C(C)CF)C)nnn1Cc1ccncc1 Cc1cc(-c2c(C=CCNC(C3CC(CN4CCC4)C3)=O)cccc2)ccc1F C(=O)(C(F)C(=O)N(C)C)NCCOCCNC(C1(CC=C)CC1)=O Cc1cc(OCC(=O)NCC2COCC2NC(C2CS(=O)C2)=O)c(C)c(C)c1 c1(OC)cc(C(N2CCCN(CC(c3ccccc3)O)CC2)=O)cc(Br)c1O C1(CNC(c2cscc2C(F)(F)F)=O)CC(F)(F)CN1C(C1C2CCCC12)=O C1(CCC)CN(C(=O)CC2CCC(C#N)C2)CC1C(=O)NCC(COC)OC Cc1cc2cccc(CN3CCOCC3c3nnnn3C)c2o1 c1(N2CC3CC(N(C)C)C3C2)ncnc(NC(=O)C2=CC3CCCC23)c1[N+](=O)[O-] C(=O)(C1=CC2C=CC1C2)N1CCC(CC(N2CCC(CC#C)C2)=O)C1(C)C c1(C(N2CC=CC2CN(C(C23CCCN(CC2)C3)=O)C2CC2)=O)nccc2ccsc12 C1(CNC(C2CC(=C)C2)=O)C(C)CCN1C(c1c(OC)nsc1OC)=O C1(NC(=O)NCC(=C)Br)CC(=O)N(C2CCCCCC2)C1 N1(C(CC2CN(C(c3c(C)ocn3)=O)CC2C)=O)CCCCCC1C C1(NC(c2cnc(C(C)C)s2)=O)CCCC(NC(=O)C(C)(C)C2CC2)C1 C12(C(C)C)CCCN1C(=O)N2.C1(CC(C)(C)C)CCC(C(F)(F)F)CC1 C(Cc1ccccc1)(CCSC)NC(CN(CC)CC)=O.C(c1nccs1)=CC=O C=C(CNC(N1CCN(C(n2cncn2)=O)CC1)=O)c1ccccc1 N1(C(C(CSC)(C)C)=O)CCC(C)C(NC(=O)CN2CCOCC2=O)C1 C1(CCNC(C(CC)C2CCC2)=O)CC(F)(F)CN1C(c1cc(F)ccc1Cl)=O c1(-c2cc(OC)c(O)cc2)nnc2n1CCN(Cc1cc(C)c(Br)cc1C)C2 c1(NC(C)=O)ccc(C(N2CC(NC(C3CCC(F)CC3)=O)CC(C)C2)=O)c(Cl)c1 c1(C(=O)NC2CC(NC(c3cnncc3Cl)=O)C2)ccc2c(c1)OCCCO2 c1(C(CC)NC(=O)Cn2cc(CNC(=O)Cn3nccn3)nn2)ncnn1C c1(CC(C)C)ccccc1Sc1ccc(CNCC(C)C#N)nc1 CCC(C)CC(C(=O)NC1CCN(CCO)C(=O)C1)NC(=O)CSC c1(C(=O)NC2CCN(C(C3(C(F)(F)F)CC3)=O)C2)ccc2c(c1)C(=O)CC2 c1(NCC2CC(CNC(=O)Cc3cccc(Br)c3)CC2O)ncnc2c1CCC2 C1(NC(=O)CC2CCC(=O)N2)C2CCC1N(C(=O)Cc1cn3ccsc3n1)C2 c1ccc(S(=O)(=O)N2CCCC(CN)C2)s1.N1(C=O)CCOC(=O)C1 c1(C(N(CCNC(C2CCC(CCCC)CC2)=O)CC)=O)ccc(F)c(O)c1F c1(C(N(CCN(C(C(C2CC2)OC)=O)C)C)=O)c(C)cc(Cl)cc1N c1(C(=O)NC2CN(C(C3ON=C(C(C)C)C3)=O)CC23CC3)cnn2c1OCCC2 c1(C(=O)NC(C(=O)NCC(C)CC2CC2)Cn2ccnn2)ccc(O)cn1 C1(C(=O)NC2CN(C(C3CC3[N+](=O)[O-])=O)C2)(CNC(=O)NC2CC2)CCCCC1 C1(C(=O)NCC2CC(NC(c3c(N)sc(C)c3C)=O)C2)CC(C(C)(C)C)=NO1 C1(CNC(C(=O)NCCn2c(C)nc(C)n2)=O)OCCOC1(C)C N1(C(C2CCCS2(=O)=O)=O)CCN(C(=O)CCc2ccc(O)nc2)C2CCCC12 c1(CC)ccc(C#N)cc1F.c12cccc(c1)CNC(=O)C1CC(O)CN1C2=O Cn1ncc2c(CN3CCSCC3C(=O)NCc3cnc[nH]3)cccc12 N1(C(c2ncc(C)s2)=O)CCCC1(C)CNC(=O)Cc1ccccc1Br CCN=c1ccc(C(=O)NC2CCC2NC(c2ccsc2C(F)(F)F)=O)c[nH]1 C1(C(N(C2(c3cn(-c4ccncc4Cl)nn3)CCC2)C)=O)CCCN1C=O CC1CC2CN(C(c3ccc(CO)s3)=O)CC2N1C(C1(C(F)F)CCC1)=O c1(C(N2C3C(NC(c4c(C(N)=O)nccn4)=O)C(C3)C2)=O)csc2c1CCCC2 N1(C(C=CC=CC)=O)CCOC2(CCS(=O)(=NC(=O)CC3(C)CC(C)C3)CC2)C1 N1(C(CC2C(C)(C)C(=O)C2)=O)CC(C(=O)NCC(N2CCOCC2)=O)C(F)(F)C1 c1(C(=O)NC2CC3CC(NC(C4(OCC)CCC4)=O)C2C3)cc2scc(Cl)c2[nH]1 CC(CF)CC(=O)N(CCNC(=O)C(F)=CCCF)CCc1ccccc1 CC1CCS(=O)(=O)CCN1C(=O)CCNC(c1ccc2ccccc2c1)=O C12(CNC(CCOCCC)=O)CN(C(c3cnn(C)c3)=O)CC1CCO2 c1(CNC(N)=O)ccc(C(=O)NC2CCCCN(C(=O)C(O)CF)C2)cc1 CCC(CC)CC(=O)NC1CCCCC1C(=O)NCCN1CCCC(O)C1 N1(C(COC(CC)CC)=O)CCC(C(=O)NON2CC(C)(C)C2CC)C1C c1(C(N2C3(CNC(C(CCC)OCC)=O)CCC2CC3)=O)cccc2c1CCO2 Cc1nc(NC(=O)NCC2CCC(=O)NC2)sc1F C1(NC(C2=C(C)OCCC2)=O)C2CCCC1CC(NC(c1ccncc1C)=O)C2 CC1(O)CCN(C(C2C3CCCCC23)C(=O)NCCC2CC2)CC1O CC1CC(C(N2CCC(CCCNC(=O)C#CC(=O)N(C)C)CC2)=O)CC(C)O1 c1(C(N2C(CNC(C(C)C)=O)CC(F)C2)=O)cccc(S(C)(=O)=O)c1F C1(C(C)N(C(=O)C=CI)C2CC2)CN(C(c2ccnc(OC3CCC3)c2)=O)CCO1 N1(C(C=CCN(C)CC)=O)C(CNC(c2ncccc2C)=O)CC2CCCC12 CC1(C)CC=C(C(=O)N2CC(CNC(c3ccc([N+](=O)[O-])cc3F)=O)C2)CC1 c1(SC)cc(F)ccc1C.Cc1cc(CC(=O)NO)on1.c12ncoc1c2=O N1(C(CCc2cc(C)[nH]n2)=O)CC2(C=C(C(=O)N3CCOCC(C)C3)CO2)C1 N1(C(C2(Cl)C(C)(C)C2)=O)CCCC(CCNC(=O)C2=CCC2)CC1 c1(C(=O)NC2C(NC(c3cc(CC(C)C)nc(O)c3)=O)C2)nccn2cnnc12 c1(C(=O)NC(C)C(C)C(=O)NC2CCC3(CC3)C2)ccn(C)c(=O)c1 c1(OC)ccnc(C(=O)NCC23CC2CN(C(C2CCC(F)(F)CC2)=O)C3)c1O CCCCC(C(=O)OCC)N1CC(NC(C2CCN(CC)C2=O)=O)C1 C(=O)(C1=CC2(CCOC2)C1)NC1CN(C(CC2C(C)=NOC2=O)=O)CC(O)CC1 C(c1ccccc1)=C(C(=O)NC(C1CCOC1)CNC(CN(C)C1CC1)=O)C#N C(=O)(C(C#N)C(C)(C)C)N(CCC)CCNC(c1ccc(C(C)(C)C)[nH]1)=O C1(C)(CC)CCC(NC(c2ccc(-c3ccccc3Cl)o2)=O)CC1 Cc1nnccc1C(=O)NC(CN(C)Cc1ccccc1)C(=O)NCCN=[N+]=[N-] C(=O)(C(C)C(O)C(C)C)NCC(CC(C)C)NC(c1ccn(C(C)C)c(=O)c1)=O C(=O)(CC(C)CC(C)C)NCc1nc(CC)sc1.C1(=O)CCC2CC(C2)N1 c1(CCCC(N2CC(O)(CN(C(C(C)SCCCC)=O)C)C2)=O)ccc(Cl)cc1 c1(N2CC(C)(C)C(NC(=O)CCCCn3ccnn3)C2)ccc2c(n1)CCC2=O Cc1nc(COC2CCCC2)cc(=NCCNCC(c2ccc(F)cc2F)O)[nH]1 C1(NC(C(C)C(F)F)=O)CN(C(=O)C=CCN(C(C)C)C(C)C)CCC1(F)F c12c(Cl)ccc(Cl)c1C(=O)N2.Cc1ccsc1CNC1CCCC1c1ccccc1 N1(CC(=O)N(C2CCC(NC(C3CCN(C)C3)=O)CC2)C)CCCNS1(=O)=O Cc1ccc(NC(=O)C(CC2CCC2)NC(=O)Cc2ccc(F)nc2)c(C)c1O C1(NC(c2scc(C)c2)=O)CC12CC(NC(=O)CC1C=NN(C)C1=O)C2 C(=O)(C1=CC2CCCC12)NCCCC(C)NC(=O)Cc1ccc(N)cc1 c1(NC(C=C(C)CNC(=O)COC(F)F)=O)ccc(O)nc1 c1(C(N2CCC(NC(C3CC34CC(F)(F)C4)=O)CC2)=O)cc2c(cn1)CCCC2 N1(C(c2ccc(C(C)C)cc2)=O)CCCC2C1CCN2C(=O)C=C1CCSCC1 N1(C(=O)CC2CCCO2)CC2CC2(C(=O)NC2(C3CC3)CC2)C1 C#CC1CN(C(=O)C(C)=C2CC2)CCN1C(=O)C=CC(C)C N1(C(C(C)SC)=O)CCCC2(CCCCC2NC(c2cn(C3CCC3)nn2)=O)C1 C(CNC(C1CC2(CCC2O)C1)=O)(CC(F)(F)F)NC(=O)Cc1c[nH]nc1O C1(NC(c2c(OCCC)cccc2)=O)CCCC2CN(C(C3CC3OC)=O)CC12 C(=O)(C(CC1CC1)NC(C1CC(C(C)C)C1)=O)N(CC(COC)O)C C1(C(=O)NC(C)CN2CCCC2)C2CC2CN1C(c1csc(O)n1)=O c1(CCCCC)nc(-c2cc(-n3cccn3)n(CC)n2)n(CC(C)(C)CO)n1 Cc1ccc(CN2CCCC(NC(N3CC([N+](=O)[O-])C3)=O)CC2)c([N+](=O)[O-])c1 CC1CCn2cc(C(=O)NCc3nc(CNC(C4COC4)=O)cc(O)n3)nc2C1 Cc1nn(C(C)C)c(C)c1C(=O)N(C)CCNC(=O)C(C)CS(C)=O C1(NC(C2N(C)C(=O)NC2)=O)CC2CC(NC(=O)COCCCF)CC12 c1(C(=O)NC(C(C)NC(C(CC#C)O)=O)(C)C)cc(Br)c(C)c([N+](=O)[O-])c1 c1(C(N(C)C)=O)ccc(CNc2cccc(NC(N3CCSCC3)=O)c2)cc1 C(=O)(C1CCN(C(=O)C(F)(F)F)c2ccccc21)Oc1cn(CC(C)C)nc1 C1(COC)(CNC2CCCN2CCCc2cscn2)CCC(F)(F)CC1 c1(C(C)=O)cc(C(N2CCC(CO)(NC(C3CC34CC4)=O)CC2)=O)c(C)nc1C C1(C(=O)NCC(CCCC)N(C)C)N(C(=O)CCCCSC)CCC1(C)C C12(NC(c3cccc(-n4ccnc4)c3)=O)CC(C1)N(C(c1cncc(O)c1)=O)C2 c1(CC)cc(C(=O)N(C(C)CNC(C2CC23CC3)=O)CC)oc1CC C(C(C)S(C)(=O)=O)(c1ccccc1)NC(c1scc(C)n1)c1nnnn1C(C)C c1(CSCC(=O)NC(C)C(C)(C)NC(C2CCCN2C)=O)cccc(Cl)c1 c1(NC(=O)Cc2ccnn2C2CCC2)cccnc1C(=O)Nc1csc(C(=O)O)n1 Cc1ccnc(O)c1C(=O)NCC1CC1CNC(=O)C(C(C)C)n1cc(C)cn1 C1(C(=O)NC(C(=O)NCC(C)NC(C=CCOC)=O)C)CC(F)(F)C1 C1(NC(C(C)OCC=C)=O)CN(C(=O)CN2CCOC2=O)CC1SC c1(CC(=O)NC(C)CN(C(=O)Cc2cnco2)C)ccc(C2CC2)cc1 C#CC(C)(C)C(=O)NC1CCCCC1Sc1cccc(OCc2ccccc2)c1 N1(C(CC(=O)OCC)=O)CCOCC2(C1)CN(C(=O)CC1CCNC1=O)CCO2 C(CC(CC)C(=O)NCC1(CNC(c2cnc(Cl)s2)=O)CC12CCC2)=CCCC C1(CNC(C2(O)C(C)(C)C2)=O)CC2CCC1N2C(c1cccc(Cl)c1)=O C12(CNC(COCCN(C)C)=O)CCCC1N(C(=O)C1CC1)CCC2 C(N=c1nc2scnc2c(NN2CCS(=O)(=O)CC2)[nH]1)c1n(CC)c(C)nc1 C(=O)(C1=C(OC)CCC1)N(CCNC(CC1(OCCCCC)CCCC1)=O)C C(=O)(C1CN(C(=O)OCC)Cc2n[nH]cc21)OC(=O)C=Cc1cc(Cl)cc(Br)c1 c1(C(N(CC(O)CNC)C)=O)cc2c(s1)CCC2=O.c1(C=O)cc([N+](=O)[O-])c[nH]1 CN1CC2CCN(C(=O)C(C)(C)CCNC(=O)Cc3cc[nH]c3)CC2C1 CC(c1ccccc1)=CC(N1C(C(=O)NC(c2ccc(O)cc2)C)CC1C)=O c1(C(=O)NC(CNC(c2cnc(C)s2)=O)CC(C)C)ccc(Cl)c(F)c1 c1(C(=O)NCCCNC(C2CC(C)=C(C)CC2)=O)ccc2n[nH]cc2n1 c1(NC(C)=O)cccc(F)c1C(N1CC(CNC(c2ccncn2)=O)C2CC12)=O C1(NC(c2c(C)nco2)=O)CC2CC(NC(=O)CC3CC(=O)NC3=O)C1C2 N1(C(c2snc(O)c2Cl)=O)CCC2CCN(C(c3cc4ccccc4o3)=O)C2C1 N1(C(C2CCN(C(C=CCOC)=O)C2c2ccccc2)=O)CCN2CCOCC2C1 N1(C(c2c(C)ncnc2)=O)CCC(CNC(c2cnc(N)cn2)=O)C(C)C1 c1(OC)ccc(C(=O)NC2CCCC2NC(c2c(C)nn(C)c2Cl)=O)c(F)c1 c1(OC)ccnc(F)c1C(=O)NC1CN(C(=O)CCC(C)(C)C#N)CC1C(F)F c1(NC(c2cnn(C3CCC3)c2)=O)ncc(C(=O)O)cc1Cl C1(C)(CNC(CC(CC)SC)=O)CN(C(=O)CC2(C)CC2(F)F)CC1C Cc1ccc(Cl)c(CN2CCC(OCc3ccc(Br)cc3)CC2)c1 N1(C(CCC(=O)N(C)C)=O)C(CC(=O)NCc2ccnc(Cl)c2)C2CCCC12 C12(NC(C3N(CC)C(=O)CC3)=O)CCN(C(c3cnc(C(C)C)[nH]3)=O)CC1C2 CCC(O)C(C)(C)C(=O)N1CCC(O)(CCNC(c2ccn(C)c(=O)c2O)=O)C1 C(C1CN(C(C23CC(F)(C2)C3)=O)CC1C(N1CC(=O)NCC1CC)=O)=CC C(=O)(C#CC(C)(C)CNC(c1sc(O)nc1C)=O)NCC(CC)CC N1(C(CC(C)F)=O)CC(NC(=O)CCc2nnc(C(F)F)o2)CCC1C Cc1oc(S(N)(=O)=O)cc1C(=O)NC1CN(C(c2cc(F)cc(F)c2)=O)CC1C c1(NC(N(C)C)=O)cc(NC(=O)Nc2ccc(-c3ncn(C)n3)cc2)cc(Br)c1 CC1(CNC(=O)C(F)=C2CCC2)CCCN(C(=O)C(c2cccc(F)c2)O)C1 C1(CNC(c2cc(OC)no2)=O)CCCC2CN(C(=O)Cc3cncn3C)CC12 C1(O)(CN(C(=O)C(c2ccoc2)NC(=O)CCOC2CCCC2)C)CCC1 c1(C(N2CCCC(CC(=O)Nc3ccc(C4CC4)nc3)C2)=O)cc([N+](=O)[O-])n[nH]1 CC(C)CS(=O)(=O)CCC(=O)N1CC2CC(C3CC3)CC(C2)C1.C1(=O)C=CC(=O)N1 c1(C(=O)NCC(C)N(C(C(C)NC(CC)(C)C)=O)C)cc2ccccc2c(O)n1 c1(C(=O)NCC(CN(C(=O)C(C#N)C2CC2)C)(C)C)cccc2c1OCCC2 C12(CCC1)CC(=O)N2.C(CC(=O)N1CCCC1)CCOC.C1C(=O)N1 N1(C(C2(C#C)CC2)=O)CCCC(CN(C)C(C2(OC)CS(=O)(=O)C2)=O)C1 c1(CC(=O)OC(c2ccccc2)C)nnc(-c2cccnc2)o1 CCC(C(=O)NC1CCCCC1NC(=O)Cn1ccnn1)C(C)O c1(C(=O)NCC2(CN3CCC(CC(=O)N)C3)CC2)ncccc1O.C1(C)CC1 C1(OC(C2CC3CC2(c2ccncc2)C3)=O)CCOC2(CCC2)C1 C1(CNC(C2(C#N)C(C)C2)=O)(CNC(=O)Cc2nn(C)cc2Cl)CCCCC1 C1(CC(=O)NC(c2ccncc2)CC)CCCN(C(=O)CC(C)(C)OC)CC1 N1(C(c2nnc(C(C)(C)C)s2)=O)CCCCC(NC(c2csc3cncn23)=O)C1 c1(C(=O)NCCCN(C(=O)C(C)CSC(F)(F)F)CC)cc(C)c(C)o1 N1(C(C2CC3(C(OC)CC3)C2)=O)CC2CCN(C(c3[nH]c(=N)ccc3Cl)=O)CC2C1 N1(C(Cc2c(C)ocn2)=O)CCCC(F)(CNC(=O)CN2CSCC2=O)C1 C1(OC(=N)O)CN(C(=O)CCSCCC(C2(Br)CC2)=O)C1 N1(C(C(C)(N(C(C(CC)C(C)C)=O)C)C2CC2)=O)CC2CN(C)CC2C1 C1(NC(C2N(CCC)CCC2)=O)CCN(C(=O)CN2CC(=O)N(C)C2=O)C12CC2 C1(CNC(N2CCC(c3nc(C)on3)CC2)=O)CCc2nc(C)cn2C1 c1(C(=O)OC)ncc(C(=O)NCCC(C)NC(=O)C=CCF)s1 N1(C(CC(C)C)=O)CCC2CN(C(=O)C(C)Cc3ccc([N+](=O)[O-])cc3)CC2C1 C12CCCC(CC1)CNC(=O)N2.c1(C(N)=O)coc(Cl)n1 C#CCCCCC(=O)NC1CCN(C(c2ccc(N)c(O)c2)=O)C1 C=CC1CCN(C(=O)CC2(C=C)CN(C(=O)CC3CCCC3C)C2)CC1 C(=O)(CC(F)(F)C(C)C)NCCN(CCC)C(C1CCOCC12CCC2)=O C(CCCC(=O)N1CCCC1CN(C)C(c1cnn(C)c1C(F)F)=O)SC c1(C(=O)OC(CC)C(N)=O)cc2c(s1)CCN(C(=O)OC(C)(C)C)C2 c1(CC(=O)NC2C(CNC(Cc3nc(C)sc3)=O)C2)cccc(C(F)(F)F)c1 n1(CC(=O)NCc2cc(Br)ccn2)ccc2c(F)cccc12.C12COCCN1C2 C1(CNC(CCCC(=C)C)=O)CC(C)(C)CCC1NC(c1ncn(C)n1)=O C1(C(=O)NCC(=C)Cl)C(C2CC2)CCN1C(C1CS(=O)(=O)C1)=O C(=O)(CCC(=O)N1CC(CC(C)NC(C2CCCC(C(C)(C)C)C2)=O)C1)OC C1(CC#C)(C(N2CCC(CCNC(c3cncnc3C)=O)C2)=O)CCCOC1 c1(CC(=O)NC2CN(C(CCCN(C(C)=O)C)=O)C(C)C2)ccc(C#N)cc1 c1(N2CC(CC(C)NC(C3CCCN(C(C)=O)C3)=O)C2)ncc(C)c(C)n1 C12(CNC(=O)CC3COCCOC3)CC1CN(C(C13CSCC1C3)=O)C2 CCCC(CC)C(=O)NC12COC(C1)C(NC(=O)CCOCc1nccn1C)C2 c1(C(=O)NC2C=CC(CNC(Cc3nc(CC)sc3)=O)C2)ccc(C#N)[nH]1 C(C(=O)NCCC1(C(N2CCCCC2CCO)=O)CC1)(C(C)C)SC c1(NC(C)=O)cc(C)cn(C)c1=O.C1(=O)C(CC2CCC2)N1C(C)C(=O)N.CO N1(C(C2(C)CCC(=O)NC2)=O)CCN(C(c2ccc(N)c(Cl)c2O)=O)C2CCC12 CON1CC(NC(=O)C(C)(C)C(=O)OC(C)(C)C)CC1=O.C1C#CCNC(=O)N1 N1(C(c2cncnc2)=O)CCN(C(C2C3CCCOC23)=O)C2CCCC12 c1(C(=O)NCC(CNC(=O)CN2C(=O)CCC2=O)OC)cc(=O)c(Br)c[nH]1 C1(C)(CNC(CC(=O)OC)=O)CC(OC)CN1C(c1cc(C2(C)CC2)on1)=O N1(C(C(c2ccccn2)C)=O)CCC(C)(CNC(C2CN(CC(F)(F)F)C2)=O)C1 C(CS(=O)(=O)CC(=O)NC1C2CC1N(C(c1ccc(N)c(N)c1)=O)C2)OC C=C(C)CCC(=O)NCC1(CNC(=O)Cc2csc(CCCCC)n2)CCC1 C1(N(C(=O)CCC2CCOC2)C)C2CN(C(c3csnc3Br)=O)CC12 N1(C(c2nc(C)sc2C)=O)CCC2CCCC(C1)N2C(c1c(C)cncc1C)=O c1(CNC(C2CC(C)(NC(C3C(C(C)(C)C)C3)=O)C2)=O)ncc(Cl)cn1 C(=O)(CC(C)(O)CC(=O)O)N1CCOCC(NC(c2c(F)ccc(C)c2Cl)=O)C1 N1(C(C2CC(NC(c3cnn(C)n3)=O)C23CCC3)=O)CCCCC2(CCC2)C1 C1(NC(C(C(C)C)NC(C)=O)=O)CC2CC1CC2C(=O)NC1CCOCC1F c1(CC(N2CC(CNC(C(CC=C)NC(C)=O)=O)C2)=O)c(C)nn(C)c1Cl C1(C(=O)NC(C)CSCCOC)(CC)CN(C(=O)Cc2ccccc2)C1 C1(N(C(c2cc(CNC(C(C)SC(C)C)=O)on2)=O)C)CCC(=O)N(C)C1 CC(O)C(C(=O)NCC1(F)CC(NC(c2cncn2C)=O)C1)NC(=O)C(F)(F)F Cc1[nH]nc2ccc(C(N3CC4(CNC(=O)C5=CCCCO5)CCC3C4)=O)cc12 C(=O)(CC(C)C(F)F)N1C(CC(=O)NC(c2onc(C)n2)(C)C)CCC1 c1(C(C(=O)NC(C)C(C)NC(C2(n3cncn3)CC2)=O)C)ccc(F)cn1 C(=O)(C1CCc2nccn21)N1C(CC(=O)OCC)CN(C(=O)CSCCOC)CC1 c1(C(=O)NC2C(CNC(C3(N(C)C)CC3)=O)C2)ccn(CC(F)F)c(=O)c1 C1(CC)CCCN(C(=O)CC2CCOC2)CC1.C12CCCC1NC2=O c1(C(=O)NC2CCCC23CN(C(C2CC(F)(CO)C2)=O)C3)ccc2c(c1)CCO2 C1(CC=C)(NC(=O)Cc2ncoc2C)CCN(C(C2(n3cccn3)CCC2)=O)C1 C(=O)(C(F)C(C)CNC(=O)CCNC(=O)CO)NCCn1ncc(CC)c1 C1(C(N(C2CCC2)C(C)C)=O)CCCN1NC(=O)C=CC(C)(C)C N1(C(c2ccc(CC)o2)=O)CC(N=c2[nH]nc(C(C)C)s2)C2(CCC2)C1 c1(C(=O)NC(C(C)NC(=O)COc2cccc(Cl)c2)C)cccc2ncsc12 Cc1ccc(C2(C(N3CCC(CF)(NC(C4C(C)C4(F)F)=O)C3)=O)CCC2)cc1 N1(C(CCN(CC)CC)=O)CC(CNC(c2coc(COC)n2)=O)CCC1C CCCC(CNC(c1cc(C#N)cs1)=O)C(=O)N(C)C(c1nccs1)C Cc1nc(C2CCCO2)ccc1C(N1CCCC(C(F)F)C1)=O C1(C)(CNC(c2cc(OC)nn2C)=O)CN(C(c2ccc(C)c(C)n2)=O)CC1C N1(C(c2ncc(OC)cn2)=O)CCCCC(NC(=O)C=C(F)c2ccccc2)C1 C(=O)(C1=NN(CCO)C(=O)CC1)NCC(C)NC(C1C2C3CCC(C3)C12)=O C(=O)(C(C(C1CCCCC1)SC)Sc1nc(C)c(C(=O)O)o1)OCC c1(OC)ccccc1C(=O)NCC1CC(n2cnnc2)C1.C1(=O)CO1.C1CO1 C1(C(N(C)CCOCCCNC(c2ccccc2Cl)=O)=O)CC2OC(=O)OC2C1 N1(C(C(N2CCOCC2=O)C)=O)CC2CCC2(CNC(=O)C(F)=CCCF)C1 c1(OC)cc(F)ccc1CC(N1CC(NS(C)(=O)=O)C(C#N)C1)=O N1(C(c2oc(CC)c(C)c2)=O)CCCC(C)(C)C1C(N1CC(CO)(OC)C1)=O c1(C(=O)NCC2CC(Cn3cc(C(C)(C)OC)nn3)C2)c(C)cnc2ccccc12 c1(OC)cc(SC(C)C(N2CCNCC2)=O)ccc1C#N c1(CNC(=O)Nc2cn(CC(=O)N(C)C)nc2C)cnc2nccn2c1 Cc1ccc2ncnc(N3CCC4C3CCCN4Cc3cccc(Cl)c3I)c2c1 c1(C(N(CCCOCCNC(C(C(CC)C)C)=O)C)=O)ccc(Cl)c([N+](=O)[O-])c1 c1(C(=O)NCC(C)(C)NC(C2(NC(=O)OC)CCCCC2)=O)cc2c(s1)CCC2 CCC(CC(F)F)C(=O)N(C1CCN(C(C23CC(F)(C2)C3)=O)CC1)CC(C)C Cc1cc2cccc(C(N3CCCC3CNS(=O)(=O)c3ccccn3)=O)c2[nH]1 c1(C(=O)NCCN(C(CCC(C)SC)=O)CCCCCC)cnc(C)c(N)c1 CC(C)C(C(=O)NCCC1CCCN(C(=O)C(C)OC(C)(C)C)C1)n1cncn1 C1(CC#C)(C(=O)N(CC(C)NC(=O)C(C)(C)C2CCCC2)C)CCCCC1 CC12CN(C(=O)CN3CCCCC3=O)C(C(N3CC4C(C(N)=O)C4C3)=O)(C1)C2 C(=O)(CC(C)C(C)(C)C)N1CCCC(N(C2CCCC2)C(Cc2c(C)n[nH]c2)=O)C1 c1(OC)c(C(N2CCC(NC(=O)CCC(C)(C)O)C(C)C2)=O)cccc1F c1(C(N2C(C(C3CC=CCC3)C(=O)OCC)CCC2)=O)coc(C)c1 Cc1oc2cc(C(=O)NC3(C)CN(C(=O)C(=O)NC(C)C)C3)[nH]c2c1C Cc1nnc(C(=O)NC2CC(F)(CNC(c3ccoc3Cl)=O)C2)s1 C(=O)(C(=O)N=S(C)(C)=O)N1CCC(O)(CCNC(C(C)NC(=O)C(C)(C)C)=O)CC1 Cc1cc(Cl)c(F)cc1C(=O)NC1CCCCC1C(=O)Nc1ccc(C#N)nc1 C(C)(C(C)(C)C(=O)N1CCCC(O)CC1)NC(c1c(C)nncc1)=O c1(C(C(N2CC(CNC(CCCC=C)=O)C(C)(C)C2)=O)C)c[nH]c2ccccc12 C1(NC(C=C(CC)CC)=O)COCCN(C(=O)C(F)=C(C)C)C1 c1(C(N2CCCC3(NC(CNS(N(C)C)(=O)=O)=O)C2C3)=O)cn2cccnc2n1 C1(NC(c2cn(CC)nn2)=O)CC(C(=O)NC2CC(CN(C)C)C2)CC1O CN1CCC2CN(C(C3CCCN3C(=O)OC(C)(C)C)=O)CCC12.C1(=O)CCN1 c1(-c2c(CN3CCN(C(C)=O)C(C)(C)C3)ccc(Cl)c2)cc2c(C)cccc2[nH]1 c1(C(=O)NCCOCCNC(C(C)SCC)=O)cccc(F)c1Br C(=O)(C1=C(CCCCl)N(CC2CC2)C(=S)NC1c1cccc(Cl)c1)OCC C(=O)(CC(C)(O)COC)NCCCCC(=O)NCc1cnc(CC)[nH]1 N1(C(C2C(C=C)C2)=O)CCC(O)(CN(C(=O)C=C(Cl)Cl)C)C1 C1CC(O)C(=O)N1.Cn1cncc1CN1CCCC1.N12CCC(C1)CC2=O C1(C(=O)Nc2cc([N+](=O)[O-])n[nH]2)C2CCN(C(C3(P(C)(C)=O)CC3)=O)CC12 n1(C(CC)C)nc(C(=O)NCC=CCNC(c2onc(Br)c2C)=O)cc1C O=C(N=c1cco[nH]1)C1CCN(C(c2ccc(F)cc2Br)=O)C1 Cc1nc(C(N2CC(NC(c3cc(C(N)=O)c[nH]3)=O)C(O)C2)=O)ccc1[N+](=O)[O-] c1(C(N(C2CCCN(C(CCCNC(C)=O)=O)C2)C)=O)cnc2ccnn2c1 C1(NC(c2n(C=C)nnc2)=O)CCC12CN(C(c1ccc(NC(C)C)nc1)=O)C2 C#Cc1cnc(C(=O)N(CC(=O)NC2C(C)C2(C)C)C)c(C)c1 c1(OC)ccc(CCCCC(=O)N2CCC(CC(C)NC(=O)C(C)O)CC2)cc1 c1(C(N(CC(C)NC(CCCC(C)O)=O)C)=O)cc(Cl)cc2ccncc12 S(=O)(=O)(c1cc(C=CC(=O)N(C)CCc2ccccc2)ccc1OCC)NCC c1(C(N2CC(CNC(=O)C(F)OC(F)(F)F)C(O)C2)=O)cc2c(s1)CCC2 C1(C(=O)NCC2(F)CC(NC(C3CNC(=O)N3)=O)C2)(CSC)CCOCC1 c1(C(=O)NC23CC(CNC(=O)C=C4CCCCC4)(C2)C3)ccc(F)c(Br)c1 C(=O)(CCC(F)F)N(C(CNC(C1CCCC1(C)C)=O)C1CC1)C C(CNC(=O)CC#N)(CC(=O)N1CCC(c2ncc[nH]2)C1)OC c1(C(=O)NC2C(NC(C3CC(C)OC(C)C3)=O)COC2)c(Cl)ccc(F)c1F Cc1cc(F)ccc1NC(=O)C(c1cncc(C)c1)N(C)Cc1ccc(F)c(Br)c1 C1(C2CCCCO2)(C(=O)OCCc2cn(CC)nc2C)CCCO1 c1(C(=O)NC(c2cc(F)cc(Cl)c2)CNC(C(C(C)C)C)=O)cccc2ncnn12 C(=O)(C(C)c1cc[nH]n1)NC(C1C(C(=O)NCCN(CCCC)C)C1)C n1(CC(=O)NC2C(CNC(C(CC=C)(C)C)=O)C2)ccc2cc(Br)ccc12 c1(C2C(C(N(C)CC3(NC(Cc4nnc(C)o4)=O)CC3)=O)C2)cccc(F)c1F N1(c2ncc(C(=O)OC(c3coc4c3COC4)=O)nc2)CC2CN(CC)CC2C1 c1(CN2CCC(CC(N3CC(C(=O)OC)C3)=O)C2)ccc(CN(C)C)c(Cl)c1 C(C(N=[N+]=[N-])C(=O)N1CCN(C(C2(COC)CC2)=O)C(C)C1)OCC CC(C)C(C(=O)NC1CC(c2ccccc2)C(O)C1)NC(=O)CN C1(C(N(C(C)CNC(=O)Cn2c(C)ccc2C)CC)=O)COC(C)(C)CO1 Cc1sc(C(=O)N(CCNC(=O)Nc2ccccc2)CCOC)nc1O C1(NC(=O)NCCNC(=O)C=CBr)CCCN(C(=O)C(c2ccc(F)cc2)F)C1 N1(C(c2c(CC)onc2)=O)CC2CC1CC2NC(c1cc(C)oc1CSCC1CC1)=O C1(C(C)(C)C)CN(C(=O)C(=O)NCC(c2ccc(F)cc2)=O)CCC1=O c1(CC(=O)N(C2CN(C(c3ccncc3C(F)F)=O)CC2O)C)cccc(Cl)c1 C1(C(N2CC(Cc3cn(CCN(C)C)nn3)C2)=O)Cc2cscc2C1 CCCC(C)C(=O)NCC1(C(N)=O)CN(C(c2cn(CC(F)(F)F)nn2)=O)C1 N1(S(Cc2nc(C3CC(OC)(OC)C3)sc2)(=O)=O)CCC(F)(CSC)CC1 N1(C(C)C)CC(C(=O)N(CCCCNC(=O)CC(C2CC2)C2CC2)C)CCC1=O C1(NCC(=O)Nc2ccn(C)n2)CC(C(=O)NCCCF)C12CCC2 C(N1CC(C)CC(C)C1)NC(COc1c(C(C)C)n(-c2ccccc2)nc1)=O C(=O)(CN=c1cc[nH]cc1)NC1C(CC)CN(C(c2ccccc2C(N)=O)=O)C1 c1(OC)cc(Cl)c(Br)cc1C(=O)NCC(C)CNC(C1(Br)CC1)=O Cc1noc(C(F)F)c1C(=O)NC1CCC(NC(=O)CC(O)CC2CC2)C1 CC1CC(=O)CC(C2CCCCC2)N1C(=O)NCc1cncn1C C1(C#N)(C(=O)NCC(CC)(C)NC(C2CCC(C)(C)CC2)=O)CC12CCC2 N1(C(CC2CC(=C)C2)=O)CC(CC(=O)NC(C)CN(C)C)C2(CC2)C1 c1(OC)cc(C(N2CC(NC(=O)C(C)(C)c3cncs3)C(O)C2)=O)cc(Cl)c1O C1(C(N2CCC(C)(NC(C3C=CC=CC=C3)=O)CC2)=O)CC2CCCCC2O1 C(C1(O)CCCc2ccccc21)NC(=O)C(=O)NC12COC(CO)(C1)C2 c1(CNC(c2cn(CC)nn2)=O)nccc(C)c1F.C12(CCCC1C)C(=O)N2 CC1(C(=O)NCC2CCC(CNC(N)=O)CC2)CCC(=O)C1.C1CC(=O)N1 Cn1nc(C(=O)NC2(C)CCN(C(c3cncs3)=O)C2)cc1C1(Cl)CC1 N1(C(C(C)CF)=O)CC(NC(c2cc(O)cnc2N)=O)CC12CCC2 c1(COC)cccc(C(=O)NCC2CC(NC(=O)C(F)C(C)C)C2(C)C)n1 C1(C(=O)NCC2N(C(C(CC)C)=O)CCCC2(C)C)CC(c2cnn(C)c2)=NO1 c1(C(=O)NC23C(CN(C(CSCC#C)=O)C2)C3)cc2ccc(Cl)c([N+](=O)[O-])c2[nH]1 Cc1cc(CC(N2CC(C(C3CCCN3C(=O)Cc3cocn3)=O)C2)=O)cc(F)c1 C(=O)(CCCCCN=[N+]=[N-])NC(C1(O)CN(C(c2cc3ncccc3o2)=O)C1)C c1(CNC(CCSCCC)=O)cc(O)nc(CNC(=O)C(c2ccnn2C)O)n1 C(=O)(C1=Cc2cccc(OC)c2OC1)N1CCC(CN(C(CSCC)=O)C)C1 C1(NC(C(C)OCCOC)=O)CC2CCC1CC2NC(=O)C1=C(Cl)CCC1 Cc1ncnc(N2CCC(NC(C3(c4ccc(Cl)cc4)CC3)=O)C(O)C2)c1Br C(=O)(C1CCCc2scnc21)NCC1(O)CN(C(C(C2CC2)OC)=O)C1 CN1C(=N)Nc2cc(ccc2)C(=O)NCC2(F)NS(=O)(=O)CCC1C(=O)N(C)C2 c1(C(N2CCC3(CC(NC(c4cnns4)=O)C3)C2)=O)ccnc2ccccc12 N1(C(C2CCN(C)C2)=O)CCC2(CCCN(Cc3cccc(I)c3F)C2)C1 C1(CC2OCCN(C(C(C)OCc3ccccc3)=O)C2)CNCC2(CCC2)C1 C1(N(C(=O)CC23CCCC2C3)C)CCC(NC(=O)CCc2cnco2)CC1 c1(CNC2CC(C)CN(C(=O)Cc3ccsc3)C2)ccc2ccc(Br)cc2n1 N1(C(c2cccc(C)c2F)=O)CC(NC(C2CN3CCCC2C3)=O)C2(CCC2)C1 C1(n2cc(CC=C)nn2)CCCN(C(C2CC(OCC)C2)=O)C1 C(=O)(C(C)(O)Cc1ccccc1)N1C(CN(C)C(c2cc(CO)[nH]n2)=O)CCC1 CCC(C)(C)C(O)C(=O)N1CCN(C(=O)Cc2nc(F)c(F)cc2F)CC1CSC CCCC(C)CC(=O)N1CCC(F)(CNC(c2ccc(CN(C)C)[nH]2)=O)C1 c1(C(=O)NCCN(C)C(c2cnsc2)=O)cc(-c2ccsc2)nn1C N12CCC(CC1)CCC2.C1(C)(C(=O)NC(CCOCCN(C)C)=O)CC(C#N)C1 N1(C(C)=O)C2CCC1CC(NC(c1ccc(-c3cccc(Cl)c3F)cc1)=O)C2 Cc1noc(C)c1S(=O)(=O)N1CCC(O)(C(N2CCCC2c2ccc(Cl)cc2)=O)C1 C(=O)(C#CC1(C)CCCO1)NC(C(=O)NCCC1CCC(C)C1)Cc1cn[nH]c1 CC1CCC(N2CCC(NC(=O)C(=O)NCCC3CCCC(C)C3)CC2)CC1 c1(C(N(CCNC(CC2CC(=C)C2)=O)C(C)C)=O)cc(F)c(Cl)c([N+](=O)[O-])c1 C(=O)(CS(=O)(=O)c1ccccc1F)N1CC(NC(C(CC)OC)=O)C(C)(C)CC1 N1(C(c2cc(-c3ccc(C)o3)[nH]n2)=O)CCCCCC(NC(C2C(C)C2C)=O)C1 C(=O)(CC(C)C(F)(F)F)N1CC(C(C)NC(c2c(C)nc(CCC)s2)=O)C1 C1(CNC(N2CC(C(CC)OC)C2)=O)CCCN1c1nccs1 N1(C(c2c(C)ccc(=N)[nH]2)=O)CCC2(CCCN2C(C2CCCCC2(C)C)=O)C1 c1(C(N2CCC(CC=C)(NC(=O)Cc3cnc[nH]3)C2)=O)cnc(Br)c(OC)c1 c1(CC(=O)NCC2(F)CC(NC(=O)CC3CCOC3)C2)cccc(Br)c1O N=c1ncc(C(=O)NC2CCCCC2NC(c2cocc2Br)=O)c[nH]1 C(=O)(C(CO)C(C)(C)C)N1C(CC)CN(C(c2c(SCC)cccc2N)=O)CC1 c1(CC)ccc(C(N2CCCC2(C)CCC(=O)NC2CCCC2OC)=O)nc1 C(=O)(CC(C)(C)C(C)=O)NC(CC)(C)CNC(=O)C(C(C)OC)N(C)C N1(C(C2C(C)(C)CCO2)=O)CCCC2(NC(C3CC4(CCC4)C3)=O)CC2C1 c1(C(=O)NCc2occ(C(N3CCC(CC(N)=O)C3)=O)n2)cc2ccccn2n1 C1(NC(C2(CCC=C)CC2)=O)CCN(C(c2cnco2)=O)CC12CCC2 c1(NC(C(N2CC3CCC2C(O)C3)c2ncc(C)s2)=O)ccc2c(c1)CCC2 C1(C)(CCC)CCN(C(C2CCCC(O)C2)C(=O)NC2CC(F)(F)C2)C1 C1(C(=O)NC(CNC(c2nc(OC)oc2)=O)(C)C(C)C)NC(=O)C2CCC12 C1(CNC(c2c(C)cncn2)=O)CC2(CCC2)CN1C(=O)CSCC#N Cc1nccc(C(=O)NC(C(=O)NCCC(=O)NCC(C)C)C2CCC2)c1N C1(NC(c2c(C)nccn2)=O)CC=C(C(=O)NCC2(C)CCOC2)C1 N1(C(c2cc(OC)no2)=O)CC2CCN(C(c3ccn(C(C)C)n3)=O)C(C2)C1 C1(n2cc(-c3ncn(C(C)C)n3)nn2)CCCN(C(=O)C(C(C)C)N(C)C)CC1 C(CCC=C(C)C)(C(=O)NCCC1CCC(F)(F)CC1)N(C(C)C)CC N1(C(C(C)(C)F)=O)CCN(C(=O)CCc2ccccc2Cl)C(CC2CCCC2)C1 CC1(C)C2CC(CN=C(NC3CC3)NC3CCN(C4CCOC4=O)CC3)CC12 c1(C(=O)NCC23C(CN(C(CCc4c(C)ncs4)=O)C2)C3)cnc(N)c(Cl)c1 C(=O)(CCCCC(=O)N(C)CC1(O)CN(C(c2ccnn(C)c2=O)=O)C1)OC C(=O)(C1=NOC2(CCC2)C1)N1CC(N(C(c2cccc(C(C)=O)c2)=O)C)C(F)C1 c1(C(c2n(C)nnn2)NC(c2ccccc2OCF)C2CC2)cccc([N+](=O)[O-])c1 C1(CC=C)(NC(=O)CC2CC=CC2)CCCN(C(=O)CCN(C)CC)C1 CC(C)(C)CC(O)C(=O)NC1CN(C(c2snc(Cl)c2Cl)=O)CC1O C12CC(O)CN(C1)ONC2=O.C1(CC)CCCCC1.CCCCC1CC1 c1(OC)cncc(C(=O)N(CCCNC(c2occc2C)=O)C2CC2)c1 Nc1c(C(N2CCCC(NC(C3(C(F)F)CCCO3)=O)CC2)=O)cc(F)cc1F Cc1noc(N)c1C(=O)NC(CCNC(c1cncn1C(F)(F)F)=O)C(C)C c1(N(C)CC2CCCN2)cnc(C#N)cn1.c1(C=O)cnc(CC2CC2)s1 Cc1ccc2cc(C(N3CC4CC3CN4C(C3OC(C)CC3C)=O)=O)[nH]c2c1 C1(C=O)CCOCC1.CC(C)(C)OC(=O)NCCOCCOCCCC c1(C(N2CCC(N(CCC)C(c3cnn(C)n3)=O)C2)=O)ccc(CC)nc1 c1(C(N2CCC(N(c3ccc(C)cn3)C)C2)=O)cncc(P(C)(C)=O)c1 C(=O)(C1=CC(C)(C)C1)N(CCCNC(C12CC1CCC2(F)F)=O)C N1(C(CCC=CC)=O)CCCCC1C(C)NC(c1cn(-c2cccnc2)nn1)=O C(=O)(C1=CC2(CN(C(=O)CN=c3cc[nH]cc3)C2)OC1)NCCC(C)(C)C1CC1 Cc1ncn(C)c(=O)c1C(N1CC2CC2(CNC(=O)CC2(C3CC3)CC2)C1)=O n1(CC(=O)N(CCNC(Cc2c(C)ocn2)=O)C(C)C)cccc(N)c1=O C12(CNC(CCC(C)(C)C)=O)CN(C(=O)C(C3CCCCCC3)F)CC1CCO2 c1(C(=O)OC)cc([N+](=O)[O-])cc(Cl)c1N1CCCC(c2ccc(F)cc2)CC1 N1(C(C2CC(=O)NCC2)=O)CC2CN(Cc3ccc(Cl)c(Br)c3)CC2C1 C(=O)(CCC(C)(C)NC(=O)C(N)=O)N1CCC(OCC=C)CC1 C1(C(N2C(C=CC(N3CCCC(F)C3)=O)CCC2)=O)CN2CCCN1CC2 n1(CC(N2CCC3C(NC(C(c4cccnc4)OC)=O)C32)=O)cccc(N)c1=O N=c1[nH]c(N2CCn3c(cnc3Br)C2)nc2ccc(Br)cc12 C(=O)(CN=c1ccc(C#N)c[nH]1)NC1C(CNC(Cc2c(C)cc(C)s2)=O)CC1 C1(NC(c2ccc(C#C)cn2)=O)C(CNC(=O)CC2(O)CCC2)CCC12CCC2 Cc1cc(=NCC2(C)CCOC2)[nH]cc1S(=O)(=O)N(C)CC1CCCN1 Cc1cc(F)ncc1C(=O)NCC(C)(C(C)C)NC(C1CCCSC1)=O Cc1cc(Br)cc2cc(C(=O)N(CC(C)CNC(=O)CC(C)(C)C#N)C)[nH]c12 CC1Oc2ccc(C(N3CC(CN(C)Cc4ccc(Cl)cc4)C3)=O)cc2NC1=O c1(C(C(=O)NC2(CCNC(C(CC)NC(N)=O)=O)CC2)C)ccc(F)c(F)c1 N1(C(C(C)OC2COC2)=O)CCC(O)(CCNC(=O)C(C)NC2CCOCC2)C1 c1(C(N2CCCCC2C(N2CC(O)C(F)C2)=O)=O)cccc2ccncc12 N1(C(c2c(-n3cc(CCC#N)nn3)cccc2)=O)CCC2(CC1)CNC(=O)NC2 c1(CCCC(N2CCC(O)(CNC(CCCC#N)=O)C2)=O)c(F)cccc1F N1(C(CCn2c(C)nc(C)n2)=O)CC(F)(F)CC1CNC(C1CCN(C)C1C)=O c1(CCC(=O)NC(C2CCCN(C(COC)=O)C2)C)cc(OC)ccc1OC C1(CNC(C2(SC)CN(C(C3CC(=C4CCC4)C3)=O)C2)=O)CCCCN1C CC(C)CCC(C(=O)NCc1cc(F)cc(F)c1)NC(c1cccc(O)c1)=O c1(C(=O)NCCN(CCC)C(C23C4CC(CC24)C3(F)F)=O)cc2c(C)noc2s1 C(=O)(C1Cc2ccccc21)N1CCC(NC(c2cccc(C)c2C)=O)CC1 S(=O)(=O)(c1c[nH]c(C(N2CC3C(CNC(=O)C=C(C)C(F)F)C3C2)=O)c1)NC c1(S)ccccc1O.c1(C(C(=O)NC(CC)CCC)OC)ccccc1 c1(CCC(C)NCCC(=O)N(CC)Cc2occc2Br)cccc([N+](=O)[O-])c1 C1(NC(C(CC#C)C)=O)C2COCC1CC(NC(c1cc(C)n(C(C)C)c1)=O)C2 CN1CC(C)(C(=O)NCCCC2CN(C(C3(CO)CC3)=O)CCO2)CC1=O C1(N(C(=O)CCc2ccsc2)CC)CCN(C(c2cc(C(N)=O)c[nH]2)=O)CC1 Cc1cccc(OC(C)C(=O)N(C)CCNC(=O)Cc2ccc(C(F)F)cc2)c1 c1(C(N(CCNC(C(c2cccc(C)c2)C)=O)C(C)C)=O)ccc(N)c(C)c1C N1(CC)C(=O)CCC1CC(=O)NC1C2CC1N(C(=O)CNC(=O)CN(C)C)C2 C1(CNC(C(CSC)(C)C)=O)(NC(c2cn(CCF)nn2)=O)CC2CCC1CC2 c1(C(N2CCC(C)C(N(C)C(c3cn[nH]c3)=O)C2)=O)nccc2n[nH]cc12 C1(C(=O)NCC2CCN(C(c3nc(C)c(C)[nH]3)=O)CC2)CCC(N=[N+]=[N-])C1 C(=O)(C1=NOC(C)C1)NCC12C(CN(C(c3c(C)sc(O)n3)=O)C1)C2 N1(C(=O)OC(C)(C)C)CCCC(CCc2nc[nH]n2)C1.C1CCCCS1 C1(O)(CNC(c2n(CC)ncn2)=O)CCN(C(C2(C)CCCC2(F)F)=O)CC1 N1(C(COC(C)C)=O)CCN(C(c2ccc(C(C)(C)C)o2)=O)C(C2CC2)C1 C1(C(NOCC(C)O)=O)CC(C)CCN1C(=O)CC1CCCC1C C1(C(=O)NC2CC(NC(c3c(C)nn(C(C)C)c3C)=O)C2)CCC2C(C1)C2(F)F C(=O)(C#CC1(CC)COC1)NC(CN(C(COCCCOC)=O)C)CC c1(C(=O)NCC2C(NC(CCOCCOC)=O)C2)ccc(F)c(C)c1C N1(C(Cc2scc(C)c2)=O)CCC2(CCN(c3nnc(CO)s3)C2)C1 N1(NC(c2c(C(C)C)cc(Cl)s2)=O)CC2CC(Nc3cc(O)nc(O)n3)CC1C2 c1(OCC#C)cccc(NC(=O)NCC(CC)(CC)NC(=O)OC(C)(C)C)c1 N1(C(c2c(C)nc[nH]2)=O)CC(C(=O)NC2C(C)C2(C)C)C(C)(C)C1 C(C(=O)N1CCCC1(C)CNC(=O)C(C)C1CCC1)(C(C)C)SCC Oc1ccnc(C2CCC(Nc3ncc(Br)cn3)CC2)n1 C1(NC(c2c(OC)cnc(Cl)c2)=O)CCN(C(=O)CC2CCCC2)CCC1CO C1(C(=O)NCCCc2c(C)n[nH]c2)CN(C(=O)CCCC2CC2)CC12CC2 c12cccc(c1O)N2.C1(CC(=O)N(CC(=O)OCC)C)CCC1OC C1(NC(C2(CNC(C3C(C)(C)OCC3)=O)CC23CCC3)=O)Cc2cscc2C1 C1(C(=O)NC(C)CN(C)C)(CO)CCN(C(c2cscn2)=O)C1 N1(C(C(CC)(C)C)=O)CCN(C2CCOCC2)C(C)C1 O=C1CC(C(=O)NC(C(=O)N2CC(SC(F)F)C2)C2CCC2)CC(=O)N1 c1(C(=O)Nc2cn(C3CCCN(C(C)=O)C3)nn2)cc(C)ccc1N N1(C(COCCC(C)C)=O)CC2CC(NC(C3CC4(C3)CC(C)C4)=O)C1C2 c1(C(N(C2CN(C(=O)CC3(O)CCCC3)C2)C)=O)cccc2[nH]nc(O)c12 Cc1cnc(CC(=O)NCCC2CC(NC(=O)C=C3CCN(C)C3)C2)o1 c1(C(N2CCC(NC(CCc3c(C)ncs3)=O)(CF)C2)=O)c(C#N)cnn1C Oc1c(CSN2CCCCC(O)(C)C2)cc(Br)cc1Br c1(C(=O)NCC(C)CNC(c2occc2CN(C)C)=O)ccnnc1O C(=O)(C(F)CCC(C)C)N1CC(SCC)C1.C12CN(C1)CC(=O)N2.CO CN(C(=S)NCCCNS(C)(=O)=O)CC1CCOC1 C1(C)(C(=O)NCC2N(C(CC(CN(C)C)O)=O)CCC2)CCC(F)(F)C1 c1(C(=O)NCCC2(O)CCCN(C(C(COC)OC)=O)C2)ccn2ccnc2c1 c1(CC(=O)NCCC(C)NC(C2CCO2)=O)c(F)cccc1F C1(CN(C(=O)CC2CCN(C(=O)C=Cc3cc[nH]c3)C2)C)CCCCO1 c1(C(=O)NCC(CNC(C(CCC)OCC)=O)OC)c[nH]c(=N)c2[nH]ccc12 c1(CN2C(C)CCC2C(N2CC(=O)NC(=O)C2)=O)ccc([N+](=O)[O-])c(O)c1 N1(C(C)=O)CCN(C(c2ccc(C)c(-c3cnn(C)c3)c2)=O)CC1C(F)F CC(C)(C)C(CO)C(=O)NC1C=CC(CC(N2CC3OCC(CO)C3C2)=O)C1 CN1CCN(C)C(C(=O)NCCC2CCC(NC(c3nc(Cl)cs3)=O)C2)C1 C1(O)(CN(C)C(C2COC(=O)C2)=O)CN(C(=O)CC23CCCC2C3)C1 c1(C(=O)NC2(CNC(CC(C)C)=O)CCOC2)cc(=O)c2cc(F)ccc2o1 c1(CNC(C(C)OC(C)=O)=O)cc(C(=O)NC(C)(CO)C2CC2)n(C)n1 c1(C(N(C(C(=O)OC)C)CC2C(C(=O)OCC)C2)=O)ccncn1 c1(N(C)C)ccc([N+](=O)[O-])c(C(=O)NC(CNC(C2COC2)=O)C2CC2)c1 c1(C(N(C2CN(C(C3C(OCC)C3)=O)C2)C)=O)cc(S(=O)(=O)N2CCCC2)c[nH]1 C(=O)(C1=NOC(C)C1)N1CCC(N(C(CC2(OC)CCC2)=O)C)C1 N1(C(CC2CC(CC)C2)=O)CC2CCC1CC2NC(c1ncc[nH]1)=O C(=O)(C(C)(C)CCCF)NCC1(C(C)NC(c2cc(C)n(C)n2)=O)CC1 N1(C(C2(OCC)CCOCC2)=O)CC2CC(C1)N(c1cc(C)nc(C(C)C)n1)C2 N1(C(C(F)(F)Sc2cn(C)nc2)=O)CC2(C1)CN(C(=O)CC1C=CCC1)CCO2 c1(C(N2CCC(NC(Cc3cc(C)[nH]n3)=O)(CF)C2)=O)ncnc(O)c1Br CC1CC(C(=O)N2CCC(N(C)C(c3c(C(F)(F)F)cnn3C)=O)C2)=NO1 c1(C(=O)NCC(C2N(C(C=CC(CC)=CC)=O)CCC2)(C)C)ccc(C)c(O)n1 C(=O)(C1=C(C)CCCC1(C)C)NCC(C(C)(C)C)NC(CC(CC)(C)C)=O c1(C(C)=O)cc(Br)ccc1NC(=O)Cc1ccc(CNC(c2ccon2)=O)cc1 n1(CC)nc(C)cc1C(=O)NC1CCC(NC(c2c[nH]c(C(F)(F)F)c2)=O)CC1 C1(C(=O)NC(C)CCNC(C2(C)CSC2)=O)CCc2cnn(C)c2C1 c1(CCC(=O)N(CC(CNC(C2C(CCOC)C2)=O)C)C)cccn1C N1(C(C)CC(C)C(N2CCC(CN=[N+]=[N-])C2)=O)CCC2(C=CCO2)CC1 C(=O)(C(F)CCC(C)C)NCC(CCOC)NC(c1ccncc1N)=O c1(NC)ccc(F)cc1C(=O)NC(C1CCN(C(=O)C(C)CSC)C1)C O(NC(=O)CCC1CCCCC1)C(=O)NCCNC(C(C)(C)O)=O Cc1cc(C(=O)N(C)CC2(O)CCN(C(C3C4COCC34)=O)C2)n(CCO)n1 CCC(CNC(C1CNC(=O)CN1C(=O)C=Cc1ccncc1)=O)CC(C)C C1(CNC(CCNC(C)=O)=O)CN(C(=O)C(C)c2ccsc2)CC1C CC12CCOC(C(N3CCC(F)(C(=O)NC4(CCF)CC(O)C4)C3)=O)(C1)C2 N1(C(c2cc3cccnn3n2)=O)CCC2CCN(c3nc(Cl)ncc3F)CC2C1 c1(C(=O)NCC(C)(C(C)C)NC(c2c(C)nc(CO)o2)=O)onc2ccccc12 C(=O)(CCCC(=O)N1CCCCC1C(=O)NCC1OCCCC1(C)C)OC c1(-n2c(C3(c4cccc(Cl)c4)CC3)nc(C(C)C3CC3)n2)cccc2cnccc12 C1(OC)CC2CN(C(=O)CCc3cncnc3)Cc3ccccc3N2C1 C(CCC)(C(=O)N1CCC(C)(NC(c2cc(OC)no2)=O)C1)=CCC C1(O)(CN(Cc2onc(CC)n2)CC)CCCN(C(=O)C(C)(C)CF)C1 C(=O)(C(CC(=O)OC)N(C)C)NCCCCNC(C(CCC)O)=O c1(NC)ncc(C(=O)O)cc1NC(C1CCCNCC1F)=O c1(N2CC3(CCC(C(N(C)CC4CCCO4)=O)O3)C2)ccc([N+](=O)[O-])c(O)n1 CC(C)C(F)C(=O)N(C)CC1(C)CCCC1NC(=O)CSc1ccc(O)cc1 C(c1ccn(C)c1)=CC(=O)NC1C(NC(CCc2scc(C)n2)=O)CC1 N1(C(c2c(C)c(F)cnc2)=O)CC(C)N(C(=O)C(C)C(C)C)C(C)C1 N1(C(CCCSC)=O)CCC2CCCC12CNC(c1cn(C)c(C)n1)=O c1(NC(C(=O)NC2C(SCC)C2)=O)cc([N+](=O)[O-])ccc1COC CCC1=NOC(C(N2CC(CNC(c3ccccc3Br)=O)C2)=O)C1 N1(C(CCOCCCNC(CC(C)O)=O)=O)CC(C2CC2)CC(C)(C)C1 C1(F)(CNC(c2c(CCC)n(CC)nn2)=O)CCN(C(c2ccc(Cl)o2)=O)CC1 N1(C(C2CCCOC2)Cc2cn(CC(=O)NC)nn2)CC2CC3CC2C1C3 N1(C(c2nc(OCC)oc2)=O)CCN(C(=O)CC2CC(OC)C2)CC1CC CC1CN(C(=O)CCN2CCN(C)CC2)CCC1NC(=O)C(C1CCC1)C1CC1 C(C)(CO)(C(=O)NCc1nc(C#N)cs1)NC(Cc1cc(C)sc1)=O N1(C(=O)CCF)CC2CC(C1)N(C(=O)C(Cc1ccccc1)C1CCCC1)C2 N1(CCC(=O)NCC(C)CNC(c2cn(C)nn2)=O)CCc2ccccc2C1 C1(NC(C(CN(C(CCCCSC)=O)C)C)=O)C(O)C2CCCC12 C(=O)(CCC(=O)NCC1CC1)NC1C(C)(CN(C(C(F)OC)=O)C)CCC1 N1(C(CSC)=O)CCC2(CC1)CC2(CO)CNC(=O)Cc1sccc1Cl c1(N)cccc(S(=O)(=O)N2CCCC2)c1.C(=O)(CP(C)(C)=O)NC(C)CCSC c1(OC)c(C)csc1C(=O)NCC#CCNC(c1cc[nH]n1)=O C1(C(N2C(C)(C)C(C(N)=O)CC2)=O)CN(C(C2CCCCS2)=O)CCC1(C)C c1(C(=O)NC(c2cccc(F)c2F)C)n[nH]c2c(=O)n(C)cnc12 C1(C(N(CC(C)CNC(=O)CSCC(N)=O)C)=O)CCC2(CCC2)O1 c1(C(=O)NC2C(C)(C)N(C(C3CC(F)(CO)C3)=O)CC2)ccnc2ccccc12 c1(CN(C)Cc2cccc(C)c2)cc(Cl)c(Cl)n1C c1(N(N2CCC2c2cn(CC(=O)O)nn2)C)cnn2c1OCC(C)(C)C2.C=O Cn1cc(CC(=O)NC2(C)CCN(C(c3ccc(O)nc3)=O)C2)c(C(F)(F)F)n1 C(CN=c1[nH]c2ccc(O)cc2s1)N(C(c1cccc([N+](=O)[O-])c1)=O)C1CC1 N1(C(c2cn(CC)nc2)C(=O)NCC2CC2)CCC(C)C2(CCC2)C1 c1(C(C(=O)NCCN(C(CCSCC)=O)CC(C)O)C)ccccc1F C(=O)(C(C)(C)C1=CCN(C(c2ccc(=O)oc2)=O)C1)Nc1c(C)cnc(Br)c1 C1(CNC(CCSC)=O)CCCCC1NC(C1CC(=C2CCC2)C1)=O C1(NC(c2nc(C(=O)OC)oc2)=O)CCN(C(c2cnc(Cl)s2)=O)C(C2CC2)C1 C1(OC)CC(CNC(=O)N(CC(C)C)C)C1(C)C.c1(OC2CC2)ccccc1 CN1CCC(C(N2CCC(CNC(=O)COC3(C)CCCC3)C23CC3)=O)C1=O C1(C)(CC)CN(C(C2CC(NC(c3ccc(C#N)[nH]3)=O)C2(C)C)=O)CCO1 C(=O)(CC1C(=O)N(C)c2ccccc21)N(C)CCN(CCO)C(C1OCCO1)=O C1(C(=O)NC2(C(=O)NCCSC(F)F)C(C)C2)CN(C)CCN1C Cc1cc2[nH]c(C(=O)NCC(C)(C)CN(C(=O)C(C)N3CC(C)C3)C)cc2o1 c1(CNC2CCC(NC(c3c(C)cccc3)=O)CC2)cncc(C#N)c1 c1(CNC(C2(OC)CCS(=O)(=O)C2)=O)cnn2c1CN(C1CC3CCC1C3)CC2 c1(NC(CC=CC=C)=O)cccc(N(C2CN(C(=O)C#CC3CC3)C2)C)c1 C1(OC)CN(C(c2cc(C)nc(C)c2)=O)C(C)(CNC(c2cc(=O)cc[nH]2)=O)C1 c1(C(c2n(CCCCCC)nnn2)NC(c2cnoc2)C)c(C)nn(CC)c1C N1(C(C(C)NC(C(C)SC)=O)=O)CCC(C(C)(O)CNC(=O)COC(C)(C)C)CC1 c1(C(C(=O)NC2(C)CCN(C(C(C)C(F)F)=O)C2)=O)cc(Cl)cc(Cl)c1 c12ccncc1S(=O)(=O)N2.c1(CCC2CCN(CC)CC2)ccc(C)cc1 c1(C(C)NC(C2CCCN(Cc3cccc(C#N)n3)C2)=O)ccc(F)c(Cl)c1F c1(OCCCC)ccc(OC)cc1.C12CCN(C1)C(=O)COCC(=O)NCC2 N1(C(COCCOCC#C)=O)CC(C(=O)N(CC(CC)CO)C)(CC)C1 c1(C(CNC(=O)Cc2cnc[nH]2)NC(c2ccc(C)o2)=O)ccc(C2CC2)cc1 N1(C(C(CNC(c2cc(Cl)cn2C)=O)N(C)C)=O)CCOC2CCCC12 C1(COC)(CNC(C2CNC(=O)N2)=O)CCCN1C(=O)CCc1ccccc1 N1(C(C(C)NS(C)(=O)=O)=O)CCOC(CNC(c2cc(CC3CCC3)c[nH]2)=O)C1 Cc1cc(F)ccc1N(C)C(=O)N(C1CC1)CC1(c2ccc(Br)cc2)CCCC1 C1(C(NOCC(=O)N(CC#C)C2CC2)=O)COCCC1C C1(C(=O)NCC2(CCNC(=O)CSc3nncs3)CC2)CC12CCCCC2 CC1CCN(C(C2CC(O)CCN2C(c2cnnc(O)c2)=O)=O)C1(C)C C1(CNC(c2c(C)nc(CC)s2)=O)CN(C(=O)C=Cc2nccs2)CCN1C c1(C(N(C2CCN(C(C)=O)C2)CC)=O)ccc(F)cc1C c1(C(C)(F)F)cccc(C(=O)NC2CCCC(NC(=O)CC3OCCCO3)C2)n1 N1(C(CCCC(=O)OCC)=O)CCC(C2(NC(=O)Cc3nnc(S)n3C)CC2)C1 Cc1cc(=NC(Cc2cccnc2)C2CC2)[nH]c(=NCc2conc2C2CC2)[nH]1 C1(C)(NCC=CC(=O)N(CCC(N)=O)CC)CCCCC1C c1(OCC(=O)NCC(C)CNC(=O)CC2(C(F)F)CC2)ccc(Br)cc1 CC1(C)CN(C(c2ccc(F)cc2F)=O)CCC1NC(c1csc(Cl)c1)=O N1(C(=O)CNc2ccccn2)CCOC(CCNC(C2CC(CF)C2)=O)C1 C1(NC(C2SCCS2)=O)CC2CN(C(=O)CC3C=CCC3)CC12 c1(NCC(C)OC)cccc2c1OCCC2NC(=O)Nc1ccco1 c1(C(N(CCC(=O)NC2CCC2C)CC=C)=O)cn(C)c(C)n1 C(=O)(C#CC1CCCO1)NC1CCCCN(C(Cn2ncc(CC)c2)=O)C1 N1(C(C2(CNC(C3C=CCCC3)=O)CC(=C)C2)=O)CCC(F)(F)C(F)C1 CN1C(=O)CCC1C(=O)NCC(C1CCCN1c1nc(C(C)(C)C)ns1)(C)C C1(SCc2cn(CC(=O)NCc3ccc(NC(C)=O)s3)nn2)CCOC(C)(C)C1 N1(C(C2(C#N)C(C)C2)=O)CC2(CC(CNC(c3ccc(F)c(C(N)=O)c3)=O)C2)C1 C1(C(=O)NC2CC(C(C)O)C2)CC2(CCN1C(c1cncc(Cl)c1)=O)CC2 c1(C(=O)O)ccc(Cl)c(Br)c1.c1(SC2CC2)cccc(C(=O)OCC)c1 c1(C(N(CCC)CCNC(C23CCC(C2)C3)=O)=O)ccc(F)c(OCC)c1F c1(C(=O)OCC)cn(CC)[nH]c1=NC(=O)c1ccc([N+](=O)[O-])cc1.C12CC(C1)C2 N1(C(c2ccc(OC)o2)=O)CCC2(CC1)CC2C(=O)N(C)CC1(N(C)C)CC1 C(=O)(CCCCC(C)(C)OC)N1CCCC(O)(CCNC(C(CC)C)=O)C1 c1(C(C)C)ccc(C(=O)NCC23CC2CN(C(=O)CCn2cccn2)C3)cn1 CC(C)C(C(C)NC(=O)CSCCN(CC(F)(F)F)C)NC(=O)CCNC=O C=C(C)CC(C(=O)NCC1OCCC1CC)NC(C1CCCCN1C)=O c1(OC)cc(C(N2CCC(C)(NC(c3ccccc3F)=O)CC2)=O)cc(F)n1 O=C(C1=NOC(CNC(=O)Cn2nc(O)ccc2=O)C1)NC1CCCCCC1 c1(C(=O)NC2CN(C(=O)CCN3CCCCC3=O)C2)cc(F)cc2nccnc12 c1(C(N2CCC(NC(C(C)c3cccs3)=O)C2)=O)ccncc1C(F)(F)F c1(C(C)CC(N2CC3CC2C3NC(=O)Cn2cnnn2)=O)ccc(F)cc1F C1(NC(C2(NC(=O)Cc3cccnc3F)CCCCC2)=O)Cc2nccn2C1 n1(C(C(=O)NCCN(CCOC)C(C2CCOC2)=O)C)cc(C)cn1 C1(CNC(CCCCOC)=O)(NC(=O)C(C)c2cccs2)CC2CCC1CC2 CC1CC(CNC(=O)C(C)Cc2cnc[nH]2)CN(C(C23CC4CC2C3C4)=O)C1 C(C1=CCCN(C)C1)NC(CC1(CNC(C(CC2CCC2)OC)=O)CCC1)=O N1(C(Cc2cc(C)sc2)=O)CC(C(=O)NCCC2CCCC2)CCC1(C)C CCCCC(CNC(c1csc(COC)n1)=O)NC(c1ccccc1Cl)=O N1(C(C2CC(C#C)(O)C2)=O)CC(NC(=O)C=Cc2cnn(C)c2)CCC1C CC1(C)CNCCN1C(=O)C(=O)Nc1ccccc1N1CCNC1=O N1(C(c2c(OC)c(C)sc2)=O)CC2CCN(C(=O)Cc3cnn(C)c3)CC2C1 N12CC(C3(CC3)C1)n1cc(nn1)CS(CC)(C)CC2=O.c1(C(CC)C=O)ccc(Cl)cc1F S(=O)(=O)(c1cc(C)ccc1-c1ccncc1)NC(CC)(C)CNC(C)=O C(CC(C)(C)C(=O)NCCc1cc(C(=O)NCC2(CCO)CCC2)no1)OC c1(C(N2CC(CNC(CC(=O)NCC)=O)C(C)C2)=O)cc(OC)ncc1F c1(C(N2C(C3(C(=O)OCC)CC3)CCCC2)=O)cc2cc(Cl)ccc2o1 C1(NC(N2CCCC2CCc2ccccc2)=O)C(O)C(O)CN1 CC(C)(C)C#CC(=O)NCC1(F)CCN(C(=O)CSc2ccccc2)C1 N1(C(C(C)OCCC#C)=O)CCCC(n2cc(CNC(=O)CCC3CC3)nn2)C1 n1(CC(=O)NC(C)CCCNC(=O)CC2CCCCN2C)ccc(=O)n(C)c1=O N(C1CSCc2ccccc21)C(CC(C)(C)C)c1ccc(Cl)cc1.C1CC(=O)N1 C1(NC(C(n2cc(Cl)cn2)C)=O)CCN(C(=O)C#CC2(C(F)(F)F)CC2)CC1C c1(C(=O)NC2C(NC(c3cncs3)=O)COCC2)c[nH]c2ccccc12 C12(C(=O)NC(CCN(C(c3cc(COC)cn3C)=O)C)(C)C)CC(C)(C1)OC2C c1(N2CCC(C(N3CC(C)OCC(C)(C)C3)C)C2)ncc(S(C)(=O)=O)cc1Cl N1(C(CNC(=O)OCC=C)=O)CCN(C(C2C=CC(CCC)C2)=O)CC1CO C1(F)(C(=O)NCCCOCCCC)CN(C(=O)C(C)n2ccnn2)C1 C1(CNC(C2(OCC)CC2)=O)CCCN(c2cncc(Cl)n2)C1 C1(C(=O)OC)Cc2cccc(NCCNC(=O)NCC(C)C)c2C1 Brc1ccc2nc(-c3cn(Cc4c[nH]c5cnccc45)nn3)nn2c1 C1(NC(CC=C=C)=O)CN(C(c2c(C)cccc2C)=O)CC(C)(C)C1 c1(C(=O)NC(C)CN(C(=O)CCn2cnccc2=O)C)cc2c(s1)CCCC2 Cc1c(NC(C2CCCC2CNC(C2(C(N)=O)CCC2)=O)=O)cccc1C#N c1(CCC(=O)NC(C2CCCN2C(C2CCC(=O)N2)=O)(C)C)ccc(Cl)cc1 c1(C(=O)NCC#CCNC(CC(=C)Br)=O)c(C)noc1C(F)F c1(C(N2CCC(NC(CCC3(C)CC3)=O)(CO)CC2)=O)cnc2n1C(C)CCC2 C1(SC(C(=O)NCCCC)CC)CNCC1(C)C CC1(C)CC(=O)NCC1C(N1CCN(C(c2c[nH]nc2F)=O)CC1CC(F)F)=O c1(C(C)(C)C)ccc(C(=O)NC2CCC2NC(c2ccccc2)=O)[nH]1 c1(C(=O)NCCOC2CN(C(C(C(C)O)N(C)C)=O)C2)ccc2cnccc2c1 CC1CC=C(C(=O)N2CC(C(=O)NC3CC(CCC(N)=O)C3)C(F)C2)CC1 c1(SCC)ccc(CC(N2CCC(CNC(=O)CCn3cc(C)cn3)C2)=O)cc1 N1(c2ccnc(C)n2)CCN(C2CCCN(C(=O)Cc3cnoc3)C2)C(=O)C1 N1(C(c2c(CC)ccc(Br)c2)=O)CCCN(C(=O)C(O)C(C)C)CCC1 N1(C(C#CC)=O)C(C(N2CCN(C(C)(C)C)CC2)=O)CC2CCCCC12 C(CC(C)C(=O)N1CC(NC(=O)CC2CCCCC2)CC1C)OC Cc1cc(CNC(=O)C(Cc2ccco2)NC(=O)CNC=O)nn1C C1(CC)CCCC1(C)C(=O)NCC(C)CN(C)C(c1cnc(C(F)(F)F)nc1)=O C1(NC(C(CC)C)=O)CCn2ccnc2C1.c12ccc(c(F)c1)CNC2=O C12CC(n3cc(CCC4(CC(C)C)COC4)nn3)CN1C2=O.C(=O)(C1CC1)OC c1(C(=O)NCC=CCNC(Cc2nc(C)sc2C)=O)ccnc(O)c1Br C(=O)(N=c1cc(C2CC2)[nH][nH]1)C1C2CN(Cc3cnn(C)c3Cl)CC21 C1(NC(c2nc(C)c(C)s2)=O)CCC12CCN(C(=O)C(O)(C1CC1)C1CC1)CC2 C1(C(=O)NCC(C)(C)OCCNC(COCCCCC)=O)NC(=O)C2CC12 C1(C(N(CCN(C(C(C)=CC)=O)C)C)=O)CCN(C2CCS(=O)(=O)C2)CC1 c1(C(N2CCC(C)(NC(c3cc(Br)no3)=O)C2)=O)ccc(-n2cccn2)c(F)c1 N1(C(c2c(CC)oc(C)c2)=O)C2CCC1CN(C(=O)C(C)(C)Cc1cnn[nH]1)C2 CC1(C)COCC(C(=O)NC2CC2NC(c2sccc2F)=O)O1 c1(CNC(N(C2CS(=O)(=O)N(C)C2(C)C)CC)=O)coc2ccc(Cl)cc12 C=CCCC(C(=O)N(C)Cc1cccc(F)c1)N.C(=O)NC=O c1(OC)ccnc(C(=O)NC2CN(C(c3cncc(C4CC4)n3)=O)CC2C)c1 C1(NC(C2(CC)CCCN(C(C3CC(CC)C3)=O)C2)=O)CCCC2(CCC2)C1 Cc1ccc(Cl)c(Nc2cc(C(F)F)cc(Cl)n2)c1.C1C(=O)N1C C=CC1CCN(C(=O)CN(C(=O)CC2CCCOC2)CC2CC2)CC1 N1(CC(N2CC=CC2CNC(c2cc(Cl)c[nH]2)=O)=O)CCCCC(O)C1=O Cc1c(C(N2CCC(NC(=O)CC3CCCC3)C3CC23)=O)cncc1Br C1(C(N2CC(C)C(NC(=O)C3=CC(C)(C)C3)C2)=O)CC2CCC(C1)S2(=O)=O c1(CNC(C2CCC(=O)NC2)=O)cnn2c1CN(Cc1ccc(O)cc1Cl)CC2 c1(C(=O)NCC2CN(C(C)=O)CC23CCC3)[nH]nc2c1CCCC2(C)C c1(CC(=O)NCC(CC)(C)NC(=O)C(F)C(F)(F)F)ccc(C)cc1C CN1CCN(C(=O)Cc2ccc(F)cc2)C(CNC(=O)CN2CCC(=O)NC2=O)C1 Cc1coc(C=CC(N2CCN(C(C3CC(C)C3)=O)CC2)=O)n1 C1(C(=O)NCC(n2cc(C(C)O)nn2)C)(Cc2ncccc2Br)CCOCC1 c1(CN2CC(CNC(=O)NCc3c(C)cccc3O)C2)ccc2c(c1)OCO2 N1(C(C(C)CN(C)C)=O)CC(C(=O)NC2(C(N)=O)CC2)CC12CCC2 N1(C(C(CC(=C)C)OC)=O)CCC2(CCCC2NC(c2cn(CC)nc2C)=O)CC1 Cc1cccc2cc(C(=O)NC34CC(NC(c5cnn(CCF)c5)=O)(C3)C4)oc12 C1(CNC(C(CC)Oc2ccccc2Cl)=O)(CO)CCCN(C(=O)CC(C)C)C1 S(=O)(=O)(c1ccc(NC2CCCCCCC2CO)c(C#N)c1)NCC(C)(C)OC Cc1nn(C)c(F)c1C(=O)NCCCC1CCCCN1C(=O)CC1C=CCC1 C12(NC(COCCCC)=O)CN(C(=O)C=Cc3ccccc3)CC1CS(=O)(=O)C2 N1(C(C2(CC#C)CCOC2)=O)CCC(C(C)(C)C)(CNC(c2nnn(C)n2)=O)C1 N1(C(C(C)O)=O)CC2CC(NC(=O)COc3ccc(F)cc3Br)CC(C2)C1 Cc1ccnc2c(C(N3CC(O)(CN(C)C(C4CCN(C)C4)=O)C3)=O)cnn12 C(=O)(CC1=CCN(C)CC1)N1CC(C(C(=O)NCC2N(C(C)=O)CC2)O)C1 C1(C(N(CC(=O)NC(c2c(C)ncs2)C)CC2CC2)=O)CCCCC(=O)N1 c1(C(=O)OCc2c(C)nns2)cc(F)c(-n2ccnc2)cc1I S(=O)(=O)(c1cccc(=NCCn2cnnn2)[nH]1)N1C(CNS(C)(=O)=O)CCC1 c1(CCC(=O)NCC(CNC(C2(O)CCOC2)=O)OC)cscc1Br CCC(O)(CNC(=O)C(C)N(C(c1cnn(C)c1OC)=O)C1CC1)CC N1(C(C(C)CN2CCOCC2)=O)CC(NC(c2c(C3CC3)cnn2C)=O)C(C)C1 c1(C(N(C)CCN(c2ccnc(C#N)n2)C)=O)cc(F)cc2nccnc12 S(=O)(=O)(c1cnccc1N1CCC2(C1)OCCO2)NCCc1ncc(C)cc1C Cc1nc(SC(F)F)sc1CC(=O)NCSCC(=O)NCCC(C)NC(=O)C(C)O C1(NC(C(CC)C)=O)CN(CC2CC(=O)N(C(C)=O)C2)CC1(C)C C(=O)(C(COC(C)C)N(C(=O)CC(C)c1ccco1)CCO)N1CC(C(=O)NC)C1 C1(CNC(c2scc(OC)c2)=O)CN(C(C2(C)CC2(Cl)Cl)=O)CCO1 C(C(=O)N=c1cc2n([nH]1)CCCC2)(C1CCCCC1)NC(c1occc1C(=O)O)=O N1(C(C2(CC)CCCO2)=O)CC2(CCCC(CNC(c3ccc(Cl)cc3)=O)O2)C1 CC(C)C(C(C)NC(=O)CO)NC(=O)CCNC(c1cc(-c2ccco2)[nH]n1)=O c1(N(CCC(N2C(C)CC(F)C2)=O)C(=O)CC2CCS(=O)(=O)C2)cccc(C#N)c1 N1(C(c2cc(CCC)[nH]n2)=O)CCN(C)C(C(=O)NC2CC=CCC2)C1 C1(NC(C=C(C)C(C)(C)C)=O)(CF)CCN(C(=O)CC2C=CS(=O)(=O)C2)C1 C1(NC(c2ccc(C)nc2)=O)CC2CN(C(c3cnc(Cl)s3)=O)CCN2C1=O c1(C(=O)NCC2CCC(NC(C(C(C)C)N(C)C)=O)C2)ccc(=O)n(O)c1 C1(NC(C2C(C(C)C)OCC2)=O)CC=CCC1C(N1CCCCC1CCO)=O C(C(C)C(C)C(=O)NCC1=CCN(C(c2cc(O)nc(OC)n2)=O)CC1)OC N1(c2n(CC(C)C)c(C3CCOC3)nn2)CCC2(CC1)C(O)CC(C(F)(F)F)O2 C1(NC(Cc2cn(CC)nc2)=O)CCC(C)(NC(=O)CC2CCC(=O)NC2)CC1 Cc1ccc(N2CC(C(=O)NCC3CCNO3)CC2=O)cc1C C(=O)(C(F)CCC(C)(C)C)N(CCN(C(c1cn(CC=C)nc1)=O)CC)CC N1(C(C(F)=CC)=O)CC(C)(C)OCC1CNC(=O)COc1cc(F)ccc1F N1(C(C(C)CC(N)=O)=O)CC(NC(=O)C(C)N2CCCC2)CC12CCCCC2 CC1CN(C(C2(F)CCN(C)CC2)=O)CCC1CO O=C(CCCC(F)C(=O)O)N1CCCCC1c1ncc(-c2cccc(Br)c2)[nH]1 c1(OCC)cccc2c1CN(C(C1CCN(C(=O)CC3=CCCC3)C1(C)C)=O)C2 CCC(C)CCCC(=O)N1CCC(C)(C)C(NC(=O)Cc2cc(C)ccc2F)C1 C1(CNC(C(C)O)=O)CCC2(CN(C(c3ccc(F)cc3O)=O)C2)O1 C12(NC(N3CC(O)(CCCCNC(c4c(C)occ4)=O)C3)=O)CCC(C)(CO1)C2 c1(C(=O)NC2CC(F)(CNC(c3[nH]nc(OC)c3Cl)=O)C2)nc(O)nc(O)c1N N1(C(C(C(C)C)SCC)=O)CC2(CCN(C(c3ccc(Cl)c(NC)n3)=O)C2)C1 N1(C(C2(C)CC2CO)=O)CCCC1(C)C(=O)NCCC1CCCOC1 C1(c2c(CC)cccc2)CCOC2(C1)CN1N(C)C(CCC2)C1 c1(C(=O)NCC2CC(NC(C(OC)OC)=O)C2)ccccc1C(C)(C)C C1(CNC(C(C)NC(C)=O)=O)CN(C(C2CC2C2(C)COC2)=O)CCC12CCC2 C1(C(N2CC=CC(C(=O)NCC(C)(C)OC)C2)=O)CCC(O)CN1C c1(C(N2C(C)CC2C(=O)N(C2CN(C3CC3)C2)C)=O)c[nH]c2nccc-2c1 C1(CCC)CN(C(=O)C=CCC2(N(C(=O)CS(=O)CC)CC)CCC2)CCO1 c1(C(=O)NCCCN(C(c2c(CC)nsc2N)=O)CC)ccn2c(C)ncc2c1 N1(c2c(SC)cnc(OC)n2)CCOC2(CN(C(c3cncs3)=O)C2)C1 c1(NCC2(C)CC2Br)cc(Br)ccc1S(=O)(=O)NCc1nc2ccc(Cl)cc2[nH]1 CC1(C)CN(C(C2CC(O)C2)=O)CC1NC(=O)CC(C)(O)c1ccccc1 CCC(COC)C(=O)NCC(CC(=O)NC(C)(CO)CO)C1CCC1 N1(C(CCC(CCC)CC)=O)CCOC2(CCSCC2)CC1 CCS(=O)(=O)NC(C)C(=O)N(CC(C)(C)NC(=O)C(C)c1ccco1)C C1(NC(c2n(CC)nc(C(C)C)c2)=O)CCCN(C(=O)C2=CCCO2)CC1 CC(C)(C)CCC(=O)N1CC2CC(C(N3CCC(c4cc[nH]n4)C3)=O)(C2)C1 c1(CC)nn(C)c(CC)c1NC(C)CNC(c1cccc(C(F)(F)F)c1)=O C(C1CCOc2ccc(Br)cc21)NCc1n[nH]c(C)c1C c1(C(=O)NCC(C)(CO)NC(C2CC3CC3C2)=O)nc2n(c1Cl)CCCC2 C12(CNC(=O)C3=NOCC3)CN(C(=O)C=Cc3cccnc3)CC1CS(=O)(=O)C2 Cc1cc(C)c(C(=O)NCCC2=CCN(C(C3(C#N)CC3)=O)CC2)c(S)n1 N1(C(C(C)Cn2cccn2)=O)CC2(CC(CNC(C3(Cl)CC3(F)F)=O)C2)C1 C1(NC(CCSCC(C)C)=O)CC(NC(c2cnn3c2CCC3)=O)C12CCC2 C1(N(C(C2C(=C)C2)=O)CC)CCN(C(=O)C=Cc2ncc[nH]2)CC1 N1(C(CSCC)=O)CCN(C(=O)Cc2cc(O)nnc2O)CC1c1ccccn1 CC1CC(NC(=O)NCCCCS)CN1C(C(=O)CC1OCCCO1)CC Cc1cc(C(N2CCC(NC(C3(N(C)C)CC3)=O)CC2C)=O)c(C)cc1Cl c1(OC)cc(C(N2CC(NC(C3(C)CCCS3)=O)C(SC)C2)=O)cc([N+](=O)[O-])c1 C1(NC(c2n[nH]c(C)c2C)=O)CC2CC1N(C(c1cccc(C(N)=O)n1)=O)C2 C1(CC)(NC(=O)CCF)CCN(C(=O)CC(O)CCNC(=O)OC(C)(C)C)CC1 c1(C(=O)NC(CCC(=O)OC)CCOC)cc2cn[nH]c2cn1 CCC(C(=O)N1CCC(NC(c2sc(-c3cccs3)nc2C)=O)C1)C(C)(C)CC c1(C(=O)NC2CC2C(N2CCS(=O)CC2)=O)cc(O)nc(O)c1 C12(C(=O)Nc3c(COC)noc3)C(NC(=O)CCC3CCC(=O)C3)C3CC1C2C3 C(=O)(CCCCCN(C)C)N(CCC(=O)NCC1CCC(CC)O1)CCCO N1(C(Cc2ccc(C#C)cc2)=O)CCN(C(=O)CSCC)C2COCC12 CC(C)(F)CCC(=O)NC1CCCC(CC(N2CCC3C(O)CC23)=O)C1 CC(C)CCCCC(=O)N1CCCC1CCC1CCCCN1C(c1cnns1)=O c1(CNC(N2CCN(S(=O)(=O)C3CC3)CC2)=O)cccc2cncn12 C1(NC(CC2CC(=C)C2)=O)CCN(C(=O)CCC2CCCN2C)CC1 C1(CC)CN(C(=O)C=Cc2cccc(CO)c2)CCC1NC(c1ccc(C)[nH]1)=O C12(NC(C(CC)OC)=O)COC(CNC(c3c[nH]nc3-c3ccncc3)=O)(C1)C2 N1(C(C(CC)CC2CCCCC2)=O)CC(NC(=O)C=CCO)CC12CCOCC2 C1(C)(C(N(C(C=C)C2CC2)C)=O)C=CCN1C(C1OCCC1C)=O C1(C(=O)NC(CNC(c2cnn(CC)c2C)=O)CO)CN(CP(C)(C)=O)C1 C1(NC(C2C(NC(C(C)=C(C)C)=O)CC2)=O)C(O)CC1O c1(NS(CCCC)(=O)=O)cnn2c1CN(C(=O)CO)CC2 C1(C(=O)NC2CCC(C)(CNC(c3cnc(C(F)F)s3)=O)C2)CCC2(CCC2)O1 C(CC(=O)NC(c1cccs1)C)N(C(=O)CN1CCCC1)CC#C C(CC(C)(C)CC(=O)NC(CCN(C)C)C(=O)N1CC(OCCF)C1)OC Cc1cnc2[nH]cc(C(C)NCC3(NC(=O)OC(C)(C)C)CC3)c2c1 CC1CN(C(=O)CC23CCCN2CCC3)CC1(C)CNC(=O)C=C(Cl)Cl C1(C(=O)NCC(N2CCC(C3(C)N=N3)C2)=O)(CC)CCCC1O Cc1cnncc1COC(C1CC1C(F)(F)F)=O C1(C(=O)NC(CNC(c2c(CC)nc(C)o2)=O)CO)CC2(CO1)CC(F)(F)C2 n1(CC(=O)NCC2CN(C(c3cc(CC)sn3)=O)C(C)C2)c([N+](=O)[O-])cnc1C Cc1c(C(N2CC(C)N(C(=O)C=CCF)CC2C)=O)oc2ccc([N+](=O)[O-])cc12 c1(C(=O)NCCCCCC2CC2)ccccc1-n1cc(-c2cccc(Br)c2)nn1 C1(C)(C(=O)NCC#CC(=O)NCCCCOC(C)C)CCCOC1 C(=O)(C(CCC1CC1)NC(=O)CSCC(F)F)NC1(C(C)C)CCC1 N1(C(c2nc(OCC)sn2)=O)CCC(NC(=O)CC(C)(C)O)CC1C N1(C(C(C)=C2CCC2)=O)CCC(O)(CNC(c2cnc(-c3cccnc3)s2)=O)C1 CC(F)(F)C(F)C(=O)NCC1(C)CCCN(C(=O)CCS(C)(=O)=O)C1 N1(C(CC(OCC)OC)=O)CC2COCC2(Cn2cc(C(C)(O)COC)nn2)C1 c1(C(=O)NC(C2CCN(C(COC(C)=O)=O)C2)C)cc([N+](=O)[O-])c2nsnc2c1 N1(C(c2c(N)ccc(C)c2)=O)CCCC2(CC(NC(C3CC(Cl)(Cl)C3)=O)CO2)C1 c1(NS(C)(=O)=O)ccc(C(=O)NCCn2ccc(NCC3CC3)n2)cc1I C12(NC(C(C)C(=O)N3CCOCC3)=O)CCC(NC(=O)CC34CC(C3)C4)(C1)OC2 C(=O)(C(F)C(=O)NC(C)C(CO)NC(c1cnn(CC(F)F)n1)=O)OCC CCC(C)C(O)CC(=O)NOC(CC(C)C)C(=O)NCC.[nH]1cncn1 S(=O)(=O)(c1ccc(NCC2CCSC2)nc1)NC(c1cnc(C)s1)C1CC1 N1(C(CCc2c(CC)cccc2)=O)CCCN(C(=O)CC(C)COC)C(C)C1 Cc1cc(C#N)nc(=NCCCC(C)NC(=O)C2c3ccccc3OC2C)[nH]1 C1(C2CCC2)(Nc2cc(N(CC(=O)NCCCC)C)nc(C)n2)CC1(F)F N1(C(C2CC(CC)N(C(c3cc(C)cc(O)n3)=O)CC2)=O)CCC12CCCSC2 c1(C(N2CC3CC(NC(C(=O)NCC4CC4)=O)C3C2)=O)cnc2c(c1)CCCC2 C1(OC)CCCN(C(=NCCC(=O)Nc2ccncc2)NC2CCCC2)C1 CC(CC(=O)N1CCOC2(CC2)C1)C(C)(C)NC(=O)CSc1nc[nH]n1 c1(C(N2CC(CNC(COCC)=O)C(O)C2)=O)ccc2[nH]c(NC(C)=O)c(C)c2c1 C1(NC(c2cccc(C)n2)=O)CCN(C(C2CCC(C)C(C)C2)=O)CC1C CC(Cc1ccncc1)C(=O)N(C)CC1(CNC(=O)C(=O)N(C)C)CC1 c1(C(=O)NCC(N2CC(O)(C(C)NC(c3csnn3)=O)C2)=O)ccc(Cl)cc1 c1(CN(C(CCN(C)CCO)=O)CCCc2ccsc2)cc(O)ncn1 C=CCC(C(=O)N1CCC(c2nnc(S)n2-c2ccccc2)CC1)C(C)C C(=O)(C(O)CCC(C)C)N1CC(C(C)NC(c2c(C)n(C)cc2)=O)C1 c1(CC(=O)NC(C2CCN(C(=O)CC(F)F)CC2)(C)C)ccc(O)c(C(N)=O)c1 N1(C(CC(C)OC)=O)CCC(CCOC)(NC(c2[nH]cnc2C)=O)C1 c1(CCC)n[nH]cc1C(N1CC(CC(C)NC(=O)CN(C(=O)C(C)C)C)C1)=O S(=O)(=O)(c1ccc(C(F)(F)F)c(F)c1)Nc1cccc(CCC#C)c1 c1(C(=O)NC(C2N(C(C3(C=C)CC3)=O)CCCC2)C)ccc(Cl)c(OC)c1 C(=O)(C(C(C)CC)NC(C1CCCN1C(N)=O)=O)NCCOCC=C c1(C(=O)NC2CCCC(CNC(C3(c4cc[nH]n4)CC3)=O)C2)ccnc(Cl)c1O N1(C(c2ccc(CC)c(N)c2)=O)CCC(C2CC2)C1CNC(CCC(=O)NC)=O C1(CC(=O)N(CCN(C)CCO)C)CN(C(=O)Cc2ccc(F)cc2)CCO1 Cc1cc(C(=O)NC2CC3CC2N(C(c2c(N)cccc2Cl)=O)C3)cc(F)c1 Cc1c(CNC(=O)C(=O)NCCC2(O)COC2)noc1-c1ccccc1 c1(SC)cc(C(=O)NC(C)C(C(C)C)NC(C2CC2CC(C)C)=O)ccc1N CCCC(C(=O)NC1CCCN(C(=O)CC=CCc2ccccc2)C1)C(C)C c1(C(=O)Nc2ccc(Br)cc2C(=O)NC2CC2)cnn2c1NCCC2 CCC(C(=O)NC(C)(C)CC(=O)NC(C)CCC1CCCC1)C(C)C C1(C(=O)NCCc2ncc(C)o2)N(C(=O)Cc2cnoc2)CCCC1(C)C C1(C(N(CCn2ncc(C)c2)C)=O)CC2C=CC1N(C(=O)CCCCF)C2 C(CNC(c1ncc(C(F)F)s1)=O)(C(C)C)NC(C(C1CCC1)OC)=O C1(CC)(CO)CCCN(C(C2CC3CC3N2C(=O)C(C)C(=O)OC)=O)C1 c1(C(N2CCCCC(NC(C(C=C)(C)O)=O)CC2)=O)oc2ccc(F)cc2c1C C(=O)(C1=NOC2COCC12)N1CC(CN=c2snc(C(C)=O)[nH]2)C(C(F)(F)F)C1 c1(C(=O)NCC2C=CCN2C(=O)CCC2CCCO2)ccc2ccoc2c1 C1(C(=O)NCC#CCNC(c2cnc(C(=O)OC)s2)=O)Cc2nn[nH]c2C(C)C1 Cc1ccc2cc(C(=O)NC3CCC(CNC(=O)C(C(C)C)C(C)C)C3)[nH]c2c1 C1(C(=O)OCC)(NC2CCCN2Cc2nn[nH]n2)CC(C(F)F)C1 C(=O)(C(=O)N=S(C)(C)=O)N(C(C)CC1CCN(C(=O)C2=NOC(C)C2)CC1)C1CC1 N1(C(CCCN(C(C)C)C)=O)CC(CNC(c2oc(C3CC3)nc2C)=O)CC1C CC1CC2CCC(C(N3CCOCC(NC(=O)C=CCF)C3)=O)CN2C1 C1(C(=O)NC2CCCC(NC(c3nncc(OC)c3)=O)C2)CN2CCN1CC2C c1(OC)ccc(OC2CCCN(CC(=O)OCC=CCl)C2)cc1 C1(C(=O)NCCCCNC(c2cnc(CC3CC3)s2)=O)CC1C1CCCCC1 Cc1cc(F)cc(C)c1C(N1CCC(CF)(NC(C2CCCCC2C)=O)C1)=O c1(OC)ccc(Cl)cc1CC(=O)NCC12CC(CN1C(C1(C)CNC(=O)C1)=O)C2 CN1CC(C)(C)CC1C(N1CCCC1C(C)(C)NC(c1cc2c[nH]nc2s1)=O)=O C1(C(N2C(CCNC(Cc3nc(C)oc3)=O)CCC2)=O)CC12CCCC2 c1(CS(=O)(=O)N(C)C)ccccc1Cc1csc(Cc2nn[nH]n2)n1 CCCCCCCNC(=O)CC1CN(C(=O)C(CO)NC(C2(CF)CC2)=O)C1 c1(C(N(CC(CC)NC(=O)CNc2ncccn2)C)=O)n[nH]cc1C1CC1 C=CC1CN(C(=O)C(C)O)CC1NC(C1CCOCC1C)=O C1(NC(=NCc2c(C)cn(C)n2)NC2CCOCC2)CC(C2CCC2)C1 Cc1cn2cc(C(=O)NCc3cn(CC(F)(F)F)nn3)nc2s1 C1(C(=O)NCCS(=O)(=O)NC)CCN(C(=O)c2ccc(OC)o2)O1 CC12CN(C(c3ccc4c(n3)CCC4)C(=O)NC3CC3)CC(CO)(C1)C2 CC1(C)CN(C(c2cccnc2)=O)C(CNC(c2nc(Cl)sc2Cl)=O)CO1 CC(C)CCCCNC(C1(CCNC(c2ccc(O)nc2)=O)CCC1)=O c1(C(=O)OC)cc2n(n1)CCCC2NC(c1ccc(C)cc1Cl)=O N1(C(=O)CCN2CCC2)CC2CCC1CN2C(c1c(Cl)csc1Cl)=O c1(CC#N)c[nH]c2ccc(C(=O)OC)cc12.c12ccc(o1)CNC2C1CC1 C1(CC)(NC(c2ncoc2C)=O)CCN(C(c2cnc(O)cc2OC)=O)CC1 CCC(C(O)C(F)F)OC(=O)Cc1ccc(F)c(OC)c1 C1(C)(CNC(COC(C)(C)C)=O)CCN(C(=O)CCN2CCCCCC2)CC1 C1(CC(N2CC(C)(CC)C2)=O)CN(C(C2(CCOC)CC2)=O)CCO1 N1(c2nccc(C#N)n2)CCC2C(C1)NC(=O)N2CCOc1ccc(Br)cc1 n1(CC(=O)NC2(C)CN(C(C3C(C)CC=CC3)=O)C2)nc2c(n1)CCCC2 c1(C2C(C(=O)NC3CC(C(C)NC(c4nc(CC)[nH]n4)=O)C3)C2)ccc(C)nc1 C1(CC(=O)NCC(C)NC(=O)C=CBr)CC(C)OC1C C1(C2CCN(C(c3csc([N+](=O)[O-])c3)=O)C2)(NC(C2CC3CCCCC23)=O)CC1 C1(C(C)C)CCOCCN1C(=O)CC(c1ccccc1)NC(c1ccnn1C)=O c1(SCC(=O)NC(CCCCCNC(CC(=C)C)=O)CO)ncnc2[nH]cnc12 N1(C(COCCC#C)=O)CCCC(N2CCN(C(=O)CCC3CC3(F)F)CC2)C1 C#Cc1cccc(C(=O)NCC2CC2NC(=O)C2=CC(C)(C)C2)c1Cl C=CC(CC)C(=O)NC(Cc1cnn(C)c1O)C(=O)NCC(F)CO C(=O)(CCC(CF)CF)N1CCC(OCCNC(CCSCC(C)C)=O)C1 CCC(F)(F)CC(=O)N1CCCN(CCNC(=O)COC2CCCC2)CC1 C1(C(=O)NCC=CC(N2CC(C(=O)OC)C2)=O)CCOCC1 C1(N(CCC)C(=O)NCc2occc2CC)CCCCC1C N1(C(c2[nH]cc(S(N)(=O)=O)c2)=O)CCC2CCC(C1)N2C(=O)CC1CCOCC1 c1(C(=O)Nc2c(C)cc(NC(C3(Cl)CC3(F)F)=O)cc2)ccn2ccnc2n1 C(=O)(CC1OCCc2ccccc21)N1C(CNC(c2nc(C)oc2)=O)CC2CC21 Cc1nc(C(C)C)oc1C(=O)NCC1(NC(C2CCCC2CF)=O)CCC1 CC1CC(=O)NC(C(=O)N(CCCC(=O)NC2(C3CCCO3)CC2)C)C1 c1(C(N2CCCC(C(C)NC(CC=C)=O)C2)=O)c(C)cc(OC(F)(F)F)cc1F C1(CNC(C(CC)OC)=O)COC(C)(C)CN1C(c1cc(C(=O)OC)cs1)=O C1(C(=O)NC2CCN(CCNC(C(CC=CC)C)=O)CC2)CC2C(C1)C2(C)C c1(C(=O)OC)cc(C)ccc1NCC1CCN(C(c2cnc(F)c(F)c2)=O)C1 Cc1ncc(C=CCNC(C2CCCC2c2ccccc2)=O)s1 c1(C(=O)NC(C2CCN(C(c3ccc(C(C)C)o3)=O)C2)C)ccnc(C2CC2)c1 C1(CC(N2CC(F)(CC)C2)=O)CC(NC(=O)CN2CCNC2=O)C1(C)C C1(NC(c2ncccc2Cl)=O)CN(C(c2ccc(CO)s2)=O)CC12CCC2 C1(CC)(CNC(=O)C(C2CCCCC2)C)CCCN1C(=O)CCn1cc(C)cn1 C(=O)(C1=NOC(C)C1)N(CC(C)O)CCNC(c1sc(N2CCC2)nc1Cl)=O CN1CCCC(C(=O)NC2CCC(CNC(=O)CC3CCCCC3)C2)C1 c1noc(C)c1C(=O)NCC.C1(NC(=O)N)CC(CCNC(=O)CN)(CF)C1.OC c1(-c2nn(CCC(C)C)c(CCC3CC3)n2)ccc(F)c(F)c1.[nH]1cncn1 C1(C(=O)O)C2CC2C2CC12.C12CCC(=CN1C(C)C)CC2 N1(C(CC2(OC)CC2)=O)CCCC(CO)(NC(C2CCCC(C)(C)C2)=O)C1 c1(C(=O)NCCC2CCCN(C(c3cc(SC)oc3)=O)C2)cn2ccnc2s1 N1(C(CCCCCCSC)=O)CC2CCCC(C1)N(C(c1cc[nH]c(=N)c1)=O)C2 c1(C(C(=O)NCCOCCNC(C(CC)n2cncn2)=O)(C)C)ccc(F)cc1 C=CCC(C(=O)NC1CCC(CCC(=O)NC(C)C(C)(C)C#N)C1)C(C)C C1(C(=O)NCCC2CC(NC(=O)COC3CC(F)(F)C3)C2)Cc2ccccc2S1 C1(CNC(=O)CC2CCC2)COC(CNC(c2cc(C3CCC3)on2)=O)C1 N(C(=NCCC(F)(F)F)NC1CCCC1)Cc1cccc(OC)c1Br C1(CN(C(CN2C(C)CC2)=O)C)CCCCN1C(c1cnccc1Cl)=O N1(C(C(c2ncn(C)c2)O)=O)CCC(O)C1C(N1CC(O)(CC(N)=O)C1)=O C=CCC(C)C(=O)NC(c1cn(Cc2scc(C(=O)OCC)n2)nn1)C c1(C(=O)NC2CN(C(c3c(OCC)nsc3)=O)CC2C)ccc(Br)c(C)c1F N1(C(CSCCC)=O)CC(CNC(c2c[nH]c(=N)cc2C)=O)C(C)(C)C1 C(=O)(C1CCCc2nccn21)N1CCCC(N)C1.C(=O)(C(F)(F)CN1CCCC1)OC c1(C(=O)NCCCN(C)C(c2ccc(C3COC3)cc2)=O)cc2n(n1)CCO2 c1(CC)cc(CNC(C2CC(C)(NC(C3CCN(CC(C)C)C3)=O)C2)=O)no1 N1(C(CCSCCC)=O)CC(NC(c2cn(CCO)nn2)=O)C(CC)C1 N1(C(c2c(F)ccc(N)c2)=O)CC2(CCCC2NC(C2CCSC2)=O)C1 Cc1ccnc(-c2cccc(NC(C3CCC3C(C)(C)C)=O)c2)n1 CCC(CC(=O)N(CCCOCCN(C)C(c1cnn(CC(F)F)c1)=O)C)C1CC1 Cc1n[nH]c(C)c1SCC(=O)NCC1C2CN(C(=O)CCCn3ccnc3)CC12 C1(NC(=O)NCC(=O)Nc2ccc3c(c2)OCO3)CNCCC12CCOCC2 c1(C(=O)OC)csc(CNC(=O)C(n2cc(CCc3ccccc3)nn2)C)c1 N1(C(c2c(NC(C)C)ccc(Br)c2)=O)CCN(S(=O)(=O)C2CCCC2)CC1C#N C1(CC(N2C(C)COCC2)=O)C2CCCC2N1C(=O)Cn1cnc(=N)[nH]1 CCC1=C(C(=O)N2CC(NC(c3ccnc(F)c3F)=O)C3CC23)CCCO1 C1(NC(CCC(=O)c2ccc(C)s2)=O)CC2CCC(C1F)N2C(=O)C(C)N(C)C CC1CN(C(=O)CC2CCCN2C(=O)Nc2c(C(F)(F)F)ncn2C)CCC1O CC(C)(C)CC(C(=O)NCc1ccc(CO)o1)NC(C1CCSC1)=O CC1(C(=O)NCC2(CNC(=O)CN3CCC(O)CC3)CC2)CCC(=O)NC1 CCC(C)(O)CCNC(=O)C(C1CCN(C(=O)Cc2ccnn2C)C1)C N1(C(c2n(CCCC)ncc2)=O)CC2(CCN2C(C2(CC3CCC3)CC2)=O)C1 c1(C(=O)NCCC(C)NC(c2ccc(F)c(CO)c2)=O)cc2c(cn1)OCCO2 c1(CC(=O)NC(C2CCN(C(c3cc(F)c[nH]3)=O)C2)C)cc(Cl)ccc1O C1(CC2(OC)CCCC2)CCN(C(=O)C(O)C(C2(F)CCOCC2)SC)CC1 c1(C(=O)NCC2(CNC(c3c(N)cc(F)cc3)=O)CC2)cc2c(=O)[nH]ccn2n1 CS(=O)(=O)C1CC(C(=O)NC2CN(C(c3cccnc3S)=O)CCC2CO)C1 c1(CC(N2CCC(N(C(=O)CSC)CC)C2)=O)cc(C)nn1C N1(C(C2=C(C)CC2)=O)CCC(C(=O)NC2(C)CCCNC2=O)CC1(C)C C1(NC(C(C2CCC2)N(C(=O)Cc2cncn2C)CC)=O)CCCCC1C C(C)(CC(C)NC(=O)CC1(C2CC2)CC1)NC(C=CC(C)C)=O C(c1cncn1C)=CC(=O)N.c1(CC)noc(CCCN(C(C2CC2)=O)C2CC2)n1 C(c1cn(C)cn1)=CC(N1CCC(C(=O)NCCCn2c(C)ncc2)C1)=O c1(C(N2CCC(CC=C)(NC(=O)C(C3CCC3)OC)C2)=O)ccc(C#C)cc1C c1(NC(C2CC2C(=O)NN2CC3CC3C2)=O)cnc(C(F)(F)F)cc1Cl c1(C(=O)NCCN(C(C2C(C=C)CC2)=O)Cc2cccnc2)cc(S(N)(=O)=O)c[nH]1 N1(C(c2c(C)scc2)=O)C(C(N2CCOC(C(N)=O)C2)=O)CC2CC12 C1(O)(CC(=O)NCC(CC)(C)NC(c2cnn(C)c2)=O)CCCN(C)C1 c1(C(NOCC)=O)cc(Cn2cc(CNC(c3cc(C#N)c[nH]3)=O)nn2)ccn1 CC(C(=O)NCC=CBr)(C1CCC1)NC(=O)Cc1ccsc1 c1(CCC)cc(C(N2CCC(CNC(=O)COCC(C)C)C2)=O)c(C)o1 N1(C(=O)CSc2ccc(Cl)nc2)CCC2(CC1)CCN(C(C1(O)CCC1)=O)C2 C1(NC(C(CCNC(=O)CCC2CCC2)OC)=O)CCn2nnnc2C1 c1(CC(=O)N(C(C)C(=O)N(C)Cc2ccco2)C2CC2)ccnn1C N1(C(C=C(C)C(F)F)=O)CC2COCCC2(NC(c2ccc(C#N)cc2)=O)C1 c1(OC)cccc(OC)c1C(c1nnnn1C)NC1CC2(CC2)C1 C1(C(=O)NCCSC)CCCCCCN1C(=O)CCCN(C)C N1(C(C2CCN2C(C2COCCO2)=O)=O)CCCC(Br)C1 c1(CC)conc1CC(=O)NC(Cc1ccco1)C(=O)NCCCF C1(NC(c2ccnc(OC)n2)=O)CC2CN(C(c3oncc3C)=O)CC12 C1(C(=O)NC(C(=O)OCC=C)(C)C)CC=CCC1NC(=O)C(O)CCSC N1(c2ncc(OC(C)C)cn2)CC2(CCCC2NC(=O)CSc2nccs2)C1 CC1(C)C2CC(C(=O)Nc3cccc(NC(=O)C(F)n4cccn4)c3)CC12 c1(C2C(C(C)NC(C3CSC3)=O)C2)ccc(Br)cc1 c1(OCC)ncccc1C(=O)NC12CC(NC(=O)COc3ccccc3)(C1)C2 C1(N(c2ccncc2F)CC2(C(=O)OC)CCCO2)CCN(CCCN)CC1 c1(C(C)C)ncc(C(N2CC(F)(CNC(=O)CCC3CCC(=O)N3)C2)=O)o1 c1(NC(C)=O)cccc(F)c1C(=O)NC1CC1CNC(=O)CCCc1sccc1C N1(C(C(c2[nH]c(=N)sc2)=O)=O)CCCCC(NC(c2occ3c2CCC3)=O)C1 C(=O)(C(C)CC(N)=O)NC(CN(C(=O)CC(F)(F)Br)CC)C C1(NC(C)=O)CC=C(C(=O)N2CCC2c2cccs2)C1 CC1CN(C(c2ccc(=O)n(C)n2)=O)CC(C)N(C(C2(NC(=O)C3CC3)CC2)=O)C1 CC(C(=O)N(C1CCN(C(C2CCC(F)CC2)=O)CC1)CCO)C(F)F c1(NCC2CC(N(C)C)C2)ccc(S(=O)(=O)N2CCC(O)C(C)(C)C2)cc1Cl C#CCC(C)C(=O)N1CC2C(CN(C)C(c3ccncc3F)=O)C2C1 c1(C(=O)NCC2(CNC(C3C(CC)OCC3)=O)CCC2)cccc(C2CC2)n1 Cc1c(Cl)cc(C(c2nnnn2-c2ccccc2)NCC2CC2(Cl)Cl)cc1Br Cc1cc2ccccn2c1C(N1C(C(=O)NOC2CCS(=O)(=O)C2)CCC1C)=O Nc1ncc(C(N2CCN(C(=O)CSC(F)F)C3CC23)=O)cc1CO C1(C(N(CCC(=O)N(C)Cc2c(C)cco2)C(C)C)=O)CCCC(=O)C1 NC(=O)CCCNC(=O)CC1CN(C(=O)N(CCCCl)CCO)C1 Cc1cc(CC(=O)N(CCNC(=O)COc2ccc(O)cc2)CC2CC2)nn1C CC(CC(=O)NCCCC1CN(C(c2ccc(F)cc2)=O)CCO1)C(F)F c1(C(=O)NCC2(O)CCN(C(C3NC(=O)C4CC34)=O)C2)cnc2ccsc2c1 N1(C(c2n(C(C)C)nnc2)=O)CCC(NC(=O)Cn2ncc(Br)n2)C(O)C1 C1(C)(CC)CC(NC(=O)Cc2ccc(OC)cn2)CN1C(c1nnn(C)c1N)=O c1(-n2c(CC(CCCC)C3CC3)nc(-c3nc(C)cs3)n2)ccc(F)c(C)c1 C(CCCCC(=O)NCC=CCC(N1CCC(CN=[N+]=[N-])C1)=O)OC c1(CC)noc(C(=O)NC2COCCC2NC(=O)COCC2CC2)c1C C(c1ccc(C(F)(F)F)cc1)=CC(=O)NCC1N(C(CC(C)F)=O)CCCC1 c1(C(=O)NC(C(C)SC)C)cccnc1CNC(C1CCOC1C1CC1)=O c1(C(N2CC=CC(NC(C(C)NC(=O)NC)=O)C2)=O)cc2ccc(C)cc2[nH]1 Cc1nc2nccc(C(N3CCOCC3CNC(=O)CC3C(C4CC4)CC3)=O)n2n1 Cc1cc(C#N)sc1C(N1CC(CNC(=O)C(F)(F)c2ccccc2)C1)=O N1(C(C(COCC)n2cc(-c3ccc(Cl)s3)nn2)=O)CC2(COC(C)C2)C1 c1(C(=O)Oc2ccccc2F)c(NC(=O)OC)cncc1Br c1(SCC)nccnc1C(=O)NCCC1CCCN(C(c2cnn(C)n2)=O)C1 C(c1ccc(Cl)cc1)=CC(=O)NCC(C1CCC1)NC(C(C)OCCC(C)C)=O C(N=c1[nH]c(=NCCSCCCO)c2sccc2[nH]1)c1cc(C)no1 C(=O)(CCCCC#N)N(CC(CNC(C(c1ccc(C(F)(F)F)cc1)C)=O)O)C Cc1ncc(CCNC(=O)CC2CNC(=O)O2)o1 C(=O)(C(F)(F)CCn1ccnn1)NC(C(C)C)CNC(C1CC1c1cccs1)=O N1(C(C2(OC(C)=O)CC2)=O)CCC2(CC1)CC2NC(C1CCN(C)C1)=O c1(C(C)=O)cc(C(=O)N(C2CCN(C(=O)CN3CCC(C)CC3)CC2)C)c(C)o1 C12(NC(C3CC(C(=O)OC)C3)=O)CCCC1CN(C(c1cncc(C)c1)=O)C2 C1(C(N2CCOCC2c2cn(CCCCF)nn2)=O)CC(=O)C12CCCC2 N1(C(=O)OCC)CCC2(CC1)CC2CNC(=O)C(C)(C)C(F)c1ccccc1 N1(C(c2c(N)ncc(C)c2)=O)CCCC(C2(NC(=O)CSCC(C)C)CC2)C1 C1(CC(=O)NCC(=C)CCNC(c2c[nH]c(Br)c2)=O)CCC(C)(C)C1 CC1CN2CCC1N=C1NC2=CC=CC(C)=CO1.C1(C=O)CCCN1C(N)=O C(=O)(N1CCCc2nccn21)C1CCC(CNC(C(CC=C)(C)C)=O)CC1 C(=O)(CC1OCCc2ccsc21)N1C(COC)(CNC(=O)C2=C(Cl)CC2)CCC1 N1(C(c2c(C)[nH]cc2)=O)CCOCC(C(=O)Nc2cn(C)nc2C)C1 N1(C(CNC=O)=O)CCN(C(=O)CC2CN3CCC2CC3)C2CS(=O)(=O)CC12 c1(CC(=O)N(C)CCOCCCNC(c2cc(CF)on2)=O)ccc(F)cc1F c1(C(=O)OC)ccc(NC2(CNC(C)=O)CC2C)cc1O C=C=C(C)CC(=O)N(C1CCN(C(=O)CSC2CCS(=O)(=O)C2)CC1)C C(CN1CCOCC1)(N=c1[nH]c(CO)c(C)s1)c1ccc(OC)cc1 C(C)(C(C)S(C)(=O)=O)CN(CC(C)C)C(=O)OC(C)C N1(C(C(C)OCCC=C)=O)CCC(C=C)(NC(c2cnc(C)c(OC)c2)=O)C1 O=C1CN(CCCN(C2CCCCC2)C(C(=O)NC2CNCCO2)=O)CCN1 c1(C(=O)NC2CC3(C2)CC(NC(c2csc(Br)n2)=O)C3)cc(I)ccc1O C(=O)(C(F)(F)C(C)(C)O)NC(COC)C(=O)NCc1ccc(C)c(C#N)c1 CC(C)CC(C)(C)C(=O)N1CCOC(CN(C(=O)C=CCF)C)C1 C12(C(N(CC(CC)NC(=O)C=C3CCC(C)C3)C)=O)CCC(C1)C2(C)C O=C(CCCCC1CC1)NC1CC(CNC(=O)C(C2(O)CCCCC2)(F)F)C1 c1(C(c2nnnn2CCOC)NCC2CC(=C)C2)cc(Br)c(Cl)s1 C(=O)(C(C)(F)C(=O)N(CCC(=O)NCCCOCCO)C)OC N(C)(C(=NCC1CCCCC1)NCc1nc(-c2ccncc2)n[nH]1)C(C=C)C C12(CNC(C(C=C)NC(C)=O)=O)CC(CO1)N(C(=O)C(C)COCC)C2 c1(C(N2CC(C(N(CC(=C)C)CC(=C)C)=O)OCC2)=O)ccc(C)nc1C CC(CCC(C)(C)C)C(=O)N1CCC(OCC(=O)NCC2(CO)CC3CC3C2)C1 Cc1cn2ccc(C(=O)N(CC(C)NC(=O)CCCC(C)C)C)cc2n1 N1(C(CC(C)NC(N)=O)=O)CCC(O)(CNC(=O)C(F)CC2CCCCC2)CC1 N1(C(CC2CC(CC)C2)=O)CCOCC1CN(C)C(c1nnsc1C)=O C1(COC)(CNC(C2(OCC)CCSCC2)=O)CCCN1C(=O)C(C)=CC1CC1 C1(C(=O)NC2(CO)CCN(C)C2)CN(C(C2CC(C)(C)CN2C)=O)CC12CC2 c1(CC)nnc(C)cc1C(N1CCN(C(=O)C#CC(C)C)C(CCO)C1)=O C(=O)(C#CC(C)(C)C)NCC(C)N(c1ncc(I)s1)C c1(C(=O)OC)coc(NC2(CNC(=O)OC(C)(C)C)CC(C)C2)n1 CCCC(CCCNC(=O)CCNC(C)=O)NC(c1ccc(F)c(N)c1)=O C=CC(F)(F)C(=O)N(C)CC1CCCN1C(=O)CSCCOC C(c1ccccc1Cl)=CC(=O)NC1C(N(C(=O)C=CC2CCCC2)C)CCCC1 C1(NC(c2c(F)ccc(Cl)c2F)=O)CC2(CCN(C(C3C4CCCC34)=O)CC2)C1 Cc1cc(Br)cnc1NC(N1CCN(CC(C)C)CC1)=O.C12CC3(C1)CC(C3)N2 c1(OC)cc(N2CCC(C)(NC(=O)C(=O)NCC3CC3)CC2)nc(=N)[nH]1 C(=O)(C(C)(CNC(C1CC(C2CC2)=NO1)=O)CC)OC.C12CN(CC1C)C2=O CCCCC(CC)CCC(=O)NCc1cccc(CNC(=O)CCC(CC)OC)c1 c1(C(N2CC(NC(C(C)OCC=C)=O)CC23CCC3)=O)cncc(P(C)(C)=O)c1 c1(C(N2CCC(NC(c3cc(COC)c(C)o3)=O)CC2)=O)ccc(Br)nc1N c1(C(N2CCCC(N(C)Cc3nnc(S)n3C)C2)=O)cc(S(N)(=O)=O)co1 C(C(=O)N1CC(CO)(NC(=O)CC2CC3(CC3)CO2)C1)(C(C)C)NC(=O)OCC C1(NC(CS(=O)(=O)NC)=O)CCCC12CN(C(c1coc(CC3CC3)n1)=O)C2 CC1CN(C(C2CCN(C(=O)Cc3ccsc3)CC2)=O)CC(=O)N1 C(=O)(N1OC2C=CC1CC2)C1CC(C)N1C(c1cnc(O)c(F)c1)=O C1(C(CNC(Cc2ncc(C)o2)=O)C)CCN(C(C2CNC(=O)C2)=O)CC1 CCCCCCCCC(C)C(=O)NC(C)(CNC(c1cnnn1C(C)C)=O)CC c1(OC)cccc2c(C(=O)NCCOCCNC(C3COC(=O)C3)=O)coc12 C=CCC(C(=O)NCC1(C(=O)NC2CNC(=O)C2)CCC1)OC N1(C(c2c(NC)nccc2)=O)CCC(C)(C(=O)NC(C)COC(F)(F)F)CC1 CN1CC(=O)Nc2cc(C(N3CCN(C4Cc5ccccc5O4)CC3)=O)ccc21 Cc1ccc(C(=O)NC(CNC(c2ccc(C(O)CF)cc2)=O)CC(C)C)cc1 C1(CCNC(c2ccn(CCOC)n2)=O)CN(C(=O)Cc2cnns2)CC(C)O1 C12(C(N(CC(C)CNC(c3n[nH]cc3Br)=O)C)=O)CCC(CC1)OC2 N12CCCCC3(CCN(C3)C(=O)C34CC5CC3(CO)CC5C4C1=O)C2.CCO C1(C(=O)Nc2n(C)nc(C3CCC3)c2)C2CCCC1N(C(=O)C(O)CC1CCCC1)C2 c1(C(=O)NCC(C2CC2)NC(C(C)C2CC2)=O)scc2c1OCCO2 N1(C(COCCCCC)=O)CCC(C)(CNC(c2c(CC)noc2C)=O)CC1 C1(NC(=O)CNC(=O)C(F)(F)F)CCCCCN(C(c2ccc(F)o2)=O)C1 N1(C(C(CCN(C)C)N(C)C)=O)CC2CCN(C(c3ccsc3Cl)=O)CC2C1 c1(C(C)C)ccc(C(N2CC(NC(=O)C(C)c3cccs3)CC2(C)C)=O)cc1F CC(Cn1ccnc1)C(=O)NCCN(C1CCCC1)C(=O)CC1CCCO1 C1(CN(CCN2CCC(CC(=O)OC)C2)C2CC2)CC2C(OC)C2C1 N1(C(C(CCCC)O)=O)CCC2C(C1)NC(=O)CN2C(=O)C=Cc1cnc[nH]1 CCC(CCOC)C(=O)NCC1(F)CCN(C(=O)CC2NC(=O)NC2=O)C1 c1(N2CCC(=CC(=O)NC3CC(=O)N(c4ccccc4)C3)CC2)cccc([N+](=O)[O-])c1 C(C(C(=O)NOC1CC1)C(C)(C)C)NC(C(CC)SC)=O C1(CNC(C(CO)N(C)C)=O)CC2CCC1N(C(=O)C=Cc1cccc(O)c1)C2 c1(N2CCOCC(NC(C(CCSC)O)=O)C2)ccn2c(Br)cnc2n1 C(=O)(C(C)(C)C(N)=O)NCCC1CCN(C(c2ccc(CSC)o2)=O)CC1 C(=O)(C1=CCCC(C)(C)C1)NC1(C)CCCN(C(CCCCCN(C)C)=O)C1 Cc1cc(C(N2CC(CNC(=O)Cn3c(C)ccc3C)C(C)C2)=O)c(Cl)cc1F CC(CCC=C(Cl)Cl)NCCCOCC(F)F.C(N)=O C(CN=c1[nH]c(C2CCCCC2)nc(=N)[nH]1)(C1(C(=O)OC(C)(C)C)CCC1)OC c1(N(C)C)nccc(C(F)F)n1.C1(=O)CCC2CC2N1 Cc1cc(C)c(C(N2CC(C3CN(C(c4cn(C(C)C)cn4)=O)C3)C2)=O)c(C)c1 c1(CC(=O)N(C2CCN(C(C(CCC)OCC)=O)C2)CC)c(F)cncc1Cl C=CCC(C)(CC)C(=O)NC1CC(CC(=O)NC2CC3C=CCC(C2)C3)C1 CC1(C)CC(NC(=O)Cn2cc(C3CCOC3)cn2)CN1C(=O)C#CC(=O)N(C)C Cc1c(Br)ccnc1C(N1CCN(C)CC1CNC(=O)COCC(F)F)=O C1(NC(C2C=CC(NC(=O)CCCCNC)C2)=O)CC12CCCCCC2 N1(C(C(C)CN(C)C)=O)CCC(C2(NC(=O)CC3CCC4(CC3)CC4)CC2)C1 N1(C(C(CC(F)F)NC(C2ON=C(C)C2)=O)=O)CC(O)C2(CCCC2)C1 C1(C)(C(N2CCC(N(C(=O)CC(C)C)CC#C)CC2)=O)CCC(C)(C)CC1 c1(CNC(c2cn(CCC34CC(CCN3)C4)nn2)=O)cc(OC(F)F)cc(Cl)c1 Cc1nc(O)c(C(=O)NC2CN(C(C3CCCCC3)=O)CC3(CC3)C2)nc1C c1(C(=O)NCCN(C)C(c2cnn(-c3ccccc3)c2)=O)ccco1.c1nccs1 CC(C)C(CCN(C)C(c1cc(C2CCC2)no1)=O)NC(=O)CO c1(OC)ncc(Cl)c(=NC2CCCC23CN(C(c2cscc2Cl)=O)C3)[nH]1 C1(C(N2CCCN(C(C(C=C)(C)CC)=O)CC2)=O)COc2ccc(O)cc2O1 N1(C(c2ccc(C)c(CO)c2)=O)CCN(C(c2cc(C#N)c[nH]2)=O)C2COCC12 Cc1cc(Cl)c(C(=O)NCC(C(C)C)NC(C2CC(O)C2)=O)cc1F N1(C(C2C(CNC(CC=CC=C)=O)C2(C)C)=O)CCC(C2(C)CC2)C1 C#CC1(C(=O)NC(CC2CC2)CO)CCN(C(c2oc(C)nc2C)=O)C1 c1(C(=O)NC2CCN(C(C3C(OC)(OC)CC3)=O)C2)cnc2nccn2c1.C(C)(=O)N N1(C(=O)NC2(c3ncc(C)s3)CCC2)CC(C)CC(C)C1C C1(C(=O)NC)CCC(NC(C2CC(N)CN2C)=O)CC1 Cn1c(O)nc2cc(C(N3CCC(CNC(=O)COCCCF)CC3)=O)cnc12 N1(C(CC(CC)CC)=O)CCN(C(=O)CNC(=O)CNC=O)CC(O)C1 N1(C(CC(CCSC)O)=O)CC2CC3CC2C1C3NC(c1cocn1)=O N1(C(C(C(CC)O)C)=O)CC2CCC1CN2C(c1sc(F)cc1Cl)=O CC1CC(CNC(c2ccc(C(F)(F)F)nc2)=O)CN1C(c1ccc(O)cn1)=O N1(C(CC2(C)CCN2C(=O)C=Cc2cocn2)=O)CC2C(C1)C2(F)F C1(N(C(c2nc(C(=O)OC)oc2)=O)C)CN(C(C2C3CCCC23)=O)CCC1C C1(NC(COCC)=O)CCCN(C(=O)CCCc2ccc(OC)cc2)CC1F C1(Cc2onc(C3(CSC)CCCC3)n2)CC(N)CC(C)(C)C1 C(=O)(CC(C)(C)C#N)N1CCC(C(C)NC(C2(C)CC(F)(F)C2)=O)C1 CN(C)N=Nc1ccccc1C(N1CCC1CNC(C1CC1C1CC1)=O)=O c1(C(=O)NC2(C)CCCN(C(C(C)O)=O)C2)cc2nn[nH]c2cc1F C(=O)(C(O)CC(F)F)NCC(c1cccc(Cl)c1)NC(CN(C)CC)=O C1(COC)(NC(C2COCC(C)(C)O2)=O)CCCN(C(c2ccco2)=O)C1 c1(CNC(C2(N(C)C(c3c[nH]cc3C3CC3)=O)CC(CO)C2)=O)cnn(C)c1C N1(C(C2N(C(c3c(OC)cccc3Br)=O)CC(C)C2)=O)CCCC2(CCOC2)C1 C1(C(N2CCC(C(C)C)C2)=O)CCCCN(C(=O)Cn2cncn2)C1 Cc1ccc(C)c(C(N2CC(CCNC(=O)CCSCC(N)=O)C(C)C2)=O)n1 N1(C(c2c(OC)scc2)=O)CC2(CCCCC2)CC1CO C(=O)(CS(=O)c1ccc(Cl)cc1)NCC1(C)CCN(C(C(C)C2CCC2)=O)CC1 Cc1cncc(CC(=O)NCC2COCC2CNC(=O)CCC(C)C)c1 c1(C(=O)NC2COCCN(C(C3C(C)C3)=O)C2)nn(C)c2ccccc12 C1(CNC(CC(CC)C)=O)CC12CCN(C(c1oc(CO)nc1C)=O)CC2 N1(c2nnc(CCC)s2)CCC(O)(C2(CO)CCC2)CC1 C1(C(N2CC(OCCC(=O)N(CC(=O)NC)C)C2)=O)CCCC1F c1(C(C)(C)C)ccc(-c2nc(CC3CCC(O)C3)n(CC(N)=O)n2)nc1 C1(C(=O)NC(C)(C)C(O)CO)N(C(c2cccc(F)c2F)=O)CCC1(C)C Cc1ccc2nc(N3CC4(CCC(=O)NC4)C3)[nH]c2c1 C1(NC(CCC(=O)NCCC)=O)CC2CCC(C1C)N2C(c1csnn1)=O C1(N(C(=O)C=Cc2ccc(Cl)s2)C)CCCN(C(=O)C(O)C(F)(F)F)CC1 C1(C(=O)NC(C)CCNC(=O)C=Cc2cncn2C)CCc2nccn2C1 CP(C)(=O)c1ccnc(N2CCN(S(=O)(=O)CC3=NOCC3)CC2)c1 N1(C(c2ccc(F)cc2)C)CC(C(N2CCCCC2CCN(C)C)=O)C(O)C1 Cn1cncc1C(=O)NC1CCN(Cc2nc(CS(C)(=O)=O)ns2)C1 c1(OC)ccc(C(=O)NCC2CC(C)N(C(=O)CN(C)CC3CC3)C2)cc1Br C12(C(=O)NCC(=O)Nc3ccccn3)CCC1CN(C(c1ccc([N+](=O)[O-])[nH]1)=O)C2 C12(NC(CCCC=C)=O)CCCCC1CN(C(c1nccc(OC)c1F)=O)C2 N1(C(C)=O)CC(CN(C(=O)CC(O)CN(C)C)C2CC2)C(C(F)(F)F)C1 C1(C(N(CCCCC=C)C)=O)CCCCC1NCc1sccc1Cl c1(OC)cccc(CCC(=O)NCC(O)CCNC(c2sncc2C)=O)n1 c1(C(=O)NCCC2CC(OC)CN2C(=O)Cc2cn[nH]c2)ccn(C)c(=O)c1 N1(C(=O)NC(CCC(C)C)C)CCN(C)C(COc2cnn(CCO)c2)C1 C1(Cn2cc(CNS(C)(=O)=O)nn2)CC2CCCCC2N1C(c1ccoc1Br)=O C12(CNC(=O)COC(F)(F)F)CCCC1N(C(c1ccc(CO)cc1F)=O)CCC2 c1(SC)ncc(C(N2CC(NC(C3CCNC3=O)=O)C2)=O)c(O)n1 c1(N2CCC(C)C(CO)C2)nc(=NCCc2ccn(C)n2)[nH]c2ccsc12 C1(CNC(C2(SCC)CN(C(c3cc(Cl)cn3C)=O)C2)=O)CC(C)(C)CCO1