SMILES O=C(C#CC1CCOCC1)N1CCSCC1C(=O)NC1CC2CC(O)C1C2 C12(C(=O)NCCCC(C)NC(c3ccc(OC)cc3)=O)CCCC1C2(F)F c1(C(C(=O)NCC(C)(C)NC(CN(CCOC)C)=O)C)ccc(C(F)(F)F)cc1 C1(NC(Cc2nc(C)sc2)=O)CCC2(CC1)CN(C(=O)COCCCF)CCO2 C1(C(=O)NCC2OCCN(C(C3(CC)CCC3)=O)C2)CCc2cc(C)ccc2O1 C1(C(=O)NCCC2C(C)C2)CCCCC1(C)NC(=O)C(Cl)Cl C=CCC(CC=C)C(=O)N(CC(C)(C)CNC(c1cn(C)nc1C(F)(F)F)=O)C c1(CC)ccc(F)c(C(N2CC3CCC3(C(N3CCC(C)(CC)CC3)=O)C2)=O)c1 S(=O)(=O)(c1cccnc1)NCC(=O)NC(CNC(c1c(CC)ncnc1)=O)CO [N-]=[N+]=NCC(C(=O)O)NC(c1cnc(-c2ccccc2Br)s1)=O N1(C(=O)NCC2CSCCO2)CCN(CC(F)(F)CO)CC1 C(=O)(CCCC(=O)c1ccccc1N)N1C(CNC(C(C2CC2)OC)=O)CCC1 c1(OC)ccccc1NC(C1(CNC(C2COCC(C)O2)=O)CC1)=O C(N=c1[nH]c(=NC(C)c2cccc(F)c2)[nH]c2cc[nH]c12)c1cnc(C)n1C C1(NC(CCCCCCC)=O)COC2(CCCN(C(c3cnn(C)n3)=O)C2)C1 N1(C(C=CCC)=O)CCC(CCC(=O)NC2(CN(C)C)CC2)CC1 n1(CC)cnc2c(NCCCn3ccnn3)nc(N3CC4COCC4C3)nc12 Cc1ccc(F)cc1CN1CC(C(c2ccccc2)O)OC(C)C1 N1(C(C(C)NC(c2cccs2)=O)=O)CC2CCN(C(C3CC=CC3)=O)C2C1 CC1(NC(c2cc(C(N)=O)[nH]n2)=O)CCCN(C(C2CCC(C3CC3)C2)=O)C1 C(=O)(C1=CCCCC1)NC(CC=C)CNC(c1sccc1-n1ccnn1)=O CC1=C(C(=O)NCC(C)CN(C)C(C2(C)CCCCO2)=O)SCCO1 c1(OC)ccc(C2CN(C(=O)NC(c3n[nH]c(=N)s3)C)CC2N)cc1 c1(C(=O)NC2C(CNC(C(C)c3ccsc3)=O)CC2)cccc2sccc12 n1(CC)c(C)cc(C(N2C3CC2CN(C(=O)CC2CC4CC4C2)C3)=O)c1C C=CC1CN(C(=O)C=Cc2ccn(C)c2)CC1NC(=O)CC12CCCC1C2 c1(CC(N2CCN(C(C=CCOC)=O)CC2C(C)C)=O)c[nH]c2c(C)cccc12 C(CCCCCCc1ccccc1)NC(c1ccc(C(F)(F)C(F)F)cc1)=O C1(NC(C=CC)=O)CCCCC12CCN(C(C1CCCC(F)C1)=O)C2 c1(C(=O)NCC(CNC(c2nc(CC)oc2)=O)F)cccc(F)c1C C1(C2CCCC(C)C2)NC(=S)N(c2ccc(Cl)c(Cl)c2)C2=C1C(=O)NC2C C(=O)(CCNC(N)=O)NCC(C)N(CC(C)(C)N1CCCC1)C CC(CCc1ccco1)NC(c1ccns1)C c1(OC)cc(CC(N2CC(NC(c3cnn(CCO)c3)=O)CC2C)=O)ccc1O c1(OC)cc(F)c(C(=O)NCC(O)CNC(c2cnc(C)s2)=O)cc1OC C(=O)(C(CCCOC)NC(c1cnccc1C)=O)NCc1onc(CC)n1 C(CCN(C)C(C1(c2cc[nH]n2)CC1)=O)(C(C)C)NC(c1cn(CC=C)nc1)=O C(=O)(C(C(C)(C)C)NC(c1cccc(C)c1O)=O)NC(CC#C)(C)C c1(CC(=O)NC23CC(C(N4CCSCC4CO)=O)(C2)C3)c(F)cc(F)cc1F Cc1cccc2sc(N(C3CC4CC3CN4)C(c3cncn3C)=O)nc12 c1(C(=O)NCC2CCN(C(C(C)=C3CCC3)=O)C2)nnn2c1CSCC2 Cc1coc(C)c1C(N1CC2CC1C2NC(=O)C(C)Oc1ccccc1)=O C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CC(=C)Cl)C(=O)N(C)CCNC(C)=O N1(C(c2nc(CS(C)(=O)=O)no2)C)CCCc2cc(OCC(C)(F)F)ccc21 N1(C(CC(CC)CN(C)C)=O)CCCN(C(c2cnnc(O)c2)=O)C(C)C1 N1(C(=O)Nc2cn[nH]c2)CC2CCC1C(Nc1ccc(OC)c(OC(F)F)c1)C2 C(=O)(C(O)Cc1cnc[nH]1)NCCOCCCN(C)C(C1COCCO1)=O C(CNC(=O)CCCOC(C)C)(C(C)(C)C)NC(c1ccc(CC)[nH]1)=O C(=O)(C(F)CCC(C)C)NC(C1CC2(C(=O)C(C)(C)C(=O)NC2)C1)COOC c1(CN2C(C(=O)OC)CS(=O)(=O)CC2)cccc2c1OC(F)(F)O2 NS(=O)(=O)c1ccc(NC(=O)CNC23CCCC(C2)NC3)cc1 C1(C(N(C)CC2OCCN(C(CCOCCOC)=O)C2)=O)CCOC(C)(C)C1 C(N=C(NCc1snnc1C)NC1CC1C)c1cc(C)sc1 C(=O)(CS(=O)(=O)CCO)N1CCCCC(CNC(CC(C=C)C)=O)C1 c1(C(=O)OC)c(Cl)n[nH]c1CNC(=O)Nc1csnc1C1CC1 N1(C(C(C)OC(C)(C)C)=O)CC=CC(NC(=O)Cc2ccn(CCF)n2)C1 C1(CNC(CC2C(OC)CC2)=O)CC(F)CN1C(C1CC1c1ccc(C)o1)=O c1(NC(C2N(C(c3c(C)ocn3)=O)CC(F)C2)=O)ccc2[nH]nc(Br)c2c1 C12(CN3CC(C)C(N=[N+]=[N-])C3)CC3CC(C1)CC(C(F)(F)F)(C3)C2 C(CCC)(C(=O)NCCC1CN(C(c2cnc(NC)cn2)=O)CCO1)=CCC CC1CN(C)CC1C(N1CCN(CCNC(=O)CCn2cnccc2=O)CC1)=O N1(C(C(CO)N(C)C)=O)CC2CCC(N)C2C1 CC1CCN(C(c2ccc(C#N)[nH]2)=O)CCN1C(=O)CN(c1ccc(Cl)nn1)C c1(CC)ccc(C(N2CCC(C)(CNC(c3snnc3C)=O)C2)=O)c(C)c1 N1(C(Cc2ncc(CC)s2)=O)CCCN(C(=O)NC2CC2)CC1 C1(CNC(CNS(N)(=O)=O)=O)CCC12CCN(C(c1nnc(O)nc1O)=O)CC2 C1(n2cc(CCOC)nn2)CCN(C(C2CC(C)(C)C2c2ccccc2)=O)CC1 c1(-c2cn(CC(=O)N(CCN(C)C)C)nn2)ccc(C2CCC2)nc1 c1(C(=O)NCC2CN(C(CSCCOC)=O)CC2(C)C)cccc(Cl)c1[N+](=O)[O-] C(C)(CCC(=O)N1CCCCC1CN(C)C(c1scnc1C(F)F)=O)SC N1(C(c2ccc(CC)nc2)=O)CCCC(COC)(NC(=O)COCC(C)C)C1 Nc1cc([N+](=O)[O-])ccc1C(N1CC2(CC(NC(C34CCC3C4)=O)CO2)C1)=O c1(OC)ccc(Cl)c(C(N2CCC(NC(=O)C=C(C)c3cccs3)C2C)=O)n1 C12(C(=O)NC(C3CCCCC3)CNC(C3(C)CCCS3)=O)C3CCC(CC13)C2(F)F Cc1ncccc1OCC(N1CCC2C(NC(=O)CCc3ccccc3Cl)C12)=O N1(C(C2SCCS2)=O)CC(CO)C2(CCN(C(C3(CF)COC3)=O)CC2)C1 N1(C(C2CC(C)NC(=O)C2)=O)CC2(CCN(C(=O)CCC3CCCCO3)C2)C1 c1(C(N2CC(CN(C)C)C2)=O)cn(CCNC(C2CC3(CC3)C2)=O)cn1 Cc1cc(F)c(C(=O)NC2CC(C)N(C(C34CC(C3)C4)=O)C2)c(F)c1 Cc1coc(C)c1CNC(=O)C(C1CCCC1)NC(C1CC1(C)C(F)F)=O C(=O)(C1=C2CCCN=C2NN1)N(C)CC1N(C(C(C(C)C)(C)O)=O)CCCC1 N1(CC(=O)NC2CNC2)CCOCC1.C1(c2cnc[nH]2)C(=O)N1Cc1nccs1 C12(OC)CCC(CC1)N(C(CO)C(=O)N)C2.C(=O)CC(C)C(=O)N(C)C[Si](C)(C)C c1(NC(c2cc(C3CCOC3)[nH]n2)=O)cccc(NC(c2ccoc2Br)=O)c1 C1(NC(c2c(C)occ2)=O)(CF)CCN(C(=O)C(c2ccccc2)NC(N)=O)C1 c1(C(=O)Nc2n(C)cc(NC(C3CC(C)OCC3)=O)n2)csc2ccccc12 c1(C(=O)NCC(C(C)C)(C)NC(c2ccsn2)=O)ccn2c1CSCC2 c1(C(N2C(C(=O)NCc3ccc(OC)cc3)CCCC2)=O)ccc(Cl)nc1Cl C12(C(N3C(Cn4cc(C(C)OC(C)(C)C)nn4)CC3)=O)CCCC1CCC2 C12(CNC(C(C)(C)OC)=O)COCCN1CCN(C(=O)C(c1ccc(C)s1)C)C2 CC1CCOC(C(=O)N(C2CCCC2)CCNC(C2CCCN(CC(F)F)C2)=O)C1 c1(-c2cnc(CCC(=O)N(CC(N3CCNCC3)=O)C3CC3)o2)cccc(F)c1 N1(C(C2CC3(CCC(C)(C)C3)C2)=O)CC2CCC(N=c3cnc(F)c[nH]3)CC2C1 C1(NC(c2cc(C)ns2)=O)CN(C(=O)Cc2cccc(Cl)c2)CC(C)(C)C1 C1(C(F)F)(CNC(c2csc(CO)c2)=O)CCN(C(=O)C(c2ccccc2)F)C1 C1(NC(C(c2ccccc2)OC(C)C)=O)CC(O)CN(C(c2cc[nH]n2)=O)C1 CN1CC(C(N2CCN(C(N3CCCC(NC(N)=O)C3)=O)CC2)=O)S(=O)(=O)CC1 N1(C(COC(CC)C)=O)CCN(C)CC1CNC(C1CCCSC1C)=O Cc1cn[nH]c(=NC(=O)c2ncc(-c3cnn(CN4CCC4)c3)cn2)c1 C1(F)(C(=O)NC(C2(O)CCN(C(c3ccnc(C4CC4)c3)=O)C2)C)CCCCC1 c1(CC(C(=O)OCC)NC(c2cn(-c3ccncc3)nn2)=O)ccc(O)cc1 c1(CNC(=O)NC(c2nnnn2C2CC2)C)conc1-c1ccccc1 N1(C(Cc2nc(=N)[nH][nH]2)=O)CCC2(C=C(C(=O)NC3CCCOC34CCC4)C2)C1 N1(C(CCOCCNC(C(CC)(C)O)=O)=O)CCC(C)(C)C1C c1(CC(=O)NC2CCC(CCNC(=O)NC3(c4nccs4)CC3)C2)cccnc1 Cc1ccnn1CC(=O)NCC(C(C)C)NC(c1scnc1C(C)(C)C)=O N1(C(c2c(C)[nH]nc2C(C)C)=O)CCN(C(C2CCCCS2)=O)CC(O)C1 C1(C(=O)NC(CNC(C(C)(C)OC)=O)(C)C(C)C)CCc2cncn2C1 c1(CNC(C2(NC(c3ccc(CO)cc3)=O)CSC2)=O)ccc[n+]([O-])c1 C(=O)(CC(CC)C1CC1)NCC(CCC)NC(=O)C(C)N(C)C(C)=O.OCC C1(C)(COC)CCN1C(=O)CONC(=O)CC1COCCO1 c1(C(=O)NCC2C(NC(CC(C)c3cccnc3)=O)CC2)ccc(F)c(N)c1 N1(C(c2cc(C)[nH]n2)C(=O)NCCCC)Cc2ccc(OC)cc2CC1C Cc1nc(CO)ncc1C(=O)NCC(O)CNC(=O)COCc1ccccc1 c1(N2Cc3c(nc(N(C)C)s3)CC2)nc(N2CCC(O)CC2)c2c(ncn2C)n1 Cc1cc(C(=O)N(CCC(C)NC(C2CC2(C)C(F)(F)F)=O)C)c(N)cc1F c1(C(=O)NCCC2CC(NC(C(CCC)=CCC)=O)C2)cc2nc(C)sc2[nH]1 Cc1cnc(C(=O)N(CC(C)(C)NC(C2CC2c2ccnn2C)=O)C)c(C)c1 c1(C(N2CCC(CNC(c3ccc(C)nc3)=O)C2)=O)cccc2ccsc12 C1(CNC(c2scc(CNC(C(COC)N(C)C)=O)c2)=O)CC(C)(C)CO1 Cc1cccc(OC(C)CN2C(=O)CN(CC3CN(C)CCO3)C2=O)c1C C12(OC)CCC(C(N3CC(N(C)C(C)=O)C3)=O)(CC1)C2.c12cn(nn1)CS2 C=CCC(C)(C)CCNC(=O)CCCC1CCCCN1C(C1CC(C)(F)C1)=O N1(C(C2N(CCC)CCCC2)=O)CC2(CCC2NC(c2ccc[nH]2)=O)C1 C#CCC(C)(C)C(c1nnnn1C(c1ccccc1)C)Nc1cnc(C)nc1C N1(C(CN2CC(C)(OC)C2)=O)CCC(NC(=O)CCNC(=O)CO)CC(C)(C)C1 Cc1cc2[nH]cc(C(c3nnnn3C)NC3CNC(=O)C34CC4)c(=O)n2n1 c1(C(N(C2CC(NC(C(c3ccccc3)SC)=O)C2)C)=O)cc(C2CC2)n(C)n1 c1(-c2cc(C)ncc2)ccc2nnc(C(=O)NCc3c(O)cccc3F)n2c1 c1(NCCN2CCCC(COC)C2)c(Br)cc(F)c(F)c1F c1(OC)cc(C(F)(F)F)ccc1CNC(N1CCCCC1Cc1cnco1)=O c1(C(C(=O)NC(C2CN(C(=O)C(O)C3CCC3)C2)C)(C)O)ccc(F)cc1 C(=O)(C1=CCC(C)CC1)NCc1c(C(=O)NCC(COC)O)nco1 N1(C(c2n(CC)nnc2)=O)CCCCC1CNC(C1CCCN1C=O)=O N1(C(C(CC#C)(C)C)=O)CC2CCC1CC2NC(c1ncn(C)c1C)=O C(=O)(CS(=O)(=O)c1ccccc1F)N1CCC2(CC(C)N(CCO)C2)CC1 Cn1ccc2cccc(C(N3CC4(C3)CN(C(=O)CCCN3CCCC3)C4)=O)c12 N1(C(C(CC(F)F)NC(c2c(CC)ncs2)=O)=O)CCCC2(CCCO2)C1 c1(C(c2n(CC)nnn2)NCCCCF)cccc(OC(C)C)c1OC Cc1nn(C)cc1C(O)C(=O)NCc1ccc(NC(=O)COCCN(C)C)cc1 C1(CNC(C2C(NC(CN3CC(C)(C)C3)=O)CC2)=O)OC2CCC1CC2 C=C(C)CC(C(=O)NCC1(CC(N)=O)CC1)NC(=O)CCC(=O)CC c1(C(=O)NC2CCC(NC(C3CC(N(C)C)C3)=O)C2)sccc1S(N)(=O)=O C=CCCC(C(=O)NCC(C1CC1)NC(=O)C(O)c1ccco1)c1ccccc1 c1(C(N(CCNC(=O)Cc2nc(=N)[nH][nH]2)CC)=O)cc2c(Cl)nccc2o1 C1(CNC(COC(CC)(C)C)=O)COCCN(C(c2n[nH]cc2C(F)(F)F)=O)C1 Cc1sc(-c2nc[nH]n2)nc1C(N1CCC1CNC(=O)C=Cc1cn[nH]c1)=O N1(C(CCOCC)=O)CCC(CCOC)(NC(=O)CN2CCCC(OC)C2)C1 c1(NC(c2csnn2)C)ccc(S(=O)(=O)NCc2cccnc2Br)c(Br)c1 CC1CN(C(=O)COc2ccc(Br)cn2)CCCN1C(=O)CCC#N N1(C(C=CCC)=O)CCC(C(F)(F)F)CC1CNC(c1ccnc(O)c1OC)=O C(=O)(C1=CCCC(C)(C)C1)N1CC(CNC(C(C)c2ccsc2)=O)C(F)(F)C1 C(=O)(C(C)CC(=O)OC)NC1CCC(CCC(N2C(C#C)CC2)=O)C1 c1(C(=O)NCCC(=C)CNC(=O)CN2CCC(C)C2)cccc(N(C)C)c1 CC1(C)CCC(O)(C(=O)NC2CC(NC(c3occc3Cl)=O)C(O)C2)CC1 C1(NC(CCc2scc(C)n2)=O)CCN(C(=O)C(O)Cc2cnc[nH]2)C1(C)C c1(C2CCN(C(CCC(=O)NC(CCCC)COC)=O)CC2)ccc(Cl)c(Cl)c1 c1(C(=O)Nc2c(C)ccc(-c3onc(C)n3)c2)cc(F)cc2cc[nH]c12 CCCCC(C(=O)NCC1C(OC)CN(C(C23CCCC2(C(N)=O)C3)=O)C1)N(C)C c1(N2CCC(COC)C2)nc(=NCCC(C)SC)[nH]c2c1COCC2 C=CC(C)(C)CC(=O)NCC1CC2CN1C2.c1(C(=O)OC)oc(CO)cc1C c1(NCCCC(C)NC(c2c(C(C)C)ocn2)=O)cc2nnc(C(C)C)n2cn1 N1(C(C=CC)=O)CCC2(CC1)CCN(C(c1cccc3nc(C)[nH]c13)=O)CC2 CC1(C)CC(CC(=O)NCCOCCNC(c2c(C3CC3)cccc2F)=O)CCO1 CCC(CC)(CO)C(=O)NCC1(NC(c2ccncc2Cl)=O)CC2CCC1CC2 N1(C2C(=O)CCC2)CCN(C(=O)C(N2CCC(N3CCCNC3=O)C2)=O)CC1 c1(CC)c(C)nc2ncnn2c1NC1CCCCCN(C(C2COC(C)C2)=O)C1 C=CC(C)(CC)C(=O)N1CCC(CCn2cc(-c3cccc(Cl)c3Cl)nn2)CC1 N1(C(CC=CC)=O)CC(CC(=O)NCc2cc(OC)ncn2)CC1(C)C CC1(C#CC(=O)N2CCCC2C2(NC(C3CN4CCN3CC4)=O)CC2)CC1 c1(C(=O)OCc2ccc(-n3cncn3)cc2)cc(C2CCCC2)ccc1Br c1(CNC(c2c(-c3n(C)ncc3)nn[nH]2)=O)ncccc1CNC(C1CC1Cl)=O C1(C)(CC(=O)OC)CCN(C(=O)C(=O)NCc2ncccc2Br)C1 N1(C(c2cc(C)ns2)=O)CCN(C(c2cnc(C3CC3)nc2)=O)CC1C N1(C(C2C(CC)C2)=O)CC2(CC(NC(=O)CCOC3CCOCC3)CO2)C1 c1(OC(C)C)ccc(F)cc1C(=O)NC1CCCC(NC(c2ncnn2C)=O)CC1 C1(C(=O)NC(CCC=C)CO)CC2(CCN1C(c1ccnc3cc[nH]c13)=O)CC2 c1(C(=O)NCC2N(C(CC(CC)OC)=O)CC(O)C2)n[nH]c2c1CCCC2 C1(C)(C(N2CCCC(N(C(c3c(C)ocn3)=O)C)CC2)=O)CC(C(F)(F)F)=NO1 N(C(=NC(C)CN(C)C)NCC1C2CCCCC12)CC1(C(=O)NCC)CCC1 N#CCS(=O)c1ccc(-c2nc(-c3ccc(N4CCCS4(=O)=O)cn3)no2)cc1 C(C)(C(=O)N1CC(CCn2cc(-c3cnsc3)nn2)C1)(C1CCC1)OC N1(C(C(C2(O)CN(C(C(CCC)(C)C)=O)C2)F)=O)CCOCC(F)(F)C1 C1(NC(c2cccc(F)c2)=O)CCN(C(=O)Cc2ccnc(F)c2F)CC1F N1(C(c2c(C)ccs2)=O)CC2CCCC1(CNC(=O)CC1CCNC(=O)C1)C2 N1(C(C(C)OCCOC)=O)CCN(C(c2ncn(C(C)C)n2)=O)CC(C)(C)C1 S(=O)(=O)(c1ccc(NCC2(C3CC3)CCC2)cc1Cl)N1CCN(CC)C(C)(C)C1 c12cc3c(cc1CN2)OC(C)C3.C1(CCOC)OCCC1C(C)C c1(C(N(CC(C)N(C)C(C2CCCC(C)(C)O2)=O)C)=O)csc([N+](=O)[O-])c1 CCCCC(C)CCC(=O)NC(COCC)C(N1CC2CCC(C1)C2(F)F)=O c1(NC(C2CCN(C(=O)COCC3COC3)CC2)C)c(Br)cc(C)cc1Br C1(CCC)CN(C(C2COCCO2)=O)CCN1C(=O)Cc1csc(Cl)n1 O=C(C1=CCCCC1)NCC1CN(C(c2cn(CC3CC3)nn2)=O)CC1(F)F N1(C(C2C(C)C2)=O)CCC2CN(C(=O)CCC3CCC(C)(C)CC3)CC12 C(C(C)C)(C(O)C(=O)N1CCCN(C(=O)C(C(C)(C)C)NC(C)=O)CCC1)OC C(C(O)CCNC(=O)CSc1nnc(S)s1)NC(C1CC2(CC2)C1)=O N1(C(CC2(OC)CC2)=O)CC2CCC1C(CNC(=O)C(C)C1(O)CCC1)C2 N1(C(c2cccc(CC)c2)=O)CC2CCCC2(C(=O)NC(C)(C)CF)C1 c1(CC)noc(CC)c1CC(N1CCC(NC(=O)CC(C)CF)C1)=O N1(C(CSCC#C)=O)CCOCC(CNC(=O)C(c2c(F)cccc2F)C)C1 n1(CC)cnc2nc(=NCC3CCCC3(C)C)[nH]c(NCC3CCCCS3)c12 N1(C(COCC)=O)CCC2(CCC2NC(=O)CC(C)c2cnn(C)c2)CC1 C1(C(=O)NCC(C(=O)OC)O)CC(O)C(O)CC1CNC(=O)CC1CC(F)(F)C1 c1(S)ccccc1.C1(C(=O)NCCOCCNC(C2(NC=O)CC2)=O)COCCO1 C(CCCC(=O)N1CC=CC1CNC(C1CCC2(CC2)C1)=O)SC c1(C(N2C(C(=O)NC(c3cc(F)cc(F)c3)C)C=CC2)=O)ncc(Cl)cc1Cl N1(C(C2(C)CCC(=O)N2)=O)CC(C2(NC(c3cncc(C#N)c3)=O)CC2)C1 C(=O)(CN=c1ccc(Cl)n[nH]1)N1CC(C(C)NC(COCC#C)=O)OCC1 Cc1cccc(C(=O)NC2CCCN(C(C3C=CCS3)=O)C2)c1F C=CCC(C(=O)N1CCC(C(=O)N(C)Cc2cccs2)CC1)N(C)C N1(C(C2CN(CC)C(=O)C2)=O)CCC(NC(c2ccccc2C2CC2)=O)C(O)C1 N1(C(C(C2CCCCCC2)OCC)=O)CC2CC(OCc3ccccc3)C(C2)C1 C1(C(=O)NCC2(O)CN(C(c3nccc(CC)c3)=O)C2)CC(C)CCC1C(C)C N#Cc1cccc(C(=O)N(c2nc(-c3ccc(Br)cc3)ns2)CCO)c1F C12CCCCC13CCN(C3)CC(=O)N2.C(C(C)=CC(=O)OC)C(=O)NC1CC1 c1(CNC(c2cc(C)oc2)=O)ncccc1CNC(=O)C(C)C#N C(=O)(C1=NNC(=O)CC1)N1C(CNC(CC(C)SC)=O)CCC1 c1(CC(=O)NCCC(CNC(C2C(C)C2)=O)O)c[nH]c2cccc(F)c12 CC(C)C(C(=O)NCC(CC(F)(F)F)NC(=O)CC1CC(=O)C1)C(C)C N1(C(C2CC(CCC)C2)=O)CC(CNC(c2cc(C)n(CC)n2)=O)CC1(C)C N1(C(C2(C#C)CCN(C(=O)CC(O)CC(C)C)C2)=O)CCC2CCCC2C1 Cc1cc(C(N2CCC(C)C2C(=O)NCC(C)(C)C2CCCC2)=O)c(O)nn1 CC1(C)CC(NC(=O)C(F)=C2CCC2)CN1C(C1CC2(CCCC2)C1)=O Cc1ccncc1C(=O)NCC(n1cc(C(C2CCCOC2)C)nn1)C c1(C(=O)C(N2CCC(N)C2)=O)cc(F)c(O)c(F)c1.C(CCl)O N1(CC(=O)N(C)C)CCCCC1c1ncc(C(F)(F)F)[nH]1 c1(NC(C2CC(C)CN(CCNC(=O)C(F)(F)F)C2)=O)c([N+](=O)[O-])cnn1C C1(NC(CN(C)C(N)=O)=O)CN(C(C2(CF)CCC2)=O)CCC1CO c1(C(N(C2CCN(C(=O)Cn3cccc3)C2)CCC)=O)cnc(OC)nc1 Cc1ccnc(C)c1C(C)(C)NC(N1CCC1Cc1c(Br)cnn1C(C)C)=O C(=O)(CC(CC(N)=O)CC(C)C)NCC(CC(C)C)NC(c1cc(C)nn1C)=O C=CCCCC(C(=O)NCCNC(=O)NCC)NC(c1cnc(O)c(C)c1)=O N1(C(C)=O)CCOC(C(=O)NCCCCCF)CC1 C1(CC)(NC(C2CC2(C)CC)=O)CCN(C(c2cc(OC)ncc2Cl)=O)CC1 c1(C(=O)NC2CCN(C(c3cn(Cc4nc(C)[nH]n4)nn3)=O)C2)cncc(O)c1 C(N(C)N1CCc2ncc(C)n2CC1)c1ccc(C(N(CC)CC2CC2)=O)cc1 C1(C(=O)NCC2(c3ccncc3)CC2)CC2CC(F)(F)CC(C1)C2(F)F N1(C(C(c2cccc(Br)c2)C)=O)CC2(CCCN(C(C3(C)C=CCC3)=O)C2)C1 C(=O)(C1=CC2CCC=CCCC12)N1CC(CNC(C2SC3C=CC2CC3)=O)C1 c1(N(C)Cc2ccn(C)n2)nc2cccnc2c(=NCCc2ncccc2C)[nH]1 Cc1ncc(C(N2CCC(Cc3nncn3C)C2)C(=O)NCCCC2CC2)s1 C1(NC(=O)OC(C)(C)C)CC1C1CCN(C(c2cc(Cl)cc[n+]2[O-])=O)CC1 c1(C(=O)NC2CCN(C(c3ccc(OC)s3)=O)CC2)ncc(Br)c(O)n1 c1(C(=O)NC2C(C)CN(C(=O)C(C)C3CCCC3)C2)ncnc2cc[nH]c12 C1(C(=O)NCCCCC#CC)CC12CCN(C(C1(C#N)CCCO1)=O)C2 N1(C(C2CCC(=C)CC2)=O)CC2CCCC2(NC(c2cnn(CCO)c2N)=O)C1 N1(C(C(=O)NCS)CCC2CCOCC2)CCC(O)(c2ccc(F)cc2)CC1 c1(OC)ccc(O)c(NC(C2(F)CCN(C(c3c(Cl)cccc3Br)=O)CC2)=O)c1 C(C)(C)(CCC(=O)NC(Cc1ccc(Cl)cc1Cl)CC(=O)N1CC(C)(C#N)C1)OC c12cccc(n1)OC21CC1.c1(OC)nc(C(=O)NC2CCN(C=O)C2)ns1.OC C1(C(N(CCCN(C(C(C)Cn2cccn2)=O)C)C)=O)CCCC(C)(C)C1 N1(C(C(C)=O)=O)CCCC2C1CCN2S(=O)(=O)c1ccccc1C N1(C(C2(C)CCOC2)=O)CC=C(CNC(C2([Si](C)(C)C)CC2)=O)CC1 c1(CNCC(F)(F)N(c2ccccc2)C)cc(F)cc(Br)c1F c1(C(=O)NC(C(=O)NC(CC)CCCO)COC(C)C)ccc2cc[nH]c2c1 C1(OCC(=O)NC(CCC)C)CCN(C(=O)CCOC(C)C)C1 N1(C(=O)NC2CCCN(c3cccc(F)c3)C2=O)CCC2C(F)(F)C2(F)C1 c1(CCC2(C(=O)NC(C)CON(C3CC3)C(c3cnn(C)n3)=O)CC2)ccccc1 Cc1cc(Cl)c(C(=O)N(C)CCOCCNC(C2CC2Cl)=O)cn1 CC1CN(C(=O)C=Cc2cccnc2)CC(C)CN1C(=O)C1=CC2CCCC12 c1(C(C)=O)cccc(OCc2cccc(C3CCCN(S(=O)(=O)C(F)F)C3)c2)c1 C(C(O)C(=O)NC1(C)CC(N(C)C)C1)NC(CCCOC(C)C)=O CP(C)(=O)C(CC(=O)N1CCCC1c1ccccn1)c1ccccc1 c1(CC)cc(C(N2CCN(C(=O)CC3CNC(=O)C3)CC2)=O)c(C)o1 C1(NC(C(c2ccn(C)c2)OCc2cccc(C)c2)=O)CCC(C2CC2)CC1 C(CCN=c1[nH]c(=NC(C)C2CCCO2)[nH]c2c1CCCCCC2)OCCOC C1(C)(Nc2nc(C(=O)NC)sc2)CCN(C(=O)CCCCNC(C)=O)C1 C1(c2n(CCCOC)nnn2)(Nc2cc(F)cc(Br)c2)C2CCC(C2)C1(C)C c1(C(=O)NC2CCCN(C(c3scc(OC)c3)=O)C2C)cc2nc(Cl)ccc2s1 Cn1cc(C=CC(N2CCC(O)(CCNC(=O)CN3CCS(=O)CC3)C2)=O)nn1 c1(SCC)cc(C(=O)NCCC2CC(NC(c3cnccc3Cl)=O)C2)ccn1 c1(C(=O)NC(C2CCCN2C(C2CC2C(C)(F)F)=O)(C)C)n[nH]cc1F C(c1cc(Cl)cc(Cl)c1)=CC(=O)NCC(CC)NC(c1cccc(F)c1C)=O c1(C(=O)NCCOCCCN(C(=O)CCn2cnnn2)C)conc1C1CCC1 NC(=O)CC(C(=O)NCC1CC(O)CCO1)NC(=O)C=CC1CCCCC1 C1(NC(C(C)(C2CC2)OC)=O)CCCCC12CCN(C(C1CCSC(C)C1)=O)C2 CC1CN(C(C2(C)CC2(Cl)Cl)=O)CCC1C(=O)O c1(C(N(CCCNC(C2CNC(=O)N2)=O)C)=O)ccc2scc(Br)c2c1 N1(C(c2n[nH]c(C)c2Cl)C(=O)NCC2CCCO2)CCCC2NC(=O)CC12 C1(C(N2CCC(C(=O)OC)C2C)=O)CC(F)CCN1C(c1conc1C)=O C(=O)(C(F)CC(CC)CC)N1CC(CC(=O)NC2CN(C(CC)=O)C2)C(C)CC1 C1(CC)C(C(N2CCC2CC2CCCC2)=O)CCN1C(c1coc(SC)c1)=O c1(C(N2C3(CN(Cc4c(OC)c(Cl)ccc4)C3)CC2)=O)ccc(C#N)cc1C CC1CCN(C(=O)CN2CCCCC2)C1C(=O)NC1(C2CCCCO2)CC1 C1(CNC(c2c(C)n[nH]c2C)=O)CN(C(c2ncnn2C)=O)CCC1C c1(C(N2CCCCC(NC(C3C(C)CC(=O)N3)=O)C2)=O)cn2cccnc2n1 Cc1ccc(O)c(C(N2CCOC(C(C)NC(=O)CC(C)N(C)C)C2)=O)c1 c1(NC(CCSC)C)[nH]c(=NCCCOc2ccccn2)nc2ncn(C)c12 C#CCCCCCC(=O)N1CC(CCNC(=O)CC2=CCCCC2)(OC)C1 CC(C)CC(C)(CNC(=O)Cc1cnns1)NC(=O)CCOCC(F)F C=C(C)C1OCCC1C(=O)NCC1COCCN1C(=O)CCNC(C)=O c1(C(N2C(CC(=O)NC3(COC)CCC3)CC2)=O)sccc1CNC(C)=O C1(=O)C(Cc2ccoc2)N1.CC(C(=O)N(C)C(C1CC1)C1CC1)N1CCCC1 c1(OCCN2CC(CNC(c3cccnc3Cl)=O)OCC2)ccc(F)cc1 n1(CC(=O)NCC2N(C(C34CC(C)(C3)C4)=O)CCCC2)cnc2c1CCCC2 C(C)(C)(CC(=O)NCC1(O)CCCOC1)N(C(C(CC)NC(N)=O)=O)C c1(C(=O)NCC=CC(=O)Nc2c(OC)cc(C)cc2)ncc(C#N)cc1C N1(C(c2c(Cl)cccc2Cl)C(=O)OC)CCn2cc(Br)cc2C1 C1(OC)CC(NC(C)CN(C)C(=O)OC(C)(C)C)N(c2ncccc2C#N)C1 Cc1cc(C(=O)NC2CC(C)(C(=O)NCCN(C)C3CC3)C2)c(C)s1 C1(C(=O)NCC2C3CC2N(C(=O)CCSC2CCCC2)C3)CCC2CCCCN12 N1(C(C(C2CCCCC2)CC)=O)CC(OC)CC1CNC(c1ccnn1CC)=O C(=O)(CC(C)C(C)(C)C)Nc1c(F)ncc(-c2cccc(NC(C)=O)c2)c1 N1(C(C)C)CCCC1C(=O)NC1CN(C(c2cnn(CC3CC3)c2)=O)C1 C(=O)(C(C1=NOC2CC12)N1CCc2cc(Br)sc2C1)NCCC(=O)OCC Cc1ccc(Br)c(C(=O)NC2COCCC2NC(=O)CCC(C)C)c1 C=C=CC(C)C(=O)N1CCCC1Cc1cn(CC(n2cccn2)C)nn1 c1(C(=O)NC(C2CCOC2)CNC(C2(C)CC3CC3C2)=O)ccc(S(N)(=O)=O)o1 CC1CN(C(=O)CC2CCOC2=O)CCN1C(C1C2CCC1(c1cnco1)C2)=O c1(N2C3CN(CC)C(C3)C2)nc2cccnc2c(=NCC2CCCN2S(C)(=O)=O)[nH]1 C1(C(N(CC(CC=C)(F)F)C)=O)CCN(C(C2CCCN2C=O)=O)CC1(C)C CCC(CCCO)N=c1cc(C)nc(N2CCOC3(CCCOC3)C2)[nH]1 c1(C(C)NC(c2n(CCOC)nnn2)c2ccc(C(=O)OC)o2)ccnc(F)c1 CC1(CNC(=O)C(N2CCCC2)C2CC2)COCCN(C(C2(CF)CC2)=O)C1 c1(CC(=O)N(C(C)CNC(c2ccnn2CC)=O)CC)nc(C)sc1C c1(CC(=O)NC2CCCN(C(C3CC4C=CC3CC4)=O)CC2)cccc(O)c1F N1(C(Cc2cc(C)no2)=O)CC2CN(C(c3c[nH]nc3[N+](=O)[O-])=O)CC2C1 C(CC(C(C)C)NC(=O)C(C)(C)c1ccsc1)N(C(Cc1c(C)scc1)=O)C C1(NC(c2ccc(CCC)s2)=O)CCCCC1NC(=O)CC(O)CC c1(OC)ccc(C(C)NC(=O)NC2CC3(CC(OC)C3)C2)cc1OC(F)F C1(C(=O)NC2(CCOC)CC2)COC(CNC(C2CC(OC)C2)=O)C1 c1(C(N(CCCNC(=O)C=C2CCN(C)C2)C(C)C)=O)cc2ccc(F)cc2o1 CN1CCn2nc(C(=O)NC3CCC3NC(=O)Cc3cc(F)ccc3O)cc2C1 C12(CNC(c3nc(CCC)oc3)=O)CC1CN(C(c1c[nH]nc1C(F)F)=O)C2 c1(OC)ccc(C(N2CCCC2CCNC(C2CC3C(C2)C3(F)F)=O)=O)c(Cl)c1 C1(CSCCNC(c2c[nH]c(=O)cn2)=O)CCN(C(C2C3CCC(F)C23)=O)CC1 C(=O)(CCC(C)(C)C#N)N1CC2C(CC(=O)Nc3cccc(N(C)C)c3)(CC2)C1 N1(C(C(C=CC)O)=O)CCN(CC2CN(C(=O)COc3ccsn3)C2)CC1 C1(NC(COC2CC(NC(c3[nH]ccc(=N)n3)=O)C2)=O)Cc2cccnc2C1 c1(C2(C(N3C(CNC(N)=O)CCC3)=O)CCC2)ccccc1Cl C(=O)(C(=O)CCC(C)(C)C)N(C)CC1CCCN1C(c1c(Cl)ccc(Cl)c1Cl)=O C1(C)(NC(C2(C)CC(=C)C2)=O)CCN(c2cc(C(F)(F)F)nc(Cl)n2)CC1 C1(CC(=O)NCC2C(C(N(CC#C)Cc3ccco3)=O)C2)CSCCO1 C1(NC(c2ccc(C)c(C)c2)=O)CCSC12CN(C(c1n[nH]cc1C1CC1)=O)C2 N1(CCOC)CC(C)N(C(=O)CNC(C2(n3cncn3)CC2)=O)CC1C C1(C(=O)NCC(CNC(C2(C)C(C)OCC2)=O)CO)CN2CCCN1CC2 N1(C(C=CCCC)=O)CC(NC(c2coc(-c3ccccc3)n2)=O)CC1.C1CC1 c1(NCC(=O)Nc2ccc(CC(=O)OCC)cc2)cnc(C=C)c(Br)c1 CCC(C)(CO)C(=O)NC1CC(CNC(=O)C(C)C(O)CC)C1 C1(C(=O)NC(CN(C(C(=Cc2ccco2)C)=O)C)C)CCCCC1CC(F)(F)F S(=O)(=O)(c1cccc(C(=O)NC2CN(C(=O)C(N)=O)C2)c1)N(CC)CC C(=O)(C1Cc2c(Cl)cccc21)NC1CCN(C(C(CCC)OCC)=O)C1C CN1CC(C(=O)NC2(Cc3nc[nH]n3)CCCCC2)CC12CCC2 C1(C(N2CCCCC(N(C(=O)CCC3CCCC3)C)C2)=O)CCCCCC1(F)F C12(CNC(c3c(C)nc(C(C)C)o3)=O)CCC(CC1)N2C(=O)CSCC1CCC1 Cc1cccc(OCC(N2CCC(CNC(c3cncc(Cl)c3C)=O)C2)=O)c1C C1CC(=O)CC2C(CC2)C(=O)N1.N1(C(=O)OC)CC(Cn2cccn2)C1 c1(C(N2CC(CNC(CS(CC)=O)=O)N(C)CC2)=O)cnc2[nH]ncc2c1 CCC(CC)CC(F)C(=O)N(C)CC1(O)CCN(C(=O)C(C)N(C)C)CC1 c1(C(C)C)ccc(C(N2CCCC2C(C)NC(C2CC23CCCC3)=O)=O)nc1 C(=O)(C1CCCc2nccn21)N1CCC(CCNC(C(N)=O)=O)C1 N1(C(C(CCOC)OC)=O)CCC(COC)(NC(=O)Cn2ncnn2)CC1 C#CCCC(O)C(=O)NCC(CC)NC(c1sc(C)cc1C)=O CC1(C)OCC2CC12C(N1CCC(NC(c2ccc(C3CC3)nc2Cl)=O)C1)=O c1(CC)ccc(C(=O)NC(C2CN(C(=O)CCn3ccnc3)C2)C)c(F)c1 N1(C(C(CC=C)C(C)C)=O)CCC2C1CCCN2C(=O)CS(C)(=O)=O c1(N(C(C(=O)NC(C)C)C(=O)O)CC(C)C)ccc(F)cc1F N1(C(c2c(-c3ccn(C)n3)n[nH]c2)=O)CCCC(CO)(NC(=O)C=CC2CC2)C1 c1(C(N(CCCNC(COC(CC)(C)C)=O)CCCO)=O)ccc2nccn2c1 N1(CCC)C(=O)CCC1C(=O)N(C1CN(C(C2CC2c2ccccc2Cl)=O)C1)C C1(NC(c2ccc(C(N)=O)nc2)=O)CC2CC1N(C(c1cnc(=N)[nH]c1)=O)C2 C1(C(=O)NCCN(C(C(C=C)(F)F)=O)C)CCc2c(cnn2C)C1 N1(CCN(C(C2CC(C(CC)CC)OCC2)=O)C(C)C)C(C)(C)CCCC1(C)C O=C(CNC1CCN(c2ccc(Cl)c(Cl)c2)CC1)NN=c1ccc(Cl)n[nH]1 C1(N(C(=O)C(C)C2CC2)CC)CCN(C(C2(C#N)CCCO2)=O)CC1 C(=O)(CCCCC(N)=O)N(C1CN(C(c2cncc(Cl)c2)=O)CC12CC2)C C12(NC(c3ncc(Br)cc3F)=O)CCN(C(=O)CCCc3ccsc3)CC1C2 C1(C(=O)NC(C#C)C(C)C)(CC)CCN(C(=O)CC2CC2(C)C)C1 C1(CC)CN(C(=O)C(c2ccccc2C)(C)C)CC1NC(=O)C(CC)OC Cc1nc(NCC23CC(NC(C4CC(=O)N(CC5CC5)C4)=O)(C2)C3)nc(C)c1Br c1(C(C(=O)N(C(c2ccncc2)C(C)C)C)OC)ccc(Br)cc1F C1(CC(=O)N(C(C=C)C2CC2)C)CCN(C(=O)CCOCC2CC2)C1(C)C C1(C(=O)NC(C#CCC)(C)C)C2CCCC2CN1C(=O)CCC(=O)NC.C(CC)N c1(NC2C3(C(=O)OCC)CCC(C2)C3)cc(C)c([N+](=O)[O-])cn1 C1(C)(C(=O)NC(CNC(C(C)OCC#C)=O)CC)CC2(C1)CC(F)(F)C2 C(c1cncn1C)=CC(N1CC(CCC=C)(C(=O)NC(C)Cc2nccs2)C1)=O C12(CNC(=O)CC3CC4CC4C3)CC1CN(C(=O)C=CBr)C2 c1(C(N2CCC(=CCNC(C(C)OC)=O)CC2)=O)cc2ccsc2[nH]1 C1(C(N(C)CC2(F)CCC2)=O)CC2(CCN(C(=O)C3=CC4C=CC3C4)C2)C1 S(=O)(=O)(c1ccc(CNC)c2cnccc12)N1C(CC)CC(O)C1.SC C1(C(N2CCC(O)(CC)C2)=O)COC2(C1)CN(C(C1CSC1)=O)C2 CC1(C2(C)CC2NC(c2cnn(-c3ccc(F)cc3)c2N)=O)CC1 Cc1nc(C)c(C(=O)NCC2CC2CNC(c2cncc(C(F)F)c2)=O)o1 CN1CCC(C(=O)OC2(CSC3CC3)CCOCC2)C1=O N1(C(c2ccc(CC)[nH]2)=O)C(C(=O)NC(CO)CC(C)C)CCC1C C1(C(N2CC(CC=C)(NC(c3cc(Cl)cn3C)=O)C2)=O)Cc2ccc(C)cc2S1 N1(C(CC=C)=O)CC2CCC(C1)N2C(=O)CC1CC(OC)(OC)C1(C)C C(=O)(CCCS(N)(=O)=O)N1CC2C(NC(C(C)Sc3ccccn3)=O)(C2)C1 C#CCC(C(=O)OC)NC(=O)CCN(C(=O)CC(C)(F)F)C(C)C C1(O)(C(N2CC(NC(C(=O)NC(C)C)=O)C2)=O)CC(C)(C)C1 Cc1ccc(NCC2CCCCC2c2cccc(Cl)c2)cc1-c1nn[nH]n1 N1(CC)CC(C(N2CC(CNC(c3cc(Br)cnc3C)=O)C2)=O)CCC1=O Cc1sc(C(N2CCCC(O)(CCNC(c3cc(O)cs3)=O)C2)=O)c(C)c1C C1(C(N(CC(C)O)CCNC(C2CC(C(=O)OC)C2)=O)=O)C=CCCC1 N1(C(c2c(C)n(CCC(C)C)nc2)=O)CCCN(C(=O)C(O)C2CCC2)CC1C Cc1ccc(S(=O)(=O)NCCNS(=O)(=O)c2cccc(F)c2)cc1C#N C#CCCC(O)C(=O)N1CCC(CNC(c2sccc2C(F)F)=O)C1(C)C N1(C(C=CCCCCC)=O)CC(NC(=O)C(C(C)C)n2ccnc2)CC1(C)C C1(OCC)CC(C)N(C(c2cn(C)ccc2=O)=O)C(C)C1 C(C)(C(=O)NCCC1CN(C(C2(CCF)CCC2)=O)C1)(C(C)C)NC(C)=O c1(C(C)=O)cccc(C(=O)Nc2ccc(NC(=O)C(C)C)cn2)n1 c1(C(=O)O)ccc(S(=O)(=O)Cc2ccnn2C2CCOCC2)cc1Cl C=CCC(CNC(c1csnn1)=O)C(=O)NCC1(C)CCCO1 C1(NC(C2C(C(C)(C)C)C2)=O)CCN(C(c2cc(N)c(F)cc2F)=O)C12CCC2 Cc1c[nH]cc(C(N2CC=CC(NC(c3c(Cl)n[nH]c3C3CC3)=O)C2)=O)c1=O C1(CCCC(=O)O)(C(N(C)CCC(=O)NC(=O)CC2CC2C)=O)CC1.C(C)(C)(C)O Cc1nc(C(N2CCN(Cc3cccc(-c4cn(CCF)nn4)c3)CC2)=O)nn1C C(=O)(CC(C)(C)CN(C)C)N1CC(NC(COC)=O)C(n2ccnn2)C1 C(=O)(CC(O)C(C)C)NCCCN(CCCCNC(c1cc(COC)on1)=O)C C(=O)(C(CNC(=O)C(C(C)C)C1CCC1)CC1CC1)NCC(C(=O)OCC)O C1(NC(C2(CCC)CC2)=O)CN(C(C2CCOC2)=O)C2(CCCCC2)C1 c1(NC(C(CCNC(C2CC2C(C)(C)C)=O)OC)=O)ccc(O)cc1Cl N1(C(c2[nH]cc(C(C)=O)c2)=O)CCCC(CNC(c2onc(Br)c2C)=O)C1 O=C1CC(CC(=O)NCC(O)CNC(C2(Oc3ccccc3)CC2)=O)CC(=O)N1 Cn1nnc2cc(C(=O)NC3CCCC(NC(C4CNC(=O)C4)=O)C3)ccc12 C1(CC(N2CC(OCCNC(C3C(CC)OCC3)=O)C2)=O)CCCS(=O)(=O)C1 N1(C(c2ccc(C#N)[nH]2)=O)CCC(=O)NC2CN(C(=O)CC3=CCCC3)CCC12 c1(CCC(=O)NC2(C)CCN(C(=O)C(F)=CCCF)C2)cccc(F)c1F C=C(Cl)C(C)(C)C(=O)N1CCCC(N(C(C2CCCCC2C)=O)CC)C1 C1(C(=O)NCC)CC2(CCC2)CN1C(=O)CCCC(=O)OC N1(C(Cn2c(CCC)nnc2S)=O)CCCN(C(c2cncn2CC)=O)CCC1 C1(CC)(OC)CCN(C(=O)Nn2cc(C(=O)Oc3ccnn3C3CC3)cn2)C1 c1(CN(CCCCS(CC)(=O)=O)C=O)ccc2nsnc2c1 CCCC(C)(C)CC(=O)N(CC(=O)NCc1cnco1)OC C(=O)(C1=CCC(NC(=O)CCN=[N+]=[N-])C1)N(CCCC)CC(N)=O C1(C)(C(F)(F)F)c2ccc(cc2)N1.c1(C(C)OC)ccc(N(C)C)cc1 N1(C(CCCCCCNC(C(C)CC2CCC2)=O)=O)CCC12CCC(O)CC2 CC1C2CC(C2Nc2ccc(Cn3ccnc3)o2)N1C(C1(c2cccs2)CC1)=O C1(C(N2CCCC(CNC(c3cc(CF)on3)=O)C2)=O)COCC2(CCC2)O1 Cc1cc(CNC(N2CC(NC(=O)OC(C)(C)C)C(O)C2)=O)cc(Br)c1 N1(C(=O)Nc2ccc(Oc3ccc(Cl)cc3Cl)cc2)CCC2(CCCCCO2)C1 c1(OC)ccc(C(=O)NCC2CCN(C(=O)C(O)C(F)F)C(C)C2)c(C)c1 N1(C(C(C)O)=O)CC2CCC(NC(c3ccc4cc[nH]c4c3)=O)(C2)C1 C(CCCC(=O)N1CCC(CNC(=O)C(C)(C)Cc2ccc(O)cc2)C1)OC Cc1[nH]nc2c(C(N3CC(N(C)C(C4CNC(=O)CC4(C)C)=O)C3)=O)cccc12 C1(C)(CNC(C2C(C)(C)CO2)=O)CCCN(C(C2(C(F)(F)F)CC2)=O)C1 N1(C(Cc2ccc(OCC)cc2)=O)C2CCC1C(NC(=O)CN1CCCC1C)C2 CN1CCC(NC(=O)Cc2ccc(O)nc2)C12CCCN(C(c1nccs1)=O)C2 CCCCC(C)C(=O)NCCNC1C=CCN1C(=O)CNS(=O)(=O)c1cccs1 Cc1ccc(CC(=O)NC2COCC2NC(C2(C#N)CCOC2)=O)cn1 c1(C(=O)NCC(c2ccc(OC)cc2)(C)O)ccc(Br)cc1OC(F)F C(=O)(CS(=O)(=O)CCO)NC1CC(CCNC(c2c(C)csc2Cl)=O)C1 C1(C(N2CCCC(CNC(C3CC(C)(C)C3)=O)C2)=O)CCc2nccn2CC1 c1(C(N(C(C)CNC(C2CC3C=CC2C3)=O)CC)=O)cccc(F)c1N N1(C(C(CC)CCOC)=O)CC(NC(=O)Cc2cc(C3CC3)on2)CC2(CC2)C1 C1(CN(C(C(C=CCCC)O)=O)CC)CCN(C(C2CCCSC2)=O)CC1 C1(NC(CCC=CC)=O)CC(OC)CN(C(C2CCCCN2CC(F)F)=O)C1 Cc1ccc(Br)cc1C(N1CC2C(NC(=O)C(C)S)C2C1)=O N1(C(C)C)CCN(CCC(=O)NCC2CC2NC(=O)CCn2ccnn2)CC1 c1(C(=O)NCC2CC(F)(F)CN2C(=O)CC2CC=CC2)ccn2nnnc2c1 c1(C(=O)NC2CCN(C(C3C(OC)CCC3)=O)C2C)ccc(C(C)=O)c(F)c1 C12(NC(=O)Nc3c(CS(=O)(=O)NC(C)C)cccc3)CCC(CC1)CO2 c1(CC)cccnc1C(N1CC(CNC(c2snnc2C)=O)C(C)C1)=O c1(CC)nc(N2CCCC(C)(CNC(=O)C(F)n3cccn3)C2)c(C#N)cc1C c1(C(C)C)cc(C(N2CCCC(CNC(c3cc(O)ncn3)=O)C2)=O)n(C)n1 O=C(CCCCCCCCCO)NC1CN(C(c2ccc(Cl)s2)=O)CCC1F C1(C(C)NC(=O)C(O)C2CCC2)CN(C(=O)CC2CS(=O)(=O)C2)CCO1 CCC(O)C(F)(F)C(=O)NCC1(CNC(C2CCN2C2CCCC2)=O)CCCC1 c1(NC(C2(F)CCN(c3nccc(OC)n3)CC2)=O)c[nH]c2ncccc12 N1(C(CC2N(C(C(CC)C(F)(F)F)=O)CC(O)C2)=O)CC2CCC(C1)C(=O)N2 Cc1ccc(CC(=O)NCC(CC(F)(F)F)NC(=O)CC(C)F)cc1F N1(C(C(C2CCCCC2)C)=O)CCC(F)(C(=O)NC(c2cccs2)(C)C)C1 c1(C(N2CCC(O)(CN(C(CCCOC)=O)C)CC2)=O)n[nH]c2c1CCSC2 C1(CNC(C(C2CN(C(c3ccns3)=O)C2)OC)=O)(CO)CCCO1 CC1COC2(C1)CN(C(C1CN(C(=O)C(C)(C)CO)CC1(F)F)=O)C2 C=C1CCC(C(=O)NC(C(=O)NCC2C(C=C(C)C)C2(C)C)C(C)OC)CC1 Cc1nc2c(C(=O)NC3CCC(C)N(C(=O)CCCN(C)C)C3)cccc2o1 c1(OC)ccc(CC(=O)NCC2CC2NC(c2cnnc(C3CC3)c2)=O)cc1Cl CC1(C(=O)NCCc2ncc[nH]2)CCN(C(C2CC2C2CC2)=O)C1 C1(C2(O)CCC2)(C(=O)NC2C(C(=O)NC3(C)CC(O)C3)CCCC2)CC1 C(=O)(C(F)(F)CC=C)N1CCCC(CCNC(C(CC=C)NC(C)=O)=O)C1 N1(C(C2(C)CCCCC2)=O)CCC2(C1)CN(C(c1ccc(O)c(F)c1)=O)CCO2 N1(C(CC2CCCC(C)(C)O2)=O)CCC2(CC1)CC2NC(=O)Cn1cnnn1 N1(C(C2(S(C)(=O)=O)CC2)=O)CC2(CCN(C(=O)C(c3ccc(F)c(Cl)c3)O)C2)C1 C1(C(N(CCN(C(C(C2CCCN(C)C2)(C)C)=O)C)C)=O)OCCN(C)C1=O C1(NC(c2cccc(C(C)(C)C)c2)=O)CCN(C(C2CC3CCCC23)=O)CC1F c1(CN(C(=O)Cn2cc(C3(O)CCC3)nn2)C(C)C)cccc(Cl)c1 c1(C(=O)NC2CC(CNC(C3(F)CCCCC3)=O)CC2O)ccc(Cl)nc1 N1(C(C(CCC)NC(C)=O)=O)CC2CCC2(C(=O)N(C)C)C1.C12CC(C1)O2 C(=O)(C(C)CCNC(C1CCOC1CNC(=O)CCc1cccs1)=O)OC N1(C(C2CC(NC(CCC(C)OC)=O)C(O)C2)=O)CCC12CCN(C)C2 N1(C(c2ncccc2C)C(=O)NCC=C)CC(CSC)CC(SC)C1 C1(C(N2CC(OCCC(=O)NC(c3scnc3C)C)C2)=O)(CC)CCCO1 C1(CNC(c2ccc(CO)c(F)c2)=O)C(O)C(O)CN1C(=O)C=CC1CC1 Cc1cc(=O)oc(C)c1C(=O)N(C)CC1(O)CCCN(C(C2(N(C)C)CC2)=O)C1 C=C(C)CN=C(NCc1cc2sccc2s1)NCc1nn(CC)cc1Br Cn1nc(Cl)c(C(N2CCN(C(C3CCOC(=O)CC3)=O)C(CO)C2)=O)c1Cl C1(CNC(=NCC=C)NCCOC)CN(Cc2cccc(CO)c2)CCN(C)C1 Cn1cnc2ncc(C(=O)NC3CCCC3NC(C3(C)CCCS3(=O)=O)=O)nc12 Cc1ncc(C(=O)NCc2nnn(C)c2C(=O)NC2COC(C)(C)C2)cn1 c1(CC)cc(C(=O)N(CCC(=O)N(CC(c2nn[nH]n2)C)C)CC)c(C)o1 C=C1CCN(C(c2cccc(C)n2)=O)C(C(N2CC(=O)NC(C(C)C)C2)=O)C1 C1(CNC(CN(CC(F)(F)F)C)=O)CCC1NC(=O)CCc1cncs1 CCC(C(=O)N1CCCN(C(c2ncn(C(C)(C)C)n2)=O)CC1)C(C)O CC1=CC(CNC(=O)C(c2ccccc2Br)N2CC3CC3C2)CCC1 c1(-c2scc(CN3CCC(C(N)=O)CC3C(=O)O)n2)c(F)cccc1F N1(C(C2CCC(C(C)C)CC2)=O)CCC(NC(=O)C=CC2CCCO2)C(C)(C)C1 N1(C(C(C)Sc2nnc(-c3ccc(OC)cc3)o2)=O)CCc2c(Br)cccc2C1 CS(=O)(=O)c1cccc(CNC2CN(C(=O)Cc3ccc(Cl)cc3)CC23CC3)n1 C1(NC(c2cc(CNC(c3c(OC)scc3)=O)[nH]n2)=O)CN(C)CCC1O c1(CCCC(=O)NCCN(C(C2(C(F)(F)F)CC2)=O)C2CC2)ccccc1Br CC1=Cc2cnccc2N2N=C1CC1CC2CCC1O c1(C(=O)NCCCCC2CN(C(C3(CCC)CC3)=O)C2)cc(C#N)ccc1N c1(C(=O)NC2CC(NC(c3n(C)ncn3)=O)C23CCC3)nnc2ccccc2n1 c1(CC(N2CCC(C(C(=O)NCC(COCC)(C)C)F)C2)=O)ccc(F)cn1 c1(OCCC#CC(N2C(C(C)C)C(O)CC2)=O)ccc2c(c1)OCO2 C1(C(=O)NCCC2CC(NC(c3cnc(=N)[nH]c3)=O)C2)CCC2(CCOCC2)O1 N1(C(COCC=C)=O)CC(CNC(=O)CCN2CCCCCC2)CC12CCC2 C1(COCC)CN(C(c2nncn2C)=O)CCO1.c12ccccc1O2 c1(C(=O)NC(CC=C)CNC(=O)CC(C)C2CC2)cc2cc(Cl)ccc2n1C c1(C(C(=O)NC(C)(C)C)N(C)CC)oc(Cc2nc(C(=O)OC)cs2)cc1Br c1(C(N(C2CCC(NC(C(CC#C)O)=O)CC2)C)=O)cnc(O)cc1C C(CCN=c1ccc(S(=O)(=O)NCc2ccc(C#N)o2)c[nH]1)N1CCCC(C)C1 C(=O)(C(C(C)CC)SC)N(C)Cc1cccc(CNC(C(C=C)(C)C)=O)c1 CC#CCCCC(=O)N1CC2(NC(c3ccc(CCC)cc3)=O)CC1C2 C1(CC(=O)NC2(C)CN(C(CC3CCN(C)C3)=O)C2)CCS(=O)(=O)C1 C1(C(C(=O)NC2(CNC(COCCOCC)=O)CCCC2)F)CCCCCC1 C1(F)(CNC(C2(C(C)(F)F)CC2)=O)CC(NC(C2(C)C=CCC2)=O)C1 Oc1nc2ccccc2n1-c1nc(-c2ccc(C3CCC3)cc2)n(CCF)n1 CCCC(C(=O)NC(C)(CNC(=O)CN(C)C)C1CC1)NC(c1ccccc1)=O c1(CN2CC3C(C(N4CCCC(F)(CC)C4)=O)C3C2)ccc(F)c2cccnc12 C1(C(=O)NCCCNC(c2ccco2)=O)CCn2c(O)nnc2C1 CC1COC(C(=O)NC2CC(CCC(=O)NCC3(F)CC(C(F)F)C3)C2)C1 c1(COC)cc(C(=O)NCC2(C)CC(C(=O)NC(=O)Cn3cnc(=N)[nH]3)C2)cs1 c1(N(CC)CC)c(C)cc(C(=O)Nc2cc(C3CC3)nn2C(C)(C)C)cc1Cl c1(C(N2CCCC(CNC(CC(CCC)O)=O)CC2)=O)ccc2c(c1)COCO2 CC1C(=O)N(C)CCN1C(=O)CN(C(=O)C=Cc1ccsc1)CC1CC1 c1(NC2C(CNC(C(CC)=CC)=O)CCCC2)cc(CC)n2ncnc2n1 C1(NC(C(COC)C)=O)CCN(C(c2ccc(OC)cc2C)=O)CC1OC C1(NC(C=C(C)C(C)(C)C)=O)CC2CC1N(C(c1ncc(C3CC3)cc1F)=O)C2 C=CCCCCCCC(=O)NC1CN(C(c2ccc(C#N)[nH]2)=O)CC1O c1(NC(C(N(C(C2C(CC)OCC2)=O)C)C2CC2)=O)cccc(C2CC2)c1 c1(NCC(=O)NCC2(CNC(C3C(C)CCO3)=O)CCC2)ccccc1[N+](=O)[O-] CC1CCC(C(=O)NC2CCCC2C(=O)NCC2CC2(C)C)O1 N1(C(c2c(C#C)c[nH]n2)=O)CCC2CC2(C(=O)NC2CC(C)(C)C23CC3)CC1 Cc1cc(=NC2C=CCCCC2)[nH]c(N2CCOCC(C3CCC3)C2)n1 C12(C(=O)NC3CC(O)C3)CCC(CC1)N2C(c1cccs1)=O.O=C(C)NCC(=O)N CCCC(C(=O)NCC1(OC)CN(C(=O)C(CC)Nc2nc(C)cs2)C1)OC C1(NC(c2c(NC)snc2C)=O)CC(NC(=O)CCCn2ccnc2)C12CCC2 N1(C(c2c(C)[nH]nc2Cl)=O)CC(C)(C)OC2(C1)CN(C(c1sncc1C)=O)C2 c1(C(N2CCC(CNC(COCC(=O)OC)=O)C(C)C2)=O)cnn2c(F)cccc12 N1(C(C(n2c(C)cc(C)n2)C)=O)CCN(C)C(CNC(=O)C(C)n2cccn2)C1 N1(C(Cc2n[nH]c(=NCC)s2)=O)CCCC2(C1)CN(C(=O)CN(C)C(N)=O)C2 C1(C(=O)NCc2scc(CC)n2)CCCCC1NC(c1cc(=O)cc[nH]1)=O C(=O)(C(O)CC(C)(C)C)N1CC2CC(NC(c3cnc(OCC)nc3)=O)C2C1 C(=O)(CC(C)(C)C(F)(F)F)N1CC(CCNC(C2(COCC)CCOCC2)=O)C1 CC1NC(=O)CCC1CNC(=O)C(C)NC(=O)C(C)(F)c1ccon1 N1(C(C2C(OC)CC2)=O)CC(NC(=O)CCCS(C)(=O)=O)CC(F)(F)C1 C(C(CC1CC1)C(=O)N1CCC(c2nn[nH]n2)C1)NC(c1scc(C)c1)=O C1(NC(=O)C=Cc2cocn2)CN(C(=O)Cc2cncc(O)c2)C2(CCC2)C1 Cc1cc(C(N2CC3CN(S(=O)(=O)c4cccs4)CC3C2)=O)ccc1[N+](=O)[O-] N1(C(c2ccc(C)cc2)=O)CCC(C)N(C(C2CCCC(F)C2)=O)CC1 Cc1nc2c(C(=O)NCc3nc(-c4ccccn4)cs3)cccc2o1 C(CC(C(=O)NC(CO)C1(C)CC1)NC(=O)Cc1cc(C)[nH]n1)OC C=C(C)CCCC(=O)NCCCCNC(C1(c2ccc(COC)s2)CC1)=O C(=O)(C(CNC(c1cncc(C#N)c1)=O)C(C)C)N1CCC(C)(N(C)CC)C1 c1(NC(=O)C(=C2CN(C(=O)CSC(F)F)C2)F)ccc(Cl)cc1F CCCCC(C)C(=O)N(C)CC1CCN(C(=O)CCc2cncc(Cl)c2)C1 C(=O)(C1=C(C)OCCC1)NC1C(NC(CC(CC#C)c2ccccc2)=O)COC1 c1(CC(=O)OC(C)(C)C)cnc(NC(C2(C)CSC2)=O)s1 C1(C)(c2cn(C(c3ccn(CC(C)(F)F)n3)C)nn2)CCOCC1 N1(C(C2(C)CC=CCC2)=O)CCC(C2CC2)(CNC(C2CCCCNC2=O)=O)C1 c1(CNCC(c2ccccc2)CNCC2(C)CCC2)cc2ccccc2cc1O c1(OC)ccc(SCC(=O)NCCCCCNC(=O)C(F)CN(C)C)cc1OC c1(C(=O)NC2CCN(C(C(COC)(C)COC)=O)CC2C)cccc2c[nH]nc12 CCC(O)C(=O)NCc1cc(CC(=O)N(CC(=O)OC)C)cs1 c1(C(N2C(CNC(CCC)=O)CCC2)=O)ccn2ncc(C)c2n1 Cn1nc(C(=O)NCC(O)C(=O)NCc2ncoc2C2CC2)cc1Cl c1(C(=O)NCC(C)CN(c2ccncc2)C)ccc(OCC(F)(F)F)c(Cl)c1 CCC(CC(F)F)C(=O)NCC1COCC1NC(=O)CCOc1ccccc1 C1(C(N2CCC(=C)C2)=O)CC=CC(NC(c2cncc(O)c2)=O)C1 C1(C(=O)NC2(CC)CCCC2)CC2CCC(C1)N2C(=O)C(F)=CCCF c1(C(=O)NC2CCN(C(c3cccc(OC)c3N)=O)C2C)c[nH]c2nccc-2c1 c1(C(=O)NC2(CCNC(CCC3CCC(C)O3)=O)CCC2)coc2c1CCCC2 Cc1ccc(C(=O)Nc2cnn(Cc3ccccc3Cl)c2)cc1O c1(C(=O)NCCCNC(c2scc(C)c2Cl)=O)cc2ccccc2cc1Cl C1(C(=O)NC(C2CCN(C(c3cnnn3C)=O)CC2)C)C2Cc3ccc(Cl)cc3C12 N1(C(C2(CC#C)CC2)=O)CCC(CF)(NC(c2ccc(NC(C)C)cc2)=O)C1 C(C(CC)C(C)C)(c1nnnn1C1CC1)N1CCCC1.c1(OCC)ccccc1 C(=O)(CS(=O)C(F)(F)F)NC12CN(C(CCC(N)=O)=O)C(CC1)C2 C1(F)(CNC(c2c(OCC)scc2)=O)CCN(C(=O)C(CO)C(C)C)CC1 C1(C(N(C(C)C(=O)NCC2CCC(F)C2)C)=O)CCC(O)CC1 C(C#CC(=O)N(C)CC1CC1(C)C)NC(COCC)=O CCC(C)(O)CNC(=O)CCC1CCN(C(C2CCC2C(C)(C)C)=O)C1 CC(C)CCC(C(=O)N1CCCCC(CO)C1)NC(c1cccc(F)c1O)=O C1(CC(=O)NCC2(O)CCN(c3ncc(C(=O)O)[nH]3)CC2)CCCC2(CC2)C1 CC1=CCC(NC(c2ncoc2NC(=O)NCC2CC2c2ccccc2)=O)CC1 C#CCC(CC(=O)N(C(C)CC(=O)OC)C)NC(=O)C(C)c1ccco1 C1(C2SCC(CC(CC)C)C2)NC(=O)CCN(CC(F)(F)F)C1=O c1(NC)cncc(C(N2CC(O)(CCNC(C3CC3c3ccco3)=O)C2)=O)n1 C#CCCN=C(NCCCN1CCOCC1C)N1CCC(C(C)C)C1 N1(C(C(CC)NC(N)=O)=O)C(C(=O)NC(C(C)C)c2nc[nH]n2)CCC12CC2 C(C1Cc2ccccc21)NC(=O)NC1COCCN(C(C)Cc2nncn2C)C1 N1(C(c2cc3scc(Br)c3s2)=O)CCC2(CCC2)C(F)C1 C1(C(=O)NCC2(CC=C)CCCCC2)CNCC1C1CCCC1 C1(OC)CN(C(=O)Cc2nnc(C)o2)CC1C(=O)NC1(c2ccccc2)CC1 c1(N(CCC(C)(C)C)C)nc2c(c(=NCc3ccc4[nH]c(=N)[nH]c4c3)[nH]1)CSC2 N1(C(c2cn(CCC)nn2)=O)CC2CCCN(C(=O)CC3CCC=CCC3)C2C1 N1(C(C(=O)N(C)CC#N)=O)Cc2cccc(C3=CCC(C(F)(F)F)CC3)c2C1 CC1CC(NC(C2CC(O)C2)=O)CN1C(c1csnc1Br)=O C(CCC(F)(F)F)ONC(C1CC(C(C)CO)C1)=O.C1(=O)CCCN1 c1(N(C)C)cc(S(=O)(=O)N2CC(NC(=O)NS(=O)(=O)c3cc[nH]n3)C2)ccc1Cl CC1CC2CN(C(C3CSC3)=O)CC2N1C(=O)CCc1nncs1 n1(CC(N2CC(C(C)NC(C3C(OCC)C3C)=O)OCC2)=O)ccc([N+](=O)[O-])n1 C1(C(N2C(CNC(C(CNC(C)=O)(C)C)=O)CC3CC32)=O)CC2CCC(C1)C2 c1(C(=O)NC2C3CN(C(C(C)SCC)=O)CC2C3)cn(C)c2c(Cl)cccc12 N1(C(c2n(C)ncc2Br)=O)CC(NC(C23CC(CO2)C3)=O)C(C2CC2)C1 N1(C(c2cnc(CC)s2)=O)CC(NC(c2cnnc(O)c2)=O)CC12CCC2 C(=O)(CCC(C)N(C)C)NCC(C)=CC(=O)NC(C)CN1CCCC1 CC1(C)OC(C(N2CC3(C2)CN(C(c2ccc(S(N)(=O)=O)s2)=O)C3)=O)C(C)(C)O1 O=C1NC(SC2COC(=O)O2)C(=O)N1CC1CCCS1 C1(c2n(C(CC)CC)nc(-c3cc(F)cc(F)c3)n2)CCSC(C)(C)C1 c1(C(N(C(CN(C(C(C2CCCCC2)OC)=O)C)C)C)=O)nnccc1C Cn1ncc(S(=O)(=O)N(C(C)(CO)C2CC2)C(=O)OC(C)(C)C)c1F N1(C(C=C(C)C(F)F)=O)CC(F)CC1CNC(c1csc(C(F)(F)F)n1)=O CC(C)(CNC(=O)CNC(=O)CC1CCCCC1)CCNC(c1cocn1)=O N1(C(C(CCC)=CCC)=O)CCN(C(=O)CCN2CCCCC2=O)CC1CF CCC(CC)CC(F)C(=O)N1CCC(C(=O)NCCC2CCN(C)C2)(CC)C1 c1(C(=O)NC(C2CCCC2)CNC(c2cc(CC)no2)=O)cnc(SC)n1C c1(COC)nc(C(C)C(c2ccc(F)cc2)C)n(-c2cnn(C)c2)n1 CCC(CC)C(=O)N1CC(CCNC(C2(c3ccc(F)cc3)CC2C)=O)C1 c1(NCC)cncc(C(=O)NCCCC(C)NC(=O)CN2CC3CCC2C3)c1 C(C(C)(CC(C)C)NC(c1cnc(OCC)s1)=O)NC(C=CC)=O CCC(C)(C)C(O)C(=O)NCC1CCN1C(c1cc(C(C)C)n(C)n1)=O c1(CC(=O)Nc2ccc(NC(C)=O)c(F)c2)n[nH]c2c1CCOC2 c12c(cccc1C)O2.C1(OC)CN(S(=O)(=O)C(F)(F)F)CC1F C1(F)(CNC(c2cc[n+]([O-])cc2)=O)CCCN(C(c2cccc(F)c2O)=O)C1 c1(C(N2C(CC(=O)Nc3ccc(OC)cc3)COCC2)=O)cnn2ccncc12 CC1CC(C(=O)NCCSCCCC2(C)N=N2)CCC1=O c1(C(C)=O)ccc(CC(=O)NC(C)(C)C(C)NC(C2CCC2c2nc[nH]n2)=O)o1 Cc1c(C(N2CCC(OCc3cc(F)c(Cl)cc3Cl)CC2)=O)oc2ccccc12 c1(SCCCCC2CC(OC)C2)ccn(C(C)Cc2nnnn2C2CCOC2)c1 c1(C(=O)OC)cc(C(=O)NC2CC(CNC(C3(C)CC3)=O)C2)cc(O)c1 C1(NC(CC2N(CC)C(=O)CC2)=O)COCCN(C(=O)CCCN2CCCC2)C1 N1(C(C(CO)NC(c2ccn(CCC)n2)=O)=O)CCC(C)(C2CC2)C1 CONC(=O)C(=O)N(CC(C)NC(=O)CC(C)CN(C)C)C c1(CC(=O)NCC(CNC(C2CN(C)C(=O)C2)=O)O)ccc(F)c(Br)c1 C(=O)(C1CCCn2cnnc21)N(C1CCC(NC(c2ncccc2F)=O)CC1)C N1(C(C2CCC(=C)CC2)=O)CC2(CCCN2C(c2cnc(COC)nc2)=O)C1 C1(C(N(C)Cc2nc(CC)sc2)=O)COCCN(C2CCCCC2C)C1 Cc1cnc2cc(C(N3CCC(C4CC4)(CNC(=O)CCC(C)C)C3)=O)ccn12 CC(=O)C(C)(C)CC(=O)NCC1CC(C)N(C(c2ccc(C(F)F)s2)=O)C1 c1(C(C(=O)NCCCSC)N(CC)CC)ccc(Cl)cc1C(F)(F)F Cc1cc(Br)cc(C)c1C(N1CCN(C(=O)CCC2CC2)CC1C)=O c1(C(=O)NC2CCN(C(CCNC(=O)OC)=O)CC2F)cc2cncn2c(O)n1 c1(N2CCC(CC=C)C2)ncc(S(=O)(=O)N(C2CCCC2)C)cc1Cl C(CCC(C)(C)C(=O)NCC1C(C(=O)NCc2ncccc2C)C1(C)C)OC C1(C(=O)NCc2c(CNC(c3c(C)cnnc3)=O)cccc2)CCCC(F)(F)C1 N1(C(Cc2nc(C)[nH]n2)=O)CCN(C(c2ccncc2C(F)F)=O)C(C)CC1C C=CCC(C)C(=O)NC1CCN(Cc2nsc(N(C)CC=C)n2)CC1 N#Cc1cc(F)ccc1C(N1CCC2CC2(NC(=O)CCCC(N)=O)CC1)=O n1(CC)nnc(C)c1CNC(c1cnc(CNC(C2CC(F)C(=O)N2)=O)nc1)=O C1(C(=O)NC(CSCC)=O)CC2CCC(C1)N2OC1CCC1.c12ccc(C)c(c1)N2 C1(C)(CNC(C2(C#C)CC2)=O)CCC(C(=O)NCC2(CO)CC2(C)C)O1 C1(CNC(C2N(CC)CC2)=O)CC2CCC(C1)N2C(C1CCC=CCC1)=O c1(CCCNC(c2cc(C(F)(F)F)sc2Br)=O)ccc(Cl)cc1 C12(CNC(C3(CC(C)C)CCC3)=O)CC(CN1C(=O)CCC1CCN(C)CC1)C2 c1(C(=O)NC(COCC)C(=O)NC2CCOC(C(C)C)C2)scc(C)c1C c1(NC(C2CCS(=O)(=O)C2)=O)ccc(CCn2cc(-c3cnccn3)nn2)cc1 c1(C(C)CC(=O)N2CCC(CN(C(=O)C3=CCC3)C)C2)ccccc1F Cc1c(C(=O)NCC2CCN2C(=O)CCn2cccn2)nn2ccccc12 c1(CNC(N2CC(C)(C(=O)OC)OCC2)=O)ccc(F)c(F)c1F c1(OC(Cc2c(CC)con2)=O)nccn2nc(Br)cc12 N#Cc1ccc(Cl)c(NC(c2cncc(NC(=O)C=CC(F)(F)F)c2)=O)c1 C=CC1CN(C(C2CC(O)C2)=O)CC1NC(c1cccc(OCC=C(C)C)c1)=O c1(C(N2CCC(NC(c3n(CCC)nc(C)c3)=O)C2)=O)c(F)ccc(F)c1F c1(C(N(CC(O)CNC(C2CCCO2)=O)C)=O)ccnn2ccnc12 N1(C(Cn2c(C)nnc2)=O)CCOC(N(C(=O)COCCOCCOC)C)C1 c1(C(C)C(N2CCC(N(C(=O)CNS(N)(=O)=O)C)C2)=O)cccc(C(N)=O)c1 N1(C(C2(C)CCC2)=O)CCCC1CC(=O)NCCCc1ccsc1 C1(NC(CC=C=C)=O)CC2CCC1CC2NC(c1c(OC)ncnc1C)=O C1(CNC(CCCOCC)=O)CCN(C(c2cc(C)cc(F)c2)=O)C12CC2 Nc1ccc(C(=O)NC2CCCC2NC(C2CC2c2cccc(Cl)c2)=O)nc1N C1(C(N2CCN(C(c3c(C)nccn3)=O)CC2CCO)=O)CCC(N=[N+]=[N-])CC1 N1(c2ccc(OC)c(C)c2)CCC(F)(F)C(C(=O)NCC2(C)CC2)C1 c1(C(=O)NCCCCCCNC(c2n(C=C)ncc2)=O)ccc2[nH]ccc2c1F C12(CCNC(c3c(C)nn(C)c3)=O)CCC1CN(C(c1ccc(CO)cc1)=O)C2 Cc1cc2nc[nH]c(=NCCCNC(=O)CCc3ccc(F)cc3Cl)c2[nH]1 CCC(CCCC(=O)N1CCC(O)CC1C1CC1)N(C(=O)Cn1cccn1)CCO C1(C(=O)NCC(=C)Br)CCCCCCN1C(c1cccc2ccnn12)=O N1(C(C(N(C)C)C2CC2)=O)CCCN(CCNC(=O)C(C2(O)CCCC2)F)CC1 C1(C(=O)NC2(c3cc[nH]n3)CC2)CC12CCN(Cc1cccc3[nH]ncc13)CC2 CCCCC(O)C(=O)NCc1nc(C(=O)NOC2CCCCC2C)c(C)o1 N1(C(C2CC(F)(F)C2)=O)CCCN(C(c2ccc(Cl)s2)C(=O)NC2CC2)CC1 c1(-c2[nH]c(=NCc3scc(NC(=O)OC(C)(C)C)n3)sc2)ccc2sncc2c1 CC1CN(C(=O)COCC(N2CCCCCC2)C)CC1NC(c1csc(=N)[nH]1)=O C(c1ccoc1)=CC(=O)NCC(O)C(=O)NCC=CCl N1(C(CC)C(N)=O)CCCC(C)(CNC(c2scnc2C(C)C)=O)C1 n1(CC(=O)Nc2c(C)c(C(F)(F)F)ccc2)ncn2cccc2c1=O c1(C2(C(=O)NCC(CC)NC(c3cnc[nH]3)=O)CC2)ccccc1C CC(C)CCCC(=O)NCc1cn(C2CCN(C(C3COC(=O)N3)=O)CC2)nn1 N1(C(C=COCC)=O)CC2CN(C(C3(n4cnnn4)CCOCC3)=O)CC12 c1(C(N2CCN(C(C3=NOC(C)C3)=O)CC2C2CC2)=O)ccc2c(n1)CCC2 C1(C)(C(N(C(C)CNC(=O)C=CCn2cncn2)C)=O)CCCCO1 C1(SCC(=O)NCCC(O)CNC(c2cn(C3CC3)nn2)=O)CCS(=O)(=O)C1 CCCCC(CC)C(=O)NCC1(O)CCN(C(C2CCOC(C(C)C)C2)=O)CC1 c1(C(N(C)CC2CCCC2(C)C)=O)n[nH]c2c1CN(C(=O)CCc1ccoc1)C2 C#Cc1cnc(C(N2CCCCC2CC(=O)NC2CNC(=O)C23CC3)=O)c(C)c1 c1(C(=O)NCCOC2CCN(C(CCC(C)N(C)C)=O)CC2)cc(N)ccc1F C1(CCNC(c2scnc2C(F)F)=O)CCCN(C(C2C3CNC(=O)C23)=O)CC1 n1(CC(=O)NC2C(NC(C=C(C)Cl)=O)CCC2)ccc2c(C(=O)NC)cccc12 N#Cc1cccc(CNC(c2cccc(N3CCCC3=O)c2)C(F)F)n1 Cc1ncc(C(N2CCC(C(C)(C)NC(c3ccc(F)cc3F)=O)C2)=O)c(=N)[nH]1 N1(C(CN(CCCCCC)C)=O)CC2(C1)CN(C(=O)C1=COCCO1)CC2CO c1(CC(=O)OC)ccc(CN2CCC(C(N3CC(O)C(F)C3)=O)CC2)cc1 c1(NC(Cc2nc(C)sc2)=O)cc(Cl)ccc1-c1nn[nH]n1 C1(c2ncc(CC)s2)CCN(C(C2OCCC2(C)C)C(=O)NCC2CC2)CC1 C1(NC(c2c(C)nsc2C)=O)CCN(C(=O)Cc2cn[nH]c2)C1(C)C c1(C(N2CCC(NC(CC(C)F)=O)C23CC3)=O)cc2c(cc1O)CCCC2 c1(NC(=O)OC)cnc(O)c(NC(C2C(C)CCCN2CCN(C)C2CC2)=O)n1 CCC(C)(COC)C(=O)NC(CNC(=O)C(C)N1CCC1)C(C)C c1(C(N2CC3CN(C(C(CO)NC(N)=O)=O)CC3C2)=O)ccc2c(c1)NC(=O)C2 CN1CCN(C(C2C3CN(C)CC23)=O)CC1C(=O)N(C)OC1CCCC1 c1(C(=O)OC)cc(C)c(Cl)cc1NC1CCC(C(F)(F)F)CC1 N1(C(C(C)N(C(C2CNC(=O)O2)=O)CC2CC2)=O)CC(CO)C(C(C)C)C1 C12(NC(c3ccnc(C4CC4)c3)=O)CCOCC1CN(C(=O)C=CC(F)(F)F)C2 c1(C(N2C(CNC(=O)COCCCF)CCC2)=O)ccc(C(F)(F)F)c(Cl)c1 N1(C(CCSCCCC)=O)CCC(C)(C)C(C(=O)NCCC(C)CCO)C1 C1(NC(C(c2ccc(C)cc2)F)=O)CCN(C(=O)CC2CC2C)CC1C N1(C(c2cc(C(C)=O)c(C)nc2C)=O)CCCC2(CNC(=O)C3CC3)CCCC12 c1(C(=O)NCC2N(C(c3c(C)nn[nH]3)=O)CC2)cc2cc(Br)cc(F)c2o1 N1(C(CC(=O)OCC)=O)CC(NC(c2oc(CO)nc2C)=O)CCCC1C Cc1nc2cc(C(N3CC=CC(NC(c4cnc(S)nc4)=O)C3)=O)ccc2n1C Cc1c(C(N2CCC(C(C)NC(=O)COC3CCCCC3)CC2)=O)ncn1C C1(CNC(c2n(CC)ncn2)=O)CCN(C(C2CCCO2)=O)CCC1(F)F c1(C(=O)NCC(CC=C)NC(C2CC(C)C2)=O)c[nH]c2c(F)c(Cl)ccc2c1=O N1(C(c2nccc(OC)c2)=O)CCN(C(C2CCCC23CC3)=O)CCC1C N1(CC)CCC(=O)N(CCSCS)C1=O.C1(C2C(=O)C2)CCC(c2ccccc2)CC1 c1(OCCC(=O)NCCNC(C2C(C(=O)OCC)CC2)=O)cccc(C)c1C N1(C(C(CO)NC(=O)CC2CC(F)C2)=O)CCC2(CNC(=O)O2)C1 c1(C(N2CCC(O)C(O)C2)C(=O)NCCCC)ccc2c(c1)OCO2 C1(CNC(=O)CCC2CC2(F)F)CCCCC1NC(=O)C=CCN1CCOCC1 CN1CCC(C(=O)NC2CN(C(c3nccs3)=O)CC(C)(C)C2)c2ccccc21 N1(c2ccnc(NCC(N3CCCCC3)C)n2)CCOCC12CC2 CC1CC(NC(=O)C=C2CCSCC2)CN(C(=O)CC2CC3(CC3)C2)C1 CC(C)CCCC(=O)N1CCC(O)(CNC(=O)Cn2ncccc2=O)C1 c1(C2N(C(=O)OCc3cc(OC)no3)CC2)ccc(Cl)cc1F C(=O)(C1=C(F)CNC1)N1CCC(C(=O)OC)(CO)C1 C1(NC(N)=O)CN(C(=O)C(C2CCCO2)NC(=O)C(=O)NCC2CC2)C1 Cc1cnc(C(N2CCC(=CCNC(C3CC(N(C)C)C3)=O)CC2)=O)c(C)c1 C=CCCC(=O)N(CCCNC(=O)C(C)NC(N)=O)CC c1(C(=O)NCC2CCC(C(=O)NCCCOCC)C2)n[nH]c(C)c1Cl CC(C)(F)C(C)(F)C(=O)N1CC(Nc2cc(Cl)ncn2)C1 C(=O)(C1=C2CCCN=C2NN1)N1C(CNC(C(COC)OC)=O)CCCCC1 n1(CC)nc(C(=O)NCC2CCCCC2NC(=O)CCC(F)F)c(Br)n1 C1(NC(c2ccccc2N2CCC(O)C2)=O)CN(C(C2(O)CCC2)=O)CCC1O C1(C)(CNC(Cc2c(C)occ2)=O)CN(C(=O)C(C)OCC2CCCO2)CCO1 c1(CNS(NCC(C)N(C)C)(=O)=O)ccc2c(c1)cc(C)n2C C1(NC(CC(C)(C)O)=O)CCN(C(C2CC3CCC2CC3)=O)C12CCC2 C1(C2CN(C(=O)C(C)CO)C2)(NC(C2CC(O)(CC#C)C2)=O)CC1 C1(CCNC(C2CCN(C(CC=C)=O)C2)=O)CCCCN1C(=O)CCCC CC1CN(Cc2cccs2)Cc2ccccc2O1.N12CCCC1CNC(=O)C2 C1(CNC(C2CC3CC3C2)=O)CN(C(=O)CN2CCNC2=O)CCO1 N1(CC)CCC(C(N2CC(CC3(CC)CC(O)C3)C2)=O)C1.c1(C(=O)N)cc(OC)ns1 C(=O)(CS(=O)c1ccc(Cl)cc1)NC(CN(C(c1nc(C)[nH]n1)=O)C)(CO)CO CC(O)(CNC(=O)C(=C1CCCCC1)F)CNC(c1cnnn1C1CC1)=O C#Cc1cnn(C)c1C(=O)N(C(C)CNC(c1sc(CC(F)(F)F)nc1C)=O)C C1(CC(=O)NC2CN(C(C34CCCC3(C(N)=O)C4)=O)C2)C=CS(=O)(=O)C1 C(=O)(C(CC(C)CC)NC(C1CN2CCN1CC2)=O)N(CCC=C)CC N1(C(c2c(OC)csc2)=O)C2CCCC1CC(CCN1CCCCC1)C2 c1(CCC(=O)NCC(C)NC(c2cscc2C(F)(F)F)=O)ccc(Cl)cn1 C(C(C)(C)CC(=O)N1CCCCC1C(C)NC(C1CCCC(=O)N1)=O)OC N#CCCCC(=O)NCc1ccnc(C(=O)NOCCNc2ccc(OC)cc2)c1 N1(C(C2CC(NC(CC(C=C)C)=O)C2(C)C)=O)CCc2ncccc2C1 C(=O)(CC(O)CCCC)NC(C(=O)N(CCSCC=C)C)C N1(C(CSCCOC)=O)Cc2occ(C(=O)NC3CC3(C)C)c2C1 N1(C(C2CN(OC)C(=O)C2)=O)CCC2(C1)CN(C(C1CC(F)(CO)C1)=O)C2 CCCC(C)CCN=c1nc2scnc2c(N(CC(C)C#N)C)[nH]1 c1(OC)cc(O)c(COC(=O)C(F)(F)c2nccn2C)cc1Cl c1(C(N2CCCC2Sc2cccs2)C(=O)N2CCCC2)nc(-c2ccco2)cs1 N1(C(C=CCOC)=O)CC(C)CCC1CNC(c1cn(-c2ccccc2)nn1)=O C1(C)(CNC(C2(C)CSC2)=O)CN(C(C2(C(C)(C)O)CCC2)=O)CCO1 c1(-c2nc(-c3c(C#N)n(C(F)F)nc3)on2)cc(Cl)cc(Cl)c1S(N)(=O)=O CCC(F)(F)C(C)(C)C(=O)NCC1CC(O)C1n1nnnc1N1CCCCCC1 C1(NC(C2(CC=C)CCC2)=O)CC2CC(C1)N(C(=O)CC(O)CCSC)C2 C1(C(=O)NCCCC(C)NC(CCc2ccc(C)o2)=O)CCC2(CCC2)OC1 CCCCC(C(=O)N1CCN(CCO)CC1c1cccnc1)NC(N)=O c1(C(N2C(C(=O)Nc3csc(-c4ccoc4)n3)CCC2)=O)ccn2ncnc2c1 C1(C#N)(C(N2CCN(c3scc(SC(C)(C)C)n3)CC2)=O)CC12CCCC2 O=C(CCS(=O)(=O)c1ccccc1)NC(CNC(C12COC(CF)(C1)C2)=O)C1CC1 C1(C2CN(C(C3CCC(F)(F)C3)=O)C2)(NC(CC2C(=O)NC(=N)S2)=O)CC1 N1(C(C2(F)CN(Cc3ccc(OC)nc3)C2)=O)CCN(C)C(C)(C)C1 C1(C(=O)NC(c2cn(CCCN)nn2)C)C2CC3C(C2N)C13.C12(C)CNC(=O)C(C1)C2 C1(NC(c2cnns2)=O)CC2CCC(C1)N2C(=O)CN1CCCC1=O O=C(CCC1=CCCCC1)N1CC(CNC(C2CC2c2ccccn2)=O)C1 c1(C(N2C(CNC(CCN(c3ccncc3)C)=O)CC2)=O)cccc(=O)n1C c1(C(=O)NC(C2CC=CCC2)C(=O)N(CC=C)CC)c[nH]nc1C C=C(C)C(C)(C)C(=O)N1CCCC(C(C)(O)CNC(=O)CC2(OC)CC2)C1 C12(C(N3CC(N(C)C(c4nc(=O)n(C)[nH]4)=O)C(O)C3)=O)CC(C1)S(=O)(=O)C2 CN=c1nc(C(N2CC3(CCC(CNC(c4nocc4C)=O)O3)C2)=O)cc(C)[nH]1 C(=O)(C1CCCc2nncn21)N1C(CNC(c2cnc(C)nc2C)=O)COCC1 C(=O)(CCCCCCC(=O)Nc1cn(C)c(C(=O)Nc2cccc(C#N)c2)n1)OC Cc1ccc(C(=O)NC2CN(C(C34CC(O)C3C4)=O)CCC2O)cc1S(C)(=O)=O CCCCCCCCN=c1[nH]c(C)cc(=NC2CCN(C3CCN(C)CC3)CC2)[nH]1 Cn1cncc1CCC(=O)NCC1CC(CNC(=O)CCc2ccccc2)CO1 C(=O)(C(CO)C(F)(F)F)N1CC2C(CCNC(C=CC=CC)=O)(CC2)C1 N1(C(CC2(CSC)CC2)=O)CCC(C(=O)NC23CCN(CC2)CC3)C(C)C1 c1(CN2C(C)(C(N3CCC(CC#N)CC3)=O)CC2)cc(F)c(F)cc1Cl C1(O)(CC(=O)N(CC=C)C)CCN(CCCCCN(C)C(=O)OC(C)(C)C)CC1 N1(C(C2C=CC(C(=O)OC)C2)=O)CCC2CCN(C(C3CCCC3)=O)C2C1 N1(C(C=COCC)=O)CC(C)N(C(=O)CCCc2ccc(F)cc2)CC1C c1(CC)cn2c(C(=O)NCC3CC(O)CN3C(=O)CC#N)cccc2n1 C1(CNC(C(CC)CO)=O)CN(C(=O)COC)CCC12CCOCC2 C#Cc1cncc(C(=O)NC2C=CCN(C(c3ccc(C)nc3OC)=O)C2)c1 C1(C(N2CCC(N(C(=O)CCC3CCC(C(N)=O)O3)C)C2)=O)CCOCC1(C)C c1(CC)ccc(S(=O)(=O)N2CCC(C(C)NC(c3n[nH]cc3I)=O)C2)cc1 c1(C(=O)NCCN(C(c2ccc(C)cc2N)=O)C)cccc2oc(C)nc12 O=S(=O)(c1cccs1)NCCN1CCC(CN2CCN(c3ccccc3)CC2)C1 c1(OC)ccc(C(N2CC(NC(C3(C(C)C)COC3)=O)C(C)(C)C2)=O)c(F)c1Cl Cc1ccc(F)c(C(=O)NC(C2CCOC2)CNC(C2(S(C)(=O)=O)CCC2)=O)c1 N1(C(C=Cc2c(C)cncc2)=O)C2CCC1CN(C(C1(F)CC1)=O)C2 C=C=CCC(=O)N(CC(Cc1ccccc1)NC(=O)CCCOCCC)C c1(CNC(C2C3(CC(NC(C4(OC)CCOC4)=O)C3)C2)=O)cccc(C)c1C C(C(=O)Nn1cccn1)NCC#C.C1(C=O)CCC2(CCC2)O1 Cc1cc(=O)c(C(=O)NC(C(=O)NC(C)C(=O)N(C)C2CC2)c2ccco2)c[nH]1 CC1(C)NC(=O)N(CC(=O)NC2CCOCC2Nc2ncc(O)cn2)C1=O N(C(=NCC(C)(C)N1CCCC1)N1CCC2(C1)CC2(F)F)C(C=C)C c1(C(=O)NCC2C(NC(c3ccc(CC)c(F)c3)=O)C2)ccc(N)cc1[N+](=O)[O-] c1(C(CNC(CCCCC)=O)NC(=O)C=CC2CC2)ccc(F)cc1F S(=O)(=O)(c1ccc(Cl)nc1C)Nc1c(C(=O)Nc2ccc(C)nc2C)nccc1 C(=O)(C1=CC2CCCC12)NCC1CN(C(C2(CC(C)C)COC2)=O)CC12CC2 C(=O)(C1CCCc2n[nH]cc21)N1CCC(NC(C(CC)n2cncn2)=O)C(C)C1 C1(C(=O)NCC(CN(C(Cn2c(C(F)F)cc(C)n2)=O)C)O)CCC(=O)N(C)C1 C(C(C)(O)CNC(c1cnn(C2CCNC2=O)c1)=O)NC(C1(COC)CC1)=O C1(NC(=O)CSC(F)F)COC2(CCN(C(c3sccc3F)=O)C2)C1 c1(CCC(=O)NC(C2N(C(CCCOCC=C)=O)CCC2)C)cc(C)nn1C C(CC(C)(C)CC(=O)N1CCC(C)(CC(=O)Nc2cc(C)cc(C)c2)C1)OC Cc1sc(O)nc1C(=O)NC1(C)CN(C(=O)C(C)n2cccc2)C1 N1(C(C(CC)CC)=O)CCC2(CC1)COC(CNC(=O)CCS(C)=O)C2 c1(CCC(C)C)ccccc1C(=O)NCC1CC(F)(CNC(=O)CNC=O)C1 C(=O)(n1[nH]c(=NC(=O)C2(C#N)Cc3ccccc3C2)c2c1CNC2)OC(C)(C)C c1(CC)ccc(C(=O)NC(C)C(C2CCCCC2)NC(=O)CC2CCC2)[nH]1 N1(C(CNC(CN(C(=O)OCC)C)=O)=O)CCC(C(=O)NC)C1c1ccccc1 c1(C(=O)NCCCC(=O)NC(C2CCCCO2)CC)ccc(SC)cc1 N1(C(C)=O)CCCC2CN(C(c3csc4c3CCCCCO4)=O)CC12 CN1CC(C(=O)NCCc2ccc(C(F)(F)F)cn2)c2ccccc2C1=O C(CCCC(=O)NCCC1CCSC1)N(C(C1C(CCOC)C1)=O)C c1(CC(N2CCC(O)(CCNC(COCC#C)=O)C2)=O)cc(Cl)c2c(c1)OCO2 CCCC(C(=O)OC)C(=O)N1C(CNC(c2cnc(S)[nH]2)=O)CC2CCCC12 CCCCCCCC(=O)NCC12CC1CN(C(C1CC3CC3C1)=O)C2 c1(C(N2CC(C=C)C(NC(=O)Cc3cn(C)nn3)C2)=O)cccc2ccncc12 c1(C(N(CC(C)C)CC(C)C)=O)cn(Cc2ccsc2)nn1 N1(C(=O)NCc2c(C)nn(CC(C)C)c2C)CC2(CC(C(=O)NC(C)C)CO2)C1 C1(O)(CC)CCN(C(C2(CNC(=O)CC3CCC(O)C3)CC2)=O)CC1 CC(c1ccco1)=CC(=O)OC(C)(C)C.N12CCN(CC1)C(=O)OCCC2 N1(C(=O)Nc2cccc(CC)c2)CC2CN(C(c3ccccc3C)=O)CC2C1 C1(F)(C(N(CCCNC(=O)C(CN(C)C)c2ccccc2)CC)=O)CCOCC1 c1(CC)nc(C(C2CC2)NC2CCC(C)(C)C2)n(-c2ccnc(C(F)(F)F)c2)n1 N1(C(C2CC(OCC)C2)C(=O)NCC(C)C)CCc2ccc(C)cc21 C(c1cccc(Cl)c1)=CC(=O)NCCCCCCNC(C1CC(O)C1)=O CCCCC(C)C(=O)N1CCC(NC(=O)C=CC(C)C)C1 c1(SC)ccc(C(=O)NC(CC)C(=O)NCC2CSC2)o1 c1(N(C)CC)[nH]c(=NCC2CC2)nc2ncn(CC)c12 c1(C(N(C2CCCN(C(CC)=O)C2)C)=O)ccc2ccc(Br)c(F)c2n1 C1(C(=O)NCCCN(C(C(n2c(C)ncc2)C)=O)C2CC2)CCn2cnnc2C1 N1(C(CCC#C)=O)CCC(N(C2CCOCC2)C(C2CCCCC2)=O)CC1 c1(C(=O)NCC(CC)NC(CCOCC)=O)cc2ccc(Cl)c(F)c2o1 CCCCCC(F)C(=O)NCc1nc(C)c(C(=O)NCC2CCCN2CC)o1 N1(C(Cc2cccc(OC)c2)=O)CCN(C(c2ccc(CF)cc2)=O)C(C)C1C c1(NC(c2c(C)c[nH]c2)=O)ccccc1N1CCN(C)CC1 c1(C(=O)NCC(C)N(C)Cc2cncs2)ccn2ccccc12 c1(CN(C(c2ccccn2)C)C)cnn(C2CC2)n1 c1(CC)ccc(OCCC(N2CCCC2C2CCN(C(=O)CNC=O)C2)=O)cc1 c1(CC)nc(C(=O)NCCN(C(=O)COc2ccc(CO)cc2)C(C)C)c(C)o1 C(=O)(CC(F)(F)C(F)F)NCCC1CN(C(C(C)C)=O)C1 C(=O)(CCCC(F)(F)F)N1CCCC(N(C(C(C)N(C)C)=O)C)C1 N1(C(C(C)NC(CC)=O)=O)CCC(O)(CNC(=O)C=Cc2cc(OC)ns2)C1 C(C(=O)NCC1CC12CCCCC2)(C(C)(C)O)NC(C=CCOC)=O C(CCCCCC(=O)N1CCCC1(C)C1CCC1)NC(c1cnc(C)s1)=O c1(-c2c(C)nc(NC(C)=O)s2)ccc2occ(Nc3ncncc3I)c2c1 Cc1cc(C(=O)NC2(CNC(=O)Cc3ccc(Br)nc3)CC2)cc(C)c1Cl CC1N(C(c2cc(CNC(C3CCCSC3)=O)ccn2)=O)CCOC1(C)C N1(C(CN(C(CC2C(C)C2)=O)C2CCC2)=O)CCC2CCN(C)CC12 C(CC(C(=O)Nc1cccc(F)c1)NC(=O)Cc1scnc1C)OC C1(C(N(C2CCN(c3nnc(CC)s3)CC2)CC#C)=O)CCCCNC1=O Cc1ccnn1CC(=O)NCC(O)CCNC(=O)CCCn1ccnn1 n1(CC(=O)NC(CCCNC(C2C(C=C)OCC2)=O)C)cnc2cc(C)ccc12 c1(OC(C)C(N2CCN(C(c3ccc(Cl)s3)=O)CC2)=O)cccc(Br)c1 C1(C(=O)NC2(C(O)CO)CCC2)CC2(CC2)CN1C(C1CC2COCC2C1)=O C#CCCCC(C)C(=O)NC(C)C(=O)NCC(C)N=[N+]=[N-] c1(OC)cc(Br)cnc1CNC1CCC(NC(=O)C(c2ccc(C)cc2)(C)C)C1 C1(NC(CC2(C)CC2(F)Cl)=O)CCC2CN(C(c3cncc(Cl)c3Cl)=O)CC2C1 c1(C(=O)NC(C)CN(C(=O)C(C)C(C)(C)C)C)cccc(S(=O)(=O)CF)c1 c1(C(N(C(C)CNC(=O)CC(F)(F)c2ccccc2)C)=O)cccn(O)c1=O C1(NC(Cc2c(C)ocn2)=O)CCN(C(=O)CSc2ccc(O)cc2)CC1F C=Cn1nccc1C(=O)NCC12CC1CN(C(c1ccccc1OCC#N)=O)C2 C1(N(C(C(C)OC(C)=O)=O)C)CCCN(C(=O)C(O)Cn2cncn2)C1 Cc1nn(C)c(C)c1CC(=O)NCC1(CNC(=O)Cn2ccccc2=O)CC1 Cc1ccc(CC(=O)NCC2CC2CNC(c2cncc(C(N)=O)c2)=O)cc1O C1(NC(C2=CN=C(OC)CC2)=O)COC2CN(C(=O)CC3(C)OCCO3)CC12 CCC(C)C(O)C(=O)NC1C2CC1N(C(c1cccc(F)c1C(F)(F)F)=O)C2 C1(NC(c2ccnnc2Cl)=O)CC2CCC1N2C(c1csc(Br)n1)=O c1(CC)ccnc(C(=O)NC(CN(C)C)C(=O)N(C2CCCC2C#N)C)c1 C1(NC(CS(CC)=O)=O)CCC2(CC1)CN(C(c1ccc(Cl)nc1N)=O)C2 c1(CN(C(C)(C)C)C(=O)NCC2CCCCC2O)cc(Cl)ncc1Cl c1(C(=O)NC2CN(C(CS(CC)=O)=O)C(C)(C)C2)cnc(O)n(C)c1=O N1(C(C)=O)CS(=O)(=O)CC1C(N1CCN(C(c2cccc(N)n2)=O)CC1CO)=O c1(C(N2CC(C(=O)OC)OC(CC)C2)C(=O)NCC=C)ccc(OC)c(C)n1 c1(C(=O)NCC(C)(O)CNC(c2cn[nH]c2)=O)cc2cccnc2[nH]1 N1(C(C(C)(C)F)=O)CCC2(CC1)CC(Nc1ncc(I)cn1)CO2 C1(N(C(C2(C)CCCN2C(c2ccc(O)nc2)=O)=O)C2CC2)CC1C1CCCCC1 N1(c2ccc(C#N)nn2)CC2(C1)C(NC(c1ccc(C3CC3)o1)=O)CCS2(=O)=O C(=O)(CCC(C(C)C)NC(C1COCC(C)O1)=O)NCCN1CC=C(C)CC1 n1(CCCC2C(C)C2)nc(-c2ccn(C)n2)nc1CCc1cccnc1 C1(CC)CC(O)CN1C(=O)C(N1CCC(NC(=O)CN2CCC(C)CC2)C1)=O C1(C(=O)NC(C)CCCCO)CN(C(=O)C=CC(=O)N(C)C)CC(C)(C)C1 c1(C(=O)NC(CNC(C(C)n2cccn2)=O)C)c[nH]c2cccnc2c1=O c12cc(n[nH]1)NC(=O)CNC2=O.C1(C2CCC2)(C(C2(COC)CC2)=O)CCC1 C1(NCC2C(Cl)c3cc(Br)ccc3O2)CC2(CCC(F)(F)CC2)C1 c1(C(=O)NCCNC(C2COC(=O)O2)=O)cc(Cl)c2n[nH]cc2c1 C(=O)(CCC(=O)N1CC(CNC(=O)C(C)NC(=O)NC)CC1C)NC N1(C(c2c(C)cc(C)o2)=O)CC(O)CCC1C(N1CCCC1C(=O)N(C)C)=O c1(CCC)ncc(C(c2nnnn2-c2ccccc2)NCCc2csc(C)n2)s1 CC#CCCCC(=O)N(C)CCNC(c1cc(Br)c(Cl)cn1)=O C1(COC)CN(C(=O)CC2C=NN(C)C2=O)CCN1C(c1cc(CCO)on1)=O c1(CC(N2CC3C(NC(c4c(C)nsc4C)=O)C3C2)=O)ccc(F)c(Cl)c1F Cc1cc(C(N2CCC(N(C)C(c3cn(C)cc3C)=O)C(C)C2)=O)c(C)c(C)c1 C(=O)(CCC(C)(C)N(C)C)NC1CC(C(N(C)CCN(C)C2CC2)=O)C1(C)C c1(C(N2CCC(C(C)NC(CNS(NC)(=O)=O)=O)C2)=O)n[nH]c(C2CC2)c1Cl C1(COC)(NC(C2(C)CC2)=O)CCN(C(C2CCCCC2c2ccccc2)=O)C1 c1(N2CCC(CC=C)(NC(C3CCCCNC3=O)=O)C2)ncnc2sccc12 c1(C(=O)NCC(C)NC(c2ccn(Cn3cccn3)n2)=O)cc2c([nH]1)CCCC2 c1(C(N(CCC(C(C)(C)C)NC(c2ccc[nH]2)=O)C)=O)cnn2c(=O)cc[nH]c12 c1(CNC(c2ccc(Br)cc2)CO)ccc(N)c(C(F)(F)F)c1 c1(C(N2C(CC)CN(C(c3cn(CC)nn3)=O)CC2)=O)ccc2sncc2c1 N1(C(c2nc(C)sc2C)=O)CC(C(=O)NC(C)CCC(F)(F)F)CC(C)(C)C1 c1(C(=O)NC(C)C(C)NC(c2ccns2)=O)ccccc1OC(F)F c1(C(=O)NC(C)(Cc2ccncc2)CO)cncc(C(F)(F)F)n1 C1(C(N2CCC(NC(C(CC)(C)CC)=O)C(C)C2)=O)CCCC2(C1)CC2(F)F n1(CC)c(=O)n(CC)c2cc(NC(N3CCSC(C)C3CCOC)=O)ccc12 N1(C(CSC(C)C)=O)CCC2CCC(NC(C3CCn4c(O)nnc4C3)=O)C1C2 CCCS(=O)(=O)C(C)C(=O)NCc1ccc(CNC(C2CC(O)C2)=O)cc1 c1(C(=O)NC2CCN(C(c3c(C(C)=O)cccc3)=O)C2C)cccc2oncc12 C1(NC(C(C(C)O)C)=O)CN(C(c2ccn(C)c2)=O)CC12CCOCC2 Cc1cc(C(=O)NC(C)(CNC(c2cnsn2)=O)C(C)C)c(Cl)cc1F C1(N(C(CC2(CNC(C(CC)OCC)=O)CC2)=O)C)CCCC(C)(C)C1 c1(CNC(C2CC(NCC3CCN(C)CC3)C2)=O)cc(Cl)ccc1F N(C(=NCC(F)F)N1CCC(C)(OC)C1)Cc1nc(CC)[nH]n1 CN1C(=O)CC(C(N2CC3C(CNC(=O)CCC4CC4(C)C)C3C2)=O)NC1=O N#Cc1cc(C(=O)NCC(C2CC2)NC(=O)CNC(c2ccco2)=O)co1 c1(CC)ccc(C(N2CC3C(NC(=O)CS(=O)(=O)NC4CC4)C3C2)=O)c(C)n1 c1(C(=O)NC2CCC(C(=O)NC(C)CCO)CC2)cc(Br)nc(Br)c1 c1(CNC(C2C(C)C2)=O)cc(O)nc(CNC(c2ccc(F)cc2)=O)n1 N1(C(C23CC(C(=O)OC)(C2)C3)=O)CCOCC(OC2CN(C(=O)C3CC3)C2)C1 C1(C(C)NC(C(C2CCOC2)OC)=O)CCN(c2nnco2)C1 C(=O)(CCCCC(=O)NCC(n1cc(-c2ccccc2N)nn1)C)OC C1(C(=O)NC(CCN(C(=O)CCc2cccc(O)n2)C)(C)C)CC2C=CC1CC2 Cc1scc(C(=O)NCC(C)(C)CNC(=O)CC23CCC(CC2)C3)c1C CC1(C)CCCCC1C(=O)NC(C(N1CCC(F)(F)C1)=O)c1ccoc1 CC(CNC(c1ccc2nc(O)[nH]c2c1)=O)CN=c1cc(Cl)nc(C(C)(C)C)[nH]1 N1(C(C(N2CCOC2=O)C)=O)CCN(C(C2CC23CCCC3)=O)CC1c1cn[nH]c1 CCCC(F)C(=O)NCCC(O)CNC(c1ccc(C(C)C)s1)=O CC1(C)CCOC(CC(N2CC3(C2)CN(C(=O)C=CC2CC2)C3)=O)C1 C1(CCNC(c2onc(C)n2)=O)CCCN(C(=O)CCOC2CCOCC2)CC1 c1(C(N2C3C(CNC(C(C)OC)=O)C(C3)C2)=O)c(F)cccc1Br Cc1nc(C(=O)NC2C=CC(CC(N3CC(CN(C)C)C3)=O)C2)c(C)s1 c1(OC)ccnc(NC(=O)CC2CCCN2Cc2cccc(CC(=O)O)c2)c1 Cc1ccnc(NC(=O)CCCCCc2ccc(F)cc2)c1Br c1(C(=O)NCC(C)CNC(C2CCC(O)C2)=O)cc([N+](=O)[O-])ccc1Cl c1(CC)nc(C)ncc1C(N1CC2(CC(NC(=O)C(C)C(F)(F)F)C2)C1)=O C1(C)(CNC(CCc2ncn(C)c2)=O)CCN(C(=O)CC(F)(F)F)C1 Cc1nc2ccccc2c(C(N2CC(CNC(c3cnsc3)=O)C(C)C2)=O)c1C C1(C)(C(c2nnnn2C2CCC2)NC(CC)COC)CCCCCC1 Cn1ccn2ncc(C(N3CCN(C(=O)C=C4CCCC4)C4CC34)=O)c12 Cc1cc(F)c(Cl)cc1C(N1CCC(NC(=O)CCCF)CC1)=O c1(C(N2CCC(N(c3scc(C)n3)C)C2)=O)cccc(I)c1F C1(C(N2CCC(C)CC2)=O)CN(C(=O)C(F)(F)CN(C)C)CCC1(C)C.CO C1(NC(=O)C=C2CC2)C2CCC1N(C(=O)Cc1ccc(-c3nnco3)cc1)C2 N1(C(c2cn(CC)nc2C2CC2)=O)CCC2(CCC2)C(CNC(C2(F)CC2)=O)C1 c1(CC(=O)NC2CCN(C(C3(C(N)=O)CCC3)=O)CC2)n[nH]c2cc(Cl)ccc12 N1(C(CC2(CNC(c3c(C)ccs3)=O)CC2)=O)CCC2CC1C(=O)N2C c1(CC(=O)NC2CN(C(C3(C(=O)OC)CC3)=O)C2)ccccc1OC C1(C(C)(C)C)CCC(C(=O)NCC2CC(NC(C3CC34CC4)=O)C2)CC1 C(=O)(CCCCC)N(CC(C)NC(c1c(CC)ocn1)=O)C c1(NCCCCC(=O)N2C(C(=O)NCC3(C)CC3)CCC2)cncc([N+](=O)[O-])c1 CCC(O)C(C)(C)C(=O)N(CCC(C)NC(=O)C(=O)NCC(F)(F)F)C N1(C(C(=O)NC(CC)(C)C)C2CCOC2)CC(C)OC(C)(C(F)F)C1 C=CCC(C(=O)N1CC(O)(CNC(c2cc(C(C)(C)C)c[nH]2)=O)C1)C(C)(C)C S(=O)(=O)(CC(=O)NCC1(C)CCC(C(=O)NC2CCCC2)C1)N(C)C.C1(=O)CCN1 CC(CCC(=O)NCCCS(C)=O)NC(C1(CO)CC(C)(C)C1)=O c12cc(ccn1)C(=O)N2.CC1(F)CC(C(=O)NC2CC(=Cc3nn[nH]n3)C2)C1 C1(C(=O)NC(c2ncc(F)cn2)C)(NC(=O)C(C)NC=O)CCCCC1 CC1CC(NC(c2cc(F)cnc2O)=O)CCN1C(=O)COc1ccsc1 O=C(C1=CC2CC(C1)CC2O)NCCN(C(c1cn(CCF)nn1)=O)CC1CC1 CC1Cc2cc(Br)ccc2CN1C(=O)NC1CCCC(F)(F)C1(C)C C1(C(NOC)=O)(C(=O)NC(C)CO)CCN(CC(c2cccc(O)c2)O)CC1 CCCC(F)C(=O)NC(CO)C(=O)NC1C2CCCCC12 C(=O)(CCC(F)(F)F)N1CCC(C(C)Nc2nccc(OCCC)n2)C1 c1(N2C(CNC(C3(CC(C)C)CCCC3)=O)CCCC2)nc2ccc(Br)cc2o1 C1(CNC(CCCCOC)=O)CCN(C(=O)Cc2ncccc2C)CC1O N1(C(CCCOC(C)=O)=O)CCC(NC(=O)Cc2cccc(F)c2)C(CO)CC1 N1(C(C(C=C=C)C)=O)CCC(C2CCN(C(C3CC(C)(CC)C3)=O)C2)CC1 c1(C(N2CC(CCCNC(C=CCC)=O)OCC2)=O)cc(O)cc(F)c1 c1(CC(=O)NCC(CC=C)NC(=O)Cn2nc(C)cc2C)ccc2c(c1)CCC2 CC(C)(C(=O)NCC(C1CCCCC1)NC(=O)CN(C)C1CC1)C(N)=O C(=O)(CC(C)C(=O)N1CCC(c2cscc2C(=O)OC)CC1)OC C1(NC(C2C(C)C2)=O)(CNC(=O)C(C)(C)c2cc[nH]n2)CCCCC1 CC(CC(=O)NCC1CCCCN1C(C1CCC(C)(C)O1)=O)C(F)(F)F N1(C(CC2CC(=O)NC2=O)=O)CCCCC(NC(C2CCC=CCCC2)=O)C1 c1(N2CC3CC(NC(=O)C(F)=C4CCCC4)CC3C2)c(F)cc([N+](=O)[O-])cc1F C1(C2(O)CCN(C(C3CCC(C)C(C)C3)=O)CC2)(NC(CCCOCC)=O)CC1 N1(CC)CCCC1C(N1CCC(C(=O)NCCC(C)(O)C2CC2)C1)=O N1(C(c2c(C#N)scc2)=O)CC2CN(C(=O)CNC(=O)NCC3CC3)C2C1 c1(C(C(=O)NC2CCC(N(C)C(=O)C3CC3)C2)=O)c[nH]c2cc(F)ccc12 c1(C(=O)NCCN(C(=O)CCc2cocn2)C2CC2)ccc(-c2nc[nH]n2)cc1 c1(CNC(C(CC)(C)C(F)F)=O)n[nH]c2c1CN(C(C1(C#N)CC1)=O)CC2 CCC(CC(=O)NC(CNC(c1cc(C2CC2)ccn1)=O)C1CC1)C1CCC1 CCC(CCNC1(CO)CCSC1)C(=O)NN1CCCC1C(=O)OCSC C(=O)(CC(C)CC(C)C)NC1CCN(C(c2ncn(CC)n2)=O)CC1O N1(C(C(C)(O)c2ccccc2)=O)CCC(CO)(Cc2ccccc2)C1 N1(C(CCC=CC=C)=O)CC(=O)NCC1C(=O)N(CC(C)O)CCF Cc1ncc(C(=O)NCC2(CCNC(=O)Cn3ccc(C(F)F)n3)CC2)c(=N)[nH]1 C1(NC(C#CC(C)C)=O)CN(C(c2ncnc3c2CCC3)=O)CC12CCC2 C1(OCCN)CCN(C(c2ncc(CCC(=O)N)o2)=O)C1.CC(=O)C1CC1N(C)C CC1CC(NC(=O)C(C)(C)C(F)F)CN(C(=O)CC2CCNC(=O)C2)C1 C1(NC(c2ncc(CC)cn2)=O)C2CCN(C(=O)CCCOC(C)(C)C)CC12 c1(C(N2CC(SC)C(NC(=O)Cn3cncn3)C2)=O)c(C(F)(F)F)cccc1F C12(CNC(C3CC3(F)F)=O)CCCC1N(c1ccnc(C3CCCC3)n1)CCC2 c1(C(N(CC(C)NC(Cn2c(C)cc(C)n2)=O)C)=O)cncc2cc(Cl)ccc12 C(=O)(C(C)(C)C(F)(F)F)N1C2CC(CNC(C=CSC)=O)C1CC2 c1(C(=O)NCC2(OC)CCN(C(c3cc(C)[nH]n3)=O)C2)cc(C(=O)OC)ccc1C N1(C(C(CC(CC)C)C)=O)CCC2(CC1)CCN(C(=O)C#CC(C)(C)C)C2 N1(C(c2c(CCNC(c3cc(CC)on3)=O)n[nH]c2)=O)CCCOC(C)C1 C(CCS(=O)(=O)c1ccc(F)cc1)NC(=NCCOC)NCC(C)(C)C1CC1 C1(NC(CCCC#C)=O)CCN(C(=O)CC(C)NC(N)=O)C12CCCC2 CCC(C)C(O)C(C)C(=O)NCC(C)=CC(=O)NCC(C)(O)CC(C)C N=c1nc(C(=O)NCC2(C(=O)NC3CN(c4ncco4)C3)CCC2)[nH][nH]1 C1(NC(c2c(CC)nns2)=O)CCN(C(C2(F)CCCC2)=O)C1(C)C CC1C2C(CCN2C(C2CCS(=O)CC2)=O)CN1C(c1cc(O)nn1C)=O Cc1noc2cc(C(=O)NCCCCN(C(=O)C=Cc3nccs3)C)ccc12 c1(C(N2CC(SC)C(NC(=O)C(CC(C)C)N(C)C)C2)=O)ccc(N=[N+]=[N-])cc1 Cc1nc(C)c(C(N2CCN(C(c3cccnc3S)=O)C(C(F)F)C2)=O)nc1C C1(C)(CCC(=O)NC2CCC(N(C)CC3CN(S(C)(=O)=O)C3)CC2)CCC(=O)N1 c1(CN(C(C2N(C(=O)OC(C)(C)C)CCC2)=O)C2CC2)cc2c(cc1Br)OCO2 C1(NC(C(N(C(C(COC)C)=O)C)C2CC2)=O)CCC2(CCC2)C1 c1(CN(C(C2CC3CC3C2)=O)Cc2nc(C)on2)ccc2nc(N(C)C)sc2c1 n1(CCN(C(C)C(=O)NCCc2cccs2)C)cc(CN)nn1 C1(O)(CCNC(C(C)=C(CC)C)=O)CCCN(C(=O)Cn2c(C)csc2=O)C1 CC1(C)CCN(C(c2ccoc2)=O)CC1CNC(c1ccnnc1O)=O Cc1ccc(C)c2c1OCCC2NCc1scc2c1OCCO2 O=S(=O)(c1cc2ccc(F)cc2s1)N1C2CCC1COC2 C(=O)(C1CCCn2ccnc21)NCc1nc(CNC(Cn2cnc(=N)[nH]2)=O)sc1 N1(C(Cc2c(C)noc2)=O)CCC(NC(=O)C(F)(F)CO)C(CO)C1 C(CNC(=O)CN(C)CCO)(CC(F)(F)F)NC(C(C)OC)=O.C(CCCC)(OC)OC CCC(C(=O)NCCCNC(C12CCCC1C2)=O)Oc1ccccc1 CC1CCN(C(C2OCCN(C)C2=O)=O)CC1NC(=O)C(C1CC(F)(F)C1)O Cc1onc(C(=O)NCC2CN(C(=O)C(O)C3CC3)C2)c1Br c1(C(=O)NCC2(NC(c3cc(CC)no3)=O)CCC2)cccc(C2(F)COC2)c1 c1(C(N2C(C(=O)O)CCOCC2)=O)cc2n(c(=O)c1)CCS2 Cc1ccc(C(N2CC(COC(C)(C)C)(NC(=O)C=CCO)C2)=O)cc1CO C(=O)(C1=CCCCCC1)N(C1CC2CCC(C1)N2C(=O)Cn1ccnn1)C c1(C(N2C(C(=O)NC(C(C)C)CCO)COCC2)=O)c(Br)cccc1Br c1(OC)ccc(CCNC(=O)CN2CCCC2CCO)cc1OCC(N)=O C1(CN(C)CC)(CNC(=O)COCC(C)C)CCCCC1.C1CC(=O)N1 Cc1cncc(C(=O)NC(C)CCN(C(=O)CSCC(C)C)C)n1 C(=O)(C1OCCn2ccnc21)N1CC2C(NC(=O)CCc3ccc(Cl)cc3)C2C1 N1(C(CCc2cc(C)no2)=O)CCN(C(C2CC(CF)C2)=O)C(CF)C1 CC1C(NC(C2CC2(C)Br)=O)CC2CCC1N2C(c1cc2ccccc2o1)=O c1(C(=O)NCC2C(NC(c3c(C)nc(C4CC4)[nH]3)=O)C2)c[nH]c2cccc(Cl)c12 N1(C(CCCN(C(C)=O)C)=O)CC2CC1CN(C(=O)Cc1ccc(C)cc1Cl)C2 C1(NC(c2scc(C(C)=O)c2)=O)CC12CC(NC(=O)CC(F)(F)Cl)C2 C1(NC(C(C)SCCOCCOC)=O)CC(C)(NC(=O)CC2CC(=C)C2)C1 C1(C(=O)O)CC12CN(C(C1CCN(S(=O)(=O)C(F)(F)F)CC1)=O)C2 c1(CC(N2CC(O)CC(OC)O2)=O)cc2ccccc2n1C CC1CN(C)C(C)CC1NC(=O)CC(C1CC1)NC(c1cnc(O)o1)=O C12(C(F)(F)F)CCC(Nc3nccc(Oc4ccccc4)n3)(CO1)C2 C1(C(=O)NCC(c2ccc(OC)cc2)NC(c2ccns2)=O)C2CCC(F)(F)C12 c1(C(=O)NC(CC(C)NC(c2c(SC)cnn2C)=O)C)c(Cl)nn(C)c1C CC1(C)CCCCC1=CC(=O)NCC1(CCNC(=O)CC(=O)N(C)C)CC1 c1(C(=O)NC(CNC(Cc2c(C)ncs2)=O)CC(C)C)csc2nccn12 CCC(C)CC(C)C(=O)N1CC(NC(=O)Cn2c(C)cc(O)cc2=O)CC1C c1(CC(N2CCC(NC(CNC(CC)=O)=O)C2)=O)c(C)cnn1C C#Cc1ccc(C(=O)NC(CNC(=O)CCc2nc(C)cs2)C(C)C(C)C)cn1 N1(C(CCSC)=O)CCC(NC(=O)CCc2cncnc2O)CC1C1CC1 c1(-c2ccc(NC(c3n(C)ncn3)=O)s2)ccc(C#N)nc1 C(=O)(CCC(C)(C)OC)NCCNC(C1CCN(CC=C)C1)=O C(C(CC(F)(F)F)NC(c1ccc(C2CC2)cc1)=O)NC(=O)CSc1ccoc1 C1(C(N2CC3(COCCO3)C2)=O)COC2CN(C(c3ccccc3Cl)=O)CC12 c1(COC)nc(N(CC(C)NC(C2(c3ccccc3F)CC2)=O)C)cc(C)n1 N1(C(CC2N(C(CC=O)=O)CCC2)=O)CC(n2cc(C3CC3)nn2)C(O)C1.NC Cc1c(NC(C2(CO)CCC2)=O)[nH]c2ccc(C(=O)N(C)CCOCCO)cc12 N1(C(c2cn(CC(C)N)nc2)=O)CC2(C)CC1(C(=O)O)C2 N1(c2c(C)nc(=N)[nH]c2C)CCC2(CC1)CC2(C)C(=O)NC1CC(O)C1OC c1(C(N2CC(NC(c3scc(C)n3)=O)C(O)C2)=O)cccc2cc(Br)cnc12 Cc1ccc(C(=O)NCCN(C(=O)C(c2ccccc2)O)C2CC2)c(F)c1 c1(-c2nc(-c3cc[nH]n3)nn2C2CCOC2)cc2sc(Cl)cc2s1 c1(SC)ccc(CCC(=O)N2CCC2Cn2cc(CO)nn2)cc1 Cc1cc(=NCCc2nc(O)n[nH]2)[nH]c(N2CCC(CN3CCOCC3)C2)n1 Cn1c(O)nc2cc(C(=O)NC3CC(CNC(c4cccs4)=O)C3(C)C)ccc12 Cn1cc(Cl)c(C(=O)NCc2nc(CNC(C3CC4(C3)CC4F)=O)cs2)n1 C1(C(N(C)CC2COCCN2C(c2cc(Cl)n(C)n2)=O)=O)CCCC12CCC2 c1(C(=O)NC23CC(CNC(C(C)OCCCC)=O)(OC2)C3)cccc2ncsc12 n1(C(C)C)c(O)nc2ccc(C(N3CC(NC(=O)C4=CCCC4(C)C)C3)=O)cc12 C12(C(=O)NCC#CC(=O)NC(C=C)COC)CCCC1OCC2 C(=O)(C1=CCCS1)NCCN(C(c1scc(OC)c1)=O)CC1CC1 Cc1cc([N+](=O)[O-])cc(C(=O)NCC2COCCN(C(c3ocnc3C)=O)C2)n1 Cc1cc(=NCC2COC(C)(C)C2)[nH]c(NCCS(=O)(=O)CC(F)(F)F)n1 CCC(CC(=O)N(C)CC=CC(=O)NC1CC1O)CC(C)C c1(C(=O)NCC2N(C(CCN(C)CC)=O)C3C(C2)C3)cccn2c(C)nnc12 C1(C(=O)OC)CN(C(=O)CCn2nc(C)c3c2CCCC3)C2(CCOCC2)C1 N1(C(COCC(=C)C)=O)CCCC2(CCC2NC(C2CCC(=O)N2)=O)C1 N1(C(CC(CC)C(C)(C)C)=O)CCC(C2(NC(C3CN(C(C)=O)C3)=O)CCC2)CC1 c1(N2C3CN(C(Cc4onc(C)n4)=O)C(C3)C2)ncnc2ccc(C(F)(F)F)cc12 N#Cc1cc(NC(C2CCCC(NCc3cc(Br)c(Br)s3)C2)=O)cc(F)c1 c1(C(=O)NCCC2CCC(NC(CCSCC)=O)C2)cc(S(N)(=O)=O)ccn1 Cc1cc(CC(N2CC(CNC(=O)COC3(C)CCC3)CC2C)=O)ccc1O C1(CC)OCCC1C(N1CCCC1C(=O)NOCc1nc[nH]n1)=O CC(C)(C)CCCCC(=O)NCC(C(=O)NCCC1CCSC1)C(C)(C)C C1(NC(C(C=C)O)=O)CC(F)CN(C(c2cccc(OC)c2OC)=O)C1 c1(OCCC(=O)NC2(CNC(C=C(CCC)C)=O)CC2)ccccc1[N+](=O)[O-] C1(NCC(C)C(=O)N(C(C)C(C)(C)CN(C)C)C)CC2CCC(C1)N2C C1(NC(CC=CCC)=O)C2CC3C(C2)C13C(=O)NCCc1ncc[nH]1 N(C1CN(C(C23CC(C#N)(C2)C3)=O)Cc2ccccc21)C(CCC(=C)C)=O C12(CNC(C(=O)Nc3cc(C)no3)=O)CCCC1CCN2C(=O)CN1CC2CC2C1 CC1(C)CC(CC(=O)NC2CC(C)(NC(c3ccnc(C(C)(F)F)c3)=O)C2)CO1 C1(NC(CCC(=O)NCCC)=O)CN(Cc2cccnc2C)CCC1C C(CCC(C(=O)N(C(C)CC1CC1)C)NC(=O)CCC(C)(F)F)OC C(=O)(C(C)CC(N)=O)NC(c1nc(C(=O)NCC2CC3(CC3)C(=O)O2)co1)C N1(C(c2ccc(S(=O)(=O)NC)s2)C(=O)NC2CC2)CCN(C(=O)OC)CCC1(C)C CC1CCN(C(c2cc(Cl)cc(Cl)n2)=O)CC1NC(c1cc(C2CC2)on1)=O c1(CNC(c2ccc3ncoc3c2)=O)ncn2c1CCCCC2 C(C(=O)NCCCCc1ccccc1C)(C(C)CC)NC(=O)OCC C(=O)(CCC1=CCCCC1)NC1(COC)CN(C(C2Cc3nccn3C2)=O)C1 N1(C(C=CCN(C)CC)=O)CCC(NC(c2ccc(CO)c(Cl)c2)=O)CC(O)C1 C(CCC(=O)NCCCNC(C1CC1F)=O)N(S(C)(=O)=O)C N1(C(COCCOC)=O)CCCC(C)(C)C1C(=O)NC1CC=C(C(C)C)CC1 N1(C(C(=O)NC(c2nnc(C(=O)OCC)s2)C)=O)CCC(O)C12CCC2 c1(CNC(C2CCCN(Cc3ccnc(Cl)c3Cl)CC2)=O)ccc(F)c(Br)c1 c1(Nc2c(C#N)ccc(C)n2)ncc2cc(F)ccc2n1 C12(CC(=O)NCCCN)CCC(CC1)OC2.C1(CO)C(=O)N1.CC(C)(C)OC(N)=O C12(CNC(C3C(OCC)C3)=O)CCCC(CN1C(c1nn(C)cc1Br)=O)C2 Cc1ccsc1C=CC(N1CCCC1CN(C)C(c1cnc(C2CC2)[nH]1)=O)=O C1(C(N2CCC(CNC(CC(COC)C)=O)C2(C)C)=O)C2CCC1(C)C2(C)C N1(C(C(c2ccc(C)s2)C)=O)CC(NC(=O)CCSC2CCCC2)CC1(C)C Cc1[nH]c2ccc(C(=O)NCc3cn(C4CC4)cn3)cc2c1C c1(C(=O)NC(CC)CNC(C2CC2(C)CCC(C)C)=O)ccc(CCF)cc1 C1(NC(C2C(CC)OCC2)=O)CCC2CN(c3nc(OC)nc(OC)n3)CC2C1 C1(C(=O)NCC(C2CCCN2C(c2ncoc2C)=O)(C)C)(CC)CC(C)(C)C1 C1(C(=O)NCCCN(C)C(C2CC3CCC2C32CC2)=O)Cc2ccccc2O1 C1(C(=O)NCCSC(C)C)(NC(CC(=O)OCCC(C)C)=O)CCCC1C N1(C(c2cc(C)[nH]c2C)=O)CCCN(C(c2ncc(Cl)cc2Cl)=O)CC1C(C)C N1(C(Cc2nc(CC)sc2)=O)CCC(CO)C(NC(c2sccc2Cl)=O)C1 Cc1cc(C(N2CC(O)CC2CNC(C2CC23CC3)=O)=O)nn1CCO c1(C(C(N2CC(NC(c3c(C)nc(C)[nH]3)=O)C(F)C2)=O)=O)ccccc1[N+](=O)[O-] C12(C(=O)NCC#CCNC(C3N(C(CCC)=O)CSC3)=O)CCCN(CC1)C2 c1(C(N2CCN(CCCCC)CC2)C(=O)NCC(=C)C)ccccc1Cl c1(C2(C(C)NC(=O)C(N3CCc4sccc4C3)=O)CC2)ccc(F)c(C#N)c1 C(=O)(CCC(=O)c1cccs1)NC1C(C(C)NC(=O)CC(C)N(C)C)CCC1 C1(NC(C=CCCC)=O)C2CC3C(C2)C13C(=O)NCc1ccc(O)cc1C C1(C(N(CC(CC)NC(=O)Cn2nccc2C)C)=O)CCc2ncsc2C1 c1(C(=O)NC(CNC(=O)CCCc2ccc(F)cc2)CO)ncnc2sccc12 C1(C(N(C(C)C(=O)NCc2ncc(C)s2)CC)=O)C2CCCOC12 CCCC(C(=O)N(C1CCN(C(c2occ(C)c2C)=O)C1)CCO)OC.C(C)(C)(C)SC c1(C(N2CCCC(CNC(=O)COc3ccsc3)C2)=O)ccc2nn[nH]c2c1 C1(C)(C(=O)NC(C=C)C)CCCN1C(c1ccc(N2CCC(C)CC2)s1)=O CC1C(C)SCCN1C(=O)C1=CCN(C(C2(C)CNC(=O)N2)=O)C1 C1(F)(C(N2CC(CCNC(CCCN=[N+]=[N-])=O)OCC2)=O)CC12CCCCC2 Cc1ncnc(C)c1C(=O)NC1CCC1CNC(C12CCC1CC2)=O C1(CNC(CSCCOC)=O)CN(C(=O)CC(C)C)CC1O C(=O)(C(C)C1CC1)N(CCCNC(C1CCSC1)=O)C.C(=O)(CC1(N)CC1)OC c1(CC)ccc(C(=O)NC(C)CNC(=O)C(F)(F)C(F)F)cc1F c1(SCC(=O)NCC(C)(C(C)C)NC(C(CC)F)=O)ccc(F)c(F)c1 c1(C(=O)Nc2ccc(Cc3ccc(Cl)cc3)cc2)cccc(C#CCO)c1 CCCCCCCCNC(=O)C(n1cc(CC(O)CN(C)C)nn1)C Cc1nn(C)c(C)c1C(C)C(=O)NCC#CCNC(C1CCNC(=O)C1)=O S(=O)(=O)(c1ccc(NC(=O)NCC(O)COC(C)C)cc1)NCC(C)(C)OC CC1(C)C(CNC(c2cnco2)=O)CCN1C(=O)CCC1CC1(Cl)Cl C#Cc1cn(C)nc1S(=O)(=O)N1CCCC2OCCCC12 CC(C)CC(C)CC(=O)NC(C1CCCCN1C(c1cc2n(c1)CCOC2)=O)C C(C)(C(=O)NNC(=O)C(C)(C)CCCCNC(C1CCCCC1O)=O)OCC Cn1ncc(CNC(=O)C(CCF)NC(c2cncnc2)=O)c1O C(=O)(C1=NOC2(CCC2)C1)OCC.O=C(CC(Cl)Cl)NC1(C)CCOC1 C=Cn1nccc1C(N1CC(OCCNC(C2CC(C)CO2)=O)C1)=O c1(CNC(=O)NC2(CO)CCS(=O)(=O)CC2)ccc2c(c1)S(=O)(=O)CC2 N1(C(CN2CCC(C)CC2)=O)CCCC2CN(C(=O)CN3CC4CC4C3)CCC12 C1(C(N(C(C)C(F)F)C)=O)CCCN1C(C1(C)C=CCC1)=O C1(C(C)NC(N(CCOC)CCF)=O)CCC1 c1(C(N2C(CNC(C(C)=CC3CC3)=O)COCC2)=O)nccc2n[nH]cc12 c1(OC)ccccc1CCNCCCCC1CCN(C(=O)OC(C)(C)C)CC1 CC1CN(C(c2cc(CCO)on2)=O)CC1C(N)=O.C12CCC(O1)NC2=O C1(NC(CC(=C)C)=O)CC2(CCC(CNC(c3cnn(C)c(=O)c3)=O)OC2)C1 C1(C(=O)NCC(C(=O)OC)(C)O)CN(C(C2(C(=O)N(C)C)CC2)=O)CCC1(C)C C(=O)(C(C)(O)Cc1ccccc1)NCCOCCCNC(CNC(CC)=O)=O N1(C(CCC(=C)Cl)=O)CC2C3CCC(C2C1)N(C(c1ccc(F)c(N)c1)=O)C3 n1(CC#C)cccc1C(=O)NC1CCCC1NC(=O)COc1ccccc1.C(=O)(N)OC C1(NC(COCCC)=O)CC2(CCC(CNC(C3(C#N)CCCO3)=O)OC2)C1 CC(C)(C(=O)N1CC2CC(NC(c3ccc(O)nc3)=O)CC2C1)C(F)(F)F c1(C(=O)NCCC(C)NC(CCc2onc(C)n2)=O)cc(F)c(O)c(F)c1 CCC(O)C(C)C(=O)N1CCOCC1c1noc(-c2cn(CC)nn2)n1 C1(C(=O)NCC(CC)NC(c2ncccn2)=O)CCCCN1C1CCCC1 C(=O)(CCCCC(C)CC)NC1C(NC(c2ccc(C#C)c(OC)c2)=O)CC1 CC(C(=O)NCC1(F)CCCN(C(=O)C(C)(C)n2cccn2)C1)S(C)(=O)=O c1(CC)cc(C(N2CCC(CNC(=O)C(c3ccc(Cl)s3)=O)C2)=O)ncn1 N1(C(C2(C)C(C)C2)=O)CC2(CC(C(=O)Nc3ccccc3CN(C)C)CO2)C1 C(=O)(CC(C)(C)CC(F)F)NC1CCCN(C(COc2c(C)cccc2)=O)CC1 C1(C(=O)NCC2C(C(=O)NC3CCN(CC)C3)CC2)OCCOC1C c1(C(N2CCC(CC(C)NC(=O)CCc3cnc[nH]3)CC2)=O)cc(N)cnc1O n1(CC)nnnc1C(c1nnc(C)s1)NCc1ccc(Cl)o1 C1(=CCNC(C(c2ccccc2Cl)C)=O)CCN(C(=O)C(F)C2CCC2)CC1 N1(C(C2(C)CCCCC2(F)F)=O)CC2(C1)CN(C(C1CC(O)C1)=O)CC2CO N1(C(c2c(C)cccn2)=O)CCN(C(=O)C(=CC2CCCCC2)F)C(C)CC1C C1(CCC)CN(C(=O)Cc2cnsc2)CC1NC(c1ccncc1NC(C)=O)=O Cc1cnccc1C=CC(N1CCC2C(NC(c3ccc(CO)cn3)=O)C2C1)=O c1(NCc2cc(CC)no2)cc(C(C)(C)O)ncn1 N1(C(c2c(Br)cc(C(C)=O)s2)=O)CC2(CCCN(C(C3C(C)C3C)=O)C2)C1 c1(C(=O)NC2N3CC(NC(C4NC(=O)CC(C)C4)=O)C2CC3)cn2ccnc2cn1 CCCC(C(=O)N(C1CCN(C(C2CC2C)=O)CC1)CC)C(C)C N1(C(CC(CC)C)=O)CC2(CCOCC2)C1C(C)C CN1CCCC(C(=O)NC2COCC2NC(c2nccc(CC#N)n2)=O)C1 c1(N2C(C)CN(C3CC3)CC2)nccc(=NCc2c(N)cccc2Cl)[nH]1 C1(NC(C(C)CF)=O)CCN(C(=O)CN2CCCCCC2=O)CC12CCC2 C(Cc1cccs1)(CC(=O)OCc1ccccc1)C(C1(c2nn[nH]c2C2CC2)CC1)=O C1(CNC(=O)CCC2CC2)CC2CCC(C1)N2C(C1Cc2nccn2C1)=O N1(C(CCN(CC)CC)=O)CCC2(CCCCC2NC(c2cnco2)=O)C1 CC(F)(F)CCC(=O)NCCC(Cc1ccccc1)NC(=O)C=Cc1ccco1 C1(C(N2CC(OCC3CC3)C2)=O)CCN(C(=O)C2CC3(CCC3O)C2)O1 C1(C)(CNC(CCSC)=O)CC(C(N2CCC(n3cnnn3)C2)=O)C1 C1(CNC(CN(CC(C)(C)C)C)=O)CN(C(=O)C(C)(C)C(=O)OC)CC(C)(C)C1 c1(CNC(C2C(C)CCC2)=O)ccccc1N1CCN(C(C2CSC2)=O)CC1 N1(C(Cc2ccc(C(C)=O)cc2)=O)CC2CC(NC(C3CCC(=O)N3)=O)CC2C1 c1(C(N2CC(NC(=O)Cc3csc(S)n3)CC(OC)C2)=O)nc2cnccc2s1 N1(C(c2c(CCCC)ocn2)=O)CCC(C)N(C(=O)CCN(C(=O)CO)CC)CC1 Cc1nn(C)c2sc(C(=O)NC3CC4CC3N(C(C3(C)CCNC3=O)=O)C4)cc12 C(=O)(CCCCCCC(=O)N1CC2CCN(C(C3CC4C=CC3C4)=O)CC12)OC CC#CCCCC(=O)N1CCC1CCNC(C)=O C=CC1CN(C(c2cccn2C)=O)CC1NC(=O)C(O)Cc1ccccc1Cl N1(C(C(C)=CC=C)=O)CCCCCCC1C(=O)NCCc1cc[nH]n1 N1(C(C(C)n2cccn2)=O)CCc2sc(CNC(=O)CN=S(C)(C)=O)nc2C1 c1(CN2CCC(NC(C(c3ccc(F)cc3)N)=O)C2)cc(F)ccc1F Cc1ccc(CCC(=O)NC(C)CNC(=O)CC2OCCC2(C)C)cc1C N1(C(=O)CCCC2CC2)CC(CO)C2(C1)CN(C(C1CCCCCCC1)=O)C2 C1(CC(=O)NCCSCCNC(C)=O)CCCC1NC(c1cn(C)cn1)=O C1(C(N2CCC(COC)CC2)=O)CC2(CCC2N(C)C)C1 C(=O)(CCCCC(N)=O)NC1C2CN(C(CCCCCOCC)=O)CC21 c1(C(N2C(CC(C)C)C(=O)NCC2)=O)cnn2cccc(Cl)c12 C1(CNC(c2cnc(CC)[nH]2)=O)N(C(=O)CC2CCC(C)C(C)C2)CCCC1(C)C Cc1cc(C(=O)NC2CC(N(C(=O)CC(C)c3cnn(C)c3)C)C2)sc1Cl C1(C(=O)NCC2CCCN(C(c3ccccn3)=O)C2)CC2CC1C1CC21 N1(Cc2ccc(CCC)o2)CCc2c(OC)ccc(N(C)C)c2C1 CC1CCN(CCC(N2CCCC(CNC(=O)CC3NC(=O)NC3=O)C2)=O)CC1 C#CCCCCCCC(=O)NC1CN(C(=O)CSCCN(C)C)CC12CC2 C1(C(=O)NCCCN(C(C(CC)NC(N)=O)=O)C)CCOC(=O)N1 N1(C(c2c(OC)csc2)=O)CCC(CO)C(NC(c2cc(Cl)ccc2C)=O)C1 C(=O)(C1=NOC(C)C1C)NCCN(C(c1cccc(CS(C)=O)c1)=O)CC c1(NC(C(C2(O)CN(C(CC)=O)C2)F)=O)ccc(CC)cc1O C1(NC(CCOC(C)C)=O)CCC12CCN(C(c1ccc3snnc3c1)=O)CC2 c1(C(N2CCC(=CCNC(C=C(CCC)C)=O)CC2)=O)cc(Cl)nnc1Cl CC(O)C(C)C(=O)NC1CC(F)(CNC(c2coc(-c3ccc(Cl)cc3)n2)=O)C1 C(=O)(CC1=NNC(=O)C1)N1CCC(C)C(NC(c2ccccc2OCCF)=O)C1 n1(-c2cn(CCOC)nc2)nc(C2CCOC2)nc1-c1ccc(C)s1 CCCCC(CC)NC(=O)C(F)CC1CN(C(c2ccc(C(N)=O)o2)=O)C1 Cc1nn(C)c(-n2ccnc2C)c1C(=O)NCCC1CCN(C(=O)C(C)O)C1 CC1CC(NC(=O)CCCc2ccccn2)CCN1CCc1ccc(Br)cc1F c1(C(N2CCC(c3cn(C4CCCCNC4)nn3)C2)=O)n[nH]c2c1COC2 CC(CC(=O)N1CC(n2cc(CNS(C)(=O)=O)nn2)CO1)NC(C1CCC1)=O Nc1cc(C(N2CC3CC2CN3C(c2ccn3c2CCC3)=O)=O)cc(F)c1 N1(C(CC(CC=C)NC(c2ccccc2O)=O)=O)CCC(O)C12CCC2 C(=O)(CCCCC1CC1)N1CCC(CCNC(=O)CO)C1 S(=O)(=O)(c1ccc(C(=O)O)cc1F)NC1CN(C(C(c2ccc(C)cc2)C)=O)C1 c1(C(N2CCN(C(C(N)=O)=O)CC(O)C2)=O)cc(Cl)c([N+](=O)[O-])cc1F Cc1cc(-c2cn(C3(NC(C4C(CO)C4(C)C)=O)CCOCC3)nn2)cnc1F c1(CC(=O)NC(C2C(C)C2)C2CC2)cc(CN2CCCC2)no1 O=C1CCN(C(=O)NC23CCC(F)(CC2)C3)CC1c1ccc(F)cc1 C(C(C(=O)NN1CCCC1)NC(=O)COc1cnn(C2CC2)c1)OCC CCC(C)C(C(=O)NCC(CO)NC(=O)Cc1cc(C)sc1C)OC C1(C(=O)NCCCC(C)(C)NC(c2ccc(O)nn2)=O)CCc2ccccc2C1 c1(CC)cc(C(=O)NC2CCCC2NC(=O)CCc2cnn[nH]2)cc(N)c1 C12(CNC(=O)NC(C)C(=O)NC3CC3)CCCNC1CCC2 N(C(=NCCSC)NCC(N1CCCC1)=O)C(C)Cc1ccccc1 C1(C)(C(=O)NC2CC(CC(=O)Nc3cc(C)no3)C2)CC(F)(F)C1 O=S(=O)(c1cccc2c1OC(F)(F)O2)N1CC(Cc2ccsc2)C1 CC(C)C(C(=O)NCCCOCOC)Oc1nnc(-c2ccn(C)n2)s1 C1(NC(=NCCOC(C)C)NCCc2ccccc2Cl)CCc2ccccc2C1 N1(C(c2c(OC)nsc2)=O)CCCC(O)(CN(C)C(C2CC2(F)F)=O)C1 CC(C)C(C)C(C)CC(=O)N1CCC(C)(NC(c2cnsn2)=O)CC1 N1(C(CC(=O)NCC)=O)CCN(C)CC1CNC(c1cc(C(N)=O)cc(Cl)n1)=O Cc1nc(C(=O)NC(C2CCN(C(=O)C(C)c3ccsc3)CC2)C)[nH]c1C C1(CNC(c2ccc3ccc(C)cc3n2)=O)CC(N=c2[nH]cnc3cnccc23)C1 C1(C(=O)NC2C3CN(C(C4(C)CCCS4)=O)C2C3)CCCCC12CC2 N(C1CCOc2ccc(Br)cc21)C(C1CC(O)CN1C(=O)Cc1cc[nH]n1)=O N1(C(C(c2ccc(C)cc2)=O)=O)CCC(O)C(NC(=O)CN2CCSCC2)C1 c1(CN2C(CC(=O)NCc3ccc(C)s3)COCC2)cnc2ccoc2c1 N1(C(C(C(CC)(C)C)O)=O)CCC2(CCCCN(C(=O)CC(C)(F)F)C2)C1 C1(CNC(C(c2ccccc2)C)=O)CC(NC(c2ccncc2O)=O)CC1O CN1CCCC(CNC(=O)C#CCNC(C2(C)CCN(C)C2)=O)C1 N1(C(c2c(CNC(C(C(CC)C)OC)=O)noc2)=O)CCCC2COCC12 C1(SCC(=O)NC(CC2CCCC2)CF)CCCNC1 c1(C(N2CC(OC)(CNc3nc(=O)n(C)[nH]3)C2)=O)ncnc2scnc12 C12CCN(CC1C)C(=O)N2.C1(CC)CCCC2CC12.C12=CC(OC)(C=C1)CNC2 CC1(C(=O)NC2CC2NC(c2c(F)cccc2Br)=O)Cc2ccccc2N1 CCCC(CC(C)C)C(=O)NC1C=CCN(C(C2(N(C)C)CCCC2)=O)C1 C1(NC(C(C)OCCOC)=O)CCCC(NC(=O)C(c2cc(C)ccn2)(C)C)C1 C(=O)(CCC(=O)N(CCCOCCNC(=O)C(c1ncccc1F)(F)F)C)NC C(=O)(C(C)CS(C)(=O)=O)N(C1CCN(c2cc(C)nc(Cl)n2)C1)C N1(C(C2(CC=C)CC2)=O)CCCC(C2CCN(C(=O)C(C)(F)C(C)(C)F)CC2)C1 C1(CNC(Cc2ccc(C(C)=O)s2)=O)CC2CCC1N2C(=O)C(F)OC C(=O)(C1Cc2ccccc21)N1CCN(C(CCCn2c(C)ccc2C)=O)CC1 CC1(C)CC(C(=O)N2CC(NC(C3CC(n4ccnc4)C3)=O)C3(CC3)C2)=NO1 N#CCCCCCC(=O)NC1CCCC1NC(C1CCCC12CCC2)=O C(CCC(C(=O)NC1CCN(C)CC1C)NC(=O)CCCN=[N+]=[N-])OC C(=O)(CCC(C)CC)NCC1(CNC(c2c(C)nc(C(C)OCC)s2)=O)CC1 C1(C(=O)NCC2CCCCN2C(c2cc(COC)cn2C)=O)(CC)CCNC1=O c1(OC)cnccc1C(N1CC2CC1(CNC(=O)CC1CCCCC1C)C2)=O c1(C(=O)NC23C(CN(C(C4(C#C)CC4)=O)C2)C3)ccc(N=S(C)(C)=O)cc1 C1(C(N(C)CC2CCCC2)=O)CCN(C(C2(N)CC2)=O)CCO1 Cc1[nH]nc(C(=O)N(C)CC2C3CN(C(=O)C(C#N)C4CC4)CC23)c1C(F)(F)F N1(C(C=CCOC)=O)CCC(C)(CNC(c2ccc(C)nc2C)=O)CC1 O(C=C(C#N)C(=O)NCC(O)CNC(=O)CC1CCS(=O)(=O)C1)CC c1(OC)ncc(NC(c2ccc(CC3CC3(Cl)Cl)cc2)=O)cc1C CCC(C(=O)N1CC(F)CC1CN(C(=O)CSc1nncs1)C)C(C)C N12CC(OCC(=O)NC3CC(C)(C(=O)OC)C3)CC(C1)C2=O.C1(COC)CCCC1 C(=O)(N=c1cn[nH][nH]1)C1CC(C)CN1C(c1ccc(N2CCOCC2)cc1)=O S(=O)(=O)(c1nc(Cl)c(C#N)s1)N1CCCC(NC(=O)OC(C)(C)C)C1 c1(C(=O)NCCOCCNC(CC2CCCC(C)(C)O2)=O)ccn2nccc2n1 C1(CC)CC(C(=O)NCCNC(=O)C2CC2)CO1.C12CC1C(=O)NC2 Cc1c(C(N2CC3(CCN(C(=O)C(C)Cn4ccnc4)C3)C2)=O)nc2sccn12 Cc1cc(C#N)c(O)nc1C(N1CCCC1CCNC(=O)CN1CC(C)(C)C1)=O c1(C(c2nnnn2CC2CC2)NCC(CC)SCC(F)(F)F)ccn(C(C)(C)C)n1 CCC(C#N)C(=O)NCC(C)N(C(c1ccnn1C1CCC1)=O)CC S(=O)(=O)(c1ccc(C)c(C(=O)NCCNC(=O)CC2CC(OC)C2)c1)NC c1(C(=O)NCC(CNC(C2CCC(O)C2)=O)OC)cnc2c(c1)CCC2 N1(C(C2C(CC)CCC2)=O)CCC(CC2CCN(C(=O)CC3(O)CC3)CC2)CC1 c1(CNC(C(CC)N(CC)CC)=O)cccc(CNC(=O)CC2C=CCC2)c1.SCC C1(NC(C(C)OC)=O)C=CCN(C(c2cccnc2N)=O)C1 c1(C(N2C(CNC(CC(=O)N(C)C)=O)COCC2)=O)c(F)cc(F)cc1Br N1(C(C(CSC)O)=O)CC(CO)C2(CCN(C(=O)CCC(=O)OC(C)(C)C)CC2)C1 C1(NC(c2nc(COC)oc2)=O)CN(C(=O)Cn2nnc(C(C)(C)C)n2)CC1O C1(N(C(c2ccc(C)nn2)C(=O)NCCCSCC)C)(OC)CC(OC)C1OC N1(C(=O)CC)CCCc2ccc(NC3COC4(CCCCCC4)C3)cc21 Cn1cc(C(=O)NCCC2CCCCN2C(C2CNC(=O)C2)=O)c2ccccc12 N1(C(c2n[nH]cc2Br)=O)CCN(C(=O)CN2CC=CC2)C(C2CCCC2)C1 CC(C)C(C(=O)NCC12CC(NC(=O)C(F)CC3CC3)(CO1)C2)n1cncn1 C1(c2nnnn2CC2CCOCC2)(NCCc2onc(CC)n2)CC2CC2C1 N1(C(CCC#CC)=O)CCC(C)CC1C(=O)NC(CCOC)C(C)C C1(CNC(=O)C(O)C2CCCC2)CC(O)(CNC(=O)Cn2cnnc2)C1 c1(N)cccc(Cl)c1.C(CSC)(C(=O)N1CC(NC(C2(NC(N)=O)CC2)=O)C1)OC C1(NC(C(CC=C)C)=O)CC2(C1)CN(C(C1CNC(=O)N1)=O)C2 C1(C(=O)NC2C(NC(=O)CNC(c3cscn3)=O)C2)CC12CC(F)(F)C2 CCCCCC(=O)NCC(N1CCOCC1)=O.C1(CN)CN(CC(=O)N)CCO1 Cn1ncc(Br)c1C(=O)NC1CN(C(=O)Cc2cc(=O)n(-c3ccccc3)[nH]2)C1 C1(C(=O)NC2CCN(CCC)C2)CC(F)(F)CCC1(C)C O(NC(=O)C(C1CC1)NC(=O)C(O)Cn1cncn1)CCC N1(C(c2nc(CCCCC)sc2)=O)C[Si]2(CCCC2)CC1C(=O)NC N1(C(Cn2c(C)nc(C)n2)=O)CCC(CNC(=O)C(CN(C)C)N(C)C)C(C)C1 N1(C(C=CCOC)=O)CC2CCCC1(CNC(C1CCS(=O)(=O)CC1)=O)C2 C1(OC)CCC2(C(N3CCCC3CN(C)C(C3CCC(=O)N3)=O)=O)CC12 c1(NC2C(C)CSC2)ccc(S(=O)(=O)N2CCN(c3ccncc3)CC2)c(Cl)c1 Cn1cc2c(n1)CCN(C(=O)CNC(=O)CCc1cn[nH]c1)C2 CC(C)C(CCNC(C1CC1(C)C)=O)NC(c1cc(=O)n(-c2ccccc2)[nH]1)=O C1(NC(c2c(OC)nsc2OC)=O)CS(=O)(=O)CC1NC(=O)CNS(C)(=O)=O c1(N(CC(C(OCC)OCC)O)CC)cc(S(=O)(=O)N2CCOCC2)ccc1C N1(C(c2c(C)cco2)=O)CCC12CN(C(c1cccc(C)c1F)=O)C2 CN1CC2(CCN(C(c3cccn3Cc3ccccn3)=O)CC2C(=O)O)C1 C(CC(O)CNC(=O)C=CCOCC(F)(F)F)NC(=O)CCN1CCCC1 N1(C(CNC(=O)NC2CC2)=O)CC2CC(NC(C3(n4ccnn4)CC3)=O)C1C2 c1(OCC)cc(C(=O)NC2CCC(C)(CNC(=O)C(C)C)C2)ccn1 C(=O)(C(C(C)C)N(C(=O)C(C)NC(c1ccccc1Cl)C)C)NCC Cc1ccccc1C=CC(=O)NC1CC1CNC(=O)COCC1(F)CC1 CCC(C)N=c1nc2c(cnn2C)c(NCC23CC(C)(CCO2)C3)[nH]1 c1(C(N(CC(C)NC(=O)C(O)CC(C)(C)C)CC)=O)cnc2nnc(O)n2c1 C(=O)(CC(C(F)F)c1ccccc1F)N1C(c2cc(COC)on2)COCC1 C1(CC)CC(C(=O)N(CC)CC2(O)CN(C(=O)CC3(CO)CCCC3)C2)CCO1 c1(C(N2C(CCC)C(=O)NCC2)C(=O)NC2CCC2)c[nH]c2ncccc12 c1(C(=O)NC2C(C)CN(C(=O)CC3CCC(C#N)C3)C2)cccn2nnnc12 C1(C(=O)NC2CC2)CN(C(=O)C(CCc2ccsc2)N2CCCC2)CCO1 C1(C(NOC(C)(C)C)=O)CC2CC1CC2NC(=O)COC(F)F C1(NC(CN(C(=O)OC(C)(C)C)C)=O)CC(F)(C(=O)OC(c2ccccc2)=O)C1 C12(C(=O)NCC3C4CN(C(c5c(OC)nsc5)=O)CC43)CCCC1C2(F)F C1(NC(C2CCOCC2)=O)CCN(C(c2cc(C(F)F)[nH]n2)=O)CCC1CO CC1(OCC(N2CCC(NC(=O)C(F)CC3CCOC3)C2C)=O)CCOCC1 N(C1CCCNc2ccccc21)C(=O)CNC1(n2cnnn2)CCSCC1 C1(C(N(CC#C)CC)=O)CCCN1C(C1CCCN1C(=O)CCNC(N)=O)=O Cc1ccc(C(=O)NCC(CC(C)C)NC(C2C(C)OC(C)C2C)=O)c(F)c1F c1(NC2C(CNC(C3(OC)CCSC3)=O)CCCC2)ncnc(Cl)c1C(C)=O C(c1ccc(C)c(C)c1)=CC(=O)NCC1C2N(C(C(C)SCC)=O)C(CC2)C1 n1(C(C)C)cnnc1C1CC1.c12coc(n1)CN(C)CCN(C)C2=O c1(C(=O)NCC(C)(C)NC(C(C)n2cccn2)=O)ccc(N2CCC(C)C2)cc1 C1(NC(=O)CCC[N+](=O)[O-])CCC2CCN(C(C3CC(=C4CCC4)C3)=O)C1C2 C1(CC)CN(C(=O)Cn2nnnc2C)CCN1C(=O)CC(=O)OC CC1CC2CN(C(=O)C=CC(C)(C)NC(=O)NC3CCN(C)C3C)CC12 C(=O)(C(C)(C)S(C)(=O)=O)NCC(CNC(C(C)(C)Cc1cnn[nH]1)=O)O Cc1cc(CNC(=O)C=CC(C)NC(=O)CCN2CCOC2=O)co1 C12(NC(C(=O)NC(C(=O)NCC)CC)=O)COC(COC)(C1)C2 N1(CC)CCC(C(=O)NC(COC)C(N2CC(C)(C)C2CSC)=O)CC1 CC1CN(C(c2nnsc2C(F)F)=O)CCC1N(C(=O)CC1(C)CC1)C C1(CNC(c2cnc(OC)s2)=O)CC12CCN(C(=O)CC1CC(C(F)F)C1)CC2 N1(C(c2cn(CCCC)nn2)=O)CCN(C(=O)CC(C)(C)O)C(CCO)C1 c1(C(N(C)CC2N(C(CSCC#C)=O)CCC2)=O)ccc(N)cc1O c1(CC)cccc(OCC(=O)NCC(F)CNC(c2cc(O)n(C)n2)=O)c1 Cc1cnc2cccc(C(=O)N(CCC(C(C)C)NC(C3CS(=O)(=O)C3)=O)C)n12 C1(CC)CN(C(=O)CC2CCCCN2C)CCN1C(=O)CN1CCC(O)CC1 CC1CCC(C(=O)CCC(=O)N2CCCC(C(N3CC=CC3CO)=O)C2)CC1 CCCCCC(O)C(=O)NCC1(C(F)(F)F)Cc2ccccc2C1 C(=O)(C(C)c1ccsc1)N(C)CC1(NC(C2(SC)CC2)=O)CC1 C1(CCC(=O)N2CCCC2)CCC(=O)N1.C12CCN(C1)C(=O)C2.CC(C)NC c1(C(=O)NCC2(C)N(C(C(CC=C)C)=O)CCC2)ccc2nc(C)ccc2c1 c1(C(N(C)CCN(C)C(C2CCCC3(CC3)C2)=O)=O)cc2c(o1)CCCNC2=O C1(C#N)(OC)CC(C(=O)NCC(O)CCNC(=O)Cn2ccc(Br)n2)C1 C12(C(=O)NC(CC=C)C(=O)OCC)CCC(C(N3CC(O)(CC)C3)=O)(CC1)C2 c1(C(=O)NC2CCCC(N(C(c3ccc(CC)o3)=O)C)C2)cc(N)c(Cl)c(O)n1 C1(C(N2CCC3CN(C(c4[nH]cc(C)c4)=O)CC32)=O)Cc2ccc(F)cc2C1 c1(C(N(CCC(=O)NC(C)CC2CCC2)CC=C)=O)coc(COC)n1 N1(C(C(C)OC(C)=O)=O)CCC(NC(c2cc(O)nc(O)n2)=O)CC(C)(C)C1 C(=O)(C1CCc2cccc(F)c21)N(CCNC(C=Cc1scc(C)n1)=O)C(C)C c1(OC)ccc(-c2ncnn2CC2COCCO2)cc1Cc1cccc(Cl)n1 c1(C(=O)NCc2nocc2C(=O)NC(C)(C)CSC)cc(OC)c(C2CC2)nn1 C12CSCN1C(=O)C1(CC1)NC2=O.c1(CN(C(=O)C(C)(F)F)C)ccccc1 c1(OCC(N2CCC(CNC(C(C)c3ccco3)=O)C2)=O)ccc(F)cc1Cl Cc1cc(C(N2CC3CC(C(N4CC5C(C4)C5(C)C)=O)(C3)C2)=O)nc(C)n1 c1(NCC(CNC(CC(n2ccc(C)n2)C)=O)O)nc(Cl)nc2sccc12 N1(C(Cc2c(CC)cccc2)=O)CCC2(CC1)CN(c1nccc(C)n1)CCO2 c1(OC)cc(NCC2CCCCC2Oc2ccccc2F)ccc1S(N)(=O)=O n1(-c2ccccc2)nc(C2CCCCO2)nc1-c1sccc1Cl Cc1nc(C(=O)NC(C)(CO)C(=O)NCC2CCCC23CC3)sc1C c1(C(=O)NC2CC3(CC(NC(c4ccc(C)cc4O)=O)C3)C2)c(Cl)cc(Br)cc1Cl c1(CNC2C(C(=O)Nc3cccc(CC)c3)C2)cccc(OC)c1Br C1(CCNC(c2c(C)c[nH]c2)=O)CCCCN1C(c1cc(O)nn1C)=O Cc1cc(N)ccc1C(=O)NCC(C)NC(c1ccc(-c2ccccc2)[nH]1)=O c1(CC)ccc(C(=O)N(CCCNC(C2C3CS(=O)(=O)CC23)=O)CCO)c(C)c1 C1(NC(c2cnnc(C)c2C)=O)COC2(C1)CN(C(C1CCC3CCC13)=O)C2 N1(C(CCCOC)=O)CCc2ccc(C(N3CC(C)N(CC)CC3C)=O)nc2C1 C(=O)(CC(F)(F)C(C)C)NC1CCN(C(CC=CC)=O)C1C(C)C C1(C(C)C)CN(C(c2cc[nH]c2)=O)CCN1C(C1SCCCS1)=O C(=O)(C1=NN(CCO)C(=O)CC1)NCC1CC(NC(C(N(C)C)C2CC2)=O)C1 C1(CC(=O)NC(CNC(c2ccn(CC(C)C)n2)=O)(C)CO)CC2CCC1O2 c1(CC)cccc(CNC(=O)CCc2cn(CC)nn2)c1.C1(C=O)COCC1CC C12(C(=O)NC(C)(C)C)CCCC1(C(N)=O)C2.C1(=O)C(=O)N(CC(C)O)CCN1 c1(CN(C(=O)COC2(C)CCOC2)C(C)C)ccccc1 c1(C(N2CCC(NC(C3N(N=O)CCC3)=O)(CO)C2)=O)ccc(CO)c(F)c1 c1(C(=O)NC(CC)(CNC(c2ccc(Cl)c(N)c2)=O)CC)nnn2c1CCCC2 Cc1nsc(NC2CN(C(=O)CN3CCN(C)CC3)C(C)(C)C2)c1C#N Cc1cc(OCC(=O)N(CC(C)N(C)C(C2CC(C)(F)C2)=O)C)ccc1Cl C1(CC=C)(NC(=O)Cc2cc(COC)no2)CCN(C(C2C=C2C)=O)CC1 C1(C2CCCCC2)(C(=O)NCC2CN(C(CCSCC(N)=O)=O)CC2O)CC1 Cc1cn2cc(C(N3CCCC(NC(C4CCN4S(C)(=O)=O)=O)C3)=O)nc2s1 Cc1[nH]ccc(=NC(=O)C2CCC(NC(=O)C(C)Cc3ccco3)CC2)c1C N1(CC(=O)NCC(C)(C2CC2)OC)CCN(C(C2(CO)CCCO2)=O)CC1 N1(C(CC=CC=C)=O)CCN(C(c2cnc(C)cc2C)=O)C(c2cccs2)C1 c1(C(N2CC(N(C)C(C3CC(c4ccccc4)O3)=O)C2)=O)c(Cl)cccc1Cl C1(C(N2CC(NC(C3(CC)CCOCC3)=O)C(O)C2)=O)CC2(CCC2)CO1 c1(C(=O)OCC)cc(C)nnc1NC1CN(C(=O)CN2CCS(=O)(=O)CC2)C1 c1(NC(C2(CC(C)C)CC2)=O)cn(C)nc1C(N)=O CC1(F)CCC(C(=O)NC2(C)CC(NC(=O)C(C)(C)c3cc[nH]n3)C2)CC1 N1(C(C(CCC)NC(N)=O)=O)C2CCC1(CNC(=O)C(F)C(C)C)CC2 c1(C(=O)NC(CC(C)NC(=O)CC2CCC(O)C2)C)cnc2c(c1)COCC2 C1(CC)CN(C(=O)Cc2ncoc2C)CCC1NC(=O)C(C)(C)c1nccs1 c1(C(=O)NCC(CO)NC(C(CC#C)C2CC2)=O)c(C)[nH]c2ccc(F)cc12 N1(Cc2c(OC)c(Cl)ccc2)CC2CCC1CN2C(c1nc(Br)cs1)=O c1(C(N(CCNC(=O)NC(c2cccc(C)c2F)=O)C)=O)cccc2sncc12 C1(C)(NC(c2c(C)nccc2)=O)CCCN(C(=O)CSC2CCOC2=O)C1 c1(C(N(C)CC2CCCN2C(=O)CCC#N)=O)ccc(S(=O)(=O)NCC(N)=O)o1 C1(NC(=O)CC2CCCCN2C(=O)CN2CC=CC2)CCCCCC1F C1(C(N2CCC(N(C(c3ccc(SC(F)(F)F)o3)=O)CC)C2)=O)NC(=O)OC1(C)C c1(OC)cc(O)ccc1Cl.c12ccccc1-c1nc(cs1)CC(=O)N2 C(CCCCNC(=O)CCCc1ccc(C)s1)N(C(C(C)SCC)=O)CC c12ccc(c(F)c1)C(=O)NC1C3CCN(C31)C(=O)C(C)S(=O)(=O)C2.C1(CO)CC1 C1(CC)CN(C(=O)CC(C)(C)SC)CC1NC(c1cnn(CCCOC)c1)=O N1(C(c2cc3cnccc3[nH]2)=O)CCN(C(c2ccc(F)cc2)=O)C2CCCC12 c1(OC)cc(C(=O)NC2CC(O)(CNC(C3CCCOC3)=O)C2)c(C)cc1O c1(C(=O)NCC(CO)NC(Cc2nc(SC)sc2)=O)cc2c(=O)[nH]ccn2n1 c1(SC(C(=O)NCC(CC)NC(c2nocc2Br)=O)C)ccccn1 CCCCC(C(=O)N1CCOC(C(=O)NCC(=O)OCC2CC2)CC1)C(C)C C1C(CC(F)(F)F)NC(=O)C(=O)N1.C1(C)(C(N(CCN=[N+]=[N-])C)=O)CCC(=O)C1 C(=O)(CC(C)CC(F)(F)F)N1CCCC(CC=C)(NC(=O)CS(=O)(=O)NC)C1 CCCCCC(CCCCC)C(=O)NC1CN(C(=O)Cc2cc(C)cs2)C1 C1(NC(c2scc(OC)c2)=O)CCCCC1CNC(c1c(C)cnn1C(C)C)=O C(=O)(C(C)C(C)O)NCCOCCN(C(c1cc(CCC)on1)=O)C N1(C(COC)C)CCN(C(C23CC2CCN3C(c2ccc(CO)nc2)=O)=O)CC1 CCC(CC(=O)N1CCC1C1CCCC1)NC(c1ccn(C)c1C)=O C(=O)(C1=NOC(C)(C)C1)N1C(CNC(c2c(C)nc(N)cn2)=O)CCC1 c1(CC)cc(C(N2CCC(NC(=O)CCC3CCCCN3C)C2C)=O)cc(O)n1 c1(C(=O)NCCC(CNC(=O)C2=CCSC2)O)nccc2c(Cl)cccc12 c1(CNC2CCCC(CO)C2)coc2ccccc12 C1(C)(CNC(C(C2CCOCC2)OC)=O)CCCN1C(c1cccc(C2CC2)c1)=O C=CC(C)CN=C(NCC1CCC1)NC1CCOC(C2CC2)C1 Cc1cn(C2CCOCC2)nc1C(N1CC(O)(CCNC(C2(O)COC2)=O)C1)=O c1(CN2C(C(=O)NCC(c3ccccc3)O)CC3CC32)c(O)cc(Br)cc1F c1(CN(C(CC=CC=C)=O)C)cnn2c1CN(C(=O)CC1CCS(=O)(=O)C1)CC2 C1(CNC(C(C(=C)Cl)(C)C)=O)CN(C(=O)C(C)NC(=O)CC)C2(CCOCC2)C1 c1(C(=O)NCC(=O)NCC2N(C(CC(C)SC)=O)CC2)ccc(C(N)=O)cn1 Cc1cc(F)sc1C(N1CC(O)CC1CC(=O)NCCC1CCCCC1O)=O CCC(CC)C(C(=O)NC(CCOC)C(=O)N1CCC(CCCO)C1)OC C1(C#N)(C(N2CC(CC(C)NC(CCN(C(C)=O)C)=O)C2)=O)CC2CCC1C2 C12(C(=O)NC(C(CO)NC(c3c(C)cccn3)=O)C)CC(C)(C1)OC2C C(=O)(C(F)C(F)(F)F)N(C1CN(C(c2cc(COC)sc2)=O)C1)C Cc1cnsc1C(=O)NCC1(O)CC(C(=O)N(CC(F)F)CC(C)O)C1 N1(C(c2cnc(C)s2)=O)CC2CC1CN2C(C1(S(C)(=O)=O)CC1)=O C1(CNC(c2ccn(CC)n2)=O)CN(C(C2CC(OC(F)F)C2)=O)CCO1 c1(C(=O)Nc2cccc(C3CCCCC3)c2)cc(Cl)c2ncccc2c1F C1(C(=O)NC)CCCC1NC(=O)NC(c1ccnn1C)C C(CCC(C)CC(=O)N(C(CNC(C1C=CC=CC=C1)=O)C1CC1)C)=C(C)C C(=O)(C(C)(C)N(C(=O)CNC=O)C)NCCOCCN(CC(C)(C)C)C C(C(O)C(=O)NC(Cc1cc[nH]n1)C(=O)NCC1CCCCO1)=CC c1(C(=O)NCC(CC=C)NC(=O)C(C)=CC)ccc(Br)c(CC)c1 C1(NC(c2c(OC)n[nH]c2)=O)CCN(C(=O)Cn2nc(C)cc2C(F)F)C(C)C1 N1(C(c2cc(C#C)c(C)cc2)=O)C2CCC1CN(C(=O)CCc1ccsc1)CC2 C(=O)(CCCCCCCNC(=O)OC(C)(C)C)N1CCC(OCC)C(C)(CC)C1 C1(CCC)CN(C(=O)C=C2CCC2)CC1NC(=O)C(C1CCC1)OC C1(C(=O)NC2CC(C=C)C2)CCCCC1(C)N c1(C(=O)NCC2(NC(C(C)n3ccnn3)=O)CCOCC2)cc2[nH]ccc2s1 c1(SC(C)(C)C)ccc(N)cc1O.N12CCC(C1)C2=O.C1CO1 c1(CNC(=O)CCOCC2CC2)ccc(C(=O)NC(C2CCSC2)(C)C)cc1 C(CC(=O)NCc1nccnc1C)(C(F)(F)F)NC(C(CCC)O)=O C1(C(=O)NC(CN(C(c2cc(C(F)F)on2)=O)CC)C)CN(CC)CCO1 C1(C(=O)NC2(CC(=O)O)CCCOC2)CC2CCC1CC2 Nc1cc(F)c(C(=O)NCC2CCCN(C(C3CC34CCC4)=O)C2)cc1Cl c1(N2C(C)CC(CNC(c3ccc(OC)cc3)=O)C2)ncc2ccnc-2[nH]1 CC(C)C(C)CCNC(=O)CC1CC(C)N(C(=O)CSC(C)(C)C)C1 C=C(Cl)C(C)(C)C(=O)N1CCN(C(c2cc(O)n(CC)n2)=O)C(CC)C1 c1(N2CCC(CNC(C3ON=C(C)C3)=O)C(C)C2)ncnc2scc(C)c12 N1(C(C(=O)N(CC(c2ccccc2)O)C)=O)CCCC2(CCC2O)C1 C1(C(N2CC(CNC(c3c(CC)scn3)=O)C(O)C2)=O)(CO)CCCCCC1 C=CCCC(C(=O)NC1CCCC1CN(C)C)NC(c1cncc(NC)c1)=O C1(CNC(Cc2cccc(C)c2)=O)CCCN(C(c2csc(=N)[nH]2)=O)CC1 C1(CNC(c2cnc(C)[nH]2)=O)CC(NC(=O)CC2(C)CC2)C1(C)C O=C1NCC2(CCCN(C(=O)NC3CCc4ccc(F)cc4O3)CC2)O1 Cc1cc(Cl)c(C(=O)NC2C3CN(C(C4CCCC(=O)N4C)=O)CC23)cc1N c1(C(=O)NC2CCN(C(CCCCOC)=O)C(C)C2)cc(C)sc1S(N)(=O)=O N1(C(C(C(=O)OCC)C)=O)CCC(C(=O)NCCOCC(=O)NC)(CC)CC1 N1(CC(N2C(CC(N3CCC(N(C)CC)C3)=O)CCC2)=O)CCCCC1C c1(CC(C(=O)N(CCn2cc(C3CCCCC3)nn2)C2CC2)O)ccccc1Cl N1(C(c2ccnc(F)c2OC)C(=O)NC(C(=O)OC)C)CCC2CN(C)CC2C1 C1(NC(CC=C(C)C)=O)CC2CCCC(C1)N2C(c1cnc[nH]1)=O C1(N(CC(=O)NCC(C2CC2)NC(C)=O)C(C(=O)NC)=O)CCOC1.C=C(C)COCC c1(C(N2CCC(C(C)(C)NC(c3ccc(C(C)C)o3)=O)C2)=O)nccc(Cl)c1F Cn1nccc1C(F)=CC(=O)NC1(CNC(C2(C(C)(F)F)CC2)=O)CC1 C#CC1(C(N2CC(O)(CC(C)C)C2)=O)CCN(C(=O)CC(CC)C2CC2)CC1 c1(-c2cc(C(=O)NCC(O)CNC(=O)C(O)CF)sn2)ccc(F)cc1 c1(C(=O)NCCCOCCNC(CC2CC(C)OC2C)=O)occ2c1CCCC2 n1(CC)cnc(C(=O)NCC(C2CC2)N(C)C(C2CCCC2OC)=O)n1 c1(CC(=O)NCC(C)NC(=O)CCC2CC2(Cl)Cl)ccc(O)nc1 n1(Cc2c(OCC=C)cccc2)cc(C#CCN2CCCC(C)C2C)nn1 N1(C(c2c(CC)scc2)=O)CC(NC(C2(CC)CCCO2)=O)CC(O)C1 c1(C(N2CCC(Cn3cc(C(CC)(O)CC)nn3)C2)=O)nccn2ccnc12 c1(C(=O)NCc2c(C(N3CCC(C(=O)OC)CC3)=O)cccc2)ccc(O)c(F)c1 c1(OC(C)C#N)cc(F)ccc1C(=O)NS(=O)(=O)Cc1ccccc1 C(=O)(CC1=CCCC1)N1CCC(N(C(C(C)NC(C)=O)=O)C)CC1 C12(C(=O)NCC3CC(C)N(C(=O)COC(F)(F)F)C3)CCC(C)(CC1)OC2(C)C C12(C(=O)NCc3c(C(=O)NCCCC=CC)con3)CCC(CC1)CO2 c1(-c2c(OC)cc(O)cc2)ccn2nc(C(=O)Nc3ccc(SC)cc3)cc2c1 CC(C)C(C(=O)NC1CCC(NC(=O)CCN2C(=O)CCC2=O)C1)NC(N)=O c1(C(=O)OC(C)(C)C)ccc(NC2CCS(=O)(=O)C2)c(Br)c1 N1(C(C(N2CCCCC2=O)C)=O)CCCC(CNC(C2(C)C=CCS2)=O)C1 C1(C(N(CC(=O)N(C(C)CCO)C)C)=O)CC2CCC2C1 CC(C)(C)CCCCC(=O)NCC1(F)CCN(C(C2CC(C#N)C2)=O)C1 C1(C(N2CCN(CCCNC(CCCN=[N+]=[N-])=O)CC2)=O)CCN2CCOCC12 N1(C(CNC(C2CCCCO2)=O)=O)CC2C(c3ccc(F)cc3)(C1)CS2=O N12CC3(CCC1CC3)C2=O.N1(C(C2(n3cccn3)CC2)=O)CC(O)C(C2CC2)C1 c1(OC)ccccc1C(C(=O)NCc1ccco1)N(C(C)C(CC)CC)C C(C(C)C(C)(C)C)(c1n(CCSC)nnn1)NCc1ccc(C)c(CO)c1 c1(OCCCOC)ccc(CN2CCCCC2C(=O)O)cc1 c1(CC)ccc(NC(C2CC2C(N2CCC=C(F)C2)=O)=O)cc1[N+](=O)[O-] C1(NC(COCCC)=O)CC2CCC1N2C(C1(F)CCCOC1)=O c1(C(N)=O)ccc(C(=O)NC23CC(CNC(C4CC4(Cl)Cl)=O)(C2)C3)o1 C1(C(N(CC(C)C)Cc2c(C)non2)=O)C2CC1(c1cccc(F)c1)CO2 C(=O)(C(CC(F)F)N(C)C(c1cccc(C2CC2)c1)=O)N(CC(C)C(C)(C)C)C C(=O)(CCC(C)OC)NCC(C1CCC1)NC(CNC(CC)=O)=O N=c1[nH]n(CC(N2CCC(N(C(=O)C#CC3CC3)CCO)C2)=O)cc1Br c1(C(=O)NC(C(=O)N(CC(COC)C)C)Cc2cnc[nH]2)ccc(=O)n(C)n1 C(=O)(CCCCC(=O)NC)NC(C(C)NC(CC=C)=O)CO C12(CNC(C(CCOC)OC)=O)CCCCC1N(C(=O)CC1CCCC1)CC2 c1(CC)cc(OC)ccc1C(=O)NCCCNC(c1cnc(OC)s1)=O N1(C(COCC(C)C)=O)CCCC1C(C)NC(=O)CC1C=CCC1 C=C(C)c1cnccc1C(c1nn(C)cc1OC)NC(c1nnnn1CCC)C C1(C2CCCN(C(c3ccc(N)c(C)c3C)=O)C2)(NC(c2cnc(C)[nH]2)=O)CC1 c1(OC)cc(C(=O)NC(C)CCNC(=O)C(F)=C2CCC2)c(Br)cc1C N1(C(CCNC(C2C(C)C2)=O)=O)CCCC(O)(CCNC(=O)C=CC2CCC2)C1 c1(C(N2CC(CNC(c3coc(Cl)c3)=O)C3(C2)CC3)=O)cnn2c(Cl)cccc12 C(=O)CCCC(=O)N1CCC(C(=O)NCc2scnc2C)C1C(C)C CC1CC(NC(C2COCCN2C(c2cc(C(N)=O)co2)=O)=O)C(=O)O1 C1(C(=O)NC2(CCOC)CCN(C(c3n(C)cnc3)=O)C2)CCC(=C(F)F)CC1 C1(C(N2CC(N3CC(C)OC(C)(C)C3)C2)=O)Cc2c(O)cccc2N1CC.C(C)(C)(C)O CCCCC(C(=O)NC1COCCC1C(N1CCC2(CCC2)CC1)=O)C(C)C C(=O)(C(C(=O)OC)OCC)N(CC)CC.C(CCCS)NC(C1CCCC1)=O N1(C(c2ccc(C)c(F)c2)=O)CC2C=CC1C(C(=O)NC1C=CCCCC1)C2 C(=O)(C1=CC(O)C(NC(=O)CC2CCSC2)C1)N1CC(C)C(C)(CO)C1 C1(NC(C2CC3(CC3)C2)=O)CN(c2nc3cccc(F)c3s2)C2CCCCC12 N1(C(=O)Cn2cnnn2)CCCCC(C2CN(C(C3CCCSS3)=O)C2)C1 c1(C(CC(CC(=O)OC(C)=O)C)C2CC2)[nH]c2ccccc2c1C C1(NC(c2cc(OC)nn2C)=O)CC(F)(F)CC1NC(=O)Cc1cccc(Cl)c1 c1(CC(=O)NCC(CC)NC(c2ccsc2C)=O)c(C)ncnc1C N1(C(c2cc(C)ncn2)=O)C2CCC(C2)C1C(=O)NCC1(F)CC1C c1(C(C(=O)NCC(CC)NC(=O)C(CC)n2ccnc2)C)c(C)noc1C C1(C(=O)NC2CC(C)(C(=O)OC)C2)C2CCN(C(c3cnncc3C)=O)CC12 N1(CC(=O)NCc2ccnc(C(=O)NCCNC(N)=O)c2)CCCNC1=O C1(C)(C(=O)NCCC2N(C(C3(C)COC3)=O)CCOC2)CCCNS1(=O)=O c1(OC)ccc2c(c1)C(C(C)C)N(C(C1CC3CCCC3C1)=O)CC2 c1(C(C)Nc2c(C)c(NCCC(F)F)ncn2)ccc2c(c1)CCCC2 c1(C(=O)OCC)c[nH]c(=NCCNC(C2CC(N=[N+]=[N-])C2)=O)nc1C Cc1ccc(Cl)c(F)c1C(=O)NC1CCN(C(C2CCC(O)C2)=O)CC1F c1(C(=O)NCC2(O)CC(NC(C3COCCOC3)=O)C2)cc(F)c(F)cc1F C1(CC#C)(C(=O)NCCC2CN(C(C3CC3c3cnc[nH]3)=O)C2)CCOC1 C=CC(C(F)(F)F)NC(=O)C=CC1CCCN1C(c1oc(C)nc1CC)=O n1(CC(=O)N(C2CCN(C(c3nocc3C)=O)C2)CC)cc(Br)cn1 c1(C(=O)NCC2C(NC(c3ccc(CCC)[nH]3)=O)C2)cnn(CC)c1C C1(C(=O)NCC(c2cncnc2)C)CC2CCC(C1)N2C(=O)Cc1cnsc1 C1(CC)(NC(=O)CCc2cn(C)nc2C)CCCN(C(=O)C(C)CN(C)C)C1 c1(-c2cnc(OC)c(C)c2)cccc2c(C(=O)Nc3ccc(C#N)nc3)[nH]nc12 N1(C(C2N(C=O)CCOC2)=O)CCCN(C(=O)CCSC(F)(F)F)CC1CO CC1(C(=O)NC2C(CNC(c3cc(Cl)c[nH]3)=O)C2)CCC(F)(F)CC1 c1(CC(=O)NC2CC(NC(C(C)(C)n3cnnn3)=O)CC2O)c[nH]c(=N)nc1O c1(CC)cc(CC(N2CCCC2CN(C(=O)C(C)=C2CC2)C)=O)n(C)n1 c1(C(N2CC(N(C(CC(C)OC)=O)C)C3(C2)CC3)=O)[nH]c2ccccc2c1C#N n1(CC)c(O)nc2ccc(C(=O)NC(c3cccc(C#N)n3)C)cc12 C1(CC(=O)N(CC=C)CCOC)CCC(NC(=O)Cn2cc(C)cn2)C1 C(=O)(C(CC)CC(C)C)NCC1CC(C)(C(=O)NC2(C(=O)OC)CCCCC2)C1 C(C(C)NC(c1cnc(C2CC2)[nH]1)=O)(C(C)C)NC(c1cnc(SC)s1)=O N1(C(c2nc(NC(=O)CCc3ncc[nH]3)sc2)=O)CCC2(CC1)CC(CO)C2 C(=O)(CCCCC(C)(C)C)N1CC(C)N(C(=O)C=CC(N2CCOCC2)=O)CC1 c1(CC)c(C(N2CC(CNC(=O)CSC(C)(C)C)CC2C)=O)oc2ccccc12 C1(NC(Cn2cc(C(C)=O)nn2)=O)CC(F)CN(C(=O)Cn2nccn2)C1 C1(NC(c2ccc(C#C)o2)=O)CC2CC1CN2C(=O)C(C)=C(C)CC c1(OC)cc(Cl)c(C(N2CC(NC(=O)CC3CCCCCO3)C(C)C2)=O)cc1Cl N1(C(Cn2c(C)cc(C)n2)=O)CCC(CO)(NC(c2cc(C#N)[nH]c2C)=O)CC1 c1(CNS(CSCC(=O)N(C(C)(C)C)C)(=O)=O)ccc(S(N)(=O)=O)cc1[N+](=O)[O-] N1(C(CCCC(C)(C)C)=O)CCCC(C2CC2NC(C2CC23CCSCC3)=O)C1 C1(C(N(CCCC(=O)NCCCOC=C)C)=O)CCC(C)(C)C1 C1(N(C)C(c2ccnc(S)c2)=O)CCCC(CNC(=O)CCc2cncs2)C1 N1(C2CCCN(C(COC(CC)C)=O)C2)CCN(C(=O)C(Br)=C(C)C)CC1=O N1(C(C=CCN(C)C)=O)CCCC2(C1)CN(C(C1(C)CC=CCO1)=O)CCO2 O=S(=O)(c1ccc(NCc2cncc(Br)c2)c(Cl)c1)N1C2CCCC1CC(O)C2 c1(NC2C(CCCC)CCC2)nc2c(c(=NCCS(=O)(=O)CC3CC3)[nH]1)CCC2 c1(CC)cscc1C(N1CCC(n2cc(C3CCOC3)nn2)C1)=O N1(CC(=O)NCC2CC(NC(C(C)CC3CCC3)=O)CC2O)C(=O)CN(C)C1=O c1(C(=O)NCC2C(NC(=O)C3=NOCC3)CC2)ccc2c(c1)C(=O)NCC2 CCC(CC(=O)NCC1C2CCC(C2)N1C(c1cc2c[nH]cnc-2n1)=O)C(F)F Cc1nc(C(=O)NCCCCCCn2cc(CNC=O)nn2)sc1C N1(CCOC)CC(C(=O)NC2CN(C(c3cnns3)=O)CC2SC)CCC1=O N1(C(CSC(C)(C)C)=O)CCN(C(S(=O)(=O)c2cccs2)=O)C(c2cn[nH]c2)C1 C1(N(C(C2C(CC)CCCN2C(=O)CC2CCCC2)=O)C)CCCC(C)(C)C1 C1(NC(C(c2cscn2)N(C)C)=O)CCC(NC(=O)C(c2ccccc2)F)C1 Cc1nscc1C=CC(=O)NCC(CO)NC(=O)C(C)(c1ccccc1)N(C)C c1(C(C(=O)NC(C)(C)C)N(C2CCN(CC)C2)CC)ccc(Cl)c(C)c1Cl C(C(C(C)C(C)C)NC(=O)C1=C(C)CCC1)NC(CC(=C)C)=O C1(CNC(c2ncccc2F)=O)CCCC(NC(c2ccnn2CC2CC2)=O)C1 N1(CC)N=C(C(=O)N2CCC(NC(c3csc(COC)c3)=O)C23CC3)CCC1=O CN1CCN(C(=O)NCc2nc(C(F)F)nn2C)c2ccccc2C1 C1(CNC(c2nc(Cl)c(Cl)s2)=O)CC2(C1)CN(C(C1CCC1)=O)C2 C=C=C(C)CC(=O)NCC1CCCN1C(C1CC2(CCC2)C1)=O Cn1nc(O)cc1C(=O)NCC1(O)CN(C(=O)Cc2cccs2)C1 N1(C(C2CCC(N(C)C)CC2)=O)CCOCC(NC(C2CCO2)=O)C1 c1(C(=O)NC2CCC(N(C(c3c(CC)ocn3)=O)C)C2)sc(C(F)(F)F)nc1C C1(NC(=O)CC2C=CCC2)CC(NC(c2cc(-c3ccccc3)no2)=O)CC1O C1(C(=O)NC(CNC(=O)CCCF)C2CCC2)CCn2nnnc2C1 C1(NC(CCC=C)=O)CCC2CN(C(C3CC(CC)=NO3)=O)CCC2C1 C1(NC(CN(C(C)C)C)=O)CCN(C(C2CCOC(=O)N2)=O)C1C1CC1 N1(C(C(C(C)(F)F)F)=O)CCC2C(CCCN2C(=O)CCCc2cccnc2)C1 c1(C(=O)NCC(C)CNC(=O)C(c2cnc(O)nc2O)(F)F)sc(C#N)cc1Cl C=C(C)CC(C(=O)NC(C)CN=[N+]=[N-])NC(=O)CCn1cccn1 CCCCCC(O)C(=O)N1CC2CC1CN2C(C1CC(O)C1)=O C12(C(=O)OC)CC1CN(C(=O)C(Cc1cc[nH]c1)NC(=O)C(OC)OC)C2 CC(F)(F)C(F)C(=O)NC(C(N)=O)C1CC1.C12(CC13CCC3)C(=O)NC2 N1(C(=O)OC(C)C)CCN(C(=O)C=Cc2ccoc2)C(C)C1 N1(C(c2ccc(CC)o2)=O)CCCC1C1CCCCN1C(=O)CC(C)C c1(C(N2C(C(C)NC(C3(C=C)CCC3)=O)CCC2)=O)n[nH]c2ccccc12 N1(C(C2C(C=CC)CN(C(=O)C(C)(C)C(N)=O)C2)=O)CC2(COC(C)(C)C2)C1 Cc1cccc(C(C)C(=O)N(C2CCCN(C(=O)C=Cc3cocn3)C2)C)c1 N1(C(C2N(C(C(C)NC=O)=O)CCOCC2)=O)CCC(F)(F)C(O)C1 C1(CNCCC2(O)CN(C(c3cnc(OC)s3)=O)C2)CCc2nc(C)[nH]c2C1 N(C1COc2ccc(Cl)cc21)c1nc(-c2n3ccc(C)cc3nc2)on1 C(=O)(N=c1cc2ccccn2[nH]1)C1(C2N(C(C(C(C)(C)C)O)=O)CCC2)CC1 C12(NC(C(c3c(C)nn(C)c3)C)=O)CCCC1CN(C(=O)CC1OCCCO1)C2 C(=O)(CCC(F)(F)Cn1cc(C(C)(O)CC)nn1)NC1C(SCC)CCCC1 CCN=c1[nH]cc(C(=O)NCC(C)NC(c2ccccc2N(CC)CC)=O)s1 C1(C)(C(=O)NCC(CCNC(C2CC(C)(O)C2)=O)OC)CCC(=O)NC1 c1(OC)ccc(F)cc1C(N1CCC12CN(C(=O)C=C(C)C)C2)=O C(C)(CNC(=O)CC1CCOC1C)(CNC(c1cc(C(C)(C)C)on1)=O)OC c1(OC)cc(C(=O)NCC2(F)CC(NC(C3CC34CCSCC4)=O)C2)c(F)cn1 c1(C(=O)NC(CC#C)(C)C(=O)N2CCN(C(=O)NC)CC2)ccn2cncc2c1 c1(C(=O)NCC(=O)NC2(CCO)CCC2)ccc2c(c1)CNC2=O c1(CNC2CN(C(c3cccc(O)c3)=O)CC2F)ccc(Br)c(Cl)c1 N#Cc1cc(Br)cnc1NCC1(O)CN(C(=O)C=CC2CCCO2)C1 c1(CCC)noc(CCCC(=O)NC(C)C(C)(C)NC(C2CC2CC)=O)n1 C(=O)(C1=CC2(CCOC2)C1)N(C)CC1CCN(C(=O)C(C)(C)n2ccc(Br)n2)C1 c12ccc(nc1)[nH]c2=O.CCC(C(=O)Nc1nc(C(=O)NC2CC2)cs1)SC CCCC(CNCC(=O)Nc1cc(C)cc(Br)c1)C(=O)Nc1ccccc1 C(CCCCC(F)(F)F)N(C(C1CCOCC1)C(C)C)C CC1ON=C(C(=O)NC2COCCC2NC(c2cccnc2S)=O)C1C C1(OC)Cc2ccccc2C1N(C)C(=O)C(C)Cc1c(C)n[nH]c1C Cc1ccc(F)cc1N(C)C(C1CC(CNC(c2cccc(C)c2O)=O)C1)=O c1(CN=C(NCc2ccc(NC)cc2)NC2CCC2)ccc(C)cc1O C=CCC(CC(C)C)C(=O)N1CCCC1(C)CNC(=O)CNC(C)=O C1(NC(=O)CSCC(N2CCCC2)=O)COCCC1NC(c1ccco1)=O N1(C(CSCC=C)=O)CCN(C(=O)CNC(=O)COC)CC1COC N1(C(COCC)=O)CCCN(C(=O)CCc2ccccc2C(F)(F)F)CCC1 C1(C(=O)NC2CCN(C(CC3C(C)(C)C3(C)C)=O)CC2F)CCN2CCOCC12 Cc1nc(O)nc(C)c1CC(N1CC(NC(c2ccc(F)s2)=O)C2CC12)=O C1(C(N(CCC(C)NC(=O)CNS(=O)(=O)N(C)C)C)=O)CCC12CCC2 c1(CC)ccccc1C(N1CCOCC1CCNC(=O)CC1CN(C)C1)=O c1(C(N2C(CC=C)(CO)CCC2)=O)ccc(C)nc1OC c1(C(=O)NCC(CC(=O)NCc2scc(C)c2)C)ncc(F)cc1N c1(CCC(N2CCN(C(C)=O)C(C(=O)O)C2)=O)csc2nc(C)cn12 C1(C)(C(=O)NCC(CN(C(c2c(C(C)C)[nH]cc2)=O)C)C)CS(=O)(=O)C1 N1(C(C2(O)CCN(C(C3(CC)CC3)=O)C2)=O)CCc2ncccc2C1 C1(NC(C(C2CN(C(C3CCC(N(C)C)CC3)=O)C2)OC)=O)CS(=O)(=O)C1(C)C c1(C(=O)NC2C=CCN(C(Cc3cnc(C)s3)=O)C2)ccc2oc(S)nc2c1 Cc1cc(C(=O)NCC2CC3CCC2N3C(=O)CC(C)(C)C2CC2)nc(C)c1 C12(CNC3C(C)N(C(=O)OC(C)(C)C)CC3)CCCC1C2(F)F c1(CNC(C2(CC(=O)NCC(O)CO)CCC2)=O)cc(C(F)(F)F)ccc1O N1(CC(=O)N(C)CCN(C)C(c2ccccn2)=O)CCCCCCC1=O CC(CCC(C)(C)C)NC(=O)CN1CCN(C(C2COCC2(C)C)=O)CC1 CCC(C)C(O)C(C)C(=O)NC(C(=O)NCc1cccc(Cl)c1)C1CCCO1 Cc1nc(Cl)cc(Cl)c1C(N1CCC12CN(Cc1cccc3occc13)C2)=O N1(C(C(C(C)C)OC)=O)CCC2(CCN(C(c3sc(CO)nc3C)=O)CC2)C1 N1(C(C2(C(C)C)N(C(c3c(OC)ccnc3)=O)CCC2)=O)CCn2nccc21 C1(CNC(=O)NC2CC(N(C)CC)C2)CCN(C2CCCCC2)C1 N1(C(c2c(CC)c[nH]c2)=O)CCC(F)(CNC(=O)C(C)CC2CCCC2)C1 CCCCC(O)C(C)C(=O)NC(CCC(=O)Nc1ccccc1F)C(C)C c1(CCC(=O)NCC2(O)CN(C(C3CC3c3cccs3)=O)C2)cccc(O)c1 C=CCC(CNC(c1cnc(O)c(F)c1)=O)C(=O)N(C)CC1CCCC1 CN1CC(NC(=O)CC2C=CC(NC(C3CCC4(CC3)CC4)=O)C2)CC12CCC2 N1(C(=O)Nc2cccc(CO)n2)CCc2nc(-c3cnn(CCF)c3)sc2C1 N1(C(c2c(CNC(COC3(C#C)COC3)=O)ccs2)=O)CCC2(CC1)CC2CO O(C1CCOc2ccc(OC)cc21)C(C1C(C(=O)OC)C=C1)=O n1(CC)nc(C(C)C)cc1C(=O)NCCCC(CO)NC(=O)CC(C)COC c1(C(=O)NC2CCCC(NC(CCSCC)=O)CC2)c(C)nc(O)nc1C CC1(O)CCC(C(N2CCOCC(NC(=O)C=CCn3cncn3)C2)=O)CC1 C1(NC(C(COC)O)=O)CC1C1CCN(C(C2(C#N)CCOCC2)=O)CC1 C(C(=O)NCc1cn(CC(=O)NC2(C(C)C)CC2)nn1)(C(C)C)SCC N1(C(CCCC#CC)=O)CCN(C(c2cc(CO)on2)=O)CC(O)C1 Nc1cnc(Cl)c(C(N2CC3CC(NC(=O)CC4CC5(CCC5)CO4)C2C3)=O)c1 c1(C(=O)NC(CCCC)CNC(=O)CC2CN(C)C2)c(F)cc([N+](=O)[O-])cc1F c1(C(=O)NCC(=O)NCCC(=O)NC(CCC)C(=O)NC)n[nH]c2c1CCC2.OCC C1(C(=O)NC2CCN(C(C=CC=CCCCCC)=O)C2)CS(=O)(=O)C12CCC2 Cc1cc(O)c(C(C)C)cc1C(=O)NCCCC(CO)NC(C12CC(C)(C1)C2)=O C(C)(C(C)C(=O)N(C1CCC(C)(C)C1)C)NC(c1cnc(OC)s1)=O Cc1n[nH]c(=NC(CNC(c2cnoc2)=O)C(C)C(C)C)s1 Cc1ccc(C=CC(N2CC(NC(C3(c4cc[nH]n4)CC3)=O)CC2C)=O)c(C)c1 N1(C(C=CC)=O)CCC(CNC(c2cnnn2C)=O)C(C)C1 c1(OC)ccc(NC(C2C(NC(C34CCCCC3C4)=O)C2(C)C)=O)cc1C c1(C(=O)NCC(C)N(C(=O)C(C)(O)c2ccccc2)C)cn(CCO)nn1 Cc1cccc(CC(=O)NC(CCOCCO)C(=O)NC2C3CCCC23)c1 c1(NC(C23C(CN(C(c4c(C)nsc4)=O)C2)C3)=O)nc(Cl)cnc1Cl c1(C(=O)NCC(C)(O)CNC(c2ccco2)=O)c(F)cc(Br)cc1Br CC1(O)CCC(C(=O)NCC2CN(c3nc(C#N)co3)CCO2)CC1 N1(C(Cc2cc(C)ns2)=O)CC(NC(C2CCCO2)=O)CC2(CCOCC2)C1 N1(C(C2C(OCC)C2)=O)CCC(C)C(CNC(=O)COc2cccc(CC)c2)C1 c1(CCC)nc(=NC2CSCC23CCC3)s[nH]1 c1(OC)ccc(C(=O)NCC23CC(C(=O)O)(CCO2)C3)c(N)c1 C1(CNC(Cc2nc(=N)[nH][nH]2)=O)CN(C(c2ncccc2Cl)=O)CCCO1 C1(C)(c2ccc(OC)c(F)c2)NC(=O)N(Cc2ccc(C)c(OC)c2)C1=O C1(C)(CNC(C(C)CO)=O)CCCN(C(=O)CCc2ccccc2C(F)(F)F)C1 C1(C(=O)NC(CCCC)CNC(C23CC(CC(F)F)(C2)C3)=O)CCC2(CC1)CC2 CCC(N=c1ccnc(NCc2ccc3nc[nH]c3c2)[nH]1)c1ncc[nH]1 c1(C(=O)NCCC(CNC(c2sccc2CO)=O)OC)ccc(C)cn1 C1(CNC(=O)CC(=O)Nc2nccs2)CN(C(c2n[nH]cc2Cl)=O)C2CC12 N1(C(CNC(c2ccco2)=O)=O)CCN(C(=O)COCc2cccs2)C(CO)C1 c1(OC)cc(F)c(F)cc1CNC(c1ccc(CN2CCC(C(N)=O)C2)cc1)=O c1(C(=O)NC2CC3CN(C(C(C(C)C)F)=O)C2C3)cnc2c(c1)CCCO2 N1(C(C2C(C)(C(F)F)C2)=O)CCCCC(CNC(=O)Cc2ccc(O)cc2)C1 C1(C(=O)NCc2cc(C)on2)(CC)CN(C(=O)CCOCC(F)F)C1 c1(CC)nc(=NC(=O)NC(c2cc(OC)c(OC)cc2O)C)[nH]s1 N1(C(CCn2ccc(C)n2)=O)CCC(NC(c2ccnnc2S)=O)C(O)C1 C1(NC(C=CCC(C)NC(CCN(CCC)C)=O)=O)CCC(C)=C(C)C1 CC1CCN(S(=O)(=O)CC(=O)NCC2(CCNC(c3ccc[nH]3)=O)CC2)CC1 N1(C(c2sc(C)c(O)n2)=O)CCCC2CN(C(=O)CNC(C3CCC3)=O)CCC12 S(=O)(=O)(c1cccs1)NCC(=O)NC1CN(C(CN(CCOC)C)=O)C2C1C2 Cc1ncc(Br)c(C(N2CCC(NC(=O)CC3CCCOC3)C2(C)C)=O)n1 c1(OC)cccc2c1C(C(=O)NC1CCCN(C(=O)C=CC3CCC3)CC1)CC2 C1(CCC(=O)NC(c2cncnc2)C)CCN(C(c2nc(Cl)cs2)=O)C1 c1(C(N(CCN(C(COCC(=C)C)=O)C(C)C)C)=O)ccnn1C(CC)CC c1(OCC)ncccc1C(=O)NCC1CC(NC(c2cc(O)n(C)n2)=O)CC1O C=C(C)CCC(=O)N1CCC(NC(c2ccc(-c3nnc(C)o3)cc2)=O)C1C C1(NC(C2(C)CCCCO2)=O)CC2CC(C1)N(C(c1c(F)cccc1F)=O)C2 c1(NCC(C)N(C(CC(n2ccc(C)n2)C)=O)C)c([N+](=O)[O-])c(C)nn1C(C)C CCCC(C)(O)C(=O)N1CCN(C(c2cccc(O)c2Cl)=O)C(C(F)F)C1 Cc1cc(Br)cc(N)c1C(=O)N(CCNC(=O)CC1CC1C)C1CC1 N#Cc1ncn(CC(=O)NC2(CNC(C3C=CCS3)=O)CC2)n1 N1(C(=O)C=CI)CC(C2CCCCN(C(c3cc4ccncc4s3)=O)C2)C1 C(C1CCCN1C(c1ccc(=N)[nH]c1)=O)=CC(=O)NCC1(OC)CCC1 c1(NC(N(CCC(F)(F)F)CC(C)(C)N(C)C)=O)nnc2c(Cl)cccn12 C(=O)(C#CC1CCOC1)NCCC1N(C(c2c(C(C)(C)F)cccc2)=O)CCC1 C=Cn1nccc1C(=O)NCc1cc(C(N2CC(c3nncs3)C2)=O)ccn1 CC(O)(Cc1ccccc1)C(=O)NCC=CCNC(c1ccc(CO)s1)=O c1(NC2C(CC)CN(C(C3CCCN(C(N)=O)C3)=O)CC2)nc(C)nc(C)c1F C(=O)(C(F)(F)C(F)(F)C(F)F)NCCCOCCNC(C1NC(=O)OC1)=O C(=O)(CC1=Cc2ccccc2C1)NCC1(CNC(CC2CCC(C)(C)O2)=O)CC1.C1CC1 c1(C=O)cc(=O)cc[nH]1.C1(CC(=O)N)(OC)CN(N(C(C)CO)C)C1 C1(NC(C(CC2CC2)OC)=O)CCCCC1NC(C1CC1c1cccnc1)=O C12(C(=O)NC3C(CC(=O)N(CCN=[N+]=[N-])C)CCC3)CCC(CC1)CC2 c1(C(c2cc(Br)nc(Br)c2)N2CC(C(=O)NCCCCC)C2)cc(F)cnc1Cl c1(NC(CCCOC)c2nnnn2C)ccc(F)c(Cc2ccccc2)c1 C(C)(c1ccc(F)cc1F)=CC(=O)N(CC(CNC(CCCCC=C)=O)O)C C12(NC(COCc3cc(C)on3)=O)CCN(C(C3(C(F)F)CCC3)=O)CC1C2 C1(N(C(=O)NCCS(CC)=O)C)CS(=O)(=O)C12CCOCC2 c1(C(N(CC(CNC(c2cc(C)nnc2)=O)(C)C)C)=O)cc(F)ccc1Br N1(C(CCCc2n[nH]c(=N)s2)=O)CCN(C(=O)NCCCCl)CC1C(F)(F)F C(=O)(C1=NN(C2CC2)C(=O)CC1)N1CC(CC=C)(NC(c2ccoc2Cl)=O)C1 C(CS(=O)(=O)CC(=O)NC(C1CN(C(C2(C)CCC(=O)C2)=O)CCO1)C)OC c1(CC(=O)NC2CCN(C(=O)CCc3cncnc3)C2)ccc(O)nc1 C1(COC)CN(C(=O)C(C2(O)CN(C(C34CC(C#N)(C3)C4)=O)C2)F)CCO1 C1(C)(CC)CC(NC(=O)CC2CCCCC2NC(c2cc(C)nn2C)=O)CCO1 c1(NC(CCC(=O)NC(C)C(=O)NC2CC2)=O)cccc(O)c1F N1(C(c2cc(C)n(C)n2)=O)Cc2ccccc2CC1CNC(C1C=CCCC1)=O C1(C(=O)NC(CCSCC)CO)COCCC1NC(=O)CC1C=NN(C)C1=O c1(COC)cc(C(=O)NCCCCNC(=O)CC2C(C)C2(F)F)n[nH]1 C#CCC(C)(CC)C(=O)NCC(C1CCN(C(C2CCCN2CCC)=O)CC1)O CC(C)P(=O)(CC(=O)N1CCC(NC(=O)C(C)(C)CC(F)(F)F)C(O)C1)C(C)C C1(C(=O)NCCSCC(=O)NOCCCCF)CC12CCOCC2 c1(C(=O)NCC2CCC(C)CN2C(=O)CC2(C)CCCC2)cnc2[nH]cnc2c1 c1(NC(C2C(NC(=O)C3=CCSC3)CCOC2)=O)cccc(Cl)c1O N1(C(C2(CC)CCC2)=O)CCCC(n2cc(C(C)NC)nn2)C1 c1(C(N2C3CN(C(C4C5COCC45)=O)CC2C3)=O)ccnc2c1OCO2 c1(C(=O)NC(C2CCCN(C(=O)COCC(F)F)C2)C)cc2c(ncn2C)s1 c1(C2C(C(=O)NC3CC(N(C(CC(=O)NCC#C)=O)C)C3)C2)ccccc1Cl N1(C(C(C)OCC2CCCO2)=O)CCC(C)(C)C(CO)C1.C1(C2CCC2)(C=O)CC1 C1(CNC(C2OCCN(C(C)=O)C2)=O)CN(C(c2cnsc2)=O)CC12CCC2 N1(C(C=CCN(CC)CC)=O)CCCC(N(C(=O)CCCOC(C)C)C)C1 N1(C(c2nnn(C)c2N)=O)CC(NC(C2CC(CC3CC3)C2)=O)CC2(CCC2)C1 CC1COC(=O)C1CC(c1ccccc1Br)N(C(C)(C)C)C(=O)O.N(C)(C)C=O C1(C2CCCN(C(=O)C3=CCCCC3)C2)(NC(CC(CC)SC)=O)CC1 C1(C(=O)NC2CCC(NC(C3CC(SC)C3)=O)C2)COCCN1C c1(CC)c(OC)cccc1C(=O)NCC1CCCCN(C(=O)COC(C)(C)C)C1 C(C(C(C)(C)C)NC(=O)CCn1ncn(C)c1=O)NC(CC(=O)OC)=O CCCS(=O)(=O)CC(=O)N1CC(NC(=O)Cc2csc(COC)n2)CCC1C n1(CC(N2CCC2c2cn(Cc3ccno3)nn2)=O)ccc2c(Br)cccc12 C1(C(N2CC(C(N3CC(=C)C3)=O)(SC)C2)=O)CCSC1(C)C c1(C(N2CC(O)(C(C)NC(=O)CCNC(N)=O)C2)=O)coc2c1C(=O)NCC2 N1(C(COCCC)=O)CCC(CNC(c2c(OC)noc2C2CC2)=O)C(C)C1 C(CC(C)C)(C(=O)NCCCC1CCCC1)NC(c1c(CC)ccs1)=O c1(C(=O)NCC(CCCC)NC(C2CC2C2CCCC2)=O)c[nH]cc(C)c1=O Cc1cc(=O)n(C)nc1C(=O)N(C)CCCCNC(c1ccc(C2CCOC2)s1)=O.N N1(C(CC(=O)OC(C)(C)C)=O)CC(CNc2cccc(CC(=O)O)c2)CC(F)C1 C1(C(N2C(CNC(c3c(C)coc3)=O)CCC2)=O)CCN(CC(C)C)CC1 C(=O)(CCC(F)(F)CSC1CC1CS(N)(=O)=O)NC(C1C(C)C1)=O CON1CCC(C(=O)NCC2(NC(c3cn(C)cc3C)=O)CCCCC2C)C1=O C1(C(=O)NCC2(F)CCN(C(C(C3CC3)SC)=O)CC2)Cc2cc(F)ccc2O1 S(=O)(=O)(c1ccc(NCc2cc(Br)ccc2F)cc1Br)NCC(C(C)(C)C)SC CCN=C(NCC1CCOCC1C)N1CCC(S(C)(=O)=O)CC1 CC(C)C(F)C(=O)N(CCNC(c1coc(C(N)=O)c1)=O)CCOCCO c1(CN=C(NCC2N(C)CC2)NCC2CCCO2)csc(S(N)(=O)=O)c1 C1(O)(CC(C)C)CCN(C(=O)C(C(C)C)NC(=O)CC2CCOCC2)C1 N1(C(CCC(C)OCC)=O)CCN(C(c2ccccc2N2CCCC2)=O)CC1C Cc1ccc(Cl)c(F)c1C(=O)NCC12CC(C1)C(NC(=O)C=CCO)CO2 CC(CCCCNC(c1coc(Br)n1)=O)NC(=O)COCCF CC1CCN(C(=O)C=CC2CCOCC2)C1C(=O)Nc1ccc(OCF)cc1 CC1(C)CCC(O)(C(=O)NCC(CO)NC(=O)Cc2c[nH]ccc2=O)CC1 N1(C(C2=CC(C)(C)C2)=O)CC2(CCC(NC(=O)CCOc3ccccc3)CC2)C1 N1(C(COC(CC)C)=O)CCC(O)(CN(C(=O)C=CC2CCCO2)C)C1 C(=O)(C(S(C)(=O)=O)C1CC1)NCCC1N(C(C(C)=C2CCCC2)=O)CCC1 C1COCCN(CC2CC2)C1.C=CCCC(=O)Nc1nnc(-c2ccccc2)o1 c1(CC(=O)OCCN)c(C)ncnc1C.C(CC(=O)N1CC(OCC)C1)OCC#C C(CCCC(=O)NC1CCOCC1NC(C12CCCC(CO1)C2)=O)(OC)OC C1(NC(=O)OC(C)(C)C)C=CCCC1(C)CO.c12cnn(c1)CCCNC(=O)N2 c1(NC(C)=O)cccc(C(N2CCCC(CNC(=O)CC34CCCC3C4)C2)=O)n1 C(CN=c1cc(C(F)F)nc[nH]1)(C1CCCOC1)NC(C1(CC2CC2)CC1(F)F)=O c1(C(=O)NC(C2CCCN(C(=O)C(C)(C)c3ccsc3)C2)C)cn(C)nc1O C1(NC(C2CCN(C(CCCCCC)=O)CC2)=O)CC2(CCCCC2)C1 N1(C(=O)NCCc2ccc([N+](=O)[O-])cc2)CCCC(C2CN(C3CC3)C2)C1 C(=O)(C1=C(Cl)CCCC1)NC1CC(C(C)NC(c2csc(C(C)(C)C)c2)=O)C1 C1(C(N(CCCNC(c2nc(=O)n(C)[nH]2)=O)C(C)C)=O)Cc2ccccc2C1C c1(NC(N(C(c2ccccc2F)C(C)C)C(C)C)=O)ccc2c(O)nccc2n1 c1(NC(CCC2N(C(COc3cc(C)nn3C)=O)CCC2)=O)cc(F)c(Cl)cn1 C1(CC)CN(C(=O)C(C)(C)CO)CCN1C(c1cc(C(C)C)n(C)n1)=O C1(C(=O)NCCN(C(=O)Cn2ccc(=O)n(C)c2=O)CC)CNC(=O)CC12CCC2 N1(C(C)C(=O)N(CCCN(C)C)CCNC(C2CC(C#N)C2)=O)C(=O)CCC1=O N1(C(CC2(NC(C)=O)CC2)=O)CC(NC(=O)C(C)(C)CN(C)C)CC12CCC2 C(CCC(C)C)(C(=O)NOCCc1ccccc1)NC(c1cccc(C)c1N)=O C1(NC(c2[nH]nnc2-c2ccccc2)=O)CCCN(C(=O)CC2CC3CC3C2)C1 N1(C(C(C=C)(C)O)=O)CCC(N=c2nc(C(F)(F)F)[nH]s2)C(C)C1 C1(C(=O)OCC)CCN(C(c2ccc(CC)s2)=O)C1.C12CCCC1CC(=O)N2.CSC C1(NC(c2c(C)n(C)nc2)=O)C(C)(C)C(NC(=O)C(C)N2CC(C)C2)C1(C)C c1(OC)ccccc1C(C)NC(=O)C(N1CCC(CN(C)C)C1)=O c1(C(=O)NC(CNC(c2nccc(OC)c2)=O)C)cc(F)c(Br)cc1N CC(C(CO)NC(=O)C(O)COCc1ccccc1)NC(=O)CN1CCOC1=O C1(C(=O)NC2(C3CN(C(=O)C4=CCSC4)C3)CC2)CCCC2(CCCCC2)C1 Cc1cncc(C(=O)NC2CC3CC(NC(c4cc[nH]n4)=O)C2C3)c1C CN1CCCC(C(=O)NC2CCC2NC(c2cn(C)cn2)=O)C1 c1(NC(C)=O)cccc2c1OCCN(C(=O)CSCC(=O)N=c1cc(C)o[nH]1)C2 C(C(N=c1[nH]c(NC(C(=COCC)C#N)=O)ncc1Br)C(C)C(C)C)C(=O)OC CC1Cn2nccc2CN1C(=O)COC1CCN(C(c2ccc(CO)cc2)=O)C1 CCC(O)C(C)C(=O)NC1(C)CCCN(C(=O)C=Cc2cnn(C)c2)C1 c1(CC)ccccc1OCC(N1CCC1COC(=O)C(C)CCNC1CC1)=O N1(C(c2ccc(C(C)C)nc2)=O)CCCC2CN(C(=O)CN(C)C(C)C)CC12 n1(CC(=O)NC(C2(CNC(=O)CN3CCOCC3)CC2)C)nc(Cl)ccc1=O c1(CC(N2CC(O)(C(C)(C)CNC(C)=O)C2)=O)nc2ccccc2[nH]1 c1(OC)c(C(=O)NCC2CC(NC(C3CC3(C)C)=O)C2)cc(Cl)cc1C N1(C(Cn2c(C)cnc2)=O)CCN(C(C2(F)CCS(=O)(=O)C2)=O)CC1CF Cc1ccc(O)c(C(=O)NCCCC(O)C(=O)N2C(CO)CC2C)c1 C1(NC(c2ccc(Oc3ccccc3)cc2)=O)COCCN(Cc2cc[nH]c2)C1 C1(C(=O)NC2C(NC(=O)C3CC3)CCCC2)Cc2ccncc2C1 CSC1=C(C(=O)N2CCCC(CCNC(C3(C#N)CCOC3)=O)C2)CCCC1 C1(C(=O)NC(CNC(c2cc(CC)ncn2)=O)C)CCC2C(CC1)C2(F)F c1(C)c(Cl)oc2ccccc12.CCCC(CCN1C(=O)OCC1)CCC.OC c1(CCC(=O)NCC(CNC(CCS(=O)(=O)NC)=O)F)ccc2ccn(C)c2c1 C(=O)(CCCCn1ccnn1)N(CC(C)NC(c1nc(CC)sc1)=O)C CN1CCN(C(=O)C=C2CCN(C)CC2)C(CNC(C2(C)CCC2)=O)C1 c1(C(=O)NC2C(CNC(C=C(C)c3ccccc3)=O)C2)cc2c(s1)CCCC2 CC(C)CC(C(=O)NCCCN1CCC(O)CC1)ONC(C1CCCCO1)=O Cc1cccc2cc(C(=O)NC3CN(c4ncc(Cl)c(O)n4)CC3(C)C)oc12 N1(C(c2ccc(Cl)cn2)C(=O)NCC)CCCc2oc(Br)cc2C1 N1(C(c2n(C)c(S)nc2)=O)CCN(C(=O)CN2CCCOC2=O)CC1CCO n1(C(C)C(=O)OCC(c2cnccn2)=O)ccc(Br)n1 c1(C(=O)NC(C2OCCN(C(c3c(CC)ncs3)=O)C2)C)cc(F)c(F)cc1F c1(CN2C(C(=O)NCc3cc(C(=O)OCC)n(C)n3)CC2)ccc(Cl)c(Cl)c1 c1(Cc2c(C(=O)NCc3ccccc3)cncc2)c(Cl)cccc1Cl c1(C(N(C2CCC2)CCC)=O)cn2c(n1)CCN(C(=O)C(C)(C)CN(C)C)CC2 c1(CC)noc(CSCC(=O)NC(CN2CCCC2)C(=O)NCS(=O)(=O)NC)n1 CC1CCC(NC(=O)CN2CSCCSC2)CN1C(C1(C2CCC2)CC1)=O C1(C(=O)NC2(COCC)CC2)CCOCC1C(=O)OC N1(C(=O)COC(F)(F)F)CC2CC(C1)N2C(c1cc(Cl)ns1)=O CC(C)C(C(=O)N=c1cc(CN)o[nH]1)NCC(F)CO N1(C(c2c(C)ncs2)=O)CCC2(CC2C(=O)NCC(C)CC(C)O)C1 CCC(F)(F)CC(=O)N(CC(O)CNC(c1cc(O)nc(N(C)C)n1)=O)C N1(C(c2c(CC)nco2)=O)CCC(C)(NC(c2cn(CCC(C)C)nn2)=O)CC1 N1(C(c2cc(OC)n(C)n2)=O)CCC(NC(=O)C(=Cc2ccco2)C)C(C)C1 c1(CNC(=O)NC23COC(N2)C3)ccc(OC(F)F)c(O)c1 CCCCCCC(C)CC(=O)N1CCC(NCC(=O)Nc2ccc(F)cc2N)C1 c1(C(=O)NC(C(C)NC(=O)CCC2CCC2)CO)ccc(C#N)cn1 C1(CNC(CCSC)=O)CCCN(c2nc(-c3ccccc3)cs2)C1 C1(C(=O)NC(c2cnc(C)s2)CC)C2CC2CN1C(c1cncc(OC)c1)=O C1(CC(=O)N(CCNC(=O)CC2CC3CC3C2)C2CC2)(OC)CCCC1 c1(N(C(C)=O)C)ccccc1C(N1CCC2C(NC(c3cc(F)n(C)n3)=O)C12)=O N1(C(CC2CN(C)C2)=O)CCC(CNC(C2CCCN2C2CC2)=O)C1(C)C c1(OCC(=O)NCCN(C(=O)Cc2nc(C3CC3)nn2C)C)ccc(Cl)cc1 c1(C(C(=O)NCC2(NC(=O)C(F)Cc3ccccc3)CCC2)O)ccc(Cl)cc1 N1(C(C(C)Cc2ccncc2)=O)CC2(COC(CNC(C3(CF)CC3)=O)C2)C1 c1(NC(=O)Nc2c(C(=O)OCC)nc(C(C)(C)C)s2)c([N+](=O)[O-])ccc(F)c1C N1(C(c2cc(C)n(C)n2)=O)CCC2(C=C(C(=O)NC3COCC(C)(C)C3)C2)C1 N1(Cc2ncc(C)[nH]2)CCN(c2cc(NC(c3ccc(C)s3)C)ncn2)CC1 C(C)(CC(C)N=c1[nH]nc(C)s1)NC(Cc1cncc(C)c1)=O C(C1CCC(C)CC1)=C(C)C(=O)NC1CCC1NC(=O)Cc1coc(C(F)F)n1 C1(C)(NC(C(Cc2ccoc2)NC(CC2CN(C(C)=O)C2)=O)=O)CCC(C)(C)C1 C1(C(C)C)COCCN1C(=O)C(O)CNC(=O)C(C)(C)CN(C)C N1(CC(=O)NC(C(C)NC(CCCCC)=O)CO)CCc2sccc2C1 Cc1nc2cc(Cl)ccc2cc1C(=O)NC(C)CNC(=O)C=C1CCC(C)CC1 CC(N=c1cc[nH]c(=NCCOC2CCOC2)[nH]1)c1cccc(Br)n1 N1(C(C2N(S(C)(=O)=O)CC2)=O)CCC(CO)C(NC(C2(Cl)CC2(F)F)=O)C1 C#Cc1ccc(NC(=O)CSc2cccc(F)c2F)cc1.C1(=O)CN1C c1(C(=O)NCC(C2CCOC2)NC(CC2CC(=C)C2)=O)ccc2ncccc2n1 C1(O)(C(N2CC(NC(COCCC=C)=O)C(O)CC2)=O)CCC(C)(C)CC1 Cc1cc(C#N)cc(C(=O)NC2CC(F)(CNC(c3ccn(C(F)F)n3)=O)C2)n1 CC1(C)CC(O)(CN2CCOC(CNC(C3COCCO3)=O)C2)CO1 C(=O)(NNc1c(F)ccc(F)c1Cl)c1n(C(C)(C)C)ccn1 C(=O)(CC(=O)NCCN(C(=O)CC1CC(F)(F)C1)CC1CC1)OC c1(C(=O)OCc2c(C)ncs2)ccc2occc2c1 C(=O)(C(O)CC(C)C)N1CCC(CC#C)(C(=O)N(CC(N2CCOCC2)C)CC)C1 C12(CNC(NCc3ncccn3)=NCC3CC3)CCCN(CC1)C2 c1(C(N2CCN(C(C3C(OCC)C3)=O)CC2)=O)cc(N)c(C)c([N+](=O)[O-])c1.C=O c1(OCC)ncc(C(N2CC(CCNC(c3c[nH]c(=N)c(C)c3)=O)C2)=O)cc1Cl C1(C(N2CC(C)(NC(COCCCC#C)=O)C2)=O)NC(=O)OC1C C1(C(=O)OC)C=CCCN1C(C1CC1NC(=O)CC1(C)CCN1C(C)=O)=O Cc1cc(C(=O)NC2CC(NC(C3CS(=O)(=O)C3)=O)CC2O)cnc1O C1(COC2CN(C(CC3(OC)CCC3)=O)C2)CC2CCC1N2C(=O)COC CCCC(CC)CCC(=O)N1CC(NC(c2cnc(S)nc2)=O)CC1(C)C N1(C(C(CC#C)C)=O)CC2CCCC2(NC(c2cnn(CCF)c2)=O)C1 O=C1CCC(CNC(c2cccc(-c3ccc(O)nc3)c2)=O)C(=O)N1 c1(C(=O)NCC(C(=O)NCC(C(=O)NC)O)(C)C)c(C)cccc1O C(c1cccs1)=C(C)C(=O)NC1CCC1NC(=O)CC(C)F CC1(C)OC(C)(C)c2ccc(C(=O)NCC3(c4nn[nH]n4)CC3(C)C)cc21 c1(C(=O)NC2C(NC(=O)COc3ccc(F)c(F)c3)CC2)ccc2cnnn2c1 c1(C(N)=O)cc(C(=O)NCC(O)CNC(=O)CN2CCCS2(=O)=O)cc(F)c1 C1(NC(c2c(C)cc(C)nc2)=O)CC2CC(C1)N(C(=O)CCc1ccccc1)C2 CS(=O)(=O)CCCC(=O)NC(=O)CC1CC1(C)C.C12(CC(N)=O)CCN(CC1)C2 N1(C(C2CCC(N(C)C)CC2)=O)C2CCC1C(CNC(=O)CCCN(C)C)C2 C1(CC#C)(C(N2CCC(C)(CNC(C34COCC(C3)C4)=O)C2)=O)CC=CCC1 C1(c2n(CC=C)nnn2)(NC2CC2c2cnn(C)c2C)CCOCC1OC C(=O)(CC(O)CCC(C)CC)NC1COCCN(C(CSCCC)=O)C1 C1(C(N2CC(C(=O)NC3C=CCCC3CO)C(F)C2)=O)CCCC2(CC2)C1 N1(C(CC2C(C)C2)=O)CCCC(NC(C2(F)CC2c2ccccc2)=O)C1 c1(NC(=O)C(=O)NC(CC=C)Cc2ccccc2)cc(C#N)cc(C#N)c1 c1(N2CCN(C(C3CCN3Cc3ccccc3)=O)CC2)nc2ccccc2s1 N(C(=NCCC(C)(C)O)NC1CCN(C(=O)Nc2cccs2)CC1)C(CC)C N1(C(C(CC)CCCO)=O)CCCC(n2cc(CC3(COCC)CC3)nn2)CC1 c1(C(CNC(=O)COC2CC2)NC(=O)C(O)Cc2cnc[nH]2)cccc(Cl)c1 CC(F)(CC1CCCC1)C(=O)NC1CC(NC(c2ccccc2O)=O)C1 CC1(C)CN(C2CC2)C1=O.C(CC(=O)NC1CC1)SCCCc1nc[nH]n1 CC1CC(C#N)(C(=O)NCC(C)NC(c2ncsc2C2CC2)=O)C1 C(=O)(N1CCC(C(=O)NC2CC=C(C)CC2)O1)C1C(C=C)OCC1 C1(NC(C(C)C)=O)C2CC3CN(C(=O)CN4CC(=O)NC5CCCCC45)C1C3C2 C(=O)(C1=Cc2ccc(Cl)cc2OC1)N1CCC(CNC(CCC(=O)N(C)C)=O)C1 c1(N2CC(CC)NC(=O)C2)nc(NC2CCN(CC)CC2)nc2c1COCC2 c1(C(=O)NC2CC(C(C)NC(C(CC)C(F)(F)F)=O)C2)cncc2ncn(C)c12 C12CCCC13CCN(C3)C2=O.c1(C(=O)NCCN2CCCC2)ccsc1Cl N1(C(Cc2nc(C)sc2)=O)CCCN(C(c2ncc(N)nc2C)=O)C(CO)C1 c1(C(=O)NCC2COCCN2Cc2ccc(Cl)cn2)cccc(OC(F)F)c1 C=CC(CCC)CC(=O)N1CCCN(C(=O)C=C(CCC)CCC)CC1 C(CN=c1nc2sccc2c(NC(C)CO)[nH]1)NCC(CC)OC1CCCCO1 c1(C(N2CC(CNC(C(C(C)C)SCC)=O)N(C)CC2)=O)ccn2nccc2c1 C12(NC(c3ncc(Br)cc3F)=O)CCCC1N(C(=O)C=CC1CC1)CCC2 c1(C(N(C2CN(C(C3CC4(CCCO4)C3)=O)C2)C)=O)n[nH]c2nccc(Cl)c12 C=CCC(CC(C)C)C(=O)NCC1CCN1C(c1cc([N+](=O)[O-])cnc1O)=O C1(C(=O)NC2CC(NC(c3cccc(CF)c3)=O)C2)CCn2nncc2C1 C(=O)(C(C)CC(C)C)N1CC2C(CNC(CC(OCC)OCC)=O)(C2)C1 n1(CC)cc(C(=O)NC(C)C(C)NC(c2csc(CO)n2)=O)c(C2CC2)c1.C(C)=O N1(CCN(C(C)CC2CC2c2ccccc2)C)CCCC1=O N1(C(c2cncc(NCC)c2)=O)CCCC(NC(c2nnc(C)s2)=O)C(F)C1 C1(C)(CC)CCC(C(N2CCC(=CCNC(=O)CCC3(O)CCC3)CC2)=O)O1 N1(Cc2ccc(C)s2)CCC2CN(C(c3ccncc3)=O)CCC12 c1(CC)ccc(F)c(C(=O)NCC2CCCCCN2C(c2n[nH]cc2OC)=O)c1 N1(C(c2ccon2)=O)CCCC(CCCCNC(C2CC(OC(F)(F)F)C2)=O)C1 C#CC1CN(C(=O)C(CCC2CC2)NC(=O)CNC(=O)C2CC2)CCO1 c1(CC(=O)NCC(F)CNC(=O)CN2CC=CC2)cnsc1 Cc1cnc(NCC(C)N(C)C)c(S(=O)(=O)NC2CCCCC2(C)C)c1 c1(C(=O)OC)ccccc1C(N1CC(C)(NC(C2NC(=O)CC2C)=O)C1)=O c1(C(=O)NC2CCCN(C(CCC=CCC=C)=O)CC2)cccc2ccsc12 N1(C(Cc2c(C)noc2C)=O)CCCC(O)(CNC(c2csc(C#N)c2)=O)C1 c12n[nH]cc1C(=O)NCC2.C(CC(=O)NCC(=O)NCCO)SC C1(NC(C2ON=C(CC)C2)c2ccccc2)CC2CC1CN2CC1CCCC(=O)N1 N1(C(C2CC(NCc3cccc(CO)c3)C2)=O)CC2(CCC2O)C1 C1(CNC(=O)Cc2ccns2)CCCCN1C(=O)COc1ccc(F)nc1 c1(C(=O)NC2C(NC(c3scnc3Cl)=O)CCCC2)n[nH]c2c1CC1CC21 C1(CCC)CC(N(CC(C)(C)CNC(C2CC23CCCC3)=O)C)CCO1 N1(C(CCCCC)=O)CCN(C(=O)Cc2cncs2)C(c2ccccc2OC)C1 c1(C(=O)NC(C)(C)CNC(=O)CSCC(N)=O)cccc2nc(-c3cccs3)[nH]c12 C12(CN(C)CC3COC(=O)N3)COC(C(F)(F)F)(C1)C2 CC(C)CCC(=O)N(C1CCC(C(=O)OC(C)(C)C)C1)S(=O)(=O)CC1CC1 c1(N2CC=C(C)CC2)nc2cccc(F)c2c(=Nc2ccccc2C(F)(F)F)[nH]1 N1(C(CC(CC)C)=O)CCC(C)(NC(=O)C=CC2CCC(C)CC2)CC1 C1(C(N(c2ccc(F)cc2)C)=O)CC12CCc1ccccc12 Cc1onc(Cl)c1C(N1CCN(CC2CCCN(C(=O)C(C)(F)F)C2)CC1)=O c1(NC(C)=O)ccc(Cl)c(C(N2CCN(C(c3cc(Cl)ncn3)=O)C3CC23)=O)c1 N1(C(c2cnc(OC)c(Cl)c2)=O)CC(C)C(NC(=O)COC(=O)CO)C(C)C1 Cc1cc(CNC2CCC(NC(c3ccc(C#N)cc3)=O)CC2)ccc1Cl N1(C(c2cnc(CCC)s2)=O)CCN(C(C2CC2F)=O)CC1c1cnn(C)c1 Cc1nc(CCC(=O)NCC=CCNC(=O)C(C(C)C)NS(C)(=O)=O)c(C)s1 c1(C(=O)NC(CCOC)CNC(c2cnc(O)n2C)=O)cn2ccc(C)cc2n1 C1(C(=O)NCCCC)C(C)CCCN1C(=O)C=CCOCCOC(C)=O c1(C(=O)NCC(C2CCCCC2)NC(=O)CC2CC2C(F)(F)F)ncncc1Cl c1(C(N2CCC(N(C(=O)C=Cc3cc[nH]n3)C)C2)=O)nc2cnccc2s1 N1(CC)CC(CNC(=O)CCC2CC(NC(c3cc(C)no3)=O)C2)CC1=O N1(C(COC)=O)CCC(C2CCN(C(c3cccc(C)c3)=O)C2)C1 N1(C(C2CN(C(CCc3ccn(C)n3)=O)CC23CC3)=O)CC2CC3CC2C1C3 c1(OC)ccc(C(=O)NCC23CC2CN(C(C2CC(C(F)(F)F)C2)=O)C3)c(Cl)c1 N1(CC)CCOCC1C(=O)NC1CCCC1CC(N1CC(N(C)C)C1)=O c1(OC)ccc2c(c1)C(C)(C)CC2NCc1ccc2ncc(Br)n2c1 O=S(=O)(c1ccc2[nH]c(=NCCn3ccnc3)sc2c1)Nc1ncccn1 Cc1cc(NC(C2CC(NC(C3CCC(=O)N(C)C3)=O)C2)=O)cnc1O c1(C(=O)NC2CC2NC(C2(C3CC(=C4CC4)C3)CC2)=O)nc(Cl)cs1 Cc1cccn2nc(C(N3CCC4(CCN(C(=O)CCCCCF)C4)C3)=O)cc12 C=CCC(C(=O)N(C)CNC(=O)C(C1CCC(CC)CC1)C1CCCC1)C(C)C c1(N2CCn3c(C)cnc3CC2)[nH]c(=NCCC(C)CCCC(C)C)nc2sccc12 C1(CNC(C(C)=C2CCC2)=O)CCN(C(c2ccn3nccc3n2)=O)C12CCC2 CC(C)CC(CC(C)C)C(=O)N(C)CCN(C(=O)Cc1cc(F)ccc1Cl)C C1(C)(NC(Cn2ccc(C)c2)=O)CCCCC1C(=O)N(C1CCCC1C#N)C c1(C(=O)NCC(C2CCCCC2)NC(CCOC)=O)cnn(C)c1C(C)(F)F N1(C(=O)OC(C)(C)C)CC(C2CN(C(=O)NC3CCCC(OC(C)(C)C)C3)C2)C1 C1(C(F)F)(OC)CCN(C(c2ccc(Cl)cc2)C)C1.n12cnc(=O)n(c1=O)CC2 N1(C(CC2C=NN(C)C2=O)=O)CC2(NC(c3n[nH]cc3Cl)=O)CCC1CC2 N1(C(C(C)CF)=O)CC2C(N(C(=O)Cc3cncnc3)C)C2C1 C1(C(=O)N(CC2(CNC(=O)CN3CCCC3)CC23CCC3)CC)CC12CCSCC2 c1(C(N2CC(NC(c3nc(C#C)sc3)=O)C(C)CC2)=O)cncc2c1CCCC2 C(C(C)(C(C)C)NC(C1CC2C=CC1C2)=O)NC(C(C)OCc1ccccc1)=O c1(CC(C(=O)NC2CC(F)(CNC(CCC=CCC=C)=O)C2)C)c(C)noc1C c1(C2C(C(N(CCCNC(CCC#C)=O)C)=O)C2)cc(Cl)ccc1Cl C1(c2nnnn2CCCOCCCN2CC=CC2)(COC)CCC(=O)NC1 C1(C(N2CC(NC(Cc3c(C)cc(O)cc3)=O)C2)=O)CCOC2(CCOCC2)C1 n1(CC(=O)NC2CCC(CC(=O)NC(CCC)(C)C)C2)ncn(C)c1=O Cc1ccc(NC(c2cccnc2C2CC2)=O)c(C)c1.C12(CC1)C(=O)NCC2 C(CNC(=O)C(=O)NC1CNCC1(C)C)(CC(C)(C)C)OC N1(C(C(C)OCC#C)=O)CCCC(N(C(=O)Cc2scnc2C)CC)C1 N1(C(c2ccc(C(=O)OC)cc2)C(=O)NC)CCCC2(CC1)CC2(F)F C1(CCN(C(=O)NCc2n[nH]c(C)c2Br)C)CCCCC12OCCO2 N1(C(C=C(C)C2CCCCC2)=O)CC(NC(=O)Cc2ccoc2)CC12CCOC2 C(CCCCC(=O)NCC1CC(C)CN(C(c2c(C)noc2C)=O)C1)=CC Cn1nc(C(=O)NC2CC(CCC(=O)NCCCN3CCCC3)C2)cc1[N+](=O)[O-] c1(CN(C(C(C)OC(C)(C)C)=O)CCCNC(c2cncs2)=O)ccccc1 C12(NC(C(C(C)C)SCC)=O)CCC(CN(C(c3cnsn3)=O)C1)C2 C(=O)(C1=C(c2ccccc2)SCCO1)NC1CC(NC(CCCC=C)=O)C1 N1(C(CS(C)(=O)=O)=O)CCC2C1CCCN2C(C1CC1c1ccccc1)=O c1(C(=O)NCC2(NC(=O)COC(F)(F)F)CCCC2)ccnc(N2CCCC2)n1 CC1=NNC(=O)C1CCC(=O)Nc1ncc(CCNC(C2CNC(=O)N2C)=O)s1 C12(NC(=O)OCC(=O)NC(C(=O)NCC)C(C)C)CCC(C)(C1)OC2 C1(F)(CNC(c2cscc2F)=O)CCN(C(C2CCC3(CCC3)O2)=O)CC1 C1(NC(C2C(C)(C)CC2)=O)CCN(C(c2cc(O)nc(Br)c2)=O)C12CC2 CCCCC(F)C(=O)NC12COC(C1)C(NC(=O)CCc1ccccc1)C2 c1(C(N2CCC(CN(C(=O)CN3CCOCC3)CC)C2)C)cc(F)cc(F)c1 C12(C(N(C)CCOCCCCNC(=O)CCC(C)(C)C)=O)CCCC(C)(C1)OC2 c1(CC(=O)NC2CCN(C(CNC(=O)OC)=O)CC2O)ccc2c(c1)CCO2 c1(NC(CCCN(C(=O)CN2CCNC(=O)C2)C)=O)ccc2c[nH]nc2c1 c1(SCC(=O)NC(CCCNC(CCC(C)OCC)=O)C)ccc2c(c1)CCC2 c1(C(N(CC2N(C(CC(CCC)C)=O)CCC2)CC)=O)ccc2cnoc2c1 C1C(C(C)C(C)C)NC(=O)CCC(=O)N1.c1(CCC(=O)OC(C)=O)ccc(O)cc1 C1(CCOC)(NC(=O)C(C)OCCOC(C)C)CCN(C(C)=O)C1 c1(C(N2CCN(Cc3ccc(OC)c(Br)c3)C3C2C3)=O)ccn2cncc2c1 C1(C)(CC(=O)NCC(Cn2cc(C3(F)CCOCC3)nn2)OC)CCSCC1 CC(CC(C)(C)C)C(=O)N1CCCCCC1C(N1CCC12CN(C)C2)=O C12(C(N3CCC(O)(C(C)C)C3)=O)CCCC1CCN2C(=O)CC(C)(C)C#N C1(NC(C(=O)NCC2CC2)=O)CCS(=O)(=O)C12CN(C(=O)CC1(O)CCC1)C2 c1(SC)cccc(C(=O)NC2(C)CCN(C(C3CCOC3)=O)C2)c1Cl c1(C(=O)NCC2CCCN(C(CCCSC)=O)C2)cc(Cl)ccc1N1CCCC1 c1(NC(=O)C2CC2)ccc(-c2ccnc(NC3CC3C3CC3)c2)cc1F c1(N2Cc3c(ccc(C)c3)CC2)nc2ccc(Cl)cc2c(=NC2CCCCC2F)[nH]1 c1(C(=O)NC(C2CCCCC2)CC)cc(Cl)cc(Cl)n1 CCCCC(CN=c1scncc1C)NC(c1coc2c1C(=O)NCC2)=O c1(CN(C(=O)CN2CCCCCC2)CCNC(c2cn(C)nc2)=O)ccc(O)cn1 CC1CN(C(=O)CC(C(F)F)NC(=O)Cc2ccn(C)n2)CCN(C)C1 C1(C(=O)NC(C2(O)CCN(C(c3scc(C)c3Cl)=O)C2)C)CCc2cncn2C1 C1(C#C)(NC(C2OCCC(NC(C3CCC(C#C)CC3)=O)C2)=O)CC2CCCC12 c1(CC(N2CC(NC(c3c(C)c[nH]n3)=O)C2)=O)c[nH]c2cccnc12 C1(NC(C2CC(n3cc(Cn4c(C)ncc4)nn3)C2)=O)CNC(=O)C(C)(C)C1 C1(CN(C(c2cc(C)sc2)=O)C)CCCCN1C(C1C(C)C1(F)F)=O C(=O)(C(C)CC(=O)NC1CCCC1NC(c1conc1C)=O)OC C1(CNC(CC2CC(OCC)C2)=O)CC(F)CN1C(C1CN(C)C(=O)N1)=O c1(COC)nc(C(C)(C)C)cc(=NCC2(CCOC3CCCN3)CC2)[nH]1 Cc1cccc(C)c1NC(=O)CN(C(C(=O)NN(C)C)c1nc[nH]n1)C1CC1 C1(NC(CCN(CCC)C)=O)CCCCN(C(c2csc(Br)c2C)=O)C1 C#CC1(O)CCCN(C(C2(C3CC3)CN(C(=O)C(O)CC3CCCC3)C2)=O)C1 C12C=CCN(C1)c1nnnn1CC1CN(CCN1)C2=O.c1(SCS)ccccc1.CO C1(C)(NC(c2c(CNC(C(COC)OC)=O)ocn2)=O)CC(C)(C)OC1=O N1(c2cc(CC)nc(CC)n2)CCC2C(CCCN2C(c2ccnn2CC)=O)C1 C(CNC(=O)C1=CCCS1)(C(C)C(C)C)NC(c1c(C(C)C)con1)=O c1(OC)cc(Cl)c(Cl)cc1C(=O)NCC1CCCN(C(=O)COC(C)=O)CC1 C1(C(=O)NC)CCN(C(=O)CCCCN(C(=O)CSCCOC)C)C1C CNS(=O)(=O)N1CCC(C(=O)OC(C(=O)NCc2cn(CC)nn2)c2cnc[nH]2)C1 Cc1cnc2n1C(C(=O)NCC1(C(C)NC(=O)CN3CC(C)(C)C3)CC1)CCC2 CCC(O)(CC)CCN=C(NC1CCC1)N(C)CCOc1ccc(F)cc1F C1(C)(NC(c2n(CCC)nnn2)C(C)(C)OC)CCS(=O)(=O)C1 c1(C(=O)NC2(C)CC(NC(CCN(CC)CC)=O)C2)ccc(Cl)c(N)c1 C1(NC(CC#C)(C)C)CCCN(C(C2CC=CC(c3ccccc3)C2)=O)C1 C12(CCCSC1)OC2.N1(C(C(=O)N(C)C)=O)CCC(CC2CC2)C1 N1(C(C(C(C)(C)C)OC)=O)C2CCC1CC(NC(c1nc3cnccc3s1)=O)C2 c1(CC(N2CC(N(C(Cn3cc(C(C)=O)nn3)=O)C)C2)=O)c(Br)cnn1C N1(C(C(C)N(C(=O)CC(Cl)Cl)CCOC)=O)CCCNC(=O)CC1 N1(CC(C)NC(c2cn(CCCOC)nc2)=O)CCN(C(=O)C(C)SC)CC1 c1(C(=O)NCCC2C(C)CCCN2C(=O)CC2CCC2)ccc2[nH]ccc2c1 CC1(C)Cc2ccc(NC(N3CCN(c4cc5cccnc5s4)CC3)=O)cc2C1 N1(C(C2(CC#C)CCCCO2)=O)CCCC2(C1)CN(C(=O)C(F)C1CCCC1)C2 c1(C(=O)NCC2OCCN(C(CC(=O)OC)=O)C2)ccc2n[nH]cc2c1C Cc1cnc(C(C(=O)NCC2CCCOC2)N(CCC#N)C)s1 c1(C(=O)NC(C2CCCN2C(=O)CCc2cnc[nH]2)(C)C)cccnc1C1CC1 n1(CC)nc(C)c(C(=O)NCc2ccc(CNC(C3C(C)C3C)=O)c(F)c2)c1C C1(O)(CNC(C(C)=C2CCC2)=O)CCN(C(=O)C(C)(O)C2CCC2)C1 N1(C(C(CCCOC)C)=O)CCC2CCC(NC(c3cccc4c3CCC4)=O)C12 c1(CC2CCCN(Cc3c(C)cco3)C2)c(C)nn(C)c1C C(=O)(C1(C)CCc2ccccc21)NC1CN(C(c2c(CC)nc[nH]2)=O)CC(C)C1 C=C(C)C1OCCCC1C(=O)NC(CNC(C1(CC(C)C)CCC1)=O)CCC C1(CN(C(C)CNC(=O)C(=O)NC2CCCOC2C)C)C(C)CCC1C c1(C(=O)NCC(CC(C)C)(C)NC(=O)C(C)CC(N)=O)nsc2c(Cl)cccc12 C(CC(C)C(=O)NCCCCC(=O)N(C)CCc1ccccn1)=CC N1(C(C(C)Cc2cncc(Cl)c2)=O)CCC2CN(C(c3ccc(F)cc3N)=O)CC12 C1(NC(C2(CC)CC2)=O)CCN(C(=O)CCc2nnc(C)n2C)CC1C(N)=O C(CCC(C)(C)C(=O)Nc1ccccc1O)NC(c1[nH]cc(C)c1C)=O c1(OCC)cc(OC)cc(CNC(C2CCN(C(c3cc(=O)cc[nH]3)=O)C2)=O)c1 C(C(O)C(=O)N1CCCC1CCNC(C1CC(c2ccccc2)O1)=O)N(C)C N#Cc1c[nH]c(=NC2C3CC2CN(C(C2(n4ccnn4)CC2)=O)C3)c2sccc12 c1(C(=O)NCC2(C(N)=O)CN(C(C3CCC(CO)O3)=O)C2)cnc2n1CCC2 N1(C(C2C(C)(C)CC2)=O)CC2CC(N=c3[nH]c4ccccc4s3)C2C1 CCC(CC(=O)N1C(CNC(=O)C(C(F)(F)F)OC)CC2CC12)CC(C)C c1(C(=O)NC(C)CCNC(C2CC2C2CCOCC2)=O)cc(=O)n2nccc2[nH]1 c1(C(=O)NC2C(CNC(C)=O)C2)cc(Br)c(C(F)(F)F)s1 C(=O)(CCCC(C)C)NCCC1(O)CCN(C(c2c(C)nn(C)c2)=O)C1 N1(C(c2c(O)cc(C)nn2)=O)CCCC2(CCCN2C(C2CCOC2C2CC2)=O)C1 C1(C(=O)NCC2(CNC(CC(C)SC)=O)CCC2)(OC)CCCCCCC1 n1(CC)nncc1C(=O)NC(C)CN(C)C(C1CC(C)(F)C1)=O N1(C(c2c(CC)cno2)=O)CC2CC1CN(C(=O)CN(S(C)(=O)=O)C)C2 CCC(C)C(=O)NC(COCC)C(=O)NCCOC1CCCC1 CCCCCC(C)CC(=O)N1CC(NC(c2cccc(=S)n2O)=O)C(C)C1 n1(C(CC)C)nc(-c2nc[nH]n2)nc1C(O)Cc1nccn1C c1(OCC)c(OC)cc(CN2CCCC2C(=O)NCC(F)(F)F)cc1Br C1(C(C)NC(c2cnc(C)[nH]2)=O)CCN(C(c2scnc2C(C)(C)C)=O)CC1 c1(NC(C23CC(NC(C4CN(C)C(=O)CC4)=O)(C2)C3)=O)cccc(C#N)c1F C1(NC(c2snnc2C2CC2)=O)C=CCC(C(=O)NCCCCCCO)C1 C1(NC(CC2CCCN(C(C3C(CC)N(C)CC3)=O)C2)=O)CCC2CCCC1O2 c1(CCCCCNC(C(C2CC(F)(F)C2)OC)=O)ccc(F)cc1 C1(CC)C(NC(=O)COCC(C)C)CCCN1C(C1CC12CCCC2)=O C1(CNC(CCCCOCC)=O)CN(C(C)=O)CCC12CCC2 C(C)(C)(C(=O)NCC1CCC(C(N)=O)O1)NC(C)=O.C12CCCC1C(=O)N2 c1(C(C)NCC(c2c(OC)cccc2)(F)F)ccc(Br)cc1OC(F)F C1(N(CC(C)(C)OCC)C)CCN(C(=O)CC2CCCC2)CC1 N1(C(c2c(C)nn[nH]2)=O)CCC2(CCOCC2)C(NC(=O)C2=CCSC2)C1 Cc1nc(C(N2CCC(O)(CNC(c3n[nH]c(C4CC4)c3Br)=O)C2)=O)sc1C C1(NC2CCC(C(=O)OCCOCCOC)C2)CCCC1OC c1(CC(=O)NC(CC(C)NC(c2cn(CC=C)nc2)=O)C)ccc2c(c1)CCO2 c1(-c2ccc(OCCCC)cc2)cnc(NC(=O)CCCC2CC2)c(O)c1 C=CCC(C)(C(F)F)NC(=O)CCC(C)NC(=O)CC(O)C1CCCC1 c1(C(N2C(CNC(c3n(C)c(O)nc3)=O)COCC2)=O)cn2ccccc2n1 C1(CCNC(CCN(CC)CC)=O)CN(C(=O)C(c2ccccc2)O)CCCO1 c1(C(N(CCOC)CCNC(=O)CC2CN(C)C2)=O)ccc2oc(C)nc2c1 N1(C(c2cc(CCC)on2)=O)CCN(C(=O)Cc2cncc(OC)c2)C2CC12 N1(CCC)CCC=C(c2cncnc2NC(c2cccc(-n3ccnc3)c2)=O)C1 c1(-c2cn(CC(CC)O)nn2)ccc(NC(=O)CNC(c2ccccc2)C)cc1 C1(C(=O)NCc2cn(CCNC(C=C(C)Cl)=O)nn2)CNC(=O)CC1C c1(CCC(=O)NCC2C(NC(C3C(Cl)(C(=O)OC)C3)=O)C2)ccccc1 c1(C(=O)NCC2CC(NC(C3C(C)CC3C)=O)C2)nc2ccccc2[nH]1 N1(C(c2c(CC)nn(C)c2)C(=O)NC(C)C)CC2(C)CCC2(C)C1 Cc1nc2c(C(=O)NCC(C)CNC(c3c(C)ccc(C)c3N)=O)ccnc2[nH]1 N1(C(C2CCN(C)CC2)=O)CC2CCC1CN(C(=O)C(C)(C)CC#N)C2 c1(C(=O)NCC(=O)NCC(CC)NC(=O)C(F)(F)CC2CC2)ccc(F)cc1 c1(C(N2CC(F)(C(=O)Nc3cn(C(C)C)nc3)C2)=O)ccc(I)c(Br)c1 C1(C(=O)NCc2ncccc2C(=O)NC(CCO)C2CCCC2)C2CCCOC12 C1(C(N(C2CC2)CC)=O)CN(C(c2noc(C)c2C)=O)CCC1(C)C c1(C(=O)NC23CC2CN(C(=O)CCC2CCOC2)C3)cccc2c1OCCC2 c1(NC2(CCC)CCCN(C(C3CCC4CC34)=O)C2)ncc2c(ncn2C)n1 C#CCC(C(=O)N1CSCC1C(=O)NCC(CC)n1cccn1)C1CC1 c1(C(N2CCCC3(NC(CC4(C)CC4)=O)C(C2)C3)=O)cc2c(nn1)OCCS2 C12(C(=O)NCC(CO)NC(c3scc(C)c3)=O)CC(C1)C(c1ccccc1)O2 C12(C)CCN(C1)CC(=O)N(C(C1CSCN1C)=O)C2c1cccs1.CCOCC C=CCC(C)(O)C(=O)N(C)CCOCCCN(C(=O)CCC(C)(C)F)C c1(CC)cc(C(=O)N(CC(C)O)CCNC(=O)CCC(=O)N(CC)CC)ccn1 CC(C)(C(=O)NCC1CCC(C(=O)NC(C2CCCCO2)CO)CC1)C(F)(F)F CCCC(C)(C)CC(=O)N1CCC(C(N(C(c2ncc[nH]2)CC)C)=O)C1 c1(C(=O)NCCC2(O)CN(C(c3c(Cl)n[nH]c3C3CC3)=O)C2)cc(F)cc(F)c1 c1(C(=O)NC(c2cn(CC3CCO3)nn2)CCC)ncccn1 CCC(O)C(C)(C)C(=O)N(C)CC1(CNC(C2CCC(=O)OC2)=O)CC1 CC1(C)CCCC(CCC(N2CCC(Nc3ccccc3)C2)=O)C1 c1(CC)ccc(C)c(C(=O)NCCC2CCOC2)c1.C12(CC1)C(=O)N2 Cc1ccc2nc(C(=O)NC(C)(CNC(C3SCCS3)=O)C3CC3)cn2c1 C1(CNC(C2CCC(CC)O2)=O)CC(O)CN1C(=O)COCc1nc[nH]n1 CC(C)C(COCCCOCCOCCNC(=O)CC1C(C)(C)C1(C)C)C=O c1(C(N2CCC(N(C)C(C3CC3C(F)F)=O)C2)=O)c(F)cc(OC(F)F)cc1F C1(C(=O)NCc2c(CO)cn(C)n2)CCN(C(=O)C(C)(C)C#N)CCO1 c1(C(N(C(C)CNC(c2cc[nH]c2)=O)CC)=O)cccc2[nH]c(C)cc12 C1(CCNC(C(C)n2ccnc2)=O)CN(C(=O)C(F)=C2CCC2)CCCO1 C1(NC(C2C(CC)C2)=O)CCOCC1NC(=O)CCSC1(c2ccccc2)CC1 c1(NC(c2cc(Cl)cc(Br)c2)c2n(CC)nnn2)ccc2scnc2c1 c1(CNC(c2n(CCCOC)nnn2)(C)CC2CCC(=O)N2)cn(C)nc1Br C(=O)(C(C)C(C)NC(c1cc[nH]c1CCC)=O)NC(CCCC)C C1(NC(CCN(C)CCO)=O)COC2(CNC(C3CC34CC(O)C4)=O)CC1C2 N1(C(CC2CN(C)C2)=O)CCc2c(CNC(=O)CCc3ccsc3)cccc2C1 c1(C(=O)NC2CCN(C(C3C(C)C3)=O)CC2C)coc2c1C(=O)NCCC2 C(=O)(CCCCCCCC)NC(CNC(C(CC=C)(C)O)=O)CC N1(C(c2c(N)ccc(OC)c2)=O)CC2CCCC(NC(=O)Cc3cnsc3)C2C1 C1(CCCC)CN(C(=O)C(C)C(C)(F)F)CCN1C(=O)C=COCC C(=O)(C1CSc2ccccc21)N1C2CC(NC(=O)Cc3cnc[nH]3)C(CC2)C1 C1(C(O)F)CCN(N2CCN(c3nccc(N4CCCCCC4)n3)CC2)C1 c1(C(N(CCNC(CC(CCC)C)=O)C2CC2)=O)cc(O)c2sccc2c1 C1(CC(=O)NC(C(=O)NCC(C)(C)O)CO)CC2(CC2)CO1 CC(CN(C)C(C1(C)CCCO1)=O)C(=O)N1CCCC1C1CC1 c1(NC(C(C(C)NC(c2c(C)scn2)=O)C)=O)cnc2[nH]cnc2c1 c1(C(=O)NCC(CC)NC(C2(c3ccc(F)cc3)CCC2)=O)cc2c(s1)CCC2 C(=O)(CC(=O)NC1(C(=O)NC(COCC)C(C)C)CC(F)C1)NCC#C c1(CC(=O)NC(CCNC(C(C=CCCC)O)=O)(C)C)cc(N(C)C)ccc1N N1(C(C=COCC)=O)CC2CCC1C1CN(C(c3occ(C)c3C)=O)CC21 N1(C(c2ccc(N)c(N)n2)=O)C2CCC1C1CC1(NC(=O)C=CC=C(Cl)Cl)C2 CC1CC=C(C(=O)NCCCN(CC(=O)N(C)C)CCC(F)(F)F)CC1 CC(C)C(CNC(=O)C(C)CO)NC(=O)C(C)OCC1CCCCO1 c1(C(C)C)[nH]nc(C(N2CCC(NC(=O)CSc3ncccn3)C2)=O)c1[N+](=O)[O-] Cc1conc1CC(=O)NC1CC(C(=O)NCc2csc(Br)c2)C1 C12(CNC(c3cc(C)[nH]n3)=O)CN(C(C3(CC4CC4)CC3)=O)CC(F)(C1)C2 CN1CCN(C(C2(C3CC3)CC=CC2)=O)CC1CNC(C1CCOCC1)=O Cc1ccc(F)c(CC(N2CC(CNC(c3cc(C4CC4)no3)=O)CC2C)=O)c1 C#Cc1cc(C(N2CCC(NC(=O)CN3CC4CC4C3)C(F)C2)=O)ccc1C Cc1cc(=NC(=O)C2(C)CCN(C(c3cc(Br)c(O)c(Br)c3)=O)CC2)[nH][nH]1 C(=O)(CCCCCC#N)NCCCCC(=O)N1CCC(N(C)C)C1 N1(C(c2nc(OC)c(C)s2)=O)CC(NC(=O)CCc2cc(C)[nH]n2)C2CC2C1 C=CCC(CNC(=O)CC1CC1C1CC1)C(=O)NCCc1cocn1 C1(NC(C2(C)CC2)=O)CN(C(=O)C(C)N2CCC2)CC1c1ccnn1C.C1CC1 c1(OCC(=O)NCC2CCC(NC(C3C(C)C3C)=O)C2)cccc(Cl)c1Cl C(=O)(CC(C)CC(C)(C)C)N1CCCN(C(Cn2ccc(C)cc2=O)=O)CC1C CP(C)(=O)C1CCN(c2nnnn2Cc2ccccc2N2CCC(CO)C2)CC1 C1(C(C)(C)C)(CNC(C2CNC(=O)C2)=O)CCN(C(=O)COC(F)(F)F)C1 C1(CC)Cc2ccccc2N(Cc2cc(F)cc(C(=O)O)c2C)C1 c1(C(C)C)ccc(OCC(=O)NC(c2ccc(Br)cc2)CSC(C)C)cc1 c1(OCC(=O)NCC(O)CNC(C2(C(F)(F)F)CC2)=O)ccccn1 N1(C(C2N(C(CC(CC)C(F)F)=O)CC23CCCC3)=O)CCC2(CCCCO2)C1 Cc1ccc(C=CCC(N2CCC(NC(c3ccnnc3)=O)C(F)C2)=O)cc1 C1(C(N(CCSC)CC)=O)CCN(C(c2ccncc2NC)=O)CCO1 c1(OC)ccc(C(=O)NCC2CCN(Cc3ccc(F)cc3)C2)cc1C(C)(C)C C1(NC(c2c(C)c[nH]c2)=O)COC2(CCN(C(c3c(O)cccc3Cl)=O)C2)C1 Cc1nn(C)cc1C1=NOC(C(N2CCN(C(=O)CCF)CC2C(C)(C)C)=O)C1 C12(CNC(C3COCCO3)=O)CCC(CC1NC(c1ccc(Br)o1)=O)C2 C(=O)(C(CO)NC(C1CCOC1)=O)N(C)Cc1sccc1CO Cc1cc(Cl)cc(C(N2CCC(NC(c3ccc(Cl)cn3)=O)C2C(C)C)=O)c1N N1(C(c2c(CC)onc2)=O)CCC(NC(=O)CS(N)(=O)=O)C(C)C1 C12CC3CCC1(C3)C(=O)Cc1cn2nn1.C#Cc1cnn(CC(=O)OC)c1 N1(C(COCCCC#C)=O)CCC2(CC1)CC2CNC(=O)C(C)NC(N)=O n1(CCOC)cc(C(=O)NCC(C)CN(C(=O)CN(C)CCO)C)c(C)n1 n1(CC(=O)NCCCN2CCCC2CCO)cc(C2(CO)CC2)nn1 C(=O)(C(F)C(C)C)N1CC(OCCC(=O)NC(C=C)CO)C1 N1(C(C(C(C)C)N(C)C)=O)CCOCC2(COCCN2C(c2ccoc2)=O)C1 c1(C(N2CCC(C)(NC(C(CC)OCC)=O)C2)=O)nc(C)n(C)c1C C1(NC(=O)C(F)C(F)(F)F)CN(C(c2cn3c(n2)CCCC3)=O)CC2(CC2)C1 C#CC1C(C(=O)N(C)CCOCCN(C)C(C2CCCO2)=O)C1(C)C N1(c2snc(CC)n2)CCN(C(c2c[nH]c3ccccc23)=O)CC(O)C1 CC(C)CC(F)(F)C(=O)NCCN(C(=O)Cc1ccc(C(F)(F)F)cc1)C(C)C c1(OC)c(F)ccc(F)c1C(=O)NCC(C)(C)NC(c1cn2cc(C)sc2n1)=O N1(C(C=Cc2c(C)nsc2)=O)CC2CC1CN2C(=O)Cc1ccc(C(F)F)cc1 CC1(C)COC(CC(=O)NCC2COC(CNC(=O)Cc3cnco3)C2)C1 c1(OC)ccc(Br)cc1C(=O)N(CC(C)NC(=O)C(n1cc(Cl)cn1)C)C C12(NC(COCC(=C)C)=O)CC1CN(C(c1ccnc(C3CC3)c1)=O)C2 CC(C)(CNC(c1cc(CNC(C2CC2Cl)=O)cs1)=O)CC(F)F N1(C(Cc2cn(C)nc2)=O)CC(NC(C2(CCO)CC2)=O)CC12CCC2 C1(C(=O)NCC(C(C)C)NC(=O)C(C(C)C)C(C)C)CCc2cnn(C)c2C1 C1(N(C(c2csc(Cl)c2)=O)CC)CCN(C(c2ccnc(CN(C)C)c2)=O)CC1 C(=O)(C1CCCc2c1ncn2C)NCCN(C(c1c(C)nc(CC2CC2)s1)=O)C CC1CNc2c(C(N3CCN(C(C4CC5(C4)CC(O)C5)=O)CC3)=O)cnn2C1 c1(OC(C)=O)cccc(C(N2CCC(NC(C34CC3CCC4(F)F)=O)C2)=O)c1C C(=O)(C(C)=Cn1ccnn1)NC(CC)CN(C)C(c1cncc(C(C)(C)C)c1)=O c1(C(N2CCCC2c2ccc(Br)s2)=O)noc(C(F)(F)CF)n1 CCCC(C(O)C(=O)NCCn1cncn1)NC(C1CN(C)C(=O)N1)=O C1(NC(C(CC)CC2CCCC2)=O)CCCC12CN(C(c1cc(F)n(C)n1)=O)C2 C1(CNC(CCNC(N)=O)=O)CCC2(CC1)CCN(C(C1CC=CCO1)=O)CC2 c1(CCN(C)C)cccc(C(N2CCC(F)(CNC(C3CCCCS3)=O)C2)=O)c1 c1(CN=C(NC2CCN(CC(F)(F)F)C2)NC2CCC2)cc2n(n1)CCO2 C1(C(=O)NCC(C)(C)OCC(N2CCOC(C#N)C2)=O)CC(=O)NC(=O)C1 C(=O)(CCCCC(C)C)NC1CCC(C(=O)NC(CCCC)C(C)O)C1 C(C(C(C)(C)C)NC(C1(C)CC(C)(C)C1)=O)NC(c1cnc(C)[nH]1)=O Cc1csc2c(N3CC4CC(NC(=O)CSCc5cccs5)CC4C3)ncnc12 C#CCC(CC(F)F)C(=O)N1CCCC(C(N2CCC(F)(C#N)C2)=O)C1 CC1(C)CCCN(C(=O)CNC=O)C1CNC(=O)CC1(C(F)(F)F)CC1 c1(NC(=O)NC(c2cc(Br)n(C)n2)C)cnc2ccc(Cl)cn12 c1(NC(C(c2cccs2)NC(C(CCOC)OC)=O)=O)cnc(C)c(C#N)c1 CC(C)C(O)C(=O)N1CCCCC1C1CCNCC1 C(=O)(CCCC(=O)N(CC(=O)NC1CN(C)CC1(C)C)C(C)C)OC OC1CCOC2(CCN(CC3CCC4(CCCOC4)O3)CC2)C1 C1(C(=O)NC2(CF)CCN(C(=O)C=C(Cl)Cl)C2)CCc2nncn2C1 c1(C(N2C(C)CCC2C(=O)NCC2CCS(=O)(=O)C2)=O)c(F)cc(Br)cc1Br C1(CNC(c2ccc(NC)s2)=O)CCC2(CCC2)C1NC(c1cccc(Cl)c1)=O c1(OC)ccc(C(=O)N(C2CCN(C(=O)C(F)(F)C(C)O)CC2)C)cc1C C1(C(=O)NCC2(C(N(C)Cc3scc(C)n3)=O)CC2)CC(C)CC(=O)N1 c1(CNC(C(C2CCN(C(C(CC#C)O)=O)C2)F)=O)ccc(O)c(C)c1 c12ccc(cc1)CN2.N1(C(C)=O)CCCC1COCCOC(C)C N1(C(C2CCC(C)(C)O2)=O)CCCCC(NC(c2ccc(C(N)=O)cn2)=O)C1 N1(Cc2c(Cl)nc(C)nc2Cl)CCC2C1CCCN2C(=O)Cc1ccc(Cl)cc1 c1(CNc2nccc(N(C)CC3(C)CCC(F)(F)C3)n2)ccc2cccnc2n1 C1(C)(C(N(C2CN(C(C(C)C(=O)OC(C)(C)C)=O)C2)C)=O)Cc2ccccc2N1 c1(C(=O)NC2CC(NC(c3cc(C)[nH]n3)=O)C2)n[nH]c(C(C)C)c1Br N1(C(Cc2ccc(C)nc2)=O)CCC(C2CC2)(CNC(C2CC(C)(F)C2)=O)C1 N1(C(C)C(=O)NC2CC(CNC(c3coc(Br)c3)=O)C2)CCCCCC1 C(=O)(C1CCCc2ccnn21)N(CCCNC(=NCCC)NC1CC1)C N1(C(Cc2nc(C)sc2)=O)CC2(C1)CN(C(C1CCc3nncn3C1)=O)CCO2 C12(CNC(COCC(C)C)=O)CC1CN(C(C1CCOC1C(F)(F)F)=O)C2 C1(CNC(c2cc(F)cs2)=O)COCCN(C(C2C=CCCC2)=O)C1 C(=O)(C(C)(C)C(C)(F)F)NC(COC)CC(=O)NC(C)C(=O)OC C(=O)(CC(C(C)OC)NC(c1cc2n(n1)CCC2)=O)NC(CC#C)CC c1(OC)ccc(C(=O)NCC(C2CCN(C(C3CCCCO3)=O)CC2)F)cc1F c1(C(N2CCC(CCNC(=O)COC3CCC3)C2)=O)ccc2c(n1)CCCC2 C1(C(=O)NC2(CC(=O)NCCC(C)(C)O)CCC2)CC2CCC2C1 c1(C(=O)NC2CCN(C(C=CCN(C)CC)=O)C2)ccc(NC)c(F)c1 c1(C(=O)NCC2CCC(N(C(C(=O)NCC)=O)C)CC2)cccc2c1OCO2 c1(N(C2CC2(F)F)CCO)ccc(F)cc1.N12CCCC(C1)NC(=O)CNC(=O)C2 CCC(C)CC(C)C(=O)NCc1c[nH]nc1C(=O)NCCC(C)(C)CC c1(C(N2CCCC(NC(C(C)(C)SC)=O)(CO)C2)=O)cccc2c1CC(=O)N2 C=C(Cl)C(C)(C)C(=O)NCC1(OC)CN(C(=O)CN2CCP(C)(=O)CC2)C1 CP1(=O)CCN(Cc2nc(-n3ccnc3)nn2-c2cccc(Cl)c2)CC1 N1(C(C)C)C(=O)CCC1C(=O)NCC1COCCN1C(=O)CN(C)C(N)=O C1(C(C)NC(=O)Cn2cnc(=N)[nH]2)CCN(C(=O)Cc2nnc(O)s2)C1 C1(CC)CN(C(=O)C(c2c(C)noc2C)C)CCN1C(c1cnc(OC)s1)=O c1(C(=O)NC2(CF)CCN(C(c3sccc3F)=O)C2)cnc2ncccc2c1 c1(C(=O)NCC(C)N(C)C(C2(CC(F)F)CCC2)=O)ccc(=N)[nH]c1Cl N1(C(C=Cc2ncc(C)[nH]2)=O)CCC(CNC(=O)CC=C(Cl)Cl)C(C)C1 c1(C(=O)NCCNC(c2cnn[nH]2)=O)ccc(S(=O)(=O)N2CCCCC2)cc1 C1(COC)CN(C(c2scc(C)c2C)=O)CCN1C(C1CC1C)=O Cn1ccc(C(=O)NCC2(O)CC(NC(C3CCC3(C)C)=O)C2)n1 c1(C(=O)NCC2OCC(CNC(c3cnsc3)=O)C2)sc([N+](=O)[O-])cc1Cl O=C(C(CO)c1ccccc1)NC1CCN(CCNc2cnn(C3CC3)n2)C1 c1(CNc2c(C(=O)NCc3c(O)cccc3O)c(F)ccc2)ccc(Br)c(F)c1F c1(C(C)NC(c2cncnc2)=O)cccc(C2CCN(Cc3cnn(C)c3)CC2)c1 N1(C2C(CN(c3ccc(SC)cc3)CCO)COCC2)CCC2NCCCC2C1 C(=O)(C(C)CCCOC)N(C(CC(=O)N(CCC)C)(C)C)C N1(C(c2nc(C)n(C)n2)=O)CC(C2CCCN(C(=O)C3=C(Cl)CCOC3)C2)C1 Cc1cc(NC(=O)CCc2ccccc2Br)cc(F)n1 S(=O)(=O)(c1ccc(S(=O)(=O)C(F)F)cc1)NC1C=CC(C(C)C)CC1 C1(C(=O)NCC2C3CN(C(CNC(=O)NC)=O)CC32)CCOC2(CCCC2)C1 N1C2CCC1CC(N(c1nnc(CC(C)C)s1)C)C2.C1(C=O)CCC(C)(C)OC1 c1(OCC)ccc(C(=O)NCc2ccsc2OC)c(OC)c1 N1(CC(=O)NC2C(CNC(=O)COC3CCSC3)COC2)CCCNC1=O CCC(CC)CCC(=O)N1CCC(CNC(C2CCCC3(CCC3)O2)=O)CC1 CCC(CC(F)(F)F)C(=O)N1CCCCC(NC(c2cc3c(s2)CCC3)=O)C1 N12CC(CC1(C)C)N(C)CC2=O.C12(NC(=O)COC3CCCC3)CCC(CC1)C2 N1(C(C=CC=CCC)=O)CCOC2(C1)CN(C(C1(C3CC3)CCCO1)=O)C2 C1(C)(C(=O)O)CCOC(C)C1.N1(CC=C)CCC(OC)C1=O Cc1nc2ncc(C(=O)NC(C)CC(C)NC(C3CCC=CCC3)=O)cc2o1 CP(C)(=O)CC(=O)NC1CCC(CC(N2CCCCC2CCO)=O)CC1 c1(C(=O)NC2CCN(C(C34C(C)OC(C)(C3)C4)=O)CC2F)ccnc2cnnn12 C12(CNC(C(N3C(C)CCC3C)C)=O)CC(CO1)N(C(=O)COC(F)F)C2 CC1CC=C(C(=O)NC2CCOCC2NC(=O)CCc2ccc(N)cn2)CC1 N1(c2c(C)cnc(C)n2)CCC2CCC(NC(C3(O)CCCC3)=O)C1C2 Cc1nc2c(C(=O)NC3CCCC3NC(c3c[nH]c(=N)cc3C)=O)cccc2o1 CC1=C(C(=O)NCC(O)CNC(=O)C=Cc2ncccc2C)C(=O)OC1(C)C N1(C(C(CC#C)O)=O)CCCC(O)(CNC(c2cc(Br)ncc2OC)=O)C1 N1(C(C)=O)CCN(C(C2(C)CCCN2Cc2ccc(OC(C)=O)cc2)=O)CC1(C)C CC1CCCCN1CC(=O)NCCOCCC(=O)NCC1CCCCC1C Nc1c(C(N2CCSCC2CCNC(=O)C(F)C2CC2)=O)cccc1[N+](=O)[O-] n1(CC)nc(C(=O)NC23CC(NC(c4ccc(CN=[N+]=[N-])o4)=O)(C2)C3)cc1C C1(CC(=O)N(CCC(C)O)C)CN(C(C2CC2C(F)F)=O)CC12CC2 C#Cc1cccc(C(=O)NC(C)(C)CCNC(=O)C(S(C)(=O)=O)C2CC2)c1 c1(CC(=O)N(C2CCN(C(C(CC)n3ccnc3)=O)C2)C)cnn(C)c1C(F)F N1(CC(C2C3CCCC23)=O)CCC(O)CC1.C1(CNC=O)CC(OC(F)F)C1 C(=O)(C1(C)CCOc2ccccc21)NCCCC(C)NC(CC(CC)(F)F)=O C(=O)(CC(C)C(F)F)NCC(CNC(CC(C)NC(N)=O)=O)O N1(C(C(=O)O)CCc2ccccc2)CCc2nnc(Cl)cc2C1 C(C1(O)CCCc2ccccc21)NCC(N)Cc1ccncc1 Cc1cc(C(=O)NCC(=C2CN(C(c3ccoc3C(F)(F)F)=O)C2)F)ccc1O C1(N(C)Cc2ccc(-n3cncn3)nc2)CCOC(C)(C)C1 c1(CNC(C2C(OC)CCC2)=O)ccc(CNC(=O)C2=C(Cl)CC2)c(F)c1 c1(CC(=O)NC(CN(C(C23CCC2C3)=O)CC)C)ccc2c(c1)OCO2 c1(NC(C(=O)NCc2c(C(=O)OC)con2)=O)cc(OC(F)F)cc(F)c1 C(=O)(C(CC(F)F)C1CCC1)NC(C1C(C(=O)Nc2c(SC)nn(C)c2)C1)C c1(-c2sc(C)c(C(=O)Nc3ccc(Br)c(C)n3)n2)cnc2ccoc2c1 n1(CC)nc(C)c(C(=O)NCC(COC)NC(=O)Cn2c(C)csc2=O)c1Cl c1(NC)cncc(C(=O)CN(C)C(C2CN(C(C)C)C2)=O)c1.C12CCN(C1)C2 c1(C(=O)NCCN(C(C2CCOCC2(C)C)=O)CC)nccc(N)c1Cl CC1(C)CN(C(C2COCCC2NC(=O)C(F)C2CCCC2)=O)CCO1 C(=O)(C1COc2ccc(F)cc21)N1CCC(NC(=O)C(F)=CCCF)C12CC2 C1(NC(CC=C)=O)CC(O)CN(C(c2cscc2C2CC2)=O)C1 C(CC(C)C)(C(=O)NC(C)CN1CCCC1)N(C(c1cc(C)[nH]c1)=O)C N1(c2ncc(C)cn2)CCCC2C1CCN2C(c1ccc2nc(O)sc2c1)=O N1(C(C2C=C(C)CS2)=O)CCCC(F)(CNC(c2n[nH]cc2C)=O)CC1 C1(O)(CNC(CC(CC)CC)=O)CCCN(C(=O)C#CC2(C)COC2)CC1 N1(C(C2N(C(C3CC(SC)C3)=O)CCOCC2)=O)CC(=O)NCC12CC2 C(=O)(C1CCCc2ccnn21)N1CCC(N(C(c2[nH]cc(CN(C)C)c2)=O)C)C1 N1(C(C2CN(CCOC)C(=O)C2)=O)CC(NC(=O)C=C(C)C2CC2)CC1(C)C C1(C(C)NC(N(C2CCCC2)Cc2cccc(C)c2)=O)CCC(F)(F)CC1 C1(CNC(CCOC)=O)CN(C(c2c(C)cc(O)cc2O)=O)CC(C)(C)C1 N1(C(c2cnc(CCCC)s2)=O)CCC(C2(NC(=O)CC(=O)NCC)CC2)C1 C(=O)(CN=c1cc[nH]cc1)NCC(C)N(C)C(C1CC1c1cn[nH]c1)=O c12sccc1S(=O)(=O)N2C.C(CCN(CCC#N)C)N(C(C)C1CC1)C Cc1c(NC(C2CCC(CNC(C3(CO)COC3)=O)O2)=O)cccc1CO c1(OCC(N2CCC(NC(c3cnc(C)[nH]3)=O)CC2)=O)ccc(F)c(F)c1 C1(NC(C2(C)N(C)CCC2)=O)C2CC1CN(C(=O)C=Cc1cccc(Br)c1)C2 Cc1cc(C(=O)NC2CC(NC(=O)C3=CCCOC3)C2)cnc1C(F)(F)F c1(C(=O)NC2C(C)CCN(C(c3cncn(C)c3=O)=O)C2)cnc2nccn2c1 C(=O)(C(C)CC(=O)N(C(C)CNC(=O)C(O)Cc1cnc[nH]1)C)OC CC1(C(=O)NCC2(C(F)F)CCN(C(c3ccncc3O)=O)C2)CCOCC1 C1(NC(c2c(OC)nccc2)=O)CC2CC(NC(c3[nH]nnc3C3CC3)=O)C2C1 c1(C(=O)NC(c2cn(Cc3cocn3)nn2)(C)C)ccccc1F Cc1ccc(Cl)c(C(=O)NCC2CC2CNC(c2cn(C)nc2C(F)F)=O)c1 N1(C(C=CC(C)=O)=O)CCN(C(=O)CCc2ccc(C)nc2)CC1CS(C)(=O)=O N1(C(c2ccc(C)cn2)=O)CCC(CO)C(NC(=O)C(C)(C)c2cccnc2)C1 Cc1ccc(C(C)(C)C(=O)NCC(C)NC(C2CCC(C)(C)CC2)=O)c(C)c1 C12CCC(CC1)C(=O)OCC2=O.Cc1cc(C(=O)N(C)C)n[nH]1 Cn1cc(C#N)cc1C(N1CC(NC(=O)C(F)=C2CCCC2)C2(CC2)C1)=O CC1(F)CN(C(=O)CC2(O)CCCCC2)CCN(C(c2cncc(O)c2)=O)C1 C1(C(=O)NCC=CCNC(C(C)(C)OCC(F)(F)F)=O)CC2COCCN2C1 Cc1ccc2cc(C(=O)NC3CC(C)N(C(=O)CCC(C)C)CC3C)ccc2c1 C1(CNC(C(C)Oc2ccc(F)cc2)=O)CC2CCC(C1)N2c1ncccn1 c1(C(=O)NCC(C2CCCN2C(C2(OC)CC2)=O)(C)C)ccnc(NC(N)=O)c1 N1(CCNC(c2c(C)cc(C)s2)=O)CCCN(C(C2CC2CN(C)C)=O)CC1 C1(NC(CSCCN(CC)CC)=O)CCN(C(=O)CCS(C)=O)CC1F c1(C(=O)NC2CC(F)(CNC(C3(Cc4cnn[nH]4)CCC3)=O)C2)ccnc(Cl)c1F CC1=C(C(=O)N(CCC(C(C)(C)C)NC(C2C(C)C2C)=O)C)C(C)(C)CCC1 N1(C(C=CCOC)=O)C2CCC1C(CNC(=O)CC(c1ccc(F)c(F)c1)C)C2 N1(C(C2(CNC(CCSCC)=O)CCC2)=O)CCCC2C1CCN2C C1(OC)CCC2(C(N3CCN(CCNC(=O)C(C)N(C)C)CC3)=O)CC12 c1(C(N(C(C)CNC(=O)C(N2CCCCC2)C)C)=O)cccc(F)c1F c1(NCCCC(=O)NCC2(NC(CNC(C)=O)=O)CC2)ccccc1OC(F)F CN1CCCCC1C1CC(C(c2cnnn2C)NC(=O)NC2CC2)C(O)C1 c1(CN(C(c2ccc(SC)cc2)C(=O)NCCOC)C)cc2c(Cl)nccc2o1 N1(C(c2c(C)nncc2)=O)C2CCCC1CN(C(C1CCCC(CF)C1)=O)C2 CC1(C)CC(CNC(c2cnsn2)=O)CN(C(=O)CCC2CC2(F)F)C1 c1(C2(C(=O)NC(C3CN(C(CC(=O)NCC#C)=O)C3)C)CC2)ccc(F)cc1C C1(NC(CN(c2ccc(Cl)cn2)C)=O)CC2CC1N(C(=O)C=C1CCSCC1)C2 N1(C(C2C(CC)C2(F)F)=O)CC2C(CNC(=O)C(C)(C)C3CCCCC3)C2C1 c1(CN2CCCC(CC(N3CCCC3c3ccco3)=O)C2)ccc(O)cc1F C(C)(N=c1[nH]c(=NC)[nH]c(=NC(C)c2cnsc2)[nH]1)c1n(CC)ccn1 C(CN=c1[nH]c(=NC2CC(C(C)C)C2)c2sccc2[nH]1)N(CCC)CCC(F)F Cc1c(O)ccc(C(=O)Nc2nnc(-c3cccnc3)s2)c1C C=CC(C)(O)CC(=O)NC(CCCC)C(=O)NCC1OCC2CCC1C2 C(C(COC)CC(=O)N1CCC(CN(C(=O)C=Cc2cncn2C)C)C1)OC c1(C(N(CC(CN(C(CC)=O)C)O)C)=O)cnn(CC2CC2)c1 C1(CC(=O)NC2CCCC2CN(C)C(C2CNC(=O)C2)=O)(CC)CCOCC1 Cc1cc(Cl)ccc1CC(N1CC(C)(NC(C2CCOC2C)=O)C1)=O N1(CC)CCCC(C(=O)N(C)CCNC(=O)CC2CCCC(C)O2)C1 C(CC1CC1)(CC(=O)N(C1CCCCC1O)C1CC1)NC(CCC=C)=O C1(C)(CNC(c2c(C)nn[nH]2)=O)CC(F)(F)CN1C(c1ccc2n[nH]cc2c1)=O N1(C(C2(SC)CCC2)=O)CC2(CCC(NC(C3CCCC3C)=O)CC2)C1 c1(C(N2C(C)COC(CO)C2)=O)cn2c(n1)CCN(Cc1ccc(Cl)s1)CC2 c1(C(=O)NC2(CC)CCCN(C(C(CC)CO)=O)C2)cnn2c1CCCC2 c1(C(N(CC2CCN(C(C=CCCC)=O)CC2)CC)=O)ccc([N+](=O)[O-])cc1 C(=O)(C(C)C(C)(F)F)NCCCN(C(c1c(OC)c(C)sc1)=O)CCO N1(CC)N=C(C(=O)N2CC(NC(c3cnn(CCF)c3)=O)C3(CC3)C2)CCC1=O C(=O)(C(O)CC(F)(F)F)N1C(CNC(CCCC(=O)OC(C)(C)C)=O)COCC1 c1(C(N2CCC(C)(NC(CC(CCC)C)=O)C2)=O)cc(F)c(F)c(F)c1F c1(CN(C(c2ccncc2)=O)Cc2ccccc2Cl)cccc2ccccc12 c1(C(N2CC(CC)N(C(=O)C=CCOC)CC2)=O)cnc2ccnn2c1C c1(C(C)(C)C)ccnc(C(=O)NCc2ncc(C(F)(F)F)cn2)c1 C(N=c1nc2c(ncn2C)c(NCc2cc(Br)ccc2F)[nH]1)C1CCN(C)NCC1 CCCCC(CC)CC(=O)N1CCN(C(C2CC(C)(F)C2)=O)CC12CCC2 C(=O)(C1=Cc2ccccc2C1O)N1CCN(C(CC(C)CF)=O)C(C)C1 C12(NC(CCSCC)=O)CCN(C(c3ccnc(OC)c3Br)=O)CC1C2 N1(C(=O)C(F)F)CCCC2(CCN(C(=O)C(C3CCCCC3)c3cccs3)C2)C1 C12(C(N3CCC(SC)C3)=O)CCC(CC1)N(C(C1CC13CCCC3)=O)C2 C1(CCC)CN(C(=O)CCC2CCC(=O)C2)CC1C(N1CC(CCC)C1)=O n1(CC(=O)N(C2CCC2)C)cnc2scc(-c3cccnc3)c2c1=O N1(C(C(C)OCCC(C)C)=O)CCOCC(NC(C2COCCN2C)=O)C1 C(=O)(CC(=O)N1CC(C(C(=O)NCC(F)Cl)OC)C1)OC C1(NC(=O)CC2CCC(F)(F)CO2)COC2(C1)CN(C(=O)CC1(O)CCC1)C2 C#CC1CCN(C(=O)CCC2CCCCN2C(C2CCCC(=O)N2)=O)CC1 C1(C2CN(C(c3cnn(CC)c3C3CC3)=O)C2)(NC(C(CC#C)C)=O)CC1 c1(C(=O)NC(CNC(C2(OC)CC2)=O)CC(C)C)nc(Cl)ccc1N N1(C(c2c(C)ccnc2O)=O)CC(N=c2ccnc(C(C)(C)C)[nH]2)C2(CCC2)C1 C1(C(N2CCN(C(C=C(COC)C)=O)CC(O)C2)=O)CCC2(CCOCC2)CO1 N1(C(COC(CC)C)=O)CCCC1C1CCN(C(=O)C(C2CCCCC2)O)C1 C12(C(=O)N)CC1Cc1c[nH]nc12.C(CCCC(=O)NCCNC(C(N)=O)=O)N N1(C(C(CO)NC(C(C)C)=O)=O)CC2CCCN(C(=O)CN(C)C(C)C)C2C1 C1(C(N2CC(CCNC(COCc3n(C)ncn3)=O)C2)=O)CS(=O)(=O)CC(=O)N1 C(=O)(C1=CCCSC1)NC1(CC=C)CCN(C(c2cnc(C)n2C)=O)C1 c1(C(N2C(CNC(C3(CC#C)CCCCC3)=O)CCC2)=O)cc(C)cc(Cl)c1N C1(NC(C(C)NC(C)=O)=O)CCCC(C(=O)Nc2ccc(CO)c(F)c2)CC1 Cc1ccc(C(N2CCC(CNC(c3ccc(C(F)(F)F)s3)=O)C2)=O)nc1 c1(CC=C)ccc(C(=O)NCC(C)N(C)C(C2CC(C)(O)C2)=O)cc1 C1(C(=O)NCC(C)(C)CNC(C2(c3ccccc3)CC2)=O)CC2CCC(C1)C2O C1(CCC(=O)NC2(C(C)N(C)C)CC2)CCN(C(=O)CC2CC(F)(F)C2)C1 C(CCC1CC1)(C(=O)N1CCN(CC2CC2)CC1)NC(c1ccnc(Cl)c1)=O CC(C)CCCC(C)C(=O)N(C)CC1COCCN1C(=O)CCc1ccc[nH]1 c1(C(N2C(C)C3CC2C3NC(c2ccccc2)=O)=O)ccc2n[nH]cc2n1 C(=O)(C1=CSCS1)NC(CNC(CCCc1onc(C)n1)=O)C1CC1 C1(CNC(=O)Cn2cc(CO)nn2)CCCCCN1C(C1CC=CC1)=O C1(NC(C2N(C(CCSC)=O)CC(F)C2)=O)CCCC2CCCCC12 C1(NC(C(n2c(C)ncc2)C)=O)CC2(C1)CC2C(=O)N(C1CCC1)C1CCC1 C1(NC(CCOCCOC)=O)CC1C1CCCN(C(C2(CC#N)COC2)=O)C1 c1(C(=O)NCC2(NC(C=CCCC)=O)CCC2)c(Cl)cc(C(F)F)cc1Cl Cc1cc(C(N2CCC(NC(c3c(F)cccc3Cl)=O)C(F)C2)=O)ccc1O c1(C(=O)NCC(C2CC2)NC(C(C=CC)O)=O)ncc(N)nc1C C1(NC(COCCC#C)=O)CN(C(=O)CCC(=O)c2ccc(CC)cc2)C2CC12 C1(NC(CCc2ncc(C)[nH]2)=O)CCCCC12CCN(C(=O)C(Cl)=CCl)CC2 CC(=Cn1ccnn1)C(=O)NCC(C)CNC(C1CCC=CO1)=O c1(OC(C)C)cccc2cc(NC(c3nnnn3C)c3ccsn3)oc12 c1(-c2c(C)ccs2)ccc2cc(C(=O)Nc3sccc3C)sc2c1 c1(-c2ccc(NC(C(=C)C(F)(F)F)=O)c(F)c2)ccc([N+](=O)[O-])cc1[N+](=O)[O-] CC(CCN(CC(c1cccs1)C)C)CC(=O)O N1(C(=O)NCCc2cc(OC)c(O)cc2)CC2CN(C)CC2C1 C#CC1CN(C(C2CCN(C(=O)CCCCC)C23CC3)=O)CC1OC Cc1nc(-c2cn(C3COCC3NC(C3(CN(C)C)CCC3)=O)nn2)ccc1F N1(C(CC2C(C)(C)OCCO2)=O)CC2CCC(C1)C(NC(=O)Cc1cnc[nH]1)C2 C12(NC(=O)CC(O)c3ccccc3)CC1CN(C(=O)COCCO)C2 n1(CC)cc([N+](=O)[O-])c(C(=O)NC2CC3CC(NC(C4CC=CCC4)=O)C3C2)n1 CCCCCCCCC(=O)NC(c1ccccc1)C(N1CCCC(CO)(CO)C1)=O C1(C(N(CC(C)N(C(=O)Cc2ccno2)C)C)=O)CC(F)C(=O)N1 C1(CC(=O)N(CCCNC(=O)CCNC(N)=O)CC)CCC(=O)C1 Cc1c(CN2CCOC(C(=O)Nc3ncncc3Cl)C2)cnn1C c1(SCC=C)ccccc1C(=O)N(C(C)CN(C)C(c1csnn1)=O)C c1(C(=O)NC2CC(CNC(C3CC(C)=C(C)CC3)=O)C2)cc2cncn2c(O)n1 c1(C(=O)NC2CC(O)(CNC(C(C)C3CCC3)=O)C2)ccc2c(c1)CCC(=O)N2 Cc1cc(C)n2ncc(C(N3CC4(CCN4C(=O)CCCC4CC4)C3)=O)c2n1 c1(C(N2CCC(N(C(CCc3cncc(C)c3)=O)C)C2)=O)cc(F)c(C)cc1Cl C1(CNC(CN2CC(=O)N(C)C2=O)=O)CC2CCC1N(C(c1sccc1F)=O)C2 C1(N(C(c2c(CC)ncs2)=O)C)CCCCN(C(=O)CNC=O)C1 N1(C(C2C(C)(CC)C2)=O)CCCC12CCN(C(=O)CNC(C)=O)CC2 C(=O)(C(O)CC(C)(C)C)NCCC(C)N(C)C(C1CC(C(F)(F)F)C1)=O C(N=c1cc(Cl)c(O)n[nH]1)C1CN(C(CCCCOC)=O)CC1(C)C C1(NC(CCC)=O)CC2CN(C(C3CCCCN3N=O)=O)CC2C1 c1(C(N2CCCC(CC)(NC(=O)CC3(CO)CC3)C2)=O)cc(S(N)(=O)=O)cn1C C12(NC(=O)C3=CCOC3)CCCC1CN(C(c1cnc3[nH]cncc1-3)=O)C2 CN1CCC(CC(=O)N(C)Cc2ccccc2CNC(C2SCCCS2)=O)CC1 C1(C)(C(N(C2(C(N(CCCC)C3CC3)=O)CC2)C)=O)CC(C)=NO1 C1(NC(CCC(=O)OC)=O)CN(C(c2cnn(CCF)c2)=O)C2(CCCOC2)C1 C#Cc1ccc(C(=O)NC(C)CN(C(=O)C(C)n2cnnn2)CC)c(F)c1 C1(C(=O)NCCOCCCC)CCCCC1NC(C1CC(=O)OC1(C)C)=O C1(NC(c2cccc(CC)c2)=O)CCN(C(=O)CCCCSC)CC1OC N1(C(CC=C)=O)CC2CCC2(CCNC(c2nscc2Br)=O)C1 C1(OC)CC(NC(c2ccc(F)s2)=O)C12CCN(C(=O)C(F)=C(C)C)CC2 N1(C(C(COC)OC)=O)CC2CCN(C(c3c[nH]nc3F)=O)CC12 CC1c2c[nH]nc2CCC1C(=O)N(CC(O)CNC(=O)C=C1CCOCC1)C C(=O)(C(C)CC(C)(C)C)NC1C(NC(C2(CC=C)CC=CC2)=O)CS(=O)(=O)C1 c1(C(=O)NC(CCCC)CC)nccc2n[nH]cc12 c1(CN2C(C(=O)Nc3cccc(C(=O)OC)n3)CC(F)C2)cc(F)c(Cl)c(Cl)c1 CC1(C#CC(=O)NC2(CNC(=O)C3=CCCSC3)CCCC2)CC1 CC1CC2CN(C(=O)C(O)C3CCC3)CC2N1C(C1CC1C(N)=O)=O N1(C(C2CC(=O)OC2)=O)CCC(n2cc(CCOCC(F)(F)F)nn2)CC1 c1(OC)ccc(C(N2CC(NC(c3cnnn3C3CC3)=O)CC2(C)C)=O)c(C)c1 CN1CCC(O)C(NC(=O)C(Cn2cncn2)NC(c2n[nH]c(O)n2)=O)C1 c1(C(=O)NC2(C)CCN(C(=O)CC3CCCCC3)C2)ccc(S(C)(=O)=O)s1 C1(C(C(=O)NC2CC(C)(NC(C)=O)C2)OC)CCC(F)(F)CC1 C(CCCCC(=O)NCC(C)N(C)C(C1(C)CCCC1(F)F)=O)OCC N1(C(C(C(C)C)CN(C)C)=O)CCC2C(CCCN2C(=O)CS(=O)(=O)C(C)C)C1 C(=O)(CCC(=O)NN(C)C)NC1(COC)CN(C(C2(n3nccn3)CC2)=O)C1 c1(CC)ccc(OC)cc1C(=O)NC1CCC1CNC(c1ccc(C)cc1N)=O c1(NC(C2C(C(=O)Nc3ccc(F)c(F)c3F)C2)=O)ncc([N+](=O)[O-])cc1I C(=O)(C1CCCc2ccnn21)NC1CCN(C(C(CC)N(C)C)=O)CC1 c1(C(N2CC(C(N3CCCC(C(=O)NC)C3)=O)(CCl)C2)=O)cccc2cc[nH]c12 N1(c2ccc(C)cc2C)N=C(C(=O)NC2CC(C)(C(N)=O)C2)CCC1=O n1(CC(N2CC(C)OCC2)=O)ccc(=NCc2cc([N+](=O)[O-])ccc2Cl)nc1O C12(C(=O)NC3CN(C(CC(c4ccc(Cl)cc4)N(C)C)=O)C3)CC(C1)S(=O)(=O)C2 N1(C(c2n(C)ccc2)=O)CCCC(CNC(C2CN(C3COC3)C2)=O)C1 C1(CCC(=O)NCCC(O)CCC2N(CC(=O)N(C)C)CCC2)CCCCCC1 C1(C(=O)NC2CCC(N(C(=O)CCCc3csc(=N)[nH]3)C)C2)CCC=CO1 C1(CNC(CCCN(C)C)=O)CN(C(=O)C(F)(F)C(C)(C)O)CC2(CCC2)O1 C1(CCCNC(=O)NCS(C)(=O)=O)CCN(CC2(CC=C)CCOC2)CC1 N1(C(CCC2CC(C)C2)=O)CCC2(CCCN(C(C3CCC(F)C3)=O)C2)CC1 N1(C(C2C3CN(C(=O)C=CCN4CCC4)CC32)=O)CC2(CO)CCC1CC2 C(=O)(C=CS(=O)(=O)CC)N1C(CCNC(CC(CC)C)=O)CSCC1 C1(N(C)C(c2cn(CC(N)=O)nn2)=O)CCCC(NC(=O)CNC=O)C1 C1(SCc2onc(C(C)C)n2)CCCCN1C(=O)CSC(C)C C12(CNC(=O)Nc3nc(C4CC4)cs3)CC(C(=O)NC3CC3)(CO1)C2 c1(C(N2CC(NC(c3cccnc3S)=O)C2)=O)cccc(=S)n1O N#Cc1cnc(NC(N)=O)c(Cl)c1.C12CCCN(C1)CC1N(CCC1)C2=O N1(C(c2c(C)nn[nH]2)=O)CCC(CF)(NC(=O)CC2CC3CCC2O3)C1 N#Cc1ccc(Cl)c(CN2CCN(C(=O)CCc3ccc(O)cc3)C3CC23)c1 C(C)(CCC#N)(c1nnnn1CCC1CCC1)CCOC.C1(C)(C)C(C)N1 O(NC(=O)CCN(C(=O)C(c1ccnn1C)O)C(C)C)C(CC)CC c1(C(=O)NCC2(OC)CN(C(=O)CCc3nnc(S)n3C)C2)cc(C)c(F)cn1 C=CC(C)C(C)C(=O)N(CC)CC1(O)CN(C(=O)CCCCCc2ccccc2)C1 N1(C(C2CC23CCCC3)=O)CCN(C(=O)CCc2cnc(C3CC3)o2)C(CF)C1 N1(C(C2OCCN(CC)C2)=O)CC2CC1CN(C(=O)CC1CCCO1)C2 O=C1CCC2(C(=O)NCC3(O)CN(C(C4CC=CCC4)=O)C3)CCCC2C1 C(=O)(C(O)CCNC(=O)CCOCC1CCC1)N(CC)Cc1ccncc1 Cn1nnc2cccc(C(N3CCN(C(=O)C(O)C4CCC4)C(C4CC4)C3)=O)c12 c1(C(=O)OC)cnc(N2CC(CNC(c3nc(C)oc3C)=O)CC2C)c(Cl)c1 C(CCCCCCC)N(C(c1cc(C2CC2)[nH]n1)C(=O)NCCOCC)CC1CC1 C(=O)(C1CCCn2cnnc21)NC1CC(O)(CNC(c2c[nH]cc(C)c2=O)=O)C1 C1(C(N2C(CC(C)C)CC2)=O)N(C(c2ncc(F)cc2N)=O)CC12CCCC2 c1(NC(C2COCCN(CC=CC(=O)O)C2)=O)ccc2c(c1)OCCO2 c1(C(=O)NC2CN(C(C(CCC#C)O)=O)CC2SC)cc(Cl)cc2ccncc12 c1(C(C(=O)NC(C)C)N(CC=C)C(C)C)ccn(C)c1 C(=O)(C1=CCCCC1F)N1C2C(C(N(CC(F)(F)F)CC)=O)C(C2)C1 c1(CC)ccc(C(N2CCC(C#N)(NC(=O)CCOC)C2)=O)c(Cl)n1 C(=O)(C(C)(C)CN(C)C)N(CCN(C)C(C1CC2COCC12)=O)C1CC1 c1(CC)cc(C(=O)NC2CCC2NC(c2ncccc2Cl)=O)ccc1Cl c1(CN(C(=O)C(=O)Nc2ccc3c[nH]nc3c2)C)nnc2n1CCNC2=O c1(C(=O)NC2(C)CC(NC(=O)Cc3ccco3)C2)ccccc1CO CC1CCCC(NC(=O)CN2CCC(CNC(=O)COCCCF)CC2)C1 c1(C(=O)NC2CCC(NCc3cccc(OC)n3)C2)ccc(C(F)F)nc1C c1(C(=O)NCCC(C)N(C(=O)CCCCC(N)=O)C)ccc2[nH]ccc(=O)c2c1 C(=O)(C1CCCc2ncc(C)n21)NC1(CCCNC(C(S(CCC)(=O)=O)C)=O)CC1 C(Cn1ccnn1)(C(=O)NCC(CO)OC)NC(C1(CCCC)CC1)=O CC1CN(C2CC2)CC1(c1nnnn1CC(F)F)Nc1cccc(Cl)c1 c1(OC)ccc(C(=O)NCCCCNC(=O)CC2CCC2(C)C)nc1 n1(CC(=O)NCCCN(C(=O)C(F)OC(F)(F)F)CCO)cc(Cl)c(O)nc1=O N1(C(c2c(C)nco2)=O)CC(F)(F)CC1(C)CNC(C1CN2CCCC2CO1)=O C#CCC(C(=O)NCc1nonc1C)NC(C1COCC1(C)C)=O C1(C)(NC(C2CC(=C)C2)=O)CCCN(C(C2CC(CC(F)(F)F)C2)=O)C1 c1(C(=O)NCC(=O)NC(C(CO)NC(C(CC)O)=O)C)ccccc1C C1(NC(C2CCC(C)C2)=O)CN(C(c2cccnc2S)=O)C2(CCOCC2)C1 c1(C(N(C2CN(C(C3(n4ccc(C5CC5)n4)CC3)=O)C2)C)=O)ccccn1 N1(C(CN2CC(=O)NCC2)=O)CCC2C(C(=O)NCCCN3CCCC3=O)C2C1 c1(C(=O)NC2CCN(C(CC(C=C)C)=O)CC2(C)C)cc2c(s1)CCC(C)(C)C2 C1(C(=O)NC2CC(OCC)C2)CCN(C(=O)COc2ccc(F)c(C)c2)C(C)C1 N1(C(c2c(C)nn(CC)c2C)=O)C(CNC(c2ccc(F)o2)=O)CC2COCC12 C1(C(N2CCC(CC=C)(NC(=O)CC(C)(C)C#N)C2)=O)Cc2c(C)cccc2O1 c1(OCC)ccc(NC(C2CN(C)CC(C)O2)=O)c2c1C(=O)N(CC)C2=O c1(CC)c(CSc2nnc(-c3ccn(C)n3)n2C2CC2)cccc1Cl c1(C(C)=O)cc(C(=O)NCC(=O)NCCc2cccnc2)n[nH]1 CCCCCCN(C(=O)C(C1CCC1)OC)CCN(C(C1CC1(F)F)=O)CC CC(C)(C(=O)NC1C(OC(F)(F)F)C1(C)C)Nc1ccccc1 c1(C(=O)NC2(CC(=O)NC3CCN(CC)C3)CC2)cccc(C#N)c1C N1(C(C2CCN(C(c3c(N)non3)=O)C2)=O)CCCC2(CC(O)C2)C1 C#Cc1ccc(C(=O)NC(C)(CNC(c2cccn3nncc23)=O)CO)cc1C Cc1[nH]cc(C(=O)NC2CC2NC(=O)Cc2c(Cl)cccc2Cl)c(=O)c1Cl C1(C(N(CC(C(C)C)C)C)=O)CN(C(c2cc(CO)[nH]n2)=O)CCC1(C)C C12(CC(=O)NCc3c(CNC(CCCC#C)=O)cccc3)CNC(=O)C(C1)C2 O=C(C1CCCc2ccnn21)NCCC1CCN(C(C2CSCCS2)=O)CC1 C1(C(=O)NCCC(COC)O)CCC(CNC(c2cnn(C)c2N)=O)CC1 N1(C(c2[nH]c(=N)sc2C(F)(F)F)=O)CCCC(NC(c2cocn2)=O)C(F)C1 N1(C(c2ncoc2CNC(C2(CO)CC2)=O)=O)CCCC2(CC2)C1 N1(C(C(CC)F)=O)CC2CC1(CNC(C1CC1c1cccc(OC)c1)=O)C2 C(=O)(C(CC)C(C)(C)CC)NCc1cn(CC(=O)NC2CC(N(C)CC)C2)nn1 CC1(C)C(C(N2CCC(O)CC2)=O)CCN1C(=O)CCOC1COC1 N1(C(CCN(C(CCC)C)C)=O)CCN(C(=O)CC2(C)CCCC2)CC1C(C)C c1(C(=O)NC(CC#CC)C)cccc2sc(C(=O)OCC)cc12 c1(OC)cccc(C(=O)NCC(C2CCC2)NC(c2cc(CO)n(C)n2)=O)c1C Cn1cncc1CCC(=O)N(CCCNC(=O)CCc1ccon1)C1CC1 N1(C(c2c(NC)cccc2)=O)CCC(O)C(C(=O)NCCC2CC(O)C2)C1 c1(C(N(CC(C)(C)NC(=O)CN(S(C)(=O)=O)C)C)=O)cc2c(cn1)OCO2 c1(NC(C2C(C(=O)NCCCCCO)C2)=O)cncc2c(F)cccc12 c1(OC)c(C(=O)NCC(CO)NC(=O)CC(C)(F)F)csc1C C(C(C)(C)C(=O)NOCCCN(C)C)N(C(=O)CN1CCCNC1=O)C O=C(C1CCCc2sccc21)NCCC1CSCCN1C(C1CCCOC1)=O O=C(CC1=CCN(C(c2ccc[n+]([O-])c2)=O)CC1)N1CCC1CF N#Cc1c(Cl)nc[nH]c1=NC1CC2CCC1N(C(C1CCCC1)=O)C2 CC(C)CC(C(=O)NC(CO)C(O)c1ccccn1)NC(c1ccc[n+]([O-])c1)=O C1(CNC(c2c(C)scc2)=O)CCC2(CN(C(C3CCCC4(CCC4)O3)=O)C2)O1 C12(CSCCNC(c3cn(CCO)nn3)=O)CCC(CO)(CC1)OC2 c1(C(=O)NC2C(NC(C(C)OC3COC3)=O)C2)csc(Cl)c1Cl c1(C(=O)NCC2(C)CC(NC(C(CCC)OC)=O)C2)ccc2oc(C)nc2c1 C1(Cc2cn(CC)nc2)CCN(N(C)C(C2CCC2CC(C)C)=O)CC1 c1(C(=O)NC2CCCC(NC(C(CC)O)=O)C2)cc2ccccn2c1 C1(NC(C=NOC)=O)CCN(C(=O)Cc2ccccc2NC(=O)C2CC2)C(C)C1 c1(C(=O)NC2C(CC)N(C(=O)CNS(=O)(=O)NC)CC2)nn(C)c(Cl)c1Cl N1(C(CN(C)C)=O)CC2CCCC2(NC(c2ccc(N(C)C)nn2)=O)C1 C1(C(N(C2CC(O)C2)C)=O)(COc2ccccc2)CC2(CC2)C1 C1(CNC(CCc2cncc(C)c2)=O)COCCC1(F)F.C12C3CN(CC13)C2=O c1(CC)cc(NC(=O)C(C(C)C)NC(=O)CCCC2(OC)CCC2)ccc1C N1(C(c2c(CC)oc(C)c2)=O)CCCC(NC(=O)CN2CCS(=O)(=O)CC2)C1C c1(OC)cc(C(=O)NCC(C)(C)CC2CN(C(c3ccc(CO)o3)=O)C2)ncn1 c1(C(=O)NCC2CN(C(=O)Cn3nccn3)CCO2)ncc2ccccc2c1O c1(CC)nnc(CNC(=O)CC(C)NC(=O)CC(C)OC)s1 N1(CCN=C(NCC(C)OC)NCC(=O)NCCCl)C(=O)c2ccccc2C1=O c1(C(N2CCC(NC(Cc3nc(C)sc3)=O)CC2C)=O)cccc2c[nH]nc12 C1(O)(CNC(c2cscn2)=O)CCCN(Cc2nc[nH]c2[N+](=O)[O-])C1 C1(C(C)(C)C)C(NC(=O)C=Cc2ccco2)CCN1C(c1ccc(C(F)F)o1)=O C(=O)(C(C)(C)CC(=O)N1CCC(N(C(=O)Cc2cccc(Cl)n2)C)C1)OC c1(C(=O)NC2CC(CO)N(C(c3ccnc(C4CC4)n3)=O)C2)cn2c(n1)SCC2 C1(C(=O)NCC2(NC(c3cc(C)no3)=O)CCCCC2C)CCCCN(C)C1=O N1(C(C2=CCCN(C(CSC(C)(C)C)=O)C2)=O)CCCC2(CC=CCO2)CC1 Cc1nc2ncnn2cc1C(=O)NC1CCC(NC(=O)C(C)n2ccnc2)CC1 N1(C(C)=O)CCC(OC(=O)NCCNC(COCC(=C)C)=O)C1 C(C)(C(=O)NOCC(C)CC)N(C(c1cc(CC)[nH]n1)=O)C1CC1 O=C1NC(C(=O)NC2CCCC2NC(c2occc2Cl)=O)Cc2ccccc21 c1(CCNC(=O)OC(C)(C)C)ncc(Br)c(N(C)C(C2CC2F)=O)n1 C1(CNC(Cc2ccc(C)cc2)=O)CCN(C(c2cc(O)cc(=O)o2)=O)CC1C C1(NC(C2C(=C)C2)=O)CC2(C1)CC(C(=O)N(C(C)COC)C)C2 N(C(=NCCC(O)C(F)(F)F)NCC(F)F)Cc1c(O)ccc(Cl)c1 C(CC(C(=O)N1CC(C)(OCC)C1)NC(c1c[nH]c(C#N)c1)=O)=CC C1(NC(CCc2cnc(C)o2)=O)CC2(C1)CC2NC(=O)CN1CCN(C)CC1 CC1(C)CC(C(=O)NC2CC2NC(=O)C=C2CCC2)CNC1=O S(=O)(=O)(c1cccs1)N(CC(=O)NCC1CC(NC(C2CCC2(C)C)=O)CC1O)C FC(F)(F)C(F)(F)CCn1cc(CCCOC2CCOCC2)nn1 Cc1nc(=N)[nH]cc1C(=O)NCC(C)CNC(c1nnn(C)c1C(F)(F)F)=O C1(C=O)CCC(C)CN1C(=O)C(C)S(C)(=O)=O.C1(COC)CCCNC1 Cc1cc(C(C)(C)CNC(C2CCC(n3cccc3)CC2)=O)n(C)n1 c1(OCC)cc(C)c(CN2CC(F)(F)CC2C(=O)NCC2CC2)cc1OC N1(C(C2=CCC(C)CC2)=O)CCC(C2(NC(=O)C(C)c3ccco3)CCC2)CC1 C1(OCC)CCC(NC(C2(NC(=O)C(C)(CC3CCC3)C3CCC3)CC2)=O)CC1 c1(N2CCN(C(=O)C(C)S(C)(=O)=O)CC2)nc(C)cc(=NCCOCC(C)=O)[nH]1 CC(O)CCCCCC(=O)NCc1cn(C2CCN(C(C3(O)COC3)=O)C2)nn1 C1(C(=O)NCC2CC(O)CN2C(=O)CN2CC3CC3C2)Cc2nccn2C1 N1(Cc2ccc(C)s2)CC2CC1CN2C(C1CCC(C(=O)OC)CC1)=O C(=O)(C1Cc2ccc(Cl)cc21)N1CC(NC(C=CC=CC)=O)CC1(CC)CC C#CCCCC(C)C(=O)N1CC(C)(C(=O)NC(C)CCc2ccccc2)C1 C(=O)(C1=CCCN(C(c2ccc(C(F)F)o2)=O)C1)NCC1CC[Si](C)(C)C1 C1(NC(C=C(CCC)C)=O)CN(C(=O)CCCn2ccnc2)CC1(C)C CC(C)CS(=O)(=O)CC(=O)N(CCCCNC(C12CC(C1)C(C)O2)=O)C c1(CC)cc(CC)[nH]c(=NCC(C)(C)CNC(c2nncs2)=O)n1 Cc1ccc(CNC(=O)N(C)Cc2ccccc2)cc1S(C)(=O)=O C12(CCOCC1)C(C=CC(=O)OCC)NC2=O.c1(C(=O)OCC)ncc(C)[nH]1 CON1CC(C(N2CCC2C(N2CCCC2C2CCOC2)=O)=O)CC1=O Cc1cc(C(=O)NCCC2CC(NC(=O)CN3CCC(C)C3)C2)cc2ccoc12 Cc1cc(C(N2CCN(C)C(CNC(=O)CN3CCCCC3=O)C2)=O)nc(O)n1 C1(C(=O)NC(C2CCCCC2)CNC(c2ccc(C)nn2)=O)CCn2nncc2C1 CN1CCN(CC(=O)NC2CCCCN(C(=O)CN(C)CCO)C2)CC1=O N1(C(CC)C(N)=O)CCCC(C2(NC(c3cnco3)=O)CC2)C1 c1(-n2ncc(NC(C(C)SC3CCCCO3)=O)c2)ccc(OC(F)F)cc1 C1(NC(CSCCC)=O)CCC(C)(CNC(c2cn(CC(N)=O)nn2)=O)C1 N1(C(c2cc(CC)ncn2)=O)CCCCCC(NC(C2CN(C3CCC3)C2)=O)C1 c1(C(N(C2CCCC2)CCCNC(CC(CC)C)=O)=O)cccc2c1CCCC2 C1(C#N)(C(=O)NC2C(C(=O)NCC=C(C)C)OCC2)CCCOC1 C(=O)(CCCF)NC1CC(CNC(C(C)NC(N)=O)=O)C1.C(C(F)(F)F)N c1(C(C)=O)ccc(C(N2CCC(O)(CCNC(=O)Cc3nccn3C)C2)=O)nn1 C(CCc1ccccc1)(C(C)NC(=O)CNc1ccc(Cl)cc1)NC(CCC)=O c1(C(C)(F)F)cccc(C(=O)NCCCNC(C2CC3CCC2C3)=O)c1 c1(CC(=O)NC2CC(NCc3ccc(Cl)nc3)C2)cc(O)nnc1O C(C(C)(C)C(=O)N1CC(CCNC(=O)Cc2ncoc2C)C1)SC c1(CNC(C2C(C(=O)NC(CC)C)CNC2)=O)ccccc1CS(=O)(=O)N(C)C C1(CC(=O)NCCN(N2CCCC2)C)CC(C)N1C(C=CC(=O)N)=O.C(C)=O C1(C)(C(N2CCC(C)(CC)C2)=O)CN(C(c2ccc(NC)cc2)=O)C(C)(C)C1 Cc1nccc(=NC(C)(CCc2nnn(C)n2)c2nnnn2Cc2ccco2)[nH]1 N1(C(CC(CC)OC)=O)CC(NC(c2ccnnc2C)=O)CC12CCC2 C1(CCNC(c2c(C)nco2)=O)COCCN1C(=O)C(C)CN(C)C c1(OC)ccc(C)cc1CC(=O)NC(CNC(C1(C)CCCS1(=O)=O)=O)C(C)C c1(OC)cccc(CO)c1C(=O)NCC1CC(C)N(C(=O)CC2CC3(CC3)C2)C1 CCC(C)(Br)C(=O)N(c1cn(-c2ccc(F)cc2)nc1C)CC(=O)OC c1(OCCC(=O)NCC(C)CNC(=O)CO)ccc(F)cc1F N1(C(CC(C)=C(C)C)=O)CCC(C2(NC(c3cc(C)cc(O)n3)=O)CCC2)CC1 N1(C(CC2N(C)CCC2)=O)CCC2(C1)CN(C(c1cc3ccsc3s1)=O)CCO2 N1(C(=O)Cc2ccccc2Nc2cnn(C3CCOCC3)c2)CC2CC2(O)C1 Cc1nc(C)n(Cc2cn(C3CC(C(=O)NCCSC4COC(=O)N4)C3)nn2)n1 C#CC1(C(N2CCC(NC(=O)C(C)=CC)C(C)C2)=O)CCCCC1 CC1(F)COCCN(C(=O)CCC2CCCN(C(=O)C=Cc3ccccc3)C2)C1 O=C1CC2C(NC(C3CC(CNC(=O)CN4CCOCC4)C3)=O)CC2O1 N1(C(C(CCC)N(C)C)=O)CCC2(C1)CN(C(c1occ(C)c1C)=O)CC(C)O2 C(c1ccccc1)=CC(C(=O)NC1(CNC(C(C2CCOC2)OC)=O)CC1)C c1(CN(C(C(=O)NCC2CCCO2)c2ccoc2)C)cccc2ccccc12 C1(CC)CC1N=c1[nH]c(=NCC(C(F)(F)F)Sc2ccccc2)[nH]c2ncn(C)c12 C(=O)(C1=COCCO1)N1CCC(N(C(c2ccc(C(=O)OC)[nH]2)=O)C)CC1 C1(C(=O)NC2CCN(C(C(C(C)C)(C)C)=O)C(C)C2)CN(S(=O)(=O)N(C)C)C1 C1(NC2(c3n(CC(F)F)nnn3)COCCOC2)CCC2COCCC2O1 c1(OC)ccc(C(N2CC(NC(=O)CCn3ccccc3=O)C(C)C2)=O)cc1O c1(CCC(=O)NC2CC(C)(CNC(c3cnc(SC)s3)=O)C2)cncnc1O c1(C(C(=O)NC2C3CN(C(c4c(C)cc(C)o4)=O)CC32)C)c(C)nn(C)c1C c1(OC)ccc(CC(=O)NC2CC(C)N(C(c3cc(C)n(C)c3)=O)C2)cc1Cl N1(C(C(CCC)N(C)C)=O)C2CCC1CC(C(=O)NCCCCCN=[N+]=[N-])C2 C=CC(C)N=c1cc(C)[nH]c(=NCCc2c[nH]c3ccc(OCC(C)C)cc23)[nH]1 C1(O)(C(=O)NC(c2nc(C(=O)NCc3ccsc3)co2)C)CC(CF)C1 c1(CC(=O)NCCC(CC)(C)NC(=O)CCc2cnoc2)cc(C)cc(C)c1 N1(C(C2C(SC)CN(C(=O)C(CN(C)C)N(C)C)C2)=O)CC(C)(C)CC1CO N1(C(c2c(C)nsc2C)=O)CC2CCC(C1)N2C(C1CCC2(CCC2)CO1)=O c1(CC)oc(C)cc1C(=O)NCc1ccc(C(N2CCCC(C(C)O)C2)=O)o1 C(CC(F)(F)F)SCC(=O)N.C(C(CC)CC)N(C(CC=C)=O)CC S(=O)(=O)(c1ccc(Br)cc1F)N1C2CCCN(C(C(CC)NC)=O)C2CC1 N1(C(c2c(CC)c(C)sc2)=O)CC(CO)C2(C1)CN(C(=O)CCOCC(C)C)C2 N1(C(CCC(=O)NCCC)=O)CC(CNC(=O)CNC(=O)C2CC2)OC(C)(C)C1 N1(C(C(CC)NC(C)=O)=O)CCC(CCOC)(NC(C2CC2(C)C(=O)OC)=O)CC1 C(CC(N)=O)(C(=O)NCC(C)N(C)C(c1cncc(C2CC2(F)F)c1)=O)OC C(=O)(CS(C)(=O)=O)NCC(CNC(c1nc(C)oc1)=O)CO C1(C#CC(=O)NCC2CCC2NC(=O)CC(c2ccccc2OC)C)(CC)CC1 S(=O)(=O)(c1ccc(Br)cc1N(C)CC1(OC)CCC1)N1CCC(CC)C1 Cc1c(C(N2CC(O)(C(C)(C)CNC(C3CN(C)C(=O)N3)=O)C2)=O)ccn1C(C)C C1(O)(CCNC(C(COC)(F)F)=O)CCN(C(c2snnc2C2CC2)=O)CC1 C(=O)(C(O)CC(C)(C)C)N1C2C(NC(c3ncc(OCC)nc3)=O)C(CC2)C1 c1(C(=O)NC(CN(C(C(C(=O)OCC)F)=O)C)C)ccc(-c2cccs2)nc1C CC1=C(C(=O)NC2CCN(C(=O)CC(C)C(F)F)CC2)COCC1 N1(C(c2cnc(C3CCC3)s2)C(=O)NCCC)c2ccccc2CC1C1CC1 C(C)(CC(C)N=c1[nH]nc(-c2ccon2)s1)NC(C(CCSC)O)=O N1(C(CN(C(C(C)C)=O)C)=O)CCC(C(O)CNC(C2CCCCN2C)=O)CC1 CC1CC(NC(=O)C=CC(N)=O)CCN1C(c1ccc(F)cc1Cl)=O N1(C(c2c(C)n(C)nc2)=O)CC2(C(N3CCCCCC3CO)=O)CC1CO2 C1(CNC(c2ccc(CC(C)C)cc2)=O)CCN(C(=O)CC#N)C12CC2 C1(NC(CN(C(=O)OC(C)(C)C)CC2CC2)=O)CCOC12CCOC2 c1(CC(N2CCC(NC(CNC(C)=O)=O)C2)=O)c(C)[nH]c2ccccc12 c1(-c2c(OC)ccnc2)cccc(CN2CCN(C(=O)OC)C(C)C2)c1F C1(C(=O)OC)(COC)CCNC1=O.C1(C(C)C)CCC(=O)N1 C1(NC(C2C(=C)C2)=O)CCN(C(c2csc(=NCC)[nH]2)=O)CC1C C1(C(=O)NC(C(C)NC(c2ccn(C)c2)=O)CO)COC(C)(C)CO1 C1(CNC(Cn2c(C)c(Br)cn2)=O)CC(C(C)(C)C)CCN1C(C1CC1C)=O C(=O)(C1CCc2cccc(F)c21)NC1CN(C(CCCNC(=O)CO)=O)C1 N1(C(C2N(CC)CCOC2)=O)Cc2[nH]nc(C(=O)N(C)Cc3csnc3C)c2C1 C1(C(=O)NC(c2cccs2)CC)CN(C(c2cc(F)ccc2F)=O)CCC1(C)C C1(C(=O)NCCCCC2CCN(C(C(C)C3CCC3)=O)CC2)CNC(=O)CC1C C1(=CC(=O)NCC(C)N(C(C2CCC(C)CC2)=O)CC)CC2CCC(C1)N2C CCCCCCCCCC(=O)NC1CCN(C(c2ncc(Br)cc2Cl)=O)C1 C(C(O)CC(F)(F)F)NC(C1=C(SC)CC1)=O.OC c1(C(=O)NC(c2cc(S(=O)(=O)NCC)oc2C)=O)ccc2c(c1)NC(=O)CS2 N1(C(CCC(C)N(C)C)=O)CC2CCOC2(CNC(C2CCCCC2)=O)C1 Cc1cc(C(=O)N(c2nnc(C)o2)C(C)(C)C)ncc1-c1cnc(N(C)C)nc1 c1(C(c2nnc(NC(=O)C(C(N)=O)c3cccc(Br)c3)s2)C)ccccc1S(C)=O c1(C(N2CCCC(CN(C(Cn3c(C)ccn3)=O)C)C2)=O)cc2sccc2cn1 c1(OC)ccc(CC(=O)N(CCCNC(c2ccsn2)=O)C2CC2)c(C)c1 C=C(CNC(=O)C(C)(C1CCC1)NC(=O)CC=CCC)C(F)(F)F C1(N(C(CCSC)C(=O)N2CCCC2)C)CCCC(F)(F)C1O C1(C(=O)NC2C(C(=O)NC3(C)CCSC3)OCC2)CC(=O)C1(C)C C1(C(=O)NCc2ccc(OC)nc2)CCCN1NC(=O)C1=NOC(C)(C)C1 c1(CC(=O)NCC2CCN(CC)CC2)c(Br)nc2n1CCOC2 N1(C(C=C(C)CC2CCCCC2)=O)CC(Nc2nnc(C)o2)CC2(CC2)C1 c1(C(N(CCCCNC(C2CCCC23CC3)=O)C)=O)cnc2ccc(F)cn12 C(=O)(CCCc1cccs1)N1CC(CC(C)NC(=O)C=C2CCC2)C1 Cc1nc(CC(C)C)c(C(=O)NCCCCNC(=O)COc2ccc(O)cc2)s1 C1(CNC(CC=C)=O)CN(C(c2c[nH]cc2Br)=O)CCC12CCC2 N1(C(C(=O)Nc2ccc(S(=O)(=O)NCC(=O)O)s2)=O)CCCN(CC#C)CC1 N1(C(C(C)N(C)C)=O)CC2(CCCN(C(C3CCn4nncc4C3)=O)C2)C1 C1(NC(N(CC(C)Cn2ccnc2)CC)=O)CCCC1 c1(C(N(CC(CNC(CCOC(C)C)=O)O)C)=O)cc2ccccc2nn1 C(C)(C)(CCCCC(=O)N1CCC(NC(C2(CC3CC3)CCC2)=O)CC1)OC N1(C(C=COCC)=O)C2CCC1CN(C(=O)C(C)CCc1ccc(F)cc1)CC2 C12(CNC(=O)CSCC(F)F)CCN(CC1)CC2.C12(CCCC1)C(=O)N2 N1(C(C2(C=C)CC2)=O)CCCOC(CCNC(c2cc(C(C)C)ccc2O)=O)C1 Cc1c(C(=O)NC23CC(NC(=O)COCC4CCOC4)(C2)C3)cccc1Br C(=O)(CCCNC(=O)OC(C)(C)C)N(C(C)CCF)C1CC1 N1(C(=O)NC2C(C)(CC)C2)CCC2(C=CCO2)C1 N1(C(c2ccc(C(N)=O)o2)=O)CCCCC1CCNC(=O)CCc1cncs1 c1(CNCc2cc(C)c(OC)c(C)c2)cc(Br)cc(F)c1F Cc1cc(=O)cc(CN2CC(C)(CCC(=O)NCC3CC4CCCC4C3)C2)[nH]1 c1(C(=O)NCC2CCN(C(C(CCOC)C)=O)C2)cc(Cl)cc(C)c1N c1(C(C)C)ncc2c(n1)CC1CCC2N1C(=O)CCc1cc2ccccc2[nH]1 Cc1cc(C=CC(=O)NCC(C)NC(c2nccn2C)=O)ccc1Br N1(C(c2ncn(CC)n2)=O)CCCC1(C)C(N1CCCC1(C)C(N)=O)=O N1(C(C2N(C)CCC2)=O)C2CCC1CC(NC(=O)CNC(c1cccnc1)=O)C2 c1(NCCC2CCN(C(C(CC)N(CC)CC)=O)CC2)cc(C)nc2cnnn12 N1(C(C2CC3(CC(=C)C3)C2)=O)CCC2(C1)CN(C(c1cccnc1CC)=O)C2 C(=O)(C(CC)NC(=O)Cn1[nH]cnc1=N)NCC1(OCC)CCC1 C1(NC(C2=C(C)OCCS2)=O)CCC2(CC1)CN(C(=O)CC1OCCO1)CCO2 c1(NCC)ccccc1C(=O)NC1CC(CNC(C2CCNC2=O)=O)CC1O c1(-c2cn(CC(C)NC(c3c(CC)cco3)=O)nn2)ccc(OC)cc1OC N1(CC(=O)OCC)CCN(C=O)CC1.C1(=O)CCCN1.c1(SCC)c[nH]nc1N c1(CC(=O)NC(C2(O)CN(C(c3coc(C4CC4)n3)=O)C2)C)nc(C2CC2)n[nH]1 CP(C)(=O)CNc1cccc(C(N2CC(NC(=O)Cn3cncn3)C(F)C2)=O)c1 c1(C(=O)NCc2c(CC)nn(C)c2)cc(C)nc2ccc(OC)cc12 CC1COCCC1N(C)C(C1(C)C=CCN1C(=O)Cc1cn[nH]c1)=O C1(NC(C2CN(CC)C(=O)C2)=O)CCCCN(c2nc(C(=O)OC)ns2)C1 C1(OC)Cc2nccnc2C1.C1(C)COCCC1.n12cc(nn1)C(=O)NCC2.C1(=O)CCN1.NC c1(OC)c(NC(=O)Cc2cc(NC(=O)OC(C)(C)C)cc(F)c2)cccc1F c1(C(N2CCN(CC(C)(C)NC(C3(C)CCCO3)=O)CC2)=O)cc2ncccc2s1 N1(C(C(C)OCCOC)=O)CC(C)(C)CCC1CNC(c1nc(C)nn1C)=O N1(C(C2CC(O)(CC#C)C2)=O)CC(NC(C2CN(C)CC(C)O2)=O)C2CCCC12 Cn1nc(C(=O)NCC(C)(CO)NC(C23CCC(C2)C3)=O)c(=O)c2ccccc12 c1(C(N2CCC(N(C)C(C3CCC(C4CC4)O3)=O)C2)=O)cc([N+](=O)[O-])cnc1N N1(C(c2c(CC)c(OC)ccc2)=O)CCC(COC(=O)C(C)C)C(F)(F)C1 Cc1ccc(C)c(S(=O)(=O)N2CC3CN(Cc4ccc(F)cc4[N+](=O)[O-])C3C2)c1 C1(C(N2CCC(CN(C(c3c(C)ccnc3)=O)C)C2)=O)OC2CCC1CC2 N1(C(C(F)OC)=O)CC(CNC(C2CCCOC2)=O)OC(C)(C)C1 C1(C(N2CCCC(CCC=C)C2)=O)CN(C(=O)CCc2ccc[nH]2)CC1(C)C N1(C(COCCC(C)C)=O)CCOCC1CNC(c1cnccc1C(F)(F)F)=O c1(C(N(CC(CNC(C23C(C)OC(C)(C2)C3)=O)O)C)=O)cc2c(s1)CCCCC2 Cc1ccc(C(=O)NC2CCN(C(=O)CCn3ncn(C)c3=O)CC2)c(F)c1 N1(C(c2cnc(C3CC3)s2)=O)CCC2(CCC2)C(CNC(C2(C(F)F)CC2)=O)C1 Cc1ccc(Cl)c(C(N2CCCCCC(NC(c3cc(O)ncn3)=O)C2)=O)c1O c1(CCC(N2CCC(C)(NC(CC3C(C)C3)=O)C2)=O)ccc2c(c1)OCO2 C=CC1(NC(C2C3CN(C(C4CN(C5CCC5)C4)=O)CC23)=O)CCCC1 C(=O)(C1=Cc2cc(Cl)ccc2OC1)NC1CN(C(C(CC)(CC)CC)=O)CC1C c1(C(=O)NC2C(CO)CCN(C(CCCCC#C)=O)C2)c(O)cc(Cl)cc1Cl N1(C(C2CCC(N(C)C)CC2)=O)CC(NC(C2(F)CCOC2)=O)CC(F)C1 Cn1nc(CC(=O)OCc2ccccc2F)c2ccccc12 Cc1nc(C2CC2)sc1CC(=O)N(CC(C)O)CCNC(C1CC2CC2C1)=O CC1=NOC(CC(N2CC(O)(C(C)NC(=O)CCc3cnn(C)c3)C2)=O)C1 c1(NC(c2snc(CC)n2)=O)c(-c2cn(C3CCOC3)nn2)cnn1C c1(C(=O)NCCC(CCNC(C(C=C)(F)F)=O)C)c(C)cccc1N C(=O)(C1OCCc2ccccc21)N1CCN(CCNC(CC(CC)(C)C)=O)CC1 n1(CCNC2CCN(C(C=CC(N3CCCC3)=O)=O)C2)ccc2ccccc12 Cc1cnc(C(=O)NC2CCC(NC(c3ccc(CO)o3)=O)CC2)cc1Cl c1(C(=O)Nc2cc(O)ccc2Cl)cc2n(c1)CCNC2 Cc1cc2sc(C(=O)NCC3CN(C(=O)CCCc4ncco4)CCO3)cc2s1 N1(C(C2CC(=C)C2)=O)CCN(C(C2(C)CCN(C(C)=O)CC2)=O)C(C2CCC2)C1 c1(OC)ccc(CC(=O)NC2CC(CNC(c3sc(C)cc3C)=O)C2)c(Cl)c1 CC(CC1CCC1)C(=O)N(CC(N1CCC1CF)=O)C1CCC1 N1(C(C2(NC(c3cc(C)sn3)=O)CCCC2C)=O)CCCCC(F)(F)C1 C1(NC(CSS(C)(=O)=O)=O)CCN(C(=O)C=Cc2ccccc2Cl)CCC1CO C1(C(=O)Nc2c(CC)n(C)nc2)C2CC(F)C(C2)N1C(c1cnsn1)=O c1(OC)cc(C(=O)NC2(CNC(=O)Cn3cc(C(C)O)nn3)CC2)cc(F)c1F C(c1ccc(F)c(C)c1)=CC(N1C(C)CC(NC(C(CC=C)CC)=O)C1)=O N1(C(c2c(F)ccc(C#C)c2)=O)CCCC(C2CN(C(=O)CC3CN(C)C3)C2)C1 Cc1nnc(CN(C)C(C2CC(C)N2C(=O)Cc2cncn2C)=O)o1 c1(C(=O)NC2C(NC(=O)CCC3CCCC3)C2)cc2c(nn1)CCC2 N1(C(c2c(C)ccc(C)c2)=O)CC2CC(NC(=O)C(C)(C)N(C)C)C(C2)C1 c1(NCC2C(C(F)(F)F)CN(C(C(COC)(C)O)=O)C2)nc(C)ccc1C#N C(=O)(C(F)C(C)CNC(c1c(C)cnn1C)=O)N(CCCC)CCO N1(C(c2n(CCC)ncc2)=O)CC(CNC(C2CC(CCO)C2)=O)CC(C)(C)C1 C1(NC(Cc2cc(=N)[nH]cc2)=O)CC2CC(C1)N(C(c1ccc(Cl)c(F)c1)=O)C2 C(CCCCC(=O)NC(C)CCC(=O)NO)NC(c1n[nH]c(C)c1C(=O)O)=O C1(CNC(N2CC(C)(Cc3nc(-c4ccco4)n[nH]3)C2)=O)CC(=O)NC(=O)C1 C1(NC(C2CC(C)C(=O)CC2)=O)CN(C(=O)CCCCO)CC2(CCC2)C1 c1(OC)cc(Br)c(CN2CC3CN(C(c4cc(C)cc(O)c4)=O)CC23)cc1O C(=O)(C1=COCC1)NC(C1CN(C(c2csc(-c3cccc(Br)c3)n2)=O)C1)C CCC(=O)N1CC(n2ccnn2)CO1.C(C(CC)CC)c1ccc(C)cc1 c1(OCC)ccc(NC(=O)C(=O)NCC23CCC(CC2)C3)c2ccccc12 c1(C(N(CC(CNC(C=Cc2c(C)ccs2)=O)C)C)=O)c(F)ccc2ccoc12 CC1(C)CCC(CC(=O)NC2CCN(c3ncc(Br)cn3)C2)C1 c1(NC(C2N(C(c3c(SC)nccc3)=O)CC2)=O)cc(F)cc(F)c1Cl c1(OCCCN(CCC)C(C2CC23CCOC3)=O)ccc(F)cc1 C1(C(N2CC(CNC(c3cc4ccsc4[nH]3)=O)OCC2)=O)CCCC2CCCN12 C1(NC(C(C)OCC(F)(F)F)=O)CC12CCN(C(=O)CS(N)(=O)=O)CC2 C12(NC(C(C)NC(CC)=O)=O)CCCC1(F)CN(C(c1c[nH]cc1CC)=O)C2 N1(C(c2cc(CCC)[nH]n2)=O)CCCCC(C(=O)NC(C)(CC)CO)C1 c1(C(=O)NCC(CO)NC(C2(C)CN(C)C(=O)C2)=O)nc2ccccc2[nH]1 CCCC(CC)CCC(=O)N1CC=C(C(=O)NCC2CSCCO2)C1 C(CC1CCC1)(C(=O)NCC(C)N(C(=O)COC(C)(C)C)C)NC(C)=O c1(C(=O)NCC2(F)CCN(C(Cc3c(C)cnn3C)=O)C2)cc(S(C)(=O)=O)cs1 C12(CNC(Cc3nc(C)sc3)=O)CCC(CC1)N2C(c1cc(C2CC2)nn1C)=O Cc1cc(F)cc(C)c1C(=O)N(CCC(C)NC(c1cn(C)nc1C(F)F)=O)C Cn1nnc2c(C(N3CCCC(NC(c4cc(N)cc(O)c4)=O)C3)=O)ccnc12 c1(OC)cc(C(=O)OCc2nc(C(=O)O)cc(C(F)F)n2)cc(CN)c1 c1(NC(C(C2CC2)SC)=O)ccc(CNC(=O)C(C)SCC2CCCC2)c(F)c1 c1(CN(CCCNC(c2ccc(C)s2)=O)C(C)=O)ccc(F)cc1 Cc1nc(=N)[nH]cc1C(N1CCC(CNC(c2sccc2C)=O)C(C)C1)=O c1(C(N2CC3C(NC(c4ccc(C)cc4N)=O)C3C2)=O)cnc(O)n(C)c1=O c1(CN(C(C)CF)C)nc2cc(Br)ccc2o1 C(=O)(C(O)CCS(C)=O)NCCN(C(CC(C)C(F)F)=O)C N#Cc1cnc(CNC(=O)NC2CCCC(C(=O)Nc3ccccc3)C2)o1 N1(C(c2c(F)cc(C)c(F)c2)=O)CCOC2(CCCN(C(C3CC(C)C3)=O)C2)C1 Cc1ccc(F)c(CNC(C2C3CN(C(c4cccc(N(C)C)n4)=O)CC23)=O)c1 c1(C(=O)NCc2cn(C)nc2)cc(C2CC2)nn1C.C1(C(=O)N)(CNC(=O)C2CC2)CC1 C1(NC(=O)NC(c2nc3c(s2)CCCC3)C)CCCCC12CCC2 c1(C(c2nnnn2C(C)(C)C)NCCCNC(C)=O)cc2ccccc2nc1C c1(C(=O)NC(C)CCCNC(c2ccn(C)n2)=O)nnc(O)c2ccccc12 C(=O)(CC(F)(F)C(C)C)NCCCC(C)NC(C(CC(=C)C)C)=O N1(C(c2c(COC)cc[nH]2)=O)CCCC1C1CCCN1C(=O)CCCC#N Cc1cc(C(N2CC(O)(C(C)NC(=O)C(C)(C)CF)C2)=O)cnn1 Cc1cnc(C(=O)NC(Cc2cn(Cc3ccccn3)nn2)CC(=O)O)c(C)c1 C12(CNC(=O)Cc3cnns3)CC(CCO1)N(C(c1ccc(O)cn1)=O)C2 N(C1CCc2ccccc21)C(C(C1(C)CC1)NC(C1C(C(C)(F)F)C1)=O)=O N1(C(c2ccc(SC)s2)=O)CCCC(C)C1CNC(c1ccc(C(F)F)cn1)=O c1(C(=O)NC2CCN(C(C3(CCOC)CCCC3)=O)C2)c[nH]c2cc(F)ccc12 Cn1cc(S(=O)(=O)N2CCC(CO)(NC(c3ccc(Br)c(C#N)c3)=O)CC2)cn1 N1(C(C(C=C)(C)C)=O)CCC2(CC1)CC(NC(=O)CC(C)C)C2 C1(CC=C)(NC(c2cnc(NC(C)=O)o2)=O)CCN(C(c2cccc(Cl)c2)=O)C1 c1(C(=O)NC(c2cccc(Cl)c2)CNC(C(CC)F)=O)oc(CC(C)C)nc1C N1(C(c2c(N(C)C)nccc2)=O)CCC2C(CCCN2C(C2CCOC2=O)=O)C1 C(=O)(N=c1[nH]nc(N(C)C)o1)N1CCCC(Cn2cc(C(CC)OC)nn2)CC1 c1(C(=O)NC(CC(C)C)CNC(C2C3CCN2CC3)=O)cccc(F)c1Br c1(C(N2CC(O)(CC=CCNC(C3C(C)(CC)C3)=O)C2)=O)c(C)nc(=N)[nH]c1C S(=O)(=O)(c1c(C)noc1C)N1C(CC(N2C(CCCC)CCC2)=O)CCCC1 Cc1noc2ncc(C(=O)NCC3CCN(C(c4ccn(C)c4)=O)CC3)cc12 N1(C(c2c(OC)cncn2)=O)CCC(C(=O)NC2(C)CC=CC2)C12CC2 N1(C(c2ccc(CNC(C(CSC)O)=O)s2)=O)CCC(F)(F)CC1 C=CCCCC(C)NC(C1CCOCC1NC(c1cc(OCC)no1)=O)=O C1(C)(C(N(CCC)C(C)C)=O)CCN(C(=O)Cc2ccc(C)o2)C1 C(=O)(C(C#N)(CC)CC)NCC(CCCC)NC(=O)C=NOC C1(C(=O)OC)CN(C(=O)CNC(c2sccc2C2CC2)=O)CC1(F)F c1(CC)nc(C)n(C)c1C(=O)NC1CC1NC(=O)CCP(C)(C)=O Cc1ccc(Br)c(CNCc2c(C)nc(C)n2O)n1 C1(C)(C(=O)NCC2(O)CN(C(C(c3ccc(C)cc3)=O)=O)C2)CCC(O)CC1 Cc1cccn2c(CC(=O)NCC3CCCN(C(C4CCCSS4)=O)C3)cnc12 C1(NC(CN(C2CCC2)C)=O)CCC(CNC(=O)Cc2ncsc2Cl)CC1 C1(CC(=O)NCC(CC)C)C(C(=O)Nc2ccccc2)CC1O CC1(C)CC(C(=O)NCc2cocn2)N(C(=O)CC2CCC(F)(F)C2)C1 C1(NC(CCC2CCC(NC(=O)CC3COCCO3)C2)=O)CCCCCC1F C1(CC(=O)NC2(C(=O)NC3CCOCC3)CC(F)C2)CC2C=CC1C2 CON(C(=O)C1CCC(C2CC2)N1C(=O)C(=O)N(C)C)C(C)C O=C(C1=NOC2(CCC2)C1)NCC1CN(C(=O)C=Cc2ccccc2F)CC1O C(=O)(C(CC(N)=O)NC(C12CCCCC1C2)=O)NCCc1onc(C)n1 C1(C(=O)NC(C=C)CO)(NC(=O)CC(C)C2CC2)CC(F)C1 CC1(C)CN(C(c2sc(C#N)cc2Cl)=O)CCC1NC(=O)C=C1CCSCC1 N1(C(CCCCCNC(N)=O)=O)CCC2(CNC(C3CCOC3)=O)CCCCC12 C1(N(C)C(C2CCS(=O)(=O)N2)=O)CCCCN(C(=O)C(c2cccnc2F)(C)C)C1 C12CCC(O1)C(=O)N1CC(C)(C1)NC(=O)CC2.C1(C)(CC)CC(C(=O)OC)C1 C(CN=c1nc(N2CCCC(CCN(C)C)C2)c2ncccc2[nH]1)C1C(F)(F)C1 c1(OCC)ccc(-n2nc(C3CSC3)nc2Cn2ccnn2)cc1Cl c1(C(C(=O)NCc2ccc(Cl)s2)NC(CSCC)=O)c(C)cccc1Br CC1CN(C(=O)COCC2CCC2)CC1CC(N1CC(C#N)(CCF)C1)=O c1(NC(CN2CCC(N(CCC)C(C)=O)C2)=O)ncc(Br)c(Cl)n1 N1(C(CCCOCC)=O)CCC(N2CCCC2C(N2CCC(CO)C2)=O)CC1 c1(C(=O)NCCC(C)C)ccc(C2CCCN(C(=O)Cc3ccc(Cl)s3)C2)cc1 n1(CC(=O)NCCC(C)N(C)C(c2snc(O)c2Cl)=O)c(O)nc2ccccc12 C1(C(N2CCC(Cc3ccoc3)C2)=O)(NC(C2CC2[N+](=O)[O-])=O)CCCC1 C1(CC)CN(S(=O)(=O)CCCS(=O)(=O)NC)c2cc(CC)ccc2NC1=O CC(CCC(=O)NCCNC(C1CCc2nccn2C1)=O)S(C)(=O)=O N12CCOC(C1)C2=O.C(C(C)S(C)(=O)=O)N(C(c1nc(CCC)oc1)=O)CC c1(C(=O)NC2CC(C)N(C(=O)CCS(C)(=O)=O)CC2)cc(S(N)(=O)=O)co1 Cc1cn(C)nc1C(N1CCN(CC(=O)N(C2CCCC(C)C2)C)CC1)=O N1(C(Cc2nc(C)sc2Br)=O)CCC(NC(=O)Cn2cnnc2O)CC1C C1(CC)CN(C(=O)CN(C)C(C)C)CCN1C(C1CC2CC2N1C(C)=O)=O Cc1c(C(=O)N(CCNC(c2nn[nH]c2Cl)=O)C2CC2)nn(C)c1N c1(CCCC(=O)N(C)CC2(O)CN(C(C(CN(C)C)O)=O)C2)cc(F)ccc1F N1(C(CCC#CC)=O)CCCC(C2CCCN(C(=O)Cc3nc(C)sc3Cl)C2)C1 CCCCCCC(C)C(=O)N1CC(CNC(c2cc(COC)[nH]n2)=O)C(O)C1 C12(C(=O)NC(c3ncccn3)CC)COCC1CN(C(c1ccc(Cl)o1)=O)C2 c1(C(=O)NC2(CN(C(C3(CCC)CC3)=O)C)CC2)cc2cccc(Cl)c2nc1C C1(c2n(CC)nnn2)(Nc2cnn(CC)c2)CCCC(C(F)(F)F)C1 C1(C(N(CC(CC)NC(c2csc(CO)n2)=O)CC)=O)CC2CC1C2 C1(NC(C2(CC)CCN(C(Cc3ncc(CC)[nH]3)=O)C2)=O)CCN(CC)C(C)C1 C1(=O)C(C(C)(C)C)OC(=O)CC2CCN1C2.N1CCC(CCOC)CC1.OC C(c1cnccn1)=CC(=O)NCC(N(C(=O)CCCn1ccnc1)C)C1CC1 c1(C(N2C(CNC(c3c(COC)noc3)=O)CCC2)=O)ccc(OC(C)C)nc1 N1(C(c2cnc(OCC)nc2)=O)CCCC(O)(CCNC(c2nn[nH]c2Cl)=O)C1 O(C1CCCc2ccccc21)CC(=O)NC(C)CNC(C1(C(F)F)CCCC1)=O c1(C(C(=O)OC)N(C(=O)CNC=O)C(C)=O)ccccc1CSC CCCCCCCCCC(=O)NC1CCN(Cc2cccnc2OC)CC1O C(=O)(CCCC(=O)NC1CC2CC(C1)N(C(C13CCCC1C3(F)F)=O)C2)OC C1(NC(C=CC)=O)CC(C2CCN(C(=O)CCS(=O)(=O)Cc3ccncc3)C2)C1 C1(CC)CN2CCC1C2=O.c1(C2(NC3CC=CC3)CC2)ccccc1.C1(=O)CN1 c1(C(N2C3CC(CC(NC(CCCCC=C)=O)C3)C2)=O)cccc2c1CCCC2 CC(C)(C)CC(C)(C)C(=O)NCC1CC2CCC1N2C(=O)Cn1cnnn1 C1(C(N2CC3(CCCC3)C2c2ccccc2)=O)CCC2(CCNCC2)CC1 c1(NC(c2cscn2)C)ccc(S(=O)(=O)NCC2(C)OCCCO2)c(Cl)c1 N1(C(C2CC(O)(CC#C)C2)=O)CC(NC(=O)C(C)C#N)CC12CCCCCC2 Cc1cc(C(=O)NC23CC(C(=O)NCCCSC(F)F)(C2)C3)cc(F)c1 N1(C(C=CC=CC)=O)CCC2(CC1)COC(CNC(C13CCC(CO1)C3)=O)C2 N12CCCC3(CCN(CC3)Cc3cccc(c3)C1)C2.c1(CC)c(O)cccc1Br C(C)(C(C)(C)C(=O)NC1CCCC1)NC(C(C(C)C)=O)=O CC1=C(C(=O)N2CCN(C(c3ccc(OC(F)F)c(Cl)c3)=O)CC2)SCCO1 C1(C(=O)NCC(CNC(c2cnc3ccoc3c2)=O)CO)OCCOC12CCC2 C1(=CC(=O)NCC2C(NC(c3occ(C)c3C)=O)C2)CCOc2ccccc21 CCCC(C(=O)N1CCC1CC(C)(C)CNC(=O)C=Cc1nccs1)OC C(CCF)(C(=O)NCCC(N)=O)NC(c1n(C)ccn1)=O Cc1cc(CNC(=O)C(C)(C)NC(=O)CC2CC(=O)NC2=O)cc(C)n1 N1(C(C2(NC(C3N(C)C(=O)OC3)=O)CCCC2)=O)CCN(C)C2(CC2)C1 c1(C(=O)NC2(C)CC(NC(C3(C)CC4CCC3C4)=O)C2)cc(O)c2ccoc2c1 N1(C(CCCOC)=O)CCC2(CC1)CN(C(C1CCC3(CC3)C1)=O)CCO2 c1(C(=O)NCC2N(C(CCOCC)=O)CC2)nn2cccnc2c1Cl C1(O)(CCC)CCN(C(C2C3CN(C(=O)C(F)(F)CO)CC23)=O)CC1 CC(C)(CCCC(=O)NCC1(CO)CCCC1)NCc1cc(C)on1.C(N)(=O)N N1(C(CC(C)OC)=O)CCCCC1CCCNC(=O)CN1CCCC1=O C12(C(C)(C)C)CN(Cc3nc4ccccc4[nH]3)CC(c3ccccc3)(C1)C2 C1(C(=O)OC)CCOC(C)(CNC(C23CC(C2)C(C(F)(F)F)O3)=O)C1 C(=O)(C(F)C(C)(F)F)NCC1(F)CC(CNC(C(c2ccccc2)C)=O)C1 CC12CCN(CC3CNCC3(F)F)CC1C2(Cl)Cl N1(C(c2ccc(C(C)C)nc2)=O)CCN(C(=O)CC2CCC2C)CC(C)C1 C1(NC(CC=CCNC(C2N(C)CCOC2)=O)=O)Cc2ccccc2C1 C(=O)(C(C(F)(F)F)C(F)(F)F)N1CCN(C(c2ccc(N)c(C)c2Cl)=O)C(C)C1 Cc1cnc(CNC(C2CCCC(NC(C3CC34CCCCC4)=O)C2)=O)c(C)c1 N1(C(C(COC)C)=O)CCCCC1C(=O)NCCC1CCC(C)CC1 Cc1cc2cccc(CNC3(CC(=O)NC4CCC5CC4C5(C)C)CCC3)c2[nH]1 c1(C(=O)NC2CN(C(c3c(OC)csc3)=O)CC(O)C2)ccnc2cc[nH]c12 Cc1ccc(OCc2cc(Br)cc(I)c2)c(-c2cccnc2-c2ccccc2)c1 c1(C(C)=O)cc(C(=O)NCC2CCCC2NC(C2CCSCC2)=O)no1 C12(CNC(C3CCCC3O)=O)CN(C(C3CCC4(CCCC4)C3)=O)CC1CCO2 C1(NC(c2cnn(CC3CCCC3)c2)=O)CC2CCC1N2C(=O)Cn1nccn1 N1(C(C2CC(C)=C(C)CC2)=O)CC2CCN(C(=O)C=C3CCOCC3)C2C1 c1(C(N(CCC(C)NC(c2c(CC)ccs2)=O)C)=O)ncc(CC)cn1 C1(NC(COC)=O)CCC2CN(C(C3(COC)CCCCC3)=O)CC2C1 c1(OC)cc(CN2CCN(CC3CCCCC(=O)N3)CC2)cc(Cl)c1OCC(N)=O C1(c2onc(C)n2)CSCCN1C(=O)CNC(=O)CCCSc1ccccc1Cl c1(C(N(C(CNC(c2c(CC)[nH]nc2Cl)=O)C)C)=O)cc2c(cnn2C)nc1O C(=O)(CCCC(F)(F)F)NC(C1CCCN1C(=O)CCN1CCP(C)(=O)CC1)C CC(F)(F)C(F)C(=O)N1CCCCC(CNC(C2CCCN2C2CC2)=O)C1 c1(CN2CC(CC#N)N(C(c3nc(C(C)C)cs3)=O)CC2)c(F)cc(Cl)cc1F N1(C(CCCNC)=O)Cc2cccn2CC(C(N2CCOC(C3CC3)C2)=O)C1 C(c1cnc2ccccc2n1)=CC(=O)NCCNC(CC1CC(CC)OCC1)=O C1(N(C(CC=C=C)=O)C)CCN(C(=O)C(N2CCCCCC2)C)CC12CC2 c1(C(=O)NCC(CC=C)NC(C2OCCC2C)=O)csc2ccccc12 Cc1cnc2n1CC(C(N1CCC(NC(=O)C=CC(C)C)C(F)C1)=O)CC2 c1(CC(=O)NC2CCC3(CC2)CN(C(C2CC2Cl)=O)C3)c[nH]c2nccc(Cl)c12 C1(NC(C(N2CCSCC2)C)=O)CN(C(c2cncc(N)c2)=O)CC1O C(N=c1cc(N)c(I)c[nH]1)c1ccc(OC)cc1C c1(NC(=O)OCC)cc(NC(C(=O)N(C2C(OCC)COCC2)C)=O)cnc1C N1(C(C(C=C)O)=O)CCC(N2CCC(CNC(=O)CC3CCS(=O)(=O)C3)C2)CC1 N1(C(C(=O)NCCc2c(OC)cccc2Br)=O)CCCC2(C1)CC2(F)F C(=O)(CS(=O)(=O)CCO)N(CC(CN(C(c1cc(OC)cc(Cl)c1)=O)C)O)C C(=O)(C(C)Cc1ccncc1)NC(CNC(COCCOCC)=O)CO N#Cc1cccc(CN2CCCCC(NC(=O)Cc3cnns3)C2)c1 C1(C(=O)NCC2CCC(NC(c3n(C)nc(O)c3)=O)C2)(N(C)C)CCC(C)(C)C1 c1(NC(C(C2CN(C(=O)Cc3c[nH]nc3O)C2)OC)=O)cnn(C)c(=O)c1 c1(C(=O)NCC(CN(C(c2c(OC)c[nH]n2)=O)C)(C)C)cc2c(cc1O)CCC2 N1(C(CN(CCC)C)=O)CC(C)CCC1CNC(=O)C(C(C)C)OCC(C)C c1(C(=O)NC(CNC(C2(C)CNC(=O)C2)=O)(C)C2CC2)ccc2c(c1)NC(=O)C2 C1(C(N2CCCC(CCNC(=O)CCc3ccoc3)C2)=O)C2CCCCCCC12 C(CO)(CCCCNC(c1cc(Cl)cnc1OC)=O)NC(CCC=C)=O N1(C(CCCNC(c2ccc(CC#N)cc2)=O)=O)CCCC(F)CC1 c1(C(=O)NCC(C)NC(c2ccc(C3CC3)nc2)=O)cc(C(F)F)n(C)n1 C1(C(=O)NCCC2CCN(C(=O)Cc3ccoc3C)CC2)(OC)CCSCC1 c1(C(=O)NCC2CCCC2NC(C2CC23CC3)=O)cccc2nccn12 N1(C(CC2(C)OCCO2)=O)CCN(C(=O)CC2C3COCC23)CC1CO C1(OC)CCN(C(=O)C(C2CC2)N(C(=O)C#CC(C)(C)C)C)CC1F C1(C(N(CCNC(c2cnc(N(C)C)o2)=O)CC2CC2)=O)CCS(=O)(=O)CC1 c1(C(N2CCC(N(C)Cc3ncc(OC)nc3)C2)=O)n[nH]c2ccc(Br)cc12 c1(CC(=O)NC2(CN(C(C(C)OCC)=O)C)CC2)cncc(O)c1 N1(C(c2c(CCNC(c3cscn3)=O)n[nH]c2)=O)CCC2CC1C(=O)O2 c1(C(N2C3CN(C(c4cc(OC)no4)=O)CC2C3)=O)c(F)ccc(OC)c1F c1(C(=O)NC(C2C(C(=O)NC3(C(C)C)CC3)C2)C)cc(O)n(C)n1 C1(NC(c2ccn(CCNC(c3c(C)nco3)=O)c2)=O)CCCCC1CCO c1(C(=O)NC2CN(C(C(COC)(F)F)=O)CC2C)c[nH]c2cccc(C)c12 C(=O)(C1=NN(C)C(=O)CC1)N(C)CC1CCN(C(=O)CC23CCCN2CCC3)C1 C(=O)(C#Cc1ccc(Cl)cc1)Nc1c(C(=O)NCCC)cc(F)nc1 Cn1ncc(N)c1C(=O)NCC1(F)CC(NC(=O)CCc2ccsc2)C1 N1(C(C(Cc2ccco2)NC(c2cncc(NC)c2)=O)=O)CC2(CCC(=O)N2)C1 c1(OC)cc(NC(=O)C(C)(C2CCC2)NC(=O)C=C(C)C)ccc1O C(CO)(CCC(C)C)NC(C(CSCC)NC(c1c[nH]ccc1=O)=O)=O C1(NC(c2ccc(C)cc2)=O)CCN(C(C2CC(CF)C2)=O)CC1CCO c1(COC)cc(C)c(C(=O)NCCCN(C(c2cc(C(F)F)cs2)=O)C2CC2)o1 C1(c2nn[nH]n2)(C(=O)OCC=CCNC(CNC(CN(C)C)=O)=O)CCOC1 c1(C(=O)NC2Cn3c(CC)nnc3CC2)cn(C)c(=O)c2ccccc12 C(=O)(CC(C)(O)c1ccccc1)N1CCC(NC(C(c2cn(C)nc2)=O)=O)C1 CC(C)C#CC(=O)NC(c1ccccc1F)CNC(c1cc(C(N)=O)cs1)=O N1(C(C(CC)SC)=O)CC2CC(C(N3C(CO)CC3CO)=O)C(C2)C1 C1(C(N(C(CC(C)C)C)C)=O)N(C(=O)CCNC(N)=O)CCCC1(C)C C(=O)(C(CCC)C(C)C)N1CCC(CNC(c2c(CCC)n(C)nc2)=O)C1 CCC(C(=O)N1CC(OC)C(NC(C2CNC(=O)C2)=O)C1)C(C)(C)CC c1(CNc2c(C(C)C)csn2)ccc(Cl)c(F)c1.C1(C)CC(=O)N1 c1(CC(=O)NC(C2CC(CC(=O)NC(C)C#N)C2)=O)ccc(C(F)(F)F)cc1 C1(C(=O)NC2C(CC)CCC2)CC(NC(c2ccc(OC)cc2)=O)CCN1 CCCCCCC(C(=O)NCc1ccccc1OC)N(C)CC1CCCCCC1 C12CCN(CC1C)C2=O.Cc1cccc(C(C(=O)O)NC(=O)OC(C)(C)C)c1 c1(-c2cc(C(=O)NC(c3ccc(O)cc3)C)c(F)nc2)cc2ccccc2o1 N1(C(C2(C(=O)OC)CC2)=O)CCN(N2CCOC(c3ccccc3F)C2)CC1 C1(CC(=O)NCC(C)(O)C(F)F)C2CCCC2N1C(c1coc(CO)c1)=O C1(S(C)(=O)=O)(C(N2CCC(NC(C3CN(CC)C(=O)N3)=O)C2)=O)CCC1 CC(C)(C#N)CCC(=O)N1CCC2(CC1)CC2NC(=O)Cc1cncnc1 c1(C(=O)NCC2N(C(=O)Cn3cccn3)CC2)cnc(C2CCC2)s1 N1(C(=O)NC(C2CCOCC2)CCO)CCCC2(C1)C(O)CC2O C1(C(N2CC(C)(OCC(=O)NC(CC(C)(C)C)C)C2)=O)CCOC(C)(C)C1 c1(C(N2CCCC(CN(C(c3ccc(C)nc3)=O)CC)C2)=O)cccc(=O)n1C N1(C(c2c[nH]nc2[N+](=O)[O-])=O)CC(NC(c2ccc(CC)s2)=O)C(C2CC2)C1 N1(CC(N2CC(C(C(=O)NCC(C)O)(C)C)(O)C2)=O)CCCCC1C c1(OC)ccccc1C(C)CC(=O)NCC(C)(C)Cn1cc(-c2ccsc2)nn1 C12(C(N3C(CNC(c4nn(C)c(Br)c4)=O)CC(F)C3)=O)CC3CC1C2C3O CN=c1cc(C(N2CC(NC(=O)C=Cc3ccccn3)CC(C)C2)=O)cc[nH]1 O=C1NCCCC12CCCN(c1cccnc1S(=O)Cl)C2 c1(C(N2CCCC(C(=O)OCC)(CC)C2)=O)ccn2ncc(CC)c2n1 c1(OCC)ccc(C(C)C(=O)N(CCC(C)NC(=O)C(C)(C)C#N)C)cc1 Cc1ccc(C(=O)NCC2(F)CC(NC(c3occc3C)=O)C2)c(Cl)c1 c1(CNC(c2cccc(CNC(Cn3c(C)ncc3)=O)n2)=O)cc(F)ccc1O c1(OC)cccc2c1C(C(=O)N1CCN(C)C(C(F)(F)F)C1)CC2 N1(C(C2C=CC(=O)N=N2)=O)CC2(CC(N3CCNC4(CC4)C3)C2)C1 c1(C(=O)NCC(CNC(C=CC(C)C)=O)O)ccc2c(c1)nc(O)n2CC1CC1 C1(NC(C23CCC(OC)C2CC3)=O)CCN(c2ncnc3[nH]ccc23)CC(O)C1 Cc1noc(C)c1C(C)NC(=O)COC1(C)CN(C(c2ccc(=N)[nH]n2)=O)C1 c1(COC)ncc(Br)cc1F.C1(C(=O)OCC)CC2CC1COC(=O)N2 c1(C(=O)NC(c2ccc(Cl)cc2)C)ncn2cc(-c3cccc(C(N)=O)c3)sc12 Cc1nc(CC(=O)NCC(C)(CO)NC(=O)Cc2ncoc2C)cs1 c1(CCC)ncc(C(=O)NCC2CC(F)CN2C(c2cc(CO)n(C)n2)=O)cn1 c1(C(=O)NC(C(C)(C)C(=O)O)=O)csc2nc(-c3ccc(C(F)(F)F)cc3)nn12 N1(C(C(CCC)(C)C)=O)CCC(C)N(C(=O)C=Cc2cncs2)CC1 N1(C(Cn2nc(C)c(Cl)c2)=O)CCC(C)C(NC(c2cnn(CC(F)F)n2)=O)C1 c1(C(=O)NCC2N(C(c3occ(C(N)=O)c3)=O)CC2)cc(C(F)(F)F)cnc1O C(=O)(C(C(C)C(C)C)NCC(O)C(C)(C)O)OCC C(=O)(NN1CCCOCC1)c1c(OCC)c(Cl)cc(C)n1 C1(NCC(C(=O)NCC(=O)NC2CCN(S(C)(=O)=O)C2)(C)C)CC2(CCOC2)C1 n1(CC(=O)NC(C2CC(NC(C3CCCC3C)=O)C2)C)nnc(C(C)(C)C)n1 C1(CCNC(C(CO)N(C)C)=O)CN(C(c2ccnc(Cl)c2N)=O)CCCO1 C1(C(=O)NC2CON(CC)C2=O)C2CCN(C(c3coc(OC(C)=O)n3)=O)CC12 N1(C(C(C)OCC(C)C)=O)CCC(CNC(=O)CS(N)(=O)=O)C(C)C1 C1(C)(C(=O)NC2C(NC(C3N(C(C(C)(C)C)=O)CSC3)=O)C2)CCC(F)(F)CC1 CCCC(C(=O)NCC)N(C(=O)CN1CCC(OCC(F)F)CC1)C c1(C(=O)NCC(C2CCCC2)NC(C2C(OC)CCC2)=O)cc(C)nnc1O c1(SC)cccc(CN2CCC3(CCCNC3)C2)c1[N+](=O)[O-] N1(C(c2cc(C(C)C)no2)=O)CC(C(=O)NCc2n[nH]c3c2CCC3)CC(C)C1 C1(CC(=O)NC(C)Cc2cnc[nH]2)COCCN1C(C1CC1Cl)=O C1(C(=O)NCC(C2CC2)NC(C23CC2C3)=O)CCNC1=O.c1(S)ccccc1 N1(C(c2c(CC)ccs2)=O)CCN(C(=O)CNC(c2cccc(O)c2)=O)C(C)C1 C(=O)(C(C)NC(=O)CC1CCCO1)N(C(C)CNC1CCC1)CC c1(CNC(=O)C(=O)NC2CCC3CC3C2)cc2c(cc1Br)OCCO2 CC1=C(C(=O)NC2CCOCC2C(N2CC(=O)NC3(CC3)C2)=O)COCC1 C1(NC(CC)=O)COCC1CNC(n1ccnc1)=O.C12CC1NC2=O CC(C)(CNC(=O)COC1CCOC1)CNC(=O)CCOCc1ccccc1 C1(Nc2snc(C)n2)CN(C(=O)C(C)(C)C2CC2)CCC1CO CC(C)(C(=O)NS(C)(=O)=O)NC(C1CC(=C2CCC2)C1)=O.C(CO)S C(=O)(C(Cn1ccnn1)NC(=O)CSCC(F)F)NCCSS(N)(=O)=O C1(C(C)(C)C)CCCCC1NCCNC(=O)NC1COC1 c1(OC)ccc2nccc(C=CC(=O)NCC(CO)NC(=O)CC(C)OC)c2c1 C1(OCCC)CN(C(=O)Cc2ccoc2)CC1C(=O)NC1CSC(C)=N1 CCC(CC(=O)N1CC(C(=O)O)CC1N(C)C)C(C)C C(CC(F)(F)F)N.C1(CCC(=O)N(CC(=O)N(CCOC)CCOC)C)CCC(C)O1 C1(NC(CC(C(C)C)O)=O)CC2CCC1N(C(=O)C(c1cc(F)cc(Cl)c1)=O)C2 c1(C2(F)C(C(=O)OC(c3ccccn3)C)C2)ccccc1 N1(C(CC=CC)=O)CC(F)CC1C(=O)NCCCCCOC N1(C(CCCNC(C)=O)=O)CC2CC1CN(C(c1nc(Cl)sc1Cl)=O)C2 C1(NC(c2ncc(OCC)nc2)=O)CN(C(C2CCC(C)O2)=O)CC1C1CC1 CC1CN(C(c2cnn(C)c2C#N)=O)C(C)CN1C(c1cc2ccccc2s1)=O Cc1ccc(C(=O)NC2(n3cc(-c4ccc5c(c4)CC5)nn3)CC2)c(I)c1 N1(C(CN(C(C(C)C)=O)C)=O)CC(NC(=O)C(C)(C)CC#N)CC12CCC2 N1(C(c2cc(SC)oc2)=O)CC2CCCC2(C(=O)NCC(C)(C)F)C1 CCCCCCCCCC(=O)N1CC2(CC(NC(C34CC(C)C3C4)=O)CO2)C1 C1(NC(C(C)OC2COC2)=O)(CNC(c2ccc(CO)s2)=O)CCCC1 N1(C(C2(COCC)CC2)=O)CC(NC(c2cn[nH]c2)=O)C2CCCCC12 c1(C(=O)OC)ccc2sc(NC3CC(C)N(C(C4CC(=O)N(C)C4)=O)C3)nc2c1 C1(CNC(=O)NCCC2(c3ccccc3)CC2)CCCC23OCCC2CC13 c1(C(=O)NC(CCCNC(Cc2ccn(CC)n2)=O)C)ncccc1C N1(C(c2ccc(-c3nc(C)on3)cc2)=O)CCN(C(=O)C2=CCC2)CC(O)C1 c1(CC(=O)N(CCCOCCNC(c2c(C(C)=O)coc2)=O)C)cn(C)nc1C N1(C(CC(C)CNC(c2cccc(F)c2)=O)=O)CCC(C)(C)C1C C(CCS(C)(=O)=O)NC(c1ccc(C(F)(F)F)cc1)(c1n(CC)nnn1)C C(C(=O)N1CCCC1CNC(C1COCCN1CC1CCC1)=O)(C(C)C)OCC N1(CC(=O)NCC2C(NC(c3c(CC)scn3)=O)CC2)C(=O)CN(C)C1=O CC(c1ccccc1)=CC(=O)N(C(CNC(c1cnc(O)c(F)c1)=O)C1CC1)C C1(c2cn(C3CC(OCC)C3)nn2)CCCCN1C(=O)Cc1ccccc1F O=[N+]([O-])c1cc(Cl)ccc1CN1CC2CCCC(C1)O2 C1(CC(=O)NCCC(C)NC(Cc2n(C(C)C)ncc2)=O)CCC12CCC2 C12(NC(c3cc(CNC(c4ncn(C)c4)=O)oc3)=O)CCN(CC1)C2 CC1CN2CC1NC(=O)c1c(nn[nH]1)C2=O.C1(COC(C)(C)C)CC12CC2 C(=O)(C1CCCc2ccnn21)N1C(C)CC(NC(C(CC)O)=O)C1 CCC(C)(CC)C(=O)N1CC(OCCC(=O)Nc2n[nH]c(C)n2)C1 c1(CNC(C(CC#C)(C)C)=O)ccc2c(c1)CN(C(=O)C(F)C(=O)OCC)C2 C1(C(N2CCC(NC(c3c(CC)oc(C)c3)=O)C2C2CC2)=O)CCCC(F)(F)CC1 N1(C(C2C(C)OCCC2)=O)CC2C3CCC(C2C1)N(C(c1nn[nH]c1Cl)=O)C3 c1(C(C(=O)NCCCF)N(C(CC)C#N)C)ccc(C)nc1 c1(C(N2CCN(CCN(C(=O)CC3CCOC3)C)CC2)=O)cc2[nH]ccc2s1 c1(C(N(C(C)CNC(C2CCC(O)C2)=O)CC)=O)oc(C)cc1C c1(C(N2CCCC2CC(=O)OC)C(=O)NCCCSCC)ccc(C)cn1 C1(CNC(Cc2c(C)ncs2)=O)CCCCCN1C(=O)CNC(C1CCCC1)=O C(=O)(C1Cc2ccccc21)N1CCC(N2CCN(C(CC(C)F)=O)CC2)CC1 c1(C(=O)NC2CC(C)CN(C(c3cccs3)=O)C2)oc2ccccc2c1Cl C1(C2(C(=O)NCC(=O)NC3CC3)CC2)CCCN1C(=O)Cn1cnnn1 C1(NC(c2ccc(C(C)(C)C)cc2)=O)C2CCC1N(C(=O)C=Cc1ccco1)C2 N1(C(CC(CC)OC)=O)C2CCC1CC(N(C(=O)CCCC1CCCO1)C)C2 c1(OC)cc(F)c(NC(C2CC3CN(CC4CCC5CC45)CC23)=O)cn1 c1(C(=O)NCC(N(C(CC(C)C)=O)C)C2CC2)cnc(Cl)c(Cl)c1 N1(C(CCCOCC)=O)CCCC2(C1)CN(C(C1(C)CCN(C)C1=O)=O)CCO2 c1(C(=O)N(C2C(C(c3cn(CCO)nn3)C)CCC2)CC)cc2ccnc(Cl)c2[nH]1 C1(C2CCCN(CC=C)C2)(NC(C2CC2)=O)CC1.c1(C(=O)OC)cnc(Cl)c(Cl)c1 Cn1nc(Br)c(C(=O)NC23CC(NC(N4CCNC(=O)C4)=O)(C2)C3)c1N N1(CCC)CCCC1C(=O)NC1C(C(=O)OC)CC1O.C12CCC1CNC2=O C(CC(C)(C)C(=O)N1CCCC(CN(C)C(C2CCS(=O)(=O)N2C)=O)C1)OC c1(C(=O)NC(C)CNC(c2cn(C)nn2)=O)cccc(NC(=O)CC(C)(C)C)c1 C1(C(=O)NCC(C(=O)OCC)C)CN(C(c2cccc(C#N)c2)=O)CC1(F)F C12(NC(Cc3c(C)cccc3)=O)CCCC1N(C(=O)C=Cc1cnc[nH]1)CCC2 c1(OC)cccc(NC(C)C(=O)NC(CNC(c2c[nH]nc2C)=O)CO)c1 C(N=c1[nH]c(=NCC(C)COC)[nH]c2ccsc12)c1sc2ccc(OC)cc2n1 C(N=c1cc(NCCC(CCCC)OC)nc(C)[nH]1)c1c(CC)cccc1 Nc1nc(Cl)ccc1C(N1CCOC(CNC(c2cc(C3CC3)on2)=O)C1)=O c1(C(N2CC3(CC(CNC(C=C)=O)C3)C2)=O)ccc2c(c1)CCCN2 c1(NCCC2CCCN(C(CCNS(C)(=O)=O)=O)C2)nc2c(cc1Cl)C(=O)OC2 c1(C(=O)NCCCCN(C(C(C(=O)NC)(C)C)=O)C)cccc2c1OCCO2 C(=O)(C1=CCCOCC1)N1CCC(C(C)NC(c2c(C)nc(C)s2)=O)C1 Cc1nnc2ccc(-c3cnc(Cl)c(C(=O)Nc4cc(Br)cnc4O)c3)cn12 C(=O)(CCCCC(C)(C)C)NC1CCN(Cc2c(O)ccc(OC)c2)CC1 c1(C(=O)NC2C=CCN(C(C(CCC#C)O)=O)C2)cc2c(C)cc(OC)cc2[nH]1 C#Cc1ccc(C(=O)NC2CCC(CC(=O)NC3CC4CCCC4C3)C2)cn1 C1(CN(C(C=CS(C)=O)=O)CC)CCCN(C(=O)CCC(=O)c2cccs2)CC1 C(=O)(C(C)(C)CC(F)F)N1CCN(C(c2c(Oc3ccccc3)cn(C)c2)=O)CC1 C#CCC(C)(C)CNC(C12CC1CN(C(C1CC(CN(C)C)C1)=O)C2)=O C1(CNC(c2ccc(C)cc2Cl)=O)CC2(CCC2)CN1C(=O)CC=CC(C)(C)C C1(C(N(C2CC(NC(=O)CC3COCCO3)C2)C)=O)CCC(c2nc(=N)[nH][nH]2)CC1 C=CCC(CC(C)C)C(=O)N1CC2=C(C1)CN(C(C1CC1CC)=O)C2 C1(CC)CCN(C(=O)C(=O)Nc2cccc(OCc3cccnc3C)c2)CC1F c1ccc(N2CCCC(O)C2)cc1.CC(CC(=O)NCC1(NC=O)CC1)N(C)C c1(OCC)ccc(Cl)nc1C(=O)NC1CC1NC(=O)CC1CC=CC1 N1(C(c2cc(=O)cc[nH]2)=O)CCCC2OCCC12.C12(CC1(F)F)Cn1cc(nn1)C2 C(=O)(C(C)S(C)(=O)=O)N1CCN(CCNC(c2cccc(C(C)C)n2)=O)CC1 C1(C2CCCC2)(C(N(CC(C)NC(C2(CC)CCNC2=O)=O)C)=O)CCNC1=O N1(C(c2cc(-c3ccccc3)on2)=O)CCC2CN(c3ncncc3F)CC2C1 C(=O)(Nn1cnnc1)C1OCCC(NC(c2ccn(CC)c2C)=O)C1 C#CCC(CC(=O)N(C)Cc1cccc(F)c1)NC(=O)C(C)C(C)C c1(C(N2C(CNC(C(CCOC)OC)=O)CC2)=O)cc(C)cc(N)c1 c1(C(N2CCC(C)(CC(C)C)CC2)=O)cc2c(Br)c(Cl)ccc2s1 c1(C(N2CCC(NC(c3cnc(C)o3)=O)CC2C)=O)cccc([N+](=O)[O-])c1N c1(C(N2CC(CC)C(NC(=O)C(C)(C)OC)CC2)=O)cc(F)c(F)cc1Cl N1(C(c2cc(CC)[nH]n2)=O)CCN(C(c2oc(CC)nc2C)=O)CCC1C C=CC(C)(CCOC)C(=O)NC(C)CNC(=O)CCOc1ccccc1F C1(CC=C)(NC(=O)CCC=CBr)CCCN(C(c2ccccn2)=O)C1 C(C)(C(=O)N1CC(C(O)C(=O)NCCn2cncn2)C1)OC(C)=O S(=O)(=O)(c1ccc(-c2cncc(F)c2)o1)N1C(c2nc(C)on2)CCC1 CS(=O)(=O)c1cccnc1NC(C1C=CC(C(=O)O)C1)=O N1(C(C2C(CC)C2)=O)CCCC1CN(C(=O)C(C)N(C1CCC1)C)C C1(C)(C(=O)NCC2CC(C)N(C(c3ccc(C4CC4)o3)=O)C2)CC2(CC(O)C2)C1 N1(C(Cc2nc(C)on2)=O)CC(NC(=O)CC2NC(=O)NC2=O)CC(F)C1 CC(C)(CF)C(=O)NCCC1(C(=O)NCCNC(=O)OC(C)(C)C)CCCC1 Cc1cn2cc(C(=O)NCC3(F)CCN(C(=O)C(O)CC(C)(C)C)C3)sc2n1 CN1CCCC1C(=O)NCCC1CCCN1C(=O)Cc1cc[nH]c1 N1(C(CC(=C)C)=O)C2COCC1CC(NC(c1ccccc1OC)=O)C2 c1(OCCC(=O)OC)cccc(C(CO)SC)c1 c1(C(N2CCCC(NC(C(C#C)(C)C)=O)C2)=O)ccc2c(=O)cc[nH]c2c1 c1(C(=O)NCC2(N(C)C(C3CCC(=O)O3)=O)CC2)ccc2c(c1)OCO2 CP(C)(=O)CC(=O)NCC1CN(C(=O)CCc2cncs2)C1 C(=O)(CN1C(=O)Cc2ccccc21)N1CC(NC(=O)C=CC=C(Cl)Cl)C(O)C1 C#CCCC(C(=O)NC(C#C)C(=O)OC)NC(C1CC2C=CC1CC2)=O C1(C(=O)NCC(C#C)OC)CCC2(CC2)N1C(c1cn(C)nc1CC)=O N1(C(C(=O)N(CCCCCC)n2cc(C)cn2)=O)CCOC(CCC(=O)OC)C1 C12(C(=O)NC3(c4onc(C)n4)CC3)CC(CO1)N(C(C1CCC1C(C)(C)C)=O)C2 N1(C(C(C(C)NC(C2CC(=C3CCC3)C2)=O)C)=O)CC2(CCC(C)OC2)C1 CCCC(C(=O)NCCNC(C1CCC(=O)C1)=O)C1CCC1 S(=O)(=O)(c1cccnc1NCC1CCCC(P(C)(C)=O)C1)NCCC(C)(C)F C(=O)(C(C)(C)CC(F)(F)F)NC1CCN(C(c2nc(C)sc2)C)CC1 c1(CNC(CC2(CC)CC2)=O)ccccc1CNC(c1cncc(OC)n1)=O C1(CCC(=O)NC2(C(=O)OC)CC2)CCCN(C(=O)CC2(O)CCC2)C1 C1(=O)CCC(=O)N2CCCC(C2)N1.c1(CC)occc1C(=O)NC1CC12CC2 C=CC1(O)CN(C(=O)C(C)N(C(c2n[nH]cc2Cl)=O)CC)C1 C(=O)(C(C)(F)C(F)(F)F)N(CCCCN(C(CS(=O)(=O)N(CC)CC)=O)C)C c1(C(=O)NCc2c(C(=O)NCC(=O)CC3CC3)cccn2)cc(F)cc(F)c1 Cc1oncc1C(=O)N(C(C)C(=O)N1CC(n2ccc(C3CC3)n2)C1)C1CC1 CCC(C)(CN1CC(F)=C(C(=O)NC(C)(C)C)CC1)C(=O)N(C)C1CC1 C(S(=O)(=O)c1ccc(Br)cc1)c1nc(CC(C)(O)C(F)F)on1 c1(C(=O)NCC2(CCNC(C3(CC(C)C)CC3)=O)CC2)cc2ccc(Cl)cc2o1 C=CC(C)(O)CC(=O)N1CCN(C(=O)CNC(C2CC2F)=O)CC1 N1(C(C(=O)NCCOCC2CC2)C2CC2Cl)CC(=O)N2CCCC2C1 C1(NC(CC2CCC(C)(C)C2)=O)CCN(C(=O)CC(=O)NC2CC2)CC(O)C1 N1(C(C(C)=CC)=O)CCN(C(=O)COc2ccc(C)cc2)C(COC)C1 C1(C(=O)O)CC2CC1N(C(c1ccc(N3CCC(O)CC3)cc1)=O)C2 N1(C(C(C=C)O)=O)CCC(C2CC2NC(c2ccccc2CC#N)=O)CC1 c1(NC(C(C)C)CN(C)C)ccc(S(=O)(=O)NCC2CCC23CCOCC3)c(Cl)c1 c1(OC)cccnc1C(=O)NC(C)(CNC(=O)C(C)NC(C)=O)C1CC1 c1(N2CCC(C)C2)nc(NC2CCCN2CCCN(C)C)nc2cc[nH]c12 C1(C(=O)NCC(CCC)C)CN(C(c2ncccn2)=O)CC1(C)C C(=O)(C(C1=NOCC1)N1CCC(N2CCCOC2=O)CC1)NCCSC CC(=O)CCCC(C)C(=O)N1C(C(=O)NCCCc2ccsc2)CCC12CC2 C12(NC(CC(COC)C)=O)CCCC1N(C(c1cc(C)c(Cl)s1)=O)CCC2 N1(C(C(c2ccc(OC)nc2)(F)F)=O)CC2CC(NC(=O)C3=NOCC3)C2C1 c1(C(=O)NC2CC(NC(C3(C#N)CC(C)C3)=O)C2)nccc2ccn(C)c12 Cc1ccc(CC(=O)NC2(C)CCCN(C(=O)CC(C)CF)C2)c(Cl)c1 c1(C(=O)NC(C2CCN(C(=O)C(C3CCCO3)C3CC3)C2)C)cnc(F)c(Cl)c1 CC(C)(C)CC(O)CC(=O)NCCOCC(N1CCCCC(C)(F)C1)=O N1(C(CC)=O)CCCC2(CNC(c3cc(OC)ccc3F)=O)CCCCC12 CCCCC(C(=O)NC1(C)CN(C(C2CCCC2OC)=O)C1)N(C)C N1(C(c2c(Cl)nc(CC)s2)=O)CCC2(CCCN2c2ncncc2Br)CC1 c1(C(N(C)CC2(O)CN(C(c3n[nH]cc3Cl)=O)C2)=O)ccc2c[nH]nc2n1 N1(C(=O)NC)CCCCC(C(=O)NCc2cc(Cl)cs2)C1 c12ccc(o1)C(=O)N(C)CCCN(C)C2=O.C1(C(=O)OC(C)(C)C)CC(CF)C1 c1(NCC)ccc(Cl)cc1C(=O)N(C(C)CN(C(=O)C=Cc1cc[nH]n1)C)C CCC(C)(C)CC(=O)NCC1CCN1C(=O)CC1CCCCO1 C(=O)(C(CN(C)C)C(C)C)N1C(C(=O)NCCCn2c(C)ncc2)CSCC1 C1(O)(CN(C)C(C2CCCS2)=O)CCCN(C(=O)CN(C)C(c2ccoc2)=O)C1 c1(CCNC(C2CN(C(=O)OC(C)(C)C)C(C)(C)C2)=O)c(F)ccc(Br)c1F C1(CC(NOC(c2ccccn2)C)=O)C2CCC(C2)N1C(C1CC=CC1)=O C(=O)(CCCC(=C)C)N1CCC(C)(CC(=O)NC(C#C)CC2CCCC2)C1 C1(CNC(c2c(C)ncn2C)=O)CN(C(c2ccc(O)nc2Cl)=O)CC12CCC2 C#Cc1ccc(C(=O)NCC2CCCCCN2C(=O)CN2CCCC2=O)c(C)c1 C1(NC(C2CCC(C)(C)OC2)=O)CCC2CC1CN2C(c1cc(N)ccc1O)=O c1(CN(C(C2CC(C)(C(=O)OC)C2)=O)C)ccc(C)nc1 N1(C(CSCCCC)=O)CCC(C(=O)NCC2CCC(CO)CC2)(CC)C1 N1(C2CCC(O)C2)CCN(C2(CSC3CC3)COC2)CC1 CS(=O)(=O)C1(C(=O)NCC2CC(O)(CNC(=O)Cc3cscn3)C2)CCCC1 c1(C(=O)NC2(CNC(C3ON=C(C)C3)=O)CCCCCC2)cnc2cc(C)nn2c1 C(=O)(CCCC(=O)NC1CC1)N1C(CNC(c2cc(SC)oc2C)=O)CCCC1 C1(CNC(=O)C=CCN2CCCC2)COCCN(C(c2ccncc2)=O)C1 c1(C(=O)NCC2C(CC(=O)NC(C)CC3CCOC3)C2)cccc2[nH]ccc12 c1(C(=O)NC)ccc(NC(=O)Cc2cc(Cl)cc(Br)c2)c(Cl)c1 c1(C(=O)NCC(C(C)C)NC(=O)CC2CC2C2CC2)cc2cccn2c(O)n1 C1(CN(C(=O)Cn2cc(Cl)cn2)C)C2CN(C(=O)CCc3nccs3)CC12 N1(C(COCC#C)=O)CCC(O)(CN(C(=O)CCCC(C)O)C)CC1 CCCCC(C(=O)N1CCC(NC(c2ccnc(O)c2)=O)C1C)N(C)C c1(NC(COC(C)C)C)nccc(N2CCC(Cc3ccccc3)C2)n1 N1(Cc2c(C)cc(SC)s2)CCC2(CCCC2C(N2CCc3n[nH]cc3C2)=O)C1 Cc1ncsc1CC(=O)NC1(CCO)CN(C(c2cnn(CCF)c2)=O)C1 c1(C(=O)OC)ccc(O)c(NC(=O)C=CC(C)NC(=O)C#CC(C)(C)C)c1 C#Cc1ccnc(C(=O)NC(CC#CC)C(=O)N2CCCOC(CC)C2)c1 C1(NC(C2(C)CNC(=O)C2)=O)CC2CCC(C1)N2C(c1cncc(C(F)F)c1)=O C(=O)(N=c1[nH][nH]c2c1CCCC2)C1(C)CN(Cc2cc(F)cc(C)c2O)C1 N1(CCOC)CCCC(NC(c2cccc(NC(=O)NC(C)(C)C)c2)=O)C1 C1(C(=O)NC2CC(CNC(CC(C)F)=O)C2)CCCN2CCCCC12 c1(OC)cc(C(=O)N(CC(C)NC(=O)CC2CCCCC2O)C)ccc1O CCC(F)(F)C(C)(C)C(=O)NC1CC(C)N(C(c2cc3ccccn3c2)=O)C1 C1(NC(CCCCCSC)=O)CCC2CN(CC3CCCO3)CC2C1 C12(CNC(C=C(CC)C)=O)CCCC1CN(C(=O)C=CCO)C2 n1(CCC(=O)NC(C2(O)CC2)C2COC2)cc(CCC2CCC2)nn1 c1(C(N2C(C)CC(NC(=O)Cn3cnc(Br)n3)C2)=O)cc2[nH]ccc2s1 N1(C(c2c(CC)scn2)=O)CC(OC)CC(NC(=O)C(n2nc(C)cc2C)C)C1 c1(N(C2CCN(C(c3ccc(CO)c(F)c3)=O)C2)C)ncc2c(ncn2C)n1 C1(NC(CCN(CCC)C)=O)CCN(C(c2cc(F)ccc2N)=O)C12CC2 CN(CC(=O)N1CCCCC1)N1CCC(COCC(F)(F)F)C1 C12(C(N(CCN(C(C(C)OC(C)(C)C)=O)C)C(C)C)=O)CC1COC2(C)C C1(O)(C(C)NC(c2ccc(F)s2)=O)CCN(C(=O)C(C)(C)c2cscn2)CC1 N1(C(C#CC(C)(C)O)=O)CCC2CN(C(c3ccc4nncn4c3)=O)CC2C1 c1(OC)ccc(C(O)CC(=O)N(C)CCNC(C2CC23CC(O)C3)=O)cc1 C1(C(N2CCC(CCNC(c3cccc(OC)c3)=O)C2)=O)(OC)CCCCCC1 C1(NC(CCC=C)=O)C2CC3C1C3C2C(=O)NCC1CN(CC)CCO1 O=C(CCCSc1cccnc1)NCCC(C1CCCC1)NC(c1cnc[nH]1)=O N12CCC(CC1)CCC2.S(=O)(=O)(C(F)F)NC(COC(C)(C)C)=O C12CN(C(=O)C=NOC)CCN1C2=O.c1(NC)ccc(F)c(Br)c1.CC C(CC(C)(C)C(=O)N(C(C)CCSC)C)NC(C=C(CC)CC)=O C1N=C2NC(=Nc3ccsc32)N2CCC1C2.CN1CCn2[nH]c(=N)nc2C1 C1(F)(CNC(C2CNC(=O)N2)=O)CCCN(C(C2CC(=O)N(C3CC3)C2)=O)C1 N1(C(C2(C)CCC(=O)C2)=O)CC2C3CCC(C2C1)N(C(c1ccccc1O)=O)C3 N1(C(C)=O)CC(O)CC1C(N1CCCC1C(C)NC(C1(N(C)C)CCC1)=O)=O Cc1cccc(OCCC(=O)NCC(O)CNC(c2cncc(C#N)c2)=O)c1C C(c1ccccc1)=CC(C(=O)Nc1cccnc1)N(C1CC1)CC1(CSC)CC1 C1(NC(CCC)=O)CN(C(=O)C=Cc2cc(C)ccc2OC)CC12CCC2 C(=O)(CC(C)CCC(=O)N1CC(O)(CCNC(=O)Cc2cc(C)cs2)C1)OC C(=O)(CCS(=O)(=O)c1ccc(OCC(F)(F)F)cc1)NC(C(CC)C)C CC1CCN(C(=O)CCS(C)=O)C(C)C1NC(=O)CCCn1cccc1 Cc1[nH]nc2c1CN(C(C1COCCN1C(c1cccc(F)c1Cl)=O)=O)CC2 c1(NC)cnncc1C(N1CC=CC1CNC(C1CC2(CCC2)C1)=O)=O C1(NC(c2c(OC)nsc2OC)=O)CN(C(=O)CS(=O)(=O)N(C)C)C(C)(C)C1 CCC1=C(C(=O)NCCCCC(=O)NCC(CC)n2cccn2)CCCO1 C12(CCCO1)C(=O)NCC2.C1(CNC(C(C)OCCOCC)=O)CC1C1CC1 C1(C(=O)NCCOC(C)=O)C2CCCC2CN1C(C1CCC(C)O1)=O N1(C(C=CC2(C)COC2)=O)CC2CCCC2(NC(=O)C2=CC3(CCOC3)C2)C1 C1(CC(=O)NCC2C(CCC)C2)CCCCC1CNC(c1[nH]ccc1C)=O c1(C(N(C2CC(NC(=O)C(c3cnn(C)c3)O)C2)C)=O)cnn(C)c1C1CC1 CCC(C)C(C(=O)N(C)CCc1ccco1)N(C)C(c1ccncc1O)=O C12(NC(c3nn(C)c(C4CC4)c3)=O)CCN(C(c3csnn3)=O)CC1C2 N1(C(C(C2CCC2)OCC)=O)CCC(C)(C)C(CNC(c2n[nH]c(C)c2Cl)=O)C1 CCCCN=C(NCc1cc(Cl)ccc1C)NC1CCN(CCS(C)(=O)=O)C1 Cc1cc(CNC2CC(Nc3ncnc4c3CCC4)C2)cc(C)c1O C12(CC(=O)NCC(C)NC(C34CC(C(C)C)(C3)C4)=O)COC(C)(C1)C2 C1(CNC(C(C=C)(C)O)=O)CC2CN(C(=O)CN(C)C)CC12 N1(C(C(C)(C)OC)=O)CCC2CN(C(C34CCCC3C4Br)=O)CC2C1 CN1CCCCC1CC(=O)NC1CC2(C1)CC2C(=O)NCCS(C)(=O)=O C(=O)(CCCCCC(C)O)N(CC(C)CNC(c1ccc(C(C)(F)F)nc1)=O)C N1(C(C2(CC#C)CCOC2)=O)CCC2(CCCN(C(=O)CCCCC#N)C2)C1 C1(c2n(CC)nnn2)(NCC2CC2(C)C)CC(C)OC(C)C1 C=C=CCCC(=O)N(CC(N1CCN(C(c2cc(C3CC3)no2)=O)CC1)=O)C C(C(C)C(F)C(=O)NCC1(O)CCSC1)NC(c1cc(CCC)on1)=O N=c1[nH]cncc1CN1CCC(OCc2cn(CC3CCCC3)nn2)C1 C1(NC(=O)CCn2ccnn2)CCSC12CN(c1ccc([N+](=O)[O-])cn1)C2 CC(C)(CC(=O)N(C)C)C(F)F.C12CCN(C1)C(c1ccccc1)C(=O)N2 O=C(CC(C(F)F)n1cccn1)Nc1ncc(C2(CO)CC2)cc1F C12(C(N3CCCC(C(=O)NC(CC#C)C(=O)NC)C3)=O)C(=O)C3CC1C2C3 c1(C(=O)NCC2N(C(C(CC)C(C)C)=O)CCCC2)ccc2nnnn2c1 Cc1ccc(C(N)=O)c(NC(C2CC2C(=O)NCc2ccncc2Cl)=O)c1 C1(C)(CNC(C(C)(N(C(c2n(CC)ncc2)=O)C)C2CC2)=O)CC2CC2C1 C(CN=c1[nH]cnc(NCCC2=CCCCCC2)c1C)c1c(OC)cc(F)cc1 C(CCNC(=O)Nc1cccc(Br)c1O)(C(F)(F)F)OC c1(CNC(COC(CNC(C=CC(C)C)=O)(C)C)=O)nccn1C C(CCO)(C(F)F)N(C(COCCNC(C1C(=C)C1)=O)=O)C c1(C(N2C(CNC(C(C)CC(F)F)=O)CC(O)C2)=O)ccnc2ccsc12 c1(C(=O)NC(CCC=C)C2CC2)oc(CNC(=O)C#CC(C)C)cc1C S(=O)(=O)(c1ccc(F)c(F)c1)NC1CCCN(Cc2cc(C)[nH]n2)C1 C1(C=C)(CC(=O)NC(CC=C)CNC(=O)CNC(C2CCCC2)=O)CCOCC1 C(=O)(C(CC(=O)NCC(C)NC(=O)C(C)Cc1ccncc1)C(C)=O)OCC C1(C(=O)NC(C2CCOC2)C#C)(CC)CCCN1C(c1cnn(C)c1Cl)=O C=CC(C)(O)C(=O)N1CCC(O)(CNC(=O)COc2ccc(Cl)nc2)C1 N1(C(c2c(CC)ncnc2CC)=O)CC2(C1)SCCC2NC(c1cscc1C)=O C1(NC)CCC(C(=O)NC2CCCC2SC)CC1.C1(=O)CCN1C.C1CCO1 C12(C(N(C(CCNC(CC=CCC)=O)C)C)=O)CCC(N=[N+]=[N-])C1C2 N1(C(c2cc3cn(C)nc3cc2)=O)CCN(C(=O)C=CC2CC2)CC(C)(C)C1 Cc1ccc(C(=O)NCC2(C)CCN(C(c3cc(C#N)on3)=O)CC2)c(F)c1Cl Cc1nnc2n1CCC(NC(CN(c1nnnn1CC(C)C)C)=O)C2 C(C(C)(C)COC1CCCCC1)(c1n(CC)nnn1)NC(C(C)C)c1cncs1 N1(C(c2ccn3cncc3c2)=O)CCC(C2CCN(C(C3CCO3)=O)CC2)C1 N1(c2cc(NCC3CCCc4ccccc43)nc(COC)n2)CCC2(CCOC2)C1 C12(CNC(C(C(C)C)OC)=O)CCC(C1)N(C(=O)C=Cc1ccc(C)s1)C2 C1(CN(C)C(c2sccc2CO)=O)CCCN1C(=O)Cc1sccc1Cl C#CC1(C(=O)N(CCC(=O)NCCCCCCO)C2CC2)CCCC1 N1(C(c2c(OC)cccn2)=O)C2CCC1C1CC1(NC(c1cncc(Cl)c1)=O)C2 C1(N(CC(C)(F)F)C2CC2)CCC(=O)N(C(C2C3CCCCCC23)=O)C1=O C1(C(N2C(CCNC(C(CC)N(CC)CC)=O)CCC2)=O)C(C)OC(C)C1C CC(C(=O)NC(CO)CCCNC(c1ccc(OC(F)F)cc1)=O)C(C)(C)C Cc1ccc(Cl)c(F)c1C(N1CCC(O)(CCNC(=O)CC(C)N(C)C)C1)=O c1(CC)nn(C)c(Cl)c1C(N1CC2(C1)CN(C(=O)CC1CCCC(C)O1)C2)=O N1(Cc2n(C)cnc2)CCC2(CC1)OCCC2NC(=O)C1=COCCO1 C1(CC)CCCC1C(=O)N(C1(C)CC1)CC(C)C.C1(=O)CCN1 C=CCC(C)(C)C(=O)NCCOCCOCCNC(c1nc(C)ccc1C)=O C1(C)(CNC(C(CC(C)C)N(C)C)=O)COCCN(C(=O)Cc2cc(Cl)cs2)C1 N1(C(C(C)c2cncs2)=O)CCN(CCSc2ccccc2O)CC1 c1(OC)ccncc1NC(=O)CC1CC1CNC(=O)C(C1CC1)C1CC1 C1(C2(NC(C)=O)CC2)CCCN1C(=O)CN(C(=O)C(C)n1cccn1)C N1(C(CNC(C(C)(C)C)=O)=O)CCCC1(C(=O)NCCC(O)C1CC1)CO C1(C)(NC(COCC(=C)C)=O)CCCN(C(C2(OCC)CCCOC2)=O)C1 c1(OC)ccc(C(=O)NC2CCCC2NC(c2n[nH]cc2C)=O)cc1 N1(CCC(N2CCCC(CNS(C)(=O)=O)C2)=O)Cc2ccccc2C1 O(NC(=O)C(C)(CO)NC(=O)CN1CCSCC1)C(C)(C)CO N1(C(C2CCn3cncc3C2)=O)CCC2(CCCN2C(C2CC23CCC3)=O)CC1 CCC(C(=O)NC1CC(F)(CNC(c2cccn2C2CC2)=O)C1)OC1CCCC1 c1(C(=O)OC(c2ncc(C)o2)C)[nH]c2ccc(Br)cc2c1F C1(C(N2CC(C=C)(CC(=O)NCc3ncc(F)cc3C)C2)=O)CC2(CCC2)CO1 c1cccc(C)c1.C1(C(C(=O)NCC(CNC=O)O)=O)(CC)COC1 CC1CC2(CCOCC2)CN1C(c1nccc2nn[nH]c12)=O n1(CC(N2C(COC)CC2)=O)cc(CNC(C2CCCC2C)=O)nn1 N1(C(c2cn(CCC)nc2)=O)CCN(C(=O)C(C)COC)C(CC(F)F)C1 c1(C(=O)NC2CCC(N(C(=O)C=CC3CCC3)C)C2)cnc(C(F)(F)F)c(F)c1 c1(C(=O)NCC(C(C)C)NC(=O)C=CSc2nc[nH]n2)ccn2ccnc2n1 C(CC(N)=O)(C(=O)N(C)Cc1ccncc1C)NC(Cc1cc(C)sc1)=O Cc1ccc(C)c(C(=O)NCC2CN(C(=O)CN3CCN(C)CC3)CCC2C)c1 c1(SC(c2cc(F)ccc2OC)CC)cccc2c1OC(F)(F)O2 CCC(C)C(C(=O)N1CC=C(C)CC1)N(C)C(C)=O.c1(C(=O)O)nn(C)cc1C N1(C(c2c(CSC)cco2)=O)CCC(O)(CNC(C)=O)C1.C1(=O)CN1C C(CCC(=O)N(CCCNC(=O)C(C)c1cncs1)CC(C)C)N(C(C)=O)C c1(NC(c2cn(C(C)C)nc2)C)ccc(S(=O)(=O)N2CC=C(Br)CC2)c(Br)c1 c1(C(N2CC(C)OC(CCNC(c3cnsc3)=O)C2)=O)cccn2nnnc12 c1(OCC)cnc(C(=O)NCc2ccc(CNC(=O)CCF)cc2)c(Cl)c1 CC(C(F)(F)CO)NC(=O)NC1CCCC(CNC(=O)OC(C)(C)C)C1 c1(CC)nc(=N)[nH]cc1C(=O)NCC(C1CC1)NC(c1nc(O)sc1C)=O N1(C(CCCN=[N+]=[N-])=O)CCc2nc(CNC(=O)COCCF)sc2C1 Cc1cc(F)cc(C)c1C(=O)NC(C(C)NC(c1nc[nH]c1C1CC1)=O)C(C)C N1(C(c2ccc(CC)s2)=O)CCCC2(CCC(NC(C3CS(=O)(=O)C3)=O)C2)C1 C(CCCCCC(=O)NCc1nc(C2CC2)no1)NC(CC=CC=C)=O C(=O)(CS(=O)(=O)N(CC)CC)NCC(C(C)C)NC(C1(C=C)CC1)=O N1(C(CCSC)=O)CC=CC1CNC(c1ccncc1)=O CCCCCCC(F)C(=O)NCC1(NC(=O)CN2CCCCC2=O)CCCCC1 C1(CC(=O)NC2C=CCCC2)CN(C(=O)CSCC(N2CCCCC2)=O)CCO1 N1(C(c2c(CC)cno2)=O)CCC(F)(CNC(c2sc(C)cc2C)=O)CC1 c1(C(=O)NC(CC(C)NC(c2ccc(C(C)(C)C)[nH]2)=O)C)cc(Cl)c(F)c(Cl)c1 Cc1cc(C#N)cnc1N1CCCC2(NC(c3ccncc3)=O)CC2C1 c1(CC(N2CCC(CN(C(=O)C(F)CC3CCOC3)C)C2)=O)cccc(O)c1 Cc1cc(C(=O)NCC2CC(NC(=O)C(C)C(C)O)C2)cc(C)c1C C(CC(C(=O)NC1CCC(Nc2cc(Cl)c[nH]2)CC1)OC)NC(=O)OC O=C(CCCCCc1cccs1)NCC(F)CNC(=O)CCN1CCOCC1 C1(NC(C2N(CCC)CCC2)=O)C2CC(NC(c3csc(C)n3)=O)CC12 c1(CC(=O)NCC(CN(C)C(C2CC(O)C2)=O)O)csc(-c2ccccn2)n1 N1(C(C(CC)n2cncn2)=O)CCCN(C(=O)CC(C2CC2)SC)CC1 C1(C(=O)NCC(C)(CO)NC(c2ccc(C)cc2Cl)=O)CC2CCC1C21CC1 c1(OCC(N2CCC(C(C)NC(=O)CC3CCOCC3)C2)=O)ccc(Br)cn1 C1(NC(COC(CNC(C(C)N2CCCC2)=O)(C)C)=O)CCCCC1O CC(CC#N)C(=O)NOCc1cn(-c2ccc(F)cc2)nn1 Cc1nn(-c2ccccc2F)cc1NC(N1CCCC1C1CCOC1)=O C(CCC(C)(C)C(=O)N1CCC(C2CC2)C1)NC(C(CCC)F)=O Cc1ccc(C(=O)NCC2CCCN(C(=O)C(c3ccc(N)cn3)C)C2)nc1C c1(C(=O)NCC2CCCN2C(=O)CCc2cnoc2)cc(Br)c(Cl)s1 c1(CNC(C=CCN(C(C2(OCC)CCCC2)=O)C)=O)nccc(C)n1 CCCCCCCOC(c1ncccc1NC(C1CCCO1)C1CC1)C Cc1c(Br)cnc(O)c1CNCc1ncnn1C1CC1 C1(SC)CN(C(c2cc(F)n[nH]2)=O)CC1NC(C1(c2ccncc2)CC1)=O N1(C(C(C)=C2CC2)=O)CCC(NC(=O)C(c2ccn(C)c2)C)CC1C N1(c2ncn(C)c(=O)c2)CCC2CCN(C(=O)OC(C)(C)C)CC12 CCCCCCCC(=O)N(C)CC1CCCN1C(=O)C(S(C)(=O)=O)C1CC1 c1(SC)cccc(F)c1C(=O)NC1CCC1CNC(C1CCC1)=O S(=O)(=O)(c1cccnc1NCC(O)CF)NCc1ccc(S(C)=O)cc1 c1(CC(=O)NCC(CNC(c2cccc(CC)c2F)=O)O)cc2ccccc2[nH]1 C12(C(N3CCC(O)(CNC(=O)CSc4cn[nH]c4)C3)=O)CCC(C1)S(=O)(=O)CC2 c1(N2CCC(N(C)C(c3cn4c(n3)CCC4)=O)C2)ncnc2cccc(F)c12 CCC(C(=O)N1CCN(C(=O)Cc2cccnc2Cl)CC1CC(F)F)C(C)C C1(C(=O)NCC2(CC)CN(C(=O)Cn3cncn3)C2)CC2(CC(SC)C2)C1 C(=O)(N=c1[nH]n(Nc2ccc(CC)cc2)cc1C#N)c1cc2cnn(CC)c2nc1 c1(C(=O)NCC(C#C)CC2CC2)c[nH]c2cc(Br)ccc12 C1(C(N2C3CC(NC(C4CCC(=O)C4)=O)(C3)C2)=O)CCC2(CCC2)CO1 C1(CC)C(NC(=O)COc2cccc(F)c2)CCN1C(=O)CN(C)C(N)=O c1(C(N2C(CNC(c3n(CC=C)ccc3)=O)CC2)=O)cccc(C(C)=O)c1 C1(C(=O)NCC(COCC)C)CC2C=CC1N(C(c1cnc(O)c(C)c1)=O)C2 N1(C(c2ccnc(OC)n2)=O)CCC2CCN(C(c3c(Cl)cnn3C)=O)CC2C1 C=C(C)CCC(C(=O)NCCC1COCCO1)N1CC(OC2CCN(C)CC2)C1 c1(NCc2cccc(-c3ccc(C(C)(C)C)o3)c2)ccsc1C#N N#Cc1ccc(C(=O)NOCC2CCOCC2)o1.N12CCCCC1NC(=O)C2=O N1(C(C2C(C3C(C)C3)C2)=O)CCC2(COC(CNC(c3ncn(C)n3)=O)C2)C1 Cc1cc(C(=O)N(CCCCN(C)C(C2C=CCC2)=O)C)c2ncccc2c1 c1(C(=O)NC(C2CCCC2)CNC(C2CSCCS2)=O)c(F)ccc(F)c1O N1(C(c2n(C)cnc2)=O)CC2CCN(C(=O)COc3ccc(Cl)nc3)CC(C2)C1 Cc1cc(F)ccc1NC(=O)C(c1cc[nH]n1)N(C1(C)CCS(=O)(=O)C1)C CC1CCOCCN1C(C1(C(C)NC(c2cnc(C(C)C)o2)=O)CC1)=O C1(CNC(=O)CC2OCCO2)C2CN(C(=O)CN3CCC(C(N)=O)CC3)CC12.C1=C(C)S1 Cc1cc(C)c(C(=O)NCC2CCCC2NC(c2cnc(S)n2C)=O)c(C)n1 CCS(=O)(=O)c1ccccc1C(=O)NC1CCCCCC1NC(c1cocn1)=O C1(C(C)(C)C)CN(C(=O)C(C2CCCCC2)F)CCN1C(c1ccc(N)cn1)=O C=CCC(CC(F)F)C(=O)NC(C1CCCN(C(c2cc(C)nc(C)n2)=O)C1)C N12CCCC(C)(C1)C2C(=O)NC(C)(C)C.c1(C(=O)NC2CCC2)csc(CO)n1 N1(C(C2(CNC(c3cn(C(C)(C)C)nn3)=O)CCC2)=O)CC2(CC=CC2)C1 c1(C(=O)NCCCN(C(=O)C(O)C(C)(C)C)CC)ccc(OC)cc1F C1(NC(C(CC=C)NC(=O)OC(C)(C)C)=O)CCC12CN(C(C1(Br)CC1)=O)C2 C(=O)(C1=NNC(=O)CC1)NCC(C)(C(C)C)NC(CNC(c1c(C)cccc1)=O)=O c1(CC)nc(C)cc(=NCC2C3CN(C(c4cnn(CCO)c4C)=O)CC23)[nH]1 C(c1c[nH]c(=N)c(C)c1)=CC(=O)NC1C(NC(C2(C(=O)NC)CCC2)=O)CC1 c1(C(N2C(CNC(C3=C(C)CCC3)=O)CC(C)(C)C2)=O)cc2cccc(Cl)c2[nH]1 C1(NC(CC2CCC(NC=O)CC2)=O)CC2CN(C(C3(C(F)F)CC3)=O)CC2C1 c1(SCC(=O)NCC2C(NC(c3c(C)cc(CC)o3)=O)CC2)cc(Cl)ccc1Cl C(=O)(CC(C)C(=O)N1CC(NC(c2oc(CC(C)C)nc2C)=O)C(C)C1)OC C1(CC(=O)NC2CC(NC(c3c(SC)cn(C)n3)=O)C2)CC2(CCOCC2)CO1 N1(C(c2c(C)cco2)=O)CC2CCCC(NC(c3cc[nH]c3C)=O)C2C1 N1(C(C2(CC)CC2)=O)CCC2(CC(NC(=O)C(c3ccc(Cl)c(F)c3)O)C2)C1 C1(NC(c2cnc(C)[nH]c2=N)=O)CCCC12CN(C(=O)C(O)CC(C)C)C2 C1(C)(CNC(c2cc(CNC(c3cnn(C)n3)=O)on2)=O)CCC(=O)N1 N1(C(C(C)SCC)=O)CC(NC(c2csc(CCP(C)(C)=O)n2)=O)CC(F)C1 C1(CCC)CN(C(C2CCC(=O)C2)=O)CC1NC(C1(CC)CCCO1)=O c1(C(=O)NC(COC)C(=O)NCCn2nc(C)cc2C)cc2ccccn2c1 N1(C(CCC=CC)=O)CC2(CCN(C(=O)Cn3ccc(C)n3)CC2)C1C(C)C C1(NC(CCC=C)=O)CCN(C(=O)CCCc2csc(=N)[nH]2)C12CCC2 N1(C(CC2CC(C)C2)=O)CC(F)(F)CC1CNC(C1(CO)CCOC1)=O C(C(C)(C)C(=O)N1CC2CC1C2C(=O)N(C(C)C(C)SC)C)OCC N1(C(c2nc(C)nn2C)=O)CCOC2(CCC(NC(=O)C(C)C(C)(F)F)CC2)C1 n1(CC(=O)NC(C)(CNC(C2CCCS2)=O)CO)cc(C(N)=O)c(O)nc1=O c1(NCc2ccc(C(=O)OC)nc2)ccc(F)c(O)c1F.N12CC3CC3(C1)C2=O N1(C(CCn2c(C)cc(C)n2)=O)CCC(NC(c2cc(Cl)n[nH]2)=O)C12CC2 C1(C(=O)NCC(C(C)C)NC(c2ccc(C(C)O)cc2)=O)CCS(=O)(=O)C1 Cc1cc(C)n(CC(N2CC3C(C(=O)NCCC4CCOC4)C3C2)=O)n1 c1(C(N2CC(NC(CC3CC(=C)C3)=O)C(SC)C2)=O)c(C)cc(F)cc1Br N1(C(=O)C=CC2CCCO2)CCN(C(c2ccc[nH]2)=O)C2(CC2)C1 c1(C(N2C(C)(CC(=O)NC(COC)CCO)CC2)=O)cnc(S)nc1 C(CNC(=O)CCn1cc(C)cn1)(CCCC)NC(COCCC=C)=O c1(CN(C(c2ccn(CCC)n2)=O)C)ccc(Cl)cc1Br c1(C(=O)NCC2(C(=O)NCCC)CCCC2)cc(C)cc(O)c1 Cc1cc(Cl)c(C(=O)NC2CCCN(C(=O)C(C)(C)C3CCOC3)CC2)cc1F C(=O)(CC(F)(F)C(F)(F)F)N1CC2CC(NC(C=CCC)=O)CC2C1 N1(C(CC2(C=C)CC2)=O)CC(C)CCC1CNC(c1ccc(C(C)C)nc1N)=O CC1CN(C(=O)COC2CC=CC2)CCC1NC(=O)C=CCOc1c[nH]c(Br)c1 Cc1ccc(C)c(C(N2CCN(C(=O)C(O)CCN(C)C)CC2CC2CC2)=O)n1 C1(CC)CN(C(C2(CN)CC3(C2)OCCO3)=O)CCN(C)C1 CC1=NOC(=O)C1CCC(=O)NC1CCC1CNC(=O)CCSCC(C)C C1(C(N2CCC(COC)C2)=O)CCCCN(C(c2c[nH]c(=N)o2)=O)C1 CC1CC(=O)NCCN1C(=O)CC1CC(NC(C2CC2F)=O)C1 Cc1cn2cc(C(=O)NCC(CO)NC(=O)CC3COCCN3C)ccc2n1 C(C(CN=c1ccn2ccnc2[nH]1)C(F)(F)F)NC(c1cn(C)c(=O)n1C)=O C1(COC)CCCC1C(=O)NC(C)CC(=O)OC(C)C C1(C(F)(F)C(=O)NC(C)CNC(c2nnn(C)c2N)=O)(OC)CCCCC1 c1(C(N2CCC2(C)OC(C2C(C(=O)OC)C2)=O)=O)nscc1C c1(SCC(=O)N(CC(C)NC(C2C(CC(C)C)C2)=O)C)nc2ccccc2s1 c1(C(C)C(=O)NC2(CF)CCN(C(=O)C(=O)N(C)C)C2)cccc([N+](=O)[O-])c1 CC1=C(C(=O)NC2CCC(CNC(=O)CCC(C)OC(C)(C)C)CC2)CCC1 c1(CNC(c2ccc(C)cc2C)C)nccc2c1[nH]c1ccccc21 C(=O)(C1=C(C)OCCC1)N1C(CNC(C(CSC)O)=O)CC(C(F)(F)F)CC1 c1(C(=O)NC23CC(CNC(C4(OC)CCSC4)=O)(C2)C3)coc2c1C(=O)NCC2 C1(C)(C(N2CC(NC(c3ccc(C(CC)=O)cc3)=O)C2)=O)CCCS1(=O)=O c1(CNC(=O)OC(C)(C)C)nnc(NC(C2CC(SCCO)C2)=O)s1.C1CO1 c1(CC(=O)NC2CC(CCC(=O)NCC3CC(OCC)C3)C2)ccccc1F c1(C(=O)NC(C(=O)NC2CN(CCC)C2)CO)csc(COC)n1 N1(C(c2c(C)snc2)=O)CCc2ccccc2C1CNC(c1ncccc1F)=O CN1CCN(C)C(CNC(C2(NC(c3cnns3)=O)CC(CO)C2)=O)C1 C(=O)(CCCC(=O)N(CC(c1ccccc1F)OC)C)N(CC(CNC)O)C C1(C(=O)OC2CCN(C(=O)NCCCCCO)CC2)CC2CCCCC2O1 Cn1nc(O)cc1C(=O)NC(C)CCCCNC(=O)C(c1ccccc1)C1CC1 c1(N2CC3C(N(CCO)CCO)C3C2)[nH]cnc2nc(Cl)cc1-2.CCC(O)C(C)C=O N1(C(CSC)=O)CCN(C(c2ccnc(C(C)C)n2)=O)CC(C)(C)C1 Cc1cc(C#N)ccc1C(N1CC(C)N(C(c2nocc2C)=O)CC1C)=O C1(C(=O)NCCn2c(C)nnc2)CCC(C2CC2)N1C(c1cnn(CCO)c1)=O C=CCCCC(C(=O)N(CC(C)C)C)NC(=O)C(=O)NCCOC(C)(C)C C1(C(C)C)CCCC1C(=O)NCC(C)(C)CNC(=O)COC(F)F N#Cc1cccc(C(=O)NC2(C(=O)NCC3(O)CC(O)C3)CSC2)n1 N1(C(C(C(=O)OCC)(C)C)=O)CCCC2(CC(NC(C3CC3C(F)(F)F)=O)C2)C1 N1(C(CC)=O)CC2(CC(C(N3CCC(O)CC34CC4)=O)CO2)C1 CC(CCc1cnn(C)c1O)N=c1cc[nH]cc1S(=O)(=O)N1CCC(C)(CO)C1 N1(C(c2c(CC)nns2)=O)CCCC(F)(CNC(=O)CC(C)F)CC1 N1(C(CC(C)(C)C#N)=O)CC2(C)CN(C(C3CCC3n3cccn3)=O)CC2(C)C1 C1(NC(C2C(C(=O)OC)C2)=O)CCCN(C(c2ncc(C)cc2F)=O)CC1 C1(C(=O)NC(C2CCCC2)C#C)C(NC(=O)CCCC)C1(C)C N1(C(C2CCN(C(N3CCCC3CC)=O)C2)=O)CCC(OCC)(CO)C1 N1(C(COCC(=C)C)=O)CCCC(N(C)C(c2cc(C(F)(F)F)n(C)n2)=O)C1 c1(NC(N2C(CC(=O)OC)CC(n3ccnn3)C2)=O)nc(C2CC2)n(C)n1 c1(SC)ccc(F)c(F)c1.C(=O)(C(Cc1cccc(Cl)c1)=NO)NCCNCCOC C=C(C)CC(C(=O)N(C1CCC(NC(C2CC2C#N)=O)CC1)C)OC C12(CNC(C3C(NC(=O)Cc4cccc(O)c4)CC3)=O)COC(C1)C(O)C2 C(C(C)(C)CC(=O)NC1CC1c1cncs1)NC(C1(C)CC(C)C1)=O C(=O)(CS(=O)(=O)CC)N(C(C(=O)NCCC#C)CC)CCC c1(C(N2CCC(CN(C(=O)C3=CCCCC3)C)C2)=O)c[nH]c2nc(Cl)ccc12 C1(CNC(c2ncc(CC)s2)=O)CC2COCC2N1C(c1cscn1)=O CN1CCOCC1C(=O)N(CCCNC(C1(C)CC=CC1)=O)Cc1ccccc1 C12CCCN(CC1)C(=O)CNC(=O)CCCOCC2.CCCCOCC.C(C)(=O)N CCC(N=c1[nH]c(=NCc2ccnc(C)n2)[nH]c2cc[nH]c12)C(C)C C1(N(C(C2(CC#C)CCCOC2)=O)CCO)CCC(F)(F)CC1 Cc1[nH]c(C(N2CC(=C(F)CNC(c3cccc(CO)n3)=O)C2)=O)c(C)c1C Cn1[nH]c(=NC(=O)c2c(S(=O)(=O)N(C)C)ccc3ccccc23)c2c1CCOC2 C(=O)(CCc1ncc[nH]1)NCCN(C(=O)CC1C=CCC1)CCC C(=O)(C(CC(C)C)C(C)C)NCCC1CCN(C(C=CC(CC)=CC)=O)C1 N1(C(c2cc(C)nc(O)c2)=O)CCN(C(c2cc(C(N)=O)[nH]n2)=O)CC(C)C1 c1(C(=O)NC2CN(C(c3cc[nH]c3)=O)CC2F)cccc(C(F)(F)F)c1Cl N1(C(C(CSC)O)=O)CCC(C(N2CCCC2C(O)CO)=O)C(C)C1 n1(CC)cnc2c(N(CCCNC)C)[nH]c(=NC(C)C(C)COC)nc12 C#CC1CCCN(C(=NCCC(=O)NC)NC2CC2C2CCOCC2)C1 C1(CS(C)(=O)=O)CN(C(=O)COC2CC2)CCN1C(C1CC(CCF)C1)=O Cc1ccc(C(=O)Nc2c[nH]nc2NC(c2cc(Br)ccn2)=O)c(F)c1 C1(NC(CCOC)=O)C(C)CCN(C(c2ncc(Cl)cc2Cl)=O)C1C C1(NC(C=CCC(C)(C)NC(Cc2c(C)ncs2)=O)=O)CCC(O)CC1 C1(CC)CN(C(c2c[nH]nc2C(F)F)=O)CCN1C(=O)C(C)c1cccs1 c1(C(=O)NC2CC(C)N(C(=O)CCCN=[N+]=[N-])C2)ccc(=O)n(CC(N)=O)c1 Clc1cc2c(cc1-n1ccnc1-c1cccc3ccncc13)OCCO2 C(=O)(CCCCC(=O)N1CC(O)C(O)C1CNC(C1(C)C(C)(C)C1(C)C)=O)NC C1(NC(c2n(CC)ncn2)=O)CC2(C1)CC(CNC(c1ccc(C)n1C)=O)C2 C=CC(F)(F)C(=O)NC1COCCC1C(=O)NCC1=CCCCC1 CC(C)CC(O)CC(=O)NCCCC(O)C(=O)NC1C2CCCCCC12 CC1c2c(F)cccc2CCN1Cc1cc2ccccc2nc1Br CCCC1C(=O)N1.C1(C(N(CCCOC)C2CC2)=O)CCCN1C(=O)OCC C1(C(C)(C)O)CCCN(N2CCC(c3ccccc3C#N)CC2)C1 n1(CC)ccc(C(=O)NCC2(C(C)NC(=O)C(C)C(F)F)CC2)cc1=O Cc1ncncc1C(N1CCC(NC(c2ccnc(C3CCC3)c2)=O)C1C)=O c1(N2C(CNC(c3cccc(CN=[N+]=[N-])c3)=O)CCC2)ccn2ccnc2n1 N1(CC)CC(CCOC(=O)NC2CC(CNC(=O)NC)C2)CC1=O.OC c1(NCC(C2COC(C)(C)O2)O)ccc(S(=O)(=O)NC(CC(N)=O)C2CC2)cc1F C#Cc1ccnc(C(=O)NCc2ccc(C(N3CCCC(F)CC3)=O)cc2)c1 c1(N(C)C)ccc(C(N2C(C(N3CCC(O)(C(F)(F)F)C3)=O)CC3CC23)=O)cn1 c1(OC)cc(CNC(c2coc(CNC(c3ncn(C)c3C)=O)c2)=O)n(C)n1 C=CC(CCC)CC(=O)N1CC=CC1C(=O)NCC1CC1c1cnccc1C C1(CNC(c2cc(CC)oc2C)=O)CC2(CC2)CN1C(=O)Cc1cccc(Cl)c1 N(C(=NCC1CCC1)N1CCC(O)C1)CCc1ccc(OC)c(OC)c1 CCC(COC)C(=O)NCc1nc(CCCNC(=O)Cn2nc(C)cc2C)cs1 CCCC(O)C(=O)NCCC(C)N(C(=O)CCOCC(=O)OC(C)(C)C)C c1(C(=O)NCC2CCN(C(CN3CC(C)(OC)C3)=O)CC2)cccc(CO)c1C c1(C(=O)NCC#CC(=O)NC(C)COCC2CC2)cn2ccccc2n1 c1(CCC(=O)N(CC(CC)NC(=O)C(C)N2CCC2)C)conc1C S(=O)(=O)(c1cccs1)NCC(=O)NCC(C1CC1)NC(=O)CSC1CC1 C1(C(=O)NC2C(CNC(=O)CN3CCC(O)CC3)C2)CN2CCCC2CO1 c1(NC(C2CN(S(CCOCC)(=O)=O)C2)=O)cnc(OC)nc1C C(CS(=O)(=O)CC(=O)N1CCC(O)(CCNC(=O)C(c2cncnc2)C)C1)OC N1(C(c2c(C)nc(O)[nH]2)=O)CC(O)(C2(CNC(C3COC(C)C3)=O)CC2)C1 C#CCCCCC(=O)N1CCC(CN(C(c2ccnn2CCF)=O)C2CC2)CC1 n1(CC(=O)NCCCOC)c(-c2ccc(Br)cc2)csc1=Nc1sc(C)nc1C C(=O)(CS(=O)(=O)C1CC1)N1C(C)CN(C(=O)C=Cc2cnccn2)CC1 C1(NC(C=CCCC2C(C)(C)C2)=O)CCCN(C(c2nonc2N)=O)C1 C1([Si](C)(C)C)(CNC(CN(CCC)C(c2cncc(OC)n2)=O)=O)CC1 C1(C#N)(C(=O)NC2(CNC(C(CCOC)C)=O)CCOC2)CCOCC1 C(CC(C)(C)C(=O)N1CCN(C)C(C(N2CC(N3CC(O)C3)C2)=O)C1)SC Cc1ccc(NC(=O)CCn2cc(C(N3CCN(CCO)CC3)(C)C)nn2)c(F)c1 CC1(C2CCCN(C(C(=O)NCCCF)C3CCCC3)C2)CC1 O=S(=O)(c1ccc(NC2CCC3(CC3)C2)c(F)c1)NC1CCn2ncnc2C1 N1(C(C(C=C=C)C)=O)CCCC(C)(CNC(c2nc(C3CC3)ncc2Cl)=O)C1 c1(CC)cccc(C(N2CCC(C)(C(=O)N(C)Cc3ccc(C)nc3)C2)=O)c1O C1(CNC(CCCCCSC)=O)CN(C(c2cnnc(C)c2)=O)CC2(CCC2)O1 c1(C(=O)NC2(CO)CCN(C(CNS(NC)(=O)=O)=O)C2)nc2cc(F)ccc2s1 Cn1cc(C=CC(N2CCC(NC(=O)CN3CCCC3CO)C2)=O)nn1 c1(C(N2C(CN(C(CCOCC#C)=O)CC)CCC2)=O)cc(OC)n(C)n1 c1(CC(=O)NC(CCNC(C=C(C)c2cccs2)=O)C)ccc2nc(O)[nH]c2c1 CCCC(C)C(=O)NCc1nc(CNC(=O)C(C)OCCOC)cs1 C1(C(=O)NOCC2CCCO2)CN(C(=O)CC2CCSC2)CC12CCC2 c1(C(N(CC(CC)NC(=O)COCCOC)C)=O)n[nH]c2ccccc12 c1(C(N2C(C(C)C)CCC2)=O)ccc2c(c1)CN(C(c1cnn3c1CCC3)=O)C2 N1(C(c2c(C(=O)OC)nccn2)=O)CC2CC1CCN2C(C1CCCN1C=O)=O C(C(C)(O)CNC(C1CC(C#N)C1)=O)NC(CC1C(C)CC1)=O C(=O)(C1CCCc2nncn21)NC1C(NC(COc2cccc(C)c2C)=O)C1 C12(C(=O)NC3COCCN(C(c4ccnn4C(F)F)=O)C3)CCCN(CCC1)C2 c1(CC(N2CCC(OCCNC(C3C(OC)(OC)CC3)=O)C2)=O)ccc(C)cc1 c1(C(N2CCC(C(CO)N(C(C(=O)N(C)C)=O)CC)CC2)=O)c(F)cc(F)cc1F c1(-n2cc(C3N(C(Cc4c(C)cccc4)=O)CCOC3)nn2)ccc(Cl)cc1F c1(OC)ncc(NC(=O)C(=O)NCCCCS(C)=O)cc1C C#Cc1ccc(C(=O)NC(C)(C)C(C)NC(C2CN(C(C)C)C2)=O)cc1Cl c1(OCC)cc(C(=O)NC(C2CCCOC2)CNC(c2cncc(C)n2)=O)ccn1 CC1=C(C(=O)N2CCC(CNC(C3(Cl)CC3)=O)C(F)(F)C2)CCCO1 c1(C(=O)NCCN(C(=O)C=Cc2nc(C)c(C)[nH]2)CC)cnc(C(C)C)nc1C N1(C(CC2N(C(c3oc(CC)c(C)c3)=O)CCC2)=O)CC(C2CC2)(OC)C1 c1(CC(=O)NCCN(C(=O)C(O)C(C)C)CCCN)ccnc(Br)c1.CO N1(C(CC2CCC(=O)NC2)=O)CCN(C(=O)C(=O)Nc2ncc[nH]2)C(CCO)C1 C1(C(=O)NCC2CCCN(c3nc(C(C)(C)C)ns3)C2)(OC)CS(=O)(=O)C1 c1(C(N2CCN(C(CC(C)(C)O)=O)CC2CO)=O)nc[nH]c2ncc(Br)c1-2 C#Cc1ccc(Br)c(C(N2CCCC2C(C)NC(=O)CC2(O)CCOC2)=O)c1 c1(CNC(=O)NC(C(=O)OCC)Cc2cscn2)cc(Cl)ccc1Cl n1(CC(=O)NCC2(F)CCC(NC(CCC#C)=O)C2)ccc(=O)c(O)c1C C1(C)(CNC(C(C=C)C)=O)CN(C(=O)C(C)C2CCC2)CC1C N1(C(C(C(C)C)F)=O)CCN(C(=O)CC(C(F)F)n2cccn2)C2(CCC2)C1 C1(CC(=O)NC(C(=O)NC(C)Cc2ncn(C)n2)CO)CCC(C(F)(F)F)C1 CC1C(NC(C2CC(N=[N+]=[N-])C2)=O)CCN1C(=O)CCn1ccc(=N)[nH]1 C1(COC)CCCN(C(C2CC(OC)CN2C(c2[nH]nc(OC)c2Br)=O)=O)C1 C1(C(=O)NC(C)(C)C=CC(=O)N(C2CCCCC2)CCO)CCCC1(C)C C12(C(=O)NC3CC(CNC(C4N(C)CCCC4)=O)C3)CCCCC1OCC2 C=C(C)CC(C(=O)N(CC(O)CN(C)C)C)NC(c1cc(OC)ncn1)=O C1(NC(C2(c3cc[nH]n3)CCC2)=O)CCOCC1C(=O)NCCC(F)F C12OCCC1C(=O)NC2.c1(C(=O)NC2CN(C)C2)cc(Cl)n[nH]1 CC1CCc2[nH]c(=NCCC(F)(F)Cl)[nH]c(=NCC3CCC4(CC4)CO3)c2C1 Cc1cc(C(=O)NCC2CCCN2C(=O)C(C)C2(O)CCC2)nn1C(C)C1CC1 c1(C(N(CC(=O)O)CC2CCOC2)=O)cc(CO)[nH]c1C1CC1 C(CC(C)C(=O)NC(C)CCC(=O)N1CC(c2nncs2)C1)OC c1(NC(C2CC(C(C)C)C2)=O)cc(CNC(=O)COC2(C)CCCC2)on1 C(=O)(CCCCC(F)(F)F)NC1(C)CCN(C(C2CCCCC2O)=O)C1 Cc1ccc(C(N2CCC(CNC(C3(Br)CC3)=O)C(C)C2)=O)c(C2CC2)c1 C(N=c1[nH]c(=NCc2ccc(F)c(F)c2)[nH]c2c1COC2)C1C(C(C)C)C1 N1(C(=O)Nc2cccc(COC)c2C)CC2CC(N3CC(F)C3)CC1C2 C1(C(C)C(=O)OC(CO)C2CC2)CCC(F)(F)CC1 C1(NC(C(C)c2cc[nH]n2)=O)CCC(NC(=O)CC=C(Cl)Cl)CC1 N1(Cc2c(C)cccc2F)CC2(CN(C(c3ccccc3Br)=O)CC2C(=O)O)C1 C1(C2CC2)(NC(c2c(C)nn(CC(F)F)c2)=O)CCN(C(=O)C(O)C(C)(C)C)C1 c1(C(=O)NC2C(NC(c3ncc(C)nc3)=O)CC2)ccc(F)c(C(C)C)c1 C(=O)(C(C)CS(C)(=O)=O)N(C1CN(C(CC2[N+]([O-])(CC)CC2)=O)CC1O)CC C1(C#N)(C(N(C2CCCN(C(CCSCCCC)=O)C2)C)=O)CC12CCCC2 c1(C(C(=O)NC(C)CCNC(=O)C(C)c2ccco2)O)ccc(C2CC2)cc1 c1(C(=O)NCC(CN(C(C2C(C)OC(C)C2C)=O)C)C)ccc(S(N)(=O)=O)o1 N1(C(C=CC(C)C)=O)CCC2(CC2C(=O)NC2CC3OC(=O)CC23)C1 C1(CCNC(CCNC(=O)NC)=O)COCCN1C(C1COC(=O)O1)=O C1(C)(C(=O)NC2CC(C)(CNC(C3(Br)CC3)=O)C2)CCC(=O)C1 C#CC1(NC(=O)C(c2ccco2)NC(=O)C(c2ccnn2C)C)CCOC1 c12cc(OC)c(cc1[N+](=O)[O-])OCCCO2.C(CCC)(N(C(C)=O)C)C1CC1 Cc1[nH]nc2ccc(C(=O)N(CC(C)N(C(=O)Cc3nnc(O)s3)C)C)cc12 CC1(CNC(C2CC3CC2C3)=O)CCC(NC(c2ccc(C(F)(F)F)nc2)=O)C1 C1(NC(CCc2cc(C)no2)=O)C=CCC(C(N2CCC(N3CC(O)C3)C2)=O)C1 C=C1COc2c(C(N3CCCC3CNC(c3ccon3)=O)=O)cnn2C1 C1(C)(N(C)C)CCCN(C(Cc2ccccc2)C(=O)NCSC2CCCCC2)C1 C=Cc1cncc(C(C(=O)NCCC(C)CC)N(C)CC2CCCO2)c1 C(=O)(C(CNC(=O)CC1CN(C(C)=O)C1)C(C)(C)C)NC(C(C(=O)OC)C)C C1(CNC(C(C)OCCCC)=O)CN(C(c2cc(Cl)cs2)=O)CCC1C c1(OC)ccc(C)nc1C(N1CC(NC(c2cc(Cl)nnc2O)=O)C2(CC2)C1)=O c1(-c2nc(COC)nn2C2CC2)n[nH]c2c1CN(C(C1CCCCC1)CSC)C2 C1(CNC(c2ccnc(Cl)c2F)=O)CCN(C(=O)Cc2cc(Br)cs2)CC1(F)F c1(C(=O)NCC(C)(O)CNC(c2csc(S(C)(=O)=O)c2)=O)cccc2occc12 Cc1ccc(C(=O)NCC(O)CCNC(=O)C(c2cnn(C)c2)O)nc1C Cn1c(C(N2C3CCCC2CN(C(=O)CCn2ccnc2)C3)=O)cc2ccsc12 N1(C(c2ccn(CCOC)n2)=O)CC(C)N(C(=O)COCP(C)(C)=O)CC1C C1(NC(C(CCN(C)C)NC(=O)C(F)C2CCC2)=O)CCC2CC1CO2 CCCCC(CC(=O)N(CC(C)(C)C)C)NC(c1coc(CC)n1)=O C1(CCC(=O)NCC(C)NC(=O)C(C)NS(C)(=O)=O)CCCCN1C C(=O)(CN=c1cc[nH]cc1)NCC(N(C)C(C1CC2(CCC2)CO1)=O)C1CC1 O=C(CN=C(NCc1ccc(F)cc1Cl)NC1CC12CC2)N1CCCCC1 c1(C(N2CC3C(NC(COCC)=O)C(C3)C2)=O)cnc2ccnn2c1 C1(CNC(C2N(S(CC)(=O)=O)CCC2)=O)CN(C(C2(n3cccn3)CC2)=O)CCO1 C(=O)(C1COc2c(C)cccc21)NC(CN(C(=O)Cc1cc[nH]n1)CC)C C(=O)(C(C)(O)C(C)(C)C)NCC(C)NC(c1ccn(CC(F)(F)F)c(=O)c1)=O CC1(C)CCCN(C(=O)CC2COCCO2)C1C(=O)NCC12CCCC1OCC2 CC1(C)CCC(n2cc(CC3CCNC3=O)nn2)CN1C(C1(CC2CC2)CC1)=O N1(C(C=CCC)=O)CCC2CC(NC(=O)CC(C)(C)CC)CCC2C1 C1(OCC(=O)OC(C(=O)NC(CC(C)N(C)C)C)C2CCC2)CCC(F)(F)CC1 C1(CC(=O)N(CCCN(C(c2cc(CN(C)C)on2)=O)C)C)OCCOC1(C)C C(=O)(C(C1=CCCSC1)N1CC(N(C)C)CCC1C)NCCC(=O)OCC N1(C(c2cc(C)nc(O)c2)=O)CC2CCCC(Nc3cc(Cl)ncn3)C2C1 n1(CC)nnc(C)c1C(=O)NCCOCCNC(C1(C)CC1(F)Cl)=O CCCC(C(=O)OC(C1CC(n2ccnc2)C1)=O)c1cccc(Cl)c1 N1(C(C(C(=O)OC)C)=O)C2CCC1CN(C(=O)CC1Cn3ccnc3NC1=O)C2 c1(C(=O)NC(C(C)NC(c2cc(C)nc(O)c2)=O)(C)C)coc2ccccc12 C(C(C)(C(C)C)NC(=O)C(C)Cc1cnc[nH]1)NC(CC1(CSC)CC1)=O CC(CC(=O)NCC1CCCCC1NC(c1ccn(C2CCC2)n1)=O)P(C)(C)=O N1(C(c2cccc(OC)n2)=O)CCC2(CC1)CCN(C(c1ccccc1C)=O)C2 C1(C)(C(N2CC(NC(c3c(C)nn(C)c3Cl)=O)C(C)CC2)=O)CCCCC1(F)F N1(C(C(C)OCCOC)=O)CC(C)(C)OCC1C(=O)NCCC(=O)NC(C)C O=S(=O)(c1ccc(OCC2CCCO2)c(F)c1)NC1CC2CNCC2C1 C(CCCN=c1[nH]c(Cl)ncc1Cl)NC(C1C(C)CC(C)O1)=O C1(C(=O)OC)CN(C(=O)C(Cl)(Cl)Cl)CCN1S(=O)(=O)Cc1ccc(OC)cc1 C1(C(N(C(C(N)=O)C2CC2)C)=O)CN(C(=O)C=Cc2nccs2)CC1F C1(C#N)(CCCCCO)CCN(C(=O)OC(C)(C)C)CC1.C(=O)(CC)NC C1(C(C)NCCC2CCCC2)CCCCN1C(c1cnnc(O)c1)=O c1(C(N2CC=CC(NC(C(COCC)C)=O)C2)=O)cccc(Br)c1[N+](=O)[O-] c1(C(C(=O)Nc2cccc(C3CC3)c2)N(C)CCO)cc(Cl)nc(Cl)c1 c1(C(=O)NC2CC(CCNC(c3cc(-c4ccco4)[nH]n3)=O)C2)cccnc1O N1(Cc2ccc(CC(=O)O)cc2)CC2CC3CC2C1C3O N1(C(COC)=O)CC(NC(=O)Cc2nc(Br)sc2C)CC1C c1(-c2onc(-c3ncc(C)c(Br)c3)n2)cnnc2ccccc12 C=CCC(C)(C)CCNC(=O)C(C1CCOC1)NC(=O)CCOCC(C)(C)C Cc1ccc(N)cc1S(=O)(=O)NCC(O)CN1CCCC(C)C1 C1(C(=O)NC(CC(=O)N(CC#C)CCO)C)CC(=O)C1(C)C c1(C(N2CCN(C(=O)CCCF)CC2CF)=O)cccc2nc(O)oc12 C1(NC(CC2(C=C)CC2)=O)CCCN(C(=O)CCOc2cc(F)cc(F)c2)CC1 c1(C(N2C(C(=O)Nc3cccc(C#C)c3)C(O)CC2)=O)cc(C)c(F)cc1C c1(C(N2C(CC)C(C(=O)NCc3ccccc3O)CC2)=O)ccc([N+](=O)[O-])[nH]1 N1(CCC(=O)NC2(CO)CCCN(C(C3C=CCC3)=O)C2)CCc2ccccc21 C1(C(N(CCCO)C(C)C)=O)(CNC(=O)Cc2ccccc2O)CC12CCC2 N1(C(C=NOC)=O)CCC(C2CN(C(c3cncc4nc(O)[nH]c34)=O)C2)CC1 C1(COC)(CNC(=O)C(CO)N(C)C)CCCN1C(=O)CCNC(=O)C=CCl c1(C(=O)NC(c2cccc(F)c2)C)ccc2c(-c3cccc(F)c3)n[nH]c2c1 N1(C(CCSCC)=O)CCCC2(CNC(=O)C=C(C)C)CCCC12 N1(C(C(CC)CN)=O)CCC(C2CNCCO2)CC1 C1(O)(CNC(C2CCN(C(N)=O)CC2)=O)CCN(C(=O)CSC2CC2)CC1 c1(CC(=O)NCC(CC)NC(=O)C(C)OCCC(C)C)nc(C)c(C)s1 c1(OC)ccc(C=CCNC(=O)NCCO)cc1OC(=O)C(F)CC(C)(C)C Cc1n[nH]c(C)c1C(C)C(=O)NC1(CNC(c2ccc(Br)o2)=O)CCCCC1 C1(C(N2CCOCC2CCO)=O)(OC)CCCN1C(=O)C(C1CCCCC1)O c1(OCCCC(=O)OC)cccc(Cn2cc(CNC(C3CCCS3)=O)nn2)c1 c1(CN2CC(C)(CC(=O)NC(C(=O)OC)(C)C)C2)cc(Br)cnc1O C1(CCNC(C2CCCC23CCC3)=O)CCCN(C(=O)C=Cc2cnc[nH]2)CC1 Cc1c(C2(C(=O)NCC(O)CNC(=O)CSc3ccccc3)CC2)cccc1F C1(NC(CC(C)C2CC2)=O)CC2CN(C(=O)CC3CN4CCC3CC4)CC2C1 c1(C(c2nnnn2Cc2nnn(C)n2)NCC=C)nn(C)cc1Cl C1(CNC(C2N(C(C)=O)CC(O)C2)=O)(NC(=O)C=CCOC)CCC(C)(C)CC1 c1(CNC(=O)NCC23CC(CO)(C2)C3)ccc(F)c2occc12.n12cc(nn1)C2 C1(C(N2CCCN(C(CC3(C#C)CC3)=O)CC2)=O)COc2cccc(OC)c2C1 c1(C(=O)NCCc2cnc(NC(C3(C)CCCN3)=O)s2)c(Cl)cccc1I c1(C(N2C(CNC(C(=O)N(C)C)=O)CC3(CC3)C2)=O)n[nH]c2c1CC(F)(F)CC2 c1(C(N2CCC(N(C(C(CSC)O)=O)C)C2)=O)cccc(-c2ccccn2)c1C C(CCCCCNC(c1ccns1)=O)NC(Cc1nc(NC=O)sc1)=O N1(C(C#CC2(C)CC2)=O)CCC(C2CN(C(=O)CCC3CCCC3)C2)C1 C1(C(=O)NCCC(C)(C)NC(CN2CCN(C)CC2)=O)CCCC1S(C)(=O)=O n1(CC(=O)OCC(C2C(OC)CCC2)=O)nnc2ccccc2c1=O O=C(CS(=O)(=O)CC1CCCO1)NCC(O)CCNC(c1ccoc1Cl)=O C12CCCC(C1)C(=O)N2.N1(C(C(C)(F)F)=O)CCOCC1CC(=O)N(C)C Cn1cncc1CCC(=O)NC(C1CCN(C(C2CNC(=O)C2)=O)C1)(C)C Cc1cc(F)c(NC(C2CCCN2Cc2cnc(C3CC3)s2)=O)cc1F C1(C(=O)Nc2nc(C3CC3)cs2)CC2C(C1)C2(F)F C1(NC(=O)CC23CCCC2C3)CN(C(=O)Cn2cc(CO)nn2)CC12CC2 N1(C(=O)CCCn2cc(CC3CCCNC3)nn2)CCCc2ccccc21 c1(NC(CCc2[nH]nc(SC)n2)=O)c(C)nn(C(F)(F)F)c1C C1(NC(C2(SCC)CC2)=O)CN(C(C23C4C5C2C2C3C4C52C)=O)CCC1(C)C C(C)(N=c1[nH]c(N2CCSCC(C)C2)nc2c1SCC2)c1c(COC)cccc1 c1(C(C(=O)N(C2CCC(NC(=O)CCC=C(C)C)CC2)C)CO)ccc(Cl)cc1 NC(=O)CCCCC(=O)NC1CCC(NC(=O)C=Cc2cccc(Cl)c2)C1 c1(N(C(=O)C(CO)NC(=O)C(C2(C#N)CCC2)N2CCCC2)C)ccccc1F N1(C(CCC=C)=O)CC2(C1)CN(C(c1cc(C(=O)OC)[nH]n1)=O)C2 C1(CNC(C(C)SC)=O)CCCC2CN(C(=O)CC3C=CS(=O)(=O)C3)CC12 c1(C(=O)NC)n[nH]c(C)c1[N+](=O)[O-].C(=O)(CCCCCN(C)C)N(CC(CC)OC)C N1(C(C2CC(C)=C(C)CC2)=O)CCCC2(CCN(C(=O)C(F)(F)C3CC3)CC2)C1 c1(CC(=O)NCC2N(C(C(C)OCC)=O)CCC2C)ccc2c(c1)CCCC2 C=C(C)CCC(=O)NC1CCCC1CNC(=O)CCC12CCC(CC1)C2 C(=O)(C(CCCOC)N1CCCC(n2cc(CSC)cn2)C1)NC c1(CC(=O)NC(C)CN(C(=O)Cc2nnc(S)n2C)C)coc2cc(O)ccc12 C(=O)(CCC(F)(F)F)NC1CC(C(C)NC(=O)C2=NOCC2)C1 c1(CN(C(CC)=O)C)ccccc1CNC(C1(C2CC2)CC1)=O N1(C(C2CC(OC)C2)=O)CCC(O)(C(=O)Nc2cn(C)nc2C#N)CC1 c1(CCC)cccc(C(=O)NC(CNC(=O)CC2CC2CC)C2CC2)c1 N1(C(CCOCCN(C)C)=O)CC2CN(C(C3(O)CCOC3)=O)CCC12 N1(c2nccc(N3CCCC(c4nnc(CC)s4)C3)n2)CCCC2CCCCC12 CC(F)CN=c1[nH]c(N(CCCN(C)C2CC2)C)nc2c1CCCC2 C1(N(C(c2cnc(OCC)s2)=O)C)CC2CC1N(C(c1ccc3nc1CC3)=O)C2 Cc1nc(SC2C(C(=O)O)C2C(F)(F)F)sc1CC(=O)OC(C)(C)C N1(C(COC(CC)C)=O)CCC(CCOC)(C(=O)NCc2cccc(Cl)c2)C1 C=CC1(C(N2CCCC(CC)C2)=O)CCN(C(c2ccc(OC)o2)=O)C1 Cc1nc(CC(=O)NCC(C)NC(=O)CCCN(C)C)c(C)s1 c1(CC)cc(C(N2CCN(C(C3CC=C(C)CC3)=O)CC2C)=O)cc(O)n1 c1(C(=O)NCC=CCNC(CCNC(=O)OC)=O)cc(C)n(C2CCC2)n1 c1(C(CNC(c2c[nH]nc2C2CCC2)=O)NC(C(C)C#N)=O)cccc(Cl)c1Cl c1(NC(C2(C)N(C(C(C)C(F)F)=O)CCC2)=O)ccc2nncn2c1 Cc1c(C(=O)N(CC(C)O)CCNC(c2ccc(C#N)[nH]2)=O)nn2c1CCCC2 c1(C(=O)NCC2CC(NC(C(C)(C)C3CC3)=O)C2)ccc(N)c([N+](=O)[O-])c1 N(C(=NCCCCl)NC)N1C(C)CCCC1.C1CC(S(C)=O)C1 N1(C(c2ccc(O)nc2Cl)=O)CCOCC2(COCCN2C(=O)C(F)F)C1 N1(CC(N2CCN(c3cc(F)ncn3)CC2)=O)CC(=O)NC1=O C1(C(=O)OCC)CC=CC(c2cn(C3CN(C(c4[nH]cnc4C#N)=O)C3)nn2)C1 N1(C(Cc2ccc(C(N)=O)cc2)=O)CCC2(NC(=O)CSC(F)(F)F)CC2C1 c1(CCNC(=O)NCc2snc(C(C)C)n2)ccc(F)c(C(F)(F)F)c1 c1(N(C(c2ccccc2)CNC(=O)CN(C)C(=O)OC)CC)ccccc1 c1(C(=O)NCCN(C(COCCCCC)=O)C(C)C)c(N)cccc1F Cc1cc(Cl)ccc1OCC(N1CCC(NC(C2CCC(O)C2)=O)C(C)C1)=O Cc1nc2ncnn2c(N(CC(C)NC(c2cnc(C(F)(F)F)cn2)=O)C)c1C N1(CC(N2C(CNC(CCC(=C)Cl)=O)CC(OC)C2)=O)CCCCS1(=O)=O N1(C(CC(C)(C)C2CCOCC2)=O)CCOCC(n2cc(C3(CO)CC3)nn2)C1 N1(C(C(CC)OC2CCCC2)=O)CCC(CNC(C2CCC(O)CC2)=O)C1(C)C C1(n2c(-c3cccnc3C)nc(C(CC)C)n2)CCS(=O)(=O)CC1 N1(S(CC)(=O)=O)CCc2cc(OC3CN(C(c4cc(Br)cnc4F)=O)C3)ccc21 C1(COC)CCCCN1C(=O)CC(=O)N1CC(N2CCS(=O)CC2)C1 Cn1cc2ccc(C(N3CC4(CC(NC(c5csc(Cl)n5)=O)C4)C3)=O)cc2n1 c1(C(=O)NC2CC(CNC(C(C)N3CCC3)=O)C2)c(F)c(F)cc(F)c1F C1(c2n(C(C)C)nnn2)(NCC2(C(C)(F)F)CC2)CCC(C#N)C1 C1(NC(c2c(CC)n(C)nc2)=O)CCC2(CCN(C(=O)C(C)N=[N+]=[N-])C2)C1 C12(C(N3C(CNC(CCOCC#C)=O)C(CC)CC3)=O)CC3CC1C2C3(F)F C(=O)(CCCCC(C)(C)C)N1CCC(C(C)NC(C(CCCC)(C)F)=O)CC1 N1(CCN(C(C(COC)C)=O)CC2CCCN2)CCCS1(=O)=O C1(NC(C=C(CCC)C)=O)C2CCC1N(C(c1cc(C)n(CC3CC3)c1C)=O)C2 c1(C(=O)NC2CCN(C(c3c(C)nn[nH]3)=O)C2)cc(Cl)ccc1OC(C)C C(=O)(C(C)(C)C1CCCN1C(=O)CC1CNC(=O)C1)N(CCCN(C)C)C N1(C(c2n(C)ccc2)=O)CC2(CC2)CC1C(=O)NOCc1cccc(F)c1 N1(C(c2onc(C)c2C)=O)CC2CN(C(c3cc(CS(C)(=O)=O)c(C)s3)=O)CC2C1 N1(C(C2C(NC(N(C)C)=O)CCCCC2)=O)Cc2ccncc2C1 c1(C(=O)NCCC2CCCN2C(=O)CCC2CCC2)c(F)ccc(O)c1F N1(C(CCOCCC)=O)CCCC(NC(c2ccncc2C)=O)C1C N1(C(CCC)=O)CC(C)C1C(=O)NC(C(F)(F)F)c1ccccc1 c1(CC)ccc(C)cc1C(N1CCC(O)C(N(C)C(C2CC(CC)C2)=O)C1)=O c1(SCC(=O)N(C2CCN(C(C3CC3C3CCCO3)=O)C2)CC)cccc(C)c1 c1(CC)c(C(=O)NCC(O)CNC(C2(C)CCCNC2=O)=O)cccc1C c1(C(=O)NC2CCC(NC(C3(C#N)CC3Br)=O)CC2)ccc(F)c2ccncc12 C1(CC)CCN(C(=O)CC2CCCOCC2)C(C(N2CCCC(OC)C2)=O)C1 Cc1ccccc1CNC(C1CCN(C(=O)C(C)n2ccnc2)C1C)=O C1(CC(N)=O)CCCN(C(=O)Nc2ccc(Oc3ccc(Cl)cc3)cc2)CC1 C1(CC)CCN(C(=O)NC2CC(OC)CC(C(C)(C)C)C2)CC1(C)OC CCCC(C(=O)N1CCC(NC(c2ccc(CC)s2)=O)C1)OCC Cc1nn2c(c1C(=O)NC1(CNC(c3c(F)ccc4occc34)=O)CC1)CCCC2 C(=O)(C(CC)C(C)(C)CC)N1CCCC(F)(C(=O)NCC(=C)Cl)C1 c1(CNC(c2nnnn2C(C)C(=O)OCC)CCC)cccc(Br)c1OC CC(C)CC(CNC(=O)C(F)C1CCC1)C(=O)NCCS(N)(=O)=O C1(CNC(c2c(CC)cccn2)=O)CN(C(c2nnsc2C)=O)CCC12CCC2 N1(CC(C(=O)NCc2cnoc2)C(C)NC(CCNC(C)=O)=O)CCC(C)CC1 C(=O)(C(C)CC(F)(F)F)N(C1CCC(OC)CC1)C(C1CC1c1cccs1)=O C#CC1(C(=O)NCC(C)SC)CCN(C(=O)CC=CCCCCC)CC1 CC1(CNC(C2(c3cncnc3)CCCC2)=O)CCN(C(C2CC2(F)F)=O)CC1 c1(C(N2CCN(CC(C3(C)CC(F)C3)=O)CC2)=O)ccc(-n2ccnc2SC)cc1.CO CCCC(C(=O)NC1(C(=O)N(C2CCCC2C#N)C)CCC1)OCC N1(C(CCCC#CC)=O)C2CCC1CN(C(=O)CCC(C)c1ccccc1)C2 Cc1ccc(C(N2CCC(O)C(NC(=O)Cc3cccc(F)c3)C2)=O)c(O)c1 CC1CCN(c2ccc(NC(=O)N(CCCN)C)cc2)CC1 CC1(C)CC(NC(=O)C(Cc2ccoc2)NC(C2CCS(=O)CC2)=O)C(C)(C)O1 C(=O)(CC1=CCCCC1)NC1CC(N(C)C(c2cncc(F)c2)=O)C1 CCCCCC(CNC(C1(C)CC1C(F)(F)F)=O)CO S(=O)(=O)(CCC(=O)N1CCN(C(C2C(F)(F)C23CCC3)=O)C(CCO)C1)N(C)C C(=O)(C(F)(F)CC(C(=O)OC)NCCC(C)N(C)C(=O)OC(C)(C)C)OCC CC1CCC(C(=O)NCC2CCC3(CC2)CC3)CN1C(c1ncc(F)cc1F)=O N1(C(c2c(C)nco2)=O)CC(C(=O)NCCN2C(=O)CCC2=O)C(C)(C)C1 c1(C(=O)NC(c2noc(-c3ccc(F)cc3)n2)CCC)cc(S(N)(=O)=O)oc1C C1(NC(C(CCC)c2cccc(Cl)c2)=O)COC2(CCN(C(=O)CSC)CC2)C1 C(=O)(CCC[N+](=O)[O-])N1CC(OCC)C(CNC(=O)CCc2cc(C)nn2C)C1 c1(C(=O)NC2C(C)(NC(C(CCC)O)=O)CCC2)ncc([N+](=O)[O-])cc1C c1(OC)ccnc(OC)c1C(=O)NC(CO)C(C)NC(=O)C(C)C1CCC1 c1(N(C)C)cc(C(F)(F)F)[nH]c(=NCCC2CCCN(C(=O)CCC(F)F)C2)n1 Cc1cnn(CC(=O)NC2C3CC2N(C(C2CC2CO)=O)C3)c(=O)c1 C(=O)(C(C(C)c1ccccc1F)NC(c1cncnc1-c1ccccc1)=O)OC C1(NC(C(C2(O)CCCCC2)(C)C)=O)CCC(=O)N(C)CC1 c1(C(=O)NC(C2N(C(CSCCC)=O)CCC2)C)cc(OCC)ccc1C c1(C(=O)NCC2CCN(C(C(COC)OC)=O)CC2)cc(N)cc(C)c1F N1(CC(N2CCC(NC(c3cnnc(Cl)c3)=O)(CF)C2)=O)CCc2ccccc21 C(=O)(C(F)C(C)C(F)(F)F)NC1(CC=C)CN(C(c2c(C)nn(CC)c2Cl)=O)C1 c1(OC)cc(C)c(CN2CC(NC(c3ccc(Br)cc3I)=O)C2)c(O)c1 Cc1nn(CCF)cc1NC(C1CCCC(NC(C2CC(F)(CF)C2)=O)C1)=O Cc1ccncc1C(=O)NC1C=CCN(C(C2(C)CCSCC2)=O)C1 Cc1ccc(C(=O)NC(C)CNC(=O)C(O)C(F)(F)F)cc1S(N)(=O)=O C1(COC)CN(C(C2CC2COC)=O)CCN1C(=O)Cc1ccc(Br)cc1 c1(OC)ccc(CN(C(c2cc(Cl)cc(Cl)c2)CO)CCO)c(Cl)c1OC C(CC(C(=O)NC(C1CCN(C(C2CC(C#N)C2)=O)CC1)C)N(C)C)SC C1(CC)C(C(=O)NCC=CC2CCC2)CCN1C(c1ncc[nH]1)=O Cc1cc(N(C)C)ccc1CC(N1CCC(COC(F)F)C1)C(=O)O c1(C(N2CCC(C3CCCN3C(c3coc(Br)c3)=O)C2)=O)ccccc1 C1(CC)(OC)CN(C(=O)CN(C2CCC2)C(c2c[nH]cc2C2CC2)=O)C1 c1(C(N2CC3C(NC(c4c(CC)nccc4)=O)(C3)C2)=O)cc2cc(C)ccc2s1 C(C(=O)NCCCOCCCNC(=O)C(F)(F)c1nccs1)(C(C)C)NC(C)=O C1(C)(C(=O)NC(C2CCOC2)C#C)CCN(C(C2CC2C(C)(F)F)=O)CC1 O=C1CCC(C(=O)NCC2(O)CN(C(=O)C=C3CCC3)C2)CN1 C#CC1C(C(=O)NCC(CC)NC(c2cccnc2OC(F)(F)F)=O)C1(C)C CCC(CC)C(C)C(=O)N1CC(C(C(=O)NC(C)C)N(C2CCCCC2C)C)C1 C1(CCNC(c2cn(CC)nc2C)=O)CCN(C(=O)Cn2cccn2)CC1(F)F c1(C(CC(=O)NC(C)CN(C(=O)C=CC2CCCO2)C)C)ccc(O)cc1 CN=c1[nH]cc(C(=O)NCC2OCCC2C(=O)NCC2CC3CCC3C2)s1 Cc1c(F)ccc(C(N2CC3CC(NC(c4ccnn4CCF)=O)C2C3)=O)c1Cl C=CCCCC(C(=O)N1CCOC(C#N)C1)NC(=O)C(SC)SC N1(C(C(COC)O)=O)CC2(CNC(c3csc(O)n3)=O)CC1CO2 c1(CC(CF)NCc2c(C(=O)OC)cco2)ccc(C#N)cc1 N1(Cc2c(OC)cc(O)cc2)Cc2[nH]nc(C(=O)Nc3cc(Br)ccc3F)c2C1 CN1CCC(N(C(=O)NCc2c[nH]nc2-c2ccc(Br)s2)CCO)CC1 C(=O)(CCN=C(NCc1ccc(-c2ccccc2)cc1)NC1CSC1(C)C)NC c1(C(=O)NCC2CC(CNC(C3(O)CC(C(=O)OC)C3)=O)C2)cc2n(n1)CCO2 c1(NC(=O)NC2CCCC(F)C2)cccc(Cc2cccc(Br)c2)n1 CC1(NC(=O)C=Cc2ccco2)CC(C(=O)NCCN2CCCC2=O)C1 C(=O)(C1CCCc2cccnc21)NC(C)CNC(=O)C(O)CC(F)(F)F CCCCCC(O)C(=O)NCC1(CNC(=O)COC2(C)CCC2)CC1 CC(C)CC(C)C(=O)N1CCSCC1CCNC(C1OCC1(C)C)=O CCCC(C)C(C)Nc1cncc(-c2ccccc2C)c1 C=C(C)CCC(C)N(c1ccccc1C)CC(=Cc1ccccc1)C C1(C(=O)NC(c2scc(C)n2)C)CC2CCCC2N1C(c1cc(F)cnc1O)=O Cn1nc(C(=O)NCC2CCC(NC(=O)Cn3cccn3)C2)cc1C#N C(CCN=C(NCCc1cccs1)NCCC1CCCO1)=CC N1(CCCC(=C)C)CCC2(CC1)CN(C(=O)C(CCC)=CCC)C2C(C)C Cc1ccc(C(C)C(=O)NCCCCC2(NC(c3ncncc3N)=O)CC2)cc1 c1(NC(=O)NC2C(NC(=O)Nc3cccc(Cl)c3Cl)C2)c[nH]c2ccc(Br)cc12 Cc1ccc(I)cc1C(N1CCN(C(=O)CS(C)(=O)=O)C2CC12)=O C1(CNC(COC(CC)(C)C)=O)CN(C(C2(C)CC2C)=O)CCN1C c1(CC)ncc(C(=O)N(C2CCCCC2N(C)C(c2cc(CC)on2)=O)C)cn1 CC(CC(=O)NC1CN(C(=O)CCCN2C(=O)CCC2=O)C1)C(C)(C)C C(=O)(C(C)CC(C)C)NCC(C1CC1)NC(c1ccc(OCCC)cc1)=O N1(C(=O)OC(C)(C)C)CCCC1(C)C(=O)NC1CC12CN(C(=O)CNC=O)C2 c1(C(N2CC3CC(NC(C=CC)=O)CC3C2)=O)cccc(C#CCO)c1 c1(C(=O)NC2C(c3n(C)ccn3)CN(C(=O)C3CC3)C2)cc(S(N)(=O)=O)cn1C C1(C(=O)NCCN(C(C2CC(OC)C2)=O)C)CCCC(C)(C)C1 N1(C(C2(CC#C)CC2)=O)CC(NC(=O)CNC(c2cccc(F)c2)=O)C(C)(C)C1 c1(NC(c2ccnn2C)CC)cc(N2CCC(CC3CCC3)C2)nc(C)n1 N1(C(CCCNC(N)=O)=O)CCC(CNC(C23CCCC2C3)=O)(OC)C1 C(=O)(C1=NN(C)C(=O)CC1)N1CCC(F)(C(=O)Nc2c(CC)csc2)C1 c1(OC)c(NC(=O)C(O)C2CN(C(C3CC4CCC4C3)=O)C2)c(C)nn1C C(N=c1nc(N(CC(C)(C)OC)C)c2c([nH]1)CCC(C)C2)c1cc(C)n(CC)c1C C1(CNC(=O)C=CCF)CN(C(c2csc(=NC3CC3)[nH]2)=O)C2(CCOCC2)C1 n1(CC)ccnc1C(=O)NC1(CN(C)C(C2(C)CCC2)=O)CC1 Cc1n[nH]c(C)c1CC(N1CCOC(C(=O)NC(C)(C)C(=O)N(C)C)C1)=O c1(NCC(=O)NCCCOC(F)(F)F)nc[nH]c2ncc(C(F)(F)F)c1-2 Cc1onc(C(=O)NC2CN(C(=O)CC3=CCCCC3)CC3(CC3)C2)c1[N+](=O)[O-] N#Cc1ccc(S(=O)(=O)N2CC3CCC3(C(=O)NC=O)C2)c(F)c1 C1(COC(C)=O)CCC(F)(F)C1.C1(=O)C(CC)NC(=O)C(C)N1CCC C1(CC(=O)NCC)CCCN(C(c2cc[nH]c(=N)c2)=O)C1.ON C1(NC(C(CC)NC(N)=O)=O)CC(CNC(C2(C(N)=O)CC2)=O)CC1O C1(CNC(c2cc(C)c(Br)cn2)=O)C2CCC1CN(C(=O)CCC(N)=O)C2 c1(OC)nccc(Br)c1C(=O)NCCN(C(=O)CNC(C1CCCC1)=O)C C1(NC(C(CCC)=CCC)=O)CC12CCN(C(=O)C(C)O)CC2 N1(C(c2cn(CC)nn2)=O)CCC(O)C(NC(c2csc(C3CC3)n2)=O)C1 C(=O)(CC(C)(C1CCC1)N(C)C)N(CCNC(=O)Cc1csc(Cl)c1)CC C1(C2CN(C(c3ccc(F)c(O)c3)=O)C2)(NC(C2CC(C)OC2)=O)CC1 C=CCN=C(NCc1ccc(S(N)(=O)=O)s1)NCc1cc(-c2ccccn2)on1 C1(C)(CC)CC(NC(=O)CCn2nc(C)nc2C)CN1C(c1[nH]c(C)nc1C)=O C(CCCCN=[N+]=[N-])N(C(C=CC(=O)N(C)C)=O)CCO.N12CCC(C1)CC2=O c1(OC)ccc2c(=NC(=O)CC3(C)COc4ccccc4O3)[nH]ccc2c1 N1(C(c2ccc(OCCO)cc2)=O)CC2(C1)CN(C(=O)C(O)C1CC1)C2 C(CNC(c1cc(Cl)c(Cl)n1C)=O)(CC(F)(F)F)NC(CC(COC)C)=O C1(NC(N2CCCC(NC)C2)=O)CC2(CC(NC3(c4cccs4)CC3)C2)C1 C(C1CCCN1C)=CC(=O)N(C)CCNC(=O)C(=O)NC1(CC2CC2)CC1 N1(C(C(C(C)C)CNC(=O)C(C)N2CCC2)=O)CC2(CCC2)CC1CO C(=O)(CCCCCS(N)(=O)=O)N1C(CNC(C2CCc3n(C)ncc3C2)=O)CC1 c1(C(N2CC3(C)CC2(CNC(=O)CCC(N)=O)C3)=O)cnn2cc[nH]c(=O)c12 CC(C)(F)CCC(=O)N1CCCCC(CNC(=O)C=Cc2cccc(O)c2)C1 Cc1cc(C=CC(=O)NC(C)(CNC(=O)C(C)(C)CF)CO)ccc1F C(C)(C(=O)N1OC2CCC1CC2)N(C(C(C)OCC#C)=O)C c1(C(N2CC(CNC(c3cn(C)nn3)=O)C(C(F)(F)F)C2)=O)cc(N)cc(Cl)c1 C1(NC(CCC(=O)NC)=O)CN(C(=O)C(C)Oc2ccc(Cl)cc2C)CC1(C)C N1(C(C(CCC)CCC)=O)CCC(C(=O)NCC(O)CC(F)(F)F)=C(F)C1 C(=O)(C(O)CC(F)(F)F)NCCOCC(=O)N(CCC)CCN(C)C C=C=C(C)CC(=O)NC(CC=C)C(=O)NC(c1nncn1C)C Cn1ncc(C#N)c1C(N1CCC(O)(CNC(c2cc([N+](=O)[O-])c[nH]2)=O)C1)=O N1(C(COc2cn(C)nc2)=O)CC(NC(=O)CC(F)(F)Br)C(O)C1 C=C(C)C(C)(C)C(=O)NCC1CC(C(N2CCC(C=C)CC2)=O)CO1 C1(NC(=O)CCc2cc[nH]n2)CN(C(c2ccc(F)cc2)=O)CC1n1ccnn1 CCCCC(O)C(=O)N(CCCCNC(C1CCC1C(=O)OC)=O)C CC1(O)CN(C(=O)C2=CCC(NC(=O)Cc3ccoc3)C2)CCC1O C(=O)(CCCCC(=O)NC1CCCC(CNC(=O)CCNC(N)=O)C1)N(C)C N1(C(C)=O)CCC(C(N2CCC(NCCc3ccccc3)CC2)=O)C(O)C1 c1(C(=O)NC2CCC2NC(=O)C(F)(F)F)cnn(C2CCCC2)n1 C#CC12CC(C#N)(CCN1C(=O)Cc1nc(C)c(C)s1)C2 Cc1cccc2nc(C(N3CCCCC3CCNC(=O)C=CC3CCC3)=O)cn12 C1(CN)CCCN(C)C1=O.n12ccnc1C(C)NC(=O)NCC2.CC N1(C(c2c(CC)nco2)=O)CCC2(C1)CN(C(=O)Cc1nc(C3CC3)nn1C)C2 C(=O)(CC(C)P(C)(C)=O)NC1C=CCN(C(CC(=C)C)=O)C1 c1(C(=O)NCC(CCCC)NC(=O)CCCC2CCOCC2)ccc(O)c(C)c1 Cc1ncc(N)cc1C(=O)NC(CCNC(=O)CCC1CCCCN1C)C(C)C c1(CNC(C(CCC#C)O)=O)ccc2c(c1)CN(C(C1(N(C)C)CC1)=O)C2 C1(NC(c2nn(CC)c(C)c2)=O)CCCCN(C(C2C(C)C2(F)F)=O)C1 C(=O)(C(F)CC(C)(C)NC(=O)C(C)c1cc[nH]n1)Nc1cn(CCC)nc1 c12ccc(cc1)OC2.C1(O)CCCO1.O=C(CNC(C(=O)COCC1CC1)=O)OC c1(N2CCCC(NC(c3c(CC)oc(C)c3)=O)CC2)ncnc2cnn(C)c12 C1(C(=O)NC(CC=C)CNC(=O)Cc2ccsn2)CC2OC(C)(C)OC2C1 N1(C(C(C)C)=O)CCN(C(C2C3CN(C4CCC5(C(C)C)CC45)CC23)=O)CC1 N1(C(c2c(CCC)nco2)=O)CC(C(=O)NCC2CC2C2CC2)CCC1(C)C c1(OCCC)c(Cl)cc(C(N2CCN(C(C3CC4CC4C3)=O)CC2C)=O)cc1Cl c1(C(N(CC(C)NC(c2ccc(=O)n(C)n2)=O)CC)=O)snc2ccccc12 C1(C(N2C(CCC)CCC2)=O)C2CC1N(C(c1cc(COCC)[nH]n1)=O)C2 C(C)(C(=O)N(C)OCC(F)(F)F)C1CCN(C(C(C)CN(C)C)=O)C1 C(CCCCCC=C)N(C(CCN(CC#C)C(C1CCCN1C)=O)=O)C(C)C C1(C(=O)NC2CN(C(CCN(C3CC3)CC)=O)C(CO)C2)CC12CCOCC2 c1(OC)ccc(NC(=O)C(=O)NCc2c[nH]nc2-c2ccc(C)cc2)cn1 CC1CCc2c(C(=O)NC3CN(C(=O)C=C4CCC4)C4(CCC4)C3)csc2C1 N1(CC(N2CC(=C(CNC(c3c(C)c[nH]c3)=O)F)C2)=O)CCC(F)CC1 C#CC(CNC(C1COC(CNC(c2cc(CC)n(C)n2)=O)C1)=O)C(C)C CC(C)C(C)C(C)CC(=O)Nc1ccc(S(=O)(=O)N2CCOCC2)cc1 c1(C(=O)NCC2(NC(C3CCC(=O)O3)=O)CCCC2)c(O)cc(Cl)cc1F C(CCC(=O)Nc1cc(C)cc(O)c1)(C(C)C)NC(c1ccc(C#C)nc1)=O c1(C(C(N2CC3C(NC(=O)C(Cl)=CCl)(C3)C2)=O)O)cc(F)cc(F)c1 C1(C(=O)NCC(CC=C)(C)C)N(C(c2occc2COC)=O)CC12CCCC2 N1(C(Cc2c(C)non2)=O)CCC(N(C(=O)Cn2cnc(Br)n2)CCO)CC1 C1(C(N2CC(CO)C(O)C2)=O)(OC)CCN(C(=O)CCc2cnoc2)C1 c1(C(N2CCCC(CNC(=O)C=Cc3cc[nH]c3)C2)=O)n[nH]c2c1CCCC2 N1(C(c2ncccc2F)=O)CCCC2CN(CCOCc3ccco3)CCC12 C12(C(=O)NC3CC(C)(NC(=O)CN4CC5CC5C4)C3)C(=O)C3CCC1C2C3 c1(C(N2CC(NC(CC3C(C)(C)C3)=O)C2)=O)ccc(F)c2c1OCC2 N1(C(Cc2ccc(C)cc2Cl)=O)CCC2(CCCC2NC(=O)C(C)C(F)F)CC1 CC(C)(F)CCC(=O)NC(C)(CNC(c1ccc(-c2ccccc2)[nH]1)=O)CO N1(C(=O)Nc2ccc(C)cn2)CC2CC(C1)N2C(C1CCC(O)C1)=O c1(COC)sc2ccc(Br)cc2c1C(=O)NCCC(N)C(F)F N1(C(c2c(OC)c(C)cs2)=O)CCC(C2CC2)(NC(c2cnn[nH]2)=O)C1 C1(C(=O)NCC(C)(O)CNC(c2conc2C2CC2)=O)CCS(=O)(=O)C1 N1(C(c2cc(OC)no2)=O)CC2CC1CN2C(C1CC(=C(F)F)C1)=O C(=O)(CCC(C)NC(C1(C)CC(F)C1)=O)NCCCC(=C)C C(N=c1ccc(OCc2cc(Cl)ccc2C)c[nH]1)c1cccc(N)c1.C(=O)OC C1(C(=O)NCC(C2CCCN2C(c2ccc[nH]2)=O)(C)C)CCOC2(CCC2)C1 C1(CNC(=O)NCCc2c(C)c(O)ccc2)CCN2CCCC2C1 c1(C(N2CC(COC)(NC(=O)CC(O)CC3CC3)C2)=O)ncnc(C)c1C C(CCCCCNC(c1cn(CCF)nn1)=O)NC(C1C(OC(C)=O)C1)=O c1(C(=O)NCC2C(NC(c3cc(F)cnc3O)=O)C2)c(O)nnc2c1CCCC2 N1(C(C(n2cc(-c3ccc(C(=O)OC)o3)nn2)C)=O)CC(C)CN(CO)CC1C C(=O)(C(CCS(C)(=O)=O)OC)N1CCCC(C2N(C(CC=C)=O)CCCC2)C1 C1(SC)CN(C(=O)CSc2ccncc2)CC1NC(=O)CN1CCOCC1 C1(C(=O)NC(C2(CO)CC2)C)(CNC(COCCC(C)C)=O)CC(C)(C)C1 N1(C(c2c(CC)onc2)=O)CCCCC1C1(NC(c2c(C)n[nH]c2C)=O)CC1 CCCCCCC(CC)NC(=O)CC1(O)CCN(C(=O)CC(C)(C)C#N)C1 c1(CN(CC(=O)NC(C)CN(C(=O)CC2(N(C)C)CCC2)C)C)ccc(Cl)cc1 c1(OC)cccc(CCC(=O)N2CC(n3cc(C4(C5CC5)CC4)nn3)C2)c1 N1(C(=O)CC2(C3CC3)CC2)CCC(CNC(C2(CO)CC2)=O)C(F)(F)C1 C(CC(=O)NCCc1ncc[nH]1)(C(C)C)NC(C1(C=C)CCCC1)=O C(=O)(CCCCCCS(N)(=O)=O)N(CCN(C(C1(CC)CCCC1)=O)C)C C(=O)(CC1=CCCCC1)NC(c1cn(C)nc1)C(=O)NC(c1ncc[nH]1)C C1(NC(C2ON=C(C(C)C)C2)=O)CN(C(C2CCS(=O)(=O)N2)=O)CC2(CC2)C1 C(=O)(CCC(C)O)N(C1CN(C(c2c(C(C)C)c[nH]n2)=O)C1)C CC(C)CCC(O)C(=O)N1CCOC(C(=O)N(CC(C)C)C)C1 Cc1ccc(ONC(C2(c3ccccc3)CC2(F)F)=O)cc1Br CC(O)CCCNC(c1ccc(CO)o1)c1nnnn1C1CCOCC1 c1(CC)cc(=NC2CN(C(c3cc(N(C)C)ccn3)=O)CC2C)[nH]c(Cl)n1 c1(OC)cccc(CC(N2CCC(N(C(=O)Cn3cnnc3)C)C2)=O)c1 C1(c2ccccc2)(C(N(C2CC(NC(c3cc[nH]n3)=O)C2)C)=O)CC1(F)F N1(C(CC(C)C2CCCCC2)=O)CCC(CO)(NC(c2cscc2Cl)=O)C1 C1(NC(C(C2CC2)SC)=O)CCC(C(=O)N(C2COCC2O)C)C1 c1(NC(C2CC(NC(C3CC(=C)C3)=O)C2)=O)cc(C)c([N+](=O)[O-])cn1 C1(CC)CC(C(=O)NC(C)(C)CN(C)C(c2oc(C)cc2C)=O)CCO1 c1(C(=O)NC(CC)(CNC(=O)CC#N)CC)cnn2ccn(C)c12 c1(CC)cccc2c(F)c(C(=O)NC(C)(CNC(=O)CC(C)OC)C(C)C)[nH]c12 C(CC(=O)O)(CC(C)C)NC(c1c(CNC(Cc2c(C)cccc2)=O)n[nH]c1)=O N1(C(c2cc(C)nn2C)=O)CCC(CO)(NC(C2C(C)C2(F)F)=O)CC1 C(c1cc(Cl)c2c(c1)OCO2)=CC(N1C(C(CC)O)CCC1)=O N1(C(CC(C)N(C)C)=O)CCCCC1CNC(=O)C(C)(C)n1cncn1 CN1N=C(C(=O)NCC2CCC(NC(=O)CC3CC4(CC4)C3)C2)CCC1=O C=C=CC(C)C(=O)NC(c1ccccc1F)CNC(c1ccon1)=O c1(CC)cc(CC)cc(C)c1.c12ccc(cc1)C(=O)OCC21CCCC1 c1(NC(=O)NC(CCC)C2CCCC2)ccc2c(c1)CCOC2 C1(C(=O)N(CCNC(C2C=CCS2)=O)C2CC2)(C2CC2)CCCO1 c1(C(=O)NC(C2CN(C(c3ncn(C)n3)=O)C2)C)ccc(C(F)(F)F)o1 c1(OC(C(=O)NC2CC(C)N(C(=O)CN3CCC3)C2)C)ccc(Cl)c(F)c1 c1(C(=O)NC2C=CCN(C(Cc3cc(C)on3)=O)C2)ccc(F)cc1Br O=C1NCc2cccc(NC3CCCN3CCC3CNCCO3)c21 N1(C(C2C(C)(C)CC2)=O)CCC2(CCC(CNC(=O)C3=NOCC3)O2)CC1 c1(C(=O)NC(C2CN(C(c3ccc(F)o3)=O)CCO2)C)ccnc(O)c1 Cc1c(Br)c(C(N2CC(N(C)C(c3nnc(S)n3C)=O)C2)=O)nn1C C1(CNC(c2cc(CC)no2)=O)CC(F)CN1C(c1cc(C2(O)COC2)on1)=O c1(C(=O)NC2CCN(C(c3c(Cl)cn(C)n3)=O)C2)cc(F)cc(F)c1N c1(NC(CCOCCNC(C=CCSC)=O)=O)cccc(Cl)c1C N1(C(c2cc(C(C)C)on2)=O)CCCC(NC(c2ccccc2)=O)C1C Cc1ccn(CC(N2CCCCC(NC(=O)C(C)(C)c3cnco3)C2)=O)c(=O)c1 N1(Cc2ccc(C#C)s2)CCCC2CCN(Cc3ccccc3)CC12 CC1CCN(C(c2c(C(F)F)cnn2C)=O)CCN1C(=O)CN1CCCS1(=O)=O C(=O)(C(C)(C)CN1CCN(C)CC1)Nc1cn(CCN(C)C)nc1 c1(CSC)ccnc(C(=O)NC(CNC(=O)CC2CCC2)CO)c1 Cc1cc(CCC(=O)NCC2C=CCN2C(c2cnsc2)=O)no1 c1(C(=O)NCCCNC(C2C(C(=O)OCC)C2)=O)ccc(CN(C)C)cc1 CCC(CNC(=O)CC1CC(=O)NC1=O)N=c1[nH]c2cc(Br)ccc2o1 CC1CCOCCN1C(C1CCOCCN1C(=O)CCN1CCOCC1)=O c1(C(=O)NCC(C2(CC)CC2)NC(CNC(=O)OCC)=O)oc(C)nc1C N1(CC(=O)N(c2ccccc2O)C)Cc2c(Br)cccc2C1=O C1(CNC(c2cc(OC)no2)=O)CCCCC1NC(C1OCCCO1)=O Cc1cc(C(=O)NC2CCC(CNC(C3(C)CC(C#N)C3)=O)C2)c(C(F)(F)F)o1 N1(C(C2(CCC=C)CC2)=O)C2CCC1C(CO)N(C(c1c[nH]c(C(N)=O)c1)=O)C2 C(CC(CC)C(=O)N1C(C(=O)NCC(O)C(C)(C)C)CCC1C(C)C)=CC C1(NC(=O)COCC(F)F)C=CCN(C(c2cccc(Br)c2)=O)C1 n1(CC)nc(C)cc1C(C(=O)Nc1ccccc1C)N(C(C)C(F)F)C O(N1CCC(CC(=O)NC(C)CCNC(c2ccc(Cl)nc2O)=O)CC1)CC Cc1cc(C(=O)NC2CC(NC(C3(C)CCCNC3=O)=O)C2)cnc1O c1(N2C(CCNC(C3N(C)CC(C)(C)C3)=O)CCC2)ncc([N+](=O)[O-])cc1F c1(C(N(CCC(C)NC(C2CN3CCN2CC3)=O)C)=O)cn(C)c2ncccc12 N1(C(=O)C2CCCc3ncnn32)CCCCCC(N=c2ncc3ccccc3[nH]2)C1 N(C(=NCCc1cnc(C(C)(C)C)nc1)NCCF)CC(CC=C)(C)C C1(C(=O)NC(CC(=O)OC)C2CC2)CC2(C1)CN(C(C1CC(F)(F)C1)=O)C2 CC(C)(C(=O)NC1(CCNC(c2cnc(-c3ccccc3)[nH]2)=O)CC1)C(N)=O c1(C(=O)NCCC(C)Nc2nccc(OCC)n2)c(Cl)cc([N+](=O)[O-])cc1Cl Cc1ccnc(C)c1C(=O)NCC1CN(C(C2CCCC(C)(C)C2)=O)CCCO1 n1(CC)cccc1C(=O)NC1CC(N(C(=O)COC)C)C1 c1(OC)c(C(=O)NC2CCCCC2NC(c2nc(Cl)cs2)=O)nc(O)nc1O CC(O)(CC(=O)NCc1nc(C(F)F)nc(=N)[nH]1)CC(=O)O CC(C)CC(C(=O)NCCCN1CCCC1C)NC(=O)C1=NNC(=O)C1 C1(CCNC(C(CC)N(C)C)=O)CCCN(C(=O)Cc2nc[nH]n2)C1 C1(C(N(C(C2CCCC2)CNC(=O)CCCC(F)F)C)=O)CCCNS1(=O)=O N1(C(C2CN(CC)C(=O)C2)=O)CC2CCN(C(c3ccsc3C(F)(F)F)=O)CC12 Cc1ccc2c(c1)CN(CC1NCC13CCC3)C(C)(C)C2 CC1(CNC(C2CCC(C)(F)CC2)=O)CCCN(C(C2(C)C=CCCC2)=O)C1 C(=O)(CC1=CCOCC1)NC(CSC)(C)C(=O)NCC1CC1Cl c1(CC)cc(C(=O)NC2CN(C(C3CCC(=C4CCC4)CC3)=O)C2)nn1CCO c1(OC)ccn2c(C(=O)NC3CC(C)CN(C(=O)C(C)C)C3)cnc2c1 Cc1ccc(F)cc1C(=O)NCC1CN(C(c2csc(C3CCCO3)n2)=O)C1 C1(C(=O)NC(C(C)C)C(=O)NCC(C)(C)C(C)(F)F)CCC(=O)C(C)C1 N1(C(c2c(C(=O)OC)coc2)=O)CCCC(CO)(NC(c2ccc(SC)o2)=O)C1 CCC(CN1CCOCC1)N=c1nc(N(C)Cc2cscn2)c2c([nH]1)CCCC2 C(=O)(CCC(=O)c1ccc(F)cc1)N1C(CNC(c2cnc(Cl)[nH]2)=O)C=CC1 N1(C(=O)Nc2ncc(-c3scc(C(=O)OC)n3)c(OC)c2)CCOC(C#N)C1 c1(CC(C)O)cn(C2c3ccc(Br)cc3NCCN2C(c2nc(C)on2)=O)nn1 Cc1nc2cc(C(N3CCCC(NC(=O)C(Cl)=CCl)C(F)C3)=O)ccc2s1 N1(Cc2cn(CCC(=O)N(c3c(C)cco3)C)nn2)CCC(OC2COC2)CC1 C(C(C)(CCO)NC(=O)C(COC)NC(c1n[nH]c(C2CC2)c1C)=O)OC N1(C(c2nnc(C(C)(C)C)s2)=O)CCC2CN(C(=O)CC3(CO)CC3)CC2CC1 N1(C(Cc2nc(COC)sc2)=O)CCC(NC(=O)CC(F)F)C(C)C1 C=C=CC(C)C(=O)NC(CC=CC)C(=O)NCC(=O)N(C)C1CC1 CCC(CC(=O)N(CCC(=O)N1CCC1CSC)C)SC C#CCC(C)(CC)C(=O)N1CCC(C(C)(C)CNC(c2cccc(F)c2)=O)CC1 Cc1cc(C(=O)NCCC(C)NC(c2cc(CO)[nH]n2)=O)on1 c1(-n2cc(C(CC)OC)nn2)ccc(Cl)c(C(=O)Nc2nccc(C)c2COC)c1 C1(CNC(c2ccns2)=O)CCCCCN1C(c1ncc(Br)cc1F)=O CCC(CN(C)C)C(=O)NCC(C1CC1)NC(c1cc(-c2ccccn2)c[nH]1)=O c1(CNC(=O)C(c2ccc(O)cc2)O)ccc(-c2cccc(Cl)c2)cn1 C(CC(O)C(=O)NC1CCCC(C(=O)NC2(C3CC3)CC2)C1)SC CCC(C)C(C(=O)NCc1cc(C(=O)NC(C2CCCCC2)C)cs1)OC N1(C(c2cncc(OC3CN(C(COC)=O)C4C3C4)c2)=O)CCC(=O)N(C)CC1 C1(C(N2CCC(NC3CCC3)C2)C(=O)NC2(C)CC2)CCC2COCCC2C1 c1(C(C(=O)NCC(CC=C)NC(c2cccnc2O)=O)C)cc(F)cc(F)c1 c1(CCC(=O)NCC#CCNC(C2CC2(F)Br)=O)ccccc1 O=C(CC1=NNC(=O)C1)NCC1CCC1CNC(=O)C(F)C(F)(F)F c1(C(=O)NCC2(C)CCCN(C(C3CCN(C)C3)=O)C2)cc(=O)n2ccsc2n1 c1(OC)c(C(=O)NCCNC(c2ccc(OCF)cc2)=O)cccc1Cl O=S(=O)(c1ccc(C2CC23COC3)cc1)C(F)(F)Br C(=O)(C1=CCCC1)N(CCCN(C)C(c1cnc(-c2ccccc2)[nH]1)=O)C C1(=O)CCCCOC(=O)Cn2cc(nn2)C2(O)CN1C2.N(CC)(CC)CC.C(C)=O CC(C)(C)C(=O)C(=O)NC1CN(C(=O)CN=S(C)(C)=O)CC1(C)C C1(N2CCCCC2)(COC)CCN(C(c2ccccc2CCCO)=O)CC1.CCO c1(N(CC(COC)(C)C)C)nc2ccsc2c(=NCC(c2ccsc2)OC)[nH]1 N#Cc1ccc(C(N2CC3CC3(C(=O)Nc3cccc(Cl)c3O)C2)=O)cc1F C1(C(=O)O)CCC(C(=O)NCCn2cc(CN3CC4CC4C3)nn2)C1 c1(C(=O)NCC(CNC(c2c(OC)cccc2F)=O)F)cc2n(n1)CCCC2=O C(=O)(CCCc1cccnc1)NCCOCCCNC=O.N=c1nc[nH][nH]1 C1(CC)C(NC(=O)CCCc2ccc(C)cc2)CCN1C(c1cccc(O)n1)=O CC1(C)CCCC(CC(=O)NCCCCC2CN(c3ccc(Cl)cn3)C2)C1 c1(CC(=O)NC(CC)(CNC(C2COCCO2)=O)CC)cc(OC)ccc1OC Cc1cc(=NCC2CN(C)CCCO2)[nH]c(N2CC3CCC(C2)O3)n1 C(C)(c1ccc(OC)cc1)=CC(N1CCCC(N(C(C(C)SCC)=O)C)CC1)=O C1(CC(=O)NCC2C(NC(COC)=O)CC2)CCCOCC1 CCCC(C)CCCC(=O)NCC(C)N(C)C(c1cnc(OC)cn1)=O N1(C(=O)OC(C)(C)C)CCC(F)(F)C(CNC(=O)NCC(C(C)(F)F)(C)C)C1 Cc1cc(C(=O)NC(C2(O)CN(C(c3cc(F)n(C)n3)=O)C2)C)nn1C(C)C CCCC(C)CC(C(=O)Nc1cccc([N+](=O)[O-])c1)N1CCC12CCC2 N1(C(Cn2nc(C)oc2=O)=O)Cc2[nH]nc(C(N3CC(N(C)C)C(F)C3)=O)c2C1 c1(CCCN(C(C)C)Cc2c(-c3cnn(S(C)(=O)=O)c3)ncn2C)ccc(O)c(O)c1 C1(CC(C)(C)C)CCC(NC2CC(Cn3cccn3)C2)(CO)CC1 N1(C(C23CCC(OC)C2C3)=O)CC2CC1CCC2NC(=O)Cc1cc(Cl)n(C)n1 Cc1cc(C(=O)NCC2CC(NC(C3CC(F)C(=O)N3)=O)C2(C)C)cc(F)c1 c1(OC)ccc(C(=O)NC(C)Cn2cc(-c3ccc(C)n3C)nn2)nc1Cl C(CCC1OCCO1)(C(=O)NCCCF)NC(=O)NC(C1CCCO1)C C1(C(N2CC(CNC(C3(F)C(C)(C)C3(C)C)=O)OCC2)=O)CC2OC(=O)OC2C1 CCCC(C)(C)CNC(c1csc(C(=O)OC)c1)c1nnnn1-c1ccccc1 C1(C(=O)NC23CC(CNC(C4CC(=O)OC4)=O)(OC2)C3)CCOC2(CCC2)C1 Cc1nc(NC2CC(NC(=O)CSCC3CCCO3)C2)cc(C(F)(F)F)n1 N1(C(CN2C(C)CCC2C)=O)CCCC(C2CN(C(C34CCC(C3)C4)=O)C2)C1 C1(CC(=O)NCC2CC(C(N(C3CCOCC3)CC)=O)C2)CC2CCC1O2 c1(OC)cc(C(N2CCC(NC(c3cc(F)n[nH]3)=O)C(F)C2)=O)cnc1OC N1(CC(N2CCN(C(c3ccc(CC)s3)=O)CC2)=O)C(=O)CN(C)C1=O CC1(O)CCCN(C(=O)C(=O)NC2C3CC4C(C3)C24CO)C1 Cc1cc(C(=O)NC2(CCNC(=O)C#CC(C)C)CCCC2)ccn1 C1(C(=O)NC2CC(CCn3cc(C(C)(C)C)nn3)C2)CC2C=CC1C2 N1(C(c2[nH]cc(CC)c2)=O)CCN(C(C2(CC3CCC3)CC2)=O)CC1CC CC1(C)CC(n2nc(-c3ccc(Cl)s3)nc2-c2cnccn2)CCO1 C(CC1CCc2ccccc21)NC(c1cc(N2CCC(OC)CC2)ncc1)=O c1(CNC(NC(COCC)CC)=NCC2CCOC2)ccc(Cl)c(O)c1 c1(OC)cc(-n2nc(Cc3cccs3)nc2-c2ccnnc2O)ccc1Cl n1(CC)c(C(=O)NC(Cc2cn(-c3ccc(O)cc3)nn2)C(=O)O)cnc1O CN1CCCC(N(C)C(C2(F)CCN(C(C3CCCC3)=O)C2)=O)C1 C(=O)(C(C)C(O)C(C)C)N(CC(=O)NCCN1CCCNC1=O)CCOC N1(CC)CC(CNC(=O)C(CN(C)C)NC(C2CCCCC2)=O)CC1=O CC1(C)CC(F)(F)CCC1CNC(=O)Nc1nc(C2Cc3ccccc3C2)cs1 C(C)(C)(C=CC(=O)NCCOC(C)(C)CNC(=O)CC1CCOC1)SC C1(C)(C(=O)NCCCC(=O)OC)CC(O)CN1C(=O)CCCC1CCCC1 C#Cc1ccc(Cl)c(C(=O)NCCN2CCN(C(=O)C(=O)N(C)C)C(C)C2)c1 C1(C(N(CC(C)NC(c2cc(C(C)C)[nH]n2)=O)C)=O)CC12CCCCCC2 C1(C(N(C2CCOCC2)CC)=O)CCOCC1NC(=O)C=CCCC(C)C C(CC(C(=O)NCCCC(=O)NO)NC(=O)Cc1nccn1C)=CC CC(CC(=O)NC(C)(CN(C(=O)Cc1cncs1)C1CC1)C1CC1)N(C)C CC1CN(C(c2cc(Br)c[nH]2)=O)CC(CCNC(=O)CC2CC=CC2)O1 CCCCN=C(NCC1=CCCCCC1)NCCOCC(C)(C)O C=CCC(CNCc1cnc(-c2cccnc2)s1)CC(C)C(C)(C)C c1(C(N2CC(N(C)C(C3CC4CC4C3)=O)C(C)(C)C2)=O)cc2ccc(F)cc2o1 C1(C(=O)NC2C=CCC(C(=O)NC(C)Cn3cccn3)C2)(CC)CNC(=O)C1 C1(C(N(CCC)C2CC2)=O)COCCN1C(=O)C(C1CC1)SC C1(C(=O)NCC(CNC(=O)C=Cc2ccsc2)F)CCCC1C1CC1 c1(C2C(C(=O)NCC3CCN(C(c4ccc(COC)[nH]4)=O)C3)C2)ccccc1F c1(NC(C2CC3(CC3)CN2C(C2C3COCC23)=O)=O)c(C(F)(F)F)cccc1O C1(CCNC(=O)CCc2cc[nH]n2)(OC)CN(C(c2csc(C)c2)=O)C1 C1(C(=O)NC(CCC)CO)(CC)CCN(C(=O)C(C2CC2)OC)CC1 N1(C(C(C)OC)=O)CC2CCOC2(CNC(=O)CC(C2CCC2)C2CCC2)C1 c1(CCC(=O)N(C2CC(NC(C(C(C)C)OC)=O)C2)C)cc(C)nc(C)c1 N1(C(C2CC(C)(C)OC2(C)C)=O)CCOC2(CCC(NC(=O)C=C(Cl)Cl)CC2)C1 C1(O)(C(=O)NCC(C2CCC2)NC(c2cc(C(F)(F)F)cs2)=O)CCSC1 c1(OC)ncc(Br)c(OC)c1C(=O)NC(CC(F)(F)F)c1cccnc1 C(=O)(CCC(C)NC(c1cccc(COC)n1)=O)N(CC(CC)(F)F)C C1(C(N2CCCC2Cc2cccnc2)=O)NCC12CC2(F)F c1(C(N(CCNC(=O)CCCSC(C)(C)C)CC)=O)cc(C)oc1C C(CC(C)C)(C(=O)NC(C1CCCN1C(c1oc(C)cc1C)=O)C)OC C1(CNC(c2c(C)n(C(C)C)nc2)=O)CN(C(=O)Cc2ccccc2)CCN1C C(=O)(C(C)C(O)C(C)C)NCC1(NC(c2cccc(C)c2Cl)=O)CCCCC1 CCC(CCCC(=O)N1CCC(CCO)(COC)C1)NC(=O)CSCC(C)C C=CC(C(F)(F)F)NC(c1ccc(CNC(C2CC23CC3)=O)cc1)=O Cc1cc(C)c(C(=O)NC2CCN(C(c3nc(=O)cc(N)[nH]3)=O)C(C)C2)c(C)c1 c1(C(=O)NC(C(=O)N(C)Cc2ncc(C)o2)CC2CCC2)ccn2ccccc12 C1(CCN(C(=O)CCCc2cnccn2)C)CCN(C(=O)CC2CCOC2)CC1 N1(C(c2c(C)ccs2)C)CCCC(CCNC(c2csc(C3CC3)n2)=O)C1 C(=O)(C(COC)OC)NCC.C(C)(C(=O)N(CC(C)OC)C)N C1(NC(C2CC(C)(C)OCC2)=O)CN(C(C2CC(F)(F)CS2)=O)CC(F)(F)C1 CC(C(F)(F)C(F)(F)F)=CC.C1(CC(=O)Nc2cnc(C)s2)(SC(C)C)CCCCC1 CCCCC(C)(CO)NC(C1C=CCN(C(=O)CN2C(=O)CCC2=O)C1)=O CC1CN(C(=O)CCOC2CC2)CC2(CCN(C(=O)CC3(C)CC(F)(F)C3)C2)O1 CC(C)(C(=O)NC1C2CN(C(c3scnc3C3CC3)=O)CC12)C(F)F CCC(F)(F)C(=O)N1CCC(C(C)NC(C2CCSCC2)=O)C1 C(=O)(C(C(C)OC)NC(=O)C(N)=O)NCc1[nH]nc(CC)n1 C1(NC(C2C(OCC)C2)=O)CN(C(=O)Cn2nnnc2C)CC1(C)C c1(OC)ccc(Cn2nc(-c3occc3C)nc2CC(C)(C)C)cc1 CC1(C)CN(C(C2CCOC2C2CC2)=O)CCC1C(=O)NC1CCCCCCC1 CCC(C(=O)NCC1CCCN1C(=O)CNC(c1cccc(C)c1)=O)C(C)O S(=O)(=O)(c1ccc(NCC2(C(O)C(C)C)CC2)c2cnccc12)NCC#CC C1(O)(CCNC(c2nc(CC)oc2)=O)CCCN(C(=O)CCOCC(F)F)C1 N1(C(C(C=C)c2ccccc2)=O)CC2CC1C2CNC(=O)C=CC1CCCCC1 N1(C(C2C(c3ccccc3F)(C)C2)=O)CCCC2(CCCN2C(=O)C=CCF)C1 C(C)(CCC(=O)NC1CCC(NC(=O)CSC2CCCCO2)CC1)SC CCC(C)(C(=O)NC(c1cccc(C)c1)CNC(C1CS(=O)(=O)C1)=O)OC c1(NC(C(CCN(C)C)(C)O)=O)ccc2cnn(C(F)F)c2c1 c1(C(=O)NC(C(C)C)C(=O)NC2(C)CCSC2)cc2ncccc2[nH]1 C1(NC(c2cc(CC)[nH]n2)=O)CCCN(C(c2cocc2C)=O)C1CC N1(C(c2cnc(CCC)s2)=O)CCCC12CCCN(C(c1ccc(C#N)[nH]1)=O)C2 C(=O)(C1CCc2c[nH]nc21)N1C(c2cn(Cc3cn(SC)nn3)nn2)COCC1 Cc1cnc(C(=O)Nc2ccc(I)cc2O)c(C)c1 C(=O)(C1=NOC2(CCN(C(c3ccno3)=O)C2)C1)Nc1cc(C)c(Cl)s1 c1(C(=O)NCC2CN(C(CCC#C)=O)CC2C)nc(Br)n2c1CCCC2 N1(C(CSCCCC)=O)CC2CCOCC2(NC(=O)Cc2c(C)noc2Cl)C1 N1(C(Cc2c(C)noc2C)C(=O)NC2CCCC2)CC2CCCCC2(CO)C1 C1(NC(C(C=C)O)=O)CC2CN(C(=O)Cn3ccccc3=O)CCN2C1=O C(C)(C)(C(C)CC(=O)N1CC(N(C)C)C(C)C1)NC(C(n1c(C)ncc1)C)=O C(=O)(CCC(=O)N(C)C)NCC(CC)N(C(Cc1c(CC)con1)=O)C N1(C(c2n[nH]c(C)c2Cl)=O)CCC2(C=C(C(=O)N3CC(OCC(N)=O)C3)C2)C1 Cc1cc(S(=O)(=O)N2CCOCC2C(F)(F)F)cc(Br)c1C N1(C(CC2C(CC)C2)=O)CCC(CNC(c2c(C)coc2C(C)C)=O)C(O)C1 c1(OC)ccc2c(c1)CCCC2N(C(=O)NC1(CN)CCOCC1)SC(C)(C)C c1(C(C(=O)NCC)N(C(C)C(=O)OC)C2CC2)cc(OC)c(Br)c(C(C)C)c1 C=C(C)C1OCCC1C(=O)N(CCC(N1CCCC1CN=[N+]=[N-])=O)C1CC1 c1(NC(Cc2ccc(C)cc2)=O)cc(Cl)ccc1C#N.C12CC(C1)CCNC2=O c1(C(=O)NCCN(CC)Cc2ccn(CC(C)C)n2)cccc(-n2ccnc2)c1 Cc1sc(-c2nc[nH]n2)nc1C(=O)NC1CCCN(C(=O)C(C2CC2)N(C)C)C1 c1(CC)nc(C)c(C(=O)NC2CCCC2(C)CNC(=O)C(C)SC)s1 C1(NC(CCCCCOC)=O)CC2CC(C1)CN(C(C1CC3CCC(C1)C3)=O)C2 N1(CCN(C(c2cncnc2)C(=O)N)C)CCOCC1.C(C)(C)SC c1(C(N2C(COC)(CNC(=O)Cc3cc(C)no3)CCC2)=O)ccc(C#N)cn1 C1(C(=O)NCC(CSC)OC)CCC(n2cc(-c3cnc(C)nc3)nn2)CC1 Cc1cnccc1CN1C(C(=O)NC(c2cn(C3CC3)cn2)=O)CCC1C1CC1 C#Cc1c[nH]nc1C(=O)NC1CCN(C(=O)CCN2CCC(O)CC2)C1 C(=O)(C1Cc2c(Cl)cccc21)N1C(CO)CC(NC(C(COC)(F)F)=O)C1 c1(OCC)cccc(CNC23CCC(NC(C4CNC(=O)C4)=O)(CC2)C3)c1F N1(C(C(C)OCC(F)(F)F)=O)CCC(N(C(=O)C=Cc2ccsc2)CCO)C1 CCN=c1cc(-c2nc(CO)n(CCc3cc(C4CC4)n(C)n3)n2)cc[nH]1 Cc1c(F)ccc(C(=O)NCC2(CNC(=O)C(F)C(C)C)CC2)c1N N1(C(C2CN(C)C(=O)N2)=O)CCCC2CN(C(=O)CCc3nccs3)CCC12 C1(COC)(CNC(=O)C=CCN(C)C(c2cn(CCO)nn2)=O)CCCCC1 C(=O)(CCCCN(C)C)NC(CC)CNC(=O)CNC(=O)OC c1(OC)ncc(S(=O)(=O)Nc2ccc(NC(c3ccsc3)=O)nc2)s1 C(=O)(CCC(=O)NC1CCC(NC(=O)CCC(=O)c2ccccc2N)C1)NC C1(CC)(NC(=O)C(COC)N(C)C)CCCN(C(c2cc(=O)n(C)o2)=O)C1 C1(OC)(CNC(=O)C=C(C)C2CC2)CCN(C(c2nonc2CC)=O)C1 C=CCCC(C(=O)NCC(C)(C)C=C)NC(=O)CCCOC N1(C(C(C)c2cc[nH]n2)=O)CCC(C2CN(C(=O)COC3CCOCC3)C2)CC1 N1(C(C2(C)CCC(O)CC2)=O)CCCCC12CC(NC(=O)CC1(O)CCOC1)C2 C1(CNC(c2ccnc(C)c2C)=O)CCCC2CN(C(C3CCCC3F)=O)CC12 C1(C)(C(=O)NCC2N(C(C(C)NS(C)(=O)=O)=O)CC2)CCCOC1 Cc1cc(C)n2nc(C(=O)NC34CCC(CN(C(C5(C)CCCO5)=O)C3)C4)cc2n1 N1(C(Cn2c(CCC)nnc2S)=O)CCC2CCC(C1)N2C(=O)CNC=O c1(C(=O)NC(C2(O)CCN(C(=O)COC3(C)CCC3)C2)C)ccc2ccsc2c1 CCC(F)(C(=O)OC)C(=O)NCC(C)(C1CC1)NC(=O)CCCC1CCOCC1 C#CCC(C)(C(=O)NC1CC2CC(O)C1C2)NC(=O)CCC(F)(F)F CC(C)S(=O)(=O)CC(=O)N1CCCC1CC(=O)NCCNC(=O)C(C)(C)C C1(c2n(CCCOC)nnn2)(NCCC2CCCCCCC2)CCCCC1F C(=O)(CCCCCN=[N+]=[N-])N1CCC(CCCCCNC(CSC(C)C)=O)CC1 C1(C(N2C(C)CC(O)C2)=O)C2CCCC1CN(S(=O)(=O)CC1CC1)C2 c1(CN2CCC(NC(c3cccn4cncc34)=O)C(O)C2)cc(Br)cc(Br)c1O C1(C(=O)OC)C=CCN1C(C1CCN(C(=O)CSC(C)(C)C)C1)=O c1(CC(=O)N(CC(C)O)CCNC(C=CC=CC)=O)cc(C(F)(F)F)n(C)n1 c1(C(=O)NCC(C)(C)NC(Cc2c(CC)con2)=O)ccc(NC)cn1 N1(C(c2ncc(N(C)C)nc2)=O)CC(NC(c2ncc(Cl)n2C)=O)CC2(CC2)C1 C1(C(C)C)N(C(=O)C(C)(C)F)CC12CCN(C(=O)CN1CC(=O)N(C)C1=O)CC2 c1(C(=O)NCC2N(C(c3n(C)nc(O)c3)=O)CC(O)C2)cc(N)c(F)c(F)c1Cl Cc1nnsc1C(=O)NCCC1CCC(NC(=O)C=Cc2ccoc2)C1 c1(CNC)cc2c3c(ccc2[nH]1)N(C(=O)Cc1cnccn1)CC3 c1(CC(=O)NCC(CNC(c2cncc(C3CC3)c2)=O)OC)ccc(C)c(Cl)c1 C1(CNC(c2n(C(C)(C)C)nnn2)c2cnn(C(F)F)c2)CC2(CC2)C(=O)O1 C1(NC(c2ccc(C3CC3)o2)=O)C2CCN(C(=O)CC3CC=CC3)C12 C1(CC)CN(C(=O)C(C)COC)CCC1NC(=O)CCc1conc1C C1(NC(CCC(C)OCC)=O)CN(C(=O)CN2CCC(C)CC2)CC2(CC2)C1 c1(CCC(N2CCC(NC(CCC(C)(F)F)=O)C23CC3)=O)n[nH]c2c1CCCC2 N1(C(CCC=CC)=O)CC(C(C)(C)C)CC(CNC(C2CC23CC(C)(C)C3)=O)C1 c1(CNC(C2(C)CC(=C)C2)=O)cccc(CNC(C2CC2[N+](=O)[O-])=O)c1 C(=O)(C1=CCC(C)(C)CC1)N1CCCC(CC=C)(NC(=O)CCC(N)=O)C1 c1(C(N2C3C(N(C(Cc4nc(C)[nH]n4)=O)C)CC(C3)C2)=O)cc2n(n1)CC(F)C2 C(=O)(C(=O)N=S(C)(C)=O)NC1(C)CC(NC(=O)Cc2nc3c([nH]2)CCCC3)C1 C1(CNC(CS(=O)(=O)NC)=O)CCN(C(=O)C(C)(C)COC(C)C)CC1O C(CC(C(N)=O)NC(=O)C(C)N(C(=O)C(c1cnn(C)c1)=O)C1CC1)OC Cc1ccc(C=CC(=O)NC2CN(C(C3CCC(C(N)=O)O3)=O)CC2F)cc1 c1(C(N2CC3CC(NC(CC(CCC)C)=O)C3C2)=O)ccc(Cl)c(F)c1F C12(NC(=O)COc3cccc(F)c3)CCCC1N(C(=O)CCOC1CC1)CC2 c1(CC)oc(C(=O)NCCC(C)N(C(=O)CC2CC3(CC3)CO2)C)cc1C C1(NC(c2c(Cl)cc(C)s2)=O)CC2CC(NC(c3ccnc(C(N)=O)c3)=O)CC12 Cc1cc(=O)c(C(=O)NC2CN(C(=O)CC3CCCCO3)CCC2F)cn1C CC1C(=O)N(CC(=O)NC2(CNC(c3csc(S)n3)=O)CCOC2)C(=O)C1C CC1CCC(C)N1CC(=O)NCCn1cc(CNC(c2cocn2)=O)nn1 Cc1cc(F)c(C(=O)N(CC(C)(C)CNC(C2CCOC2C2CC2)=O)C)cc1F c1cc2ccccc2s1.C1(CC=C)CCCC1(c1nnnn1C)NCCS(N)(=O)=O N1(C(c2ccoc2C)C(=O)NC)CCN(c2ncccc2Cl)CC1 C1(C(=O)NCCOCCCC#C)CN(C)CCN1C(c1nc(C)sc1C)=O N1(C(C(=O)NCc2ccc(Br)cc2)C2CCOC2)CCC(O)(CCF)CC1 C(=O)(CCCCC(C)(C)OC)N(C1CCN(C(=O)CN2CCOC2=O)CC1)CC C#Cc1cc(F)ccc1CN1CCN(Cc2cccc(C#N)n2)CC1C(C)C Cc1nc(CCC(=O)N2CCC2CNC(=O)C(C)(C)CN(C)C)oc1C C1(CC)CN2CCN1C(=O)C1CC(C1)SCC1(CC2=O)CC1.C1(CC2CC2)CC1 Cc1cccn(CC(=O)NC2CC(C)(NC(=O)CC34CCCC3C4)C2)c1=O C1(CNC(c2cccc[n+]2[O-])=O)CC2(CCC2)CN1C1CCCNC1=O C(C(C)(C)CC(C)O)NC(C1C(CC)CCN1C(C1CCCC(O)C1)=O)=O C1(C(=O)NC2(c3ccccc3)CC(NC(=O)CC3(CO)CC3)C2)CCCOCC1 C1(CNC(C2C(CC)N(C)CC2)=O)CN(C(c2nccc(Cl)c2F)=O)CCC1C C1(NC(C(CC)CN(C)C)=O)CC2CCC(C1)N2C(=O)CCN1CCCCC1 N1(C(CCC(=O)Nc2nccs2)=O)CC2(C1)CN(C(C1OCCCO1)=O)CCO2 Cc1cc(-c2ccnc(NC3CCOC3C)n2)cc(C)c1 C1(c2nc(C)[nH]n2)CCCC12CCN(CC(=O)NC(C)CCCC(C)C)CC2 C1(NC(CSCC(C)C)=O)CCN(C(=O)COCCCF)C(C)C1 c1(C(N(C(CCNC(c2c(C)nc(C)[nH]2)=O)C)C)=O)ccccc1S(C)=O N1(C(=O)OC2(COCO)N(C(C(C)S(N)(=O)=O)=O)CC=C2)CC2(CCC2)OCC1C Nc1cccc2cc(C(=O)N(C3CCCN(C(=O)C=CCF)C3)CCF)cnc12 N1(C(CC(=O)OCC)=O)CCCC2(CNC(=O)CSSC)CCCC12.CC(N)=O C12(C(=O)NCC(c3ccccc3)NC(C(CC)N(C)C)=O)CCC(O)(CC1)CC2 C1(NC(CCOCC)=O)CN(C(=O)CCc2csc(=N)[nH]2)CC1C(F)F C1(NC(CCn2ccc(C)n2)=O)CC2CCC1CC2NC(c1nc(Cl)cs1)=O C1(CNC(C#C)=O)CCC2(CCC2)C1NC(c1ncccc1OC)=O C#Cc1cc(C2CC2C(=O)NC2CN(C(=O)CCC(=O)NC)CC2C)ccc1C C#CC1(CNC(C2C=CC(NC(=O)CC3CCCC(=O)N3)C2)=O)CCCC1 CC(C)C(CC1CCCC1)C(=O)NCCCC(C)(C)NC(=O)C(C)N1CCC1 c1(C(=O)NC(CNC(C2=CC(C)(C)C2)=O)C2CCC2)cc(F)cc(Br)c1O C1(CCNC(C(C)CN(C)C)=O)CCN(C(C2(C(F)(F)F)CNC(=O)C2)=O)CC1 N1(C(C#CC(C)C)=O)CC2C3CCC(C2C1)N(C(c1cc(Cl)c(F)cc1F)=O)C3 c1(C(N2C(C(=O)Nc3c(OC)nn(C)c3)CCCC2)=O)cc(Br)cc(F)c1F Cc1cc(C)c(C(N2CC(C(C)NC(c3ncccc3C)=O)C2)=O)o1 C(=O)(CC(C)(C)F)NC1(CN(C(=O)CCCSc2ccccc2)C)CC1 c1(NCC2C(C)(C)C2)ccc(S(=O)(=O)NC(c2cccc(F)c2)CO)cc1Cl C1(O)(C(C)NC(Cc2c(C)nc[nH]2)=O)CCN(C(c2ccc(CO)cn2)=O)C1 c1(C(N2CCN(C(c3cc(Br)c(Cl)cc3F)=O)CC2)=O)cc(Br)c2cn[nH]c2c1 CC1CC2CN(C(=O)CCCC3(NC(=O)CC4CCC4)CC3)CCN2C1 c1(C(=O)NCC2CCCCN2C(c2cccs2)=O)cc(Br)ccc1O C1(C(N2CCC(N(C)C(c3nnc(C)s3)=O)C2)=O)(COCCOC)CCCCC1 N1(C(C(C)C)=O)CCCC1(CNC(c1csc(-c2ccccc2)n1)=O)COC N1(C(CC=C)=O)CCc2ccccc2C(NC(C2(CC(F)F)CC2)=O)C1 C1(CNC(CCC=C(C)C)=O)(NC(=O)C2=C(C)OCC2)CC2CCC1CC2 C(c1ncco1)=CC(=O)NC1C(NC(C2(CCC)CCC2)=O)CC1 C1(N(C(C2CCN(C)C2=O)=O)C)CCCN(C(c2cncn2C)=O)CC1 CC(CNC(=O)Cc1ccn(C)c1)C(=O)NOCC=CCl N1(C(C(C)C)=O)CCC(C(N2CCC(O)C(C)C2)=O)C(F)C1 Cc1ccnc(O)c1C(N1CCC1NC(=O)C(O)C(C)c1ccccc1F)=O Cc1cc(C)c(C(=O)NCC2CCCN(C(c3cccc(C)c3N)=O)C2)c(C)n1 CC(N=[N+]=[N-])C(=O)NCC1(O)CN(C(c2ncc(F)cn2)=O)C1 C(C)(C(=O)NC1(CC(=O)NC)CSC1)N(CC)CC.C1CC(=O)N1C.C(N)(=O)N N1(C(=O)OC)CCCC(Nc2ccnn2CCCc2ccccc2)C1 c1(COC(C)(C)C)ccc(C(=O)OCCOCCOCC)cc1 Cc1cc(-c2ccc(CC(=O)N(C)C)cc2F)ccc1SCCCn1ccnc1 c1(NC(C)=O)cc(C(=O)NCC2CCC(NC(c3cocn3)=O)C2)ccn1 c1(N2CCC(=C(F)Cl)C2)nc(=NC(C)c2cnn(CC(F)(F)F)c2)[nH]c2c1SCC2 c1(NC(C2(C(F)(F)F)CCCNCC2)=O)cccn2nnnc12 C1(C)(CNC(C(C)c2ccsc2)=O)CCCN(C(=O)C(Cl)=CCl)C1 C(CC)(CCC(=O)NCc1noc(COC)n1)NC(c1c(CC)non1)=O CP(C)(=O)CN1CCCC(C(=O)NCCC2CN(C(=O)CCC(N)=O)CCO2)C1 CC1(C2CN(C(C3C=CC(NC(c4ccc(C#N)cn4)=O)C3)=O)C2)CC1 S(=O)(=O)(c1cnccc1N(C)Cc1ncc(CC)s1)NCC(c1ccc(C)s1)O C(CCCCC(=O)N1CCOCC1C(=O)NCC1(SCC)CC1)OC CCC(C)C(=O)C(=O)N1CC(OCCC(=O)NCC(C)(O)CC(C)C)C1 [N-]=[N+]=NC1(C(N2CCC(CCCO)C2)=O)CCN(C(=O)C(=O)CCCCC)C1 CC1CC=C(C(=O)NC2(C3CC3)CCN(C(C3CC(C)(O)C3)=O)C2)CC1 C(CCNC(c1ccoc1Cl)=O)(C(C)C)NC(CC=CCC)=O S(=O)(=O)(c1cccc(C)c1)NC(CC)CNC(=S)NCCC(F)(F)C(=O)O c1(OC)cc(C(=O)NCC2CCCC2NC(C23CCC2CC3)=O)ccn1 Cc1ccc(C=C2C(C#C)C2)cc1.N1(C(c2cc(F)n(C)n2)=O)CCCC(C=O)C1 c1(C(=O)NC(C(=O)NCCS(CC)=O)CO)ccn(C)c1C c1(C(=O)NCC(CN(C(=O)CSc2cccs2)C)(C)C)cn(C)[nH]c1=N C1(C(C)(C)NCc2nc(COCC)sc2)CCc2nccn2C1 N1(C(C(=O)N(CCN2CC(C)C(C)C2)CCO)=O)CCC2(CC1)CN(C)CCN2C c1(CC)noc(C(=O)NCC2C(C)CCN2C(c2cc(OC)ccn2)=O)c1C O=C1CCCN1C1CCN(Cc2sccc2F)C1 c1(C(N2CCC(C(N(CCC=C)CC)=O)CC2)=O)ccc2[nH]ccc2c1 C1(CCNC(c2c(CC)nn[nH]2)=O)CSCCN1C(=O)C(F)C1CCCC1 c1(CC)conc1CC(=O)N(CC(C)O)CCNC(=O)Cc1nonc1C N1(C(CC2C(C)(C)N(C(C3CC4(CCO3)CC4)=O)CC2)=O)CC2(CCCCC2)C1 c1(C(N(C2CCN(Cc3c(Br)ccnc3Cl)C2)C)=O)ccnc2c1OCO2 c1(NC)cncc(C(=O)NCC2COCC2NC(c2cc(C(N)=O)[nH]n2)=O)c1 N1(C(CCN2CCC(C)CC2)=O)CCC(C2CCN(C(C34CC(C)(C3)C4)=O)C2)C1 CC1(CC(N2CCC(O)(CNC(C3CCCN3C(N)=O)=O)C2)=O)CCS(=O)(=O)N1 Cc1nc(C(N2CCN(C3CCN(C(c4cnc(S)nc4)=O)C3)CC2)=O)cn1C C1(C(N(CCN(C(C(=O)OC)C)C)C)=O)CCCN(C2CCC2)CC1 c1(C(=O)NCC(=C)CCNC(=O)C(C2CC2)OCC)cnc(OCC(F)F)cn1 c1(SCC)c(C(N2CCCC(CN(C)C)C2)=O)n[nH]c1C1CC1 C(=O)(CCC=CBr)NC1C(CNC(CC(=O)OCC)=O)C1 C1(C(=O)OC)C2CCC(CC2)C1NC(=O)CC(=O)NCc1c[nH]c(C(C)(C)C)c1 N1(C(C2C(=C)C2)=O)CC2CCCC(NC(C3(COC)CCC(O)CC3)=O)C2C1 c1(OC)cccc(Cl)c1C(=O)NC1CCN(C(c2cccc(Cl)c2Cl)=O)C1 N1(c2snc(CC)n2)CCC2(NC(c3nc(C)c(C)nc3C)=O)CCCC12 C1(CNC(=O)CSc2cccc[n+]2[O-])CC2CCC1N(C(c1cc[nH]n1)=O)C2 N1(C(c2c(NCC#C)nccc2)=O)C(C)C2CC1C2NC(C1(OC)CC1)=O O=C(C1=CCCCC1)NC12CC(C1)N(C(c1ccc(F)c(Br)c1)=O)C2 C12(CC(=O)NCC(CNC(c3ccccc3)=O)OC)CCCC1C2 c1(CNC(C2(CNC(=O)CCc3ccsc3)CCOCC2)=O)ccc(F)cc1O c1(C(N2CC(NC(c3cnc(COC)s3)=O)C3C(C2)C3)=O)c(C)cc(O)nc1C C(C(C(=O)N1CCC(O)(CNC(C23CCC(CC2)CC3)=O)C1)C(F)(F)F)OC C(=O)(C(CNC(c1cnn[nH]1)=O)C(C)(C)C)N(c1ccc(O)cc1)CC#C C12(C(=O)NC(C3(CCF)CC3)C)C3C4C1C1C2C3C41C(=O)Nc1ccc(O)cc1 N1(C(C2C(C)CCO2)=O)CCCC2(CCC2NC(c2cc(C3(C)CC3)on2)=O)C1 c1(C(=O)NC(C(=O)NCC)C2CC2)cc(C(=O)OC)cc(Br)c1 CC1(C)CC(C(=O)NC2CCC(NC(C3(O)CCOCC3)=O)CC2)C1C(F)(F)F c1(CNC(N2CCC(C)C2C)=O)ccc(F)cc1N N1(C(C=C(C)C(C)C)=O)CCCC(C2CC2NC(=O)Cc2cncn2C)C1 CC1=C(C(=O)N2CCC(C)(C)C2CNC(C2CC2[N+](=O)[O-])=O)CCCO1 c1(C(N2CC3C(CNC(C4ON=C(C)C4)=O)(C3)C2)=O)csc2c1CCCC2 c1(C(=O)NCC(C(N2CC(CC)OCC2)=O)O)cnn2c1OCC2 N1(C(COC)=O)CC2(CCN(C(c3cccc(OCCN(C)C)c3)=O)CC2)C1 N1(C(COCCCC#C)=O)CC2CC(C(=O)NC(CCF)C(=O)OC)C(C2)C1 N1(C(CSCC(N)=O)=O)CC2CC(NC(c3cc(C(N)=O)cs3)=O)CC2C1 N1(C(c2cc(Br)nn2-c2ncccc2Cl)=O)CC(O)C2(CCC2)C1 Cc1cc(C)c(C=CC(=O)NCC2CCCC2NC(=O)CSS(C)(=O)=O)c(C)c1 c1(C(=O)NC(CCNC(C2(C=C)CCC2)=O)C)cnc2cc(C)nn2c1 N1(C(=O)NCC2CC3C=CC2O3)CC2CS(=O)(=O)CC2C1 C(=O)(CS(=O)c1cccc2occc12)NS(c1ccc(OC)c(C(=O)O)c1)(=O)=O C=CCCC(C)(C)C(=O)NCC(O)CN(C(=O)CCCC(OC)OC)C N1(CC(=O)N(CCN(C2CCCC2)C(=O)CC2CC2COC)CC)CCC(C)C1 C(C)(CNC(=O)CNC(c1ccsc1)=O)(C(C)C)NC(c1cnc(C)[nH]1)=O C#Cc1cnc(C(=O)NC(C)(CNC(=O)C(O)CCN(C)C)CC(C)C)c(C)c1 CCCCC#CC(C)(C)NC(c1ccc(C2CCCO2)[nH]1)=O C1(C(N2C3C(C(=O)NCC4(CC(C)C)CCC4)C(C3)C2)=O)CC12CCOCC2 c1(C(N2CCCCC(NC(=O)CC3CCCO3)C2)=O)ccn2ncc(Br)c2c1 c1(NC(C2CCN(C(CSC(C)=O)=O)CC2O)=O)cc(Cl)cc(Cl)c1[N+](=O)[O-] CCCCC(F)(F)C(=O)NC1CCN(C(c2nn(C)cc2CC)=O)CC1OC c1(C(N2CC(CNC(C(C)=CC)=O)C(C)(C)CC2)=O)cc2cc(Cl)ccc2o1 N1(CC(N2CC(O)(C(C(=O)NCCCOC3CCC3)F)C2)=O)CCOCC1=O C1(=CCNC(CCc2scc(C)n2)=O)CCN(C(=O)Cc2occc2C)CC1 C1(CC(=O)NCC23CC(NC(C4CC(CCC)C4)=O)(C2)C3)CCC(F)(F)C1 c1(CC(C(=O)NCCC2CN(C(COCC#C)=O)C2)O)ccc(C(F)(F)F)cc1 c1(OC2CCCN(CC(=O)NC(COC)C)C2)cc(C)cc(C)c1 c1(C(=O)NCC2CC(NC(C3C(OC)CCC3)=O)C2)ccc(Cl)c(O)c1 C(=O)(CS(=O)(=O)C1CC1)N1CC(CCCCN(C(C(C(C)O)C)=O)CCO)C1 N1(C(C2CC2F)=O)CC(CNC(=O)C(c2ccc(F)c(Cl)c2)(F)F)C2(CC2)C1 c1(C(N2CC(O)(CNC(C(C)C)=O)C2)=O)ccc(CNC(=O)C(C)O)cc1 c1(CC)cc(F)ccc1C(N1CCC(N(C(=O)COC(CC)CC)C)C1)=O C(=O)(Nn1cccn1)C1CN(C(CC(CC)OC)=O)CC1CC C1(CNC(=O)CCCF)CC2(CC2)CN1C(=O)CCC1CCCO1 c1(SC)ccccc1CC(=O)NC1CCC1CNC(c1csnn1)=O N1(C(c2ncn(C(C)(C)C)c2)=O)CC2CCC1CN2C(c1cnn(C2CC2)n1)=O C(=O)(CC(C)CC(C)C)N1C(CNC(c2cc(C)nn2C)=O)C(O)C(O)C1 c1(CC(=O)N(C(CNC(COC(CC)C)=O)C2CC2)C)cncn1C1CC1 N1(C(C2C(=C)C2C(=O)OC)=O)CCOC(C(=O)NC2(C(=O)OC)CC2)CC1 N1(C(c2c(C(=O)OC)[nH]cc2)=O)CCN(Cc2ncccc2Br)CC1 N1(C(CC2CC(=O)OC2)=O)CCCC(CNC(C2CCC(=O)O2)=O)C1 CCCS(=O)(=O)CC(=O)NCC1CCN(C(C2(CF)CC(=O)C2)=O)C1 c1(CNC(C(CC)NC(=O)C(C)NC(N)=O)=O)ccc(Br)cn1 c1(C(=O)NCC(n2cc(-c3cc(C4CC4)no3)nn2)C)cc(Cl)nc(Br)c1N N1(CC2C(C(C)C)C3CCC2C3)CCCOC(CCN)C1 Cc1[nH]nc(C(=O)NC(C)C(=O)NCc2ncc(CO)o2)c1C c1(C2(N(C3CCC(NC(C(C)C)=O)CC3)C(=O)C3CC3)CC2)cccc(C#N)c1 c1(COC)ccc(C(=O)NCC2(F)CN(C(C3CCC3C(=O)OC)=O)C2)nc1 C(=O)(C(F)(F)C(C)(C)O)NC1C(SC)CN(C(=O)CCCNC(=O)C2CC2)C1 C(=O)(C(C)(C)CCC(=O)NCC(C1CC1)NC(C1CCC(C)(C)CC1)=O)OC c1(CC(=O)N(C2C3CN(C(C4(OC)CC(C)C4)=O)CC32)C)ccc(Cl)cc1Cl Cc1ccc2c(c1)CC(C(=O)NCC(C)CNC(c1sccc1C)=O)S2 C12(NC(C3N(C(c4cccc(CC(C)C)c4)=O)CC3)=O)CCCC1OCC2 c1(C(=O)NCC2C(NC(C3(C(=O)NC)CCC3)=O)C2)cocc1C C1(C)(C(=O)NCC(CN(C)C(c2ccnc(OCCO)c2)=O)O)CCCCCC1 N1(c2nnc(CCC)s2)C(CNC(c2ccnn2CCOC)=O)CC2COCC12 C12(NC(C=C(C)Cl)=O)CCCN(C(c3ccc(NC(N)=O)cc3)=O)CC1C2 CC(=O)CCCCC(=O)N1CCCC1CCC(N1CCC(O)C1(C)C)=O N1(C(c2cc(C)sc2C)=O)C2CCC1CN(C(C13CC(CN1C1CC1)C3)=O)C2 C(C(=O)NC(C)CNC(c1ccn(-c2ccccc2Cl)n1)=O)(C(C)(C)C)OC c1(OC)cccc(C(=O)NC2(CCNC(=O)CC(C)C3CCCO3)CCC2)c1 C=CC1(CC(=O)NC2CC(N(C)C(c3cnccc3C)=O)C2)CCCCC1 N1(C(CS(CC)(=O)=O)=O)CC2CCC1C(C(=O)Nc1nonc1C1CC1)C2 N#CC1CCN(C(=O)C(=O)Nc2ccc(N3CCCC3=O)cc2)C1 CCC(CCCC(=O)N1CC2CC(C1)N(C)C2)NC(=O)C(F)(F)C1CC1 C1(CNC(C2CCC(OC)C2)=O)CC2(CCN(C(=O)CC3(C)CC3(F)Cl)C2)CO1 c1(C(N2C3CCC2C(F)C(NC(=O)CC2CC2)C3)=O)ccnc2c(F)cccc12 c1(C(=O)NC2CC(CNC(C3CCCN3C3CC3)=O)C2)[nH]ccc1CC1CC1 C(CNC(=O)Cc1nc[nH]n1)(C(=O)NCC(C1CC1)N(C)C)N(C)C C1(NC(=O)NC(C(c2ccc(C3(C(F)(F)F)CC3)cc2)C)=O)CC(S(C)(=O)=O)C1 N1(C(C2N(C)CCOC2)=O)CCN(C(=O)CNS(N)(=O)=O)CC(CO)C1 c1(C(N2CCC(CCNC(C(C3CC3)OCC)=O)CC2)=O)cncc2[nH]ccc12 CCCCCCCC(=O)N1CC(C(=O)Nc2cccc(F)c2C)C(C)C1 Cc1[nH]nc2ncc(C(N3CCOC(CNC(C4CC(N(C)C)C4)=O)C3)=O)cc12 Cc1[nH]nc(NC2CCC2c2cccc(OC(F)(F)F)c2)c1C(=O)O c1(C(C(=O)NCC(=C)C)N(C(CC2CC2)C(=O)OC)C)sccc1Br C=CCN=c1[nH]c(C(N2CC3CC2CCC3NC(=O)CN2CCCC2=O)=O)cs1 CCCCCC(c1nnnn1C(C)C)NCC(c1ccc(C)cc1)C c1(C(=O)NC2CCN(C(C3(CC)CCCC3)=O)CC2C)cc(N)c(Cl)c(O)n1 c1(C(=O)NCC2CN(C(c3ccc(OCC)cc3)=O)CC2C)cccn(C)c1=O C(CCC(C)C)(C(=O)NC(C)CC1(O)CCC1)NC(C1CC(CC)C1)=O C(CCCCNC(c1coc(Br)c1)=O)NC(CN(C)C1CC1)=O c1(OC)cc(C(=O)NC2CCC2CNC(=O)C(C)Sc2ccccn2)on1 N1(CCNC(=O)NCCC(C=C)C)c2ccccc2NS1(=O)=O N1(C(c2cnc(C(=O)OC)s2)=O)CC(C)(C)CC1CNC(=O)CSC(F)F Cc1cnccc1C(=O)NC1CCC(CNC(=O)CC2CCC3CC23)CC1 N(C(=NCCCCl)NC1CCN(CC2CC2)CC1)C(C)COC1CCOC1 c1(CN(C(=O)CN(C2CCCC(C)C2)C)CC)cc(Br)ccc1[N+](=O)[O-] Cc1nc(CC(N2CCCC2CN(C(=O)C(C2CCCCC2)O)C)=O)n[nH]1 N1(c2n(CCC(=O)NC)c(C3CC(F)(CO)C3)nn2)CCN(CC(N)=O)C(=O)C1 N1(C(c2c(C3(C)CC3)cccc2)=O)CCCC(F)(CNC(=O)CN2CC(C)(C)C2)C1 N12CCc3nc(ncc3CC1)NC2=O.C(CCN1CCOCC1)(C(C)C)OC N1(C(c2ccc(CCC)[nH]2)=O)CCCC(O)(CNC(=O)Cc2cn(C)nc2C)C1 c1(NC(CN(C(CCC#C)=O)C2CC(C#N)C2)=O)cc(CO)cc(F)c1 c1(C(=O)NC2CN(C(C3CCOC3)=O)CCC2CO)ccc2cccc(O)c2c1 C1(NC(C(n2cc(C)nc2)(C)C)=O)CN(C(C2CC2F)=O)CCC1C C(=O)(CC1=CSC2=NCCN12)NC1C(C)CCN(C(=O)C(C2CCCCC2)O)C1 Cc1cnc2n1CC(C(N1CC(NC(C3CC(=C4CC4)C3)=O)C(F)(F)C1)=O)CC2 CC(C)C(CNC(c1cc(Cl)cs1)=O)NC(=O)CCOC1CC1 Cc1cc2n[nH]cc2cc1C(=O)N(CC(C)O)CCNC(C1CS(=O)(=O)C1)=O c1(SC)ccc(O)c(C(N2CC(NC(C3CCCCN3C)=O)C3CC3C2)=O)c1 c1(C(=O)NCCN(C(=O)CCOc2ccc(Cl)cc2)C)cccc2nc(O)oc12 C1(OC)CC(C(=O)OC)N(C(=O)NC(c2csc(C(C)OC)n2)C)C1 c1(C(=O)NCC2CCN2C(c2cc3ccncc3[nH]2)=O)nncc2ccccc12 c1(C(N2CCCC(CNC(Cc3c(C)n[nH]c3)=O)C2)=O)ccc(P(C)(C)=O)s1 c1(C(=O)NC23COC(CNC(C4CCCSC4)=O)(C2)C3)cc(F)c(F)cc1F N#Cc1ccncc1C(=O)NC(C(=O)NOCC1CCOC1)C1CC1 C1(C(=O)NCC(CNC(C2(O)CCC(C)CC2)=O)(C)O)CC2(C1)CS(=O)(=O)C2 C1(C(=O)N(C2CCOC2)C2CC2)(NC(=O)NC(C)C)CCSC1 c1(-n2ncc(CN3C(C(N4CC(C)OCC4)=O)CC(O)C3)c2)ccc(C#N)cc1 C(=O)(C(F)C(F)(F)F)NC1CC(F)(CNC(c2cccc(C(F)F)c2F)=O)C1 C1(C(=O)N(CC(C)(C)CNC(C2CCOC2C)=O)C)(OC)CCS(=O)(=O)C1 C1(NC(CCN(CC)CC)=O)CC2CC1CN(C(c1ccc(CF)cc1)=O)C2 c1(OCC)ccc(CN2CCC3(CC3C(=O)Nc3cc(C)nn3C)C2)c(OC)c1 CC1C(C)SCCN1C(C(=O)N(CCC(=O)OC(C)(C)C)CCl)C(C)C1CCOC1 C(=O)(C(CC(C)C)NC(c1c[nH]c(C#N)c1C)=O)NC(C=C)C1CCC1 C12(CC(=O)NC3CCCC34CC4)CCC1CN(C(C1CC1F)=O)C2 c1(C(N(C)CC2CCCN2C(=O)C=CCO)=O)ccc2cc(Cl)ccc2c1 C1(NC(CCC=C(C)C)=O)CN(C(C2(C)CCCCO2)=O)CC12CC2 C(CC(C)C)(C(=O)N1CCN(C(c2nc(C)n(C)c2C)=O)CC1C(F)F)OC C=CC(C)(O)C(=O)NCCC1CSCCN1C(=O)CCc1ccoc1 O=C(C#CC1CCOC1)NC1CCSC12CN(C(c1cnc[nH]1)=O)C2 C(=O)(C1CCC(=O)c2cccn21)NC1CCCN(C(c2c(C)scc2)=O)C1 C(C)(CNC(=O)C=Cc1cocn1)(CNC(=O)Cc1ccn(C)n1)OC N1(C(C(CC(C)C)=O)=O)C(C(=O)Nc2cnc3c(c2)CCC3)C2CC(O)C1C2 C(CC(C)N=c1[nH]c(OCC)ncc1Cl)N(C(=O)C(CC)CC(C)C)CC C(=O)(CC(O)CC(C)(C)C)NCC(CCNC(=O)CC1CCCCC1)OC c1(CC)cc(C(=O)NC(C2CCCN2C(=O)C(CC)C(C)C)C)cc(O)n1 c1(OC)c(C(N2CCOCC2C(=O)NC(c2nc(C)oc2C)C)=O)cnn1C c1(C(=O)NC2CC(CNC(C3(F)CCCC3)=O)C2)n[nH]c2cccnc12 C1(CC)CN(C(=O)C(Cn2cccn2)NC(c2scnc2Cl)=O)CC1F c1(Nc2ccn(COC)n2)ncccc1S(=O)(=O)N1CC(C)N(C)C(C)C1 N1(C(C2CCCC(OCC)C2)=O)CCCC2(C1)CN(C(C1(C(=O)OC)CC1)=O)C2 CC1(C)CC(NC(=O)COCCF)CN1C(c1cnsn1)=O O=C(CCCCCn1cnnn1)NCC1(NC(c2ccc(Br)s2)=O)CC1 c1(OC)cc(CN2CCC(F)(C(=O)NC3COC(=O)C3)C2)c([N+](=O)[O-])cc1OC n1(CC)nc(C(=O)NC2C3CC2N(C(=O)CC2CC(C(C)(C)C)C2)C3)ccc1=O c1(C(=O)NCCC(C)NC(c2cc(C3CCCC3)n(C)n2)=O)cn2c(n1)CCC2 C(=O)(CC(C)C(F)(F)F)N1CCCC(CNC(c2ccc(OCC)cc2)=O)CC1 CCC(COC)C(=O)NCC1C2CC1N(C(=O)CCOc1cccc(C)c1)C2 C1(C(C(=O)NCC2C(C(C)C)C2)(C)C)CCCN(C(c2ccncc2)=O)C1 N1(C(CNC(C)=O)=O)CC2COCC2(C(=O)NCC2CCCN2C)C1 c1(OCc2cccc(C(=O)OC(C)(C)C)c2)ccc2[nH]c(=O)c(=O)[nH]c2c1 c1(OC)cncc(C=CC(=O)NCCN(C(C2CNC(=O)CC2(C)C)=O)CC)c1 C1(CC(=O)N(CC)CC2CCCN2C(c2ccccc2Cl)=O)CCCNC(=O)C1 Cc1cc(C(N2CCC(c3ccncn3)CC2)C(=O)NC(C)C)ccc1Br c1(C(N2C(CCCNC(C3C(CC)C3)=O)CCC2)=O)cnc(O)c2ncccc12 c1(C(N(C)CCn2cc(-c3ccc(F)c(F)c3N)nn2)=O)scc2c1OCCO2 c1(SCC(=O)NC2CN(C(C(C#C)(C)C)=O)CC2C)ccc2ccccc2c1 C1(NC(c2ccc3ccnn3c2)=O)CCC2(CC1)CN(c1ncncc1Cl)C2 N(C1CCOc2cc(Br)ccc21)C1OC(=O)N(c2ccccc2C(F)(F)F)C1 C(=O)(CCCC(N)=O)NCC(CO)NC(c1ccc(CSC)cc1)=O N1(CC)CCOCC1C(=O)N(C)CCN(C(=O)CCC1CCCC(=O)N1)C(C)C C1(CNC(C2CC2F)=O)CCC2(CC1)CCN(C(c1c[nH]cc(Cl)c1=O)=O)CC2 N1(C(Cc2c(O)ccc(C)c2)=O)CCOC2CCN(C(=O)C(C)C(C)C)CC12 Cc1cc(=NCC2(CNC(C3CC(C4CC4)C3)=O)CCCC2)[nH]c(C(F)(F)F)n1 N1(C(C2C(C=CC)CN(C(=O)C(C)CC(C)C)C2)=O)CCC2(CC(F)C2)C1 C#Cc1ccc(C(=O)NCCSC2CCCN(C(=O)C=CCF)CC2)nc1 C=C(C)CC(C)C(=O)NCC(C)(C)CN(C)C(c1ccc(O)cc1F)=O CC(C(=O)N1CCC(C(=O)NC2CCCCC2N=[N+]=[N-])O1)c1ccn(C)n1 c1(CN2C(C(=O)Nc3cn(C(C)(C)C)nc3)CCC2)ccc2ncnn2c1 C1(CNC(C2(C)C(C)C2)=O)CCC2(CC1)CC(NC(c1cc(O)n(C)n1)=O)C2 c1(C(=O)NC2C(NC(Cc3nc(C)[nH]n3)=O)CC2)cc(C)c2ccccc2n1 c1(C(=O)NC(C)C(C)(C)NC(=O)CN(C2CCSC2)C)nccc(Cl)c1O C1(CNC(C(C)(C)OCC)=O)CCC2CN(C(c3ccnc(CC)c3)=O)CC12 Cn1cc(OCC(=O)NC2CCC(NC(=O)Cc3c[nH]nc3O)C2)cn1 Cc1nc(C(F)(F)F)cc(C(N2CC(NC(=O)C(=O)C3CCCC3)C2)=O)n1 C1(NC(c2c(CC)c(C)sc2)=O)CCCN(C(c2ccc(N(C)C)cn2)=O)C1C CC1(C)Cc2ccc(C(=O)NCC(C)NC(c3cc(Cl)ccc3F)=O)c(O)c2O1 c1(CC(=O)N(C2CCN(C(C=C3CCC(C)C3)=O)C2)C)ccc(C(N)=O)nc1 N1(C(N2CCC(Cc3nc[nH]n3)CC2)=O)CCCCC1CCCO c1(C(=O)NC(C)(C)CCNC(=O)CC2CCCO2)ccc(Cl)c(C#N)c1 CC1c2cc(F)cc(Cl)c2CCN1C(=O)NC1CCN(c2ccccc2C#N)C1 C12(C(=O)NC3CN(C(C=Cc4c(C)n(C)nc4)=O)C4C3C4)CCC(F)(CC1)CC2 C1(CNC(=O)COCC2CCCOC2)CN(C(C2CC23CC3)=O)C2(CCC2)C1 c1(C(N2CCC(O)(C(=O)NCCCC=CC)C2)=O)nc(C)ncc1Br CC(C)C(C)CC(=O)N1CC2CC(C(N3CCCC3C(C)O)=O)(C2)C1 N1(C(=O)OC(C)(C)C)CC(O)CC1(C)CNC(c1csc(O)n1)=O CCCC(C)(C)CC(=O)N1CCC(F)(CNC(C2CC23CCCCC3)=O)C1 N1(C(c2cnc(CC(C)C)[nH]2)=O)CC(CNC(C2CC(O)C2)=O)CC12CCC2 CC(C)C(O)CCN=c1[nH]c(=NC(C)c2ccsc2)c2[nH]ccc2[nH]1 CCC(CC(=O)NC1CCCC1CNC(C1(CSC)CCC1)=O)C1CCC1 C1(C(=O)NC2C(CNC(CC(C)=C(C)C)=O)C2)CCCCCCC1 C(=O)(C1=CCCCC1C)NCC1N(C(c2cnc(CC(C)C)[nH]2)=O)CCC1 c1(C(=O)NC(CCOC)CNC(=O)C(C)(O)C(C)C)ccc2nn[nH]c2c1 n1(CC)cc(C(=O)NC2CCN(C(=O)CC3C=CS(=O)(=O)C3)C2CC)c(C)n1 C(=O)(CC(C)CNC(=O)C(CC1CC1)NC(=O)Cc1ccnn1C)NC c1(SCC)cccc2cccnc12.c12nc(n(-c3cnn(C(C)C)c3)n1)CC2C CC1(C(=O)NC2CCCC2NC(c2cncc(C(F)(F)F)c2)=O)CC=CCC1 N1(C(C=CC=CCC)=O)CC(C)(NC(=O)CC2CCCN2C(C)=O)C1 N1(C(C2(C)CC(C)C2)=O)CCC2CN(C(c3cc4cscc4s3)=O)C2C1 C1(C)(C(=O)NC2CN(C(C(c3cccnc3)OC)=O)CC2C)CC2CCC1C2 N1(C(c2cc(C)n(C)c2)=O)CC(C)N(C(c2nnn(C(C)(C)C)n2)=O)CC1C Cn1cnc2cccc(C(=O)NCc3nc(CNC(C4SC5C=CC4C5)=O)cs3)c12 C=C1CC(C)(C(=O)NC2CC(N(C(=O)CC(C)OC)C)C2)C1 c1(OCC(=O)NC2CCC(NC(c3cc(C(F)F)no3)=O)CC2)ccccc1O N1(C(c2c(C)c(N)cnc2)=O)CCN(C(=O)Cc2cn(C)nn2)CC12CCC2 CC1CCOC(C(=O)N(C)CCOCCNC(c2cnn(CCO)c2)=O)C1 C(=O)(C(CCSC)NC(=O)CC1CCCC1)N.CCC(CN1CCCC1)OC c1(C(=O)NC2(C)CCN(C(c3nnc(Cl)cc3N)=O)C2)ccc2oc(S)nc2c1 C1(C(=O)NC(C(=O)OCCC)C)N(C(=O)C(C)N(C)C)CC12CCCC2 c1(NCCC(=O)NC2(CN(C(=O)Cc3cc[nH]c3)C)CC2)ccccn1 N1(C(c2n[nH]cc2I)=O)CCC2(CCCN2S(=O)(=O)c2c(Cl)cccc2Cl)CC1 Cn1ncc2c(O)cc(C(N3C4CCC3CN(C(=O)Cc3csnn3)C4)=O)cc12 C1(F)(C(N(CCOc2cccc(C)c2)C)=O)CCCN(C(=O)CN2CCCC2)C1 C1(C(N(C)CCN(C)C(C2CC3(C2)CS(=O)(=O)C3)=O)=O)CC2CCCC(C1)C2=O c1(C(N2CC(C)CC(NC(CCc3ccc(C)s3)=O)C2)=O)ccc2nc[nH]c2n1 C(=O)(CCCCCn1cc(Cc2ccc(F)cc2)nn1)N(C(C(=O)OC)C)C C1(CNC(COCCOC)=O)CN(C(c2cnc(C)nc2O)=O)CC12CC2 c1(C(N2CCC(CC3COCCO3)C2)=O)cc2[nH]c(-c3cccs3)cc(=O)n2n1 C(=O)(CC(C(F)(F)F)OC)N1CC(NC(CCC)=O)C(C)CC1 C1(NC(=O)CCC2CCC2)CCCC(NC(=O)CCn2cc[nH]c(=O)c2=O)CC1 N(C1CCSc2ccc(F)cc21)C(CCC(C(=O)OC)(C)C)=O C1(O)(CNC(CC(CC)SC)=O)CC2CCC(C1)N2C(=O)C(C)(C)C(C)(C)C n1(CCC)cc(Cl)c(C(=O)NC2CC(O)(CNC(=O)CC3C=CCC3)C2)n1 C1(NC(c2nn(C)c(C3CC3)c2)=O)CCN(C(C2(C(N)=O)CC2)=O)CC1CO C1(NC(c2c(CCC)nns2)=O)CC(O)CN(C(c2onc(C)c2C)=O)C1 c1(CC)ccccc1OCCC(=O)NC(C)(CC)CCNC(=O)CCCF C1(C(N(C)CC2(O)CN(C(C(C)OC3CCCCC3)=O)C2)=O)Cc2nccn2C1 c1(OC)c(C(F)(F)F)n[nH]c1Cc1noc(C2(C)CC2)n1 c1(CC(=O)NC2C(CNC(CC(CN(C)C)O)=O)CCCC2)cc(Cl)ccc1O N1(C(c2ccn(COC)n2)=O)CCC(C2CC(NC(=O)CCCOC(C)C)C2)C1 C(N=c1[nH]cnc(C)c1F)C1(NC(CNS(CC)(=O)=O)=O)CCCCC1C C1(C(NOCCCC)=O)CC(C)N1C(=O)CN=[N+]=[N-] C1(N(C(c2c(CC)occ2)=O)C)CN(C(=O)Cc2ncn(C)c2C)CC1F N1(C(c2cnc(COC)s2)=O)CCCC2(C1)CN(C(=O)C(F)n1ccnc1)C2 Cc1c[nH]c(=NCCNC(=O)C(c2ccc(Cl)cc2)(C)O)c([N+](=O)[O-])c1C Cn1c(O)nc(N2CC3(CCC3)CC2CNC(C2CC2c2ccsc2)=O)cc1=O N1(C(CCc2cnn(C)n2)=O)CC2CCC(C1)N2C(c1ccc(C2CC2)s1)=O CCC(C)(COC)C(=O)N1CCCC(N(C(=O)C=CCN2CCCC2)C)CC1 C1(CNC(C(F)=CC)=O)COC(C)(C)CN1C(c1cc(C)c(C)c(F)c1)=O C=CCC(C(=O)NCC(CC(C)C)NC(c1cccc(C(F)F)c1)=O)OC N1(C(C=CCC)=O)CCC(C)C1CNC(C1(COC)CC1)=O C=CC(CC)CC(=O)NCc1ccoc1C(N1CCOC(C2(C)CC2)C1)=O Fc1ccc(CNC2COCCN2c2cc(-c3ccccc3)ncn2)cc1F C1(NC(CN(C)Cc2cn(C3CCC4CCC34)nn2)=O)CC(C(=O)O)C12CCC2 C(=O)(C(CCC1CCCC1)N1CCCC1CC1CCC1)NC(C)C C1(C(N2CCC(C)(NC(c3nnn(CC)c3C)=O)C2)=O)CC(C)(C)CN1C c1(C(=O)NCc2c(CN(C(C(CC=CC)C)=O)C)cccc2)cn2c(n1)CCC2 c1(CN2CC(C(=O)Nc3c(CC)noc3C)C2)ccc(OC)c(Br)c1 N1(C(C2CC2NC(C)=O)=O)CC2CCC(C1)N2Cc1c(-c2cccs2)noc1C N1(C(c2cccnn2)=O)CCC(F)(C(N2CCC(O)(CO)C2)=O)CC1 N1(C(C(CCC)N(C)C)=O)CC(CNC(=O)C(=O)Nc2ccccc2)C(C)(C)C1 C12(NC(CCCC)=O)CC1CN(C(C1CCCC1C(=O)OC)=O)C2 C(CN=c1[nH]nc(O)s1)C1N(C(=O)CCCc2cnn[nH]2)CCCC1 C1(C)(CC)C=C(C(=O)N2CCOCC(NC(=O)CCn3cncn3)C2)C1 N1(C(CCCCOCC)=O)CCC2(CCC2NC(C2CCCO2)=O)CC1 c1(C(=O)NC2CC(C)N(C(=O)Cc3cncn3C)CC2)cncc2n[nH]cc12 C1(NC(C23CC(NC(CCc4cc(C)on4)=O)(C2)C3)=O)(CO)CCC(C)C1 C1(C(=O)NC(CC)CC(=O)OC)CCCCC1(C)NC(=O)C=CC(F)F C(C(C)(C)C(=O)NCC=CBr)NC(CC(C)C1CCCO1)=O C1(OC)CC2(C1)CC(C(=O)NC1CN(C(c3ncccc3F)=O)C3CC13)C2 c1(OC(C)C)cc(C(N2CCN(C3CN(C(C4(C)CC4F)=O)C3)CC2)=O)ccn1 c1(C(=O)NCCC2CN(C(C3CC=CCO3)=O)CCCO2)c[nH]c2ncccc12 c1(C(=O)NC2CC(NC(C3CNC(=O)O3)=O)C2)cnc2c(Br)cccn12 c1(C(=O)NCC2C(CNC(c3cn(C(C)(C)C)nn3)=O)C2)cc(N)c(F)cn1 C1(C(c2ccccc2)C)CCN(C(=O)OCC(C)(C)C)CC1 C(CCCC(=O)NN1CCCC1C(=O)N(C(c1ccccc1)CO)C)OC CCC(C)(C)CCCC(=O)N1CC2CC2(CNC(=O)CCCc2nncn2C)C1 N1(C(c2cnn(C)c2Cl)=O)CC2OCC(C(N3CCC(c4cnco4)C3)=O)C2C1 N1(C(C2CC(CC3CC3)C2)=O)CC2(C(=O)NC3CCCC(O)CC3)CCC1CC2 c1(C(N2CCCN(C(=O)C(O)C3CC3)CC2)=O)ccnc2c1CCC2 C(=O)(C(C)(C(F)F)c1ccccc1)NC1CCN(C(c2c(C)oc(Cl)n2)=O)CC1 C1(N(CCOC)C(c2ccc(Cl)cc2)C)COC2(CCNCC2)C1 C(=O)(CC1OCc2ccccc21)NCC12N(C(C(CCC)C(C)C)=O)CC(C1)C2 N1(C(C(C2CCCCC2)N(C)C)=O)CC2COCC2(NCC=CCl)C1 c1(CC(=O)NC(C2OCCOC2(C)C)C)c(Br)cccc1Br c1(OC)cc(C(N2CC3CC2CC3NC(=O)CC2(OC)CCC2)=O)cnc1O C1(C(N2C(C#C)CC2)=O)CC12CCN(C(c1noc(C)c1C)=O)C2 N1(Cc2ccc(CC)cc2)CCN(c2cc(N(C)CC)nc(CC)n2)CC1(C)C n1(CCC)nccc1C(=O)NC1C=CC(C(=O)NOCC2CCC3CC23)C1 c1(C(=O)NC2CCC(N(C(=O)Cc3cncs3)C)C2)ccc(S(C)(=O)=O)o1 N1(c2nnc(C(N(CCCCCC)CCOC)=O)s2)CCN(C)CC1 CCC(CCC(=O)NCC1CN(C(c2[nH]ccc(=O)c2C)=O)C1)OC N1(C(c2c(SC)ccs2)=O)CCN(C(c2cc(C)cs2)=O)C(C)CC1C C(=O)(C(C)C(=O)N1CCCC1(C)C(N1CCN(C(=O)C2CC2)CC1)=O)OC C1(NC(CN(C(=O)OC)C)=O)CCC(C)(C)N(C(=O)CN(C)C(N)=O)C1 C1(C(F)(F)F)(C(=O)NCC(CC)NC(c2cncc(N)n2)=O)CC=CCO1.CC Cc1ccc2c(c1)C(CC(=O)NCC(C)(C)CNC(c1cccs1)=O)C(=O)N2 C(=O)(C#CC1(C)CC1)N(CC(C)N(C)C(c1csc(C2CC2)n1)=O)C C(CCCC(C)NC(=O)C(c1cnn(C)c1)C1CC1)NC(C(COC)C)=O Cc1ccc2c(C(=O)NCC(CC(C)C)NC(=O)Cc3ncc(C)s3)coc2c1 c1(C(N(C)CC2CCCN(C(C(CC)SC)=O)C2)=O)cccc(=S)n1O c1(NC(C2(C)CCN(C(C3C(C)C3C)=O)C2)=O)cccc(N=[N+]=[N-])c1 C1(C(N2C(C(=O)NC3(CC#C)CCC3)CCC2)=O)CC(=O)N(OC)C1 n1(CC(=O)N(C2CCN(C(=O)C(CC)NC(C)=O)C2)CC#C)cc(Br)c(C)n1 CC1=C(C(=O)NCCC(C)NC(=O)Cc2sccc2Br)SCCO1 N1(C(CC(C(C)C)O)=O)CCC2C(CCCN2C(=O)Cc2ccc(F)cc2Cl)C1 C1(C#CC(=O)NCC2CCCC2NC(c2cnc3ccnn3c2)=O)(CC)COC1 N1(C(CCc2cc(C)[nH]n2)=O)CCC(C)(CNC(C2(C)CCCCC2C)=O)CC1 CC(C(=O)NCCC(C)N1CCC1)C(C)NC(c1ccnnc1O)=O CCCC(C)(O)C(=O)NCCCCCCNC(C1C2C3CCC(C3)C12)=O Cc1nc(C)c(CCC(N2CC(NC(C3(N(C)C)CCC3)=O)C3CC23)=O)c(O)n1 c1(C(=O)NC(C2CCCCCC2)CC)ccc(-n2cc(CCOC)nn2)cc1C c1(C(N(CC(C)NC(c2nn(C(CC)C)c(C)c2)=O)C)=O)c(C)nc2sccn12 c1(C(=O)NCC2CCCN2C(=O)C(c2ccc(Cl)s2)=O)cccc2oncc12 C(c1cnc(O)nc1O)=CC(=O)NCC1(NC(c2c(C)[nH]c(C#N)c2)=O)CCC1 C12(CNC(c3cnsc3)=O)CCC(CC1)N2C(C1CC2(C1)CC(O)C2)=O c1(NC(C(=O)NCC2(CO)CC3CCCC3C2)=O)cccc2ccccc12 N1(C(c2ccccc2F)C)CCC(C2(NC(=O)Cc3cccs3)CC2)CC1 C12CC3(CCN(CC3)C1)CO2.c1(CNC(CC=C)=O)csc(-c2ccncc2)n1 C1(CNC(C(C=C)C)=O)CCN(C(=O)C(C)NC(C)=O)CC1 N1(C(c2cc(C)sc2C)=O)CCCN(C(=O)CN(C2CCC2)C)C(C)C1 c1(C(=O)NC2CN(C(=O)C#CC3CCCC3)CC2F)cc2cc(F)ccc2o1 C1(NC(c2c(CCC)n[nH]c2)=O)CC(NC(=O)C(CC)C2CCC(=O)N2)C(O)C1 n1(NC(C(C)N(C)C)=O)cc(Cl)cn1.C12CN(C1)C(=O)C(C)N1CC(C1)C(=O)NC2 C1(C(=O)NC2CC3N(C(c4c(OC)nsc4)=O)C(CC3)C2)CCc2cnc(C)n2C1 c1(CC(=O)NC2C3CCN(C(C(C)n4ccnn4)=O)C32)ccc2c[nH]nc2c1 C(=O)(CCS(C)(=O)=O)N1CC(CNC(c2c(CCC)n(CC)nn2)=O)C2C1C2 C1(=CC(N2CC3C(NC(Cc4nc(=N)[nH][nH]4)=O)C(C3)C2)=O)CCCCCC1(F)F C1(NC(Cn2c(C)cnn2)=O)CN(C(=O)C(C)N2CCCC2)CC1C(F)F c12c(cc(Cl)cc1C(=O)N(C1(C)CCOCC1)C)C(=O)N2.N(C)(C)C(=O)OC c1(C(C(N2C(CO)CC(NC(CCCOC)=O)C2)=O)C)nc(F)ccc1Cl C1(C(=O)NC(c2ccsc2)C)CSCN1C(c1cnsc1)=O c1(OC)c(C(=O)N(C)Cc2ccc(O)c(C)c2)cccc1C1CC1 N1(C(C(C2CCOC2)OC)=O)CC(CNC(=O)C(C)CSC)(OC)C1 c1(CC)ccc(C(N2CCC(CNC(C3CC(C)C3)=O)C(C)C2)=O)cc1N c1(C(N)=O)ccc(N2CCN(Cc3ccc(-c4ccccc4)s3)CC2)nc1 CCCCC(C)C(=O)NCc1c[nH]nc1C(=O)N(C)Cc1scnc1C CC1(C)CN(C(C2CC2C2CC2)=O)C(CNC(c2cc(N)cc(F)c2)=O)CO1 C1(NC(C2(CCOC)CC2)=O)C=CC(C(=O)NCCCn2cccn2)C1 CCC(C(=O)NC(C)C(C(=O)N(CC(C)(C)O)CCO)C(C)C)C(C)(C)CC c1(C(N2C3CCC(NC(c4c(C)nc(CC)o4)=O)(C3)C2)=O)cc(S(N)(=O)=O)cs1 C(=O)(CC(CCCCCNCC1CCCC12CC2)C(F)(F)F)OCC(=O)O C12(Nc3nccc(CC)n3)CCN(CC1)C2=O.C1(C)(SC)CC1 N1(C(c2c(OC(F)F)cc(C)s2)=O)CCN(C(C2CCC2)=O)CC(CO)C1 N1(C(C2CCC(OC)CC2)=O)CCOCC(NC(C23CCC(OC)C2C3)=O)C1 c1(C(c2nnnn2Cc2ccco2)NC(=O)NC2CCCO2)ccc(F)cc1 c1(C(=O)NC(CN(C(C2CCOC2SCC)=O)C(C)=O)C)[nH]cnc1C N1(C(C(c2scc(C)n2)C)=O)CC(NC(=O)CCC23CCC(CC2)C3)C(C)C1 C(=O)(C1=CC(O)C(NC(=O)C(c2cncn2C)O)C1)NCCCC(=C)C CC1CN2CCC1NC(C(C)O)C2=O.c1(CNC(=O)OC(C)(C)C)ccccc1 C(=O)(C(F)C(F)(F)F)NCCC1N(C(CCc2cncc(OC)c2)=O)CCCC1 C1(NC(CC2CC(N(C)C)C2)=O)CC(O)CN(C(C23CCC(C2)C3(C)C)=O)C1 c1(CC(=O)NCC2N(C(Cc3nc(C)sc3)=O)CCC2)c(C)nn(C(F)F)c1C C(=O)(C(C)(C)CCNC(C1CCC1COC)=O)NC(CC)C(C)(C)O Cc1nnc2cc(N3CCC=C(CNC(c4cccc(F)c4F)=O)C3)ncn12 CCCC(C(=O)N1CCC(O)C(NC(=O)CCc2ncc[nH]2)C1)C(C)C Cc1nc(N)cnc1C(=O)NCCCN(C)C(C1(C)CCCO1)=O C=CCC(CCCCC)C(=O)NCCCCC(C)NC(=O)Cc1cc(C)no1 N1(C(c2nc(C)n(C)n2)=O)CCN(C(c2cccn2C)=O)CC1c1ccccc1 Cc1nn(CC(=O)NC(C)CCC(=O)N2CC(C)=C(C)C2)c(=O)o1 C1(CC)C(NC(=O)Cc2cc(C)nn2C)CCCN1C(=O)COC1CC=CC1 C1(C(C(N2CC(N(C(C(C)OCc3ccccc3)=O)C)C2)=O)O)CCCCCC1 N1(C(CS(CC)=O)=O)CC2CN(C(c3cccnc3C3CC3)=O)CC2(C)C1 c1(C(=O)NCC2(O)CCN(C(C(CCC)OC)=O)C2)c(C)nn(C)c1OC Cc1ccc(C(=O)NCC2CC(C)N(C(c3nc(C(C)C)oc3C)=O)C2)c(F)c1 N1(C(CC(C)(C)OC)=O)CCN(S(=O)(=O)N2CC(C)OC(C)C2)CC1 C(=O)(C1=Cc2cc(F)ccc2OC1)NC(N1CCN(C2CCC(OC)C2)CC1)=O c1(C(=O)NC(CC)CC(=O)NCC23CCC(CC2)C3)cccc(O)c1F C1(C(=O)NC2CC(NC(Cc3ccc(C#N)nc3)=O)C2)CC2CCC1CC2(F)F Cc1cc(O)ccc1CC(=O)NC1(C)CCN(C(c2cnn(C)c2)=O)C1 N1(C(C)=O)c2ccccc2CC1C(=O)NCC1([Si](C)(C)C)CC1 C#CC1CC(NC(=O)C(C)CN(C(=O)CCC2CCCOC2)C)C1 N1(C(C(c2cnn(C)c2)C)=O)CC(O)CC1C(=O)NCc1cncc(Cl)c1 C1(C(=O)NC(CC)C(=O)NCC2CC3(CCO2)CC3)CC2(CCO1)CC2 c1(OC)ccccc1C(C)NC(=O)C(=O)NC(C1CCCO1)COC c1(C(=O)NCC2OCCN(C(c3onc(C)c3C)=O)C2)ccc2occ(C)c2c1 C1(NC(C=Cc2nc(C)sc2)=O)CN(C(=O)CCc2ccccc2)CCC1CO C1(C(N(CCCNC(=O)CCC(=O)c2cccnc2)C)=O)CNC(=O)CC1(C)C c1(NC(C2C3(CC(C)(NC(=O)OC(C)(C)C)CC2)CC3)=O)cccc2ccsc12 N12CCC1C2=O.C1(CC#C)(C(=O)NCCOC(C)C)CCC1 C1(NC(C2C3CCOCC23)=O)CC2(C1)CN(C(=O)CCc1nnc(S)nc1O)C2 C1(C(=O)NCC(C(=O)NCC2(CF)CC2)N(C)C)CCN(C)C1=O C1(C)(C(=O)NCCN(c2ncc(C(=O)OC)cn2)CCC)CCCCCC1.C(C)(=O)OC c1(C(N(C)CC2CCCN2C(C2OCCOC2(C)C)=O)=O)ccnc2[nH]nnc12 N1(C(CC#C)=O)CCN(C(c2cc(C)nc(C)n2)=O)CC1C Cn1c(-c2ccc(Cl)cc2)nnc1C1CC(=O)N(C(C)(C)C)C1 C1(NC(CC(=O)OCC)=O)CC2CN(C(=O)COCCO)CC2C1 c1(CC)cc(=NC(C)C2COc3ccccc32)[nH]c(-c2ccoc2)n1 C(=O)(C1=CCC(NC(C2CCCCCC2)=O)C1)NCC(c1ccsc1)C C1(C(=O)NCc2cscn2)CN(C(=O)Cc2ccc(Cl)cn2)CCC1O c1(CN(CC(=O)O)C(C2CCC(=O)N2)=O)cn(CC2CCCO2)nn1 c1(C(=O)NCC(CNC(CCSCC)=O)O)cc2c(OC(F)(F)F)cccc2[nH]1 c1(CSCC2(CNC(C(N)CC3CCCCO3)=O)CC2)ccc[n+]([O-])c1 C1(SCC(=O)NCC2CCCC(NC(c3c(C)cco3)=O)C2)CN2CCCN1CC2 c1(C(N2C3C(NC(CCCCCC)=O)(CCC3)CC2)=O)ccc2c(c1)C(=O)NC2 CS(=O)(=O)C1CC(C(N2CCCC(Nc3cc(O)nc(O)n3)C2)=O)C1 C1(C(=O)NCC(C)(C)NC(COCC(=O)NC)=O)CSCC1C CC(CO)C(=O)NCCC(C)(C)NC(=O)C(C)COc1ccccc1 C(=O)(N=c1[nH]oc2cnccc12)C1N(C(c2cc(C(C)=O)[nH]n2)=O)CC2(CC2)C1 C(CCO)(C(=O)N1CC(CCNC(c2cc(-n3ccnc3)ccn2)=O)C1)N(C)C c1(C(=O)NC2CCN(CCNC(C(C)=C(CC)C)=O)CC2)cccc(F)c1F CCCC(CC)C(=O)NCc1cc(C(=O)N(C)CCc2ncccn2)cs1 C(=O)(C#CC1CCOC1)NCCN(CCOC)C(C1COCC(=O)N1C(C)C)=O C1(C)(CNC(C(CC)O)=O)CCCN(C(=O)C(c2ccc(Cl)cc2)=O)C1 N1(C(c2n(C)cnc2)=O)CCC(O)(C2CCN(C(=O)C(=O)NC3CC3)CC2)C1 Cc1ccc2nc(C)cc(C(=O)NC3CN(C(c4ccn(C)c4)=O)C3)c2c1 C(C)(C)(CCC(=O)NCCC(=O)NCC(C)SC1CC1)NC(C)=O Cc1cc2c(NC(C3CC3C(=O)NCc3c(Cl)cccc3Cl)=O)cccc2s1 C1(C(N(CCC)CCCCCNC(=O)COC(C)(C)CC)=O)CCCN1C=O C1(NC(C(C(C)C)CNC(c2sccc2CO)=O)=O)CCC2CCCC1O2 Cc1ccc2c(c1)C=C(C(=O)NC1CCC(CS(N)(=O)=O)C1)CO2 Cn1c(C(=O)NCC2CC(C(=O)NC3CCN(C4CC4)C3)C2)cnc1O C(C(C)C)(C(O)C(=O)N(C)CCOCCC(=O)NC1CC(F)(F)C1)OC C1(NC(Cc2c(Cl)cn(C)n2)=O)CC2(NC(c3ccn(C(F)F)n3)=O)COC1C2 N1(C(C(C)Nc2scc(C)n2)=O)CCC(C2CC2)(CNC(C2(Cl)CC2)=O)C1 O=C(C#CC1CCOC1)NC1CCC12CN(C(c1ncc(F)cc1F)=O)C2 c1(C(N2CCC(CN(C)CC)CC2)=O)cc(F)cc(Cl)c1.CCCC=CC(=O)O N1(C(C(CC2CC2)NC(c2c(CC)ncnc2)=O)=O)CCC12CCN(C)C2 c1(C(=O)NCCC(C)NC(c2ccn(CCC)n2)=O)cnc2n1CCC(C)C2 N1(C(C(CSC)OC)=O)CC2CCC1CN2C(C12CCN(CC1)C2)=O N1(C(COc2cc(C)on2)=O)CCC(CO)(NC(C2CCC(N(C)C)C2)=O)CC1 C(=O)(C1COc2ccc(Cl)cc21)NC(CCC)CCCNC(=O)CCC(=O)NC N1(CC2(OC)CCC2)CCCCC1c1cn(CC(O)CNC(C)=O)nn1 c1(CNC(c2ccc(C)cc2)C(=O)O)ccc2cc(F)ccc2n1 c1(C(N(CCN(C(C(C(COC)C)C)=O)C)C)=O)cncc(S(C)(=O)=O)c1 c1(C(N)=O)ccc(NC(=O)CC2CCCN2C(c2ccc(O)nc2Cl)=O)cc1Cl N1(C(=O)CCC2CC2)CCC2(CCCN2C(=O)Cc2nc[nH]n2)C1 C(CC(=O)N1CC(CO)CC(C)(C)C1)(C(F)(F)F)NC(C=CC(CC)C)=O C1(C(=O)NCCN2CCC(NC(c3c(C)nsc3N)=O)CC2)CCCCNC1=O N1(C(C(F)OC)=O)CCCC2(CCCN(C(c3cnc(O)c(Cl)c3)=O)C2)C1 CCC(CC)CCCC(=O)NCC1CC12CCN(C(=O)Cc1ccc(C)o1)CC2 n1(CC(C)NC(c2cc(C(F)(F)F)co2)=O)cc(CCC2CCOCC2)nn1 C1(CNC(C2C(CC)CCC2)=O)CCN(C(C2CCSCC2)=O)C1(C)C c1(C(=O)NCC2CN(C(C(C)(C)C3CCCC3)=O)C2)ccc2cccc(Cl)c2n1 C(c1cccc(O)c1)=CC(N1CCC(O)(CNC(c2scnc2C2CC2)=O)C1)=O Cc1nn(CC(=O)NC2CC3CC(NC(=O)C=C4CCC(C)C4)C2C3)c(=O)n1C C1(CC(=O)NCCN(C(=O)C(c2ccccc2)O)CCOC)COCCO1 c1(C2(C(=O)NCC(c3ccccc3)CNC(c3c(C)cno3)=O)CC2)cccnc1Cl c1(C(=O)NCC(CNC(C(C)NC(C)=O)=O)(C)F)cccc(F)c1F.CC(F)(F)F c1(C(=O)NC(CNC(C(C(C)C)C)=O)CC(C)C)ccc2occc2n1 C1(NC(c2ocnc2C2CC2)=O)CC12CC(NC(C1CC13CCCC3)=O)C2 c1(CNC(CC2CC(=C)C2)=O)cccc(CNC(C2COC(C)C2)=O)c1 CC1=C(C(=O)N2CCN(C(=O)C=C(Cl)Cl)CC(C)C2)CCC(C)(C)C1 c1(C(N(C2CCN(C(c3c(NC)cccc3)=O)C2)C)=O)cc(C2CC2)ccc1F C#Cc1ccc(F)cc1C(N1CCOCC1CNC(=O)CCC(C)SC)=O CC1=NOC2(C1)CC(C(N1CC(O)(C(C)NC(C3CC(C)CO3)=O)C1)=O)C2 N1(C(c2cc(C(C)=O)on2)=O)CCC2(CCN(C(C3(N(C)C)CC3)=O)C2)C1 CC(N)CCC(=O)NNC(=O)CC1(C(F)F)CC2(CCC2)C1 Cn1nccc(C(=O)NC2CCCN(C(C3(C)CC(C#N)C3)=O)CC2)c1=O C1(NC(C(C(C)C)OCC)=O)CC1C1CCCN(c2nnc(C)s2)C1 CC(C)(C)CC(O)C(=O)N1CCN(C(=O)CS(=O)(=O)N2CCOCC2)C(CO)C1 c1(CC(C)NC(C2(n3cc(-c4ccccc4Cl)nn3)CC2)=O)cccc(F)c1 C1(C(C)C)CN(c2ccc(C(F)(F)F)cn2)CCN1C(C1(C)CCCCC1)=O CCC(O)C(C)(C)C(=O)NC1CC(N(C(C=CCOC)=O)C)C1.C1CCC(=O)N1 c1(CC)ccc(C)c(NC(=O)NC2CN(C(=O)C(CC(C)C)N(C)C)C2)c1 N1(C(c2c(N)ccc(F)c2)=O)CCC2CN(C(c3cn[nH]c3)=O)CC2C1 N(C(=S)N1CC(C)C(O)C(C)C1)c1c(C)csc1 Cc1cc(C)nc(SCC(N2C3(C(=O)NCC4CCCC4)CC(C)(C2)C3)=O)n1 c1(C(=O)NC(CC)CNC(CCC)=O)cccc2ncccc12 C12(C(=O)NCC(C(=O)NC)(C)C)CCN(C(=O)C(C3CCCCC3)C)CCC1C2 C(C(O)CC(C)(C)C)NC(c1cc(CNC(CN(C(C)=O)C)=O)nn1C)=O C(=O)(CC1=CCCCC1)N1CC(NC(c2c(NC(CC)=O)cccc2)=O)C(C)C1 C(=O)(C1=NOC2COCC12)NCCCCN(C(=O)C1=CS(=O)CCC1)C C1(NC(c2cncc(C)c2)=O)CCC2(CCN(C(=O)C(C(C)C)C(C)C)C2)C1 N1(C(c2ccc(N(C)C)cc2F)=O)CCN(C(=O)CCCC2CC2)CC(C)(C)C1 N1(C(=O)OC(C)(C)C)CC(CNC(C2CCOCC23CCC3)=O)OCC1(C)C C1(NC(C2=C(C)OCC2)=O)CC2CCC1N(C(=O)C(C1CCOCC1)F)C2 C=CC(C)(CCOC)C(=O)N(CC(C)NC(c1cc(F)ccc1SC1CC1)=O)C Cc1nc(C2CC2)nc(S)c1C(=O)NC(C)CC(C)NCCN(C)C C1(C2CCN(C(c3n[nH]c(C)n3)=O)C2)(NC(C(Cn2ccc(C)n2)C)=O)CC1 C1(CNC(CC=C)=O)CCN(C(=O)Cc2ccn3ccnc3c2)CC1(F)F N1(C(CC=CCC)=O)CCC(O)(CN(C(=O)C(O)C(C)CC)C)CC1 N1(C(C2(CC#C)CCCC2)=O)CCCC(N(C(=O)CCCC2CCCC2)C)CC1 C1(C(=O)NCC2OCCN(CC)C2)CC(C)CN(C(C2(C#N)CC2)=O)C1 c1(C(N2CCC(C(N3CC(N(CC=C)C)C3)=O)(CC)C2)=O)ccc2nccn2c1 c1(NCC=CCC(=O)NC(CC#C)C)cn(C)nc1CC C(=O)(C(F)C(C)CNC(c1cn(CC)nn1)=O)NC(C#C)CC1CCCC1 C1(C(=O)NCC(C)(C2CC2)NC(C2CC2c2ccco2)=O)CCc2nncn2C1 C(=O)(C#CC1CC(F)(F)C1)NC(C1CCN(C(c2ccnn2CC#N)=O)C1)C CC(C)CCC(F)C(=O)N1CCC(CNC(=O)CCCC(C)C)C(C)C1 C(=O)(C(C)C(CC)CC)NCC1ON=C(C(=O)N(C2CCCC2)CCC)C1 c1(N2CCC(N(C(=O)Cc3ccc(=N)[nH]c3)C)C2)ccc(Br)cc1 CC1CCOC(C(=O)NC2(CF)CCN(C(c3nn[nH]c3C(F)(F)F)=O)C2)C1 C1(C(=O)NC(CNC(C(C)N2CCCC2)=O)(C)C)CCC12CCOCC2 CC(c1ccccc1)=CC(=O)N(C(C)CN(C)C(c1cn(C)c(=O)n1C)=O)C C1(C(=O)NC2(CO)CCN(C(c3n(CC)ccc3)=O)C2)Cc2cc(C)ccc2S1 c1(NC2CC(C(C)NC(C(CC)n3cncn3)=O)C2)ncnc2scnc12 c1(C(N2CC3(C2)CN(C(=O)Nc2c(F)cccc2F)C3)=O)ccc(B(O)O)cc1 N12CCC(NC(=O)CSC(F)F)C(C1)C2=O.c1(C(N)=O)cnc(N2CCC2)nc1 C1(NC(CNS(NC)(=O)=O)=O)CCN(C(=O)COCCC2CCCC2)C(C)C1 c1(C(CC)N(C2CC2)CC)cccc(-c2ncccc2OC)c1.CCN C=C(C)C(C)(C)C(=O)NCCCCCNC(C1CC(=O)N(C(C)C)C1)=O C1(CNC(C(C2CCC2)NC(c2cccc(OCC)c2)=O)=O)CC12CCCCC2 c1(C(=O)NCC23C(NC(CCCCC=C)=O)CC(CC2)C3)nc(Cl)c(=O)[nH]c1N c1(C(C)=O)ccc2ncc(C(=O)NCCN(C)C(c3ccc(CF)cc3)=O)n2c1 CC1(C)CCN(C(c2sccc2C#N)=O)CC1CNC(C12COCC1C2)=O C(=O)(CN=c1[nH]c(N2CCCC3(CCSCC3)C2)nc2cccnc12)NCC N1(C(=O)CCOCC2CC2)CCC(O)(C(C)(C)NC(C(=CC2CCCC2)C)=O)C1 c1(C(=O)NC(C)C(C)(F)F)ccc2c(c1)OCCO2 c1(N2C(CNC(c3c(CC)n(C)nc3)=O)CCC2)nc(Cl)nc(CC)c1C C1(C)(C(=O)NCC(CN(C)C(C23CC(CC(F)F)(C2)C3)=O)O)CC2CCC1O2 c1(C(N2CCCC(NC(c3c(C)oc(Cl)n3)=O)CC2)=O)ccnc2[nH]cnc12 C(CN=c1[nH]c(Cl)ncc1C)OC1CN(C(CCc2scc(C)n2)=O)C1 C1(CC)C(CC(=O)NC2CC(CCNC(=O)C(C)NC(N)=O)C2)C1(F)F C1(NC(=O)COCC2CCC2)CCC(C(=O)Nc2cnncc2Cl)CC1 Cc1[nH]c(C(=O)NCC2CC2NC(C2(c3ccn(C)n3)CC2)=O)c(C)c1[N+](=O)[O-] C(=O)(C1Cc2ccc(Cl)cc21)NCC1(F)CC(NC(C2CCC(CC)CC2)=O)C1 N1(C(COC(CNC(C(C(=O)OC)(F)F)=O)(C)C)=O)CC(C2=NOC(C)C2)C1 C(CCC(C)(C)NC(=O)CCCN(C)C(C1(OC(C)=O)CCC1)=O)OC C1(NC(C(C)N2CCC2)=O)CC2(CCN(C(c3ccc4nsnc4c3)=O)CC2)C1 N1(C(C(CC=C)CC)=O)C(C)CN(C(=O)C=Cc2ccccc2C#N)CC1C c1(C(N2CCCCC(NC(CC(=O)NC3CC3)=O)C2)=O)c(F)ccc(Cl)c1F c1(-c2cc(C)nn2C)csc(=Nc2cccc(Cl)n2)n1-c1c(C)cccc1F C12(C(N3CCC(NC(CCNc4cccc(C)c4)=O)C3)=O)CC(CO)(CCO1)C2 C(=O)(C(CCCOC(C)(C)C)N(C)C)N1CC(C#CC)C1.c12ccccc1CO2 c1(C(=O)NCC2N(C(c3ccc(C)cc3C)=O)CC=C2)cccc2c1COC2 N1(C(CSCCC)=O)CCC(F)(CNC(=O)Cc2nc(C3CC3)n[nH]2)CC1 C1(CNC(C=CCN(CC)CC)=O)C=CC(NC(C2CCCCO2)=O)C1 CC1=NN(C)C(=O)C1CC(=O)NCCC1COCCN1C(C1CC(C)(O)C1)=O S(=O)(=O)(c1cnc(NCCCCC)c(Cl)c1)NCCN1CCC(CC)C1 Cc1ncnc(C(C)(C)NC(CC(=O)OCc2ccccc2)C)c1Br c1(C(N2CC(NC(C3C(C(C)C)OCC3)=O)C2)=O)cc2ccc(Cl)cc2o1 c1(OC)ccc(Cl)c(C(=O)NC2C3CC2N(C(=O)C(C)(C)C(C)O)C3)n1 CC1CC(C(=O)NCC2CC(NC(c3scc(F)c3Cl)=O)C2)=NO1 n1(NC(=O)NC(C)C(=O)N(CC(F)(F)F)C)cc(C2CCOCC2)nn1 Cc1c[nH]c(C(=O)NC(C(=O)NC2(c3nc[nH]n3)CC2)C2(C)CC2)c1 CC(C)(C)C(O)C(=O)N(CCNC(c1ccsc1C#N)=O)Cc1ccc(Cl)nc1 C1(C(=O)Nc2cc(C(=O)N(C3CCN(CCF)C3)C)n[nH]2)(NC(C)=O)CCCC1 CCC(O)C(C)C(=O)NC1CCC(CNC(C2OCCN(C)C2=O)=O)CC1 c1(C(=O)NCC2CCC(NC(c3n(CC)ccn3)=O)C2)ccc(=O)oc1 c1(C(=O)NC2CC23CCN(C(C2C=CCS2)=O)C3)cccc2nncn12 c1(C(N2CC(CNC(C(C)C)=O)C(F)(F)CC2)=O)ccc2nnn(C(C)(C)C)c2c1 n1(CC)cc(Cl)c(C(=O)NCC(C(C)(C)C)NC(c2[nH]nnc2C2CC2)=O)n1 C1(CC)CCC(C(=O)NCCC2CCCN2C(=O)CSCC(F)(F)F)C1 C(=O)(C(C)(C)C(F)(F)F)N1CC(C(N(CC(O)COC)CC)=O)OC(C)C1 CCC(C)(CC)C(=O)NCC(C)(C)CN(C)C(c1cn(C)c(O)n1)=O Cc1c(CNC(C2(F)CCN(C(C3CCC(N(C)C)C3)=O)C2)=O)nnn1C N1(C(C2(c3c(C)c[nH]n3)CC2)=O)CCN(C(=O)CSc2cn[nH]c2)CC1 CC1(C)CN(C(=O)CCCN=[N+]=[N-])CCN(C(=O)CNC(c2cccs2)=O)C1 C1(CNC(C(C(C)C)N(C)C)=O)CC2(CCN(C(c3scnc3Cl)=O)C2)CO1 C(CCC(C)CC(=O)N1CC2CCC(CNC(=O)COC3CC3)C2C1)=C(C)C C1(SCC)CCC(C(=O)NCC=CCNC(C2CC2c2ccccc2)=O)CC1 Cc1cc(C(=O)NC2CC2C(=O)Nc2cc(F)cc(Cl)c2)ccc1C#N C1(C(N2CC(CC(C)C)C2)=O)C(C2CC2)CCN1C(c1ccc(C(F)F)o1)=O c1(C(=O)NCCCN(C2CCCC2)C(=O)C(=C2CCCCC2)F)c[nH]ccc1=O CON(CCC(=O)NC1CCCC(O)CC1)C(=O)CC1CCOC1 N1(C(Cc2cn(CC)nn2)=O)CCC(C)(CNC(c2nc(C)ccc2F)=O)CC1 C(C(CC(C)C)C(=O)NCC1(O)CCN(C(c2oc(CO)cc2C)=O)C1)OC N1(C(COCC(C)(C)C)=O)CCC(C)(CNC(C2(C#N)CC3CC3C2)=O)CC1 C1(C(N(CC(C)(C)CNC(c2ccc(O)c(Cl)n2)=O)C)=O)CC2CCCCCCC12 c1(N2CCC(CCN(C)C)C2)nc2c(c(=NC3CC4(COCCO4)C3)[nH]1)COC2 C1(C(=O)NCc2cccc(NC(C3(C)CC3)=O)c2)Cc2ccccc2O1 C1(CN(C)C(C2CCOC2)=O)CCCCN1C(c1c(Br)nnn1C)=O C1(C(=O)NC(C2(C(=O)NCCC(=C)C)CC2)C)NC(=O)OC1C N1(C(c2cnc(C)s2)=O)CC2(C1)CN(C(C13CC=CCN1CCC3)=O)CC2CO C1(CCC)CCCC1C(=O)NCCN(c1nc(CCOC)ns1)CC1CCCC1 C(=O)(CC(C(F)(F)F)C(=O)NC(C1CSC1)C)N1CC(CF)C1 Cc1cccc2c(CCC(=O)N3CC(CNC(=O)C(C)C(F)(F)F)C3)c[nH]c12 c12nc(c(C)o1)C(=O)NC2.N1(C(c2c(CC)ccs2)=O)CCSCC1CO N1(C(C2(CC)CCCCC2)=O)CCN(C(C2CCCCC(=O)N2)=O)C(C(C)C)C1 C1(NC(C2CCCC(C)CC2)=O)CC2CC(C1)CN(C(c1cc(N)ccn1)=O)C2 c1(C(=O)NCC2C(C)CN(C(=O)C(=O)NCC(F)(F)F)C2)c2c(nn1C)CCC2 Cc1cccnc1C(F)(F)C(=O)NCC1CCC1NC(C1CC1C#N)=O C1(C(=O)Nc2n(CCN(C)C(=O)OC(C)(C)C)ccc2)CCCC1C N1(Cc2c(C)sc(Br)n2)CCC(NC(=O)C(=O)Nc2ccccc2Cl)C(O)C1 C1(C(c2nc3ccccc3[nH]2)=O)CCC(N=c2ccc3cc(Br)cc(Cl)c3[nH]2)CC1 C1(O)(C(=O)NC(CCN(C(c2c(C)cccc2)=O)C)C(C)C)CCCC(C)CC1 C1(CN(C(=O)COc2ccc(C)cc2)C)CC(F)CN1C(C1CC=CCC1)=O C(CCCCC(=O)NC1CC2CC1N(C(=O)CCc1nncn1C)C2)OCC C(=O)(C(F)CCC(C)C)N1CCC(C(CO)NC(C(CC2CC2)OC)=O)CC1 C1(C(N2C(CCC)COCC2)=O)CN(C)CCN1C(c1cccn1C)=O c1(CNC(C2CC3OCCC23)=O)ccc(Cl)cc1Sc1ccccc1 CN1CCCCC(C(N2CCC(O)(CNC(C3C4CN(C)CC34)=O)CC2)=O)C1 N1(C(C=CC=CCC)=O)CC2CC1C2NC(=O)CC(C)(C)c1ccccc1 CC(C)(CS(N)(=O)=O)C(=O)NC1CC(CNC(C2OCCC2(C)C)=O)C1 C1(CNC(C2COC2)=O)CCCN(C(c2ccc(-c3cccc(Cl)c3)s2)=O)C1 c1(OCC(N2CCC(NC(C(C)(C)O)=O)C(CO)C2)=O)cccc2ccccc12 C(=O)(C1CCCn2cnnc21)N1CCC(C)(CNC(COC(CC)CC)=O)C1 C#CCCC(O)C(=O)N1CCN(C(=O)C2=CCCC2)CC1c1cccc(OC)c1 N1(C(C2C(C(N)=O)C2)=O)CC2(CCC(NC(=O)Cc3ccc(F)cc3F)CC2)C1 C1(C)(CNC(C(CC)(F)F)=O)CCC(NC(=O)CCO)C1.c1(=O)ccc1=O.C1CC1 C1(CNC(C(C)(C)N2CCC2)=O)CC2(CCN(C(=O)C#CC3CCOC3)CC2)C1 Cc1c(C(=O)NCC2(NC(=O)CN(C)C(N)=O)CCCCC2)cnn1CCO c1(C(=O)Nc2c(CC)cccc2)cc(F)cnc1NC(c1c(I)ccnc1F)=O Cn1cc(C(=O)NCCCCCNC(=O)Cc2ccccc2C(F)(F)F)c(Cl)n1 C1(C(N(C(C(=O)OC)C2CC2)C)=O)CCN(C(C2CCC(C)C2)=O)C1 N1(C(C(CC)OC)=O)CC(CNC(c2csc(-c3cnccn3)n2)=O)CCC1C N1(C(CCC=C(C)C)=O)CCN(C(c2ccc(O)nc2C)=O)C(CC(F)F)C1 c1(CNC(C2(C)CCCO2)c2nnnn2CC(O)(CO)CO)ccccc1Br C1(C(=O)Nc2cnc(C)nc2)CCC(C)(C)N(C(c2[nH]ccc2C)=O)C1 C1(C)(C(=O)NC2CC(C(C)O)C2)CCN(C(c2c[nH]ccc2=O)=O)C1 C1(C)CN(CC(=O)N(C)C)CC(C)O1.Cc1sc(O)nc1C(=O)NC1CC(OC)C1 C(=O)(C(CNC(C1(C)CC=CC1)=O)C(C)C)NC(CC)C C(=O)(C(C)(C)CC(=O)NC(CC1CC1)C(=O)N1CCCC1C(C)(C)C)OCC C12(C(=O)NCCN(C(c3c(SC)nn(C)c3)=O)CC3CC3)CCC(CC1)OC2 Cc1nc2ccccc2nc1C(=O)NC1CCC1NC(=O)C(c1cncnc1)C c1(OCC)ccc(CC(C)C(=O)N(CC(O)CNC(c2cnns2)=O)C)cc1 c1(C(C)C)cc(N(CC(C)NC(C2CCC(C)(C)O2)=O)C)nc(C(C)C)n1 C12(NC(COC(CC)C)=O)CCOCC1CN(C(=O)Cn1cc(C)cn1)C2 C1(OC)CN(C(C2CC(O)(CNC(=O)OC(C)(C)C)C2)=O)CC1c1nccn1C CN=c1nc(N2CCC(SC)C2)[nH]c(=NCCNC(=O)OC(C)(C)C)[nH]1.C(Cl)CC C1(CNC(C2CCC(C)O2)=O)CCN(C(=O)C=C(C2CC2)C2CC2)C12CC2 Cc1ncc(N)cc1C(N1CCC(C(N2CC(OC(=O)N(C)C)C2)=O)CC1)=O N1(C(c2[nH]cc(C(C)=O)c2)=O)CC2(C1)CN(C(=O)Cc1csnn1)CC(C)(C)O2 CCC(CC)CCC(=O)N1CCC(O)(CCNC(C2CN(C3CCOC3)C2)=O)C1 c1(C(=O)NC(C)(CO)C(=O)O)noc2c1CC(F)(F)CC2 C1(CC)CCC(O)(C(=O)N(C)CCN(C(=O)Cc2ccon2)C)C1 CCN=c1[nH]c(C)c(C(N2CCN(C)CC2CNC(=O)C(CCO)N(C)C)=O)s1 N1(C(c2cc(C(C)=O)on2)=O)C2CCCC1CN(C(C13CCCC1C3)=O)C2 c1(OCCN(CCCN(C)C)C)ccc(CNC(=O)NC2CCC(C)O2)cc1 C1(CO)(NCCCn2cncn2)CC2CCC1CC2 N1(C(CSCC(N)=O)=O)CCCC(O)(CCNC(C2(F)CC=CCC2)=O)C1 c1(N(C)C)cccc(C(N2CCN(C(=O)Cn3cnc(C(N)=O)n3)CC2)=O)n1 C(=O)(C(C)(F)C(=O)N1CCC(c2ccccc2CNC(C)=O)CC1)OC C(=O)(C(CN=[N+]=[N-])NC(C1CC1(Cl)Cl)=O)N(C)Cc1ccnn1C N1(C(C(COC)O)=O)CCN(CC(C)NC(=O)C(C)(C)CSC)CC1 C1(C(=O)Nc2cccc(CNCc3cnc(OC)nc3)c2)CCCCC1(F)F CC1C2=C(C(=O)N1C)C(c1cncn1C)NC(=O)N2CCF C1(C(=O)NC(c2nc(C)oc2)C(N2CCC=C(Cl)C2)=O)CC2CCC1CC2 c1(C(N2CC(=C(CNC(C(CCSC)(C)C)=O)F)C2)=O)ncc(Cl)c(N)c1Cl N(C(=NCC(C)N1CCCCCC1)NCC(C)(O)Cc1ccccc1)C1C(C)C1 c1(C(=O)NC(CNC(CCOC)=O)CC(C)C)c(C)ccc(Cl)c1N C(=O)(CS(=O)(=O)C1CC1)N(C)CC1N(C(C2CCC(C(=O)OC)O2)=O)CCOC1 C1(CNC(C2(OCC)CC2C(C)C)=O)CC(F)(F)CN1C(=O)CCN(C)CCO CC(CN(C(=O)OC(C)(C)C)C)C(F)C(=O)NCCOCCS C#Cc1cn(C)nc1C(N1CCCC(NC(c2ccc(N)cc2Cl)=O)C1)=O C1(C(N(C2CN(C(CSCCC)=O)C2)C)=O)CCc2ccccc2O1 N1(C(c2ccn(CCC)n2)=O)CCC(C(N2CCOCC2CO)=O)(CC)C1 Cc1noc(C)c1C(C)C(=O)OC.C12(F)CN(C1)C(=O)C=CC=C(Br)C(=O)NC2 C1(C(=O)NCC2(O)CN(C(CC(COC)C)=O)C2)CN2CCCN1CC2 N1(C(CC=CC(C)(C)C)=O)CC2CCC(C(=O)NCC3COCC3(C)C)(C2)C1 c1(C(=O)NCCNC2CN(C(C=CC)=O)C2)n[nH]c2cc(Cl)ccc12 c1(-n2c(C)cc(C)n2)ccccc1S(=O)(=O)N1CCNC(C)C1C Cc1ncc2n1CCC(C(=O)NCC1CCN(C(=O)CCOC3CC3)C1(C)C)C2 C(CC(=O)NCC1(CCNC(=O)C(C)(C)c2cccnc2)CC1)(C(F)(F)F)OC n1(CC)ccnc1C(N1CCC1(C)CC(=O)NC(c1ccn(C)n1)C)=O NS(=O)(=O)c1sccc1C(=O)NCC(c1ccccc1)NC(=O)Cn1cnnn1 c1(C(N2CCC3CN(C(=O)COc4cccnc4)C3C2)=O)ccc2sncc2c1 C1(CC(=O)NC(C=C)CO)CC(C)N(C(=O)CN2C(=O)CCC2=O)C1 C1(C(N2CCC(F)(CNC(=O)C=CC3CCCO3)CC2)=O)CCC2CCCCN12 N1(C(c2cc(CN(C)C)ncc2)=O)CCCC2CN(C(=O)CCC[N+](=O)[O-])CC12 CN1CCCC(C(=O)NCCC2(O)CCN(C(=O)CC3CCC(F)(F)C3)C2)C1 Cc1nscc1CO.C(=O)(CC(C)N1CCCC1=O)N1CC(CC2C(=O)N2C)C1 c1(C(=O)NCCC2N(C(CS(=O)(=O)NC)=O)CCC2)cccc2c1CCOC2 c1(N2CC3C(C(=O)OC)C3C2)cc(C)[nH]c(=NCCC2CC(C)(C)NC2=O)n1 O=C(C(O)C1=CCCCC1)NCC1OCCC1C(=O)NCCCC(F)F c1(C(=O)NCC2N(C(CCC3(C#N)CC3)=O)CCC2)cccc(-n2cncn2)c1 c1(CC(=O)N(C)CCNC(c2snnc2C2CC2)=O)csc(-c2ccccc2)n1 C1(CC(=O)NC2CCCN(C(c3cccc(=O)o3)=O)C2)CC(C2CC2)C1 N1(C(C(C)NC(C)=O)=O)CCCN(C(c2csc(Cl)n2)=O)C(C)C1 C#Cc1ccc(C(=O)NCC(CC(C)C)NC(=O)C=Cc2cn[nH]c2)nc1 CC(C)C(CNC(C1C2CC(=O)CC12)=O)C(=O)NCC(C)(C)C1CC1 O(NC(=O)C(C)(C)CCNC(C1CCC(OC)CC1)=O)CCCC C1(NC(c2c(C)nc[nH]2)=O)(CNC(=O)C(F)(F)Sc2cnn(C)c2)CCCCC1 C=C(C)CC(C)C(=O)N1CC(C)(NC(c2cnc(CC(C)(C)C)s2)=O)C1 c1(CNC(CC2CC3(CN(C(CC4ON=C(C)C4)=O)C3)C2)=O)ccc(C)n(C)c1=O C1(NC(CNC(CCC(C)C)=O)=O)CCN(C(C2(CF)CCC2)=O)CCC1CO S(=O)(=O)(c1cccnc1Cl)N1CC2(N(C(CNS(C)(=O)=O)=O)CC2)C1 c1(CN(C(=O)CC2CC2CNC(=O)COC2(C)CCC2)C)n[nH]c2c1CCC2 c1(N(C(CN(c2cnc(=N)[nH]c2)C)=O)CC2CC2)ccccc1Cl N1(C(CC(CC)C2CCC2)=O)CCOC(C(=O)NCCCCCN=[N+]=[N-])CC1 C1(C2CCCN(C(C(C#N)C3CC3)=O)C2)N(C(c2cccc(Cl)c2)=O)CC12CCC2 n1(CCC(=O)NCCC2CCN(C(c3n(CC=C)ccc3)=O)C2)c(C)ccc1C C(=O)(C(=O)C(C)(C)C)NC1(CC=C)CCN(C(C2CCCC(O)C2)=O)C1 c1(C(=O)NC2CC(N(C(CC(n3c(CC)ncc3)C)=O)C)C2)csc2nccn12 N1(C(C2N(C(CC)=O)CCC2)=O)CCC(NC(=O)C=Cc2nccs2)C(CO)C1 c1(C(N(CC(=O)NCC(O)COC2CCCC2)CCC)=O)sccc1CC c1(NC(C2CC3CC2C2CC32)=O)cc2ncccc2[nH]1 C(C(C)(C)CCNC(c1ccnc(C)c1)=O)NC(CCN(CCCCC)C)=O N1(C(C(C(=O)OCC)F)=O)CCC(NC(C2(C)CCCC2)=O)CC(C)(C)C1 C1(NC(=O)CCc2nnc(O)nc2O)CCCC12CCN(C(=O)CC1CCC1)C2 c1(C(N(CCSC)NC(C#C)CNC(C2CC2CC)=O)=O)cccnc1 C1(C(=O)NC2CC(C)(CNC(=O)CN3CCSCC3)C2)(CC)CC1(F)F c1(OC)ccc2nc(C)c(C(=O)NCC3CCCCN(C(C4CSC4)=O)C3)n2n1 Cc1nn(C)cc1C(=O)NC1CCC(C(=O)NN2CCC(N(C)C)CC2)C1 Cc1nnc(CCOC(C2CCOCC2)=O)s1.C12CCN(C1)C(=O)C(C)N(C)C2 CC1CCCCC1CC(N1CCC(CNC(C2CC(C#N)C2)=O)CC1)=O C1(CNC(C(c2ccn(C)c2)C)=O)CC2(C1)CN(C(c1csc(O)n1)=O)C2 C1(NC(CCCOCCC)=O)CC12CC(C(N1CCC(SC)CC1)=O)C2 C#Cc1cccc(C(=O)NC2(CC(N3CCC(C)(COC)C3)=O)CCC2)c1 N1(C(c2n(CC)ncn2)=O)CCN(C(c2cc(OC)cs2)=O)CC12CCC2 CS(=O)(=O)CC(=O)NC1CC1C(=O)N(c1ccc(C(F)(F)F)nc1)CCO Cc1cnc(Nc2cccc(F)c2F)c(S(=O)(=O)N(CCCOC2(C)CC2)C)c1 c1(C(N2CC3CN(C(c4cc(SC)ncc4)=O)C3C2)=O)cnc2ccc(C)cn12 C1(CNC(C=CSC)=O)CCC2CN(C(=O)C=Cc3cncn3C)CC12 N1(CC(=O)NCC2C(C(N(C3CC(OC)C3)CC)=O)CCC2)CCCCC1=O C1(CNC(C2CC2(Cl)Cl)=O)CN(C(c2nocc2C2CC2)=O)CCO1 c1(NC(C2CCN(C(c3ccc(O)cn3)=O)CC2)=O)cccc(F)c1F Cc1cccc(-c2ccc(NCc3cccc(C(F)(F)F)c3)nc2)c1F c1(C(N2CCC(CC)C2CNC(C2OC3CCC2C3)=O)=O)ccc(NC)cc1C C1(NC(c2nccc(C#C)c2)=O)CC12CCN(C(C1CCOC(=O)CC1)=O)CC2 C1(C(=O)NCC23CC(CO2)N(C(=O)CC2CCCC2)C3)CCOC2(CCCC2)C1 C1(C(=O)NC(C2(O)CN(C(C3CNC(=O)N3)=O)C2)C)COCC1(C)C CN=c1cc(C(=O)NOCC(N2C3CCC2COC3)=O)cc[nH]1 c1(C(=O)NC2(CNC(C(C)Oc3c(C)cccc3)=O)CC2)cc2n(c1)CCCC2 c1(OC)c(F)cc(C(C(=O)NC(c2cccc(C)c2OC)C)OC)cc1Br Cc1ccc2c(-c3nc(CC(C)C)nn3Cc3ccccn3)coc2c1 c1(-n2cc(OCCOCCC=C)nn2)cc(OC)c(F)c(F)c1 C1(NCC(=O)Nc2ccc(C)cc2)CN(C(=O)CCCCN(C)C)CC(C)(C)C1 c1(N2CCN(C(=O)Nc3ncc(SC)nc3)CC2)cccc2c[nH]nc12 C=CCCCC(C(=O)NCc1cnc2c(c1)CCC2)NC(=O)C(CC)SCC Cc1coc(-c2ccccc2)c1C(=O)NCCCNC(=O)CCc1cc(Cl)no1 Cc1cc(CCC(=O)NC2CCC2NC(c2cccc(O)n2)=O)ccc1Cl c1(C(N2CCC(N(C(C3C(C(=O)OC)CCC3)=O)C)C2)=O)cnn(C)c1C1CC1 C(=O)(CCC(C)(F)F)NC(C1CCN(C(C(C)OCC)=O)CC1)C c1(CCNC(=O)CCOC2CN(C(C34CCCC3C4)=O)C2)cccc(O)n1 C(=O)(CCS(=O)(=O)c1ccccc1)N(C(C)CN(C(=O)C=CC1CCCO1)C)C C1N=C2N=CC(=CN2)C(=O)N2CCCC(C)C12.CC(=O)CC1CC1.C(C)(C)(C)O Cc1ccc(CCC(=O)NCC23CC(NC(=O)COc4cnn(C)c4)(C2)C3)o1 C1(C(N2CCC(F)(C(=O)NCC3(C#N)CC3)C2)=O)C2CC3C(C2=O)C13 C1(NC(C(C)OC2CC2)=O)CN(C(=O)C(O)CC2CCCCC2)C2CCCC12 CC(C)CC(=O)NC1CCC(Cn2cc(Cn3cncn3)nn2)C1 c1(C(N2CCC(O)(C(C)NC(C3CCCCC3)=O)C2)=O)cc2n(c1)CCOC2 Cc1cc(C(N2CC(C(=O)NCC3(C)CC(F)(F)C3)CC2(C)C)=O)ccc1C#N c1(C2C(C(=O)NCC3(F)CC(NC(C=C(C)C(C)(C)C)=O)C3)C2)ccc(F)cc1 C1(C(=O)NC2(CNC(c3nn(CC)nc3C)=O)CC2)CCOC(=O)CC1 O=C(C1=NOC2(CCC2)C1)NC1CC2CCC1CN2C(=O)C#CC1CCOC1 C(C(CC(F)(F)F)NC(=O)CC1CC2(CCC2)C1)NC(=O)CCn1ccnn1 C1(NC(C(C2CC2)SC)=O)CN(C(=O)CC2CN(C)C2)CC12CC2 C1(C(N2CCN(S(=O)(=O)c3ccc(Br)cn3)CC2)=O)C2CC3CC(C2)CC1C3 N1(C2C(=O)NCCCC2)CCOC2(CCN(C(C3CC(F)(CO)C3)=O)CC2)C1 c1(C(=O)OC)ccc(CC(=O)NC2CCC(NC(C3CCOCC3)=O)CC2)cc1 C(=O)(CN=c1cc[nH]cc1)NC(CN(C)C)C(=O)N(C)Cc1nnc(O)o1 c1(C(=O)NCC(CNC(CCc2ccc(SC)cc2)=O)O)cc2cccnn2n1 C(=O)(C1=CCC2CCC1N2C(=O)CCc1nccs1)N1CC(C)OC(C)C1 c1(OC)ccc2[nH]c(=NC(C)CCn3cncn3)nc(N3CCOC(C)CC3)c2c1 N1(C(C(CC)Sc2ccccc2)=O)CC(CNC(=O)C(C)NC(C)=O)C(C)(C)C1 C12(NC(CCOCCOC)=O)CCOC(CNC(=O)CC(C)CF)(C1)C2 C1(C(=O)NC2C(NC(C3=C(C)CC3)=O)CC2)CCCC(C)(C)C1 c1(C(=O)NCC(C(C)C)NC(C(C)OCC#C)=O)cc(Cl)c(Cl)c(Cl)c1 C(N=c1cc(C2CC2)nco1)C1CCN(C(C=CCCC)=O)C1 C1(NC(CCC#C)=O)C2CN(C(c3cc(Br)n(C)c3)=O)CC12 N1(C(c2occ(C)c2F)=O)CCN(C)C(CNC(=O)C(F)Cc2ccccc2)C1 CC1CCN(C(=O)C(=O)NC2CCC2CNC(C2(C)CCCS2)=O)CC1 Cc1cnc(CNC(=O)NCCSCc2ccc(Cl)s2)cc1Br c1(C(=O)NC(CNC(C2(NC(N)=O)CC2)=O)CO)cscc1C(N)=O Cc1cnn(C)c1CC(=O)NCC(C(C)(C)C)NC(c1cc(Br)c[nH]1)=O C1(NC(c2cnc(-c3cccs3)o2)=O)CN(C(c2cnc[nH]2)=O)CC1C1CC1 c1(CCC(=O)NCC(=C)CCNC(=O)C=Cc2nccs2)cc2ccccc2o1 C1(NC(CCC(C)OC)=O)CCN(C(c2sc(C)nc2C)=O)CCC1(F)F N1(C(=O)OC(C)(C)C)CC2(C1)SCCC2Nc1nccc2occc12 CN1N=C(C(=O)NCC(O)CCNC(c2cc(C#N)n(C)n2)=O)CCC1=O Cc1ccc(C=CC(N2CCCC2CN(C)C(c2nc(C)ncc2Cl)=O)=O)cc1 C(CC(N)C(=O)NC(C)CN1CCOCC1)SC C(C)(CCC(=O)N1CC=CC(NC(=O)C(C)(C)O)C1)OC(C)=O C1(NC(C2(CN(C)C)CC2)=O)CC(CC(=O)NCCCC2CCCC2)C1 C1(CCNC(CCCC=C)=O)CCCN(C(C2CSCC(=O)N2)=O)CC1 N1(C(C(C#N)=CC2CC2)=O)CC2C(CNC(=O)CC3CCC(C4CC4)O3)C2C1 c1(C(CNC(=O)CC2CC(F)C2)NC(c2c(CC)c[nH]c2)=O)ccc(F)cc1F C1(C(=O)NCCCOCC(C)C)CCCC(NC(=O)CN=[N+]=[N-])CC1 N1(C(Cn2ncc(C)c2)=O)CCCC(C)(C)C1CNC(=O)CC1CCC(=O)C1 c1(C(=O)NCC2C(CN(C)C)C2)cc(CNC(=O)C(O)C2CCCC2)ccn1 n1(CCN(C)C)cc(C(=O)NC2CC(C)(NC(=O)CCc3ccccc3)C2)cn1 c1(CC(=O)NC(CC)CNC(C2CN(C)C(=O)N2)=O)ccc([N+](=O)[O-])cc1F C1(c2cc(CC)no2)CCN(C(c2cc(C(C)=O)c[nH]2)=O)CC1 O=S(=O)(C(F)(F)F)N1CCOC(C2CCC2)C1.c12cccc(n1)CCCNC2 C1(C(=O)NC(C(=O)NC)CC)CC2CC2N1C(C1CC(OC)(OC)C1)=O C1(C)(C(=O)NC2CC3C(NC(c4c(C)nc(N(C)C)s4)=O)C3C2)C(C)(C)C1(C)C c1(C(N2CCN(C(=O)CO)CC2)C(=O)NC2CC2)ccc(Cl)cc1Cl Cc1cnc2cccc(C(=O)NC3(C)CC(NC(=O)CCNC(=O)CO)C3)n12 C(=O)(C1CCOc2ccc(F)cc21)NC1CCN(C(CSCC(C)C)=O)C1(C)C N1(CC(=O)Nc2ccc(CO)cc2)CCCC(CNC(c2nnc(CO)s2)=O)C1 C(=O)(CCC(=O)NCCC1CCC(C(=O)NCCCn2nccn2)C1)NC C(=O)(C1=CC2CC(C1)CC2O)N(C1CCN(C(c2cc3cccnc3[nH]2)=O)C1)C C1CC(=O)N(C)CC2CN(C(=O)C(C)O1)C2.C(C(=O)NCC)(C1CCC1)OCC.NC C1(CC)COCCN(C(=O)N(C2CCS(=O)(=O)C2)C)C1 C1(CCCCCNC(C2(CC)COC2)=O)CCN(C(C2(C)CCCC2C)=O)CC1 N1(C(C=CC(C)C)=O)CCN(C(=O)CN2CCC(C)C2)C(CC(F)(F)F)C1 C1(CC(=O)NCC2(OC)CN(C(C3CC3C)=O)C2)CSc2ccccc2NC1=O S(=O)(=O)(c1ccc(O)cc1)N1C(CC(N2C(C#N)C3CC3C2)=O)CCC1 C1(NC(c2n(C(CCC(C)(C)C)SC)nnn2)CC(C)C)CC2(COCCO2)C1 Cc1cc(O)ccc1CC(=O)NCC1CN(C(C2COCCC2(F)F)=O)C1 CCCC(C(=O)NC(C)COc1cccc(Br)c1)c1ccccc1 C(=O)(CCCCN=c1ccnc(N2CCC(c3cnn[nH]3)C2)[nH]1)NC C(N=c1[nH]c2c(c(=NCCN(S(=O)(=O)c3ccccc3Cl)CC)[nH]1)COC2)C1C(C)C1 c1(C(N2CC(CC(N3CCCC(C(=O)O)C3)=O)C2)=O)c[nH]ccc1=O c1(OC)nccc2c(C(=O)Nc3cc(Br)c(C(=O)OC)cc3C)csc12 CCC(C)C(C(=O)N(CC(C)CNC(=O)CCCC1CCCO1)C)OC C1(C(=O)NC(CC(=O)NC)C)C(C)OCCN1C(=O)CC1CCCC2CC12 c1(CC(=O)NC2CC3(CN(C(C4(C(=O)OC)CC4)=O)C3)C2)ccc2occc2c1 c1(OC)c(C)nc[nH]c1=NCC1(CNC(C2CCCC(O)C2)=O)CC1 c1(NC2C(C)COC2)nc(=NCc2cnn(Cc3ccccc3)n2)[nH]c2c1CSC2 C1(NC(C(C=CC)O)=O)CCN(C(C2CCC(C)(O)CC2)=O)C(C)C1 CN1CC(NC(=O)CC2(NC(=O)C=CC3CCC3)CCC2)C(C)(C)C1 CC(C)CCCNC(CNC(C)=O)=O.C(=O)(CC(C)C)NCC(C1CCOC1)S C(=O)(C(F)(F)C(O)C1CC1)NCC1CC(NC(Cc2cc(C)n(C)n2)=O)C1 c1(CN(C(c2ccnc(OC)n2)C(=O)NCC=C)C)ccccc1COC N1(C(c2ccc(OC)cn2)=O)CCCC(F)(C(=O)NC(C)CS(C)(=O)=O)C1 Cc1cc(F)cc(C)c1C(N1CCC(O)(C(C)NC(=O)CCCCO)CC1)=O N1(C(c2c(CC)ccs2)=O)CCOCC1CC(N1CCC(CCF)CC1)=O C1(C(N2CC(CNC(=O)C=CC3CCC3)OCCC2)=O)CC2(CCOCC2)CO1 c1(C(=O)Nc2cc(OC)nc(Br)c2)cccc(S(=O)(=O)C(F)(F)F)c1 C(CC(N)=O)(C(=O)N1CCCC(F)CC1)NC(c1c[nH]c(=NC)o1)=O c1(C(N2CCN(C(C(C)C(F)(F)F)=O)CC2C2CC2)=O)cc2c(ncn2C)[nH]1 Cc1ccc(C(=O)NCCOC(C)(C)CN(C(C2CCC(F)C2)=O)C2CC2)cn1 C(N(C)N1CC2(CC(F)C2)C1)c1c(C)cccc1C C(c1ccc(F)c(Cl)c1)=CC(=O)NC1CC2CN(C(c3n(CC)ncn3)=O)C1C2 c1(CC)[nH][nH]c2ncnc(=NC(CCc3ccccc3)C(C)C(C)C)c1-2 Cc1[nH]c(=N)nc(O)c1CC(N1CC(NC(=O)CN2CCSCC2)C(C)(C)C1)=O C1(NC(=O)CCC2CCC2)CN(C(=O)C=Cc2ccc(Cl)c(Cl)c2)CC12CCC2 C=C1CCN(C(=O)C(COC)OC)C(C(=O)NCC2CC(=C3CC3)C2)C1 C1(C(N(C(C(C)C)C)C)=O)CN(C(c2cc(Cl)cn2C)=O)CCN1C C1(C(=O)NC(C2CCOC2)C#C)CC2CCC1CNC2 c1(COc2c(-c3nc(-c4ccc(C)o4)on3)nccc2)cc(F)ncc1C Cc1cc(NC(c2csc(CNC(=O)C(C)(F)F)c2)=O)cc(CO)c1 C12(CCN(C(=O)C(O)CN3CCCC3)CC1)C(=O)N2.C1(CC(=O)OC)(COC)CC1 C1(Cc2c(-c3nnc(C(C)(C(C)C)OC)o3)non2)CC2(CCOCC2)CO1 c1(OC)ccc(C(N2CC(CNC(=O)CC3CC(F)C3)C2)=O)nc1Cl C1(C)(C(=O)NC2CC(NC(c3c(CC)cco3)=O)C2)Oc2ccccc2NC1=O c1(NC2CC(F)(CNC(=O)CC3CCC4CC34)C2)cc(=O)n2ccccc2n1 C(=O)(C(F)(CNC(c1cnc(C)c(C)c1)=O)C(C)C)N1CCC(OCCC)CC1 c1(C(=O)NCC(C2CC2)NC(CCCOCCOC)=O)cccc(CSC)c1 C1(CCNC(C(C)NC(COCC#C)=O)=O)CCCC2CC12 n1(CC(=O)N(C2CC(=C)C2)C)cc(CNC(=O)C=CC)nn1 Cc1c(CN2CCCC2(C)C(=O)Nc2cc(O)nc(Cl)n2)cccc1O C1(CC(C)NC(C2CC(=C3CC3)C2)=O)CCN(C(C2(N(C)C)CC2)=O)CC1 C(=O)(C(CCC(N)=O)N(C)C)N1CCN(C(c2c(C)oc(Cl)n2)=O)CC1CC1CC1 c1(C(=O)NCCN(C(c2cnc(C(C)=O)s2)=O)C)ccc2ccccc2n1 N1(C(C(c2ccc(OC)cc2)C)=O)CCN(C(c2cnn[nH]2)=O)C(C2CCC2)C1 c1(CCC(=O)NCC2CC2CNC(=O)Cc2cn[nH]c2)cccc(F)c1Br CC1CC(C)N(C(c2cn(CCO)nn2)=O)CCN1C(=O)CCC1CCOCC1 c1(SCC(N2CC(C(=O)OC)N(C)CC2)=O)cn2cc(C)cc(C)c2n1 C1(C)(C(=O)NC(C)Cc2nncn2C)CCCN1C(C1(n2cccn2)CC1)=O C1(C(=O)NCC(CC)NC(C2(Nc3ccccc3Cl)CC2)=O)COC(C)(C)CO1 Cc1ccc(C(N2CCC(C(=O)NC3CC(O)C3O)C23CC3)=O)cc1F Cc1nn2c(c1CNC(=O)Cc1cccs1)CN(C(=O)Cn1cccc1)CC2 CCC(CC)CC(F)C(=O)NC12CCC(NC(=O)C(C(C)C)SC)(CC1)C2 N1(C(c2c(C)onc2CO)=O)C2CCC1CC(NC(=O)C(F)CC1CCOC1)C2 N1(C(CONC(CN2CC(C)(OC)C2)=O)=O)CCC2C(COC)C2C1 Cc1ccc(CC(=O)NC2CCCC2NC(c2[nH]ncc2C#N)=O)cc1Br C1(CC(=O)NC2CCN(C(=O)C=C3CCSCC3)CC2CO)CN2CCC1CC2 Cc1c(C(N2CC3CC(NC(=O)C4=CCOCC4)C2C3)=O)ccc2cncn12 c1(C(=O)OCC)ccc(CC(N2CC(F)CC(NC(C)=O)C2)=O)cc1F C(N=C(NC1CCC1)N1CCCC(CC)C1)C1CCC(OCC)CC1 C1(C(N(CCC(=O)N(CC)CC)CC=C)=O)CC12CCOC2 C12(CNC(C3(SC)CCC3)=O)CCCC1N(C(C1(C)CCN(C)C1=O)=O)CCC2 Cc1ccc(C)n1CCC(=O)NCC1CC1NC(c1ccc(NCCO)cc1)=O Cc1cc(C(N2CCCC2C2(C(N3CC(OC(F)F)C3)=O)CC2)=O)ccc1O N1(C(=O)NC2CCCC(C)CC2)CCC2(CC1)C(=O)NCc1ccccc12 C=CCC(C)(C(=O)N1CC(F)(CNC(=O)CC2CCOC2)C1)N(C)C N1(C(C2(CC#C)CC2)=O)CCN(C(c2onc(Br)c2C)=O)C(C)C1 c1(CS(C)(=O)=O)ccccc1NC(=O)NC1CC1.c1(N)cccc(-c2cccc(Cl)c2)c1 C(=O)(C(C)C(CC)CC)N1CCCC(CN(C(c2cnc(CC)nc2C)=O)C)C1 C1(C(=O)NCC2CC(C)N(C(c3nscc3N)=O)C2)CNC(=O)C(C)(C)C1 C(=O)(CCCC(=O)N1CCCC1c1nc(C(=O)NC(C2CCOC2)C)cs1)OC Cc1ccc(CCC(N2CC(NC(c3ccc(C)n3C)=O)C3CC23)=O)cc1C c1(NC(=O)CC2(NC(c3ccc(CO)cn3)=O)CCC2)cccc([N+](=O)[O-])c1Br N1(C(c2n(CC)ccc2)=O)CCN(C(=O)C(c2c(C)noc2C)C)CC12CC2 N1(C(C2(CC)CC2)=O)CCC2C(C1)NC(=O)CCN2C(=O)CC1CNC(=O)C1 C1(C(C)=O)CC(O)CN1C(=O)C(F)=C(C)C1CC1.C c1(N(C)C)cc(C(N)=O)ccc1C(=O)NC1C2CN(C(CCOC)=O)C1C2 C(=O)(C(CC(F)F)c1ccccc1)NC(C1CCCC1)CNC(C(C)C1CC1)=O C(CS(=O)(=O)CC(=O)N(C)CC1(NC(c2ccc(C)c(C(C)=O)c2)=O)CC1)OC c1(C(=O)NC2C(NC(C3N(CCC)CCC3)=O)CC2)[nH]c2ccccc2c1C c1(CC)c(C(=O)NCC(O)CNC(c2nccn2CC)=O)oc2ccccc12 C12(C(=O)NC3C(SC)CN(C(c4cncc(C)n4)=O)C3)CCC(CC1)C2(C)C c1(C(=O)NCC(C)NC(CCC=C(C)C)=O)ccc(Cl)c2c1OCCO2 Cc1oc(C(C)C)cc1C(=O)NCC1CC(NC(=O)C=CC(=O)OC(C)(C)C)C1 C(=O)(CC(C)CNC(=O)Cn1cccnc1=O)NC(c1cccnc1O)C c1(NC2C(C=C)COC2)nc2cccc(Br)c2o1 Cc1cc(NC(C2CC2C(N)=O)=O)ccc1NC(C1(C)CCCO1)=O c1(C(N(C2CCN(C(=O)C#CC3CCCC3)C2)C)=O)ccc2nc(Cl)nn2c1 C1(CCC)(CO)CCN(C(c2cnc(OCc3ccc(C(F)(F)F)cc3)s2)=O)CC1 N1(C(=O)CC(F)(F)F)CCCN(C(c2cccc3cc[nH]c23)=O)C(CO)C1 c1(N2CCN(CC)CC2)nc2ccsc2c(=NCCC2CCC(C)CC2)[nH]1 c1(NC(C2(CCNC(CC3C(C)OCC3)=O)CCC2)=O)cncc(C2CC2)c1 C#CC1(C(N2CCCC(NC(N)=O)C2)=O)CCN(C(=O)Cc2nc(=N)[nH][nH]2)CC1 c1(C(C(F)F)OC(c2c(Cl)cc(C)c(F)c2)=O)cccc2ccccc12 C1(C(=O)NC(C)CCNC(C2(C#N)CCCC2)=O)CC(c2ccc(F)cc2)=NO1 CCC(CN(C)C)CC(=O)NCC1(C)CCN(C(=O)Cn2cnc(C(N)=O)n2)C1 N1(C(C23CC(OC)C2C3)=O)CC2CC(C1)N(C(=O)C(N)=O)C2 C(CCC(C)(C)C(=O)N1CCC=CC1COC)NC(C(CC)C(C)C)=O c1(CNC(C(c2ccc(C)s2)N(C2CC2)CC)=O)ccc(Cl)s1 n1(CC)nccc1C(C(=O)NCc1ccco1)N(CCC#N)CC1CC1 c1(C(N2CCC(NC(C=COCC)=O)CC2C2CC2)=O)cc(F)cc2cc[nH]c12 N1(C(C(C)SCC)=O)CC(C)(C)C1C1CCN(C(c2[nH]c(C)nc2C)=O)CC1 CCC(CCCO)NC(=O)CC1CCN(C(c2nonc2N)=O)C1 c1(C(N2CC(O)(CN(C(C3(Cl)C(C(C)=O)C3)=O)C)C2)=O)ccc(C)c(Cl)c1N C1(NC(c2cc(CC)ncc2)=O)CCN(C(=O)Cc2ccccc2OC)CC1O C1(CNC(C(CC)n2ccnc2)=O)CN(C(=O)C(C)n2cccn2)C2(CCC2)C1 c1(C(=O)NC(CC)(C)CNC(=O)CCc2cnco2)nc(C(C)C)oc1C C1(C(=O)NC(C(=O)OC)Cc2cc(O)ncc2Br)CCC(=O)CC1(C)C C(=O)(C1=CCCSC1)NCC(CCC)NC(C1CCCCC1C(=O)OC(C)(C)C)=O c1(C(=O)OC)cnc2c(c1)S(=O)(=O)NC=N2.C12(OC)CC(CO)CN1C(C1CC1)N2 N1(C(c2onc(C)c2C)=O)C2CCC1C(F)C(NC(=O)Cc1ccc(F)cc1)C2 N1(C(CC(CNC(C2N(CCC)CCC2)=O)C)=O)CC(F)(C2CC2)C1 C1(N(C(C(C)(C)OC)=O)C)CCC(NC(c2nccn2C)=O)CC1 C=C(CNC(C1CC(C(F)(F)F)(OC)C1)=O)CCNC(=O)Cc1nocc1C N1(C(C2C(=C)C2)=O)CCCC12CCCN(C(=O)CC1CC1)C2 O=C(CS(=O)(=O)CCO)N1CCC(O)(CNC(C2Cc3cccnc3C2)=O)CC1 Cc1cc(=NC(=O)C(=O)NC2CCN(C(C3COC(=O)N3)=O)C23CC3)[nH]o1 c1(OC)coc(C(=O)NCCC2CN(C(C3CC3(F)F)=O)C2)cc1=O C(=O)(CC(C)C(=O)NC(C)C(C)C(=O)N(C1CCOC1)C1CC1)OC O=C(N=c1cc(Br)[nH][nH]1)C1CN(C(C2C3COCC23)=O)CCN1 C1(NC(c2c(C(C)C)ocn2)=O)CN(C(=O)CC(C)F)CC1n1cccn1 CC(F)(CNC(=O)CN1CCSCC1)CNC(C1CCCOC1)=O c1(C(=O)NCC2CCN(C(C(C)C3CC3)=O)C2)cnc2ncn(C)c2n1 C=CC(C)C(C)C(=O)N1CCC(N2CCC(C(=O)OCC)C2=O)CC1 c1(C2CCN(C(=O)NCc3ccc(CCCCC)o3)CC2)cncc2nnnn12 CCC(C(=O)Nc1cccnc1)NC(=O)Cc1sccc1C c1(CCNC(CNS(NC)(=O)=O)=O)cnc(C)cc1C C1(N(C(=O)CC=C(Cl)Cl)C)CCCN(C(C2(O)CC2(C)C)=O)CC1 C(CCCCCn1nc(-c2cccc(N)n2)nc1-c1ccc(OCF)cc1)OC C1(C(=O)OCC2COCCO2)CCc2ccccc2O1 N1(C(=O)NCc2ccc(C(F)F)o2)CCC(NC(=O)C=Cc2cn[nH]c2)CC1 C1(CCC)CCN(C(=O)C(c2cnn(C)c2)NC(c2c[nH]cc2CC)=O)C1 c1(C(=O)NC2CC(C)(C)N(C(=O)Cn3ccnn3)C2)cccc2sccc12 c1(NC(C(C2CCCC2(C)C)N(C)C)=O)ccc(OCF)cc1 c1(OCCCC)ccc(CC(N2CC(CNC(=O)C3=CCSC3)(OC)C2)=O)cc1 Cc1ccc2c(C(N3CC(C(=O)NC4(C)CCOC45CC5(F)F)C3)=O)coc2c1 CC(C)CC(C(N)=O)N(C)C(c1n[nH]cc1CNC(C1CC1c1ccco1)=O)=O C1(C(c2cccs2)N(C)C(=O)OC(C)(C)C)CC2C=CC1N(C(C1CCC1)=O)C2 CC1(C(N2CCCC(C(=O)Nc3cccnc3C3CC3)C2)=O)CC12CCNCC2 C(CNC(=O)CNC(c1cccnc1)=O)(C(C)(C)C)NC(C(F)=CC)=O N1(CCOCCC=C)CCCC(NC(=O)CCCCCO)CC1 C1(NC(C=CCOC)=O)CCN(C(=O)C(N2CCOCC2)C)C1C CCC(C)(C)C(=O)C(=O)N1CCC2(CC2NC(c2ccc(CO)s2)=O)C1 c1(N(c2ccccn2)C)ccc(NC(=O)CN2CCOC3CC23)cc1 CN1CC2(CCN(C(C3(F)CCN(C(C4CC4C(C)(F)F)=O)CC3)=O)CC2)C1 c1(C(=O)NC(C)CC(C)NC(=O)C(N2CCSCC2)C)ccccc1[N+](=O)[O-] C1(C)(NC(C2N(CC)CC2)=O)CCN(C(=O)C2=CCOC2)C1 N1(C(C2CN(C)C(=O)N2)=O)C2CCC(C2)C1CC(=O)NCCc1csnn1 c1(C(=O)NCC(CNC(CN(C(=O)OC)C)=O)O)cc(O)nc(Cl)c1 N1(C(C2(CC#C)CCCO2)=O)CCOC2CN(C(=O)CN3C(=O)CCC3=O)CC12 CCS(=O)(=O)CC(=O)N1CCC(O)(CCNC(c2c[nH]cc(Cl)c2=O)=O)C1 c1(C(N2C(CNC(c3ccnc(C)n3)=O)CCC2)=O)cccc2cc[nH]c12 c1(CC(=O)NC2CC(F)(CNC(C(C3CCCCC3)OC)=O)C2)ccc(C)nc1 c1(C(=O)NC(C2CCN(C(C(CC#C)C)=O)CC2)C)cc(F)c(F)c(F)c1 CC(O)C(C)CNC(=O)CCOCCN(C(=O)C=CC1CCCC1)C c1(C(N(C(C)C)CCNC(c2ccc(N)c(N)n2)=O)=O)ccc(F)c(Cl)c1F C1(CCCC)(C(=O)NC(CN(C(=O)C(C)C2CCOC2)CC)CC)CCC1 CC(C(=O)N1CCC(C(N)=O)C1)(C1CCC1)NC(c1cc[nH]n1)=O Cc1ccc2c(C(=O)NC3CC3NC(c3ccc(C(C)(C)C)s3)=O)csc2c1 Cc1ccc(N(C)C(C2CN(C(=O)COCCC(C)C)CC2(C)C)=O)cc1C c1(C(=O)NC(C)C(C)NC(=O)CCc2nc[nH]n2)cc(-c2ccco2)no1 C1(CC#C)CCCC1NC(c1ccc(CNC(C2CSC2)=O)o1)=O C1(C(N(CC(C)NC(CCCC(C)C)=O)C)=O)CC2CC1CC2(F)F C1(C(=O)NC)(CC)CCCC1.C1(C(=O)N(C)CCN(C)C)CCC1(OC)OC S(=O)(=O)(c1ccc(Br)c(F)c1)N1CC2CCN(C(CN(C)C)=O)CC2C1 CCC(C(=O)NC(C1CC(NC(c2coc(C)c2)=O)C1)C)C(C)(C)CC c1(C(=O)NCC2(C)C(C)CN(c3snc(C(C)=O)n3)C2)cnc2ccnn2c1 C(=O)(CC(O)C(Cl)(Cl)Cl)NC1CC(C)(NC(C2N(C)CC(C)(C)C2)=O)C1 C(=O)(CCS(=O)(=O)NC)NCC12C(CN(C(C=CC=CC)=O)C1)C2 c1(NC(c2c(NC(C)=O)cncc2)=O)ccn2nccc2n1.C12CC1CNC2=O N1(C(C2CCC(C)C2)=O)CC(CNC(=O)C(C)(C)CC2CC2)CC(C)(C)C1 C(=O)(C(C(C)C)n1cc(C)cn1)N1CC(CC(C)NC(C=C(CC)CC)=O)C1 CC1(C(=O)NCCC2CCCN2C(C2(C)C=CCC2)=O)CCNC(=O)C1 N1(C(c2ccc(C)o2)=O)CC(NC(C2(CC3CC3)CCOCC2)=O)CC12CCC2 N1(C(COC(CC)C)=O)CC(O)(C2CCCN2C(C2CC2F)=O)C1.C(C)(C)(C)O N1(C(c2ccnc(C(C)C)n2)=O)CCN(C(=O)C(O)C2CCCC2)CC1CO C(C)(C)(CC(=O)NCC1CCCCO1)N(C(CC(C)n1cccc1)=O)C N1(C(c2c(OC)ccnc2)=O)CCC2CCC(NC(=O)CCN3CCCCC3)C12 N1(C(c2c(SCC=C)cccc2)=O)CC2CCC(C1)C(NC(=O)CCC)C2 C(C)(CC(=O)OCc1cc(F)ccc1N1CCOCC1)(C(C)(C)C)N(C)C N1(C(c2onc(C)c2C)=O)CCC(NC(c2ccc(NC(N)=O)cc2)=O)C(O)C1 CC(C)(C)CCC(=O)N1CCC(O)(CNC(c2ccc(-n3ccnc3)nc2)=O)C1 C(N=c1[nH]c2c(C)cccc2o1)C12OCC(NC(CSCCC)=O)(C1)C2 Cc1cccc(S(=O)(=O)N(C2(C(N)=O)CCNCC2)CC2CC3(CCNCC3)C2)c1 c1(C(=O)NC2C(C)N(C(c3ccc(Cl)c(F)c3)=O)CC2)cc2n(n1)CC(O)CO2 c1(C(=O)NC(C2(O)CN(C(C3ON=C(CC)C3)=O)C2)C)c(F)cc(Cl)cc1F C1(C(=O)NCCSCC(=O)NCc2c(CC)nn[nH]2)CCOC(C)C1 C1(C(=O)NC(CC(=O)OCC)C)CCCCN(C(c2cncs2)=O)C1 N1(C(C(=O)C2CC2)=O)CCN(c2ccc(I)cn2)CC1 C1(C(=O)NCCC2(O)CN(CCn3cnnc3)C2)(CC)CCCC1 c1(-n2cc(CNC(C3(C#N)C(C)(C)C3)=O)nn2)ccc(C(F)(F)F)cc1F Cc1nnnn1CC(=O)NCCN1CCCC1CNC(C1CC1C1CCCC1)=O c1(-c2cn(CC3N(C(CNC(N)=O)=O)CC=C3)nn2)ccc(F)cc1F N1(C(C(c2cccnc2)C)=O)CCC2(C1)CN(C(C1CC(S(C)(=O)=O)C1)=O)C2 N1(C(CCCC(=O)NCC)=O)CCC2(NC(=O)C=CS(C)(=O)=O)CCCC12 c1(C(=O)OC)cc(Br)c(F)cc1NC(C1C2CC1N(C(=O)CC(=O)OC)C2)=O Cc1cc(=O)c(C(N2CCC(C(=O)N(C)CCn3ccnc3C)C(C)C2)=O)c[nH]1 C1(C(N(C(C)CCNC(C2CCC=CCC2)=O)C)=O)CN2CCN1CC2 CCCC(CC)C(=O)NC(CO)C(C)NC(=O)CCCc1csc(=N)[nH]1 C1(CNC(C(C)S(C)(=O)=O)=O)CC2(CCC2)CN1C(c1ccoc1Br)=O C1(NC(CCCOC)=O)CN(C(C2CCC(=O)C(C)C2)=O)CC2(CCC2)C1 CC(O)(CC(F)(F)F)C(=O)NC1CC2(C1)CN(C(=O)CC1CCC1)C2 O=C(CS(=O)CCC(F)(F)F)NCC1C2CN(C(c3nc(Cl)cs3)=O)CC12 C(=O)(C(=O)C(C)(C)C)NC(C1CCN(C(CCOc2c(CC)cccc2)=O)C1)C c1(NC(C2C(c3cc(-c4c(OC)cccc4)[nH]n3)C2)=O)c(C)nc(O)nc1O C1(CCSC)C(=O)N1.C(CC(=O)N(C)CCC1CN(C(=O)C(C)C)C1)NC(=O)OC CCCC(C)CCCC(=O)N(C1CCN(C(C2CCOCC2)=O)C1)CCO C1(C(=O)NCCCN(C(=O)C(C)CF)CC)COc2c(F)cc(F)cc2C1 N1(C(C(N2CCOCC2)C)=O)CCC2(CC1)CN(C(C13CC1COC3(C)C)=O)C2 c1(CC(=O)NCC2CC(NC(c3c(CC)[nH]cc3)=O)C2)cccc(C)c1C C1(C2CCCCC2)(C(=O)NC(CNC(=O)CC(C(F)F)n2cccn2)CO)CC1 N1(CC2N(C(=O)OC(C)(C)C)C(C)(C)CC2)CCC2(CC1)OCCO2 c1(C(N(CCNC(=O)CCCNC(=O)C(C)(C)C)CC)=O)oc(C(F)F)cc1C N1(C(C(C)(C)CC2CC2)=O)CC(C2CCCN(C(=O)C(C)(O)C(C)(C)C)C2)C1 N1(C(c2cn(CC(C)C)nc2)=O)CCC(NC(c2[nH]nnc2C2CC2)=O)C(O)C1 N1(C(CCCCN(C)C(C23CCCC2C3)=O)=O)CCCC(C2(C)CC2)C1 N(C(=NCCOc1ccco1)NC(C)COC)CC1(C)CC(=C)C1 C(=O)(C(O)C(CCC)NC(c1sccc1Cl)=O)N1CCC(CCC)C1 N1(C(CC(CNC(C2COC(C)C2)=O)OC)=O)CC2CCC2(C)C1 N1(C(C2CCC(C(=O)OC(C)(C)C)O2)=O)CC(O)Cc2cc(Br)ccc21 N(C(=NCCC(=O)N1CCC(Cc2ccccc2)C1)NC(C)C)CC(CCC)C N1(C(C)C)C(=O)NC(CCN(C)C(c2ccccc2)C)C2(CCCCC2)C1=O C1(NC(CC2CCCC(C)(C)O2)=O)C2CC3CN(C(C4CCCCS4)=O)C1C3C2 Cc1cc(F)c(Br)cc1C(=O)NCCCn1cc(-c2cc(F)ccc2Cl)nn1 c1(N(C(=O)CC)CC)cc2cc(OC(c3ccccc3[N+](=O)[O-])=O)ccc2[nH]1 N1(C(C(C(=O)O)OCC)=O)CCC(Nc2cc(OC(C)(C)C)cc(F)c2)C(C)C1 N1(C(C(C)N(C)C)=O)CCC2(NC(c3ccc(C(F)(F)F)cc3)=O)CCCCC12 C1(CN(CCCCC=C)C)CCCN(C(=O)CCCn2cccc2)C1 C1(C(=O)NCC(=O)OCC)CCCN(C(C2CCS(=O)C2)=O)CC1 C1(F)(CNC(c2nccc(C)c2)=O)CCCN(C(C2(c3nccs3)CC2)=O)C1 CC1C(C(=O)N(CCCOCCO)C)CCCN1C(c1c[nH]nc1Cl)=O c1(CCNC(=O)NC(c2cc3ccccc3o2)C)c[nH]c2c(Br)cccc12 N1(c2cc(C)ncn2)CCCC(C)(C(=O)NC2C3CCCCCC23)C1 Cc1cn(C)nc1C(=O)NCC(C)(C)OCC(=O)NC1C2CCCC12 c1(OC)ccc(F)c(CNC2CC2NC(c2nc(-c3ccco3)n[nH]2)=O)c1 C1(C(=O)NC(CN(C(Cc2cnc(C)o2)=O)C)(C)C)C2CCN(CC2)S1(=O)=O Cn1cc(C(N)=O)cc1C(=O)NCC1(O)CN(C(=O)CCc2cccn2C)C1 C1(C(=O)OC)C(O)C(O)CN1C(c1cnc(Br)n1C)C(=O)NCc1cccs1 c1(OC)ccc(C(O)CN(C)CC2CC2(C)C)c(OC)c1 CCCCCCCC(C)(c1nnnn1CCSC)NCCS(=O)(=O)CC1CC1 C1(CNCC(CC2CCC(C(=O)OC)CC2)O)CC2(CCC2)CO1 c1(-c2ccc(CC(=O)Nc3c(SCC)cccc3)cc2)nnc2cnccn12 C1(C)(C(N(CC(C)(C)CNC(=O)C=CS(C)=O)CC)=O)Cc2ccccc2C1 C(C)(CCC(=O)NCCN(C1CCCC1)C(c1cc(-c2ccco2)no1)=O)OC c1(CC)ccc(F)c(C(=O)N(CC(CC)NC(=O)C(CC)N(C)C)C)c1 C(CCCC(=O)NC1(C(=O)N(CC(C2CCCC2)O)C)CCSC1)OC c1(N2CCC(CCN(C)C)C2)nc(=N)[nH]c(=NCC2CCC3(CC2)CC3)[nH]1 C1(CC#C)(C(=O)NC2CC(NC(c3cc(C(N)=O)co3)=O)C2)CCCOC1 c1(NC(c2ccc(O)nn2)=O)ccc(C(F)F)c(N2CCNC2=O)c1 N1(CC(=O)N(C)CC2(O)CN(C(c3c(C)coc3)=O)C2)CCN(C)CC1 CN1CCC12CN(C(C1CC(NC(=O)C(C)(C)F)CCO1)=O)C2 C1(C(=O)NCCCC(C)(C)NC(C(CN(CC)CC)F)=O)CCn2nncc2C1 CC1c2ccccc2OC1CC(=O)N(CCCCNC(=O)CN(C1CCC1)C)C c1(CN(C(=O)C(N2CCC(F)(CO)C2)=O)C(C)C)cc(C#N)n(C)c1 Cc1cc(F)cc(C(N2C(CNC(C3CC(=O)N(C)C3)=O)CC3CC23)=O)c1N C=CC(C)(O)CC(=O)N1CCCCC1CNC(C1CC1C)=O Cc1ncc(CNC(C2(NC(=O)C(C)C3CCCC3)CCSC2)=O)n1C C1(CNC(CCC#CC)=O)CC(NC(C2SCC=C2C)=O)C12CCC2 c1(OC)ccccc1C(C(C)C)NC(c1cnc(OCF)cn1)=O C#CC1(C(N2CC(CO)C(CNC(=O)CCC)C2)=O)CC(=O)C1 c1(C(=O)NC2C(NC(C=C(CC)C)=O)CCC2)c(-c2ccccc2Cl)noc1C c1(C(N2CCCC(NC(C(C)n3cnnn3)=O)C2)=O)cn2ccc(CO)cc2n1 N1(C(c2cc(C)no2)=O)CCC(OC2CN(C(C3C=CCS3)=O)C2)CC1 c1(C(N2CCC(NC(C(CCCC)CC)=O)C23CC3)=O)cc(C)nc2ccnn12 N1(C(C(c2cn(C)nc2)(F)F)=O)CC2CCC(C1)N2C(=O)CC1(O)CC1 C1(C(=O)NC2CCN(C(CCC(C)OC)=O)C(C)C2)CCn2ncnc2C1 C(=O)(C(CC(C)C)N(C)C(C1CCCN(C)C1)=O)NCc1ncc(C)n1C CCCCC(C)N=c1[nH]c(=NCCc2ccc(N)cc2)[nH]c2c1CCCCC2 CCC(C)(C)CC(=O)NC1CCN(C(c2c(C)coc2C)=O)CC1F C(=O)(C1=COCCO1)N(C1CCC(NC(c2snnc2C2CCC2)=O)C1)C C1(NC(C)=O)CCC(C(=O)N(CC(O)CNC(=O)CC2CCCCC2C)C)CC1 CC#CCCCC(=O)NC1CCC(C)N(C(=O)Cn2cnc(Br)c2)C1 CC1=NOC(C(N2CCC(CC(=O)NC3CC3(C)C(F)F)C2)=O)C1 CCC(C)(C(=O)N1CC=CC(NC(=O)C(C)CO)C1)OC N1(C(c2cc(NC(C)=O)c(C)cc2)=O)CC2CCC(C1)N(C(=O)CC(C)C)C2 CC(C)CC(CC(=O)NCC1CC(O)CCO1)NC(C1(C2(O)CCC2)CC1)=O c1(SCC)ccccc1C(=O)NC1COCC1NC(=O)CC1CCCC1 N1(C(c2cc(C#N)on2)=O)CC(NC(C2CC2Br)=O)CC(F)C1 Cc1cc(NC(c2csc(C(=O)NCCO)n2)=O)c(C)s1.C12CC(C1)CNC2=O c1(C(=O)NCC(C2CCOC2)(C)C)ccc2nnnn2c1 N1(C(C2CC(C)C2)=O)CCC2(CCCCN(C(C34CCC(C)(CC3)OC4)=O)C2)C1 C1(CNC(CC(CCC)O)=O)CCC(C)(C)CN1C(=O)CC1(O)CCOCC1 c1(C(N2CCC(NC(C(CC)C#N)=O)C2)=O)c(C)n(C)c2ccccc12 C#CCCCCN=C(NCc1ccsc1)NC1CCOCC1 C(N=c1[nH]cnc2c1COC2)C1CCN(C(=O)CCCC(F)(F)F)CC1CO c1(C(=O)NCC(CC=C)NC(c2csnn2)=O)cc2cc(F)cc(F)c2[nH]1 N1(C(c2cc(C)oc2)=O)CCC(C(=O)NCc2oc(CO)nc2C)CC1 CCC(C)(CCNC(=O)C(O)C(C)C)NC(C1CCCS1(=O)=O)=O C1(OCC(O)Cn2cc(Cc3ccccn3)nn2)(CNC=O)CCSC1 c1(OC)cccc(C(=O)NC2CC(CNC(C3(C)CNC(=O)C3)=O)C(O)C2)c1F N1(C(=O)C=Cc2ccccn2)CCC2CCCC12C(N1CCC2(CCC2)CC1)=O C1(CNC(c2ccon2)=O)CC2(CC2)CN1C(=O)CC(O)Cc1ccccc1 c1(NC(c2n(C)nnn2)C2CC2c2ccco2)ccc2nscc2c1 c1(C(=O)NCC2CN(C(C(C=CC)O)=O)C2)ncc(C2CC2)cc1C C=Cn1nccc1C(=O)NC1CCC(CCC(=O)N(C2CCCCC2C)C)C1 C1(F)(C(=O)NC(CC)C)CCN(C(=O)CS(=O)(=O)NC)C1 N1(C)C(=O)CCN(CCC2OCCOC2(C)C)C1=O.C(c1ccccc1)=CCNC C12(NC(CCc3nnc(C)o3)=O)CCCC1N(C(c1cc(C(F)F)no1)=O)CC2 c1(C(=O)NC2C(NC(Cn3nnc(C(C)(C)C)n3)=O)C2)cccc(Cl)c1O c1(C(=O)NC(C(=O)NC(c2cscn2)C)(C)C)cccc(OCC(N)=O)c1 c1(C(N2CCC(CCNC(c3c[nH]c(=NC)o3)=O)C2)=O)cccc2nncn12 c1(-c2onc(-c3cccc(C)c3)n2)cc2scc(Cl)c2[nH]1 N1(C(CCc2cc(C)on2)=O)CCC2CC1CN(C(=O)C(C)OCCN(C)C)C2 C(=O)(C(C)CCC(C)(C)C)N1CCC(C2N(C(CC(=C)C)=O)CCC2)CC1 CCCCCCCCOCC(=O)NCC1CCCC1NC(c1cnc(S)n1C)=O C1(C2CCCO2)(C(=O)NCCCOCCNC(Cc2cn(C)nn2)=O)CCCO1 N1(C(C(F)=CC)=O)CCC(O)(CNC(c2nc(C)n(-c3nc[nH]n3)n2)=O)C1 C1(C)(CC)C=C(C(=O)NCCCN(C(=O)C(C)(O)C2CCC2)C2CC2)C1 C1(C(=O)NCc2cccnc2O)(NC(CC#N)=O)CCc2cc(Br)ccc2C1 Cc1noc(C)c1S(=O)(=O)N(CCCNC1(Cc2ccccc2)CCOCC1)C c1(OC(C)C)c(C(=O)NCC2CCN2C(=O)CC(C)O)cccc1N c1(C(=O)NCC2CCC(NC(C(C3CCC3)OCC)=O)C2)ncc(C)nc1OC N1(C(C2(CC=C)COC2)=O)CC(C2CCCN(C(c3cc(C)ccc3F)=O)C2)C1 C12(CNC(C(N3CCOCC3)C)=O)COC(CNC(C3CCC=CO3)=O)(C1)C2 C1(C)(C(=O)NCC(c2ccccc2)N(C)C(c2nccs2)=O)C=CCC1 Cc1nc(N2CC(NC(=O)C(C)S)C(C#N)C2)ncc1F C1(CCN(C(c2scc(C)c2)=O)C)CCCCN1C(C1CN(C(C)C)CCO1)=O CC1CCC(C(N2CC(NC(=O)Cn3cc(Cl)cn3)C3CC23)=O)CC1 N1(C(C=CCCC)=O)CCCC(C2CN(C(=O)C=Cc3ccccc3C#N)C2)C1 c1(NC(C(N2CCN(C(=O)NC3CCCC3)CC2)C)=O)cn2ccsc2n1 N1(C(Cc2cn(CC)nc2)=O)CCN(C(=O)CCCN2CCCC2)C2CC12 c1(C(=O)NCCC(C)N(C(=O)CCC2CC2(C)C)C)ccc(=O)n(CCO)c1 C1(CNC(C(C)NC(C)=O)=O)CC2CN(C(=O)COC3CCCCCC3)CC12 CCCC(F)(F)C(=O)N1CCOCC(C(=O)NC(C)Cc2nn[nH]n2)C1 C1(C(=O)NCC(CNC(c2nc(C)oc2C)=O)F)CC(C)OC(C)C1 N1(C(C=C(C)C)=O)CCC(C(=O)NCc2ccn(C)n2)(OC)C1 C1(SCC(C2CCCOC2)OC)CC2OC(C)(C)OC2C1 C1(CC)C(=O)NCCN1C(C1CCN(C(=O)Cn2ccnc2)C12CC2)=O c1(C(=O)NC(CC=C)C(=O)N(C)CC2(C)CCCO2)cncc(C=C)c1 c1(C(N2CCCC(N3CCN(C(C(C)(C)C)=O)CC3)C2)=O)cc(Cl)c(Cl)cc1F CC1CC=C(C(=O)NC(C)(C)CCCNC(=O)C2=CCCC2(C)C)CC1 c1(C(=O)NC(CNC(c2cccc(C(C)=O)c2)=O)CC(C)C)ccc(F)c(Cl)c1 c1(C(N(C)CC2N(C(C=CCCC)=O)CCOC2)=O)c(Br)ccc2c1OCO2 c1(C(=O)NCC(C)(C)OCC(=O)NC(CCC)CO)cc(N)cc(F)c1 c1(C(=O)NC2C3(CN(C(CC4ON=C(C)C4)=O)C3)CC2)c[nH]c2c(C)cccc12 O=C1CC(C(=O)NC2CN(C(=O)Cc3cc(F)cc(Cl)c3)CCC2F)CCCN1 CC1CCc2ncc(C(=O)NCC(O)CNC(c3cnn4cccnc34)=O)n2C1 C(N=c1nc2c(Br)csc2c[nH]1)C1(C)CCCN(C(=O)CC2(O)CCOC2)C1 c1(C(=O)NCCCC(C)NC(C2CCC(C)(CC)O2)=O)cc(C)nc(N(C)C)n1 C(=O)(C(C)C(O)C(C)C)N1CCC(CNC(c2nccc(OC)c2N)=O)C1(C)C C1(NC(c2cncc(C)c2Cl)=O)CCN(C(=O)C(C)n2cccc2)CC1(C)C Cc1ccc(C2CC2C(=O)NC23CC(C2)N(C(=O)C(F)C(C)(C)O)C3)cc1C N1(C(C=Cc2nc(C)sc2)=O)CCC(CNC(c2ccn(CC#N)n2)=O)CC1C c1(C(=O)NCCC(=C)CNC(c2ccc(C)o2)=O)cn(C)c(C)n1 N1(C(C(CC)N(C)C)=O)CC(C2CCCCN(C(c3nc(Cl)sc3C)=O)C2)C1 C1(CNC(c2c(C(N)=O)nccn2)=O)CCCC12CCN(C(C1CC1F)=O)CC2 N1(C(c2c(C#N)cn[nH]2)=O)CCC2CN(C(=O)C=CCOCC(F)(F)F)C2C1 C12(C(=O)NCC3(CN(C(C(CC)(C)O)=O)C)CC3)CCOC(C)(C1)C2 CCC(CC)(CO)C(=O)NC1CCC(O)CN(C(c2cnn(C(C)C)c2N)=O)C1 C#CCCCC(C)C(=O)N1CC2CC(C(=O)NC(CCC)C(F)(F)F)C(C2)C1 c1(OC)cc(CC(=O)NC(Cc2nonc2C)C(=O)O)ccc1Br C12(C(N(C3CCCCCC3)CC)=O)CC1CCN2C(=O)CCC1CC1 c1(C(N(C)CC2CCN(C(C3C(C=C)OCC3)=O)C2)=O)ccc(OCC)c(F)c1 N1(C(c2cnc(NC)s2)=O)CCC(CNC(C2CC(n3cccn3)C2)=O)C(C)C1 c1(C(N(C)CC2CCCN(C(C3CCN(CC)C3)=O)C2)=O)cc2cnccc2[nH]1 N1(CCCCCNC(C(c2n(C)ncc2)O)=O)CCN(C(=O)CNC(N)=O)CC1 N1(C(Cc2cc(C)on2)=O)CCCN(C(c2ccnnc2)=O)CCC1 Cc1cc(CCC(=O)NC(C)CN(C(=O)C(O)Cc2[nH]cnc2C)C)on1 Cc1cc(C)c(C(=O)N(CCC(C)NC(c2ocnc2C(F)(F)F)=O)C)o1 N#Cc1cccc(CN2CCC(C(N3CCC(O)C(O)C3)=O)C2)c1Cl c1(C(N2C(CNC(CC3(COCC)CC3)=O)CC(O)C2)=O)cc(Cl)cc(F)c1F c1(C(N2CCCC(CF)C2)C(=O)NCCC2(C)CC2)cc2c(cc1OC)CCC2 C1(CNC(c2c(OC)cccc2)=O)CC2CN(C(=O)CCc3cn(C)cn3)CC12 CCC(CCCC(=O)Nc1cnn2cccnc12)NC(=O)C(C)N(C)C c1(C(=O)NC2CCC(NC(=O)Cn3nnc(=O)[nH]3)C2)ncncc1Br N1(c2snc(COC)n2)CCC(F)(F)C(CNC(C2(C)CC2Br)=O)C1 c1(C(N2CCC(OCCC3(C(C)NC(N)=O)CC3)C2)=O)ccc(N)cc1 O=C(CC1=CCCC1)NC(CNC(c1cncc(Cl)c1Cl)=O)CO c1(NC(C2CC(NCc3c(C)cc(O)cc3C)C2)=O)ncnc2ccccc12 CCC(C)C(=O)C(=O)NCC(C(C)(C)C)NC(C1CCN(CC)C1)=O C=CCC(Cc1ccccc1)C(=O)OCCC(=O)NC(=O)Nc1ccccc1 CCC(C)(C)CC(=O)NC(c1ccc(F)cc1)CNC(=O)CCCN(C)C(C)C C(CCCCCNC(C1(SC)CC1)=O)n1cc(C(CC)(C)C)nn1 CCC(C)(C)C(O)C(=O)N(CCN(C)C(c1ccc(C(C)(F)F)nc1)=O)C(C)C c1(C(=O)NC2CCN(C(C3(C(O)C(F)(F)F)CCC3)=O)C2)cc(Cl)c(Cl)s1 C1(CC#C)(C(=O)NCCOC2CN(C(c3nc(Cl)cs3)=O)C2)CC=CCC1 C(CN=[N+]=[N-])(C(=O)NCCC1CC(C)=NO1)NC(CCCNC(=O)OC)=O c1(NC(C2CN(C(c3scc(C)c3)=O)C2)=O)n[nH]c2ccc(Cl)cc12 Cc1nc[nH]c1C(c1nnnn1CCC1(C)CC1)NC(C)C(=O)OCC1CC1 Cc1cccc(C(F)(F)C(=O)Nc2cccc(CNC(c3cnc(O)s3)=O)c2)c1 C1(NC(c2[nH]cc(C)c2)=O)CN(C(=O)CSc2nncs2)CC(C)(C)C1 c1(C(C)C)cccc(C(c2nnnn2C2CCC2)NC2CC(NC(N)=O)C2)c1 N1(C(CC)C(=O)NCCN(C(=O)C=C(C)C2CC2)C)CCOC(CCF)C1 c1(Cc2nc(C)sc2)cn2cc(C(N3CCC(S(C)(=O)=O)C3)=O)ccc2n1 N1(S(CC)(=O)=O)CC2(CN(C(C3CC3Cc3ccccc3)=O)CCO2)C1 CN1CCOC(C(N2CCC(F)(CNC(C3(C(F)F)CCCC3)=O)C2)=O)C1 C(=O)(CC(C)(C)CC(F)(F)F)NC1(C2CCN(C(COCC(=O)OC)=O)C2)CC1 N1(C(CCN(C(=O)CC2CC3CCC2C3)C)=O)CCC=C(F)C1 N1(C(C=CC(C)(C)SC)=O)CC2CC3CC2C1C3C(=O)Nc1cnc(C)nc1SC C1(C(=O)NC(C#C)CC2CC2)CC12CC(NC(=O)COCCSC)C2 C(CCCCCNC(=O)CCN(CCCCC)C(C)C)NC(C(C)=CC)=O C(=O)(C(C)(C)CC(=O)OC)NC(C1CC(CC)NC(=O)C1)=O.C1C=CCN1 c1(OCC)cnc(C(=O)NC(C)C(C)NC(c2cc(C3CC3)ccn2)=O)c(Cl)c1 Cc1cc(C(N2CC(NC(=O)C(O)C3CCC3)C(O)C2)=O)c2cccnc2c1C N1(C(CN2C(C)CCC2)=O)CCC(C)(CNC(=O)Cn2cc(N)cn2)C1 C1(C)(C(N(CC(N)=O)C(C)C)=O)CC12CCN(C(C1(N)CCCC1C)=O)CC2 N1(C(C(C)OC)=O)CCC2(CC2)CC1C(=O)NCC1(C)C=CCCC1 C1(NC(c2ccnc(OC)n2)=O)CCC2CCN(C(=O)CC3(C(F)F)CC3)C1C2 C1(C(=O)Nc2cccc(C(=O)O)c2)CC2(C1)OCCO2 C1(CCOC)CN(C(=O)C=CS(C)=O)CCN1C(c1nn(C(F)F)cc1Cl)=O C1(C(=O)NCCC2C(CNC(C(C)SCCCC)=O)C2)(N(C)C)CCCC1 C(CN(C(=O)CC12CCCC1C2)C)(CO)(CO)NC(C(C1CC1)OCC)=O CC1CC(C(N2CC(CC(C)NC(=O)C3=NOC(C)(C)C3)C2)=O)Cc2nn[nH]c21 N1(C(CC(C)(F)F)=O)CC(C2(NC(=O)CC(C)(C)C)CC2)C1 C(=O)(C1OCCc2cc(O)ccc21)N1C2CC(NC(c3n[nH]cc3Cl)=O)C2CC1 Cn1cccc1C(N1CCC(CCNC(c2csnc2-c2ccccc2)=O)C1)=O C(=O)(C1=CCCOCC1)NCC(C)(CNC(c1nc(C)ccc1F)=O)OC C(=O)(CCCN=[N+]=[N-])N1CCC(N(C)C(C2COC(=O)N2)=O)CC1 C1(CNC(CCCCN(C)C)=O)CC2CCC(C1)N2C(=O)C(O)c1ccco1 c1(C(N2C(C)C(NC(=O)CN(C)CCO)CC2)=O)ccc2[nH]ccc2c1 CC1(C(=O)NC2CC(CNC(=O)C=CC(F)(F)F)C2)CCCS1(=O)=O CCC(C)CCC(=O)Nc1c(Oc2cnn(-c3ccccc3F)c2)ncnc1C CCC(C)(O)C(=O)NCCCCCCNC(c1nnn(C)n1)=O c1(OC)n[nH]cc1C(=O)NC1CC(CC(=O)NCC2CC2C(C)C)C1 c1(OCCOC)ccc(C(=O)N(C)CC2CCN(C(=O)CCC(C)SC)C2)nn1 Cc1nccnc1C(N1CCOCC1c1cn(Cc2cccnc2F)nn1)=O c1(C(=O)NC2CC(NC(C(C)CN(C)C)=O)C2)ccnc2c(F)cccc12 C(=O)(CCCCCN=[N+]=[N-])N(C(C)=O)C(C)C1CC1.C(=O)(C(CC(C)C)O)OC N1(C(Cc2c(C)nc[nH]2)=O)CC2(CCNC(=O)CCc3ccncc3)CCC1C2 C1(CNC(CCCN(C)C)=O)(NC(C2CCCN2C)=O)CC(F)(F)C1 c1(CCC)cccc(NC(C2CCC(CNC(C3C4CCCC34)=O)O2)=O)c1 Cn1cnc2nc(NCc3ncc[nH]3)nc(N3CCC=C(Cl)C3)c12 N1(C(CC(=O)OC)=O)CCC2CCCN(C(=O)Cn3ncn(C)c3=O)C2C1 c1(C(=O)NC(C2(CNC(c3ccns3)=O)CC2)C)ccc(N2CCC2)nc1 C1(C(C)C)N(C(=O)C2CC2)CC12CCN(C(=O)C(F)(F)c1cscn1)CC2 c1(C(=O)NCC(C)N(C(C(C)OCCCC)=O)C)ccnc2ncnn12 C1(CNC(c2[nH]nc3cnccc23)=O)CN(C(=O)CC2CCCC2)C2(CCC2)C1 n1(CC)cc(C#N)c(=NC(=O)C2(C)CCN(C(c3cc(Br)c(F)cc3Br)=O)C2)[nH]1 c12nc(c3c(n1)CSC3)N1CCC(CO)(C1)CN2.c1(CSC)ccc(N2CCC2)o1 C(N=c1[nH]c(N2CCCC(C(C)(C)C)C2)nc2cccnc12)c1n(CC)ccn1 c1(C(=O)NC(C(=O)N(CC#C)CCF)CC2CCCCC2)cc(C)oc1CC C1(NC(C2C(CC)C2)=O)CN(C(c2csc(C(F)F)c2)=O)CC12CCOCC2 C1(C(N(CC(=O)NCCc2onc(CC)n2)C)=O)C2CCC(=O)C12 CC(C(=O)N(C1CCN(C(C2(C(C)(F)F)CC2)=O)C1)C)C(C)(C)C c1(OC)cc(C(=O)NC(C)CNC(=O)C(C2CCOC2)SC)sn1 c1(C(C(=O)NCc2cccs2)N(CC(C)(C)CO)C)cc(C2CC2)ccc1F Cc1ccc(C2CCC2)c(C(=O)NCCCCNC(=O)C(F)C2CCC2)c1 c1(OC)ccc(CC(=O)NC2CC(O)CN(C(c3csnc3OC)=O)C2)cc1F O=C(C#CC1CCCOC1)NC1(C2CN(C(=O)CN3CCCCC3)C2)CC1 CN1CCN(C(=O)CCF)C(CNC(C2CC(F)(F)C2(C)C)=O)C1 CC1CC1(C(N1CC(C(=O)N(C)C)C1)=O)NC(=O)CC1CCOC1 CCCCC(C(=O)NCC1(O)CCSC1)NC(=O)COC(C)C C(C(C(=O)N1CCCCC1C(C)(C)C)C(C)(C)C)NC(C=C(C)C1CC1)=O N1(C(C2CCCN(C(c3ccnc(O)c3)=O)C2)=O)CCC(C2=NOCC2)C1 c1(OC)ccc(F)c(C(=O)NCC2(CNc3ncc(Br)cn3)CCC2)c1 C12(CCCO1)NC2.C1CC(=O)N1.C(C(=O)N(C)CCO)SC C12(C(N3CC(C(=O)OC)C3)=O)CCC(CF)(C1)OC2.c12cc(cs1)OC2 c1(C(=O)NCc2nc(CNC(CCCCC#C)=O)sc2)cc(S(N)(=O)=O)c[nH]1 C1(C(=O)NCC2(NC(CCNC(=O)OC)=O)CCOC2)OCCC1(C)C C12(C(=O)O)CC1CCCN2Cc1cccc(-c2cn(-c3cncc(F)c3)nn2)c1 CC1(NC(=O)CCC2CC2(C)C)CCN(C(C2CCC3CC3CC2)=O)CC1 C1(C(=O)NCc2cscc2C)(CC)CCN(C(=O)CCC2CCCC2)CC1 c1(C(=O)NC2CCC(COC)C2)cc(CNC(=O)C(O)C(C)C)nn1C c1(OC)ccc(CC(=O)N(C(C)CNC(=O)C=C2CCC(C)C2)C)cc1O CN1C(=O)C(=O)c2cc(NC(c3onc4c3CCCC4)=O)ccc21 C1(C(=O)NC(CCNC(c2cncc(C)n2)=O)C)CC2(CCOCC2)C1 C1(C(=O)NC2COCCN(C(C(CCC)C(C)C)=O)C2)CNC(=O)CC12CCC2 c1(CCC)nc(C)c(C(=O)NC2CC(CCNC(c3cccnc3CC)=O)C2)s1 Cc1cc(C)c(C(N2CCCN(C(=O)CCc3ccc(=N)[nH]c3)CC2)=O)cn1 C1(NC(c2ccc(CSC)cc2)=O)CCCCN(C(C2CC(C)(C)CO2)=O)C1 c1(OC)cnc(C(=O)NCC(O)CNC(=O)CC2(C)CCCC2)nc1 C12CCN(C1CC)C(=O)N2.c1(C(=O)NC)nocc1CC.C(C)(C)(C)O c1(CNC2CCN(OC)C2)noc(NC(=O)N(S(C)(=O)=O)C)n1 Cc1nnc(N2CC(O)(C(C)NC(c3cccc(C4(C)CC4)c3)=O)C2)nc1C CCCCC(C(=O)N1CCC(C(=O)NCC(CC)CC)C1(C)C)C(C)C Fc1ccccc1-c1csc(NCc2csc(-c3ccccc3)n2)n1 c1(C(=O)NCCCNC(c2c(CC)ocn2)=O)c(Br)c2ccccc2n1C CCCC(C)(CCC)C(=O)N1CC(O)(C2CCCN2C(=O)Cn2cncc2C)C1 N1(C(C=C(C)c2ccsc2)=O)CCCC(O)(CNC(C2CC3C(C2)C3(F)F)=O)C1 N1(C(C2C(C(C)C)CCC2)=O)CCC(CNC(c2coc(Cl)c2)=O)CC1 c1(OC)cccc(C(O)CNC(=O)N(CC(C)Cc2nc(C(F)(F)F)cs2)C)c1 c1(OC)cc(CNC(C2CN(C(c3csc(Br)c3)=O)CCO2)=O)ccc1[N+](=O)[O-] C1(NC(CC#N)=O)CC12CCC(NC(C1(C3CCCO3)CCCO1)=O)CC2 Cc1cc(-c2cc(O)ncc2Br)cc(C)c1F C(=O)(C(CNC(C1(C)COC(=O)N1)=O)C(C)(C)C)N1CCC(C)(N(C)CC)C1 c1(C(C(=O)NC2CC2)N(c2ccsn2)CC)cccc2c1OCO2 c1(C2CN(C(CCO)=O)C2)ccc(N)cc1.N1(CC)CCOC1=O.CN1CC1 C1(C(=O)OCC)N(C(=O)C=Cc2ncccc2C)CC12CCCC2 N1(C(C)=O)CS(=O)(=O)CC1C(=O)NC1(C)CCN(C(c2cnccn2)=O)C1 Cc1c(C#N)c(=NC2CC23CC(NC(N2CCOCC2)=O)C3)[nH]c2ccccc12 N1(C(C=C(CC)C)=O)CCN(C(C2CCC(=O)C2)=O)CC1c1cccc(Cl)c1 CCCCC(C)C(=O)NCC1(NC(C2CC3C(C2)C3(F)F)=O)CCC1 N1(C(C2ON=C(C(C)C)C2)=O)CCn2nc(CNC(=O)Cc3cncs3)cc2C1 c1(CONC(c2cn(-c3ncccn3)nn2)=O)ncc(O)cn1 C(=O)(C(CC(N)=O)NC(c1ccc(Br)c(C)c1)=O)OCC C1(NC(c2cnn(CC)c2C)=O)CCN(C(=O)CC2(C3CC3)CC2)CC1F c1(C(=O)NCC(N2CCN(C(CC(C)OC)=O)CC2)C)cccc2c(C)n[nH]c12 C(=O)(CC(C(F)(F)F)NC(C1CC2(CCC2)CO1)=O)N1CCN(CCC)CC1 c1(C(C)NC(=O)NC2C(c3cn(CC)nc3)OCC2)cn(C)nc1NC(C)=O c1(C(N(C2CCCC2)CCCC)=O)[nH]ccc1CNC(c1coc(C(F)F)c1)=O C(=O)(C1Cc2ccccc21)NC(CNC(C(F)=CC)=O)(C)CSC C(CCCCNC(=O)COCc1ccccn1)N.CC1CN(CC(=O)NCCO)C1 c1(C(N2CC(OCCNC(c3ccc(CC)cc3)=O)C2)=O)ncc(C)cc1OC N1(C2CC2)CCOCC1CN(C(=O)CCOC)C.c1(COC)nn[nH]c1C=O C1(C(=O)NCC(C)C#N)N(C(c2cc(N)cc(F)c2)=O)CCC1(C)C N1(C(CCOCC#C)=O)CCCC2(C1)CN(C(C1CCCN1C1CCCC1)=O)C2 c1(CC)ccc(C(=O)N(CC(O)CN(C(=O)CCc2csc(=N)[nH]2)C)C)c(C)n1 c1(C(=O)NCC(CNC(C(C)(c2ccccc2)OC)=O)O)n[nH]c(C)c1F c1(NCC2(OC)CCCCCCC2)ccc([N+](=O)[O-])c(OC)n1 N1(C(C2(C)CCC2)=O)CCC(NC(C2CC2c2ccc(Cl)s2)=O)C(CO)C1 c1(OC(C)C)ccc2c(c1)CCC2NCCS(=O)(=O)c1cnn(C)c1 CC1CCN(C(c2cnccc2Cl)=O)CC1NC(C1(C(F)(F)F)CCC1)=O C1(NC(CC(C)SC)=O)CCN(CCC2CC3CCC2C3)CC1 c1(N)ccc2nnnn2c1.O=CN1CCN(C(N2CCC(C(=O)C3CC3)C2)=O)CC1 N1(C(c2c(C)nns2)=O)CC(=O)NCC1C(=O)NCC(C)C1CCC1 c1(NCC)ccccc1C(N1CC2CC1C2CNC(=O)CCCC1CC1C)=O N1(C(C(c2ccc(OC)cc2)=O)=O)CCN(C(C2CC(C)C2)=O)C2COCC12 N1(C(C(=O)Nc2cc(C(F)(F)F)ccc2Cl)=O)CCC2CCCC2C1 N1(C(C2ON=C(CC)C2)=O)CCN(C(=O)C2=NOC(C(C)(C)C)C2)C2CCC12 C1(N(C(C2CC2C)=O)CC)CCN(C(=O)CCC(C)C)CC1 c1(C(C)C)ccc(C(=O)NC(C)C(=O)N2CC(c3cc[nH]n3)C2)o1 n1(CC(C)C)cc(C(C(=O)N(C)C)N(C)CC2CCOCC2)cn1 C1(CC(=O)NCC2CC(=O)NCC2)CC2(CCOCC2)CO1 N1(C(C(CC=CC)C)=O)CC2CCC2(CNC(=O)COCCCF)C1 C1(C(N2CC(C(N(C)Cc3ccon3)=O)C(F)C2)=O)CC(=O)NC(=O)N1 CC(C)CC(C)(CNC(=O)C1=CCCCC1)NC(C1CCCCS1)=O C=C(C)c1ccccc1NC(C1(C)CC(NC(=O)C(C(C)C)OC)C1)=O CC1CCc2ncc(C(=O)NC3CC3CNC(c3sccc3C#N)=O)n2C1 C1(CS(=O)(=O)NC)CCCCN(C(=O)NCC2(C3CCCCC3)COC2)C1 n1(CC(=O)NC2CCCCC2NC(c2cc(Cl)cnn2)=O)ncc2ncccc12 C(c1ccc(=N)[nH]c1)=CC(=O)NCC1OCCN(C(c2c(C)ncn2C)=O)C1 N1(C(C2C(C(=O)OCC)CC2)=O)CC(NC(=O)Cc2cncnc2)C(C)(C)C1 c1(CC(=O)NCC2(O)CN(C(C(CC=C)(C)N(C)C)=O)C2)cn2cc(C)sc2n1 C1(NC(c2ccc(OC)c(F)c2)=O)CCN(C(C2CCC2C)=O)CC(C)(C)C1 CC1=NC(C)(CNC(C(=O)NCc2ccccc2NS(C)(=O)=O)=O)CS1 c1(C(N2CC(NC(CCOCC)=O)(CF)C2)=O)cccc2ccnn12 c1(OC)ccc(C(=O)NC(C)C(C)NC(=O)C(F)(F)c2nccs2)cc1O C12(NC(CNC(CC)=O)=O)CCN(C(c3ccn(CC)c(=O)c3)=O)CCC1C2 C1(C2CC2)(CN2CCC(C(N3CCC(c4c(N)non4)C3)=O)C2)CC=CC1 C(=O)(C1COc2ccc(Cl)cc21)N(CCCNC(C1CC(C)(C)CCO1)=O)C CC(O)CCN=c1[nH]c2c(c(=NCC3(CF)CC34CCOCC4)[nH]1)CSC2 C(=O)(C1=CCC2CCC1N2C(=O)CCC1CC(C)C1)NCc1c(C)nc[nH]1 C(CCCCCC(=O)NCP(C)(C)=O)NCC1C(C(=C)C)OCC1 CCCCCCC(C)C(=O)NC1CC2CC1N(C(=O)C(=O)NC1CC1)C2 N1(C(C(C)OCCC#C)=O)CCC2(C1)CN(C(c1cc(C(F)F)no1)=O)CCO2 C12(NC(C(C)CF)=O)CCCC1N(C(c1cc(-c3ccncc3)on1)=O)CC2 CCC(O)C(F)(F)C(=O)N1CCCOC(CCNC(=O)CCN2CCCC2=O)C1 C1(C(=O)NC2CCOCC2NC(C2CCN(C3CC3)CC2)=O)(OC)CCOCC1 N1(C(CCC)=O)CCCCC1C1(NC(c2ccccc2Cl)=O)CC1 CCC(CC(F)(F)F)C(=O)N(C)CCNC(c1ccc(SC)cc1OC)=O C1(C(=O)NC2(C)CC(NC(C(C)NC(CC)=O)=O)C2)CCN(C)C1CC CC(C)C(C(=O)N(C)C)N(C(=O)CCCc1ccncc1)C.C12CC1NC(=O)NC2 C1(NC(CN(C(=O)C(C)COC)CC)=O)CCCC1CN(C)C C(N=c1[nH]c2c(c(=NCCOC(F)(F)F)[nH]1)COC2)c1ccc(SC)cc1C C1(NC(c2c(C)csn2)=O)CCN(C(c2ccsn2)=O)C1c1ccccc1 C1(NC(Cc2c(C)n[nH]c2)=O)CN(C(=O)CCC(=O)C2CC2)CCC1C CC1(C)C2CCC1(C(=O)NC1CCCC(C(=O)NC3CCOCC3F)C1)C2 C1(n2c(-c3c(C)n(C(C)C)nn3)nc(-c3cccc(C(N)=O)c3)n2)CCCC(C)(C)C1 CN1CC2CCCC(CC1=O)N2C(c1cc(Cl)ncc1Cl)C(=O)NC(C)(C)C c1(CC(=O)NCC(CO)NC(CC2CCC(=O)NC2)=O)cccc2ncccc12 c1(C(=O)NC(CC)CNC(=O)CCC2CCC(=O)N2)c(F)ccc(C)c1Cl c1(C(=O)NCC(C)CN(C(=O)CC2CC3(CC3)C2)C)ccc2c(c1)COB2O CC1(C)CCC(O)(N(c2ccccc2)C(=O)NC2(NC(N)=O)CC2)CC1 C1(C(=O)NCC=CCNC(C2(C(F)(F)F)CCO2)=O)CCC1(F)F C1(CCC)(NC(C2CC3C=CC2CC3)=O)CCCN(C(=O)CC2CC2(C)C)C1 C1(CCNC(c2cnc(N(C)C)s2)=O)CN(C(C2OCC2(C)C)=O)CCS1(=O)=O C1(C(N2CCN(CCNC(C(CC=CCC)C)=O)CC2)=O)CCCC1C1CC1 C1(C(C)(C)OC)CC(C)(C)CN1C(=O)C=Cc1ccc(SC)s1.C1(C(=O)N)CC1CF c1(C(N2CC(CNC(COCC#C)=O)N(C)CC2)=O)c(F)c(F)c(F)c(F)c1F C1(CNC(CC(CC)OC)=O)COCCN(C(c2ccnc(OC3CC3)c2)=O)C1 C1(C(C)C)CN(C(=O)COCc2nc[nH]n2)CCN1C(c1cnc(C#N)s1)=O [N-]=[N+]=NC1CC(C(=O)NC(Cc2ccco2)C(=O)NC2CCCC(O)C2)C1 C1(NC(C(C(CC)C)O)=O)CC2CN(C(c3sc(CC(C)C)nc3C)=O)CC2C1 N1(C(c2c(OC)n[nH]c2)=O)CC2(CCOCC2)CC1CNC(C1CC1C(C)C)=O Cc1cc(C(N2CC3CC3(CNC(=O)C=CC3CCCC3)C2)=O)c(N)cc1F Cc1cc(C(=O)N(CC(=O)NC2(C(F)F)CC(O)C2)C(C)C)ccc1F C=C1c2ccccc2C(=O)N1CC(N1C(CNC(=O)Cc2ccoc2)CC1)=O N1(CS(CC(Cc2ccccc2)OCC)(=O)=O)CCC(F)(c2ccc(F)cc2)CC1 C1(CC2(O)CCC2)CN(C(=O)CN(C(=O)CC2CCCC2)OC)C1(C)C C1(C(N2CC(C(=O)NC3COCC3C)(CC)C2)=O)CC2(C1)CC(O)C2 Cc1ccc(C)n1CC(N1CCC(CN(C(=O)C(O)C(F)F)C)C1)=O N1(C(c2ccc(F)cc2Cl)C(=O)NCC=C)CC(=O)N(C)CC1CC C1(CC)(CC)CCCN1C(=O)CC1CCCN(C(=O)C(C)C)C1 C12(C(=O)NCC(CNC(c3cn(C(C)(C)C)nc3)=O)O)COC(C1)OC2 C(c1cccnc1)=CC(=O)NC1CCC(N(C(C=C(C)I)=O)C)C1 C(=O)(CCCCCN(C(=O)C(C)OCCC(C)C)C)NC(C(CC)(C)C)C c1(C(N2CC(COC)(CNC(C3CCNC3=O)=O)C2)=O)cnc2sc(C)c(C)n12 C=C(Cl)C(C)(C)C(=O)NCC1CN(C(c2cccs2)=O)CC12CC2 c1(C(=O)NCCN(C(c2cc(C#N)c(N)cn2)=O)CC)ccc(S(N)(=O)=O)cc1 N1(C(C(C)CC2CCCCC2)=O)CCN(C(=O)COC(=O)CO)CC1C(C)(C)C Cc1ccc(CN=C(NCC2CCCCC2)NC2CCCC(F)C2)cc1 C1(C(N2CCC(N(C(=O)CCC3CC3(C)C)C)C2)=O)CCC(F)(F)CC1 C1(C(=O)NCC(C(=O)OC)C)CN(C(=O)CN(C2CCCC2)C)CCO1 n1(C(C)C)ccnc1C(=O)NCCCCCNC(=O)CC1CC(CF)C1 C=CCC(C)(CC)C(=O)NCCOCCCNC(c1ccnn1CC1CCC1)=O N1(C(=O)NC2CC=CCC2)CCCCC1CC(F)(F)F c1(CN2CCC(NC(=O)NCCc3ccccc3F)C2)ccc2ccsc2c1 C(=O)(C#CC1CCCC1)N1CCN(C(c2ccc(C(O)CF)cc2)=O)CC1CF c1(C(=O)NC23CC(CNC(CCN(C)CC)=O)(C2)C3)ccc(CO)c(Cl)c1 Cc1ccc(C(=O)NC23CC(C2)N(C(=O)CCC2CCC(O)CC2)C3)cc1N C1(C(N2CC(NC(c3c(C)nc(C(C)OC)s3)=O)C2)=O)CNC(=O)CC1(C)C C(=O)(CCC(=O)C(C)(C)C)NC(C=CC(=O)NC(C#C)CC1CCCC1)C c1(C(N2CCC(N(C(=O)CCN3CCCC3)CC)C2)=O)cc(F)cc2nn[nH]c12 Cc1noc(C)c1CNC1COCC1NC(N)=O.c12cc(ccn1)CNC2=O C1(NC(C2CCC(CNC(CNC(C(CC)C)=O)=O)C2)=O)CC2OC1C1CC21 N1(C(Cn2c(C)cc(C)n2)=O)CCN(C(c2cnc(O)s2)=O)CC1c1ncc[nH]1 c1(NCc2c(C)cc(C)s2)[nH]c(=NCCn2cccn2)nc2sccc12 N1(C(CCCN(C)C)=O)CCCCC1C1CCCN(C(=O)Cc2n[nH]c(=N)s2)C1 Cc1cccc2cccc(C(=O)NCC3(C)CCN(C(=O)C4=CCSC4)CC3)c12 C1(NC(C2C(C(C)C)OCC2)=O)CCCCCC1C(=O)N1CCCO1 c1(C(C)(C)C(N2CCN(C(c3ccc(S)cc3)=O)C3CC23)=O)ccc(C#N)nc1 C(c1nc2ccccc2o1)=CC(=O)NC(C(C)C)CNC(=O)C(CO)C(C)(C)C C1(C(=O)NCC2CN(NC(C3CC(CF)C3)=O)C2)CCN(C2CCCCC2)CC1 c1(C(N2CCC(C)(CCNC(C3N(C)C(=O)CC3)=O)C2)=O)ccc2ccoc2c1 c1(OC)cc(CCN2CCCC(C(=O)N(C)C)CC2)cc(-c2cccc(N)n2)c1O N1(C(c2c(CC)csc2)=O)CCC2(CCCN2C(=O)C(COC)N(C)C)C1 CC1C2CCC(C2)C1C(=O)N(CCn1cc(C2CCCO2)nn1)C1CC1 C1(CNC(C2C(CCC)C2)=O)COCC1NC(=O)CNC(C1CCCCC1)=O C1(CNC(C(c2cncnc2)C)=O)CCN(C(=O)C(=O)Nc2ncc[nH]2)C1 N1(C(C(c2ccccc2F)OC)=O)CC2(CCN2C(=O)C(C)(C)C(C)C)C1 N1(C(C2C(C)OCC2)=O)CCC(NC(c2ccc(-n3cnnn3)cc2)=O)C1(C)C C1(C(=O)NC(c2nocc2C(=O)NCCS(C)(=N)=O)C)CC(=O)C1(C)C C(=O)(CCCC(C)(C)C)N1C(CNC(c2nc(C)[nH]n2)=O)C(C)CC1 c1(OCC)ccc(C(N2CCC2C(=O)NCCc2ccc(Cl)cc2Cl)=O)cc1O C1(CNC(c2c(F)ccc(C)c2)C)(CO)COCC2COCCN12 C1(C(N2CC(NC(=O)C(F)(F)CC3CC3)CC(F)C2)=O)Cc2cc(Cl)ccc2O1 C(=O)(C(C)C(C)S(C)(=O)=O)N1CCC(C(C)Nc2ncc3c(n2)COC3)C1 c1(CC)nccnc1C(=O)NCC1CCCC(NC(c2ccc(Cl)cn2)=O)C1 C1(CC(=O)NCC2(CC)CCC2)(CNC(c2c(CC)c[nH]n2)=O)CNC(=O)C1 C(=O)(CC(O)CNC(C12CC1CCN2C(=O)Cn1cncn1)=O)OC c1(COC(C(=O)OCC(c2ccccc2)OCC)C)ccc(Cl)cc1 CC1=NC(C)(CNC(=O)C(CCN(C)C)NC(=O)C=Cc2cnn(C)c2)CS1 C1(CNC(CNC(=O)OC)=O)N(C(C2CCCN2C(C)=O)=O)CCCC1(C)C C12(CNC(COC)=O)CC(CNC(C3(CC(C)C)CCNC3=O)=O)(CO1)C2 C=C(Cl)CC(C(=O)Nc1ccc(CC)nc1)NC(=O)C(C)C1CCC1 c1(C(c2n(CC)nnn2)NC(C(C)C)C2CCC2)nccc(Br)c1C N1(C(CCC#C)=O)CCN(C)C(C(N2CCN(C(C)=O)CC2)=O)C1 O=C(C1=CC2C=CC(C1)C2)NC1(CF)CCN(C(=O)C(O)Cc2cnc[nH]2)C1 N1(C(CC=CCC)=O)CCC2(CO)CN(C(c3cc(OC)ccc3C)=O)CC2C1 C(=O)(C(F)CC(C)(C)C)NC(C)C(C)C(=O)Nc1ccc(N(C)C)cc1 C(C(C)(C(=O)N(CC(C)CNC(=O)C=Cc1nccs1)C)OC)OC C(=O)(C(C)Cc1cnn(C)c1)NC(CNC(C1(SC)CCC1)=O)C1CC1 C1(CN(C(C2CC2OC)=O)CC)CCCCN1C(c1[nH]c(COC)nc1C)=O C12(NC(c3c(C)cc(F)s3)=O)CCN(C(c3coc(CO)c3)=O)CCC1C2 c1(OC)cnc(C(=O)NCC23CC(CN2C(C2(OC)CCC(C)C2)=O)C3)c(F)c1 CCCC(CC)CCC(=O)NC1CC(F)(CNC(=O)Cc2ccn(C)n2)C1 c1(C(=O)NCCNC(C2(C(=O)OCC)CC2)=O)c[nH]c2ccc(F)cc12 Cc1cc(C2(C)CC2)oc1C(=O)NNC(=O)N(C)CCO C1(CNC(CCSCC)=O)C2CN(C(=O)CCCOc3ccccc3)CC12 c1(C(=O)NCCCOC)cn(C2CCOC2)nc1SCc1ccccc1 C=CCCCC(=O)NCC1CN(C(=O)Cn2cc(C)c(C(F)(F)F)n2)C1 c1(CCC(=O)NCCCCCc2cn(C3CCN(C)C3)nn2)ccncc1Br N(C1CCCc2ncc(C(F)(F)F)cc21)C(=O)CCc1cc(Br)cs1 C12(CC)CC(C(=O)NCC(O)CNC(=O)C=Cc3ccn(C)c3)(CO1)C2 CC(C)C(C)CC(=O)N1CCOCC1CN(C)C(c1cn[nH]c1)=O Cc1ccc(I)cc1C(=O)NC1C2CN(C(C3CCC(C(=O)O)CC3)=O)CC12 CC(CCCNC(c1coc(C2CC2)n1)=O)NC(=O)CCn1cc(Cl)cn1 O(N1CCC(N(C(c2csc(C#N)c2)C(=O)NC(C)C)C)CC1)CC CC1CN(C(=O)CC2CCCS(=O)(=O)C2)CCCN1C(c1cccnc1Cl)=O N1(C(C)=O)CCC(N=c2nc(N3CCC(F)C3)[nH]c(N3CC(F)(F)C(F)C3)n2)C1 c1(CC(=O)N(C)CCN(C)C(c2ncn(C)n2)=O)c[nH]c2cccc(Cl)c12 N1(C(CNC(=O)CCC2CCCO2)C2CC2)CCN(C(=O)CCOC(F)F)CC1 CCCC(O)CC(=O)NC1CCC(NC(C23CCCC(C2)OC3)=O)CC1 C(N=c1[nH]cc([N+](=O)[O-])c(O)n1)C1CCCN(C(CC2C(C)=NOC2=O)=O)C1 C1(C(N2CC(NC(C3CCN(c4n(C)ccn4)C3)=O)C2)=O)CCC(C(N)=O)CC1 c1(C(N2CC(C)(NC(C(c3n(C)cnc3)O)=O)C2)=O)ccc(F)c(F)c1 C1(CNC(C(=O)N(C2CCCCC2)NC(C)=O)=O)OCCC1NC(=O)C(C)(C)C c1(-n2cc(CCCN(C(COC)=O)C3CCC3)nn2)ccc(S(N)(=O)=O)cc1C CC(C(=O)NCC1CC(NC(c2ccncc2N)=O)C1)C(F)F CC(C)C(C)(O)CNC(C1(NC(=O)CCc2ccn(C)n2)CCSC1)=O c1(C(=O)COC(=O)C(F)C2CC2)cccc2cccnc12 C1(CNC(C=CC(C)C)=O)CC2(CCN(C(=O)C=C3CCN(C)CC3)C2)CO1 C(C(CNC1(c2nnnn2CC(F)F)CC(CO)C1SC)C(C)C)OC N(C1CCc2c(F)cccc21)C(c1ccccn1)C c1(OC)cnc(Cl)[nH]c1=NC(=O)c1sc(=NCc2ccccc2[N+](=O)[O-])[nH]c1C c1(CNC(C2CC(NC(=O)COCC(F)(F)F)C2)=O)c(F)cccc1F C1(CC(N2CCC(CNC(CSS(C)(=O)=O)=O)C2)=O)CC2CCC1O2 CCC(C)C(C(=O)NC(C)=O)NC(c1nnc(-c2ccncc2)o1)C C1(CNC(CCn2c(CCC)ncc2)=O)(OCCC(=O)NCC)CCCCC1C O=C(C1=CC(O)C(NC(=O)C2=C(Cl)CCOC2)C1)NCC(C1CCCCCC1)O N1(C(C2=CCCN(C(C(C)OCC(C)C)=O)C2)=O)CCC2(CCN(C)C2)C1 c1(C(=O)NCC2C(NC(CCc3cc(C)no3)=O)CCCC2)cccc(O)c1F C1(NC(C2CCC(CC)CC2)=O)CCN(C(=O)C2=CC(C)(C)C2)CC1O c1(NCC2(OC)CCC2)ncc(C)cc1S(=O)(=O)NC(C1CCOC1)c1cccs1 N1(CCC(N2CCC(N(S(C)(=O)=O)CCN)C2)=O)C(=O)c2ccccc2S1(=O)=O c1(C(=O)NCCC2(O)CN(C(c3c(OC)oc(C)n3)=O)C2)ccc2c(c1)NCC2 c1(N(C(C)=O)CC)ccc(NC(=O)C(=O)NCC2(C)CSC2)cc1 N1(C(C(C=C)OC)=O)CCC(C)(NC(c2cncnc2C)=O)C1 C1(CCC)CN(C(C2(C(=O)NC3CC3)CC2)=O)CCN1C(=O)C=CS(C)=O C(=O)(C(C)C(C)c1ccccc1Cl)N(CCCNC(c1cnn[nH]1)=O)C(C)C c1(C(NNC(=O)C2CCCS2)=O)n[nH]c2ccccc12 c1(C(=O)NCC(CNC(C2CCC(=O)N2)=O)O)cc2nccc(C(F)(F)F)n2n1 N1(C(C(CCOC)OC)=O)CCC(C(N2CC(N3CCCC3)C2)=O)C12CC2 c1(N2C(COC)(CNC(=O)CC(C)N(C)C)CCC2)c(Cl)cccc1[N+](=O)[O-] c1(OCC(=O)N(CCCCN(C(CC2(C=C)CC2)=O)C)C)c(C)cc(Cl)cc1C c1(C(=O)NC(CNC(C2C(C(=O)OCC)C2)=O)C)cc(C)c(F)cc1Cl C#Cc1cccc(C(N2CCC(NC(c3cc(C)ccc3N)=O)C2C)=O)c1C c1(CC(=O)NC2CCC(NC(C3N(N=O)CCC3)=O)CC2)ccc2[nH]ccc2c1 c1(CC)nc(C(N2CCC(CCNC(c3occc3Br)=O)C2)=O)c(N)s1 N#Cc1ccc(C(N2CCC(NC(C3C=CCS3)=O)C2)=O)o1 C1(CNC(C(C)(C)O)=O)(NC(=O)COCC2CCCO2)CC2CCC1CC2 c1(C(=O)NC(CN(C(=O)CCc2cn[nH]c2)CC)C)cc2c(C)nn(C)c2s1 CCCCCCC(C)CC(=O)NC1(C)CCN(C(c2cc3c([nH]2)CCCC3)=O)C1 C1(C(=O)NCC2(F)CCN(C(c3cccc(C)n3)=O)C2)Cc2nnsc2S1 Cc1ccc2oc(N3CC4CC(NC(=O)C(C)(C)N(C)C)CC(C4)C3)nc2c1 c1(OC)ccc(C(=O)NC2COCCC2NC(=O)Cc2ccno2)c2[nH]ncc12 C1(OCC)CC2CN(C(=O)C=CC(C)NC(C3CCCN3C)=O)CC12 C(=O)(CCCC(C(C)C)NC1CC2(C1)CC2N)OC C1(n2cc(CCOC)nn2)CCCN(C(=O)CC(C)n2ccnc2)CC1 C1(C(N2CCC3(CC(NC(C=CC)=O)C3)CC2)=O)CC12CCc1ccccc12 N1(C(N2CCC3CC(C(=O)OC)C3C2)=O)CCn2c(Cl)ccc2C1C N1(C(c2c(C)nc[nH]2)=O)CC2CC(O)C1C2NC(c1ccc(C(C)C)o1)=O n1(CCC)cc(C(=O)N(CC(C)CNC(c2cc(OC)n(C)n2)=O)C)c(C)n1 C1(CNC(CC(C)c2cnn(C)c2)=O)Cc2ccccc2CN1C(=O)C1CC1 N1(C(C2CN(CC)C(=O)N2)=O)CCC2CCN(C(c3cnc(C)nc3C)=O)CC12 c1(C(=O)NCCCN(C(C=C(CCC)C)=O)C(C)C)c(C(C)C)cccc1C CC1CN(C(c2cccc(=O)o2)=O)CC1n1cc(C2(C)CCCO2)nn1 C1(NC(C2(CCOC)CCCC2)=O)CC(C2CCN(C(=O)CNC=O)C2)C1.C(C)(=O)O CC1(C)CCCN(C(=O)CC2CC2)C1CNC(=O)C(O)Cc1c(F)cccc1Cl c1(C(N2CC(CNC(CC(C)F)=O)N(C)CC2)=O)cncc2n[nH]cc12 c1(C(N2CCC(C(C)NC(=O)CCCC3CCCCC3)C2)=O)cccc(N)c1O C(=O)(CC(C)C(=O)N1CCC(C)(NC(=O)CSc2cccc[n+]2[O-])C1)OCC C1(N(C(=O)CC2CC3CC3C2)CC#C)CCN(C(C2CCCOCC2)=O)CC1 Cc1c(C(N2CCN(C(C3CN(C(N)=O)C3)=O)CC2C)=O)cncc1F c1(C(N2CCC(C(C)NC(c3cc(COC)sc3)=O)C2)=O)cccc(C)c1OC CC(CCC(=O)N(CCNC(=O)Cc1ccc(Br)nc1)C1CC1)N(C)C N1(C(CNC(C2N(C)CC(F)C2)=O)=O)CCC(C2(C)CC2)C1 C1(NC(c2ccc(C(N)=O)o2)=O)CC2CN(C(C34CC5CC3C4C5O)=O)CC2C1 c1(NC(C2C(=O)C3C(C2)C3)=O)nc(Br)ccc1Cl c1(C(N(C2CC(NC(=O)CCOc3cccnc3)C2)C)=O)cnn(C)c1Cl c1(OC)cc(C(C)NC(C2C3CNC2C3)=O)ccn1 C(c1cccc(Br)c1)=CC(=O)NCC(C)(C)NC(C1(C2CCCCO2)CC1)=O Cc1nc(Br)sc1C(=O)N(C)CCOCCCNC(=O)C(C)C(C)C Cc1nc(C(C)(C)C)sc1C(=O)NC1(C)CCN(C(=O)C=CC2CCCCC2)C1 N1(C(CCc2ccn(C)c2)=O)CC2CN(C(c3[nH]nc4ncccc34)=O)CC2C1 CON(C)C(=O)CCCCCNC(c1cc(Cl)ccc1C)=O n1(CC(=O)NCC2N(C(COCC(C)C)=O)CCC2C)ncc2ncccc12 N1(C(=O)CC2CC(NC(c3ccc4n[nH]cc4c3)=O)C2)CCN2CC(O)CC2C1 C(=O)(C1CSc2ccccc21)N(CCC(C)NC(C1CCC1)=O)C c1(CC(=O)NC(C(C)NC(C2C(CCC)CCC2)=O)C)cccc(C(F)F)c1 N1(C(C(C)CO)=O)CCC(NC(c2ccn3c(O)nnc3c2)=O)C2(CCC2)C1 N1(C(=O)CC2OCCO2)CC2(C(=O)NCC(O)C(F)(F)F)CC1CO2 N1(C(c2c(C)cco2)=O)CCCC(C(C)NC(c2ccc(C(C)C)o2)=O)C1 C1(NC(C(C)OCC)=O)CC(O)CN(C(=O)Cc2cc(Cl)cnc2C)C1 c1(C(COC)OC(Cc2ccc(C(COC)=O)s2)=O)ccc(F)cc1F c1(N2CC(CC=C)(C(=O)OC)C2)cc2nncn2cn1.N12CCC(=CC1)CC2 C1(CNC(c2csnn2)=O)CN(C(=O)CC(C(F)F)n2ccnc2)C2(CCC2)C1 n1(CCCOC)cc(C2COC2)nn1.C1(C(=O)NCCC)CCC(CN)C1 c1(C(C(=O)NC2CCOC2)N(CCSC)CC)ccsc1C CC(C)(CC=CC)N.c1(C(=O)NC2CCC2)cn(CCOCCO)cn1 c1(OC)ccc(C(N2CCOC(C(N3CCC(CCO)C3)=O)C2)=O)cc1 c1(CC(=O)NC2CCN(Cc3cc(C(F)(F)F)ccn3)C2)cccc(Cl)c1 CN1N=C(C(=O)NCC(C(N2CCCC(CCO)C2)=O)N(C)C)CCC1=O C1(C(N2CCN(c3ccnnc3)CC2)C(=O)NCCC2CC2)CC(C2CC2)=NO1 CC1(C)CC(NC(=O)Cc2nc(C3CC3)cs2)CCN(C(C2(CF)CCC2)=O)C1 C1(NC(C2(CC)CCCO2)=O)(CC2CC2)CCN(C(C2CCC2(C)C)=O)CC1 O=C1COc2ccc(S(=O)(=O)Nc3ncnc4[nH]c5ccccc5c34)cc2N1 c1(C(=O)NC2C(CNC(CCc3cnn(C)n3)=O)C2)cnc2cc[nH]c2c1 N1(C(C2CC23CCCC3)=O)CC2CN(C(=O)CC3=CCCCC3)CC2C1 c1(C(=O)NC(C)CCCCNC(c2ccn(C3CCC3)n2)=O)cccc(Cl)c1F c1(C(=O)NCC2C(C(=O)NC(c3ccn(C)n3)CC)CC2)cc(OCC)ncn1 C1(F)(CNC(c2c(C)snc2)=O)CCCN(C(=O)CCOCC(F)F)C1 CCCC(CCC)C(=O)NC(CC(=O)NCC1(CC)CCOC1)C1CC1 c1(C(N2CC(N(C)C(c3ccc([N+](=O)[O-])o3)=O)C2)=O)c(Cl)ccc(F)c1Cl C(=O)(C#CC1CCOC1)NC(CN(C(=O)Cc1nc(C)sc1C)CC)C c1(C(C(=O)OCC)(F)F)n[nH]c(=NC(=O)N2CC3(C2)CN(C(C)=O)C3)s1 N1(C(c2c(C)cno2)=O)CCC(NC(C2CCN(C)CC2)=O)C(O)C1 c1(CN2CCC(CC(N3C(C(=O)OC)CCC3)=O)CC2)c(OC)cc(Br)cc1F C1(CC)(NC(=O)CC(C)(C)C)CCN(C(C2CCNC2=O)=O)CC1 N1(C(c2nccc(SC)n2)=O)CCCC2(NC(c3coc(C4CC4)n3)=O)CC2C1 c12c(cc(Cl)cc1Cl)N(CC(F)(F)F)CCO2.C#CCC C12(NC(C(=O)NCC)=O)CCC(CN(C(=O)C(C)Oc3ccc(Cl)cc3)C1)C2 N1(C(c2c(C)c(CC3CCCC3)on2)=O)CC(C)OCC1c1ccccc1 C1(N(C(c2cnn(CC)c2Cl)=O)C)CCN(C(=O)C2=COCCC2)CC1C C1(CNC(C(C)(C)CF)=O)CCC2CN(c3ccnc4ncnn34)CCC2C1 C1(C2CCC2)(CNC(C=CCN(C(C2(CCC)CC2)=O)C)=O)CC1 C1(NC(C=CC)=O)CCN(C(c2ccc(CN=[N+]=[N-])o2)=O)C(C2CC2)C1 c1(SCCc2nc(NC(CC(=O)NCCN(CC)CC)CC)on2)ccc(Cl)cc1 C(=O)(C#CC(C)C)NC(CCNC(Cc1nc(-c2ccc(C)o2)sc1)=O)C c1(C(=O)NCCN(CCC)C(c2cccc[n+]2[O-])=O)cccc2cccnc12 C1(OC)(CNC(=O)NC(C)CC(=O)N2CCCCC2)CCSCC1 C1(CC(=O)N(CCC(=O)NC(=O)C(C)N(CC)CC)C)CCCC1CC C1(NC(C)=O)CN(C(=O)CCc2cccc(Cl)n2)CC2(CC2)C1 CC(N=c1nc2c(cnn2C)c(NC2CCCC2CO)[nH]1)c1ccc(Cl)cc1 C1(CNC(C2CCOC2)=O)CN(C(C2CC=CC2)=O)CC12CCOCC2 N1(C(C2N(C)CCCC2)=O)CC2CCC(C1)N2Cc1cn(CCCCCCO)nn1 c1(-c2cn(CC3OCCN(C(C4C(C)(C)OCC4)=O)C3)nn2)cccc(F)c1F c1(C(=O)NCc2c(NCC)cccc2)cc[nH]c(=N)c1[N+](=O)[O-] C(=O)(C(=O)N=S(C)(C)=O)NC1CN(C(c2ccc(CN(C)C)o2)=O)CC(O)C1 c1(CN(C)C(C2CCCS2)=O)cccc(CNC(=O)CCN2C(=O)CCC2=O)c1 C1(CNC(C2C(CC(C)C)C2)=O)COC(C)(C)CN1C(c1nccc(Cl)c1F)=O N1(C(c2cc(SCC)oc2)=O)CCCC(N(C(=O)C(C)C2CCC2)C)C1 CC1CCN(C(C2CCC3(CC3)N2C(c2n[nH]c(O)n2)=O)=O)CCS1 N1(C(c2cnc(=N)[nH]c2)=O)CC2CC(NC(=O)C3=CS(=O)CCC3)CC1C2 Cc1nccc(C(N2CCC(CO)C(c3ccccc3)C2)=O)c1C c1(C(=O)NC2C(CNC(C3C(C=C)OCC3)=O)C2)c(N)cc(C)cc1F S(=O)(=O)(c1ccc(N(C)CCn2cccc2)c(Cl)c1)NCc1ncc(C)s1 O=C(CC(C(F)(F)F)NC(c1ccc(Cl)cc1)=O)NCc1cccnc1F c1(CCC(N2CCC(CN(C(C=CCC)=O)CC)C2)=O)ccc(Cl)cc1Br C(=O)(C1(C)CCOc2ccccc21)NC1CN(C(C(C)=C2CC2)=O)C1 c1(C(=O)NC2C3CN(C(c4c(OC)cc(N)cc4)=O)C2C3)nccn2cnnc12 N1(C(c2c(CC)cno2)=O)C(C)CC2CN(C(C3(OC)CCC3)=O)CC12 c1(C(=O)NC2C(CNC(c3cc(CCO)on3)=O)COC2)cc2ccccc2o1 c1(C(CNC(C2(CCC=C)CC2)=O)NC(=O)CNC2CCC2)ccc(F)cc1 N1(c2cccc(CN3CC(=O)NC3=O)c2)CC2CC1CN2C(=O)C1CC1 N1(C(c2c(C)cc(O)nc2)=O)CC2CCC(C1CO)N2C(=O)C1=NOC(C)C1 c1(CNC(C(=O)N(CCOC)Cc2cnn(C)c2)=O)nc2cccc(C)c2n1C CC1(NC(C2CC2(C)Br)=O)CCN(C(C2CC(n3ccnn3)C2)=O)C1 CC1(C)CC(NC(=O)CCC2CCCN2C(C23CCC(C2)C3)=O)C(C)(C)O1 N1(C(=O)NCc2[nH]nc(CC)n2)CCC(C)(CN(C)C)C1 C1(C(=O)NC2(C)CN(C(c3c(OC)c(Cl)ncc3)=O)C2)CC12CCC1(CC1)CC2 c1(CC(N2CCC(C)C2CNC(c2nnn(C)n2)=O)=O)cc(F)cc(Br)c1 C(=O)(CC(CC)C(F)F)NCCN(C(=O)C(C)S(N)(=O)=O)CC C1(NC(C(C)OC2CCOC2)=O)COCCN(C(C2CN(C)CCN2C)=O)C1 N1(C(CC(c2nc3ccccc3[nH]2)=O)=O)CC2(CC(NC(=O)C(O)C(F)F)CO2)C1 C1(NC(C(=Cc2ccco2)C)=O)CC2CN(C(=O)C3=CCCS3)CCN2C1=O C(=O)(C1=C(C)OCCC1)N(CC(CC)NC(=O)CC1CCCN1CC)C C1(NC(C2CC=C(C)CC2)=O)CC2CCC(C1)N2C(=O)C(F)(F)C(C)(C)O N1(C(CNC(CC)=O)=O)CCCC1(C(N1CCC(C(C)O)CC1)=O)CC c1(NC(C2(C)CCN(C(C3C(C(=O)OC)C3)=O)C2)=O)cc(OC)cc([N+](=O)[O-])c1 C(C)(C(=O)NC1CCC1NC(c1ccc(-c2ccncc2)s1)=O)(C1CC1)OC c1(C(=O)NCC2C(NC(CC(C)(C)O)=O)CCC2)coc2c1C(O)CCC2 C1(C2CCN(C(c3ccc(C4CC4)nc3)=O)C2)(NC(c2n(CC)ncc2)=O)CC1 c1(C(N2CCC(F)(NS(CC)(=O)=O)C2)=O)c(Cl)cc(F)cc1Cl C#Cc1ccc(C(=O)N(C)CC2CCN(C(c3cc(C(C)=O)c[nH]3)=O)C2)cc1 NS(=O)(=O)c1cnc(NC(=O)NCc2sccc2S(N)(=O)=O)nc1 N1(C(c2cc(C)c(Br)cc2)=O)CCC2(CCN(Cc3cc(Cl)cc(Cl)c3)C2)C1 c1(CC(N2C3C(NC(C4CC4F)=O)C(C3)C2)=O)cccc2sccc12 Cc1c(C(=O)NCC(C)(C(C)C)NC(=O)C=Cc2cncn2C)noc1C1CC1 N1(C(c2c(C)scc2)=O)CCCC(CCNC(c2ccc(CC3CC3)cc2)=O)C1 C1(C(COC)NC(CCC)=O)CCN(C(=O)C(COC)N(C)C)CC1 N(C(=NCC(C)(C)S(C)(=O)=O)N1CCC(O)C(C)(C)C1)Cc1n(C)cnc1 N1(C(c2c(CC)nn(C)c2)=O)CCC(CO)C(NC(=O)C(C)C(C)C)C1 c1(C(C(=O)NC)N(C)Cc2ccc(C(F)(F)F)s2)cc(CO)no1 CC(CC(C)(F)F)C(=O)N1CCC(OCCNC(c2cc3n(n2)CCCN3)=O)C1 N1(C(CCN(C)CC)=O)CCOC(CCNC(c2ncncc2F)=O)C1 CCS(=O)(=O)CC(=O)NCc1nnn(C)c1C(N1CC(F)CC1CO)=O c1(C(=O)NC2CN(C(CCCCC=C)=O)CC2O)sc2cccc(F)c2c1Cl c1(C(N2CC(C)(CNC(=O)CO)OCC2)=O)ccc2cccnc2c1 c1(C(N2CC=CC(NC(CCNC(=O)CO)=O)C2)=O)ccc2ncc(=O)[nH]c2c1 C1(C(=O)NCC2C(OCC)C2)C(C)CCN1C(=O)CCSC(C)C c1(C(N2CCC(CNC(c3c[nH]ccc3=O)=O)CC2)=O)cc(O)nc(C2CC2)n1 CCS(=O)(=O)CC(=O)N1CC2(CCN2C(c2ccn(C3CCOCC3)n2)=O)C1 CC1C(NC(c2cn(C(C)(C)C)cn2)=O)CCCN1c1nnc(CO)s1 c1(NC(C(CNC(=O)OC(C)(C)C)C)=O)ccc(F)cc1F N(C1CCC(C)(C)c2ccccc21)Cc1ncc(C(=O)OC)cn1 c1(CC(=O)N(CCCNC(=O)C(N)=O)C)ccc2oc3ccccc3c2c1 Cc1nc(C(N2CCC(C)(CNC(C3CCCC(N(C)C)C3)=O)C2)=O)sc1C C1(C2(O)CN(C(C3CCC(F)CC3)=O)C2)(CNC(=O)CCc2cncnc2)CC1 c1(C(=O)NCCCC2N(C(C(CC)C#N)=O)CCCC2)cc(SC)ccc1C C1(c2ccc(OC)cc2)C(C(=O)NC2COCCC2NC(=O)CO)CC(=O)N1C CC1CN(C(=O)C=C2CCCCC2)CC(CCNC(c2cc(C#N)cn2C)=O)O1 c1(C(=O)NCC#CCNC(C(c2cccc(Cl)c2)CC)=O)noc(C2CC2)c1C C(=O)(C1=NOC(C)C1C)N1CC(COC)N(C(=O)CSc2ccccc2C)CC1 C(C(=O)NOCCOC)(C(C)C)NC(CC1ON=C(CC)C1)=O C1(NC(c2ccsn2)=O)CN(C(c2cn3ncccc3n2)=O)CCC12CCC2 c1(C(N2CCC(CC(=O)NC(CC)CCCO)C2)=O)ccn2nccc2c1 CC1OC2CCC1(NC(c1sccc1CNC(c1cc(O)cc(=O)o1)=O)=O)C2 C=C1CC2CCC(C1)N2C(=O)C#CCNC(C1CCCC(=O)CC1)=O C1(C(C)C)COCCN(C(C2COCC2NC=O)=O)C1.C1(C)CCC(=O)C(C)C1 c1(C(=O)NC(CN(C(COCC#C)=O)C)(C)C)cccc(Br)c1Cl CC1(C(=O)NCCC2CCN(C(C3COCC3C(N)=O)=O)CC2)CCC(=O)N1 c1(OC)cccc(F)c1C(=O)NC1C2CN(C(=O)CSc3nc[nH]n3)CC12 C#CCC(C)(C)C(=O)NCCCCC(C)NC(c1ccn(C)c(=O)c1)=O C12(C(N3CC(C(C)C)OCC3)=O)CC(CCO1)N(C(c1cnns1)=O)C2 c1(C(C)(C)C)ccc(O)c(C(N2CC(CNC(C3CS(=O)(=O)C3)=O)C2)=O)c1 Cn1cnc2c(NC(=O)C(=O)NC3(CO)CCCC3)[nH]c(=N)nc12 C1(C(=O)NC(CCOC)CO)CC(F)(F)CN1C(=O)CN(C1CCCC1)C N1(C(C2(F)CC(C(=O)OC)C2)=O)CCC2(CC1)C(NC(C1CSC1)=O)CS2(=O)=O c1(C(=O)NC(C)CNC(=O)Cc2ccc(N)cc2)coc2c(F)cc(F)cc12 c1(OC)cnc(CNC(=O)CC(CNC(C2(C)CCCC2)=O)OC)nc1 c1(C(c2n(CC)nnn2)NC2(n3cc(Br)cn3)CC2)ccc(Br)c(C(F)(F)F)c1 C1(C2(O)CN(C(c3cnn(C(F)F)c3)=O)C2)(CNC(c2c(CC)n[nH]c2)=O)CC1 n1(CCCC)nc(C(=O)NCC2CC3(CC3)CN2C(=O)C(C)CCO)ccc1=O Cc1cc(C(=O)NCC2(C)CC(NC(c3coc4c3COC4)=O)C2)cc(C)n1 C(=O)(NN1CCCC1C(N1CCSC(C)(C)C1)=O)c1n(CC)ncc1C C1(NC(c2nc(OC)c(C)s2)=O)CN(C(=O)Cc2sccc2C)CC2CC12 C1(NC(C2(NC(C)=O)CC2)=O)CC(C(=O)N2CCC(O)C(F)C2)=CC1O N1(C(C(CCCOC)C)=O)CCC(C2(NC(=O)C(F)CC3CCCC3)CC2)C1 CC1(C)CCCCC1CC(N1CCN(C(=O)Cc2ccns2)C(CC(F)F)C1)=O c1(CC(N2CC(NC(Cn3ncc(C)c3)=O)C(C)C2)=O)c[nH]c2c(C)cccc12 c1(COC)sc(C(=O)OCCC2(C#N)CCC2)nc1C c1(C(N2CCC(NC(CC3CCN(CC)C3)=O)CC2)=O)ccc(F)c(CO)c1 C1(CC(=O)NCC(CO)NC(=O)CCc2ccco2)CCC(F)(F)CC1 c1(-c2c(CN3C(C(=O)NCCC(CC)O)CC3)cccc2)ccc(OC)cc1 c1(C(=O)NC2C(OC)CN(C(=O)CC(C)NC(C)=O)C2)cc(F)cnc1O CC1CCCC(O)(C(N2CC(O)(C(C)NC(c3cnn[nH]3)=O)C2)=O)CC1 C=CC(C)(CCOC)C(=O)N1CC2CN(C(=O)Cc3cn(C)nc3Cl)CC2C1 c1(NOCC)cnc(C(C)C)nc1.C1CC(=O)N1.C12(CC1)N(C)C2=O c1(C(N2CC(C(C)NC(CCCCOC)=O)OCC2)=O)ccc2c(c1)C(=O)NC2 C1(CC(C)NC(C2(OCC)CCC2)=O)CCN(C(=O)CC(C)SC)CC1 n1(C(CC)(C)CC)cc(CNCCOC(c2cc(CCC3CC3)[nH]n2)=O)nn1 N1(C(Cc2c(SC)cccc2)=O)CC(NC(c2ccn(C)c(=O)c2)=O)CC(F)C1 C1(NC(C(C)=CC)=O)CC12CCN(C(C1(COC)CCC1)=O)CC2 N1(C(c2nc(C)sc2)=O)CCC(N(C)C(C2CC2(C)C)=O)C2(CC2)C1 N1(C(C=C(C)C(C)(C)C)=O)CC(F)(F)CC1(C)CNC(C1(F)CCC1)=O c1(C(N2C3CN(C(CC(COC)C)=O)C(C3)C2)=O)cc2c(F)ccc(Cl)c2[nH]1 CN1CC=C(CC(=O)N2CC(NC(c3cncs3)=O)CC23CCC3)CC1 N1(C(CC2CC(=C)C2)=O)CCC(OCCNC(=O)CC2CN(C)C2)C1 C1(CC)C(NC(c2c[n+]([O-])c(C)cn2)=O)CCCN1C(C1CCCCS1)=O c1(C(=O)NCC(C)CN(C)C(c2c[nH]c(=N)o2)=O)nccc2nn[nH]c12 C(=O)(C1CCCc2ccnn21)NCC1(CNC(c2c(C)noc2)=O)CC1 N1(C(CCC#C)=O)C2CCC1CN(C(C13CCC(CC1)C(C)O3)=O)C2 Cc1cc(C(=O)NCCCCC(C)NC(C2CNC(=O)CC2C)=O)cnc1F CCC(C)(CNC(C1CN(C(C2C3CCCCC23)=O)CC1F)=O)C(N)=O c1(C(=O)NCC2C(CNC(c3nc(C)oc3C)=O)C2)n[nH]c2c1CCSC2 N1(C(C2N(C)C(=O)OC2)=O)CCOCC(CNC(c2ccccc2CO)=O)C1 CC1(C)CCN(CC(=O)NC2CCCCC2CNC(=O)C(=O)NC2CC2)C1 C1(CC(=O)N(C2CCCN(C(C(C)(C)CF)=O)C2)CCF)CCOCC1(C)C CN=c1ccc(C(=O)NC2CC(C)N(C(c3cocc3C)=O)C2)c[nH]1 c1(CC)oc(C(N2CCC(CC)C2)C(=O)NC)cc1C(=O)OC.C1(C(=O)OC)CC1 C1(CC(=O)Nc2c(CC)nsc2)CC(C)(C)CN1C(=O)CCC1CC1(C)C N1(C(c2cnc(COCC)s2)=O)CC2(CCCC(CNC(C3CC3(F)F)=O)O2)C1 c1(C(N2C(CCCNC(C3CNC(=O)N3)=O)CCC2)=O)coc2c(Cl)cccc12 Cc1cnc2n1C(C)N(C(=O)Nc1ccc(F)cc1O)CC2 N1(C(C(n2ccc(C)n2)C)=O)CCCC(NC(=O)CC2CCC(=O)N2C)C1C C(=O)(CCCCN1C(=O)CCC1=O)NCC1C(NC(C(C)=CC2CC2)=O)C1 C1(CC(=O)NC)CCC2(CN(C(N3C(CO)CC4OCCC34)=O)C2)O1 c1(OC)cc(CNC(c2cccc(O)c2Cl)=O)c(OC)c2ccccc12 C(C(CO)C(F)(F)F)c1nc(-n2c(C)nc(C(F)(F)F)n2)[nH]n1.C(=O)O Cc1cc(C(=O)NOCC(=O)Nc2cc(=O)n(C)cn2)c[nH]c1=N c1(C(=O)NC2CC(SCC)C2)ccc(N2CCCC2)cc1.C12(CC1)C(=O)N2 C1(OC)CC2CC(C(N3CCN(CC(C)NC(c4coc(C)c4)=O)CC3)=O)CC12 CC1CN2CCN1C(C(=O)NCC1CC1CNC(C1CCC(=O)N1)=O)C2 c1(C(N2CC(COC)N(C(=O)C=CC3CCCC3)CC2)=O)nccc2cc[nH]c12 N1(C(C(C)NC(C)(C)C)=O)CC(O)(CNC(=O)C(C)C2CCCO2)C1 C=CCCCCC(=O)N1CCCC(F)(CNC(=O)C(C)C2CCCC2)C1 c1(CCNC(=O)OC(C)(C)C)ccc(Br)cc1F.CC1C(C(=O)NC)C1 O=C(C#CC1CCC1)OCC(=O)Nc1ccc(CC2(SC(F)(F)F)CC2)cc1 c1(CCCNC(NC(c2nc(N(C)C)n[nH]2)C)=S)cccc(Cl)c1 C(C(=O)NN(CNC(=O)OC(C)(C)C)CC(C)C)c1c(OC)cnc(Cl)c1 n1(C(F)(F)F)cc([N+](=O)[O-])c(=NC2C34CCC(C3)C24)[nH]1 CC(C)C(C)C(CNC(=O)Cc1cccnc1F)NC(=O)CCc1ccn(C)c1 Cc1nn(C)c(Cl)c1CC(=O)NCCC1CC(NC(C2(C)CC=CC2)=O)C1 CC(C)CC(C)C(=O)N(CC(C)(C)CNC(C1OCCCC1(C)C)=O)C C1(C(=O)Nc2ocnc2C(N2CC(OCCO)C2)=O)(OC)CC(C)(C)C1 C(C(=O)Nn1nnc2c1CCCC2)C1(N(C(c2cn(CC=C)nn2)=O)C)CC1 C(C(C)(C(=O)NCC(C)(C)CN(C(=O)CC=C(Cl)Cl)C)OC)OC N1(C(CC(CC)O)=O)CC2(CCN(C(c3cnn(CCO)c3)=O)C2)C1 c1(-c2cn(C3(NC(c4c(C)n(C)cn4)=O)CC3)nn2)cc2ccccc2[nH]1 c1(OC)cc(C(=O)NCC23CC2CN(C(C2(OC)CCSC2)=O)C3)cc(F)c1F n1(C(C)C)cc(C(=O)NC2CC(CNC(C3(F)CCC3)=O)C(O)C2)ccc1=O c1(C(=O)NCCC2CCN(C(C(CNC(C)=O)(C)C)=O)C2)cn2ccsc2n1 C1(CNC(Cn2c(C)cnc2)=O)CCC2(CCN(C(c3ccno3)=O)CC2)CO1 C1(SCC(=O)NCc2nccc(C3CC3)n2)CCC(C(C)(C)O)CC1 C1(C(N(CC)Cc2nnnn2C)=O)CCN(C(=O)CSc2ccccc2)CC1 c1(CNC(CC2N(C(C(C)Oc3ccccn3)=O)CC2)=O)ccccc1O N#Cc1ccc(F)c(C(N2CCC(NC(=O)C(F)n3cccn3)C(F)C2)=O)c1 N1(C(c2cccn(C)c2=O)=O)CC2(CCN(C(c3c(O)ccc(F)c3F)=O)C2)C1 c1(C(C)NC(C2(CNC(C(C)C)=O)CCC2)=O)cccnc1F CC1CN(C(=O)CC2CCCCN2C)CCN1C(=O)CNC(N)=O N1(C(Cc2ncc(CC)[nH]2)=O)CCN(C(=O)CCCCOC(C)C)C(C)C1C C1(CNC(C(C2CC2)SC)=O)CC2CCCC2N1C(=O)Cn1ccccc1=O c1(OC)nc(C)cc(C)c1CN(C)C(=O)C1CC1.C1(CN)CC(O)(CO)C1 c1(C(=O)NCC(CNC(C(CCOC)C)=O)O)cc(C)c(C)c(S(N)(=O)=O)c1 c1(N(c2nc3cc(Br)ccc3o2)C)ccnc(S(N)(=O)=O)c1 n1(COCC(C2(CNC(C3CC3C(=O)OC)=O)CC2)=O)cc(C(C)(C)OC)nn1 CC1CCCCN(C(c2ccc(C(F)(F)F)c(-n3cncn3)c2)=O)C1 Cc1ccn(CCC(=O)NCc2occc2C(=O)NCCC2CCN(C)C2)n1 N1(C(C2C(COC)C2)=O)CC(NC(C23CC(CO)(C2)OC3C)=O)CC2(CC2)C1 N1(C(c2c(CCC)nns2)=O)CCC(C2CN(C(C3(C)CCC(C)C3)=O)C2)CC1 N1(Cc2cnn(CC)c2C)CCn2ncc(SC)c2C1 c1(C(=O)NCC(CC)NC(c2cnc(SC)nc2)=O)ccc2ncccc2c1F Cc1ccc(C)n1CCC(=O)N1CC(OC2CCN(C(C3CC(O)C3)=O)CC2)C1 N#CC1(C(N2CC(Cn3cc(CN4CCCC4CO)nn3)C2)=O)CC12CCCC2 C#Cc1cc(C(=O)NCCOCCNC(=O)CSCC)ccc1Cl Cc1cc(C(N2CCN(C(C3CCN(C)C3=O)=O)CC2c2ncc[nH]2)=O)c(C)n1C c1(NC(C(C)N(C(c2cnc[nH]c2=N)=O)C2CC2)=O)ccc(CO)cc1 Cc1c(F)ccc(C(=O)NCC(C2CC2)NC(C2NC(=O)C3CC23)=O)c1N C(=O)(CCC(c1cccnc1)NC(=O)NOCCC1CC1)OC c1(C2(C)CC2)c(C(N2CC3C(NC(C4C(CC5CC5)C4(C)C)=O)C3C2)=O)cnn1C n1(CC(C)C)cc(CC(=O)NCC(O)CN(C(=O)C(F)C2CCC2)C)cn1 c1(CC(=O)NCCCCCNC(C2C3CCC2CC3)=O)ccc(Br)c(F)c1 C#CCCCCCC(=O)NCC(O)CC(=O)NC1CCC(O)C(O)C1 C1(C(=O)NCCC(C)N(CCC)C)CC=CC(NC(C2CC23CCC3)=O)C1 N1(C(C(CC#C)(C)C)=O)CC2CC(C1)N(C(c1cc(CC)c(N)cc1F)=O)C2 S(=O)(=O)(c1cc(OC(F)F)ccc1C)NC(c1cccc(C)c1)CO Cc1nc(C2CC(c3occc3C(N3CCC(c4cc(C)no4)C3)=O)C2)cs1 C1(C(=O)NCC2OCCN(C(C3(CCCC)CCCC3)=O)C2)CCCC(F)(F)C1 N1(CC2CCCN(c3c(OC)cccc3)C2)CCC(N=[N+]=[N-])(CO)C1 c1(CC(=O)NCC2C3CN(C(c4ccc(N)cc4F)=O)CC23)cc(F)cc(F)c1 C(=O)(C(C)CO)N1CC(OCCC(=O)N(C(C)CCO)C)C1 CCC(C)C(C(=O)NC(CCOC)C(=O)N1CC(CO)C1)NC(C)=O C1(N(C(CN(c2ccccc2)C(C)=O)=O)C)C2CN(C(c3cnc(Cl)[nH]3)=O)CC12 C1(C)(CC)CCC(C(=O)NC(C2CCCCC2)CNC(c2[nH]c(C)cc2C)=O)O1 C(=O)(C#CC1CCCO1)NCC(CNC(Cc1c(C)nn(C)c1C)=O)C C1(CN(C(C2CC(OCC)C2)=O)C)CN(C(c2ccnn2CC2CCC2)=O)CCO1 c1(C(N(CCC(C)NC(c2cnn(C)n2)=O)C)=O)ccc2nonc2c1 O=S(=O)(c1cnc[nH]1)N1CCC(C2CCCC2(F)F)C1 N1(C(C)C)CCC(CNC(=O)CNC(=O)C(C)NC(N)=O)C1 C1(NC(c2cc(C)no2)=O)CC2CCC1CN2C(=O)C(O)Cn1cncn1 c1(C(N2CCC(O)(c3cccc(F)c3)C2)C(=O)NCCC)cccn2ccnc12 N1(C(C(CCNC(c2c(CC)n[nH]c2)=O)O)=O)CC(CO)CC(C)(C)C1 c1(C(=O)OC)nc(NC(=O)NC23CC(C4CCS(=O)(=O)C4)(C2)C3)sc1C(F)(F)F c1(C(=O)NC(CCCNC(C(C(C)C)SC)=O)(C)C)cnc2n1CC(C)CC2 C(=O)(C1=C(C)N(C)c2nnnn2C1C)NCC1N(C(CCC=C)=O)CC2(CC2)C1 c1(C(=O)NCC2CCN(C(C3(COC)CCC3)=O)C2)c(C)noc1C1CC1 C1(C)(C(N2CCC(C(C#C)C)CC2)=O)CN(C(=O)C(O)C(C)CC)C(C)(C)C1 C(CO)(C(C)NC(=O)CCc1ccc(Cl)s1)NC(C1(CC)CC1)=O Cc1nc(CCC(=O)NCCC2(CNC(=O)CC(C)(C)F)CC2)oc1C CS(=O)(=O)CC(=O)NC1CN(C(C2CC2c2ccccc2)=O)C1 C1(CCC(=O)N(CC(C)(C)O)CC)CCCCN(C(=O)C(C)C(F)F)C1 C#CCCC(C(=O)N(C)CC1(O)CCC1)NC(C1CC1C(C)(C)C)=O C=CC(C)(CCOC)C(=O)N1CC2(CCN(C(C34COCC3C4)=O)C2)C1 C1(C(=O)NC23C(CN(C(c4ccc(C(C)C)o4)=O)C2)C3)CCc2n[nH]cc2C1 c1(NCC2(NC(=O)CP(C)(C)=O)C(C)CCCC2)ccc([N+](=O)[O-])cc1F C(=O)(C(C)(C)C1CCCO1)NCC(CC)NC(=O)Cc1ccnn1C1CCC1 C12(CNC(c3n(C)nnc3)=O)CC(NC(=O)C(F)=CC3CC3)(C1)C1(CCC1)O2 C12(CNC(=O)CNC(c3ccc(Br)c(Cl)c3)=O)CCCCC1C2(F)F c1(C(=O)NCC(C)N(C(c2onc(CC)n2)=O)C)ccc(F)cc1 C1(C(=O)NC2CCN(C(C3(C)CCCCC3)=O)CC2F)CCc2nnc(O)n2C1 C12(C(N3CC4(CN(C(C5CCC(=O)NC5)=O)C4)C3)=O)CCOC1CCOC2 c1(C(=O)NCCN(CC(C)O)C(c2cc(F)ccc2Cl)=O)cccn2cnnc12 C(N=C(NCc1cc2ncn(C)c2cc1)N1CCC(CF)C1)NCc1ccccc1 C1(C)(C(=O)NC2CC(C)(NC(Cc3c(C)noc3Cl)=O)C2)CCN(C)CC1 c1(C(=O)NC2C(CC)CN(C(C3CSC(C)=N3)=O)CC2)cc2nc(C)sc2[nH]1 C1(C(=O)NCC2C(C)CN(C(C3CCCC(F)(F)C3)=O)C2)CCCCCS1(=O)=O N1(C(c2c(C)scc2)=O)CC(O)(C2(CNC(C34CCOC3CCOC4)=O)CC2)C1 c1(C(=O)NCC(CNC(C(N)=O)=O)CO)ccc(CC2CC(=O)NC2=O)cc1 N1(C(C2(C)CC(=C)C2)=O)CCC(C2(NC(=O)C(N3CCSCC3)C)CC2)C1 C1(C(N(CC=C)C)=O)(OC)CCN(C2CN(C)CC2O)CC1 C1(CNC(c2conc2CNC(C2CC3CC3C2)=O)=O)CC12CCCCC2 c1(CC(=O)N(C(CNC(c2c(CC)[nH]cc2)=O)C2CC2)C)ccc(C(C)=O)cc1 CCCCC(C(=O)NCCn1cc(C(N2CC(N3CCCCC3C)C2)=O)nn1)OC c1(C(N)=O)ccn(CC(=O)NC2(C)CC(NC(=O)Cc3cn(C4CC4)cn3)C2)n1 N1(C(c2c(C)c[nH]n2)=O)CCC(CO)C(NC(=O)C(N2CCSCC2)C)C1 CCC(CC)(C(=O)NCC1CC(NC(=O)CCn2ccnn2)C1(C)C)OC N12CCSCC1C2=O.C(=O)(CCCSc1ccccc1)OCC(C)C C(=O)(C(C)(C)CC(F)(F)F)NC(CC)(CNC(=O)C(C(C)(C)C)N(C)C)CC C1(CNC(C2CC(C)(CNC(CCCC3C(C)C3)=O)C2)=O)COCCN1C CC1(C)CC(NC(=O)CC2(O)CCCCC2)CN(C(c2cccc(Cl)c2F)=O)C1 c1(SC(c2noc(Cc3ccccc3)n2)C)nc(O)c2c(C3CC3)csc2n1 C(C(CC(C)C)NC(=O)CC(C)(C)O)NC(c1c(CC)noc1)=O Cc1cc(C#N)cnc1C(=O)NCC1CCCCN1C(c1nc2cccnc2s1)=O CC1(CC(=O)NCC2(NC(c3cc(C(C)(C)C)c[nH]3)=O)CCCC2)CCCO1 c1(C(N2CCC(C(=O)NC(CCC)CO)C2)=O)ccc(C)c(O)n1 N1(CCN(C(=O)CC2CC2(Cl)Cl)C)CCN(C(=O)C(c2cccnc2)C)CC1 N1(C(C=Cc2n(CC)ncc2)=O)CCCC(CCC)(NC(=O)Cc2cc[nH]c2)C1 C#Cc1ccc(C(=O)NC(C2CN(C(=O)CCSCC)CCO2)C)c(C)c1 c1(CCC(=O)NC(C(C)N(CC)CC)=O)cccc(N(C)C(C)=O)c1.C(C)(C)(C)O C1(NC(C(C)=CC)=O)CC2CN(C(c3c(C)noc3C(F)F)=O)CC2C1 C1(NC(c2c(C)nc(CC)o2)=O)CCN(C(c2cnc(C)n2C)=O)C12CCC2 N1(CCN(C(=O)C(CCO)=C(C)C)C(C)C)CCC(C(N2CCCC2SCC)=O)C1 c1(-c2occ(C(N3C(C(=O)OCC)CC3C)=O)n2)ccccc1F Cc1cncc(C(N2CC3CC2C3)C(=O)NC2COC2)n1 N1(C(Cc2c(OC)ccc(C)c2)=O)CCC2(CCCC2NC(c2ccon2)=O)C1 N1(C(C2CC2NC(=O)C(CC(F)F)c2ccc(F)cc2)=O)CC2(CCC2)C1.CC c1(C(N2CCNC(CO)C2)=O)cc(C(N2CC(N3CCCC3=O)C2)=O)nc(Cl)c1 c1(OC)ccc2nc(C)c(C(=O)NC3C4CN(C(=O)CCC5CC5)CC34)n2n1 C1(C(=O)NNC(=O)C2SCCS2)(OC(=O)NCC)CCCCC1 C1(NC(c2c(F)ccc(C)c2)=O)CC2CC1CN(C(=O)CCSC(F)(F)F)C2 N1(C(C(C)(C)NC(=O)OC)=O)CC2C(C(=O)NC(C)Cc3cc(C)no3)C2C1 C(=O)(C(C)(C)C(=O)NCCN(CC(C)O)C(=O)COC1(C)CCCC1)NC c1(C(N2C(CCC#C)CCC2)=O)ccc(Cc2ncccn2)nc1 C=C(CNC(c1cccn1-c1ccccc1)=O)CCNC(c1ccncn1)=O N1(C(C(CCC=C)NC(=O)CC(=O)OCC)=O)CCCN(C)C(=O)C1 CC1CN(C(=O)CC2CC3CC3C2)C(C)CN1C(c1cc(O)ccc1Cl)=O c1(N2C(CNC(c3c(CC)c[nH]c3)=O)CCC(C)(C)C2)nc2ncc(Cl)cc2o1 CC1CCC(C(=O)NCCC(C)(C)NC(c2ccc(-c3ccco3)s2)=O)C1 N1(C(c2ccc(Br)c(F)c2)C(=O)NC2CCCCC2)CCn2ncnc2C1 C1(C(=O)NCC2CC(NC(C3CCN(C(CC)=O)C3)=O)C2)CCc2nc[nH]c2C1 Cc1nc(N)cnc1C(=O)N(C)CCNC(=O)CSc1cccc(Br)c1 c1(C(=O)NCC2C(NC(CN(C)C(=O)C3CC3)=O)C2)cn(C2CCCC2)nn1 c1(C(=O)NC(CN(C(c2cc(Cl)ns2)=O)CC)C)cncc(O)c1Cl C1(C#N)(C(=O)NC2CC(NC(c3ncn(CC)c3)=O)C2)CC2CCC1C2 c1(C(=O)OC)cccc([N+](=O)[O-])c1NCC1CC(NC(=O)Cc2cc[nH]n2)C1 c1(OC)nc(C(N2CC3C(NC(C4(CO)CCC(=O)N4)=O)C3C2)=O)sc1C N1(C(CCc2cnc(C)s2)=O)CC2(CC(NC(=O)C(C)(C)F)CO2)C1 c1(C(=O)NCC2CCN(C(COC)=O)CC2C)ccc2c(c1)C(=O)CCS2 CC(CCNC(C1CCOC(C2CC2)C1)=O)N=c1[nH]cnc2cnccc12 N1(C(c2cc(OC)n[nH]2)=O)CC(CNC(C2CC(=C3CC3)C2)=O)N2CCC1C2 Cc1cc(C(c2nnnn2C)Nc2ccc(-c3cnn[nH]3)cc2)cc(C)c1 c1(-n2cc(CN(C(C(CCC)F)=O)C)nn2)ccc(OC)cc1OC C1(NC(c2c(CC)nns2)=O)CCC2(CC1)CC2NC(C1CCCN(CC)C1)=O C1(CNC(C2CCCC2)=O)C2CN(C(c3ncc(C(F)F)s3)=O)CC12 CCCC(O)(CCC)CC(=O)NCC1(OC)CCN(C(=O)C(O)C(C)(C)C)C1 c1(C(=O)NCC2C(CNC(c3csc(C)c3N)=O)C2)cc2ccnc(Cl)c2s1 c1(OC)ncc(CNC(=O)CCn2cc(-c3cnccc3Cl)nn2)cc1C C(=O)(CCCCC(C)CC)NC1(CC=C)CN(C(C2CC2(Cl)Cl)=O)C1 Cc1ccc(C(=O)NC(C2CC(C)(C)C2)CO)c2ccccc12 N1(C(C2CCCC=C2Br)=O)CC(F)(F)CC1Cc1cn(CC(O)C(F)(F)F)nn1 c1(C(=O)NCCC2CCN(C(=O)C(F)F)C2)nncc2ccccc12 N1(CC)CCCN(C(=O)C(C(C)OC)NC(=O)C(C2CC2)OC)CC1 C#CCC(C)(C(=O)NC(CCO)C(C)(C)C)NC(c1[nH]cnc1C)=O C(=O)(C(O)C(C)CC)NC(c1cc(F)cc(Cl)c1)CNC(CC=CC)=O C12(C(=O)NC3CCC(CNC(c4c(C)nsc4N)=O)C3)CCCCC1C2(F)F n1(COC)nccc1C(N1CCC1C(=O)NCc1cnc[nH]1)=O C1(CC=C)(NCC(=O)NCc2nc(C)cs2)CN(C(=O)C(=C2CCCCC2)F)C1 C(=O)(C(CC(F)F)NC(c1nnn(C)c1N)=O)NCc1cncc(CC)c1 C=CC(C)(C)CC(=O)NC1CN(C(=O)C(c2cc(Cl)ccc2Cl)(F)F)CC1(C)C CC(CCNC(C1(NC(c2csc(=N)[nH]2)=O)CCCC1)=O)C(F)(F)F N1(C(C2N(CC)CCOC2)=O)CCC2C(C(=O)NC3CCCC3F)C2C1 c1(C(C(=O)NC2(CNC(C3(C4CC4)CC3)=O)CCOC2)=O)ccc(F)c(Cl)c1F C1(C(=O)NC2CCC(CNC(Cc3cn(C)nc3)=O)C2)CCC(=O)NC1 c1(OC)ccc(F)cc1CC(=O)NCC1(C(C)NC(C2(C)CC(C)=NO2)=O)CC1 c1(C(N2CC(O)(CNC(c3c(C#N)cn[nH]3)=O)C2)=O)ncnc(O)c1Cl c1(CC(C(N(Cc2cn(C(CC)C)nn2)O)=O)=O)ccc(-n2ccnc2)cc1.OC Cc1cc(C(N2CCN(C(=O)C=C3CCSCC3)CC2CCO)=O)c(C)cn1 N1(C(C(C)OCCC(C)C)=O)CCC(C2CC2)(CNC(c2cnns2)=O)C1 N1(C(C2C(OCC)C2)=O)CCC2(CC1)CN(C(c1cnc(O)c(C)c1)=O)CCO2 CC#CCCCC(=O)NC1CCC(C)N(C(c2ccc(C(C)(C)C#N)cc2)=O)C1 N1(C(CSC)=O)CCC(CO)C(NC(=O)CCOc2ccc(Cl)cc2Cl)C1 C1(C(C)C)(C(=O)N(CC(C)OC)C)CCN(C(=O)C(C)OCc2ccncc2)C1 Cc1nc(C(N2CCC(NC(=O)CC3CC(C)C3)C(O)C2)=O)ccc1[N+](=O)[O-] C1(OC)CCCCCC1NC(=O)C(F)C1CC(NC(=O)COC(C)C)C1 c1(C(=O)NC(C2N(C(CCC(=O)OC)=O)CCC2)C)coc2cc(C)c(C)cc12 CP(C)(=O)c1ccc(C(N2CCCC2CNC(=O)C2=COCCO2)=O)s1 C1(C(=O)NCc2n(CCC)ccn2)CCC(O)CN1C(C1CC2(CC2)CN1C)=O N1(C(=O)Nc2scc(C(=O)OCC)n2)CCC(C)(F)C1 c1(CC)ccc(C(N2CC(CNC(c3ccoc3C(F)(F)F)=O)C2)=O)c(C)n1 CC(C)CC(C)C(=O)NCCN1CCCN(C(=O)C=Cc2cscn2)CC1 Cc1c2cccc1C(=O)O2.C1(N(C(C)C)CC2CC2)(C(C)C)CCCN1 c1(N2C(CNC(C#CC)=O)CCC2)ncc2ccccc2n1 c1(CNC2(c3nnnn3CCCF)CC(CC)C2)cc(OC)c(C)cc1C c1(C(N2CC(C)CC(NC(c3c(C)nsc3)=O)C2)=O)cc(C)nc2[nH]nc(O)c12 C=CC1(C(=O)N(CC(C)O)CCNC(=O)CSc2c(C)n[nH]c2C)CCOCC1 N1(C(CC2C(C)C2)=O)CC2(CCC(CNC(=O)CC(=O)NCc3nccs3)O2)C1 C1(OC)CN2CC1C2=O.C1(NC(=O)C=Cc2ccnn2C)C2(CC2)C12CC2 N1(NC(N2C(Cc3ccc(OC)c(OC)c3)CC2)=O)CCC2(O)CCCCC2C1 N1(C(C2C(C(N)=O)C2)=O)CCN(C(C2(CF)COC2)=O)CC1C1CCCC1 c1(C(N2C3CC(NC(C4CCC(CC)CC4)=O)C2CC3)=O)cc2ncccc2o1 c1(C(=O)NCC2CCCCN(C(COCC=C)=O)C2)nccn2cc(C)nc12 C1(CNC(=O)C(N2CCCCC2C2(O)CCC2)=O)CCc2ccccc2C1 Cc1ccc(-c2ccc(-c3cnccn3)cc2)cc1N c1(C(C(=O)N(CC(C)NC(=O)CCc2ccoc2)C)(C)O)ccc(Cl)cc1 CCCCS(=O)(=O)Cc1noc(Oc2ccc(C(F)(F)F)cn2)n1 C1(NC(c2ncc(C)c(Cl)c2)=O)CC2CCC(C1)N2C(=O)CC1CCCCO1 C(C(=O)NCCC1CCC(=O)N1)(C(C)C)NC(C(C)NC(COC)=O)=O C1(C#N)(CS(=O)(=O)Nc2ccc(NC(C3CCC(C)C3)=O)nc2)CCOCC1 N1(C(C(CC)C)=O)CCN(C(c2cncc(C(N)=O)c2)=O)C(CCOC)C1 CC1CN(C(=O)Cc2ccc(F)cc2F)CCCN1C(C1(C)C=CCC1)=O C1(CCNC(C(C)OC2COC2)=O)CCC2(CN(C(=O)CC3=CCCCC3)C2)O1 C(C)(CC(=O)NCCc1nccn1C)NC(CC=C(C)C)=O C(=O)(CCC(O)C(C)(C)C)N1C(CNC(C2CC(C)OC2C)=O)CCC(C)C1 N1(C(C(C)NS(CCC)(=O)=O)=O)CCc2cc(C(N)=O)ccc2C1 CCCCCS(=O)(=O)CC(=O)N1CCN(C(C2CCCC2)=O)C(C)C1C N1(C(C2C(C)(C)C(NC(c3ccc(=N)[nH]c3)=O)C2)=O)CC2(CC=CC2)C1 N1(C(C23C(CN(C(C4(CCC)CCC4)=O)C2)C3)=O)CC(=O)NC(=O)C1C C1(CN(C(=O)CC2(C)CC2(F)F)C)CCC(NC(=O)C(=C2CCCCC2)F)CC1 c1(N2CCC(C)(COC)C2)nc(=NCC2(CO)CC(C)(C)C2)[nH]c2c1CCCC2 Cc1cc(CC(=O)NC2(C(=O)NOCC(C)(C)C)CCSC2)cc(F)c1 C(C(C)(C)CC(=O)NC1CCCN(Cc2ccccc2Cl)C1C)OC C(C(CC(C)C)NC(C12CC(F)(C1)C2)=O)NC(C(C)NC(C)=O)=O Cc1ccc(C)c(CC(N2CCCCC(NC(c3sccc3C)=O)C2)=O)c1 N1(C(c2cc(CC)[nH]n2)=O)CCCC(C2CN(c3nc(C)ns3)C2)C1 C1(NC(Cn2ncc(C)c2)=O)C2CC1CN(C(c1ccc(CO)s1)=O)C2 c1(C(N2CC(OC)C(NC(=O)CCNC(N)=O)C2)=O)cc2c(C)cccc2[nH]1 N#Cc1ccc(S(=O)(=O)N2CC3CC2C3C(N2C3CCC2CNC3)=O)cn1 C1(C(=O)NCC(CC)NC(=O)C(N2CCN(C)CC2)(C)C)CC(C)OC1=O C(=O)(C(C)(C)CC(=O)NC1COCC1NC(c1c(C(=O)OC)cco1)=O)OC c1(NC(C2N(C(c3c(OC)ccnc3)=O)CSC2)=O)cnc2ccnn2c1 c1(C(C)NC(c2n(CC=C)nnn2)C2(n3ccnn3)CC2)c(F)ccc(C)c1F C1(C(N(CCC(=O)NC(CC(=O)OCC)C)C)=O)CCCCC1(C)C C#CC1(C(=O)N(C)Cc2cc(C)nn2C)CN(C(=O)CC2CCN(C)C2=O)C1 C1(C(=O)NC2(CNC(C3(OC)CCCCCC3)=O)CCC2)CCCC2(CCC2)C1 C1(NC(CCCc2onc(C)n2)=O)C2CC1N(C(c1cc[nH]c1C)=O)C2C CN=c1cc(C(=O)N(C)CC2CCCCN2C(=O)CC(C)(C)F)cc[nH]1 CC1CCC(CNC(=O)N(C2CC2)CC2CCOC2)Cc2ccccc21 CCCCCC(F)C(=O)NCC(C1CC1)NC(c1cc2cccnn2n1)=O C=C1CCN(C(=O)CCCCC2CC2)C(C(=O)NCC2CCC2CO)C1 c1(CC(C)C(=O)N2CC(NC(C3(C)CCNC3=O)=O)C2)ccc(F)c(F)c1 CCCC(CNC(C1CC(=O)C1(C)C)=O)C(=O)NC1CCCC1N=[N+]=[N-] c1(OCC(=O)NCCC(CNC(CC(=C=C)C)=O)O)cc(C)ccc1F c1(CC)ccc(C(=O)NC2(CCNC(C3CC(CF)C3)=O)CC2)cc1 C1(N(CC)CC)CCCC1(C)C(=O)NNC(=O)C1CCOC(c2ccncc2)C1 C(CC(CC)C(=O)NC1CCCC1C(N1CC2CCC2(C(=O)OC)C1)=O)=CC Cc1ocnc1CC(=O)NCC1CCC1C(=O)NCCS(N)(=O)=O Cn1cnc(C(N2CC3CC2C3NC(c2ccc(C3CCC3)cc2)=O)=O)cc1=O c1(OC)cccc(C(=O)NC2CCC(N(C(=O)CC3COCCN3C)C)C2)c1O c1(C(N2C3(CN(C(c4c(OC)cccc4C)=O)C3)CC2)=O)ccc(F)c(C)c1N C1(F)(CC)CCN(c2nnc(-c3ccc(C)s3)n2Cc2ncnn2CCF)CC1 CC(CC(=O)NCCCOCCC(N1CCC2(CCCN2)C1)=O)C(F)F C(CCN=c1[nH]c2c(cc1C#N)CN(C)CC2)NC(C(C)OCCOCC)=O C(C(=O)N(C(C)C(C)(C)C)CC)(C(C)C)NC(c1ncn(CC)c1)=O C1(CC)(NC(=O)CCOC)CCN(C(C2CCC(C)NC2=O)=O)CC1 C12(NC(C)=O)COCCC1CN(C(=O)CCc1nnc(-c3ccsc3)o1)C2 c1(C(=O)NCc2nc(CNC(C=CCOC)=O)sc2)cccn2nccc12 C1(NC(=O)C=CCOCC(F)(F)F)C2CN(C(c3cscn3)=O)CC12 N1(C(c2c(C)ncnc2)=O)CCC(N=c2[nH]c3ncc(Cl)cc3s2)C1 C1(NC(C2CC(O)C2)=O)CN(C(c2cn3c(n2)CCCC3)=O)C2(CCC2)C1 CC(C)(C)C(C(=O)N1CCOCC1c1cccnc1)C(F)(F)F C1(C(N2C(C)(C)CC(CNC(=O)CC#N)C2)=O)CC2CCCCCC12 C(=O)(C(C)C(C)(C)C)NC12CC(NC(c3c(SC(C)C)cccc3)=O)(C1)C2 N1(C(CC)=O)Cc2nccn2CC(NC(c2c(C)cc(OC)cc2F)=O)C1 Cc1nn(C)c(=O)c(C(N2CCN(CCNC(=O)CC34CC(C3)C4)CC2)=O)c1C Fc1ccc2c(c1F)CN(C1CC1c1ccccc1C1CCCCC1)C2 C1(CC(=O)NCC(CC=C)NC(=O)CCSC)CC(=O)c2ccccc2C1 N1(C(CC2CC(CC)C2)=O)CC2(CNC(C3CCCS3)=O)CCC1C2 c1(OCC)ccc2c(CC(=O)N(C(=O)COc3cn[nH]c3)C)coc2c1 c1(C(N(CCNC(c2c(OC)ccnc2)=O)CC2CC2)=O)ccc(OC)cc1F O=C(CC(F)(F)C(F)F)N1CCC(NC(C2(C3CCC3)CC2)=O)C(F)C1 c1(OC(C)C)ccc(C(=O)NCCCC(C)(C)NC(c2cccnc2)=O)cc1 Cc1cc(C(N2CCN(C)C(CNC(=O)Cn3cnnc3O)C2)=O)ncc1N C(=O)(C(F)C(C)(C)O)NC(CO)C(C)(C)C.C12(CCOCC1)N(C)C2=O C1(C)(CN(C(Cn2c(C)ncc2)=O)C)CCCC1NC(c1cncs1)=O Cn1cc(Cl)c(C(=O)NC(CO)C(=O)NCC2CC(C)(O)C2)n1 Cc1ccc(C(CNC(=O)CCc2cccc(C)n2)NC(=O)C#CC2CC2)cc1 N1(CCNC(CC2C(CC)C2)=O)CCN(C(c2coc(C(F)F)n2)=O)CC1 Cc1nn(C(C)(C)C)c(C)c1C(=O)NCCC=CC(C)C C1(C2CCCN(C(C3(CC(F)F)CCC3)=O)C2)(NC(C(F)OC)=O)CC1 N1(C(C2(OC)CCSCC2)=O)CC2(CCC2NC(c2ccc(Cl)cc2)=O)C1 C1(NC(C2CCOC2C2CC2)=O)CN(C(C2(c3ccccc3)CC2)=O)CCC1F C1(S(N)(=O)=O)(C(N(CCNC(CC2(C(=C)F)CCC2)=O)C2CC2)=O)CCC1 CN(C)S(=O)(=O)N1CCC(CC2CCCCC2)=C(F)C1 C1(N(C(C2CN(C(C)C)C2)=O)C)CC2CCC(C1)N2C(C1CCC2CC12)=O C1(CC(=O)N(CCN(C(CCC=C)=O)C)C)Cc2ccccc2C1=O N1(C(C)=O)C(C)CCCC1C.CC1CNCCC1CCNC=O c1(C(CO)NC(C(C)(C)NC(c2nc(CCC)oc2)=O)=O)ccc(C)cc1 c1(C(=O)NCC23OCC(NC(c4c(C)cns4)=O)(C2)C3)cc2c(O)cccc2[nH]1 N1(C(c2c(CC)noc2)=O)CC2CC(C(N3CCC(O)(C(C)C)C3)=O)C(C2)C1 C#CCC(C(=O)N1CC(CCCCC)C1)NC(=O)C(C)OCC Cc1cc(O)c(F)cc1NC(C1(C2CC2)CN(C(c2cc(C3CC3)on2)=O)C1)=O c1(CCNC(N2CC(c3n(CC)cnn3)C2)=O)csc2ccc(F)cc12 C(CO)(CC(F)(F)F)NC(CC1(OC)CN(C(=O)Cc2cnc(C)s2)C1)=O C1(C(C)N)CC2C=CC1C2.c1(NC(N(CCOC)CC)=O)ccsc1 C(=O)(C(O)CC(F)(F)F)N1CCC2C(C(N3CCC(OCC4CC4)C3)=O)C2C1 c1(C(=O)NC(C(N2C(COC)C=CC2)=O)CC2CC2)ccc(C#N)cn1 c1(C(N2C(CNC(CC(C)OC)=O)CC(C)(C)C2)=O)nnn2c1C(=O)NCC2 N1(CC=C)CCc2ccc(NC(=O)CCCC(F)(F)F)cc2C1 Cc1nocc1C(=O)N(C(C)C(=O)NCCCC(F)F)C1CC1 C(CS(=O)(=O)N=S(C)(C)=O)NC(C(C)CCCO)c1nnnn1C c1(C(C)C)nocc1C(=O)NC(Cc1cc[nH]n1)C(=O)NCCCc1nccs1 c1(C(N2CCN(C(CC(C)CF)=O)C(C3CCC3)C2)=O)nc2ccccn2c1F N1(C(C2N(CC)CCC2)=O)CCC2(CCCCC2NC(=O)C=CC=C(Cl)Cl)CC1 N1(C(CC2C=NN(C)C2=O)=O)CC2(CC(C(=O)NCC3CCC3CO)CO2)C1.OCSC C=CC1(C(=O)NCC2CCC2CO)CCN(C(=O)CS(=O)(=O)NCC)C1 C1(C)(CNC(C2(OC)CCCC2)=O)CCN1C=O.C1(CCC)(CF)CC1 N1(C(C2N(C)C(=O)NC2)=O)C2CCC1CC(N(C)C(c1cccs1)=O)C2 N1(C(C=CSC)=O)CCC(C2CCN(C(C3CN4CCC3(C)CC4)=O)CC2)C1 c1(C(N2CC(CNC(C3COCCOC3)=O)C(C(F)(F)F)C2)=O)ncc[nH]c1=O N1(C(C(COCC)C)=O)CCCC(CCC(=O)NCCc2ccn(CC)n2)C1 Cc1nc(N2CCOCC(CNC(=O)CCC3CCCO3)C2)cc(C#N)n1 N1(C(=O)CN2CCCCC2)CCN(CC(=O)NC2CCC3(CC3)C2)CC1 C1(OC)(CC(C)C)CCN(N2CCC(c3cc(O)n[nH]3)CC2)C1 N1(C(CNC(=O)C(C)(C)CC)C2(CC=C)CC2)CCCC(C)(C(N)=O)C1 N1(C(C)=O)CCN(C(C2C3CC4C(C3)C24)=O)C(C)C1.c12n[nH]cc1SCC(=O)N2 N1(C(COc2ccn(C)n2)=O)CC2(CCCN(C(=O)C(O)C3CCC3)C2)C1 C1(NC(C(C)OCCC=C)=O)CN(C(c2snnc2C)=O)CC12CC2 C1(CC)CN(C(=O)C(C)(C)CNC(C2(C)CCOC2)=O)CCN1C c1(CC(=O)NC2CCCCC2NC(c2cc(C3CC3)on2)=O)c(F)cccc1F C1(CNC(C2CC(O)(CNC(COc3cc(C)on3)=O)C2)=O)CC12CCOCC2 C1(C2(O)CCC2)(C(=O)NCC(CC(C)C)NC(C(CC)N2CCCC2=O)=O)CC1 Cc1cc(O)c(Cl)cc1C(=O)NCC1(NC(=O)C(O)C2CCCC2)CCCC1 CC1CC(NCc2cc(OCCCCl)ccc2Br)c2ncnn21 Nc1c(C(=O)NCCC2CCN(C(=O)C(F)=CC3CC3)C2)cnc2ccnn12 C1(CC(=O)NCc2ccc(CC)s2)N(C(=O)CCc2cccnc2)CCC1(C)C c1(C(C(=O)NCCCOC)N(C)Cc2ccccc2)cc(OC(F)F)cc(C)c1 C(=O)(C(C)CC(C)(F)F)N1CCC(N(C(c2c(C)nn(C3CC3)c2Cl)=O)CC)C1 N(C(=NC)N1CCC(C)(C#N)CC1)Cc1cc(OC)c(OC(F)F)cc1 N1(C(c2cnn3c2N(C)CC3)=O)CC2CCCC2C1C(N1CCOC2C(O)CC12)=O N1(C(CNC(=O)CC2CCCC2)=O)CC2(CCCC2NC(=O)CC23CCCC2C3)C1 C(=O)(CCCCCNC(C1CCCC1C1CC1)=O)N(C)Cc1nncs1 C1CCCC(=O)NOC2CCCN1C2.Cc1ccnc(NC(C23CC(CO)(C2)C3)=O)c1N c1(NC(C(C)NS(c2c(C)noc2C)(=O)=O)=O)ccc2c(c1)CCOC2 N1(C(c2nncc(CCC)c2)=O)CC(O)CCC1C(=O)NCc1nc(N(C)C)n[nH]1 c1(OC)cc(C(=O)NC(C)CN(C)C(c2ccc(Cl)cc2C)=O)cc(Cl)c1OC c1(C(N2CCC(OC)(CNC(C3CNC(=O)C3)=O)C2)=O)ccnc(Cl)c1O c1(OC)ncc(C(=O)NCC(CC2CC2)C(=O)NCC(N2CCCCC2)C)cn1 S(=O)(=O)(c1ccc(C(N2CCCC2c2nncn2CC2CC2)=O)cc1)NCC CCCC(C(=O)OC)C(=O)Nc1ccc(NC(=O)CC2(OCC)CC2)cc1C C#Cc1nc(C(=O)NC2CC(CNC(c3cscc3Br)=O)C2)cs1 c1(C(N2CC(C(C)NC(C(C(C)C)OC)=O)C2)=O)c(F)c(C)cc(N)c1F c1(C(N(CCCCCCNC(C2CC(SC)C2)=O)C)=O)ccc(C#N)cc1O CC1CN(C(=O)Cc2ccncc2Cl)CC(C)CN1C(c1cscc1F)=O C(N=c1[nH]c2cc(F)ccc2o1)C1(C)CN(C(C(CC)C2CCC(=O)N2)=O)C1 C1(C(=O)NC(C2CCCC2)CNC(Cc2nc(COC)sc2)=O)CCC2CC1CO2 N1(C(c2nc(OC)c(C)s2)=O)CCCC1C1CCCCN1C(=O)Cc1cnc[nH]1 n1(C(C)C(=O)NCc2ccc(F)cc2[N+](=O)[O-])cnc2c(N)ncnc12 c1(C(=O)NC2C(CNC(C3(CC#C)CC3)=O)C2)ccccc1Cc1ccccc1 c1(C(=O)NC2CC3C(NC(C4C(C)(C)COCC4)=O)C3C2)cc2cccnc2[nH]1 Cc1cc(C(C)C(=O)NCC(CNC(=O)CSC(=O)N(C)C)N(C)C)c(C)o1 N1(C(CN(C)C)=O)CCN(C(=O)COCC2CCOC2)CC1c1ccccc1Cl c1(NCC(C)(O)CO)ccc(S(=O)(=O)NC2CCCC=C2Br)cc1Cl C1(C)(CNC(C2CC(C)OCC2)=O)CC2(CC(O)C2)C1 C(CC(=O)NCC(O)CN(C)C(C1CC1C(C)C)=O)SC Cc1cc(O)ccc1C(=O)NCC(C)(C)CNC(c1c(Br)nnn1C)=O C12(NC(C3(C)CN(C(c4ccccc4NC(N)=O)=O)C3)=O)OCCCC1C2(F)F C(N=c1[nH]c(N(CC(Cl)Cl)C)nc2cc[nH]c12)c1c(C)nc(CC)o1 C1(CC(N2CCC(NC(CC(CC)O)=O)CC2)=O)CCC(=O)NC1=O Cc1cncc(C(=O)NCC23CC(NC(=O)CC4CCC(C)C4)(CO2)C3)c1Cl c1(OC)ccc(C(=O)NCCC2CN(C(C3(F)CCOC3)=O)CCO2)cc1F N1(C(c2cc(C)[nH]n2)=O)CC2(CCN2C(C2CCCN2Cc2ccccn2)=O)C1 C1(CC(=O)NCC(C)CNC(=O)CNc2cccs2)OCCC1(C)C Cn1nc(O)cc1C(N1CCC(n2cc(-c3c[nH]nc3CO)nn2)C1)=O CC1CC(C(=O)NCCCc2cn(C)cn2)N(C(c2ccco2)=O)C1 C12(C(=O)NCC(c3ncc[nH]3)C)CCC(CC1NC(=O)Cc1ccnn1C)C2 S(=O)(=O)(c1ccc(NCc2cn(C3CC3)nn2)c(F)c1)NC(CC(=O)NC)C Cc1nnc(CCC(=O)N2CC(CNC(C3(C)CC3F)=O)C2)n1C CC1(C2CCCN(C(C3CCC(O)CN3C(=O)C(N)=O)=O)C2)CC1 C1(C)(NC(C(c2cccnc2F)(C)C)=O)CCCN(C(C2(CC(F)F)CC2)=O)C1 CC(O)(CC(=O)NC1(CNC(=O)C(=Cc2cscn2)F)CCOCC1)C1CC1 c1(C(=O)NCC(C)NC(c2c(C)ncn2C)=O)ccc(-c2cccs2)cc1F N#Cc1cc(=NC(=O)N2CC(C3CC3)(Cc3ccccc3)C2)[nH][nH]1 Cc1cc(C)c(C(N2CCN(C(c3cc4n(n3)CC(F)C4)=O)CC2C)=O)c(C)c1 CCCCC(O)C(=O)N(CCCOCCN(C(=O)CC1(C)CC(F)(F)C1)C)C c12[nH]c(cc1Br)CNC2=O.C1(CC)(Cc2ccccc2)CCOC1 c1(CCC(N2CC(C(C(=O)N(CC)CC)C)C2)=O)cn(C)cn1 c1(C(=O)NC2C=CC(C(=O)NCc3ncc(Cl)cn3)C2)cc(O)cc(O)c1 C1(NC(C2N(C(CN3CCC(OC)C3)=O)CCOC2)=O)CCCCC1N=[N+]=[N-] C1(NC(CSCC)=O)C=CC(C(=O)N(C(CO)C(C)C)C)C1 c1(C(N2C3CC(CNC(=O)Cc4cc[nH]n4)(OC3)C2)=O)cc(F)c(Cl)cc1Cl N1(c2n(CCOCC=C)c(C(c3ccc(C)cc3)O)nn2)CCC(C2CCC2)C1 c1(CC(=O)Nc2nc(C3CC3)cs2)nccc(Br)c1Br c1(C(N2CCC(CNC(c3nc(C)[nH]n3)=O)C2)=O)cc(Br)c(C)cc1F c1(C(N(Cc2n(C)c(O)nn2)CC2NC(=O)CC2(C)C)=O)c2ccccc2nn1C S(=O)(=O)(c1cccnc1)N1CCC(CC(=O)Nc2cccc(C#C)n2)C1 Cc1cc(F)ccc1C(=O)N(CCCCC(=O)NC(CO)C1CCC1)C CCCCC(O)C(C)C(=O)NC(CC=CC)C(=O)N1CC(C(C)CC)C1 n1(CC=C)cc(C(=O)N(CCCN(C)C(c2ccoc2C)=O)C)cn1 C#Cc1cccc(C(=O)NCC2CCN(C(=O)CC3(OC)CC3)CC2C)c1Cl Cc1sncc1C(=O)N(CCNC(=O)C(N1CCNC1=O)C)CC1CC1 Cc1ccc(N(C(C2CN(C(=O)Nc3ncc(C)cn3)C2)=O)C(C)C)cc1 C1(C(=O)NCCc2cnc(NC(=O)CCOCc3ccco3)s2)CCC2(CC2)C1 Cc1c(Cl)ccc(C(=O)NCC2(O)CN(C(c3cc(CO)ccc3Cl)=O)C2)c1N C(C)(CCCCN=c1ncc(F)c[nH]1)NC(c1cccc(C(C)(F)F)n1)=O C(C)(C)(CC(=O)N1CCCC1(C)CNC(c1ccn(-c2ccc(F)cc2)n1)=O)OC Cc1cc(Cl)c(N(C2CCCNC2=O)C(=O)CCC2CCC(O)CC2)cc1C C1(NC(=O)COc2cncc(Cl)n2)CCCCC12CCCN(C(c1ccoc1)=O)C2 N1(C(C2C(C=C)C2)=O)CCC2(CC1)CN(C(=O)CCc1ccncc1)CC(C)O2 C(=O)(CCC(C(C)C)NC(=O)COC)N(CC)CC1CCCCC1 O=C(CC1=CCCCC1)NCCNC(=O)CNc1ccc(O)cc1 c1(CC(=O)NC(CNC(C(C2CCC2)OC)=O)C)c(F)cc(Br)cc1F c1(C(=O)NC(C(=O)NCC2CCN(C(C)=O)C2)CC2CC2)cc(C#N)n(C)n1 c1(CNC(C2(OC)CN(C(CCN(CC)CC)=O)C2)=O)cnccc1C C1(CNC(Cc2c(C)nc(C)s2)=O)CN(C(C2CC2C(C)O)=O)CCC12CCC2 C1(C)(CC)CCN(C(c2coc(C(C)NC(c3n[nH]c(C)c3O)=O)n2)=O)C1 C#CCCCC(C)C(=O)NC(CO)C(N1CCC(CC)(CO)C1)=O N1(C(CC(C)OC)=O)CCC(CCNC(c2[nH]ccc2C)=O)CC1C C1(=O)CCCN1.C1(C(=O)NC)(CNC2C3CC32)CC1.S(C)(=O)(=O)NC1CC1 c1(C(N2CC(CNC(C3CCc4ncnn4C3)=O)C2)=O)ccc2c(c1)CNC2=O C1(N2C(=O)CN3CC(C3)C2)CCCCCC1.C(=O)(CC(F)(F)F)NC c1ccc(CO)cc1.c1(C(C)NCC2CC(C(=O)OC)C2)cn(C2COC2)nn1 c1(C(=O)NCCNC(CS(=O)(=O)NCC)=O)cc(Cl)c(C)c(Br)c1 C1(CCC)(NC(=O)C=C2CCC2)CCCN(C(=O)CC2(C)CCOCC2)C1 c1(C(C)=O)ccc(C(=O)NC(C)CCCNC(=O)Cc2c[nH]nc2O)o1 N1(C(C(C)N)=O)CCC2(CC(O)c3ccccc3O2)C1 c1(C(=O)NCCN(C(=O)C(C)C2CC2)CC)ccc(Sc2ccc(C)cc2)nc1 C12C3CN(CC13)C2=O.C(C)(CCC(=O)NCC)N(C(C(OCC)OCC)=O)C.OCC c12ccc(cn1)CO2.C(C)(C(=O)NCCC(=O)NC(C)C)OCCOC N1(C(CCOCC)=O)C2CCC1CC(CC(C)NC(=O)C1=CCCOCC1)C2 c1(OCC)ccc(C(=O)NC2CN(C(C3(CCF)CC3)=O)CC2C)cc1 CS(C)(=O)=Nc1cccc(C(N2CCCCCC(S(C)(=O)=O)C2)=O)c1 CC(O)(CNC(=O)Cn1ccnn1)CNC(c1ccc(Cl)o1)=O C1(C(=O)NC(CC=C)CO)CC(NC(c2c(C)c[nH]c2CC)=O)CCO1 c1(C(N2CCC(N(C(C(CN(C)C)O)=O)C)C2)=O)cc(Br)c(F)cc1N N1(C(C)C)CC(N(CC2CCN(C)CC2)Cc2cccnc2)CC(C)(C)C1 c1(CC)ncccc1C(=O)NC1CN(Cc2ccc(Cl)cc2)C1.c12csc(n1)C2 CC1=C(C(=O)NCC(CO)NC(=O)COCc2nccn2C)S(=O)(=O)CCO1 c1(C(=O)NC(C2CCN(C(=O)CCc3nc[nH]n3)C2)C)ccc2c(c1)CCN2 N1(c2nccc(P(C)(C)=O)n2)CC2(CC(O)C(O)CO2)C1 C1(NC(c2c(CC=C)cccc2)=O)(CO)CCCN(C(c2c(C)nsc2C)=O)C1 Cc1cccc(C(N2CSCC2C(=O)NCC2C3CCCOC23)=O)c1F.C1CC1 C1(C(N2CC(OCCC(=O)NCC(c3ncccn3)C)C2)=O)CCOC(=O)CC1 c1(C(N2CCC(Cc3ccnc(Br)c3)C2)C(=O)NCCC)ccc(C(F)F)cc1 N1(C(CCCN(C)C)=O)CC(NC(C2CCCC2(F)F)=O)CC2(CCOCC2)C1 c1(C(=O)NC23CCCN(C(CC4CC(=O)C4)=O)CC2C3)cnc2ncnn2c1O C1(CNC(C2(C)CCC2)=O)CC2(CCN(C(c3ccc4nonc4c3)=O)CC2)C1 c1(OC)ccc(C)c(C(=O)NCC(C2CC2)NC(=O)C(F)Cc2ccccc2)c1 CCC(CNC(c1cnnc(C)c1)=O)(CC)NC(C1CC1CC(C)C)=O CCC(O)C(F)(F)C(=O)N1CC2CCC1C(NC(=O)C(CC)SC)C2 C1(CNC(C=CC(=O)OC)C2CC2)CC2(CCCCC2)CO1 CC1Cc2cccc(C(=O)NCC3(F)CN(C(=O)CSCCC(F)(F)F)C3)c2O1 N1(C(CSc2ccc(C)cc2)=O)CCCC(C)(NC(=O)Cc2nc(=N)[nH][nH]2)C1 CCC(CO)(C(=O)N1CCC(C)(CNC(C23CCC(OC)C2C3)=O)C1)OC C1(NC(c2ccc(C)o2)=O)CCCCC1NC(c1ccc(Br)cc1)=O CC1(C)C(c2cccc(F)c2)CCN1C(=O)NCc1ccn(C2CCCCO2)n1 N1(C(c2scc(C(=O)OC)c2)=O)CCOC2CN(C(=O)CCCC(C)=O)CC12 c1(C(C2N(C(C3CSC(C)(C)OC3)=O)CCC2)=O)ccc2c(c1)S(=O)(=O)N=C2Cl c1(C(=O)NCC(C)NC(c2cc(C(F)F)ccn2)=O)cc(F)ccc1C(F)(F)F O=C1CCC(C(F)CNC(=O)Nc2c(N3CCN(CCO)CC3)cccc2)CC1 N1(C(COc2cn(CC)nc2)=O)CCN(C(c2cccc(F)c2)=O)C(C(F)F)C1 CP(C)(=O)C1CC1.c1(N)snc(Oc2ccccc2)c1Cl c1(CNC(C(=O)Nc2c(C(=O)OC)nc(C)cc2)=O)cc2cccc(C)c2[nH]1 c1(NC(Cc2c(C)noc2)=O)ccc(C2CCC(=O)N2)cc1 N#Cc1nc(Cl)ccc1NC(=O)Cc1ccnc(F)c1 CC(C)C(C#N)C(=O)N1CC(S(=O)(=O)N2CCN(C(=O)C(O)C(F)F)CC2)C1 C1(CCNC(C2(CC)CCCC2)=O)CCCN(C(=O)C=CC=C(C)C)CC1 C(N=c1ccnc(NCC(C)OC)[nH]1)c1cn(-c2ccc(CC)cc2)nn1.C(=O)NC C1(N(C(C2C(OCC)CC2)=O)C)CC2CC1N(C(C1CC(C(=O)OC)C1)=O)C2 N1(C(COCCCCC)=O)CCN(C(c2c[nH]c(C(N)=O)c2)=O)C(CC)C1 C(=O)(CC(COC)NC(=O)CC1CCCO1)NC(COC)(C)C N(C1CCc2c(F)cccc21)C(N1CCc2sccc2C1)=O CCC(CCC(=O)NOCCCF)NC(c1sccc1C)=O C(C)(CN=c1nc2c(cnn2C)c(NCC2(F)CCC(CO)C2)[nH]1)OC(C)C C1(CC(=O)NCC(CCC)C#N)CN(C(=O)C2=C(C)OCC2)C(C)(C)C1 c1(CNC(N2CCC(NCc3cnn(C)n3)C2)=O)ccc(I)c(F)c1F N1(C(CC=C=C)=O)CC2(CCN(C(C3Cc4ccccc4S3(=O)=O)=O)CC2)C1 C1(C#N)(NC(CCc2scc(C)c2)=O)CCN(Cc2ccc(Cl)c(F)c2)C1 N1(C(c2ccc(CC)c(F)c2)=O)CCC(C)(C)C(NC(=O)C=Cc2cscn2)C1 C#Cc1cccc(C(=O)NCC2CC(NC(=O)CNC(=O)C3CC3)C2(C)C)c1F C#CCC(C)(C)C(=O)N1CC(C(C(=O)N(C)CCN2CCOC2=O)OC)C1 c1(SCCC(=O)NCCCN(C(=O)C=C2CCC2)CC)ccncc1 N1(C(c2cnc(OC)s2)=O)C(CNC(C2(CC)CC(OC)C2)=O)CC2CC12.c1ccccc1 N1(c2ccc(COC)cn2)CCC2C(CCCN2C(=O)C(C)OCCC(C)C)C1 c1(C(=O)NCC(C2CCN(C(C)=O)CC2)F)c(C)nn(-c2ccccc2)c1C Nc1cc(F)c(Cl)cc1C(N1CC(O)(C(Cl)(Cl)Cl)C1)=O C=C(Cl)CC(C(=O)NC(C)CC(C)C(F)F)NC(c1nnccc1C)=O N1(C(c2c(C)n(C3CCC3)nc2)=O)CCCC(C)(NC(C2CCCC2(C)C)=O)C1 C12(NC(c3cc(C)on3)=O)CCCC1N(c1nc(Cl)nc3[nH]ccc13)CCC2 c1(C(=O)NC2C(CNC(C(CC#C)C)=O)CCC2)n[nH]c2c(C)cccc12 c1(N2CCC(N(CC#C)C(c3ccnn3CC)=O)CC2)cnc(C#N)c(C#N)n1 C1(OC)COCCC1CC(=O)NCCCCCN(C)C(c1oc(C)cc1C)=O N1(C(c2cncc(SCC)n2)=O)CC2CC1CC2CNC(C1CCS(=O)(=O)N1)=O c1(N2C(C)CC(NC(=O)C3=CCC3)C2)cc(=O)n2cc(Cl)ccc2n1 Cc1cc(C(N2CC(NC(c3ccnn3CC#N)=O)C(C)C2)=O)[nH]c1C N1(C(c2nccc(C(C)(C)C)c2)=O)CCCC1C1CCCCN1C(=O)CC(F)F CCC(CCC(=O)NCC1CN(C)CCO1)NC(=O)CCC(=O)CC C1(C(=O)NCCC2CC(C(=O)NCCN3CC4CC4C3)C2)CC2(CCC2)CO1 C12(NC(c3c(C)ccs3)=O)CCC1CN(C(=O)CCOc1cccc(CO)c1)C2 C1(CC(=O)N(C2CN(C(C=C(C)C(F)F)=O)CC2(C)C)C)Cc2ccccc2O1 N1(C(c2cc(C)[nH]n2)=O)CCCN(C(C2CCCCNC2=O)=O)CC1 c1(NC(C(c2sc(C)c(C)c2Br)N(C2CCN(C)C2)CC)=O)ccc(F)cc1C c1(C(=O)NCCC2CC(NC(C3(C)CC(C)C3)=O)C2)cc(F)cc2nc(S)[nH]c12 C(=O)(CCC(O)C(C)(C)C)NC(C)CN(C(=O)Cn1cc(C(F)F)cn1)C c1(C2(CC)CC2)ccc(Cl)cc1.C1(CO)CCOC(C)C2(CC2)CN(C)C(=O)N1 C1(C(CC)C)CCN(C(c2cncc(Cl)n2)=O)CC1 N1(C(c2c(CCC)n[nH]c2)=O)CC=CC1(C)C(=O)NCCSCCO C1(C(=O)NCC(=C)CC)CN(C(c2cc(C)nn2C)=O)CCN1C N1(C(C(CC)(C)C#N)=O)CC2CCC1C(CNC(c1csnc1C)=O)C2 C1(C)(C(=O)NC(c2ccc(Cl)cc2)C)CCCN(C(C2CC(O)CCN2)=O)C1 C1(NC(c2n(CC)cc(Cl)c2)=O)CC2CCC(C1)N2C(=O)C=CC1CCCN1C c1(C(=O)NC(c2cnc(C)o2)C)cncnc1O C(=O)(NNC(=O)C12CC(n3cc(C4(CCO)CC4)nn3)C1C2)C1C(C)(C)C1 C1(=O)CC(C)N1.C(C(C)NC(=O)C=CCOCCO)N(C(C)=O)CC Cc1cc(C(=O)NC(C)CN(C)C(c2ccc(C(N)=O)nc2)=O)ccc1O C1(C(N2CCN(C(=O)CC3CC4(CC4)C3)CC2C2CC2)=O)CCOC2(CCC2)C1 c1(CNC(C2C(C(=O)NCCCOCCCC)C2)=O)ccco1 N1(C(CC=CC)=O)CCN(C)CC12CCCCC2 c1(C(CNC(=O)CC2(CSC)CC2)NC(C2N(CC)CCC2)=O)ccc(F)cc1 c1(OC)cc(OC(C)C)cc(CCC(=O)NC(C2CN(CC3CCCO3)C2)C)c1 CC(CS(C)=O)N=c1nc(N2CCC3(CCC3)CC2)c2c([nH]1)CCCC2 c1(N2CCC(S(CC)(=O)=O)C2)nc2ccsc2c(=NCCC(C)SC)[nH]1 Cc1cc(C(=O)NCC2CCOC2C(=O)NC(C2CCOCC2)(C)C)ns1 C(=O)(C1=CCCSC1)NCC(C(=O)NCC1(C)CCOCC1)O C(C(C)C(=O)NCc1n[nH]cc1C(=O)NCCn1ccnc1C)OC c1(C(=O)NC2CC3(C(NC(c4c(Cl)c(C)n(C)n4)=O)C3)C2)cc2ccncc2s1 C#CCCN=C(NCc1ccc2nc(C)[nH]c2c1)NC1CCCN(C)C1=O S(=O)(=O)(c1cccc(NC(C2CC3(C2)CN(C(C)=O)C3)=O)c1)N(CC=C)CC=C CC(O)C(C(=O)N(CCCOCCNC(=O)C(C)(C)C1CC1)C)NC(N)=O O(N(C)C(=O)CNC(=O)C(F)CC1CN(C(c2cc[nH]n2)=O)C1)CC C1(C(NOCC=C(C)C)=O)CCC(NC(=O)COCC(F)F)CC1 c1(-c2cn(C(C)C)nn2)nc(-c2cccc(Cl)n2)nn1CCCCO N1(CCCNC(CCc2cn(C)nn2)=O)CCN(C(=O)Cn2ncnn2)CC1 COC1CC(NC(=O)NCCCCN2CCCCC2)c2ccccc21 C1(CC=C)(OCC)CN(C(=O)C(C)C#N)C1.C12(C=CCC1)C(=O)NC2 N1(C(c2cncc(C#C)c2)=O)CC2CCC1C(CNC(=O)C(C)CC(F)(F)F)C2 C1(C(=O)NCC2ON=C(C)C2)CC(=O)CN1C(C1CCSCC1)=O N1(C(c2c(C)nc(CO)s2)=O)CC(CNC(=O)CC(=O)NC2CC2)C(C)(C)C1 C(C1=CCN(C(c2cc(N)ccc2C)=O)CC1)NC(CCN(CCC)C)=O c1(CNC(C2CCCN(CCc3cc(C)on3)C2)=O)c(Br)ccc(C)c1F c1(CNC(CCC(C)C)C(=O)O)ccc2c(c1)C(=O)N(C)C2 Cc1cccc2c(C(N3CCCOC(CNC(C4(O)CCOC4)=O)C3)=O)coc12 N1(C(=O)NCC)CCC2(CC1)CC2(C)C(N1CC(O)C(N=[N+]=[N-])C1)=O N1(C(=O)COCC2CC2)CCCC(C2CN(C(=O)CSc3cn[nH]c3)C2)C1 c1(CNC(C2CC2CN=[N+]=[N-])C)cc2occc2s1 c1(N(C)C(c2cn(CCN(C)S(N)(=O)=O)nn2)C2CC2)cccc(OC(F)F)n1 C1(C)(NC(C2(C3N(C(CC=CCC)=O)CCC3)CC2)=O)C(C)(C)C1(C)C c1(C(N)=O)cccc(C(=O)NC2CCOC(c3cccc(F)c3)C2)n1 C1(C(=O)NCCCCC#C)COCCN(Cc2ccc(F)cc2)C1 c1(C(=O)NC2C(CNC(C(CC)OC)=O)C2)cccc(S(=O)(=O)N2CCOCC2)c1 c1(C(=O)NC(C2CCN(C(CC3(C)CC3)=O)CC2)(C)C)cc2ccccn2c1 C1(SCCNC(=O)OC(C)(C)C)CC(C)(C)CCC1NC(=O)CC1CCOCC1 c1(OC)ccc(F)c(C(N2CC(NC(=O)C(F)C(C)(C)O)C(C)C2)=O)c1 c1(OC)cc(Cl)c(Cl)c(Cl)c1NC(=O)Cn1c(C2CCC2)nc2ccccc12 N1(C(c2c(CC)ncnc2)=O)CCC(C)C(C(=O)NC2CCCCC2C#N)C1 C#Cc1cccc(C(=O)NCCN(CCC)C(C2CC(=O)N(C)C2)=O)c1 C(=O)(C1=C(Cl)CCC1)NCCN1CCC1N(C)C.C12(CC(C(F)F)C1)C(=O)N2 c1(OC)cccc2c(-c3cn(CSC4CC5CCC4(C(=O)O)C5)nn3)c[nH]c12 Cc1ccc(C(=O)NC(C)CN(C(=O)CC2CCC(C)CO2)C)c(F)c1F C(=O)(C(CCC(N)=O)N1CCOC1=O)N1CCC(NCc2ccc(OC)s2)CC1 CC(C)CCCCC(=O)NCCC1CN(C(c2nc(=O)n(C)[nH]2)=O)C1 C=Cc1cncc(C(=O)NC2(C)CCCN(C(=O)Cc3ccc(OC)cc3)C2)c1 CC(C)(C)CC(O)CNC(=O)CC1(C)CCN1C(c1cc(O)cs1)=O C12(NC(C(CC)=CC)=O)CCCCC1N(C(=O)Cn1ccc(=O)n(C)c1=O)CC2 C1(C(N(CCC2N(C(=O)OC(C)(C)C)CCC2)C2CC2)=O)CC12CCOC2 c1(C(=O)NCC(C2CC2)NC(CNC(N)=O)=O)cc(=O)c2ccc(O)cc2o1 C1(CNC(CC(C)C)=O)CCN(C(c2nonc2N)=O)CC1(F)F c1(C(=O)NC(CSC)C(C)(C)C)ccc(C)c(C)c1Cl c1(C(N2CC(C)C(CNC(=O)Cc3nnc(O)s3)C2)=O)csc2ccc(F)cc12 c1(C(=O)NC23CCN(C(c4cnc(C(N)=O)s4)=O)CC2C3)cnc2ncccn12 c1(C(N2CCC(CCNC(=O)C3=CCSC3)CC2)=O)cnc2c(c1)OCC(=O)N2 c1(NCC2(C(=O)OC)CC2)ccc(NC(=O)CC2(C)CC2(F)Cl)c(Cl)c1 c1(CCC)c(C(=O)NCC(C)(C2CC2)NC(=O)C=C(C)C(F)F)nnn1CC C1(C(=O)NC2CCC(O)C2)C2CCCC1CN(C(=O)Cn1cc([N+](=O)[O-])cn1)C2 n1(CC(N2CC=CC(NC(C(CC(C)C)(F)F)=O)C2)=O)ccc2c(N)cccc12 Cc1cc(C(=O)NCC2(O)CCCN(C(=O)C(O)(C3CC3)C3CC3)C2)ncc1F C1(NC(CCOCC)=O)CCN(CCCNC(C2CCCC2)=O)C1 C1(NC(CC)=O)CC(C)CN(C(c2csc(-c3csc(C)n3)c2)=O)C1 C1(CNC(CC(C)OC)=O)C(O)C(O)CN1C(=O)CCC(=O)NCc1nccs1 c1(C(=O)NCC2(NC(C(OC)OC)=O)CCOC2)cc(C)nc(O)c1 c1(C(=O)NCC2C(NC(C(=O)NCCC(N)=O)=O)CCCC2)cccc2c1CCN2 N1(CCC)CC(C(=O)NC2CC3C(NC(C4CCO4)=O)C3C2)CC1=O C(=O)(C=CS(F)(F)(F)(F)F)NC(C)(C)CNC(c1ccccc1C(=O)N(C)C)=O C1(CNC(C2CC(C)=C(C)CC2)=O)CC(N=c2[nH]nc(C(F)(F)F)s2)C1 C1(NC(C2CCCCS2)=O)CCSC12CN(C(C1CCC(C(F)F)CC1)=O)C2 C1(NC(C2(C#C)CCC2)=O)CCN(C(=O)CC2OCCC2(C)C)CC(C)(C)C1 N#CC1(C(=O)NC2CCCCCN(C(C34CC(F)(C3)C4)=O)C2)CCCC(=O)C1 C(C1(O)CCCc2ccccc21)C(=O)Nc1cc(C)cc(C(N)=O)c1 N1(C(C2C=CCS2)=O)CCOCC1C(N1CCSCC1)=O O(C1CCCc2ccc(OC)cc21)Cc1nn(CC)c(-c2ccns2)n1 N1(C(=O)C2=NOC(CO)C2)CCC2(CCN(C(c3cc4ncccc4[nH]3)=O)C2)C1 c1(C(C(N2CCC(CNC(=O)COCC3(F)CC3)C2)=O)O)ccccc1F C1(C(=O)NC(C)C2CC2)CCC(NC(c2ccon2)=O)C1 C(=O)(CC1COc2ccccc21)NC1CC(NC(C2CC(=O)NC2)=O)C1 c1(C(=O)NC(C2CCCN(Cc3scnc3Cl)C2)C)cccc(F)c1F C1(C(=O)NCC2CC(CNC(C(C)NC(C)=O)=O)C2)CCCC2(CC2)C1 CC1CCOC1CCNC(c1ncoc1CNC(=O)CC1CCOC1C)=O N1(C(c2c(CC)nn(C)c2)=O)CC(NC(C2CCOC2)=O)CC12CCCC2 C1(CC#C)(C(N2CCC(NC(=O)Cc3csc(SCCSC)n3)C2)=O)CCCC1 C1(C(=O)NCC(c2ccccc2)CNC(=O)C=CCF)C(Cl)(Cl)C12CC2 C=CCN=C(NCC(C)(C(C)C)OC(F)F)NCC.C12(CCOC1)OC2 C1(C(N2CCCC(CC(N3CCC(COCC)C3)=O)C2)=O)CCCCCCC1 C(=O)(CC1=NNC(=O)C1)NCCCCNC(C(C)C1CCCO1)=O C1(F)(CNC(CC(=O)NCC#C)=O)COCCN(C(=O)Cc2ccoc2)C1 C1(=O)N2CCC(O2)C(=O)O1.N1(C(=O)OC(C)(C)C)CCC(C(=O)COC(=N)O)C1 N1(C(c2c(NC)snc2C)=O)CC2CCN(C(=O)CC3CCCCN3C)C2C1 C=CC(CC(=O)NC1CC1NC(=O)CCN(C)C1CC1)c1ccccc1 CCCCC(CNC(=O)C(C)=C1CCCC1)NC(C1(C)CCCCO1)=O c1(CNC(=O)CCCC2(C(=O)OC)CCC2)cc(OC(C)(C)C)cc(O)c1 c1(NC)ccc(NC2(C(=O)Nc3ccnc(Br)n3)CC2)cc1NC(C1CC1F)=O Cc1ccc(CCNC(C2CC(=O)CN2C(C2CC(C)N(C)C2)=O)=O)cc1 C1(CN(C(=O)C=CBr)C)CN(C(c2cc(-c3ccco3)on2)=O)CCO1 CCCCCCCCCC(CC)C(=O)N(CC(=O)NOCCC(C)C)C FCCCN=C(NCCN1CCOCC1)NCc1ccccc1N1CCCCC1 C(=O)(C(F)(F)CCn1cccn1)NC1C2CN(C(C(C=C)O)=O)CC21 c1(C(=O)NC(C2CCOC2)C#C)ccc(CNC(c2ccsc2Cl)=O)cc1 c1(C(=O)NCCOCCN(C)C)cn(C2(Cc3cc(Cl)c[nH]3)CC2)nn1 CC(C)S(=O)(=O)CC(=O)NC(CNC(c1cnn(C)c1)=O)CO.c1(C)cc[nH]c(=N)c1 C(C)(C(C)C(=O)NC(C1CCC1)C)NC(c1c(CC)ocn1)=O N1(C(C2N(C(C(CC(C)C)N(C)C)=O)CC2)=O)CCOCC(C)(C)C1 C1(C(=O)NCC2(C)CCN(C(CCCOCCOCC)=O)C2)CC12CCCCC2 CONC(=O)C(=O)NCCN1CCC(OC)C1.C1(C)C(C)C(=O)O1 C#Cc1ccc(C(=O)NCC2OCCC2C(=O)NC2CCN(OC)CC2)c(C)c1 C1(CNC(=O)C2CC2)CCCCN1C(C(=O)OC)c1nccs1.CC(Cl)Cl c1(CCC(=O)NC)ccccc1-n1cc(CN(C(C)COC)C)nn1 c1(C2(C)C(C(=O)NC(c3ccc(O)cc3)CC)C2)ccc(F)c(F)c1 c1(CC(=O)N(CC2CC(NC(=O)Cc3ccco3)C2)C2CC2)cncc(Br)c1 C(=O)(C(F)(F)CC)NC(CCC)CNC(=O)C(O)CN1CCCC1 C1(C)(C(N2CC(C)C(NC(c3ccn(C)c3)=O)C(C)C2)=O)CCCCCNC1=O CC(C(=O)NCC1CCCCC1NC(=O)CCC(C)(C)O)C(F)(F)F CC(CC(=O)NC(C(=O)N(C)CC1CC(F)(F)C1)C1CCCO1)C1CC1 N1(C(C(C(=O)OC)C)=O)CCCN(C(c2cccnc2)=O)CC1 c1(C(=O)NCC(C)(CO)NC(C(CC)C(C)(F)F)=O)cc2ccccc2cc1Cl C1(CC2CCC(=O)N2)CCC(CC(N2CCC(c3ccc(CO)cc3)C2)=O)CC1 C1(NC(CCOCCC)=O)CCC2CC1CN2C(=O)Cc1ccnc(F)c1 c12ccc(nc1)[nH]2.N1(CCCNC(N(CC#C)CC2CC2)=O)CCOCC1 n1(CC(N2C3CN(C(c4ccc(C)o4)=O)C(C3)C2)=O)ccc2nc(O)nc(O)c12 c1(CCC(=O)NCC2CCC(C(=O)NC3C(C)(C)C3)CC2)cc(F)ccc1Br Cc1ccc(F)cc1CC(=O)NC1(C(=O)NC2CCOC(C)C2)CCC1 OCCCCCCCCNc1cc(-c2ccccn2)cc(F)c1 C1(C(N2CCC(N(C(=O)Cc3nc[nH]n3)CC)C2)=O)CC2CCC1C2 c1(NC(C(C2(C)CC2)NC(c2c(CC)ncnc2)=O)=O)ccc(O)c(C)c1 C1(CNC(=O)OCC)CN(C(=O)CC2CC2C(F)(F)F)CCO1 c1(C(N2C3C(NC(C4CCC5(CCC5)O4)=O)C(C3)C2)=O)occ2c1CCCC2 CC(O)C(C)(C)C(=O)N1CCCC2(CNC(=O)CCC(F)(F)F)CC12 C(=O)(CS(=O)(=O)C(C)C)N1CCC(CCC2CCN(C(CC)=O)C2)CC1 C1(C(=O)NC(C=C)C(=O)N2C(C(=O)OC)CC2C)CC2(CCO1)CC2 c1(C2(N(CC(C)(C)C)C(C)CNS(C)(=O)=O)CC2)ccccc1 CCC(CC)C(C(=O)N1CC2CC2C1C(=O)Nc1cccc(O)c1)OC c1(C(=O)NCc2scc(C(=O)NCCCC(CC)CC)c2)cc2ccccn2n1 c1(OC)ccc(CN2CCN(C(c3c[nH]nc3C)=O)CC2C)cc1Br C(=O)(CCCC(C)=O)NC(C1CC=CCC1)C(=O)NC(CC=C)CC c1(C(CC(=O)NCC(C)N(C(CCCC#C)=O)C)C)c[nH]c2ccccc12 C(C(=O)NNC(=O)CNCCCCCF)c1ccc(OC)cc1 C12(C(=O)NCC(C)S(C)(=O)=O)CC(CO)(CN1C(C1CCCC(=O)CC1)=O)C2 C1(CNC(c2c(CC)occ2)=O)CN(C)CCN1C(c1nscc1N)=O N1(C(CNC(C2COC(=O)O2)=O)=O)CCN(C(C2CCOC2C(F)(F)F)=O)CC1 C1(C(=O)NC2CCCC(NC(C(CSC)(C)C)=O)C2)Cc2nncn2C1 C(=O)(CCC(C)(C)[N+](=O)[O-])N(C(C)C(=O)NCCN1CC(CF)C1)C C1(C(N2CC(CC)N(C(=O)C=CCO)CC2)=O)CCc2nn(C)cc2C1 Cc1c[nH]cc(C(=O)N(C)CC2(CNC(C3(CO)CCOCC3)=O)CC2)c1=O Cc1nc(Cl)cc(=NCC(C)C2CCNCC2)[nH]1 N1(C(C(CC=CC)C)=O)CC(NC(c2cnn(CCF)c2)=O)CC12CCC2 C1(CC)CCC(C(=O)NC(C(=O)N2CC(OC)C2)c2cccs2)O1 N1(C(c2ccc(Cl)o2)=O)CCC2(CCC(NC(C3(CO)CCC3)=O)C2)CC1 C1(C(=O)OCC)(C(=O)NC2CCCC(F)C2)CCCCC1.N12CCC(C1)C2=O c1(N(C)C)nc(NCc2nc(-c3cccnc3)no2)c2cc(C(C)(C)C)sc2n1 c1(C(=O)NC2CN(C(c3cc(Br)ccc3Br)=O)CC2F)cc(Br)c(F)cc1F CC1(C)CCCN(c2ccc(-c3cccc(Cl)c3)nn2)C1 CC(C)(CCC(=O)N1CCC(CCC(=O)NC(C(C)(C)O)C2CC2)CC1)[N+](=O)[O-] N1(C(COCC)=O)CCCN(C(C2(c3cc(Cl)ccc3F)CC2)=O)CC1C N1(C(C2(CCC)CC2)=O)CCOC2(C1)CN(C(=O)CCC1CC1(Cl)Cl)C2 c1(C(C2CC2c2ccccc2)C)nc(-c2cc(I)nn2C)n(CC2CC2)n1 c1(C(=O)NCCCN(C(=O)CCOCCN(C)C)CCC)c(C)nsc1N C1(CNC(C(N2CCOCC2)C)=O)C(NC(c2csc(F)c2)=O)CC1O CN1CCN(C(=O)C=C2CCCC2)C(CNC(=O)CCCN2CCOC2=O)C1 CC(C)C(C(=O)NCCCN(C(=O)CCc1nccs1)CCO)NS(N)(=O)=O N1(C(c2cc(C(C)=O)[nH]n2)=O)CC(C(=O)NCC(C)O)OC(C)C1 N1(C(C2CC(N(C)C)C2)=O)CCC2(CNC(=O)CCCC(N)=O)CCCC12 C(=O)(C(N)CCC(C)(F)F)NCc1cccc(NS(C)(=O)=O)c1 C1(C2(c3cn(CC(=O)NC(c4cnoc4)C)nn3)CCC2)OCCC1(C)C Cc1nc(CNC(=O)C(CNC(c2cocc2C(N)=O)=O)CC2CC2)cc(O)n1 c1(NC(c2n(CCC)nnn2)c2cc(C3CCC3)no2)cc(F)ccc1SC N1(c2nc(=N)nc(N3CCN(S(CC)(=O)=O)CC3)[nH]2)CCC2(COC(=O)N2)C1 C1(NC(C2CC(CC)(CC)C2)=O)CC2CC1CN(C(=O)CC1CC1(Cl)Cl)C2 CCCCC(C)C(=O)NCC(C)NC(c1ccc(N)c(O)c1)=O c1(CSC)cc(C(N2CCC(O)(CN(C)C(c3csnc3C)=O)C2)=O)ccc1F CC(C)(C)C#CC(=O)NCc1ncoc1CCNC(=O)C(C)(O)C1CC1 C#CCC(C)C(=O)NC1CC(CNC(=O)COCc2ccccc2C)C1 C(CC(=O)N1CC(O)(c2cn(CCN3CCSCC3)nn2)C1)(c1cccs1)NC c1(C(=O)OOC(=N)O)ccc(Cn2cc(C(C(C)O)NC(N)=O)nn2)cc1 C(=O)(C1SCCc2ccccc21)N1CC(C(C)NC(c2cn(C)c(=O)n2C)=O)C1 c1(C(=O)NC2C(OC)CN(C(C3CCC(C)(C)OC3)=O)C2)cc2c(s1)CCOC2 C1(NC(C=CC(=O)N(C)C)=O)CCCCN(C(=O)CCC2(C#N)CCC2)C1 Cc1ccc(=O)n(CC(=O)NC2CC3CC2N(C(C2CCS(=O)(=O)C2)=O)C3)c1 Cc1nn(C)c(C(=O)NC2CCCCN(C(=O)CC3CCCCO3)C2)c1Cl c1(C(=O)NCCC2CN(C(CSC)=O)CC2C)cc(C)n(-c2cccnc2)c1C CN1CC(O)(CN(C(=O)C(O)C2CN(C(c3ccccc3)=O)C2)C)C1 N1(C(CCc2n(C)ccc2)=O)CC(C(=O)NCc2ccccc2)C2(CCC2)C1 n1(CC)cc(C(=O)C(=O)N(C)CCOCCSc2n[nH]c(O)n2)cn1 c1(COc2c(=O)cc(C(=O)OCc3ccc(F)cc3)oc2)cc(F)c(Br)cc1Cl C(=O)(CC(C)CF)NC(C1CCCC1)CNC(c1c(C(C)C)ccs1)=O C1(NC(=O)C=CCC(=O)NCCN2CCC2)CCN2CCCC2C1 Cc1nc(C)c(CCC(=O)NCC2CCN(C(c3c[nH]c(=O)cn3)=O)C2)c(O)n1 C=CCCCCC(=O)N1CCC(F)(C(=O)NCC2SCCS2)C1 C1(CCCC(N2CC(C)(NC(c3nc(COC)oc3)=O)C2)=O)CCC(C)C1(C)C c1(C(=O)NC2CCC(NC(c3scc(C)c3)=O)C2)cnc(Cl)cc1Cl C1(CNC(C(C)N(CC)CC)=O)CC2(CO1)CN(C(c1cccc(Cl)c1)=O)C2 C(=O)(C1=CCC(C)(C)CC1)NC1CCN(C(CCCCC)=O)CC1F C1(C(=O)NC(CC)COC)CCCN(C(=O)CCN(C)CC)C1 CC(CNC(c1ccc(C2CC2)s1)=O)(CO)NC(=O)C(c1ccccc1)F Cn1c(C(c2nnnn2-c2cccc(OCF)c2)NC(CF)C2CC2)cnc1Br c1(C(=O)NC(CC)CN(C(=O)CCC2CCCO2)CC)cc(Br)cn1CC N1(C(C(n2cc(Cl)cn2)C)=O)CC2(CCCC(CNC(c3nccs3)=O)O2)C1 C1(C)(CC)NC(=O)C2=C1N(CC1CC1)C(=O)NC2c1ccc(C)c(CC#N)c1 C1(NC(C(CC(=C)C)OC)=O)CCN(C(=O)CCCCCF)CC12CCC2 CC1CC(=O)NC(C(=O)NC2CCC(NC(=O)CC3CCCC4(CC4)C3)CC2)C1 c1(C(=O)NC(C2CCC3(CN(C(=O)C(Cl)=CCl)C3)O2)C)c(N)cccc1[N+](=O)[O-] N1(C(c2ccn(CC)n2)C(=O)NCCOCC)CCOc2ccc(Cl)cc2C1 c1(C(=O)NC(C(C)NC(c2ccc(=O)oc2)=O)C)cnn2ccc(O)nc12 N1(C(C2CCN(C(=O)NC)CC2)=O)CCC2CCN(C(=O)CC(=O)NC3CC3)CC12 C1(NC(CCCCCC)=O)CCN(C(c2nccc(Cl)c2C)=O)CC(C)(C)C1 c1(CN2CCC(NC(c3ccc4cccnc4n3)=O)C2)cccc([N+](=O)[O-])c1Cl N1(C(=O)CN2CCOC2=O)CCC(CC(N2CCCCC2)=O)CC1 c1(CC(=O)NC(C(=O)N(C2CC(OC)C2)C)CC2CCC2)ccc(C)cc1 c1(CN2CC3CN(C(c4ccc(O)cn4)=O)CC32)ccc(F)c(O)c1F C1(O)(CNC(=O)CC2CC(NC(c3nc(Cl)cs3)=O)C2)CCCCCC1 C(=O)(CCC(C)SC)N(CCCCCC)CCNC(=O)CC(C)O c1(C(CC(CNC(c2ccco2)C)OC)C2CC2)nnnn1C1COC1 C1(COC)CNC(=O)CN1C(C1(N(C(=O)C(C)N2CC(C)C2)C)CCC1)=O C(=O)(C(O)(C(F)(F)F)c1ccccc1)N(C(CNC(=O)C(C)(Cl)Cl)C1CC1)C c1(OC)ccc(C(C)C(=O)N(C)C2CC2)cc1F.C12(O)CCN(CC1)C2=O c1(NCCc2cc(C)n(C)n2)[nH]c(=NC2CCC(C(N)=O)CC2)nc2sccc12 N1(C(CC=CCC)=O)CC(NC(C23COCC2C3)=O)C(C2CC2)C1 Cc1nc2cccc(C(=O)NCC(CNC(=O)C(C)(C)c3cscn3)CO)n2n1 C1(NC(C2C(C=C)C2)=O)CC(F)(CNC(=O)CCC2CCCCC2)C1 C(c1cccn1C)=CC(=O)NC1CC(c2ccccc2)(CNC(C2(C)CC2)=O)C1 N1(C(c2cncs2)=O)CCCC(C2CCN(C(c3cccc4cncn34)=O)CC2)C1 C(=O)(CC(C)(C)O)N(C)CCOCCC(=O)NCc1nc[nH]n1 CCC(F)(F)CC(=O)NC(CCN(C)C)C(=O)N1CCCCC1CC(N)=O C1(C(=O)NC(C2CCN(C(c3ncc(CC)s3)=O)CC2)(C)C)CC2CCCC2C1 C1(N(C(=O)C=C(Cl)Cl)CCOC)CCN(C(=O)C(c2ccc(C)o2)C)CC1 c1(C(=O)NC2CC3(CCN(C(C4C(C)C4)=O)CC3)C2)nc(O)c2ccccc2n1 N1(C(CCCOCC#C)=O)CC(C(=O)NCC)OC(C)C1.N1(CC(=O)N)CC=CC1 C=Cc1ccc(C(N2CC(OCC=CC(=O)NCC)C(C)C2)=O)cc1.C1CO1 c1(C(c2nnnn2C2CCC2)NCc2cc(C)on2)nc2ccccc2[nH]1 N1(C(C=CCOC)=O)CCN(C)C(CNC(=O)CC2(C)CCS(=O)(=O)N2)C1 N1(C(C(C)n2ccnn2)=O)CC2CCC(C1)C2CC(N1CCCC2(CCO2)C1)=O c1(C(N2CCC(CCOC)(NC(C=CSC)=O)C2)=O)c(SC)nc(O)nc1C n1(CCC(N2CCC(C(C(=O)NC3(C(=O)OC)CC3C)C)C2)=O)c(C)ccc1C CCC(C)(C)C(O)C(=O)N1CCC(C2CCC(C)(C)N(C(=O)CS(N)(=O)=O)C2)C1 C1(NC(C(CC)SC)=O)CCCCN(C(=O)CCc2nc[nH]n2)CC1 c1(C(=O)NCC2C(NC(C(CSC)c3ccccc3)=O)C2)cncc(C#N)c1 N1(C(CC2CCN(C)C2)=O)CCOC2(CCN(C(c3cc(O)ccc3O)=O)C2)C1 C(=O)(C(C)C(O)C(C)C)NCC1CC2(CN(C(C3(OC)CCSC3)=O)C2)C1 C(N=C(NC1CCOCC1)N1CC2C(C(F)F)C2C1)c1n(C(C)C)ncn1 C(=O)(CC(C)(C)CC(=O)NCC(O)CNC(c1ccsc1C)=O)OC Cc1c(C(=O)Nc2ncc(-c3ccccc3)s2)cnn1C(C)(C)C N1(C(=O)CCc2ccoc2)CCC(F)(CNC(C2C(C(C)C)(CC)C2)=O)C1 CCC(C(=O)NCCN(CC(C)O)C(C1(CF)CC1)=O)n1ccc(C2CC2)n1 CC1(NC(C2CCCS(=O)(=O)C2)=O)CCCN(C(=O)C(C2CC2)C2CC2)C1 N1(C(c2cn(C)nc2C2CCCNC2)=O)CCC(CO)C(O)C1 C1(NC(CCN(CC)CC)=O)CCCN(C(c2cc(CF)on2)=O)C1 c1(OC)ccc2c(c1)OC(NC(=O)CC1CCC(C)(C)C1)C2 C12(CNC(c3nc(COC)oc3)=O)CC(CO1)N(C(C1CCCC(C)(C)O1)=O)C2 CC1(C(N2CCC(c3cn(CC4CCOC4)nn3)CC2)=O)CC2CCC1O2 N1(C(c2ccnn2-c2ccccc2)=O)CCC2(C1)OCC1CC21 c1(COC)ncsc1C(=O)NCCCC1CCCN1C(=O)CCC1CCOC1 N1(C(CNC(c2cccc(C)c2)=O)=O)C2CCC1C(NC(=O)C(C)(C)C(C)C)C2 CS(=O)(=O)c1cccnc1N1CCCC(NC(=O)C=Cc2nccs2)CC1 C(CCCC(=O)NCC1(CO)CN(C(=O)Cc2sccc2C)C1)OCC C(C)(CCC(=O)N1CC2CC1C2CNC(c1ccc(C(F)(F)F)o1)=O)OC N1(C(C(C2CCOC2)NC(CCOCC#C)=O)=O)CCN(Cc2nncs2)CC1 N1(C(C=C(CC)C)=O)CCC(C(C)(C)C)(CNC(=O)C(O)Cc2[nH]cnc2C)C1 c1(N(C)C)ccc(C(=O)NCC(O)CCNC(c2cc(CO)on2)=O)nn1 C(CCCC(C)C)N(C(C(=O)NC1(CC)CC1)c1ccoc1)C N1(C(c2c(C)[nH]cc2)=O)CC=C(CCNC(=O)CC(C)C(F)F)CC1 c1(OC)c(C)cc(C(=O)NC(C)CNC(=O)CC2C(C)(C)C2(C)C)cc1C c1(CNC(C2(C)C(C)(C)C2)=O)ccc(CNC(C2(CO)CCCO2)=O)cc1 CC(C)CS(=O)(=O)CCC(=O)NC1CCN(C(=O)C(O)CC2CCCCC2)C1C c1(C(C(=O)NCc2ccco2)N(C(C)CC(C)C)CCOC)sc(C)cc1C N1(C(c2cc(SC)oc2)=O)CC2CC(NC(=O)Cn3ncn(C)c3=O)C2C1 CC1(C)CCN(C(C2CC(NC(c3ccc(F)cn3)=O)C2(C)C)=O)C1 c1(OCCOC)cccc(C=CC(=O)NC(C)Cc2cccc(C)n2)c1 c1(OCCN(C)C(C2CC(O)(C#N)C2)=O)cccc(Cl)c1 N1(C(=O)Cc2cn(C3CN(C(c4ccc(N)cn4)=O)C3)nn2)CC2CCC(C1)O2 C1(C(=O)NCC(CNC(c2cnc(O)c(F)c2)=O)F)CCCC12CCOCC2 C1(C(N2CC(O)(CCc3cn(Cc4cocn4)nn3)C2)=O)CCS(=O)(=O)N1 C1(C)(CCC(=O)NCCOCCCNC(C(C)c2ccsc2)=O)CC1(F)F c1(C(=O)NC2CC3CN(C(C4ON=C(CC)C4)=O)C2C3)ccc2nsnc2c1 N1(C(C(CN(C)C)(C)C)=O)CCC2CC2(NC(c2cccn3nnnc23)=O)CC1 N1(C(CC=C)=O)CCCCC(N(C(=O)C(c2cccnc2)O)C)C1 CC(C)C(C(=O)N1CCN(C(=O)CC2CCCC3(CC3)C2)CC1CO)C(C)C N1(C(C2C(NC(CC3CCC(C)CO3)=O)C3CCC2C3)=O)CCCOCC1C N1(CCC(=O)NNC(=O)c2ccc(Cl)cc2F)CC2C3C=CC(C3)C2C1=O c1(CC(=O)NC23CCC(CNC(C=NOC)=O)(OC2)C3)csc2cc(C)sc12 C1(COC)(NC(C2CCOC(C)(C)C2)=O)CCCN(C(c2c(C)noc2N)=O)C1 Cc1nc2ncnn2cc1C(N1CC(NC(c2ccc(Cl)s2)=O)CC1(C)C)=O C1(N(C(C(C)NC(=O)NC)=O)C)CN(C(c2cncc(C(C)C)c2)=O)CC1(C)C C=C1CC2CCCC(C1)N2C(=O)C(C)(Cn1cccn1)NC(=O)C(C)C1CC1 C=CCC(C)(CNC(=O)C(C)N(C)C(C1CCOC1CC)=O)CO C(CC1=CCN(C(=O)C(C)CF)CC1)NC(c1c(CC)nc[nH]1)=O C12(NC(=O)CC3CC(NC(c4cccc(O)c4)=O)C3)CCCC1OCC2 C1(C(=O)NC(c2ccccc2)C(=O)N(CCC(F)(F)F)C)CC2CCC1CC2 c1(C(N(CCNC(CC2(C(=O)OC)CCC2)=O)C)=O)cc2cnccc2cc1F O=C(NNc1ccccc1C(F)(F)F)C(F)(F)Br.C1CCN1 c1(C(=O)NCCNC(C2CC(CC)(CC)C2)=O)ccn2[nH]c(=N)nc2c1 C(=O)(C(C)C(C)c1ccn(C)n1)NC(CNC(c1nnc(C)s1)=O)C C1(NC(c2c(C)nncc2)=O)CCCC12CCN(C(C1(O)CCC1)=O)C2 Cc1ncc([N+](=O)[O-])n1CC(=O)NC1CN(C(C2CC(C)(C)O2)=O)CC1(C)C N1(C(C(C(CC)(C)C)O)=O)CCCC2(CCN(C(=O)C=Cc3cn(C)nn3)C2)C1 C(N(O)C(=O)CC1CCN(C(=O)NC)CC1)c1cn(CCC=C=C)nn1 c1(SC(C)CC(N)=O)nc2ccccc2n1CCNC C#Cc1cn(C)nc1C(=O)NCC1CC(NC(=O)C(F)CC2CCC2)C1 N1(C(Cc2cc(C)no2)=O)CCn2c(C(=O)NCC3CNC(=O)CO3)cnc2C1 C(CC(C)C)(C(=O)N1CC(NC(c2cnns2)=O)CC(F)C1)NC(C)=O c1(OC)cncc(C(=O)NC2CCC(NC(c3cc(N)ccc3F)=O)CC2)c1C C1(C(=O)NC2(CNC(c3ccc(C(C)=O)nn3)=O)CC2)CC2CCC(C1)C2 c1(CC)cccc(C(N2CCC(O)(CNC(C3(C)CC(C)(C)C3)=O)C2)=O)n1 C12(C(=O)NCC3(O)CN(C(C4COC4)=O)C3)CCC(CC1)C2 Cc1ccncc1C(=O)NCCn1cnc(C(=O)NC2(C(F)F)CCCC2)c1 Cc1conc1CC(=O)NCCCC(C)NC(=O)COCCc1cccs1 C1(C2CCN(C(=O)C=C=C(C)C)CC2)(NC(C(C)OCCCCCC)=O)CC1 c1(C(=O)NC(C(C)C)CNC(C23CC2CCC3(F)F)=O)ccc(O)c([N+](=O)[O-])c1 C1(NC(c2cc(C)[nH]n2)=O)CN(C(c2ccc(C(=O)NC)nc2)=O)CC2CC12 C1(C(=O)NCCC2CCC(NC(CCP(C)(C)=O)=O)C2)CCc2nncn2C1 c1(CNC(C2CCCCCN2C(c2cccnc2)=O)=O)cccn2nccc12 c1(C(=O)NC(c2ccccc2)(CC)C)occ2c1CCC2 Cc1c(C(N2CCCN(C(c3ccc(F)s3)=O)CCC2)=O)[nH]c2c(C)cccc12 N1(C(C(c2cnccn2)C)=O)CCC2(CC(NC(C34CCCC3CCC4)=O)C2)C1 C1(C(N2C(CC(=O)NC(CCC=C)CO)CCC2)=O)CCC(C2CC2)C1 C(=O)(C(C)(O)CC(F)(F)F)N1C(CNC(CCN(C)CC)=O)CC1 N1(C(C(C(CCC)NC(C2CCC(=O)CC2)=O)O)=O)CC2C(=O)NC(=O)C2C1 N1(C(c2ccnc(-n3ccnc3)c2)=O)CC2CC(C1)N(CCn1cccn1)C2 c1(C(=O)NC2CC(NC(C(CC)OCC)=O)C2)sc2ccc(F)cc2c1C C(=O)(C(F)(F)C(F)(F)C(F)(F)F)NCCNC(=O)CCC(=O)c1ccc(F)cc1 N1(C(C)=O)CC2CC2(NC(c2c(Cl)n[nH]c2C2CC2)=O)C1 C1(C(N(CCNC(c2nc(CC)sc2)=O)C2CC2)=O)(CC)CCC(O)CC1 C(=O)(C(C(C)O)N(C)C)N1CC(C(=O)NCCSC(F)F)(OC)C1 CC(C)C(C)CC(=O)N(C(C)C(=O)Nc1cnn(C(C)(C)C)c1)C N1(C(c2cc(CNC(CCC#C)=O)sc2)=O)CC2COC(=O)C2C1 N1(C(c2c(NC)scn2)=O)CCN(C(=O)C(C)OC2CCCC2)C2CCC12 c1(C(=O)OC)cccn(CC(N2CSCC2C(N2CCCCC2)=O)=O)c1=O c1(N(C2CCN(C(c3ccc4[nH]ccc4n3)=O)C2)C)nccc(S(C)(=O)=O)n1 N1(C(c2cc(C(C)(C)C)on2)=O)CC2(CCCCN2C(C2(CO)CC2)=O)C1 c1(CC)nc(C)oc1C(=O)NCCc1ccc(CNC(C2CCCC2C)=O)cc1 C1(C(=O)NCCCN(C(C)=O)CC)CCN(C(C2CC=CCC2)=O)C1 N1(C(c2n(CC)ccn2)=O)CC(NC(c2cnc(C)cc2Cl)=O)CC(C)C1 C(=O)(C(CNC(C1(C)CNC(=O)N1)=O)C(C)(C)C)NC(C)C(F)F N1(C(Cc2c(C)ncnc2C)=O)CCCC1C1CCCN1C(=O)CCOC1CC1 c1(CSCC(=O)OC(c2ccc(F)cc2)C(=O)OC)ccc(C#N)cc1F N1(c2ncc(C)c(C(N3CC(CO)C3)=O)n2)CCCC(C)(c2ccccc2)CC1 C1(NC(c2c(C)cc(Cl)cc2)=O)CC2CC(C1)N(C(=O)CCc1ccncc1)C2 c1(C(=O)NCc2c(CCNC(c3c(C)onc3)=O)ocn2)cc(O)ncc1Br C(=O)(C1=NOC(CNC(=O)CCC2CCCC2)C1)NC(c1ncc[nH]1)C N1(C(C(c2ccc(C)cc2)C)=O)CCN(C(c2n[nH]c(C)c2F)=O)C(CCO)C1 C1(CNCC2C(NC(=O)OC(C)(C)C)CCOC2)=NN([SH](=O)=O)CCCC1 C(C(O)C(=O)NCCN(C(=O)CSc1nccn1C)CCOCCO)N(C)C CN1N=C(C(=O)NCC(CC(=O)NC2CCCC3(CCC3)C2)C2CC2)CCC1=O C#Cc1ccc(C)c(NC(=O)CCC2CCCN2C(=O)Cc2ccc(F)cc2)c1 N1(C(c2cc(S(C)(=O)=O)sc2)=O)CCC2CCC(C1)N2C(=O)CC1CCOC1=O C1(C(N2CCC(C(C)Nc3cc(O)ncn3)C2)=O)CC(=O)N(C2CCCC2)C1 C(C1=CCCN(C(=O)CCC(N)=O)C1)NC(c1c(CC)nn(C2CC2)c1)=O C1(NC(C(CC)(C)O)=O)CN(C(=O)CCn2cnc3ccccc23)C2(CCC2)C1 N1(C(C(C#C)(C)C)=O)CCC(CC)(NC(c2ncccc2CC)=O)CC1 C1(CNC(c2ncn(C)c2)=O)CC2(CC2)CN1C(=O)CC(=O)NC1CC1 N1(c2cc(C)c(C#N)cn2)CCC2(CN(C(c3ccn(C)c3)=O)CC(C)O2)C1 Cc1ccc(-c2cn(C3CCN(C(=O)C(C)CF)CC3)nn2)cc1F C1(NC(c2n(C(CC)CC)ncc2)=O)CCN(C(=O)CCC2CCCO2)C(C)C1 N1(CC(COC(COC)C)O)CC=C(CNC(C2CCC(C)CC2)=O)CC1 C#CCC(CC#C)NC(=O)CC1CCCN(C(C2CC(C)N(C)C2)=O)C1 C1(C(N2CCC(C)(NC(CC3CCC(C)(C)C3)=O)CC2)=O)CC2(C1)CC1(CCC1)C2 CC(C)(C)C(O)C(=O)NCCC1(NC(c2cc(C(C)(F)F)on2)=O)CCOCC1 N1(CC=C)CCC(O)CC1CC(=O)NCCSCC(=O)OCC C(=O)(CCC(=O)NCCCN(C1CCCC1)C(c1ccsn1)=O)NCC C1(NC(c2ccc(SC)o2)=O)CCC2(CC1)CN(C(=O)CC(C)SC)CCO2 c1(-c2cn(-c3cccc(CN4CCN(C=O)CC4)c3)nn2)c(F)cc(Cl)cc1Cl c1(OC)cc(C(N2CC3CC3(C(=O)NC(C)(C)CC(C)C)C2)=O)ncn1 C1(N(C(=O)CC2(C)CC2(Cl)Cl)C)CCCCC1NC(c1cn(C)c(O)n1)=O CCC(CC(=O)NC(CC1CC1)C(N1CCN(C(C)(C)C)CC1)=O)CC(C)C C(=O)(N(CCC(=O)NCC(c1ccco1)N(C)C)OC)c1ncc(OC)nc1 N1(C(C2(COC)C=CCC2)=O)CC2CCC(C1)C2NC(c1cnc(C(C)C)o1)=O c1(CC(=O)NC2CC(CNC(C(C)C3CC3)=O)C2)ccc2c(c1)CCCS2(=O)=O C(CCNC(c1nc(C)c(C)s1)=O)(C(=O)NC(c1cnc[nH]1)C)OC C1(CNC(c2c(CC(N)=O)scc2)=O)CCCCN1C(C1C=CCCC1)=O N1(C(COCC(C)C)=O)CCN(C(=O)CC(O)CCc2ccccc2)C(CO)C1 Cc1cccc(C(=O)C(=O)NC2(CO)CCN(C(=O)C=CC3CCCN3C)C2)c1 N1(C(C(N2CC(CC(C(=O)NC3(CCC)CCC3)F)C2)=O)=O)CCC(C)CC1 Cc1cc(Br)ccc1C(=O)NCC1COCCN(C(=O)CC(C)O)C1 Cc1ccnc(OCCN(C(=O)CC2(CS(C)(=O)=O)CC2)C)c1 C(=O)(C(CC(F)F)NC(=O)CC1(C)CCC1)NC(c1n(C)ncc1)CO c1(CC(=O)NCC=CC(=O)NC(CC)(C)C)csc(C)c1 c1(C(=O)NC(C(C)NC(C2CN3CCN2CC3)=O)CO)[nH]nc2ncnc(O)c12 c1(CNC(NC(C#C)Cc2ccccc2)=NCCOCC)cccc2sccc12 Cc1cnn(CC(=O)NC2(CNC(=O)CSC3CCOC3=O)CCCC2)c1 c12ccc(cc1)OCC(=O)N2.CC(C)S(=O)(=O)NC(C1CCN(CC(=O)O)C1)C c12ccc(cc1)CCNC(=O)NC2CCC.c1(C(=O)NC(C)(C)C)cnn(C)c1F C1(N(C(COC(CC)C)=O)CCF)CCCN(C(C2COCCN2CC)=O)C1 C(=O)(C1=CC2(CCOC2)C1)NCCn1ncc(C(N2CCC(C)(N(C)C)C2)=O)c1 CC(CC(=O)N1CCC2(CC2)CC1C(=O)NCC(C)N(C(C)C)C1CC1)C(C)(C)C C=CCC(CNC(=O)C=CC1CCC1)C(=O)NC1(CC(C)C)CC1 C=CC(C)(CC)C(=O)N1CCC(CNC(c2cnn3c2OCC3)=O)CC1 N1(C(CNC(=O)OC)=O)CC(CNC(C2CC3CCC2CC3)=O)OC2(CCC2)C1 Cc1cc(C(N2CCCC(CO)(NC(=O)C=C3CCC3)C2)=O)c2ccccc2n1 CC1CCC(CC(N2CSCC2C(=O)NC(C)(CO)C2CCCC2)=O)CC1 CC(CCCCNC(C1CC(=O)N(O)C1)=O)N(C(C1(CCS(N)(=O)=O)CC1)=O)CC N1(C(Cc2cc(CC)no2)=O)CCC=C(C(=O)NCC23CCCCC2C3)C1 C12(OC)CC1CN(C(c1cnc(CO)o1)=O)C2.C(=O)(CC1(CO)CC1)N Cc1cc(C(=O)NCCCOCCCNC(c2cncs2)=O)c2c(c1)CCO2 C1(CC(=O)N(C)C)CC2(CCN(CC(=O)NC3CCC3)CC2)CO1 c1(NC(c2nc(C(C)OCC)sc2)=O)ccccc1-c1noc(C(F)(F)F)n1 c1(C(N2CC(SC)C(NC(c3conc3C(C)C)=O)C2)=O)cc2c(ncn2C)s1 C=CCC(C(=O)NC(C)(C)C(C)CC(=O)NCC(c1ccccc1)F)C(C)C C1(CC)CN(C(c2cc(CNC(=O)CCOC(C)C)ccn2)=O)CCS1 CC1(C(=O)NCC(=O)NC2CC2)CCC(=O)C1.C1C(=O)NCCO1 C(C(=O)NCC1(CN(C)C(C2(C)CCCN2C(C)C)=O)CC1)(C(C)C)SCC C(=O)(C1c2ccccc2C2CC1C2)N1CCN(C(C2CCCC(C)C2)=O)CC1C C=CC(C)CC(=O)N1CCCC(CCNC(c2ccn(C(C)(C)C)c2)=O)C1 N1(CC(=O)N(c2ncc(C)cc2Cl)CCO)C(=O)NC2(CCCC(C)(C)C2)C1=O N1(C(c2ccc(OCCOC)cc2)C(=O)NC2CC2)CCOCC(O)C1 C(CS(C)(=O)=O)(C(=O)O)n1cc(NC(CSCC(=O)NC2(C)CC3(CC3)C2)=O)nn1 c1(N(CCNC(C2(C)CCCCO2)=O)CC)ncnc2c1nnn2CCOC C(=O)(CC(O)CC(C)(C)C)N(CC(C)(C)CNC(C1(C)CC(C)(C)C1)=O)C C1(Nc2cc(C#N)sc2)CN(C(c2cn3ccccc3n2)=O)CCC1(F)F C(=O)(CCCC(F)(F)CO)N1C(C(C)NC(=O)CC2CC2(C)C)CCCC1 N1(C(c2nc(CNC(C3(CC#C)CCCO3)=O)oc2)=O)CC2(CCC2O)C1 C(CNC(=O)CC1CC(SC)C1)(C(C)(C)C)NC(C1CC(C)(CC)C1)=O N#CC1(O)CC(C(N2CCCC2C2(NC(c3ccoc3)=O)CC2)=O)C1 C1(C(=O)NC(C(C)SC)C)CC2(CCC2)CN1C(=O)C(C)N(C)C c1(OC)cc(C)c(C(N2CC(C)=C(C)C2)C(=O)Nc2ccccc2)c(C)c1 C=CCCCC(=O)N(CCC(C(C)C)NC(c1ccn(C2CCC2)n1)=O)C c1(OC)nc(C)cc(=NC2CC(n3ccnn3)C(O)C2)[nH]1.C1(=O)CCN1 C1(NC)CCCCC1CCO.C(=O)(C(=O)N1CC(OC)C1)NC O=S1(=O)CCCC(n2nc(-c3cccnc3)nc2-c2cc(C3CC3)no2)C1 CC1CCN(C(=O)C(F)C2CCCC2)C1C(=O)Nc1cnn(C)c1C(N)=O C(=O)(CC(F)(F)F)NC1C(CNC(=O)C=Cc2cn[nH]c2)C1 c1(N2CCOCC(NC(c3cnc(CC)nc3O)=O)C2)nc2ccc(F)cc2o1 C1(C(C(=O)NCCC2CC2)N(CCN=[N+]=[N-])C)CCCCC1(C)C c1(NC(=O)NC2CCCC2CNC(=O)NCC(F)(F)F)ccc(O)nc1 C(CC(C(C)C)(c1nnnn1Cc1cccs1)NCC1CCN(C(C)=O)C1)OC C(=O)(C(O)CCCNC(c1cnnn1C)=O)NCCc1cn(C)nn1 N1(C(C2OCCN(C)C2)=O)CC2C3CCC(C2C1)N(C(c1cc(N)ccn1)=O)C3 c1(C(=O)NCC2N(C(C(COC)N(C)C)=O)CCN(C)C2)nccn2ccnc12 c1(C(=O)NC(C(=O)Nc2c(C)nc(F)cc2)C)cnn2ccccc12 C(=O)(C(F)(F)CF)N(C1(CNC(CN2CC(C)C2)=O)CCCC1)C1CCCC1 N1(C(C(CCC)OC)=O)CC(NC(=O)C=Cc2ccsc2)C2(CC2)C1 C1(=CC(=O)NCCC(C)NC(=O)C2=CCCS2)CCCCCC1(F)F c1(C(=O)NC(CCC)C(=O)NCC#CCCO)cnn2c1OCC2 c1(CNC(C=CC(=O)OCC)=O)n[nH]c2c1CN(C(=O)CN(C)C(N)=O)CC2 C(=O)(C1CCCc2ncc(C)n21)N1CC(CC)N(C(=O)COCCF)CC1 C(=O)(C1=CCCC1(C)C)NCC(CCNC(c1nc(C)nn1C)=O)(C)C C#CC1(O)CC(C(=O)NCC(C)CN(C)C(c2cc(CC)oc2C)=O)C1 c1(SC)ncc(C(F)F)c(CN)n1.c12ccc(cc1)OCCSC2.SCC CC(C)CC(CSc1ccccc1)C(=O)NC(c1cc(C(C)(C)C)on1)=O c1(C(=O)NC(C)CC2CN(C(C3CSCCS3)=O)C2)cc2c(cn1)OCCO2 N1(C(C2N(C(C(C)(C)NC(=O)OC)=O)CC(O)C2)=O)CCC(O)CC1C C1(CC=C)(C(=O)N(CCCCCNC(=O)C(O)Cc2[nH]cnc2C)C)CCCC1 CC(C)C(F)(F)CC(=O)N(C1CCN(C(=O)CCC2CC2(Cl)Cl)CC1)CC1CC1 C(=O)(CCC(=O)c1cc(C)sc1C)N(CC(CC)NC(=O)CS(N)(=O)=O)C C(=O)(C(C)=CCNC(=O)COC1(C)CCC1)N(CCCNC)C C(=O)(CCCC(F)F)NCC(C)CN(C)C(c1ccc[nH]1)=O c1(C(=O)NC(CNC(CC(CC)C)=O)C2CCC2)cc([N+](=O)[O-])c2nsnc2c1 Cc1cn2c(=O)c(C(N3CCN(C(c4ccnn4C)=O)C(CO)C3)=O)cnc2s1 CC(O)(CC(=O)NC1CC(CNC(C2CCCC2S(C)(=O)=O)=O)C1)C(F)(F)F c1(C(N2CCC(c3n(CCOC)c(S)nn3)CC2)=O)cc2c(Br)cccc2[nH]1 c1(OCC)cc(C(=O)NC2CC2C(=O)NC)ccc1OC.c1(SCC)ccccc1I C1(N)Cc2cccc(Br)c2C1.c1(C(=O)NCC)cccc(CNC(=O)OC(C)(C)C)c1 c1(C(=O)NC(C2CN(C(C3(C)CCSCC3)=O)CCO2)C)cc2n(n1)CCC2 c1(C(=O)NC(C)Cn2cc(CCC3CCCCO3)nn2)ccc(OC(F)F)cc1 c1(SC)nc(N2CCCC2CC2CCCN(C(=O)C#CC3CC3)C2)cc(C)n1 N1(C(N)=O)CCN(CC(c2cn(CCC3CCO3)nn2)C2CCCC2)CC1 C(=O)(N1CC(C)(O)CO1)C1CC(NC(C(COC)(C)OC)=O)C1 c1(NC(=O)NCC(C)(C)C2=CCCC2)ccccc1S(=O)C(F)(F)F c1(C(N2C(CNC(C(C=CCCC)O)=O)CC2)=O)ncc2ccccc2c1N c1(CNC(=O)NCc2cccnc2-c2cncc(F)c2)ccc(O)c(Br)c1 Cc1nn(C)c(Cl)c1C(=O)NCC(CO)NC(c1cnsn1)=O C#CCC(C(=O)NCC1(CNC(C2C(C)C2(F)F)=O)CC1)C1CC1 C12(C(=O)NC(C)CCC(=O)NCC3CCC3(F)F)CC(C)(CCO1)C2 N1(C(c2cc(CC)nn2C)=O)CCN(C(=O)C=Cc2cscn2)C(CO)C1 N1(C(C(=O)NC2C(C)CN(C(=O)C=CC3CCC3)C2)C)CCP(C)(=O)CC1 C1(CNC(C2C(C)(C)C2)=O)C2CCC(C2)N1C(c1csc(N(C2CCC2)C)n1)=O C(CC(C(=O)N1CC(C(=O)NCC2(C#N)CCCC2)C(C)C1)OC)OC Cc1ccc(C(O)CCNC(=O)CCc2nc(C(C)(C)C)no2)s1 Cc1cc(C(N2CC(NC(c3nsnc3O)=O)CCC2C)=O)cn(C)c1=O C1(C(=O)NC2CCC(C(=O)NCCCC(C)C)C2)(OC)CCSC1 Cc1cc(C)c(C(N2CCN(C(=O)C3=NOC(C)(C)C3)CC2)=O)c(S)n1 C(=O)(C1CCCc2c(I)n[nH]c21)N1Cc2c(cc(OC)c(OC)c2)C1 S(=O)(=O)(c1ccc2ncsc2c1)N1CC2CN(C(C(C)NC(C)(C)C)=O)CC2C1 N1(C(C2C(OC)CCCC2)=O)CCN(C(C2CN(C(=O)NC)C2)=O)C(C(C)C)C1 c1(OC)cncc(C(=O)NCC2CCCC(NC(=O)CCOC(C)C)C2)c1 N1(CCC)CCCCC1C(=O)NCCCN(C(c1cc(C(=O)OC)cs1)=O)CC Cc1ccc(-c2noc(CNC3CC(NC(C4CCCO4)=O)C3)n2)cc1 N1(C(C=C(C)C)=O)CCCC2(CCC(NC(=O)Cc3cncs3)C2)C1 C1(CNC(CCCCOC)=O)C2CCC(C2)N1C(c1cccc(Cl)c1F)=O C1(C(=O)NC(COC)C(=O)OC)CCN(C(c2conc2C)=O)C12CC2 c1(C(=O)NCC(CNC(C(C)c2ccon2)=O)O)ccc(O)cc1 C=CCC(C(=O)N(CC(C1CCC1)OC)C)NC(c1cccnc1S)=O C(CCCCC(=O)NC(C(F)(F)F)C1CC1)NC(C1N(CC)CCOC1)=O C1(C(NOCc2cn(-c3ccc(C)nc3)nn2)=O)CC(=O)NC1(C)C C(CCCCC(=O)N1CC(C)(C)CC1CCO)N(C)C(c1ccccc1F)=O c1(CC(=O)NC2CC(C(=O)NCC3(CCC)CC3)C2)ccccn1 c1(C(=O)NCC(CC=C)NC(=O)CN2CCOCC2)ccc(CC)c(F)c1 c1(NCC2CCCC3CN(C(CCCC)=O)CC32)nc[nH]c2ncc(C(N)=O)c1-2 CC1CC(NC(=O)C(F)(F)c2ccccn2)CN1C(=O)CN1CCC(C)(C)C1 Cc1nc(=N)[nH]c(=NCC(C)C(=O)Nc2cnc3cnc(Cl)cc3c2)[nH]1 C=CCC(CNC(c1ccnc(C)c1N)=O)C(=O)NCCN(C)C1CC1 N1(C(CN2CC(C#N)C2)=O)CCC2(NC(=O)Cc3ccc(C(N)=O)cc3)CC2C1 c1(N2C(CNC(C(c3ccccc3F)(C)OC)=O)CC2)cc(=O)n(C)c(=O)n1C N1(C(C(C)OCCC=C)=O)C(CNC(=O)COCC2CCCO2)CC2CCCC12 C1(CC)(CO)CCCN1C(=O)NC(C1CCOC1)CO c1(C(C(=O)NCCC2CC(NC(c3nc(CC)sc3)=O)C2)O)ccc(Cl)c(Cl)c1 c1(CNC(=O)NCc2c(OC)ncc(Br)c2)ccc2c(c1)CCCO2 N1(CC(=O)N(CCNC(=O)Cc2cccs2)CC)CCC(C)(O)C1 N1(C(CSCC#C)=O)CC(C(NCP(C)(C)=O)=O)CCC1C c1(C(N2CCC(OCCNC(=O)CCC3CCC3)C2)=O)cc(F)cc([N+](=O)[O-])c1 CC(C)C1=NOC(C)(C(=O)NC2CCCC(NC(=O)Cc3cnoc3)C2)C1 C1(C)(C(=O)NCCCCCNC(c2c(OC)ncnc2)=O)Cc2ccccc2N1 C12(CNC(CC(c3ccccc3F)C)=O)CCC(NC(=O)CC3(C)CC3)(CO1)C2 C=C(C)C1OCCC1C(=O)NCCCC(N1CCN(C)CC1C)=O c1(C(=O)NCC2(C)CCCN2C(C2CC(C(F)F)C2)=O)nc[nH]c2ncnc1-2 CC1CC(CNC(=O)C(F)n2ccnc2)CN(C(=O)CCSc2ccccn2)C1 C(CN=C(NCC1C(c2cn(C)nc2)OCC1)NC1CCC1)SC1CC2(CC2)C1 N1(C(CC2(C=C)CC2)=O)CC2CCCC2(NC(c2cc(N)c(Cl)c(O)c2)=O)C1 Cn1cc(C=C(F)C(=O)NCc2ccc(CNC(C3C4COCC34)=O)cc2)cn1 N1(C(c2onc(C)c2C)=O)CC(NC(=O)CC2(C)CCCO2)CC2(CCC2)C1 CS(=O)(=O)c1ccc(Cl)c(S(=O)(=O)N2CCCC2c2ncon2)c1 N1(C(c2n(C)ccn2)=O)CCCN(C(c2cc(C(F)(F)F)ns2)=O)CC1 C1(NC(c2cc(C)ncc2)=O)CCN(C(C2CC2C2CC2)=O)C12CCC2 N1(C(COCC(N)=O)=O)CCC2(CNC(=O)CNc3ccccn3)CC2C1 C1(CC#N)CCCN(C(=O)Nc2ccc(OCCCc3ccc(Cl)cc3)cc2)C1 C(CS(N)(=O)=O)NC(CCC1(C)CC1)=O.C12(CCC1)CC=CC(=O)N2 c1(C(=O)NCC2CCCN(N3CC(CCCCSC)C3)C2)ccc(OC)cc1N c1(OC)cc(C(=O)NCC(C2CCCCC2)NC(=O)CC(C)F)cc(OC)c1O C=C(C)C1CN(C(C23CC(C)(CN2C(c2ccnnc2)=O)C3)=O)CCO1 C(=O)(CC(C)CC(F)(F)F)N(C(CCCC)CNC(=O)C(C)(C)C(=O)NCC)C c1(CC)cc(-c2ccc(C(N3CC(F)CC3C(=O)OC)=O)nn2)ccc1F C1(CC(=O)NC2CC3CN(C(C4(O)CCSC4)=O)CC3C2)CCCC2(CCC2)O1 C1(O)(CNC(c2c(OCC)ccs2)=O)CCCN(C(c2scnc2Cl)=O)CC1 C(=O)(C(C)(C)CCCO)NCC(CCOC)NC(C1COCCC1(F)F)=O C(=O)(C1CCc2cc(F)ccc21)N1CCC(F)(CNC(C2C(=O)NCC2)=O)CC1 C12(NC(c3c(C)n(CC(F)F)nc3)=O)CCCN(C(=O)CSS(C)(=O)=O)CC1C2 c1(CC(=O)NCCCOCCNC(C2CSCCS2)=O)noc2cc(F)ccc12 c1(C(C)NC(C(Cc2cc[nH]n2)NC(CC=C=C)=O)=O)ccccc1F C(CC(N)=O)(C(=O)NCCN1CC2CCC1C2)NC(C1(C#N)CCOC1)=O CCC(C)CC(=O)NC1CCCC1CC(=O)NCc1ccncc1Cl C1(C(=O)NC2C3CN(C(C4C(C)(C)CCC=C4)=O)CC32)CCC(C2CCCO2)O1 c12ccccc1C(=O)N2.c1(C(C(=O)OCC)OC)cn(C2COCC2O)nn1 c1(OC)cc(C)cc(C(=O)NC2CC(NC(c3cc(C(C)=O)c[nH]3)=O)C2)c1C C1(O)(CNC(=O)CC2CCOC(=O)N2)CCCN(C(=O)CC(=O)NC2CC2)C1 n1(C(C)C)ncc2c1C(NC(=O)C(N1CCC3(CNC(=O)C3)C1)=O)CCC2 CC(C(=O)NC1CC(C)(NC(c2cc(-c3cccs3)on2)=O)C1)S(N)(=O)=O C12(NC(C3CCCC3)=O)CCCN(C(=O)CCc3cc(Cl)cs3)CC1C2 C1(C2CC2)(C(=O)NCC2CCC(=C)CC2)CN(C(=O)CC(C)n2cccn2)C1 C1(F)(CNC(CN(C(=O)CC2CC2)C)=O)CCC1 C1(CNC(=O)CC2CCC=CCC2)CCC2CN(C(c3ccc(F)cc3)=O)CC12 C#Cc1cccc(NC=O)c1Cl.N12CCCN(C(C)C1)CC2.S(C)(=O)(=O)N N1(C(C(CC=CC)C)=O)CCOCC(C(N2CC(OCC(C)C)C2)=O)C1 C(=O)(C(C)(C)C1CC1)NCCC1CC(C(N(CCOC)CC)=O)C1 C(=O)(CCCC#N)N(CCCN(C(=O)CCC1CC1(Cl)Cl)Cc1ccccn1)C c1(C(N(C2CN(C(C(=O)NCC)=O)CC2O)C)=O)ccn2c(C)cnc2c1 c1(N(C2CNCC(F)(F)C2)C(=O)Cc2c(Cl)cccc2Cl)ncc2[nH]ccc2n1 N1(CC(=O)N(CCSC)CC)CC(=O)Nc2ccccc21 C1(NC(c2cccnc2F)=O)CCC2CN(C(C3CC4C(C3)C4(F)F)=O)CC2C1 CC(C)C(C)(CNC(C1CC(C)N1C(=O)CCNC(=O)CO)=O)C(C)C c1(C(=O)NCC(C)N(C(=O)C(Cl)=CCl)C)ccnc(N2CCC(C)C2)c1 CCCC(C(O)C(=O)NC1(C(C)C)CCC1)NC(c1coc(CC)n1)=O.C(C)=O Cc1ccc(CC(N2CCC(N(CCO)C(C3(C)C=CCC3)=O)C2)=O)c(Br)c1 Cc1ccc(CC(=O)NCC2CN(C(=O)CC3COC(=O)C3)CCO2)c(Cl)c1 N1(C(CCc2c(C)n(C)nc2)=O)CCC(NC(=O)C(=O)NCC2CC2)CC(O)C1 c1(SCC(=O)N(CC)Cc2ccccc2)cncc(C(=O)OC)c1 N1(Cc2ccc(NC(=O)OC)nc2)CC(NC(C2CCC(=O)N2)=O)CC(F)(F)C1 N1(C(Cc2c(OC)cccc2)=O)CCC2(CC2C(=O)NCCCCF)C1 N1(C(c2ncc(C)nc2)=O)CC2CCN(C(=O)CC3CCS(=O)(=O)C3)CC2C1 n1(CC(=O)N(C(C)C(=O)N(C)CC2(C)CCCO2)CC)cc(Cl)cn1 C1(C(N2CCC(NC(C(CC=C)C)=O)(CC)CC2)=O)CCCCC(F)(F)C1 CCC(O)CC(=O)NCCCOCCC(=O)Nc1cccc(Cl)n1 Cc1cc(O)ncc1C(=O)NCCCN(C)C(C1CCCN1C1CCC1)=O C1(C)(C(=O)NC(C2CN(C(=O)CC(c3cccs3)N(C)C)C2)C)CC(C#N)C1 C(c1ccc(F)cc1F)=CC(=O)NCC(CNC(c1cnnc(O)c1)=O)OC c1(C(N2C(C(=O)NC(C#N)C(N)=O)CC2)=O)c(F)cc(Br)cc1Cl C1(C(N(C(C)C)CCNC(=O)C(C)CF)=O)C2CC1(c1ccccc1)CO2 N1(C(CCCCC=C)=O)CCC(C2CC2)(CNC(c2nnc(C)s2)=O)C1 C1(COC)CCCCC1N(C)C(c1cc(CCNC(c2nc(Cl)cs2)=O)on1)=O c1(CNC(C(F)=C(C)C)=O)ccc(C(=O)NCCN2CC3CC3C2)o1 C1(C(=O)NC(C(=O)N(CC=C)CC)CO)CC12CCOCC2 c1(C(=O)NCC2(F)CN(C(CC3CC(=C)C3)=O)C2)ncncc1OC c1(NC)c(N=[N+]=[N-])cnnc1O.c1(CCCC)ccccc1 c1(C(C(=O)O)NC)ccccc1.C(C(CC1CCCC1)CO)NC(C(=O)OCC)=O C(C(CC)(CC)NC(=O)CC1CCC(=O)NC1)NC(C(CC)C1CCC(=O)N1)=O c1(C(C)(C)C)cccc(C2(O)CN(C(=O)Nc3c[nH]nc3C3CCOC3)C2)c1 C(CC(C)(C)C)(C(=O)NCc1cncc(C(N2CCC(C)(C)C2)=O)c1)OC c1(N2CC(C3(N4CCN(C)CC4)CC3)C2)nc(NCC(=O)NC)c2ccsc2n1 C1(C(=O)NCC2(O)CCN(C(Cn3c(C)ccn3)=O)C2)CN2CCN1CC2C CC(CC(N)=O)C(=O)NC(C1CCCN(CC2CN(C3CCOCC3)C2)CC1)=O C1(C(N2C(CCNC(CNC(C3C(C)C3)=O)=O)CCC2)=O)CC2(CSC2)C1 CN1CC2(CC2)CC1C(=O)NC(CC1CCCC1)C(=O)NCC1CCCC12CC2 c1(NC(C(CCOC)NC(c2ccc(CC)[nH]2)=O)=O)cc(F)ncc1OC(C)C N1(C(CSC)=O)CC2CCC2(CC(=O)N(CCCC(F)(F)F)C)C1 c1(C(=O)NC2C(C)CCN(C(c3nncn3C3CC3)=O)C2)ccn2nnnc2c1 C(=O)(CC(C)(C)CNC(C1CN2CCC1CC2)=O)NCC1CCCC(C)C1 c12cn(nn1)CCCN2CC.c1(C(=O)NC)cc(CC)no1.C1(=O)C(O)N1.CCO C(=O)(C(C)C(F)(F)F)N(C1CCN(C(c2coc(SCC)n2)=O)C1)CC#C C1(C(=O)NC2C(NC(C(c3ccc(OC)cc3)O)=O)CCC2)COCC(C)(C)O1 C12(NC(c3n[nH]c(C)c3Cl)=O)CCCN(C(=O)C(C)(C)C(N)=O)CC1C2 C(=O)(C(CNC(C1CCCCO1)=O)N(C)C)NC1(C(C)C)CC1 CN1CCCC(CN(C)C(c2conc2CNC(c2cc(C3CC3)[nH]n2)=O)=O)C1 CC1CCC(C(=O)NC2CCC(C(N3CCCC3CCC(C)(C)C)=O)C2)O1 N1(S(CC(=O)OCC)(=O)=O)CC(NC(c2c(F)cccc2I)=O)CC(C)C1 C(=O)(C(CC1CCCC1)NC(C1CC1C(=O)OC)=O)NCC=CC Cc1ccc(C(C)N(C(=O)CNC(=O)CCCN(C)C)C)c(C)c1 c1(COC)cccc(CC(=O)NC(C)(C)C(C)NC(c2coc(C3CC3)n2)=O)c1 C(=O)(C1=CCOCC1)NCC(N(C(=O)C(=O)Cc1cccc(Cl)c1)C)C1CC1 N1(C(C(c2cc(C)oc2C)C)=O)CCC(O)C(NC(=O)CN2CCC(C)(O)C2)C1 CC(C)C(C)CC(=O)N1C(=O)CCC1COC(c1cccc(O)c1)=O c1(CC)cccc(CC(=O)NCCC2CC(OC)CN2C(=O)C=C(C)C(F)F)c1 C(CNC(=O)CSCC1CCCO1)(CC(F)(F)F)NC(=O)CC1CC1 Nc1cc(C(=O)NCC2(NC(=O)CC(F)(F)F)CC2)cc(O)c1Cl C1(NC(CSCC#C)=O)CCN(C(c2csc(C(=O)NCC)n2)=O)CC12CCC2 c1(C(=O)OCCCC)ccc(Cl)cc1NC(=O)NC1CCC(C(C)C)C1 C1(NC(=O)OC(C)(C)C)(CN(CCOC)CC)CCCC(C)(C)C1 n1(CC)nc(C(=O)N(CC(C)O)CCNC(=O)C(O)c2cnc[nH]2)c(C)n1 C#Cc1cnc(C(=O)NC(CC)CCC(=O)N2CCC(N3CCCC3)C2)c(C)c1 C12(C(=O)NCCc3cocn3)CCC(CC1)N(C(C1(O)CC3CCC1C3)=O)C2 c1(CC(=O)NCC2C(NC(=O)CCc3nncs3)CC2)ccn(C(F)F)n1 n1(CC(N2CC(NC(C34CCC(C3)C4)=O)CC2CO)=O)ncc2ncccc12 N1(C(=O)CCn2ccc(O)nc2=O)CCCC2(C1)CN(C(=O)CC1=CCCC1)C2 c1(C(C)C)cccc(C(N2CCC(NC(c3cc(Cl)c[nH]3)=O)C(C)C2)=O)c1N Cc1cc(Cl)c(C2CCOC2)cc1C.C(C(O)CO)N(C(CN1CC1)=O)C C12(CCS(=O)(=O)C1)C(=O)N2.c12nc(cs1)C2.N1(C(=O)OC(C)(C)C)CCCC1 Cc1cc(=NC2CCc3cccnc32)[nH]c(=NCCc2ccco2)[nH]1 C(=O)(C1CCCn2ccnc21)N1CC(C)N(C(c2ccc[nH]2)=O)CC1C c1(C(=O)NC(C(=O)NC(COC)CO)c2ccco2)cnc(C)nc1C c1(C(N2CC(CC)N(C(=O)COC(C)C)CC2)=O)cc2c(s1)C(C)(C)CCC2 NC1CC12CCN(C(c1ccc(C3(C(F)(F)F)CC3)cc1)=O)CC2 S(=O)(=O)(c1ccccc1C(F)(F)F)NC1OCN(C)C(C(F)(F)F)C1 CC(C)CC(O)C(C)C(=O)N1CCC(NC(c2ccc(CO)s2)=O)C1C(C)(C)C N1(CC2CCCC(C(=O)OC)C2)C2CCC1CC(=O)NC2 C1(NC(c2cccc(OC)c2)=O)CC2CN(C(=O)Cc3nncn3C)CC2C1 CC1(C)CN(S(=O)(=O)N2CCC(C(=O)OC(C)(C)C)C2)CC(CCO)O1 C(=O)(C1SCCc2ccccc21)N(C)CCN(C(=O)C1=NOC2(CCOC2)C1)C C1(CNC(C2C(CC)C2)=O)CCN(C(=O)CCC(=O)c2ccccn2)C12CC2 N1(C(C(C(C)C)O)=O)CCC2(CCOCC2)C(NC(=O)CC2CC3CCC2O3)C1 C#CCC(C(=O)NC(C)CCNC(c1cnc(Cl)n1C)=O)C1CC1 S(=O)(=O)(c1cccnc1N1CCC(F)(F)C(F)C1)NCC(OC)OC N1(C(c2n(CC)nnc2)=O)C(C(=O)N(c2ccccc2)CCO)CCC1C c1(C(=O)NC2C(CNC(=O)CCc3nc[nH]n3)COC2)cc2ncccc2o1 CCC(CC)CC(c1nnnn1CC1CC1)NCc1ccoc1C C(CCCC(CO)NC(=O)CC(=O)N(C)C)NC(c1cccc(OCCC)c1)=O Cc1cccn(CC(=O)NC2CN(C(=O)C=C3CCC3)CC2(C)C)c1=O C(=O)(C1=CCC(NC(C2(O)CCC2)=O)C1)NCC(CC)N1CCCC1 c1(OC)ccc(F)cc1-c1cn(Cc2cc(C(C)(C)C)n[nH]2)nn1 S(=O)(=O)(c1cccc(F)c1)N1CCC2(C(NC(c3ccc(C)cc3C)=O)C2)CC1 CCC(C)CCC(=O)NCC1C=CCN1C(c1nn(C)cc1Cl)=O CCCCC(=O)NC1CCN(C(C23CSC(C2)C3)=O)C1 Cc1csc2c1CN(N1CC(c3c[nH]c4cnccc34)C1)CC2O CCCN=C(NCC(O)CN1CCCC1)NC1CC(OC(C)(C)C)C1.OC c1(C(N(CCCNC(C2CC(C3CCC3)C2)=O)C)=O)ccc(S(N)(=O)=O)cc1F n1(C(C)C(=O)NCC(C)(C)CC2CC2)cc(Br)c(CC2CC2)n1 c1(C(=O)OC)cc(=NCC(C)SC)nc(-c2ccncc2)[nH]1 C1(C(C)NC(C23CC(C#N)(C2)C3)=O)CCCN(C(=O)Cn2cnnc2O)C1 C1(NC(CCCOCCOC)=O)CCC(C)(CNC(c2csc(S)n2)=O)C1 C1(CC)CC(O)CCN1C(=O)CCCC(C)NC(=O)CC1OCCO1 CC1(C)CC(NC(c2ncoc2C2CCCO2)=O)CN1C(c1ccccc1O)=O c1(NC(c2c(-c3c(C(=O)O)scc3)cccc2)=O)c(OC(F)(F)F)cccc1O C1(NC(c2ncc(OC)nc2)=O)CCC2CN(C(=O)Cc3n[nH]c(C)n3)CC2C1 N1(C(C(C)SCC)=O)CC(C(=O)NC(c2ncc[nH]2)C)C2(CC2)C1 c1(C(=O)NCC2CN(CC(=O)N(C(C)C3CC3)C)C2)cc2cccnn2n1 c1(C(N(C)CC2CCN(C(c3c(CC)c[nH]c3)=O)C2)=O)cc(F)ccc1C(F)F Cc1csc2ncc(C(N3CC(C(C)NC(c4coc(C(C)C)n4)=O)C3)=O)n12 c1(CC(N2CCC(c3cccs3)CC2)=O)cnc2ccccn12 N1(C(C2C(C)(COC)C2)=O)CC2(C1)CN(C(=O)CSc1cccc[n+]1[O-])C2 N1(C2CN(C(C)C)C(=O)C2)CC=C(COc2cc(-c3ccccc3)ncn2)CC1 C(C1=CCN(C(=O)CN2CCCC(CC)C2)CC1)NC(C(CCOCC)OC)=O c1(CCNc2cc(C(=O)OCC)ncn2)c(Cl)nc2sccn2c1=O CC1C(C(=O)NCC2(F)CC(NC(=O)C(C#N)C3CC3)C2)C1(F)F Cc1cc(CC(=O)N(CC(C)NC(c2c(Cl)csc2Cl)=O)C)cc(C)c1 C(=O)(CS(=O)(=O)CCO)N(C1CCCN(C(=O)CCc2cncs2)C1)CC c1(C(=O)NC(CN(C(c2cccc(SC)c2)=O)CC)C)ccc(N)c(F)c1F C1(C(=O)NC2CCC(N3CCOCC3)C2)(O)CCCC1.CC(C)(C)OC(=O)NC c1(CC(C)C)ncc(C(=O)NC(CO)C(C)NC(c2ccc(C3CC3)o2)=O)s1 c1(OC)cc2c(cc1C(=O)NC1CC1NC(c1ccccc1F)=O)CCC2 C1(CNC(CN(C)CC)=O)CCN(C(=O)COc2ccc(F)c(Cl)c2)C12CC2 C1(C)(CNC(C(C)c2ccco2)=O)CCC(NC(=O)C=Cc2ccsc2)CC1 C(CN=C(NCc1ccco1)NCC1CC2CCC1CC2)SC c1(SC)ccc(C(=O)N(CC(C)N(C)C(C2CCN(C)C2=O)=O)C)c(Cl)c1 N1(C(C2CC23CCOCC3)=O)CCC(O)C(F)(F)C1.c12c[nH]nc1CCNC2=O C1(C(=O)NCc2ncccn2)CCC2(CC2)N1C(=O)C=Cc1cccnc1 C1(O)(CN(CC(O)(CO)CO)C(=O)NC(C)(C)C)CCCN(Cc2n(C)c(Cl)cn2)C1 c1(C(=O)NCCCC(C)NC(c2cc(SC)oc2)=O)cccc2c1NCC2 N1(C(C(C)Cn2ccnc2)=O)CCCC(C)(NC(C2CCCC(C)(C)O2)=O)C1 C1(NC(C(c2cn(C)nc2)=O)=O)CC2CCC1C(NC(=O)C(F)CC1CCC1)C2 c1(C(=O)NCCC2(NC(CN(CCC#C)C)=O)CC2)snnc1C c1(CC(=O)NCC2CC2CC2CN(C(=O)C3=CCCC3)CCO2)cc(F)cc(Cl)c1 C1(C(C)NC(C2C(OCC)C2)=O)CCN(C(C2CCN(C(C)(C)C)CC2)=O)CC1 N1(C(C(CC)OC2CCCC2)=O)CCC(CNC(c2ccc(C#N)o2)=O)C1(C)C N1(C(CN(CCC)C)=O)CCC(C)(C)C(NC(=O)CCC2CCCN(C)C2)C1 CN1CCCC(O)(CC(=O)NCC2CCC(NC(=O)CC3CSCCS3)CC2)C1 CCCCC(CC)CC(=O)N1CC(F)CC1C(N1CCN(C2CC2)C(C)C1)=O N1(C(C(C)(C)F)=O)CCC2(CCCN2C(C2CCC3CC23)=O)C1 c1(C(=O)NC2CC(NC(c3c(C)onc3Cl)=O)C2)cc2ccccc2oc1=O CC1CCCC=C1C(=O)N1CC2CCC(C(=O)NCCc3ccon3)(C2)C1 c1(NC(=O)NCCCCCC)cccc2c1NC(=O)CC2 C1(C(=O)NCC2CN(C(c3nnc(CC)s3)=O)CC2C)CC(C2CC2)=NO1 N1(C(c2n(COC)ncc2)=O)CC(NC(=O)C(C)(C)Br)C(SC)C1 C1(NC(C(C)OC(C)=O)=O)CN(C(=O)CCC2(C)CC2)CC1n1ccnn1 C=CCCCCC(c1nnnn1C1CC1)Nc1cc(Cl)c(Cl)c(Cl)c1 C1(CC(C)NC(=O)C(c2cncnc2)C)CCN(C(=O)C2=CCSC2)CC1 c1(C(=O)NC(C(CO)NC(CCSC)=O)C)cnn(Cc2cccs2)c1C c1(C(=O)NCC2N(C(C3C(C)CC=CC3)=O)CCOC2)ccc2nonc2c1 N1(C(c2cnn(C(C)C)c2N)=O)CCN(C(=O)Cc2ccc(Cl)s2)CC(O)C1 c1(C(N2C(CC(=O)NCCC(C(C)C)N(C)C)COCC2)=O)cc(O)cc(F)c1 CC1CN(C(=O)Cn2ccnc2)CC(C(=O)NCC2(CO)CCCCC2)O1 C(C(C)C(F)C(=O)N1CC(C)(C#N)C1)NC(CC1CC(SC)C1)=O c1(-c2c(OCCCC)cccc2F)nc(C(=O)NC(C)(C)CO)n2ccccc12 C=CCC(C)C(=O)N(C1CCN(C(c2cc(C3(Cl)CC3)n(C)n2)=O)C1)C N1(C(c2nc(COC)oc2)=O)CCCC(O)(CNC(c2ccc(C)c(C)c2)=O)C1 C1(CNC(C2(COC)CCCCC2)=O)CN(C(=O)CCc2ccsc2)CCCO1 N1(C(C2CC(CN(C)C)C2)=O)CC2(CCN2C(=O)Cc2cc[nH]n2)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CCC(C)C)C(=O)NCCCSC(F)F Cc1cn(C(C)C)cc1C(=O)NC(C)CCCNC(c1nncs1)=O c1(NC(C(C)NC(c2c(C(C)C)n(C)nn2)=O)C(C)C)cnc2ccccc2n1 C12(CNC(=O)CCc3cncnc3)CC1CN2C(c1ccc(C2CCC2)cc1)=O Cc1nc(C(=O)NCC(C)(CC(C)C)NC(c2nc(C)oc2C)=O)cc(O)n1 C#CCC(O)C(=O)NC1CCN(C(=O)C(c2ccc(F)cc2)(F)F)C1.C1CNC1=O C1(C(=O)OC)CC2CCC1CC2NC(=O)NC(c1ccccc1)c1cscn1 S(=O)(=O)(CC(C)(F)C(C)(C)F)NC(c1cc(Cl)ccc1Cl)CC C1CC2C(C1)C2(F)F.N12CCCC1C(=O)NC1CCC(C1)C2=O.CS c1(C(=O)NC2CC3CN(C(C(C4CC4)OCC)=O)CC32)ccc2nnc(O)n2c1 C1(C(N2CC(CNC(c3c(C)ncs3)=O)OCC2)=O)COCC(=O)N1C(C)C CC1C(NC(c2nncn2C2CC2)=O)CCCN1C(C1CCCS(=O)(=O)C1)=O N1(C(CNC(=O)CNC(=O)Cc2c[nH]nc2O)=O)CCC2OCCC2C1 Cc1cc(-c2ccc(C(=O)Nc3ncn(C4CC4)n3)nc2)cnc1C#N c1(-n2c(Cc3cccc(C)c3)nc(CO)n2)cc(Cl)ccc1F.CO C1(F)(CNC(c2ccc(Cl)cc2Cl)=O)CCCN(C(=O)CSC2CCOC2)C1 C(CCCCCNC(c1ccc(C2CCOC2)s1)=O)NC(C1(CC#C)CCC1)=O CCCS(=O)(=O)c1ccccc1C(=O)NCC1COCCN1C(=O)CC1CSC1 CC1(C(=O)NCC2(CNC(c3cccnc3O)=O)CC2(F)F)CCC2CC2C1 C(CC(N)=O)(C(=O)NC(CC(C)C)C(N)=O)N(C(N)=O)C.CC(C)CC=O N1(C(c2cc(C3C(C)C3)on2)=O)CC(C2(NC(=O)Cn3cnc(C#N)n3)CC2)C1 c1(C(=O)NC(CC=C)CNC(=O)CNS(N)(=O)=O)ccnc(SC(C)(C)C)c1 c1(OC)c(Cl)cc(C(=O)N(C2CCN(C(=O)CC(C)SC)C2)C)nc1Cl C1(C(N(CCCN(C(C(C)NC(N)=O)=O)C)C)=O)CC1C1CCCC1 C(=O)(CCC(C)(F)F)NCC1N(C(C2(OC)CCC2)=O)CCC1C N1(C(C2C(CC(C)(C)C)C2)=O)CCCC(CCNC(=O)COC2CC2)CC1 C1(CNC(C2CCN(C)C2)=O)CN(C(=O)C=C2CCC(C)(C)CC2)CC(C)(C)C1 c1(NC2(c3ccc(OC)cc3)CCCC2)nc2cc(Br)cnc2s1 C1(C(N2CCC(C(C)(C)NC(c3n(C)ccc3)=O)C2)=O)CCCN(S(C)(=O)=O)C1 c1(C(=O)NC2(C)CC(NC(C(C)OCCCC)=O)C2)cc(SC)nn1C c1(OCC)cc(NCCN(CCOC)C(c2c[nH]c(Br)c2)=O)nc(C)n1 CC(O)C(N)C(=O)NCC1(CO)CC2CC2C1 c1(C(C)=O)cc(C(=O)NCC(C)(C)CNC(=O)CCOCC(F)F)cnc1C c1(C(=O)OC)cc2c(s1)CCS(=O)(=O)C2.c12cnc(cn1)Cc1nc-2no1 C1(NC(N2CCC(CC(C)(C)C)C2)=O)CC(=O)N(C)C1c1ccccc1 n1(CC(=O)NC(C2(CNC(=O)C(CCO)NC(N)=O)CC2)C)cnc([N+](=O)[O-])n1 C(CCNC(C12CC(n3cc(C4(O)CCCC4)nn3)C1C2)=O)(C(F)(F)F)N(C)C c1(C(=O)NCC2C(NC(Cc3cccc(CC)c3)=O)CC2)cc(O)ccc1Cl c1(NC(c2c[nH]c3nccc-3c2)=O)ccc(F)c(Cl)c1F n1(CC(=O)NC(CCNC(C2C(C)=CCC=C2)=O)C)nc2ccccn2c1=O N1(C(C(CO)N(C)C)=O)CCC(CC(=O)NCC2CCN(C3CC3)C2)C1(C)C CC1CN(C(=O)CC2(C)OCCO2)CC(C)N(C(c2ncccc2F)=O)C1 N1(C(CC2CC(OCC)C2)=O)CC2CCCC(CNC(=O)C#CC3CCC3)C2C1 N1(C(C(C)(C)OC)=O)CCC(O)(C(=O)NCCCCOc2ccccc2)C1 Cc1cc(C(N2CCCC(NC(=O)CNS(=O)(=O)N(C)C)C2)=O)nc2ccccc12 C(=O)(CCCCCC(C)O)NC(c1ccc(CNC(=O)CC=C(Cl)Cl)cc1)C C1(CC(=O)NC(C(C)NC(COC)=O)C)CCC(F)(F)CC1 N1(C(C2(C)CCC(C)C2)=O)CC2CCC1CN2C(c1ncoc1Br)=O C12(NC(=O)C3CC3)CCCC1N(C(=O)Cc1ccoc1)CC2 CCC(C)C(O)C(=O)N1CCC(F)(CNC(=O)Cc2cc(F)ccc2C(F)(F)F)C1 c1(OC)ccc(F)c(CN2CCCC(NC(C3(O)CC3)=O)C2)c1 Cc1cc(C)c(CC(N2CC3(C2)CN(c2cc4nncn4cn2)C3)=O)c(C)c1 Cc1cn2cc(C(N3CCC4CN(C(=O)CCCC(C)C)CC4C3)=O)ccc2n1 Cc1ccc(C2CC2NCCC(N2CCC(N3CC=CC3)CC2)=O)c(Br)c1 N1(C(C(C)OCCOCC)=O)CCC(CNC(=O)CC2CCCC23CC3)C(C)C1 c1(CNC(=O)NC(c2cccnc2)CN(C)C)[nH]nc2c1CCC2(C)C C#Cc1ccnc(C(N2CCCC(C(C)C(N3CCC(N(C)CC)C3)=O)C2)=O)c1 C(=O)(C(C)CC(C)(F)F)N(C)CC1OCCN(C(C(COC)(F)F)=O)C1 CCC(O)C(F)(F)C(=O)NC1CCCC(NC(=O)Cc2cccnc2)C1 N1(C(Cc2cccc(CC)c2)=O)CCN(C(=O)COC2CCOC2)CC1CC1CC1 C1(NC(c2coc(C(F)(F)F)c2)=O)CN(C(c2ccon2)=O)CC2(CC2)C1 CCCCCC(O)CC(=O)NCCC1CC(NC(c2cc(C3CC3)n(C)n2)=O)C1 c1(C(=O)NC2COCCN(C(=O)OC(C)(C)C)C2)cc(O)nc2ccccc12 CC(C)C(F)(F)CC(=O)NCC1(CNC(C2(C)CC3CC3C2)=O)CCC1 N1(C(c2cc(OC)cc(OC)c2Br)C(=O)NCC(=C)C)CC2CS(=O)(=O)CC2C1 C1(CC(N2CC(N(C(CC(CCSC)O)=O)C)C2)=O)CCCC(C)(C)CC1 C1(C(=O)Nc2n(C)c(Cl)cn2)CCN(C(=O)C(C)(C)CF)C1(C)C C(C)(C(C(=O)Nc1cc(Cl)ccc1O)C(C)C)NC(C(CC(C)C)=O)=O C1(CNC(c2cc(CC)[nH]n2)=O)CCN(C(c2c(C)cnn2C)=O)CC1C Cc1cc(C(=O)NCCCOCCNC(c2ccoc2C)=O)c(C)n1NC(N)=O c1(OC)ccc2c(CC(N3CCCC(N(C(=O)C(C)CF)C)C3)=O)coc2c1C CC(C)(O)C#CC(=O)NCC1CCCN(C(C2CN3CCN2CC3)=O)C1 C=CCCC(C(=O)N=c1ccn(C2CC2)[nH]1)NC(=O)C(O)C(F)(F)F C#CCCCCC(=O)NC1CCN(C(=O)C=CBr)C(C)C1 N1(C(CSCC=C)=O)CCC(O)(CCNC(=O)C(C)Sc2ccccn2)C1 C1(C)(OC)CCCN(C(C2CN(C(C3COCOC3)=O)CCO2)=O)C1 c1(CC(=O)NCC2N(C(C3C(C(=O)OCC)C3)=O)CC2)cc(F)ccc1O c1(C(N2CC(C(N3CC(OC(C)=O)C3)=O)C2)=O)ccc(-n2cccn2)cc1 C(CCCC(=O)NCCN1CCC(NC(=O)C2CC2)C1)NC(CC1C(C)C1)=O C1(NC(c2cc(OCC)n[nH]2)=O)CCC(C)(CNC(c2conc2C)=O)C1 Cc1ccc(C(N2CC(NC(=O)Cc3ccnn3C)C3CC23)=O)cn1 C#Cc1ccc(C(=O)N(CCNC(=O)C(C)(C)C#CC)CCOC)c(C)c1 C(=O)(CC(CC(C)C)NC(C1CCCC(CF)C1)=O)NC(C#C)C c1(C(=O)NC2CN(C(C3C4CC4C4CC34)=O)C2)c[nH]c2cccc(Br)c12 C1(F)(CNC(c2c(C(C)C)n[nH]c2)=O)CCN(C(c2ncoc2C2CCC2)=O)C1 c1(OC)cc(Br)c(C)nc1NC(C1CC1C(=O)NCCn1cc(Br)cn1)=O N1(CC(=O)N(C)C)CC(C(=O)NCCN2CC=CC2)CC1=O C(=O)(C(F)C(C)(C)O)NCC(C)CC(=O)NCCC1OCCC1(C)C c1(C(=O)NC2(CO)CCN(C(=O)CC3(O)CCCC3)CC2)ncc2[nH]ncc2n1 N1(C(C2CCC(CC)CC2)=O)C2CCC(C2)C1CNC(C1CC12CCC2)=O C12(C(=O)NC3CC(OCC)C3)CC1CN(C(=O)CC1CC1C1CC1)C2 Cn1cc(C#CCNC(C2OCCC2NC(C2CCC3(CC3)C2)=O)=O)cn1 N1(C(C(C)=C2CC2)=O)CCCCCCC1C(=O)NC(c1ccns1)C CCC(C)(CO)C(=O)NCC(CNC(c1csc(N2CCCCC2)n1)=O)OC N1(C(C=CC=CC)=O)CCN(C(=O)C(C)Cc2ccc(F)c(F)c2)CC(O)C1 c1(C(=O)NCC2(C)CCC(NC(C=CCC)=O)C2)cn(CC#N)c2ccccc12 Cc1cn2ccnc(C(=O)NCC(C)N(C(=O)CC3CCCO3)C)c2n1 N1(C(CN(C)C(=O)OC(C)(C)C)=O)CCC(C)C1C(=O)N(c1cnncc1Cl)CO Cc1noc(C(C)C)c1C(N1CCC(C)(NC(=O)C(C)c2ccco2)C1)=O C(=O)(C1=NOC(C)(C)C1)NC(C(C)C)C(C)NC(c1cc(Cl)c(F)cc1Cl)=O CCC(CNC(C1CN(C(=O)CC2CCCSC2)CC1C)=O)(CC)OC c1(C(=O)NCCC2CCN(C(C3CC3CN3CCCC3)=O)C2)ccnc(CO)c1 c1(C(=O)NCC2CN(C(c3c(C)csn3)=O)CC(C)C2)cnc2ncccn12 c1(C(N2CCN(C(CC(C)CN(C)C)=O)CC2CF)=O)ccc2c(c1)CCN2C C#CCC(O)C(=O)N(C(CNC(c1cc(C(N)=O)co1)=O)C1CC1)C N1(C(c2c(CC)c[nH]c2)=O)CCC(F)C(NC(=O)C(C)C#N)C1 n1(C2(NC(=O)CC3CC3C(F)(F)F)CC2)nccn1.C1(C)CC(=O)N1CCOC.N CS(=O)(=O)c1cccc(Cl)c1C(=O)NC1CC(O)CN(C(=O)Cc2cnns2)C1 c1(C(=O)NCC2CN(C(=O)C3=CCCC3)CCO2)cc(Br)nc(Br)c1 Cc1cccc(Cl)c1C(=O)NC(C)CC(C)NC(C1(CCN(C)C)CC1)=O Cc1sc2ccc(F)cc2c1C(=O)N(CCCN(C)CC1CCN1C(C)(C)C)C c1(C(=O)NCCC(C)N(C(=O)Cn2cnnn2)C)cnc2n1CCOC2 C(=O)(C(CO)C(F)(F)F)NCC(CC)(C)C(=O)NC1CCCCCC1(C)C c1(C(=O)NCC2COCCN(C(c3cccc(C)n3)=O)C2)cc2c(s1)COCC2 c1(C(=O)NCCCCc2nn[nH]n2)ccc2cnnn2c1 N1(C(c2c(C)ccc(F)c2)=O)CC2(CCN(C(=O)C(F)C(C)C(F)(F)F)CC2)C1 C(CCC(=O)NCC(N1CC=CCC1)=O)NC(COCCC=C)=O Cc1nc(CCNC(=O)CC2CCCC2NC(=O)C(O)CN(C)C)cs1 C1(NC(C2CC3(CSC3)C2)=O)CN(C(C2CCS2(=O)=O)=O)Cc2ccnn2C1 Cc1cc(N2CC=C(CCNC(=O)C(C)Cc3ccco3)CC2)n2ncnc2n1 C1(NC(CCCOC(C)C)=O)C(C)CN(C(c2ccnn2C(C)CC2CC2)=O)CC1C N1(C(=O)CC2CCC(NC(C3C4C5CCC(C5)C34)=O)CC2)Cc2cccnc2C1 C1(NC(C(CC)SC)=O)CCN(C(=O)C(C2CC2)OCC)CC1CO N1(C(c2ccn(C(C)C)n2)=O)CCC(CO)C(NC(C2CC2C#N)=O)C1 c1(OCC)c(F)c(C(N2CCN(C(=O)C(C)C(C)C)CC(O)C2)=O)cc(F)c1F c1(CC(=O)NCC(C)N(C(C2(CC)CC2)=O)C)cc(F)ccc1F c1(C(=O)NCC(CN(C(C(C)OCCCC)=O)C)O)ccc(C(C)C)nc1 C1(NC(CSC(C)C)=O)CCCC1C(N1CCC1C1CCCC1)=O c1(CNC(CN(C)C(C2CCCO2)=O)=O)cccc(COc2ccccc2)c1 C1(CNC(N2CCC(n3cnnn3)C2)=O)CCC(F)(CC2NC(=O)NC2=O)CC1 c1(CC(=O)N(C)CC2CCN(C(CC(C(C)C)O)=O)C2)ccc2nsnc2c1 C1(CC(=O)N(CCCC)CCO)CCCN(C(=O)C2=NOCC2)C1 C(CC(C)C)(C(=O)NS(CC(=C)C)(=O)=O)OC(CNC(=O)NC(C)(C)C)=O N1(C(c2c(C)n(C)cc2)=O)CCCC(C(=O)N(C2CCC2C)C)C1C c1(OC)c(C(N2CCC(C(C)C(=O)N(CCN=[N+]=[N-])C)C2)=O)cnn1C C=CC(C)(C)CC(=O)NC(CNC(=O)C(F)(F)c1cscn1)C(C)(C)C CN1CCCC1C(=O)NCC(CNC(C1CC(F)(F)C1)=O)CO C1(CNC(C2(CC(C)C)CCOCC2)=O)CN(C(=O)CCS(N)(=O)=O)CCC1C C1(NC(C2(C=C)CNC2)=O)CC2OCCCC12 C(=O)(CCCCC(=O)NC1CCN(C(c2cnc(S)nc2)=O)CC1C)NC CCCCCC(O)C(=O)N(CC(=O)Nc1ccc(O)cc1)C Cc1cnc2c(C(=O)NC(C)CCCNC(c3cnc(C#N)s3)=O)cccc2n1 c1(C(=O)NC2CCC(CNC(C(CCOC)(C)C)=O)C2)coc2cc(O)ccc12 N1(C(C(CC#C)C2CC2)=O)CC2CCC2(CNC(=O)COCCC)C1 CP(C)(=O)C1CCC=C1C(=O)NC(c1ccc2c(c1)CCCC2)C(=O)O C=CCC(C)(C)CC(C(=O)NC)N1CCC(C)(C)C(c2ccccc2)C1 C=CCC(CC=C)C(=O)NC1CCCN(C(C2CC(C)(C)CN2C)=O)C1 Cc1ccc(N(C(C2CCOC(C)C2)C(=O)NCCOC(C)(C)C)C)nc1 C1(CC)CN(C(=O)Cn2cnc(C(N)=O)n2)CCN1C(C1CCC(C)(C)CO1)=O C1(C)(N(C)C)CCN(C(=O)C(C)(C2CCC2)NC(=O)CCc2cccn2C)CC1 C(=O)(C(C)C(F)(F)F)NCC1CN(C(CCCN(CCC)CCC)=O)CC1C C1(NC(c2ccc(CN(C)C)[nH]2)=O)CC2(C1)CN(C(c1cnn(C)c1Br)=O)C2 C(N=C(NCCOC)N1CCN(CC)C(C)C1)c1ccc(C(=O)OC)cc1.C(COC)OC C1(CCCC)CCCN(C(=O)C=CC(C)NC(=O)CC2CCCC2OC)C1 N#Cc1cccnc1NC(c1cc(C(F)(F)F)ccc1Cl)=O C(C(C(=O)NC1CCCOC1)C(C)(C)C)NC(C(C)CC1CC1)=O C1(C)(C(N(CC(C)NC(C2(C)N(C(CCC)=O)CCC2)=O)C)=O)CCCCCC1 c1(NCC2CCN(C(C(CCC)NC(N)=O)=O)C2)cc2nc(CCC)nn2cn1 c1(C(N2CCC(NC(c3cnc(OC)nc3C)=O)C2C)=O)cccc2c1NCC2 CC1(CNC(C2CNC(=O)C2)=O)CCN(C(=O)CCSCc2ccccn2)C1 C1(CNC(c2c(C(C)C)ccs2)=O)CCN(c2nccc(CC#N)n2)C(C)C1 C1(NC(CC(CC)C2CCC2)=O)CC(C(=O)N2CCCC2(C)C(C)(C)C)=CC1O CN1CC(NC(=O)C=CCNC(C2CC2(Cl)Cl)=O)C2(CC2)C1 c1(CNC(N2CCC(c3nnc(SC)s3)C2)=O)ccc(Br)cc1F C1(C(=O)NC2CC(F)(CNC(c3c(CC)n(C)nc3)=O)C2)CC12CCCCC2 CCCCC(CNC(c1cnn(C)c1)=O)NC(c1cccc(CC(F)(F)F)c1)=O C1(C(N(C(COC)C)C)=O)CCCC1CNC(C12COCC1C2)=O c1(C(=O)NCC2(F)CN(C(=O)C=CC3CCOC3)C2)c(Cl)csc1Cl c1(C(=O)NC2(CNC(C3C(C=C)C3)=O)CCOC2)ccc(C2CC2)nc1O C1(C(=O)NCC2CC(O)CN2C(=O)CN2C(=O)CNC2=O)CC12CCCCC2 Cc1ccc(F)cc1-n1cc(CC2CN(C(c3cc(Br)n[nH]3)=O)C2)nn1 N1(C(CC(=O)OC)=O)CC(C)OC2(CCN(c3ccc([N+](=O)[O-])cc3Cl)CC2)C1 C(c1cnc(O)nc1O)=CC(=O)NC(CNC(CCC=C(C)C)=O)CC(C)C C1(C(=O)NCC2C=CC(NC(CCc3c(C)ncs3)=O)C2)CCCNS1(=O)=O c1(NCC2(CSC)CC2)ncc(C)cc1S(=O)(=O)N1CCC(C)CC(C)C1 Cn1nc(O)cc1C(N1CC(F)CC1CNC(c1cnnc(Cl)c1)=O)=O c12cc(ccn1)C(=O)N2.C1(C(=O)NC(CN(C)C2CC2)C2CCC2)CCS1(=O)=O CC1OC(C)C(C(=O)NCC2CN(C(=O)CCn3cncn3)CCO2)C1C C1(N(C(C(c2ccccc2)NC(c2nc(C)oc2)=O)=O)C)CCN(C)C1=O C1(NC(COC2CCCC(C)C2)=O)CN(C(=O)CCC(F)(F)F)C2(CCC2)C1 CC1CCCC1(NC(=O)NC(C)(C)C)CN(C)S(N)(=O)=O CC(C)(C(c1nnnn1C1COC1)NCC1(SC)CC1)C(N)=O N1(S(CC)(=O)=O)CCCC1C(=O)NCCCCNC(C1CC1(C)Br)=O c1(-c2nc(C)sc2)ccc(CCNC(=O)NCCC2CCC(=O)N2)cc1 C1(C(N(CCO)CC)=O)CCCCC1n1cc(C2CC3CCC2C3)nn1 C1N=C2C=CC(=CN2)S(=O)(=O)C(C)N2CC1C2.c1(C2(NCC(C)C)CC2)cccs1 n1(CC)cc(C(=O)NCC2CC2NC(=O)CN2CCC2C)c(C2CCOCC2)n1 c1(C(c2nnnn2C(C)(C)C)CCCN)cccc(N(C)C)n1.CNC N1(C(c2ccc(CC)nc2)=O)CC2CCC(C1)N(C(=O)C(Cl)CCC)C2 C12(NC(c3ccncn3)=O)CCCC1N(C(c1cc(=O)cc(Cl)[nH]1)=O)CCC2 C1(NC(C(C=CC)O)=O)CCC(O)CN(C(=O)CCOc2cc(F)ccc2F)C1 C=CC(C)(C)CCCNC(c1[nH]ccc1CNC(C1CC(Cl)(Cl)C1)=O)=O c1(-c2n(C(COC)C)nc(-c3ccccc3C)n2)cnc2c(c1)nc(O)n2C c1(CC)scnc1C(=O)NC1CC(C)(NC(=O)CCc2csc(C)n2)C1 C(=O)(C#CC1CCOCC1)NCC(C)C(F)C(=O)NCC1=NOC2CCCC12 Cc1c(Cl)ccnc1C(=O)N(CCNC(c1ccc(C#N)cc1)=O)C(C)C C1(C(=O)NCC(CNC(=O)Cc2nncn2C)OC)C(F)(F)C12CCC2 C1(CNC(c2c(CC)c[nH]n2)=O)CC(C(=O)Nc2cnc(OC)nc2)=NO1 CCC(CC(F)(F)F)C(=O)N(C1CCCN(C(=O)C2=C(Cl)CCC(C)C2)CC1)C c1(NC(C2(CCCC)CCCC2)=O)cccc(NC(C2COCCO2)=O)c1 c1(NC(c2nc(C)c(Br)s2)=O)ncc(F)cc1Cl N1(C(c2cccc(C)c2F)=O)CCN(C(C2CC2F)=O)C(C#N)C1 c1(CN2CCCC(CNC(c3cc(C)n(C)n3)=O)C2)ccc(Cl)c(I)c1 CCC(C)(C)CC(=O)N1CCC(c2ccccc2)(CNC(=O)C(F)OC)CC1 Cc1cccc(-n2nnnc2C2(NC(C)COC(C)(C)C)CCCC2)c1 c1(NC(C2C(C#N)C2)=O)nc2c(s1)CC(NC(=O)CC1CC1)CC2 c1(OC)cnc(C(=O)NCC2C3CC2N(C(=O)C(C(C)C)SC)C3)nc1 c1(NC(=O)NC2(C(F)(F)F)CC2)ccc(CN2CCCCC2C2CCCC2O)cc1Br N1(C(=O)NC2CCN(C(C)C)C2)CCCCC1(C)CO Cc1cc(-c2cccc(C(C)NC(C(c3ccccc3)C(N)=O)=O)c2)cnn1 C1(CC)CN(C(c2ccc(OC)c(F)c2)=O)CCN1C(=O)Oc1onc(C)c1C C(=O)(C1=CC2CCC(C1)C2)N(C1(C(N(C2C(C)COCC2)C)=O)CC1)C c1(CC)cc(C(N2CC=CC(NC(=O)C(c3ccccc3Cl)C)C2)=O)cc(O)n1 c1(-n2c(CC(CC)C)nc(CCC(C)C)n2)ccc(F)cc1F N1(C(C2CCN(CC)C2)=O)CC2CC(C(=O)NC(CC)CO)(C2)C1 N1(C(C(C)=CC)=O)CC2CCC1C(NC(=O)C=CC1CCCC1)C2 C=C(Br)CN=c1nc2c(cnn2C)c(NCC2CC(C#N)C2)[nH]1 c1(C(=O)NCC(C)N(C(c2c(CC)nco2)=O)C)cc2cc(F)ccc2s1 C12(CNC(C3N(CC(C)C)CCC3)=O)CC(CCO1)N(C(=O)CC1C=CCC1)C2 c1(C(=O)NCCC(C)NC(=O)CCCCc2ccc(F)cc2)ccc(N)c(F)c1 c1(C(=O)NC(CCNC(c2nn(CC)c(C)c2)=O)C)cn2cc(Cl)cc(Cl)c2n1 c1(C(=O)NCCC(C)NC(c2ncccc2O)=O)ccc(S(N)(=O)=O)o1 N1(C(C)C)CCC(C(=O)NCCCCNC(c2cscn2)=O)CC1 N1(C(CC(C=C)CC)=O)CCC(NC(=O)C2=CCCC2)C2(CCC2)C1 c1(CCNC(C2(C)CCCO2)(C2CCCO2)C)nnnn1CCC1CC1 C1(NC(COC(C)C)=O)C2CC3CC(C2)CC1(CO)C3.c1(C(=O)N)cnn(C2CC2)c1 C12(C(=O)NC3CCN(C(=O)C(c4ccc(F)cc4)O)C3)CCN(C1)S(=O)(=O)C2 C1(NC(=O)CCc2cncnc2)CCN(C(=O)Cc2ccccc2)C12CCC2 C=CCC(CC)C(=O)NCC(CC(F)(F)F)NC(c1cnc(S)nc1)=O C=C(Cl)C(C)(C)C(=O)N(CC(C)(C)NC(=O)CC1CCC1C)C C(CC(=O)NCCc1cccc(O)c1)(C(F)(F)F)NC(C1(C#N)CC(C)C1)=O c1(C(N2CC(CC(N3CCC(O)(CC)C3)=O)C2)=O)cc2ncccc2[nH]1 c1(C(=O)NCCN(CCOC)C(C2CC23CCCC3)=O)ccc(C)c(Cl)c1F C(C(=O)NC1CC(C#N)C1)(C(C)(C)C)NC(c1ccc(C)nn1)=O Cc1cc(C(N2CCN(Cc3ccc(Cl)s3)CC2)C)cc(Br)c1 C1(NC(c2ccc(Br)cc2Cl)(c2n(C)nnn2)CCC2CC2)C(=O)NCC1(C)C C=CC1(NC(c2csc(Cl)c2)c2nnnn2CCCC2CC2)CCOCC1 N1(c2c(OCC)cccc2)CC2CC1CN2C(=O)Cc1cc[nH]n1 c1(C(N2CC(NC(c3cn(C4CC4)nn3)=O)C2)=O)ccc(C(F)F)nc1 CC(=O)CCCCC(=O)NC1(CNC(=O)CC(C)C(F)F)CCOC1 C1(NC(C=CC(C)C)=O)CC2CC(NC(=O)CCCC(=O)NC(C)C)C1C2 N1(CC(=O)NC(CC=C)CNC(c2ccc(C#N)cc2)=O)C(=O)C(C)C(C)C1=O C12(C(=O)NC3CCC(O)C3)CCC(n3cc(CN4CCCC4=O)nn3)(CC1)C2 C1(C(=O)NC2(C#C)CC(F)(F)C2)CCN(C(=O)C(C(C)C)NC=O)CC1(C)C c1(C(=O)NCC(C)CNC(=O)C(=O)N(C)Cc2ccc(F)cc2)ccnc(Cl)c1 C(=O)(C(F)C(C)C(F)(F)F)NC(CC(C)NC(C(C(C)C)F)=O)C c1(C(N2CCC(N3CCCC3)C2)=O)ncc(C(F)F)cn1 CCC(CC(=O)N(CC(=O)NC(CC1CCCC1)CO)C)C(C)(C)C C(CCN1CCCC1(C)C)(C(C)C)OC.C1(C)CCC(=O)N1 C(c1c(F)cccc1F)=CC(N1CCC(C)C1CNC(=O)COCCF)=O c1(C(=O)NCCN(C(=O)C(C)CN(C)C)CC)cccnc1OC CCC(C)(O)C(=O)N1CCC1CNC(=O)C(C)(C)C1CCCC1 c1(C(=O)NCC2(O)CN(C(C(CO)N(C)C)=O)C2)cc(F)ccc1C(F)F Cc1ccc2[nH]cc(CCC(N3CCN(C(c4cc(Cl)c[nH]4)=O)C(C)C3)=O)c2c1 C(C(=O)NC(C(=O)N(C)CC1(CO)CCC1)c1ccco1)(C(C)C)OCC C(=O)(C1=C(C)OCCS1(=O)=O)NC(C(C)(C)NC(CC=C)=O)C Cc1ncnc(O)c1C(N1CCN(C(C2(F)CC=CCC2)=O)CC1)=O c1(OC)ccc(C(C)C)c(C(=O)NCCN(C(=O)CCN2C(=O)CCC2=O)C)c1 c1(C(=O)NCCCC(C)NC(=O)C=C2CCSCC2)c(Cl)ccnc1F C(CC(O)CNC(c1ccc(-c2ccncc2)o1)=O)NC(C1(F)C(C)C1)=O C1(NC(c2n(CCC)ncc2)=O)CCCCC1CNC(=O)CC1CSC1 n1(CC)nc(C(=O)NCc2csc(C(=O)NCC(c3ccsc3)C)c2)c(C)n1 Cc1ccc(C(=O)NCCC2CN(C(=O)CC3CCC(=O)O3)CCO2)cc1C N1(CCN(C=O)CC2CC2)CCCOCC1 C=CC(C)C(C)C(=O)NCCNC(c1cnc(C(=O)N(C2CCC2)CCO)s1)=O CC1(C(N2CCOC(C(N3CC4CC3C4)=O)C2)=O)CC(C#N)C1 C(=O)(C1=CCCOCC1)NC1C(CC(C)(C)C)CN(C(C2CC(O)C2)=O)C1 c1(C(=O)NC2CC(N(C(Cn3c(C)nnn3)=O)C)C2)cncnc1C1CC1 C(=O)(CCCCCNC(=O)C(CC)CCC)NC(CCCC)COC C1(CC(=O)NC2CCC(NC(c3c(C)c[nH]c3)=O)C2)CCOCC1(C)C c1(C(=O)NC2CCN(CC(C)(C)O)C2)cccc2cnccc12 C12(C(N3CCCCC(C(=O)Nc4ncc(C#C)s4)C3)=O)CCC(CO)(CC1)CC2 c1(C(=O)NC2CCN(C(C3(C(=O)OC)C=CCC3)=O)C2)ccnc(O)c1Br C12(NC(CCC(C)OC)=O)CCOC(CNC(C3CCC(C)(O)CC3)=O)(C1)C2 c1(C(N(C2CN(C(=O)Cc3cc[nH]c3)C2)C)=O)nc(C2CCCCC2)sc1C Cc1ccc(CCC(=O)NCC2CCCN(Cc3ncc(Br)s3)C2)cc1 CCC(C(=O)NCC(O)C(=O)NCCc1csnn1)n1ccnc1 CC1CC(C(=O)NC2CCCC(NC(C3CN(C)C3)=O)C2)CC(C)(C)C1 C(C)(C)(CC(=O)N1CCC(C(C)(C)NC(c2cc(N(C)C)ccn2)=O)C1)SC C12N(CCC1(C)C)C(=O)C2.c1(NC(=O)NC2C(C(=O)OC)CC2)cccnc1 C(=O)(C(C)(C)Cc1ccc(Cl)cc1)NC(CNC(C1(C)C=CCC1)=O)C1CCC1 n1(CC)c(=O)n(CC(=O)NNC(=O)c2ccncn2)c2ccccc12 Cc1nn(C)c(C(F)(F)F)c1C(=O)NCC1CCCN(C(c2cn[nH]c2)=O)CC1 N1(C(CC2C(NC(C(=CC3CCCC3)C)=O)CCC2)=O)CCCC2(CCOC2)C1 c1(OC(C)C)cccc(C(=O)N(C2CCCNC2=O)C)n1 C1(N(C)C(C2CC3(CCC3)C2)=O)CC2CC1N(C(C1C=CCCC1)=O)C2 c1(C(N(C(CN(C(CCc2cncc(C)c2)=O)C)C)C)=O)cccc2ccsc12 Cc1ccc(C(=O)N(CCC(=O)NCC2CCCC(=O)N2)C(C)C)nn1 C1(CNC(C2(OCC)CCOC2)=O)CCN(C(=O)C2=COCCO2)C12CC2 N1(C(c2ncc(OC)nc2)=O)CC(C)CN(C(=O)C2Cc3ccccc32)CC1C C(=O)(C(F)(F)C(F)(F)OC(F)(F)F)N1CC(C)C(C)(N(C)CCOC(F)F)C1 C(=O)(C(CCC(C)C)NC(c1ccnc(O)c1)=O)N(CC(CCC)O)C N1(C(C)=O)CCC(CNC(=O)NC(c2cn(C)nc2CSc2ncc[nH]2)=O)C(C)C1 C(=O)(C(F)C(C)CNC(=O)CN1CCOCC1=O)N(CC(C)C)CCO C(=O)(CC(O)CC(C)(C)C)N1CCC(C(=O)NCC2CC(OCC)C2)C1(C)C C1(NC(C2(CC)CN(C(C3CCCC(C)(C)C3)=O)C2)=O)C=CC(C)(C)CC1 N1(C(c2cn(C(C)C)nn2)=O)CC=C(CC(=O)NCC2CCOC2=O)CC1 c1(OC)cncc(CCC(=O)NC2CCC(NC(C3CCOC(=O)N3)=O)C2)c1 C1(CNC(C2(C)C(C)(C)C2(C)C)=O)CN(C(=O)Cn2cccc2)C2(CCC2)C1 C1(C(=O)NCC2C(C)C2C)CC2CN(C(c3cc(Cl)n(C)n3)=O)CC2C1 C1(N(C(N2CCCC2)=O)C2CC2)CCCN(C(C2CCC3(CC3)C2)=O)C1.O=C1CN1 c1(-c2n(C(CC)CC)ncc2)nc(C2COc3ccccc32)nn1CCC(C)C C1(NC(=O)C#CC2CCCCC2)CCCCC12CCN(C(c1ccsc1Cl)=O)C2 C(C(C(=O)N1CC(c2ccco2)C1)C(C)C)NC(C(OC)OC)=O N1(C(C(C)=C2CCC2)=O)CCCC1C(C)(C)NC(=O)CCNS(C)(=O)=O C#CC1C(C(=O)NCC2CCCN2C(=O)CN(C)C(C)=O)C1(C)C c1(C(C(=O)NCc2cn(-c3cccc(Br)c3)nn2)O)cccc(Cl)c1Cl c12[nH]nc(c1Cl)C(=O)N1CC(C1)N(C)C2=O.c1(CC)nc(-c2ccco2)sc1C c1(C(=O)NC2C(CNC(COCCOCC)=O)CCC2)cccc(N(C)C)c1 C(=O)(C(C(C)C)c1ccccc1)NCCN(C(COC(CC)C)=O)CCOC C1(NC(C(C)SC(C)C)=O)CCN(C(C2(c3ccccc3)CCCC2)=O)CC1 c1(NC)cncc(C(N2CCOC(CCCNC(=O)CC3(OC)CC3)C2)=O)c1 N1(C(CC2(C#N)CCC2)=O)CCC2(CCCN(C(C34CCCC(CO3)C4)=O)C2)C1 C(=O)(CCC(C)=O)NC(C(=O)NCCSCC(C)C)CC1CCOCC1 CCC(CC)CC(F)C(=O)NC1CC(OCC)C1.N12CC3(CC3)CC1OCC2=O c1(C(=O)NCC(CC)NC(c2c(C)ccn2C)=O)cc(N2CCCC2)nc(Cl)c1 C1(C(N2CCC(CCNC(c3c(C)ocn3)=O)C2)=O)CN(C)CCN(C)C1 C1(CS(=O)(=O)NCC(c2ccccc2)C)CCC2(CCOCC2)CO1 n1(C(C)(C)C)ccc(=NC(=O)C(=O)NCC2CSC2)[nH]1 Cc1nnsc1C(=O)NCC(C)NC(c1cn(CCO)nn1)=O C(=O)(C(C)(C)CF)N(C)CCNC(c1ncoc1C(C)(C)C)=O N1(C(CC23C(CN(C(c4ccc(CO)[nH]4)=O)C2)CC3)=O)CCCC2(CCCO2)C1 N1(C(CC2ON=C(C)C2)=O)CC=CC(C(=O)N(C)CC2COCCO2)C1 CS(=O)(=O)C1CCCC1C(=O)NCC1CN(C(=O)Cn2ncnn2)CCO1 c1(CCCC)ccc(CC(=O)O)cc1.c12cn(nn1)C(C)C(=O)N(CC)CC2 CN=c1cc(C(=O)NC2CCOC2C(=O)NCC(C)(C)C(F)F)cc[nH]1 c1(C(C2CC3CCC2C3)NC(=O)NCCN2CC=CC2)cccc(F)c1 N1(C(C2CC(C)C2)=O)CC2CCC(NC(c3ncc[nH]3)=O)CC2C1 C1(COC)CCC2CN(C(=O)C(F)(F)CC3CC3)CCC2C1.C1(=O)CCCC1=O c1(C(=O)NCC2N(C(CCN(C)CC)=O)CCCC2C)sc2cccnc2c1Cl Cc1ccc(C(F)(F)C(=O)NCc2nccn2C(c2ccccc2)C)c(Br)c1 C1(C)(CC)CCCN(C(c2ccnc(C(=O)NC)n2)C(=O)NC2CC2)CC1 c1(CC(N2CCC(N(C)C(C3CCCS3)=O)C2)=O)cc2ccccc2c(=O)o1 c1(C(=O)NC(C)CNC(c2ccc(C(C)(C)C)cn2)=O)cc2cc(Cl)cnc2o1 C1(CC(N2CC(O)(C(C)NC(c3nc(C)c(C)s3)=O)C2)=O)CN2CCC1CC2 C(=O)(CC(C=C)CC)N(CC(=O)NCCCCCC#C)C1CC1 CC(C)CC(C(=O)N(CCCOCCN(C)C(c1n[nH]cc1Cl)=O)C)C(N)=O N1(C(CC2N(C)CCOC2)=O)CC2CCCC2(NC(=O)CCCCC2CC2)C1 C1(NC(CC(C(C)C)O)=O)CC2(CCN(C(C34CCOC3CCOC4)=O)CC2)C1 C(CCCCCCCO)NC(C1N(c2nc(C)c(Br)cn2)CCC1)=O C1(N(C)C(c2cc(C3CC3)no2)=O)CCC(NC(C2CCCCC2F)=O)CC1 C1(C(C)C)CN(C(=O)CC(F)(F)F)CCN1C(CC(C)(C)C)=O.C1(NC)CCC1 Cc1ncc(CCN(C(c2snnc2C)C(=O)NCC2CCCO2)C)[nH]1 c1(C(=O)NCC2CCN(C(C3CC(=C)C3)=O)C2(C)C)oc2c(Cl)cccc2c1C CNS(=O)(=O)N1CCN(C(=O)NC(c2cnccn2)C)CC1 c1(C(=O)NCC(=O)N(C2CC(C)OC(C)C2)C)ccc(Cl)c([N+](=O)[O-])c1 c1(C(=O)NC(CC)CNC(=O)CN(C)Cc2cncn2C)ccc2nncn2c1 C(C(C)(CC(C)C)NC(C1CC=CC1)=O)NC(C(CC)(C)OC)=O C1(CC(=O)NC(C)CO)CCCCC1NC(=O)CC=Cc1ccccc1 c1(SCC)cccnc1C(=O)NC1(CCNC(c2ccncc2CC)=O)CCC1 C12(C(=O)NCC(C3CC=CC3)O)CCC(CC1NC(c1ccncc1F)=O)C2 O=C(C#CC1CCCCO1)NCC(CNC(c1cccn2cncc12)=O)CO c1(CSC)ccc(NC(C)C=CCc2ccccc2)cc1 C1(C(=O)NC(C2CCCN2C(c2sccc2C(F)F)=O)(C)C)CN2CCN1CC2 c1(C(=O)NCC(C)(C2CC2)NC(C2CCCC(O)C2)=O)cncc(C(F)F)c1 C(=O)(C(Cc1cnc[nH]1)NC(C1CCN(C)C1)=O)NCCN(CCC)CC C=CCCC(C(=O)NCCc1ncccc1F)NC(=O)CCC1OCCO1 c1(NC(N2CCC=C(C)C2)=O)ccn2nccc2n1 C1(NC(CCCC)=O)CC2CCC(C1)N2C(c1c(C2CCC2)cnn1C)=O Cc1cncn1C.c12cc(on1)CN(C)C2C(=O)NCC(F)F N12C3CCCC1CN(C3)CC2=O.c1(N)ccccc1F.C1(CSC)(C)CC1 Cc1nnc(NCC(C)NC(=O)C2=CCSC2)c(C#N)c1C N1(C(CSCC(C)=O)=O)CC2COCCC2(NC(c2cnc3ncccn23)=O)C1 C(=O)(CCCCC1CC1)NC1C=CC(C(=O)NC)C1.C12COCC1NC2=O N1(C(C2CC(C)(NC(CC3(OCC)CCC3)=O)C2)=O)CC2CC2(C(=O)NC)C1 C1(C(=O)NCCCCNC(C(C2CCCCCC2)(C)C)=O)OCC2CCCCC12 C1(C(C)NC(C2(F)CCC2)=O)CCCN1C(C1CCC(=O)N1)=O c1(C(=O)NC2CCC(CNC(C(CCN(C)C)O)=O)CC2)cccc2cncn12 N1(C(CCCC#C)=O)CC2CCC2(C(=O)NCC(c2ccc(C)cn2)O)C1 N1(C(c2ccc(C)cn2)=O)CCCC2(NC(=O)CCc3ccncn3)CC2C1 Cc1nc(C(=O)NC(C)(Cn2cc(Br)cn2)c2nn[nH]n2)oc1C c1(-c2cncc(NC(c3nc(CC)sc3)=O)c2)cc(F)c(OC)c(F)c1 N1(c2cc(NC(C)CC(N)=O)nc(COC)n2)CCN2C(=O)C(=O)NCC2C1 c1(C(=O)OC)csc(CNC(=O)Cn2cc(C(C)N(C)C)nn2)n1 c1(C(N2C(CNC(C=Cc3c(C)ccnc3)=O)C=CC2)=O)cncc2c1CCC2 C(=O)(C(F)(F)CO)NCCC1(C(N2CC(C(=O)OC)(CC)C2)=O)CC1 N1(C(CN2CC(=O)NCC2)=O)CCCCCC1C(N1CCC2(CCC2)C1)=O Cc1cccc(Cl)c1C(=O)Nc1cnc(F)c(-c2cscc2C(=O)OC(C)C)c1 CC1C(NC(c2nccc(N)c2Cl)=O)CCCN1C(C1C2CCCOC12)=O C1(CNC(C2(C(=O)OC)CC2)=O)CCN(Cc2cc(Cl)ccc2Cl)CC1(F)F c1(C(=O)NCC2N(C(C3C(C4C(C)C4)C3)=O)CCCC2)cccc([N+](=O)[O-])c1 C1(=CC(=O)NC2CC(C(=O)OC)CC2O)CCCCC1(C)C c1(C(=O)NCCN(C)C(c2cc3sccc3[nH]2)=O)cc(Cl)ccc1C(F)F CCCC(C(=O)NCC=C(C)C)NC(C)=O.C1(O)CC(NC(=O)COc2ccsn2)C1 c1(C(=O)NCCCN(C(=O)Cc2ccc(C(N)=O)cc2)C)cnc([N+](=O)[O-])n1C c1(C(N2CCC(CN(C(c3c(C)nns3)=O)C)C2)=O)ccc(F)c(C)c1N c1(C(=O)OC(C#C)CC2CCOCC2)nn(C)c2c(Br)cncc12 c1(C(=O)NCCN(C(C(C)C2CCOC2)=O)C2CC2)cnc2c(c1)CCCO2 c1(CC)onc(C(=O)NC2(C)CC(C(N3CCOC(CC(C)C)C3)=O)C2)c1C c1(COC(c2c(OC)nc(C(=O)OC(C)C)cc2)=O)cc(C#N)cc(C#N)c1 C1(COC)CN(C(=O)CC2SC(=N)NC2=O)CCN1C(=O)COCCC(C)C c1(NC(C2(C)CCN(C(C(=C)F)=O)C2)=O)ccc(C)cc1C O=C(CC(C(F)(F)F)n1ccnc1)NCC1CCC1NC(c1cnn[nH]1)=O c1(COOCC(N2CC(CC(C)NC(C(C)SC)=O)C2)=O)nc(C)no1.C C(c1cccc(F)c1)=CCC(=O)NC1C2CCN(C(C3COC(=O)N3)=O)C12 c1(C(=O)NC2(C)CN(C(C(CCSC)NC=O)=O)C2)ncc(F)cc1C C(C(CC1CCCC1)C(=O)Nc1c(C)nsc1C)NC(CC=C=C)=O N1(C(C(c2ccccc2)C)=O)CCCC(C(C)(C)C(=O)NCCS(C)(=O)=O)C1 c1(NCC(=O)NC2C=CC(CNC(C(=Cc3cnc[nH]3)C)=O)C2)ccc(F)cc1 C12(C(=O)NCCN(C(C3(CC(F)F)CC3)=O)C3CC3)CC(C(N3CCCC3)=O)(C1)C2 C1(CNC(C(C)(F)c2ccccc2)=O)(CNC(=O)C(O)c2ccsc2)CC12CCC2 C1(CNC(CC(C)F)=O)(CO)CCCN(C(c2cn(C)[nH]c2=N)=O)C1 C1(CNC(c2nnc(C)s2)=O)CN(C(c2cc([N+](=O)[O-])c[nH]2)=O)CCC12CCC2 N1(C(c2c(C)ncs2)=O)CCCC2C(CCCN2C(=O)Cc2ccon2)C1 C1(C(N(C2(C#C)CC2)C)=O)C(CNC(c2cncn2C(C)C)=O)C1(C)C n1(C2C(C(=O)NC3(CC)CC3)C2)cc(C(N2CCC(c3nn[nH]n3)C2)=O)c(C)n1 C1(CC(=O)NC(c2ncn(C)n2)C)(OC)CN(C(=O)CC2CCCCO2)C1 N1(C(C(=O)NC(=O)NC)C)CC2CCC(NC(c3cscn3)=O)C2C1 Cc1cc(C(C2CC2)NC2COCC2C)nc(Cl)c1 c1(OC)ccc2sc(C(c3nnnn3C(C)C)Nc3ccccc3)c(C)c2c1 C=CC(C)(CC)C(=O)N1CCCC(CN2CCN(C(c3csc(C)n3)=O)CC2)C1 C1(NC(c2cc(C)sn2)=O)CC2CCC(C1C)N2C(c1ccc(O)nc1C)=O c1(CC)cnc(CC(=O)NCCC2(NC(c3cccnc3)=O)CCC2)[nH]1 N1(C(C(CC)(C)COC)=O)CC2CC(C)N(C(c3cccc4ccoc34)=O)C2C1 Cc1cnc(NC(C)CC(C)(C)C)c(S(=O)(=O)N2CCN(C(C)CO)CC2)c1 Cc1csc(CCC(=O)NC(C)CC2CN(C(c3cncn3C3CC3)=O)C2)n1 C1(C(=O)NCC(CNC(=O)C=CC2CCC2)F)C2CC3C(C2=O)C13 c1(CCOC)ccc(NC(=O)C(COC)OC)cc1.N12CCC(C1)OC(C)C2=O N1(C(C=CCOC)=O)CCCCC2(CCN(C(C34COC(COC)(C3)C4)=O)C2)C1 C1(CN(C(=O)C(c2ccccc2)F)C)CCCN(C(=O)CC2CCNC2=O)C1 N1(C(c2nc(C(C)C)oc2)=O)CC(NC(=O)CSc2ccccn2)CCC1C N1(C(CC2CC(C)(C)C2)=O)CC2CN(C(c3cc(O)cc(F)c3F)=O)CCC12 Cn1cc2ncc(C(=O)NCC3(CNC(c4cnc(=N)[nH]c4)=O)CCC3)cc2n1 C(=O)(C1=CCC(NC(=O)CC2CCSCC2)C1)NCc1ccc(C)s1 c1(CCC(=O)NCCOCCNC(CSCC=C)=O)ccc(F)c(F)c1F c1(OC)ccc(C(N2CCCCC2CN(C(=O)C2=NOCC2)C)=O)c(F)n1 C1(CC(=O)NC2CN(C(c3cc(Br)nc(Br)c3)=O)CC2F)CCCCC1(F)F N1(C(CS(N)(=O)=O)=O)CCC2(CCCN(C(C3Cc4ccncc4C3)=O)C2)C1 N(C1CCNc2ccc(Cl)cc21)C(c1ccn(C2CCOCC2)n1)=O C#Cc1ccnc(C(=O)N(C2CN(C(c3cnccc3Cl)=O)CCC2C)C)c1 C(C(C(C)(C)C)NC(c1cc(C(C)(C)C)n[nH]1)=O)NC(C1CCC(C)O1)=O N1(C(CC(C)(C)NC(COCC(C)(C)C)=O)=O)CC(O)(C2CC2)C1 N1(C(C2COC(=O)O2)=O)CCC2(CCCC2NC(c2csnn2)=O)CC1 C1(C(=O)NCCC(=C)CNC(C2(CCF)CCC2)=O)CCCC1C1CC1 c1(OC)ccc(C=CC(=O)NC2CC(NC(C3(c4ccnn4C)CC3)=O)C2)cc1F C1(C#CC(=O)N2CCCC(NC(c3sccc3OC)=O)C2)(CC)COC1 O=S1(=O)NC(=NCCOC2CCC2)c2ccccc21 C=C(Cl)CC(C(=O)N1CCC1(C)C(=O)OC)NC(c1ncon1)=O c1(OC)ccc(C)cc1C(=O)NC(C1(O)CN(C(c2cc(C)nc(O)c2)=O)C1)C c1(C(=O)NC(CC=C)CNC(C2CC(C(F)F)C2)=O)ccc(-c2csnn2)cc1 Cc1cccc(NC(=O)C(C)SCCNC(=O)Cc2ccnn2C)c1 N#Cc1ccnc(CNCC(N)Oc2ccccc2)c1 C1(NC(C=CCOC)=O)CN(C(C2CCCCC(=O)N2)=O)Cc2nccn2C1 c1(NC(=O)NC2CCN(CCC(C)F)C2)ccc(Br)c(F)c1F c1(C(N2CC(C(F)Cn3cc(C4CC4)nn3)C2)=O)occ2c1CCC2 C(=O)(CCS(C)=O)NC(CCCNC(C(C)NC(C)=O)=O)C C(C(C)(C)CNC(=O)C(F)C1CCOC1)N(C(C1C(C)C1)=O)C C(=O)(CCCC(F)(F)CO)NC1CC(C)(NC(c2cc(C)c(OC)c(C)c2)=O)C1 O=C1CCSc2ccc(C(=O)OCC3CC(=O)N(Cc4ccccc4)C3)cc21 N1(C(c2cc(CC)ncc2)=O)CCCCCC1C(=O)NCc1ncoc1C1CC1 C(=O)(C1=NOC(C(C)(C)C)C1)N1CC(SC)C(NC(=O)C(C)(C)CC2CC2)C1 C#CCC(C(=O)Nc1cccc(C(N)=O)c1)NC(=O)Cn1cnc(C#N)n1 N1(C(C(C)(C)CF)=O)CC2CCC1C(CNC(c1snc(O)c1Cl)=O)C2 c1(SC)sccc1C(=O)NCC1CC1NC(c1ccc(C2CC2)s1)=O C1(NC(C(C(C)O)(F)F)=O)CC2CC(NC(=O)Cc3cnc[nH]3)CC2C1 C1(NC(CC2(OC)CCC2)=O)COC2(C1)CN(C(=O)C=C(C)c1cccs1)C2 N1(C(c2c(C)n(C)nc2)=O)CCn2nc(CNC(=O)C=CCO)cc2C1 N1(C(C(C)NC(=O)C(c2ccc(Br)cc2)O)=O)CC2CCC1C2 N1(C(CCC)=O)CCC(NC(c2ccnc(F)c2)=O)C1C N1(C(c2c(CC)nn[nH]2)=O)CCOCC(CNC(C2(C)CCCCCC2)=O)C1 c1(N(CCOCCOCCOC)C)cc(N2CCC(c3ccnn3C)C2)ncn1 c1(OCC)ccc2c(c1)nc(CS(=O)(=O)C1CCC(C)C1)n2CC CCCCCCN1CCC(C(=O)NCC2CC(OC(F)F)C2)C1 c1(C(=O)NCC(C)(CC)NC(c2cn(CC=C)nn2)=O)cc(F)c(C)cc1Cl C(=O)(CCC(F)(F)C(F)(F)F)N(CC(CO)(CO)NC(=O)CCOC(=O)CO)C c1(C(N2CCCCC(CNC(C(CC)O)=O)CC2)=O)cc(Cl)c2c(c1)OCCO2 C1(CNC(C(C)(C)OCC)=O)CN(C(C2CC2c2ccccn2)=O)CCCO1 c1(C(N2CC(N(C(C3C(=C)CC3)=O)C)C3(C2)CC3)=O)ccc(Cl)c(F)c1N C1(COC)(CNC(=O)Cn2nnnc2C)CCN(C(=O)CC(C)(C)C2CC2)C1 CCS(=O)(=O)c1ccccc1C(=O)NCC1(NC(=O)CNC(c2ccoc2)=O)CC1 C1(NC(CCCN(Cc2ccccc2)C)=O)C(C)CCN1C(=O)OC(C)(C)C.CC CC(C)(CN=c1nc(N2CCC(F)C2)c2c([nH]1)CSC2)N1CCCC1 C(=O)(CCCC(C)(C)C#N)NC(C(=O)N(C)CC1CCCC1)(C)C1CCC1 Cc1nc(CC(=O)NC2CCCC2CC(N2CC(F)(F)C2)=O)co1 c1(C(N2C3(CNC(C(C)C4CCC4)=O)CCC2CC3)=O)c[nH]c2cc(F)ccc12 c1(CC)nccnc1C(=O)N(C)Cc1cccc(CNC(=O)Cn2cnnn2)c1 CC1CCC=C1C(=O)N1CC(F)CC1CNC(=O)CCC1CCCC1 C1(F)(CNC(CN2C(C)CC2)=O)COCCN(C(=O)CCCNC(=O)C2CC2)C1 c1(OC)cccc(-c2cc(CNCC34CCCN(CC3)C4)n[nH]2)c1F C(c1ccc(C)nc1)=CC(=O)NC(CCNC(c1c(OC)cc(C)s1)=O)(C)C N1(C(C2(CCN=[N+]=[N-])CC2)=O)CC(=O)CC1C(=O)NCC1CC2(CC2)CO1 C(C(=O)NCCC(C(C)C)NC(=O)CCCn1ccnn1)(C(C)(C)C)SC C(C(=O)N(C)CCOCCNC(C1CC(C)(O)C1)=O)(C(C)(C)C)OC c1(C(=O)NCCCCCCN(C(CC(=O)NCC)=O)C)ccc(F)c(F)c1N c1(C(=O)NC2CCN(C(=O)CO)C23CC3)cc2sc(Br)cc2[nH]1 C(=O)(C1Cc2ccccc21)N(CCCCCCNC(C1CCC2CC1CO2)=O)C c1(CCC(=O)NC(C(C)NC(CNC(=O)OC)=O)C)c(C)noc1Cl C(=O)(C(C)C(C)O)N1CC(CC=C)(NC(C2(C(F)F)CCCC2)=O)C1 c1(C(=O)NCC(=O)NCC#C)cccc(C#C)c1C c1(C(=O)NCC(CC)NC(C2CC2(C(C)C)CC)=O)cc(OC)nc(F)c1 C(CC(C(=O)N=c1ccn(CC)[nH]1)NC(c1ccc(CC)cc1)=O)OCC c1(C(=O)NCc2c(CCNC(c3nn(C)c(O)c3)=O)ocn2)cccc(F)c1Cl c1(SC)nc(C)cc(NC(c2c(CO)cccc2)c2nnnn2C)n1 N1(C(=O)NC2CCCN(c3nn[nH]n3)C2)CCC(O)(C2CC2)CC1 C12(NC(c3c(OCC)nccc3)=O)CCCC1CN(C(C1CNC(=O)C1)=O)C2 Cc1ccc(C(=O)NC(C(=O)NCC(C)C2CC2)C2(O)CCC2)cc1C Cc1cc(C(=O)OCC2(C)CC2Br)c(N)c(F)c1 C(CC(C)(C)C(=O)Nc1ccc2c(c1)CC2)NC(C(CC)NC(C)=O)=O C(=O)(C(O)CCCc1ccccc1)NC(c1ccnn1C)COC C1(CCCC)NC(=O)CCN(Cc2cnc(-c3ccc(F)cc3)s2)C1=O c1(C(=O)NCC2CN(C(=O)C(=Cc3c[nH]cn3)F)C2)cc2n(c1)CCOC2 C1(C(N2C(CNC(c3ccc(C(F)(F)F)cn3)=O)CC2)=O)COCCOC1 Cc1c(C(N2CCC3CN(C(=O)CC(C)C)CC23)=O)ccc(Br)c1F c1(CNC(C2CC(N(C)CC3C(C)C3)C2)=O)cccc(Cl)c1Cl N1(C(c2cc(C)ncn2)=O)C2CCC(C2)C1CC(N1CCC(C)(CN(C)C)C1)=O C1(CC)CN(C(=O)CCc2c(F)cccc2F)CCC1NC(=O)C(C)=CC1CC1 C(=O)(CCC(=O)C(C)(C)C)N1C(C(=O)NC(CCCC)CC)CC2(CCC2)C1 c1(OC)cc(CC(=O)NC2CC2CNC(=O)C=Cc2cocn2)ccc1C CC1(C)CCCC(O)(C(=O)NC2CC2CNC(=O)CC2(C)OCCO2)C1 c1(N2CC(C)C(N(C)C)CC2)nc2ccsc2c(=NCC2(C(F)(F)F)CC2)[nH]1 C12(CC)COC(CNC(N3CCC(C4CCCN4)C3)=O)(C1)C2 C1(C(=O)NCC(CC)(C)O)CC2(CC(NC(c3n[nH]cc3[N+](=O)[O-])=O)C2)C1 Cc1c(Br)c(C(N2CCOCC2CNC(c2c(F)cccc2Cl)=O)=O)nn1C N1(C(C23N(C(CCCC)=O)CCC2C3)=O)CCN(C)CC1CC CCC(CNC(C1CC(C)=NO1)=O)(CC)NC(=O)C(C)SC C1(CNC(C2CCN(CC)C2)=O)C(C)CCCN1C(c1coc(SC)c1)=O C(=O)(C1=CC2CCC1C2)NCC1CC(C)(C)CN1C(c1nc2ccccc2[nH]1)=O c1(C(=O)NCCCOCCNC(C2C(=C)C2)=O)cnc(P(C)(C)=O)cn1 c1(OC)ccc(C(=O)NC(C)C(C(C)C)NC(c2ccc(C(C)C)nc2)=O)cn1 CC1=NN(C)C(=O)C1CC(=O)N(CC(C)CNC(c1cc(CO)[nH]n1)=O)C c1(C2CCC(=O)N2)cccc(Nc2ccc(C3CC3(F)F)cc2)c1 c1(C(=O)NCCCCC(C)NC(c2nocc2Br)=O)ccc2[nH]ccc2c1 N1(C(C2(SC)CN(C(C3CC(C)C3)=O)C2)=O)CC(C)CCCC1C C1(C(N2C(C)C(C)N(C(=O)C3=CC(C)(C)C3)CC2)=O)CC2(C1)CC1(CCC1)C2 C1CC(O)C(=O)N(C)C(CC)C(=O)N1.C(C)(C)(C)OC(N)=O N1(C(C2C(C)OCC2)=O)CCCCC(NC(=O)CCc2cnc(C3(C)CC3)o2)C1 C12(NC(=O)Cn3cccc3)CN(C(=O)Cc3cc(C4CC4)no3)CC1CS(=O)(=O)C2 n1(CCC(=O)NCC(CC=C)NC(c2ccns2)=O)nc(O)c2ccccc12 C(C(C)C(C)C)NC(CNC(CN(C1CC1)CC)=O)=O C1(c2ccc(N(C)C)cc2)C(NC(=O)CSCCC(=O)O)CC(=O)N1C1CC1 C(=O)(CCC(C(C)C)NC(=O)CC1(CSC)CC1)NC(COC)(C)C(N)=O CS(=O)c1ccccc1C(N1CCC2(C1)CN(C(=O)COCCO)C2)=O CCCCCC(O)CC(=O)NC(C1CC(NC(C2(CC(C)C)CC2)=O)C1)C N1(C(CS(CC)=O)=O)CC(C)CN(C(C2CCN(C)C(=O)C2)=O)CC1C c1(CCCC(=O)NC(CC2CN(C(=O)NC)C2)C(C)(C)C)ccc(Cl)c(C)c1 c1(C(=O)NCC2CCCN(C(c3sccc3Cl)=O)CC2)cc2n(n1)CC(F)C2 CCCCCCC(=O)NC1CN(C(=O)CC23CCCN2CCC3)C(C)(C)C1 C1(NC(C2CC(C)C2)=O)CCCCN(Cc2ccc(Cl)nc2)C1 C1(C(c2nnnn2C2CCOCC2)NCC=CC)CCOC1C C1(CNC(CN2CCC(C)C2)=O)CCN(C(c2cncc(N(C)C)n2)=O)C12CC2 C=C(C)CC(C(=O)N1CC(CCO)(CC)C1)NC(c1ccc(C)c(C)n1)=O C(=O)(CC(C)(C)C)NCC(=O)NC(C(=O)NC(CN(CCCC)C)C)(C)C C1(C(=O)NC2CCCCN(C(C(C)n3ccnc3)=O)C2)C2CCC(C2)C1(C)C N1(C(c2ccc(C)o2)=O)CCC(C)C1CNC(=O)C=CCN1CCCCC1 C=CCCCCC(=O)NC1CC(NC(=O)C=Cc2ccccc2)C12CCC2 N1(C(COCCNC(c2cc(C)c(O)nn2)=O)=O)CCCC(C)(O)CC1 C1(NC(CCNC(COC)=O)=O)CC(C)N(C(=O)CCC(=O)OC)C1 C1(C(=O)NCC(C2CCCC2)NC(c2coc(Br)c2)=O)CC2CCC(C1)O2 CC1COC(C(=O)NC2CC(NC(c3nccn3C)=O)C2)C1 C(=O)(CCC(C)N(C)C)NC1(CC)CN(C(=O)C=Cc2scnc2C)C1 N1(C(c2ccc(-c3nc(SC)[nH]n3)cc2)=O)CCCC(C)(C)CC1 C1(C(N(CCCNC(c2cncc(OC)c2)=O)C)=O)CCc2nc(=N)[nH]cc2C1 c1(C(CO)NC(C2CCN2C(C2(C(=O)OC(C)(C)C)CC2)=O)=O)cccnc1 N1(C(C2C(C)CCC2)=O)CCCC(C)C1CNC(=O)Cn1ccnn1 C1(C(=O)NCCn2c(CC)ncc2)CCN(C(=O)COCC(C)C)C12CC2 Cc1ccc(NCC(N2CC(OCCNC(=O)CSc3ccccn3)C2)=O)cc1 c1(C(N2CCC(NC(CC3(CC=C)CCCC3)=O)C2)=O)cccc(C)c1C#N C1(CNC(c2c(CC)nns2)=O)CC(C)N(C(=O)CNC(=O)Nc2ccoc2)C1 c1(OC)cc2c(cc1CN1CCCC(c3n[nH]c(C)n3)C1)OCO2 C1(NC(CCCC(C)NC(c2cc(C(F)F)[nH]n2)=O)=O)CC12CCCCCC2 C1(c2n(CCCOC)nnn2)(NCC2CCC=CO2)CCN(C)CC1 C(=O)(CC(C)(C)CC(C)=O)N.C1(C(=O)N(C(CC2CC2)c2ccon2)C)(OC)CCSC1 c1(CNc2c(C(=O)OC)cnn2C2CCCCO2)cc(Br)ccc1Br N1(c2nnc(C)o2)CCC(NC(c2cccc(-n3c(C)cnc3O)c2)=O)C(O)C1 C(=O)(CC(CCCC)NC(c1nnc(S)n1C)=O)NC(C#C)CC N1(C(c2ccc(C)c(O)n2)=O)CCCN(C(C2CCCOC2)=O)CCC1 CCCCCCC(C)C(=O)NC1CCCC1C(=O)NCc1cccc(CO)n1 CCC(C)CCCC(=O)NCCN(CCOCCO)C(C1CCCOCC1)=O CCCCC(CC)CCC(=O)N1CCC2(C1)CN(C(=O)CCC(C)SC)C2 c1(C(=O)NC2CC(C(=O)NCC(C3CCC3)OC)OCC2)ccn2cncc2c1 N1(C(c2c(CC)c[nH]n2)=O)CCCC1(C)C(N1CC2C=CC2C1)=O C1(CNC(C(CC=C)OC)=O)CCCCCN1C(=O)C(COC(C)C)OC n1(CC)nc(C(=O)NCCOC2CCN(C(C3CCS(=O)CC3)=O)C2)cc1C CCCC(=O)NNC(=O)NC1CCN(C(C)=O)CC1 c1(NC(C2(C)CC(NC(C(C=CC)O)=O)C2)=O)ccnc(CC)c1 N1(CCCOC)CCCC(NC(=O)C(=O)NCCOC2CCCCC2C)C1 N1(CC(=O)NC2CC3CCC2C3)CCCc2n[nH]cc2C1 C1(CCNC(COC(CC)(C)C)=O)CN(C(=O)C2=CCSC2)CCO1 N1(C(CC(=O)NC)=O)CCCC(CNC(C2(COC)CCOC2)=O)C1 Cc1n[nH]cc1C(C(=O)C(=O)CN(CC#N)C(C)C)N.C1(SCO)CCCO1 c1(C(N(C)CC2CCCC2NC(=O)CCn2ccnn2)=O)ncn2c1CCC2 C1(CC(=O)N(C2CCN(C(C(=O)NCC)=O)C2)C)CCC2(CCC2)O1 C1(C(N2CCC(C)CC2)=O)CCCN(C(C2(F)CCOC2)=O)CC1 N1(C(c2c(C)occ2)=O)CCC(CC(=O)N(CC(=O)NC2CC2)C)CC1 CCCC(CCCNC(C1(C(C)C)CCCO1)=O)NC(c1csc(=NC)[nH]1)=O C=C(C)CC(C(=O)NC1(CC(=O)N(C)Cc2ccns2)CCCC1)OC C(=O)(CCCCCC(C)C)NC1C=CC(C(=O)NCCC2(OC)CCC2)C1 CCCCC(CC(=O)N1CCOC(CCO)C1)NC(=O)CC1COCCCO1 N1(C(CCC#C)=O)CCC(CO)(COC)C1.C1(=O)CCC2CC(C2)N1 N1(C(C2CC(CC)C2)=O)CCC2CCCC12C(N1CC2CC(C)C1C2C(=O)O)=O Cc1cc(Br)cnc1CCNC(=O)C(N1CCCC1CC1CCOCC1)=O c1(OC)ccc(I)cc1CN1CCN(C(C2CCCN(C)C2)=O)C(C)C1 C1(CNC(CC(=O)OCCC(C)C)=O)CCN(C(=O)Cc2ccoc2)CC1 c1(C(=O)NC2CN(C(CCC(C)C#N)=O)CC2C)ccc2[nH]c(=O)c(=O)[nH]c2c1 C1(C(=O)NCC2(O)CCC(C)C2)CC2(CC2)CN1C(c1cnsc1)=O c1(C(N2C(CN(C(=O)C=CC3CC3)C)COCC2)=O)cc2cccc(O)c2[nH]1 C#CCCCC(C)C(=O)NC(CC1CCC1)C(N1CC(OC)CC1C(=O)OC)=O N1(C(C2N(CCC)CCC2)=O)CC(NC(=O)CCNC(=O)COC)CCC1C N1(C(C2CC(C)(C)N(C(=O)CCC(=O)C3CC3)C2)=O)CCC2(CCC2)C(CO)C1 CC1CC(CNC(=O)CCN(C(=O)C(=Cc2cn[nH]c2)C)C)CCO1 C(=O)(C(C)(C)C(O)CC)N(CCN(C(C1C(CCC)C1)=O)C)C.c12nnn(n1)C2 CCCCCC(C)c1nc(CC(CC)OC)nn1-c1ccc(C(C)C)cc1 Cc1ccc(NC(N2CC3C(C2)N3C(=O)Cc2ccc(O)cc2)=O)c(I)c1.C C(=O)(C1=CCC2CCC1N2C(c1csc(Cl)n1)=O)N1C(C)(C(=O)NC)CC1 c1(CCC(=O)NC2C(CNC(c3nc(N(C)C)oc3)=O)CC2)c(Cl)cccc1Cl CC1(C)OC2(CNC(C3(C)CCC3)=O)CC1(NC(=O)CCC1CCCCCC1)C2 C(=O)(C(C)C1=CCCC1)NCCCCC(C)NC(c1cccc(C(=O)OC)c1)=O CCCC(C(=O)NCCN(C(=O)C(C)OCCOC)C)c1cccc(Cl)c1 CCCCCCC(F)C(=O)N1CC(F)(CNC(=O)Cc2ccc(OC)cc2F)C1 C(C(C(C)(C)C)NC(c1nc(O)c(C)s1)=O)NC(Cn1ncc(C(=O)OC)c1)=O C(=O)(CC1OCc2cc(Cl)ccc21)N1CCC(O)(C(N2C(C)COCC2)=O)CC1 N1(Cc2c(C)cc(C)[nH]2)CC2CC1CN2C(c1ccc(Sc2cccc(Cl)c2)o1)=O c1(C(=O)NC2C(NC(C3CCN(C(C)=O)C3)=O)CCC2)ccc(F)c(Cl)c1N C12(NC(CCSCCC)=O)CC(CNC(C3CCCNS3(=O)=O)=O)(C1)OC2C c1(CN2CC(NC(c3ccccc3OC(F)F)=O)C2)ccc(F)cc1Cl c1(C(=O)NCC(C)CNC(=O)CNC(=O)CC(F)(F)F)cnc2c(c1)COCC2 Cc1cccc(C(C)(C)C(N2CC(NC(c3nc(C)c(C)[nH]3)=O)CC2C)=O)c1 c1(C(=O)NC2C(CNC(C3(NC(=O)OC)CCCC3)=O)C2)ccc(Cl)c(F)c1 N1(C(c2c(C)nco2)=O)CCN(C(c2cc3c(s2)CCC3)=O)C2CCCCC12 C=C(F)C1(CC(=O)NCc2ccc(C(=O)N(C3CCC3)CCN(C)C)s2)CCC1 c1(CCC)ccccc1C(=O)NC(C)CCN(C(=O)CCC1CCOCC1)C C1(C2CCN(C(c3ccc(F)nc3F)=O)C2)(NC(=O)C(=Cc2c[nH]cn2)F)CC1 Cc1ccccc1Cn1cc(C(C)NC(=O)CCn2cccn2)nn1 C1(NC(=O)CCc2cscn2)CCOC(C(N2CCSCC2CO)=O)C1 c1(NC(=O)CCc2cc(F)ccc2[N+](=O)[O-])ccc2ccccc2n1 C1(N(C(c2c(CC)cns2)=O)CCO)CCN(C(C2(OC)CS(=O)(=O)C2)=O)CC1 c1(NC(C2N(C(c3cc(C)c(F)cc3)=O)C3C(C2)C3)=O)c(C)cc(Cl)nc1Cl c1(OC)ccc(CC(N2CCCC(C(F)F)C2)C(=O)NCCCF)c(OC)c1 CC1CC(C)N(C(c2cc(F)c[nH]2)=O)CCN1C(c1csc2c1CCCC2)=O Cc1cc(OCC(=O)NC2CCN(C(=O)COCC3CCC3)CC2C)cc(C)c1 c1(C(=O)NC2(C)CCN(Cc3nc(C(C)OC)sc3)C2)n[nH]c2c1COC2 c1(C(N)=O)cnc(Cl)[nH]c1=NCCC1CCN(C(c2ccc(F)cn2)=O)C1 C(=O)(C(=O)C(C)(C)C)N1C(CN(C)C(c2cccnc2F)=O)CCC1 c1(C(=O)NC2CN(C(C(C(C)O)NC(N)=O)=O)C2)cc2cccc(F)c2o1 C(CCCCCNC(=O)CC1CC(C)=NO1)NC(c1cc(OCC)n[nH]1)=O C1(C(=O)NC(C)CCCl)C2CN(C(c3cccnc3C(=O)N(C)C)=O)CC12 c1(C(=O)NCC2C(CNC(CC3(CC)CCC3)=O)C2)ccc(OCCF)cc1 C(=O)(C1=CCN(C(C2(CC3CC3)CCCCC2)=O)CC1)NCC(NOCC)=O C1(NC(c2c(CNC(C3(C)CCCN(C)C3)=O)cc[nH]2)=O)CCc2nncn2C1 C1(C(C(=O)NC(CC)CNC(=O)CCn2ccnn2)C)CCC(=O)N1 c1(-c2nc(C3CC4(c5ccccc5C4)OC3)on2)n[nH]c(=NC2CCCCC2)o1 c1(CC)ccc(C(=O)C(=O)NCc2c[nH]nc2C2CCN(C(C)C)C2)s1 S(=O)(=O)(C(F)(F)F)NCCC(=O)N(CC(O)CNC(=O)CC1CC=CC1)C C1(CC)CN(C(c2nc(Br)cn2C)C(=O)NC2(C)CC2)CC1N(C)C c1(CC)nnc2n1CCCC2C(=O)N1CCCC(N(C)C(C2OCCO2)=O)CC1 c1(CC(N2C(CCC(=O)NC(C)(C)C(N)=O)CCC2)=O)cccc(F)c1F N1(C(C(CC=C)C)=O)CC23CCCC2(C1)CN(C(c1cc(O)cc(O)n1)=O)C3 N1(C(CCN(CCCCC)CC)=O)CC(CNC(=O)CSCC(N)=O)CC1(C)C C1(NC(C(C)SC(F)(F)F)=O)CCCCC1NC(=O)C=Cc1cocn1 CC1CN(C(C2(CF)CC2(F)F)=O)CC1NC(C1CCC(n2cccc2)CC1)=O C#CCC(CC(=O)NCCC(C)O)NC(C1CCCC1O)=O c1(C(N2C(CCNC(C3(C)CC(=C)C3)=O)CCCC2)=O)cc(C)cc(F)c1 c1(C(c2nnnn2CCN2CCOCC2)NC(c2nncn2C)C)nn(C)cc1Br C1(CCC(=O)N(C(CC)C)C)CCN(C(=O)CSc2ccncc2)C1 C1(C(NOCC)=O)(OC2CC(=C)C2)CCN(C(c2ccc(=N)[nH]c2)=O)CC1 N1(C(CCC=CCC=C)=O)CC(NC(=O)Cc2c(Cl)cnn2C)C(O)C1 C(CC)(CC(=O)NC)N(C(c1cccc(I)c1)C(=O)NCCCC)C C1(NC(c2c(C)oc(Cl)n2)=O)CCC2CN(C(=O)CCn3cnc(=N)[nH]3)CC2C1 n1(CC(=O)NCC2CC(F)(CNC(=O)C(F)C3CCC3)C2)ncccc1=O C(=O)(CCCS(N)(=O)=O)N1C2CN(C(C3N(CCC)CCC3)=O)CC1C2 C12(NC(Cn3ncc(C)c3)=O)CCCC1CN(C(c1cccc3[nH]ccc13)=O)C2 N1(C(c2nccc(C#C)c2)=O)CC2(CCCC2)C1C(=O)NC1CCCC(C2CC2)C1 N1(C(CCC#C)=O)CCC2(CC1)CC(C)N(C(c1ccc(OC)c(CC)c1)=O)C2 c1(-n2cc(C(=O)NCC3OCC(CNC(CCC)=O)C3)nn2)ccc(Cl)cc1Cl N1(C(C2CN(C(C)C)C2)=O)C2CCC1CN(C(=O)C(F)(F)CO)CC2 C=CC1(C(=O)NCC2CC23CC3)CCN(C(c2cn(C3CC3)cn2)=O)C1 c1(OC)cc(F)ccc1C(N1CC2CC2(C(=O)Nc2ccc(N(C)C)cc2)C1)=O Cc1c(NC2CN(C(=O)CCCn3ccnc3)C2)ncnc1Cl C(=O)(C1=CCC2(COC2)OC1)N(C)CC1CCCN(C(=O)Cc2csc(S)n2)C1 c1(CCC)[nH]ccc1C(=O)NCC1(F)CC(CNC(C2(CC)CC2)=O)C1 c1(CC(N2CC(C)C(n3cc(CN4CC5CC5C4)nn3)C2)=O)cnc(O)nc1O N1(C(C2N(C(COCC(C)C)=O)C3C(C2)C3)=O)CCOCCC1C(C)C c1(C(N2CCC(Nc3nc(C)c(F)cn3)C(F)C2)=O)ccc([N+](=O)[O-])c(C)c1 C1(CNC(C(COC)(C)C)=O)COCCN1C(=O)CC1COC2CC1C2 C(CC(C)CCNC(C1CC2C=CC1C2)=O)NC(c1cc(CC)no1)=O CC(C)(C)C(CC(=O)NCCN(C(=O)Cc1c[nH]ccc1=O)CC1CC1)C(F)F c1(CNC(c2scc(C)c2)=O)cc(C)c(C(N2CC(C)(CF)C2)=O)o1 Cc1cccc(CC(=O)NC2CN(C(=O)CN3CCOCC3)CCC2CO)c1Cl Cc1cc(C(=O)NCCC2CCN(C(=O)CCC3CC3C)C2)nn1C(F)F c1(C(=O)NC2CN(C(c3[nH]cc(C#N)c3)=O)CC2O)c(F)cc(Cl)cc1F C(c1cccc(O)c1)=CC(N1C(C(C)NC(=O)CC2CCCC2O)CCCC1)=O C1(NC(=O)CCc2ccsc2)CCCN(C(=O)CCCn2ccnc2)C1 c1(C(=O)NC2CC2(F)F)cc(F)cc(F)c1.N12CCCC1C1(CC1)N(C)CC2=O CC1CN(C(c2ccnnc2S)=O)CCC1NC(=O)CC(=O)NC1CCCC1 N1(C(CC(CC)SC)=O)CC(C(=O)NCc2ccnc(C#N)c2)CC(C)(C)C1 CC(c1ccc(F)cc1F)=CC(=O)N(c1ncc2cccnc2n1)CC(C)C C1(C(=O)Nc2cc(C)c(Cl)cn2)CCC2(CN(Cc3cc(F)cc(Br)c3Cl)C2)O1 C12(COC(c3cccc(C4CCC4=O)c3)=O)CC3CC(C1)CC(Cl)(C3)C2 N1(C(C(c2scc(C)n2)C)=O)CC2(CCC(CNC(=O)C(C)NC=O)O2)C1 N1(C(c2ccn(C)c2)=O)CCC2CN(C(c3ncc(Cl)cn3)=O)CCC12 C(=O)(C(C)(C)CCCNC(=O)C=CCn1ccnc1)NC(C)C=CC(F)(F)F c1(C(N2CC(C(C(=O)NC(C)CC(C)C)OC)C2)=O)c[nH]ccc1=O c1cn(C)c2cc(F)ccc12.CC1CN(C2CC2)CCN1C(=O)C(=O)N CCC(Cc1ccccc1)C(=O)NC1CC(NC(c2c[nH]nc2C(C)(C)C)=O)C1 C1(C(N(C(CC)CNC(C2CSCCS2)=O)C)=O)CCS(=O)CC1 c1(C(N(CCC(N2CCCC(C(C)C)C2)=O)C2CC2)=O)cc2ccccc2o1 CC(=O)C(C)CC(C)C(=O)N(C(C)C(=O)NCC12CCC(CC1O)C2)C1CC1 C1(CC=C)(C(=O)NCC(O)CNC(c2nnc(Cc3cc[nH]c3)s2)=O)CCCC1 Cc1nonc1CNC(C1(CCNC(=O)C(O)CC2CCCC2)CCCC1)=O C1(CC(N2CC(NC(=O)NC)C2)=O)CCN(C(C2CC(SC)C2)=O)C1(C)C C(=O)(C(C)(O)CCc1ccccc1)NC(CNC(c1c(C)ncn1O)=O)CC(C)C Cc1ccc(S(=O)(=O)N2CCN(CCC(C)Sc3cccc(F)c3)CC2)s1 C1(NC(=O)CCCC2CC2)CN(C(C2(C3CCC3)CC2(F)F)=O)CC2(CC2)C1 C1(CC)CCCN(C(=O)CS(C)(=O)=O)C1C(=O)NC1CCCC(C(C)C)C1 c1(C(=O)NCCC2N(C(=O)CCC(F)(F)F)CCC2)cc2ccncc2[nH]1 CCCC(C)(CC)C(=O)NCC1(NC(C2OC3CCC2C3)=O)CCOCC1 C(C(=O)N(C)CCNCC(CC)O[Si](C)(C)C)OC(C)C Nc1c(C(=O)NCC2CCCN(C(=O)CCC(F)F)C2)cnn1-c1ccncc1 N1(C(c2cc(=NCC)[nH]cc2)=O)CCC2CCCN(C(=O)Cc3cnns3)C2C1 C1(CC)C(NC(=O)C2=NNC(=O)C2)CCCN1C(=O)CC1CCCCC1O c1(C(=O)NC2C(C(=O)NC(c3cccc(I)c3)C)C2)ccc2[nH]c(=N)sc2c1 C1(C(=O)OCC)CCN(C(=O)C(C2CC2)NC(=O)CC23CCCC2C3)O1 Cn1nc(O)cc1C(N1CC(C)(c2cn(Cc3ccc(I)cc3)nn2)C1)=O N1(C(CSC(C)C)=O)CCC(C2CCN(C(C3C(C)OC(C)C3C)=O)CC2)C1 c1(C(C)=O)sc2ccccc2c1C(=O)NC(C(=O)O)c1cnsc1 c1(CC)nc(C)[nH]c1C(=O)NCc1cn(CC(C)NC(C2CC3CC3C2)=O)nn1 N1(C(CCC2CCN(C(c3c(CC)cncc3)=O)CC2)=O)CC2COC(=O)C2C1 N1(C(C=C(C)Cl)=O)CCN(C(=O)Cc2csc(=N)[nH]2)C(c2cc(F)ccc2F)C1 C1(O)(CNC(C2C(C)CCC2)=O)CCN(C(=O)CN2CC(C)(C)C2)CC1 C#Cc1cccc(C(=O)NC(C)CCCNC(=O)C(C)CC(C)C)c1Cl c1(C(N2CC(NC(C(C(C)C)OC)=O)C(C)CC2)=O)ccccc1S(C)(=O)=O C1(NC(C(C)S(C)(=O)=O)=O)CCCCCN(C(=O)Cc2cc(F)ccc2Cl)C1 C(=O)(CC1=CCN(C(c2cccc(I)c2)=O)CC1)NCc1nccc(C)c1 c1(C(N2CC3C(CN(C(CC4(C(=C)F)CCC4)=O)C)C3C2)=O)cnn(C)c1C#N c1(C(=O)NCC(C2CCCC2)NC(c2coc(C(F)F)n2)=O)ccc(F)cc1F c1(C(N2CCC(C(C)NC(=O)C(N)=O)C2)=O)ccc(C2=CCOCC2)cc1 C=C(C)CCCC(=O)Nc1ccc(Cl)c(O)c1.C1C(F)(F)C(=O)N2CCN1CC2 C1(C(=O)NCC2(F)CN(C(C(CCOC)C)=O)C2)CN(CP(C)(C)=O)C1 N1(C(C(CCF)NC(C2CCOC2C2CC2)=O)=O)CCCC(F)(F)CC1 CCCCC(CNC(C1CCCN1C1CCCC1)=O)NC(c1ccccc1)=O c1(OCC(=O)NC(CC2CN(C(C3C(C(=O)OC)C3)=O)C2)C)cc(C)c(Cl)c(C)c1 C1(NC(COCCC)=O)CCCN(C(C2CCCC(C(N)=O)C2)=O)C1 c1(C(=O)NC2CCCN(c3c(C(=O)OC)cccn3)C2)ccc(Br)c(F)c1F C1(C(=O)NC2CC3(CCCO3)C2)CCCCCCN1C(=O)CCc1ccc[nH]1 C1(C(N(CC(C)OC)C)=O)CCN(C(=O)OC(C)(C)C)CC1C C(=O)(C(CC1CC1)NC(C1CCC1(F)F)=O)N(CC(C)(F)F)C C1(NC(C2(O)CC2)=O)CCC2CN(c3cc(O)nc(O)n3)CC2C1 c1(-c2n(CCC)ncc2)ccc(NC(c2ncc(-c3ccccc3)cn2)=O)nc1 C(C(C)(C)C)N(C(=O)N(CC#N)CCOC(C)(C)C)C CC(C)(F)C(C)(F)C(=O)NC1CCC(CNC(c2ocnc2C(F)(F)F)=O)CC1 c1(NC(c2ccc(=N)[nH]c2)C)[nH]c(=NCCC(C)(C)CO)nc2scnc12 C(CN=C(NCc1cnc(C2CC2)[nH]1)N1CCC(C2CCCC2)C1)OCC=C c1(C(=O)NC2CCN(C(c3n[nH]c(C)c3F)=O)CC2O)cccc2occc12 N1(C(CSC)=O)C2CCC1CC(N(C)C(C1CCC3(CCCO3)O1)=O)C2 c1(C(N2C(C)CC(Nc3ncc(C(=O)OC)cn3)C2)=O)cc(F)ccc1C C1(C(=O)NC(c2cnn(C)c2)CO)(NC(CN2CC(C)(OC)C2)=O)CCN(C)C1 C1(Oc2cccc(OCc3ccccc3)c2)CCC2CNCCC2C1 c1(C(N2CCN(CCCNC(c3ccccn3)=O)CC2)=O)[nH]cc2c1CCC2 CCC(C)(C)CCCNC(=O)Nc1cc(O)cc(F)c1 C1(NC(C(CSC)C)=O)CCN(C(=O)CCC(C)(C)C)C(C)C1 Cc1nn(C)cc1CCC(=O)NCC1CN(C(c2csc(C)c2C)=O)CC1O C1(COC)(NC(=O)CN2CCC(C)C2)CCN(C(c2ccc(N)cc2F)=O)CC1 Cc1c[nH]cc(C(=O)NC(C2CCCCC2)C(C)NC(c2nnn(C)n2)=O)c1=O c1(NC(c2ccc(CCNC(c3ccncc3O)=O)cc2)=O)cc(F)ncc1Br c1(C(=O)NC2(C)CN(C(=O)C(C)(C)c3cc[nH]n3)C2)c(Br)ccc(F)c1F C1(C(N(C(CC)CC)CC)=O)CCCN(C(=O)CCC2CCOC2)C1 Cc1cccc(C(O)C(N2CCC(C)(NC(c3cnn(CCF)c3)=O)C2)=O)c1F N1(C(=O)N(C(=O)C2CC2SCc2cccnc2)C2CC2)CCOC(C2CC2)C1 C(C1C(C(=O)NCC#CCNC(C2(N3CCOC3=O)CC2)=O)C1(C)C)=C(C)C C1(NC(CCN(C(C(c2ccn(C)n2)C)=O)CC2CC2)=O)CC(=O)N(C)C1=O C1(C(=O)NCC2CCCC(C(=O)NC(CCC)C3CC3)C2)CC12CCCCC2 Cc1cc(C)c(NC(C2CC(C)CN2C(C2CCOC2C(C)C)=O)=O)cc1C N1(C(C(COC)(C)C)=O)CC(CO)CC1(C)C CN=c1cc(C(=O)NCCNC(c2onc(C)c2C)=O)cc[nH]1.c12cnc(s1)NC2 CC1(C)OC(=O)CC1C(N1CCOC(CC(=O)NCC2C3CCCC23)C1)=O CC1C(NC(=O)C(O)C2CN(C(c3cc(C(N)=O)co3)=O)C2)CCCC1C(N)=O C1(C(N(CCC=C)CCO)=O)CN(C(c2ccc(OC)cc2)=O)CCC1O N1(C(c2c(OC)cncc2)=O)CCN(C(C2CCOC2(C)C)=O)CC12CCC2 c1(C(=O)NCC2CC(NC(C(COC)C)=O)C2)cccc2nc(N(C)C)oc12 c1(C(N2C3CCC(NC(C=CC)=O)C(C3)C2)=O)cccc2c1OCCC2 N1(C(c2nncc(C)c2)=O)CCCCC(NC(C2NC(=O)CC2C)=O)C1 C(=O)(C1=NN(C(N)=O)C(=O)CC1)NC1CCC(N(C)C)CC1 N1(C(c2cc(C)cc(F)c2)=O)CCC2(CCCC2NC(=O)C=C2CCCC2)CC1 C12(NC(C(C)(C)O)=O)CCOCC1CN(C(=O)CS(=O)(=O)C(C)(C)C)C2 c1(SCC)ccc(CC(=O)N(CCNC(=O)CC2CC3C=CC2C3)CC)cc1 c1(Cl)ccc(CO)s1.c1(C(=O)NCC2CC2CC(=O)NCC2CC2)c[nH]nc1C1CC1 c1(C(N2C(CC)CN(C(=O)CC3CCC(F)(F)C3)CC2)=O)cc(C)c(F)c(C)c1 C1(O)(CCNC(c2cncc(COC)c2)=O)CCCN(C(=O)CCS(C)=O)C1 c1(C(=O)OC)cc2ccccc2[nH]c1=NC(CNC(=O)C=C(C)Cl)C(C)C(C)C CCC(CC(=O)NC1CCC1NC(=O)C(=O)N(C)C)C(C)C CCS(=O)(=O)CC(=O)N1CC(NC(c2cccc(Cn3ccnn3)c2)=O)C2CC12 C(=O)(C1=NN(C)C(=O)CC1)NC(COCC)C(=O)NC1Cc2ccccc2C1 C1(CC)(NC(=O)C(n2cnc(C#N)n2)C)CCCN(C(c2ccncc2C)=O)C1 c1(C(=O)NCC(C)N(C)C(c2cc(C(F)F)no2)=O)ccc(Cl)cc1O c1(C(=O)NCC2N(C(C3C(=C)C3)=O)CCC2)cncc(C(F)(F)F)n1 C1(CNC(CN(C2CC2)CC)=O)OCCC1C(=O)NC1(C)CC1C C(=O)(C1=CCN(C(=O)C(CC)CC(C)C)CC1)N(C1CCN(CC)C1)C C=C1CCC(CN2CCCCC2)CC1.C(=O)(C(=O)N)NCC=CCO C(=O)(C1=CC(c2ccccc2)NC(=O)N1)NC(CCCC)CSc1ccccc1 C=Cc1ccc(C(=O)N(CCCNC(c2ccc(COC)[nH]2)=O)C)cc1 CC(CC(=O)N1CC(CC(C)NC(C2(C(N)=O)CC2)=O)C1)CC(F)(F)F c1(OCC(N2CCCC(CNC(Cc3cnc(C)[nH]3)=O)C2)=O)c(Cl)cccc1Cl C1(CCOC)CN(C(c2cncnc2)=O)CCN1C(=O)C(C(C)(C)C)SC CC1C(NC(C2CC(O)C2)=O)CC2CCC1N2C(=O)CN1C(C)CCC1C Cc1nc2ccccn2c1C(=O)N(CC(N)=O)Cc1cc(C(=O)O)no1 C1(C(=O)NC(COC)C(=O)NC2CC2(C)C)C2(CC2)C12CC2 N1(C(CCC2(C#N)CCC2)=O)C2CCC(C(N3CCn4nccc4C3)=O)C1CC2 c1(OC)cc(C(=O)NC2CCC2NC(C2CC(C)=NO2)=O)cc(F)n1 c1(C(=O)NC2CN(C(C3(COC)CCOC3)=O)C2)cc(Cl)cc(C)c1N C1(C)(C(N(C2CCN(C(C(Cn3ccc(C)n3)C)=O)CC2)C)=O)CCC(=O)NC1 c1(NC2CCN(C(CCN(C)CC)=O)CC2C)cc(=O)n(C(C)C)c(O)n1 O=S(=O)(c1ccc(Br)cc1Cl)N1CCN(Cc2cnc(-c3ccccc3)s2)CC1 C#Cc1ccc(C(N2CC(C)(C)C2C2CCN(C(=O)COC)CC2)=O)cc1 c1(C(=O)NC2C(SCC)CCCC2)ccn2nnnc2c1.C1(=O)CS(=O)(=O)N1 Cc1ccc(C(=O)O)cc1NC(c1ccc(SC(F)(F)F)cc1F)=O C(=O)(CC1CCOc2ccccc21)NC1CCC(NC(=O)Cn2cnnn2)C1 N1(C(N(C)C)=O)CCCN(C(=O)NC2CCC(F)CC2)CC1 c1(C(=O)NC2CN(C(C3C(CC)C3)=O)CC2C)ccc2[nH]c(C)c(C)c2c1 C1(C(=O)NCc2cc(C(N3CC(CN=[N+]=[N-])OCC3)=O)no2)CCCC(F)(F)C1 O=C(C#CCNC(=O)C=CC1CC1)NC1CC(F)(F)C1 C(=O)(C(C)(C)F)NC(CN(C(c1csc(CC(F)F)n1)=O)CC)C C1(CC#C)CCCCN1C(c1ccc(CNC(c2ccco2)=O)s1)=O N1(C(CC(CC2CC2)OC)=O)CCC12CCN(C)C2 C1(C(=O)NC2C(NC(C3(C)CCC3)=O)CC2)CCN(c2ccccc2)C1=O C#CCCCC(=O)NC(C1CCN(C(C2CCOC(CCC)C2)=O)CC1)C N1(C(C2(CC=C)CCC2)=O)CC(CNC(c2c[nH]nc2C(F)F)=O)CCC1C C(=O)(C(C#N)C(C)(C)C)N(CC(C)NC(=O)C1=CC2C=CC1C2)C c1(C(=O)NCC(CC)NC(C2C3CC(F)(F)CC23)=O)cc(C)c(O)c(N)c1 C1(NC(=O)Cc2cnsc2)(CO)CCCN(C(=O)CN2CCCC2CO)C1 N1(Cc2n(CC)ncn2)CCOCC(C(=O)NC(C)CCSc2ccccc2)C1 CN1CCC(C(=O)NC2CC2NC(c2cocc2C(N)=O)=O)CC1=O c1(C(N2CC3(CN(C(CCC=C)=O)C3)OCC2)=O)ccc2c3c(cccc13)CC2 N1(C(N2CCC(C(=O)Nc3ccc(CC)nc3)(CC)C2)=O)Cc2ccccc2C1 S(=O)(=O)(c1ccc2nc(O)[nH]c2c1)N1CC(C)(C(N2C(COCC)CCCC2)=O)C1 CCC(C)(CNC(=O)CCCCNC(N)=O)C(=O)N1CCC1(C)C C(=O)(C(F)(CNC(=O)C=C(C)CCC)C(C)C)N(CCOCCOC)C c1(C(=O)O)cccnc1OC(F)F.C12=CC=C(C=C1)C2.N12CCCC1C2=O c1(C(N2CCN(C(C(CC#C)C)=O)C(CC(F)(F)F)C2)=O)c(C)cc(Cl)cc1C C1(CNC(c2c(CC)onc2)=O)CCC(C=O)CC1.N(CCO)C1CC1 c1(OC)ccc(C(=O)NC2CCC2NC(c2ccnn2C2CCOCC2)=O)cn1 CC1CC(NC(C2CCN(C(=O)Nc3ccco3)C2)=O)CN1c1ccccc1 C1(O)(CNC(C2(CC)CCC2)=O)CCN(C(=O)CC2CCCC(=O)N2)C1 N(C1C(O)CCCc2ccccc21)c1[nH]c(=NC(CF)c2ccccc2)cc(C)n1 N1(C(C(C(C)(C)C)C2CCCCC2)=O)Cc2ccc(CNC(=O)C3CC3)cc2C1 Cc1cc(CCC(=O)N2CC(NC(c3nnsc3C(F)F)=O)C2)no1 CC(C)CC(C(=O)NC(C)(C)CC(N1CCCC(C)(C)C1C)=O)C(N)=O c1(C(=O)NCC(C)(C)NC(C=C(C)c2ccco2)=O)ncnc(O)c1Br c1(C(=O)OC(=O)NC(CC=C)CNC(c2cccc(CO)c2)=O)c(Cl)nn(C)c1Cl Cc1ccc(C)c(SCC(=O)NCC2CCCCN2C(=O)C(F)CC2CCC2)c1 C1(NC(c2c(CCC)[nH]cc2)=O)CC(C(=O)NC2CCCCC2CC)CC1O C1(N(c2nc(-c3cccc(Cl)c3)cs2)C)CC(C)(C(=O)OCCO)CC1(C)C S(=O)(=O)(c1cc(F)c(Br)cc1F)NC(C1N(Cc2nccs2)CC2C(C)(C)C21)=O C(C(COC)CC(=O)N1CC(F)(CNC(C2CN(C)CC2C)=O)C1)OC c1(N2CCC(C=C)C2)nc(=NCc2sccc2Br)[nH]c2ncn(CC)c12 c1(Cc2[nH]nnc2C2CC2)ccccc1F.N12CCOCC1NC(C)C2 C1(NC(Cn2cc(CNC(C3(C)CCCO3)=O)nn2)=O)COCCC1O c1(OC)ccc(C(=O)NCC2CCCN(C(=O)Cn3cnccc3=O)C2)cc1 C1(C(=O)NCCCNC(c2ccc(CO)o2)=O)CC2CSCC(C1)C2(F)F C(=O)(CCCOC1CCC1)NC1CC(N(C(C(C)n2ccnn2)=O)C)C1 n1(CC)nnc(C(=O)NC(C)(CO)C(=O)NC2CC(=O)N(C(C)C)C2)c1C O=[N+]([O-])c1cc(Nc2ccccc2-c2nc[nH]n2)c2c(c1)OCCO2 C(=O)(C1=C(C)OCCS1)NCCN(C(=O)CC12CCCN1CCC2)CC C1(C(c2n(CCSC)nnn2)NCC2CC(C)C2)CC2CCC1CC2 c1(NC(c2nc(C(F)(F)F)n[nH]2)C)cc(N2CCC(c3nc(=N)[nH][nH]3)C2)ncn1 C(c1cncnc1O)=CC(=O)NCCC(C)(C)NC(C1N(C)CCC1)=O N1(C(C(CC)O)=O)CC2(CC(CC(=O)Nc3ccc(Br)cc3O)C2)C1 C(CC1CCC1)(C(=O)NC1CC(CCC(=O)N(C)CCN2CCCC2=O)C1)OC N1(CCc2cn(-c3c(C)cc(C#N)cc3)nn2)CC2CCCCCC2(C#N)C1 c1(N2CCOCC(C)C2)nc(N2CCc3ncccc3C2)c2c(ncn2C)n1 C1(C)(C(=O)NC(CN(C(=O)Cn2ncccc2=O)C)(C)C)CCCC1(F)F c1(CN2CCCC(C(=O)CCN)C2)cc(Cl)cnc1Br.c1(O)ccccn1 C1(NC(CCc2onc(C)n2)=O)CC2CN(C(c3ccc(C(F)F)o3)=O)CC12 C1(=O)N=C2C=CN(N2)CCN1.c1(CNC(=O)OC(C)(C)C)cscc1Br c1(CN2CC3N(C(c4c(CCC)onc4C)=O)C3C2)ccc([N+](=O)[O-])c(F)c1 N1(C(c2ccc(CC)s2)=O)CCCCCC(NC(=O)Cc2sccc2Cl)C1 C=Cn1nccc1C(=O)NC1(CNC(c2ccnn2C2CC2)=O)CCCCC1 C1(N(C(c2[nH]cc(C(C)=O)c2)=O)C)CCCCN(C(C2CCC(C)O2)=O)C1 c1(C(c2nnnn2CCCO)NCC(C(=O)OCC)OC)cc(Cl)c(Cl)[nH]1.C(C)S C1(C(=O)NC2(COCC)CC2)CC(O)CCN1C(c1[nH]cc(C)c1C)=O C(=O)(C1=CC2(CCOC2)C1)N1CCN(C(c2cccc3c2CCC3)=O)C(CF)C1 C1(C(=O)Nc2cc(-c3ccccc3)sn2)CN(C(c2cnon2)=O)CC12CC2 C1(C)(C(=O)NCCC(N2CCN(C)CC2)C)CCCN(CCC2CCCCC2)C1 c1(CC(N2CC(CNC(C(C)CN(C)C)=O)OCC2)=O)ccnc(Cl)c1F N#CC1CN(C(=O)CC2CCCC(NC(=O)C(F)C3CCCC3)C2)CC12CCC2 C12(COC)CC(CNC(C3(C(N)=O)CCC3)=O)(CN1C(=O)C1=CCCCC1)C2 c1(C(=O)NCC(C(C)C)NC(C2Cc3cscc3C2)=O)ncc([N+](=O)[O-])n1C c1(C(=O)NCC(C)(CO)NC(C2CCN(C)C2=O)=O)ccc2nonc2c1 Cc1cn2c(C(=O)NCC=CCNC(C3CCC(=O)N3)=O)cnc2s1 C1(OC)CCC2(CCCN(C(=O)C(=O)NC(=O)Nc3cnn4ccn(C)c34)C2)C1 C1(=CC(=O)NCCN(C(C23CC(C)C2C3)=O)CC)CCN(C)C1 C1(NC(C(c2n(C)nnc2)(F)F)=O)(CO)CCCN(C(C2CSCC(=O)N2)=O)C1 C1(C(N2C(C(=O)NCC#CCCO)C=CCC2)=O)CC2CCC(C1)C2 C1(CNC(C=CC(=O)OCC)=O)CCC(C(=O)NCCCN2CCC2)C1 c1(CC(=O)NC(CC)CNC(=O)COC2CC=CC2)cncnc1 C1(CC(N2CC(SCC)C2)=O)COCCN(C(=O)CCC23CCC(CC2)C3)C1 c1(C(=O)NCC(CC)NC(C23CCC(OC)C2CC3)=O)c(F)ccc(Cl)c1[N+](=O)[O-] CCCC(C(=O)OC)C(=O)N1CC(CN(C(=O)CC2CC=CCC2)C)C1 N1(C(CCc2cc(C)n(C)n2)=O)CC2(NC(=O)Cc3ccncn3)CCC1CC2 N1(C(CC=CC=C)=O)CCC2(CC2NC(=O)CC2CCCC(O)C2)C1 c1(OC)ccccc1SCC(=O)NCC1CC(NC(=O)CCc2ncc[nH]2)C1 C1(C(=O)NC(C)C(C)n2cccn2)CC2(CC2)CN1C(=O)CC1CCOCC1 N1(C(c2c(C)ccc(F)c2)=O)CCCC2(CCN2S(=O)(=O)C(C)C#N)C1 CC1CN(C(c2cccc(F)c2)C)CCC1NC(c1cc(Cl)c[nH]1)=O C(=O)(C1CC(O)c2ccccc21)NCC(CC)NC(c1cc(C)ccc1NC)=O C1(NC(c2cc(-c3ccccc3)no2)=O)C2CCC1N(C(C1CCCO1)=O)C2 N1(C(CC(C)(CC)NC(CCC=C=C)=O)=O)CC2(CNC(=O)N2C)C1 c1(OC)ccc(C(N2CC3CC2C3)C(=O)NC2COC2)cc1Cl C1(O)(CNC(C2CC=CC2)=O)CCCN(C(c2ccccc2-n2cccn2)=O)C1 S(=O)(=O)(c1ccc(NCc2ncnn2C)c(Br)c1)NCC1CC(C)C1 N1(C(Cc2c(C(N(CC)CC)=O)cccc2)=O)CCC(O)(CC2CC2)CC1 CC(F)(F)C(F)C(=O)NC1CCOCC1C(N1CC(OCCF)C1)=O N1(C(=O)NCCOc2ccccc2F)CCC2(CNC(=O)N2)C1 c1(SC)cc(N2CCOC(C(C)NC(C3Cc4cscc4C3)=O)C2)nc(SC)n1 N1(C(c2c(CC)c[nH]n2)=O)CCC(N(C(=O)COCC(=O)OC)CCO)CC1 C1(CNC(=O)C(F)=C2CCCC2)CN(C(=O)C=CC2CCOCC2)CCC1(F)F c1(C(=O)OC)cc(C(=O)NC2CC(F)(CNC(C3CC=CCC3)=O)C2)c(C)s1 CC1(C)CC(C(=O)NCCCN2CCC(F)(F)CC2)CN(C(c2csnn2)=O)C1 N1(C(CC(C)(O)C2CC2)=O)CCN(C(c2nc(O)[nH]c(=O)n2)=O)C2(CCC2)C1 Cc1c(N)ccc(C(=O)N(C(C)CNC(C2(C(C)C)CCCO2)=O)C)c1Cl C12(CNC(C3(C)CC3)=O)CCCC1CCN2C(c1cc(-c2ccncc2)[nH]n1)=O C(=O)(CC(C)C(F)(F)C(F)(F)F)NC(CCCNC(c1n(CC)c(O)nc1)=O)C C1(C(N2CCC(N(C(c3cscc3OC)=O)CC)C2)=O)COC2CCCCC12 C1(NC(C2CCOC2)=O)CCN(C(=O)Cc2cn3ccsc3n2)CC1O c1(C(N2C(C)CC(NC(C3(O)CC3)=O)C2)=O)cc2cc(Br)cn2cn1 Cn1cc(CNC(c2cn(C3CCCC3CNC(=O)CO)nn2)=O)ccc1=O N1(CC)C2CCC1CN(C(=O)NCc1cc(C)cc(O)c1)C2 c1(C(=O)NCC2CCC(NC(CC3(C)CCC3)=O)CC2)onc2c1CCCC2 N1(C(C(CC=CCC)C)=O)CCC2(C(N3CCC3C)=O)CC2C1 CCCCC(CNC(=O)CC1CCC1)NC(=O)CC1CCC1 CCC(C)C(C(=O)N(CCCNC(=O)C=Cc1ccco1)CC)OC c1(OCC#C)ncccc1C(=O)NCCC(C(C)C)NC(=O)Cc1cnco1 c1(C(c2n(C(C)C)nnn2)NCC2CC23CCC3)ccc(C#N)cn1 C(=O)(C(C)(O)CCC)N1CC(CNC(c2cc(CCCC)oc2C)=O)C1 C(=O)(CCCCCCNC(=O)Cc1csc(C)n1)NCCC(C(C)C)OC N1(C(C=CC=CCC)=O)CCCC(NC(=O)C=CC2CCOCC2)CC1 CCC(O)C(C)C(=O)NCC1(C)CCCN1C(=O)C(C)n1ccnc1 Cc1nc(C(=O)OCC2OC(=O)NC2(C)C)c(=O)[nH]c1C C1(NC(=O)C=CC2CCCO2)CCCC12CN(C(C1(C(F)(F)F)CC(O)C1)=O)C2 c1(OC)cccc(NC(C2(NC(=O)C(=CC3CCCC3)C)CCCCC2)=O)c1 N1(C(C(C)C2CCCO2)=O)CC(C)N(C(=O)CSCc2ccccc2)CC1C C(=O)(CCN(OC)C(=O)c1cc2ccccn2n1)NC(CCC(=C)C)C C1(O)(C(=O)NCC(CCNC(C2CCOCC2C)=O)OC)CCCCCC1 C1(NC(Cc2n(C)cnn2)=O)CC12CCN(C(=O)CC1CCC1(C)C)CC2 c1(C(N2CC(C(N)=O)(CNC(C3OCC(=O)C3)=O)C2)=O)cc(Br)ccc1F c1(OC)ccc(Cl)c(C(=O)NCCOCCCNC(=O)Cc2ccnn2C)n1 C=CC1(C(N2CCC(COC)C2)=O)CCN(C(=O)CC2(O)CCCC2)CC1 N1(C(c2cccc(OCC#C)c2)=O)CCN(C(c2snnc2C)=O)C(C)C1C c1(OC(c2c(Br)cn(CCOC)n2)=O)ccc(C#N)c(Br)c1 N(C1COc2ccc(Br)cc21)C(=O)NCC(CC=C)c1ccccc1 c1(OCC)ccc(NC(c2cc(C#N)cs2)c2nnnn2C2CCC2)c(C)n1 Cc1cc(C(N2CCC(NC(=O)CP(C)(C)=O)C(C)C2)=O)ccc1C(N)=O Cc1ccc(C(N2CC(NC(=O)Cc3cccc(O)c3)C2)=O)cc1NS(C)(=O)=O N1(C(c2cncc(OC)c2)=O)CC(NC(c2cnn(C(F)F)c2)=O)C2CC2C1 C1(NC(CCn2c(C)ncc2)=O)C(C)CN(C(=O)C=Cc2cccs2)CC1C C1(C(=O)N(C)CC2CCCS2)(OC)CCN(C(=O)C=Cc2ccoc2)C1 C1(C(=O)NC2(C)CN(C(c3cc[n+]([O-])cc3)=O)C2)CC2CCC1CC2 C#CC1(C(N2CC(=O)NCC2CC)=O)CCN(C(=O)CC)CC1 C(=O)(C1CCCc2ncccc21)OC(CCCC)CCC C(=O)(C1=C(F)CN(C(=O)C(F)C(C)(C)O)CC1)N1C(COCC)CCC1 CC1(NC(c2cc(Br)co2)=O)CCCN(c2ncnc(Cl)c2CO)C1 c1(CN(C(=O)CCC2CC(NC(C3(N(C)C)CCC3)=O)C2)C)ccncc1 N1(C(C(C)CC2CC2)=O)CC2COCCC2(NC(c2cc(C3CC3)cs2)=O)C1 C1(C(=O)NCC(CNC(c2nccnc2N)=O)OC)CCN(C)C(=O)C1 N1(C(C(CC)C#N)=O)CCCC(CO)(NC(=O)CCc2cc(C)n(C)n2)C1 C1(CC=C)(C(=O)NCC(C)C(C)O)CCN(C(c2cc(OC)cnn2)=O)C1 c1(OCC(=O)OC)ncc(C(N2CCC(NC(=O)Nc3ccccc3)C2)=O)cn1 N1(C(c2ccc(C)nn2)=O)CC2CCCC(NC(=O)C3=CC4CCCC34)C2C1 c1(C(=O)NCC2C(C)CN(C(=O)C(C)(C)CO)CC2)cc(S(N)(=O)=O)c(Cl)o1 CC1(C)CCN(C(=O)CCS(=O)(=O)N2CCOCC2)CC1NC(C1(CF)CC1)=O c1(C(N2CCC(NC(=O)C(=Cc3c[nH]cn3)F)C23CC3)=O)cc2ccccn2n1 CC1(C(c2nnnn2CC2CCOCC2)NCc2nncs2)CC2(C1)CC2(F)F N1(C(C(C(C)(F)F)F)=O)C(C(N2CC3CCOC3C2)=O)CC2CCCC12 C1(NC(C=C(CCC)CCC)=O)CCCCC12CCN(C(C1(C)COC1)=O)C2 N12CC3CC(CC1C3)OC(CCC)CC2=O.C(=O)(C(CC(C)C)OC)NCC Cc1ccnc2sc(C(=O)NC3CC(NC(=O)CS(=O)(=O)C(C)C)C3)c(C)c12 C1(NC(c2ccc(C)s2)=O)CN(C(=O)C=CC2CC2)CC1c1ccnn1C c1(OC)cccc(C(N2CCCC(CO)(NC(C3CC3C(F)F)=O)C2)=O)c1O Cc1nc(O)ccc1C(=O)NC1(CN(C)C(C2OC3CCC2CC3)=O)CC1 C1(NC(C23CN(C(CN(C)C)=O)C(C2)CO3)=O)CCCCCC1(C)C C1(C(N2CC(CNC(c3c(OC)csc3)=O)OCC2)=O)CC(C2CCC2)C1 C12(NC(c3c(Cl)cnc(C)n3)=O)CCCC1N(C(=O)Cn1cc[n+](C)c1)CCC2 c1(C(N(C2CCN(C(=O)CCCC3CCCS3)C2)C)=O)cccc(CO)c1 C(CN=c1cc[nH]cc1C#N)C1C(C)CCCN1C(c1coc2ccccc12)=O c1(C(=O)NC2CC(C)N(C(C3(C#N)CC4CCC3C4)=O)C2)ccc2n[nH]cc2n1 c1(CC(=O)NC(C(=O)N(C)CCC2CC2)C2CCC2)ccccc1 c1(CC)cncc(C(=O)NC2CCCC(N(C)C)C2)n1.C12CCCN(C1)C2=O Cc1cc(C(=O)NC(C)(C)C)nn1C c1(CCC)cc(C(N2CCC(O)(CNC(=O)CC3CC(C)=NO3)C2)=O)sc1C CCC(C)(C)C(=O)NCC(c1ccccc1)CNC(c1ccn(C)c1)=O c1(C(N2CCCCC(NC(=O)CC3CCC4CC34)C2)=O)ccc2cccnc2c1 C1(O)(CC(=O)NCC(CC)NC(=O)CCC2CCCCO2)CCCOC1 n1(CC(=O)NC2(C3N(C(c4nc(CCC)sc4)=O)CCC3)CC2)ncn(C)c1=O N1(C(c2ccc(C(C)C)cc2)=O)CCCCCC(NC(C2CC(O)C2)=O)C1 C1(C(N2CC(C(CC)C)C2)=O)CCN(C(=O)Cc2n[nH]c(C)n2)C1C(C)C CCC(C)(COC)C(=O)N1CCC(N(CCO)C(c2cnc(O)n2C)=O)C1 O(S(=O)(=O)CCCCCF)C1C(P(C)(C)=O)CCCC1 CCCS(=O)(=O)CC(=O)NC1CC2CC(NC(=O)C(F)CC3CCCCC3)C2C1 c1(-n2cc(CCSC)nn2)ccc(Cl)cc1F.C1C(C)(C)C(=O)N1 C(=O)(CN=S(C)(C)=O)N1CCC(C)C1CNC(=O)C(F)(F)C(F)F C1(C2CN(C(C3(CCF)CC3)=O)C2)(NC(=O)C(O)Cc2ccc(Cl)cc2)CC1 C12(C(=O)NCCCCC(C)NC(c3cc(COC)no3)=O)CCC(O)(CC1)CC2 C1(NC(C(CCC)=CCC)=O)CN(C(c2cn[nH]c2)=O)CCC1C(F)(F)F N1(C(c2nc(CC)oc2C)=O)C2CCC(C2)C1CNC(=O)C(c1cccnc1)O N1(C(c2ccc(C)cc2)=O)CCC2(CCCC2NC(=O)C=CCO)C1 C1(C(N2CCC(CNC(Cc3c(CC)cccc3)=O)C2)=O)CCn2nccc2C1 c1(N2CC(C(=O)OC(C)(C)C)(COC)C2)ccc(SC)cc1[N+](=O)[O-] C1(C(=O)NCC2N(C(c3cnc(OC)c(Cl)c3)=O)CC=C2)CC2CC1CC2(F)F N1(C(CSCC=C)=O)CC(C(=O)NCC(C2CCCCC2)O)CC12CCC2 c1(C(=O)NCC#CC(=O)NC2(CO)CC3CCC2C3)ccn2ccccc12 C1(NC(C=CC(=O)OCCCC)=O)CC2CCC(C1)N2C(c1ccc(SC)o1)=O CN1CCN(C(C2CC2c2ccc3c(c2)OC(F)(F)O3)=O)c2ccc(Cl)cc21 C1(C)(CCC(=O)NCC(C)CNC(=O)CCOCC(C)(C)C)CCC(=O)N1 n1(CC)nccc1C(C)NC(=O)CCC1(NC(c2cncnc2)=O)CCCC1 C#CCCC(O)C(=O)N1CC(NC(=O)C(C2CC2)SC)C1 N1(C(C2(CC(=O)NC)CCC2)=O)CC2CCN(C(=O)C3=NOCC3)CC2C1 N1(C(CC(c2c(C)noc2C)C)=O)CCCC(N=c2[nH]c(Cl)ncc2Br)CC1 C12(CNC(C(C)C3CCCC3)=O)CCCC1CN(C(=O)Cn1ccnn1)C2 C1(CNC(COCCC(C)C)=O)CCN(C(c2cnc(S)n2C)=O)CC1(F)F N#Cc1ccc(C(=O)NCc2cc(C(N3CCCOCC3)=O)n(C)n2)s1 C(C(CC(=O)N(OC)C(C)C)OC(C)=O)NC(c1cc(COC)[nH]n1)=O c1(CNC(CC)=O)ccc(CNC(c2ccc(C)cc2C(C)(C)C)=O)cc1F c1(CCCC(=O)NCC(C)(CO)NC(C(CC#C)C)=O)cc(C)ccc1C n1(CC(=O)NC2(CN(C)C(C3CCCC3(C)CO)=O)CC2)ncn(C)c1=O C(C(C)NC(c1cc(Br)nn1C)=O)(C(C)C)NC(C1(C(=O)OCC)CC1)=O c1(C(=O)NC(C)CNC(C2(C(C)(C)C)CC2)=O)ccc(C(F)(F)F)cc1Cl N1(CC(=O)N(C(CCNC(c2n(C(C)C)ncn2)=O)C)C)C(=O)CCCC1=O N1(C(C(C)(F)F)=O)CCCC2(NC(c3cnc(C4CC4)[nH]3)=O)CC2C1 C1(C(=O)NC(COC)(C)CO)CCCN(C(=O)Cn2cncn2)CC1 C(CCCC(CO)NC(c1ncsc1C)=O)NC(c1c(Cl)cn(CCOC)n1)=O C(=O)(C(C)(C)C1=CCSCC1)N(C(CCNC(C(CCC)C)=O)C)C C1(NC(C2(CC(=O)OC)CC2)=O)CC(NC(C2CCN(C)CC2)=O)C12CCC2 C1(CNC(=O)OC(C)(C)C)CCCN1N1CCC(c2cccc(Cl)n2)C1 C(C1CN(C(c2[nH]nnc2CC)=O)CC1C(=O)NCc1ccc(OC)o1)=CC CCCCC(C(=O)NC(C(=O)NC1(CO)CCC1)C1CCC1)C(C)C C1(CNC(C(C)Cn2cccn2)=O)CCN(C(c2ccn(C3CC3)n2)=O)CC1 C12(CCOC)CCN(CC1)C2=O.c1(CNC(=O)Cc2cnoc2)cc(Cl)ccn1 C=C=CC(C)C(=O)N(C(CNC(=O)Cc1csc(=N)[nH]1)C1CC1)C c1(C(=O)NCC2CC(OC)CN2C(C2CNC(=O)N2)=O)coc2c(F)cccc12 C1(C(N2CC(OCCNC(c3n(CC#C)ccc3)=O)C2)=O)COCCC1(F)F N1(C(c2cc(C)cc(O)n2)=O)CCC2CCCC12CNC(C1(C)COC1)=O n1(CC(=O)NCC23CC(CN2C(c2ccc(CO)o2)=O)C3)nnc2ccccc12 C1(CC(N2CC3CC(Nc4ncnc(Cl)c4CO)C3C2)=O)CCCC(F)(F)C1 CC(C)C(C(C)NC(=O)COC1CCC1)NC(c1nc(Cl)cs1)=O c1(NC(c2c(NC(c3c(C)coc3)=O)cccn2)=O)ccc(C)c(Cl)c1 c1(CCC)ccccc1S(=O)(=O)C(=O)NCCc1ncnn1SC(C)(C)C c1(C(=O)NC2CCN(C(Cn3c(C)nnn3)=O)CC2C)cc2n(c1)CCCC2 C=CCC(C)(C)CC(=O)N(C1CN(C(c2ccc(C#N)c(O)c2)=O)CCC1C)C C1(CNC(Cn2c(C)ccc2C)=O)CCC2(CCC2)C1NC(C1(N(C)C)CCC1)=O c1(C(N2CCC(C(F)(F)F)C(CO)C2)C(=O)NCCOCC)ccc(C)c(Br)c1 C1(C(=O)NC2C(CNC(Cc3cn(C)nc3Cl)=O)CC2)CCc2nn[nH]c2C1 Cc1cc(C(N2CC(N3CCCS3(=O)=O)C2)=O)cc(C)c1 C(C(O)CCNC(=O)CC1(CNC(c2nscc2C)=O)CC1)OC N1(C(C(COCC)C)=O)CCOC(C)C1C(=O)NCC(C1CCCCC1)C CC1CCN(C(c2ccc(C(N)=O)s2)=O)CC1NC(=O)CCc1cnoc1 CCC(CC)(C(=O)NCC1CCC(C(=O)NCc2noc(C)n2)C1)OC c1(CC(=O)NCC=CCNC(C2C(c3cn(C)nc3)OCC2)=O)ccc(O)cc1 N1(C(CC(C)F)=O)CCN(C(C2NC(=O)OC2(C)C)=O)C(c2ccc(F)cc2)C1 C(=O)(CC(O)CC(C)C)NC1C(C(=O)NCCC(=O)OCC)CCCC1 CCCS(=O)(=O)C(C)C(=O)NCCCCC(C)NC(=O)C(C)(C)C1CC1 N1(C(COc2c(C)nc(-c3ccccn3)nc2O)=O)CCC2OC(=O)OC2C1 CC1=C(C(=O)NC2CCC23CN(C(=O)C(F)C(C)C)C3)CCCC1 C(=O)(C(C(=O)N(CCC(C)NC(=O)CN1CCOCC1)C)C1CC1)OCC C1(NC(C(C=C)O)=O)CN(C(c2cc(N)cc(F)c2)=O)CC12CCC2 C=CC(C)CC(=O)N1CC(OCCC(=O)Nc2nc(OC)c(C)s2)C1 C1(C(=O)NC(CNC(c2nn(CC)c(C)c2)=O)C2CCC2)CCc2nnnn2C1 c1(OC)cccc(F)c1CC(N1CC(CNC(c2nccn2C)=O)CC1C)=O C1(CNC(COCCSC)=O)CCN(C(C2(C)COCCO2)=O)C1(C)C C1(NC(C2OCC(C)C2)=O)CC2(CCCN(C(=O)CCC3CCCO3)C2)C1 C1(CC=CCCC)(C(=O)N(C2CCN(C(=O)OC(C)(C)C)C2)C)CCSCC1 c1(OCC(C)C)ncccc1C(=O)NC1CC(CNC(C2CCCC(C)C2)=O)C1 C(=O)(C(C)(C)C(C)(F)F)N1CC(C=C)C(NC(c2nc(O)c(C)s2)=O)C1 C1(O)(CC(=O)N(C2CCN(C(=O)COCP(C)(C)=O)C2)CC)CCOC1 CC(=O)CCCCC(=O)N1CCCC1OCc1c(C)cccc1Cl n1(CC)cnc(CCNC(=O)Cn2cc(CCNC(c3coc(C)c3)=O)nn2)c1 c1(C(N(C(C(N)=O)C2CC2)C)=O)c[nH]nc1CNC(=O)C=CC1CCOC1 C1(CCNC(CC#N)=O)CCCCN1C(c1cnc(-c2cnccn2)s1)=O Cc1c(C(N2CCC(O)C(C(=O)NC(CO)C(F)(F)F)C2)=O)cccc1Br CCCCCCCC(=O)NC1CCCCC1NC(C1(F)CC=CCC1)=O C1(C(=O)Nc2cncc(OC)c2)CCC(C)N(Cc2nnc(-c3cccs3)o2)C1 C1(C(N2CCC(NC(c3c(Cl)cc(C)s3)=O)C2C)=O)CNC(=O)CC1C c1(C(=O)NC2C(CNC(c3c(C)ccc(OC)c3)=O)C2)cn2nc(C)sc2n1 N1(C(=O)OC(C)(C)C)C2COCC1CC(NC1(C)CC1)C2.C123CC(C1)(C2)C(=O)N3 c1(N(C(=O)Cn2cc(CC3CCCC3=O)nn2)C)nccnc1Cl Cc1noc(C)c1C(C)C(=O)NCC1CCCN1C(c1cnn(C(C)(C)C)c1)=O C(=O)(C(C)CC(=O)NC1CCCC1C(N1CCN(CC2CC2)CC1)=O)OC c1(C(N2CCCC2c2ccccc2Br)C(=O)NCCCC)ccc(C(F)F)cn1 C(=O)(C(C)(C)CC1CC1)NCC(COC)NC(=O)CC(C)C1CCCO1 N1(C(CC(CNC(CCCOCCC)=O)C)=O)Cc2n[nH]cc2C1CO C(=O)(C(C(C)(C)C)N1C(=O)CCC1=O)NC1C(NC(c2scc(COC)c2)=O)C1 c1(C(N(C(CCNC(c2n(CCC)ncc2)=O)C)C)=O)ccn2nccc2n1 C=C(Cl)CC(C(=O)NCCN(CCCF)C)NC(c1cccc(O)c1F)=O C1(=CC(=O)NC2CC(CCC(=O)NCC(O)CN3CCC3)C2)CCOCC1 CC(C)(CCCNC(C1(F)CC=CCC1)=O)NC(=O)CC1CCOCC1 c1(CC)nnc(O)c(C(=O)N(CCC(C(C)C)NC(c2cc[nH]n2)=O)C)c1CC c1(NC(c2nccn2C(C)(C)C)C)ccc([N+](=O)[O-])cn1 C1(OC)CCC2(C(=O)NCC3CCC3NC(=O)Cc3ccoc3C)CC12 c1(C(=O)NCC2CN(C(=O)CCc3cnc[nH]3)C2)ccc(Cl)c2ccccc12 C1(c2nc(COCC)nn2-c2cc(F)ccc2C)CCc2ccnn2C1 CC(C)CC(O)C(=O)NCCCN1CCC(NC(=O)Cc2cnns2)C1 c1(C(=O)NCC(C)CN(C)C(c2n[nH]cc2Cl)=O)ccc(CO)nc1 C(=O)(C(CC)CC(C)C)NCC1(C(=O)NC(C(=O)OCC)CC)CCCC1 c1(C(C(=O)NCC(=C)C)N(CC(c2ccncc2)C)C)csc(C(C)(F)F)n1 O=C(C#CC1CCCCO1)N1CCC(CNC(C2(O)COC2)=O)C12CC2 c1(C(N2CC(NC(c3cc(CC)c(C)s3)=O)C(F)CC2)=O)nc2cccnc2s1 C1(OC)CC(CO)N(C(=O)CCN(CCO)C(c2cc(CO)oc2C)=O)C1 c1(CC)cc2c(NC3CC4CN(C(=O)CCCC5CCC5)CC34)ncnc2s1 N1(C(c2ccc(OC)cc2)=O)CCC(CC(=O)NCCC(C)(C)C)C1(C)C C1(NC(C(CC)(CC)CO)=O)C(C)(C)CN(C(=O)CCNC(=O)CO)CC1(C)C C(C(C)(C)CNC(=O)CC1C=CCC1)N(C)C(C1(CN2CCCC2)CC1)=O N1(C(C2CC(C)OC2)=O)CCCC2(CCN(C(c3cnn4ccn(C)c34)=O)C2)C1 c1(OC)ccc(C(c2nnnn2C)Nc2ccc(-n3nc(C)cc3C)cc2)cc1Br N1(C(CNC(c2c(C)noc2N)=O)=O)CC2CC(O)CC2C1 c1(NC2(c3n(C(C)C)nnn3)CCC(C)(C)CC2C)ccc2c(c1)C(=O)NCC2 n1(CC)cc(C2CN(C(=O)NC(=O)N(C)C)CCO2)c(C(F)F)n1 C1(C(=O)NC23CN(C(CCCC#CC)=O)C(C2)C3)CC12C(=O)Nc1ccccc12 C(=O)(C1=CCC(C)CC1)NCC(CNC(c1ccc(C)cc1Br)=O)CO c1(CSCC(C)(C)C)cccc(C(N2CCC(NC(N3CCCCC3)=O)C2)=O)c1 C#CCC(C)(CC)C(=O)NCc1cncc(C(=O)NC(C)C=C)c1 c1(C(C)C)cccc(CC(=O)NCCCNC(C2(C3CCCO3)CCCC2)=O)c1 CCCCC(CC)CC(=O)NCCC(C)(C)NC(=O)CSc1nccn1C(C)C CC1CCC(C(=O)NCC2C3CCCOC23)N(C(c2cnc(=N)[nH]c2)=O)C1 N1(C(C(C(CC)C)O)=O)CCC2(CCN(C(=O)CNC(c3ccccc3F)=O)C2)C1 C1(C(=O)NCc2cc(C)c(C)o2)CCN(C(C2(C)CC(=O)N(C)C2)=O)C(C)(C)C1 c1(CN(C(C2C(NC(c3cnccn3)=O)C2)=O)C2CC2)ncoc1C1CCOCC1 C(=O)(CCC(C)(C)NC(C1(C#N)CCCC1)=O)NCC(CCN(C)C)O N1(C(c2c(CCC)n[nH]c2)=O)CCC(C(=O)Nc2cnn(C)c2C(N)=O)C(C)C1 N1(C(c2cn(CC)nc2C)=O)CC(CNC(=O)CC(C)F)C(F)(CO)C1 C1(C(C)(C)C)CN(C(=O)CCSC(F)F)C1.C(C(F)(F)F)NC(=O)C O(N(C)C(=O)CNC(C1(C)CN(C(=O)Cc2nc(=N)[nH][nH]2)C1)=O)CC C(=O)(C(C(C)C)OCCOCCC1(CNC(=O)CSC)CCCC1)NCC N1(C(CC(C)OC)=O)CCC(C)(CNC(C2(c3cccs3)CCCCC2)=O)C1 Cc1ccc(O)c(CNC(=O)Nc2ccc(OC3CCOC3)cc2)c1 C(=O)(C(F)CC(C)C)NC(C1CCOC1)CNC(c1c(CC)onc1C)=O CCCCC(C)C(=O)N(CC(O)CN(C)C(c1ccc(OC(F)(F)Cl)cc1)=O)C CC1CCCN(C(c2sccc2CO)=O)C1CNC(C1CC12CC(O)C2)=O C1(CC)C(NC(=O)C(C)c2cncs2)CCN1C(c1cnn(CCOC)c1C)=O C1(NC(C(CC)=CCCC)=O)CN(C(C2CC2COC)=O)CCC1O N1(C(C2N(C(C)=O)CCC2)=O)CC(NC(=O)CCC(N)=O)Cc2ccccc21 CCCC(C)(CCC)C(=O)NC(CNC(c1cc(N)c(F)cc1C)=O)CC(C)C c1(C(N(C(C)CNC(=O)C(C)(C)N(C)C)C)=O)ccc(F)cn1 S(=O)(=O)(c1cccc2ccccc12)N1CC(NC(c2cc(OC)ncc2)=O)(CO)C1 CCCC(C)CCCC(=O)N1CCCOC(CNC(c2cc(F)cc(Cl)c2N)=O)C1 C1(C(=O)NCC(CCSC)NC(C2C3(CC3)C23CC3)=O)CCCC(C)(C)CC1 Cc1ccnc(NC(N2CCSCC2C2CC2)=O)n1 C=CC1CN(C(C2CCCC2O)=O)CC1NC(=O)CC1CC=CC1 C1(C(=O)NCCCN(C(C23CC(C4CCOC4)(C2)C3)=O)CC)C2CCCC12 N1(C(C=CC)=O)CCOC(C(C)CNC(=O)CCCn2ccnc2)C1 c1(C(=O)NC2C(NC(CC3(C(=O)OC)CC3)=O)CCCC2)cccc(O)c1F c1(NC(CCN(C(=O)C(C)C2CCCO2)CC)=O)cc2ccccn2n1 N1(C(CC)C)CCC(NC(=NCc2cccc(OC)c2)NCC)CC1.CC(F)(F)F N1(C(Cc2nc(C)oc2)=O)CC(NC(=O)Cc2nnc(C)o2)C2CC12 C=CCC(CC(=O)N(CCCCOC)CC)NC(C1CC1C(F)(F)F)=O C1(NC(CN(C)CC)=O)CCN(C(=O)C(C(C)C)NC(=O)OC(C)(C)C)CC1O Cc1ccc(CC(=O)NC(C2CCN(C(C3CC3c3cnn(C)c3)=O)C2)C)cn1 C(CS(=O)C(F)(F)F)NC(C(N1CCN(CC)CC1)c1ccc(Cl)cc1)=O c1(C(=O)NCC=CCNC(c2n(C)ccc2)=O)cc2c(nc1O)CC(C)(C)CC2 C1(C(=O)NC(CC(=O)NCc2onc(C(C)C)n2)(C)C)CC(=O)NC(C)C1 N1(C(C(C)C2(O)CCC2)=O)CCCC(C2(NC(=O)CCn3cncn3)CC2)C1 C1(C(=O)NCC(C2CCC2)OCC)(NC(c2[nH]ccc2CC)=O)CCCC1C Cc1ccn2c(C(N3CCSC4(CCC4CNC(=O)C=CCO)C3)=O)cnc2c1 N1(C(CC(C)NC(=O)C2=C(Cl)CCOC2)=O)CC(NS(C)(=O)=O)C(N=[N+]=[N-])C1 N1(C(C(CNC(C2(CC)CCC2)=O)CC2CC2)=O)CCC(C)(C#N)C1 C1(CC=C)(NC(=O)C=C(C)C)CCN(C(=O)C=CC2CCOCC2)CC1 CC1CN(C(=O)CCn2ccnc2)CC(C)N(C(c2ccc(F)c(O)c2F)=O)C1 N1(C(CNC(=O)OCC)=O)CC(O)CC1C(=O)NC(c1cn(C)nn1)(C)C c1(C(=O)NCCCNC(C2CCC(C)O2)=O)ccc(C(=O)OC(C)(C)C)cc1 C1(C(N(CCC)CCNC(=O)C(O)CC(C)C)=O)CC2C=CC1CC2 c1(C(=O)NCC2OCCN(C(CCC3CC(C)C3)=O)C2)ccc(N)c(Cl)c1 c1(OCC)ccc(-c2nc(-c3ccc(-c4cccs4)o3)n(CC3CCC3)n2)cc1 Cc1cccc(CC(=O)NCC(CO)NC(C2(C)C=CCCC2)=O)c1 c1(C(=O)NC(=O)CC2(N3CCCC3)CC2)ncc(Cl)nc1Cl.N12CCCC3(CC13)C2 c1(NC(C(=O)N(CC)Cc2ccccc2)=O)cc(OC(C)C)cc(O)c1 C=CCCC(F)(F)C(=O)NC1CC(F)(CNC(c2ccnc(C3CC3)c2)=O)C1 C1(C(COC)NC(=O)CCCCn2cc(-c3cn[nH]c3)nn2)CCC(F)(F)CC1 C1(NC(CCCOCCC)=O)CCCCN(C(c2cnc(C(C)C)s2)=O)CC1 C=CCC(CC=C)C(=O)NCC1(F)CCN(C(C2CC2C(C)C)=O)C1 c1(C(=O)NCC2(CNC(=O)CCC3CC4CCC3C4)CC2)cnc(O)c(F)c1 CCCCC(C)C(=O)N(C)CCOCCNC(=O)C(CC)c1ccccc1 O=S(=O)(N1CCCCC1)N1CCCC(n2ccnn2)C1 CC(C)(C)CC(=O)NC1CC(NC(=O)C(C)(C)Cc2ccc(O)cc2)C1 N#Cc1cc(C(=O)Nc2cccc(-c3ccc(CO)cc3)n2)ccc1O C(=O)(C(C)(C)CCCF)NCC1C(C)CCN(C(c2nccnc2N)=O)C1 C1(C(=O)NC(C2CN(C(c3cc(C)nn3CCO)=O)C2)C)CCCC(C)CC1 C1(C(=O)NCC(c2ccccc2)CNC(CCCCC)=O)OCCN(C)C1=O C1(CNC(C(=O)NCC)=O)CCC(F)(CNC(=O)CC(C)COCC)CC1 N1(CCCNC(C(C2CCCOC2)N(CCOC)C2CC2)=O)CCN(C)CC1 c1(OC)ccc(N)c(C(=O)NCC2(O)CN(C(C3(CO)CCOC3)=O)C2)c1 Cc1cc(C(=O)NC(C2CN(C(=O)C(C)(C)SCCNS(C)(=O)=O)C2)C)n(C)n1 C#Cc1cccc(C(N2CC3CCN(C(c4cc(Cl)no4)=O)C3C2)=O)c1C c1(C(N(CCCNC(C(C)CC)=O)CC)=O)cc(OC)c(OC)c(OC)c1N c1(C(=O)NCC=CCNC(C2(c3ccc(Cl)nc3)CC2)=O)ccc2occc2c1 C#Cc1cnc(C(N2CC(N3CCC(O)C3)C2)=O)c(C)c1.C12CCC(C1)NC2=O CC(C)CC(O)C(=O)N1CCC(NC(=O)C)C1C.C(CC(C)c1cn[nH]c1)CC=O c1(CC)ncc(C(=O)NCC2CCN2C(c2cc(N(C)C)ccn2)=O)cn1 C(C(C)(C)C(=O)N1CC(CF)C1)N(C)C.C1(=O)C(C2CC2)N1C c1(SC)c(-n2cc(C(C3CCCN3)(C)N)nn2)cnn1C N1(C(C23N(C(CCCOCCC)=O)CC(C2)C3)=O)Cc2ccncc2C1 C1(OC)CN=C(N2CCN(C3C4CCCC34)CC2C)N1 C1(C(N2CC(NC(C(CC)OC)=O)C(O)CC2)=O)CC2(CCOCC2)C1 c1(C(N2CC3C(CNC(c4c(CC)cccc4)=O)C3C2)=O)cccc(Cl)c1N c1(N2CCC(NC(C(F)(F)C3(CC)CC3)=O)C(F)C2)ncnc2c(Br)cccc12 c1(C(N2CCC(C)(NC(C3CCC(COC)C3)=O)CC2)=O)cc(S(N)(=O)=O)c[nH]1 N1(C(C23CC(NC(C4C5CCCCC45)=O)(C2)C3)=O)CCc2c(ccnc2C)C1 C=C(C)CC(C(=O)NCC1CCCC12CC2)NC(=O)CCc1cnoc1 N1(C(=O)OC)CCC(OCCOCCCCNC(=O)CC2CC2C)C1 c1(CNC(=O)COC(F)F)ncoc1CCNC(c1csc(Br)n1)=O C=CCC(CC(C)C)C(=O)N1CCC(CF)(NC(=O)C(CO)NC(=O)C(C)C)C1 c1(C(=O)NCC(C)NC(=O)Cc2cnc[nH]2)cnc(N(C)C)cn1 N1(C(c2ccn(CCOC)n2)=O)CC(NCc2cc(Br)c[nH]2)CC(F)C1 C1(C(C)NC(=O)C=CCN2CCOCC2)CCN(c2cc(C3CC3)ncn2)CC1 C1(C)(CC)C=C(C(=O)NCc2csc(C(=O)Nc3ccc(OCF)cc3)c2)C1 C(C)(CO)(C(=O)NC(C)CSC)NC(CCOCCCOC)=O C1(c2cn(C(C(=O)NCCCCC)C)nn2)CCC(C(=O)O)CC1 C1(C(=O)NC2CCC(NC(CC(=O)NCC)=O)C2)CC(=O)NC2CCCCC12 c1(OC)nc(C)ncc1C(N1CC(NC(=O)CN2CC(=O)NC2=O)CC1C)=O CCCCCC(CC)C(=O)N(C)CCN1CCN(C(=O)CCCCOC)CC1 c1(C(C2CCCO2)N(CC(C)(C)C)C(COCCOC(C)=O)=O)cccs1 CC1CN(C)CCC1NC(=O)C=CCN(C)C(C1CCCSC1C)=O C(=O)(CCCCCCCCCO)NC1C(C)N(C(=O)CC(C)(C)O)CCC1 C1(NC(CC(CC)C2CC2)=O)CCS(=O)(=O)C12CN(C(=O)CS(=O)CC)C2 C1(F)(C(=O)NCCOCCCN(C)C(C2(C)CCCS2)=O)CCCN(C)C1 c1(CO)ccc(CNC(c2cc(Cl)sc2Cl)c2nnnn2CC2CCOC2)cc1 C=C1CC2(C1)CC(C(=O)N(C(C)CNC(=O)C(c1ccccc1F)CC)C)C2 CC1CN2CCN1C(C(N1CC3(CC(NC(C4CCN(C)C(=O)C4)=O)C3)C1)=O)C2 c1(CNC(C(C)SC)=O)cnn2c1CN(C(=O)CCc1cscn1)CC2 N1(C(c2n(CC)ncc2)=O)CC(C2CN(C(=O)CC3CC(O)C3(C)C)C2)C1 CC1CCN(C(C2N(C(=O)CC(F)(F)F)CCCC2(C)C)=O)CC1(C)C Cc1ccc(F)cc1C(=O)NCC1(F)CC(NC(=O)CC2C=NN(C)C2=O)C1 C=C1CCC(C(N2CCOC(CNC(c3ccncc3Br)=O)C2)=O)CC1 CC1CC(C)(C(N2CCC(F)(CNC(c3ccoc3Br)=O)CC2)=O)CCO1 C1(C(N(CC=C)CC=C)=O)CCCCN1Cc1ccc(OCC)cc1 N1(C(CC2(OC)CC2)=O)CCOC(CNC(=O)CC2(C)OCCO2)C1 C1(NC(c2cc(C)c(C)o2)=O)CC(F)CN(C(=O)C(C(C)O)N(C)C)C1 Cc1cn2ccc(C(N3CCCC3(C)CNC(=O)CC3CC4CC4C3)=O)cc2n1 N1(C(CSC)=O)CC2C(CC(=O)NCc3nnc(C4CC4)o3)C2C1 Cc1sc(Cl)nc1C(=O)NCC(C)(C)NC(C1(C(=O)Nc2ccccc2)CC1)=O O=C(N=c1cnc(Cl)c[nH]1)C1CC1C(N1CCOC2CC12)=O CC(C)(C)C1=NOC(C)(C(N2CC3CCC3(CNC(C3CC(O)C3)=O)C2)=O)C1 C1(CCC)CN(C(C2C3C2CCOC3)C(=O)NCCCF)CC1C(=O)OC C1(CNC(C(c2ccc(C)cc2)C)=O)CN(C(c2occc2F)=O)CC12CC2 Cn1c(CNC2CC2c2ccc(Br)o2)nc2ccccc12 n1(CC(=C)C)nnnc1C(c1ccnn1CC)NC(c1ccc(Cl)s1)CC c1(C(=O)NC2(CF)CCN(C(=O)CCc3cnco3)C2)ccc2c(c1)COC2 C1(NC(=O)C(F)C2CCCC2)CCC2(CCN(C(c3ccon3)=O)CC2)C1 CC(C)(CO)CCCNC(C12CC(CO1)N(C(c1cc(F)cnc1O)=O)C2)=O c1(N(C2CCCC2)CCCNC(=O)Cc2cnsc2)ncnc2cc(C3CC3)nn12 Cc1c(C(=O)NCC(O)CCNC(c2coc(C(F)F)n2)=O)cccc1[N+](=O)[O-] Cc1ccc(CNC(=O)C(n2cc(CN3CCNC3=O)nn2)C)c(Cl)n1 C1(NC(CCC2CC(C)C2)=O)COC2CN(C(c3ccc(Cl)c(N)c3)=O)CC12 CCC(CC(=O)NC12CCC(CC1)N(C(c1sc(CO)nc1C)=O)C2)C(F)F CC(C)CC(CNC(c1cc(CF)on1)=O)NC(=O)C(N1CCSCC1)C Cc1nc(NC2CCCC2C(N2C(C)C2C)=O)ncc1Br CC(C)CCCOCC(N1CCCC1c1cn(C2C=CCCC2)nn1)=O C1(CNC(C(C)CF)=O)CC2CCC(C1)N2C(=O)C(C)(C)c1ccn(C)n1 Cc1cccc(-c2cn(C)nn2)c1.C1(=O)CC(C)(O)C2C(C2)CN1Cc1ncon1 C1(NC(C(C)SCCCC)=O)CC(F)CN(C(=O)CCC(=O)N(CCO)CC)C1 N1(C(CC(=O)NCC)=O)CC(OC)CC(NC(=O)C(O)C(C)(C)C)C1 CCC(CC(=O)NCC1CC(F)(CNC(c2cccn3cncc23)=O)C1)C(F)F C(=O)(C1CCc2ccccc21)N(CCCNC(=O)CC(C)P(C)(C)=O)CC C#Cc1ccc(CC(N2CCCC(C)(NC(=O)Cn3cncn3)C2)=O)cc1 Cn1nccc1C=CC(N1CCCC1CCCNC(C1C=CCC1)=O)=O N#Cc1cc(Cl)c(C(=O)NC2(C3CN(C(=O)C(O)Cn4cncn4)C3)CC2)s1 CCCC(F)(F)C(=O)NC(C)C(=O)NC(c1cn(CC)nn1)C c1(C(N2CC(NC(c3c(OC)cc(C)cc3)=O)C(C)C2)=O)cc(C)c(Cl)c(N)c1 c1(C(C(=O)NC(C)CN(C(=O)CSC(F)F)C)C)c(F)cccc1F C1(CCC(=O)NCC(N(OC)C)=O)CCCCN(C(=O)COCC2CCOC2)C1 CN1CCCC1(C)C1CCN(C(=O)C(=O)NCCC2CN(c3ccccn3)C2)C1 C1(C(N2CCC(CC(=O)NC(C#C)C(C)SC)C2)=O)(NC)CCCC1 CN1CCN(C(=O)C=C2CCCCCC2(F)F)CC1CNC(c1cnc(Cl)s1)=O C(C)(C)(CC(=O)N1CCOCC1CNC(c1ccn(C2CC2)c1C)=O)OC N1(C(Cc2n[nH]c(=N)s2)=O)CCC2COC(CO)C2C1.N12CC(CF)OC(C1)C2 CN1CCC(C(=O)N(C(CNC(c2csc3cncn23)=O)C2CC2)C)CC1=O c1(OC)ccc(F)c(-n2nc(C(O)CC)nc2C(C(C)C)OC(C)(C)C)c1 c1(N2CCC(N(C(c3c(C)nc(O)[nH]3)=O)C)CC2)nc2cc(Br)ccc2o1 C#CCC(C)(C)C(=O)NCc1ccsc1C(=O)NC1CC(C)(C)OC1=O c1(C(N2CCC(CCNC(C=CC(CC)=CC)=O)C2)=O)ccc[n+]([O-])c1 N1(C(c2c(N)non2)=O)CC(CNC(=O)CC(F)(F)F)C(O)C1 C1(C(N2CCCC(C)(NC(c3ccc(C)c(F)c3)=O)C2)=O)CC(C2CCCC2)C1 c1(C(N2CC(CCNC(C3CCCC3O)=O)(OC)C2)=O)cccc(SCC#N)c1 C1(CC(=O)NC2CC(C(C(=O)NC(C3CCCC3)(C)C)F)C2)CCCC2CC12 c1(CN2CCC(NC(c3sccc3F)=O)C(F)C2)cnc2ccccc2c1 N1(Cc2c(F)ccc(C)c2)CC2CCC1CN(C(c1coc(Cl)n1)=O)C2 CC(CC(=O)NCCn1cnc(CCO)c1)C(C)(C)NC(c1cncnc1)=O C1(C#N)(C(=O)NCC(c2ccccc2)NC(C(N2CCSCC2)C)=O)CC2CC2C1 C1(C(N2CC3(C(C)NC(=O)O3)C2)=O)CCC(C)(C)N(C(=O)CN(C)C(N)=O)C1 CON=Cc1ccc(C(=O)NCC(C)(C(C)C)NC(=O)COCCCF)cc1 N1(C(Cc2cn(CC)nn2)=O)CCCC(N(C(=O)CC2CC=CC2)C)CC1 N1(C(=O)OCC)CSCC1C(=O)NCCN(C(C1CCCO1)=O)C1CC1 C1(C)(C(N(CC(C)C)CC(=O)NC2CCSC2C)=O)CCCCC1 C1(NC(c2cc(C)nnc2O)=O)CN(C(=O)C(C)CF)CC12CCC2 C(C(C)(C(=O)N1CCOC(CNC(=O)CCN2CCOCC2)C1)OC)OC N1(C(c2cc(CNC(c3c(CC)cns3)=O)ncc2)=O)CCc2nn(C)cc2C1 C1(C(N(C)CC2(O)CN(C(Cc3c(C)noc3)=O)C2)=O)CCC(C)(C)C1 c1(C(=O)NCC2C(NC(C(CC)(C)O)=O)C2)c[nH]c2cc(Br)ccc12 c1(C(N2C(C)CN(C(C(C)C)=O)C(C)C2)=O)cccc(N=S2(=O)CCCC2)c1 c1(CC)nccn1C(C)CC(=O)N(CCC(C)NC(C1(C(F)F)CC1)=O)C c1(C(N(CCOCCNC(CC2CC(=C)C2)=O)C)=O)nc(C)c(C)s1 Cn1nccc1C=CC(N1CCCC1C(N1CCC(CCF)CC1)=O)=O.CC=O C1(CC(=O)NCCOCCN(C2(n3cccn3)CC2)C)CCCOC1.C1(O)CCCC1 C12(NC(CC3(NC(C)=O)CC3)=O)COC(C1)C(NC(=O)CSC1CCOC1=O)C2 Cc1cc(C(N2CC3C(N(C)C(c4cc(CO)[nH]n4)=O)C3C2)=O)cc(C)n1 C1(C(C(=O)N(C)C)N(C)Cc2cc(C)c(C)s2)Cc2ccccc2C1 c1(CN(CCC(N2CC(Cc3c(C)ccs3)C2)=O)C)ccc(F)c(F)c1 C1(CNC(CCN(C)CC)=O)CN(C(=O)C(n2ccnc2C)C)CC1(C)C CCC(C)CC(=O)NC1(CC(N2CCOC(CC(C)C)C2)=O)CCCCC1 Cc1sc2ncnc(C(N3CCCCC3c3ccnn3C)=O)c2c1C C1(NC(c2cc(C3CC3)no2)=O)CN(C(c2cc(Cl)no2)=O)C2CC12 N1(CC2CCCC(C)C2)C(=O)CCN(Cc2ccc(-c3cccc(F)c3Cl)o2)C1=O C1(CC=C)(NC(C2CC2CCC)=O)CCN(C(c2c[nH]ccc2=N)=O)C1 c1(C(=O)NC2CC(NC(C(c3ccc(Br)cc3)C)=O)C2)cnc(O)n1C Cc1c(-n2ccnc2CC(=O)Nc2cccc(F)c2)cccc1Cl c1(OCC)cc(CN2CCOC(CC(=O)NCc3ccsc3)C2)c(Br)cn1.CO C1(C(N(CC(CC)(C)OC)C)=O)CCC(C)(C)N(C(=O)C(O)C(C)(C)C)C1 c1(N2CCCCC(SCC)C2)ccc(S(=O)(=O)NC2CCS(=O)CC2)cn1 C(=O)(C(CNC(=O)CNc1ccccn1)CCC)N1CCC(CCCC)C1 N1(C(CSCc2nc(C)[nH]n2)=O)CCSCC1CCNC(=O)CC(F)F CCCCC(CNC(=O)CP(C)(C)=O)NC(C1CCN(c2nc(C)cs2)CC1)=O c1(OC)nscc1C(=O)N(C1CC(NC(=O)COc2ccn(C)n2)C1)C c1(N(c2ncc(Cl)cn2)C)ccc(Br)cc1[N+](=O)[O-] Cc1nc(O)ccc1C(N1CCC(C(C)NC(=O)C(c2cncn2C)O)C1)=O N1(C(=O)OC(C)(C)C)CC2CCC2(NC(N2CCOCC23CC3)=O)C1 CC1(C)CC=C(C(=O)NC(c2ccccc2)C(=O)NC2CCC3CC23)CC1 c1(C(N2CCN(C(C(CC=C)NC(C)=O)=O)CC2CC)=O)cc2n(c1)CCSC2 C1(COC)CCN(C(=O)COCCNC(=O)Cn2nnnc2C)CC1 Cn1ncc(C(=O)NC2CC(NC(C3CCC3(C)C)=O)C2)c1-n1cccc1 N1(C(c2n(CC)ccn2)=O)CCCC(C)C1CCNC(c1cscn1)=O Cc1ccc(C(N2CCC(C)(C)C2C(=O)NCC(O)C2CCC2)=O)c(C)n1 c1(OC)ncccc1CC(=O)NC1CCC(CNC(c2cccc(F)c2)=O)C1 CCC(CC)C(C)C(=O)NC1(CN2CCN(C(=O)C(C)=C(C)C)CC2)CC1 c1(OC(C(N2CC(CC=C)(NC(=O)Cc3ccccn3)C2)=O)C)ccc(C)cc1 C(=O)(CCCC(C)(C)C#N)N1C(CC)C(NC(c2cccc(Cl)c2OC)=O)CC1 C1(C2CC2)(NC(CCC=C(C)C)=O)CCN(C(C2CCCC(C)(C)C2)=O)C1 CN1CCOC(C(N2C(C(=O)NCCC(C)(C)C)CC3CC23)=O)C1 N1(C(CNC(C)=O)=O)CC2CC(CNC(c3c(C)cc(O)nc3C)=O)CC1C2 C1(=O)CCCC2(CC2)N1.C1(C(NOCC(=O)OC)=O)CC=CCC1 C(=O)(C(F)CC(C)(C)C)NC1CC2(C(NC(c3cc(C)nc(O)n3)=O)C2)C1 C(=O)(CC1=CCCC1)NCCOCCC(=O)N(C(C)C)CCc1ccccc1 C1(C)(c2n(-c3c(C)cc(F)cc3)nc(CCO)n2)CC(C(C)C)=NO1 N1(C(C=NOC)=O)CCC2CC2(NC(c2ccc(-n3cc(Br)cn3)cc2)=O)CC1 c1(CN2CCC(C(N(CCn3c(C)ncc3)C)=O)C2)ncccc1Cl C(=O)(C(COC)CC)NCC(C)N(C(C1CC(CC)(CC)C1)=O)C c1(C(N(CCn2cc(C3CCCCO3)nn2)CC)C)ccc(OC)cc1 N1(C(C2C(C)OCC2)=O)CCC(CNC(c2cccc(C3CCC3)c2)=O)C1(C)C C1(C(N(C)CC2CCN(C(Cc3c(C)nc[nH]3)=O)C2)=O)CCc2ncccc2C1 C1(OC)CN2CCCC2(C(=O)NCCC2CCCN(C(=O)CC3(CO)CC3)C2)C1 c1(OC)cc(C(=O)O)ccc1C(=O)OC.c12ccc(cn1)CN1CCC(C1)CN2 N1(C(C2CC(C)C2)=O)CCC2C(NC(C3OCCCO3)=O)C12 N1(C(C(C)N2CCCC2)=O)CCC2CN(C(C3CC3C3CCC3)=O)CC2CC1 N1(C(c2ccc(C)s2)=O)CCC(CF)(NC(C2CN(CC(C)C)C2)=O)C1 C1(CN2CCC(C=C)C2)CCCC(C)(C)CC1 C1(COCCOCCN(C(c2cc(CC(=O)NC)on2)=O)CC)COCCN1C Cc1ccc(F)cc1C(N1CCC(O)(CNC(c2cnc(Cl)[nH]2)=O)C1)=O n1(CC(N2C(CNC(C3CN(CC(F)(F)F)C3)=O)CC2)=O)nc2c(n1)CCCC2 N1(C(c2cc(C)nc(O)n2)=O)CCC2CCC(NC(=O)C=Cc3cnc[nH]3)C12 n1(CC(=O)NC(C2CCCC2)CNC(C=CC(C)C)=O)nc(C)n(C)c1=O Cc1cc(C(=O)N(C)CC2CCCN(C(=O)C(C)N(C)C)C2)cc([N+](=O)[O-])c1Cl c1(C(=O)NC2C(NC(CCOCC#C)=O)CC2)ccc(C(F)F)nc1O Cc1cc(C)nc(-c2cccc(-c3n[nH]c(CNC(=O)CC(C)(C)NC)n3)c2)n1 Cc1cccc(C(=O)NCCNC(c2cccnn2)=O)c1 Cc1cc(C#N)c[nH]c1=NC1CN(C(c2ccc(Br)o2)=O)CCC1C C1(C(=O)NC(CC)CN(C(=O)CCCCS(C)=O)C)CCc2c(nnn2CC)C1 N1(C(C2(C#N)C(C)(C)C2)=O)CCC2(CC1)CC2NC(c1cc(CF)on1)=O C12(C(=O)NCC3(O)CCN(C(=O)CC4(O)CCC4)CC3)CCC(CF)(CC1)CC2 CC(C(=O)NC1CC(CNC(C2(C#N)CCOCC2)=O)CC1O)S(N)(=O)=O c1(CC)ccc(C(=O)NCC2CCCCC2NC(=O)C(F)(F)C2CC2)cc1F C1(NC(C2(OCCCC)CCCC2)=O)CC(CO)N(C(c2cc(OC)n[nH]2)=O)C1 C(C(C(=O)NCc1nnnn1C)C(C)C)NC(C1(Cl)C(C(C)=O)C1)=O C(C)(C(=O)NC(CNC(N)=O)CO)NC(COCCCC)=O N1(C(CC)CC)CC(C(=O)NCCCN(C(=O)COC2(C)CCCC2)C)CC1=O C(=O)(C(C)(F)C(F)(F)F)N1CC(OC)C(NC(c2ccnc3c2CCO3)=O)C1 Cc1cc(C2(N(C)C)CCC2)no1.c12cnnn1C(=O)NCCCC1(CC1)NC2=O CC1CN(C(C2(O)CC2)=O)CCN(C(=O)CCCC2CCC2)C1 C1(CCC)CN(C(=O)CN(CC(=O)OCC2CC2F)C)CC1C(=O)NC c1(C(n2ncnc2C)=O)ccc(Cl)cc1.C(=O)(CC(C)C1CCCO1)OCC c1(CNC(C(CNC(C(C)OCC=C)=O)C)=O)cnn(C)c1C c1(C(N2CCOCC(CNC(CCC#C)=O)C2)=O)ccc(S(=O)(=O)NOC)cc1 c1(C(=O)NCC(C)CN(C)C(c2cc(F)cnc2Cl)=O)ccc(=O)n(CCF)n1 c1(C(N2C(CNC(C(C)=C3CCC3)=O)CCC2)=O)cc(Br)nn1C N1(C(CCOCCN(C(=O)CCCCN(C)C)C)=O)CCCC(O)(C2CC2)C1 c1(CC(=O)NC2CC(C)(NC(Cc3n(C)ccn3)=O)C2)cccc2nsnc12 C1(C(=O)NC(CC)C(C)(F)F)CN(C(c2sccc2CO)=O)CC(C)(C)C1 C1(NC(c2c(C)nc(C(C)(C)C)s2)=O)CC2CCC1N(C(=O)C(C)(C)F)C2 CCC(CC#N)N=c1[nH]c(=NCC2CC3CCC2CC3)[nH]c2cc[nH]c12 C(=O)(C(C(C)O)N(C)C)NC(C1CN(C(CN(C2CCCCC2)CC)=O)C1)C C1(C(=O)NCC2C(NC(CC(=O)OC)=O)CCCC2)Cc2ccccc2CCO1 C1(CN(C(=O)C=CC2(C)COC2)CC)CCCN1C(=O)CC1CN(C)C1 N1(C(c2c(CC)ccs2)=O)CCCCC1C1CCN(C(C2(C)CC2Br)=O)C1 C1(C(=O)NC2CCC(C(N3CCC(O)(CC)C3)=O)C2)(CC)CCNC1=O C1(C2CCCN(C(c3c(F)ccnc3F)=O)C2)(NC(=O)CC2(O)CCOC2)CC1 C1(C(C)C(=O)NC(C)(C)CC)CCN(C(c2ccn(C)n2)=O)C1 c1(C(=O)NCC(C)(C)OCCNC(c2ccc(C)c(Br)c2)=O)n[nH]c2c1CCCC2 C(CCNC(=O)C=Cc1cccnc1)(C(=O)NC1CC1CC(C)C)OC C1(CN(C(c2coc(N(C)C)n2)=O)CC)CCCN1C(c1scnc1C)=O CC1(CNc2cccc(CNC(=O)CC3CC4CC4C3)n2)CCOCC1 N#Cc1c(C(=O)NCc2cn3cc(Br)ccc3n2)[nH]c2cc(Cl)ccc12 c1(C(N2CCCC(NC(c3cn(CC=C)nc3)=O)C2C)=O)nccn2nccc12 c1(CCC2N(C(C(N3CCC(C)C(CO)C3)=O)=O)CCC2)c[nH]c2ccccc12 c1(C(=O)NC(CC)CNC(=O)C(C)Oc2ccccc2F)cc(C)n(C)c(=O)c1 c1(CNc2cccc(NC(Cn3c(C)cnc3)=O)c2)c(Cl)oc2ccccc12 C1(C(=O)NC2(CC#C)CCCCC2)CCN(C(c2cc(=O)cc(C)[nH]2)=O)CCO1 N1(C(C(C)OCC=C)=O)CCCC2C1CCN2Cc1ccc(F)c(Br)c1 c1(C(CCOC)NCC2CCCC2)ccc(O)cc1.C1(N)CC(n2ccnc2)C1 CN1CC(C(=O)NC2COCC2NC(=O)CC2(C)CC(F)(F)C2)CCC1=O N1(C(c2c(N)cn(C)n2)=O)CCC2(CCCN(C(C3CC(F)C3)=O)C2)C1 c1(C(=O)NCC2CCCC(CNC(CCS(C)=O)=O)C2)cccc2nc[nH]c12 c1(C(=O)NCC2(OC)CCN(C(c3csc(C)c3C)=O)C2)cnccc1C#N N1(c2ncnc(C)c2F)CCCC(C)(C)C1CNC(=O)CCc1ccn(C)n1 Cc1ccccc1COCC(=O)NCCC1(NC(=O)CCC(C)C2CC2)CC1 C1(C(=O)NC2C(NC(=O)Cc3cscn3)CCCC2)CN2CCN1CC2 Clc1ccc2c(c1)CN(c1nccc(N3CCC(OCCF)C3)n1)CCN2 C(=O)(C(C)(C)CS(N)(=O)=O)N1CCC(NC(c2cc(C)n(C(C)C)n2)=O)C(C)C1 C(=O)(C(COC(C)(C)C)O)N(CCC(C)C)CCC1CCOCC1.C(CC#N)NC=O C(=O)(C1CC(=O)c2ccccc21)N(C)CC1CN(C(C2(CO)CC2)=O)CCO1 c1(C(=O)NCCOCC(N2C(CCC)C(=O)NCC2)=O)cncc2[nH]ccc12 N1(C(C(CCC)NC(CN(CCC)C)=O)=O)Cc2cccc(C)c2C1 N1(CC(=O)NCC2N(C(c3c(C)ccs3)=O)C3C(C2)C3)CCP(C)(=O)CC1 N1(C(C2(CNC(C3C(OCC)C3)=O)CCC2)=O)CCN(CCOC)CC1 C#Cc1cncc(C(N2CCC(CN(C)C(C3CC(C(C)C)C3)=O)C2)=O)c1 Cn1cnn(CC(=O)NC2(CNC(c3coc(C(F)F)n3)=O)CCC2)c1=O C1(C(=O)NC2C(C)CN(C(C3CC3(C)Br)=O)C2)CCc2ccccc2O1 C1(NC(c2cccnc2)=O)CC2CC(C1)N(C(c1sncc1Br)=O)C2 CCC(CC(C)C)C(=O)N(CCNC(c1ccnc2cc[nH]c12)=O)C1CC1 C(=O)(CCC(C)(C)F)NCC(C)CC(=O)NC(C(F)(F)F)C1CC1 C1(CNC(c2c(C)nc(C)s2)=O)C2CCC(C2)N1C(=O)CNC(=O)CN(C)C CC(CC(=O)N1CCN(C(C2CC(F)(F)C2)=O)CC1CC(F)(F)F)CC(F)(F)F CS(=O)(=O)c1ccc2c(c1)CN(C(=O)C=C1CCSCC1)CC2 C1(CNC(C(CCC)N(C)C)=O)Cc2ccccc2CN1C(=O)CN(C)C(C)=O CCC(C)(C#N)C(=O)NCC(C(=O)N(C1CC1C)C)N(C)C c1(C(=O)Nc2ccc(-c3nc(O)n[nH]3)nc2)cnc(O)c(Br)c1 N1(C(CCOCCOC)=O)CCS(=O)(=O)C(CCNC(=O)C(F)C2CCC2)C1 C(CCC(C)C)(C(=O)NC12CCC(CC1)C2)NC(C1ON=C(CC)C1)=O C1(CC(=O)NC2(CCOC)CC2)CC(O)C1(C)C.C(C(O)CNC)O N1(C(c2nnn(C(C)(C)C)n2)=O)CCC(CC(C)(C)NC(c2cnc[nH]2)=O)CC1 c1(NCC(C)OC)cc(Br)ccc1S(=O)(=O)NC(C1CN(C)C1)C C1(CC)CCOC1C(=O)NCC(F)CNC(c1[nH]nnc1-c1ccnn1C)=O c1(C2(C(=O)NC3CCN(C(C4CC(C(=O)N)C4)=O)C3)CC2)cc(F)ccc1C.CO C(C)(C(N=c1nc(C2CCCC2)[nH]s1)C(C)C)NC(Cc1c(C)nsc1)=O N1(C(CCOC)=O)CCC(C(=O)NC(C23CCC(CC2)C3)C)(COC)CC1 C1(CN(C(C2CC(F)C(=O)N2)=O)CC)CCN(C(C2(CN(C)C)CC2)=O)CC1 N1(C(C2CC23CCC3)C(=O)NCC(F)F)CCN(CC2CCOC2)CC1 Cc1nc2ccccn2c1C(=O)N(C)CC1(NC(c2cccc(=S)n2O)=O)CC1 c1(N(C)C)ncccc1OC(C1CCN(c2ccccc2)C1=O)=O CCC(C)(C(=O)NCC(C)CNC(=O)CCNC(N)=O)C(N)=O CCC(C)CC(C(=O)N1CC2C=CC1CC2)NC(=O)C=C(C)c1ccccc1 C(=O)(CC(N)CCS(C)(=O)=O)N1CCC(c2ncc(CC)s2)C1C c1(OC)cc(C(=O)NC2CC(C)(NC(C3CC(C)C3)=O)C2)c2ccccc2n1 N1(C(c2cn(CCOC)nc2C)=O)CCC(NC(=O)C(C)SC(C)C)C(C)(C)C1 C1(NC(C(CNC(c2onc(CC)n2)=O)C)=O)CN(C)CCC1O N1(C(=O)Nc2cc(C)on2)CCC(NC(=O)CNS(C)(=O)=O)C(C(C)C)C1 C1(C(N(CC#CC)C)=O)COCCN1C(c1n[nH]cc1C)=O c1(C(=O)OC)cc(S(=O)(=O)NCCF)c(F)cc1Br Cn1cc(C(=O)NCc2ccc(N)cn2)c(C(F)F)n1 N1(C(c2cc(C)cc(C)c2N)=O)CCN(C(c2cc(C)n(C)c2)=O)CC(C)(F)C1 Cc1cn2nc(C(N3CC4C(CNC(C5(C(C)C)CC5)=O)C4C3)=O)cc2c(=O)[nH]1 N1(C(C(C)NC(CC)(C)C)=O)CC(NC(c2cccc(C)n2)=O)CC12CCC2 C(=O)(CC(C(F)(F)F)c1ccon1)NCC1N(C(c2cc(C)[nH]n2)=O)CC=C1 C12(NC(C3(OC)CCC3)=O)CC(CNc3ccnc(-c4nccs4)n3)(C1)OC2C CC(CC(C)(C)C)C(=O)NCC1CCCN(C(c2cc(C(F)F)[nH]n2)=O)CC1 c1(SC2CCC(N(C(CN(C(=O)CCC3CC3)C)=O)C)C2)ccccc1Cl C1(NC(C(C)N(CC(F)(F)F)C)=O)CC2CCC(C1)N2C(=O)CCc1cccs1 Cc1ccc(CN(C(c2ncc(Br)s2)C(=O)NCC2CC2)C)s1 c1(C(=O)NCC2(F)CC(NC(C3C(CC)CCO3)=O)C2)nc(C)c(C)[nH]c1=O Cc1sc2ccccc2c1C(N1CC2CC(NC(=O)CC3CCC3(F)F)C1C2)=O c1(C(=O)NCCCCNC(C2C(C(C)C)(CC)C2)=O)ccc(OC)c(F)c1F c1(C(=O)OCC)cc(N2CC(NC(c3cc(C(F)(F)F)on3)=O)CC2C)nc(Cl)n1 N1(C(C2C(CNC(c3ccc(O)cn3)=O)CC2)=O)CC2CCC(O)CC2C1 c1(OCC)ccc(CC(=O)NC(CN(C(=O)CN2CC3CC3C2)CC)CC)nc1 c1(C(=O)NC2CC3CN(C(c4onc(COC)n4)=O)CC32)cnc2ncccn12 c1(OC)nc(C)ccc1C(=O)NCCC1CCCN(Cc2c(C)noc2Cl)C1 C1(NC(C=CCOC)=O)CCC(C)(CNC(C2(n3cnnn3)CC2)=O)C1 C1(C(=O)NCCN(C(C(C)=C(CC)C)=O)C2CCCC2)CCc2ncccc2C1 C(=O)(C1CCC(=O)c2ccccc21)N(CCNC(c1cccc([N+](=O)[O-])c1)=O)CC c1(C2CN2)c(F)ccc(I)c1Br.Oc1csc(CN2CCCC2)c1 C(=O)(C(C)C(C)(C)C)N1CC(NC(c2cc(C(=O)OC)[nH]c2)=O)C(C)C1 c1(OC)cc(Br)c(C(c2nnnn2CC(F)F)NC2CC2CC2CC2)cc1Cl c1(CCC)ccccc1NC(=O)CNC(c1cc[nH]n1)=O c1(CC)ccc(C)c(C(N2CC(CNC(=O)C(C)SC(F)(F)F)C(C)C2)=O)c1 c1(COC)cc(C(=O)NCc2cn(CCNC(=O)C(C)C3CC3)nn2)on1 CCC(C)(C(=O)O)NC(=O)CS(=O)(=O)N1CCN(C)CC1 C(=O)(CCCSC)N(CC=CC(=O)N(CC#C)CCOCC(C)(C)C)C N1(C(C(C)OCCOC)=O)CCOC(CCNC(=O)CC(C)(C)c2cccs2)C1 C1(CCC)CN(C(=O)C(CCSC)OC)CCN1C(C1(C)COC1)=O c1(CNC(c2c(C)nc(COC)s2)=O)cc(OC)cc(C)c1OC c1(CC(N2CCC(NC(C(C)OC)=O)C2C2CC2)=O)cc(Cl)cnc1C n1(CC(=O)NCC2CC(NC(c3sccc3F)=O)C2)ccc(-c2ccccc2)n1 c1(C(=O)NCCCNC(CC2CC(OC)C2)=O)sc(C2CCCC2)nc1C(F)F c1(CNC(C2COCCC2NC(=O)CCc2ccsc2)=O)cccnc1F C1(C(N2CCN(C(C)=O)CC2)=O)CC2CCC(C1)N2C(=O)C(C)NC(=O)C1CC1 N1(C(CC(=O)OCC)=O)CCC(NC(C23CCC(CC2)C3)=O)C(CC)C1 c1(C(=O)NCCOC(C)(C)CNC(C2CC23CC(O)C3)=O)cccc2c1OCC2 c1(C(=O)NCC(CNC(=O)CCCc2ccccc2)O)cc2c(s1)COCC2 c1(CC(=O)NCC(CN(C)CC=C2CN3CCC2CC3)O)ccc(S(C)=O)cc1 C=CCC(C(=O)NCC1CC(C(=O)NC(C)CS(C)(=O)=O)C1)OC C(CC1CCC1)(C(=O)NC1(CNC(c2cc(CO)on2)=O)CC1)OC C1(C(=O)NCC2(F)CN(C(c3[nH]c(=N)sc3)=O)C2)CC(F)(F)CS1 c1(C(C)Nc2nccs2)ccc(OC(F)F)c(-c2cccc(C(F)(F)F)c2)c1 Cc1ccc2[nH]nc(C(=O)NCC(C)(CO)NC(c3sccc3C#N)=O)c2c1 C1(NC(C(C)NC(COC)=O)=O)Cc2ccccc2C1NC(c1cnccn1)=O N1(C(c2ncn(C(C)C)n2)=O)CC(O)CC1CNC(C1COCCO1)=O c1(C(CNC(c2c(C)nn(C)c2)=O)NC(c2cncn2C)=O)cc(F)cc(Cl)c1 N1(C(C2CCCS2(=O)=O)=O)CCCCC1C1(C(=O)NCCn2cncn2)CC1 N1(C(CSC)=O)CC2C3CCC(C2C1)N(C(C1CCC2(CC1)CC2)=O)C3 N1(C(C(C)(CO)OC)=O)CCC2(C1)CN(C(=O)C=CC1CCCCC1)CC(C)O2 N1(c2ncn(C)c2)CC2CCC(NC(c3n[nH]c4c3CCCCC4)=O)CC2C1 CN1CCN(C(=O)CN2CC=CC2)C(C(=O)N(C)CC2CCCCC2O)C1 C(N=c1nc(Cc2ccccc2)[nH]s1)c1cccc(NC(C=C(C)Cl)=O)c1 c1(SC)ccc(CCCNC(=O)N(C2CCC2)CC2CC2)cc1 c1(C(=O)NCC2N(C(Cc3cnc(C)s3)=O)CC=C2)cc2n(n1)CCCO2 CCCC(C)C(=O)NCC(C)CN(C(=O)CCCN(C)C(c1ccccc1)=O)C c1(C(=O)NC2C(CNC(CCC(=C)C)=O)COC2)cccc(O)c1Br c1(C(N2CCC(N(C(C3ON=C(C)C3)=O)C)C2)=O)c(C(F)F)nc2n1CCCC2 c1(C(=O)NC2CC3(C(NC(CSc4cccc(C)c4)=O)C3)C2)cccc2c1CCC2 c1(CC)ccc(-c2cc(NC(=O)NCCOCCC3CC3)on2)cc1 c1(OC)ccc(S(=O)(=O)Cc2ncccn2)cc1Br N1(C(=O)Cn2cnc(C(F)(F)F)c2)CCCC2(C1)CN(C(c1ccncn1)=O)C2 CC1(C(=O)NC2CC(CNC(=O)C(c3ccsc3)C3CC3)C2)CC1(Cl)Cl CC1=NN(C)C(=O)C1CC(=O)NCC(C1CC1)NC(=O)CSc1ccccc1O C(=O)(CCCC(CC)NC(=O)C(O)C1CC1)NCCOCC(=C)C N1(C(c2cnc(CC)[nH]2)=O)CCN(C(=O)CN(C)CC)C2(CC2)C1 C1(NC(c2c(Cl)ccc(C)c2)=O)CCC2CCN(C(=O)C(Cl)=CCl)C1C2 n1(CCC#C)c(N(C2CC2)CC2CC2)nnc1C1CC1C CCC(C(F)(F)F)NC(=O)C(CCOC)NC(=O)CC1CC2C=CC1C2 C(=O)(CC(C)(C)C(F)F)N1CCC(C(C)(C)CNC(=O)C(O)C(C)(C)C)CC1 C1(C(=O)N)C(c2csc(COC)n2)C1(C)C.C(C)(C(=O)N1CCC1C(=O)OC)OCC CCC(C)(CCNC(=O)Cn1cnnc1)NC(C1CCCOC1C)=O N1(C(c2cccc(C3CC3(F)F)c2)=O)CC2(CCN2C(=O)CSc2cccs2)C1 C1(NC(c2cc(C3CC3)on2)=O)CS(=O)(=O)CC1NC(c1cc(Cl)cnn1)=O Cc1occc1C(=O)NCC(c1ccccc1)N(C)C(C1(C)CC(C)C1)=O CC1CCCCC1(C)n1cc(CCC2CN(C(c3cc([N+](=O)[O-])n[nH]3)=O)C2)nn1 c1(CC)nc(N2CC(CCOC)(NC(C3CCOC3CC)=O)C2)c2ccsc2n1 CC(C)(C)C(=O)N(c1nc(C(=O)Sc2cocn2)cs1)C(=O)O.c12cn(nn1)C2 C1(CNC(c2cnc(COC)s2)=O)CC2CCC(C1)N2C(C1CC(SC)C1)=O C(=O)(CC(C(F)(F)F)OC)N1CC(CC)(NC(c2cc(C(N)=O)c[nH]2)=O)C1 c1(CC(=O)NC(C2CCN(CC3CC3)C2)C)ccnn1Cc1nc(C(F)F)no1 c1(C(=O)NC2CC2NC(c2cnc(C(F)(F)F)o2)=O)cc(Cl)c(F)c(Cl)c1 CCCCCCCCCCC(=O)N1CCC(NC(C23CCC(C2)OC3)=O)C1(C)C c1(C(=O)NC2C3CN(C(C(CCCOC)C)=O)C2C3)ccc2c(c1)NC(=O)C2 C#CCC(C)(C(=O)NCC(C)C(=O)OC)NC(=O)CCNC(=O)OC C1(C(N2CC(O)(C(C(=O)NC3(C=C)CCCC3)F)C2)=O)CC2(CCC2)CO1 CC(CCN(C)C)C(=O)NC(C)C(C)NC(=O)COCP(C)(C)=O C1(CC)(NC(c2ccnnc2Cl)=O)CCN(C(=O)C(C)Oc2ccccn2)CC1 c1(C(=O)NC2CCCC(NC(C(C)=C3CCCC3)=O)C2)occ2c1CCOC2 C12(C(N(CC(=O)NCC)C)=O)CC1CN(C(c1cn(C3COC3)nn1)=O)C2 C1(C(=O)NCC(CN(C)C(C2C3(CC3)C23CC3)=O)(C)C)C2CCC(C2)S1(=O)=O Cn1ncc(C(=O)NC2CC(NC(=O)Cc3ccc(Br)s3)CC2O)c1N c1(C(=O)NC2CC(F)(CNC(C(CC)C#N)=O)C2)coc(S(N)(=O)=O)c1 Cc1ccc(C(C(=O)NCC(CO)NC(=O)CCn2cnnn2)C(C)C)cc1 C#Cc1ccc(Cl)c(SCC(=O)NCc2cccs2)c1.C(CCOC(F)F)N C1(CNC(c2ncc[nH]2)=O)C=CCN1C(=O)CCCc1cc[nH]n1 O=C(C1=NOC2(CCN(C(=O)Cc3ccc(Cl)s3)C2)C1)Nc1ncc(F)c(Cl)n1 c1(SC(CNC(c2cccc(OC)c2)=O)OC)ccc(Cl)cc1Cl Cc1cc(C(N2CCC(NC(C3(F)CCCOC3)=O)C(C)(C)C2)=O)cc(N)c1O c1(C(=O)NC2C(NC(C(C)Sc3nnnn3C3CCCC3)=O)CC2)sccc1Cl N1(C(C2C(C)CCN2C(c2cc(CO)[nH]n2)=O)=O)CC2(C1)CC(C)(O)C2 CC1CN(C)CC(C(=O)NC(C(=O)NCC2COC(=O)N2)c2ccoc2)O1 C1(CN(C(=O)CCn2cccc2)CC)CCCN1C(=O)CCc1csc(=N)[nH]1 N1(CC(=O)NC2C(N(C)C(c3nncs3)=O)C2)CCCCCC1 C1(CNC(C(CCSC)C)=O)CC(C)(C)CN1C(=O)C(C)NCC1CCCO1 c1(C(=O)NCC(N(C(=O)C(F)(F)CC2CC2)C)C2CC2)ccc2ncnn2c1 CC1(C)CNC(=O)C1NC(C1CCCCN1C(=O)CCC1CCCO1)=O c1(C(=O)O)cc(CN2CC3(CC3)CC2C(N2CCOCC2CO)=O)ccc1O C1(NC(C2C(NC(c3c(C(C)=O)coc3)=O)CCC2)=O)CC(C)N(C)CC1C CC(CC(=O)N(C(C)(C(=O)NCCc1ccccc1)C1CC1)C)n1cccc1 C1(NC(CC2(C)CCCCC2)=O)CN(C(c2cc(Cl)ccc2F)=O)CC1C#N c1(C(N(CC(C)N(C(C(CC=CC)C)=O)C)C)=O)ccc(N)cc1Br n1(CC)cc(C(=O)NCC(C)(C)CNC(=O)C(C)(C)CC)c(-c2ccccc2)n1 C12(C(N3CC(C)(NC(C4C(COC)C4)=O)C3)=O)CCC(CC1)C2(C)C c1(C(=O)NC(CC=C)CNC(C2CCC(F)CC2)=O)cc(O)cc(Br)c1 C(=O)(C(F)(F)C(O)C(C)C)NCC1OCCN(C(CC2CC(C)C2)=O)C1 Cc1cc2c(C)n1C1C(N(C)C)CCN(C1)C2=O.C1(C(=O)C2CC2)(CF)CC1 CN1CCN(C(=O)CCC(C)(F)F)C(CNC(c2ccn(C3CC3(F)F)n2)=O)C1 C(=O)(CC1=NNC(=O)C1)NCC1CCCN(C(C(c2cc(C)c(F)cc2)=O)=O)C1 c1(NCc2c(Br)ccc(C)c2)ccc(S(=O)(=O)NCCCCF)cc1Br CN(C)S(=O)(=O)N1CC(C(=O)NCCNC(C2CCCC(O)C2)=O)C1 C1(CC(=O)NCC2CCN(C(c3nc(CC)[nH]n3)=O)CC2C)CC2(CCCC2)CO1 C1(NC(C2(CC#C)CC2)=O)CCCC(NC(=O)CC2CC(=O)NC2=O)C1 C1(Nc2scc(CC(N)=O)n2)CCOC(c2cccc(F)c2)C1 C1(NC(CNC(C)=O)=O)CCN(C(=O)C(c2ccccc2F)C)C1C N1(C(CNC(c2ccc(C)s2)=O)=O)CCCCC1CNC(=O)CCC1(C)CC1 C1(C(=O)OC)CC(C(=O)N(C2CC(NC(=O)C(C)NC(C)=O)C2)C)C1 C(=O)(C(F)CCC(C)(C)C)NC(C)C(N1CCC(F)(F)C1)=O C(=O)(C(F)(F)c1nccs1)NCC(C)NC(C1CC(n2ccnc2)C1)=O c1(C(=O)NC(CNC(CNC(C)=O)=O)(C)C2CCC2)cc(C#N)on1 Cc1nc(C(N2CCC(C(C)(C)NC(C3CCCC3C)=O)C2)=O)c2ccccn12 N1(C(C(CN(C)C)(C)C)=O)CC2CC(NC(c3cnn4c3NCCC4)=O)CC2C1 c1(OC)cc(C(=O)NCCNC(C2(C)CC2F)=O)ccc1-n1cccc1 c1(CCC(=O)NCC2N(C(C(CC#C)C)=O)CC(O)C2)ccc(OC)c(C)c1 CC(N=c1cc(Oc2ccccc2)nc(C(F)(F)F)[nH]1)c1cc(Br)ccc1Cl O(P(C)(=O)CCNC1C(=O)OCC1C)CC c1(C(=O)NC2(CC=C)CCCN(C(=O)C(F)C(=O)OC)C2)cc(F)c(F)cc1Cl C=CCC(CC(C)C)C(=O)NCCC1CC(NC(c2ccncc2Br)=O)C1 c1(CN=c2scc(C=O)[nH]2)c[nH]c2ccc(F)cc12.NC1CCc2ccccc21 C12(C(N(CCC(C(C)C)NC(C=CCC)=O)C)=O)CCCN(C1)S(=O)(=O)C2 C1(CNC(c2ccncc2Cl)=O)CN(C(=O)COCC2CC2)CC1C(F)(F)F CC1CCC(CC(=O)NCC2COCC2NC(c2cc(C3CC3)on2)=O)O1 Cc1cc(C(=O)NC(C)CCNC(=O)COCCO)ncc1C#N C1(C(N2CCC(NC(C3CC3c3ccco3)=O)(CF)C2)=O)CCCCC12CCC2 c1(C(=O)NCCCCNC(c2cc(C3CC3)ns2)=O)cc(Cl)ccc1Cl c1(C(N2C(C(N3CC4CC4C3)=O)CC(C)C2)=O)cn2cccc(Br)c2n1 N1(C(CCCOCCC)=O)CCC(CNC(=O)CCc2cccn2C)C1(C)C c1(C(=O)O)cc(C(=O)O)cc(C(=O)NCCc2nccn2-c2ccccc2)n1 N1(C(C(C)OCC)=O)CCC2(CC1)CC(NC(c1c(C)noc1C(C)C)=O)CO2 N1(C(c2nnc(CC)s2)=O)CCC2(NC(c3nc(C)sc3C)=O)CCCC12 C1(CCC(=O)NCC2CCCC23CC3)CCCCN1C(=O)CCCn1ccnc1 c12cc(C)nc(n1)NC(=O)c1ncncc1-2.c1cccc(C(F)(F)F)c1F.CS Cn1ccc2[nH]c(C(=O)NCCCNC(C3CC3F)=O)cc12 N1(C(C(C)N(C(=O)CCOC2CCC2)CCC)=O)CCn2ccnc21 C1(NC(C(CCC)C)=O)CCC(O)CN(C(=O)C=Cc2nc[nH]n2)C1 Cc1cc(C)cc(S(=O)(=O)N2CCC(CC(=O)NC3CCC(F)(F)C3)C2)c1 Cc1ccc(C2CC2C(=O)NC2CCCN(C(C3C4CNC(=O)C34)=O)CC2)c(Cl)n1 c1(CCC(=O)N(C2CN(C(=O)C3=NOCC3)C2)C)nc2cccc(F)c2[nH]1 Cc1cc(C(=O)NCCOCCNC(c2ccn(C(=O)OC(C)(C)C)n2)=O)n[nH]1 C(=O)(C1CCCc2ccc(O)cc21)NC1C(NC(C=CC=CC)=O)CCCC1 C1(CNC(CN(S(CC)(=O)=O)C2CC2)=O)(NC(=O)CC2CCOC2C)CCCCC1 c1(OC)cc(CO)ccc1-c1cc(C(=O)NCc2cc(O)cc(O)c2)n[nH]1 C(=O)(CC1COCc2ccccc21)NCC1CCN(C(CC(=O)OCC)=O)CC1 n1(-c2ccn(CC)n2)nc(-c2cccc(CO)c2)nc1CSC1CCC2(CC2)C1 N1(C(C(C2CC2)SC)=O)C2CCC1C(CNC(=O)CC1CC1)C2 N1(C(=O)NC(=O)NC(C(CC)O)C)CC(C)OC2(CCC2)C1 c1(C(=O)NCC(C(C)C)NC(c2coc(Cl)n2)=O)ccnc2c1CCC2 C(CN=c1[nH]c(=NCCCC(=O)NC)c2ccccc2[nH]1)SCCNC(CC)=O c1(NCC2C(C(=O)Nc3c(C(=O)OC)cccc3O)C2)cc(C)cc2[nH]ncc12 c1(OC)cc(C(=O)N(CCn2cc(-c3ccccc3F)nn2)CC)n(C)n1 CC(CCC(=O)NC1C(C)C1C)NC(=O)C(O)Cn1cncn1 C1(CCC(=O)NCCCOCCCC)CCCN(C(C2CC3CC3C2)=O)C1 c1(OC)cccc2c1C(C(=O)NCC(C)(C)NC(c1cnsn1)=O)CC2 Cc1ncccc1C(N1CC(F)CC1C(=O)NCc1ccc(I)cc1)=O c1(N(CCCc2cccc(Cl)c2)CCOC)ncc([N+](=O)[O-])o1.c1(=O)c(=O)[nH]1 N1(C(C2C(C(C)C)N(C(c3ncncc3N)=O)CC2)=O)CC(C)C(C)C1C CS(=N)(=O)C1CC(NC(C2CCCC(F)(F)C2)=O)C1 c1(C(C)C)nnc(C=CC(=O)NC2C=CCN(C(C3CC4CCC3O4)=O)C2)o1 S(=O)(=O)(c1ccc(N(C)CC)cc1Br)NCCCNC(n1ccnc1CCC)=O C1(OC)CN(C(=O)CC2CCC(C)(C)C2)CCC1NC(c1cccc(C#N)c1)=O C(=O)(CCC(=O)Nc1ccn(CCO)n1)NCC C1(C(N(C)CC2CC=CCC2)=O)CC2CCC(C1)N2C(=O)C1=C(Cl)CCCC1 c1(C(=O)NC(CC)CNC(=O)C(N2CCC(OCC)C2)=O)ccnc(F)c1N c1(C(=O)NCCCNC(C2C(C#C)C2(C)C)=O)cc2c(nc1O)CCCC2=O C(CCCCC(=O)N(CCN=[N+]=[N-])C)N(C(=O)CC1CC(=O)NC1=O)C N1(C(C(CC=C)C)=O)CCCCC12CC(NC(=O)CCC(=O)c1cccnc1)C2 c1(C(=O)NC23C(CN(C(CNC(C(CC)C)=O)=O)C2)C3)ccc(N)c(C)c1C c1(CC(C)C(N2CC(NC(=O)CSC3CC3)C(CO)C2)=O)ccc(F)cc1F C(=O)(C1CCCc2cncn21)NC1CN(C(C=CCC)=O)CC2(C1)CC2 c1(CC)nc2n(n1)CC(C(=O)NC)CC2.N12CC(C1)C(OC)C2=O c1(OCC(=O)NCCC2(O)CCN(C(C(C)=C(CC)C)=O)C2)cccc(Cl)c1Cl C1(O)(CCNC(C(C#C)(C)C)=O)CCCN(C(c2c(N)cccc2Cl)=O)C1 C1(NC(C(CC)NC(C)=O)=O)CC2CCC1CN(C(c1ccc(F)c(OC)c1)=O)C2 C1(c2cncnc2)(C(=O)NC(CC)CNC(=O)Cn2ncnn2)CCCC1 Cc1ccc(C(=O)NCC2CCN(C(=O)C#CC(=O)O)C2)cc1C c1(N2CCC(C(COC)C)CC2)nc(C)ccc1C c1(C(=O)NCC2CN(C(CCCC)=O)C2)ccc(F)c(C(C)(C)C#N)c1 Cn1nnc(C(=O)NCCCCC2CCCC2)c1C(=O)NOCC1CCOCC1 N1(C(=O)CC2CC2(Cl)Cl)CCN(CCNC(C2(CO)CCC2)=O)CC1 c1(C(N2C(CCC)CN(C(=O)C(CC)OC)CC2)=O)c(N)cccc1[N+](=O)[O-] c1(OC)cccc(Br)c1CN1CCC(Oc2cnn(-c3ccccc3)c2)CC1 N1(C(C2(NC(N)=O)CC2)=O)CC2(COC(CNC(c3ccc[n+]([O-])c3)=O)C2)C1 Cn1ncc(Cl)c1NC(C1(C(=O)NCC2CC(F)(CNC(N)=O)C2)CC1)=O Cc1nc(C2CCOC2)sc1C(=O)N(C)CC1CCN(C(=O)COC(C)C)C1 C(C1CC1)(C1CC1)=CC(=O)NC(CC)CNC(c1cnn(CC(F)(F)F)c1)=O C1(NC(C2CC(N(C)C)C2)=O)CC(O)CN1C(=O)C(c1ccccc1)O N12c3ccccc3C(n3cc(nn3)C1=O)C2(C)C.CC(C)(C)SCC(=O)OC=CCl N1(C(COCC)=O)CC(C2CCCN(C(c3coc4c(F)cc(F)cc34)=O)C2)C1 c1(C(=O)NCC(C)(C2CC2)NC(c2noc(CC)c2C)=O)cc2ncccc2o1 C(=O)(CC(CN)C(F)F)N1C(c2n(C)ncc2)CCCC1 C1(NC(c2cccs2)=O)CCN(C(=O)C(c2cccc(Cl)c2)(F)F)CCC1CO N1(C(c2nc(OC)c(C)s2)=O)CC2CC1CN(C(=O)C(C1CC1)OC)C2 C(=O)(CCC(CC)NC(=O)C1=CCCCO1)NCC(C1CCC1)OCC CC(C)C(C)(O)C(=O)NC1CC(C(F)F)(NC(C2CC3CCC(C2)O3)=O)C1 N1(C(C2(C)C(C)(C)C2)=O)CC2(C=C(C(=O)NC3CCCC4(C3)N=N4)CO2)C1 C(=O)(CS(C)(=O)=O)NCC(C(C)C)NC(C(C)NC(=O)NC)=O CC1CNC(=O)C1NC(=O)NC(c1ccccc1Cl)CC(N)=O C(=O)(CCCCCCBr)NC1CC(CN(C2CN(Cc3ccccc3)C2)C)C1 c1(C(=O)NCCCN(C(c2n(CC)ccn2)=O)C)cc(F)c(CO)c(F)c1 N1(C(C(C(c2ccc(C)cc2)C)O)=O)CCC(N=c2nc(C(C)C)[nH]s2)C(C)C1 N1(C(c2ccc(C)cc2)=O)CCC(NC(=O)CSS(C)(=O)=O)C(C)(C)C1 Cn1nnnc1CNC(N1CCC(NCCCn2ccnn2)C1)=O C=CCC(C)(C)CC(=O)NC1C=CC(CC(=O)Nc2cc(C)cc(C#N)c2)C1 C1(C(C(=O)NCC2C(C(=O)OC)C2)F)CCCCC1.C12CC1C(C)NC2=O C1(C(c2n(CCC(=O)OCC)nnn2)NC(C2(CC)CC2)(C)C)CCCOCC1 c1(CN2CCC(N(C(c3cccc(C(N(C)C)=O)c3)=O)C)C2)ccc(C#N)cc1 C1(CC(=O)NC(C2CN(CC(COC(C)C)O)C2)C)CCCNC(=O)C1 C(=O)(CC(O)C(C)(C)C)NC1(COC)CCCN(C(c2coc(C)n2)=O)C1 C1(C(=O)NCc2cc(CC)no2)(CNC(C2CCC2)=O)CCOCC1 c1(NC(=O)C=C(C)CNC(C2C(CCOC)C2)=O)cccnc1.C1(N)CC1 C1(C(=O)NCC2N(C(C3C(C=C)C3)=O)CC2)CCC(=O)N1CC c1(C(N(CCCNC(c2c(CC)noc2C)=O)C2CC2)=O)cc(C)cc(F)c1N c1(SC)cccc(C(=O)NCCCOCCNC(c2cc(Cl)ccn2)=O)c1 C=C(C)C(CC(=O)NC(C(=O)Nc1cnc(C)c(C)c1)C1CC1)OCC C1(NC(CC(CC)C)=O)COC2CN(C(=O)COCC(F)F)CC12 CC1CCC(NC(c2cc(N)cc(O)n2)=O)CN1C(=O)CCC(N)=O c1(CC(=O)N(CCNC(C(C2CCCCC2)OC)=O)C)ccc2ccccc2c1 C1(CN(C(C(c2ccccc2)C)=O)C)CCCN1C(c1cn(C2CC2)nn1)=O C(=O)(C1=CC2CC=CCC12)NCc1cn(-c2c(OC)cccc2C)nn1 N1(C(C2CN(C(CNC(=O)OCC)=O)CC23CC3)=O)C2CCC1CC(=O)NC2 Cc1ccc(C(=O)NC2CCCC2(C)CN(C)C(C2COCCO2)=O)c(N)c1F c1(C(=O)Nc2nc(-c3ccccn3)cs2)cc(O)c2occc2c1 Oc1cc2c(nn1)CN(Cc1ccccc1-c1cc(F)cc(F)c1)CC2 c1(OC)ccc(O)cc1C(=O)NCCC(C)(C)NC(C1CCCC(C(N)=O)C1)=O C1(C(=O)NCCC(=O)NCC)COCC1NC(C1(Cl)CC1(F)F)=O C1(CC(N2CCC(CC=C)(NC(C3CCCCC3)=O)C2)=O)SC2=NCCN2C1=O CCC(C(=O)N1CC(N(C)C(c2ccnc(OC3CC3)c2)=O)C1)C(C)(F)F C1(C(C(N2CC(CCC)C2)=O)C)CCCN(CC2CC(=O)C2)C1 N#Cc1ccc(N2CCC(=CCNC(C3CC3F)=O)CC2)nn1 N1(C(c2cccc(SC)c2)=O)CC2CCCC2(CNC(=O)C2=CCC(C)CC2)C1 c1(C(=O)NCC2(C)N(C(=O)C=C(C)C)CC(OC)C2)cccc2c1OCCC2 N1(C(C(n2cc(-c3ccc(Cl)cc3)nn2)C)=O)CCCC2CC1C2(C)C c1(C(N(CC(CNC(c2cc(COC)sc2)=O)C)C)=O)ccc(N)c(Cl)c1 C12(CC(=O)NC3C(NC(c4ccc(C)cn4)=O)COCC3)CCCN1CCC2 C(C(O)C(C)(C)C)NC(CCN(C(c1n(CC)ccc1)=O)C(C)C)=O C1(C(=O)NC2(C(=O)NC(c3nccs3)C)CSC2)CCC(C)(C)OC1 CC1CCC(N(C)C(c2cccnc2OCC2CC2)=O)CC1 c1(OCC(C)(C)Nc2cnc(C(C)(C)C)o2)cccc(-c2ccno2)c1 N1(C(c2ccc(COC)o2)=O)CCC(C)(CC(=O)NCC2CC[Si](C)(C)C2)C1 C(=O)(CCC(CC)OC)NC(CCC)CNC(=O)CC1CC(C(F)F)C1 N1(C(c2n[nH]c(C)c2O)=O)CC2CCCC2(NC(=O)CSc2nnc(S)s2)C1 C1(O)(CC#N)CCN(C(c2cc(C3CC3)no2)C(=O)NC2CCCCC2)C1 c1(OC)ccccc1CC(N1CC(OC)CC1CNC(c1ncccc1O)=O)=O CC1(C)CCc2cccc(C(=O)NCCC3(NC(C4CCC4F)=O)CCC3)c2O1 N1(C(C(C)CN2CCOCC2)=O)CCCC(N(C)C(c2ncccn2)C)C1 c1(OC)cccc(C(C)=CC(N2CCOCC2CNC(c2nocc2C)=O)=O)c1 C(C)(C(C)(C)NC(=O)CCF)NC(C(SCCC(C)C)SC)=O C1(NC(c2c(OCC)scc2)=O)CC2CC1CN2C(=O)C=C1CCCCC1(C)C Cc1ccc(C(=O)NCC2(O)CCCN(C(C3(C)CSC3)=O)C2)c(C)n1 c1(C(N(CCN(CC)CC)CC)=O)cccc(CNC(=O)CC(C)O)c1 C1(C(=O)NCC=CCNC(CC)=O)CCc2nnc(C)n2C1 C#Cc1ccc(C(N2CC3C(CN(C)C(c4cn(CCC)nn4)=O)C3C2)=O)cn1 C=C(CNC(=O)C(F)C1CC(NC(=O)C(=O)NCC(F)F)C1)C(F)(F)F c1(C(N2C(C)(C(=O)NC3(CC=C)CCOC3)C=CC2)=O)cc(C)nc(C)c1 N1(C(C(C)OC)=O)CC2=C(C1)CN(C(c1ccc(-c3ccc(C)o3)s1)=O)C2 N1(C(CC2(C)CC2)=O)CCOC2CN(C(C3CCCS3)=O)CC12 c1(CN(C(=O)COC2(C)CCCC2)C)ccc(CNC2(Cl)CC2(F)F)cc1 C1(NC(C(c2ccnn2C)NC(c2c(C(C)C)nco2)=O)=O)CCCC(F)(F)C1 C1(C(=O)NCCCCCCNC(c2c(OC)nccc2)=O)OCC2CCCC1C2 CC(C)CC(CO)NC(=O)C(=O)NCCC1CCN(C(=O)CCc2cnoc2)C1 C(CN=c1c(Br)c[nH]cc1[N+](=O)[O-])C1C(C)CCCN1C(c1ccco1)=O c1(C(N2CC=CC(NC(C(C)SCCCC)=O)C2)=O)cc(F)cc2cccnc12 C(=O)(CC(=O)NC1CC(NC(=O)CC(C)n2ccnc2)C1)OCC C1(NC(N2CCC(CN(C=O)CC)CC2)=O)COc2ccccc2O1 C1(CC)CCN(C(=O)CSCC(N)=O)C(C(N2CCCN(C(C)=O)CC2)=O)C1 c1(C(=O)NCCC2CC(C(=O)NCC(C)(C)C(N)=O)C2)ccc2cncn2c1 c1(C(=O)NC2CCCC2NC(C2CCC=CCC2)=O)cnc(O)cc1C(F)(F)F c1(SCC(N2CC3CCC3(Cc3cn(CC)nn3)C2)=O)ccc2nc[nH]c2c1 N1(C(Cc2ccn(C(C)C)n2)=O)CCN(C(=O)C(CO)N(C)C)C(CC(F)F)C1 N1(C(c2c(C)ncnc2)=O)CC(NCc2ccc(Br)cc2C(=O)O)CC(C)C1 C1(NC(=O)C2=COCCO2)CC12CCC(NC(C1CCCOC1)=O)CC2 C1(C(=O)OC(c2c(C)cc(C)c(C)c2)C)CC2CCCCCCC12 Cn1nc(C(N2CCC(O)(CNC(=O)CCC[N+](=O)[O-])C2)=O)c2ccccc12 N1(C(C2(COC)CC(=C)C2)=O)CCOC(C2CC(F)(F)C2)C1 C12(C(=O)NC3(C(N(C)CC4CC(O)C4)=O)CC3)CCC(C)(C1)OC2 C(c1cn(C)nn1)=CC(=O)NCC(CNC(=O)C(CO)OC)OC CON(CCC(=O)N1CCC2CC12C)C(=O)C1CCC(=O)O1 N1(C(CCc2ccc(C)nc2)=O)CC2CCCC2(CNC(=O)C2=CCCC2)C1 CC1CC(=O)NC(C(=O)N(CCCNC(C2(C)CCCNC2=O)=O)C)C1 N1(C(C(C(C)C)NC(C)(C)C)=O)C2CCC1C(C(=O)Nc1scnc1C(N)=O)C2 c1(C(N(CC(C)C(=O)NC2CCC(=O)NC2)C)=O)ccc(O)cc1 CCCCCCC(F)C(=O)N1CC2CCCC1(CNC(c1cccnc1N)=O)C2 C(C)(C)(CCCNC(=O)CC1CC(C)N(C(=O)CN(C)C)C1)OC C1(CN(C(=O)C=CC2CC2)CC)CCCN1C(=O)CC(c1ccccc1)OC C1(C(C)NC(c2cnc(CC(C)(C)C)s2)=O)CCN(C(c2cc(F)cs2)=O)CC1 C1(C(=O)NC2C(NC(C3(S(C)(=O)=O)CCC3)=O)CC2)Cc2ccccc2C1 c1(C(=O)NC2C(OC)CN(C(=O)CCc3nc(C)c(C)[nH]3)C2)cc(O)nc(C)n1 N1(CC2COCC(C)(C)O2)CC(CNC(=O)NN2CCOCC2)C2(CCC2)C1 N1(C(C2(C(C)C)N(C(c3cncc(C)n3)=O)CC=C2)=O)CCOC(C)C1C c1(CNCC2N(C(c3nncc(OC)c3)=O)CCC2)ccc(Br)c(C#N)c1 Cc1ccc(=NCCC(=O)N2CC(CC(C)NC(=O)C(CO)C(C)(C)C)C2)[nH]c1 C1(NC(c2cnsc2)=O)CCCCCN(C(c2ccncc2C(F)(F)F)=O)C1 c1(C(=O)NCC(N(C)C(C2CC3CCC(C2)C3)=O)C2CC2)ccn2c1CCCC2 C(=O)(C1CCc2cccc(O)c21)N1CCC(C)(CNC(c2c(C)cco2)=O)C1 C1(NC(C2CC(OC)C2)=O)CCCCCN(C(=O)Cc2cnc3ncccn23)C1 N#Cc1cc(F)c(C(=O)NC2CN(Cc3ccc(I)cc3)CC2O)c(F)c1 c1(OC)cccc2c(C(=O)NC3(CO)CCN(C(C45CCC4C5)=O)C3)cnn12 O=S(=O)(c1c(Cl)cc(Br)cc1Cl)N(c1nc2cc(Cl)ccc2s1)C1CC2(CNC2)C1 C(=O)(C1CCc2ccc(Cl)nc21)N1CCCC(C)(NC(CCNC(C)=O)=O)C1 c1(C(N2CC3C(CNC(c4ccc(Cl)s4)=O)(C3)C2)=O)nc2ccccc2[nH]1 c1(-c2nc(-c3c(C)cc(C(=O)OC)s3)on2)c(F)ccc(C)c1F c1(OC)cc(C(N2CCC(NC(=O)C(C)Sc3ccccn3)C2)=O)ccc1Cl C(c1cccc(Cl)c1Cl)=CC(=O)NCc1nc(-c2cccc(OC)c2)oc1 C(C(C)(C(=O)NCC1CCCC(CO)C1)NC(C1CCC(F)(F)C1)=O)SC C1(CNC(C(C)C2CCCC2)=O)CN(C(c2cc(N)cc(O)c2)=O)CCCO1 Cn1nc(C(=O)OC(C)(C)C)cc1N.C1(C)(O)CNC(=O)N1CCO c1(C(N2CC(C)CC(NC(C(C)OCCC=C)=O)C2)=O)ccc2sc(C)nc2c1 CS(=O)(=O)c1ccc(C(N2CCCC(CCNC(C3CC(=O)N3)=O)C2)=O)o1 n1(CC2CC(OCC(=O)NC3C(C)COC3)C2)cccnc1=O c1(C(=O)NC(C)C(C)NC(=O)CCC2CC2(Cl)Cl)ccc(-c2ccco2)o1 N1(C(c2c(C)con2)=O)CC2CC1CN(C(=O)Cc1c(F)cc(F)cc1F)C2 C(=O)(C(C)C(=O)NCC#CC(=O)N(C1CCCC1(F)F)C)OC c1(C(N2C(CNC(CCC#C)=O)CC3CC32)=O)n[nH]c2c1CCCC2 C(=O)(C(C)(C)n1cnc(C)c1)NCC(C1CCCC1)NC(C(C)=C1CCC1)=O CCC(C)(CCNC(c1cc(C)n(CC)n1)=O)NC(=O)Cc1cncn1C1CC1 S(=O)(=O)(c1cccs1)N(C(C1(c2ccccc2)C(C)C1)=O)CC1CC1 c1(COC)ccc(C(N2CC(CNC(=O)C(C)SC3CCC(=O)N3)(OC)C2)=O)s1 c1(C(N2CC(SC)C(NC(=O)C(C)(C)C(C)C)C2)=O)ccc(C#N)cc1C c1(SCC(=O)NCC2CC2NC(c2cncc(O)c2Cl)=O)nc2ccccc2s1 c1(C(C(=O)NCCSC)NC(=O)CC2CC=CC2)cccc(C(C)(C)C)c1 C1(C)(CC(N2CC(F)(C(=O)OC)C2)=O)CCN(C(=O)CCOC(C)C)C1 C1(C(=O)NC(CNC(C2CCC(C)S2)=O)(C)C)COCCOC1 Nc1c(C(=O)NCC2(O)CCCN(C(c3cc(F)n[nH]3)=O)C2)ccc(Cl)c1O S(=O)(=O)(c1ccc2oc(=O)c3ccccc3c2c1)NC1C=CC(OC)C1(C)C c1(NCC2(CCO)CCC2)ccnc(N2CC3C(Br)C3C2)n1 c1(C(=O)NCC(C)NC(C(C)NC(CC)=O)=O)ncc(Cl)n1C c1(N(C(=O)Cn2ccc(COC)n2)CC)ccc(CN2CCS(=O)CC2)cc1 C(C(CC1CC1)C(=O)NC1CC(=O)N(CC2CC2)C1)NC(c1c(C)c[nH]c1)=O N1(C(COCCC)=O)CCCCC1C(C)(C)CNC(=O)CCn1cnnn1 c1(C(=O)Nc2cc(C)c(NC(C3CC3C3CC3)=O)cc2)nncc2c1CCCC2 C1(NC(c2c(NC)scn2)=O)CC(C(=O)NCC(N2CCCCC2)=O)C12CCC2 C(=O)(CCC(CF)CF)N1CC(CNC(C(C)SC)=O)OCC1 c1(C(=O)NCc2onc(CC)n2)ccc(CNC(c2cc(OC)n[nH]2)=O)nc1 c1(C(=O)NC(C)CNC(=O)C(C)(C)Cc2cnn[nH]2)ccc(O)nc1Cl CCC(C#N)C(=O)NCC1CCC(CNC(C2CN(C3CCOC3)C2)=O)CC1 N1(C(c2c(C(CC)(C)C)cccc2)=O)CCC(NC(=O)CS(N)(=O)=O)C(O)C1 C(=O)(C(F)(F)CC(C)C)N(C(C)CNC(=O)C(C)Sc1ccc(F)cc1)CC C1(C(N(CC(C)(C)NC(C2(C)CC2(F)F)=O)C)=O)CCc2nccn2CC1 c1(C(N2CC(F)(CNC(c3c(CC)cco3)=O)C2)=O)cc2c(C)c(C)ccc2[nH]1 Cc1nn2ccccc2c1C(=O)NCc1nc(C(=O)Nc2ccnc(O)c2)sc1 C(=O)(C(F)CC(C)(C)NC(=O)C(CO)C(C)(C)C)NC(c1c(C)nc(C)[nH]1)C N1(C(C(CC#C)C2CC2)=O)CCC(NC(c2ncsc2C)=O)CC(C)(C)C1 CCC(C)(O)C(=O)NCC1CCOC1C Cc1ccc(N2CC(NC(=O)CC3COCCN3Cc3cscn3)CC2=O)cc1 C1(NC(CN(CCOC)C)=O)CN(C(=O)CC2CCCCO2)CC1CO N1(C(CC(CCC)O)=O)CCC(C2CC2)(NC(c2coc(-c3ccsc3)c2)=O)C1 S(=O)(=O)(c1cccc(N2CCC(C(C)C)C2)n1)NCc1ccc(OC)nc1 N1(C(=O)Cn2nnc(=O)[nH]2)CCOC2(CCN(C(C3(n4cncn4)CC3)=O)CC2)C1 C(=O)(CCC(=O)NN(C)C)N1C(C(N(C)CC2CC(=C)C2)=O)C=CCC1 C#CC1CCCC(NC(C2CN(C(=O)CCCc3cccs3)CC(C)O2)=O)C1 C1(NC(CNS(N)(=O)=O)=O)CC2(CCN(C(C34CC(O)C3C4)=O)CC2)C1 CCC(F)(F)C(=O)NCCC1CN(C(C2CC(N3CCCC3)C2)=O)C1 Nc1ccc(C(N2CC(CO)(NC(=O)CC3CC34CC4)C2)=O)c([N+](=O)[O-])c1 CCCC(C(=O)NC1CCC(NC(C2(CC(C)C)CC2)=O)CC1)C(C)C N1(CC2N(C(C(n3c(C)ccn3)C)=O)CC2)CC2C3CCC(C3)C2(C)C1 C(C(C)CC(=O)Oc1ccccc1C(=O)NC1CCCC(F)C1)OC N1(C(Cc2cc(C)no2)=O)CC(CNC(=O)CC23CC(C2)C3)OC2(CCC2)C1 c1(C(N2CC(NC(C3C(OCC)C3)=O)(CF)C2)=O)ccc(C(N)=O)nc1 C1(NC(C2C(CC)N(C(c3cc(C)c(CC)o3)=O)C2)=O)CC2(C1)CC(CO)C2 C1(NC(C2CC(OC)C2)=O)CC(C)CN(C(=O)Cn2ccc(C)cc2=O)C1 CC1CC(NC(=O)CC2C=CCC2)CN(C(=O)COc2ccc(O)cc2)C1 C(=O)(C1=C(Cl)CCC1)N1CCC(OCCNC(c2cnc(C(C)OC)s2)=O)C1 C1(CN(CC(=O)N(C)CC2CCCC2)C)CCCN1C(C1(C2CC2)CC1)=O C1(C(=O)NC)CCN(C(=O)CCCc2cccc(C(N(CCCO)C)=O)c2)C1C C1(C(=O)NCC(CCC)NC(=O)Cn2ncc(=O)cc2C)CC(=O)NC(CC)C1 c1(C(=O)NC(CC(=O)NC(CC=C)(C)C)C2CC2)ccc2c[nH]nc2c1 N1(C(COCCCC)=O)CC(CNC(=O)CSc2nc(C)cc(C)n2)CCC1C C1(CNC(c2ccc(Cl)cc2)=O)CN(C(=O)C=C2CC2)CCO1.C12(CCCO1)CC2 C1(CNC(C2CCN(C(C3(C)CCC4CC4C3)=O)C2)=O)CCn2ncnc2C1 N1(CC(C)C)CCN(C(C2C(NC(=O)CCc3ccn(C)c3)C2(C)C)=O)CC1 C1(N(CC(C)C)C(C2CC=CCC2)=O)CCN(C(=O)C(C)N2CCCC2)CC1 C(=O)(CS(=O)c1ccc(Cl)cc1)NC1CN(C(Cc2cn(CC)nn2)=O)C1 C1(COC)C=CCCN1C(=O)CC1C(NC(C2(SC)CC2)=O)CC1O C(=O)(C(C)CC(C)CC(C)C)N1C(CC)CN(C(c2oc(SC)cc2C)=O)CC1 c1(CN(CC(=O)OC)CCN(C(c2coc(Cl)c2)=O)C2CC2)ccccc1 c1(C(N(C)CCNC(c2csc(Cl)c2)=O)=O)cccc(C2CNC(=O)C2)c1 c1(C(N2CC(CC(=O)NCC3CCNC(=O)C3)OCC2)=O)ccc(Cl)c(F)c1 CCC(C#N)(CC)C(=O)N1CCC(NC(=O)C(C)C2CCOC2)CC1 Cc1ccc(F)cc1CNC(=O)CC1CCN(C(c2cccc[n+]2[O-])=O)C1 C1(C(C)C)CC2(C1)CN(C(c1cc(Cl)cs1)=O)C2.C12CCCCC1(C)NC2=O Cc1nc(C(=O)NC(C2CCCC2)CNC(=O)CC2CN(C)C2)cs1 Cc1nc2cccc(C(=O)NC3(C(F)F)CC(NC(C4CCS(=O)(=O)C4)=O)C3)n2n1 c1(C(=O)NCC2CC(OC)CN2C(=O)COC(F)(F)F)cnc2n1C(C)CCC2 C#Cc1cnc(C(N2CCN(C(c3cc(C)co3)=O)C(CC)C2)=O)c(C)c1 n1(CCNC(C2C(CNC(C=CC(C)(C)SC)=O)CCO2)=O)nc(C)c(Cl)c1C C(=O)(C1=COCCC1)NC(C)CCCCNC(=O)CS(C)(=O)=O C(=O)(CC(C)C(F)(F)F)NCCC1(C(N(C(CC)C2CC2)C)=O)CCC1 C(C)(C(=O)NNC(=O)c1ccccc1S(=O)(=O)N1CCCC1)OC CC1CC(CNC(c2n[nH]c3c2COC3)=O)CN(C(C2CC2Cl)=O)C1 C(CCC(C(=O)N(Cc1ccco1)OC)NC(=O)CCN(C)CCO)OC Cc1ccc([N+](=O)[O-])c(NCC23CC(CNC(=O)C=CC4CCC4)(CO2)C3)c1 C1(CN(C(CCCOC(C#C)=O)=O)C)CC(F)CN1C(C1CCOC1CC)=O N1(C(C(C)C)=O)CC2(CCOCC2)CC1CNC(c1ccn2nccc2n1)=O CC1C(NC(=O)CCc2ccc(Cl)s2)CCN1C(=O)CC1(CO)CC1 N#Cc1ccc(CC(=O)NCc2cn(CC3CC(C(N)=O)=NO3)nn2)cc1F N1(C(CCC(C)OCC)=O)C2CC1CN(C(C1C3COCC13)=O)C2 c1(C(N2CCC(O)(CNC(=O)Cc3cnsc3)CC2)=O)coc2cc(O)ccc12 C1(NC(C(C)(C)C2CCOC2)=O)CN(C(c2cccnc2O)=O)CCC1O c1(NC2C=CC(NC(=O)OC(C)(C)C)CC2)cc(=O)c2ccccc2[nH]1 c1(C(=O)NCC2(O)COC2)ncn2cccc(C3=CCSCC3)c12 CC(C)C(C(=O)NCC(=O)NCc1ncc(CO)s1)Sc1ccccc1 C1(CNC(=O)CNC(N2CCCC2)=O)CC2COCC2N1C(c1cccnc1)=O Cc1noc(C(N2CC(F)(C(N3CC(CCN(C)C)C3)=O)C2)=O)n1 Cc1c(C(C)NC(CCCC#N)c2nnnn2CC2CCOCC2)cnn1C C12(CC)CN(C(=O)CCNC(=O)C(N)=O)C(CNC(=O)Cc3cccs3)(C1)C2 N1(C(COCC)=O)CC2C(C1C(N1CCOC(C#N)C1)=O)C2(C)C Cc1cccc(C(=O)NC2CC=C(C(=O)NC34CC(C3)C4)C2)c1N C1(N(C)C(C2CS(=O)(=O)C2)=O)CCN(C(=O)CC2CC2C(F)(F)F)CC1 c1(C(=O)NC(C2(O)CCN(c3nccc(C#N)n3)C2)C)cnc2[nH]cncc1-2 C(=O)(C(C)C(F)(F)F)NCC(CNC(CCN(CCCCC)C(C)C)=O)(C)O C(CCF)(C(=O)NCCC1(C)CCOCC1)NC(CC1(OCC)CCC1)=O c1(OC)cc(OC)c(C(=O)NC(C)CNC(=O)C(O)C(C)(C)C)cc1N Cc1cc2c[nH]nc2c(C(N2CCC(NC(C3CCCOCC3)=O)C2)=O)c1N c1(C(=O)NCC(CNC(c2ccc(NC)c(F)c2)=O)(C)C)cncc2ccsc12 C1(C)(C(N2CCC(NC(C(COC)O)=O)C(O)C2)=O)CCC(C)(C)CC1 N1(C(c2n(CC)cc(Cl)c2)=O)CC(CNC(c2cnc(C)s2)=O)CC(C)C1 c1(NCC2CCCN(C(C(C=C)NC(=O)OC(C)(C)C)=O)C2)cc(Cl)ncc1Br C(=O)(N=c1cc(C(F)(F)F)[nH][nH]1)C1N(C(C(C)(C)OC)=O)C2C(C1)C2 C1(NC(CSC)=O)CC2CN(C(=O)Cc3cccc(OC(C)C)c3)CC2C1 C1(C(N2C(CN(C(=O)C=CCO)CC)CCC2)=O)C(F)(F)C12CCC2 n1(C(C)C)ccc2c(C(=O)OCC(c3ccc(F)nc3)=O)cccc12 Cc1cc(C(=O)NC(C)C(C)NC(=O)C(=O)Nc2ncc[nH]2)n(C2CC2)n1 C1(C(=O)NC2CCC(NC(Cc3ncc(C)o3)=O)CC2)CCC(C)(C)CC1 N1(C(=O)Cn2ccnn2)CCC2C(CCCN2c2ncc(F)cn2)C1 C1(OC)(CNC(c2cc(C)cnc2C)=O)CCN(C(c2c(C)csc2Cl)=O)CC1 C1(C(C)(C)C)CC(NCc2nnc(CSc3ccccc3)o2)CC(C(C)(C)C)C1 C(=O)(C(CNC(=O)C(F)CC1CCCC1)OC)OCC1N(CC)CC1 N1(C(C(C)CC2CCC2)=O)CCOCC(CNC(c2cccc(C3CC3)n2)=O)C1 C(C)(C)(CC(=O)N(CCCCN(C)C)C)NC(C1C(CC)CCO1)=O O=C(C1=CCSC1)NCCCCCNC(C1CC(=O)N(c2nccs2)C1)=O c1(CC)cc(Sc2cccc(C)c2)ccc1CC(C(=O)O)n1ccnc1 Cc1ccc(C(=O)NC(C)CNC(=O)CC2CCC(=O)N2C)c2c1NCCC2 Cc1cc(Cl)c(C(N2CCCC(CCNC(=O)C=Cc3cn(C)cn3)C2)=O)cn1 CCC(CC)(CO)C(=O)N1CC2CCC2(NC(=O)Cc2ccc(Cl)c(C)c2)C1 N1(Cc2c(OC)cc(Br)cc2C)CCn2nc(CNC(=O)OC)cc2C1 CC(C)CS(=O)(=O)CCC(=O)NCCOCCNC(c1ccnc2ccsc12)=O N1(C(C2C(C3C(C)C3)C2)=O)CC2CC(NC(c3cc(C(C)(C)C)no3)=O)CC1C2 c1(C(N(C2CCCN(C(C(N3CC(C)C3)C)=O)C2)C)=O)cnc2[nH]c(O)nc2c1 C(CC(=O)NCc1ccc(F)nc1C)(C(C)OC)NC(C1(CSC)CC1)=O c1(CC)csc(CC(=O)N(C2CCN(C(=O)CCc3ccccc3)C2)C)n1 C1(C(N(C)CC2CCN(C(c3c(C)cn(C)c3)=O)CC2)=O)COCC(C)(C)O1 N1(C(Cc2cc(C)no2)=O)CCCC1(C)C(=O)NCC1CCCC1N(C)C c1(C(N(CC(CC)NC(=O)Cc2nocc2C)C)=O)conc1C C=CCCC(C)(C)C(=O)NCc1ccnc(C(=O)NCc2ccc(Cl)nc2)c1 N1(C(c2c(C)cc(Cl)cc2)=O)CCC2CCCC(C1)N2C(=O)CNS(N)(=O)=O Cc1cccn2cc(CC(N3CCN(C(=O)CCOC4CC4)CC(O)C3)C=O)nc12 n1(CCC(=O)NCC(C2CC2)NC(c2cc(COC)[nH]n2)=O)cc([N+](=O)[O-])cn1 C1(C(N2CCC(COCC)C2)=O)CCCC(NC(=O)CCC2(C#N)CCC2)C1 CS(=O)(=O)c1cncc(-c2cncnc2C(=O)NCC=CC2CC2)c1 C=CCCCCCCCC(=O)NC1(CN(C)C(c2ccnc(C)c2C)=O)CC1 C1(NC(c2cc3n(n2)CCO3)=O)CC1C1CCCN(C(C2(O)CCC2)=O)C1 c1(C(=O)OC)ccccc1C(=O)N(C1CCN(C(=O)CSC(C)C)CC1)C Cc1cn2nc(C(=O)NC3COCCN(C(C4(CO)COC4)=O)C3)cc(C)c2n1 c1(C(N2C(CCCNC(c3cnc(C)o3)=O)CCC2)=O)nccn2c(C)nnc12 c12cc(cc3c1OCCO3)C=CC(=O)N1CCN(CC(OC)C1)C2=O.CON Cc1cccc2[nH]cc(C(=O)NC3CC(F)CN(C(C4CC=CCC4)=O)C3)c12 C(C(CC(F)(F)F)NC(=O)CN1CCCC1C)NC(C1(OC)CCOCC1)=O c1(CN2CCC(O)(C(=O)NCCCCCCCC)C2)ccc2c(c1)CCO2 CCC(CC(=O)N(C1CN(C(C2CNC(=O)CC2C(F)(F)F)=O)C1)C)C(C)C Cc1cc(F)ncc1CNC(=O)C(C)(C)NC(=O)C=CC1CCCN1C C(=O)(C(CCC)N(C)C)NCC=CC1C(C(=O)NCC=CCCC)C1(C)C C=C(Cl)CC(C(=O)N1CC(C)C1(C)C)NC(=O)CC(C)(C)SC N1(C(C(CSCC)NC(=O)CCCCN(C)C)=O)CCC=CC1CC c1(OC)ccc(CO)cc1C(=O)NCC1CC(NC(C2CC3C=CC2CC3)=O)C1 C1(CNC(c2cn(C(C)(C)C)nc2)=O)C2CN(C(=O)Cn3cccc3)CC12 c1(CCC(N2CC(C)C(NC(=O)C(F)=C3CCC3)CC2)=O)nc2ccccc2o1 C=C1CC(C(=O)NCC(C)(C)C2CCC2)(CNC(=O)CC2(OC)CC2)C1 N1(C(C(CNC(C2C3CCC(F)C23)=O)O)=O)CCC12CCOCC2 C1(C)(C(N(C2(C(=O)O)CC2(C)C)C)=O)CCCCO1 c1(CN(C(=O)CC2CCCCN2)C(C2CCC2)C)cccc(F)c1 c1(C(=O)NC2CN(C(C3CC4(CSC4)C3)=O)CC2C(F)F)cc(=O)cc(Cl)[nH]1 c1(C(=O)NC2(CNC(C(CC)(C)C(N)=O)=O)CCCC2)ccc2c(c1)CCN2C CN1CC(C(=O)NCC2CCN(C(=O)COC3COC3)C2(C)C)CCC1=O S(=O)(=O)(c1ccc(N(C)Cc2ccno2)c(Br)c1)NCC1(C)C(C)OCC1 C(CCCCC(=O)N1CCC(C)(C(=O)OC)C1)N(C(=O)COC1(C)CCC1)C N1(C(c2n(C)nc(C)c2F)=O)C2CCCC1CC(NC(=O)C1=NNC(=O)CC1)C2 CC1CCC(C)N1C(c1cc(NC(c2cccnc2I)=O)cn1C)=O Cc1ncc(C(=O)NC(C(=O)NCc2nnc(C)o2)C2CCCC2)c(C)n1 N1(C(C2(C(C)NC(C3CC34CCOC4)=O)CC2)=O)CCC2(C1)CN(C)C2 CC1CCC(C)(C=CC(=O)NC2CCC2)C1(C)C.C12CN(CCC13CCC3)C2 Cc1sc2ccccc2c1CNC(=O)Nc1ccc(=O)n2c1CCC2 Cc1cc(C)c(C(N2CC(NC(=O)C(=O)NCC3CC3)CC(O)C2)=O)c(N)c1 c1(OC)ccc(S(=O)(=O)N2CCN(CC(N3CCCOC(C)C3)=O)CC2)c(F)c1 N1(C(C(C)SCCCC)=O)C2CCC(C2)C1CC(=O)N(C(C)CC1CCCC1)CC c1(C(N(C(c2c(C)c[nH]n2)=O)C)=O)cc(C(N)=O)ccc1[N+](=O)[O-].C12(CC1)CN2 C12(CNC(CC(N3CCCCCC3)C)=O)CC(CNC(=O)C=C3CC3)(CO1)C2 N1(C(c2c(Cl)cn(CCC)n2)=O)CC2CC(NC(=O)Cc3csc(C)n3)C1C2 c1(NC(C)C)ccc(C(=O)NCC2(NC(=O)CSCCC#N)CCOC2)cc1 c1(C(=O)NC(C(=O)NCCN(C(C)=O)CC)COC(C)(C)C)c(Br)c(C)nn1C Cc1ccc(C(=O)NC23CCCC2CN(C(=O)C2=NOC(C)(C)C2)C3)c(O)c1C N1(C(C(CC)CC(C)C)=O)CC2(C1)CN(C(=O)C=Cc1cccnc1C)CCO2 Cc1cccc(CC(N2CCC(C)(CNC(C3(C#N)CCCO3)=O)C2)=O)c1 Cc1c(CC(=O)NCC(CC(=O)NCCc2ccccc2)C2CCC2)ncn1C C1(CC)CC(CNC(=O)CCSCc2ccccc2)N(C(=O)C2=CCOC2)C1 c1(OC)cc(C(=O)NCC2CN(C(c3snnc3C)=O)CCO2)cc(Cl)c1 Cc1ccc(C(N)=O)cc1C(=O)NCC1CC(O)CN1C(=O)CCC1CC1(F)F C(C(C)CC(F)(F)F)NC(C1(C)N(C(CCCOC)=O)CC=C1)=O CCC(C)(C#N)C(=O)N(C)CC1(O)CN(C(c2ccc(CC(C)C)s2)=O)C1 N1(C(CCOCCOC)=O)CC2CC(NC(=O)CSC3CCCCO3)C2C1 C12(NC(C3CCCC3)=O)CCCN(C(c3coc(Br)c3)=O)CC1C2 C1(CNC(C2CC(OC)C2)=O)CC2(CC2)CN1C(=O)CCCN(C)C c1(CC(C)NC(c2cnc(COC)s2)=O)ccc(CNC(=O)CC(C)(C)O)cc1 c1(C2C(F)(C(=O)NC3C(NC(c4cnco4)=O)C3)C2)ccccc1 C(CC(C)C)(C(=O)N1CC(N(C(=O)CC=Cc2ccc(F)cc2)C)C1)NC(C)=O C1(CNC(c2nn(CC)c(C3CC3)c2)=O)CN(C(C2CSCCS2)=O)C(C)(C)C1 C(=O)(C(O)CC(F)(F)F)NC1CC2(C(NC(c3ncc(CC)cn3)=O)C2)C1 C(=O)(C(CNC(C1(NC(C2CC(C)=NO2)=O)CC1(C)C)=O)OC)OC N1(C(=O)NC(CC)CC)CCCC2(COc3ccccc32)C1 C1(CCC)CCCC1(c1nnnn1CCSC)NCC(S(C)(=O)=O)C1CC1.O(C)CC Cc1cc(O)ncc1C(=O)NC1CN(C(C2CC2C)=O)CCC1F C1(N=[N+]=[N-])(C(=O)NCC(N2CCC(C(=O)OC)CC2)=O)CCNCC1 C#CCC(CC(F)F)C(=O)N1CCC(C(=O)NCC2(C(O)CO)CC2)C(O)C1 C=CCC(C(=O)NCC(O)CN(C)C)NC(C1(C)COC1)=O c1(C(N2CCC(F)(CNC(CC(C)F)=O)C2)=O)cc(Cl)cc(Cl)c1 C1(C(=O)NC2CCN(C)CC2C)(CC)CCCN(C(C2CC3C=CC2CC3)=O)C1 c1(C(=O)NCC2C(C)CN(C(=O)CN3CCC(C)(O)C3)C2)ccc(C#N)c(O)c1 N1(C(c2cc(C)cc(Cl)c2)=O)CC2OCC(NC(=O)CS(=O)(=O)C(C)C)C2C1 C(=O)(C#CC1(C)CCCO1)NCCC(C)NC(=O)C1CCc2c[nH]nc21 N1(C(C2C3(CCN(C(C(C)(C)OC)=O)C3)C2)=O)CC(C)(C2CCC2)C1 N1(CC(=O)OCCc2c(OC)ccc(Cl)c2)C(=O)NC2(CCC(C)C2)C1=O Cc1c(C(N2CC=CC(C)C2)=O)cccc1N1C(=O)NC(C)C1=O C(N=c1ncn(Cc2ccccc2OC(F)F)[nH]1)C1C(C)CCCC1 Cc1c(C(=O)NCCN(C(=O)CC(C)CF)C)oc2c1ccc1ccccc21 c1(C(=O)NCCC2CN(C(c3c(C)nc(O)[nH]3)=O)C2)ccc([N+](=O)[O-])s1 N1(C(C2CC(=C)C2)=O)CCCC1C(C)NC(=O)C(C1CCOCC1)F c1(C(CC)C)nc(NCCOC2CCN(C(c3ccn(CC)n3)=O)C2)cc(C)n1 c1(C(=O)NCC2C(NC(C(c3ccccn3)C)=O)CCC2)cnc(Cl)c(Cl)c1 N1(CC)CCC(N2CCC(CNC(=O)C(C)Cc3ccco3)CC2)C1=O Cc1ncc([N+](=O)[O-])n1CC(=O)NC(C)(C)CNC(=O)C(C1CCOCC1)F C(=O)(CCC=CC)N1CC(CCCCNC(CSCCCC)=O)C1 N1(C2CCN(C(C(C)(C)SC(F)(F)F)=O)C2)CCN(C(c2cc(O)no2)=O)CC1 n1(CC)ncc(Cl)c1C(=O)NCC(CNC(=O)CCC1CC1C)OC c1(C(=O)NC2CN(C(C3(C)C(C)OCC3)=O)C2)ccc(N)cc1F Cc1nn2cc(C(=O)NCCCCCN(C)C(c3ccc(C(N)=O)[nH]3)=O)nc2s1 CN1CC(C(N2CC(CNC(c3ccoc3C(F)(F)F)=O)C2)=O)OCCC1=O C1(NC(c2n(CC)ncc2Cl)=O)CCCN(C(C2CC23CC(C)(C)C3)=O)CC1 c1(C(=O)NC2(C)CCN(C(c3ccc(C(C)=O)[nH]3)=O)C2)cncc2cccnc12 C1(C(N(CC(O)CNC(C2CC2Cl)=O)CC)=O)CCCCC1COC Cc1nc(C2CC2)sc1CC(=O)NCC(C1CC1)NC(c1cc(C(N)=O)cs1)=O c1(CC(=O)NCC2(OC)CN(C(C3(Br)CC3)=O)C2)ccc(C)cc1Cl N1(C(CNC(=O)C2CC2)=O)CCC(CCNC(c2cn[nH]c2)=O)CC1 CN1C(=O)OCC1C(N1CCC1CNC(c1coc(-c2cccnc2)n1)=O)=O N1(CC(C)(C)N(c2ccccc2Cl)CC)CCCOC(CN)C1 C1(CC)CN(C(=O)C(CCC2CCC2)NC(C2CC(F)C2)=O)CCO1 C(CCN=c1[nH]c2c(c(=NCC(C)(C)n3cccn3)[nH]1)CSC2)OC=C C1(F)(CNC(C(COC)OC)=O)CCN(C(=O)CCCCc2cnn[nH]2)CC1 c1(C(N(CCNC(=O)CNc2nccs2)CC)=O)cc(F)cc(N)c1N CC1=C(C)CC(C(N2CCC(C)(C)C2C(=O)NC2CC3C=CC2C3)=O)CC1 c1(C(N2C(CCNC(C3C(C)C3)=O)CSCC2)=O)cc(Br)cc(F)c1F CC(O)C(C)(C)NC(=O)C(C1CCN(C(=O)C(F)C2CCCC2)C1)F C(=O)(C(C)(C)NC(C1C(CN)C1(F)F)=O)OC(C)C(=O)N(S(C)(=O)=O)CCO N1(C(CC2CC(OC)C2(C)C)=O)CC2CCC(C1)N2C(=O)C(C)(C)N1CCCC1 C1(NC(=O)Cc2ccc3ocnc3c2)CC2CCCCCC2C1 CC(C)CC(Cn1cc(-c2ccccc2)nn1)NC(c1ccsn1)=O C1(CNC(CC(CC)C2CCC2)=O)CC12CCN(C(C1CN(C(N)=O)C1)=O)CC2 C1(C(=O)NCCCC(=O)OC(C)(C)C)CC12CCN(C(C1CC3(CC3)C1)=O)CC2 C12(NC(c3cnn4c3CCC4)=O)CCCC1CN(C(c1cc(Cl)ns1)=O)C2 c1(C(N2C(CNC(=O)CC3CCC(O)C3)CCC2)=O)cc(Cl)c2c(c1)OCCO2 C1(NC(=O)Cn2cc([N+](=O)[O-])cn2)CC2CCC(C1)N2C1CCN(C2CC2)C1=O c1(C(C(=O)NC2C(n3cc(CN(CC)CC)nn3)CCC2)(F)F)ccc(C)cn1 c1(C(N(CC(CNC(C(c2ccccc2)SC)=O)O)C)=O)cccc2c1CCO2 N1(C(CCNC(=O)OC)=O)CCC2CCN(C(c3ccc(C(N)=O)o3)=O)C2C1 N1(C(=O)NC(C)Cn2ncc3ccccc23)CCOCC12CCCCC2 C(=O)(C1=CC2C=CC(C1)C2)NCCCOCCNC(C(C(CC)CC)C)=O Cc1cc(C(=O)NC(CNC(C2CCCC2(C)C)=O)CO)nn1CCO N1(C(=O)Cc2c[nH]nc2O)CCN(C(=O)C=Cc2ccoc2)C(C(F)F)C1 c1(C(N2CC3CC2CS3=O)C(=O)NCCC2CC2)ccc(Br)c(Cl)c1F C(N(C)N1CCc2sccc2C1)c1ccc(OCc2ccc(CCC)cc2)cc1 c1(C(=O)NCC2(CNC(=O)Cn3cnccc3=O)CCCC2)cc(Cl)ncc1Cl c1(C(N2CCN(C(=O)OC)CC2)C(=O)NC(c2nccs2)CC)ccc(C)cn1 Cc1noc(C(F)F)c1C(N1CCC1CNC(=O)C=CCn1cncn1)=O n1(CC(N2CCC(N(C(=O)COC3COC3)C)C2)=O)nc2c(n1)CCCC2 c1(CN2CCN(CC(N3CC(O)CC3CO)=O)CC2)cc(Cl)cnc1Br C(=O)(C1=CC2CCCC12)N(C)Cc1cccc(CNC(C2(CC)CCC2)=O)c1 C#CCC(C)C(=O)N1CCCC1C(C)NC(c1cnn(C(C)C)c1Br)=O C(=O)(C(O)CCSC)NC(C12CCC(CC1)C2)C(=O)NCc1cn(CC=C)nn1 CC(C)(C)C(O)C(=O)N1CCCCC1CNC(C1C2CNC(=O)C12)=O CCCC(C)(C)CC(=O)NC1CC2(C1)CC2C(=O)N(C)Cc1cn(C)nn1 Cc1ccccc1C(=O)NCCOCCCN(C)C(c1ncc[nH]c1=O)=O C1(C(=O)Nc2ccc(C(=O)NCCC(F)(F)F)nc2)CCc2nc[nH]c2C1 c1(C(=O)N(C2CCN(C(=O)C(C)(C)F)C2)C)ccccc1F.CO C1(CC#C)(C(=O)NC2C=CCN(C(C3CCC4(CC4)C3)=O)C2)CCCOC1 N1(C(C2C(CC)CCC2)=O)CCCC(NC(c2ccc(O)c(C)c2)=O)CC1 C=CC(C)(C)CC(=O)N1CCC(CC(=O)N(CC(C(C)C)OC)C)C1 CC1CC(C)(C)CCC1NC(=O)CCC1(C)CN(C(c2cc(Cl)no2)=O)C1 C(CCC(C)C)(C(=O)N1CCCC1CN(C)C(C1(C(F)F)CCC1)=O)NC(C)=O c1(CCCC)cccc(-n2cc(CC3CCN(C(=O)COCCO)C3)nn2)c1 N1(c2ncc(C(=O)NCC(c3ncccc3F)C)s2)CCN(C)CC1 N1(C(COCCNC(c2cccc(OC)c2)=O)=O)CCN(C)C(=O)C1 CC1CCCn2ncc(C(=O)NCC3(C4CC4)CCN(C(=O)C=CBr)C3)c21 N1(C(CC(C(=C)C)OCC)=O)CC2CCC(NC(c3cnoc3C)=O)(C2)C1 Nc1ccc2oc(C(N3CCC(CO)C(NC(=O)C4=CCOCC4)C3)=O)cc2c1 C12(CNC(C=Cc3c(C)n[nH]c3)=O)CCC1CCN2C(c1csc2cncn12)=O CCCC(C)(CC)C(=O)N1CC(NC(c2cccc(C#N)c2C)=O)CC(C)(C)C1 C(C)(C)(CC(F)C(=O)NCc1n[nH]c2c1CCC2)NC(CCNC(=O)NC)=O C1(O)(C(C(=O)NCC(CNC(C2C(C)(CC)C2)=O)C)(F)F)CCOCC1 C1(N(C(=O)CC2CCOC2)C)CCCN(C(C2(C)CC2(Cl)Cl)=O)CC1 C(=O)(C1CCc2cc(F)ccc21)N(CC(C1CCCCC1)OC)C CC(=O)CCCC(C)C(=O)NC1CCCN(C(c2nccnc2C)=O)C1C CC1CCCC1(C(=O)NCCN1CCCCC1=O)NC(=O)CCC(C)N(C)C Cc1cc(C(N2CCC(F)(CNC(=O)C(C)S(C)(=O)=O)C2)=O)cc(C)c1N C(C(CNC(c1sccc1C(=O)OC)=O)C(F)(F)F)NC(CCCC)=O C1(NC(Cc2ccc(C)s2)=O)CCC(C)N(C(c2sc(C)cc2C)=O)C1 N1(C(C2CCCN(C(C3(C#C)CCCC3)=O)CC2)=O)CCC(C)C2(CCC2)C1 C1(NC(=O)C=Cc2ccco2)COC2(CCCN(C(=O)NCc3ccccc3)C2)C1 C(CN=C(NCc1ccnn1C)NCC1CCCN(C(C)C)C1)c1c(C)cn(C)n1 C1(C#N)(C(c2n(CCC=C)nnn2)NCCN(C)C(=O)OC)CCOCC1 c1(C(N(CCCNC(=O)C(F)CC2CC2)C2CC2)=O)nccn2nccc12 C1(N(C(CSCCOC)=O)C)CCC(NC(=O)Cn2nnc(C(C)(C)C)n2)C1 CC1=C(C(=O)N2CCN(C(=O)C=CC(C)C)CC(C)(C)C2)CCC(C)(C)C1 c1(CC)cn2c(C(=O)NC(C)C(C(C)C)NC(C3COC(=O)O3)=O)cccc2n1 C1(C(N2CCC(CNC(C3(C(N)=O)CC3)=O)C23CC3)=O)CCC2(CCOCC2)O1 CC1(C)CCN(C(=O)Cc2cccnc2O)CC1CNC(c1cccc(=O)o1)=O Cc1cc2c(NC(C3(CNC(c4ccnc5ncnn45)=O)CC3)=O)cccc2o1 C(C)(CC(C)(C)CO)NC(CC(C)(C)n1cc(CCNC(COC)=O)nn1)=O c1(C(=O)NC(C2CCN(C(COC(C)C)=O)C2)(C)C)cc(O)ccc1Br C1(C(=O)NCCCOCC)CCCC12CCN(C(c1cscn1)=O)C2 C=CCC(C(=O)N1CC(SCC=CC(=O)NOC2CC2)C1)OC Cc1[nH]nc2cc(C(N3CC(O)C(O)C3CNC(c3ccn(C)n3)=O)=O)ccc12 CC1CN(C(C2CC2(C)C)=O)CCC1C(=O)NC(C)(C)C(O)C(F)F C=CCCC(CC(C)C)C(=O)N1CCN(C(=O)CC2CCN(C)CC2)CC1CO N1(C(c2n(CC)c(O)nc2)=O)CCN(C(c2ccc(N)cc2F)=O)C2CC12 c1(C(=O)NOC(C2(CN3CCC3c3ccccn3)CCO2)=O)ccccc1 C(=O)(CCC(C)(C)C)NC(c1cccc(OC)c1)CNC(=O)C(C)NC=O N1(C(C2(CC)CCCC2)=O)CCC(C(F)F)(CNC(=O)C=C(C)C2CC2)C1 c1(C(=O)NC2CN(C(CCC)=O)CC2c2ccccc2)nc(C)c(C)nc1C c1(C(N2CC(NC(=O)COCCCF)C2)=O)nc(C2CCC2)ncc1Br c1(C(N2CCC(OCCNC(Cc3c(C)non3)=O)C2)=O)ccc(P(C)(C)=O)cc1 CC(=O)CCN=C(NCC(C)(C)CCN(C)C)N1CCc2cccc(Cl)c2C1 c1(CC)nn(C)c(Cl)c1C(=O)NCCC1CCCN(C(C2(C)CC=CCC2)=O)C1 C(=O)(C(C)CC(C)(F)F)NCC(CC)(CC)NC(=O)C=Cc1ncc(C)[nH]1 CC(C(C)C(=O)NC1CC(=C2CC2)C1)NC(=O)Cn1ncn(C)c1=O CC1(C)CN(CC(=O)NCC2(C(=O)NCC(CC3CC3)CO)CCC2)C1 CC(C)C(CC(=O)N(C1CCC2(C1)CC2(F)F)C)C(=O)OCC(C)(C)C CN=c1ccc(C(=O)NC2CCCC2NC(C2CCCN2C2CCCC2)=O)c[nH]1 Cc1nc2n(n1)CCN(C(=O)C(C(C)C)NC(=O)C1=C(Cl)CCOC1)C2 C(=O)(C(C)C(O)CC)N(C)Cc1ccc(CNC(c2onc(COC)n2)=O)cc1 c1(C(N(c2ccccc2)CCNC(CN(C(C)=O)C)=O)=O)cc(C)nc(O)n1 N1(C(c2c(C)cccn2)=O)CCCC2(NC(C3CCCCN3C)=O)CC2C1 N1(C(c2csc(C(F)F)n2)C(=O)NCCC2CC2)CCN(c2cncnc2)CC1 C12(CNC(CC3C(C)C3(F)F)=O)COCCN1CCN(C(=O)Cc1ccns1)C2 C#CCCCC(=O)N1CCC(CCOC)(NC(=O)C(CO)OC)C1 C1(NC(c2cc(C)n(C)c2)=O)CC2(CCN(c3cc(-n4cncn4)ncn3)CC2)C1 C(C(CNC(C1(C(C)NC(=O)CC2CC(C)=NO2)CC1)=O)CO)OC C12(C(=O)NCC(C)(F)CNC(c3cccnc3S)=O)CCOC1CCOC2 O=C(C1CCCn2cnnc21)NCC1CCN1C(=O)CC1OCCCO1 c1(C(N2C(C(C)NC(C3(CC)CC3)=O)CCC2)=O)cncc(C(F)F)c1 C(C1OCc2ccccc21)NC(=NCCC)NCC1(OC(C)C)CCSCC1 N1(C(CC(c2cccc(F)c2)C)=O)CCN(C(C23COC(CF)(C2)C3)=O)C(C)C1 CC1CN(C(c2ccccc2OC2CC2)=O)CCN1C(=O)C#CC1(CC#N)CC1 c1(C(=O)NCCS(C)(=O)=O)n[nH]c2c1CN(C(c1cc[nH]n1)=O)C2 CC1(C(N2CCC(CCNC(=O)Cn3nccn3)C2)=O)CCCO1 Cc1nc2cc(C(N3CC=CC(NC(C4CC(=O)NC(=O)C4)=O)C3)=O)cnc2[nH]1 C1(CC)CC(=O)N2CC=CC2(C)C(=O)N1.C1(C2N(CCC)CC2)CCCCC1 N1(C(c2[nH]cc(C)c2)=O)CCC(CNC(=O)CCc2cc(C)nn2C)C(O)C1 CCC(CC(=O)NCC(N1CCN(C(C2CC(OC)C2)=O)CC1)=O)C(C)C CC1CCC(C)(C(N2CC(NC(=O)C=CC3(C)COC3)C(C)C2)=O)C1(C)C c1(C(N(C(CCSC)C)C)=O)csc(CNC(=O)OC(C)(C)C)n1 C(CC)(c1ccccc1)=CC(=O)NC(CC#C)C(=O)NCCC(C)N(C)C c1(C(=O)NC2C(NC(CCOCCCOC)=O)CCOC2)cc2sc(Cl)cc2[nH]1 c1(NCC(C(CC)C)O)ccc(S(=O)(=O)NCc2c(C)cc(C)cc2C)cc1Br C1(CCC)CN(C(=O)C(C)NC(=O)CCCC(C)C)CCN1C(c1cccs1)=O c1(OCCC(=O)NCC2CCCCN2C(=O)C(F)(F)C2CC2)ccc(F)cc1 N1(C(C=CCC)=O)CCN(C(=O)C(C)(C)C2CCC2)CC1C1CC1 C1(CNC(C(C=C=C)C)=O)CCCC2(CN(C(=O)C#CC(C)(C)O)C2)O1 N1(CCC)CCN(C(c2cscc2C)C(=O)NCCOCC2CC2)CC1 C1(OC)CC(CNC(C2(C(C)(C)O)CC2)=O)N(C(=O)C(C)CSC(F)(F)F)C1 C1(C(=O)NCC2CC(O)CN2C(=O)Cc2ccsc2Cl)CCC=CCCC1 c1(C(C)CNC(N2CCC(CC3CC3)C2)=O)cccc(Cl)c1F c1(NC(C2N(C(CC=C)=O)CC(O)C2)=O)ccc(C)c(Br)c1 CC1CCC(CNC(C2(C(F)F)CC2)=O)CN1C(=O)CCCn1c(O)nnc1O c1(C(N2C(CNC(CCC#C)=O)CC(C)(C)C2)=O)cc(C)cc(Cl)c1N CCC(CC)C(C)NC(=O)CC(=O)NCC(CSC)OC c1(C(=O)NC(COCC)C(=O)NCCc2noc(C)n2)cnc(O)c(C)c1 N1(C(C2(COC)COC2)=O)CCCCC1C(=O)Nc1cccc(C)n1 Cc1c(C(=O)N(CCCCCNC(C2CC2C2CCCC2)=O)C)sc2nccn12 S(=O)(=O)(c1ccccc1F)N1CCN(CCNC(c2cnc(C3CC3)[nH]2)=O)CC1 N1(CC(=O)N(CC(C)C)CCO)C(=O)NC2(CCc3ccccc32)C1=O.CC(C)CS CC(C)CC(C(=O)N1CCOC(CNC(c2cc(S(N)(=O)=O)c[nH]2)=O)C1)C(N)=O Cc1oc(C#N)cc1C(=O)NCCOC1CCN(C(=O)CC(C)CF)CC1 c1(CN(C(C(=O)NCC(CC)O)=O)CC)ccc(N2CCCC2=O)cc1.SCC CC(CC1CCC1)C(=O)NCC1CCOC1C(=O)NCC1C=CCC1 c1(SC)cc(C(N2CCC(C(C)NC(=O)CCC(N)=O)C2)=O)c(C)o1 C1(C(N2CCN(C(C3OCC(C)(C)C3)=O)CC2)=O)CC2CCC(C1)O2 C(CCC1CC1)(C(=O)N)OC.C1(C(F)C(=O)NCCSC(F)F)CC(SC)C1 c1(NC)cc(C(N2CCC2CNC(C2CC(C)=NO2)=O)=O)cc(C(F)(F)F)c1 CC1OCCC1(C)C(=O)NCC=CC(N1CC(CC23CC(C2)C3)C1)=O C1(NC(c2c(C)oc(C(C)C)n2)=O)CN(C(=O)CSc2cnn(C)c2)C(C)(C)C1 N1(C(c2nnn(CC)c2C)=O)CCC(CNC(c2cccc(=O)o2)=O)C(C)C1 c1(N(C2CCNCC23CC3)C(Cc2cc(C)on2)=O)cnc2ccc(F)cc2c1 C1(CC(=O)N(CCN(C(=O)C(CSC)N(C)C)CC)CC)CCCC12CC2 N1(C(CCCn2c(C)ncc2)=O)CC2CN(S(=O)(=O)C(Cl)(Cl)Cl)C2C1 C(=O)(C(CC1CC1)NC(=O)Cn1nccn1)NCC1(SCC)CC1 N1(C(C(C)NC(c2ccc(C)s2)=O)=O)CCC(C)N(C(=O)CC(C)C)CC1 c1(C(=O)NCC2CCN(C(=O)C(F)n3cccn3)C2)ccc2c(c1)CCCC2 C(CN(C)C)(CC(=O)N1CCCC(CC)C1)NC(C=CCN(C)CC)=O C1(C#N)(C(=O)NCc2c(C(=O)NCC(c3nc[nH]n3)C)c[nH]n2)CCCOC1 C1(OCC)CC(N(C)C)(C(N2CCOCC2(C)C)=O)C1(C)C N1(C(c2c(C)nn[nH]2)=O)CC(C)CN(C(=O)C(C2CCC(=O)N2)C)CC1C C12(C(=O)NCC(CC)NC(=O)CCn3ncn(C)c3=O)CC(C(F)(F)F)(CO1)C2 c1(C(=O)NC23C(CN(C(C4C(C=C)C4)=O)C2)C3)nnc(O)c2c1CCCC2 C1(C(N2CC(NC(c3ccc(-c4cn[nH]c4)cc3)=O)C2)=O)CN2CCCC1CC2 Cc1cc(C)c(C=CC(=O)NC2CCC2CNC(C2CCCO2)=O)cc1C N1(C(C2(CO)CCN(C(=O)Cc3ccccc3F)C2)=O)CC2(CCNC2=O)C1 CC1(C)CCC(C(N2CCC(CNC(=O)Cc3ccncc3Cl)C2)=O)C1 N1(C(c2cnc(C(C)C)o2)=O)CC(F)CC1CNC(c1cc(C2CC2)ns1)=O C(=O)(C(C)(C)C(F)F)NC(C)C(C)NC(=O)Cc1cccc(C(F)(F)F)c1 C1(C(=O)NCCNC(c2ccoc2)=O)C=CCN1C(=O)CCCn1ccnn1 C(=O)(N1OC2CCC1CC2)C1(COC)CN(C(=O)CCCCCF)C1 c1(C(=O)NC(CNC(=O)Cc2ccccc2F)CO)nnn2c1C(=O)NCC2 CC#CC1CCN(C(=O)C(C)(C2CCC2)NC(c2cnc(C)nc2)=O)C1 Cc1ncc(Cl)c(C(=O)NCC(C2CCCC2)NC(C23COCC(C2)OC3)=O)n1 C1(CNC(CP(C)(C)=O)=O)CN(C(C2CC(=O)NC(=O)C2)=O)C2CCN1C2 C1(C(=O)NC2CN(C(C3C(C)CC(C)O3)=O)CC(C)(C)C2)CCc2ccccc2O1 C1(NC(c2c(C)n[nH]c2C)=O)CCN(C(c2csc(C(N)=O)n2)=O)C(C2CC2)C1 C(CCC(=O)NCCNC1(NC(=O)CSc2n[nH]c(O)n2)CC1)SCC C1(C)(C(N(CCC(N2CCCCC(COC)C2)=O)C(C)C)=O)CC(=O)N(C)C1 Cc1[nH][nH]c(=N)c1C(=O)N(CCCCN(C(=O)CCCOc1ccccc1)C)C c1(OC)noc(C2CC2)c1C(=O)N(CC(O)CNC(c1cc(C(N)=O)co1)=O)C C(=O)(CCCCC(=O)NC1CC(C)(CNC(C2CC=CCC2)=O)C1)OC CC1OCCCC1C(N1CC(CC(C)(C)CNC(c2sccc2Cl)=O)C1)=O C(CCC(=O)NC1CC(CNC(C2CC2C(C)SCC)=O)C1)OCC Cc1ccc(C)c(C(N2CCCCC(C(=O)NCCCC(F)F)C2)=O)n1 c1(-c2c(C)ccc(OC3CCCC3)c2)ncnc2sc3ccccc3c12 N1(C(=O)CC(F)(F)C(F)F)CCN(C(c2ccc(Cl)cc2F)=O)C2CCCCC12 O=C1CCOC(C(N2CCCC(C(=O)NCCOc3ccncc3)C2)=O)C1 c1(NC(C2CCCN(C(c3c(CC)nco3)=O)C2)C)cc(OC)nc(OC)n1 C1(=O)C(N(C)C)C(C)NC(=O)CCC2CCN1C2.C(C(C)C)N(CCOC)CC Cc1cc(N)c(C(N2CCC(O)(CN(C)C(C3OCCC3C)=O)C2)=O)c(F)c1 N1(CCC2(C)CC2)CCC(=O)N(C(C2(N(C)C)CCOCC2)C2CC2)C1=O CC1CN(C(=O)Cn2ccccc2=O)CC1C(N1CCC(O)(C(N)=O)C1)=O c1(-c2c(CNCC(CO)F)c[nH]n2)cccc(Br)c1 c12ccc(cn1)CNC2=O.c1(C(=O)OC)coc(CNC(=O)CC2CCCC2)n1 c1(C(=O)NC2CN(C(=O)C(F)C(F)(F)F)CCC2CO)ccc(Cl)c2occc12 N1(c2nccc(C)n2)CCCC(C2(NC(C3CCC(=O)N(C)C3)=O)CC2)C1 C1(CNC(C(c2ccc(N)cn2)C)=O)CC2CC1CN2C(c1cnnn1C)=O c1(OC)cccnc1C(=O)NC1CC1CNC(c1cccc(-c2nnco2)c1)=O C1(C(N2CC3(CN(C(=O)Cc4ccnn4C4CC4)C3)C2)=O)CNc2ccnn2C1 c1cc2n[nH]cc2cc1-n1cc(C2CCN2CC2CCSC3(CCC3)C2)nn1 n1(C(C(C)C)C(=O)OC(C)C(c2ncccn2)C)cc2c(n1)CCCC2 CC(C)(C)C(C(=O)NCCC1CCCO1)NC(C1COCC1(C)C)=O c1(CC(=O)NC2CN(C(C(CC)COC)=O)CC2O)cc2ccccc2s1 CC(C)CCC(=O)C(=O)NC1CC2(C1)CC(C(N1CCC(O)C(C)C1)=O)C2 O=S(=O)(c1ccc(N2CCCCCCCC2)c(Br)c1)NC1CCN(CCF)C1 c1(C(N2CCC(C(F)C(=O)N3CC(C4CCOCC4)C3)C2)=O)ccc(O)cc1F C(CCC(=O)NC(c1ncccn1)C)NC(C=CC=CCC)=O C1(CNC(c2ccc(C3(O)COC3)cc2)=O)CN(c2nccc(Br)n2)CCO1 CC(CN(C)C)CC(=O)NC1CCC(NC(C2CC(=O)N(CC3CC3)C2)=O)CC1 C(C(N=[N+]=[N-])C(=O)N1CCCCC1CNC(c1cnc(Cl)s1)=O)OCC N=c1cc(C(N2CCCC2c2c(F)cccc2Cl)=O)c(F)c[nH]1 C12(C(=O)NCC(COC)(O)CO)CCC(CC1)N(C(=O)C(c1ccnn1C)C)C2 C(=O)(CC(C)C(=O)N1CCC(CNC(=O)CC(C)C)C(C)C1)OC CC(C)C(CNC(=O)COCCc1ccc(Cl)s1)NC(=O)C(C)CF CCC(C)C(C(=O)NC1COCC1O)NC(=O)C(F)OC(F)(F)F c1(CC)nncn1NC(=O)C(CN(C)C)NC(C1C2(CC2)C12CC2)=O CC(C)C(F)(F)CC(=O)NCCCCN(C)C(c1ccc(C(N)=O)o1)=O c1(C(=O)NC(C2N(C(C3OCCN(C)C3)=O)CCC2)(C)C)coc(S(N)(=O)=O)c1 O=C(CCC[N+](=O)[O-])NCCOC1CN(C(=O)Cc2ccnn2C2CCCC2)C1 c1(C(=O)NC2C=CCN(C(C(CC)C#N)=O)C2)cc(Cl)ccc1O CCC(C)(Cl)CNC(=O)COCCNC(=O)CCC1CC1(C)C C1(C(=O)NC2(C(F)(F)F)CC3CCC2C3)CCC12CCOCC2 C1(C(=O)Nc2ccc(OC)cc2)CN(Cc2cccc(O)c2Br)CCC1O C(CN=c1[nH]c(SC)ncc1NC(C)=O)N1CCN(C(CC(C(N)=O)OC)=O)CC1 c1(C(=O)NCCCOCCNC(C(COC)(F)F)=O)ccc(F)c(F)c1F N1(C(CN(C(C)=O)C)=O)CCC(=CCNC(C2CCCC2F)=O)CC1 c1(CN2C(C(=O)Nc3cc(F)ccc3Cl)CC(=C)C2)ccc2cc[nH]c2c1 C1(CC(=O)NCC(C2CC2)NC(=O)C=CCn2cncn2)CC(O)C12CCC2 C1(NC(c2nc(C)n(C(F)F)c2)=O)CCCCN(C(C2OCC3CCCC23)=O)C1 c1(C(N(CCCNC(=O)COCC(F)(F)F)C)=O)csc(C(C)(F)F)n1 N1(C(c2ccc(COC(C)=O)o2)=O)CCCCC1.C(=O)(CC(C)(C)C)NC(=O)CN N1(C(CC(CCCC)O)=O)C2CCCC1CC(NC(=O)CCC1OCCO1)C2 C#CC1(C(=O)NCC2C(C)CCN2C(=O)C(COC)COC)CCCC1 CC1CC(=O)NCC1C(=O)N(C1CN(C(=O)Cc2cc(C(F)(F)F)co2)C1)C C1(NC(=O)CCc2ccon2)C2CC(O)C1N(C(C1(CC(F)F)CC1)=O)C2 c1(C(C)C(=O)NCC(O)CCNC(c2ccoc2)=O)ccc(Br)c(Cl)c1 C(=O)(C(O)CC[S+](C)C)NCCC1CCCN(C(C(C)Cc2cnc[nH]2)=O)C1 C1(C(=O)NCc2conc2C)(CC)CCN(C(c2cncn2C(C)C)=O)CC1 CC1(C)Cc2[nH]nc(C(N3CCC(NC(=O)C4=CC(O)CCC4)C3)=O)c2C1 N1(C(c2c(C)ncnc2)=O)CC2(CCC(C(=O)Nc3ccc([N+](=O)[O-])cc3)O2)C1 C#Cc1cnn(C)c1C(=O)NCC(F)CNC(c1ccc(C(=O)C2CC2)cc1)=O C=CCC(CNC(=O)CCN(S(C)(=O)=O)C)NC(=O)CC(C)F C1(CCOC(=O)N(C(C)(C)C)CCS)CCCCN1CC(F)F C(c1ccc(F)c(OC)c1)=CC(N1C(CNC(C(C)=CC)=O)CC(O)C1)=O N1(C(CCC)=O)CC(NC(c2ccc(O)cc2Cl)=O)CC12CCCC2 C1(C(N2CCC(F)(F)C(F)C2)=O)C2CCCC2CN1C(c1cc(Cl)n[nH]1)=O c1(-c2onc(-c3ncc(C(F)(F)F)o3)n2)ccc2c(c1)C(=O)CCC2 C1(C(C)C)C(=O)NCCCN1C(C1(C)CCN(C(=O)CN2CCOCC2=O)C1)=O C1(NC(c2ccc(CC)cn2)=O)CN(C(=O)CSCC(=O)NC)CCC1C C1(C(N2C(CNC(C(C)OCC3CC3)=O)CCC2)=O)CCN(C)C(=O)C1 N1(C(CS(CC)(=O)=O)=O)CC2(CCCC2)C1C(=O)NC1CC2CCC1O2 c1(CC(N2CC(C(C(=O)N(C(C)COC)CC)OC)C2)=O)ncc(C)o1 N1(C(C(C)N(C(=O)Cc2ccc(O)cc2)CC)=O)CCC2(CCCN2C)C1 N1(C(CN(C2CCC2)C(c2c(C(C)C)ocn2)=O)=O)CC(O)C2(CCCC2)C1 N1(C(COCCC=C(C)C)=O)CCCCC1C1CCCN(C(=O)CO)C1 c1(CCC(=O)NC2C(C)N(C(=O)CCN3CCC3)CC2)cc(F)ccc1F C1(C(N2C(CNC(C=C(C)C(C)C)=O)CC(O)C2)=O)CC12CCCCC2 C(=O)(C(CC(C)C)c1ccc(Cl)cc1)NCC(CO)NC(c1c(C)scn1)=O c1(NCC(=O)N(C2CCN(C(c3n[nH]cc3F)=O)C2)C)ccccc1 C1(CNC(=O)CC2CCSC2)CCCCN(C(C2CCC(F)(F)C2)=O)C1 CCC(C(=O)NC1CC(NC(c2nocc2C)=O)C(O)C1)C(F)(F)F C(CN=C(NCC1(C)CCCCC1)NC1CCCS(=O)(=O)C1)OC c1(C(=O)NCc2sc(C(=O)NC3C(CC)CCC3)c(C)n2)ccnc(N(C)C)c1 C1(CCNC(c2c(C)scn2)=O)CN(C(C2CC3(C2)OCCO3)=O)CCCO1 C(=O)(CCCN(C)N=O)NCC1C2CN(C(CCN3C(C)CCCC3)=O)CC21 c1(C(=O)NC2(CC(F)(F)F)CCN(CCCOCC)C2)nc(C(C)C)ncc1Cl C(N=c1[nH]c(=NC(C)CCCCCO)[nH]c2c1CSC2)C1C(C(=C)C)OCC1 c1(CC)c(NC(=O)NC2CCC(Nc3ccc(F)c(C)c3)C2)ncnc1Cl c1(C(=O)NC2CCCN(C(C3CC(C#C)(O)C3)=O)CC2)nc(C)[nH]c2nccc1-2 c1(C(=O)NC2CCCCN(C(C(C)CC3CC3)=O)C2)cc2cccc(Br)n2c1 c1(C(C(=O)NC2C(NC(C(CC=C)CC)=O)CCC2)O)cccc([N+](=O)[O-])c1 c1(COC)ncc(C(=O)NCC(CO)NC(c2nnc(C)s2)=O)c(O)n1 C12(C(=O)Nc3cccc(CO)c3)CCN(C(C34CSCC3C4)=O)CCC1C2 NS(=O)(=O)C1CCc2ccccc2C1NC(N1CC2CC(C1)C2O)=O N#Cc1cncc(NC(C(=O)O)C2=CCCS2)c1 C(=O)(C1CCCc2nc[nH]c21)N(C1C(N(C(c2c(C)snn2)=O)C)CCCC1)C C1(C(=O)Nc2ccccc2Cl)CN(C(=O)COc2ccccc2)CC1O c1(C(=O)NC2CCCCN(C(c3ccc(C)n3C)=O)C2)cc(O)c2sccc2c1 C(CC(=O)N1CC=C(CO)CC1)(C(C)(C)C)NC(c1scc(OC)c1)=O Cc1nc(NCC2CSCCO2)cc(=NCc2ccc(OCC(C)C)nc2)[nH]1 CN=c1[nH]c(N(CC(=O)OC(C)(C)C)NC(C2CCCCC2)=O)ncc1Br Cc1ccnnc1C(=O)NC1CCCC(C(=O)N(C2CCCCC2C)C)C1 c1(C(=O)Nc2n(C)ncn2)ccc(Cl)cc1Nc1ccc(-c2ccno2)cc1 C1(CNC(C2C(NC(Cc3cc(CC)no3)=O)C2(C)C)=O)CCOC(C)(C)C1 C1(NC(C=COCC)=O)COC2(CCCN(C(C3CN(CC(F)(F)F)C3)=O)C2)C1 n1(CCCC)ncc(C(=O)NCC2(CNC(C3COC(=O)N3)=O)CCC2)c1C C1(CCNC(C2(CC#C)CC2)=O)CCCCN1C(=O)CCn1cc(Cl)cn1 CC1CC(C(N2CCOC(C)(CNC(c3cc(Cl)no3)=O)C2)=O)CCN1C N1(C(c2nc(COC)oc2)=O)CCN(C(=O)C(c2cnn(C)c2)OC)CCC1C c1(OC)cc(Cl)cc2[nH]c(C(=O)NCC(c3ccc(F)cc3)N(C)C)cc12 c1(C(N2CCC(NC(C(C=C)(F)F)=O)C2C)=O)cc(C)c(C)c(F)c1 C=CCC(F)(F)C(=O)NCC1CC(NC(=O)C(CCF)NC(=O)OC(C)(C)C)C1 N1(C(=O)NCC2CCC3(CCCC3)O2)CCN2CCNCC2C1 O=C(CCCCN1CCCC1)NC1CN(C(=O)Cc2ccccc2Cl)C2CC12 c1(C(N2C3C(NC(C=C(CC)C)=O)CC(C3)C2)=O)ccc(Cl)c(C#N)c1 c1(OC)ccc(C)cc1S(=O)(=O)NC1COCCN(C(=O)C(C)=CC2CC2)C1 C(=O)(C(C#N)C(C)(C)C)NC(CC#C)CC(=O)N(C)CC1CC(O)C1 C1(C(CN2CC(CN(C(C3(SC)CC3)=O)C)C2)=O)CCOC(C)C1 N1(C(CNC(CC(C)(C)C)=O)=O)CCCC(C)(CNC(=O)COC2CCOC2)C1 c1(C(=O)NCC(CCOC)NC(COCCOC)=O)ccc(CCF)cc1 N1(C(C2C(C(=O)OC)C2)=O)CC2CC(NC(c3cnc4[nH]cncc3-4)=O)CC2C1 Cc1cc(N)cnc1C(N1CCC(C(O)CNC(=O)C(C(C)O)N(C)C)CC1)=O c1(C(CC)C)ccc(NC(=O)CC=C(C)C)cc1.N12CC(CC1C)C2=O C1(NC(CN(C(C)=O)C)=O)Cc2ccccc2C1NC(=O)CC1CC1(Cl)Cl N1(C(c2nccc(CNC(C3C(C)(C)C3(F)F)=O)c2)=O)CCCC(O)CC1 C1(N(C(c2c(COC)n(C)nc2)=O)C)CCCN(C(=O)C(=O)NCC(F)F)CC1 C1(NC(C)=O)CN(C(=O)Cc2cccc3ccoc23)C2(CCCOC2)C1 CC1NC(=O)CCC1C(C1CCC1)NC(C1CC2(CC2)CN1C(=O)CC#N)=O c1(C(=O)NC2CCN(c3c(C)ccs3)C2=O)ccc(CF)cc1 C=CC(C(=O)NCC1CCC1C(N1CCC(C2(C)N=N2)C1)=O)OC S(=O)(=O)(c1cccc(C(N2CCCC2C(C)(C)O)=O)c1)NC(C(C)C)C1CC1 c1(C(=O)NC2(C)CN(C(c3ccc(F)c(Cl)n3)=O)C2)ccc(N)c(Cl)c1O N1(C(C2(C#C)CC(=O)C2)=O)CCC(C)C(CC(=O)NCCN2CCCCC2=O)C1 c1(C(N2CCC(C(=O)NCC(C)CCO)C2)=O)cccc(CO)c1 c1(C(N2CCC(N(c3c(C(=O)OCC)cncc3)C)C2)=O)cccc(C)c1F Cn1c(C(=O)NCC(C2CCCC2)NC(=O)COC2CCOC2)ccc1[N+](=O)[O-] c1(C(C)(C)C(=O)NCCCNC(c2ccn(CC(F)F)n2)=O)c(F)cccc1F c1(OC)cnc[nH]c1=Nc1ccc(C(F)F)c2ccccc12 C12(CC=CCC1)C(=O)NC2.c1(CC2CCCO2)cccc(O)c1.OC c1(SC)ccnc(C(=O)NCC2C(C)CCN2NC(C2CC2C(C)O)=O)n1 C(=O)(CCCCC#N)Nc1c(C)oc(CO)c1.C12CC(NC1=O)C(=O)Nc1cn2nn1 c1(C2CCN(NC(=O)C(c3ccc(F)cn3)N)C2)ccc2sc3ccccc3c2c1 C1(C(N(CC(C)NC(c2c(CC)c[nH]c2)=O)C)=O)CCC(CC)CC1 c1(NC(C2CCN(Cc3ccc4ncoc4c3)CC2O)=O)cc(Cl)cc(Cl)c1Cl C1(N(C(CC2ON=C(C)C2)=O)C)CCCCN(C(=O)CN2CCSCC2)C1 C(=O)(C1=CC(C)(C)C1)NC1C(OC)CN(C(=O)Cc2nocc2C(C)C)C1 c1(C(CNC(C(C)N(C)CC)=O)NC(=O)COC2(C)CCC2)ccccc1F N1(C(CC2CCC(C)O2)=O)CCC2(CC2C(=O)Nc2ccnc(C3CC3)n2)C1 N1(CCNC(C(F)(F)C2(OC)CCC2)=O)CC=C(CN)CC1.C(C)(C)O N1(C(c2c(CC)nc[nH]2)=O)CC2CCCC1(CNC(c1cc(C)cc(O)c1)=O)C2 CC(C)CCCCC(=O)NC(C1=CCCCC1)c1nnnn1-c1ccc(F)cc1 C(CCCCSC)NC(CCN(C(=O)C(C1CCC(=O)N1)C)CC#C)=O C1(NC(Cc2scc(C)c2)=O)CC2(C1)CC2NC(c1nc(C(C)C)oc1C)=O CCCN(OC)C(=O)C(c1cccnc1)NC(=O)CC(C)(C)O c1(C(N2CCN(C(C(C)S(C)(=O)=O)=O)C(CF)C2)=O)ccc2c(c1)NC(=O)C2 C(=O)(C(C)(C)CC(C)(C)C)N1CC(C(N(CC(CC)(C)OC)C)=O)C(C(C)C)C1 CC1Cc2sc(NC(=O)NCC(c3ccc(F)cc3F)O)c(C#N)c2C(C)C1 c1(C(N(CCCCNC(C2(C(F)(F)F)CCC2)=O)C)=O)cc2cccc(Cl)c2s1 c1(C(N2CCCC(N(C(CCCC)=O)CC)CC2)=O)ccc(P(C)(C)=O)s1 C(C)(C)(CCCNC(=O)COC(C)(C)C)NC(C1CCC(OC)C1)=O c1(C(=O)NCC(C(C)C)NC(C2(CC#C)CCC2)=O)cccc2c1nc(O)n2C c1(NC(C2N(C(C(CC)(C)O)=O)CCC2)=O)nc(F)c(Br)cc1Br N1(C(C2(OC)CC(C)C2)=O)CC(C(=O)NCCn2ccnn2)C(C)C1 CC1(CCCOC(=O)CCC2CCCO2)CC1(F)F Cc1cccc2c1OC(C(=O)NCCCCCCNC(C1(C(C)C)COC1)=O)C2 N1(C(c2c(C)sc(O)n2)=O)CCC(F)C(NC(c2cc3occc3s2)=O)C1 Cc1ccc(F)cc1C(=O)NC1CC2CN(C(=O)CC3CC(=O)NC3=O)CC12 N1(C(C(CC#C)C)=O)CCN(C(c2cnc3n2CCS3)=O)CC(C)(F)C1 N1(C(c2nc(Cc3nc(C)sc3)sc2)=O)CCN(C(=O)COCC2CC2)CC1C Cc1cc(C(=O)NC2CC(F)(CNC(C3C=CCCC3)=O)C2)no1 CC1COC(C(=O)NC2(C)CC(NC(=O)CN3CCSCC3)C2)C1 C(CC(=O)NCCOCCNC(=O)CC1(C)CC1)(OCC)O.CCCF.OC c1(C(=O)NC2(C)CN(C(C3CC(C)C(C)CC3)=O)C2)nnc2n1CCCC2 C1(C(N2CC(C)(CC(=O)NC3C(NC(=O)OCC)C3(F)F)C2)=O)CC12CCOCC2 C1(NC(=O)C(c2ccc(F)cc2)F)CCC12CN(C(=O)CC1COCCOC1)C2 N1(C(C(C)N2CCCC2)=O)CCC(NC(C2C=CCCC2)=O)C12CCC2 c1(CC(=O)NCCCN(C(C=Cc2c(C)cccn2)=O)C)c[nH]nc1S(N)(=O)=O c1(CC(N2CCOCC(CNC(C(CC#C)O)=O)C2)=O)nc2c(o1)CCSC2 C=C(C)CC(C(=O)NCCC(=O)NCCOC)NC(=O)C=C1CCC(C)CC1 C#Cc1ccc(C(=O)N(C)CC2CCN(C(c3ccc(O)nc3C)=O)C2)c(C)c1 CC(CNC(C1CC2CC2N1C(c1ccc(F)nc1)=O)=O)C(C)(F)F CC(C)(F)C(=O)NCCOC1CCN(C(=O)CN2CCOC2=O)C1 Cc1ccc(C(N2CC(F)(C(=O)NCc3ncccc3Cl)C2)=O)c(O)n1 C1(NC(=O)CC2COC(=O)C2)CC2CCC1CC2NC(C1(CO)CC1)=O N1(C(CC)=O)CCCCC1C(N1CCC(CCNC(C2CC(=O)N2)=O)C1)=O C1(NC(CC2(CC)CCC2)=O)CC2CC(C1)N(C(=O)Cc1ccc(F)cc1)C2 N1(c2ncc(C)cn2)CC23CCCC2(CN(C(=O)Cc2csc(C)n2)C3)C1 N1(C(CN(C)CC)=O)CCN(C(=O)CC2CCCCCC2)C(c2nccn2C)C1 c1(C(=O)NCCC(=O)NCCCC2(C(N)=O)CCCC2)ncccc1O C(CN=C(NCC(c1ccccc1)N(C)C)NC1CCOCC1)c1scc(C)n1 C1(NC(C=Cc2cnc(C)s2)=O)CCC12CN(C(=O)C(C)NC(N)=O)C2 c1(C(N2CCC(N(C(=O)CC3=CCCC3)C)C2)=O)cc2scc(Cl)c2[nH]1 c1(NC(C(C)(N(C(CSC)=O)C)C2CC2)=O)cccc2c1OCC2 C1(N(C)C)CN(C(C(=O)NCc2ccc(F)cc2)C2CCOC2)CC1C1CC1 C1(CC(=O)NCCSCCOC)CC(C)(C)CN1C(=O)CCN1CCCCC1 c1(C(=O)NCCCCC(C)NC(c2c(C)nc(CO)s2)=O)c(O)cccc1O CN1CC(C)(C(=O)N(CCCNC(C2C3CCC(C3)C2(C)C)=O)CCO)CCC1=O C1(NC(c2cccc(COC)c2)=O)CCN(C(=O)C=C(C)C(F)F)C(C2CC2)C1 N1(C(C(CC)(C)C(=O)OC)=O)Cc2c(OC)ccc(OC)c2C(O)C1 CC(C)CC(C(=O)N=S(C)(=O)c1nccn1C)NC(c1cncnc1)=O C#CCCC(O)C(=O)NCC(CNC(c1cc2occc2s1)=O)C(F)(F)F N1(C(c2cnc(NC(C)=O)s2)=O)CCC(C)(C)C1C(=O)NC1CCC(F)(F)C1 N1(C(CCC#C)=O)CCCN(C(c2ccc(F)c(CO)c2)=O)C(C(C)C)C1 Cc1[nH]c2ccccc2c1C1CC1.C1(=O)C(Cc2nonc2C)N(C)CCCO1 C1(NC(C(C(C)(C)C)OC)=O)CN(C(c2ccc(C)cc2Cl)=O)CC2CCCC12 C1(C)(CNC(CCN(C)CC)=O)CCCN(C(C2(Br)CC2)=O)C1 C1(C(N2CCN(C(=O)CCc3ccncc3)CC2CO)=O)CCCC(F)(F)CC1 c1(C(=O)NCC2(C(F)F)CCN(C(C(C)(C)OC)=O)C2)c(F)ccc2[nH]ccc12 N1(C(CNS(CCCC)(=O)=O)=O)CCCOC(CCNC(C2CCCC2)=O)C1 N1(C(CC(CNC(C2CCC(CO)CC2)=O)OC)=O)CC(O)CC(O)C1 C(=O)(CC(F)(F)C(F)F)NCC(C(C)(C)C)NC(=O)CC1CCCS(=O)(=O)C1 C(=O)(CCCCCCN=[N+]=[N-])NCC1C(NC(c2nccc(C(=O)OC)c2)=O)C1 N(S(=O)(=O)N1CCC(c2ccccc2C(=O)O)CC1)C1CC(C)(C)SCC1 N1(C(C2C(=C)C2)=O)CC(NC(C2CC(=O)CO2)=O)C(n2ccnn2)C1 C1(N2C(C(=O)OC)CCC2)CCN(C(C2(CC(=O)O)CCOC2)=O)CC1 C1(NC(C(C(C)C)NC(C(CO)OC)=O)=O)CCCCC12CC2 Cc1cc(C(N2CC(NC(=O)CC3CCS(=O)(=O)C3)C2)=O)c(N)c(Cl)n1 N1(C(C2C(C(C)C)OCC2)=O)CC=C(C(=O)NOCC2CCOCC2)CC1 c1(CC)ccc(-c2nc(C)c(NC(c3n[nH]cc3-c3ccc(F)cc3)=O)s2)cc1 Cc1c(C)n(CCC(=O)N2CCCC2)c2ncnc(NC3CCCSC3)c12 c1(CNC(C2CCC(n3cc(CCNC(C)=O)nn3)C2)=O)cccc(C)c1 C1(OC)CN(C(=O)CCc2ccncc2)CC1NC(=O)CC1CCC(=O)N1 Cc1cc(NC(=O)CC2C3CCCC3N2C(C2CCCSC2)=O)ncc1F c1(N2C3CN(C(CC(C)n4cccn4)=O)C(CC3)C2)ncc2cccnc2n1 c1(NC(=O)C=Cc2cnccn2)nc2c(s1)CC(NC(C1CCSCC1)=O)CC2 C(=O)(C#Cc1ccccc1)NCC1OCCN(C(=O)OC(C)(C)C)C1 CC1(C)CCC(C(=O)NCC2(O)CCC2)CN1C(C1CCC(=O)N1)=O Cc1ncn(C)c(=O)c1C(=O)NCCCC(CO)NC(c1c[nH]c(=N)o1)=O CC(CCC(=O)N=c1ccn(C(C)(C)C)[nH]1)NC(c1cnc2cc[nH]c2c1)=O CC(C(=O)N1CCC(F)(CNC(C2CCCC3(CC3)C2)=O)CC1)S(C)(=O)=O C(c1c(Cl)cccc1Cl)=C(C)C(=O)NCC(F)CNC(=O)CCP(C)(C)=O C(=O)(C(C#N)C(C)C)N1CC(C)C(C(=O)NCCn2cccnc2=O)C1 Cc1ccc(-c2cn(CCOCC3CC(F)(CO)C3)nn2)cc1.C(=O)(C(F)(F)Cl)NCC CN1C(=O)N(C)C(c2ncc(C3OCCO3)s2)C2=C1CCN(CC1CC1)C2=O C(=O)(CC1=CCCC1)NCCN(C)C(C1CCCC(Cc2ccccc2)O1)=O c1(C(=O)NC2C(CNC(c3c(C)occ3)=O)COC2)cnc2c(C)cccc2c1 N1(CC(=O)NS(c2cn(C)nc2CO)(=O)=O)CC(CO)Cc2ccccc21 C(=O)(C(C(C)NC(=O)COC1CCOCC1)C(C)C)NCC(CC)C(C)(F)F c1(C(=O)NCC2(C)CCCC2NC(=O)Cc2cnc[nH]2)cccc2oncc12 C(=O)(C=C(Cl)Cl)NCC1CC(NC(C2(N(C)C)CC2)=O)C1 C1(NC(COC)=O)CCCC(CO)C1.c1(CC)nocc1C(=O)NC1CCN(C=O)C1 c1(OC)ccc2nc(N3CCC(CO)C3)[nH]c(=NCCC(C)(C)C)c2c1 Cc1cn(CC(N2CCN(Cc3n[nH]cc3Cl)C3CC23)=O)c(=O)nc1O N(C(=NCCCF)NCC1(c2c(Cl)cccc2Cl)CC1)CCCN(C)C C1(CC(=O)N(CCCF)C)CCCN1C(c1nocc1Cl)=O c1(C(=O)NC(C(C)NC(=O)CCN2CCN(C)CC2)CO)cccn2ccnc12 N1(C(=O)CC2COCCN2C2CC2)CCC2(CCC(c3ccccc3)CC2)C1 CC1CC(C(=O)NC(C)CN2CCN(C(=O)CCc3cc[nH]n3)CC2)CCO1 Cc1ccc(C(=O)NC2CCN(C(=O)Cc3cnns3)C23CC3)cc1C(F)(F)F C12(C(=O)NC(C3CCN(C(C4(CC#C)CCC4)=O)CC3)CO)CC=CC(C1)OC2 N1(C(C(C(C)C)NC(c2c(CCC)n[nH]c2)=O)=O)CCC(CO)C(C)(C)C1 c1(CN(C(C(=O)NC(c2c(OC)nccc2)C)=O)C2CC2)ccc(F)c(C)c1 c1(C(=O)OCC)cccc(C(=O)NCC2CC(C(F)(F)F)CCN2C(C)=O)c1 c1(C(N2CCC(O)(CNC(CCCCSC)=O)C2)=O)cc(Cl)cc2c1NCCC2 CCC(CC)C(=O)N1CCCCC1c1cn(-c2cnn(C)c2)nn1 c1(OC)cc(NC(c2cscc2-c2cc(F)ccc2I)=O)c(Cl)cn1 c1(NC(=O)CC2CN(Cc3ccc(I)cc3Br)C2)c(I)cc([N+](=O)[O-])cc1I C12(F)CCCN(C1)C(=O)C(OC)C1CN(C1)C2=O.CCC(O)COC c1(C2CCN(C(c3c(OC)scc3)=O)CC2)ccc2c(c1)S(=O)(=O)N=C2Cl C1(CN)CCCCN1C(c1cc(CO)[nH]n1)=O.c1(C2(OC)CC2)c[nH]c(C(=O)OC)c1 C1(OC)C(CNC(=O)C=CCOc2ccccc2)COC12CCC2 C1(C(N(C2CN(C(c3csc(-c4ncccn4)n3)=O)C2)C)=O)CC(C)(C)CN1C c1(CN2CCC(O)(C(=O)NC(c3c(C)cc(Br)cn3)C)C2)cc2ccccn2n1 N1(C(=O)COC(F)F)CCN(C(=O)COc2ccccc2Cl)C(CCOC)C1 C1(=O)CCCC(=O)N1.C(=O)(C(CC1CCC1)C(=O)OC(C)(C)C)N(CCOC)C Cc1csc(C2CCCN2C(CC(N2CCCC2)=O)=O)n1 c1(C(N2C3CC(NC(C(C)n4ccnc4)=O)C3CC2)=O)noc2c1CCCCC2 c1(C(=O)NC(CN(C(C2(OC)CC(C)C2)=O)C)(C)C)ccc2cc(C)ccc2n1 O(NC(=O)C(F)C(C)CNC(=O)C1=CCCC1)CC(=C)Cl C1(NC(C(C)(N(C)C(C2CC3(CCCO3)C2)=O)C2CC2)=O)CCCC(O)C1O N1(C(C(N2CCCC2)C)=O)CC2CCC(C(=O)NCCCCC3CC3)(C2)C1 c1(NC(C(N2CCC(Cc3sc(C)c(Cl)n3)C2)CC2CC2)=O)ccc2c(c1)CCC2 CC(C)CC(C(=O)NCC(=O)N(C)O)NC(c1cc(Cl)c[nH]1)=O c1(C(=O)NC(C(C)NC(C2(C)CS(=O)(=O)C2)=O)CO)ccc2c(c1)CC(C)(C)O2 N12CCN(CC1)Cc1cn(nn1)C1(CC1)C2=O.c1(CO)ccc(C)nc1OCC c1(C2C(=O)N2)nc2cc([N+](=O)[O-])ccc2o1.C(CN(C)C)SC C(=O)(C(C)(C)C(O)C(C)C)NC1C2CC(CNC(c3c(C)[nH]cc3)=O)(C2)OC1 c1(C(=O)NC2CC(NC(c3cnc(OCC)s3)=O)C2)cc(F)cc2cnccc12 C(=O)(C(C)(C)CCCNC(c1nnccc1C)=O)NC1CC(OC)C1(C)C C1(NC(C(C)CF)=O)CCC2CN(C(c3cc(O)ccc3Cl)=O)CCC2C1.C1(C)CC1 CCCCCCC(CC)C(=O)N1CCC1(C)C(=O)Nc1cncc(C(=O)OC)c1 N1(C(c2ncc(C)nc2)=O)CCC2(C1)CN(C(C1CC(CC3CC3)C1)=O)CCO2 N1(C(C2C(CC)C2)=O)CC(CN(C)C(c2cc(F)sc2Br)=O)C2(CC2)C1 CCC(COC)C(=O)NCCCN(C)C(c1snnc1C1CC1)=O C1(C(=O)NCCN(C(C(C)OCC(C)C)=O)CC(C)O)OCC2CCCCC12 CC1CC(NC(=O)C(CCC2CCC2)NC(C2CCSC2)=O)CC(C)C1 C(CCN=C(NCc1cnc(CC)o1)NC(c1ccco1)C)c1nnc(CC)s1 C(=O)(C(CNC(=O)C(C)CO)(CC)CC)NCc1ncc(OCC)nc1 C1(C(=O)NC(CNC(Cn2c(C)ncc2)=O)(C)C2CCC2)CCCCN(C)C1=O C1(NC(C)=O)CN(C(c2c(Cl)cc(Br)cc2Cl)=O)CC12CCOCC2 O=C(CC(F)(F)F)NCC1(O)CN(C(=O)C(F)OC(F)(F)F)C1 N1(C(C(=O)OC(C)(C)C)=O)CCCCC(CC2C(OC)CC2O)C1 C1(C)CCC(=O)N1.C(CC(F)(F)F)N(C(COC)=O)CCO c1(C(N2CCC(N(C(C3(COC)CCOC3)=O)C)CC2)=O)ccc(Cl)nc1O N1(C(COC(CC)C)=O)CCC(C)CC1CNC(=O)Cc1nc(Cl)cs1 CC1CCCCC1(C)CNC(C1(c2cncc(F)c2)CCC1)=O C1(OC)CN(C)C(C)(C(N2CCC(CN(C)C(c3cccc(N)c3C)=O)C2)=O)C1 N#Cc1ccc(O)c(C(=O)NCC(O)CNC(C2CC2c2cncc(Br)c2)=O)c1 C(C)(C)(CC(=O)Nc1ccc(C(C)(C)C)cc1)OC N1(C(c2cncc(CC)c2)=O)C2CCCC1CN(C(C1CCC(=O)N1C)=O)CC2 c1(C(N(CCC(C(C)C)NC(c2scc(C)c2)=O)C)=O)ccc2c(c1)CCCO2 N1(C(c2cccc(CO)c2)C(=O)NC2COC2)CC2CC1C(O)(C(F)(F)F)C2 CN1CCN(C(=O)CN2CCCCC2=O)CC1CNC(c1ncccc1F)=O c1(C(N(c2c(C)ccc(C)c2)C2CNCC(C)C2)=O)cccc2c1OCO2 C1(C(=O)NCC(COC)(C)C)CCN(C(C2COC(=O)N2)=O)CC1C c1(C(C)NC(N2CCC3(COC)C(C2)C3)=O)cc2ccccc2o1 c1(OC)nn(C)cc1C(=O)NCCCC(=O)N1CCC1C(C)C CC1CCC(C(N2CCCCC2CCNC(=O)CN2CCCOC2=O)=O)CC1 C12(NC(C(CC)C)CO)C3CC1C1C(C(=O)Nc4ccnc5ncnn45)C3C21 C1(CNC(C2C(C)C2)=O)COCCN1C(C1CCCCC1C(F)(F)F)=O C1(C(C(=O)N(c2cccc(F)c2)C(C)(C)C)O)CCCN(C=O)C1.CO C#CCCC(O)C(=O)NCC1CC(NC(=O)C(C)=C2CCC2)C1 CC(C)CC(O)C(=O)NCCC1CSCCN1C(=O)CCCc1ccncc1 C(CC(C)CC(C)(C)C)NCC(c1ccccc1C(F)(F)F)C c1(NCCC(c2nnnn2C2COC2)N)ccc(F)cc1.C1(C(C)(F)F)(C)CCC1 CCCCC(O)CC(=O)NC1CC(NC(=O)C(F)Oc2ccc(Cl)c(F)c2)C1 N1(C(C(C2CCOC2)OC)=O)CC2(CCN(C(c3ccc(O)nn3)=O)C2)C1 C1(NC(COc2cc(C)on2)=O)CC2CC(C1)N(C(=O)CC1CC3(CCC3)C1)C2 N1(C(C(C2(C)CC2)NC(c2ccc(OC)nc2)=O)=O)CC=C(C(C)(C)C)CC1 CCCCC(C(=O)N1C2CCC1C(CNC(=O)Cc1nnc(O)s1)C2)NC(N)=O N1(C(=O)CCCCN2CCOCC2)CCN(C(=O)CCc2ccon2)C(CO)C1 C1(C(N2CC(O)(C(C)NC(=O)CC3CC4CCC3C4)C2)=O)CCC(C)(C)CC1 C1(OC)CCN(C(=O)OC2(C(=O)NC(C)C)CCOCC2)C(c2ccccc2)C1 CCC(N=c1ccc2nnc(C(c3ccccc3)C)n2[nH]1)C(C)C Cc1cn(CC(=O)NC2CC2CNC(c2cc(C3CC3)[nH]n2)=O)c2ccccc12 CC1CCCCCCN1C(=O)C=CC1CCCN1C(C1CN(C(N)=O)C1)=O C1(CNC(c2ccc(C(F)F)o2)=O)CC(O)CN1C(=O)Cc1sccc1Cl C1(C(N2C(CCC=C)CCC2)=O)CN(C(c2cc(C(C)=O)on2)=O)CCC1(C)C c1(C(=O)NC(c2nc(C)on2)C)cc(CNC(=O)C(C)c2ccsc2)ccn1 N1(C(C)=O)CCN(C(=O)CCc2cncs2)C(COC)C1 N1(C(C2C3CCC2(c2cncs2)C3)=O)CCN(C(=O)Cn2cccc2)C(CO)C1 c1(OCC)nc2ccc(C(N3CCCC(NC(=O)C(=O)C4CC4)C3)=O)cc2[nH]1 C(=O)(C1=CCCN(C(=O)CCOCC(C)C)C1)Nc1ccc(C)c(O)n1 c1(OC)ccc(C(=O)NCC(C)(C)CNC(C2COC3(CCC3)C2)=O)c(OC)n1 c1(CC(=O)NC2CCN(C(c3cnn[nH]3)=O)CC2)csc2c(F)cccc12 c1(C(=O)Nc2cccc(Cl)c2CO)c(F)ccc(Br)c1Cl C(=O)(C1=NNC(C(F)(F)F)C1)NCC1OCCN(C(c2ccc(N)cn2)=O)C1 c1(OC)ccc2c(ccn2CCCC(=O)N2CCC2C(=O)Nc2c(Br)n[nH]c2C)c1 Cc1ncnc(C(N2C(C(=O)N(C)CC3(C)CC3)CC2C)=O)c1C C1(C(N2CC(N(C(c3cc(SC)c(C)o3)=O)C)C(F)C2)=O)CCCCNC1=O CC1(C)CCC(n2cc(C3CC3(c3ccc(Cl)cc3)CO)nn2)CO1 N1(C(c2c(OC)ccc(Br)c2)=O)C2CCC1C(F)C(NC(=O)C(F)OC)C2 C1(NC(C(C)Cc2ccco2)=O)CCCCC1NC(c1ccnn1C)=O C1(C(=O)NC(C)C2CC2)CCN(C(=O)CC2CC2C2CC2)CC1 c1(C(N(C(CCNC(C2CCN(C(C)=O)C2)=O)C)C)=O)cc2cc(Cl)ccc2o1 CC(C(=O)NC1CC2CCC(C1)N2C(c1cc2n(n1)CCCO2)=O)C1=CCCC1 C=CCC(C)C(=O)NC(CC1CC1)CC(=O)N1CC=CC1 c1(-n2cc(CCCC#N)nn2)ccc(CNC(=O)C(c2ccccc2)F)cc1 C(c1ccc(C)c(C)c1)=CC(=O)NCC(CC=C)NC(c1nn(CC)nc1C)=O N1(C(C(C=C)C)=O)CC2(C)CC1(C(=O)NCCC1COCCO1)C2 Cc1cn2cccnc2c1C(=O)NC1COC2CN(C(=O)CC3CCC3)CC12 c1(CNC(C2(C(C)NC(=O)Cc3ccon3)CC2)=O)cccnc1 CN1CCCCC1C(=O)NC(C)(CNC(=O)C=CC1CCOC1)C1CC1 C(C(CC(C)C)C(=O)N1CCn2nccc21)NC(c1n(CC)nnc1)=O N1(C(C(CCO)N(C)C)=O)CC(NC(c2c[nH]c3ccncc23)=O)C2(CCC2)C1 c1(OCC)cc(C(=O)N(CCNC(=O)CCc2cnco2)CC2CC2)ccc1C CCC(CNC(C1(C)CC=CCO1)=O)(CC)NC(=O)C(C)(C)C.C1(=O)C(C)N1 N1(C(C(C)(C)C(F)(F)F)=O)CCCC2(C)CCCC12 c1(CNC(C2CCN(C(C(C)=CC=C)=O)C2)=O)oc(C)nc1C c1(C(COC(=O)C(F)(F)F)=O)cccc(Cl)c1N.CC1C(=O)N1 c1(CC)ccc(C(N2Cc3nc(Br)sc3C2)=O)cc1C#N c1(OCC)ccc(CNCC(CSC)CNC(=O)OC(C)(C)C)cc1 C1(C(=O)NC2CCSC2)(CNC(c2ccnn2CCF)=O)CCCO1 C12(C(N3CCCN(C(c4c(C)oc(Cl)n4)=O)CC3C)=O)CCC(F)(CNC1=O)C2 N1(C(C2N(C(CC)=O)CSC2)=O)CC(NC(c2ccc(C3CC3)s2)=O)C2(CC2)C1 C12CCN(CC1)N(C(=O)OC1CCC1)CCc1nc2n[nH]1.c1(SC)ccccc1 c1(C(=O)NC(CNC(C(F)=CC)=O)C(C)(C)C)c(C2CC2)nc2sccn12 C1(CNC(CC(C)N(C)C)=O)CN(C(c2ccnc(O)c2)=O)CC(C)(C)O1 C(c1cc2ccccc2n1C)=CC(=O)N(C1CN(Cc2ccccc2)CC1(C)C)C O=C1CCOCC(C(N2CCCC(C(c3ccccc3)C(=O)NC3CC3)C2)=O)C1 C1(C(=O)NCC2(CC(C)C)CC2)CC1C1CN(C(C2C3CCC(F)C23)=O)C1 c1(C(N(CCCNC(CC(C)SC)=O)CCO)=O)ccc2ccncc2n1 CC(CC(=O)NC1CC(O)(Cn2cc(CC3CCC3)nn2)C1)C(C)(C)C n1(CC)nc(C)cc1C(N1C(C(=O)NC2CC(C(F)F)C2)CCC1C1CC1)=O c1(C(N2CCC(=CC(=O)Nc3nc(F)ccc3Br)CC2)=O)nc(O)nc(O)c1F C1(n2cc(C3N(C)CCC3)nn2)(C(=O)NCC(F)(Br)Br)CCCCC1 c1(C(=O)NC(CN(C(c2cnc(O)c(F)c2)=O)CC)C)c(F)c(C)cc(N)c1F Cc1cccc(C=CC(=O)NC23CC(CNc4ncc(I)cn4)(C2)C3)c1 c1(C(=O)NCCN(C(=O)C2=C(C)OCC2)CCOC)cc(C)c(Br)c(C)c1 Cc1ccc(C(N2CC(F)(CNC(=O)Cn3nnnc3C)C2)=O)c(Br)c1 C(C1=CCN(C(=O)CN2C(C)CCC2C)CC1)NC(C(C)=C(CC)C)=O C(=O)(CC(CCCC)NC(=O)Cn1cccc1)N(CC(CCCC)CC)C N1(C(C(C)(C)C2CCC2)=O)CCCC2(C1)CN(C(=O)CC1CCOC1)CCO2 CC1(C)CCN(C(c2cccc3oncc23)=O)CC1NC(=O)CSC(F)(F)F C1(C2CCCN(C(c3ccc(Br)s3)=O)C2)(NC(C(C)(C)F)=O)CC1 c1(N(CCC)CCNC(=O)CC2CCC(=O)N2CC)ncnc2sccc12 CC1CC(C(N2CCC(O)C2)=O)N(C(=O)CCN(CCO)Cc2ccccc2)C1 c1(C(=O)NC2CC(C)N(C(=O)Cc3cnsc3)C2)ccn(CCO)c(=O)c1 C(CCCCCN(C(C)=O)C(C)C)NC(CCOCC)=O.c12csc(n1)NC2=O N1(C(Cc2cnc(C)s2)=O)CCN(C(=O)C=CC(C)(C)C)CC1 C1(C(=O)NCC2(C)N=C(C)SC2)CC(C)(C)CN1C(=O)NC(=O)C(Cl)(Cl)Cl c1(CSCc2cccc(OC(C(=O)OC)C)c2)cc2ccccc2s1 CN1C(=O)CCC1(C)CC(N1CCC1CNC(=O)CC1CC=CCC1)=O c1(CC)nc(C(=O)NC(CNC(C2(CO)COC2)=O)CC)cs1 C#CCC(C(=O)NC1CC(CC(=O)NC2C(=O)OCC2CO)C1)C1CC1 c1(OC)cccc(C(=O)NCCC(O)CNC(=O)CCC(=O)N2CCCC2)c1 N1(C(CNC(CCC)=O)=O)CCCC1(C(=O)NCC(C)O)C(C)C C1(CC)(CC)CN(C(=O)Nc2nc(-c3ccc(F)c(F)c3)cs2)CCS1 C1(NC(C23OC(C)C(C2)C3)=O)CN(C(=O)CC(=O)N(C)C)CC2(CCOCC2)C1 C(CCCOC)(C(=O)NCc1cccc(Cl)n1)NC(C(C1CC1)OCC)=O C1(C2(O)CCC2)(C(=O)NCC#CCNC(=O)CCCCNC(=O)C2CC2)CC1 N1(CC(N2CC(N(C(C(F)(F)N(CC(=O)NCC)C)=O)C)C2)=O)CCCC1CC C1(NC(CC2(OC)CC2)=O)CC2CCC1CC2NC(=O)Cc1nc(C)no1 c1(C(N2C(C)CC(NC(C(CC#C)CC#C)=O)C2)=O)n[nH]c2ccc(F)cc12 CC(O)C(C(=O)N1CCCCC1c1cn(C(C23CC(CO2)C3)C)nn1)N(C)C Cc1cc(C)nc(-c2cn(CCCC(=O)NCC3CCOC3C)nn2)n1 C1(C)(CNC(C2CCN(C(CCOCC)=O)C2CC)=O)CC2CCC1C2 c12cccc(n1)C(=O)N2.C1(SC)CCCC1C(=O)NC1CC1C(=O)N(C)C1CC1 C(C(N=c1nc(C2CC2)[nH]s1)C1CCC1)NC(c1ccc(Cl)cc1)=O C1(C(N(CCNC(CCCNC(=O)OC)=O)C)=O)CCCCC(=O)N1 N1(C(CCC(C)(C)NC(CCC(C)N(C)C)=O)=O)CCCC2(CCC2)C1C C(C1=NOC2CN(C(C3(F)CCCC3)=O)CC12)NC(c1cccc(CO)c1)=O c1(C(N(CCNC(c2c(C)cncc2)=O)C)=O)coc2c(F)cc(Cl)cc12 N1(C(C(C2CCCC2)OCC)=O)CC(OC)CC1CNC(C1(O)CC1)=O c1(C(N2C3CC(NC(C4CCN(C)C4=O)=O)(C3)C2)=O)ccc2cc(Cl)ccc2n1 Cc1[nH]ccc1C=CC(=O)N(C1CCC1NC(=O)CC1CC1)Cc1ccccc1F C1(C(N2CCC(C)(O)C2)=O)CCCCCN1C(=O)C=CCN1CCCC1 N1(C(c2cc(COC)no2)=O)CC(CNC(c2c[nH]nc2OC)=O)C(O)C1 C1(C)(C(=O)NC2CN(C(c3c(C)c(F)ccc3)=O)C2)CCOC12CC2(F)F c1(C(N(C(CNC(CC(C)OC)=O)C)C)=O)[nH]cc(C(C)=O)c1C C1(NC(C(CCN(C)C)NC(C)=O)=O)CC(F)CN(C(C)=O)C1 Cc1cc(C(=O)N(CCCN(C(C2CC2F)=O)Cc2ccccc2)CC)sc1C c1(C(=O)OC(c2cc(C)sc2C)C)ccc(Br)cc1F N1(C(c2ccc(OC)cc2Cl)=O)CC2(CCCN(C(=O)Cc3csc(C)n3)C2)C1 C#Cc1cccc(C(=O)NC2C=CC(C(=O)Nc3cnc(C)c(C)c3)C2)c1 Nc1cc2[nH]cnc2cc1C(N1CCOC(CCNC(c2ccns2)=O)C1)=O C(CC(=O)NCc1ccccc1Cl)(C(F)F)NC(C(CO)OC)=O C(=O)(C(C)(C)C(F)(F)F)NCCC(C)N(C(=O)C1=NOC(C)(C)C1)C C(=O)(C(C)C1=CCCC1)NC(CN(C(c1cc(CC)ncn1)=O)CC)CC CCC(C)(CO)C(=O)N1CCCC1Cn1cc(-c2nnc(C(=O)O)s2)nn1 C1(C(N(CCNC(c2ccccc2SC(C)C)=O)CC)=O)CCC12CCCO2 C1(=CCNC(Cc2n(C)ncc2)=O)CCN(C(=O)CCNC(=O)CC2CC2)CC1 N1(C(=O)CSCc2ncc[nH]2)CCN(C2COCC2NC(=O)CCCF)CC1 c1(CCC(=O)NCCCN(C(c2ncsc2C)=O)CC)ccc(F)nc1 c1(NC(C2CCCN(C(C3(C(=O)OC)CC3)=O)C2)=O)ccc(F)c(F)c1Cl c1(OCCC)ccc(C(=O)NCCCCC(C)NC(C2(O)CCSC2)=O)cc1 N1(C(c2c(C)nn(C)c2C)=O)CCCC2CN(C(C3(C)CCC34CCC4)=O)CC12 N1(CC(=O)NCC(CCOC)O)CCN(C(=O)C(C)O)CC1 c1(C(N2CCC3(C(C(=O)Nc4cc(CC)no4)C3)C2)=O)nccc2[nH]ccc12 c1(C(=O)NCC(CN(C(C(CN(C)C)O)=O)C)O)sc(F)cc1Cl N1(C(c2cc(C(C)=O)no2)=O)CCN(CC(C)NC(=O)CSC(C)(C)C)CC1 CC(C)CC(CO)NC(C1CCC(C2CC2)N1C(=O)Cc1cccnc1F)=O N1(C(=O)NC2CCCN2C(C2CC2C(F)(F)F)=O)CCN(CC(F)F)CC1 N1(C(C(C)CNC(=O)N(C)C)=O)CCC(C)C(C(=O)OC(C)(C)C)C1 N1(C(c2nc(OCC)oc2)=O)CCN(C(c2cc(COC)on2)=O)CC1C C(=O)(C(C)N=[N+]=[N-])NC(CC(=O)NC(c1ccco1)COC)C1CC1 CCC(CC)CCCC(=O)NCC1COCC1NC(=O)C(C)(C)C1CCCCO1 c1(SC)cccc(-c2cccnc2C(=O)Nc2cnn(CCO)c2)c1 N1(C(C(CC)=CC)=O)CC=C(C(=O)NCC2CCC(C)(CC)O2)C1 C1(C(=O)NCC(C)(O)CNC(=O)CCn2ccnc2)CSC2(C)CCC(=O)N12 C(C(CC(C)C)NC(=O)CC1CN(C)C1)NC(COC(CC)(C)C)=O N1(C(c2cc(C)sc2Br)=O)CCCC12CCN(C(=O)C(F)(F)C(C)O)C2 c1(C(N(C2CCCN(C(=O)Cc3cn(C)cn3)CC2)C)=O)ccccc1C#N c1(C(N(C2CCN(C(=O)C(O)CCS(C)=O)CC2)C)=O)nnn2c1CSCC2 c1(C(=O)NC2CC(C(=O)NCCOCCOC)C2)cncnc1C C(N=c1nc(N2CCCC(CO)CC2)c2c([nH]1)CCCCC2)C.CC1C(N)C1(F)F c1(OC)ccnc(C(=O)NCC(CNC(c2ncnc(O)c2F)=O)OC)c1F N1(C(C=CC(=O)N(C)C)=O)CCN(C(=O)C(C)(C)C)CC1c1cccc(F)c1 CCS(=O)c1ccccc1C(=O)N(C)CC1CCN(C(C2(COC)CC2)=O)C1 C1(NC(c2c(C)n[nH]c2C)=O)CCN(C(C23CCC2C3)=O)C12CC2 N1(C(C(CCC)N(C)C)=O)CC(CNC(=O)CNC=O)CC12CCC2 c1(C(=O)NC(CN(C(=O)CCC2CCOC2)CC)C)cc2cccc(Br)n2c1 C1(C(N2CCCC2CCNC(C2(F)CC2)=O)=O)CC2CCC1CC21OCCO1 c1(NC(CC(=O)NC2C(NC(COC3(C)CCCC3)=O)COC2)=O)ccc(F)cc1 N1(C(c2cc(C)c(O)cc2)=O)CC(NC(=O)C=Cc2ccc(Cl)s2)CC2(CC2)C1 c1(C(N2CC(C)C(CNC(=O)CSC(C)(C)C)C2)=O)cc2c(ncn2C)s1 c1(C(N2CCN(c3cccs3)CC2)C(=O)NCCC)nccc2cc(Cl)ccc12 C1(C(N(C(C)C(=O)OC)CCC)=O)CC2CCC(C1)N2C(c1cnc(C)c(C)c1)=O N1(c2ccc(S(=O)(=O)N3CCCC3)nc2)CCc2cc(F)cc(Cl)c2C1 C1(NC(C2(NC(C)=O)CC2)=O)CN(C(=O)CCc2ccc(Cl)nc2)CC1O C1(CCCC(=O)OC(C)(C)C)CCCCN1C(N1C(C(C)O)CCC1)=O CC1CC2(CC2)CN1Cc1cc(-c2ccccc2)no1 C#CCCC(O)C(=O)NC(C1CCCC1)CNc1cc(C(=O)OC)nc(C)n1 C1(NC(c2cnc(C)n2C)=O)COC2(C1)CN(C(C1CCCN1C1CC1)=O)C2 CC1(CNC(c2csc(C(F)F)c2)=O)CC(NC(C2(C3CC3)CC2)=O)C1 C1(O)(C(C(=O)NCC2C(CNC(=O)Cc3csnn3)C2)(F)F)CCCCC1 n1(C(C)C)nnc(C(C)NC(N2CCC(OCC34CC(CN3)C4)C2)=O)n1 C(N=c1[nH]c(=NCC2(CN(C)C)CC2)c2ccccc2[nH]1)c1nc(OC)sc1 c1(CC#N)ccc(C(=O)NCCCN(C(=O)Cc2ccccc2)C2CC2)cc1 O=C1Nc2cc(C(=O)NC3CCN(C(c4c[nH]nc4F)=O)CC3O)ccc2C1=O C(=O)(C(CC)(CC)CO)NCC(CC)NC(c1ccnc(OC(C)C)c1F)=O C1(CC=C)(C(=O)NC)CCCN1C(=O)CCN1CCCC1=O.C(C(F)(F)F)=CC C(C(CNC(=O)CC1CC(F)C1)C(F)(F)F)NC(C1(OCC)CCCC1)=O Cc1cc(Cl)cc(C(=O)NC(CNC(C2CC(C(C)C)=NO2)=O)C(C)(C)C)c1N C1(CCNC(CC2(C=C)CCC2)=O)CN(C(C2CCC(=O)C2)=O)CCO1 c1(NC2(CO)CCCN(C(C(CSC)(C)C)=O)C2)ncnc2sc([N+](=O)[O-])cc12 Cc1ncnc(C)c1OCC(=O)NC(C)(CNC(=O)CC1NC(=O)NC1=O)CO N1(C(C(C)=C(CC)C)=O)CCC(CNC(c2ccc(C(C)O)cc2)=O)(COC)C1 c1(C(N2CCC(OCC3CC3)C2)C(=O)NC)nc(C)c(C(C)(C)C)s1 c1(OC)ncnc(C)c1NC(=O)OC(C)(C)C.c12cncc(c1)C(=O)N2 c1(C(=O)NCCN(C(C2C(C)OC(C)C2)=O)C2CC2)cc(N)cc2c1OCCO2 N1(C(C)C)CCC(CC(=O)NC(C)C(C)NC(c2ccccc2)=O)CC1 C1(CCN(C)C)CCN(C(C2CC2CNC(c2cn(C)cn2)=O)=O)C1 c1(C(=O)NC2(C3N(C(C4(C)CCCO4)=O)CCCC3)CC2)c(Cl)nc2ccccn12 N1(C(C(F)=C(C)C)=O)CC2CCC(C(=O)NC(C3CCCC3)CC)(C2)C1 c1(C(=O)NC2C(NC(CC(C)C)=O)CCC2)cc(NC(=O)OC(C)(C)C)ccn1 c1(C(=O)NC2(C)CN(C(c3c(C)nccn3)=O)C2)cncc2nc[nH]c12 c1(CN(C=O)NC(=O)OCC)cccc(CO)c1.c12nc(cs1)SCC2 C(=O)(CCC(=O)NCCCC(C)NC(=O)C(C)N(S(C)(=O)=O)C)NCCC c1(NCC#CCNCc2cn(CC=C)nc2)sc(C)cc1C C1(CNC(C2CCN(C)CC2)=O)(NC(c2cnn[nH]2)=O)CCC(F)(F)CC1 C(=O)(C1=CS(=O)CCC1)N1CC(C)(N)C1.C(C(=O)Nc1ccccc1)(C(C)C)SC N1(CCC#C)CCC(C(N2CCOCC2CNC(C2(CC3CC3)CCC2)=O)=O)CC1 C(N=c1nnc(CC)c(OC)[nH]1)C1CN(C(Cc2c(CC)cccc2)=O)CC1C CN1N=C(CC(=O)N2CC(NC(c3ccoc3Br)=O)C(C)(C)C2)CC1=O N1(C(C2C(C(=O)OC)C2)=O)CCC(C2CC2NC(C2(CC(C)=O)CCC2)=O)CC1 C(=O)(C1COc2ccc(Cl)cc21)NC(c1cn(-c2c(C)ccnc2)nn1)C C1(NC(C(C2CC2)OCC)=O)CC1C1CCCN(C(=O)C2=CCCCC2)C1 c1(NC2C(c3ccc(OC)cc3Br)OCCC2)cc(C=O)ccc1OC C1(C(N(CC)OC)=O)CCC2(CCN(C(c3cc(CO)ccn3)=O)CC2)O1 c1(OCC(=O)NC)ccc(C(=O)NC2CC(CCl)C2)cc1 CS(C)(=O)=NC(=O)C(=O)N1CCN(C(C2Cc3cccnc3C2)=O)CC1 C1(C(=O)NC2CC(CCC(=O)N(CCOCC)C3CC3)C2)OCCOC1C N1(C(c2c(CC)noc2)=O)CCC(CNC(c2scc(C)c2OC)=O)(SC)CC1 n1(CC)cnc2c(NC(CN(C)C)CCO)nc(N3CCC=C(C)C3)nc12 c1(NC(C2CN(C(c3c(OC)csc3)=O)C2)=O)cc(C)c(Br)cc1F c1(C(=O)OCC(=O)NC2C(C(=O)OC)CCC2)nc2ccccc2nc1C C1(C(=O)N(c2ncncc2Cl)CC(F)F)CSc2ccccc2O1 c12ccccc1CO2.c1(CC(=O)NC(CN(C(C(C)OC)=O)C)C)ccccc1 c1(OC)ccc(CN2CCCC(C(=O)N(C3CCOCC3)C)C2)cc1[N+](=O)[O-] c1(C2C(CNC(=O)NCC)CC2)ccc(C)cc1.c12csc(n1)COC2=O C1(C)(CC(N2C(C)(C(C)C)CC2)=O)CCN(C(c2ccon2)=O)C1 n1(CC(=O)NC(CCCNC(CC2(COC)CC2)=O)C)cnc2c1CCCC2 C(C)(CN(C)C)(C(=O)N(C1CCCC1C#N)C)NC(C(N1CCOC1=O)C)=O C1(N(CCCO)CC2CN(S(C)(=O)=O)C2)CC2(CC2)C1 N1(Cc2c(C)nn(C)c2)CCCC(NC(c2ccc(Cl)c(Cl)c2)=O)CC1 O=C(CCC[N+](=O)[O-])N1CCN(C2CCCN(C(C3CCCCCO3)=O)C2)CC1 c1(C(=O)NC2CCC(N(C(CC(C)CF)=O)C)CC2)cnc(O)n(C)c1=O c1(NC(c2c(NC)nsc2)=O)nc(Cl)ccc1C(=O)NCCC1CCCCO1 C1(O)(C(C)NC(CNC(CC)=O)=O)CCN(C(=O)C(C)(C)C2CC2)C1 c1(N(C)C)ccc(N2CCN(C(C3(C)COC(=O)C3)=O)CC2)cc1Cl C(CC(C(=O)NC1CN(C(c2ccc(F)cc2)=O)CC1F)NC=O)SC Cc1cccc2cc(C(=O)NCCC(C)NC(C3(C(C)C)CCCO3)=O)oc12 CC1CCCN(C(=O)C=CC(=O)N(C)C)C1CCNC(=O)COC1CCCOC1 c1(C(N2CCC(C)(NC(Cc3c(C)noc3)=O)C2)=O)ccc2nonc2c1 CCS(=O)(=O)CC(=O)N1CCC1C(N1CCOC(C)CC1)=O N1(C(C2CC(C)CN(C(=O)C(C3CC3)C3CC3)C2)=O)C2CCC1CC(F)C2 C=Cc1cc(C(=O)NCCOCCCN(C)C(C2(CC(F)F)CC2)=O)cc(F)c1 CC1(CO)CN(C(c2ccc(NC(c3ccc(Br)c(Cl)c3F)=O)s2)=O)CCC1O N1(C(CC2C(CC)C2(F)F)=O)CCC(NC(=O)CC(F)(F)F)C(F)(F)CC1 C(=O)(C1c2ccccc2C2CC1C2)N1CCC(F)(CNC(C=CC)=O)C1 N1(C(C(CN(C)C)NC(C)=O)=O)CCCCCC1CNC(=O)C(O)C(C)C C1(CNC(CCSC)=O)CN(C(C2CC(N=[N+]=[N-])C2)=O)CCO1 C1(F)(C(=O)NC2(CC=C)CN(C(C3CCOC3C=C)=O)C2)C(C)(C)C1(C)C N1(C(C=C(COC)C)=O)CCC2CCCC12CNC(=O)Cc1cc(C)no1 N1(C(CCOCC)=O)CC(NC(=O)C(C)(C)CN2CCN(C)CC2)C(C)C1 N1(C(C=C(C)Cl)=O)CC2CC2C1CNC(=O)Cc1sc(O)nc1O N1(C(c2cc(C)c(Cl)s2)=O)CCOC2(CCCN(C(C3CC3F)=O)C2)C1 c1(OC)ccccc1C(C)C(=O)NCC1C2CN(C(=O)CCCC3CC3)CC12 C1(C(=O)NC2CCC(N(C)C)C2)CC2CC2N1Cc1cnn(Cc2ccccc2)c1 CCC(C)C(C)C(=O)NC(C1CC(NC(C2(CC3CC3)CCCO2)=O)C1)C C1(NC(C2(C#C)CCC2)=O)CCC(C)(CNC(C23CC(F)(C2)C3)=O)C1 C1(C2CCN(C(c3cccc4sccc34)=O)C2)(NC(CC=CC=C)=O)CC1 C(=O)(C1=C(F)CN(C(=O)CCCCCF)CC1)Nc1c(OC)cccc1 C=CCC(C)C(=O)NC1CC(C(C)NC(C2CCCC2(C)C)=O)C1 C1(C(N2CCC(=CCNC(=O)CC3COCCN3C)CC2)=O)(OC)CCCSC1 C(=O)(C1=C(C#N)CCC1)NCC(C(=O)NC(COC)C(=O)N(C)C)C c1(CN(CCNC(C)=O)CC)cnn(C)c1O CN1C(=O)C(=O)N(CC(=O)NC2CCN(C(C3CCCOC3)=O)C23CC3)C1=O CCC(C)(C(=O)NCCC1CCN(C(c2ccc(Br)o2)=O)C1)C(N)=O C1(NC(C(C(=O)OCC)F)=O)CCC2(CC1)CC2NC(=O)CCNS(C)(=O)=O CCCC(O)CC(=O)N(CC(C)(C)CNC(=O)CCC)C c1(Oc2cccnc2F)cc(F)cc(Br)c1Cl.N12CCCC1Cn1cc(nn1)C2 C1(NC(C(C=CCCC)O)=O)CCCN(C(=O)CC2(N(C)C)COC2)CCC1 N1(C(C2C(C)CN(C(=O)Cn3cnnc3O)CC2)=O)CCC(C2CCOC2)C1 C1(CN(C(=O)C(O)CC2CCOCC2)C)CCCN1C(c1csc(Br)c1)=O C1(CNC(c2c(COC)n(C)nc2)=O)CCN(C(=O)CN(C)C(=O)OC)CC1O N1(c2nnc(C(c3occc3)N3CCCC3)n2CC2CC2)CC(C)OC2(CCC2)C1 CON(CCC(=O)NCCCSC(F)F)C(=O)C1CC1(C)C c1(NC(CNC(c2nc(C)c(C)s2)C)=O)cc(F)cc(F)c1 C1(OC)(OC)CC2CC(C(c3nnnn3C)NC3CCCCCC3)CC2C1 C1(CC)CN(C(=O)C=CBr)CC1NC(=O)C(c1cnn(C)c1)O C1(NC(N2CC(CS(C)(=O)=O)OCC2)=O)CCCCCC1F C=Cn1nccc1C(=O)NCc1csc(CNC(c2cc(C)sc2N)=O)n1 C(=O)(CCC(C)(C)C#N)NCCC1CN(C(C2(CC(C)C)CCC2)=O)C1 N1(C(C(C)OC)=O)CCCC(C2CN(C(=O)Cn3cc(Br)cn3)C2)C1 Cc1cc(C(=O)NCCN(C(=O)C2=CCCC2C)C2CC2)c2[nH]cnc2c1 C1(NC(c2cc(-c3ccccc3F)no2)=O)CCCC(CO)CC1 c1(C(=O)NCCCCC(C)NC(c2cc(Cl)nnc2O)=O)ccc(F)c(F)c1F C1(CN(C(c2cnc(O)o2)=O)CC)CCN(C(c2cc(C(C)(C)C)no2)=O)C1 N1(C(CN(CC#C)C(c2cnncc2O)=O)=O)CC(C)(C)C1COC N1(C(C=C(C)C)=O)CCN(C(=O)Cn2nccc2C)C(c2nccn2C)C1 CC1CN(C)CC1NC(C1OCCC1CNC(c1nnc(S)n1C)=O)=O CC(=O)CC(C)(C)C(=O)NCc1cccc(NC(C23CCCC2C3)=O)c1 N1(C(=O)C(F)=C2CCCC2)CCC(Nc2nc3cccnc3s2)C2(CCC2)C1 C(=O)(C#CC1(C)CCCO1)N1CC(C(C)C)N(C(c2cnn(CCF)c2)=O)CC1 Cc1ccc([N+](=O)[O-])c(C(N2CC3CC3(CNC(c3cncnc3)=O)C2)=O)c1C N1(C(C(c2scc(C)n2)(F)F)=O)CCC(O)C(NC(C2(C)CNC(=O)C2)=O)C1 c1(C(=O)NCC(CNC(C(C)OCC)=O)(C)O)cc(OC)c(OC)cc1F CN1CC(C)(C(=O)NCC2(CNC(c3csnn3)=O)CC23CCC3)CC1=O c1(C(N(CCOCCC(=O)OCC)CC)=O)cc(C(C)=O)on1 c1(OC)cccc(C2CC2C(N2CC(CO)(CC3(C(F)(F)F)N=N3)C2)=O)c1 c1(C(=O)NC2C3(CN(C(CCC(C)OC)=O)C3)CC2)cc(Cl)c(F)cc1Cl C(C(=O)NCC1CC(=O)N(C2CN(CCn3ccc(C)n3)C2)C1)(C(C)C)SC C(CC(C(=O)N1CCC1CC(=O)OC)NC(=O)CC(C)(C)C)OC N1(C(CSC(C)C)=O)C2CC1CN(C(c1ccoc1)=O)C2 C12(NC(=O)CN3C(=O)CNC3=O)CCN(C(c3ccncc3C(F)F)=O)CCC1C2 C=CC1(CC(=O)NCc2ncccc2C)CN(C(C2(OC)CCOC2)=O)C1 Cc1nc(C)sc1C(=O)O.C(C1CCCO1)=C.C12CN(C1)C2 N1(C(C2C(C(C)NC(c3ccc[nH]3)=O)C2)=O)CC2CC3CC2C1C3 N1(C(C(C(C)C)O)=O)CCC2CN(C(=O)Cc3cc(Br)cs3)CC2C1 C1(NC(c2c(CC)nns2)=O)CCCCCC1C(=O)NCC(C)C1CC1 c1(C(=O)NC2(CNC(c3cnn(C)c3CO)=O)CC2(F)F)cccc([N+](=O)[O-])c1 c1(C(N2CC3C(CNC(C4CC4F)=O)(C3)C2)=O)cccc(F)c1C1CC1 O=C(CCCCC(F)(F)F)NCC1CCN1C(c1cccn1C1CCCC1)=O C1(C(=O)NC(c2c(CCC)nns2)C)CCN(C(=O)C(=O)N2CCOCC2)O1 c1(CNC(=O)NCC(c2cccc(N(C)C)c2)O)cccc2c1OCCCO2 Cc1ccc(OC(=O)C(C)C2CCC2COC(=O)COc2ccccc2)c(O)n1 c1(CC(=O)NC(CCNC(C2(CC)CC2(F)F)=O)(C)C)ccccc1OC c1(C(N2CC3C(CNC(c4ccncc4)=O)(C3)C2)=O)cc(F)cc(F)c1Br c1(OC)cccc(C(=O)NCC(C2CCCC2)NC(=O)C=CC2CCOC2)c1N CC(CN(C)C)CC(=O)NCC1(F)CC(NC(=O)C=CC(=O)N(C)C)C1 N1(C(C(C)Oc2cccc(CO)c2)=O)CCOCC(CNC(C2CCCN2C)=O)C1 c1(NC(c2ccc(CSC)nc2)c2nnnn2C(C)C)cc(C(N)=O)ccc1C N1(C(C(C(COC)C)C)=O)CCCCC1C1CCCN1C(C1CCOC1)=O Cc1ccc(C(=O)NCC(F)CNC(=O)CCc2c(C)n[nH]c2C)c(O)n1 Cc1nn(C)c(C)c1CC(N1CCCC1CN(C(=O)Cc1cnc[nH]1)C)=O c1(C(=O)NCC2C(NC(CCC=CC)=O)C2)cccc([N+](=O)[O-])c1NC C1(OC)CC2(C(=O)N(CCC(C)NC(c3cccn3C(C)C)=O)C)CC12 c1(CC)ccccc1CCNC(=O)Nc1coc(SC)n1.C12(CC)CC(CO1)C2 C1(C#N)(C(=O)NCC(C)CNC(=O)C=Cc2cnc[nH]2)CC2CC2C1 N(C)(S(=O)(=O)N(C)C)CC(=O)NCC1(F)CC(NC(C2C(C)(COC)C2)=O)C1 C1(CC)CN(C(C2(CC)CCCO2)=O)CCC1NC(c1nc(C)no1)=O c1(C(=O)NCC2CC(NC(c3cnc(=N)[nH]c3)=O)C2)cccc(Cl)c1Br Cc1ccc(SCC(=O)NCCN2CCN(C(C3CC3F)=O)CC2)cc1 C(=O)(C(C)CC(C)C)COCCOCCN(C(=O)C(CC)OCCCOCC=C)C Cc1ccc(CNC(=O)C(=O)NCc2ccc(O)cc2F)c(F)c1F C1(CC)(NC(c2cccc(N)n2)=O)CCCN(C(=O)C(CC)c2ccccc2)C1 C(CCCS(C)=O)NC(C(C)NC(COC)=O)=O CC(C)C(CNC(c1cccn1Cc1ccccn1)=O)NC(=O)CC(C)F c1(C(N2C(C)(CC)CC(NC(=O)C(C)(C)C)C2)=O)c[nH]c2ccc(F)cc12 C1(CNC(CC=CCC)=O)CN(C(c2cnc(C3CC3)[nH]2)=O)CC12CCC2 C1(C(=O)NCC(F)CO)CCCN1NC(=O)CSC1CCSCC1 C(N=C(NC(C1CC1)C1CC1)N1CCOC(C2CCC2)C1)c1c(CC)n(C)nc1.C1CC1 c1(C(N(CC(CNC(C(C2CCC2)OC)=O)O)C)=O)conc1C1(C)COC1 C(=O)(C(CO)C(C)(C)C)N1CCC(C(C)C(=O)N(C)Cc2ccco2)C1 N1(C(c2cc(C)nc(O)c2)=O)CC2CCC(C(=O)N(C)C3CC3)C2C1 c1(C(N(CCN(C(CCN(CCC)C)=O)CC)CC)=O)cccc(C)c1 C#Cc1ccc(C(=O)NC(C2CCCN(C(=O)Cc3cccs3)C2)C)cc1 C1(OCC)CCC2(CC1)CCN(C(=O)N=c1cnn(Cc3ccc(Cl)cc3)[nH]1)C2 Nc1c(-c2noc(C3CCCN3c3cccnn3)n2)cnn1-c1ccccn1 N1(C(=O)OC(C)(C)C)CCC(OC(CC(C=C)O)=O)C2(CCC2)C1 N1(C(C=C(C)C)=O)CCC(N(C(=O)CN2CCCCC2=O)CC2CC2)CC1 N#Cc1c[nH]c2ncnc(N(C3CNCCOC3)Cc3nc(Br)ccc3F)c12 C1(O)(CNC(C(=O)N(C)C)=O)CCN(C(=O)CC(F)(F)F)C1 N1(c2c(C)cncn2)CC2CC(NC(=O)Cc3ccc(S(C)=O)cc3)CC2C1 N1(C(CC2(C)CC2)=O)CCN(C(c2ccnn2C)=O)C(CC#N)C1 c1(-n2cc(C3(C)N(C(c4c(C)nsc4)=O)CCC3)nn2)cc(Cl)cc(Br)c1 Cc1ccc(C(=O)NCCC2CCC(C(F)(F)F)O2)c(I)n1 c1(CCO)ccccc1.c1(C=O)coc(Br)n1.CC(C(=O)N1CC(C)C1)N(C)C Cc1ccc2c(c1)CCC2C(=O)NCCC1CC1C1CC1 C1(CNC(C(n2c(C)ccn2)C)=O)CC(F)(F)CN1C(c1cccc(F)c1O)=O N1(CC(N2CCCC(C(C)C)C2)=O)CCCNC(=O)C1C c1(C(N2CC(C(C)NC(C=CSC)=O)OCC2)=O)cc(F)c(C)cc1Cl c1(CC(=O)NC(C)CN(C)C(c2cncnc2)=O)ccc2c(c1)CC2 C1(NC(=O)C(O)C2CC2)COCCN(C(=O)CCC2CCCCC2)C1 N1(C(C2N(CC)CCCC2)=O)CC2(CC(CC(=O)NCC3CCCCC34CC4)C2)C1 c1(NC(C2CCN(C(=O)CCc3cncnc3)CC2O)=O)nc(Cl)cnc1Br C1(O)(CNC(CCCCNC(N)=O)=O)CCCN(C(c2cc(O)nc(Cl)c2)=O)C1 c1(CN2C(C(N(CC(=C)C)Cc3ccccc3)=O)CC(F)C2)ccc(Br)c(F)c1 C12(NC(c3nc(COCC)sc3)=O)CCCC1CN(C(C1CC(SC)C1)=O)C2 CCC(CC(=O)NCCCC(=O)Nc1ccc(O)cc1)C(C)C c1(C(N(C(C)C)CCNC(=O)C(C)n2cccn2)=O)ccc(O)c2ncccc12 Cn1cnc2c(NCc3nc[nH]n3)nc(N3CC(C)(C)OC4(CCC4)C3)nc12 C1(C(=O)NCCC2(OC)CN(C(=O)Cc3nnc(C)s3)C2)OCCN(C)C1=O S(=O)(=O)(c1c[nH]ccc1=NC1CCN(C(C)C)C1)NC(c1ccc(OC)cc1F)C c1(CC(=O)NC2C3CN(C(=O)CC4CC5CC4C5)CC23)ccc(F)c(Cl)c1 CC(CCC(=O)N1CCC=CC1C(=O)NC(C1CC1)C1CC1)C1CCC1 C(=O)(CC(C)(C)C(C)=O)N1CCC(NC(C2C(C(=O)OC)CCO2)=O)(CO)CC1 C1(C(=O)NCCC2(O)CN(C(CCC(=O)NC)=O)C2)CCN(S(N)(=O)=O)CC1 Cc1nc(C)c(C(N2CC(C(C)NC(=O)CC(C)(C)F)C2)=O)[nH]1 C1(NC(CC=C(C)C)=O)CCN(C(=O)C(=Cc2cccc(F)c2)F)CC1CO N1(C(c2nc(-c3cn(C)nc3)oc2)=O)CC(CNC(=O)CC(F)F)CC12CCC2 C(=O)(CC(O)CC(C)(C)C)N1CC(C)(CC(=O)NCC(C(C)C)C2C(C)C2)C1 CC(C)C(O)C(=O)N(C)CC1CN(C(C2(C)CC2(Cl)Cl)=O)C1 c1(CN(C(=O)CC2C(NC(=O)COC3CCCCC3)CC2O)C)cnnc(O)c1 c1(C(=O)NC2CCCN(C(CCc3c(C)n[nH]c3C)=O)C2)cc2n(n1)CCO2 Cc1cc(=O)c(C(=O)NOC2CN(C)CC2O)c[nH]1.C12(CCC1)C(=O)N2C1CC1 CC1CN(C(=O)Cc2cc(Br)ccc2O)CCN1C(c1cccc(=O)o1)=O C1(CC(C)(C)C)CN(C(=O)CCn2cncn2)CCN1C(C1CCCC1F)=O N1(C(C2C3N(C(COCCCC#C)=O)C(CC3)C2)=O)CC2(C1)CC(C)(F)C2 Cc1cn2ccnc(C(=O)NC3CN(C(c4cn(C)nn4)=O)CCC3C)c2n1 c1(C(c2nnnn2CCOC)NC(C(=O)NCCOC)=O)nc2ccccc2s1.C(Cl)N Cc1sc(Br)nc1-c1cn(-c2cccc(COC(C)C(=O)O)c2)nn1 N1(C(C=CCCCC)=O)CCCC1C=CC(=O)NC1CN(C(C)(C)C)C1 N1(C2N(C(C3=C(C)OCC3)=O)CC2)CCC(N=c2[nH]c3ncc(Cl)cc3s2)CC1 C1(CNC(c2ccn(C(C)(C)C)n2)=O)CCN(C(=O)COC2CCC2)CC1 C1(NC(C2CCC(=C)CC2)=O)CC2CC(NC(c3c(Cl)sc(C)c3C)=O)CC2C1 C=CC1CCCCN1C(C1CN(C(c2cn(C)c(=O)n2C)=O)CC1(F)F)=O C1(C(=O)NC2(C(=O)Nc3cccc(C4CC4)c3)C(C)(C)C2)CCCC(=O)C1 C1(C(=O)NCC(CC)NC(=O)CN(C(=O)COC)C)CCCC(F)C1 Cn1nc(C(=O)NCC(C2CC2)NC(c2ocnc2C(F)(F)F)=O)cc1Br c1(C(C2CC2(Br)Br)NCC2(CO)COC2)nnnn1CCCF c1(C(C(=O)NC2(CCNC(=O)CC3CC=CC3)CC2)F)ccc(F)cc1 N1(C(CCC(C)N(C)C)=O)CCN(C(c2ccc(C(F)F)o2)=O)C(C)C1 C(=O)(C(F)C(=O)N(C(C)C(=O)NCCCn1cc(C)cn1)C)OCC CCCC(O)CC(=O)N1CCN(C(C2(C(=O)NCC3CC3)CCC2)=O)CC1C Cc1sc(Br)nc1CNC1CCC(NC(c2ccc(Cl)cc2)=O)C1 N1(C(CC2C(C)C2)=O)CCC2(NC(=O)COCC3CCOCC3)CCCCC12 C1(NC(c2c(CC)non2)=O)CCCN(C(C23CCCC2C3)=O)C1 CC1CN(C(=O)C(C2CCOCC2)F)CC1(C)C(=O)N(C)CC1CCC1 c1(C(=O)NC(c2cn(CC3CCCO3)nn2)CCC)cccc2c1CNC2=O CC(C)(CCCC(=O)N1CCC(=C(F)F)CC1)NC(=O)C=Cc1nccs1 C1(C)(C(N2CC(C(C)NC(C3CC(OC(F)(F)F)C3)=O)OCC2)=O)CCC(F)(F)C1 c1(C(N(CCNC(C(COCC)C)=O)CC2CC2)=O)cccc(S(=O)(=O)CF)c1 C(CC(C)(C)CC(=O)N(C1CCCC1)CCCNC(c1cc(C2CC2)on1)=O)OC C(CC(=O)NC1CCCC(NC(c2cscc2Cl)=O)C1)(C(N)=O)NC(C)=O c1(NC(C(C)Oc2ncccc2-c2ccc(F)s2)=O)ccccc1C#N C(=O)(CCCCCCCO)Nc1cccc(C(=O)OC)c1.c12cn(nn1)CCS2 CCCC(C)(O)C(=O)NCC1CCCC1C(=O)NC1CNC(=O)C1 C(=O)(C(C)(C)CS(C)(=O)=O)N1C(CNC(c2cc3nnn(C)c3s2)=O)CC1 c1(C(N(CC(C)NC(C(C)CC(F)(F)F)=O)C)=O)coc2c1NC(=O)CCC2 c1(OC)cc(C(=O)NCc2cc[nH]c2C(=O)NC2CC(CO)N(C)C2)n(C)n1 Cc1cnc(NCC(C)Cc2cccs2)c(S(=O)(=O)NC(c2nccn2C)C)c1 C12(C(N(CC(C)(C)C)CCO)=O)CC1CN(C(=O)Cn1cccc1)C2 c1(C(N2C(CN(C)C(C3(C)CCC(=O)N3)=O)CC2)=O)cc(Cl)c(N)c([N+](=O)[O-])c1 C1(C2CCN(C(c3cc(C4CC4)nc(Cl)c3)=O)CC2)(NC(=O)CCC2CC2)CC1 C(=O)(C1=C(C)OCCC1)NC(CC)CNC(=O)CN1C(C)CCC1C c1(C(=O)NCC(CC)(CC)NC(C2CCCS2)=O)c(Cl)cncc1Cl CCC(F)(F)CC(=O)NC1CN(C(C2(c3ccc(F)cn3)CC2)=O)CC1F N1(CC2(c3cn(CCC(c4ccc(C)cc4)(C)C)nn3)CC2)CC(=O)NC(=O)C1 Cc1ccc(OCC(=O)NCC2CC(NC(c3cc(Br)[nH]n3)=O)C2)cc1 c1(CC)cc(NC(=O)C(C2CC2)NC(C2CCC3(CC3)C2)=O)ccc1C C12(NC(CCN(C)CCO)=O)CC(C1)N(C(c1ccc(NS(N)(=O)=O)cn1)=O)C2 C1(CNC(C(COCC)n2cc(Cn3cccc3)nn2)=O)CC(C(C)(C)C)=NO1 C(=O)(C1=C(F)CN(C(=O)CC(C)c2ccco2)CC1)N(CC(C)C)CCOC N1(CC(=O)NC2(C(=O)NC3CC3C(F)(F)F)CCCCC2)CC(=O)NC1=O N1(C(c2cccc(CCC)c2)=O)CCC12CN(C(=O)C(c1ccnn1C)O)C2 Cc1cc(NC(c2cc(Br)sc2C)=O)ccc1NC(C1CCCO1)=O C1(NC(CCC=CC(C)C)=O)CC=C(C(=O)NC(C)(C)CO)C1 c1(CNC(C(N(C(C(C)NC(CC)=O)=O)C)C2CC2)=O)cc(C)ccc1F N1(C(C=Cc2cn(C)nn2)=O)CCN(C(=O)C2CC2)C2(CCC2)C1 c1(C(=O)NC2CCC(CCNC(CC3(C)CC3)=O)C2)cc(C(N)=O)ccn1 c1(C(N2C(CN)CC(C)(C)C2)=O)cc(F)cc2cccnc12 Cc1cc2c[nH]nc2cc1C(=O)NC(C)CNC(c1c(F)ccc(C(F)F)c1F)=O c1(C(=O)NCC(CNC(C(C(=C)C)(C)C)=O)F)cc2ccc(SC)cc2[nH]1 C1(C(=O)OCC(c2ccc(N(C)C)cc2)=O)CN2CC(CCC2=O)O1 Cc1ncc(C(=O)NC(C)CNC(C2(C)CC=CCC2)=O)cc1Cl N=c1c(C(=O)NC2CCCC(NC(=O)C=Cc3ccncc3)C2)c[nH]cc1Br N1(C(C)=O)CCCC1C(=O)NC(C)CC(=O)NCc1nc(N(C)C)n[nH]1 c1(NCCSC)cc(O)cc(=O)o1.N12CCOC(C1)CN(C)CC=CC2=O c1(CC)[nH]nc(Cl)c1C(=O)NCCNC(=O)Cc1scnc1C1CCCC1 c1(C(=O)NC2(CO)CC2)ccc(F)c(N2CCC2)c1 C(=O)(C1=NOC2COCC12)NCC(C)N(C(c1c(C)c(F)cc(Br)c1)=O)C N1(CC(COCCCC)O)CCC(N2CCCC2=O)CC1 C1(NC(c2cnn(C)n2)=O)CN(C(c2ccc(F)cc2F)=O)CC2CCCC12 Cc1cnn(C)c1C(=O)NCC1(C(C)NC(=O)Cc2cc(C3CC3)no2)CC1 C(C(C)C(F)C(=O)NOCCCN(C)C)NC(c1c(OC)nsc1)=O c1(OC)cc(C(=O)NC2CC2CNC(=O)C=C2CCC2)cnc1OC.C1(C)CC1 Cc1ccc(C(N2CCC(O)(C(C)NC(=O)Cc3cnnn3C)C2)=O)cc1F c1(CC(=O)NC2C(NC(c3cnc(C)[nH]3)=O)CCOC2)cccc(C)c1Br N1(C(C(CC2CN(C(C3CC(=C)C3)=O)C2)F)=O)CCCC(C)(C)C1C N1(C(C(C#C)(C)C)=O)CC2CC(NC(c3ccc4c(c3)CC4)=O)C(C2)C1 Cc1sc2ncc(C(=O)NCC3(CNC(C4CCC5C4C5(F)F)=O)CC3)n2c1C C1(C(N(C(c2ccccc2)C)C)=O)CCCN(C(c2cc(Cl)ns2)=O)C1 C12CCN(C1CC)C2=O.CCC(COCC1CC1)NC(C1CN(C2COC2)C1)=O c1(C(=O)C(=O)C2CC2)[nH]c2cc(CNc3cc(OC)c(Br)cc3)ccc2c1C CCC(CN=c1cc(C)nc(NCCOc2ccc(F)cc2)[nH]1)OC.OCC C(=O)(C1=CCCCC1C)N(CC=CC(=O)N(CCn1c(C)ncc1)C)C C1(C(N2CC(n3cc(C4C=CCCC4)nn3)C(O)C2)=O)CCCC2(CC2)C1 C1(COC)(CNC(c2ccc(C(C)(C)C)s2)=O)CCN(C(C2CC2[N+](=O)[O-])=O)C1 CC1CCCCN1CCC(N1CC(O)CC1CNC(c1cnc(S)n1C)=O)=O C1(C(C)C)CCOC1C(=O)NC1CCC(CCNC(=O)C2CC2)C1 C(C12CCSCC(CC1)C2)NC(CCO)c1nccs1 C1(C(=O)NCC2CC(OCC)C2)C2CN(C(=O)C(c3ccccc3C)C)CC12 c1(C(N2C(CNC(CC3ON=C(C)C3)=O)CC2)=O)cc2c(C)cc(C)nc2s1 C(=O)(CS(N)(=O)=O)NCC1N(C(CN(C)C(c2ccccc2)=O)=O)CC=C1 N1(C(CC(=C=C)C)=O)CCC2CN(C(c3ccc(CO)nc3)=O)CCC12 C(c1ccc(C)c(Cl)c1)=CC(=O)NCC1CCCN(C(C(CCC)(C)O)=O)C1 CC1(C)CCc2cc(Br)ccc2N1C(=O)NC12CCCC1NC(=O)CC2 c1(-c2ccc(CC(N3C(C(=O)OCC)CCCC3)=O)nc2)ccc2c(c1)CC2 c1(NC(c2c(C(C)NC(Cc3cc(CC)no3)=O)noc2)=O)ccc[n+]([O-])c1 C(CCCCC(=O)N1CC(O)CC1(C)C(=O)NCCCNC(=O)OC)OC CCC(CO)C(=O)NC1CCN(C(C2CC2c2ccc(OC(C)C)cc2)=O)CC1 c1(C(=O)NC2CN(C(c3n[nH]c(C4CC4)c3Cl)=O)C2)cc2c(cc1O)OCO2 C12CN(CCO1)c1nnc2s1.C=CC1CC1(C(=O)OC)C(F)F c1(N2C(C)CC(NC(c3n(C(CC)C)ncc3)=O)C2)nc(C)nc(O)c1C C1(C(C)C)CN(C(C2(Cc3cccnc3)CC2)=O)CCN1C(=O)CN=S(C)(C)=O c1(C(N2C(CC(N3CC(F)C(F)C3)=O)C3CCCC32)=O)ccc2c[nH]nc2c1 C#CC1(O)CCN(C(C2CCC(O)CN2C(c2csc(Cl)n2)=O)=O)C1 Cn1ncc2cc(C(=O)NCC3CC3CNC(C3CCc4ccnn4C3)=O)sc12 CCC(C)C(O)CC(=O)N1CCCC(C)(C(=O)NC2CC3(CCC3)C2O)C1 c1(C(=O)NCC2CC(NC(C(CC#C)C)=O)C2)c(Cl)ccc([N+](=O)[O-])c1Cl CCC(CC(=O)N(CCC(N1CC2(CCC2)CC1CO)=O)CC)CC(C)C C=CCC(C(=O)NCCOCCCNC(c1cn[nH]c1)=O)c1ccccc1 c1(C(=O)OC)ccc(C(=O)NC2CN(C(C3(C4(C)CC4)CC3)=O)C2)c(C)c1 C1(C(N2C3CC(N(C(C(C)OCC)=O)C)CC2CC3)=O)CN(S(=O)(=O)N(C)C)C1 N1(C(C(c2ccccc2)OC)=O)CCCC1N(C)Cc1ncns1 C1(N(C(CCC=C=C)=O)C)CN(C(c2cc(SC)oc2C)=O)CC12CC2 c1(CNC(C(C)(C)OCC)=O)c[nH]nc1C(=O)NOCC1CCCC1 N=c1nc(N2CCCC(F)(F)CC2)[nH]c(=NCCN2CC=CC2)[nH]1 N1(C(C2CC(CCC)C2)=O)CC(F)CC1CNC(=O)Cc1ccoc1 c1(OC)ccc(CO)cc1-c1cccc(-c2nn[nH]n2)c1.C12CC1C(=O)N2 N1(C(CSc2n(C)ccn2)=O)CC2(CCN2C(C2CC23CC3)=O)C1 Cc1cncc(C(N2CCN(C(C3CC4(CCC4O)C3)=O)C(C)C2)=O)c1Cl C1(C(N2CC3(C(NC(CS(=O)(=O)NC)=O)CC3)C2)=O)Cc2ccccc2S1 Cc1ccnc(NCc2cc3n(n2)CCCC3)c1C#N c1(C(=O)NC2CCCC(NC(CNS(NC)(=O)=O)=O)C2)cc2ncccc2s1 Cc1cc(C(=O)NC2CCC(C)N(C(=O)CCc3cn(C)cn3)C2)c(F)cc1F S(=O)(=O)(c1cc(C)cnc1NCC(CC)CC)N1CC(N2CC(F)C2)C1 c1(NC(C2CCCC(NC(=O)CC3CCCC3)C2)=O)ccc(O)c(F)c1 CCC(C(=O)NC(C)(C)C(C)NC(=O)CNC(=O)NC1CCOCC1)C(C)C O=C(CC1CC(=O)Nc2ccccc21)NCC#CCNC(C12COCC1C2)=O C1(C)(OC)CCN(C(=O)CC(C)n2ccc(C)n2)CC1.n1(C)cccc1C(=O)OCC Cc1ncnc(C)c1NC(C1CCCN1C(=O)C(C)n1cccn1)=O N1(C(C(CCCC)(F)F)=O)C2CC=C(C(=O)NOC3CCCN(C)C3)C1CC2 c1(C(N2C(C)CC(NC(C34CCN(CC3)C4)=O)C2)=O)ccc2c(c1)OCO2 Cc1ccc2c(c1)SC(C(N1CCCC(N(C(=O)C3=C(Cl)CCC3)C)CC1)=O)C2 C(CC(O)C(=O)N(c1ccc(C)cc1)C)NC(C1(OC(C)=O)CC1)=O C1(C(C)NC(c2cnn(C3CC3)c2)=O)CCCCN1C(c1cc(CO)on1)=O N1(C(=O)OC(C)(C)C)CCN2CC(NC(=O)C(F)(F)CC(C)=O)CCC2C1 c1(C2(NC(=O)Nc3scc(C(C(=O)OC)(C)C)n3)CCC2)c(F)cncc1Cl Cc1nc2ccc(C(=O)NCC(C)(C)CCNC(C3CCOC3C)=O)cc2o1 C(C)(C(=O)NCc1csc(CNC(=O)Cc2cccnc2)n1)(C(C)C)NC(C)=O c1(-c2cn(Cc3cc(C)no3)nn2)cnn(C)c1CNC(=O)C(C)O Cc1ccc(C(C)(C)C(=O)NC2CCC2CNC(=O)C=Cc2sccc2C)cc1 c1(C(N(C2CCCN(C(C(C)C)=O)C2)C)=O)nnc(O)cc1O CCC(CC)C(=O)N1CCC(C(=O)NC2(c3noc(C)n3)CC2)(C(C)C)C1 C1(NC(C2(CC=C)COC2)=O)CCOC(CNC(=O)CC2(O)CCC2)C1 c1(CC)nn(C)cc1C(=O)NC1CC(F)(CNC(c2cccc(OC)c2)=O)C1 c1(CC)[nH]nc(C(=O)NC(CNC(=O)CC2COCCN2C)C(C)C)c1[N+](=O)[O-] c1(CC)c(NC(=O)C=CC2CCCN2C(=O)CN2CCCC2C)cnn1C CC(C(=O)NCC1CCN(C(=O)C=Cc2ccc(O)cc2)C1)C(C)(F)F N(C(=NCc1ccoc1)NCC1CC(=C2CCCC2)C1)Cc1n(C)ncc1 C1(C(N(CCCC(=O)NC(C(=O)OC)CO)C)=O)CN(C)C(=O)N1 c1(CC(N2C(C)CCC(NC(c3cnc(C)[nH]3)=O)C2)=O)cccc2ncccc12 N1(C(C(CC)CC)=O)CCC(C2CCN(C(C3(N(C)C)CC3)=O)C2)CC1 c1(OCC)ccc(C)nc1C(=O)Nc1cccc(CNC(=O)C=CSC)c1 C#Cc1cnc(=NCCCCC(C)NC(c2ncoc2C2CCC2)=O)[nH]c1 C(=O)(C(O)CCS(C)=O)NC12CC(NC(C=CC(=O)N(C)C)=O)(C1)C2 C1(C)(CCNC(C2(CC(C)C)CC2)=O)CCN(C(C2CCCCO2)=O)C1 C(=O)(CCCCC(N)=O)N1CCC2(NC(CCC(=O)NCCC)=O)C(C1)C2 Cc1cn(C)cc1C(=O)NC(C)C(c1ccccc1)NC(=O)Cc1ccn(C)n1 C(=O)(CC(O)CCSC)NC1C(NC(c2c(CC)nccc2)=O)CC1 c1(C(=O)NC2CCCCC2CO)ccc2c(c1)CCO2.C12(CC1)C(=O)N(C)C2 C=C(F)C1(CC(N2CC(C(=O)NCCNC(C3(C)CC(O)C3)=O)C2)=O)CCC1 N1(C(CSCC=C)=O)CCCC2CN(C(=O)CCCCC(CC)CC)CCC12 C1(CC)CN(C(=O)C(=O)Nc2cc(F)ccc2OCC(=O)OC)CC(C)(C)C1 c1(CC)nc(=N)[nH]cc1C(=O)NC1CC12CC(NC(=O)Cn1cccn1)C2 c1(NC(C2(CCC)CCC2)=O)ccc(NC(c2cc(OC)ccc2F)=O)c(C)c1 c1(C(=O)NCCOCCNC(CC2CCC(C)C2)=O)cc(CO)n(C)n1 C1(C2CCN(C(c3cnco3)=O)CC2)(NC(=O)COc2ccc(Cl)cc2F)CC1 N1(C(CN(C(c2ccsc2Cl)=O)CC)=O)CCCCC(F)(F)C1 CCC(CC(=O)N1CCCC1(C)C(=O)Nc1ccc2nccn2c1)CC(C)C N1(C(C(=O)NC(C)C)=O)CCC(C(F)F)(CNC(C2CCN(C)C2C)=O)C1 C12(C3C(C)C3)CC(CN1C(=O)CN1CCN(C(=O)Cn3cnc(CO)n3)CC1)C2 C(=O)(CCCC(CC)NC(=O)Cc1c(C)n[nH]c1C)NC1(C=C)CCCCC1 C1(CNC(CCC(=C)C)=O)CN(C(c2sc(C(C)(C)C)nc2C)=O)CCC1(C)C C1(N(C(c2cn(CCC)nc2)=O)C)CCCN(C(C2CC3OC2C2CC32)=O)CC1 Cc1ccc(C(C)C(N2CCCC2CC(=O)NCCCO)=O)cc1 c1(C(=O)NC(CC#C)C(=O)NCCN2CCCNC2=O)cnc(O)cc1C c1(C(=O)NC(C(C)NC(C=CCCC=C(C)C)=O)C)cc(C(F)(F)F)cc(Cl)c1 CC1SCCCC1C(N1CC(CCNC(=O)CC(=O)NC2CC2)C1)=O C(=O)(C(C)(CO)NC(c1ns[nH]c1=O)=O)N(C1CC1C1CC1)C N1(C(C(CCSC)O)=O)C2CCCC1CN(C(=O)CC=Cc1ccccc1)C2 C1(NC(c2ccc(Cn3ccnc3)[nH]2)=O)CS(=O)(=O)CC1O CC1CCCCC1(C)C(=O)NCc1cc[nH]c1C(=O)NCCCSC(F)F C1(NC(=O)CN2CC3CC3C2)CCC(CCC(=O)NCCCOCC(F)F)C1 c1(SCC(=O)NCC23C(CN(C(C4C(C)C4)=O)C2)C3)c[nH]c2ccccc12.CN N1(C(c2ccc(C(C)C)s2)=O)C2CCCC1CC(NC(=O)CNC(=O)C1CC1)C2 N1(C(C=CCOC)=O)CCC(C(C)NC(C2CC2(C)C(C)C)=O)C1 c1(C(=O)NC(CNC(CC(CCC)C)=O)(CC)CC)cc2c(cn1)OCCC2 c1(OC)ccc(C(C)C(=O)NCC2CN(C(c3cc(C)c(Cl)s3)=O)C2)cc1OC C1(CCCNC(c2cnn(C(F)F)c2)=O)CCN(C(C2C3CCCCC23)=O)CC1 C(=O)(C1CCOc2ccc(F)cc21)N(C1CCN(C(=O)CS(C)(=O)=O)C1)C c1(NC(CN(C(C=CCCC)=O)C)C)c(C)cc(C(=O)OC)cc1[N+](=O)[O-] Cc1c(Br)noc1C(=O)NC1(CNC(=O)C(F)(F)c2cnn(C)c2)CC1 Cc1c(F)ccc(C(=O)NC(C)CNC(=O)CCS(N)(=O)=O)c1N N1(C(CSc2n(C)nnn2)=O)CCN(C(C2CCCCC23CCC3)=O)CC(O)C1 N1(C(C(=O)OCC)=O)CC(C(N2CCC(NC(C)=O)C2CC)=O)C2(CCC2)C1 C1(C(=O)NC2CC3C(NC(C4(C)COC(=O)C4)=O)C3C2)CC2CCC1C21CC1 C(=O)(CS(=O)(=O)C1CCCC1)N1CC(CNC(c2ccc3nc(C)oc3c2)=O)C1 Cn1ncc(CC(C)CC(N2CCCC2)C)c1O.C(=O)(C(O)CC1CCCC1)N c1(C(N2CCCC(NC(c3c(C)cc(CO)o3)=O)C2)=O)ccc2c(c1)OCC2 CCC(C)(C)CCCC(=O)N1CCCC12CCN(C(C1CCC(F)C1)=O)C2 C1(C(=O)NCCN(C(CCC)=O)C)CCC(=O)N1n1ccc(C2CC2)n1 c1(C(=O)NCC2C(NC(c3cccc4occc34)=O)C2)c(Cl)cccc1[N+](=O)[O-] Cc1cc(NNC(=O)NCc2cccnc2N(C)C)nnc1C c1(C(=O)NCC2N(C(C(C)SCC)=O)CC(OC)C2)ccc(C)cc1CC C1(C(=O)NC2C(SC)COC2)CC2C=CC1N(C(c1nnc(S)n1C)=O)C2 CCC(C)(C(=O)N1CCC(O)(CCNC(c2c[nH]nc2OC)=O)CC1)C(N)=O C(C(C)(C)CN=[N+]=[N-])NC(c1ccc(CNC(C(C)c2ccco2)=O)o1)=O Cn1[nH]c(=NC(=O)C2CC3(C2)CC2(CCC2)C3)n(-c2ccccc2C(F)(F)F)c1=O C(=O)(C1=CS(=O)CCC1)NCC(CC)NC(=O)Cc1cc(F)ccc1OC c1(C(=O)NCC(CNC(C(=O)NCCNC(C)=O)=O)(C)C)nccc2[nH]ccc12 C1(CC(=O)NCCCCCNC(c2c(CCC)occ2)=O)CCC(=O)N1C C1(C(=O)NC2C(C)N(Cc3nnc(C4CC4)s3)CCC2)Cc2ccncc2C1 N1(C(=O)Cc2csnn2)CCc2c(ccc(Br)c2F)C1 S(=O)(=O)(c1ccc2[nH]c(=NCC(C)CCOC)ccc2c1)N(CCSC)CC Cn1ncc(NCc2cnc(-c3ccccc3)[nH]2)c1C(F)F C1(C(=O)NCc2ncc(C)o2)CC(F)CCN1C(=O)Cn1cncn1 C(CCC1CC1)(C(=O)N1CCCC1CCO)N(C(C(C)N1CCCC1)=O)C c1(C(N2CC(NC(C3OCCN(C)C3=O)=O)C3(C2)CC3)=O)ccc2nn[nH]c2c1 CS(=O)(=O)CCN(C(=O)NC1COCC1C(F)F)Cc1ccns1 CC1CN(C(C2CCC(F)(F)CC2)=O)CCC1N(C(=O)CN=S(C)(C)=O)C C1(CNC(C(CO)OC)=O)CN(C(=O)C=Cc2ncc(C)[nH]2)CC1(C)C CC(C(=O)N1CCCC2(NC(=O)CC3C=CCC3)CC2C1)C(C)S(C)(=O)=O c1(C(N(CC(C)CNC(=O)CCCN2CCCC2)C)=O)cnc2[nH]cnc2c1 c1(OCC(N2CCC(F)(CNC(C(C)SCCCC)=O)C2)=O)ccc(Cl)c(C)c1 c1(CC)nc(-c2cc(Cl)c(CC)cc2F)n(C2CCC(=O)N(C)c3ccccc32)n1 CC(C)(F)C(=O)N1CCC(NC(C2CC2F)=O)C1 C1(C(=O)NCc2ccncc2)CC12CN(c1ncc(Br)cn1)C2 C(=O)(CCCCCCCC(=O)OC)NCC(N(C(CSCC=C)=O)C)C1CC1 Cc1cnc2c(C(=O)NC(CC3CCCCO3)C(=O)O)cccc2c1 Cc1ccc2oc(=NC3CN(C(=O)CSc4ccccc4)CC3C)[nH]c2c1 C12(OC)CCC(C(=O)NC3CCN(C(c4coc5c4COC5)=O)C3)(CC1)C2 C1(NC(Cc2nc(C)oc2)=O)CN(C(c2cn(C)c(C)n2)=O)CC(C)(C)C1 C1(C(C)C)CN(C(=O)CSc2cnn(C)c2)CCCN1C(=O)Cc1cscn1 C12(CNC(c3cccc(C)c3)=O)CC(C1)C(NC(=O)C(c1cncn1C)O)CO2 c1(NC(=O)NCC(=O)OCC=C)cn2cc(Cl)cc(C)c2n1.OCC C(C)(C(=O)N=c1cc[nH]cc1[Si](C)(C)C)n1cc(-c2c(C)ocn2)nn1 c1(C(CC(=O)NCc2csc(-c3cnn(C)c3)n2)N(C)C)ccccc1F N1(CC)CCOC(C(N2CCC(C(C)(C)CNC(=O)CC(C)F)CC2)=O)C1 C1(C)(NC(C=NOC)=O)CCCCC1C(N1CC2CCC(C1)O2)=O c1(C(N2CC3CC3(C(=O)NCC(O)CO)C2)=O)ccc(Cl)cc1O N1(C(CCCC)=O)CC(CO)C2(C1)CN(C(=O)CCCC1CCCCC1)C2 c1(C(=O)NCCC=CC)cc(C(=O)OC)cs1 c1(OC)cc(CC(N2CC(CNC(c3cnn(C4CC4)c3)=O)C(C)C2)=O)ccn1 N1(C(C(CC)C)=O)CCC(NC(c2ccnc(Br)c2N)=O)CC1C c1(OC)ccc2c(C(N3CCC(C)(NC(c4cc(C)co4)=O)C3)=O)n[nH]c2c1 N1(C(c2nn(C)c(F)c2)=O)CCCC(O)(CNC(=O)C=C2CCCC2)C1 CCC(CC(=O)NC1CC(NC(C2(c3ccno3)CC2)=O)C1)C1CC1 C(c1ccc(C(F)(F)F)cc1)=CC(=O)NC1C2CC1N(C(c1cscn1)=O)C2 C(=O)(CC(C)C(C)(C)C)N(CC(=O)N(C)CCF)CCOC c1(NC2(C(N3CCC(C(=O)OC)C3)=O)CC2)cc(N(S(C)(=O)=O)C)ccn1 c1(C2(NC(CN(C(CC3(OC)CCC3)=O)C3CC3)=O)CC2)nncn1C C1(NC(c2n(C=C)ncc2)=O)CCN(C(C2CCCNS2(=O)=O)=O)CC1(C)C C1(C)(CNC(CC(C=C)C)=O)CCCN(C(=O)C(CO)OC)C1 N1(C(=O)NC2CC(CC)(CC)C2)CCC(C)(CC(=O)NC)C1 CCC(CC)C(F)C(=O)NCC(C(=O)N1CCC(C(=O)NC)C1)C(C)(C)C C(c1ccc(Cl)cc1Cl)=CC(=O)NCC(C)CNC(C1CCOC(=O)CC1)=O C1(C(=O)NCCC2(N(C)C)CC2)CCN(C(=O)C2CC2)O1 N1(C(c2coc3c2CN(C(=O)OC(C)(C)C)C3)=O)CCC2CCNCC2C1 CC1CCN(C(c2cnc(=N)[nH]c2)=O)C(C(=O)NCC(c2ccnn2C)O)C1 c1(C(=O)NCC(C)(O)CNC(=O)Cc2cocn2)ccc(C2(O)COC2)cc1 c1(NC(C2CC2N)=O)ccc([N+](=O)[O-])c(O)c1.CC1(C)CC1 C(=O)(CC(C)(C)O)NCC1(CNC(c2c(CC(=O)OC)scc2)=O)CC1(F)F C=CCC(CC(=O)N(C1COCC1OC)C)NC(=O)CC1CCCSC1 CC1CN(C(=O)Cc2sccc2Cl)CC(C)C1NC(=O)CCF C(=O)(C1=NN(CCO)C(=O)CC1)N(C1CC(NC(CC(=C)C)=O)C1)C N1(C(C)=O)CCCCCCC1.C(=O)(C(F)(F)CN(C)C)NC1CCN(S(C)(=O)=O)C1 C(=O)(C1=CCCN(C(=O)CCOCC(F)F)C1)NC1CCCC(OC)CC1 Cc1ccc(S(N)(=O)=O)cc1NC(=O)Nc1ccsc1CO c1(C(N(CC(CNC(Cc2ccc(OC)s2)=O)O)C)=O)sc(C)cc1Cl c1(NC(C)=O)cc(Cl)ccc1C(=O)NCCC1CN(C(C2(C)CC2)=O)CCO1 c1(CC(=O)NC(CC(C)C)(C)CNC(=O)OC(C)(C)C)ccc2ocnc2c1 CC(C)(F)CCC(=O)NC(CNC(=O)CCNC(=O)NC1(CO)CC1)C1CCC1 C1(NC(C=CC2(C)COC2)=O)CC=C(C(=O)NC2CC(O)C2)C1 CC(C)(C)CC(C)(C)C(=O)N1CSCC1C(=O)NC1CN2CCC1(F)CC2 Cn1cncc1C(O)C(=O)NCCC1(NC(c2cccs2)=O)CCC1 C1(C(C)C)CCN(C(=O)C(c2ccoc2)NC(C2C3CC4C(C3)C24)=O)CC1 N1(C(c2nnn(C)n2)C(=O)NCc2cc(O)nn2C)CC2CCC(C1)C(=O)N2 N1(C(C2(CCC)CC2)=O)CCN(C)C(C(=O)N(C2CC(SC)C2)C)C1 C1(C(=O)NCC(C)NC(CN(CCOC)C)=O)CC(OC)C1.C(C)(=O)O C=C(C)CC(C(=O)NCC1(C)CN(C(c2c(C)cccc2N)=O)CCO1)OC Cc1cc(C#N)cnc1-c1ccccc1C1CC=CCO1.N1(C2(c3ccccc3)CC2)CCC(C)C1CC.C(C)C=O c1(OC)ccc(F)c(CNC(C2CC(F)CN2Cc2cc(C)no2)=O)c1 N1(C(CCC=C)=O)CCC(C(=O)NCc2ccc(OC)nn2)C(O)C1 CCC(C)(C)C(O)C(=O)Oc1ccc(OC(C)CNC(=O)CS(=O)(=O)C2CC2)cc1 C(=O)(CCCC(C)(F)F)N(CC(C)NC(=O)Cc1cncnc1)CC c1(C(N2C(CCNC(c3n(CC)ccc3)=O)CCCC2)=O)c[nH]c2cccnc12 C1(NC(C2C(C)=C2)=O)CC2CCC(C1C)N2C(=O)C(F)(F)c1ccccc1 N1(Cc2cccc(CCNC(c3c(C)ccnc3)C)c2)CC(C)(C)OC1=O c1(C(=O)NC23CCN(C(=O)CNS(=O)(=O)C4CC4)CC2C3)c[nH]c2ccncc12 N1(CCNC(C(CCC)C)=O)CCN(C(c2cnc(Cl)cc2N)=O)CC1 Cc1cc(NC(C2(F)CC=CC2)=O)ccc1NC(=O)C(F)C(C)(F)F C1(CNC(C=CC=CC)=O)CCCN(C(=O)C(C)OCCN(C)C)C1 c1(C(N(C(C(=O)NCC(COCC)C)C2CC2)C)=O)ccnc(C)n1 c1(CC)ccc(F)c(C(=O)NCC(CNC(C2(CC)CCCO2)=O)OC)c1 C1(NC(CCCCCN(C)C)=O)CN(C(c2ccco2)=O)C2(CCOCC2)C1 n1(C(C)C)cc([N+](=O)[O-])c(=NC2CC(NC(=O)CCCc3ccsc3)C2)[nH]1 CC(C)C(CNC(=O)Cc1ccc(Br)s1)NC(=O)CNC=O C=CCCCCCN=c1cc[nH]cc1S(=O)(=O)N1CCCC(O)C1C N1(C(COCC)=O)CC(CNC(C2CCN(CC(C)(C)O)CC2)=O)C(C)C1 c1(C(C(N2C(C(=O)NC(CN(CC)CC)C)CSC2)=O)=O)ccc(C)cc1 N(C1CCc2c1cnn2Cc1ccc(Br)cc1)C(CNC(C(CC)CC)=O)C c1(SCc2ccccc2)nocc1C(=O)NC1(C)N(C(C(C)NC(N)=O)=O)CC1 C=CCC(C(=O)N1CCCC1(C(=O)NCC(=O)NC(C)C)C(C)C)C(C)C CCC(CC(=O)N1CC(N(C)C(C2(Br)CC23CCC3)=O)C1)OC c1(C(N(C2C3CN(C(C(C(C)C)OC)=O)CC32)C)=O)cc2c(o1)CCCC2 Cc1cc(C)c(C(O)CNC(=O)NCC(F)(F)CC2CCOCC2)c(C)c1 C(=O)(Nn1cnnc1)c1nc(-c2c(C)nn(-c3cccc(Br)c3)c2)n(C)n1 n1(CC)cc(C(F)(F)C(=O)NCC(C2CC2)N(C)C(C2CCO2)=O)cn1 C1(C(=O)NCCN2CCCN(C(c3ccoc3Cl)=O)CC2)CC2(CCC2)CCO1 c1(CC(COc2cn(Cc3ccc(C)cc3)nc2)=O)cccc(F)c1C#N C1(C(=O)NC2CCCC2)CCCN1N=O.CC1(C)CNC(=O)CO1.C(CN)O.O Cc1oc(C(=O)NCCn2cc(CNC(=O)Cc3cccs3)nn2)cc1CO C#Cc1ccc(CC(=O)NC(CO)C(=O)NCC(C)S(C)(=O)=O)cc1 N1(C(C2(C(=O)OCC)CC2(F)F)=O)CC(NC(c2ccn(CC)n2)=O)C(C)C1 C=CCC(C)C(=O)NC1CC1NC(c1cccc(OCC=C(C)C)c1)=O c1(C(N2C(C3(NC(CNC=O)=O)CC3)CCCC2)=O)cccc2cnnn12 c1(CC)ccc(C(=O)N(C(C)C(=O)N2CC(N3CC(C)(O)C3)C2)C2CC2)cn1 C(=O)(CP(C)(C)=O)N1CCCC(CCC(=O)NCC2(CC)CCCC2)C1 C1(CCOCC)CN(C(=O)C(N2CC3CC(C)C3C2)=O)CCCO1 C1(C(=O)NCCCNC(C2(c3c(C)c[nH]n3)CC2)=O)CCCCC1O c1(C(=O)NC(CNC(CC2(OC)CCCCC2)=O)CO)ccc2nccnc2c1 CC1CCCC1(C(=O)N(C)CCc1cnn(C)c1)NC(=O)CN(C)C c1(C(=O)NC(C)CC2CN(C(=O)C(C)n3ccnc3)C2)ccc(C(F)F)nc1 C(=O)(C(C)CCCC(C)=O)NCC1C(NC(CCC(CC)OC)=O)CCC1 N#Cc1ccc2ncnc(N3CCn4c(CC(F)(F)F)nnc4C3)c2c1 c1(C(N2C(C)CCC(NC(c3c(C)cns3)=O)C2)=O)noc2cc(Cl)ccc12 C1(CN(C(=O)CC#N)C)CN(C(c2cn(-c3ncccn3)cn2)=O)CCO1 N1(C(C2CC(C)(CC)C2)=O)CCCCC(C(=O)NCc2nccn2C)C1 n1(CC=C)c(=O)cc(Cl)n(CC2CC2c2ccc(C3(COC)CCC3)o2)c1=O c1(C(=O)NCC(CC=C)NC(=O)C(C)N(C)C)cc(CC)n(-c2ccccc2)n1 CN1CCN(C2CCCN(C(=O)NC3CCN(C4CCCC4)C3)C2)C1=O c1(C(=O)NCC(C)CNC(=O)CCCOCc2ccccc2)cc(Cl)nc(Cl)c1 CC1(C(N2CC3CCC2C3NC(=O)C=CC2CCOCC2)=O)CCCNC1=O N1(C(CCOCCCOC)=O)CCC(C)C1CNC(c1ccccc1CC#N)=O N1(C(C2C(C)(C)C2(F)F)=O)CCN(C(c2ccoc2Br)=O)C(CC2CC2)C1 c1(NC(COCC)=O)cc(N2CCC(OCCC(C(F)F)SC)CC2)nc(C)n1 N1(C(C=C(CC)C)=O)CCCCC1CC(=O)NCCN1C(=O)CCC1=O Cc1nc([N+](=O)[O-])cn1CC(=O)NCC1(F)CCN(C2CCSC2)CC1 c1(C(=O)OC(N(CC(O)C(=O)OCC)CC)=O)ccc(O)c(C(C)(C)C)c1 C(=O)(N1OC2CCC1CC2)C1C(C)(C)C1NC(=O)CCCC#N C#CCC(C)(C)C(=O)NCCC1CCN(C(C2C(C(F)(F)F)C2[N+](=O)[O-])=O)CC1 N1(C(C2CC(=O)NC2)=O)CCC(CNC(c2csc(CO)n2)=O)C(F)(F)C1 N1(C(CCCC#C)C(=O)Nc2c(C)cc(C)cc2C)CC(=O)N(C)C2(CCC2)C1 c12ccc(nc1OC)CNC2=O.c1(OC)cccc(SCC(=O)NC2CC2F)c1 Cc1cc(CC(=O)NCCn2cc(C(=O)N(CCC(O)C3CC3)C3CC3)cn2)no1 C(=O)(CCCC(=O)N1CCC(CN(C(=O)C(C(C)C)c2ccc(C)s2)C)C1)OC Cc1cccc(C(F)C(=O)NC(CNC(c2scnc2C)=O)CO)c1 C1(CCNC(c2cccc(-c3cc[nH]n3)c2)=O)CSCCN1C(C1CC1CF)=O O=C1CN(C(=O)COc2cccnc2)C(C(=O)NCC2(O)CCSC2)CN1 CCC(C)C(C)C(=O)N1CCCOC(CCNC(=O)CC(=O)N(C)C)C1 C(=O)(C(C)(C)CC(C)(C)C)NCC(CC=C)NC(=O)C#CC(C)(C)C c1(CC)ccc(OCCOC(c2cccc(C(F)(F)Cl)c2)=O)cc1 N1(SCC2C(NC(=O)NC(c3ccco3)c3cccs3)CCO2)CCCOCC1 Nc1c(C(=O)NC2(CN)CC2)cc(Cl)nc1Br.C12CN(C1)C(=O)C2=O.C1(CC)CC1 c1(C(=O)NCCN(CCC)C(C2(CO)CCCC2)=O)cc(C)cc(Br)c1 C#CCC(CC(=O)NCc1ccc(CC)s1)NC(C1(CC)CCCO1)=O C(=O)(C(F)CCC(C)C)N1CC(C(=O)NCC(COC)(C)O)N(C)CC1 Cc1ccc(S(=O)(=O)NCCOCC#CCN2CCCCCC2)c(C)c1C(=O)O C1(CNC(CC(C)SC)=O)CC2(CCN(C(=O)Cc3cnc(O)nc3O)C2)CO1 CC12CCCC(C(=O)NC3CC(CNC(c4ccc(Br)cn4)=O)C3)(CO1)C2 c1(C(N2CC(NC(C3(Cl)CC3(F)F)=O)CC2(C)C)=O)cnc2c(c1)NCC(=O)N2 N1(C(=O)CCn2cncn2)CC2CC1CN2Cc1ccn(-c2ccccc2)n1 Cc1nsc(C(=O)NC(C)CCC=C(C)C)c1I CN(CCCC(=O)N(CCCNC(C1(CO)CCCCC1)=O)C)N=O C(=O)(CS(=O)(=O)CCCc1ccccc1)NCC1CCC(NC(C)=O)C1 C1(CC(=O)NC(CCCNC(Cc2scc(C)c2)=O)C)OC(C)(C)OC1=O C(=O)(CC(C)(C)COC)N1CC(C(C)NC(c2c(SCC)cccc2)=O)OCC1 C1(N(S(=O)(=O)CCOCC(=O)OC)CCOC)CC2CC1CN2C1CC1 c1(C(N(CC(CC)NC(=O)CCn2nc(C)nc2C)C)=O)ccc(O)c(F)c1 C1(C(=O)NC2CCN(C(CN(C)C(=O)C3CC3)=O)C2)CCC2CC2CC1 c1(C(=O)NCCC(C)NC(=O)CC2(O)CCCC2)cc(Br)c2[nH]nnc2c1 C1(C(=O)NC2C(CN=[N+]=[N-])CCC2)C=CCN(C(=O)C=Cc2ccncc2)C1 c1(COC)ccc(-c2nc(CN(C)C)nn2CCCO)cc1.c1(CC)ccccc1F CN1CCCC(C(=O)NC2CN(C(=O)CCCn3ccnc3)C2)C1 C(=O)(C(CC)C(C)(C)CC)N1CCC(CC=C)(NC(=O)C2=NOC(CC)C2)C1 C1(CC)CN(C(=O)Cc2cccc(C)c2Cl)CCC1NC(c1nc(C)n(C)n1)=O c1(CC)cnc(O)c(C(=O)NC2CC(C)(NC(c3ccc(OC)o3)=O)C2)c1 c1(C(CNC(c2nc(CC(N)=O)no2)C)OC)cccc(Br)c1 C12(CC(=O)NCCCN(C(C(C)NC(C)=O)=O)CCO)CC3CC(CC(C3)C1)C2 N1(C(c2c(CC)nc(C)o2)=O)CC(NC(c2cnc(C)s2)=O)CC2(CC2)C1 c1(C(N(C)Cc2cn(CC3CCOC3)nn2)=O)n[nH]c2c1CSCC2 Cc1cnc(Br)c(NC(C2CC3(CC3)CN2C(c2ccc(I)c(F)c2)=O)=O)c1 c1(CC(N2C(CCNC(CC(C)CF)=O)CCCC2)=O)c[nH]c2cc(F)ccc12 C1(C(=O)NC23OCC(C(N4C(C)C(C)CCC4)=O)(C2)C3)CCc2cnnn2C1 C(C(C(=O)NCCNC(=O)CCc1n[nH]c(=N)s1)OC)OC c1(CC(=O)NCC(CNC(C2CN(C(N)=O)C2)=O)OC)cn(C)cn1 N1(C(C(COCC)C)=O)C2CCC1CN(C(=O)C(C)(C)C(F)F)C2 CC1OCCOC1C(=O)NCC(C)(C)CN(C(=O)CCc1ccccc1F)C c1(CC(=O)NC(CNC(c2ccc(O)c(F)c2)=O)CO)c(F)cncc1Cl C(C(=O)N(C)OC)NC(C1C(NC(COCC(C)C)=O)CCC1)=O N1(C(c2c(CC)cc[nH]2)=O)CCOC(C(=O)NC2COC(C(F)F)C2)CC1 C(N=c1cc[nH]c(C#N)n1)C1OCC(CNC(CSCCCC)=O)C1 n1(CC(=O)NCC2CN(C(c3c(Br)cn(C)n3)=O)CC2O)cccc(N)c1=O c1(OCCC)ccc(C=CC(=O)NC2CN(C(C3(C)CC(F)C3)=O)CC2C)cc1 c1(C(=O)NCC2CC(C)N(C(C3CC3(F)F)=O)CC2)snc2ccccc12 C(CC(=O)N(C(CSC)CC)CCNC)OCCOCC#C c1(C(=O)NC(C)C(C)NC(C2(C)CC(C#N)C2)=O)cccc(Br)c1Cl C=CC(C)CC(=O)NC(CNC(c1ccc(Cn2ccnc2)o1)=O)CO C#CC1(O)CCN(C(=NCc2ccc(Cl)cc2)NCC(=O)Nc2ccccc2)C1 Cc1cc2cc(NC(C)CCCSCc3ccccc3)[nH]c2cc1Cl Cc1c(F)ccc2c(=O)c(C(=O)NC3CCCC34CN(C(=O)CCF)C4)c[nH]c12 Cc1cccc2c(C(N3CCC(C)C3CNC(c3cccc(Cl)c3F)=O)=O)n[nH]c12 Cc1nc(C)c(C(=O)NC2CCOC(CNC(=O)Cc3ccccc3O)C2)o1 c1(CC)c(C(=O)N(C)CCNC(=O)CSC(C)C)cnn1-c1ccccc1CC CN1C(=O)CCC1CC(=O)NC1CC2C(NC(c3cnc[nH]c3=N)=O)C2C1 C12(C(=O)NC(=O)NC3C(C)CCCC3)CCCC1N(CC#N)CC2 N1(C(C2(C=C)CCC2)=O)CCCC2(NC(=O)C(C)Oc3ccccc3)CC2C1 n1(C(C)C)ccnc1C(=O)NC1CCC(CNC(c2cnc(C3CCC3)o2)=O)C1 C#CCCC(O)C(=O)N1CC(NC(=O)C(C)=C(C)C)C(C)C1 c1(OC)cccc(C(C(=O)N(CCNC(=O)CC(C)c2ccco2)CC)OC)c1 Cc1ccc(C(=O)NC(C)CCc2ccnn2C)c(-n2ccnc2)c1 C1(C(=O)NCC(n2cc(-c3nccn3C)nn2)C)Cc2ccccc2OC1CO CC1(C)COCC1CNC(=O)NCc1nnc(Cc2ccc(Cl)cc2)o1 c1(C(=O)NC2(C3CCCN3C(c3cnsn3)=O)CC2)ccn2nccc2n1 c1(NCC(C2C(C(=O)OC)C2)NC(C2CC2c2ccco2)=O)nccc(C#N)n1 C1(NC(CSC)=O)CCCCC12CCN(C(=O)CC(=O)OCCC(C)C)CC2 C(=O)(C1=CS(=O)CCC1)NC1CC2CC(NC(c3ccc(CN(C)C)o3)=O)CC21 c1(CC)nc(C)ccc1NC(=O)NCc1ccc(C)c(OC(F)F)c1 c1(-c2nc(C3CCC(F)(F)C3)nn2C2CCOC2)cnc2cnccn12 C1(CN(C2COC(C3CCOCC3)C2)C(c2cnnn2C2CC2)=O)CCC=CCC1 N1(C(Cn2nc(C)c(Cl)c2)=O)CC(C)CCC1CNC(=O)CC1CN(C)C1 N1(c2ccnc(NC(CC(CC)C)=O)n2)CCc2[nH]nc(CO)c2C1 C1(O)(CN(C(C(C2CCCC2)OC)=O)C)CCN(C(=O)C=C2CCN(C)C2)C1 c1(C(=O)NC(C(=O)N(C)CC2CC(=C)C2)c2ccoc2)ccc(C)nc1O C1(C)(C(=O)NCC2C(NC(C(C(C)C)O)=O)CCC2)CCN(C)CC1 Cc1c(Cl)c(C(=O)NCC2(O)CCN(C(c3c(Cl)cncc3Cl)=O)C2)nn1C c1(C(=O)NC2CC(NC(C(C)CC3CCCCC3)=O)C2)cccn2[nH]c(=N)nc12 C1(CNC(=O)Nc2cccc(C(C)C)n2)CCC2(CCCCCC2)O1 Cc1ccc(CNC(N2CC3(CN(C)C)CC2(C)C3)=O)c(O)n1 N1(C(CNC(CCC)=O)=O)CCSCC1CCNC(C1CS(=O)(=O)C1)=O C=CC(C)(CCOC)C(=O)NC(C)CC(C)NC(c1ncnn1C)=O CC1C(C(=O)N2C3CCC2C(C(=O)NCC24CC(F)(C2)C4)C3)=NOC1C C1(CNC(c2n(CC)ccn2)=O)CN(C(C2CCCC2O)=O)CCC1(C)C C1(C(N2C(CN(C(=O)C(F)CC3CCC3)C)COCC2)=O)CC2CCCC(C1)C2 CC(CN1CCOCC1)C(=O)N1CC(C(C)(C)O)(CNC(C2CC2C(C)O)=O)C1 C(=O)(C#CC1CCCCO1)N(C)CC1CCN(c2snc(CC)n2)CC1 C1(CC)CCN(C(C2CC=CC(O)C2)=O)C1C(=O)N(C)Cc1ccn(C)n1 c1(OC)ccc([N+](=O)[O-])cc1NC(=O)CC1C(=O)Nc2ccccc21 C1(NC(c2c(C)cns2)=O)CC2CN(C(c3cc(O)cc(N)c3Cl)=O)CC2C1 N1(C(=O)CCN2CCC2)CCC(C2OCCC2NC(=O)CSCC(F)F)CC1 c1(OCCN(C(=O)C(C)C)CC(C)C)cc2c(Cl)cc(Cl)cc2[nH]1 Cn1ncc2cc(-c3ccc4ncc(C(=O)NC(C)(C)CO)n4c3)ccc12 c1(NC(C2(CC)CCCN2C(C2C3CCCCCC23)=O)=O)cc(C)cnc1C c1(OC)cccc2c(C(=O)N(C(C)CCNC(=O)CSC)C)n[nH]c12 N1(C(C2N(C)CCC2)=O)CCC2(CCCN2C(c2ccc(C(C)(F)F)nc2)=O)C1 N1(C(c2cn(C)nn2)=O)CC(NC(=O)C2=COCCO2)C(S(C)(=O)=O)C1 CCC(C)(CO)CN=c1cc(C)nc(N2CCOC3(C)CC2CNC3)[nH]1 Cc1c(C(=O)NCC(O)CNC(C2C3(CC3)C23CC3)=O)ccc(Br)c1F C1(N(C)C)C2CN(c3ccnc(N4CCC(c5ccccc5)C4)n3)CC12 C(=O)(C1=CCCCCC1)Nc1c(NC(C(C)OCCOC)=O)c(F)ccc1 C1(O)(CCCNC(c2nc(CC)sc2)=O)CCCN(C(C2(CN(C)C)CC2)=O)C1 C12(C(C)=O)CCC(C(=O)N(C3CC(NC(=O)C(C)O)C3)C)(CC1)OC2 CC1=C(C(=O)NCCC2CCCN(C(=O)CCc3ncc[nH]3)C2)SCCO1 Cc1scc(C(=O)NCC(C2CC2)NC(c2cc(C(N)=O)cs2)=O)c1C c1(C(N2CCOCC2COC)C(=O)NCCC(=O)OCC)cc(Cl)c(OC)cc1Cl c1(C(c2n(CCCC)nnn2)Nc2c[nH]nc2OC)cc(F)c(OC)cc1F CCCCC(CC)C(=O)NCCCOCCNC(=O)C(C)c1ccco1 c1(C(N2C(CNC(CC(CCSC)O)=O)C=CC2)=O)cc2cc(F)ccc2s1 N1(C(C2ON=C(C)C2)=O)CC=CC(NC(=O)CCC(=O)N(C)CCN(C)C)C1 N1(C(C(c2ccc(F)cc2)(C)O)=O)CCCCC(NC(=O)C=C2CCCC2)C1 N1(C(C2N(CCC)CCC2)=O)CCCN(C(=O)CN(C2CCCC2)C)CC1CO C1(CCC)CN(C(c2coc(C(C)=O)c2)=O)CC1NC(C1CCCC1CC)=O c1(C(=O)NCCC(=C)CNC(C2CCC(C)C2)=O)cc2ccc(OC)cc2o1 C1(C(N2CCC(NC(C(C)=C(C)C)=O)C2C)=O)CCC(C)C(C)C1 C1(NC(CC(=O)NCCN(CCCOC)C)=O)CC1C1CCCC1 C(=O)(C(C)(C)C(C)C)NCC1CC(NC(Cc2c(C)nsc2)=O)C1 C1(NC(C2N(C(C(=O)OC)=O)CCC2OC(C)(C)C)=O)CCOC12CCOCC2 N1(C(c2ccc(OC)s2)=O)CC(NC(=O)CCCNS(C)(=O)=O)CC(F)C1 C1(C(=O)NC2C(CNC(Cc3cc(C(C)C)no3)=O)COC2)OCCN(C)C1=O c1(C(=O)NC(C2CCCCN2C(=O)CSCC(N)=O)C)ccc([N+](=O)[O-])n1C C1(CC)CN(C(c2ccncn2)C(=O)NC(c2ccccc2)C)CC(C)S1=O C1(CCNC(C2(CC#C)CCCO2)=O)CCN(C(=O)Cc2ccc(C)s2)C(C)C1 C(C(=O)N1CC=C(C)CC1)(C(C)(C)C)NC(CSCCC=C)=O N1(C(C2CC(CC)(CC)C2)=O)CCN(CCC(=O)NC2CCC(CC)CC2)CC1 N1(C(c2n(C)nc(CNC(c3nsnc3O)=O)c2)=O)CCCC12CCOCC2 c1(-n2cc(C(C)OC)nn2)ccc(OCCOc2ccccc2)cc1 C1(C(=O)NCC(C(=O)NC)O)CC2CCC(C1)N2C(=O)COC(C)C C1(C(=O)NCCN(C(=O)CCc2ccccn2)CC(C)O)(CCF)CCOCC1 c1(CC)onc(C(N2CC(C(=O)N(CCC(C)C)CCO)(CC)C2)=O)c1C c1(Cn2cc(C(N(CCNC(C3CCCOC3)=O)CC)=O)nn2)ccc(F)cc1 C(=O)(C(F)(F)CCn1ccnn1)NCC(CC)NC(=O)C(C)n1ccnc1 C1(NC(c2c(C(C)C)ocn2)=O)CCCCCC1NC(C1CC(C(F)(F)F)C1)=O C1(O)(CN2CCCC(CNC(=O)CCc3ccoc3)C2)CCCCCC1 N1(C(CN(C2CC2)CC)=O)CCC(C)(NC(=O)C(c2ccccc2)C)CC1 C1(C(N2CC(OC(CC)=O)C2)=O)C2CC3C(C2NC(=O)C(C)CC2CCCC2)C13 N1(C(c2scc(C(N(CC=C)CC=C)=O)n2)=O)CCN(c2ccc(Cl)cc2)C(=O)C1 C(=O)(C1=CC(C)(C)C1)N1CC(CCNC(c2c(C)cc(CO)o2)=O)C(C)C1 c1(OC)cccc2c1OC(C(=O)NCCCCN(C(=O)C(O)CC(F)(F)F)C)C2 C#Cc1cc(C(=O)NC2COC3(CCC3)C2)cc(F)c1 N1(C(Cc2cc(C)n(C)n2)=O)CCC(C2CC2)C1CNC(C1(C)CCC1)=O N1(CC)CCCC1CC(=O)NC1(C)CC(NC(C2CC2C(C)(F)F)=O)C1 c1(CC)ccc(F)c(C(=O)NC2CCN(C(=O)C=CCOC)C(C)C2)c1F Fc1cc(CSc2cc(C3CC3)cnc2F)c2ncccc2c1 N1(C(C(CC=C)C(C)C)=O)CCC2(CC1)CN(C(c1ccc(CO)o1)=O)CCO2 C=CCCC(=O)NCc1ccc(C(=O)NCC(F)Cl)s1 C1(C#CC(=O)NCC2CC(C)N(C(=O)CCCC(C)=O)C2)(CC)COC1 c1(NCC2(C)NC(=O)NC2=O)ccc2[nH]c(C(F)(F)F)cc2c1 N1(C(CC(CC)C2CC2)=O)CCCC12CCN(C(C1COC3COCC13)=O)C2 c1(OCC(=O)NC(C(C)NC(Cc2c(C)noc2Cl)=O)C)nc(O)nc(O)n1 N1(CC(=O)N(CCCNC(C2(C3CC3)CCCO2)=O)C)CCC(=O)NC1=O c1(C(=O)NC(C2CCN(C(c3c(C(C)C)c[nH]n3)=O)C2)C)ccc(S(C)(=O)=O)o1 C(=O)(C1=NOC(C(C)(C)C)C1)N(C1(CNC(CCN(C)CCO)=O)CC1)CCCO CCCC(C(=O)NCC1CC2(CCC2)C1)NC(=O)CN1CC2CC2C1 c1(CN2CC(C)S(=O)CCC2)c2c(nn1C)CCOC2 c1(C(N(C(C)=O)CC)=O)ccc(N)cc1OC.C1(NC(N)=O)CCN(C(=O)CN)CC1 C1(C(=O)NCc2ccnc(C)n2)CC2(CC2)CN1C(c1coc(N(C)C)n1)=O C1(C(N2CC3C(CNC(C(c4ccn(C)n4)(C)C)=O)C3C2)=O)C2CCC(F)(F)C12 C1(CN(C(c2c(CC)cco2)=O)C)CCCN(C(C2(C#N)CC2)=O)C1 c1(N2CC(C#N)C(NC(c3ncccn3)=O)C2)ccn2ncc(Br)c2n1 C1(NC(CC(C)C(F)F)=O)CN(C(c2cc(C#N)n(C)n2)=O)CC1C1CC1 C12(C(=O)NC3(C)CC(NC(Cn4ccc(C)cc4=O)=O)C3)CCCC1CC(=O)C2 CCC(C(=O)NCC(C)NC(=O)Cn1cnc(Br)c1)Sc1ccccc1 C(=O)(C(C)(O)C(C)C)NC(c1cccc(OC)c1)CNC(CC(COC)C)=O CC(C)(C)CC(C)(C)C(=O)NC1C2CCC1N(C(=O)C(O)C(F)(F)F)C2 C(=O)(C1=CS(=O)CCC1)NC1CCC(CNC(CCn2c(C)cc(C)n2)=O)CC1 N1(C(c2n(CC)nnc2)=O)CCCC(CO)(CNC(c2ccc(O)nc2)=O)C1 c1(C(=O)NCC2C(NC(=O)CCc3nccs3)C2)cc2c(F)c(F)ccc2s1 C(=O)(C1CCCc2ncnn21)NC1CC(CNC(c2cnc(C3CC3)nc2)=O)C1 c1(NC(C(C)C)=O)ccccc1C(N1CC(O)(CNC(C2C3CCCC23)=O)C1)=O N1(C(CCC(C)=O)=O)CC2CC(C(=O)NC(C(C)C)C3CC3)CC2C1 C(=O)(CCCC1CCCC1)N1CC(C(C(=O)NC(COC)COC)O)C1 n1(CC)ncc(Cl)c1C(=O)NC1CCCC1NC(c1nc(Cl)oc1C)=O c1(CC2N(Cc3c(C(F)F)cccc3)CCC2)cnc(Cl)cc1Br c1(C(=O)NCCNC(=O)C(=O)Nc2ccccc2C(=O)O)cc(Cl)ccc1F C1(C(=O)OCCN(CCC)C(C2CCS(=O)(=O)C2)=O)Cc2ccccc2N1C(C)=O Cc1c(C=CC(=O)NCC2(F)CN(C(c3cnnn3C3CC3)=O)C2)cnn1C C#CCC(C(=O)N1CC[Si](C)(C)C1)NC(c1ccc(F)cc1)=O C1(NC(c2ccc(C(N3CCCC3)=O)cc2)=O)NC(=O)N(CCOCC=C)C1=O C(CN=c1[nH]c2c(c(=NC3CCN4CCC3CC4)[nH]1)CCCCC2)OC(F)F c1(OC)nc(C(=O)NC(CNC(C2(C)CC2(C)C)=O)C2CC2)sc1C C(N=C(NC(C)COC(F)F)NC1CC(C)(F)C1)c1cnc(C)o1 CCC(C(=O)NC1CCN(C(c2ccc(F)c(O)c2)=O)CC1F)C(C)C N1(C(c2c(C)nns2)=O)CCC2(NC(=O)C(C)Oc3cccnc3)CCCC12 C(=O)(CS(=O)(=O)C(C)C)NC1CC2(CC(CNC(CCC(C)SC)=O)C2)C1 C1(NC(CC=C=C)=O)C(C)CN(C(=O)C=CCOC)CC1C c1(N2CCC(NC(c3ncc4ccccn34)=O)CC2)ccc(Br)c2ccccc12 Cc1nn(CC(N2CC(O)CC2CNC(C2CCCCN2N=O)=O)=O)c(=O)n1C C1(O)(CNC(C(C)OC(C)(C)C)=O)CCN(c2ncc(Br)cn2)C1 C1(CNC(C2CC(OCC)C2)=O)CN(C(=O)C#CC2CCCOC2)CCC1(C)C N1(C(C(CC)NC(=O)OC)=O)CCN(CC(N2CC(C(C)N(C)C)C2)=O)CC1 c1(NC(=O)NC2CC(CS(C)(=O)=O)C2)cccc(S(=O)(=O)CF)c1 CC(C)(C)C(CNC(=O)CSCCC#N)C(=O)Nc1cccc2c1CCO2 CN1CCN(C(C2Cc3nnsc3S2)=O)C(CNC(=O)Cc2ccnn2C)C1 C(=O)(C1OCCc2ccccc21)NCCN(C)C(c1nnc(O)cc1O)=O n1(CC)nc(C)cc1C(=O)NC(C1CC1C(=O)NCC1CC12CCOC2)C c1(NC(COCC(=O)NC(c2ccccc2)C(C)NC(C)=O)=O)ccccc1F N1(C(C(=O)N(C(C)C)C(C)C2CC2)C)CCC(c2cnn(C)c2)CC1 CC(CC=Cc1ccccc1)C(=O)NC1CCC1CS(N)(=O)=O C(C(C)C(=O)NC(C)CN(C(=O)Cc1cnn(-c2ccccc2)c1)C)OC c1(C(=O)NC(C2CC2C(=O)NC(c2cncc(F)c2)C)C)cc(Cl)n(C)n1 C=C1CCC(C(=O)NC(C)(CNC(c2ncn(C(C)C)n2)=O)C2CC2)CC1 c1(C(=O)NC(C(=O)NCC2CCN(CC)CC2)C2CCCO2)occ2c1CCC2 N1(C(C2(C#N)CCCC2)=O)CCOC(C(N2CCOCC2CO)=O)CC1 C(=O)(CS(=O)(=O)c1ccccc1Cl)N1CCC(CNC(C2CC(C)(CC)C2)=O)C1 n1(CC(=O)NC2CC(CCn3cc(C4OCCO4)nn3)C2)ncc(Br)n1 CC(C)C(C(=O)NCC1CC(NC(C2COCCN2C)=O)C1)Nc1ccccc1 C1(=O)C(C(C)C)CN1CCC.C(CC(C)C)OCCNC(C(C)NC(C)=O)=O N1(C(C=C2CCC(C)C2)=O)CCC(NC(c2ccc(OCCF)cn2)=O)C1C c1(C(=O)NC2CCN(C(c3c(N)nccn3)=O)CC2CO)nc[nH]c2ncnc1-2 C1(C(=O)NC(C2CCCO2)Cn2cc(CC=C)nn2)CCC(C(=O)O)CC1 N1(CCC(=O)NC(C2CCCN(C(C(CC)CC)=O)C2)C)CCSC(C)(C)C1 Cc1ccc(NC(=O)C(N2CC(O)(CCNC(C3CCC4CC34)=O)C2)=O)c(C)c1 C12(NC(c3c(CC)ocn3)=O)CCCC1CN(C(C13CCC(CC1)OC3)=O)C2 C(C(CC1CC1)C(=O)N(C1CCSCC1)C)NC(C=CC(C)C)=O Cc1cc(C(=O)NCCOCC(N2CCCC2(C)C(C)C)=O)[nH]c1C c1(COC)c(C(N2CC(O)(CN(C(=O)C(F)(F)CC3CC3)C)C2)=O)cnn1C Cc1cnsc1C(=O)NC(CC1CCOCC1)C(=O)NCc1cccs1 c1(C(=O)NCCN(C(C2=CC(C)CC2)=O)C2CC2)cc2c(F)c(F)c(F)cc2[nH]1 CC(CC(C)(C)C)C(=O)NC1CC(CNC(c2cccn2CC2CC2)=O)C1 c1(Nc2ccc(S(=O)(=O)Nc3c(C)ncs3)cc2)cc2cc(F)ccc2o1 c1(C(=O)NCC2CC(NC(C3C(C)(CC)C3)=O)C2)nnn(C)n1 CC1(N=c2[nH]nc(-c3ccccc3)o2)CCN1C(C1CCCSC1)=O C1(C)(CNC(C2CN(CCC)C(=O)C2)=O)CCCN(C(C2CC(=O)N(C)C2)=O)C1 N1(C(C2CC(CC)(CC)C2)=O)CC2CC1CN2C(C1CC(C(C)C)=NO1)=O c1(CNC(C=C(CC)CC)=O)cccc(C(=O)NC2CC2(C)C(C)C)n1 C1(C(=O)NC(C2CCN(C(c3cc(Br)c[nH]3)=O)CC2)C)CCC(=O)CC1C N1(C(CC(C)SC)=O)CC2(CCN(Cc3cn4ccccc4n3)CC2)CC1C C1(NC(c2n(C3(C)CC3)nnn2)c2conc2CO)(CSC)CCC(C)(C)C1 N1(C(c2cnc(C)c(N)c2)=O)CCOC2(CCCN(C(=O)C(O)CC(C)C)C2)C1 c1(OC)ncc(-c2cncc(C(=O)Nc3cncnc3Cl)n2)cc1C N1(C(CC2ON=C(C)C2)=O)CCCCC(C(=O)NC2CC(C(N)=O)C2)C1 Cc1cnc(C(=O)NC2(C)CC(NC(=O)CCC3CCCC(O)C3)C2)cn1 c1(C(N2CC(C(N)=O)(CNC(c3ccc(OC)nn3)=O)C2)=O)c(C)oc(C)c1C CCCC(C(=O)N1CC2CC(NC(=O)CCCCCSC)C(C2)C1)C(C)C c1(N2CCC(C)CC(C)C2)nc(=NCCSC(F)(F)F)[nH]c2cccnc12 c1(C(=O)NCCC2N(C(CC(C)C3CC3)=O)CCSC2)c(Cl)cc(C#N)cc1Cl c1(C(N(CCOCCNC(C(C)c2cccs2)=O)C)=O)cccn(O)c1=O Cc1cc(NC(c2nnnn2C)c2cocn2)cc(S(C)(=O)=O)c1 C(C(C(=O)Nc1cccc(Cl)c1O)C(C)C)NC(C(=CC1CCCC1)C)=O c1(SC)ccc(C)c(C(=O)OCC2=CCCCCC2)c1 c1(CC)ccc(C(N2CCC(O)(C(C)NC(=O)CCc3nncn3C)C2)=O)nc1 C1(CC(N2CC(c3cc(O)n[nH]3)C2)=O)CC(C)(C)CN1C(C(C1CC1)OC)=O C1(CNC(=O)C(O)C(F)F)CN(C(c2c(O)cccc2F)=O)CC12CC2 N1(C(C(CC)F)=O)CCC2(NC(C3C(c4ccccc4)C3(C)C)=O)CCCC12 C1(NC(CCCc2onc(C)n2)=O)CC12CCN(C(=O)CC(C)C(C)C)CC2 c1(SCCN(C)CC2CCN(C(CC)=O)C2)cc2ccc(C)cc2nc1Cl c1(C(=O)OC)ncccc1NC(N1CCCC(Cn2cc(CCCO)nn2)C1)=O CC1CN(C(=O)CC2CCN(Cc3cc[nH]c3)CC2)CC(C)O1 Cc1ccc(F)c(OCC(=O)N(C(CNC(C2CC3CC3C2)=O)C2CC2)C)c1 c1(C(=O)NCCN(CCC)C(C2COCC2C(N)=O)=O)ncoc1C1CCCO1 C1(CC(=O)NC2C(NC(CCN(CC)CC)=O)CCOC2)CCCC(C)(C)O1 N1(C(c2ccc(CCC)s2)=O)CCC2CCN(C(c3nccc(C)n3)=O)CC2C1 c1(C(N)=O)cc(Br)ccc1NC(C1CC(F)CN(Cc2ccnc(F)c2Cl)C1)=O c1(C(=O)NCCN(C2CC2)C(C2(C3(C)OCCO3)CC2)=O)c(F)cccc1F S(=O)(=O)(CC(C)(C)CC1N(C(=O)OC(C)(C)C)CC=C1)NC(=O)NCC1CC1 C1(NC(C(c2cccnc2)NC(C(C)C)=O)=O)CC2CC1C(O)C2O C(=O)(C1CNC(=O)c2ccnn21)NCC1N(C(c2scc(CC)n2)=O)CCCC1 Cc1ccc(CCC(N2CCCC2CNC(=O)C(O)C2CC2)=O)cc1Br C(C(CNC(=O)CC(=O)OC(C)(C)C)OC)NC(COC)=O c1(C(N(C2CCN(C(C3(C)CCCC3)=O)C2)CCC)=O)cc(F)c[nH]1 c1(-c2n(CC=C)nc(-c3ccc(Cl)nc3)n2)cc(C(=O)O)nc2c1CCCC2 CC1=NS(=O)(=O)NC=C1C(=O)NC(CNC(=O)CS(=O)(=O)CCOC)C1CC1 c1(OC)cnc(C(N2CCC(C)C2CNC(=O)Cc2c[nH]nc2O)=O)c(F)c1 C(=O)(CC1=NN(C)C(=O)C1)NCC1CCCN(C(C2(CC(C)C)CCC2)=O)CC1 c1(C(=O)NCC2(F)CC(CNC(CC3(C=C)CC3)=O)C2)nc(C2CC2)oc1C c1(CC(N2CCC(CN(C)C(C3CC3F)=O)C2)=O)csc2ccccc12 c1(OCC)ccc(CC(C)C(C)NC(=O)NC(=O)C2CC2)cc1.C1(=O)CN1 C1(C)(NC(CCCN(C(=O)OC)C)=O)CCN(C(=O)C(C(C)C)N(C)C)C1 c1(C(=O)NC(C2CCCC2)CNC(C(F)OC)=O)cn(Cc2ccccc2)nn1 N1(C(C(C)(N(C(CSCC)=O)C)C2CC2)=O)CCn2c(cnc2C)C1 C12C=CCN(C1)C2=O.C(=O)(C(CC1CCC1)OC)N(CCC(N)=O)CC N1(C(CC(C)(C(F)F)N(C)C)=O)C2CCCC1CC(NC(c1nccn1C)=O)C2 N1(CCOC)CCN(C(=O)C(CNC(=O)C(F)n2ccnc2)CC2CC2)CC1 C1(NC(c2cc(C(C)(C)C)sc2)=O)CCCC(NC(C2COCCO2)=O)C1 C1(NC(C(C2CCC2)NC(c2ccc(C(N)=O)[nH]2)=O)=O)CC(F)(F)C1 C1(OC)CC(C(=O)NC2CCOCC2F)N(C(=O)C(C)c2cc[nH]n2)C1 CC(CNc1ccccc1F)CS(N)(=O)=O.c12ncnc(n1)N2CCO CC(=O)CCCC(=O)N1CCC(C)C1C(=O)NCc1ccccc1C#N C1(C(=O)NCc2cn(CC)nn2)CN(C(C2CCC2C)=O)CC1C(C)C c1(C(N(C(C)CNC(c2cnn3ccncc23)=O)C)=O)ccc2c(c1)NCCC2 N(C)(C1CCCc2cccnc21)COC(C(c1ccnn1C)C)=O CC1OC(C)C(C(=O)NCC(c2ccc(CO)cc2)O)C1C C1(C)(NC(=O)NCc2onc(C(=O)OCC)n2)CC(O)CN1C c1(C(N)=O)nccnc1NC(C1CN(C(C2CC2(F)F)=O)C1)=O c1(NC(c2ccc(OC)c(NC(C)=O)c2)=O)cc(O)c2ccsc2c1 c1(C(=O)NCCNC(CC(c2ccc(C)cc2)(C)C)=O)c(C)ccc2nonc12 c1(C(c2ccccc2)NC(C(CC2CCCCC2)OC)=O)ccccc1F c1(C(N2CCC(=CCNC(C3CCCCC3)=O)CC2)=O)cnc2c(c1)CCOC2 N1(C(C(c2cccc(Br)c2)(C)C)=O)CC(NC(=O)C=CC=C(Cl)Cl)C(O)C1 CC(C(C)(C)O)N(C)C(C1CCN(C(=O)C=CC2CCOC2)C1)=O c1(C(=O)NC(c2cn(-c3cnncc3F)nn2)(C)C)ccc(Br)cc1Br c1(C(N2CC(CC)CN(C)CC2)=O)cc2cccc(C)n2n1 C(=O)(CCCCC(N)=O)N1C(C(C(=O)NC(c2cncnc2)C)(C)C)CCC1 C1(C(N(CC(COC)(C)C)C)=O)C2CC2CN1C(C1CCS(=O)CC1)=O c1(NC(c2cccc(-n3nccn3)c2)=O)cccc(Cl)c1CO N1(C(C#CC(C)C)=O)CCC2CN(C(=O)C(C)C(F)(F)C(F)F)CCC12 CC1(C)CCN(C(C2CCC(=O)NC2)=O)C(C(=O)NC2(CO)CC(F)(F)C2)C1 c1(C(=O)NCC2C(C)CCN(C(=O)Cn3nccn3)C2)cccc2c1nnn2C C(CCCCCC(=O)NCCN(C)C)N(C(C(CCC)C)=O)C c1(OC)ccc(F)c(C(=O)NCC2COCCN2C(=O)CN2CCS(=O)CC2)n1 C1(C(=O)NCc2n(CC)cnc2)CC(F)(F)CN1C(=O)C(=O)NOC CCC(CCCC(=O)NCC(O)CC(C)C)NC(C1C2CCC(F)C12)=O C(=O)(C1CCCn2nccc21)N1CC(C)CC(NC(c2cnc(C)s2)=O)C1 c1(C(=O)NC2C3(CCN(C(c4c(C)n(C)nc4)=O)C3)C2)cccn2ccnc12 c1(C(N2CCC(Cn3cc(-c4c(C)nc(C)s4)nn3)C2)=O)cc(N)c(C)cc1Br c1(CNC(CCCN(CCO)CC)C(=O)OC(C)(C)C)c(C)cccc1Br C1(NC(=O)CCCC2CCOCC2)CN(C(C2CC(F)C2)=O)CC2(CCC2)C1 c1(C(N(CCNC(C(CC)C#N)=O)C)=O)cc2cc(C)cc(C)c2[nH]1 C1(C(N(CC(C)(C)CNC(c2[nH]ccc2C2CC2)=O)CC)=O)CCCC(C)CC1 C(=O)(C(CCC)NC(c1ocnc1COC)=O)N(C(C#C)C1CCC1)C C(C(N)=O)(C(C)(C)C)ONC(c1c(C)n(-c2ccccc2Cl)nn1)=O C1(CNC(C(=O)NC(C)C)=O)CN(C(=O)C(N)CCC(N)=O)CCC12CCOC2 C=CCC(C(=O)N1CCC(C)(CNC(=O)C=Cc2ccccc2)C1)NC(C)=O c1(C(N2CC(C)(C)C(NC(C3CCCCC3)=O)C2)=O)cnc2nc(Cl)ccc2c1 C1(SC)COCC1NC(=O)CC1CCN(C(=O)C=CC(C)C)C1 NC(=O)CCC(C(=O)NCC1CC1c1cn(CC2CC2)nn1)n1ccnc1 C1(NC(C=COCC)=O)CCN(C(c2nn(C)c(C)c2Cl)=O)CC1C N1(C(c2c(COC)noc2)=O)CC=C(C(C)(C)C(=O)Nn2cnn(C)c2=S)C1 C1(NC(=O)CC2CC2(Cl)Cl)CN(C(=O)Cc2ccc(-c3ncon3)cc2)CC1F C1(O)(CNC(C2CCCS2)=O)CCCN(C(=O)C(O)COCc2ccccc2)C1 c1(CCCC)cn(CCCNC(c2ccnn2CC2CCCN2CC)=O)nn1 N1(CC(=O)NCC2(C)N(C(C3C(OC)CCC3)=O)CCC2)OC(C)(C)CC1=O Cc1cc(F)c(C(=O)NC23CC(C2)N(C(C2(c4cccs4)CC2)=O)C3)cc1F c1(C(=O)NC(C2CCN(C(C3(CCOCC)CCC3)=O)C2)C)c(Cl)nn(C)c1Cl N1(C(Cc2ccc(C)cc2)=O)CCOC2(CCN(C(=O)C(O)C(C)(C)C)C2)C1 N1(S(C(C)C#N)(=O)=O)CCC2CN(C(C3CC=CCC3)=O)CCC12 CCC(CC)C(F)C(=O)NC1CCN(C(=O)Cn2ccnc2C)C1 c1(CC(=O)NCC(C2CC2)NC(=O)CSc2ccccc2)ccnc2[nH]ncc12 C(=O)(N(CCC(=O)NCC(=O)NC)OC)C1(CC)CCCC1 C(C(=O)C1CCOc2ccccc21)OC(Cn1nc(C)c(Cl)c1)=O C#Cc1ccc(CNC(=O)C(=O)NC(C2OCCC2(C)C)C)cn1 CCCN(OC)C(=O)Cn1nc(C(C)CC)nc1-c1cc(OCC)cc(OC)c1 C(=O)(C1CNC(=O)c2ccnn21)N1CC(C)(C)OCC1CNC(C1(C)COC1)=O C=CC(C)(C)C(=O)NCC1CC(F)(CNC(=O)CNC(=O)OC)C1 C1(C)(C(=O)NCCN(C(=O)CC2(COC)CC2)CCC)CCN(C)C1=O C1(NC(C(C)NC(N)=O)=O)CN(C(c2cc(O)cc(O)n2)=O)C2CCCC12 c1(NC(C23C(CN(Cc4ccc(C#C)s4)C2)C3)=O)cc(F)c(F)cc1F C1(C(N2CC(C(CC)CC)C2)=O)CC2COCC(C1)C2.C(=O)(CC(C)CC(=O)OC)N c1(OC)ncc(-c2cscc2C(=O)NC2CCCC2)cc1Cl.N1(C)CCCCC1 C1(N(C(C2N(C)CCC2)=O)C)CC2CCC(C1)N2C(=O)CNC(=O)CN(C)C n1(C(C)C)cc(Br)c(C(=O)NC2CC(NC(C3CC3F)=O)C2)n1 c1(C(C)C)cccc(C(N2CCC(NC(=O)CCc3cncs3)C(F)C2)=O)c1N C1(C(=O)NCCOCCN(C(=O)CCc2ccncc2)C)COC2(CO)CC1C2 Cc1nc(C)c(CC(=O)NC2CC(C)(CNC(=O)CN(C)C(C)C)C2)s1 Cc1c(NCc2cccc(C(C)C)n2)nc[nH]c1=NCC1(C2CCC2)CCC1 C1(O)(CNC(=O)NC)CCN(C(C2C(C)(C)C2(C)C)C(COC)OC)C1 C1(C(c2n(C(CC)C)nnn2)NCc2cc(COC)cs2)CCC2(CC2)C1 C=CC1OCCC1C(=O)N(C)CC1CCN(C(c2cc(COC)ccn2)=O)C1 C(=O)(C1CCc2cc(Br)ccc21)NC(C(C)(C)NC(C=CC(C)C)=O)C c1(N2C(CCC(=O)NC(C(C)C)CO)CCC2)ccc([N+](=O)[O-])cc1Cl c1(C(N2CC(C)OCCC2)=O)cc(S(=O)(=O)N2CCSCC2)c[nH]1 C(=O)(C(C)(C(F)F)c1ccccc1)N1CCC(NC(Cc2c(C)non2)=O)CC1 C1(CNC(C2CN(CC)C2)=O)CC(C(=O)NC2CC(n3ccnc3)C2)CO1 CC(C)C(O)C(F)(F)C(=O)NC1CCC(NC(=O)C(F)C(F)(F)F)CC1 C1(C2CCN(C(C3CC4CCCC34)=O)CC2)(NC(CSCC(C)=O)=O)CC1 c1(C(N2CC3CN(C(Cn4ncc(C)c4)=O)C3C2)=O)cc(Br)cc([N+](=O)[O-])c1F C1(C(=O)NC(CN(C(C)=O)CC)C)CC1C1(C)COC1.C1(=O)CN1.C1(=O)CN1 C1(NC(C(C=C=C)C)=O)CCN(C(=O)Cn2ncc3ncccc23)CC12CCC2 C1(C)(COC)CC(NC(c2ncc(C(F)F)s2)=O)CN1C(=O)Cn1nnnc1C CC1CCCC(O)(C(=O)NC2(CNC(=O)CCF)CCCC2)CC1 c1(C(N)=O)ccc(CC(=O)NCC2(NC(=O)CC3CCC(=O)O3)CCC2)nc1 C(CCCCC(=O)NCCCCC(N)=O)N(C)C(c1cc(O)nc(O)n1)=O c1(C(CNC(c2c(C)ncs2)=O)NC(=O)C(O)CC2CC2)ccc(F)cc1F CCC(C(=O)NC1CCC1NC(=O)C(C)(C)n1ccc(Cl)n1)n1ccnc1 C1(C(N2CCC(C)C2CNC(C2CCC(=O)N2C)=O)=O)CCc2nnc(O)n2C1 c1(OC)ccc(F)c(N)c1C(N1CC(NC(=O)C(F)(F)c2cccnc2)C1)=O Clc1cc(Br)c(C(c2nnnn2CCCC2CC2)NCC2CC23CCC3)s1 c1(C(=O)OCC)ccc(NC(=O)Cc2cccc(Br)c2F)cc1Cl c1(COCC(=O)NC2(C(N)=O)CSC2)ccnc(O)c1.C1(=O)C(O)CN1 C(C(C(=O)N1Cc2cccnc2C1)C(C)(C)C)NC(c1ccc(NC(C)=O)o1)=O c1(C(N2C(CNC(CCCC(C)=O)=O)CN(C)CC2)=O)cn(C)c(=O)nc1O N1(C(c2cnn(-c3nccs3)c2)=O)CCc2c(OC(F)(F)F)cccc2C1 N1(C(C2CC(C#C)(O)C2)=O)CCC2(CC1)CC(C)N(C(c1coc(CC)n1)=O)C2 c1(NCC2CCCN(C(CCOC(C)C)=O)C2)ncnc2scc(Br)c12 Cc1cc(NC(=O)C(=O)NCCC2CCCN2C(=O)N(C)C)c(C)o1 c1(C(C)CC(=O)NCC(CO)NC(C2(O)COC2)=O)c[nH]c2ccccc12 CN1CCC(C#N)(CNC(c2[nH]ccc2CNC(=O)C2=NNC(=O)C2)=O)C1 c1(C(=O)NCC2CC3(CN(C(CC(=C)C)=O)C3)C2)cc(F)c(O)c(F)c1 C(C1=CCN(C(=O)C=CC2CCCO2)CC1)NC(=O)CSc1ccccn1 N1(Cc2cnn(C)c2C(N2CCCC2)=O)CC2CCCC(C1)C(=O)N2 C1(C)(C(=O)NC2CCC(NC(C3C(C)(O)CCC3)=O)CC2)CCCCNC1=O c1(CC)c(C(=O)NCC2C=CCN2C(=O)CN2CC(C)C2)cnc2ncnn12 O=S(=O)(c1ccc(N2CCC(CCO)C2)cc1Br)NCCN1CCCCC1 c1(NCc2cccc(NC(C)=O)c2)c(N)sc2cccnc12 n1(CC)cc(C(N2CC(C)(NC(C3COC(C)C3)=O)C2)=O)c(C(C)C)n1 N1(C(CC(C)CNC(=O)CCOCC(F)F)=O)CC2(CCC1CO)CC2 Cc1cc(=O)ccn1CC(=O)NC1CCC(N(C)C(c2cc(C(F)F)no2)=O)C1 c1(C(=O)NC(C)CC2CCC2)ccc2cn(C(F)F)nc2c1.c1(=O)c(=O)[nH]1 N1(C(C(c2ccc(F)cc2)C)=O)CC(CNC(=O)Cn2nnc(=O)[nH]2)CC1(C)C CCC1=C(C(=O)NCC2CC(C(N)=O)=NO2)CCCO1 c1(C(N2CC3C(NC(CP(C)(C)=O)=O)(CCC3)C2)=O)ccc2c(c1)CCC2=O Cc1cc(C(=O)NCCC2CC(NC(=O)C(C)OC3CCCC3)C2)ccc1Cl CCCCC(C)(F)C(=O)NC(CNC(=O)CCNc1cncnc1)CC N1(C(C(COC)OC)=O)CC2(CC(NC(c3cc(Cl)ccc3N)=O)C2)C1 N1(CCC)C(=O)CCC1C(=O)NCC1(NC(C2(C(N)=O)CCC2)=O)CCOC1 Cc1cc(F)sc1C(=O)NC(C)C(C(C)C)NC(c1cnn(C)c1Cl)=O CS(=O)(=O)C1CC(C(=O)NCCC2(O)CN(C(=O)CC3CCC(F)(F)CC3)C2)C1 c1(C(C(=O)NCCCC)N(C)C(c2cccc(O)c2)C)cc(S(N)(=O)=O)co1 C1(CNC(c2c(C(C)C)onc2)=O)CCC2(CCC2)C1NC(C1CCOCC1)=O c1(C(=O)OC)cnc(NC(C)CNC(c2cccc3occc23)=O)c2ccsc12 c1(OC)cc(O)ncc1C(N1CC2CC2(CNC(C2CC3(CC3)CO2)=O)C1)=O C1(CC)CCOC(CNC(=O)NCC2(c3ccno3)CC2)C1 c1(C2C(C)(C(=O)NCC(=O)NCC(C)O)C2)ccc(F)cc1F C(=O)(CCCC(=O)NCC1(NC(C2C=CCS2)=O)CCOC1)N(C)C C12(NC(N3CC(F)(CC)C3)=O)CC(CO1)N(C(=O)OC(C)(C)C)C2 C1(CN(c2nc(=N)nc(N3CCC4(CCCO4)C3)[nH]2)C)CC2OC(C)(C)OC2C1 C(=O)(C1SCCc2sccc21)N(C)CC1CCCN(C(=O)C2=CCCO2)C1 C=CC1CN(C(C2CC3C=CC2CC3)=O)CC1NC(=O)COCCCCC c1(C(=O)NC2CC(NC(CC3CCN(C)C3=O)=O)C2)cc(F)ccc1N Cc1nn(C)c(C)c1C(=O)NCC(C)(C)CNC(=O)CCc1cn(C)cn1 C1(C)(NC(C(c2ccc(C)o2)C)=O)CCCN(C(=O)CCCCC2CC2)C1 C(=O)(C(C1=CCSC1(C)C)N1CCCC(O)(C2CC2)C1)NCC(=C)C c1(CC(=O)NC(CC)C(c2ccc(C(F)(F)F)cc2)O)ccc(Br)c(F)c1 C1(C(=O)NCCCC(=O)NC(C2CCCC2)C#C)CCC(=O)C(C)C1 N1(C(c2cn(CC)nc2-c2ccccc2)=O)CC(C2CN(C(=O)C3=CCC3)C2)C1 N1(C(C)CN(C)C(C)C)CC2(CCC(CCN)O2)C1.N1(C(C(=O)N)C)C(=O)CCC1=O c1(NC(C2(C)N(Cc3cccc(OC)c3C)CC2)=O)c(O)cccc1C#N N1(C(C=CC(C)NC(=O)CCN(C)C)=O)CCC(CN(C)C)CC1 C(C(C)(C)CC(=O)NC1(CCNC(C2CC2c2ncccn2)=O)CCC1)OC c1(CC(=O)NC2(CF)CCN(Cc3nc(C)oc3)C2)c[nH]c2c(C)cccc12 C1(C(=O)NCC(c2nccs2)C)CC2CCCC2N1C(=O)C1=COCCC1 CCC(O)C(=O)NC1CCCC1NC(c1nocc1Cl)=O c1(CCC(N2C(C)CC(Nc3nccc(C(C)(C)C)n3)C2)=O)ccc(Cl)c(Cl)c1 C1(C(=O)NC(CC(N)=O)C2CC2)CCC2(CC2)N1C(=O)CC1COCCO1 c1(C(N(C)CC2CCN(C(C3CNC(=O)N3)=O)C2)=O)ccnc2[nH]nnc12 c1(CC)cc(C(=O)NC(C)(CNC(=O)COC(F)(F)F)C2CCC2)ccc1F Cc1nc(O)ccc1C(N1CCC(F)(CNC(c2cn(C)c(=O)n2C)=O)C1)=O C1(NC(CN2CCC(C)C2)=O)CN(C(C2(CC(F)F)CCC2)=O)CC1CO N1(C(Cc2cc(C)[nH]n2)=O)CCOCC(C(=O)N(C2CCCC2C#N)C)C1 C1(OC)(OC)CC2(CCN(c3cc(NC4CC(n5cncn5)C4)ncn3)C2)C1 C12(C)CC(CC)(CN1C(C)=O)C2.N1(CCC(=O)NCCCOC)C(=O)CCC1=O N(C1CCc2c(Br)ccc(Cl)c21)C(C(N1CCC(OC(CSCC)C)CC1)=O)=O CC1CN2CCN1CC2C(=O)NCCOCCN(C(=O)C(C)(C)CO)C C12(CNC(c3c(C)sc(Cl)n3)=O)CCCCC1CN(C(=O)C(F)(F)C(C)O)C2 C12(C(=O)NCCN(C(c3cn(C4CCOC4)nn3)=O)CC)CCC(CC1)C2(C)C N1(C(CN2CCC(OC)C2)=O)C2CCC(C2)C1C(=O)NC(c1ncn(C)n1)C c1(N(C2CC3CNC2C3)C(C(OCC)OC)=O)ccc(C#N)cc1 CCC(CC)(CO)C(=O)N(C(C)C(=O)N1CC(OC2CC2)C1)C N1(C(CCCn2ccc(C)n2)=O)CCC(C)C1CNC(c1cccc[n+]1[O-])=O c1(N2CCN(CCCN(C(c3cccc[n+]3[O-])=O)CCO)CC2)ncc2c(n1)COC2 C(CCC1CCC1)(C(=O)NC(c1cccc(C)c1)C)NC(C1C(C)=CCS1)=O Cc1ccc(C=CC(=O)N(CC(=O)NCC2CC23CCOCC3)C2CC2)cc1 CC(C)C(C(=O)N1CCC1C(=O)NCC1CCCN(c2cnccn2)C1)N(C)C C1(C(=O)NC2CCCN(C(CC3C(CC)C3)=O)C2)CCCCCN1C C1(S(C)(=O)=O)(C(N(C(CNC(C2(CO)CC2)=O)Cc2ccccc2)C)=O)CCC1 Cc1[nH]nc2ncc(C(N3CC=C(CNC(C4C(F)(F)C45CC5)=O)CC3)=O)cc12 c1(OC)cccc([N+](=O)[O-])c1C(N1CC(NC(=O)C(C)(O)C(F)(F)F)C(C)C1)=O c1(C(=O)NCC(CCOC)NC(c2cc([N+](=O)[O-])n[nH]2)=O)ccn2c1CSCC2 C(C1CCCCC1)=CC(=O)N(C1C2CN(C(C3CCOC(=O)C3)=O)CC12)C N1(C(Cc2c(=N)[nH]cnc2)=O)CC2(C1)C(NC(c1ccsc1)=O)CCS2(=O)=O N12CCN1C(CCO)C2.N1(CC=O)CCCCCC1.C(CC(F)(F)F)SCC=O N1(C(CCCOC)=O)CCC(CNC(=O)C2=COCCC2)C12CCC2 N1(C(=O)NC2C(CS(C)(=O)=O)C2)CCC(OCCNC(C2SCCCS2)=O)CC1 c1(NC2CC(C)CN(C(=O)C(C)(CO)CO)C2)ccc2ncccc2c1 N1(C(=O)OCC)CCC(c2ncc(C(=O)NC(C)CO)s2)CC1 C(C(C)(O)CCOC)NC(C(C)(C)N(C(=O)CS(=O)(=O)N(C)C)C)=O CCCC(C)(C)C(=O)N(CC(=O)N(C)Cc1cn(C)nn1)C C(c1ccccc1Br)=CC(=O)NCCCN1CCN(C(=O)OC(C)(C)C)CC1 c1(OC)ccc(C(=O)NC2CCCC(N(C)C(c3cc(C)sn3)=O)C2)c(OC)n1 C(CC(C)C)(C(=O)NC1CC(CNC(C2CNC(=O)O2)=O)C1)NC(C)=O C1(C(=O)NC2CC(CCNC(=O)Cc3ccns3)C2)CC2CCC1O2 c1(C(=O)N=c2ccn(CCC(F)(F)F)[nH]2)cc2c(O)ccc(F)c2cc1Cl CCCCCCC(=O)N1CCC(C(=O)NCC2(C)CC(F)(F)C2)C12CC2 Cc1ccc(=O)n(CC(=O)NCC2(CNC(=O)CCCC(N)=O)CCCC2)c1 c1(OC)c(C(N2CCCC(C(=O)N(C)Cc3cn(C)nn3)C2)=O)cnn1C C(=O)(C1C(OC)CCC(C)N1C(c1[nH]nnc1-c1ccccc1)=O)OC c1(C(C)C)ncc(Cl)c(C(=O)NC(C)C(C)NC(=O)CCC2CCN(C)C2)n1 C1(CNC(=O)Cn2cnnn2)CN(C(=O)C(O)Cc2cnc[nH]2)CC12CC2 N1(C2C(C(=O)NC(c3c(OC)ccc(F)c3)CO)C2)Cc2ccccc2C1 c1(OC)ccc2c(=NC(C)N3CC=CCC3)[nH]c(-c3ccccn3)nc2c1 Cc1nccc(C(=O)NC2CCC(NC(=O)C(C)(C)n3cnnn3)C2)n1 C(=O)(C(C)(C)CCNC(=O)CC1CCSC1)NC(c1c(C)nccn1)C Cc1cc(C(=O)NC2CC(O)CN(C(=O)CC3CC4(CCC4)C3)C2)cc(N)c1Cl C1(C(C)C)CN(C(C2(NC(=O)CC3OCCC3C)CCC2)=O)CC(=O)N1 C(=O)(C(C)(C)CC(F)F)NC1C(CC)CN(C(=O)C=Cc2cnn(C)c2)C1 C#Cc1ccc(C(=O)OCC(=O)Nc2ccc(Cl)c(Cl)c2C)cc1C c1(C(=O)NC2C(F)CCN(C(c3[nH]n(C)c(=O)n3)=O)C2)cnc2c(n1)CCCC2 N1(C(C(C)OCCCC)=O)CCSC(C(=O)NC(C)C#N)C1 c1(OC)nc(C(=O)NCCNC(=O)COc2ccc(F)cc2C)cc(O)n1 O=C(CCC(CF)CF)NC1CCCCC1NC(c1ccc2c(c1)CCC2)=O c1(C(N2C(C(N(CC(F)F)C)=O)CC2)=O)cn(C)cn1 C1(NS(CC(C)C)(=O)=O)CCN(C(=O)CC2CCC(=O)NC2=O)CC1F c1(CC(=O)NCC(C)N(C)C(c2cncn2C2CC2)=O)ccc(F)cc1Br C1(NC(CCOCCC)=O)CCOCC1NC(=O)Cc1cnoc1 N1(C(C(=O)NC(=O)OCC)=O)CCCCC1C(=O)Nc1cnc(CCC(C)C)s1 C1(C(=O)NC(C(C)(C)NC(c2c(C)c[nH]n2)=O)C)CCCN(Cc2cccs2)C1 C1(CCC)(NC(C2CC(F)(CF)C2)=O)CCCN(C(c2ccsc2C)=O)C1 c1(OC)cnc(Cc2nccn2C)c(C(=O)NCCN(C(=O)CSC(C)C)C)c1 C(=O)(C(F)C(C)CC(C)(C)C)NC(C)CCCNC(C1Cc2ccccc2O1)=O C1(CC)(CC)CC(NC(C2CC(C)(C)CN2C)=O)CN1C(=O)Cc1cn(C)nn1 N1(C(c2ccc(Cl)[nH]2)=O)CC2=C(C1)CN(C(c1cnc(C(F)F)cn1)=O)C2 C(CC(=O)NC1CCC(=O)NC1C)(C(F)(F)F)NC(c1c(NC)cccc1)=O N1(C(C(CC)F)=O)CC2CC1CCC2NC(c1ncn(-c2ccccc2)n1)=O C(=O)(CC1=CCOCC1)N(C(C)C(=O)NCC1(C)CCCC1O)CC c1(CNc2ccc(CNC)cc2)cc(C)ncc1Br c1(C(=O)NCC2(F)CC(NC(CN3CCC(C)(O)C3)=O)C2)ccc2c(c1)NCC2 C(=O)(C(CNC(C1CCOC1C1CC1)=O)CC1CC1)NC(C=C)C C1(CCn2ncc(C)c2)CCN(C(=O)CC2CCC(C)O2)CC1.N1(CC)CCCCC1 N1(C(=O)OC(C)(C)C)CCOC2CN(CC3(c4ccc(F)cc4F)CCCC3)CC12 c1(-c2nc(C(=O)NCCOC3CN(C(=O)CC4CC4)C3)sc2)ccccc1F C1(NC(c2cnn[nH]2)=O)CCC2(CC1)CN(C(=O)CN1C(=O)CCC1=O)CCO2 N1(C(C(C)=C(CC)C)=O)C2CC1CN(C(c1ccccc1Cl)=O)C2 C1(c2n(C)ncc2)CN(C(c2cncs2)=O)CCN1C(C1CCCCS1(=O)=O)=O N1(C(c2c(CC)n[nH]c2)=O)CCC(C(=O)NC(C)C(=O)OC(C)C)CC1(C)C C1(CC(=O)NC2CN(C(C3(CCOCC)CCCC3)=O)C2)CCn2cncc2C1 Cn1cncc1C=CC(=O)NC1CC1CNC(c1cn(-c2ccccc2)nn1)=O N1(CC(=O)NC2(c3ccc(Br)s3)CCC2)CC(c2ccc(Br)cc2)CCC1=O C1(SC(C(c2cccc(-c3nn[nH]n3)c2)(C)C)=O)Cc2ccccc2C(=O)O1 CCCC(C(=O)N1CCCCC1CNC(C1(c2ccccc2)CCOC1)=O)OC c1(CC2C(NC(=O)Nc3c(NC)cccn3)CCC2)c(C#N)cnc2ccnn12 CN1CC(O)CC1C(=O)NC1CCC(C)(CNC(=O)Cc2cn[nH]c2)C1 N1(C(c2nn(CC)nc2C)=O)CC2CC1C2NC(=O)CC(C)CN(C)C C1(NC(=O)NCC2CC3(C2)OCCO3)C2CC3CC1CC(O)(C3)C2 Fc1cc(F)c2[nH]c(=NCc3cn[nH]c3)[nH]c(=NCCc3ccc(Br)cc3)c2c1 C(=O)(CCCC(C)(C)C)N1C(CNC(C2C(C(=O)OC)CC2)=O)CCCC1 CC1=C(C(=O)NCC(C)(C2CCC2)NC(=O)C2=C(Cl)CCCC2)SCCO1 C(=O)(C1=CCCS1)N1CC(OCC(=O)NC(C2CCOCC2)C)C1.C(CF)O N1(C(c2csc(C(C)(C)C)c2)C(=O)NCC(=C)C)CCC(C(F)F)(OC)C1 CC(C(=O)NC1CC(NC(C2(C(F)(F)F)CCCC2)=O)C1)S(C)(=O)=O c1(OC)ccc(=NCC2(CNC(c3c(C)cccc3F)=O)CCC2)[nH]c1OC C1(CC)(NC(=O)CC2(C)CC2)CCCN(C(C2CCC2c2ccc(F)cc2)=O)C1 C(=O)(CCC(F)(F)C(F)F)NC1CCC2(C(NC(C(C)NC(N)=O)=O)C2)CC1 c1(OCCNC(C(=O)NC2(C)ON=C(C)C2)=O)ccc(CS(C)(=O)=O)cc1C c1(OC)ccc(C(=O)NCC2CN(C(=O)C(C(C)C)NC(C)=O)C2)cc1 C(C(C)NC(C1(CCNC(=O)CSCCOC)CC1)=O)OCC C1(NC(c2ccc(C)nc2)=O)CCN(C(=O)Cn2c(C)csc2=O)CC1F N1(C(C(C)NC(=O)OC)=O)CC2CS(=O)(=O)CC2(NC(c2ccns2)=O)C1 C=CCCCC(C)(C)C(=O)NC(CC1CC1)CC(N1CCCC2(C1)N=N2)=O CCCCC(O)C(C)C(=O)NC(C(N1CCCCC1)=O)c1ccoc1 CON1CCC(CC(=O)N(CC(C)N(C)C(C2C(F)(F)C23CC3)=O)C)CC1 CC(C)CCCCCC(=O)NC1(C(N2CC(c3nc(=O)o[nH]3)C2)=O)CCOCC1 C#CCCCCCCC(=O)N1CCC(C#N)(NCc2ccc([N+](=O)[O-])c(Br)c2)C1 C(C)(C(=O)NC1CCC1C(=O)NC1(c2ccsc2)CC1)(C1CC1)OC c1(C(N2CCN(C(CC(C)CF)=O)C(CO)C2)=O)ccc2ncccc2c1 C1(NC(c2n(CC)ncn2)=O)COC2(C1)CN(C(c1coc(Br)n1)=O)C2 C(=O)(CCCCCCCCCO)N1CC(C(C)NC(C2CCC2)=O)OCC1 c1(C(=O)NC2CC3N(C(C(CC)=O)=O)C(CC3)C2)ccc2c(C)[nH]nc2c1 CC1(NC(=O)CC2CCCCC2(F)F)CCN(C(c2ccc(C3CC3)s2)=O)CC1 c1(COC)cc(C(=O)Nc2nc(-c3ccc(Cl)s3)cs2)n[nH]1 CCC(C)(CNC(C1(F)CCN(C(C2(C)CCC(=O)N2)=O)C1)=O)CO N1(C(CC(C(F)F)NC(CCc2cc(C)no2)=O)=O)CCOC2COCC2C1 Cc1cc[nH]c1N(C1CCCCC1)C(N1CCC(Cc2ccncc2)C1)=O C1(O)(CC)CCN(C(C2CCN2C(C2CCCC3(CC3)C2)=O)=O)CC1 N1(C(c2c(N)c3c(cn2)cccc3)=O)CCN2CCN(C(C3CCSC3)=O)CC2C1 c1(C(N(C(CNC(COCCCC)=O)C)C)=O)cnn(CCN(C)C(C)C)c1C CC1=C(C)CC(C(=O)NC2CC3(C2)CC(NC(c2cc(Cl)no2)=O)C3)CC1 C1(CCNC(C2CC(CCC)C2)=O)CCN(C(=O)CCOC(C)C)C1 C#CCC(CC#C)NC(=O)C=CCN(C(=O)C(O)CC1CC1)C c1(OC)ccc(NCc2ccsc2C)cn1.C1(C)C(=O)OC(=O)N1 N1(C(C2CC3CN(C(COC(C)C)=O)CC2C3)=O)CCC2CCNC(=O)C12 N1(C(C2N(CCC)CCC2)=O)CC2CCC(NC(c3ccc(=O)n(C)c3)=O)(C2)C1 N1(C(CCSCC)=O)CC(NC(C2C=C(C)CS2)=O)C(CC)C1 C1(CCNC(C(COC)O)=O)CCCCN1C(c1csc(C(N)=O)n1)=O C1(NC(CSSC)=O)CN(C(c2cnn3cccc(Cl)c23)=O)C2(CCOCC2)C1 Cc1c(C(=O)NCC2CN(C(C3(N=[N+]=[N-])CC3)=O)C2)cc(C2CCCC2)n1C C1(C(=O)NCC(C2CCN(C(c3cccn3C3CC3)=O)CC2)C)CCCOCC1 C(C(N)=O)(C(N)=O)N(C(=O)Nc1ncc(C(C)C)s1)CCO N1(C(c2c(COC)nn[nH]2)=O)CCCC(C)C1CNC(=O)C(C)C(F)(F)F C1(NC(C=CCN(CC)CC)=O)CN(C(c2cnnn2C)=O)C2(CCOC2)C1 C#CC1(C(=O)NC(CC)CO)CCN(Cc2ccccc2Cl)CC1 CCCCS(=O)(=O)CC(=O)N(C1CCCN(C(C2CC2(C)C)=O)C1)C C12(CNC(c3nc(C(C)C)sc3)=O)CC1CN(C(C1(C)CC(C#N)C1)=O)C2 c1(OC)ccc(C(=O)N(C2CN(C(C3CC=CCO3)=O)C2)C)cc1O c1(CC)n[nH]cc1C(=O)NCC1(N(C)C2CC2)CCC1.c12coc(c1)NC2=O c1(C(N2CC(C(C)NC(C3CC(C(F)(F)F)C3)=O)OCC2)=O)ccc(F)cc1Cl c1(OC)nccc(C(=O)N(CC(C)(C)CNC(C2CCCC(C)C2)=O)C)n1 N1(C(C(CC)C)=O)CCCC(CCNC(C23CC(C2)C(c2ccccc2)O3)=O)C1 c1(C(=O)NC2CCN(C(C)=O)CC2)cnc(S(C)(=O)=O)nc1 C1(C(N2CC(C3(CNC(C(C(CC)O)C)=O)CC3)(O)C2)=O)CC2(CCCCC2)C1 CN1C(=O)CCC1CC(=O)NCC12CC(NC(C3CCC(N(C)C)CC3)=O)(C1)C2 C1(C(=O)NC(C2(CNC(=O)CCC(C)(C)C)CC2)C)C(O)C(=O)N(C)C1C C1(C2CCN(C(C3CCC3)=O)CC2)(NC(C(C)Cc2ccc(F)c(Cl)c2)=O)CC1 CCS(=O)(=O)C=CC(=O)N1CCOC(CN(C(=O)C(F)C2CCC2)C)C1 N1(C(c2ncc(CC)nc2)C(=O)NCC2COC2)CC(C)CC(C)C1 C1(NC(c2occc2Cl)=O)COC2(C1)CN(C(=O)CCc1cccc(F)c1)C2 N1(C(C2ON=C(C)C2C)=O)CCCC(NC(c2cccc(C(F)(F)F)c2)=O)C1C C1(C(=O)NC(c2nc(C3CC3)cs2)C)CC(CNC(C2CC3(CC3)CO2)=O)C(O)C1 N1(C(C(C2CC2)OCC)=O)CCN(C(c2ccc(Cl)c(Cl)c2)=O)CC1CC C(C(O)CC(=O)NCC1CN(C(c2ccnc(C(N)=O)n2)=O)CC1O)N(C)C C1(NC(c2ccc(CNC(C)=O)cc2)=O)CCCCCC1NC(c1cso1)=O C(=O)(C(C(C)C)N1CCN(c2cccs2)CC1)NC1CCN(CCOC)CC1 N1(C(C2CC(OC)C2)=O)CC2CN(C(c3conc3C(F)(F)F)=O)CCC12 C1(COC)CN(C(C2(c3cccc(Cl)c3)CC2)=O)CCN1C(=O)CCC(N)=O C#CC(CC(C)(C)C)NC(C1(C(C)NC(=O)C(O)CN2CCCC2)CC1)=O C1(C(N2CCC(C(C)(C)C(=O)NC3CC=CCC3)C2)=O)CCCC(=O)CC1 S(=O)(=O)(c1ccc(NCC(C)OC(C)(C)C)c(F)c1)NC(c1cncc(C)c1)C Cc1cccc(C(CNC(C2CC(=O)N(C)C2)=O)NC(c2csc(O)n2)=O)c1 CCCCCC(O)C(=O)NC1CCN(C(C2(C(N3CCCC3)=O)CC2)=O)C1 c1(C(N2C(CNC(c3cccc(CC)n3)=O)CCC2)=O)nc(Cl)ccc1OCC N1(C(CNCCC)=O)CCc2ccsc2C1C c1(C(=O)OC)cc(F)ccc1OC.n12ccc(n1)C(c1nnnn1C)NC21CCC1 CC1CCCC(C)N1NC(=O)CC1CCCN1C(=O)OC(C)(C)C C=C(C)CC(C(=O)Nc1cnn(C)c1CC)NC(C1CC(C)C1)=O C1(n2cc(C3CCN(C(=O)CC45CCCC4C5)C3)nn2)CCC(F)(F)CC1 C1(NC(C(CSC)(C)C)=O)CCC(C)(NC(C2CC3CCC(C2)O3)=O)CC1 CCN=c1[nH]cc(C(N2CCC(O)C(NC(C3CCC3(F)F)=O)C2)=O)s1 c1(C(=O)NCC(CO)NC(c2nc(CCC)sc2)=O)ccc(-n2ccnc2)cc1 C(CC(C)(C)C(=O)N1CCC(CN(C(=O)CCCCO)C)C1)OC c1(OC)ccc2c(c1)CCC2C(=O)NC1(C)CCN(C(=O)C(Cl)=CCl)C1 N1(C(C2(SC)CCC2)=O)CCC(CC(=O)NC2C=CCCCC2)CC1 C1(NC(C(C)NC(C2CCCC2)=O)=O)(CO)CCCN(C(=O)C(C)CF)C1 N1(C(CCCC(C)=O)=O)CCCC2(CCCN2C(c2csc3ccccc23)=O)C1 CCC(C)CCCC(=O)NC(C)C=CC(N1CCNC(=O)C1C)=O c1(C(N2CC3CCCC3(Nc3ccon3)C2)=O)ccc2cccc(CO)c2n1 N12CCC(C1)C(C)CNC(=O)C1CC(C1)SCC2=O.N(CCOC)(CC)CC c1(C(C)(C)C)cccc(CC(N2CCC(N(CCO)C(C3CCC(=O)O3)=O)C2)=O)c1 c1(C(=O)NC(C2CC2C(N2CC(F)CC(F)C2)=O)C)cnccc1C#N C(=O)(N(CCC(=O)N(C1CCCC1)CCCO)OC)C1C(C(=C)C)OCC1 C1(NC(C2CCCO2)=O)CC2CCC1CN(C(C1CC(O)C(F)C1)=O)C2 N1(C(CCCc2cc(C)sc2C)=O)CCCCC(CNC(=O)C2=NNC(=O)C2)C1 C#Cc1cc(N(C2CC2)CCOC)cc(N)c1.N12CCOC(C)(C1)C2=O c1(CC(=O)NCCNC(CN(C)C(=O)OC(C)(C)C)=O)cccc2ccccc12 C(=O)(C1=CCCOC1)NC(C(=O)N(C)CC1C(C)CCC1)CCF c1(C(N(CCNC(C2CC3CCC2C3)=O)CC)=O)ccc2c(c1)C(=O)NC2 C1(NC(C(CCOC)C)=O)CC2CCC1CC2NC(C1CCCN(C(C)C)C1)=O C(=O)(CCCCCCNC(c1cccc(C)c1C#N)=O)NCC(CC)CC(C)C CC(O)(CC(=O)N1CC(N2CCN(C(C3(N(C)C)CCCC3)=O)CC2)C1)C1CC1 C(=O)(C(CC)C(=O)NCC(C)N(C)C(c1occ(Br)c1C)=O)OCC N1(C(C=CC(CC)C)=O)CCC2(CC2)CC1C(=O)NC1(CO)CCC(C)C1 CC1CCCC(C)N1C(=O)C(=O)NC1C2CC1N(C(=O)C=Cc1cncc(O)c1)C2 c1(C(=O)NCCC(C)NC(Cc2ccc(C)c(O)c2)=O)cc2ccc(O)nc2s1 C1(C(N(CC(CCC)O)C)=O)(CNC(=O)CC2CC3CCC2C3)CCCCC1 N1(C(c2c(NC)nccc2)=O)CC(CO)C2(C1)CN(C(C1CC(C(F)F)C1)=O)C2 C1(CCC)(NC(C2CC2F)=O)CCN(C(C2CCCOCC2)=O)CC1 c1(N(CCC)CCNC(=O)C(=O)NC2CC2)cc2c(cn1)C(=O)CCC2 C1(NC(Cc2c(C)ncs2)=O)CCN(C(C2(C)CC2C)=O)CC1F c1(C(=O)NCC(CC=C)NC(=O)CC(C)n2ccnc2)c(Br)cnn1C c1(C(=O)OC)ccc(O)cc1F.C12CCCC(C1)CNC(=O)N1CC(C1)C(=O)N2 C(C(C)CC(=O)N(CC(=O)NC(c1nnnn1C)C)C)OC C1(CNC(C(C=C)O)=O)CCCCN(C(c2c[nH]c(=NC)o2)=O)CC1 C(=O)(C(C#N)C(C)(C)C)NC(C)C(CO)NC(c1ccc(SC(F)(F)F)cc1)=O C1(CN(C)C(C2CC2c2cccc(O)c2)=O)CCCN(C(=O)C=CCF)C1 N1(C(=O)NC)CCC(C(=O)NCC2CC(C(=O)O)C2)CC1C1CC1 N1(C(CC(CC)C2CCC2)=O)CCN(C(c2ccncc2)=O)CC1c1ncc[nH]1 C1(C(=O)NCC(CNC(C2(CC3CC3)CC2)=O)CO)CC2(CCCC2)CO1 C1(CC)(NC(C2CCCN(C)C2)=O)CCCN(C(=O)CC2CCC(C)C2)C1 c1(C(=O)NC2CN(C(C(CC#C)O)=O)C2)cn2c(Br)cnc2s1 C1(C(C(=O)N(C2CN(C)C2)C2(C(=O)OCC)CC2)C)CCCCN1CCO Cc1ccc(CC(C(=O)NC(C)(CNC(c2occc2Cl)=O)CO)N(C)C)cc1 N1(C(C=CCCC)=O)CC2CCCC(CNC(=O)C3Cc4ccccc43)C2C1 C1(OC)CCN(C(C2CC2C(=O)NCCCC(=O)OC)=O)C1 c1(NCc2n(C(C)C3CC3)ccn2)c[nH]c2c(-c3ccnc(F)c3)cccc12 CCS(=O)(=O)C=CC(=O)N1CCN(C(c2ccc(C(F)(F)F)c(O)c2)=O)CC1 CCCC(C)CS(=O)(=O)N(CC(C1CCCCC1)O)C c1(C(N2CCC(C)(NC(C(CCOC)OC)=O)C2)=O)cc(F)c(Cl)cc1F C12(NC(CCCc3c(C)ccs3)=O)CCOC(CNC(c3cnco3)=O)(C1)C2 C=Cn1nncc1S(=O)(=O)Oc1ccc(C(=O)OCC(C)C)cc1 C(=O)(CCC(CC)NC(=O)COC1CCCCC1)Nc1cccc(OC)c1 C(c1cnc(OC)nc1)=CC(=O)N(C(CCNC(CC(CC)C)=O)C)C c1(CC)cccc(CNC(=O)C(=O)N2CC(OCc3ccc(Br)cc3)C2)c1Br C(=O)(CC(F)(F)Br)NC(CC)C(=O)NCCNC(=O)OC(C)(C)C C(=O)(C(O)CCN(C)C)N1CCC(NC(c2cnc(OCC)s2)=O)C1 c1(C(=O)NCCC(C)N(C)C(C2CCCC2(F)F)=O)nccc(Cl)c1F CC1CN(C(=O)CC2CC(=O)NC2=O)CCN(C(c2c[nH]nc2F)=O)C1 c1(C(C)=O)cc(NCC(C)NC(c2ncoc2C2CC2)=O)ccc1[N+](=O)[O-] C(N=c1cc[nH]c(C#N)n1)C1CCCN(C(CC(C)OC)=O)C1 C(=O)(N1CC(O)CO1)c1c(CNC(CC2(OCC)CCC2)=O)cnn1C N1(C(C(CCC)OCC)=O)CC2(CCN(C(c3nc(Cl)cs3)=O)CC2)C1 c1(C(=O)NC2C(NC(C(C)OCCOC)=O)CCCC2)csc2c(C)cccc12 C(N=c1[nH]c(N2CCOC(c3ccco3)C2)nc2c1COC2)C1C(C)(C)NC(=O)O1 C(CC(O)C(F)F)NC(C1N(C(CCOCC)=O)CC1)=O c1(C(=O)NCCOCCCN(C(C2(C(=O)NC)CC2)=O)C)sccc1Cl N1(C(C(C(C)C)Sc2ccccc2)=O)CCCC(O)(C(N)=O)C1 CCC(CO)(C(=O)NCCC1CCN(C(c2ccn(CO)c2C)=O)C(C)C1)OC N1(C(c2cc(C)n(C)c2)=O)CCN(C(c2ccc3nccn3n2)=O)C2(CCC2)C1 C1(NC(Cc2c(C)cc(C)s2)=O)CCN(C(C2CCC(C)(C)CO2)=O)C12CCC2 CC(C)CCCCCC(=O)NCC(C(=O)NCC1(O)CC(C)(C)C1)N(C)C CC1(C)CC(CNC(C2(CO)CCOCC2)=O)N(C(c2ccnc(Cl)c2O)=O)C1 N1(C(c2cc(=NC)[nH]cc2)=O)CCC(C)(C)CC1C(=O)NCCC[Si](C)(C)C C(CC(O)(CC)CC)NC(=O)NC.N12CCN(CC1)C(C=C)C2=O c1(C(=O)NC(C)CCCNC(C2CC(CF)C2)=O)ccc(O)cc1Cl C(=O)(CS(=O)(=O)C1CC1)N1C(CC)CN(C(=O)C(C)(C)Nc2ccccn2)CC1 C1(C(N(CC(C(=O)NCc2nnc(C)s2)C)C)=O)CC2COCC2C1 CC(C)(CCCNC(C1CC2(C1)CC(O)C2)=O)C(=O)NC1CC1c1ccco1 c1(CC(c2nnnn2-c2cccc(Cl)c2)(C)NCCOCC)ccc(F)cc1Br Cc1cccc(SCC(=O)NC(C)(C)CNC(c2cnn(CC3CC3)c2)=O)c1 N1(C(CNC(=O)O)C)CCCCC1.C1CC(=O)NCC(=O)N1CC.C1(SC)CCCO1 c1(C(=O)NC2CC(CNC(Cc3ccc(C)s3)=O)C2)nn2cccnc2c1Cl c1(SC)cc(C(N2CCCC2CN(C(=O)CCC2CC2)C)=O)c(Cl)cc1Cl N1(C(C(C)C2CCCC2)=O)CCC(F)(N2CCOCC2)C1 c1(SCC)ccccc1C(N1CCOC(CCNC(C2(F)CC2)=O)C1)=O C(=O)(C1=NN2CC(C)CN=C2N1)NCC(C1CC1)NC(C1CCC(CC)CC1)=O c1(C(c2ccccc2)NC(C2(F)C3CCCC23)=O)ccccc1Cl C1(NC(c2c(OC)ccs2)=O)CC2CC(C1)N(C(c1c(F)cc(O)cc1F)=O)C2 C(C#Cc1ccccc1)N(C1CCC(c2cc(O)[nH]n2)C1)C N1(C(c2c(C)snc2)=O)CCCN(C(=O)C(F)CC2CCCCC2)C(C)C1 C(=O)(CCCS(N)(=O)=O)NC1C(CNC(CSC(C)(C)C)=O)CCCCC1 C(=O)(C(C#N)C(C)(C)C)NC(C(=O)NCC(C)Cn1cccn1)c1cccs1 N1(C(C2(CC(C)C)CNC(=O)C2)=O)CC2(CCN(C(=O)Cc3cscn3)CC2)C1 C1(CC)CN(C(c2csc(C(C)(C)C)n2)=O)CC1NC(=O)C(C(C)C)SC N1(C(C(CC)OCC)=O)CCC(C2CC2)C1C(N1CCC12CC(C)(C(N)=O)C2)=O C(CC(C(C)C)NC(=O)C(N1CCSCC1)C)N(C(C(c1ccc(Cl)s1)C)=O)C c1(C(=O)NC2CCCC(NC(=O)Cn3nccn3)CC2)ccc2ncccc2c1 C1(CNC(Cc2c(C)con2)=O)CCC2CN(C(c3ccc(N)c(F)c3)=O)CC12 O=C1NCC2CN(Cc3ccc(Cn4cc(I)cn4)cc3)CCC2N1 c1(C(N2C(C)CCN(C(C3C(C)C3(F)F)=O)CC2)=O)cc(F)cc2cc[nH]c12 CC1(NC(c2ccsc2-c2ccccc2)=O)CCN(C(C23CCC(C2)C3)=O)C1 CCC(C)(C)C(=O)NCCCCCN(C(=O)CC(C)(C)c1ccccc1)C N1(C(C(CCSC)OC)=O)CC(CNC(c2coc(C(F)F)c2)=O)CC12CCC2 c1(C(C)=O)cnc(N2CCCC2C(N2CCC(C3CCCNC3)CC2)=O)c(C)c1 CCCCC(CC)CC(=O)NCC1CC(F)(CNC(c2nn(C)c(N)c2C)=O)C1 Cn1cc(NC(=O)CSC)cc1C(N1CCCC1Cc1ccccc1O)=O CCC(CC)C(F)C(=O)N1CCC(CC(=O)NCCC2OCCC2C)CC1 c1(C(=O)NC2CCC(C)N(C(=O)CCC3CCCC3)C2)ccc(P(C)(C)=O)s1 C1(NC(C)=O)CCC2(CC1)CCN(C(=O)NCC1CN=C3N=CNN3C1)CC2 Cc1cnc(C(=O)NC(C)C(=O)NC2CCCCC2(F)F)c(F)c1 C12(NCC3C(c4n(Cc5ccccc5)nnn4)OCC3)CCCC1CCC2 C(=O)(C(N)CCC(=O)C(C)N1CCCCCC1(C)N)OCC CN1N=C(CC(=O)N2CCC3(CCCN3c3nc(C4CC4)ns3)C2)CC1=O c1(C(N2C(Cn3cc(CCCC)nn3)CCC2)=O)cnc2[nH]cc(C)c2c1 C1(CNC(Cc2cn(C)nc2)=O)CCCC(Cn2cc(C3COCC3O)nn2)C1 N1(C(CC(C)C2CCCO2)=O)CC2(NC(c3cc(Br)c[nH]3)=O)CC1C2 c1(C(=O)NC(CN(C(C(C)OCC=C)=O)C)C)c(Cl)csc1Cl N1(C(C(C=CC)O)=O)CC2CCCC(C1)N2C(=O)C(C1CC(F)(F)C1)O C1(C(=O)NC2C(CNC(c3ccn4ccsc34)=O)CC2)CC2(C1)CC(O)C2 CCC(CC(=O)NCCCOCCNC(c1ccnc(O)c1)=O)c1ccccc1 c1(CC(=O)NCCN(C2CCCC2)C(C2CC23CCC3)=O)cn2ccsc2n1 c1(C(N2CC(N(C(=O)CC3C=CS(=O)(=O)C3)C)C(C)(C)C2)=O)ccc(Cl)c(C#N)c1 CC1C(N(C)C)CCN1C(=O)CCCCN(C)C(C1CCC(=O)NC1)=O C(=O)(C1=C(CC)CCCC1)NC(CCC)CCCNC(c1ccc(O)c(C)c1)=O CCC(C)CC(=O)NCC(C)N(C(=O)C(c1ccccc1OCC)(C)C)CC C1(C(=O)NCc2cnc(COC)s2)CC(F)CN(Cc2cncc(C)c2)C1 C(C1=CCN(C(C2CCN2CC)=O)CC1)NC(C1CC(SC)C1)=O C12(C(N3C(CCOc4cccc(OC)c4)CCCC3)=O)C3C4C1C1C2C3C41C C1(CNC(=O)CCOC2CC2)CC2CN(C(c3cccnc3O)=O)CC12 c1(C(C)=O)cc(NC2CCN(C(C3CC(=O)N(O)C3)=O)CC2)ccc1[N+](=O)[O-] N1(C(CCN(CC=C)C(C2CCCOC2C)=O)=O)CCCC2NC(=O)CC12 C1(NC(C(C)OCOC)=O)CC2(C1)CN(C(C1CCCN(C)C1)=O)C2 N1(C(CC(=O)OC)=O)CCCC1C1CCCCN1C(c1cncc(C)c1C)=O C=CCCCCCCC(=O)NCCCN(C(C1CCCN(C(=O)C2CC2)C1)=O)CC N1(C(CN(C2CCCCC2)C)=O)CC(F)(F)CC1c1nc(-c2cccc(F)c2)no1 CCCC(O)CC(=O)N1CCC(C(C)NC(=O)CN2C(C)CCC2C)C1 O=C(CCCCn1ccnn1)NCC1CCCN(CC2CC2CC(=O)OC)C1 N1(C(c2c(CC)n(CC)nc2)=O)CCOC2(CCN(C(=O)C(C)C3CC3)C2)C1 C(C1CCCC1)=C(C)C(N1CCC(CCC(=O)NCCC#CCO)C1)=O C1(C(=O)NC(CNC(c2c(SC)cc(C)cc2)=O)(C)C)CCCC2CCCN12 N1(C(C(N2CCC(N(C(CSc3nc(C)[nH]n3)=O)C)C2)=O)C)CCOCC1=O c1(C(N(C(C(=O)N(C)Cc2cc(CO)[nH]n2)(C)C2CC2)C)=O)nncn1C c1(SC)nccc(=NC(=O)c2cncc(CNC(=O)CN3CCCC3)n2)[nH]1 S(=O)(=O)(c1ccncc1)N1CC(F)CC(C(=O)Nc2cc(C)cc(Br)c2)C1 c1(-c2ccc(NC(c3ccc(C)c(F)c3)=O)cn2)csc2ccncc12 c1(NCC(C)NCc2c(C)cc(C(F)F)o2)c(Cl)cc([N+](=O)[O-])cc1Cl C1(CC#C)CCN(C(C(=O)NCC(=C)C)C2CC2(Br)Br)C1 CCC(C(=O)N(CC)CC1CN(C(=O)Cc2cc[nH]n2)C1)N1CCCC1=O C1(NC(CCCC)=O)C2CC1N(C(=O)Cc1cc(C(F)(F)F)co1)C2 C1(O)(CCNC(c2cc(C)n(C)c2)=O)CCN(C(=O)CC2C(=O)NN=C2C)CC1 c1(C(=O)NC2CCC(NC(C=CS(C)=O)=O)C2)ccc2c(c1)CCCC(=O)N2 C1(NC(=O)C(c2cc(C(F)F)no2)N2CCC(c3cnco3)C2)CCOCC1 N1(C(CC(=C=C)C)=O)CC(C(N2CC(OC(F)F)C2)=O)C2(CC2)C1 Cc1cc(C(=O)NC2C(C(=O)NCC3C(C)C3C)C2(C)C)ccc1O CC1SCCCC1C(=O)NC1COCCC1C(=O)N(CC(C)(C)C#N)C C12(NC(c3c(C)onc3C3CC3)=O)CCOCC1CN(C(=O)C(C)C#N)C2 c1(N2CCN(C(C)CO)CC2)nc2c(c(=NCC3CC=CC3)[nH]1)CSC2 Cc1nc2c(o1)CCCC2CC(=O)NC1(CNC(=O)C#CC(C)(C)C)CC1 C1(C(=O)NCc2ccco2)(CNC(C(CC)C)=O)CC12CCC2 N(C(=NCCN(CC(C)C)CC)N1CCC(CC)C1)CC(CC=C)CO.OC O=C(N1CC(n2cc(-c3cnn(C(F)F)c3)nn2)CO1)c1ncc(C(F)F)cn1 C1(CC)CN(C(C2CC23CCCCC3)=O)CCN1C(=O)C=Cc1ncco1 N1(C(c2ncc(CC)nc2)=O)CC2CCN(C(=O)C(C)CCOC)C2C1 c1(N(CC(=C)C)C)nc2cccnc2c(=NCC(C)C(Cl)(Cl)Cl)[nH]1 CC(C)CC(C)CC(=O)NC1CCCC12CN(C(c1cnn(C3CC3)c1)=O)C2 c1(OC)nn(C)cc1C(=O)NC1CC(CCNC(=O)CC2CC2)C1 N1(C(CNC(Cc2cn(C)nc2)=O)=O)CCCC(C)(O)C1 C(=O)(C#CC1(C)CC1)N1CC(CN(C)C(=O)OCC)C(N2CCCC2)C1.C(C)(C)(C)O C1(CNC(c2c(SC)cccc2)=O)CC12CCN(C(=O)Cn1nnc(C)n1)CC2 CN1C(=O)NCC12CN(C(=O)C(O)CNC(=O)C=CC1CC1)C2 Cc1ccc(F)c(NC(C2(CNC(c3cnn(CCF)c3)=O)CCCC2)=O)c1 C(=O)(C(CC1CCC1)N1CC(Cc2cnccn2)C1)NC(C)C N1(C(c2n[nH]c(C)c2Cl)=O)CC2CCC(NC(=O)C=CC(=O)NC3CC3)CC2C1 c1(C(N2C(CNC(C(CC)n3ccnc3)=O)CC3CC32)=O)cc2cccnc2s1 C1(NC(CS(=O)(=O)NCC)=O)CCC12CCN(C(=O)C(C)C1CC1)CC2 C1(CC(=O)N(C2CCCN(C(c3ccnc(CO)n3)=O)C2)C)CCCN(C)C1 C1(C(N2CC(CN(C(=O)C(F)(F)CN(C)C)C)OCC2)=O)CCOCC12CCC2 C1(CNC(c2c(CC)[nH]nc2Cl)=O)CN(C(=O)CCCOC(C)(C)C)CC12CC2 C(C(C)(C)CC(=O)N1CCCC1C(C)NC(=O)CCc1cncc(OC)c1)OC Cc1cc(Br)ncc1NC1CCCCN(C(=O)OC(C)(C)C)C1 [N-]=[N+]=NCCCCCCCS(=O)(=O)NCC1CN(c2ncc(Br)cn2)CCO1 C(CCNC(C1(F)CCOC1)=O)(C(=O)NC1CC(C(C)(C)O)C1)OC N1(C(C2(F)CCCCC2)=O)CCC2CCN(c3nc4cc(Br)ccc4o3)CC2C1 C#CCC(O)C(=O)N(CCNC(C1(NC(=O)OC(C)(C)C)CCOC1)=O)C1CC1 c1(OC)cccc(S(=O)(=O)N2CCC(C(C)Nc3ncc(F)cn3)CC2)c1 c1(CC)nsc(N)c1C(=O)NC1CC(CCNC(=O)CCc2ccccc2)C1 N1(C(c2c(CC)occ2)=O)CCCC1C=CC(=O)NCC(O)C1CC1 c1(C(=O)NCC(CN(C(c2c(C)nc(Br)o2)=O)C)O)c(C)nc(=N)[nH]c1C c1(C(=O)NC(C(C)NC(=O)Cn2ccc(C(F)F)n2)C)c(F)ccc(C#N)c1F C1(C)(C(=O)NC2CC(CCNC(CN(C)C(c3ccsc3)=O)=O)C2)CC=CCC1 N1(C(c2cc(C)oc2)=O)CC2CCC1C(CNC(c1cccc3c1COC3)=O)C2 C1(CC=C)(C(=O)NCC(c2ccccc2)F)CCCN1C(=O)COC(C)(C)C c1(C(N2C(CNC(CC(C)F)=O)CCC2)=O)ncsc1S(N)(=O)=O C1(C(C)NC(c2n(CC)cnn2)=O)CN(C(=O)Cc2ccnc(F)c2)CCO1 c1(C(=O)NC2CCCC(C(=O)NCC(=C)C)C2)ccc(OC)c(F)c1 N1(C(c2c(C(C)C)[nH]cc2)=O)CCN(C(=O)Cn2nccn2)C(CS(C)(=O)=O)C1 c1(C(N2CC(COC)(NC(=O)Cc3cncnc3)C2)=O)nc(C)n2ccccc12 C1(CNC(C2C(C)(C)C2)=O)CC12CCN(C(=O)CNC(=O)C1CC1)CC2 C(CNC(c1csc(S(N)(=O)=O)c1)c1nnnn1C1CCC1)(CC(C)(C)C)OC NS(=O)(=O)C(C(=O)NC1C=CCN(C(c2ccn(C3CC3)n2)=O)C1)c1ccccc1 C(=O)(CC(O)C(C)CC)NCC(CC(=O)NCc1[nH]nc(COC)n1)O C1(C#N)(C(=O)NCC2C(NC(c3cc(OC)n(C)n3)=O)CCC2)C2CCCCC12 C1(NC(CCOC)=O)(CNC(C2CC3C=CC2C3)=O)CCC(C)(C)CC1 C=C1C(OC(=O)C(=O)Nc2ccccc2C(C)(F)F)CC2CC1C2(C)C C1(CNC(CNC(CN(C)C)=O)=O)CCCCN1C(c1csnc1Cl)=O N1(C(Cc2n(C)cnn2)=O)CCC2CN(C(c3ccsc3)=O)C2C1 N1(C(c2c(COC)cco2)=O)C2CCC1CN(C(C1(C(C)(C)C)CCC1)=O)CC2 C1(NC(c2ccc(CO)o2)=O)CCCC(C(=O)NCc2nc[nH]n2)C1 C(=O)(C(C)C(C)(F)F)NCC1(C(F)F)CCN(C(C(N2CCN(C)CC2)C)=O)C1 CC1=C(C)CC(C(=O)NCC2(NC(C3CCN3S(C)(=O)=O)=O)CCCCC2)CC1 c1(N(CCCC(=O)NC2CCC2)C)ccc(F)cc1Cl N1(C(CC2(C#N)CC2)=O)CCC2(CCOC2)C(CNC(C2CCCC(O)C2)=O)C1 C(=O)(C1=CCCN(C(=O)C(C)(C)OC(C)C)C1)NC(CC(=O)NC)C1CC1 C1(C(=O)NC2C(CC=C)CCC2)CN(C(C2CCCNC2=O)=O)CCC1(C)C c1(C(N(C(C)CNC(C2CC(O)C2)=O)C)=O)csc2ccc(F)cc12 C1(NC(C(C)(C2CC2)OC)=O)(CNC(c2cnc(C3CCC3)[nH]2)=O)CCCCC1 CC1CCC(F)(F)CN1C(C1(CCNC(=O)CCP(C)(C)=O)CCC1)=O C(=O)(CCCC(C)(C)C)N(CC(c1ccc(Cl)c(Cl)c1)O)C C1(NC(c2c(C)cccc2)=O)COC2(C1)CN(C(=O)C1=CC3CCCC13)C2 C1(OC)CCN(C2CC2)CC1.C12(NC(=O)C=CC3CCC3)CN(C1)C(=O)CC2 C1(CC(=O)NCc2cc(-c3ccccc3)n[nH]2)CCN(CC=C2CCOCC2)C1 C1(NC(C=CC(C(CN(CC)CC)C)=O)=O)(NCCc2ccco2)CCC1 C(CCCCCNC(=O)CCc1nc(C)no1)NC(c1cnc(OCC)s1)=O c1(C2N(C(C(=O)NCC)C3(CC)CC3)CCOC2)cc(O)ncc1Br c1(CN(C(C(c2nc(C(C)C)sc2)N2CCCC2)=O)C2CC2)ccc(Br)cc1 c1(C(N2C3CN(C(c4ccnc5ncnn45)=O)CC2C3)=O)ncn2cccnc12 c12nn(C)c(c1Cl)NC2=O.c1(CN2C3C(CC)C(C3)C2)cc(Cl)ccc1OC N1(C(c2c(OC)nc(C)cc2)=O)CC2CCC1CC2NC(C1COCC(C)O1)=O CC1CC(NC(=O)CSCC(c2ccccc2)=O)CN1C(C1CC2(CC2)C1)=O c1(SC)ccc(C(=O)NCC2CC(NC(=O)Cn3nnnc3C(C)C)C2)o1 N=c1nc(C(N2CC(c3cn(CC(=O)Nc4ccc(Cl)cc4)nn3)C2)=O)cc[nH]1 S(=O)(=O)(c1ccc(N2CCC(c3ccc(C)cc3)C2)c(Cl)c1)NCC=C=C C1(c2nnnn2CCOC)(Nc2ccc(SC3(CC)CC3)cc2)CCCC(C)C1 C1(NC(c2ccc(C)c(C)n2)=O)CCC2CN(c3cc4nnnn4cn3)CC2C1 n1(CC)cnc2nc(=NCCSC)[nH]c(NC(CC3CCCCC3)CO)c12 CCCCC(=O)NC(C)(C)CN(C(=O)Cc1cnn(CC)c1)C N1(C(Cc2ncc(C)o2)=O)CCC(O)C(NC(C23CC(C)C2C3)=O)C1 Cc1ccc2[nH]c(C)c(CCNCCCOC(C)C)c2c1 c1(C(=O)NC(C(=O)OC)CC2CCOC2)ccnc2cc(Br)ccc12 N1(C(CCc2n(C)ncc2)=O)CC2(C)CN(C(=O)CC3(O)CCC3)CC2(C)C1 C1(C(N(CC)CC2CCS(=O)(=O)C2)=O)CN(C(c2oncc2C)=O)CCC1(F)F C(=O)(CCC(F)(F)C(F)F)N1CC(CC(C)NC(c2ccc(C)c(C)c2O)=O)C1 c1(CC(N2C3CC(NC(CC4CCN(C)C4=O)=O)(C3)C2)=O)cccc(C#N)c1 CCC(CC)C(C)C(=O)NCCCN(C(=O)CN(C1CCS(=O)(=O)C1)C)CC N1(C(C(=O)NCc2nn(CC)c(NC)c2)=O)CCCC12CCOCC2 C#Cc1cccc(CNC(=O)CN(C(=O)COC(C2CC3CCCC3C2)=O)C)c1 N1(C(C2(Br)CC2)=O)CCC(N2CCCC2c2cc(F)c(F)c(F)c2)C2(CC2)C1 c1(OCC)ccc(NC(=O)C(C)=C(C)C)cc1C.C1(=O)C=CC(C)N1 c1(CNC(CCCCC(=O)NC)=O)n[nH]c2c1CN(C(=O)C(C)C(F)(F)F)CC2 N1(C(c2c[nH]c(=N)s2)=O)CC2OCC(NC(c3ccc(O)nc3)=O)C2C1 C1(C(=O)NCC(CNC(C2N(C(CCC)=O)CCC2)=O)O)(CC)CCCCC1 C1(NC(C(C)=C(CC)C)=O)(COC)CCCN(C(c2cc(C)c[nH]2)=O)C1 O=C1COCC2(CNC(c3ccc(Cl)s3)c3nnnn3C3CC3)OCCN12 Cc1cncc([N+](=O)[O-])c1NC(C1CC1Cc1ccc(F)cc1)=O C1(NC(CCc2onc(C(C)(C)C)n2)=O)CN(C(=O)C=CBr)C2CC12 c1(C(N2CC(OC)C(OC)C2)=O)cc(C(N(C(=O)OC)C)C)cc(Cl)c1 Cc1c[nH]c(C(=O)N(C)CCOCCNC(=O)C(C)n2cnnn2)cc1=O N1(C(CC2CC(F)(F)C2)=O)CC2CCC1C1CN(C(C3(C=C)CCC3)=O)CC21 CC1CN(C(=O)C=CCN(C)C)CC(CCNC(=O)C(C)(C)N2CCCC2)O1 c1(C(N2CCC(N(C(C(C)OCC#C)=O)CC3CC3)C2)=O)c(F)ccc(Cl)c1F C(N=c1[nH]cnc2c1COC2)C1N(C(C2C(C)CC(=O)N2)=O)CCCC1 C=CC(C)(C)CC(=O)NC1(C)CCN(C(C2(CC=C)COC2)=O)C1 C(=O)(CCc1csnn1)NC.C(=O)(C(CCNCCO)C1CC1)CCC c1(NC)cc(C)[nH]c(=NCC(CNC(c2[nH]c(C)nc2C)=O)C(F)(F)F)n1 c1(C(=O)NC2C=CCN(C(c3cnc(C(C)=O)s3)=O)C2)c(F)cc(F)cc1F C#CCC(CC(=O)OCC)Nc1nocc1C(N1CC(F)(C#N)C1)=O C1(NC(COC2C(CC)CCCC2)=O)CC(C)CN(C(c2[nH]cc(C)c2C)=O)C1 c1(OC(c2ccccc2)CNC(c2ccc(OC)cc2)=O)cnn2cccnc12 c1(OCCC(N2CC(NC(c3c[nH]cc3Br)=O)C(F)C2)=O)ccc(F)cc1F C1(CNC(CN(CCC)C)=O)CN(C(c2sc(CCC)nc2C)=O)CCC1C Cc1nnc(O)c(C(=O)NC2CC(CNC(=O)CCC3(C)N=N3)C2)c1C c1(C(=O)NCCC2CCCN(C(c3coc(Br)c3)=O)C2)cc2cnccc2[nH]1 O=C(N=c1ccc(-n2cncn2)n[nH]1)c1csc(-c2cc(Br)cs2)n1 C=CC(C)(O)CC(=O)NC(C)(CC)CCNC(=O)C(C)=CC1CC1 N1(C(C(C)C(C)(F)F)=O)CC(C)(C)CCC1CNC(c1ccc(C(F)(F)F)[nH]1)=O c1(OC)ccccc1C(=O)NCC(C)(C)CCNC(c1snc(Cl)c1Cl)=O N1(C(c2c(N)nc(Cl)cc2)=O)CCC(C2CCCN(C(C3(F)CCCC3)=O)C2)C1 C1(NC(c2ccco2)=O)CCC(F)(CNC(C2(C3CCCO3)CCCC2)=O)C1 C(C(=O)NC(C)CC=CCSCC)(C(C)(C)C)NC(C(C)SCCC=C)=O Cc1nn(CC(N2CC(CNC(=O)Cc3cnc(C4CC4)[nH]3)C2)=O)cc1Br N1(C2CCCN(CC3C(C)(C)CCC3)C2)CC(O)C(C)(C)C1 Cc1cccnc1CCC(N1CCOC(CNC(=O)C=CC2CCCO2)C1)=O c1(OC2CCN(C(CC=C)=O)C2)ccc(CNC(C2(C)CS(=O)(=O)C2)=O)cc1 C1(C(CO)NC(C2N(C)CCC2)=O)CCN(C(=O)C(O)c2ccco2)CC1 C1(C(=O)NCC2(O)CCOC2)CCC2CCC1N2C(c1cc2ccccn2n1)=O N1(CC2CCN(CC(c3ccccc3OC)OC)CC2)CC(C)(C)OC1=O N1(C(C2C(C)(C)OC(=O)C2)=O)CCN(C(C23CC(CN2C2CC2)C3)=O)CC(C)(F)C1 Cc1cc(C(=O)NCC#CC(N2CCN(C(C)C)C(C)C2)=O)nc(C)n1 Cc1nc(Br)oc1C(=O)NCC1CN(C(=O)C(c2ccccc2)C)CC1C Cc1cc(NC(=O)C(=O)Nc2ccccc2-c2ccco2)cc(F)c1 O=C(CCCn1ccnn1)N1CC(CCCCOCCSC23CCCC2C3)C1 N1(C(c2c(C)coc2C)=O)CC(C2CCCCN(C(C3(C)CCC(=O)O3)=O)C2)C1 Cc1nc(CNC(C)(CCCO)c2ccccc2)sc1C(c1ccccc1)=O Cc1c[nH]c2ncc(C(N3CC(N(CCO)C(C4CC4(C)Br)=O)C3)=O)cc12 N1(C(COCC(C)C)=O)CCC(NC(c2ccn3ncccc23)=O)C(F)(F)CC1 N1(C(C2(N(C)C)CC2)=O)CCC2CCN(C(=O)C(C(C)(C)C)c3cc[nH]n3)CC12 N1(C(c2c(C)cncc2C)=O)C2CCC1CN(C(=O)Cc1ccc(F)cn1)C2 C(=O)(N=c1ccn(CCCCO)[nH]1)Nc1ccc(C)cc1-n1ccnc1C C(=O)(C(CNC(=O)C(C1CCCCC1)F)CC1CC1)NC(CC)COC c1(C(=O)NC2CC(NC(C3(CC)CCOC3)=O)C2)cc(C(C)C)cc(F)c1 N1(C(C=CC(CC)=CC)=O)CC2(C1)CN(C(=O)C(CC(C)C)NC(=O)OC)C2 c1(C(=O)NCC2CN3CCC2C3)cnc(S)n1-c1ccccc1 C1(NC(c2c(C)nn(-c3ccc(Cl)cc3)c2)=O)CCc2c[nH]nc2C1 Cc1cc(Br)cc(C(N2CC(CNC(=O)C(C)(C)C)C3CC23)=O)c1N C(=O)(CCC(C)(C)C#N)NCC1C(NC(c2c(C)cnnc2O)=O)CC1 C1(OC)CN(C(C2CC(=O)CC(=O)C2)=O)CCC1NC(=O)COC1CC1 CCC(C)C(C(=O)N1CCOC(C(N2CCC(C)(OCCC)C2)=O)CC1)N(C)C C1(C(=O)NC(CC(C)NC(C2(COC)CC2)=O)C)CCC2(CC1)CC(O)C2 N1(C(c2cn(C)c(=O)cc2)=O)CCC(C2(NC(=O)Cc3cncnc3)CC2)C1 C1(C)(CCOC)CN(N2C(C)CC(O)C2)CCO1.C1(CC=O)CCCC2CC12 c1(C2(NC(c3c(C(C)C)noc3)c3nnnn3C3CC3)CC2)ccc(Cl)cc1 c1(SC)ccc(C)c(C(=O)NC(C)(C)CNC(=O)Cn2cncn2)c1 c1(OC)ccc(C(O)C(=O)NC2CCCC2NC(C23CC(C)C2C3)=O)cc1 c1(SC)cc(C)c(C(N2CCC(N(C(=O)CSCCC#N)C)C2)=O)s1 CC1OCCC1C(=O)NCC1CC1CNC(c1nc(-c2ccccc2)cs1)=O C(CCCS(=O)(=O)CCCCCO)N(C1(CC)CC1CCO)C c1(OC)c(F)cc(C(N2CC(O)CC2C(=O)Nc2nnc(C3CC3)o2)=O)cc1F C(CC(C(C)(C)C)NC(C1(C(C)NC(=O)COCC2CCCO2)CC1)=O)N(C)C CN1CCOCC1CC(=O)NC1(CNC(=O)CCCC#N)CC1 C1(NC(=O)C=CCOC2CC2)COCC1NC(=O)C(=O)NC1CCNC1 c1(CC)cc(OC)ccc1C(=O)NCCCN(C)C(c1csc(C(C)C)n1)=O N1(C(C(CN(C(c2c(NCC)cccc2)=O)C)C)=O)CCC(C)(N(C)C)CC1 Cc1nc(NC(=O)CC2CN(C(=O)NCCN3CCCC3C)C2)c(Cl)cc1C#N CCCC(C(O)C(=O)NCc1cnc(Cl)c(C)c1)NC(=O)CC(C)(C)C(F)F CC1CC(CNC(=O)CN2CCCCCC2)CN1C(=O)COC(C)(C)C c1(NC(C2CN(C(C3(Br)CC3)=O)CCC2O)=O)cccc(F)c1F C1(C(=O)NCc2c(C(N(C)Cc3c(CC)noc3)=O)scc2)CCCC(=O)C1 N1(C(C2CCCC2NC(C2CCC(F)(F)C2)=O)=O)CCCN(CCO)CC1 Cc1c(C(=O)NC2C3CCN(C(c4ncc[nH]c4=O)=O)C23)ccn1CCO C1(C)(CNC(c2n(CC)nc(C(C)C)c2)=O)CN(C(=O)CSCC#N)CCO1 N1(C(c2ccc(NC)nc2)=O)CCC2CCCC12C(=O)NC1(C2CCC2)CC1 C1(C(N2CC(C(C)NC(c3nonc3N)=O)OCC2)=O)CN2CCCN1CC2 c1(C(N2C(CNC(C(C)CC3CCC3)=O)CCC2)=O)ccn2ccnc2n1 C1(NC(=O)C2=CCSC2)CC(F)(F)CC1NC(c1csc(Br)n1)=O N1(C(c2c(C)ncnc2C)=O)CCCC2CN(C(C3(F)CCOC3)=O)CC12 c1(C(N(CC(C)NC(=O)CCC2CCCCO2)C)=O)cnc(C(F)(F)F)nc1 N1(C(CC(=O)NCC)=O)CC(NC(=O)C(CCOC)OC)CC2(CC2)C1.N(CC)CC N1(C(C2C(C(=O)O)C2(F)F)=O)CCCC(n2cc(-c3cscn3)nn2)CC1 Cc1cnn(C)c1C(N1CC2CC1C2C(=O)NOCC(C)(C)O)=O C(=O)(C(C)(CO)NC(=O)C(C)O)NCc1cc(C(=O)OC)n[nH]1 C(CC(=O)N1CCN(CC(C)C)CC1)(C(F)F)NC(C(CC)COC)=O c1(N(C)Cc2cc(NC(C)=O)ncc2)nc2cc[nH]c2c(=NCCC(F)F)[nH]1 C#CC1(NC(C2CC(NC(=O)C3=CCCC3)CCO2)=O)CC2CCCC12 N1(C(C(C(=O)OCC)F)=O)CCCC12CCC(NC(c1c[nH]cc1CC)=O)CC2 C1(NC(C2CCC(CNC(C(C(C)C)SC)=O)CC2)=O)CCCCC1C#N C1(CNC(CP(C)(C)=O)=O)CN(C(=O)C=Cc2ccccc2)CC1(F)F CCC(C)C(C(=O)N1CC(CCNC(=O)C(C)(C)CCF)C1)c1ccccc1 N=c1nc(N2CCC(C3N(Oc4ccncc4)CC3(F)F)CC2)cc(N)[nH]1 c1(C(=O)NC(C(C)C)C(C)NC(C2(C)C(C)(C)C2(C)C)=O)cccc2occc12 C1(C)(C(=O)NCC=C)CCCN(c2ccc(CC(=O)O)cn2)C1 c1(OCC(C)C)ccc(C(=O)NC(CNC(C2CCOC(=O)N2)=O)C(C)C)cc1 c1(C(=O)NCCC(=O)NC2C(C)CN(C(C3CCC3)=O)C2)ccc([N+](=O)[O-])cc1 N1(C(c2nc(C)sc2C)=O)CCC2CN(C(=O)CCC3CCCOC3)CCC12 CC(C)C(C(=O)N1CCOC(CNC(C2C=CCC2)=O)C1)C(C)C c1(CN(CCNC(c2c(NC(C)=O)cncc2)=O)C)ccccc1C#N C12(CNC(C3C(=O)NCC3)=O)CCCC1CN(C(=O)Cc1c(F)cccc1F)C2 CN1CC2CCC1C(NC(C1(NC(C3C=CCC3)=O)CC1(C)C)=O)C2 N1(C(C2(C)CC2)=O)CCC2(CCC2CNC(=O)CON=C2CCCCCC2)CC1 Cc1nc(C(N2CC(C(O)C(=O)NC3CCCSCC3)C2)=O)c(C)o1 c1(C(N2CC(CC)(CO)C2)=O)ccc2c(n1)CN(C(c1n[nH]c(O)n1)=O)CC2 c1(CN(CC(C)(C)CN)CC)ccc(C(C)C)c(C)c1 C(C(N=[N+]=[N-])C(=O)N1CC2CC1(C(=O)NCc1nccs1)C2)OCC N1(C(CCC(=C)C)=O)CC(NC(c2cnccc2C(F)F)=O)CC1(C)C N1(C(C(C(=O)OCC)(C)C)=O)CC2(NC(C3CCCS(=O)(=O)C3)=O)CCC1CC2 c1(C(=O)Nc2ccc(NC(c3c(C)cc(C)s3)=O)nc2)cccc(C#N)n1 n1(CCNC(=O)C(F)=CC2CC2)ccc(C(=O)NC(c2cccnc2)CO)c1 c1(C(N2CCN(CC)CC2)=O)n[nH]c2cc(C(=O)NCCCCCC)ccc12 c1(C(N2CCC(F)(CNC(c3c(C)ocn3)=O)C2)=O)ncnc(O)c1Br c1(C(=O)NC2CCN(C(C=CC)=O)CC2CO)cnc2cc(C)nn2c1C c1(C(N2CC3C(C(=O)NC4C(C(C)C)C4)C3C2)=O)cc2ncccc2[nH]1 Cc1ncc(C)c(=NCC2CN(C(C3CCN(C)CC3)=O)CCC2C)[nH]1 c1(C(N2CCC(NC(c3c(C)onc3C3CC3)=O)C2)=O)c[nH]cc(Br)c1=N C1(C(=O)NCC2CC(CNC(CCC(C)OCC)=O)C2)CC2CC(=O)C1O2 C1(C(=O)NC(CC)CSC)CCCCCCN1C(=O)CC1(OCC)CCC1 c1(C(N(C)CC2C(NC(CC(CN(C)C)O)=O)CCC2)=O)cc(F)cc(Cl)c1N N1(CC#N)CCOCC(C(=O)NC2CC3OCCC23)C1 Cc1cc(C(N2CC(C3CN(C(C4CC5COCC5C4)=O)C3)C2)=O)c(N)c(C)c1 c1(C(N2CCC3C(C2)CN3C(C2CCC3(CC2)CC3)=O)=O)cccc2c1COC2 c1(C(=O)NCC(C)(C2CC2)NC(C(CN(C)C)N(C)C)=O)cccc(CC#N)c1 C1(NC(C(c2ccc(F)cc2)C)=O)CCN(C(C2CCCC(F)(F)C2)=O)CC1O CCCC(C)C(C)NC(c1c(CNC(=O)CSCC(N)=O)nnn1C)=O c1(-n2cc(C(C)NCCc3ccccc3C(=O)O)nn2)cncc(CO)n1 n1(C(CC)C)nnnc1C(c1cncn1C(C)C)Nc1cnn(CC(C)C)c1 C1(CNC(CN2C(C)CC2)=O)CC(F)CN1C(=O)CSC1CCS(=O)(=O)C1 C#Cc1ccc(C(=O)NC2(C(=O)NCC3CN(C4CC4)C3)CC2C)nc1 C1(C(CNC(C(F)=CC)=O)O)CCN(C(=O)CSC)CC1.C12(CCSC1)OC2 N1(C(C(Cc2ccc(N)cc2)OC)=O)CCC2(C)C(C1)C2(Cl)Cl N1(C(c2c(C)ccc(=N)[nH]2)=O)CCC2(C1)CN(C(=O)CCC(C)(C)C)C2 N1(C(COCC(C)C)=O)CCC2CN(C(C3CCCC3(C)C)=O)CC2C1 c1(C(=O)NC(C(C)NC(C2CCC(C)CC2)=O)CO)ccc2cc[nH]c2c1F C1(CNC(C(CCC)NC(C)=O)=O)CN(C(=O)CSC(F)F)CCCO1 N1(C(C2C3(CC(C)OC2)CC3)=O)C2CCC1CC(CN1CCC(O)C(F)CC1)C2 c1(C(N2C(C(N3CC(S(C)(=N)=O)C3)=O)CC2)=O)nccc2cc[nH]c12 C(C(=O)NCC1(NC(=O)COC(C)(C)CC)CC1)(C(C)(C)C)N(c1ccsc1)C C1(NC(C(c2ccc(C)cc2)C)=O)CC2CN(C(=O)CCC(N)=O)CCN2C1=O c1(C(=O)OC)cc(C2CCCN(C(=O)CCc3csc(=N)[nH]3)C2)cc(F)c1 C(=O)(C(=O)N=c1ccn(CC)[nH]1)N1CCC(CCN(CC(C)C)CC)C1 C=CC1CCN1C(=O)CC(C)N(C(=O)CSCC(N)=O)C CC(C1OCCc2sccc21)N(C)CCC1C(C)(C)C1(C)C Cc1cccc(C(=O)NC2CC(NCc3ccc(OC(F)F)nc3)C2)n1 c1(SC)nc(N2CC3CN(C(C4CCN(C)CC4)=O)C3C2)c2ccccc2n1 C12(C(=O)NC3(CNC(CC4CCC(C)(C)C4)=O)CC3)CCCN(CC1)C2 N1(C(c2n(C)nc(CC)c2Cl)=O)CCC12CCN(C(=O)C(C)COC)CC2 CCC(C(=O)NC(C)(C)CCNC(=O)Cc1ccsc1Br)N(C)C N1(C(Cc2ccc(C)c(C)c2)=O)CC(NC(C2(C)CC2(F)F)=O)CC12CCC2 C=CCC(C(=O)NCC1(C(=O)NCC2(C3CC3)CCCO2)CCCO1)OC N(C(=NCCC(C)=O)NCC1(CCO)CCCO1)CC1(OCC)CCOC1 C12(NC(CCC=C)=O)CCCC1(F)CN(C(=O)CCc1cnn(C)c1)C2 Cc1cc(C(=O)NC(C)CCNC(c2cnns2)=O)c2c(c1)CCO2 c1(C(=O)NCC2C(NC(c3ccc(CC)cn3)=O)C2)cccc(Br)c1O N1(C(c2cc(OC)ncn2)=O)CCCCC(CNC(c2cnco2)=O)C1 CC1OC2CCC1(C(=O)NCC1CC1C(N1CCCSCC1C)=O)C2 n1(CC(=O)NCC(C)NC(c2cnn(C)c2Br)=O)cc(C#N)c(O)nc1=O C1(NC(c2cnn(CCC)c2C)=O)CN(C(=O)CC2CCC(=O)NC2)CC12CC2 Cc1csc(C=CC(=O)NC2CC(NC(c3ccc(Br)cc3)=O)C2)n1 c1(C(=O)NCCN(C(C(C)SC)=O)C2CC2)ccc(-n2ccnc2)cn1 c1(C(N2CCN(C(CCCOC)=O)CC2C)=O)cc2occc2n1C c1(C(=O)NCCN(C(=O)C(O)c2ccco2)C)cccnc1N.C1(OC(=O)O)CC(N)C1 N1(C(CN)=O)CC(C2CCN(C(=O)CC(Cl)Cl)CC2)C1 N1(C(=O)C(c2ccc(C(F)(F)F)c(Cl)c2)=O)CCN2CCc3ccccc3C2C1 C(=O)(C1=CC2(CCOC2)C1)N(CCCN(C(=O)C(C)(C)N1CCOCC1)C)C C(C(=O)NOCC1CCOC1)=CCNC(C1C(C)C1)=O C(=O)(C1(C(=O)NC2CN(C(C3CCC34CCC4)=O)C2)Cc2ccccc21)OCC C(=O)(CCC(=O)N(C)C)NCCN1CC=C(C)CC1.C1C(=O)N1CCOC c1(-c2ncc(CNC(C(CC)C)c3nnnn3CC(F)F)s2)ccccc1C c1(C(=O)NC(CNC(c2c(CC)ccs2)=O)CC)nc(O)nc(O)c1F C=C=CCCC(=O)NCCCOCCOCCNC(c1ccnn1CC(F)F)=O N1(C(c2ccc(COC(C)=O)cc2)=O)CC2CC1CN2C(=O)CCF c1(C(c2n(CCCF)nnn2)NCc2conc2C2CC2)cc(Cl)ccc1F c1(N(C2COCCN(C(=O)C(C)(C)Cn3cccn3)C2)CC)cc(CO)cc(C)c1 c1(C(N2C(CC)CN(C(C3(O)CC3)=O)CCC2)=O)cc2ccccc2nc1C C1(NC(C=CCC)=O)CCCC(NC(c2cc(O)ccc2OCCCC)=O)CC1 c1(C(C(=O)NC(CN(C(=O)CC(C)C2CC2)CC)C)(C)C)ccccc1C C1(C2(O)CN(C(=O)CN3CCN(SC(F)F)CC3)C2)(CNC(=O)CC2CC2)CC1 N1(C(C2C(c3n(C)ccn3)C2)=O)CCCCC(NC(C2C=CCCC2)=O)C1 N1(C(CN(C(=O)OCC)C)=O)CCCC2(CNC(C3OCCC3C)=O)CCCC12 S(=O)(=O)(CCC(=O)N1CC(F)(F)CC1CNC(=O)CCC1CCC(C)O1)NC CCCCC(O)C(C)C(=O)NCC(C)CN(C)C(c1cccnc1OCCO)=O c1(C(N(CC(CNC(C23C(C)OC(CO)(C2)C3)=O)O)C)=O)ccc2nn[nH]c2c1 Cc1ccn(C)c1C(=O)N(CCCCN(C(=O)C(C)Cc1ccccc1)C)C N1(CCC(=O)NCC(CC)NC(c2cnn(CC)c2)=O)CCCCC1C c1(N2CC(C)C(NC(c3cn(C4CCC4)nn3)=O)CC2)ncc(Br)cc1[N+](=O)[O-] C#CCCCCCCC(=O)NC1CC(O)CN(C(c2ccoc2C(C)C)=O)C1 N(C1CCCc2cn(C(C)CC)nc21)C(=O)NC1CCC(C(CC)(C)C)CC1 N1(C(C(C)N2CCC2)=O)CC(NC(=O)CCc2cscn2)CC12CCC2 CC1(C)CN(C(C2COCCO2)=O)CC(CNC(c2ccc(F)c(C#N)c2)=O)O1 N1(C(c2ccc(C)nc2C)=O)CCC2(CC1)CC(NC(C1CCC1(F)F)=O)CO2 c1(C(=O)NCC2(F)CCN(C(C(C)(C)C(N)=O)=O)C2)cc2cccnn2c1 C=CC(C)(C)CC(=O)NCCC1CCCN(C(=O)Cc2c(C)nn(C)c2Cl)C1 C12(C(=O)NCC3C(C(N(C4CCN(C)C4)CC)=O)CCO3)CC1CNC2=O c1(CC(=O)NCC(C)N(C)C(c2ccc(C(F)F)s2)=O)cccc2cnccc12 c1(COC(C)C(=O)OCCCCc2ccccc2)nc2ccc(O)cc2s1 c1(N2CC(NC(CC(C)(C)OC)=O)CC(C)(C)C2)cc2nnc(C)n2cn1 c1(C(=O)NCCCCC(C)NC(c2c(Cl)cnc(C)n2)=O)cc2ccsc2n1C C1(C(N2CCC(COC)(NC(c3nccnc3N)=O)C2)=O)CC(S(C)(=O)=O)C1 c1(CC)nn[nH]c1C(=O)NCCN(C(c1cncn1C)=O)C(C)C C1(CNC(=O)NC(C(=O)NC)CSC)CCCC(C)C1 CCC(CCC(=O)N(C)CCc1ccc(Cl)cc1Cl)OC CC(N=c1cccc(S(=O)(=O)NC(C)CCCO)[nH]1)c1ccccc1 O=C(CCCC(F)(F)CO)NCC(F)CNC(=O)C(c1cccnc1)O N1(C(C2CCC(CN(C)C)O2)=O)CC2CCC2(CNC(c2ccc(F)cn2)=O)C1 CC(C)(Cl)C(=O)NCC12CC(NC(c3cc(-c4csc(=N)[nH]4)c[nH]3)=O)(C1)C2 C1(NC(C2C(NC(C(CC3CCC3)OC)=O)C=CCC2)=O)CN2CCCC1C2 C1(CNC(C2N(C)C(=O)NC2)=O)(NC(c2cccc(Cl)c2)=O)CC2CCC1CC2 C1(NC(C2(CC)CC(F)(F)C2)=O)CCC(F)(F)CC1.C12CC(O)(C1)CNC2=O N1(C(C=C)=O)CC2(CCC2)CC1CNC(c1csc2nnsc12)=O N1(C(c2ccc(C=C)cc2)=O)CCC(C(=O)N2CCCCC(C)(F)C2)=C(F)C1 N1(C(CCC=CCC=C)=O)CC(C)(C)CC1C(=O)N(C)Cc1ccon1 C1(C(=O)NC2CC(CCNC(C(C)N(C)C)=O)C2)CCN(C2CC2)C1=O C1(C(=O)NCC(=O)NC)CC2(CC2)CN1Cc1cc(O)cc(F)c1 CS(=O)(=O)C1CCN(c2cc(NCCOCCC3CCCO3)nc(C(F)F)n2)C1 CC1CN(C(c2nnc(S)n2C)=O)CCC1NC(c1coc2c1COC2)=O C1(CC(=O)NC2(CCC)CCC2)CCN(C(CC)C(=O)O)C1 c1(C(N2C(C)CC(NC(C=CSC)=O)C2)=O)cncc2c1CCC2 c1(C(C)NCCNC(C(C)OCCOCC)=O)cn(CC(N)=O)nn1 C1(CNCC(CN(C(C)C)C)O)CCCC(C(F)F)CC1 O=CN1CCCC1C(=O)NCC1COCC1NC(c1ccccn1)=O N1(C(c2c(C)[nH]c(=N)s2)=O)CCC2(CO)CN(C(c3ccccc3Cl)=O)CC2C1 c1(C(N2CCCC2C2CCN(C(c3cncnc3)=O)CC2)=O)cccc(Cl)c1 N1(C(CCC=C)=O)CCN(C(=O)CN(C(=O)C(C)C)C)CC1c1cnn(C)c1 N1(C(c2cc(C)n(C)n2)=O)CCC(C(=O)NCC(O)C(C)O)C12CC2 C1(NC(=O)CC2CCCC2(F)F)(CO)CCCN(C(=O)CCCC2CCCC2)C1 CC(O)C(C(=O)NC1CC1)NC(c1cscn1)=O.C1(CCO)(CNC(=O)CS)CC1 c12cccc(c1)C(=O)OC(=O)C2.CC(C(C)NC(C1CCCS1)=O)C(=O)O c1(C(=O)OCC)cc(S(=O)(=O)NC2(NC(=O)OC(C)(C)C)CCC2)ccc1OC c1(CC)cc(NC(C2CC2CF)=O)ccc1C.C12CCCN1C(=O)CNC2 N1(c2ccc(NC(C3CCO3)C)cn2)CCC(CNC(=O)OC(C)(C)C)S1(=O)=O c1(-c2cn(CCCOCC(=O)NC(CC)(C)C)nn2)cc(C)nn1C CC(CC(N)=O)C(=O)NCC=CCNC(c1ccnc(C(F)(F)F)c1F)=O CC(CC1CC1)C(=O)NC1CCC1CNC(c1cnc(O)o1)=O N1(C(C(CC)NC(N)=O)=O)CCCCC(NC(=O)COC)C1 c1(CC(=O)NCC(C(=O)N2CC(CC)(CC)C2)CC(C)C)c[nH]c2cnccc12 C1(C(=O)NCC(=C)Cl)CN(C(=O)C(CC)OCC)CC1C n1(CC(=O)NC(C2CCN(C(COC(CC)C)=O)C2)C)nc(C)cc1C(F)F Cc1ccc(C(=O)N(C(C)CC(=O)NC2CC(=O)NC2=O)C)cc1F Cn1cc([N+](=O)[O-])cc1C(N1CCC(CCNC(=O)C(F)OC(F)(F)F)CC1)=O N1(C(c2c(C)ccs2)=O)CCOCCC1C(=O)NCC1(O)CCC(C)C1 c1(CCC(=O)NCC2COCC2NC(C2CC23CCC3)=O)cccc(Br)c1 Cc1ccc(C(=O)NCC(O)CNC(C2CC(C3CC3)=NO2)=O)c2c1CCC2 c1(NC(N(C2CC2)CC)=O)cc2c(cn1)C(=O)N2.c1(OCC)[nH]ccc1C(C)C C=C(C)CCCC(=O)NC1CN(C(c2cccc(OC(C)C)c2F)=O)C2CC12 C=Cc1ccc(C(=O)N(c2cc(Br)ccn2)C2CCC2)cc1 CC(C)C(C(C)C)NC(=O)C(C1CC1)NC(=O)CN1CSCC1=O c1(NC(=O)Cn2cc(C3(OC(=N)O)COC3)nn2)nncc2ccccc12 CCCC(C(=O)NCC12CC1CN(C(=O)COCC=Cc1ccccc1)C2)C(C)C C(C)(N=c1[nH]c2ccc(F)cc2o1)C1CCN(C(c2ccc(OC)nn2)=O)CC1 c1(C(=O)NC2C(NC(=O)CCCCc3cnn[nH]3)C2)cc(F)ccc1F c1(NCC(C2CC2)NC(C2CC(CF)C2)=O)ncc2c(Br)cccc2n1 C12CC(C)(C1)NC2=O.c1(C(CNC(C2CCOCC2)CC)=O)cnn(C)c1 c1(-c2cn(CC(CCNC(C(C)(C)O)=O)F)nn2)cccc(-c2ccco2)c1 C(CN=c1[nH]c(=NCCOCCO)[nH]c2cc[nH]c12)N1C(C)COCC1 C(=O)(CCCC(=O)N1CC(C)CCC1C(=O)NCc1ccc(F)cc1F)OCC N1(C(=O)COCC2CCCCC2)CCN(C(c2cccc(F)c2O)=O)C2(CC2)C1 N1(C(CC(=O)OCC)=O)CC2(CC(CNC(c3cncc(C)c3)=O)C2)C1 C12(NC(=O)CC3(C(F)(F)F)CC3)CCCC1N(C(c1ccnc(Cl)c1F)=O)CC2 c1(OC)ccc(O)c(C(N2CCN(C(=O)Cc3cnc(C)s3)CC2CC#N)=O)c1 C(=O)(C1CCCc2nn[nH]c21)NCCC1S(=O)(=O)CCN(C(C(C)(C)OC)=O)C1 C1(CNC(C2(SC)CC2)=O)CCCN(C(=O)Cc2cc(CC(C)C)on2)CC1 Cc1ccc2c(n1)C(C(N1CC(c3cn(CC(N)=O)nn3)CC(C)(C)C1)=O)C2=O N1(C(CC(CC)C)=O)CCC2CCN(C(=O)C(O)Cc3ccccc3)CC2C1 C1(OC)CN(C(C2CC(F)C2)=O)C(C)(CNC(=O)CCc2cnc[nH]2)C1 S(=O)(=O)(c1cccc2cccnc12)N1C(C(=O)NCC2COCCO2)CCC1 C1(CNC(c2cc(C)[nH]n2)=O)COCC2(CCN(C(=O)CN3CCCCC3)C2)O1 C1(CC)CN(C(=O)CSCCNC(c2ccn(C3CC3)n2)=O)CCS1 C(=O)(C1=CC(C)(C)C1)N1CC(CNC(c2ccc(C(C)C)cc2)=O)C2C1C2 C(C(CC(F)(F)F)NC(=O)C(N1CCCC(C)C1)=O)NC(c1c(C)csc1Cl)=O Cc1cnc2ccc(C(=O)N(C3CC(NC(=O)CC4=NNC(=O)C4)C3)C)cn12 c1(C(c2n(C(CC)(C)C)nnn2)NCC(C)Cn2cccn2)cncc(C)n1 Cc1ccc(F)cc1C(=O)NC1CCCC1CNC(C1CCC(N=[N+]=[N-])C1)=O c1(CN2CCCC(C(=O)NC3CC(O)(Cc4cnccn4)C3)C2)cnc(O)nc1O N1(C(C(CC=CC)C)=O)CC(C(N2CCCC2CNC(N)=O)=O)C(F)(F)C1 C=Cc1ccc(C(=O)NCC2CCC(NC(=O)CC(C)C3CC3)CC2)cc1 Cc1ccc2sc(=NC(C)C3CN(C(=O)CCC4CC4(F)F)CCO3)[nH]c2c1 c1(C(=O)NCC2(O)CN(C(CCC)=O)C2)ncc(Br)cc1F c1(C(=O)NCCN(C(=O)C(C)SC(F)(F)F)CCOC)cc(N)cc(O)c1C C(=O)(C(CC(C)C)n1nnnc1C(C)(C)N)NC1(CF)COC1.c1(OC)ccc(Cl)cc1 N1(C(c2c(C)cc(C)cc2Br)=O)CCN(C(=O)CC(C)(C)C)C(C)CC1C C1(NC(=O)COC2CN(C(C3CN4CCC3C4)=O)C2)CCC2CC1CO2 C(CCC(=O)NCCOCCNC(=O)Cn1ncnn1)NC(=O)CC1CC1 C(=O)(CCCCCC(=O)OC(C)(C)C)N(C(CCC#CC)=O)C(C)(C)C c1(C(=O)NCC(=O)NCCCn2cccn2)cc(CO)on1 C(=O)(C(C)(F)C(C)(C)F)NCC1(CN=c2snc(C(=O)OC)[nH]2)CC1 C12(C(=O)NC(C)(C)COC3CCCCC3)CC(CO)(CCO1)C2 CC(C)CC(CNC(C1CC2CC2C1)=O)NC(=O)COC(CC(C)(C)C)=O N(C(=NCCCF)NC1CCc2sc(Cl)cc21)Cc1c(C)ccs1 N1(C(C2CCC(CCC)CC2)=O)CCC(CNC(C2CC(F)(CO)C2)=O)CC1C c1(-c2c(CNC(c3ccc(N4CCCCCC4)nc3)=O)c[nH]n2)cccc(Cl)c1 O=S(=O)(c1ccc(Br)cc1N1CCC(F)(F)CC1)N1CC2CC2C1 N1(C(C(C)NC(N)=O)=O)CCC(CNC(=O)CCc2nc(CO)no2)C1(C)C C(=O)(C1=CCCCN(C(=O)OC)CC1)N(CC(C)NC(CCS(=O)(=O)NC)=O)C c1(CC(=O)NCC(C)N(C(=O)Cc2ccc(CO)cc2)C)cccc(Br)c1 CC1CCN(CC(=O)NC(Cc2cc[nH]n2)C(=O)NC(c2nncs2)C)CC1 C=C(C)CC(C(=O)N1C2CCC(C2)C1CNC(c1cnccc1C)=O)OC C1(NC(C2(OC)CCCC2)=O)CCN(C(C2CCCN2C(C)=O)=O)C1C(C)C C1(CC)C(C(=O)NCC(C)(C)n2ccnc2)CCN1C(=O)CCc1ccc[nH]1 c1(NC(CNC(C2C3CCC2CC3)=O)=O)cc(Cl)ccn1.C1(F)(CN)CC(CO)C1 C1(C(=O)NCc2cn(CC)nc2)CC2(CCN(C(c3nc(C)c(Br)s3)=O)CC2)C1 N(C(=NCCc1ccc(Cl)cc1Cl)NCCNC1CC1c1cccs1)C1C(C)C1 c12ccc(cc1)NOCCCCn1nc(CCO)nc1-2.C=CC c1(C(=O)NCc2c(C)nc(C)[nH]2)c[nH]c2ccncc12.C12CC(O)CN1C2=O Cc1ccc(C(N2CCN(C(=O)Cc3c(Cl)cccc3Cl)C3CC23)=O)c(I)c1C c1(C(N2C(CNC(C3(CCCC)CC3)=O)CCCC2)=O)cc(OC)ccc1C C1(CCNC(c2ccsc2Br)=O)CCCN(C(=O)CC2CCOC2)C1 C12(C(N(CCNC(c3coc(Cl)c3)=O)CC)=O)CCCC1CC(F)(F)CC2 C1(C(N2C(CCNC(c3cnc(C4CC4)o3)=O)CSCC2)=O)C2CC3C(C2=O)C13 C1(CC#C)(C(=O)NC(C2CCN(C(C3(C#C)CC3)=O)CC2)C)CCCCO1 c1(C(N2C(C(=O)NCC(=O)N(C(C)(C)C)C)CC(=C)C2)=O)cc(F)ccc1F CC1(C)CC(NC(=O)C=CCNC(C2CC2(C)C(F)F)=O)C1 C1(C(=O)NC(C=C)C(F)(F)F)CC(C)CCN1C(=O)CCC1CC1(C)C C1(CN(C(c2ccc(CSC)o2)=O)C)CN(C(C2(C(F)(F)F)CC2)=O)CC12CC2 N1(C(C=Cc2n(CC)ccn2)=O)CC2=C(C1)CN(C(=O)CCC1CCCO1)C2 c1(C(=O)NC2(CN(C(c3c(OC)c(F)ncc3)=O)C)CC2)cc(F)c(F)cc1F C12(C(=O)NC3CCN(C(Cc4n[nH]c(=N)s4)=O)C3C3CC3)CC1Cc1c[nH]nc12 C1(C(N(CCOCCCN(C(CC(=O)N(C)C)=O)C)C)=O)CCCC2CCCN12 Cc1ccc(CC(N2CC3(CC3)CC2CNC(c2cn[nH]c2)=O)=O)cc1F C12(CNC(c3n(CC)cnn3)=O)CCCC1N(C(C1(COC)COC1)=O)CCC2 c1(N2CCN(C(C(=O)Nc3c(C)[nH]nc3Cl)=O)CC2)ccn2nccc2c1 N1(C(C2C(C)CC(C)O2)=O)CC2(C1)CN(C(c1ccc(=O)n(C)n1)=O)C2 N1(CCN)CCOCCC1=O.n1(CC(c2ccccc2)OCCC)ccnc1C CN1CCC(C)(C(=O)NCC2CC2NC(c2cncc(-n3ccnc3)n2)=O)C1 N1(CC(=O)NC(=O)C(c2ccccc2)Sc2ccccc2)CCN(CCCO)CC1=O N1(C(C2(c3ccc(C)cc3)CCCCC2)=O)CCCC(NC(C2CC2C)=O)C1C c1(C(=O)NCC(C2N(C(CCC#C)=O)CCC2)(C)C)ccc(-c2ccsc2)cc1 C1(C(N(CC(C)NC(CC2(OCC)CC2)=O)C)=O)COC(=O)N1C N1(C(CCC(=O)NCC)=O)CCCN(C(=O)C(C)(C)NC(c2ccccc2)=O)CC1 Cc1cc(F)cc(C(N2CC3CC2CN(C(=O)CCC2CC2(C)C)C3)=O)c1N C1(CNC(c2c(C(C)C)cco2)=O)CN(C(=O)C(O)CC(F)(F)F)CC(C)(C)O1 N1(c2nc(OC(C)C)c(Br)cn2)CCC2CN(c3ccnc(C)c3C#N)CC12 C1(O)(CNC(c2cnc(SC)s2)=O)CCN(C(=O)CNC(=O)CC(F)(F)F)CC1 C=C(C)CCCC(=O)NCCCCCC1CCN(C(C2(CC)COC2)=O)CC1 c1(C(N2CCN(C(c3c(Cl)cnc(CC)n3)=O)CC2)=O)noc2cc(Cl)ccc12 C1(CC(=O)Nc2cnsc2)(NC(=O)CC2CCC2)CCC1 C1(NC(c2cc(C(=O)OC)sc2)=O)CC(NC(=O)C(C)C(C)F)CC1O CC1CCN(C(=O)C(=O)C(C)(C)C)CCN1C(=O)CCOC1CCN(C)CC1 c1(NC2CCCC(NC(c3cnc(CC4CC4)s3)=O)C2)ncnc2cccnc12 O=C(CCC(=O)NCC(F)CNC(=O)CC1CC(Oc2ccccc2)C1)OC C(=O)(C1SCCc2sccc21)N(CCNC(c1ccnc2ncccc12)=O)CC CC#CC1CN(C(C2C=CCN(C(=O)C(O)COC)C2)=O)C1 C1(C(N2CCCC(C(C)C)C2)=O)CC2(CCN1C(=O)C(F)(F)F)CC2 c1(CC)c(N2CCN(C(=O)C(C)N(S(=O)(=O)CC)CC)C(C)C2)nc(C)nc1Cl C(=O)(C1CNC(=O)c2ccnn21)N1C2CN(C(C=CC(CC)=CC)=O)CC1CC2 CC1CCCN(C(=O)C(=O)NCC2CCCN2C(=O)C=Cc2ccnn2C)C1 C1(C(=O)NC(c2ccc(F)cc2)CNC(C(C)(C)OC)=O)CCSCN1C CCCCC(CC)C(=O)NCC1(CO)CCN(C(=O)C(CCO)N(C)C)CC1 C12(C(=O)NCCC(CC)(F)F)CCCC1CN(C(=O)CCn1cncn1)C2 Cc1noc(C)c1C(C)C(=O)N(C)CC1CCN(C(c2cnc(=N)[nH]c2)=O)C1 C(=O)(CCC(=O)N1CC2CC2(NC(c2csc(C(C)(C)C)c2)=O)C1)OCC c1(C(=O)NC(CC)CN(CC(C)(C)C)C)sc(N(C)C)nc1C C(=O)(CC(C)CNC(C1CCN(C(=O)CCC2CCC2)C1)=O)NC C(=O)(CC(C)CNC(=O)OC(C)(C)C)NCC1(CC)CN(C)C1 c1(C(=O)NCCN(C(=O)CCc2ccn(C)n2)CC)cc(F)cc(S(N)(=O)=O)c1 C#Cc1ccc(CC(=O)NC2CC(F)(CNC(C3(C)CCOC(C)C3)=O)C2)cc1 NC1(C(N2CCOCC2CC2CCCO2)=O)CCCCCC1 CC1(C)CCCC(C)(NC(=O)CNC(=O)CC2CCCC23CC3)C1 c1(NC(=O)NCC2CC2)nn(C)c2c1CN(C(=O)CCC(=O)NSCC(C)C)CC2 c1(C(N2CCCC(NC(C(C)(C)N(C)C)=O)CC2)=O)cccc(C#CCO)c1 N1(Cc2cccc(C)c2)CCC2C(CCCN2C(=O)Cn2ccc(C)n2)C1 CCC(C)C(=O)C(=O)N1CCC(COC)C1NC(=O)C(C)(C)CC CC1N=C2NC(=NCC(CC)C3C1CC3)Nc1ccsc12.c1ccc2c(c1)CCO2 C(=O)(CCCCCCNC(=O)C(C)(O)C1CC1)N(C)CC1CCN(C)C1 c1(CC)ncccc1C(N1CCC(NC(c2[nH]c(O)nc2C)=O)C1)=O CCCC(C(=O)N(CCCNC(C1CC(=O)N(c2cn[nH]c2)C1)=O)C)OC C1(C(=O)NC(C(CC)C)CO)CCCCC1(C)NC(c1ccc(O)cn1)=O C1(N(CC(C)C)CC(=O)NC(c2cn(-c3ccccc3)nn2)C)CCS(=O)(=O)C1 N1(C(C2=C(C)OCC2)=O)CCC12CCCN(C(c1ccn(C)n1)=O)C2 C(C(=O)NCC#CC1CC1)(C(C)(C)C)NC(C(CC)N(C)C)=O Cc1cc(N)n2ncc(C(=O)N(C)CC3(O)CCCN(C(=O)C(F)F)C3)c2n1 c1(OC)ccc(NC(=O)Nc2ccc(OC(C)C)nc2)c(F)c1.C1C(O)CN1 N#CC1CN(C(=O)CCC=Cc2cccs2)CC1NC(=O)C1=COCCC1 Cc1ccc(C)c(C=O)c1O.c1(N)cc(C)c(F)c(C)c1.N12CC3C(C1)N23 C1(NC(COCCC#C)=O)CCCCC1C(=O)NC1CC(CN(C)C)C1 C(=O)(NNc1cccc(-c2nn[nH]n2)c1)OC(C)(C)C C(=O)(CCC(=O)c1ccccc1N)N(C)CC1(NC(C(C)SC)=O)CC1 OCCCC(Cc1ccc(F)cc1)n1nnc(-c2cscn2)n1.c1ccc(Cl)cc1 C1(CNC(CN(C(C(C)C2CCCC2)=O)CC2CC2)=O)CC2OC1C1CC21 C1(NC(c2n(C)nc(Br)c2)=O)CN(C(C2CCO2)=O)Cc2nccn2C1 N1(C(CCOCC#C)=O)CC2CCC1CN2C(C1CC1(F)C(=O)OCC)=O CCCS(=O)(=O)CC(=O)NCC(C)(C)CNC(=O)CSc1nnnn1C c1(C(N(CC(C)N(C(C2C(OC)C2)=O)C)C)=O)ccnc(NC(C)=O)c1 CCC(C)C(CC(=O)NCCCOC(=N)O)NC(c1c[n+]([O-])c(C)cn1)=O CC1OC(C)CC1C(N1CC(CCCCNC(C2CC(=O)N2)=O)C1)=O c1(NC(C2(SC)CN(C(=O)CC3CC4(CC4)CO3)C2)=O)cn(C)c(=O)cc1C Cc1cc(C(N2CC(O)CC2C(=O)NCCCCCC2CC2)=O)nn1C C1(CCN(C(=O)CC(C)(C)F)C)CCCCN1C(=O)C=Cc1cc[nH]n1 N1(C(c2n(CCC)nc(C)c2)=O)CC(OC)CC(NC(=O)CCC2CC2(Cl)Cl)C1 CCC(CC)CC(=O)N1CC2(CNC(C3C(C)(C)C3(F)F)=O)CCC1C2 C(=O)(C1CCCc2ccc(C(=O)OC)cc21)NC1CC(O)CCN(C(CC)=O)C1 CCC(CC(=O)N1CC(O)(C(F)C(=O)NCCc2cccc(O)n2)C1)SC n1(CCC)nc(CSC)nc1-c1cc(Br)c(Cl)[nH]1 CC1CCC(CNC(c2ccncn2)=O)N(C(=O)CC2(C#N)CC2)C1 C1(C(N(C(CC)=O)C(C)C)=O)CCCN1NC(=O)c1ccc(C)nc1 c1(C(=O)Nc2cccc(-c3onc(C)n3)c2)ccnc2c1ccn2C c1(OC)ccc(Br)c(C(N2CCCC(CNC(=O)CCC3CC3)CC2)=O)c1 c1(SCC)nc(C)c(C(CC)C(=O)NCCNC(C2(F)CC2)=O)s1.c1(S)ccncn1 N1(N(C(CC2CCN(C(c3cc(C)ns3)=O)C2)=O)C)CC(C)OC(C)C1 c1(OC)cc(CNC2(c3ccccn3)CCCC2)c(C)cc1C CCC(CCCC(=O)NCC1(CO)CC(C)(C)C1)NC(c1coc(OCC)n1)=O CC1CN(C(C2COCCN2C)=O)CC1NC(c1cc(CO)on1)=O c1(C(=O)NC2CC(NC(C3CC4CC4C3)=O)C2)cc2cc(Br)cn2cn1 C=C(C(=O)NCC1CN(C(=O)Cc2ccc(C)nc2)CCC1(F)F)C(F)(F)F C1(CC(=O)N(C(C)COC)CC)C2CCCC2N1C(=O)C=Cc1cc[nH]c1 C1(CCNC(Cn2c(C)ncc2)=O)Cc2ccccc2CN1C(=O)C(=O)NC(C)C CC(C)CCCC(C)C(=O)NCc1nc(C(=O)NC(C)Cc2nncn2C)co1 C1(C(=O)NCc2ccc(CC(=O)NCC3ON=C(C)C3)cc2)CC(C)(C)CN1C n1(CC(=O)N(C2CCN(C(=O)C=CCOCCSC)C2)CC)ncc(Br)n1 C1(C)(C(N2CC(c3c(CNC(CC=C)=O)nco3)C2)=O)CCCCCC1 Cn1nc(C(F)(F)F)c(I)c1CNC1CC(c2ccc(Br)cc2)C1 c1(C(=O)NCC(C(=O)NC2COC(C(C)C)C2)OC)ccc(O)cn1 c1(C(C(=O)NCCCCCC)N(C2CC2)CC)nnc2n1CCC2 c1(CC(=O)NC2C(NC(CCS(C)=O)=O)C2)cccc2nsnc12 C(=O)(C1=CC2(CN(C(C3(C)CCCC3O)=O)C2)OC1)NCCOCC#C C1(CSC)(NC(c2nnnn2C(C)(C)C)c2csnn2)CCCC1 c1(NC(=O)NC(C#C)CC)oc2ccc(Br)cc2c1C C1(NC(C2C(=C)C2)=O)CN(C(c2ccccc2COC(C)(C)C)=O)CC1(C)C C1(C(N(C)CC2(NC(c3cnc4n3CCS4)=O)CC2)=O)CN(CP(C)(C)=O)C1 c1(NC(C(c2ccccc2)OC)C)nc(C(F)(F)F)ccc1C#N N1(C(CN(CCC)C(c2cccc(=O)o2)=O)=O)CCOC(CCC)C1 C1(CC(=O)NCC(C)CNC(C2CS(=O)(=O)C2)=O)CC2C=CC1CC2 N1(C(c2nc(OC)nc(O)c2)=O)CC(NC(c2cn(C)c(C)n2)=O)CC2(CC2)C1 C1(C(c2n(CC)nnn2)NC(CCO)C2CCC2)CCC2(CCC2)O1 c1(C(=O)NCCCC2OCCN(C(C(CC=CC)C)=O)C2)cc([N+](=O)[O-])oc1C c1(NC(C23C(CN(Cc4c(CC)cccc4)C2)C3)=O)ccc2c(ccn2C)c1 N1(C(CCC#N)=O)CC2CC1CCC2NC(=O)CCC1CCOC1 c1(C(C)=O)cc(=NC(=O)N2CCCC(Cn3cc(C(C)(C)O)nn3)C2)[nH]n1C C1(COC)(NC(=O)CCCc2ccccc2)CCCN(C(=O)C(C)(C)CO)C1 c1(C(=O)NC2(CO)CCN(C(C(COC)(C)O)=O)C2)ccc(OC)cc1OC c1(CNC(CC(C)N(C(C(C)=O)=O)C)=O)csc(COC(C)C)n1 N1(C(C(CCC)C)=O)CC(NC(=O)CN2CCCCCC2=O)CC(F)C1 N1(C(c2cc(CC)no2)=O)CCC(C(=O)NCC2C(=O)NN=C2C)C(O)C1 C(C)(C(CC(=O)N1CCSC2(CC2)C1)NC(c1cc(C)nc(C)n1)=O)OC C1(COC)CN(C(c2cnn(CCO)c2)=O)CCN1C(=O)Cc1cccc(F)c1 c1(C(N2CCN(C(C(CC)COC)=O)C(C)C2C)=O)ccc2nc(CO)[nH]c2c1 N1(c2n(Cc3n(CCOC(C)C)ncc3Br)nnn2)C2CCC1CC1(C2)N=N1 C1(O)(C(N(C(CNC(=O)Cc2csc(=N)[nH]2)C2CC2)C)=O)CCOCC1 Cc1nc(Cl)ccc1CC(=O)NCC1CN(C)CCN1C(=O)CCC(N)=O C(CO)(C(C)N=c1nc2sccc2c(N2CCN(C(=O)NC(C)C)CC2)[nH]1)SC N1(C(CS(N)(=O)=O)=O)CCC(NC(C2CN3CCN2CC3)=O)C(C(N)=O)C1 C(=O)(C(C)(C)CC1CC1)N1CCC(N(C(C(N2CCCCC2)C)=O)C)C1 c1(C(N2CC(C)C(c3ccccc3F)C2)=O)nc(NC2CC2)ncc1Br C(=O)(C(O)CCNC(C1CC(C)N1C(C1CC=CC1)=O)=O)OC c1(CNC(C2C(C(C)NC(C=C(C)c3ccco3)=O)C2)=O)ccn(C)c(=O)c1 c1(N(C)C)nc(C(=O)NC2(C)CCN(C(C3(Cl)CC3)=O)C2)[nH]c(=N)n1 c1(CC)cccc2[nH]c(C(=O)NCCCCC(C)NC(=O)COC(C)C)cc12 C1(C)(C(=O)NCC2(F)CCN(C(C3CCC(=C)CC3)=O)C2)CCCNC1=O N1(C(C(CC)C(C)C)=O)CC2=C(C1)CN(C(=O)Cc1ccc(Cl)cc1C)C2 C1(NC(C2C(C(C)(F)F)C2)=O)CC(C)(NC(=O)CCn2cnnn2)C1 c1(N2CCN(CCNC3CSC3)CC2)ncc(C)cc1S(=O)(=O)NC.CC c1(NCC2(NC(C3CCN(C(C)C)CC3)=O)CCC2)ccc(=O)n(CC(C)O)c1 c1(C(=O)NCc2ccc(CNC(C3CCC(OC)C3)=O)cc2)cc(N)ccc1Cl N1(CCNC(C=CC)=O)CCCN(C(c2cn(C)nc2-c2ccccc2)=O)CC1 C1(C(C(=O)NC(C)CCNC(c2cc(Cl)n(C)n2)=O)C)CCC(C)(C)CC1 CC(C)(CNC(C1COCC1C(N)=O)=O)CNC(C1(CC2CC2)CCCO1)=O C1(N(c2nnc(COC)s2)CC2CC2)CCN(C(c2cncc(F)n2)=O)CC1 N1(C(c2ncn(C(C)C)n2)=O)CCCC(CCCCNC(=O)CCS(C)=O)C1 c1(C(=O)NCC(C)(CC(C)C)NC(Cc2c(C)occ2)=O)nc(O)nc(O)c1F C(=O)(C(CC(C)C)ONC(=O)Cc1ccnc(O)c1)N(C12CCN(CC1)CC2)CC C12(CC(=O)NCC(CC)NC(c3c(Cl)c(C)nn3C)=O)CCCN1CCC2 c1(C(C)C)cc(O)ccc1NC(=O)C(CCF)NC(=O)CO.C1(CN)CCC1 C1(C(N(C)CC2CCN(C(CC3CCN(C)C3)=O)C2)=O)COCCN1C N#CC1(C(N2CCC(F)(C(=O)NCC(O)C(F)F)C2)=O)CC2CC2C1 C1(NC(COCC(=C)C)=O)CN(C(=O)C(c2cccnc2)O)CC1O N1(C(c2cc(C)c(O)cc2)=O)CCN(C(=O)CCc2cc[nH]n2)C2COCC12 N1(C(C2OCCC(C)(C)C2)=O)CCC2(C=C(C(=O)N(C3CCCC3)CC(N)=O)C2)C1 C1(CC(=O)N(CCOC)CCOC)CCC(NC(=O)CN2CC=CC2)C1 c1(C(=O)NC)cncc(-c2ccc(C3(NC(c4sc(Cl)nc4C)=O)CC3)cc2)c1 c1(OC)cc(C(N2CCC3(CC3C(=O)NCCC3CCCC3)C2)=O)cc(Br)c1 c1(C(=O)NCC23N(C(C(C(COC)C)C)=O)CC(C2)C3)cnc2ncccn12 N1(C(C2(C(C)NC(C3CC(=C4CC4)C3)=O)CC2)=O)CC(C2CC2(F)F)C1 Cc1cc(F)ccc1C1CC(Nc2cc(C(F)(F)F)ccc2N(C)C)C1 c1(CCC(=O)N(CCN(C(CCNC(=O)NC)=O)C)C)ccc(F)cc1F C1(NC(CC(CN(C)C)O)=O)CN(Cc2ccccn2)CC1N=[N+]=[N-] Cc1cc(C(=O)NC(c2cn(C)nn2)C(N2CCC(O)C2)=O)ns1 C1(NC(C2CCC(CNC(C3(CCOC)CC3)=O)C2)=O)Cc2cncn2C(=O)N1 Cc1cccn2ncc(C(N3CC(NC(=O)C=C4CCCCC4)CC(C)C3)=O)c12 C(=O)(C1COCc2ccccc21)NCCNC(Cc1cccc(C)c1F)=O C(C)(CC(=O)N1CCC1CNC(=O)C(C)N1CCCC1)SC c1(C(N2CC(O)(C(C)NC(=O)CC3COCCO3)C2)=O)cc(N)c(Cl)cn1 N1(C(CC(COC)(C)O)=O)CC2(C1)SCCC2NC(=O)CN1C(=O)CNC1=O C12(OC)CCC(C(=O)NCC3(CCNC(=O)Cc4ccncc4C)CC3)(CC1)C2 C12(C(=O)NC3CCCC3C3CC3)COCC1CN(C(=O)CCN1CCCCC1)C2 C1(CNC(=O)C=C2CCC2)CCCN(C(=O)Cc2ccc(F)nc2)CC1 C(C(CC(C)C)C(=O)NC(CC(=O)NCC1(CO)CC2CC2C1)C(F)(F)F)OC c1(N(C(C2CCOCC2)C(=O)OC)C)cc(C#N)cnn1 C1(NC(C=CC(C)NC(c2nc(C)n(C)c2)=O)=O)CCCCCC1C C1(C(N(CCNC(c2cnc(C)[nH]2)=O)C2CC2)=O)CC1C1(C)COC1 C1(C(=O)NCC=CCNC(C2CCCN(CC)C2)=O)CCc2nncn2CC1 Cc1ccccc1NNC(=O)C(C)Cn1c(C)nc2ccccc12 CCS(=O)(=O)C1(CNc2cc(N3CCOC(COC)C3)ncn2)CC1 C(CN=c1[nH]c(=N)[nH]c(=NCC(c2ccccc2F)OC)[nH]1)OC(CC)(C)C N1(C(C(C2CN(C(C3(OC)CCCC3)=O)C2)O)=O)CC(C)CCCC1C C(=O)(C1=NOC(c2ccccc2)C1)N1CC(OCCNC(=O)CC2(CO)CC2)C1 C12(C(=O)NCc3cccc(CNC(Cc4cc(C)no4)=O)c3)CC1CCC2(F)F C1(CCC)CN(C(c2cnc(O)o2)=O)CC1C(=O)NCCC1CC(C)C1 C1(NC(C(C)CO)=O)CC2(CCCCN2C(=O)C(N2CCSCC2)C)C1 c1(C(=O)NC2CCC(CNC(c3ccc(CC)o3)=O)C2)ncc(C)cn1 c1(CC(CNC(C2CC2C(F)F)=O)N(C)C(C2(C)COC2)=O)ccccc1 c1(CN(C(CN(CCC(C)NC(C2CC=CCO2)=O)C)=O)C)ccccc1 N1(c2nnc(-c3c(C)cc(COC)o3)n2CC(C)C)CCOCC(C)(F)C1 N1(C(C(C)CC2CC2)=O)CCC(CNC(c2nccn2C)=O)C1(C)C c1(CNCC2CC(C(C3C(NC(C4(SCC)CC4)=O)C3)=O)C2)ccccc1 C1(CN(C(=O)CC2CNC(=O)O2)C)CN(C(C2C=CCS2)=O)CCO1 N1(C(C2CCC(CC)O2)=O)CC(C(=O)NC(C)(CO)C(C)C)CCC1(C)C c1(C(=O)NC(CNC(C2(C(F)F)CC(F)(F)C2)=O)C2CC2)cccc2sccc12 CCCCCC(=O)NCC(=O)N(C)CCN(C(=O)C(O)CN1CCOCC1)CC c1(C(=O)NCCCCNC(c2ccc(F)c(F)c2F)=O)ccc2nc[nH]c2n1 C1(C)(CNC(CCCN(C(C)=O)C)=O)CCN(C(C2(C(=O)OC)CCCC2)=O)C1 C1(CC=C)(NC(c2nccs2)=O)CCCN(C(=O)Cn2nc(C)cc2C)C1 c1(Nc2ccc(C(N3CC(C(=O)OC)C(O)CC3)=O)c(N)c2)ccc(C)c(CO)c1 Cc1cccc(C(C)CNC(c2cccc(C)n2)c2nnnn2C(C)C)c1 c1(C(N2CCC(C)(CNC(C3CCCOC3)=O)CC2)=O)ccn2[nH]c(=N)nc2c1 CCCC(CC(C)C)C(=O)NCCN(C(=O)CC(C)(C)C(F)(F)F)C1CC1 N1(C(C(C)(C)N(C)C)=O)CC2(CCC(C(=O)NCc3ncccc3F)O2)C1 c1(NC(=O)NCC2CC(F)(CO)C2)ccncc1OC.C1(OC)CC1(F)F.O=CCN c1(OC2CCN(C(c3ccc(COC)o3)C(=O)NC)C2)cccc(C)c1 C1(C(N2C(N)CCC2)=O)CCCN(S(=O)(=O)C(F)(F)F)C1 N1(C(c2c(CC)con2)=O)CCCCC(NC(=O)C(C)NS(C)(=O)=O)C1 c1(CC)c(C(N2CCC2CNC(=O)CCc2ccnc(Cl)c2)=O)cnn1C Cc1[nH]nc(C(N2CC3CC2C3NC(c2ccc(Cl)cc2)=O)=O)c1Cl c1(CC(=O)NCCC2(O)CN(C(C3(CCF)CCC3)=O)C2)c(F)cccc1F c1(OC)cc(C)c(C(N2CCC(CN(C)C(C3(C#N)CCCO3)=O)C2)=O)c(C)c1 c1(C(N2CC(F)CC(NC(CCCNC(C)=O)=O)C2)=O)cnc(C)c(C#N)c1 C(=O)(CCC(F)(F)F)NCC(CO)NC(c1cn(CC)nc1C(C)(C)C)=O c1(C(N2CC(C)(CC(=O)Nc3ccc(F)c(CO)c3)C2)=O)cc(F)c(O)c(F)c1 C12(C(N3CCCC(CNc4nccc(OCC)n4)C3)=O)CC3CC(C(=O)N1)C2C3 N1(C(CN(CCC#C)C)=O)CC(NC(=O)CSc2nccn2C)C(C(F)F)C1 O=C(C#CC1CCCC1)NC12COC(C(=O)Nc3cc4ccncc4[nH]3)(C1)C2 CCCCCC(F)C(=O)N1CC(CNC(=O)C(F)(F)F)CC2COCC12 N1(CCCc2c(C(C)C)[nH]cc2)CCC(c2nc(C3CC3)no2)(c2ccccc2)C1 Cc1cc(Cl)ccc1C(=O)NC(C)(CNC(c1cc(F)n(C)n1)=O)CO c1(CNC(=O)Cc2ccccn2)cccc(C(=O)NC2(c3ccc(Cl)cc3)CC2)c1 c1(NC(C(CC)=O)=O)cnc(Cl)cc1C(=O)Nc1ccccc1C(N)=O N1(C(C2(CCC)CC2)=O)CCC=C(CNC(C23CCC(O)C2CC3)=O)C1 N1(C(CCc2c(OC)ccc(F)c2)=O)CC2(C1)CN(C(=O)C(F)C(C)C)CCO2 c1(C(=O)NC2CC(NC(c3cc(C(C)=O)sc3)=O)C2)ccc(O)c(Cl)n1 C1(C(=O)NC(C(C)C)CCNC(=O)CCCc2cccs2)CC12CCOC(C)C2 C1(CCNC(C(N(C(C(C2CC2)SC)=O)C)C2CC2)=O)CCCCCC1 C12(C(=O)NC(CCC(=C)C)C)CCC(CC1NC(=O)CC13CCCC1C3)C2 CC1=C(C)CC(C(=O)NCC2COCCN(C(=O)CCCCCN(C)C)C2)CC1 C1(CO)CCCC(N=c2ccc3c([nH]2)CCCC3=O)C1 C12(NC(C3C(C(C)NC(C(C)C4CCC4)=O)C3)=O)CCCN(CCC1)C2 c1(N(CC)CC)ccc(NC(=O)C(=O)NCC(C)N(C)C)cc1.c1(S)ccc(I)cc1 c1(C(=O)NC2(C)CC(NC(=O)CC(F)(F)F)C2)ccc(OC(F)F)c(F)c1 c1(CNC(C2CCCN2C(=O)COC2CCOC2)=O)cc(F)cc(F)c1 C(=O)(CCC(=O)NCCOCCCOCCNC(C1CCOCC1)=O)OC C1(N(C(=O)C(C)(C)NC(=O)Cc2cccs2)C)COC(C)(C)C1 c1(C(N2CC3CCC(C2)N3c2ccncn2)=O)ccc([N+](=O)[O-])nc1 N1(C(CN(CC)CC)=O)CCC(F)(F)C(CNC(c2cc3cnccc3o2)=O)C1 C1(C)(NC(C(C=C)OC)=O)CCCCC1C(=O)N(CC(=O)OCC)CC C1(O)(C(C)NC(Cc2cc(C)sc2)=O)CCN(C(C2(c3cccnc3)CC2)=O)C1 CCC(CC(=O)NCC1(OC)CN(C(=O)C(C)(C)CC2CCOC2)C1)SC c1(C(=O)NCCN(C(=O)CCOC2CCCOC2)CCOC)cc(O)n(C)n1 N1(C(C(C)C(F)F)=O)CCC(NC(=O)C=Cc2ccncn2)C12CCC2 N1(C(C2C(=C)CC2)=O)CCC(C2(NC(=O)C(O)C(C)(C)CC)CCC2)CC1 c1(C(=O)NCC2OCCN(C(C3(COC)CCCCC3)=O)C2)nccc(Cl)c1C c1(C(=O)NCCS(CC)=O)cnc(CNC(C2(C)CCCCC2)=O)nc1 CC1CCCN(C(C2(C)CCN2C(c2cccc(Cl)c2)C2CC2)=O)CC1 C=CCCCC(C(=O)NC(C)CS(N)(=O)=O)NC(c1cnc(CC)o1)=O c1(NC(=O)NC2C(OC)(OC)C2C(=O)O)c(C)cccc1C c1(OCC)cc(C(=O)NCCC2CCN(C(C3CC3CF)=O)C2)cc(Cl)c1O C1(NC(c2onc(C)c2C)=O)COC2(CCN(C(c3cccc(Cl)c3Cl)=O)C2)C1 C(CS(C)(=O)=NC(=O)c1nc(-c2ccc(Br)cc2)cs1)OCC C1(NC(c2ccc(Cl)nn2)=O)COC2(C1)CN(C(C1C(F)(F)C13CCC3)=O)C2 C1(C(C(=O)NCC(=C)CC)C)CCCN(C(c2cnn(CC)c2C)=O)C1 C(N=c1cc(C2CC2)nc[nH]1)c1c(CNC(CC2ON=C(CC)C2)=O)cccc1 c1(C(=O)NCC(CNC(c2c(C(C)C)ncs2)=O)(C)F)cccc(O)n1 C1(CCC)(NC(c2ccc(OC(F)F)cc2)=O)CCCN(C(C2CC2CF)=O)C1 N1(C(c2onc(OC)c2Br)=O)CCC(NC(=O)Cc2csnn2)C(F)C1 c1(C(=O)NC2COCCN(C(c3c(CC)ocn3)=O)C2)ccc2nncn2c1 c1(C(N2CC3C(CNC(C(C(C)C)SC)=O)(C3)C2)=O)cnc2n1CCS2 N(C1CCCOc2ccc(Br)cc21)(CC#C)C(=O)NC12CCC1S(=O)(=O)C2 C(=O)(CCCC(C)OC(c1ccn(C2CCC2)n1)=O)OCC CC1CN(C(c2ccc3c(n2)CCOC3)=O)CC(C)N(C(C2CC=CCO2)=O)C1 C(CC(C)C(=O)N1CCCC1CNC(c1cc[nH]c1C(C)C)=O)OC N1(C(Cn2cc(C(=O)OC)nn2)=O)CC2CC(NC(c3cnn(C)c3OC)=O)C1C2 Cc1cc(C)c(C(=O)NCC2CCN(C(c3ccnn3CC#N)=O)C2)cc1C N1(CC)CCC(C(=O)NC2(C)CN(C(=O)Cc3ccccc3O)C2)CC1 C1(C(=O)NCCOCCNC(C2CCN(OC)CC2)=O)CCC(=O)N2CCCC12 C1(O)(CNC(CCCC#C)=O)CCN(C(c2c(C)ncn2OC)=O)CC1 N1(C(C)C)CC(C(=O)NC(C)(C)CCCNC(C2CC2F)=O)CC1=O Cc1csnc1C(=O)NC(C)CCN(C)C(C1CCCCS1)=O CC#CC1CCN(C(=O)C(C(C)C)NC(c2cscc2OC)=O)CC1 C(C(=O)N(CCNC(C)=O)CC1CC1)(C1CCCC1)SC.C1COC1 CCCCC(O)C(=O)NCC1CN(C(C2CN(C)C(=O)N2)=O)CCCO1 c1(C(N2CC(C(N3CCOC4(CC4)C3)=O)C(F)C2)=O)nccc2cc[nH]c12 c1(C(C)=O)cc(=NCC2CCCN2C(=O)CCNC(c2ccccc2)=O)[nH]cn1 c1(N(CC(C(C)C)c2ccnn2C)C(C2CCN2CC(F)F)=O)ccnc(Cl)n1 C=CC(C)(C)C(=O)N1CC2CC1C2NC(=O)Cc1c(C)noc1C C1(C)(C(=O)NCC(c2ccccc2)N(C(C(CO)OC)=O)C)CCC(C)(C)CC1 c1(C(=O)NCCn2ccnn2)csc(Cc2ccco2)n1 c1(S)ccccc1F.Cc1[nH]ccc1C(=O)NC(C1(CC2(C=O)CCC2)CC1)C C1(NC(c2cnc3[nH]cncc2-3)=O)CN(C(C23CC(CO2)C3)=O)C2(CCC2)C1 N1(C(CN2C(CC=C)CCCC2)=O)CCN(c2ccccc2)C(C)C1=O c1(C(N2CC(CC)N(C(c3ccsc3)=O)CC2)=O)cn2nc(C)sc2n1 CN1CCN(C(C(=O)NC2(C)CC2)C2=NOCC2)CC12CCOC2 C12(NC(c3[nH]nc(OC)c3Cl)=O)CCC(C1)N(C(=O)CC1SC(=N)NC1=O)C2 c1(NC(C(C)(C#N)c2ccccc2)=O)cc(Br)ccc1F N1(C(CC(C)N(C)C)=O)CCN(C(=O)CC2CCC2(C)C)CC(C)(C)C1 C1(NC(C(CC)=CCCC)=O)CCSC12CN(C(C1CCCN1S(C)(=O)=O)=O)C2 C#Cc1cccc(OC)c1.N12CCN(C(=O)CCCC(=O)N(C)CC)C(C1)C2=O CC(CCCNC(=O)CCN(CCO)CCO)NC(C1(F)CCOC1)=O N1(CCNC(CN(C(=O)C(O)(C2CC2)C2CC2)C(C)C)=O)CCNC(=O)C1 C12(NC(Cn3nc(C)n(C)c3=O)=O)CCCC1N(C(=O)CC1CCC(=O)N1)CC2 c1(C(C(=O)OCC)(C)C)ccc(NC(c2nccnc2N)=O)c(Cl)c1 c1(CC)cccc(C(=O)NCC23CC(NC(=O)C=CC(N4CCCC4)=O)(C2)C3)c1 c1(C(N2CC(C)(NC(C3CC34CCOC4)=O)C2)=O)nnn2c1C(=O)NCC2 c1(C(=O)NC(C2(NC(C)C)CCC2)C)ccc(N(C)C)cc1 c1(C(N2CCC(CC(=O)NC(CCSC)CO)C2)=O)ccc(O)nc1C C1(CNC(CCn2c(C)ncc2)=O)CN(C(=O)C(C)C(C)(C)C)CC1(F)F Cc1ccc(C(=O)NCC2(O)CN(C(=O)C=CCOC3CCOCC3)C2)c(N)c1Cl C(=O)(C(CCC1CC1)NC(c1cc(CCO)on1)=O)NCCc1cc(C)on1 C1(C(=O)NC2CCC2C(F)F)CC2(CC(C(=O)NCC3CCCO3)C2)C1 CCC(CCC(=O)N(C1CCCN1C(=O)CC1CC2CC2C1)C)NC(C)=O c1(C(N(CCCNC(CCCOC(C)=O)=O)C)=O)ccc(N2CCOC2=O)cc1 C(=O)(CC(C)(C)C1CC1)N1CCC(N(CC#C)C(C2CC(OC(C)=O)C2)=O)CC1 N1(C(c2ccc(CCCC)cc2)=O)CCN(C(=O)C(C)C(O)CC)CC1COC c1(NC(C2CC(NCc3c(CO)nn(C)c3O)C2)=O)c([N+](=O)[O-])ccc(Cl)c1Cl c1(SC)ccc(Cl)c(C(=O)NC23CC2CN(C(c2cccc(C)c2F)=O)C3)c1 C(=O)(C#CC1CCCOC1)N1CCCN(C(C2(F)CCCCC2)=O)CC1CO c1(C(N2CCC(NC(c3ncc(C)nc3)=O)C2)=O)ncccc1[N+](=O)[O-] c1(C(=O)N(C(CC(C)NC(CCC2(C)CC2)=O)C)CC)cc(C)ccc1N1CCCC1 N(C(=NCCCCl)NCC1CC=CCC1)CC1N(Cc2cc(C)on2)CC1 c1(CC(C(=O)NC(C)CCO)NC(C(C2CCCC2)OC)=O)ccccc1Br CCCCC(C)C(=O)N1CC(CNC(=O)CCc2nnc(C)n2C)C(C)C1 C1(NC(c2ccsn2)=O)CCN(C(C2(F)CCCC2)=O)CC1F C(=O)(C1CCc2cccc(O)c21)NCC1CN(C(=O)Nc2ccc(SC)cc2)C1 C=C(Cl)CCC(=O)N1CCC=CC1C(=O)NC1CC(CC(N)=O)C1 C1(CN(C(C2(COC)COC2)=O)C)CCN(C(c2cncn2C2CC2)=O)CC1 c1(CNc2ccc(NC(C3C4COCC34)=O)cn2)cc(F)cnc1Cl C1(CNC(c2nccc(CC)c2)=O)CCN(C(c2sc(C)cc2C)=O)C12CCC2 c1(CNC2CCCC(C(N3CCC(O)C3)=O)C2)ccc2cc[nH]c2c1Cl c1(CC(=O)N(C2CN(C(C3(CCF)CCC3)=O)C2)C)ccc(C(F)(F)F)cc1 N1(C(C2CC(C)NC(=O)C2)=O)CCN(C(=O)Cc2c(F)cccc2F)CC(O)C1 c1(CN2CC3(C(C(=O)Nc4nccc(C)c4)C3)C2)ccc(I)c(F)c1F Cc1c[nH]c(CC(N)=O)c1C(=O)NC1(CNC(C2CCCCN2C(C)C)=O)CCC1 N1(C(c2cnc(C(C)O)s2)C(=O)NC(CC)(C)C)CC(C)S(=O)(=O)C(C)C1 CCC(CC(=O)NCCC(C)N(C(=O)C(C1CC1)OC)C)SC C(CCCOC)(C(=O)N1CCC(C)(OCC)CC1)NC(CC=CCCCCC)=O N1(C(C2CCN(C)C2)=O)CCC(C2(NC(C3OCCOC3(C)C)=O)CCC2)CC1 c1(OC)ccc(S(=O)(=O)NC(c2ccccc2)CO)cc1C=CCO C(CC(=O)N1CC2CCN(C)C2C1)(C(F)(F)F)NC(c1c(CC)cccn1)=O C12(C(N(CCOC)C(C)C3CC3)=O)CCC1CN(C(c1cc(N)cc(F)c1)=O)C2 CN1CCC(CN(C)C(C2COC(CNC(=O)Cn3[nH]cnc3=N)C2)=O)C1 N1(C(c2c(C)nc(C3CC3)s2)=O)CC2CC1CC2NC(=O)C=C1CCC1 C12(NC(c3cc(CC)on3)=O)CCC1CN(C(C13CC(C)C1C3)=O)C2 N1(C(CC2CC(=O)C2)=O)CCN(C(C2CS(=O)(=O)CCO2)=O)C(CO)C1 c1(C(N2CC(NC(c3nc(C)n(C)c3)=O)C(F)CC2)=O)cc(O)cc([N+](=O)[O-])c1 N1(C(C)=O)CCC2(C1)CN(C(=O)C=Cc1ccncc1C)CCO2 c1(C(N2CC3CCCC(C2)N3C(C2CC2F)=O)=O)c(F)cccc1[N+](=O)[O-] c1(C(=O)OC)cn(C2CCN(C(=O)C(F)=CNC(CSCC=C)=O)C2)nn1.CCOC Cc1ccccc1C(C)(C)CNC(C1=CCCC1)c1nnnn1C1(C)CC1 Cc1cc(C(=O)NCCCN2CCC(NC(c3cc(F)n(C)n3)=O)C2)cn1C Cc1c(C(=O)NCC2(O)CN(C(C3(Cl)CC34CCC4)=O)C2)cncc1Br CC1C(NC(c2c[nH]c(=O)cn2)=O)CCN1C(=O)CC1CSCCS1 c1(CNCCC)ccc(-c2cnc(O)s2)c(F)c1F C1(C(N2CC=C(C)C2)=O)CCC(C)CN1C(=O)CC1(O)CCCOC1 CC1(C)C=C(C(=O)NC2CCC2NC(c2cc(Br)cn(CCO)c2=O)=O)C1 N1(c2nnc(-c3c(C(=O)OCC)csc3C)n2C2CC2)CCCC(CC)(CO)C1 c1(CC)ccc(O)c(NC(=O)C=CCNC(C2CCCC2C(C)C)=O)c1 C1(C(N2C(CCNC(C(C)OCC3CC3)=O)CCCC2)=O)CC2CCC(C1)C2 Cc1cnccc1C=CC(N1CC(O)(CCNC(=O)C(n2cc(C)cn2)C)C1)=O Fc1ccc2c(CNC3CC(c4cncc(Br)c4)C3)n[nH]c2c1F CC(C)C(C(=O)OC(C)(C)C)NC(=O)CCC1CCCCN1Cc1cnccn1 C1(C#N)(SC)CN(C(=O)CC(CNC(C2CC(CF)C2)=O)C2CCC2)C1 CCCCC(CC)CC(=O)NC(CN(C(c1cc(C(C)(F)F)on1)=O)CC)CC CCC(CCCO)NC(C1CN(C(c2nnc(S)n2C)=O)CCO1)=O C1(C(=O)NC(C2CCCN2C(=O)CC2CC2)(C)C)CCC(F)(F)CC1 Nc1cccc(C(=O)NCC2(NC(=O)CCCc3cnn[nH]3)CCCCC2)c1 C(=O)(C(CCF)NC(=O)C1=CCCC1)NC(c1cccc(Cl)c1)C CCCCC(O)C(=O)NCCCN1CCC(NC(c2cncnc2C)=O)C1 N1(C(C=COCC)=O)CCN(C(c2cnn(C)c2C)=O)C(CC#N)C1 c1(SC(C)(C)C)n[nH]c(=NCC2CCC(NC(=O)C=CC3CCCCC3)C2)s1 Cc1cccc(C(N2CCC(N(C(=O)C(Cc3cccc(Cl)c3)=NO)C)C2)=O)n1 C1(NC(c2cn(C)nn2)=O)CN(C(c2ncc(F)cn2)=O)CCC12CCC2 C1(C(=O)NCCCc2cn(CC3CCC3(C)C)nn2)(OC)CCOCC1 c1(OC)ccccc1C(=O)NCC1CN(Cc2csc(Br)c2)C1 N1(C(CCCc2scc(C)n2)=O)CCCC(c2cn(CC3CCC(=O)O3)nn2)C1 c12ccc(cn1)[nH]2.C1CC(=O)NC(=O)C12CC2.C(C)(C(C)n1cncn1)OCC N1(C(c2c(OC)cncc2)=O)CCN(C(=O)Cc2cccc(C)c2F)C(C)C1C c1(C(=O)NCC2(CNC(C3(COC)CCCCC3)=O)CC2)cc2cccnn2n1 N1(C(=O)CCn2cnc([N+](=O)[O-])c2)CC2CCC1CN2C(C1CCC(F)C1)=O C(CCC(C(=O)NC1(c2ncsn2)CC1)NC(C1CCC(O)CN1C)=O)OC c1(OC)ccccc1CC#N.C1(S(N)(=O)=O)(CN2C(=O)NCC2)CC1 c1(C(=O)NCC(CC)NC(=O)C(c2cccc(C)c2)(F)F)cc2n(c1)CCC2 Cc1cc(C(=O)N(C2CCCN(C(C3(C)CCCCO3)=O)C2)C)nn1C N1(C(CC(C)OC)=O)CCC2(CC1)CCN(C(=O)CCCC(C)=O)CC2 N1(C(CCCOC(C)=O)=O)CCC(CCN(C(=O)Cc2cc(Cl)n(C)n2)C)CC1 N1(C(C2C(OC)CC2)=O)CCCCC1C1(NC(C2CCN(C)C2)=O)CC1 CCCCCC(C)(CC)C(=O)N(CCNC(=O)CN1CCCC1=O)CC c1(CC)cc2c(Cc3ccc(F)cc3)ncnc2s1.C12(CCCC1)NC2 C1(C(N(C2CC2)CC2N(C(c3n[nH]c(C)c3N)=O)CCC2)=O)CCCCC1(C)C c1(-c2n(CCC#N)c(N3CCN(C)C(C4CC4)C3)nn2)c(F)c(F)cc(F)c1F c1(NC(c2ccn(CC)n2)c2nnnn2C2CCOCC2)c(F)cc(Cl)cc1Br c1(C(N2CC(CC(CNC(CCC3C(C)C3)=O)(C)C)C2)=O)c(Cl)cncc1Cl c1(OC)ccc(C)nc1C(=O)NCC1CCN(c2nc(SC)ns2)C1(C)C N1(c2c(C)cc(CC)c(C)n2)CCC2(CCCN(C(=O)CC(C)C)C2)C1 c1(CC)ccc(C(N2CCCC(NC(C3CSCC(=O)N3)=O)C2)=O)cc1N CCCC(C(=O)N1CCC(OCC(=O)NCC2(F)CCCCC2)C1)OCC CC1(C)CCC(C#N)=C(C(=O)NCC2C=CCN(C(=O)CCP(C)(C)=O)C2)C1 C1(CC(=O)N(CCCCN(C(CC2CC(=C)C2)=O)C)C)CCCCO1 CCC(C)CC(=O)C(=O)N1CC(n2cc(CC3CN(c4ccccn4)C3)nn2)C1 c1(C(=O)NC(CC)(C2CC2)C2CC2)conc1C(C)NC(=O)CCCn1ccnn1 N1(C(c2cn(CCC)nc2)=O)CCN(C(=O)C(CC)C(C)C)CC1C C(CC(F)(F)F)SCC(=O)NCCN(C(=O)CC1CCOC1)Cc1ccccc1 Cc1cc(N2CCC(CN(C)C)CC2)nc(N2CCC(C(F)F)C2)n1 C(=O)(C1Cc2ccccc21)NCCN(C(C(C(C)C)(C)O)=O)C1CCCCC1 C(c1ccc(O)c(O)c1)=CC(=O)Nc1ccc(F)c(C(=O)O)c1 N1(C(C2CC2C2CCCCO2)=O)CCC2(CC1)CN(C(=O)CCCN1CCCC1)C2 N1(C(C2CC(=C)C2)=O)CC(NC(C2(C(=O)O)CC2C(F)(F)F)=O)CC(F)C1 N1(C(C(=O)N(C)C)=O)CC2CC2(NC(C2CCC3CC23)=O)C1 N1(C(c2c(OC(C)C)cccc2)=O)CCN(C(=O)CC2CC2)C(CCOC)C1 c1(OC)ccncc1C(=O)NC1CC(C)N(C(c2sccc2CO)=O)C1 c1(C(N2CC(C)OCC(C)(C)C2)=O)c(F)ccc2ccncc12 Cc1cc(C(=O)N(CC(C)(C)C(=O)NCCc2ccns2)C)cc(C)c1 c1(COC)cccc(C(=O)N(C)CC2CCN(C(=O)C(C)N3CCC3)C2)n1 O=C(C1=CS(=O)CCC1)NCC1C2CN(C(=O)CCc3cc[nH]n3)CC12 C1(C)(CNC(C(c2ccc(OC)cc2)C)=O)COCCN(C(=O)CC(C)(C)O)C1 C1(N=c2cc[nH]c(O)n2)(CNC(C(CC)CC2CCCC2)=O)CCCCC1 C12(C(=O)NCCC3(O)CCN(C(c4ncn(CC)c4)=O)C3)CCCC(C1)OC2 C(C)(C)(CCCC(=O)N1CCSCC1C(=O)NCCCC1C=NNC1=O)OC C(=O)(C1=CCCCC1C)NC1(C(=O)Nc2nc(C)nc(O)c2)CCC1 n1(CCNC(C2CCC(c3cn(CCn4ccc(C)n4)nn3)C2)=O)cccnc1=O C(=O)(CC(C)(C)C(=O)OC)NC1C(=O)NC1.C(CC(C)(C)C)OC Cc1[nH]nc2c1CCC(C(N1CC3COCC(C1)C3NC(=O)CCC(C)C)=O)C2 CCC(CCC(=O)NC(COC)CCO)NC(=O)C(C)CSC N1(C(C(CO)OC)=O)CC(=O)CC1C(=O)NC(CCO)C1CCC1 N1(C(c2cccc(C#C)n2)C(=O)NCC(C)C)CCC2(CC1)CC(N(C)C)CO2 N1(C(C2CC(CC)(CC)C2)=O)CC2CCCC2(NC(=O)Cc2csc(Cl)n2)C1 C#CC1(O)CCN(C(=NCC2C(C)(C)C2(F)F)NCC(F)F)C1 c1(C(N2C(C(=O)NC(COC)COC)CC3CC32)=O)ccc(Cl)c2ccccc12 C(=O)(C1=CCCCC1)N(C)CC1CCCN1C(=O)CCCOC(S(C)(=O)=O)=O C1(NC(COCCC)=O)CC2CCC1(NC(=O)CC(=O)N(C)C)C2 C1(C(N2CC(N(CCOC)C)C2)=O)CC12CC(NC(C1CCC(C)(C)C1)=O)C2 C#CC1(C(=O)NC(C)C(C(C)C)NC(c2coc(N(C)C)n2)=O)CCCC1 c1(C(=O)NC2C(NC(C3(OCC)CCCC3)=O)COC2)cnn2c(Cl)cccc12 C(CC(C)(C)C#N)NC(C1CCC(NC(c2cn(CC=C)nn2)=O)C1)=O C(=O)(C1=CCCC1)NCc1cn(CC(=O)NC(C2CCCCC2)C)nn1 C1(NCc2ccc(OC(F)(F)F)cc2Cl)CCCCC12CCCC2 C(=O)(CC(C)C(F)F)NC(C(=O)Nc1ccc(C(C)=O)cc1)CC1CC1 c1(OCCOC)cc(C(=O)NSc2nc(N3CCCC3)ccn2)cc(C)c1 c1(NC2CCN(C(C3(C4CCCO4)CC3)=O)C2)ccc([N+](=O)[O-])c2cccnc12 c1(C(N2CCC(C)(NC(C(C(CC)C)O)=O)CC2)=O)c(OC)cc(OC)cc1N N#Cc1ccc2[nH]cc(C(N3CC(Nc4ccncn4)CC(F)(F)C3)=O)c2c1 c1(OC)ccc2c(N3CCC(O)(CC(=O)OCC(=O)N(C)C)CC3)ncnc2c1 O=C(CCCNc1ncccn1)NC1CCN(C(=O)CCc2ccoc2)C1 c1(C(N2CC(N(C)C(C3CCCCN3C)=O)C2)=O)cc2c(s1)CCSC2 N1(C(C(n2ncc(C)c2)C)=O)CC2CCC(C(N3CC4C(C(N)=O)C4C3)=O)(C2)C1 C1(C(N(CCC)CC)=O)CCCCCN1C(=O)COc1ccccn1 Cc1cc(C)c(C(N2CC3CC3(NC(=O)CC3CCSCC3)C2)=O)cc1N c1(NC(C(CCCOC)NC(=O)Cc2cncn2C)=O)cccc(C#N)c1C C1(C(=O)NCC2CC(C)(C)OCC2)CCN(C(=O)CCCC2CCC2)C(C)(C)C1 C1(C(=O)NC(C)CCCNC(=O)C#CCN(C)C)COCC(C)O1 c1(NC(=O)NCC2C(=C)C2)cnc2ccc(F)cc2c1 c1(OC)ccc(C(=O)NC2CCN(C(C3CC4(C3)CC4F)=O)C2C)c2sccc12 c1(C(=O)NCCC(C)(C)NC(C2CCCC(OC)C2)=O)cc(F)c(Cl)cc1Cl CCC1=NOC(C(=O)NCc2cn(CCNC(=O)Cc3cnn(C)c3)nn2)C1 C(c1nc(C)cs1)=CC(=O)NCC(C)(CO)NC(c1c(CC)c[nH]n1)=O Cc1cccc(C(=O)NCC2(C)CCN(Cc3cscn3)CC2)c1I C(=O)(C(C)C(O)C(C)C)NC(CCC)C(=O)NC12CCC(C1)OC2C N1(C(=O)Cc2ccc(O)nc2)C2CCC1CN(C(C1(Br)CC1)=O)CC2 c1(C(N2C(C)CC2C(=O)N(C)CCc2nccs2)=O)cccc2c1CCC2 Cc1cc(=NC(=O)C(=O)NCC23CC(CN2c2nccc(C(N)=O)n2)C3)[nH]o1 Cc1c(C(=O)NCC2CCCC(NC(C34CC(F)C3C4)=O)C2)ccc(F)c1F c1(CC(C)C)ccc(C=CC(N2CCN(C)CC2CNC(c2cnc[nH]2)=O)=O)cc1 C1(CNC(COCC=C)=O)CCCN(C(=O)CN(CC)CC)C1 CC(C)CC(O)C(=O)N1CC(C(N2CCC(OCCF)C2)=O)CC(C)C1 c1(OC)ccnc(C(=O)NCCC2(O)CN(C(C3(CC4CC4)CCC3)=O)C2)c1C C(=O)(CCC(=C)C)NCCCOCCCNC(C1C(CC#C)CCO1)=O O(NC(=O)C(C)(C1CC1)N(C(=O)C=C1CCOCC1)C)CCC(C)C.c1(=O)cn1.C C1(C(=O)NCCN(CCC)C(c2cc3scnc3[nH]2)=O)CCCC1S(C)(=O)=O C1(C(=O)NCC(CC)N2CCCC2)CCN(C(=O)CN(C)CCOC)C(CC)C1 c1(C(=O)NCC(C)(CO)NC(c2cc(C)ns2)=O)cc(S(C)(=O)=O)c(C)o1 C(=O)(C1=CC2CCC1C2)NC1(C)CN(C(c2c(C)[nH]c(C#N)c2)=O)C1 c1(C(=O)NCCOCCNC(C2CC2F)=O)ccnc(CO)c1 N1(C(c2c(C)c(C(F)(F)F)n[nH]2)=O)CCCN(C(C2CCC(C)O2)=O)CC1 c1(C(N2CC(OC)C(NC(c3cncc(F)c3)=O)C2)=O)ccc2nsnc2c1 c1(C(=O)NC2C(NC(C(CC#C)C3CC3)=O)C2)nccc(Cl)c1C C1(CNC(c2c(O)ccc(C)c2)=O)CC2(CCN(C(C3CCOC3C)=O)CC2)C1 C1(NC(C2CC(CNC(c3cccc(F)c3)=O)C2)=O)CCCN(C(C)=O)C1 c1(C(=O)NC(C)CN(C)C(c2csnn2)=O)ccc(C(F)(F)F)cc1C(F)F C1(NC(C(CC)=CCCC)=O)CCN(C(=O)C(C)c2ccco2)C1C C(CC(=O)NCC(C)C(C)C)(CC(C)C)NC(c1ccc(C)c(C)c1)=O N1(C(C=C2CCC(C)C2)=O)CCCC2(C1)CN(C(=O)Cc1cncc(F)c1)C2 N1(C(c2c(CC)cncc2)=O)CC(C)C(NC(=O)C=Cc2cnc(C)s2)C(C)C1 CC(CCCNC(c1cn(Cc2ncccn2)nn1)=O)NC(c1csc(Cl)c1)=O C12(C(=O)NCCC3(COC)CC3)CCCC1(C=O)C2.c1(C(=O)NC)coc(C(C)C)n1 C1(C)(C(=O)NCC2(COC)CC2)CCCN(C(C2CC23CNC3)=O)C1 c1(CC(=O)NC2CCC(F)(CNC(Cc3cn(C)nc3)=O)C2)ccc(F)c(F)c1 c1(OCC)cncc(C(N2CCC(C(=O)N(C)Cc3ccccc3)C2)=O)c1 C(=O)(CCCC(=O)NCCC1CCCN(C(=O)CCCCSC)C1)OCC c1(OC)cc(NC(=O)CCC2CCCN(C(=O)CCCOC)C2)ccc1C C1(CC(N2CCN(C(c3csnc3Cl)=O)CC(O)C2)=O)Cn2ccnc2NC1=O C1(C)(C(NOCC2(COC)CC=CC2)=O)CCCCC1 C12(SCC)C(N)CC1C2(F)F.c12nc(cs1)C(OCC)C(=O)NCC2.C(=O)(CC)N.CC c1(CC(=O)NC2CC(C)(CNC(C3OCC(C)(C)C3)=O)C2)ccc(Br)cc1O c1(CCNC(C2CC(C(C)=O)CN2C(=O)OC(C)(C)C)=O)c(Cl)cccc1Br Cc1cc(Cl)c(C(N2CCC(C)(CNC(=O)Cn3ccsc3=N)C2)=O)s1 c1(NC(C(N2CC(c3cccc(C)c3)OCC2)=O)=O)c[nH]c2ccccc12 c1(-c2nc(-c3cc(-c4n(CCCCC=C)ccn4)on3)on2)ccc(OC)cc1 O=C(CSC1C=CCCC1)NNC(=O)Nc1ccc(-c2nn[nH]n2)cc1 c1(CC)ccc(C(=O)N(CC(C)CNC(=O)C(O)Cc2ccco2)C)cc1CC c1(OCC(=O)N(C)CC2CCN(C(C3(CC=C)COC3)=O)C2)ccc(OC)cc1 N1(C(=O)NC2C(n3cc(C(C(C)C)(C)C)nn3)CCC2)CCC(C)(CC#N)C1 c1(C(=O)NCC2CCN(c3snc(CCC)n3)C2)ccnc2[nH]nnc12 C1(NC(CCNC(=O)NCC)=O)CC2CC1CN2C(=O)C(CC)OCC Cc1cc(C(N2CCCC(C(=O)NCCN(CCO)CCO)C2)=O)cc(C)c1Br c1(N(C(C2CCNCC2)C)Cc2c(C)cccc2Br)ncnc2cc[nH]c12 C(=O)(CC1=CCCC1)N1CCC(NC(C(C)OCC)=O)CC1 c1(C(N2CCC(SCn3cc(C(C)OC)nn3)C2)=O)ccc(OC(F)F)c(F)c1 c1(C(=O)NC(CNC(C(CC)(C)OC)=O)C2CC2)cc2nc(F)ccc2o1 C1(CNC(CC=C(C)C)=O)CN(C(=O)CCOC2COC2)CCC12CCC2 CC1CCCCC1(CNC(c1cnc(C(C)(C)C)[nH]1)=O)NC(=O)CC1CN(C)C1 C1(NC(C=CC(CC)C)=O)C(CC(=O)N(C(C)CN(C)C)C)C1(C)C O(NC(=O)CC1C(NC(=O)CCc2ncccn2)CC1O)CCSC Cc1ccc(CCNC(=O)C(N2CCOC(c3cccs3)C2)=O)c(Br)c1 CC1(C(N2CC3CC3(CNC(c3ccnnc3O)=O)C2)=O)CCNC1=O c1(C(C)C)noc(CCC(=O)NCCC2CN(C(c3coc(Br)c3)=O)C2)n1 c1(-n2c(-c3n(CC)nc(C)c3)nc(-c3cnn(CC)c3)n2)cccc(Cl)c1C CCC(C)C(C)C(=O)NCC(C)CN(C)C(C1(CC)CCCC1)=O c1(N2CCC(CNC(CC=C)=O)(CO)CC2)ncc(C)c(OCCC)c1C N1(C(=O)CC2CN3CCN2CC3)CC2CC(NC(COC(CC)C)=O)C2C1 c1(OC)c(NC(=O)CNC(Cc2ccco2)CO)cc(C)cc1C c1(C(=O)NCC2(NC(C34CCCC3CC4)=O)CCC2)cccc([N+](=O)[O-])c1 C(C)(C(C(=O)NCC1CCCC1O)NC(=O)CCCC1CC1)OC N1(CC(=O)NC(CCN(C(c2c(C)cno2)=O)C)C)CCC(CO)CC1 CCCCC(O)C(C)C(=O)N1CCC(O)(CCNC(C2(C)COC2)=O)CC1 CCCC(CCc1ccccc1)C(=O)N(CCNC(=O)C=CC=CC)C1CC1 C12(CNC(C(C)OCC)=O)CCCCC1N(C(c1cc3ccc(C)cc3o1)=O)CC2 C1(C(N(CCCO)CC#C)=O)CC(C)CN(C(=O)CC23CCCC2C3)C1.C1CC1 C(C(CC1CCCC1)C(=O)N(c1csnc1C)C)NC(c1ccc(C(C)=O)[nH]1)=O N1(C(c2cccc(CC)n2)=O)CCN(C(c2c(C)csc2Cl)=O)C(C)CC1C C#CCC(C)(C(=O)NCC(C)CO)NC(=O)C(O)CN(C)C C1(C(N(C(C)CNC(C2CC2c2cnnn2C)=O)C)=O)COC(=O)C1 CCC(CC(=O)NC(C(=O)NCCCC(C)(C)C)C1CC1)C(C)(C)C N1(C(C(C(C2CN(C(C3(C(N)=O)CC3)=O)C2)O)=O)=O)CCn2cnnc2C1 C(C(CC(C)C)C(=O)NCCOC(C)(C)CNC(=O)C(C)(C)C(N)=O)OC Cc1cc(C(=O)NCC2COCCN2C(c2cc(C(C)C)sn2)=O)sc1Cl N1(C(C2CCC(OC)CC2)=O)CC2CC1CC2C(N1CC(O)C1)=O CCCCC(CCCC)NC(C1(C)CC(O)CN1C(=O)C=C(Cl)Cl)=O N1(C(c2scc(C)c2C)=O)CCC(C(N2CC(CO)CC2CO)=O)C12CCC2 C1(NC(C2C(Oc3ccc(C(=O)OC)cc3)CCC2)=O)CCCS(=O)(=O)C1 N1(C(CC(C)SC)=O)CCN(CC(C)NC(=O)CCCCN(C)C)CC1 C1(C(N(CCCN(C)Cc2ccc(OC)c(Br)c2)C)=O)CCc2ccccc2O1 Cc1ccc(NC(=O)NCC2CC(=O)N(C(C)C)C2)cc1C(C)C C1(NC(Cc2cn(CC)nc2)=O)CC2(C(=O)NC34CCCC3CCC4)COC1C2 C(=O)(CC(C)(C)C(=O)OCC)N1CCCC(C)(CNC(C(C(=C)C)(C)C)=O)C1 N#Cc1c(NC(=O)Cc2csc(Nc3ccc(F)cc3)n2)cc(Br)cc1F C1(CC(N)=O)CCN1C(=O)C(=O)NCCONCCCC(=O)OC(C)(C)C.CC.C N1(C(C2(C)N(C(c3cncc(C)n3)=O)CC=C2)=O)CCC(O)C(C)(C)C1 Cc1cc(Cl)c(NC(CCC(C)C)c2nnnn2C2CCC(OC(C)(C)C)C2)s1 n1(CC)cccc1C(=O)NCCC1CC1C(=O)NCCc1cn(C)cn1 c1(C2(C)CNC(=O)N2)ccc(F)cc1Br.C(CCC(=O)OC(C)(C)C)SC C1(NC(c2cn(CCOC)nn2)=O)CCCN(C(c2ncc(F)cc2F)=O)C1C C1(C(N2CCN(CCOCC)CC2)=O)CC(=O)N(C)C1c1cnn(C)c1 c1(N(C(C)C)CCNc2ccc(C(C)(C)C)cc2)ccccc1[N+](=O)[O-] n1(SSCCNCC(N2CCC(CC(C)(C)C)CC2)C)ncccc1=O Cc1nn(C)c(C)c1C(C)C(=O)NC1CCCC1NC(c1n[nH]cc1F)=O C1(NC(=O)C=Cc2cscn2)CCN(C(=O)CC2(C(F)(F)F)CC2)CC1CO N1(CC2C(N)CC2)CCC(C(=O)NCC)CC1.C(=O)(C(C1CCC1)OC)N.C1(C)CC1 C(=O)(C#CC(C)(C)CNC(C1CC2(CCC2)C1)=O)N(CC(O)C1CC1)C C(CC(C)(C)C(=O)NCC(C)(C)OCC(=O)NC(C(C)C)c1nc[nH]n1)OC C1(NC(CC2(C(=O)OC)CC2)=O)CC(F)CN(C(c2ccc3c(c2)CC3)=O)C1 C(C(C(F)(F)F)N1CCN(C(=O)CO)CC1)NC(c1ccc(SCC)nc1)=O c1(CC(N2C(C(N3CCCC(N(C(C)=O)C)C3)=O)CCC2)=O)cc(Br)ccc1Cl N12CC3CCC(CC3C1)C2=O.Cn1nnc(=NCc2ccn(CC(F)(F)F)n2)[nH]1 c1(NC(C2CCC(CCNC(C(C)(C)SC)=O)C2)=O)nc(C(C)C)cc(C)n1 N1(C(C(C)(F)F)=O)CC2CCC1C1CN(C(=O)CN=c3ccc(C#N)c[nH]3)CC21 N1(C(c2nc3ccccc3s2)C(=O)NC2COC2)CCOC2(CCCSC2)C1 C=CCC(CNC(=O)CC1(OC)CCC1)C(=O)N1CC(NC(C)=O)C1 C(=O)(CC1COCc2ccccc21)NCC(C)N(C(c1cc(Cl)c(F)cc1O)=O)C Nc1nonc1C(=O)NC1CCC(CCNC(=O)CNC(c2cccs2)=O)C1 C(C(CNC(=O)C=CCOc1ccccc1)C(F)(F)F)NC(C1CCC(C)O1)=O C(=O)(C1CCc2ccccc21)Nc1n(-c2ccc(C)cc2)c2c(n1)cccc2 c1(C(C)NC2CC3CCC2CC3)cccc(N=[N+]=[N-])c1 Cc1ccc(SC2(C)CC2)cc1NC(=O)Nc1cc(Cl)cc(I)c1 c1(N(C(C(C)CC2CC2)=O)CCO)cc(N2CCN(S(C)(=O)=O)CC2)ccn1 N1(C(C(CC(=C)O)OC)=O)CCCCCCC1C(=O)NOCC(O)C(C)(C)C N1(C(C2N(C(c3ccc(N)c(F)n3)=O)CC(O)CC2)=O)CCN2C(=O)OCC2C1 Cc1nc2ccc(C(N3CC(NC(=O)C(C)(C)CCCO)C(C)C3)=O)cc2o1 C(c1sccc1Br)=CC(=O)NCC1CCCCN1C(=O)Cn1nccn1 Cc1cccc2c1OC(C(N1CCC3CN(C(c4nc(Cl)cs4)=O)CC3C1)=O)C2 N1(C(C(C)OCC2CCCO2)=O)CC(O)CC1CNC(c1ncc(F)cn1)=O c1(C(=O)NC2CC(C)(NC(C(C)CC3CC3)=O)C2)cc(S(C)(=O)=O)ccc1O Fc1cccc2c1CCCC2NCc1cnc2n1CCCCC2 C(c1c(C)nn(C)c1Cl)=CC(=O)NC1CC(NC(C2(COC)CCC2)=O)C1 CCCC(C)CC(=O)N1CC(C2(NC(c3ccc(=NC)[nH]c3)=O)CC2)C1 c1(OC)ccc(C=CC(N2CC(CCNC(C3CCC(C)(C)O3)=O)C2)=O)cc1O N1(C(CC(CC)C)=O)CCCC(C)(NC(c2cc(OC)ccn2)=O)C1 O=C1CC(CC(=O)N2CCOC(CNC(C3(N4CCOCC4)CC3)=O)C2)=NN1 C12(CC(=O)NC3CC(C)CN(C(=O)CS(N)(=O)=O)C3)CCCN1CCC2 C1(NC(C2CC3C=CC2CC3)=O)COCCN(C(C2CC3(CCC3)CO2)=O)C1 C(=O)(CC1=CCCCC1)N1C2CC(CNC(=O)CSCc3ccncc3)C1CC2 N1(CC(=O)N(C(C(=O)OC)C)C)CCN(C(=O)CCc2cc(C)cs2)CC1 C#CCC(O)C(=O)NCC(F)CNC(c1ccc(-n2[nH]c(O)nc2=O)cc1)=O C1(CNC(c2ccc(C(N)=O)[nH]2)=O)CN(C(c2ccnc(S)c2)=O)CC12CC2 C1(C2(N)CCC2)(C(=O)NC(c2cccc(Cl)c2)CC)CC1 CC1CCCN(C(=O)C(C2CCN(C(c3ccc(-c4cc[nH]n4)o3)=O)C2)C)C1 CCCC(C(=O)NCC(CC)NC(C12CCCN(CC1)C2)=O)S(N)(=O)=O N1(C(C(=O)NCCCOC)=O)CC(OC(C)(C)C)C(F)(F)C1 C1(C(N2CC(NC(c3cccc(C)c3C)=O)C(C)CC2)=O)CCCC2CCCN12 C#CC(CC)(CC)NC(=O)C(CNC(=O)CCC1CC1(C)C)N(C)C C1(O)(CC=C)CCN(C(=O)CCN(C)C(c2ccncc2NC)=O)CC1 CC1(C)CN(C(C2CCC(=O)N2)=O)CCC1C(=O)NC1CCCCC1 CCC(CC)(CC(=O)OC)C(=O)NCCCCCCNC(=O)CN1CCNC1=O c1(C(=O)NC2C(N(C(=O)CC(=O)NC3CC3)C)CC2)cnn2c(Cl)cccc12 c1(N(CCCN(C)C(C2OCC2(C)C)=O)C)ncnc2cnccc12 N1(C(C=CC(C)NC(=O)CN2CCCC2)=O)CCC(O)CC1C N1(C(c2nc(C)oc2C)=O)CCC(C2(NC(=O)CC3CC3C(F)(F)F)CC2)CC1 c1(CNC(C2C(C)(C)C2(C)C)c2n(CCC)nnn2)c(Br)c(CC)nn1C Fc1cc(CN2CCOC(c3n[nH]c(C(F)(F)F)n3)C2)c2ncccc2c1 n1(CCC)nc(C)c(N(C(=O)CCOCCNC(=O)C(F)C(C)C)C)c1C N1(SCC)OCC(NC(=O)C(=O)NC2CC(OC(C)(C)C)C2(C)C)C1=O c1(C(N2CCCC(O)(CNC(CCOCC#C)=O)C2)=O)ccc(O)c(C)c1C CN=c1cc(-c2nc(CC3CCOCC3)nn2Cc2ccccc2)cc[nH]1 C1(C(=O)Nc2ccc(CC)cc2)CCCN(C(=O)C(C)(C)CN(C)C)C1CC c1(C(C)C)cc(C(=O)NCC=CCNC(=O)C(O)C(C)C)nn1-c1ccccc1 CCC(CC)CCC(=O)NCC1CN(C(c2ccc(O)c(CO)c2)=O)CC1C c1(CC)cn2c(n1)CCC(C(N1CCN(C(c3cc(C4CC4)cs3)=O)CC1)=O)C2 C1(NC(C2(C)CC(C)=C(C)CC2)=O)CC(N=c2cc(C(F)(F)F)nc(Cl)[nH]2)C1 N1(C(C2(CN(C)C)CC2)=O)C2CCC1CN(C(=O)CC1CCCC1O)C2 C1(NC(C2(C)CCCC2(F)F)=O)CC12CCN(C(c1cnc(C3CC3)s1)=O)CC2 C(=O)(CCCC(=O)N(C)C)N1C(CNC(c2c(C)n(C)nc2)=O)C=CC1 Cc1cc(NC(C2CC(C)N2C(=O)C(N2CCCCC2)C)=O)cnc1O C1(C(=O)NC(COC)(C)CO)CCC2(CC2)N1C(=O)CCc1csnn1 CN1C(=O)OCC1C(N1CCN(CCCCCNC(=O)CSC2CC2)CC1)=O N1(C(c2cc(CC)sn2)=O)CC2CCC1CN(C(=O)CC1CC(F)(F)C1)C2 C(CCn1c(N2CCC(C)(C(N)=O)C2)nnc1-c1n[nH]c(C)n1)(C(C)C)OC C1(CNC(C(c2cccs2)OC)=O)(NC(=O)CNC(=O)CNC(C)=O)CCOC1 C1(NC(C2C=CCCC2)=O)CCCCN(C(c2ccnc(S)c2)=O)C1 c1(C(=O)NCC2N(CC(C)C)CCCC2)cc(Br)cc2c1OCCC2=O Cc1cc(C(=O)OCCc2cccc(C)c2)ncn1 c1(OC)nc(C(C)C)ccc1C(=O)NNC(=O)NCN1CCCC1 C1(OC)(CNC(c2ccc(Cl)nc2N)=O)CCN(C(=O)CC2COCC(C)O2)CC1 C1(NC(=O)NCCCNc2ccc(O)cc2)CCCCC1c1cccnc1 C(=O)(C(C)C(C)NC(=O)C=CCCC)NCCOCCC#C Cc1cccc(C(N2CC(NC(c3cccc(-c4ccco4)c3)=O)C(F)C2)=O)c1 C1(C)(CNC(CCC#CC)=O)COCCN(C(c2sc(C)cc2OC)=O)C1 c1(CC)ccc(CC(=O)N(CC(C)CNC(c2cnccc2C)=O)CC)cc1 C(CCC(=O)NCCN(C1CCCCC1)C(=O)C(C)c1cc[nH]n1)SC C1(OC)COCCC1CC(=O)NCC(=O)N(C)CCN1CCOCC1 c1(C(N2C3C(CNC(C4CCCCS4)=O)C(C3)C2)=O)nccc2occc12 C12(NC(C(C)C#N)=O)CCCC1CN(C(c1ccc(OCC(F)F)cc1)=O)C2 c1(C(N2CCC(O)(CNC(C(CCC#C)O)=O)C2)=O)ncnc2ccsc12 CCC(CC)CC(=O)N1CCC(C(=O)N(C)CC23CCC(CC2)C3)C1CC c1(C(N2CCC(N(C(=O)C3=CCN(C)C3)CCC)C2)=O)cncc2ccccc12 C1(NC(=O)COCCCF)CCN(C(=O)Cc2ccco2)C1c1ccccc1 Cc1cc(C(=O)NC(C2CCN(C(=O)C=CC(F)(F)F)C2)(C)C)cc(C)c1Cl CC1CC(NC(C2CCCN2C)=O)CN(C(c2cn(C3COC3)nn2)=O)C1 C1(C(N(CC(CNC(C(C)OC(C)(C)C)=O)O)C)=O)CCCOCC1 C(=O)(C(F)C(=O)NCc1nc(C(=O)N(CCCCO)C)co1)OCC c1(C(C)=O)c(NCCC2CC(NC(=O)CS(N)(=O)=O)C2)nc(C)nc1Cl CC1CN(C(=O)CCc2c(N)n(C)c(=O)n(C)c2=O)CC(C)N1CC#N C(C(C)(O)CC(=O)NCC1(CNC(=O)C(c2ccnn2C)C)CC1)OC c1(CN(C(C(=O)NCc2nc(COC)on2)(C)C)C)ccc(C)cc1 C1(NC(c2ccc(C)n2C)=O)CN(C(=O)C(F)(F)c2ccnn2C)CC12CC2 C1(C(=O)NCc2c(C(N(CCCCCCC)C)=O)cccn2)CC2(CCC2O)C1 Cc1cnc(CO)c(C2CCN(C(=O)NCC(C3CC3)C3CC3)CC2)c1 CCN=C(NCC(C)(C)C(F)F)N1CCC2(CCCC2)C1 C1(C2CCN(CCN(CCC)C)C2)COCCN1C(=O)OCC C1(CNC(C2CN(C(=O)NC)C2)=O)CCCN(C(c2cccc(O)n2)=O)CC1 CCC(C)C(C)C(=O)NCCC1CCN(C(=O)Cc2cncn2C)CC1 c1(C(=O)OCC)cc(=NC(C)(C)CNC(=O)CCOCC2CCCO2)[nH]cn1 c1(C(=O)NCC2CN(C(C3(C#N)CCC3)=O)CC23CC3)ccn2cnnc2c1 C=CCCCCCCCC(C(=O)NC1CCC1)N1CC(C)Oc2cc(Cl)ccc21 c1(C(=O)NC2CC(C)(NC(CCCCC=C)=O)C2)cc2ccc(F)cc2nc1C Cc1cc(Br)ccc1-c1noc(C(C2CCC2NC(=O)OC(C)(C)C)C2CC2)n1 C1(NC(c2c(C)n(C)cn2)=O)CCC2(CC1)CN(C(C1CNC(=O)N1)=O)CCO2 CC12CC(C1)C(=O)N2.C1(CNC(C23CC(C2)C3)=O)C(CO)C1(C)C c1(C(=O)NC2CC3(C(NC(CC4CC(OC)C4)=O)C3)C2)cccc2[nH]cc(Cl)c12 C1(CC)CCCN(CC(=O)NC(C)CCCNC(=O)CCc2cncnc2)C1 C1(C(N2CCCCC2c2cn(Cc3cc(Br)cs3)nn2)=O)C(Cl)(Cl)C12CC2 CC1(C)COC(CCC(=O)NCC2(NC(=O)CCCc3ccc(F)cc3)CC2)C1 N1(C(C(CCCC)N(C)C)=O)CCC2(C1)CN(C(c1nc(C)n(C)c1C)=O)C2 C=Cc1ccc(C(=O)CNC2N(C(C3CC4(CCC4)CO3)=O)CCC2(C)C)cc1 c1(C(=O)NCCC2(NC(C(C)OCC3CCCO3)=O)CC2)ccc(C(N)=O)nc1 C1(CC(=O)NCCC(C)N(C(=O)CCC2CCCO2)C)C=CCCC1 c1(C(N2CCC3CN(C(C4=NNC(=O)C4)=O)CC32)=O)cc(O)cc2ccccc12 c1(C(=O)NCCNC(C(C)NC(=O)OC(C)(C)C)=O)ccnc2[nH]c(O)nc12 C1(CNC(C2CC2CNC(=O)OC(C)(C)C)=O)OCC2CCC1C2 C1(CCC)C(=O)NCCN1CC(=O)Nc1cccc(F)c1 Cc1cc(C(N2CC(F)(c3cn(-c4ccc(C(C)C)cc4)nn3)C2)=O)ccc1Cl c1(NCCCCOCC)ncc(S(=O)(=O)N2CCCC3(CCSCC3)C2)cc1Cl N1(C(c2ccc(C)cc2C)=O)CC2(CCCC2)C1C(=O)NCC(O)C(F)F C(CCc1ccccc1)(C(=O)O)NCc1ccc(C(C)(C)C)cc1 C1(CNC(C=CC)=O)CCCCN1C(c1cc(-c2cccc(Cl)c2)ns1)=O C12(CNC(c3cc(C)n(C)c3)=O)CC(CCO1)N(C(=O)CC1(C(F)(F)F)CC1)C2 C(=O)(C1=CCCC1)N(CCCNC(C1CC(C)(C)C1C(F)(F)F)=O)CC c1(-n2c(-c3cc(O)ncc3)nc(-c3ccccc3Br)n2)ccc2c(c1)CCC2 O=C(C#CC1CCOC1)NCC1(O)CC(NC(C2Cc3nccn3C2)=O)C1 CON1CCC(C(=O)NC23CCN(C(C4(O)COC4)=O)CC2C3)CC1 C(=O)(C(S(C)(=O)=O)C1CC1)NCC(CC)(CC)NC(=O)CC1CC2CCC1O2 c1(C(=O)NCc2c(-c3c(C)cncc3)c[nH]n2)ccc(Br)c(Cl)c1F c1(-n2c(-c3cc(C4CCOC4)[nH]n3)nc(CCOC)n2)ccc(C)c(F)c1 N#Cc1ccc(=NCC2(F)CC(NC(c3sccc3Cl)=O)C2)[nH]n1 c1(C(=O)OC(c2nnc(C3CCC3)o2)C)ccc(Cl)c2cccnc12 N1(C(C2CC(=O)NCC2)=O)CC2CCN(C(c3cc(Br)cnc3Br)=O)C2C1 CN1CC(CO)N(N2CCC(O)(C(F)(F)F)CC2)CC1=O N1(C(C2(C(C)C)COC2)=O)CCCN(CCNC(=O)CC2CC2C)CC1 c1(C(N2CC(O)(CNC(C3(OCC)CCSCC3)=O)C2)=O)cc(N)cc(O)c1F c1(C(=O)OC)cc([N+](=O)[O-])ccc1NCC(F)C(F)(F)F N(C(=NCc1ccc(C(N)=O)cc1)N(C)Cc1ccn(C)n1)C(CC)CC C1(CCNC(CC=C)=O)CN(C(c2nc(C(F)(F)F)sc2C)=O)CC1C C=CC1CN(C(C2CN(C(=O)C(=O)NC(C)C)CC2C)=O)CC1O c1(COCC(C2CC2)NC(C)CN2CCCCC2)cccc(CO)c1 C1(NC(COCCCC#C)=O)CC2CCC1CN2C(=O)C(c1ccc(C)o1)C N1(C(c2n(C)ccn2)=O)CC2(NC(c3cn4ccnc4s3)=O)CCC1C2 c1(C(NCC2N(C(c3cccc(Cl)c3O)=O)CCOC2)CCO)cccc2ccncc12 N1(C(c2cccc(F)c2F)=O)CC=C(C(=O)N2Cc3ccncc3C2)CC1 C1(O)(CCNC(C2(C=C)CC2)=O)CCN(C(=O)CC2CC(=O)NC2=O)C1 N1(C(Cn2c(C)ncc2)=O)CCOCC(CNC(=O)C(C)S(C)(=O)=O)C1 c1(C(N)=O)ccnc(C(=O)NCCC2CCCN2C(=O)C(c2ccccc2)F)c1 C(c1cc(OC)ccc1OC)=CC(=O)NCCN(C(C(C)OCC)=O)C1CC1 c1(NC(C2C(NC(c3cc(CC)no3)=O)C2)=O)cccc(NC(C)=O)c1 C(=O)(CC(C)(C)C(F)F)NC(C(=O)NC(c1c(C)nc(C)[nH]1)C)c1ccoc1 C(=O)(C(CN=[N+]=[N-])OC)N1CC(COC)(NC(c2cc(OC)n[nH]2)=O)C1 c1(OC)ccc(OC)c2c1CCN(C(c1cc(C)ncn1)C(=O)NC1CC1)C2C C1(NC(Cc2cc(C)sc2C)=O)CC(F)CN(C(c2ccc(C(C)O)cc2)=O)C1 c1(CC(=O)NC(CCN(C(c2ccc(C(C)=O)cn2)=O)C)C)cccc(C)c1F c1(OC)cc(CNC(C2CC(F)CN(C(=O)C(C3CC3)SC)C2)=O)ccc1C c1(C(N2CC(NC(CN(C)CC)=O)C2)=O)ccc(C)nc1OC c1(C(=O)NCCCC(O)C(=O)N2CC3CC3C2)cnn2ccc(Cl)c(F)c12 CCCC(CC(C)C)C(=O)NCc1ccc(Cl)o1 Cc1cc(C(N2CC(NC(=O)CC3CC(F)C3)CC23CCC3)=O)c(N)c(Cl)c1 Cc1nn(CC(N2CCOC(c3ncc[nH]3)C2)=O)cc1Br C12(NC(CS(=O)(=O)N(CC)CC)=O)CCCN(C(=O)C(C)NC(N)=O)CC1C2 C1(NC(CSC(C)(C)C)=O)CCN(C(=O)CCCc2ccccc2)CC1F C1(C(=O)NC(C(=O)NC2CC(CC(=O)OC)C2)C2CC2)CC(=O)CCO1 C1(N(CC(=O)OC)C)CCN(C(c2cccc(N3CCNC3=O)c2)=O)CC1 c1(C(=O)OCC(c2cccs2)=O)ccc2c(c1)OC(F)(F)CN2 CC(C)C(N=[N+]=[N-])C(=O)N1CC2CCC(C1)N2C(=O)Cc1cc(F)ccc1Cl N1(C(C=CC=CC)=O)CC(NC(=O)Cc2cnsc2)C(c2ccc(F)cc2)C1 C1(CC)CN(c2cc(N3CCC(CO)CC3)ncn2)CC1NC(=O)N(C)C N1(C(C(Cc2cc[nH]n2)NC(C(C)=C2CCC2)=O)=O)CC2C(C)C2C1 c1(CCNC(C2CC(C(F)(F)F)C2)=O)ccnc(C(F)(F)F)n1.C12CCN1C2 C1(C#N)(C(=O)NCCC2(O)CN(C(Cc3nc(C)oc3)=O)C2)CCCC1 N(C1=C(C(=O)O)CCC1)C(C1C(CC(N2CCN(C)CC2)C)N(C)CC1)C(=O)OC C1(NC(C(C)OCC)=O)CCCN(C(c2csc(C(N)=O)n2)=O)CC1 N1(C(c2c(CC)[nH]nc2Cl)=O)CCC2(CCCC2NC(=O)C=CC(=O)NC2CC2)C1 c1(OCC(=O)NC2(CC)CCN(C(=O)C(C)c3cc[nH]n3)C2)ccc(F)c(F)c1 C1(NC(c2nc(C)oc2C)=O)CC2CCC1(NC(=O)CC1(C)OCCO1)C2 N1(C(c2cc(CC)oc2C)=O)CCC(NC(=O)CCCc2sccc2C)C(C)C1 C12(NC(C(CC3CC3)NC(C3CC(C)(C)C3)=O)=O)CCN(CC1)C2 CC1=CCC(C)(NC(C2(CNC(C3C4CCCC34)=O)CC2)=O)CC1 C1(C(=O)NCCN(C(=O)C(C)(C)Cc2ccc(O)cc2)C)CCC(C(N)=O)CC1 N1(C(c2c(OC)cccn2)=O)CC2(CCCC2NC(c2nnc(C)s2)=O)C1 O=CN1CCN(C(=O)CC2CCN(C(=O)CCOc3cc(Cl)cc(Cl)c3)C2)CC1 CCC(O)CCNC(C1(CNC(=O)C(C2CCOCC2)C)CCC1)=O N1(C(CC(C)CN(C)C)=O)CC(NC(c2cn3c(n2)SCC3)=O)CCC(O)C1 C1(C(N(CC(CN(C(c2ncn(C(C)C)n2)=O)C)O)C)=O)CCC2C(C1)C2(F)F c1(C(=O)NCC2CC(NC(c3ccc(Cl)s3)=O)C2)ccc(SC2CC2)c(F)c1 N1(c2nnc(C)s2)CCCC(CCCNC(=O)CC23COCC(C2)C3)CC1 C(=O)(C1=NNC(=O)C1)NCC#CC(=O)NC1(CC(=O)OC)CCC1 C1(C(=O)NCCC2N(C)CCCC2)CCN(C(c2cncn(C)c2=O)=O)CC1O c1(C(=O)NC2C(CNC(C(CC#C)C3CC3)=O)CCC2)ccc(C)cc1CC c1(CN(C(c2c(SC)cc[nH]2)=O)C)ccc2c(c1)CCC2 C1(NC(C2(CC(C)C)CC2)=O)CCN(C(=O)CN2CCCOC2=O)CC(O)C1 c1(C(=O)NC(c2ccn(C)n2)CC)cnc(CNC(c2sc(O)nc2C)=O)nc1 C(=O)(C(COC)CC(C)C)NCCCC(CCC)NC(c1onc(Br)c1C)=O N1(C(c2ccc(OC)cc2)C(=O)NCCSC)CCC(S(=O)(=O)C(C)C)C1 C1(NC(C2CC=C(C)CC2)=O)CC2CC1N(C(c1cc(Cl)ccc1O)=O)C2 C1(C(C)(C)C)(CNC(=O)CC2CCS(=O)(=O)C2)CCN(C(=O)C2=COCC2)C1 c1(C(N2C(CCNC(C(COCC)N=[N+]=[N-])=O)CCC2)=O)cc2cccnc2[nH]1 C(=O)(CC(C)C(=O)N1CC(CNC(c2cc(F)ccc2C)=O)C1)OC N1(C(CNC(C(COCC)n2cc(COC)nn2)=O)C)CCOC2(CCCC2)C1 C1(N(C(c2ccc(COC)cc2)C(=O)NCCCC)C)CCCC(C)(C)C1 Cc1noc2cc(C(=O)NC(C3CCCN3C(c3cnc(O)s3)=O)C)ccc12 C(C(C)(CC(C)C)NC(=O)CCC1CC1(F)F)NC(c1cnc(NC(C)=O)o1)=O N1(C(CC(CC)O)=O)CC(NC(=O)Cn2ncn(C)c2=O)C(C)(C)C1 N1(C(CCN(C(C2C(OC)(OC)CC2)=O)C2CC2)=O)CCCC(C2(C)CC2)C1 N1(C(C2=C(C)CCCC2)=O)CCC2CC1CN(C(C1CCC(CO)CC1)=O)C2 CC(C)C(F)(F)CC(=O)N(C)CCC1CCN(C(c2cnc3n2CCS3)=O)CC1 C=CCCCCCCC(=O)C1=CC=C(F)C=CC(N2CCCCC2)CC1 C12(NCC(=O)NCC3N(C(CN4C(C)CCC4)=O)CC3)CC3CC1C2C3 N1(C(CCC(CC)C)=O)CCn2ncc(CN(C(=O)CC3COC(=O)C3)C)c2C1 c1(SC)ccc(C(=O)NN2CCCCC2C)cc1.c12cn(nn1)C1CCN(C1)C2 N1(C(=O)NCCCC)CCN(C(c2noc(C3(c4cccs4)CC3)n2)=O)CC1 C1(CNC(CCOC)=O)CN(C(c2cc(F)cc(Cl)c2Cl)=O)CCC12CCC2 N1(C(CC(CC#C)NC(c2occ3c2CCC3)=O)=O)CCSCC(C)C1 N1(C(c2c(CC)cccc2)=O)CC(F)(F)CC1C(=O)N(CCC(C)C)CCC(C)C C1(C(=O)NCCC2(O)CCCCC2)CC(O)CN1C(=O)Cc1cccc(O)c1 C(=O)(C(CCF)NC(c1cnc(C2CC2)o1)=O)N1CCC(=C)C1 CCC(C)C(C(=O)NC(C)CCCC(=O)NC1(C)CCCCC1)OC c1(C(=O)NCCC2CCC(NC(CCOC)=O)C2)cc(N(C)C)cc(C#N)c1 n1(CC(=O)NC(c2occc2C)CC)cc(C2CCCC2)nn1 c1(C(=O)OC(Cc2c(C)non2)C(=C(Cl)Cl)C(=O)ON)c(-n2cccc2)sc(C)c1C Cc1cc(S(N)(=O)=O)cc(C(=O)NC(C)C(C)NC(=O)CN2CCCCC2)c1C CCC(C)CCCCC(=O)NC1(CCO)CN(C(c2cc(Br)n(C)c2)=O)C1 c1(OC)nn(C)cc1C(=O)N(C)CC1CC(F)CN1C(c1nc(Cl)sc1C)=O CC(C)CC(C(=O)N1CC2(CCC2)CC1C(=O)NC12CC(F)(C1)C2)C(N)=O C1(NC(CC(C(C)C)OCC)=O)CN(C(c2ccc(C#N)o2)=O)CC12CCCC2 C1(CCC(N2CCC(C(C)C)C2)=O)CCCN(C(C2C3CN(C)CC23)=O)C1 Cc1ccc(=N)[nH]c1C(N1CCC(C)(CCNC(C2CC23CCCC3)=O)C1)=O CCC(CC(=O)NCC12CC(CO1)N(C(=O)C1=NOCC1)C2)C(F)F N1(C(=O)OC(C)(C)C)CCC(C(N2CCN(CC(O)C3CC3)CC2)=O)(C(F)F)C1 c1(Nc2nccc(CNC)n2)n[nH]c2c1CCC(F)(F)C2 C1(C(=O)NCC(C)CC2CC2)CCC=CC1NC(=O)CC1CCCC(=O)C1 C(=O)(CC(C)(C)C(=O)N1CC(CC(C)NC(=O)C=CBr)C1)OC c1(OCC(C)C)ccc2[nH]c(C)c(C(=O)NCCNC(C34CC(O)C3C4)=O)c2c1 C1(NC(c2cc(C(C)C)c(Br)cc2)=O)CC12CCN(C(C1CCCOC1)=O)CC2 CC1=NOC(C)(C(=O)NC(C)CCCNC(C2CC2c2ccc(OC)nc2)=O)C1 C(CC(=O)NC1CCCC(CNC(=O)COc2ccsn2)C1)(C1=CCCC1)OC CC(CC(=O)N1CCC(CNC(C2(C(C)(C)C)CCC2)=O)C12CC2)C(C)(C)C c1(NC(CC2OCCN(C(C3=CCCC3C)=O)C2)=O)cccc(C#N)c1F c1(C(=O)NCCn2cc(CNC(C(C)(C)SC)=O)nn2)cn2cccnc2n1 CCCC(C(O)C(=O)N1CC(N(C)CCOC)C1)NC(=O)Cc1csc(C)c1 C(=O)(C(C#N)C(C)(C)C)NCC1(CNC(C(C(C)C)n2ccnc2)=O)CC1 C1(NC(c2nnc(C)o2)=O)CCN(C(=O)C(C)Cc2ccc(Br)cc2)CC1O C1(CNC(=O)Cc2ccccc2F)CN(C(c2csnn2)=O)CCC12CCOC2 c1(C(=O)OCC)nnc(SC)nc1N1CCC1CN(C)C.c1(C)cccnc1C N1(C(C(Cn2ccc(C)n2)C)=O)CC(C)CN(C(=O)C(C)CC2CCC2)CC1C c1(C(=O)NCC(C)NC(=O)C(N2CCC(O)CC2)C)c(F)ccc(Br)c1F c1(OC)cc(F)c(F)cc1NCc1cc(O)cc(Br)c1 C(c1cccc(CO)c1)=CC(N1CC(NCc2cccc(Br)c2)C2(CC2)C1)=O C1(C(=O)NCC2(O)CCN(C(Cn3c(C)nnn3)=O)CC2)CCc2nnnn2C1 c1(C(=O)OC)csc(C(=O)OCC(Cc2ccccc2)C2CC2)c1 C(=O)(C1=COCCC1)NC1CN(C(C2(CC#C)CCCO2)=O)CC1CCC C1(NC(C(N(C(CCC(=C)Cl)=O)C)C2CC2)=O)CCOC(C)(CC)C1 N(C1CCCc2ccoc21)c1nccc(N(C)CC2CCCCC2)n1 CC1CCc2[nH]nc(C(=O)NC3CCN(C(C4CS(=O)(=O)C4)=O)CC3C)c2C1 c1(NC(C2C(C(=O)OC)C2)=O)cc(C)c(F)cc1OC.N12CCC1(C)C2=O c1(C(=O)NC2C(CNC(CCC3(C)CC3)=O)CCCC2)ccc2c(c1)NCC2 c1(N2CCCC(O)CC2)nc(N2CCOCC3(CCC3)C2)c2ccsc2n1 Cc1c(C(N2CCC(F)(C(=O)NCC3COCC3(C)C)C2)=O)cccc1F Cc1cnc(C(=O)NCCC2CCN(C(C3(F)CCC3)=O)CC2)cn1 C(=O)(C1=C(Cl)CCC1)NC(C1C(C(N2CC(COC)C2(C)C)=O)C1)C c1(C(=O)NCC2(C)CCN(C(Cc3nnc(C)o3)=O)C2)ccc(F)cc1Br c1(C(c2nnnn2C2(C)CC2)N)c2c(nn1C)CCCC2.C(C(C)OC(C)(C)C)SC C1(CNC(CCC#C)=O)CCC2(CCN(C(=O)C(F)C(F)(F)F)CC2)CO1 c1(C(N2CC(NC(CCCN(C(C)=O)C)=O)C(C)C2)=O)cc2occc2s1 C12(C(=O)NCN3C(=O)CN(C(=O)CN4CCC4)CCC3)CC3CC1(CO)CC3C2 c1(C(=O)NCC2(C)C(NC(COCC(=C)C)=O)CCC2)cc(OC)cnc1F c1(C(N2CC(CNC(CSc3n(C)nnn3)=O)C3C2C3)=O)nc2c(s1)COCC2 c1(C(CN(C(c2c(C)sc(O)n2)=O)C)O)ccc(S(C)(=O)=O)cc1 CC(CNC(=O)CC1(C)CCC1)C(F)C(=O)Nc1cncc(C2CC2)c1 N1(C(CC(COC)C)=O)CCC(C)(NC(C(=O)NC2CC(CO)CCC2)=O)CC1 c1(OCOC)ccc(C(=O)NCC(C)=O)c2[nH]c(CC(=O)OC)cc12 C1(OC)CCCC(CNC(=O)CN(C)C(c2ccc(C(F)F)o2)=O)C1 C1(NC(C(C=C)O)=O)CCCC(NC(c2cc(Sc3ccccc3)nn2C)=O)C1 c1(C(=O)NC2(CNC(Cc3cnc(C)[nH]3)=O)CCCCC2)cc2sccc2n1C C(C)(CCC(=O)NC1CC2(C1)CC2NC(=O)CC1(N)CCCC1)OC C12(CNC(c3cccc(NC(=O)OCCC(C)C)c3)=O)CCCN1CCC2 Cn1ccc(=O)c(C(=O)NC2CCC(CNC(C3CC4(CCC4)C3)=O)CC2)c1 c1(C(C)(C)C(=O)NCC2CCCC2NC(=O)C(F)=CCCF)ccccc1Cl c1(C(N2C3(CNC(C(C)(C)OCC)=O)CC(C2)C3)=O)cc(C)nc(Cl)c1N N1(C(C(C)OCC=C)=O)CC(C(=O)NCC2CCC3(CC3)CO2)C2(CC2)C1 C(C(C)CC(=O)NC1CC(F)(CNC(c2coc(-c3ccccc3)n2)=O)C1)OC C1(C2CCCN(C(=O)C=C3CC3)C2)(NC(Cc2ncc(C)s2)=O)CC1 C1(NC(=O)OC(C)(C)C)CC2CN(C(C3(C#N)CC34CCC4)=O)CC12 N1(C(Cn2c(C)nnn2)=O)CC2(CCN(C(=O)C=C3CCN(C)CC3)C2)C1 C1(CCCC(=O)NN(CC(=O)NCCOCCCNC(N)=O)C)CCCC(=O)N1 Cc1ccc(CC(N2CC3CC2C3CNC(=O)CC(=O)N(C)C)=O)cc1 c1(C(CC)(C)C)ccc(CNC2(C)CCN(C(C3COCC34CC4)=O)C2)cc1 c1(C(=O)NC2CN(C(c3cnc(SC)s3)=O)CC2F)cc2ncccc2[nH]1 CC1CN(C(C2(C)CC(O)CN2C)=O)CC(C)N(C(C2CNC(=O)CC2C)=O)C1 C1(C(N2CC(CCC=C)(C(N3CCC(CC4CC4)C3)=O)C2)=O)CC2CCCC2C1 CC(C)(CC(F)C(=O)N1CC(O)CC(C)(C)C1)NC(C1CCCOCC1)=O C1(CC(N2CC3(CCN(C(C4C(C)C4)=O)C3)C2)=O)CCC2(CC1)OCCO2 C1(NC(N(C2CC2)Cc2cn(C)nc2)=O)CC(N)CC(C)(C)O1 c1(C(=O)NC(C2CN(C(c3cnc(O)c(F)c3)=O)CCO2)C)cc2cscc2s1 C=CCC(C(=O)NCC1(CNC(C2CC(O)CN2C)=O)CCC1)c1ccccc1 C1(NC(C2CCC3(CC3)N2C(=O)CC2CC(=O)NC2=O)=O)CCCN2CCCC12 O=C(NOCc1ccccc1)C(O)CNC(c1ccc(C2CC2)o1)=O CC1Oc2c(C(=O)NC3CC4(CCC(C)(C)CC4)C3)cccc2C1C Cc1cc(Cl)cc(C(=O)NCC(O)CN(C(=O)CC2CCCC2)C)c1O C12(CNC(c3ccc(C(C)C)s3)=O)CC(NC(C3CCCC3O)=O)(C1)C(C)O2 C1(CC(=O)NCCC(C)NC(c2ccc(C(C)(C)C)cn2)=O)OCCOC1(C)C N1(C(C2C(=O)OCC2)=O)CCCC(N(C(=O)CCn2cccn2)CC2CC2)C1 N1(CCO)CC2OCCCC2(NC(=O)CCN2CCN(c3ncccn3)CC2)C1 c1(C(=O)NC(C2CN(C(C3C(=C)C3)=O)C2)C)ocnc1-c1ccccc1 N1(C(Cc2nc(C)sc2)=O)CC(CC(=O)NC(=O)CC2CN(C(C)C)C2)CC1C Cc1ccc2nsnc2c1C(=O)NCC12CC1CN(C(c1cnncc1O)=O)C2 Cc1ccccc1C(=O)NCCCCCNC(C1CCCS1)=O FCCN=C(NC1CC1)NC1CC1c1ccc(-n2cccn2)cc1 C1(OC)CC(CCNC(=O)C(C)NC(C)=O)N(C(c2cc(C)n(C(F)F)n2)=O)C1 CCCC(C(=O)NC1(CNC(=O)CN2CCCC2CO)CC1)N(C)C Clc1ccc(C2=CCN(c3cccnn3)CC2)cc1 Cc1cc(F)ccc1CNC(C1CCCC(NC(=O)CSc2ccccn2)C1)=O CN1CCN(CC(=O)NC2CCC2NC(c2ccn(C3CC3)n2)=O)CC1=O C1(NC(=O)NC(C2(CSC)CCCC2)=O)CCN(C(=O)C(=O)NC2CC2)C1 C1(C(C(=O)NC(C2CCCC2)C#C)C)CCN(C(=O)Cc2cncn2C)C1 CN1CC=C(CC(=O)N(C2(C(=O)NC3(C4CCCO4)CC3)CC2)C)CC1 c1(CC)ccc(C(=O)NCC2(C)CCC(NC(=O)CNC(=O)CN(C)C)C2)nc1 c1(OC)cccc(N(C(=O)C(C)CNC(=O)Cc2ccoc2)C)c1 c1(C(N2CCC(CNC(C3C(SC)CCC3)=O)C2)=O)cc2ccccc2[nH]1 C1(CC)CN(C(=O)CCSCC(N)=O)CCN1C(C1CC2CC2C1)=O C=CCCCC(C)(C)C(=O)N1CCC(C(N2CCOC3COCC23)=O)C1 CC(C)(O)C(F)(F)C(=O)N1CC2CC(NC(c3csc(Cl)c3Cl)=O)CC2C1 C1(CNC(C)=O)CN(C(C2CC(=O)N(c3ccc(F)cc3)C2)=O)CCCO1 c1(OC)ccc(CN(C)C(C2CCCN(C(=O)CO)CC2)=O)cc1OCCCl C1(O)(CNC(=O)C(Cl)=CCl)CCCN(C(c2ccc(OC(F)(F)F)nc2)=O)C1 N1(c2c(C)cncn2)CCCC2C(NC(c3ccc(C(N)=O)nc3)=O)C12 C1(C(=O)NCc2cnns2)(CNC(C2C(=C)C2)=O)CC=CC1 Cc1ccncc1C(=O)NC(c1nocc1C(=O)NC1(C(C)(F)F)CCC1)C C(c1ccc([N+](=O)[O-])s1)=CC(=O)N(CC(C)O)CCNC(C(C1CC1)OC)=O C1(NC(C2(C)CC(=C)C2)=O)CC2CCC(C1C)N2C(c1csc(=NC2CC2)[nH]1)=O CCC(C(=O)N1CCC(CN(C)C(C2CC(n3cnnc3)C2)=O)C1)OC1CCCC1 C=C(C)C1OCCC1CNC(=O)C(Cn1ccnn1)NC(=O)COc1cc(C)on1 C(=O)(CCCC(C)(C)C#N)NC1CCN(C(c2ccc(OCC)nc2)=O)CC1C N1(C(C(=O)NC2Cc3c(nc(C)s3)CC2)=O)CC2(C)CN(C)CC2(C)C1 Cc1ccc(Cl)c(O)c1C(N1CCC(C(C)NC(c2cc(Cl)cs2)=O)CC1)=O C1(CNC(CC(CC)C)=O)CCN(C(=O)Cc2ccnc(OC)c2)C12CCC2 Cc1ccccc1OCCCC(=O)N(CCNC(=O)CS(N)(=O)=O)C1CC1 N1(C(C2CCC(CCCCC)O2)=O)CCOC(CNC(C2(C(=O)NC)CC2)=O)C1 N1(C(C(C)SC(C)C)=O)CCC2(C1)CN(C(c1ccccc1CC(F)(F)F)=O)C2 CC1CN(C(=O)Cc2ccccc2)CCC1CNC(c1csc(CO)n1)=O C1(NC(COCCOCC#C)=O)CN(C(=O)C(C)(C)c2cccnc2)CC1C CC1(C(=O)NC2CC2C(F)(F)F)CC(O)(CO)C1 Cc1cccc2c1ccn2CC(N1CCN(C(=O)C=C(Cl)Cl)C(CO)C1)=O C1(O)(CNC(C2C(NC(C3(OC(C)C)CC3)=O)CCOC2)=O)CC2CCC1O2 c1(CC(=O)NC2CN(Cc3cncc(F)c3)CC2O)ccc(Br)cc1Br N1(C(c2cc(CCC)[nH]n2)=O)CC(C(=O)NCCN(C)CC)C(C(F)F)C1 CCCCC(C(=O)NCCCNC(C)=O)NC(=O)Cc1c(C)cccc1C N1(C(C(=O)NC2CCN(C(c3ccc(COC)o3)=O)C2)C)CCCC(O)C1 C(C)(CCC(=O)OC)N(CCCC(C)C)OC.c1(C)cn(CC(=O)N(C(C)(C)C)C)nn1 C(=O)(C1=CC2CCC(C1)C2)NC1C(CC)CN(C(=O)CCc2nc(O)n[nH]2)CC1 O=C1CN(C(c2cc(O)cs2)=O)C(C(N2CCC(CCO)C2)=O)C1 CN1CCC(C(N2CC(O)CC2C(N2CCCC2CN2CCCC2)=O)=O)CC1 C=C=CCN=c1nc2ncn(C)c2c(NCC(C(F)F)c2ccccc2)[nH]1 NC(=O)CCCCC(=O)Nc1cn(CCOc2cnc(F)c(C(F)(F)F)c2)nn1 N1(C(c2oc(CC)c(C)c2)=O)CC(CNC(c2ccc(C)cc2)=O)C2(CCC2)C1 c1(C(c2ccc(F)cc2)NC(N(CCC#C)C)=O)ccc(F)cc1 N1(C(C=CC(=O)OC)=O)CCC(F)(CNC(C2CCCN(C(C)=O)C2)=O)C1 c1(CC)[nH]nc(C(=O)NCC2(CC(C)C)CC2)c1-c1nn[nH]n1 C(=O)(C#CC1CCOCC1)NC1CC(CNC(c2c(C)cc(O)nn2)=O)C1 c1(C(=O)NCCC(C)NC(C2(C3CCCO3)CC2)=O)cc(O)nc(C2CC2)n1 C(=O)(CS(=O)(=O)CCC(F)(F)F)N1CCC2(N(C(CC(CC)C)=O)CCC2)C1 C(=O)(C(CNC(=O)CNC(=O)C(C)(C)C)CC(C)C)N1CCCN(CC)CC1 C(=O)(C(CNC(=O)C(C)(C)C)CC1CCCC1)NCc1[nH]nc(COC)n1 c1(C(=O)NC(C(=O)NCC(C(C)O)C)(C)C)ncn2c1CCC2 N1(C(CC(C)(C)n2cc(-c3ccc(C)cc3C#N)nn2)=O)CCC(O)CC(C)(C)C1 Cc1cc(NC(C2(NC(c3coc(C(N)=O)c3)=O)CC(CO)C2)=O)cc(Cl)c1 C1(CNC(c2cc(OCCOC)ncc2)=O)CCN(C(=O)CC=C(C)C)CC1C C(=O)(C1CCc2nnc(C)n21)NCCC(C)NC(c1cc(CC)on1)=O C1(NC(c2c(CC)c[nH]c2)=O)CCN(C(C2CC2F)=O)C(C)C1 N1(C(c2c(CC)onc2C)=O)CC2CC1CC2CNC(c1ccns1)=O Cc1cccc(C2=CCN(CC3CCCC3(C)C)CC2)c1C C1(NC(C(CC)OCC)=O)C2CN(C(=O)CC(C)(C)c3cccs3)CC12 c1(OCC(=O)NCCCNC(CC=CCCCCC)=O)ccc(C(N)=O)cc1 c1(-c2cn(CC(CNC(C(C)NC(N)=O)=O)(C)C)nn2)cccc(F)c1F Cc1cccc(C(=O)NC(CNC(c2cccc(-n3cccn3)n2)=O)CO)c1 C(=O)(CCCC(=O)N(CCCNC(C12CC(N=[N+]=[N-])C1C2)=O)C)NCC CCC(C)CCCC(=O)N(C(CNC(c1ccnn1COC)=O)CC)C c1(C(N(C(C)CNC(C2CC(N(C)C)C2)=O)C)=O)cnc(Cl)c(N)c1 C1(NC(C(C)N(C)C)=O)CC12CCN(C(c1c(F)cc(O)cc1F)=O)CC2 Cc1ccn2ncc(C(=O)N(C3CCCC(NC(c4cnc(O)s4)=O)C3)C)c2n1 CC(C)C(C(C)NC(=O)CCCN(C)C)NC(c1ncccn1)=O c1(SCC)cccc(C(N2CCC(C)(NC(C3CCCC3)=O)C2)=O)c1 c1(C(N2CCC(NC(CC=CCCC)=O)C(O)C2)=O)cc2ccccc2oc1=O CC#CCC(C(=O)N(C)Cc1ccncn1)NC(=O)COCC1CCCO1 N1(C(C=CCCC)=O)CCC2(CCCN(C(=O)C(F)C(=O)OCC)C2)C1 C1(C(N2CCN(C3CN(CC)C3)CC2)=O)CC(C(F)(F)F)CCN1C C1(NC(CC2CC(CC)C2)=O)CCN(C(=O)CC(F)(F)Cl)C1C N1(C(C(Cc2ccccc2)NC(=O)OCC)=O)CC2(C1)OC1(C)CC2(C#N)C1 CN1CCCC(CC(=O)NCC2CCCN(C(=O)CC3(C)N=N3)C2)C1 Cn1[nH]c(=N)cc1C(=O)Nc1cccc(CN2C(=O)C=CC2=O)c1 CCCCCC(O)C(=O)NCC1(OC)CN(C(C2CC3(CCC3)CO2)=O)C1 C1(CNC(C(C)n2ccnc2)=O)CCCCC1NC(=O)CC1CSC1 C12(NC(C(C(C)C)OCC)=O)CCCC1(F)CN(C(=O)C=C1CCOCC1)C2 c1(C(=O)NCC(CCOC)NC(C2CCCN2C=O)=O)sc(OC)nc1Cl C=CCC(C)(C)C(=O)NC1CCN(C(c2ccn(C3CC3(F)F)n2)=O)CC1CO N1(C(CC2C(C)CC2)=O)CC2CC1CC2CNC(c1coc(Cl)n1)=O C1(C(c2ccc(O)cc2)NC(=O)NC2C(OC)(OC)CC2)CCS(=O)(=O)CC1 C(=O)(CC(O)(CCC)CCC)NC1CC2CN(C(CC(CCC)O)=O)CC1C2 C12(CNC(CC3ON=C(CC)C3)=O)CCCC(CN1C(=O)C(F)=CCCF)C2 CC1(C(N2CCC(C(N)=O)C2)=O)CN(C(=O)C(F)n2ccnc2)C1 c1(N2CCN(C(C(C)C3CCCO3)=O)CC2)nccc2sccc12 C1(C(=O)NCCCN(C(c2ccccc2)C(=O)NC)C)CCCCC1(C)C c1(OCCCC)ccc(C(C)NC(=O)NC2(c3ncccn3)CCOCC2)cc1 CCCC(C)(C)CC(=O)NCC(O)CCNC(c1ccc(CSC)cc1)=O c1(-c2n(CC=C)c(N3CCC(C4CC(N)CCO4)CC3)nn2)ccc(O)c(F)c1 N1(C(C2CSC(C(F)(F)F)C2)=O)CC(O)(CCC(F)(F)F)C1.c1(CO)ocnc1C C1(NC(c2ccncc2Cl)=O)CCC2(CC1)CC2NC(c1ccc(=O)oc1)=O C1(CNC(C2(CO)CN(c3nc(C4CC4)nc(=N)[nH]3)C2)=O)CCc2nnnn2C1 c1(C(=O)NC(C(C(C)C)NC(CCCCCSC)=O)C)c(C)ncn(C)c1=O c1(C(=O)NC2CC(F)(CNC(C(CC)(C)C(F)F)=O)C2)ccc2nnc(O)n2c1 CCC(CC(=O)NC1COCCC1NC(=O)Cc1cncc(O)c1)CC(F)(F)F Cc1ccc(-c2nc(C(N3CC(CC(C)NC(C4OCCO4)=O)C3)=O)cs2)cc1 CC(C)(C(=O)NCC1CCCC1C(=O)NC1CC2CC2C1)c1cnsc1 C1(C(=O)NCC(C(C)O)C)(CNC(=O)CN2CCNC2=O)CCCCC1 c1(OCC(=O)NCC(C)(C2CCC2)NC(C2CCC(CC)C2)=O)ccccc1Cl C(=O)(CC(O)CCCCC)N1C(C#C)CN(C(=O)C=CC(C)C)CC1 Cc1cnn2cc(C(=O)NCCC(C)CCNC(c3ccc(=O)oc3)=O)cnc12 N1(C(c2cc(COC)[nH]n2)=O)CCCC2(C1)CN(C(=O)CC1CC=CC1)C2 C1(CNC(C2C(C)(C(N)=O)C2)=O)CC(F)(F)CN1C(=O)CCOC1CCCCC1 S(=O)(=O)(c1ccc(C)c2nsnc12)NCC(CC)CO C1(CNC(C2(C)CCC2)=O)CN(C(=O)CC2C=CS(=O)(=O)C2)C2(CCOCC2)C1 C=CCC(CNC(c1c[nH]cc1C)=O)C(=O)NCCCCN(C)C(C)C Cc1ccc(CNC(C2C3CC3CN2C(c2cc(C)ccc2F)=O)=O)c(O)c1 N1(C(C(CCN(C)C)N(C)C)=O)CCCC(F)(CNC(c2cc(O)ncn2)=O)C1 C#CCCCCCC(=O)NCC1CCN(C(c2n[nH]c(C)n2)=O)CCC1(F)F N1(C(C(c2scc(C)n2)C)=O)CC23CCCC2(C1)CN(Cc1cnn(C)c1)C3 N1(C(C(C)SC(C)C)=O)CCCCC(CNC(=O)CN2CCCC2C)C1 c1(NC(C2CC2C2CC2)=O)ccnc(-c2cccc(CO)c2)n1 CCCCC(CN1CCCC(C#N)C1)CC N1(C(C(C)(C2CC2)OC)=O)CC(NC(c2nccn2C)=O)C2(CCCC2)C1 C1(NC(C2(C(NOCCOCCOC)=O)CC23CCC3)=O)CN(C)CCN1C c1(C(=O)NC2CC(CNC(C3C(C)(C)CO3)=O)C2)ccc(CC2CC2)cc1 CCC(C)CC(C(=O)Nc1cc(CO)cc(F)c1)NC(c1cnnn1CC)=O C1(NC(C(C=CC)O)=O)CN(C(c2ccnc3ccnn23)=O)CCC12CCC2 C1(OC)CC(NC(=O)C(F)C(C)C)CN(C(=O)C(CC2CCC2)NC(C)=O)C1 Cc1cc(C)c(C(=O)NCC2C3CN(Cc4c(C)noc4C)CC23)c(O)n1 C1(NC(C(CC)C2CCC(=O)N2)=O)CN(C(c2c(C)nsc2C)=O)CC1OC C#CC1CCC(NC(C2CCN(C(=O)C=Cc3ccccc3)CC2)=O)C1 c1(SCCC)ccc(C(=O)NC2CN(C(C3CCC3)=O)CC2O)cc1 c1(N2CCS(=O)CC2)cccc(S(=O)(=O)N2CCCC2CF)n1 C1(CCNC(c2cnc(CC)s2)=O)CCN(C(c2cc(C(C)C)nn2C)=O)CC1 Cc1nn(C)c(C(=O)NCCOCCCN(C(=O)CCC(=O)OC)C)c1Cl c1(CC)cc(NC(CNC(c2cnn(C)c2Cl)=O)C(C)C(C)C)nc(C)n1 c1(C(N(C2CCCN(C(c3nnn(C)c3C)=O)C2)CC)=O)cc(Br)c(C)o1 C1(CNC(CCN(CC=C)C(C2CC=C(C)CC2)=O)=O)CN(CC)CCCO1 c1(C(C)C)cnn(C)c1C(=O)NCc1scc(CCN2CCOCC2)n1 N1(C(c2c(SC)nccc2)=O)C2CC1CN(C(=O)CC1CC(F)CN1)C2 C1(c2nc(C(=O)NCCCOC)nn2-c2ccc(Br)nc2)CCC2CCCCN12 CCC(C)CC(C)C(=O)NCC1(CNC(c2ncccc2NC)=O)CCC1 Cc1nn(CC(N2CCCCC2CN(C(=O)Cc2cc[nH]c2)C)=O)c(=O)n1C N1(C(C(CCC)NC(N)=O)=O)CCC(NC(c2[nH]c(C)nc2C)=O)C(O)C1 c1(CC(CC)O)nc(-c2cccc(Br)n2)nn1-c1cccc(OC)c1 c1(C(=O)NCc2nc3ccccc3[nH]2)ccc(F)c2ccsc12 CCCC(CCC)CC(=O)N1CC2CCN(C(c3cc(CC)c(CC)o3)=O)CC2C1 N1(C(c2ccccc2Cl)=O)CCC(O)(CNC(=O)C(F)(F)C2(O)CCC2)C1 C(CCC(=O)NC1(c2cn(CC3(c4ccccc4)CCCC3)nn2)CC1)C1C(C)C1 N1(C(C(C(C)C)SC)=O)CC2CCN(C(c3cccc4nc[nH]c34)=O)CC2C1 N1(C(CCP(C)(C)=O)=O)CCC2C(CCCN2C(c2ccns2)=O)C1 C1(C(=O)NC(C)Cc2cn[nH]c2)CCN(C(c2cnn3c2OCC3)=O)C12CC2 N1(CP(C)(C)=O)C#CC1.C=C(F)C1(CC(=O)NCC(F)(F)F)CCC1 c1(C(=O)NCC(CN(C(=O)CCC(F)(F)F)C)O)cccc2nc[nH]c12 C(c1ccc(C(F)F)o1)=CC(N1CCC(CN(C(c2c(C)cns2)=O)C)C1)=O C#Cc1ccc(NC(C)C)cc1.C1(C(=O)O)CCN(C(=O)OC(C)(C)C)CC1C Cc1c(F)ccc(C(=O)NC2CCN(C(=O)C=CC3CCCCC3)C(C)C2)c1N c1(NC(C(C(C)NC(c2c(C)ccnc2C)=O)C)=O)cnc(C)nc1C C(C)(C(C(=O)N1CCCC1CCNC(C1CC=CCC1)=O)N(C)C)OC CC(C)(C#N)C(=O)Nc1cccc(CNC(=O)Cc2nnc(S)n2C)c1 Cc1nc2cc(CC(=O)NCC(C)NC(=O)C=CCN(C)C)ccc2o1 c1(C(C)=O)nc(N2CCC(N3CCOCC3)C2)ncc1C.C12C3CN(CC13)C2=O C1(OCC)(CN)CCCN(C(=O)C(=O)NC(C2CCCCN2C)(C)C)C1 Cc1c(CC(N2CCOC(CCNC(c3cncs3)=O)C2)=O)cnn1C CC1(C)C2CCC1(C(N1CCC(C(=O)NC(C(O)CO)C3CC3)(CO)C1)=O)C2 N1(C(c2c(OC)c[nH]n2)=O)CCC(NC(c2ccc(C(C)(C)C)nc2)=O)C(C)C1 N1(C(=O)OC(C)(C)C)CCOC(C)(C(=O)NCC2CC3(C2)CC(O)C3)C1 C=CCC(F)(F)C(=O)N1CC(C)(OCC(=O)NCc2noc(COC)n2)C1 CCC(CC(=O)N1CCC(CNC(=O)COCCN(C)C)C12CC2)C(F)F C(=O)(CC(C(F)(F)F)NC(=O)CN1CCC(=O)NC1=O)N1C(C2(C)CC2)CCC1 N1(C(c2c(C)nns2)=O)CC(CO)C2(C1)CN(C(=O)COC1CCOCC1)C2 Cc1cc(C(N2CCC(C)(C)C(NC(=O)C3=C(Cl)CCCC3)C2)=O)cc(=O)n1C C1(NC(CC2CC(OC)C2)=O)CN(C(c2cncc(C3CC3)c2)=O)C(C)(C)C1 N1(C(CC2(OC)CC2)=O)CCC(C(=O)NCCCC2C=NNC2=O)CC1C CN1CC2CCN(C(C3(CF)CCN(C(C4COC(=O)N4C)=O)C3)=O)CC2C1 N1(C(CCCOCC=C)=O)CC(F)(F)CC1(C)CNC(=O)CC1CCSCC1 Cc1nn(CC(N2CC(C(C)NC(=O)CCc3cncnc3)C2)=O)c(=O)n1C C(=O)(C(C(C)(C)C)NC(=O)C(C)CCN(C)C)NCCCc1nc(C)[nH]n1 C1(C(=O)OCC(C(C)C)OCCN(C)C)CCN(C(c2ccccc2)=O)CC1 Cc1cncc(C(=O)NCC2CCCC(CNC(=O)CC3CCOC3=O)C2)n1 C1(C(N(CCCNC(=O)C=Cc2ccco2)CC)=O)CSC(c2ccccc2)=N1 CC(N=c1nc2sccc2c[nH]1)C(O)c1ccc(Cl)c(Cl)c1 C1(O)(c2cn(CCCN(C(=O)CCC3(N(C)C)CCCC3)C)nn2)CCCCC1 c1(N)ccc2nccn2n1.C(=O)(CCOCCNC(C1(N(C)C)CC1)=O)N N1(CCNc2cccc(OCCC)n2)CC(C)OC(C)C1 c1(OC)cc(C)c(CN2CC(C(N3CCC(CF)CC3)=O)C2)cn1 C1(OC)(CNC(=O)CC2CCCOCC2)CCN(C(=O)C#CC2(C)CC2)CC1 c1(CNC(CC2CCC(=O)N2)=O)ccccc1CNC(C1(F)C2CCCC12)=O C(=O)(C(C)(C)NC(C1CCOC1C1CC1)=O)NC1(CC=C)CCC1 c1(C(N2CC(O)(CNC(C(=O)OCC)=O)C2)=O)cc(COC(C)(C)C)nn1C c1(C(=O)NCC(CCOC)NC(C2CC=CCC2C)=O)c[nH]ccc1=O Cc1ccc(O)cc1C(N1CCC1(C)CC(N1CCC(C(N)=O)C1)=O)=O CC1(C)CCC=C1C(=O)NC1CCN(C(c2cc(C(C)(C)C)[nH]c2C)=O)C1 c1(C(N(C2CCCC(NC(=O)C3=COCCC3)C2)C)=O)cc(O)cc(O)n1 C=Cn1nccc1C(=O)NCCCCC1CCCN(C(=O)CN(C)CC)C1 C1(CN(C(=O)CC2CCC(=O)N2)C)C2CN(C(c3cccc(C(F)F)n3)=O)CC12 C1(NC(=O)C2CC2)CCN(C(c2cc(C)cc(O)n2)=O)CC12CCC2 c1(CC)nn(C)c(C(=O)NCC2CC3CC3N2C(c2csnc2C2CC2)=O)c1Cl CC1CCN(C(C2CC3(CC3)C2)=O)CCN1C(=O)CCCCCc1ccccc1 N1(C(CN(CCOC)C)=O)CCCN(C(=O)Cc2ccc(C)cc2)CC1C c1(CC)cc(C(=O)NC2CC(CNC(C3CCCCC3F)=O)C2)c(C)nn1 C#CC1CN(C(c2ccccc2O)=O)CCN1C(=O)COCC(=C)C Cn1ccc2c(C(N3CCCC(C)(CNC(=O)Cc4cnoc4)C3)=O)cccc12 C1(C#N)(OC)CC(C(=O)NC(CO)C(C)NC(C2CN(C)C2)=O)C1 C(=O)(C1CCc2ccc(C)cc21)N1C2(CCN(C(C(C3CC3)OCC)=O)C2)CCC1 C1(CC(=O)NCC(C)N(C(=O)C(O)C2CC2)C)CC1(C)C c1(NC(N2CCC(C(C)(O)C(F)(F)F)CC2)=O)c(O)ccc(F)c1Br N12CC3C4CCC(C3C1)N(C4)CCC2.Cc1cc(OC2CCCC2)no1 c1(NCC(CC)CCO)[nH]c(=NCc2cccc(Br)c2C)nc2c1ncn2C Cc1cccc(NC(C)C(=O)Nc2ccsc2C(=O)NCCCCC(F)(F)F)c1 C1(NC(C=C(C)c2ccccc2)=O)CCC(N=c2nc3[nH][nH]cc-3c(O)n2)CC1 C1(C(=O)Nc2cccc(I)n2)CC2CCCCC2N1Cc1cccc2[nH]ncc12 Cc1cc(NC(c2coc(Br)n2)c2nnnn2CC2CCCO2)ccc1O C1(CC(=O)NCC2(O)CN(C(c3c[nH]c(=O)s3)=O)C2)CC2CCC1O2 C1(C(N2C(CNC(c3c[nH]nc3C3CCCO3)=O)CC2)=O)CCc2c[nH]nc2C1 C12(C(N3CCC(C(=O)NC)CC3)=O)COCC1CN(C(=O)CCc1cn(C)nn1)C2 Nc1cc(C(=O)NCC2CCCC(NC(=O)COC3CCCC3)C2)cnc1N C1(c2ccccc2)(NC(c2cc(F)cs2)=O)CCN(C(c2ccnnc2)=O)C1 C=C=C(C)CC(=O)N1CCC(CCN(C)C(C2CC2CCOC)=O)CC1 Cc1cc(C#N)cc(C(N2CC(CCNC(C3COCCO3)=O)C2)=O)n1 c1(CCC(=O)N(CC(C)CNC(=O)C=CC(F)(F)F)C)ccncn1 c1(C(N2CCCC(CNC(C(CO)NC(N)=O)=O)C2)=O)ccc(F)c(CO)c1 CN1C(=O)CC(NC(C2CC2CNC(=O)C(=O)C(C)(C)C)=O)C1=O C1(N(C(COCC)=O)C)CCCCC1N(C)C(c1oc(C(=O)NC)cc1C)=O CCCCCC(C(C)(C)C)NC(N1CCCC(C(O)C(=O)O)C1)=O Cc1ccc2nc(C)cc(C(N3C4CCC3C(CNC(=O)C=C3CC3)C4)=O)c2c1 N1(c2c(C)c(NCc3nc(Cl)cs3)ncn2)C2CCC1CN(C)C2 C(CC(=O)NCn1ccnc1)N(C(=O)CN1CCCC1)CC#C N1(C(C2C(C(=O)OC)C2)=O)CCC2(CC1)CCN(C(=O)CCc1ccoc1)CC2 c1(C(=O)OC)c(C)cc(C)nc1NC1CC(F)(CNC(C2(C3CCCO3)CC2)=O)C1 n1(CCCC)cc(C(=O)NC(CNC(c2cccnc2C(F)F)=O)CO)c(C)n1 C(C(C)C)(C(O)C(=O)NC(COC)C(=O)NCc1ccc(F)cn1)OC CC(CO)N(C(=O)CC1(N(C)C)CC1)C.C12(CC1)C(=O)N(C)C2 N1(C(c2cnc(CC)[nH]2)=O)CCC(NC(c2cc(C3CC3)nn2C)=O)C(C)C1 c1(OC)ccc(O)cc1CNC1CC(F)CN(C(C2CC3C=CC2C3)=O)C1 N1(CC)CCOCC1C(=O)NCC(=O)NCc1cn(-c2ccccc2C)nn1 C(N=c1ccnc(NC2CCCC(C3CC3)O2)[nH]1)C1(C=C)CCOCC1 N#Cc1ccccc1CC(N1CC2(C1)CN(C(c1cccc(C3CC3)c1)=O)C2)=O C1(NC(CSC(C)(C)C)=O)CCC2CN(c3nnc(-c4ccccc4)o3)CC2C1 c1(C(=O)NC(c2ccc3c(c2)CN(C(=O)CC#N)C3)C)ccnc2c1ccn2C C(=O)(C(F)C(C)CC(C)(C)C)NC(CC)CNC(=O)CC=C(Cl)Cl CCC(C)C(C)C(=O)NC(C)(C)CCCNC(c1cncc(C)n1)=O N1(C(CCC)=O)CCC(CC(C)NC(C2CN(C(C3CCC(=O)N3)=O)C2)=O)CC1 c1(CNC(C2CCC(=C)CC2)=O)n[nH]c2c1CN(C(c1cscn1)=O)CC2 c1(OC)ccccc1C(=O)NC(C)CCCNC(=O)CCCOC(C)(C)C c1(CC)nc[nH]c1C(=O)N(C1CCN(C(C2C(C(=O)O)C2(F)F)=O)C1)C C12(C(=O)NCCC=C)CCC(CC1NC(=O)NC(C(=O)OCC)CC)C2 C(CC(C)(C)C(=O)N1CCCC(C(C)NC(=O)CC2CCCC2)C1)SC N1(C(C(C(=C)C)(C)C)=O)CC(NC(C2CC23CCC3)=O)C2(CCCC2)C1 C1(C(N(CCCCC(=O)NCC(O)C(F)F)C)=O)CCC(C#N)CC1 c1(NC(Cc2cn(CC(COC)(C)C)nn2)=O)cccc(Oc2ccncc2)c1 C=C=CCCC(=O)N(CCC(C)NC(c1c[nH]c(C(N)=O)c1)=O)C c1(C(=O)NCCC2(C)CCN(C(C3COCCO3)=O)CC2)ccc(S(N)(=O)=O)o1 O=C1Cc2cc(C(=O)NCC3CCCN3C(c3cccnc3Cl)=O)ccc2N1 c1(OC)ncc(C(=O)NCCCCCOC(F)F)cn1 C1(NC(CCc2n(C)ncc2)=O)CCN(C(=O)CCCc2cnn[nH]2)C12CC2 N1(C(C2C(c3ccc(C)nc3)C2)=O)CCC2(CC1)CN(C(=O)CC(O)C(C)C)C2 c1(C(=O)NCC(=C2CN(C(=O)CCN3CCNC(=O)C3)C2)F)ccncc1Cl c1(CC(=O)NCC23OCCC(NC(CCSC)=O)(C2)C3)c(O)nc(=N)[nH]c1C N1(C(C2C(COC)C2)=O)CC2CCC(C1)N2C(c1cc(C2CCOC2)[nH]n1)=O C(=O)(N=c1[nH][nH]c2cc(Cl)ccc12)c1cc(OC)ncc1OC(F)F Cc1cc(C(=O)NC2CC(C(F)C(=O)NCCC3CCCC3)C2)cc(C#N)c1 c1(N(CC(C)NC(c2cc(OC)c(Cl)cc2)=O)C)cc2nncn2cn1 C(=O)(C1=CS(=O)(=O)CCC1)NC(c1ccc(C)cc1)CNC(=O)Cn1cccn1 C(C(=O)N=c1ccn(C(C)C)[nH]1)(C(C)(C)O)NC(c1c(C)nc(C(C)C)o1)=O C1(C(=O)OC)N(C(C2CCC3(CC2)CC3)=O)CC12CCCC2 c1(C(=O)NCCCN(C(=O)CC(C)C2CCCO2)CC)ccccc2c(C)[nH]c1-2 C1(C(N(CCCNC(=O)Cn2cnnn2)C)=O)CCCCC1C(F)(F)F.CC C(=O)(C1CCc2ccccc21)NC1(C)CCCN(C(c2oc(C)c(CO)c2)=O)C1 N1(CC(=O)NCCC2CC(NC(C34COCC3C4)=O)C2)CCCOC1=O c12ccc3c(c1)CCN(C3)Cc1cccc-2c1F.SC C1(Cc2nc(CCOCC)[nH]n2)CCCN1S(=O)(=O)N(C)C c1(N2CC(C)C(NC(=O)CCc3nc(O)n[nH]3)CC2)nccc(C#N)c1[N+](=O)[O-] Cc1csc(C(c2nnnn2CCCF)NC(Cc2cccnc2)C(=O)O)n1 C12CCN(C3(CCC3)C1)C2=O.C1(C(=O)OC)CN2CCCN1CC2 Cc1ccc(=O)n(CC(N2CCCC(NC(=O)C(S(C)(=O)=O)C3CC3)CC2)=O)n1 C1(C(C2CCCC2)SCC(C)O)CCOC1 Cc1ccc(C(N2CCC(CNC(=O)C=Cc3cc[nH]c3)C(C)C2)=O)c(C)n1 c1(OC2(C(=O)NCC(CNC(=O)Cn3cc(Cl)cn3)F)CC2)ccc(Cl)cc1 c1(NC(C2SCCN(Cc3c(C)cccc3Br)C2)=O)nc(Cl)c(F)cc1C#N CC(C)C(C#N)C(=O)N1CC(CO)(NC(=O)C(Cc2ccccc2)C(C)C)C1 c1(CC)c(C(=O)NC(C)CCNC(=O)CCc2ccc(Cl)cc2)csc1C N1(C(c2cnc(COC)[nH]c2=N)=O)CCN(C(=O)C(O)CC)CC12CC2 C1(C(N2C(CCCC)CCC2)=O)CCCC(NC(C2CCN(OC)CC2)=O)CC1 N1(C(c2cc(CC)n(C)n2)=O)CCCN(C(C2CC3CCCCCC23)=O)C(C)C1 c1(OC)cccc(CN2CCC(N(C(=O)CC3CCCC3)C)C2)c1Cl c1(OC)cccc(C(=O)NC(C2CCCN2C(=O)CC(C)NC(N)=O)C)n1 N1(C(C(CNC(c2c(CC)occ2)=O)C(C)C)=O)CCOCC2(CCC2)C1 c1(NC(COC)(C)CCOC)nc(C)ccc1[N+](=O)[O-] c1(COC(CC(C)(C)F)=O)ccccc1S(=O)C(F)(F)F C(=O)(CC(F)(F)F)N1CC(CNC(C(CC)OC2CCCC2)=O)C1 c1(CC)nc(NC2CCOC2(C)C)c2scc(C)c2n1 N1(C(C(C)C#N)=O)CCC2(CCCCN(C(c3cnc4n3CCS4)=O)C2)C1 Cc1sc2ccc(Cl)cc2c1C(=O)NCC1CN(C(c2ccc(CN(C)C)[nH]2)=O)C1 c1(NC(N2CC(CN(C(C3C(C)C3)=O)C)C2)=O)[nH]ccc1-c1cccs1 C(=O)(C(O)C(F)(F)F)NCC(C)CC(=O)NCC1CC(C#N)C1 N1(C(C(C2CCC2)OCC)=O)CC2(CCN(C(C3NC(=O)C4CC34)=O)C2)C1 N1(C(C(CC2CC2)OC)=O)CCCN(C(=O)C=Cc2ncc[nH]2)C(C)C1 c1(C(=O)NC2CN(C(C(CC=C)C)=O)CC2C)c([N+](=O)[O-])c(C)nn1C N1(C(c2cc(CC)ncc2)=O)CCN(C(=O)C(C)P(C)(C)=O)CC1C1CCC1 n1(CC(N2CC(OCCNC(CN(C(C)=O)C)=O)C2)=O)ncc(O)nc1=O C1(C)(C(=O)NCCCOC)CCCN(C(=O)Cc2ccccc2C#N)C1 N1(C(c2c(NCc3cccc(CC)c3)ccs2)=O)CCc2ccccc2CC1 C(=O)(CC1=CCOCC1)NCC(C)(C(C)C)N.CC(C)CSCC(=O)NCCS C12(NC(c3c(SC)c[nH]n3)=O)CC(C1)N(C(c1csc(-c3ccco3)n1)=O)C2 Cn1nc(C(=O)NCC2CC2NC(c2cnncc2O)=O)c2c1CCSC2 Cc1cc(C(=O)NC2(CCNC(c3cc(C4CCC4)on3)=O)CC2)ncc1F CC1CC2(CCN(C(=O)Cc3cnns3)CC2)CN1C(=O)C(O)C1CC1 C1(CNC(=O)C=CC2CCOC2)CC2COCC2N1C(c1ccc(O)nc1Cl)=O c1(C(=O)NCC(CNC(CSc2cccc(C)c2)=O)F)ccc2nc(Cl)nn2c1 C1(NC(CC2CCC(NC(COCCSC)=O)C2)=O)CC2CSCC2C1 N1(C(C=C2CCC(C)C2)=O)CCCCC1CNC(C1CC(O)C1)=O C(=O)(C(C)CNS(=O)(=O)CC1CCC(NC(=O)OC(C)(C)C)C1)OCC Cc1nc(O)nc(O)c1CC(=O)NCCCC1(NC(C2(C)CCCC2)=O)CC1 C12(CNC(N(c3ccc(C(=O)OCC)cc3)C)=O)CC(C)(C1)OC2C c1(C(=O)NCC#CCNC(C(C(CC)C)C)=O)cc2c(cc1Br)OCO2 C1(CC)(NC(c2oc(Br)nc2C)=O)CCN(C(=O)CC2(O)CCCC2)CC1 n1(CC(N2CC(O)(CCNC(c3cccc(F)c3)=O)C2)=O)ncc2ncccc12 N1(C(COC2(C#C)COC2)=O)CC2(C1)CN(C(=O)C(CC)SC)CCO2 C(=O)(CCCCC(C)(C)C)N(CCCCCC)CCNC(C1CCC2(CC2)C1)=O Cc1cc(CN2CCCC(NC(=O)CCN3CCCCC3)CC2)ccc1F C(CCC(C)(C)NC(=O)C(c1ccc(C)o1)C)NC(c1ncn(CC)c1)=O N1(C(C(COC)COC)=O)CCCC(CO)(NC(c2ccc(F)cc2F)=O)C1 c1(C(=O)NC2C(NC(c3cnc(COC)s3)=O)COCC2)cc(C#N)ccc1O CN1CC2(C)CN(CC3CCCCO3)CC2(C)C1 c1(CCNC(C(C2CC2)SCC(=O)OCC)=O)cnc(-c2ccccc2)n1C.CN Cc1cc(C(=O)NC2CCCCC2NC(=O)CC2CCCO2)cc(N)c1 C1(C(N2CCC(C)(NC(=O)CCSCC(N)=O)CC2)=O)CCC2(CCC2)CO1 c1(C(=O)NC2CC(F)(CNC(c3cnn[nH]3)=O)C2)cccc2nsnc12 C1(C(=O)NCc2cc(CC)nn2C)CCCN(C(c2cc(CO)[nH]n2)=O)C1C CC1CC(C)N(C(c2cnco2)=O)CCN1C(c1cc2nccc(Cl)c2s1)=O C(N=C(NCC1(O)CCCCC1)N1CCC(OC)C(C)C1)c1ccc(C#C)cc1 C(=O)(C(CO)C1CC1)N(CCNC(C(C)C)=O)C C1(NC(c2[nH]cc(C)c2)=O)CC2C1CCN2C(=O)Cn1nc(C)n(C)c1=O c1(C(=O)NCCOC2CCN(C(c3cnc(N(C)C)s3)=O)C2)c(Cl)nn(C)c1Cl CC1CC(=O)NCC1C(N1CCN(C(=O)C(c2ccccc2)C)CC1C)=O CCCC(CC)CCC(=O)NCC1CC(NC(=O)C2=CCCC2)CCO1 C1(NC(C2(NC(C3C(NC(C)=O)CC3)=O)CC=CC2)=O)CCC(C)(C)CC1 N1(C(Cc2c(C)n[nH]c2C)=O)CC2CCCC2(CNC(C2CC2F)=O)C1 C1(C(=O)NCc2ncn(C)c2)CCN(C(=O)C23CC(C#N)(C2)C3)O1 n1(CC2N(C(C(n3cc(C4(C)CSC4)nn3)C)=O)CC2)cc(F)ccc1=O C(C(CC(F)(F)F)NC(=O)C(C(C)(C)C)C1CCC1)NC(CC=C)=O c1(C(N2CCC(CNC(Cc3cc(C)sc3)=O)(CF)C2)=O)ccc(=O)n(CCO)c1 C1(CN(C(CC(C)c2ccco2)=O)C)COCCN1C(=O)Cc1cncs1 CCC(C)(CNC(=O)CCCCCSC)C(=O)NC1CN(C(C)C)C1 C1(C(=O)NCC2N(C)CCC2)CC(O)CN1C(=O)CC1CC2(CC2)C1 c1(N2CCCC(OC(CC)C)C2=O)cc(OC)cc(C(=O)OC)c1Cl c1(NC(C(=O)NC(C(=O)NCC(C)C)C)=O)cccc2c1CNC2=O C1(CC)CCC(C(=O)NC(C2CCCCN2C(c2scnc2C2CC2)=O)C)CC1 CCC(C)C(=O)NC(C)CC1CN(C(=O)C=C2CCC(C)C2)C1 CCC(C)CCCC(=O)N1C2CCC1C(C(=O)NCc1nc(C)c(C)[nH]1)C2 c1(CNC(C2(F)CN(C(CCc3cnc(C)s3)=O)C2)=O)ccc2[nH]ccc2c1 c1(C(COC)(C)O)cn(CCCC(=O)NCc2nc(C(N)=O)co2)nn1 C1(C(=O)NCCn2cnnc2)(CC)CCN(C(C2CSC2)=O)CC1 C12(C(=O)OCc3cccc(OCC)c3)CC(Cc3ccccc3)(C1)OC2(C)C Cc1cccc2ccc(C(=O)N(CC(C)NC(=O)C(Cl)=CCl)C)nc12 c1(C(N2CCCC(CN(C(C3(C=C)CC3)=O)CC)C2)=O)cc(C)[nH]c(=NC)n1 c1(-c2nc(CN(CC#C)C)on2)ccccc1F.C(F)(F)F c1(C(N(CCCN(C(=O)CSC2CCCC2)C)CCO)=O)ccc(N)c(F)c1 N1(C(C(=O)NC(C)C)=O)CC2CC2(NC(=O)CCC(C)N(C)C)C1 C=Cc1cnn(C)c1C(N1CCCC(CNC(=O)C(CC)SC)C1)=O c1(C(=O)NC)cccc(C(=O)NC2CC(C)(NC(=O)Cc3ccncc3Cl)C2)c1 C1(NCCCC)C2CC3C1C3C2C(=O)NC(=O)C(C)N(C(C)CC)C(C)C c1(NC(c2ccc(OC)nc2)C)nccc(=NC(C)C2CCCC2)[nH]1 CC(C)(C)C(C#N)C(=O)N1CCS(=O)C2(CCC2)C1 C=CCCCCCC(=O)NCC12CC1CN(C(=O)CC1CCCC1(F)F)C2 C12(C(N3CCC(COC)CC3)=O)COC(C1)C(NC(=O)Cn1nccc1C)C2 N1(C(c2n(CC)c(O)nc2)=O)CCC2(CC2C(=O)NC(C)(C)CC2CCC2)C1 Cc1noc(C)c1C(=O)NCC1(O)CC(N)C1.N1(C(=O)C2CC2)CC1 C(=O)(C1=CCCN(C(C(=O)NC2CC(F)(F)C2)C(C)CC)C1)OC NC(=O)CC(C(=O)N1CCC1c1ccccc1)NC(=O)CCCn1ccnc1 Cc1ccc(I)c(C(=O)NCC2CCN(Cc3ncsc3C)C2)c1 C(CC(=O)NNC(=O)C1CCCC2(CC2)C1)SC.N1(CCO)CC1 C1(CNC(C(C)c2ccco2)=O)C(C2CC2)CCN1C(c1cncn1C)=O CCCCC(CC)C(=O)N1CC(F)(C(=O)NC(C2CSC2)C)C1 C12(NC(Cn3ncc(C)c3)=O)CCCC(CN(C(=O)CCc3ncc[nH]3)C1)C2 c1(C(=O)NC(CC)CNC(C2CC2C2CCCO2)=O)ccc(N)c(F)c1 CC(CCCCNC(c1cnn(C)c1C(F)F)=O)NC(=O)CC1(O)CCCOC1 C(=O)(CC(O)CC(C)C)N1C(C(=O)NCCNC(=O)C(C)C)(CC)CCC1 CCCCCCC(=O)N1CCCC(O)(CN(C)C(c2occc2Br)=O)C1 c1(CNC(C2CCC(CC)O2)=O)ccc(C(=O)NCC2(O)CCCCC2)cn1.C1CC1 Cc1nc(=N)[nH]c(C)c1C(=O)NCC1(O)CN(C(C23CCCN(CCC2)C3)=O)C1 N1(C(c2cccc(CC=C)c2)=O)CCN(C(=O)CC(C)COC)CC(C)C1 C1(NC(CC=CC)=O)CN(C(=O)C(CC)C2CCC(=O)N2)CC1(C)C Cc1ncc(NCc2nnn(C)c2C(F)(F)F)cc1C(=O)O C#Cc1ccc(C(=O)NC(CNC(c2nocc2C(C)C)=O)C(C)C(C)C)cc1 c1(C(=O)NCCC(C)CCNC(C2(C)CCC2)=O)nnc(O)nc1O CC(C)C(F)(F)CC(=O)N1CCC(CCNC(C2CC2(C)C)=O)C1 N1(C(c2c(CCC)nco2)=O)C2CCC(C(=O)Nc3ccc(CF)cc3)C1CC2 O(N1C(=O)c2ccccc2C1=O)CC(=O)N(C)Cc1ccc(CO)cc1 C1(CNC(C(C)(F)F)=O)CCC2(CCN(C(C3CC(C)(O)C3)=O)CC2)CO1 N1(C(c2cc(C)c(C)s2)=O)CC(NC(c2ccn(C(C)C)n2)=O)CC(F)C1 C1(CC)C(C(=O)NCc2cc(OC)ns2)CCCN1C(c1ncn(C)n1)=O C=C(C)C(CC(=O)NCC(CCCC)NC(=O)CCCCCC1CC1)OCC CON(CCC(=O)NC(C)CC(=O)N(C)C)C(=O)C1C2CCC(F)(F)C12 c1(C(N2C(C)CCC(NC(c3cnn[nH]3)=O)C2)=O)cc2ccc(F)cc2s1 Cc1c(C(=O)NC(C)C(C)NC(c2ccc(Br)cc2)=O)cnn1C(C)(C)C c1(C(=O)NC(CC)(C)CNC(=O)C(C(C)O)N(C)C)ccc(=NC)[nH]c1 c1(NC(C(=O)NC(CNC(CC2N(C(C)C)CCC2)=O)(C)C)=O)ccc(Cl)cc1 c1(NC(=O)C(=O)N(C)C)cccc(Br)c1F.C12(CCC1)N(C)C2=O CCCCC(O)C(=O)N1CCCC1C1(C(=O)NCCC(C)(C)O)CC1 N1(C(C2CCC(=O)C2)=O)CCC(C2CC(NC(C3CCCCC(=O)N3)=O)C2)CC1 c1(C(=O)NC(C(C)NC(c2ccc(-c3ccco3)s2)=O)CO)ccc(O)nc1 C(CCCC(=O)NC(C1(O)CCN(C(C2CS(=O)(=O)C2)=O)C1)C)OCCC=C c1(-c2cccc(CSCCOC(=N)O)c2)nc2c(s1)CCCC2 c1(C(N2CCCC(O)(CNC(C(C)OCC)=O)C2)=O)cnc2c(c1)COCC2 N1(C(C2(O)CC(C)(C)C2)=O)C2CCC1CN(C(C1CC1c1ccc(F)cn1)=O)C2 CCC(C)(CO)C(=O)N1CCN(C(c2ccc(C)c(Cl)c2)=O)C(C(C)C)C1 N1(C(C=Cc2c(C)coc2C)=O)Cc2ccccc2C(NC(C2C=CCS2)=O)C1 c1(C(C(=O)NCC(C)(C)CNC(=O)CSC2CC2)(F)F)cc(F)cc(C#N)c1 Cc1cnc(-c2cn(CCC3CN(C(=O)C(c4ccc(Cl)cc4)C)C3)nn2)nc1 CN1CCN(C(c2cncnc2)=O)C(CNC(c2csc(C(N)=O)n2)=O)C1 c1(CC(=O)NC2(CF)CCN(C(COCCCC#C)=O)C2)ccc(C)cc1Cl c1(OC)n[nH]cc1C(=O)NC(CO)C(C)NC(C1CC1c1ccoc1C)=O CC(C)C(C(=O)NCC1CCCCC1NC(c1ccc(Cl)nn1)=O)n1ncc(N)n1 c1(C(=O)NCC2(COC)COC2)cc(-c2ccc(NS(C)(=O)=O)cc2)cnc1F C1(C(=O)NC2CCCN(CC(=O)Nc3scc(C)n3)C2)CCS(=O)(=O)C1(C)C C1(CC(=O)NC(CC)CC(=O)OC)CCN(C(=O)CC2C(=O)NN=C2C)C(C)C1 C1(C(N2CC(OCC(=O)NC)C2)=O)COC(CNC(=O)Cc2ccnn2C)C1 CN(CCNC(C1CCCCC1)=O)N1CC2CCCCCC2C1 C(=O)(C(C)(C)CC(=O)NCC(C(N1CC(C2(C)CC2)C1)=O)N(C)C)N(C)C C=CCCCCCCC(=O)NC(C)(C)C(C)CC(=O)NCC12CCCC1CCO2 C1(CNC(C(CCO)N(C)C)=O)CCCCN(C(=O)C(N)=O)C1 CCCCC(C(=O)NCC1CC(NC(C2CSCN2C(C)=O)=O)C1)C(C)C C(=O)(C1Cc2ccccc21)NCC(C)(C)CNC(c1c(F)cccc1Cl)=O C(=O)(C1=CS(=O)(=O)CCC1)NCCC1N(C(C2(C)COC2)=O)CCSC1 c1(C(=O)NCC2C3(CCN(C(C=NOC)=O)CC3)C2)cc(S(N)(=O)=O)cn1C c1(OC)cc(F)c(C(N2CC(CNC(c3cccnc3)=O)C2)=O)c(F)c1 N1(C(C(C2CC2)SC)=O)CCOCC(CNC(=O)COCCF)C1 C1(C(=O)NCCC2CN(C(C3(F)CCOC3)=O)C2)CCC(NC2CCC2)CC1 C1(OCC(=O)NCC2CC2CNC(=O)CN2CC3CC3C2)CCCCCC1 c1(NC(=O)NCC(c2cccc(Cl)c2)(CC)O)ccc(CC(=O)OC(C)C)cc1 Cc1ccc(C(=O)NCCN(C)C(c2ccc(C3CC3C)o2)=O)c(C)n1 C(=O)(CC(C)C(F)F)NCCC(=C)CNC(=O)COc1cccc(CC)c1 CCC(CC)(CC)C(=O)NC1CN(C(=O)CSc2ccc(F)cc2)C2CC12 N1(C(C2(C(N3CC(N=[N+]=[N-])C3)=O)CC(=C)C2)=O)CCOC(C)C1C C(=O)(C(C)(CO)OC(F)(F)F)OC(C)(C)C.c12cnccc1C(=O)N2 C(N=c1cc(C(F)F)nc(S(C)(=O)=O)[nH]1)C1CC2N(C(CCSC)=O)C(CC2)C1 c1(C(=O)NC2C(NC(C(CC)N(C)C)=O)CCCC2)c(N)cccc1[N+](=O)[O-] c1(OC)cc(OC)cc(CNC2(c3nnnn3C)CCCCC2CC#N)c1 N1(C(C2(C(C)(C)C)CCCC2)=O)CCOCC(NC(c2cccc(N)n2)=O)C1 c1(C(=O)NC2(CC(=O)NC(CC3CC3)C3CC3)CC2)cnccn1 C1(C(N(CCNC(CN(S(CC)(=O)=O)C)=O)C2CC2)=O)CCCC1C(F)F CCS(=O)(=O)C=CC(=O)N1CC2(CCN(C(=O)Cc3cc(Cl)ccc3Cl)C2)C1 c1(C(=O)NC2CC(F)(CNC(C(C)N(C)C)=O)C2)cnc2c(cnn2C)c1 Cc1ccc(F)c(S(=O)(=O)NCCOC(=O)NC23CC(C)(C2)OC32CCC2)c1 c1(Oc2ccc(COC(COC)C)cc2)ccc(S(=O)(=O)CCCO)cc1 CC(C(=O)NCC1CCC1NC(=O)CCOc1cccc(Cl)c1)C(F)(F)F C(=O)(C1=CC2CCCCCC12)NC(CNC(c1c(C)c(F)c(F)cc1)=O)(C)C C1(C)(OC)CN(CC(=O)NC2CC(OCCSc3ccccc3)C2)C1 C1(C(=O)NC(c2cccnc2)C(=O)NCCC2(C)CCCC2)CC1C1CCC1 N1(C(CCN(C(C2CCCC(OC)C2)=O)CCO)=O)CCC2(CCCCC2)C1 Cc1cc(C(N2CCC(CNC(=O)CC3CCCN3C)C(O)C2)=O)c(N)cc1F C1(C(=O)NC2(COC)CC2)CCN(C(c2ccccn2)=O)C1C(C)C C1(NC(c2c(C)csn2)=O)CCC2CCN(C(c3cnc(C(C)C)o3)=O)C12 Cc1cc(CC(=O)N(C)CCOCCN(C(=O)CCF)C(C)C)cs1 c1(C(=O)N(CCCCNCC2CCC(C(=O)OC)CC2)CCO)cccc(Cl)c1Cl c1(CNC(C2OCC(C(=O)NC(c3n(C)ccn3)CO)C2)=O)cc(Cl)ccn1 N1(C(c2c(C)nn[nH]2)=O)CCCC2(NC(C3CC=CCO3)=O)CC2C1 N1(C(CCC(=C)Cl)=O)C(CC(N2C(C(=O)OC)CC2C)=O)C2CCCC12 CC1CCC(Cl)=C(C(=O)NCC(C)(O)CNC(=O)Cc2ccncc2Cl)C1 C(=O)(C1=NOC2(CCC2)C1)NC1(COC)CCN(C(=O)CCN2CCCC2)CC1 CN1C(=O)CCC(CNC(C2CC(C)N2C(=O)CCC(=O)N(C)C)=O)C1=O c1(CC)nc(C)ncc1C(=O)NC(C)CC(C)NC(c1ccc(OC)nc1Cl)=O c1(C(N2CC(NC(c3cnn(C4CCC4)c3)=O)(CO)C2)=O)cccc2[nH]ccc12 CC(CC(C)(F)F)C(=O)N1CC2CC(O)C1C2NC(c1ccn(CCN(C)C)n1)=O Cc1ccc(O)c(C(N2CCC(N(C)C(C3CCOC3C(C)C)=O)C2)=O)n1 C1(C(=O)NC(c2ccncc2)C)CCN(C(c2cn(C3CC3)nn2)=O)CC1O Cc1ccc(CCC(=O)N(C(C)CNC(=O)C(C)C2CC2)C)s1 c1(SC)ccccc1CC(N1CC(NC(c2nnccc2C)=O)CC1C)=O N1(C(C(C)OCC)=O)CC2CC1CCC2NC(C1(O)CCCCCC1)=O C1(C(N(C2CN(C(C3(C(F)F)CC3)=O)C2)C)=O)CCC(=O)N(C2CC2)C1 C=CC1(NC(=O)C(CC2CC2)NC(C2CN(C(C)=O)C2)=O)CCCCC1 N1(C(CN(C(=O)CC#N)C)=O)CCC(O)(C(=O)Nc2ccc(NCCO)cc2)C1 C1(OC)CCC(NC(=O)C(C)N(C)C(c2sccc2Cl)=O)C1 C(=O)(C#CC1(CC)COC1)N1CC2C(C(=O)NC3(CC=C)CCCC3)(C2)C1 C1(F)(c2cn(CC3N(C(CS(C)(=O)=O)=O)CC3)nn2)CCC(F)(F)CC1 N1(C(C23C(C)OC(C)(C2)C3)=O)CCN2C(=O)C(NC(c3cnn(C)c3)=O)CC2C1 C12(CCNC(c3cc(C)on3)=O)CCC1CN(C(=O)C=C(C1CC1)C1CC1)C2 c1(C(N(C2CCCC(NC(=O)C(C)(C)n3cnnn3)C2)C)=O)cnc(=N)[nH]c1 CN1C(=O)CC(C(N2CCCN(CC(C)(C)C)CC2)=O)C1c1ccccc1 C(=O)(C(C)(O)C(C)C)NC(CC(=O)Nc1ccc(OC)cc1)C1CC1 N1(C(C(C)(C)C2CCC2)=O)CCC(NC(C23CSC(C2)C3)=O)C(C)(C)C1 S(=O)(=O)(c1cc(Br)c(Br)s1)NCCC1CCCN(C(C(C(C)(C)C)O)=O)C1 Cc1nc(NC(c2ccccc2)CC#N)cc(=NCC2CC2Cl)[nH]1 C(=O)(CC(CCC)NC(=O)CCCCCF)N1CC(OCC#C)C1 C1(OC)CCCC(C(N2CCC(C)(NC(=O)Cc3n[nH]c(C)n3)C2)=O)C1 N1(C(c2c(CC)cc[nH]2)=O)CCC(C(=O)NCC2CC3(CC3)CO2)CC1CC C1(C)(C(N(CCC#C)CC)=O)CCCN(C(c2ccc(F)s2)=O)C1 c1(C(N2CC3CC3(c3nc[nH]n3)C2)C(=O)OC)ccc(Cl)cc1.N12CCC(C1)C2 C=CC1(CC(=O)N(C2CCCC(NC(=O)CC3CCC3)C2)C)CCCCC1 Cc1sc(C)c(S(=O)(=O)N2CC(NC(=O)C(F)(F)F)CC2C)c1C C1(C(=O)NCC(C)NC(C2CC(n3cccn3)C2)=O)CCC(C)C1 c1cc2[nH]c(NCC3CCNC4CCC34)nc2cn1 c1(OC)ccc(C(=O)NCC2CN(C(C3(C#N)CC3)=O)CC2O)c(F)c1F C(=O)(C(C(C)C)n1ccc(C2CC2)n1)N1C(C(=O)N(c2c(C)nsc2)C)CCC1 C1(NC(C=COCC)=O)CCCCC1OC.C1(CNC(=O)CN(C)C2CC2)CC1 C(=O)(CC(C(C)OC)NC(C1CC2C=CC1O2)=O)N(CC(CC)OC)C C(CN=[N+]=[N-])(C(=O)NCCCc1ncn(C)n1)NC(c1c[nH]c(=NC)s1)=O C1(NC(c2nc(-c3c(C#N)ccnc3)sc2)=O)CCOC12CCOC2 c1(CC(N2CCC(CC(=O)NCc3cccc(Cl)n3)C2)=O)cc(F)cc(Br)c1 C(CCN(C(=O)CCC1CCCC(O)C1)C)(C(C)(C)C)NC(c1c(C)nns1)=O C1(C(=O)NC(CNC(CCCC(=O)OC)=O)CO)CCn2ncnc2C1 C1(NC(C2CN(CC)C2)=O)CCN(C(=O)CCP(C)(C)=O)CC1(C)C C#CCC(C)(C)C(=O)NC1CC(C)CN(C(=O)CCCc2ccc(F)cc2)C1 c1(-c2cn(CC3OCCN(C(c4ccc(OC)o4)=O)C3)nn2)ccc(SC)cc1 C(=O)(CC(P(C)(C)=O)P(C)(C)=O)N1CCC(C)C(CNC(=O)CCCN=[N+]=[N-])C1 Cc1cc(C)n2nc(C(=O)NC(C)C(C)(C)NC(c3c[nH]c(=O)cn3)=O)nc2n1 C1(N(C(=O)CC2CCC(C3CC3)O2)CC)CCN(C(C2(F)CCC2)=O)CC1 C1(N(C(CC=CCNC(C2N(CC)CCCC2)=O)=O)C)CCCCC1(C)C CCCC(CC)CCC(=O)NCCNC(C1CCCCN1CCC)=O CCCC(F)C(=O)NCCC1(NC(C2CCCN(CCC)C2)=O)CCC1 c1(CC(=O)NCC2CN(C(CC(C)c3cccs3)=O)CC2O)cc(F)ccc1O n1(CC(C)C)ccc(CC(N2CCC2CNC(C2CCOC2=O)=O)=O)n1 C(c1ccccc1[N+](=O)[O-])=CCNC(C1CC(O)C1n1cccn1)=O C(C1(O)CCc2ccccc21)NC(NNC(=O)OC(C)(C)C)=O c1(C2(NC(CCOC(CC)C3CCC3)=O)CC2)ncnn1C.N12CC(C1)C2=O c1(C(N(CC(CN(C(CCCC(C)=O)=O)C)O)C)=O)cc2c(F)ccc(F)c2[nH]1 C(=O)(C(CC)C(=O)N(CCCOCCNC(=O)CCc1ncc(C)[nH]1)C)OCC NC(=O)CCC(=O)N1CC(OCCNC(=O)Cc2cn[nH]c2)C1 C1CCC(=O)NC12CCC2.c1(C(=O)NC2N(C)CC2)ccnn1C1CC1 CC1(C)CCC(CC(=O)NC23CCN(C(c4sccc4C(F)F)=O)CC2C3)CC1 C1(C(=O)N(CCCC(C)O)C)(CC)CCCN(C(=O)C=CCF)C1 C(=O)(CCCCCSC)NC1CCCC(C(N(CC(CC)C)C)=O)C1 c1(C(C)C)cc(O)nc(NCc2cc(N3CCCC3)ccn2)n1 CC1(C(=O)N2CC=CCO2)CCCN(C(C2CCC(O)C2)=O)C1 S(=O)(=O)(c1cc(F)ccc1C(=O)O)NC(c1ccc(C(F)(F)F)cc1)C c1(OC)ccnc(C(=O)NCCNC(=O)CCSC(F)(F)F)c1OC N1(C(CC(CC)C)=O)CCC2(CC1)CN(C(c1nc(Br)c[nH]1)=O)CCO2 Cc1cccc(C)c1C(C)Nc1cc(C2CC2)cnc1Cl C1(NC(=O)CSc2cnn(CO)c2)CCN(C(C2CC(=C3CCC3)C2)=O)CC1F c1(C(=O)NCC2N(c3nccc(OC)n3)CCCC2)ncc(C#N)cc1C S(=O)(=O)(c1csc(C(=O)NC2CC(C)(CNC(c3ccn(C)c3)=O)C2)c1)NC Cc1cc(C(F)F)n(CC(=O)NCC2COC(CNC(=O)C(F)(F)C3CC3)C2)n1 c1(C(=O)NC2(CCCNC(C(C)OCC#C)=O)CC2)ccc(Br)c(N)c1 C1(C)(NC(C2(CCNC(C3CC(OC)C3)=O)CC2)=O)CC1(C)C CC(CCCNC(C1(C)C=CCC1)=O)NC(c1cc(C2CCCC2)no1)=O CC1(C(=O)NCC2CCC(NC(=O)C(F)(F)CC3CC3)C2)CC2CC2C1 n1(CC(=O)NCC2CC2C(N2CCOC(CC3CCC3)C2)=O)cccnc1=O C(=O)(CC1=NNC(=O)C1)N1CCN(C(CC(CC)C2CC2)=O)CC1C(=O)OC CCC(C)C(O)C(C)C(=O)N1CC(F)(F)CC1(C)CNC(=O)CC1CCCN1C C12(C(N(C(CCCC)C)C)=O)CCC(NC(c3cccc(C)c3)=O)(CC1)C2 N1(C(C)=O)CCC2CN(C(=O)C(C3CCCCC3)C3CC3c3sncc3C)CC2C1 c1(CCC(=O)NCC=CCNC(=O)COCC2CC2)ccccc1Cl c1(C(=O)NCC=C(C)c2cccs2)ccc(=O)n(CC2CCCC2)c1 N1(C(C(C)Cn2cccn2)=O)CCN(CCC(=O)NO)CC1.C1C(=O)N1 c1(SC)ccoc1C(=O)NC(C)CC(C)NC(C1CC(n2cnnc2)C1)=O c1(C(=O)NCC(CO)NC(CCc2ccc(C)s2)=O)ccc2sccc2c1 C=CCS(=O)(=O)CCNC(=O)NC1CC(C)(C)CN1 C(=O)(C(C(C)O)NC(=O)CC1CCCC(=O)C1)N1C(C)CCC1 C1(CC(=O)Nc2ccc(CNC(COC(CC)C)=O)nc2)COCC(C)(C)O1 CC1(C)CCC(C(=O)NCC2CCC2)(NC(C2C3CCC(F)(F)C23)=O)C1 N(C1CCCc2occc21)Cc1cc(C)n(-c2cccc(C(F)(F)F)c2)n1 N1(C(CCCCCN(C(=O)C(Cl)Cl)C)=O)CCC2CCCC2CC1 c1(OC)ccc2c(c1)OCC(C(=O)N1CCC1CNC(=O)CC1(O)CCC1)=C2 c1(OC)ccc2c(=NC(C)c3cc[nH]n3)[nH]c(=NCC(C)(C)C(F)(F)F)[nH]c2c1 N1(C(c2cc(CC(=O)OC)on2)=O)CCC2(NC(C3CCC(C)(C)C3)=O)CC2C1 N1(C(C(C)=CC)=O)CCCC(CCNC(=O)CCN2CCOC2=O)C1 c1(CC=C(C)C)cc(=NC(=O)C2CCCN2C(=O)Cc2ccc(O)nc2)[nH]n1C C(c1ccc(F)c(Cl)c1)=CC(=O)NCC#CCNC(c1c(C)nn(CC)c1C)=O C1(C#CC(=O)NCCCOCCN(C)C(C2(C)CCCN2C)=O)(CC)COC1 CCC(CN(C)C)CC(=O)N(C(C(=O)N(c1cccc(F)c1)C)C1CC1)C C1(C)(CNC(COCC=C)=O)CC(F)(F)CN1C(=O)C=Cc1cccnc1 C1(NC(C23CC2CNC3=O)=O)CC(O)(c2cn(CCF)nn2)C1 Cc1nc(C(C)C)oc1C(=O)NC(C)CC1CN(C(C2COC(C)C2)=O)C1 CC1CC(N=c2[nH]c(N3CCC(N4CCC4)(CO)CC3)nc3c2CCCC3)CS1 Cn1cc(C(=O)CNC(=O)C(F)(F)c2nccn2C)cn1 c1(C(=O)OCC)cccc(C#CCNC(CCO)C(C)(C)C)c1 C12(CC(=O)NCC(C)(O)CNC(c3ccc(F)s3)=O)CCC(CC1)C2 c1(N(C)C)ncc(C(=O)NC2CN(C(=O)CCNS(C)(=O)=O)CC2CO)cc1Cl CC(C)CCCC(C)C(=O)NC1(C(=O)NCCCCCC2CC2)CCC(C)(C)C1 CC1(C)CC(=O)NC1CNC(C1CC2(CC2)CN1C(C1CC(N(C)C)C1)=O)=O C(CCNC(C1COC1)=O)(C(C)C)NC(C(C)(C)OC)=O C=CC(C)(C)CC(=O)NCCN(C(=O)C(C)Sc1ccccc1)CC1CCCC1 Cc1cc(C(=O)NCCC2CC(NC(C3(CF)COC3)=O)C2)cs1 C(=O)(N=c1[nH][nH]c2c1CN(C(=O)C(F)(F)Cl)C2)c1cccc(C#C)c1 CN=c1nc(N(C)CC2CCCS2)[nH]c(=NCc2ccc(CCC)cc2F)[nH]1 C1(CNC(CC(=O)NCC2CC2)=O)CCC2(CCC2)C1NC(C1CCCC1)=O CC1CC2CN(C(c3ccc(F)cc3N)=O)CC2N1C(C1COCC1C(F)F)=O Cc1cccc(C)c1NC(=O)C(Cc1cc[nH]n1)NC(=O)CN1CC2CC2C1 CCC(CCOC)C(=O)N1CCC(O)(C(C)NC(=O)CCCCC2CC2)CC1 Cn1c(C(N2CC(C(=O)NCC3CC3[N+](=O)[O-])CC2(C)C)=O)cccc1=O C1(C(=O)NCC(C)NC(=O)CCCC2CCOCC2)(CO)CCO1 CCCCCCC(C)C(=O)NC(C)CNC(c1cc(F)c([N+](=O)[O-])cc1F)=O N1(C(COCCOCC)=O)CC(NC(=O)CSc2cccc(Cl)c2)CC1(C)C C1(CNC(CCc2ccn(C)c2)=O)(CO)CC12CCN(C(c1csnn1)=O)CC2 N1(C(c2c(SC)cccc2)=O)CC(NC(=O)CC2(C)CCCO2)C2(CCC2)C1 n1(CC(=O)NCC(C)NC(C2CC23CCOCC3)=O)cc(C#N)c(O)nc1=O N1(C(CCCC#C)=O)CCN(C(=O)Cc2cc(F)cc(F)c2)CC(C)(F)C1 C(CCCCC(=O)NC)NC.N1(C(CN(C)CC)=O)CCN(CC2CCCCC2)CC1 O=S(=O)(c1cccs1)N(CCCCO)Cc1cccc(OCC(F)F)c1 C=Cc1ccc(C(N2CC(NC(C3CC34CC(C)(C)C4)=O)CC(F)C2)=O)cc1 C1(CC(=O)NCC2(NC(C3COCCO3)=O)CCC2)CCCC(F)(F)C1 C1(NC(c2c(CC)cc(Cl)cc2)=O)CCN(C(C2COC(=O)O2)=O)C1(C)C C#CCC(C(=O)N1CC(F)(F)C1C1CC1)NC(=O)CC1CSCCO1 O=C(C=C(Cl)Cl)NCCC1CC(NC(=O)CCn2cnnn2)C1 c1(N2CCN(C(c3cc(Cl)ncc3Br)=O)C(CC#N)C2)ncnc2n[nH]c(Br)c12 CCC(C(=O)NC(c1ccccc1)C1CCCC1)N1CCCC1=O C(C(O)C(=O)NC1CC(O)C1CC(=O)N(C)Cc1c[nH]nc1C)=CC C1(CNC(NCC(F)=CC)=NCC2CC2)COC2(CCCCC2)O1 Cc1cc(C)c(CCNC(=O)Cn2cnc(C(F)(F)F)n2)c(C)c1Br N1(C(c2c(C)noc2)=O)CCCC(C)C1CNC(c1coc(O)n1)=O c1(C(=O)NC2C(C)N(C(C3CCC3)=O)CCC2)ccc([N+](=O)[O-])c2cccnc12 Cc1cc(C(=O)NCCC(C)(C)NC(=O)C2=NNC(C(F)(F)F)C2)ncc1F C1(NC(C2N(CCC)C(=O)CC2)=O)CC(O)CN(C(=O)CN2CCNC2=N)C1 c1(C(N2CC(NC(C(CCOC)C)=O)C(C(F)F)C2)=O)cc2c(C)cccn2n1 C(=O)(CC(F)(F)Cc1cccc(Br)c1)OCC(C1CC2CCC1CC2)OC CC#CCC(C(=O)N(C(C)CSC)C)NC(C1C2CCCCCC12)=O C1(COC)CN(C(c2ccc(CO)cc2F)=O)CCN1Cc1ccnc(Br)c1 C(=O)(C(CC)N(C(C)(C)C)CC)N(CCNC(C(COCC)C)=O)CC C1(C(N2C3C(NC(C4(OC)CC4)=O)C(C3)C2)=O)CC1C1CCCC1 c1(C(N(C(C)CNC(=O)CSCC(N)=O)CC)=O)cnc2n1CCS2 C1(CC(=O)NC(C#C)(C)C)CCN(C(=O)C=CC=CCC)C1(C)C C1(Cn2cc(C3(OC)CCCC3)nn2)CCN(C(=O)CC2NC(=O)NC2=O)CC1 C#CCCCCC(=O)NC1(CNC(C23CC2COC3(C)C)=O)CCCCC1 Cn1cc(Cl)cc1C(N1CCC(OCCNC(c2cncc(C3CC3)c2)=O)C1)=O c1(C(=O)NCC2(O)CC(NC(C(CC#C)C3CC3)=O)C2)ccn(CC)c(=O)c1 c1(C(=O)NC(C)CC(C)NC(C2CCOCC2)=O)ccc(C)c(C#N)c1 c1(CNC(C2CCCCCN2C(=O)OC(C)(C)C)C)ccc(S(=O)C(C)C)cc1 c1(CNC(C(CNC(C2CC3CC(=O)C2C3)=O)CC2CC2)=O)cc(F)cc(F)c1 c1(C2C(C(N(CC(C)NC(C(CCC)O)=O)C)=O)C2)cccc(Cl)c1Cl O=C(NNC(=O)C1CCCCC1)c1cc(-n2cncn2)on1.N12CCC(CC1)C2 C1(C(=O)NCCCCN(C)C(c2cccn2C)=O)CCC1(F)F N(C1CCc2c(F)cccc21)C(N1C(C(=O)OC)CC(F)(F)C1)=O Cc1c(N)ccc(C(N2CCCC(NC(C3CCc4n[nH]cc4C3)=O)C2)=O)c1C CCCC(CC)CCC(=O)NC(C)(CO)C(=O)N1CC(O)CC1C(C)C Cc1ccc(F)c(C(=O)NC2CC(=O)N(C3CN(C(=O)C=CCO)C3)C2)c1 C1(CNC(CCOCC(C)C)=O)CCN(C(c2coc(C#N)c2)=O)C1(C)C N1(C(COCCC#C)=O)CC2CCCC2C1C(=O)NCC1CCOCC1(C)C N1(C(c2ccc(C)c(O)c2)=O)CCC2CCCC12C(=O)N(CC(C)O)C CCCCC(C(=O)N(CCC)CCC)NC(c1cc(O)cc(Cl)c1)=O CCC(C(=O)N(CC(O)CN(C)C)C)c1ccco1.C1CO1.C(CN)O Cc1cc(C)n(CC(C)NC(C2CC2c2ccc(-c3ccsc3)cc2)=O)n1 N1(C(=O)NC2CCC(C(C)=O)CC2)C2(CC(N(C)C)C(O)C2)CC1(C)C c1(CC2(C(=O)NCCN(C(=O)CCC3CCCC3)C)CC=CC2)ccc(F)cc1 c1(C(=O)NCC(CCC)NC(c2[nH]cnc2C)=O)ccc(F)cc1F c1(C(N2CCC(c3cnn(C)c3)C2)C(=O)NCCOC)c(C)cnn1COC c1(C(N2C(CC(=O)NCC3(OC)CCCOC3)CC2)=O)cc[nH]c2nccc1-2 c1(CN2CC(CNC(c3ccc(CC)c(Cl)c3)=O)C2)ccc(F)c2ccccc12 c1(NC2C(CNC(c3c(C)ncn3C)=O)CCC2)ncc([N+](=O)[O-])cc1F N1(C(CCC=C(C)C)=O)CC(NC(=O)Cc2cc(Cl)ccc2O)CC12CCC2 CC1CC(NC(=O)CCc2cncs2)CCN1C(=O)C=Cc1ccoc1 c1(C(=O)NC2C(NC(CS(CCOC)(=O)=O)=O)CCC2)ccc2sc(C)nc2c1 N1(C(C(C)S(C)(=O)=O)=O)CC2CCCN(C(c3ncsc3S(N)(=O)=O)=O)C2C1 C(=O)(CC(CC)C(C)(C)C)NC(c1cccc(F)c1)C(N1CC(CC=C)C1)=O c1(C(=O)NC2CC(Nc3ccnc(Cl)n3)C2)cc2c(nc1O)CCCC2 N1(C(C2C3CC(=O)CC32)=O)CCC2C(C1)CN2C(=O)Cn1cc(C2CCC2)nn1 CC(C)(O)C(C(=O)Nc1ccc(OCCO)cc1)NC(=O)CCn1ccnn1 N#Cc1ccc(CN2CC(C(=O)Nc3ccsc3CO)CC(F)C2)c(Br)c1 CC(CC(F)F)C(=O)N1CCC(CN(C(=O)CCCC2CCCC2)C)C1 C(=O)(C(C)(C)C(F)(F)F)N(CC(C)NC(=O)CC(C(F)F)n1cccn1)CC C(=O)(C(=O)C(C)(C)C)NCC(CC(=O)N1CCC(C(C)C)C1)N(C)C c1(C(=O)NC2CC(CO)N(C(C3CC3F)=O)C2)cc(C2CC2)nc(O)c1 c1(CC)cc(CC)[nH]c(=NCCN(C(=O)CSC2CCS(=O)(=O)C2)CC)n1 c1(OC(C)C)cnc(N2CCNCC2NC(c2cc(CO)ccn2)=O)nc1 N1(C(C2C(CC)OCC2)=O)CC(CC(=O)NCc2ccsc2)CC1(C)C C(C(C)(O)CC(=O)NC1CCC1NC(=O)C=CCN(C)Cc1ccccc1)OC c1(C(=O)NC2C=CCN(C(c3c(C)c(Cl)cnc3)=O)C2)c[nH]c2nc(Cl)ccc12 c1(C(N2CC(C=C)C(NC(=O)C(C3(O)CCCC3)F)C2)=O)nccn2ccnc12 Cc1csc(CCC(=O)NCCCCNC(C2(CO)CCCO2)=O)n1 CC1CCCN(C(=O)C=C2CCOCC2)C1CNC(=O)COC1CCCC1 c1(C(=O)NC23CCN(C(C(C)(C)OC)=O)CC2C3)cc2sccc2n1C N=c1[nH]c(C(F)(F)F)ncc1C(N1CCC1CNC(c1cc(C2CC2)[nH]n1)=O)=O C1(C(=O)NC(C2(C(=O)NC3CC4CCC3O4)CC2)C)CC2(C1)CC21CC1 N1(C(C(CC)N(C)C)=O)CCC2CN(C(=O)Cn3cc(C#N)cn3)CC12 c1(C(C(N2C(C(N3CCC(O)CC3)C)CCC2)=O)C)c[nH]c2ccccc12 Cc1cc(CNC(=O)C(F)C2CCC2)oc1C(=O)NCCc1cscn1 c1(CC)noc(C)c1C(=O)NCC1CCC(C(=O)N)CC1.C1(CC2CC2)CC1CF c1(CC)c(N(CCNC(=O)Cc2ccc(C)cc2)CC)nc(C)nc1Cl c1(C(N2CC(NC(c3n(CC)nc(C)c3)=O)C(F)CC2)=O)[nH]nc2cnccc12 Cc1cc(C(N2CCOCC2CN(C)C(c2csc(C(N)=O)n2)=O)=O)cc(C)n1 c1(C(N2CC(C(N3CC(CCO)C3)=O)OCC2)=O)ccn2nccc2c1 C12(NC(c3c(C)cco3)=O)CCC(CNC(=O)C(O)(C3CC3)C3CC3)(C1)OC2 C(=O)(C1CCCc2cncn21)N(CCCN(C(=O)CC1CCCN1C)C)C c1(C(N(CC)CC)=O)cccc(CC(C)N)c1.c12ccc(cc1)N(C)C2 CCCCC(CC(=O)NC1CN(C)CC1(C)C)NC(=O)CNC(N)=O N1(C(C2C(C(=O)OC)C2)=O)CCCC(C(N2CC(n3ccnn3)C2)=O)C1C C(=O)(CCCn1cccn1)N(C1CCC(NC(=O)Cc2csnn2)C1)C Cc1[nH]nc(C(=O)NC2CC(CNC(C3(C#N)CC3(C)C)=O)C2)c1[N+](=O)[O-] C(C)(C(=O)N(CCNC(C1(C2CC2)CC1)=O)C1CC1)(C(C)C)NC(C)=O N1(C(c2c(C)onc2)=O)CCC2(CCOCC2)C(NC(C2C3COCC23)=O)C1 C1(CO)CCCCC1N=c1[nH]c(=NCc2cccc3ccsc23)[nH]c2c1CSC2 c1(C(=O)NC2CCCC(NC(C3CC(CC)(CC)C3)=O)C2)cc(Cl)cnc1C Cc1nc(C(=O)NCCOCCNC(=O)C(c2ccccc2F)O)c(Br)s1 CN1CCC(CC(=O)N(CC(O)CNC(c2nocc2C2CC2)=O)C)C1 c1(CNc2c(C(=O)Nc3cnc(C)c(Br)c3)nc[nH]2)cccc2c1OCC2 C1(C(=O)NCC(CC=C)NC(c2ccc(CO)o2)=O)(Cn2cccn2)CCCCC1 N1(C(c2c(C)scn2)=O)CC(C)(C)CC1CNC(c1ccon1)=O C1(CNC(c2ccc(CNC(C)=O)o2)=O)CCN(C(=O)CC(C)F)CC1(F)F C(C(C)(CC(C)C)NC(C1CC2CCC(C1)S2)=O)NC(C1(CC)COC1)=O c1(CNC(CC)(C2CC2)C2CC2)nc(-c2ccccc2)ncc1F C1(C2CC2)(CNC(CCC(=O)N(C)C)=O)CCN(C(C2(C)CC(C#N)C2)=O)C1 S(=O)(=O)(c1ccc(N2CCC3(CC2)N=N3)c(C#N)c1)NC(CC)COC c1(SC)cccc(F)c1C(N1CC2CC2(CNC(C2(O)CCC(C)(C)C2)=O)C1)=O C1(C)(CNC(C2(C(F)F)CC(=C)C2)=O)CCCN(C(c2cnc(N)cn2)=O)C1 N1(C(c2ccn(C)n2)=O)CCC(C)(CNC(c2cnn(CC3CC3)c2)=O)C1 N(C(=NCCNCCCS(C)(=O)=O)N1CCCC1)CCN(CCOC)CC N1(C(COCC#C)=O)CC2CC1C2C(=O)NN1C(c2ccccc2)CCC1 CCCC(C#N)C(=O)NC1CN(C(=O)NC2(C)CC(C(F)(F)F)C2)C1 C=CCC(CC=C)C(=O)NCCOC(C)C.c1(NCC)cc(O)cc(F)c1 C(C(C)(C(=O)NC1CCCC1(C)COC)NC(=O)CNc1cccnc1)SC C1(NC(C(C(C)C)=O)=O)CC(C)CN(C(c2cnn(CCF)c2)=O)C1 C1(C(C)(C)C)(CNC(=O)CNC(=O)C2CC2)CCN(C(=O)Cn2ncnn2)C1 c1(C(=O)NCCN(C(c2cccc(C(=O)OC)n2)=O)CC)cnccc1C(F)F C1(F)(C(C(CNC(CCNC(=O)OCC)=O)(C)C)=O)CCCC1.C(CF)OCC.NC Nc1c(C(N2CCC(O)(CCNC(c3coc(O)n3)=O)C2)=O)cc(Cl)[nH]c1=O N1(CCC)CCCCC1C(N1CCN(C2CC2)CC1)=O.C12CN(CCO1)C2=O N1(C(c2c(C)ccs2)=O)CC(C2(NC(=O)CCCN3CCCCC3)CC2)C1 Cc1nc(CCC(N2CC3CC3(CNC(=O)CN3CCSC3)C2)=O)oc1C C1(COC)(CNC(=O)C=C(C)C)CCCN1C(C1CCCO1)=O N1(C(CCC=CC)=O)CCCC2C1CCN2C(=O)C(c1ccncc1C)C c1(C(C(=O)NCC(CNC(c2nc(CCC)sc2)=O)(C)O)C)c(C)noc1C CCC(C)(F)C(=O)NC(c1ccc(C)cc1)CNC(c1cnc(S)n1C)=O Cc1cc(Cl)cc(NC(C2CC3CC3N2Cc2ccn(CCF)n2)=O)c1I Cc1cc(F)cc(C(=O)NCC2CCN(C(c3ccncn3)=O)CC2)c1C C#CCC(C)(CC)C(=O)NCC12CC(NC(c3scnc3COC)=O)(C1)C(C)O2 C1(C(N2CCC(C(=O)N(C)C)C2)=O)(NC(CCC2(C)N=N2)=O)CC(O)C1 Cn1c(C(=O)NCC2(F)CN(C(C3CC(=C4CCC4)C3)=O)C2)cc2sccc12 C(=O)(CC1=CCCCC1)N1C(CNC(C(C)Cc2ccc(F)c(F)c2)=O)CCC1 N1(C(COCC)=O)CCC(C(=O)Nc2cnc(Cl)cc2C(N)=O)C(O)C1 CC12CC(C(=O)NCCNC(=O)CC3(n4cnnn4)CCOCC3)C(CO1)C2 N1(C(C(CC)=CC)=O)CCC=CC1C(=O)ON1CC(N(C)C2CC2)C1 N1(CCC)CCCC1C(=O)NC1COCC1C(=O)Nc1cnn(CCC)c1 c1(C(=O)NCC#CCNC(C2C(C)C2)=O)cccc(N2CCCCC2)c1 C(=O)(CCN(CCO)C(=O)NC(C)C1CC1)NC(c1nncs1)C CN1CCC(C(N2CCCC2C2CCN(C(=O)CCOCC(F)F)CC2)=O)C1=O n1(CCOC)nc(C(=O)NCC2CCC(C)CN2C(=O)C2=C(C)OCC2)ccc1=O C1(CNC(=O)CCc2ccoc2)CCN(C(=O)Cc2cccc(F)c2O)CC1O c1(C(=O)NC(CCOC)CNC(c2ccn(C)n2)=O)ccc(C(=O)OC)cc1F N(C(=NCC(=C)C1CCOCC1)N1CCC(S(C)(=O)=O)CC1)CCC=C c1(CN(C)C)cc(C(=O)N(C2CCCN(C(C3(CO)CCC3)=O)C2)CCF)ccn1 c1(C(=O)NC2(C)CCN(C(C3CCC3)=O)C2)cc2c[nH]cnc-2n1 N1(C(CN2CC(C)C2)=O)CC2(CCN(C(c3cnc(O)cc3O)=O)CC2)C1 C1(CNC(COCC(=C)C)=O)CC(F)CN1C(=O)CC1CC(C)C1 CCCCC(CN=c1nc(C2CCCC2)[nH]s1)NC(c1cc(C)on1)=O Cc1ccc2c(c1)CCCC2N(C)C(C(C)(C)OC(C)(C)CSC)c1nnnn1C c1(CC)c(C(N2CC(C)(NC(c3ccnn3CC)=O)C2)=O)cnc2ncnn12 c1(C(=O)NCCCNC(c2c(C)nn(C)c2C)=O)ccc2nc(N(C)C)[nH]c2c1 N1(C(CC2CC(OC)C2(C)C)=O)CCC(NC(c2cc[n+]([O-])cc2)=O)CC(O)C1 C1(C(=O)NCCC2CCN(C(=O)CN3CCSCC3)C2)CC2CCC1O2 C(=O)(C(C)(C1CCC1)NC(=O)CC1COC(=O)C1)NC(C1CCCC1)C#C c1(C(N2CCC(SC)C2)C(=O)NCCCC)ccc(F)cc1Cl c1(OC)ccc2c(c1)CCCC(NC(C1CC(CN)C1)=O)C2 C(=O)(C1SCCc2sccc21)NCC1(NC(c2cc3n(n2)CCC3)=O)CCCC1 CC1(C)CC(C(=O)N(C2CCCC2)CCNC(C2(C#N)CC2C(F)(F)F)=O)=NO1 C1(CC(=O)NCC(CC)NC(C23CCCN2CCC3)=O)CC(C)(C)C(=O)N1 N1(C(C=C(CC)C)=O)CC2(C1)SCCC2NC(C1CC(=O)N(C(C)C)C1)=O Cc1c(CC(=O)N(C(C)CCNC(=O)CC2CC2(C)C)C)oc2ccccc12 CCC(CC)(C(=O)N1CC2CC(NC(C3(C(C)C)CC3)=O)CC2C1)C(C)C C=CCN(OC)C(=O)C1=NOC2(CCN(C(c3cccc(C)c3C)=O)C2)C1 c1(C(=O)NC(C(C)NC(c2ccc(C)cc2O)=O)C)ccn2c(C)cnc2c1 CN1C(=O)CCCC1C(N1CC(CC(=O)NCC(CO)C2CCC2)C2(CC2)C1)=O O=C(CCCCC1CC1)NCC1(NC(C2CCCC(F)C2)=O)CCCC1 N1(C(C23CCC(OC)C2C3)=O)CCC(CCOC)(NC(=O)CCC(C)(C)F)CC1 N1(c2n(CCOC)c(-c3ccc(C)c(C)n3)nn2)CCOC2COCC12 C(C(C)(C(F)(F)F)NC(=O)C(C)OC(c1cccc(OC)c1)=O)OC N1(C(c2n(C)ncc2Cl)=O)CC(NC(=O)CNc2ccccn2)CC(O)C1 C(CO)(CCCCNC(=O)C(C)(C)COC)NC(C(=O)Nc1cccc(OC)c1)=O Cn1nc([N+](=O)[O-])cc1C(N1CCC1CNC(C1CC2C=CC1O2)=O)=O C1(CNC(C=COCC)=O)(CNC(C2(c3cccs3)CC2)=O)CC12CCC2 c1(C(=O)NC(C)CC(C)NC(=O)CC2(C#N)CC2)ccccc1S(C)=O N1(C(c2n[nH]c(C3CC3)n2)=O)CCN(C(C2CN3CCN2CC3)=O)C2(CCC2)C1 C1(NCC(C2CCCC2)C)CC2OC(C)(C)OC2C1 C(O)CC(CO)NC(C1(C)CCN1C(C1CCC(N(C)C)C1)=O)=O c1(C(N2C(CNC(C(c3ccc(Cl)cc3)C)=O)CC2)=O)cnc(=NCCF)[nH]c1 c1(CC(=O)NCC(CNC(C(=O)NCC)=O)(C)O)ccc(F)cc1C c1(CNC(C2CC(NC(C(C)Cc3cnco3)=O)C2(C)C)=O)n[nH]c2c1CCC2 N1(C(C(=O)NCC)=O)CCCC2C(NC(=O)C=C3CCCC3)C(C)(C)C12 c1(NC2CCN(C(C3CCCN3CCF)=O)C2)ccnc(-c2ccccc2)n1 c1(C(=O)NC2CN(C(C3(OC)CCCC3)=O)C(C)C2)ncnc2sccc12 N1(C(C2(C)CN(C(C(n3c(C)ncc3)C)=O)C2)=O)CCC2(C=CCO2)CC1 c1(NC(c2cccc(CC(C)C)c2)c2n(CC(=C)C)nnn2)ccc(Br)cc1Cl c1(C(N2CC(CNC(C(C)n3ccnn3)=O)OCCC2)=O)cc(C#N)ccc1F C1S(=O)(=O)CCN=C2NCC(CCCO)CC3(CCC1N2)OCCO3 CC(C)(Cc1cnn[nH]1)C(=O)NCCNC(C1CCCCC1F)=O C1(C(=O)OC)CCCC(C(=O)NC2(C)CCN(S(=O)(=O)C3CC3)C2)C1 c1(C(=O)NC(C2CCCCN2C(=O)CC(=O)NC2CC2)C)cncc2sccc12 N1(C(COC)=O)CCC2CCCN(C(=O)COC3CCOCC3)C2C1 C#Cc1ccc(C(N2CCN(C(=O)CC3CCCOC3)CCC2C)=O)c(C)c1 Cc1nn(C)c(C)c1CC(N1CC(CC(C)NC(=O)C(=Cc2cnc[nH]2)F)C1)=O c1(C(C(=O)NC2CC2)N(C(C)CC(N)=O)CC#N)c(F)cccc1Br CN1CCN(C(C2CC(=O)NC(=O)N2)=O)C(CNC(=O)C(C)(C)C2CCCO2)C1 N1(C(C(C)OCCOC)=O)CC2(CC(NC(c3cc(C(C)C)no3)=O)C2)C1 C1(C(=O)NC2(C(=O)NCC(c3cn(C)nc3)O)CCCC2)CN2CCC1C2 c1(NC(CC(=O)OCC)C2=CCCC2)nc(Cl)cn2ccnc12 Cc1csc(Cl)c1C(N1CC(NC(=O)C(C(C)C)c2ccn(C)n2)C(O)C1)=O C(=O)(C(C)(O)C(F)(F)F)N(CCCNC(C1CCN(C2CC2)C1=O)=O)CC N1(C(c2c(C)snn2)=O)C2CCC1CC(NC(C1CC3C(C1)C3(F)F)=O)C2 N12CC=CCC1C2=O.C1(NC(=O)OCC)COCCC1C(=O)NC1CC(SC)C1 c1(C(N2CCOC(C3CC3)C2)C(=O)NCCCOC)ccc(C#N)s1 C(=O)(CCCCC(=O)N1CCC(CC(C)NC(c2cocc2C)=O)CC1)OC c1(C(=O)NCC2C(NC(c3occ(C)c3)=O)CCC2)sc(F)cc1Br C1(CNC(C(C)=C(C)C)=O)CC2CCC1N2C(=O)C(C)n1ccnc1 c1(OC)ccc(F)c(C(N2C(C(N3CC4CC3CO4)=O)CCC2C)=O)c1F C=CCCCC(C)(C)CNC(c1cn(CCNC(C2(CC(C)=O)CC2)=O)nn1)=O C(CN=c1[nH]c2c(c(=NC3CCOC(C)(C)C3)[nH]1)COC2)OC(C)C C1(C(N(CC2=CCCOC2)C)=O)CN(C(C2(C)SCCCS2)=O)CC1(C)C c1(NC(N2CCCC2)=O)ccc(Nc2cc(Br)cnc2O)cc1 N1(C(COCCC#C)=O)CC2CCCCC2(NC(=O)CC2(OC)CC2)C1 CC1CN(C(c2ccoc2C2CC2)=O)CC1CNC(=O)COCC(F)(F)F c1(OC)oc(C)nc1C(=O)NCC1CCC(NC(c2cc(CCCO)on2)=O)C1 C1(CNC(C(C(CC)O)C)=O)CN(C(c2[nH]nnc2C)=O)CCC12CCOCC2 Cc1cc(C#N)cnc1C(N1CC(NC(C2CCCC(=O)N2)=O)CC1C)=O C1(OCCC#N)CCN(C(C2CC2)C2CC2)CC1.C(=O)(NNC(=O)N)C1CCC(F)C1 C(=O)(C1=COCCO1)N1CCN(c2c(CNC(C(C=C)O)=O)cccn2)CC1 C1(CC(=O)Nc2ccc(-c3cn(CCOC)nc3)s2)Cc2ccccc2C1O S(=O)(=O)(c1ccc(Cl)cc1)Nc1c(-c2ccc(C(=O)O)s2)ccc(F)c1 Cc1ccc(C(=O)C(=O)NCC(C)NC(C2(Cc3cccc(F)c3)CC2)=O)cc1 N1(C(C(C)N(C(C(C)OCCOC)=O)C)=O)CCCC(C)(C)C1C Cc1cc(F)c(CN2CC3CC3(C(=O)NCCOc3ccccc3)C2)cc1Br C12(CNC(CC(=O)NCC#C)=O)CCCC1N(C(c1ncccc1Cl)=O)CCC2 N1(C(c2ccc(C(N(C)C)=O)cn2)=O)CC2(CC2C#N)C1 c1(C(=O)NC2C(NC(C3(C#C)CCC3)=O)CC2)ccc(F)c(OC(F)(F)F)c1 N(C1CCCn2cnnc21)C(C1(NC(c2c(C)noc2)=O)CCCC1)=O C(C(C)(C)CC(=O)NC1C2CC1N(C(c1cnn(CCO)c1C)=O)C2C)OC C(=O)(C(C(C)(C)C)OC)NCCC1(O)CCN(C(c2c(OCC)nccc2)=O)C1 N1(C(C(C)n2cccn2)=O)CCC(CCNC(=O)CCC(C)(C)C)C(F)(F)CC1 c1(C(=O)NCC2CN(C(C3COCC(C)O3)=O)C2)ccc(Cl)c(F)c1F c1(NC(C(CC)(C)CNC(=O)CC2CNC(=O)O2)=O)ccc2nc[nH]c2c1 C12(C(=O)NCCNC(=O)CNc3ccccc3F)CCC(C(F)(F)F)(CC1)C2 c1(C(N2C(CNC(c3cncn3C)=O)CC(OC)C2)=O)ccc(Cl)nc1N c1(C(=O)NCc2c(C(=O)NCC3C(CC)CCO3)n(C)nn2)cccn(C)c1=O c1(CC)nc(C)[nH]c1NC(=O)NCC1CCN(C(c2ccccn2)=O)C1 C(C)(N=c1[nH]c(=N)[nH]c(=NCCc2ccc(Cl)cc2C)[nH]1)c1ncc(C)cn1 CN1CCN(C(=O)C(F)C2CCC2)C(C(=O)Nc2ccc(OC(F)F)nc2)C1 c1(CC)ccc(C(=O)N(C)CC2(C(=O)NC3(c4ccn(C)n4)CC3)CC2)cc1F C(=O)(C(C(=O)NCC=CCC(=O)N(C1CCC2CC12)C)OC)OC C(=O)(CCC(C)(C)OC)NCC(CC=C)NC(c1cnc(CC(C)C)[nH]1)=O N1(C(C(CC)F)=O)CCC(CNC(=O)C=Cc2ccncn2)C(F)(F)CC1 N1(C(C2CCC(N(C)C)C2)=O)CCC2(C1)CN(C(c1ccnc(O)c1F)=O)C2 CCCS(=O)(=O)C(C)C(=O)N(CC(C)NC(=O)Cc1cccnc1F)C C=C(C)CCN(Cc1ccc(CC2CC2)cc1)N1CC2CCOC2C1 C=CCCCC(C)(C)C(=O)NCC(C)(C)OCC(=O)NC(C)(C)C(O)CO CC1CCCCC1NC(=O)C(N1CCOC(CCN)C1)=O C1(O)(CCNC(c2c(CC)ncs2)=O)CCN(C(=O)COc2cccc(F)n2)C1 C1(C(=O)NCCN(C(C23CC(O)C2C3)=O)CC2CC2)C2CCC1(c1cscn1)C2 c1(C(=O)NCC2(NC(c3cc(O)cs3)=O)CC2)ccc2c(=O)ccoc2c1 CC1CCN(C(c2cn(C(C)(C)C)nn2)=O)CCN1C(C1CCCCC(=O)C1)=O c1(N(C(C(CC(C)C)O)=O)C(c2ccc(F)cc2)CO)ncnc2cccnc12 N1(C(c2nc(C)oc2)=O)CC(C(=O)NCCC2COCCO2)C(F)C1 CC1(c2ccccc2)CN(C(=O)NCC2CCCC23CC3)CCO1 c1(C(=O)OCC)c[nH]c(=NCC2(C)CCCN(C(c3sccc3F)=O)C2)cn1 N1(C(C(CC(=O)OC)C)=O)CCC2CN(C(c3cn(CCO)nn3)=O)C2C1 CC(=O)CCCC(=O)NC1CCCC1CNC(C1(C)CC1(C)C)=O c1(C(CNC(=O)CO)NC(c2nc(C)n(C)c2)=O)ccc2ccccc2c1 C1(C(=O)NC2C(NC(=O)CC3(O)CCCC3)CC2)Cc2nccn2C1 c1(C(N2C(CN(C)C(C3CC3C3CC3)=O)COCC2)=O)ccc(F)c(CO)c1 C1(NC(Cc2cc(C)on2)=O)CN(CC(N2CCCCC2)=O)CCC1C C1(N=c2nc(C(F)(F)F)[nH]s2)(CNC(C(C)(C)OC)=O)CC1 c1(C(N(C(CCNC(Cc2nnc(C)o2)=O)C)C)=O)ccc2occc2c1 N1(C(C(C)=C2CCC2)=O)CCC(NC(=O)C(C)n2cncn2)C(F)C1 N1(CC(N2C(CCNC(=O)C=CC3CCCC3)CCCC2)=O)CCS(=O)(=O)CC1 C1(C(N2CCC(C(F)F)(CNc3cnc(F)cn3)C2)=O)COc2ccccc2O1 N1(C(C2(COC)CC=CCC2)=O)CCC2CN(C(=O)CSC(F)F)CC2C1 N1(CCC(=O)Nc2cc(OC)cc(OC)c2)CC2CC(F)CC2C1 Brc1ccc2oc(-c3ccc(NCC4CCN4C4CC4)s3)cc2c1 N1(C(=O)CC2CCC=CCC2)CCN(C(=O)CCCC(F)(F)F)C2CCCCC12 C1(CNC(c2cc[nH]c2)=O)(CO)CCCN(C(C23CCCCC2C3)=O)C1 N1(C(c2c(C)[nH]cc2)=O)CCC(C2CC(NC(C3CCC=CCCC3)=O)C2)CC1 n1(CCC(N2CC(C)(NC(C(C)N(C)C)=O)C2)=O)cc(C#N)c(O)nc1=O c1(OC)ccc(S(=O)(=O)N2CCOC(CSC3CCC4(CC3)OCCO4)C2)cc1 C1(NC(C2C(C(N)=O)C2)=O)COC2(C1)CN(C(c1c[nH]c(=S)cn1)=O)C2 N1(C(Cc2nc(C)[nH]n2)=O)CCC(NC(=O)CN2CCCC2=O)CC1C NS(=O)(=O)c1ccc(C(N2CC3(CCCN3C(C3(O)CC3)=O)C2)=O)s1 Cn1ccn2ncc(CNC(C3CC4(CC4)CN3C(=O)OC(C)(C)C)=O)c12 C12(NC(C(C)O)=O)CCCC1N(C(=O)CCCOc1ccc(Br)cc1)CC2 c1(C(N2CC(C)C(CNC(=O)C=CCO)CC2)=O)cnn2c1CCCC2 C1(NC(C(C)SCCCC)=O)CCC(NC(c2cccc(CC(C)C)c2)=O)CC1 c1(C(N2C(CCOC)CN(C(=O)CC3CC3(C)C)CC2)=O)cc(S(C)(=O)=O)co1 c1(C(=O)NCC(C)N(C(c2c(OC)nn(C)c2)=O)C)c(Cl)ccc(C)c1N N1(C(C2CC(=C)C2)=O)CCCC2(NC(=O)CC3CCC34CCC4)CCCC12 Cc1cc(C(=O)O)ccc1CN(C)CC1CCC(F)C1 C(=O)(C#CC1CCCC1)NC(C(N1CCCC(C)(C)C1)=O)Cn1cncn1 C(=O)(C(CCCSCC)N1C(c2ccccc2)CCC1C)NCCOCC N1(C(CSc2ccc(C)cc2)=O)C(C(N2CCCC2C(N)=O)=O)C2CC(O)C1C2 c1(NC(C2CCCN2C(=O)Cn2cncn2)=O)ccc(O)c(CO)c1 c1(C(=O)NCC2CC(NC(C3CCC3(F)F)=O)C2)ccc2nc(C3CC3)oc2c1 C1(NC(c2cc(Cl)cc3c2OCC3)=O)CN(C(=O)C(F)F)CC2(CCC2)C1 c1(C(=O)N)ccoc1C(=O)O.c1(CCN(CCCO)C)ccccc1 C1(NC(C(C)N(C)C)=O)CC2CN(C(c3cc(Cl)cc(Br)c3)=O)CC2C1 c1(C(N)=O)cc([N+](=O)[O-])ccc1NC1CC(F)(CNC(c2ccnc(F)c2)=O)C1 c1(C(N2CC(NC(C(C)NS(C)(=O)=O)=O)C(F)CC2)=O)ccc2ccn(C)c2c1 c1(OC)ccc(CC(C)C(=O)N(C)CCN(C)C(c2ccc(Cl)cn2)=O)cc1 N1(C(c2cnc(OC)s2)=O)CC(C2(NC(=O)Cc3ccncc3Cl)CC2)C1 C1(CNC(c2cc(C)nn2C)=O)CN(C(=O)CC2CCC(C)CO2)CC12CC2 Nc1ccc(C(=O)NCCC2CN(C(C3CCC(O)C3)=O)CCO2)nc1N N1(C(C23CC(CO)(CN2)C3)=O)CCOc2c(Br)cccc2C1 C1(CNC(c2c(CC)c(C)sc2)=O)CN(C(C2CCC(=O)C2)=O)CC12CC2 C1(CC(=O)NCC(C)(C)NC(=O)CO)CNC(C)(C)CO1 C1(C(N2CC(NC(C(C)=C3CCC3)=O)C2)=O)CC(c2cccnc2)=NO1 C1(C)(CNC(CC2N(C(C)C)CCC2)=O)CCCN(C(C2CC(F)C(=O)N2)=O)C1 Cc1nc(CC(N2CC(c3csc(C4COCC4n4cccn4)n3)C2)=O)co1 C(=O)(C1=CCCCCC1)NC1CCC(CNC(c2cnc(CC(C)(C)C)[nH]2)=O)C1 C1(CC(=O)NCCCN(C(c2ccnn2CC2CCC2)=O)CC)CNC(=O)O1 Cc1ccc(F)c(C(=O)NC2CCCCC2NC(=O)CC(C)(C)C2CC2)c1F C(C)(C)(C(=O)NCCn1ccnn1)C1(C)CC1.C12CCC(C1)NC(=O)C2 C(=O)(C(CC(C)C)NC(c1ncncc1OC)=O)NCC(CCOC)O c1(C(N2CC(O)(CNC(c3ncncc3F)=O)C2)=O)ncccc1F C1(C(C)(C)NC(c2ccncc2)=O)CCN(C(c2coc(C3CC3)n2)=O)CC1 C12CC13CCN(C3)C2=O.c1(C(=O)Nc2ncc(CC)s2)cccc(C(F)F)c1 C1(C(=O)NC2CN(C(CCN(C)CC)=O)CC(O)C2)C2CCC3(COC(=O)C13)O2 C(=O)(C(C)(C#N)CC)NCC(C)NC(CN(C(=O)OC(C)(C)C)CC)=O C(C)(CC1CC1)(C(=O)Nc1cccc(F)c1)Oc1c(OC)cccc1 C(=O)(C(C(C1CC1)OC)N(CCCOC(C)C)C)NCCC Cc1cccnc1C(C)NC(C1C=CCN(C(=O)CC2CCCCC2)C1)=O N1(C(c2nc(CC)oc2)=O)CCN(C(=O)C(C)S(C)(=O)=O)CC1C N1(C(c2c(CC)nccc2)=O)CC(C(=O)NCc2ccc(O)nn2)CC(C)(C)C1 c1(C(=O)OC(CC)C#N)cc(C)n(C)c(=O)c1 C1(NC(c2cn(Cc3cnc(-c4ccccc4)s3)nn2)O)CN2CCCC2CO1 c1(CC(=O)NCC2CC(NC(C(CC)N(C)C)=O)C2)cc2ccccc2nc1O c1(C(=O)NCCCCC(CO)NC(CCCC(=C)C)=O)nccn2cc(C)nc12 C1(C(N(CC(N2CC(OCCN(C)C)C2)=O)C)=O)Cc2ccccc2C1(C)C C(CCCCO)N(C)C(C1(NC(c2ccn(C)c2)=O)CSC1)=O C1(O)(CNC(C(C)C2CCCC2)=O)CN(C(=O)CC2CCCC2O)C1 C1(C(=O)NCC(C)CN(C(=O)Cc2cccc(F)c2)C)CCC12CCC2 C1(NC(C=CCC)=O)C2CCC1N(C(C1(OCC)CCCC1)=O)C2 n1(CC)c(C(=O)NC2(C(=O)NC(C)C(C)n3cncn3)CCC2)cnc1O N1(C(c2c(OC)noc2C)=O)CCC2(C1)CN(C(C1CCC3(CC3)C1)=O)CCO2 c1(NC(c2cc(SC)oc2C)c2nnnn2C(C)C)ccc(C(N)=O)c(C)c1 c1(C(c2nnnn2CC)CC=C2CCO2)cccc(F)n1.CS(=O)(=O)CC1(CO)CC1 c1(NCC2N(C(=O)OC(C)(C)C)CC(F)(F)C2)c(Cl)cc(O)cc1Cl CON1CCC(C(=O)NCC2COCC2NC(C2(S(C)(=O)=O)CC2)=O)CC1 C1(C(=O)NC(C(=O)NCCNC(C)=O)CC2CCCC2)CCCCO1 C12(C(N3C(CSC)CCC3)=O)CC(CO)(CN1C(=O)C(c1ccn(C)c1)C)C2 C1(C(=O)NCC(C2CCC2)NC(c2c(CC)nc(C)o2)=O)CCCCC1(C)C C1(C(N(CCC)CC2CC2)=O)(CC)CCN(C(c2ccoc2CC)=O)CC1 C#CCC(C)(C)C(=O)N1CCN(C(=O)CC(c2ccccc2)NC(C)=O)CC1 N1(C(C(CC)C#N)=O)CCC(O)(C(C)N(C(=O)C(=O)N(C)C)CC)CC1 C1(NC(C2C(C)(Br)C2)=O)CN(C(c2cnn(C(C)(C)C)c2)=O)CC2(CCC2)C1 C1(COC)(COCC(C)Cc2cccs2)CCC1.C1C(OC)CN1 c1(CC)[nH]nc(Cl)c1C(N1CC(C)(NC(=O)C(C)OCC(C)C)C1)=O N1(C(C2(c3n(C)ncc3)CC2(C)C)=O)CCC(CNC(=O)Cc2ccsn2)CC1 c1(CC)nnc(CNC(c2n[nH]c(COC)n2)c2nnnn2CC(F)F)s1 C(=O)(C1=CSCCO1)N1CC2C(CNC(=O)Cc3cnoc3)(C2)C1 C(CCC1CC1)(C(=O)N1CC2(CCC2)C1)NC(c1ccc(C)o1)=O N1(C(c2cn(CCC)nc2)=O)CCC(NC(=O)C(N2CCCC(C)C2)=O)C(C)C1 C1(N(CC#C)C(c2ccco2)=O)CCN(C(C2CC(c3ccccc3)C2)=O)CC1 c1(CC(=O)NC2(C)CC(NC(C=CC(CC)C)=O)C2)cccc([N+](=O)[O-])c1C CN1CCOC(C(N2CC3CC3(CNC(c3ccsc3)=O)C2)=O)C1=O C(=O)(C1=CCCCC1)N(C1CN(C(C2C3CC(=O)CC23)=O)C1)C C1(C(=O)NCCCC=C)COC2(CCN(Cc3cc(Br)c(C)cn3)CC2)C1 C1(C(=O)NCC(CNC(c2ccn(C(C)(C)C)c2)=O)CO)CC2CCC2C1 C1(C(=O)NOCCOC(C)C)(CC)CCN(C(=O)CC(C)COC)C1 CCC(C(=O)NC1CC(NC(C2(OC(C)=O)CCC(C)(C)C2)=O)C1)C(C)(C)CC c1(C(C(=O)NCC2CCCO2)N(C(CC=C)C)C2CC2)cnc(OC(C)(C)C)s1 C(=O)(CC(F)(F)F)N1CC(CC=C)(C(=O)NCc2nccn2C2CC2)C1 c1(CNC(C(C)OCCOC)=O)ccc(C(N2CC(N(C)C)C2)=O)cc1 c1(C(=O)NCCC(C)NC(c2cccc(NCC#C)c2)=O)ccc(C)cc1F c1(CNC2C(C(=O)Nc3c(C)cncc3)CCC2)ccc(Br)nc1Br C12(C(=O)NC3C4(CN(C(=O)C(F)=C5CCC5)C4)CC3)CC3CC(C1)CC(O)(C3)C2 N1(C(C(C=CC)O)=O)CC(NC(c2cc(C(N)=O)no2)=O)Cc2ccccc21 Cc1cc(Cl)c(C(=O)N(CC(O)CNC(=O)C=CC2CCOC2)C)cc1[N+](=O)[O-] Cc1cc(=O)n(C)nc1C(N1CCC(C2(NC(c3cccc[n+]3[O-])=O)CC2)C1)=O CC(=O)CCCC(=O)NC(C1CCOC1)CNC(c1cccc(C(C)(F)F)c1)=O C#Cc1ccc(CNC2CCCCC2C(=O)NCC2CCC(F)(F)C2)cc1 C12(C(=O)NCC(N)=O)COCC1CN(c1nnc(SCC3CCCO3)s1)C2 c1(C(=O)NC2C(NC(COCC(=O)NC)=O)CC2)csc(=NC2CC2)[nH]1 c1(C(C)NC(c2cnc[nH]2)=O)ccc2c(c1)CN(C(C1C(C)(C)C1(C)C)=O)C2 c1(NC(c2ncccc2NC(c2ccc(Cl)nc2F)=O)=O)ccc(Cl)c(I)c1 N1(C(C(C=C)O)=O)CCCC(C2CN(C(=O)C(C#N)CC)C2)C1 C1(C(=O)NCC(O)C(=O)NCC(C)C2CCC2)(CC)CCNC1=O C=C(C)CC(C(=O)N1CC(O)(C(F)(F)F)C1)NC(=O)C(C)c1cccs1 N1(C(C(C)C#N)=O)CCCC(C2CN(C(=O)Cn3nnc(C4CC4)n3)C2)C1 C1(NC(c2c(C)n3c(s2)cnc3)=O)CCC12CCN(C(c1cnc(S)[nH]1)=O)CC2 C1(C(=O)NCCC2(O)CCC2)CCCN(C(C2COCOC2)=O)CC1 CC(C(CO)NC(=O)C(C)(C)C1CCCCO1)NC(c1cc(C2CCC2)[nH]n1)=O c1(C(CC)OC)cn(Cc2ccc(C(=O)NCC3CC3(F)F)o2)nn1 N1(C(CCCC=C)=O)CCN(C(=O)CCc2nccn2CC)C2CCCC12 C(C(=O)NCC(C)CC1CC1)(C1CN(C(c2nccs2)=O)C1)OC C1(NC(C=C(C)C(F)F)=O)CCOC12CCN(C(c1ccc(CO)cn1)=O)CC2 c1(COC)ccc(CN(C(c2ccccc2)(C)C)Cc2ccco2)cc1 C1(C(=O)NC2CC(C)N(C(C3(C)CCCCC3)=O)CC2)CCc2nnnn2CC1 C1(C(N(C)CC2CCN(C(C=CCCC(C)C)=O)C2)=O)C2CC3C(C2)C13 c1(OC)ccc(CC(N2CC(C3CC3)OC(C)C2)=O)c(C(=O)O)c1 Cc1cc(NC(=O)C(C)CN2CCOC(C(C)(C)C)CC2)cc(C)c1 CC1CN(C(=O)C(C)O)CC(C(=O)NCCC2CC2C2CC2)O1 C(=O)(C(C)(C)C(C)(F)F)N1CC(C)C(NC(=O)C(C#N)C(C)(C)C)C1 N1(C(C=CC(C)(C)C)=O)CCCCC12CN(C(C1(Cl)CC1(F)F)=O)C2 C1(CNC(=O)CN2CC=CC2)(CO)CCCN(C(c2n[nH]cc2Cl)=O)C1 N1(C(C(=O)NC(c2ccc(C(C)C)cc2)C)=O)CCc2ncccc2C1C c1(C(N(CC(CC)C)C)=O)ccc(CNC(C2C3CC(=O)CC23)=O)cc1 c1(C(N2CC(O)(CNC(c3nc(CCC)oc3)=O)C2)=O)cc(C2CC2)nc(Cl)c1 C(Cc1c[nH]nc1O)(C(=O)O)NC(c1cnn(C2CC2(F)F)c1)=O C(=O)(C(C)(C)CCCF)N1CCCC(CC=C)(NC(=O)C(C)OC)C1 c1(C(N(C)CC2CCN(C(=O)CC(O)CN(C)C)C2)=O)cc2c(ccn2C)[nH]1 c1(NC(C2C(c3onc(COC)n3)C2)=O)ccc(Cl)cc1Cl C1(NC(c2c(C)ocn2)=O)CCC(F)(CNC(=O)C(C)(O)C2CCC2)C1 C1(NC(CC(C)Oc2ccc(F)cc2)=O)CC2CN(C(c3cn[nH]c3)=O)CC2C1 C1(O)(C(C)C)CCCN(CC2(CN)CNC2)C1 c1(C(=O)NCC(C)NC(=O)CC2CCC(=O)NC2)ccc(Cl)c(C(F)(F)F)c1 N1(C(CN(C(C)=O)C)=O)CCOCC1CCNC(c1cc(O)n(C)n1)=O C#CCS(=O)(=O)CCNC(=O)Nc1cccc(C(=O)OC)c1 N1(C(C2CCOC2)=O)CCN(C(C2(Cl)CC2)=O)CC1c1ccc(F)c(F)c1 C1(C(N(CC(N2CC(Sc3ccccc3Br)C2)=O)C)=O)CC2CCC1O2 N1(C(CC2(CNC(C3(O)CCSCC3)=O)CC2)=O)CC(O)C(O)C1 CC(C)(C)C(=O)NCCC(=O)NCCCOCC(=O)NC1CC1F.O C(N=c1[nH]ccc(=NCc2ccc(C(C)(F)F)cc2)[nH]1)c1c(C)cco1 Cc1ncc(C=CC(=O)N(CCCNC(C23CC(C)C2C3)=O)C(C)C)s1 CC(C)C(C(=O)N1CC2CC1(CNC(C1CCC1)=O)C2)NC(N)=O Cc1ncc(Cl)c(C(N2CCC(O)(C(C)CNC(c3cc(C)sn3)=O)C2)=O)n1 CCCC(CO)NC(=O)CC=CCNC(c1coc(C2CC2)n1)=O c1(NCC2(CC)CCCC2)ccncc1S(=O)(=O)NCCCN(C)CC c1(NCCCOC(CC)(C)C)cc(=NC(C)Cc2cnc[nH]2)[nH]c(C)n1 Cc1cn(-c2ccccc2)nc1C(=O)Nc1cnn(C2CCS(=O)(=O)C2)c1 N1(C(CC(=C)Br)=O)CC2(COC(CNC(c3cnc(C)cn3)=O)C2)C1 Cc1cccc(C(O)C(=O)NC2(C)CN(C(C34CCC(CO3)C4)=O)C2)c1F c1(OC)cc(C(N2CCC(CNC(=O)C(C)CSC)C2)=O)ccc1OCC(C)C C1(C(=O)NC(C2CN(C(Cc3nc(C(C)C)sc3)=O)C2)C)CC1C1CC1C c1(C(C)C)cc(C(=O)NC2CCCC2CNC(=O)COC(F)(F)F)ccc1F N1(N(C(=O)CSC(F)F)C)CCN2C(=O)NCC2C1.C1(C=O)CCCCC1C CC1(C)CC(C(=O)OC2CCC3(CCC3)C2)C(C)(C)O1 C(=O)(CC(C)(C)C)NCC(CN(C)C(c1cc(C2CC2)on1)=O)(C)C c1(C(=O)OC)c(C(=O)NCC(C)NC(c2ccc(CSC)cn2)=O)cccc1F CC(F)(CNC(=O)Cc1nc[nH]n1)CNC(c1cc(Cl)n[nH]1)=O CC(CO)C(=O)NC1(C2CCCN2C(c2ccn(-c3ccncc3)n2)=O)CC1 c1(C(N(CCn2cc(C(C)O)nn2)CC2CCC(=O)N2C)=O)cc(C2CC2)nn1C N1(C(C(C2N(C(C=C(C)C(C)C)=O)CCCC2)C)=O)CC2CC(C1)N(C)C2 c1(C(N2C(C(=O)NC(C34CC(CO3)C4)C)CCC2)=O)ccncc1Cl c1(SC)ccc(CNCc2ccn(CC(F)(F)F)n2)o1.C12CCC(C1)C(=O)N2C CC(C)C(N=[N+]=[N-])C(=O)NCc1nocc1C(=O)NCC1C(C)C1C c1(C(=O)NC(COCC)CO)coc(CNC(=O)C(C)OC2CC2)n1 C12(NC(C=Cc3cnc(C)s3)=O)CCC(CNC(C3OCCCO3)=O)(C1)OC2 c1(C(N2CCC(N(C)C(C3CC3CF)=O)C2)=O)[nH]c2ccccc2c1Br c1(OC)ccc(C(=O)CN2CCCC2C(N2CCCC(O)C2)=O)cc1 C(=O)(C(CCN(C)C)NC(c1coc(CO)c1)=O)NCC1(CO)CC(C)C1 N1(C(C=CCC)=O)C(C(=O)NC2COCCC2OC)CCC12CC2 C(=O)(CC1=CCOCC1)NC(CC)CN(C(=O)C(c1cn(C)nc1C)O)C CC1CN(C(C2C(C)C2C)=O)CCCN1C(=O)CCCSc1ccc(Cl)cc1 CCC(COc1sccc1CN1CCCCCC1)CC(F)F.C1(C)C(=O)O1 C1(OCC)CC2(C1)CC2C(=O)NCC1(NC(=O)Cc2cc(C)nn2C)CCCC1 C1(C(=O)NC(CSCC)C(=O)NCCN2CCOCC2)CC12CCCCC2 Cc1ccc(O)c(CC(=O)NCC2CCN(C(=O)CCF)CC2)c1 C1(NC(CCC#C)=O)CC2(CCN(C(=O)CC3COCC4(CCC4)O3)CC2)C1 N1(C(C2(OC)CCCCC2)=O)CC2CCC(C1)N2C(=O)CCc1cnc[nH]1 C1(C(=O)NC(C)CCCNC(c2nnc(S)n2C)=O)(CC)CCC(O)CC1 Cc1cc(C(=O)NCC2CC2C(=O)NCC(C)(C)C(=O)N(C)C)ccn1 C(=O)(CCCN(C(=O)C(C)OCCCC)C)N(CCCC)CCO C1(C(c2nnnn2C2CCOC2)NCCCSCC=C)C2(CCC2)C12CCC2 C1(C(=O)OC)CCN(C(c2ccc(CNC(c3ccc(Cl)o3)=O)nc2)=O)C1C c1(CC(=O)NCC(CNC(c2cc(C)sn2)=O)O)ccccc1CC(N)=O N1(C(CCC(C(=O)OC)(C)C)=O)CC2CCCC1CN(C(c1csnc1Cl)=O)C2 C(=O)(CCCCC(C)=O)N1CCC(C(=O)N(C)CC2CCOC2)(OC)C1 N1(C(c2sc(C)c([N+](=O)[O-])c2)=O)CC2(C1)CN(C(=O)C1=COCCC1)CCO2 C1(C(=O)NCCN(C(=O)C2=COCCO2)C(C)C)CCC2(CC1)NC(=O)NC2=O C1(CNC(CC2N(C(COCCC=C)=O)CC2)=O)(CO)CC=CC1 c1(NCC(N2CCCC(c3nc4ccccc4[nH]3)C2)=O)csc2cc(Cl)cnc12 C1(CNC(C(C)=C(CC)C)=O)CN(C(=O)C(C)(C)CCC)CCN1C C12(C(N3CCC(CC(C)NC(c4cc(CC)[nH]n4)=O)CC3)=O)CCOC(C)(C1)C2 c1(C(=O)NCC(CC)(C)NC(=O)Cc2c[nH]nc2O)cccn2c(O)nnc12 c1(NC(=O)N(C2CCC(n3cccc3)CC2)CC2CNCCO2)cccc(F)n1 N1(C(CC(C)CF)=O)CC2CCCC2(CNC(c2ncn(C)n2)=O)C1 c1(CNC(C=CC)=O)n[nH]c2c1CN(C(=O)CCCc1ccc(O)c(F)c1)CC2 C1(C(=O)NC2CCNC2=O)(NC(c2coc(CO)c2)=O)CCCCC1 CC(C)CC(CNC(C1(CNC(=O)CSC2CC2)CC2(CC2)C1)=O)CO C1(NC(C2(COC)CC2)=O)CS(=O)(=O)C12CCN(C(=O)C(C(=O)OC)OC)CC2 c1(C(=O)NC(C2CCN(C(=O)CC(O)C3CC3)CC2)C)cc2ccccc2n1C N1(C(COC)=O)CCCC(NC(=O)CCOc2cncc(NC(C)=O)c2)CC1 C1(C(C)NC(Cc2nc(C)[nH]n2)=O)CCN(C(=O)CC2CC2(Cl)Cl)CC1 N1(C(c2c(OCC)scc2)=O)C2CCC1CN(C(=O)CC(C)(C)C(=O)OC)C2 C1(CNC(C(CC)F)=O)(COC)CCN(C(C2(C(C)(C)C)CCC2)=O)C1 N1(C(CN(C)CC)=O)CC(NC(C2CC2C(C)(C)O)=O)CC12CCCCCC2 C1(NC(=O)COCc2nc[nH]n2)CCC(CCNC(c2cnn(CCF)c2)=O)C1 CC1(C(N2CCN(C(c3cc(C(N)=O)[nH]n3)=O)CC2)=O)CCC12CCC2 c1(OC)ccc(C)nc1C(N1CCSCC1CCNC(=O)CCc1cscn1)=O n1(CC(=O)NCC(C2CCC2)NC(C(C)C2CCC2)=O)ccc([N+](=O)[O-])n1 C(=O)(CCC1C(=O)Nc2ccccc21)NCC(CNC(C(C)=C1CC1)=O)O C(=O)(C(F)CCC(C)(C)C)NC(C(=O)NC(C=C)CO)(C)CO Cc1coc(C(C)C)c1C(=O)NCCC1CCCCN1C(=O)C(F)OC(F)(F)F C(=O)(C1=NNC(=O)CC1)N1CC(C#N)(CNC(C2=C(C)CCC2)=O)C1 c1(SCc2cn(C(C)NCC(C)(C)CC3CCCCC3)nn2)c(Br)c(C)nn1C c1(CC(N2CC3C(CNC(C4(C)COC(=O)N4)=O)C3C2)=O)ccc2sccc2c1 C1(C(=O)NCC)(CNCc2ncc(-c3ccc(F)cc3)[nH]2)CCOCC1 c1(C(=O)NCCNC(c2ccc(CN(CC=C)C)cc2)=O)cc(C)cc(Cl)c1 c1(C(=O)NC(CNC(C(CCC)NC(N)=O)=O)C)cc(C)cc(Br)c1O n1(CC)nc(C)cc1C(N1CCN(CCN(C)C(C2CS(=O)(=O)C2)=O)CC1)=O Cn1cnc([N+](=O)[O-])c1NC(=O)C(=O)NC1CCC(C)(O)CC1 N1(C(C(CC)(C)C)=O)CCC(C2(NC(c3cnc4sccc4c3)=O)CC2)C1 C1(NC(C=CSC)=O)COC2(CCN(C(C3(C4CCCCC4)CC3)=O)C2)C1 C1(OC)(CNC(C2OCCOC2C)=O)CCN(C(c2ccc(CO)nc2)=O)C1 N1(C(C2(C)CCC(=O)NC2)=O)CC23CCCC2(C1)CN(C(=O)Cn1cnnn1)C3 N1(C(c2cc(OC)no2)=O)CC12CC(O)(CNC(=O)CCC(N)=O)C2 Cc1cn2nc(C(N3CC(NC(=O)CCC(F)(F)F)C4(CC4)C3)=O)cc(C)c2n1 c1(NCc2cc(OC)nn2C)[nH]c(=NC(CCO)C(F)F)nc2c1ncn2C c1(C(=O)NC(CN(C(c2c(SC)scc2)=O)C)C)ccc2c(C)noc2c1 O(NC(=O)C(CCOCCO)NC(c1ncncc1Cl)=O)CC(=O)N(C)C c1(-c2cc(C(F)F)[nH]n2)nc(-c2nc[nH]n2)nn1Cc1ccncc1 C1(CNC(CN(C)CCO)=O)CC(O)CN1C(=O)CCNC(C1CCCO1)=O C1(C2CCCCC2)(C(=O)NC2C(NC(CN(S(C)(=O)=O)C)=O)CS(=O)(=O)C2)CC1 CCCCC(CC(=O)N(CC1=CCCOC1)C)NC(=O)C(C)c1ccco1 Cc1noc(C(=O)NCC2(Cc3ccccc3)CC2(C)C)n1.N12CC(CCl)(C1)C2=O C(=O)(C(C)CS(C)(=O)=O)C=O.n1(C(N(CCN(C(C)C)N)C)=O)cc(C2CC2)cn1 c1(C(N(CC(O)CNC(c2cnc(C3CC3)s2)=O)C)=O)cccc(CF)c1 c1(C(=O)NC2CC3C(NC(=O)CC4CC(F)(F)C4)C3C2)ccc2ccnn2c1 CC(C)C(C(=O)NC(C)CF)NC(=O)CN1CCCNC1=O C1(NC(CCOC(C)=O)=O)CN(C(C23CCC(C)(C2)OC3)=O)CCC1C C1(CC(=O)NCCC2N(C(CCN(CC)CC)=O)CCC2)CCC(=O)N1C Cc1ccnnc1C(=O)NC(C)(CNC(c1ccc(CN(C)C)[nH]1)=O)C1CCC1 C=CCCCC(C(=O)NCC(C)(O)C1CCCC1)NC(=O)CCCCSC N1(C(CNC(CC(C)C)=O)=O)CC2C(CNC(=O)Cc3nccn3C)C2C1 c1(OC(C)C)cnccc1CO.CC1C(=O)N2CC(C2)C(O)C(=O)NN1C1CC1.N(C)C c1(OC)cnc(F)c(C(N2CC(NC(c3cn(C4CC4)nn3)=O)CC2C)=O)c1 c1(C(N(C)CC2CCN(C(C=C(C)C)=O)CC2)=O)cc(Cl)cc2nc(C)[nH]c12 C1(C(N2CCC(CC(C)NC(c3cnc(N)cn3)=O)CC2)=O)CCC(=O)N(C)C1 c1(C(N(C(c2ccccc2)CNC(=O)CSC(C)(C)C)C)=O)cc(F)n(C)n1 C1(NC(C2CN(C(=O)OC)C2)=O)CN(C(c2cc(F)cc(C#N)c2)=O)CCC1(F)F c1(C(=O)NC2CCC(N(C(=O)Cc3csc(S)n3)C)C2)cc([N+](=O)[O-])cnc1O c1(C(N(CCCCNC(C2C3(CC(OCC)C3)C2)=O)C)=O)occ2c1CCCC2 C1(CNC(c2n(C)ccc2)=O)CCCC2(CN(C(C3CCCCC3(C)C)=O)C2)O1 C1(CC(C)NC(c2ccc(CCC)s2)=O)CCN(C(c2cnccc2C)=O)CC1 C(=O)(C1=C(Cl)CCOC1)N1C(CNC(C2CN3CCC2CC3)=O)CC(O)C1 Cc1oc(S(N)(=O)=O)cc1C(=O)NC1CC(NC(=O)Cn2cn[nH]c2=N)C1 c1(C(N2CC(NC(c3ccc(OC)s3)=O)C3C2C3)=O)ccc([N+](=O)[O-])c(C)c1 c1(C(=O)NCCCO)ccc2c(c1)CN(Cc1cc([N+](=O)[O-])ccc1O)C2 N1(C(=O)C=Cc2cccs2)CC2CCC(C1)N(C(C1COC1)=O)C2 CN1N=CC(CC(=O)NCC(C2CC2)NC(c2cccc(C(C)(F)F)c2)=O)C1=O N1(CC(=O)NCCC(C)(C)NC(c2c(SC)scc2)=O)CCCCCCC1=O C1(NC(C2OCCC(NC(C=CCN(C)CC)=O)C2)=O)CCCC1(C)CC1CC1 C1(C(=O)NCC2CCN(C(Cc3c(C)scc3)=O)C2)CC12CC(F)(F)C2 Cc1cc(C)c(C(=O)N(C2CC(NC(=O)COCCCF)C2)C)cn1 CCC(C)C(CC(=O)NCc1ccc(Cl)nc1)NC(c1cccc(CC#N)c1)=O c1(NC(=O)NCC(CC)(C)Cl)ccc(OCCOC(C)CC)cc1 Cc1cc(N)cnc1C(N1CCOC(C(N2CCC(C)(C(C)C)CC2)=O)CC1)=O c1(CC2(OCCCN(C)CNc3cccnc3)CC2)cc(F)ccc1F C1(C(N2CC(CN(C)C(c3cc(CC(C)C)ncn3)=O)C2)=O)(CC)CCNC1=O c1(C(N(CCN(C(C(C)CC2CCCO2)=O)C)C)=O)[nH]ncc1C#N C1(NC(CCOC)=O)COCCN(C(c2cn(C)nc2-c2ccco2)=O)C1 c1(OC(C)C)ccc(C(C)C(=O)Nc2ccc(C(F)(F)F)nc2)cc1 c1(C(=O)NCC2CC(C)N(C(=O)CCCN=[N+]=[N-])C2)cnc2c(c1)NCC2 C#Cc1ccc(F)c(C(=O)NC(CNC(c2cc(Cl)c(C)c(OC)c2)=O)CC)c1 c1(C(N2CCC(C)(CN(C)C)C2)C(=O)NCCOCC)ccc(F)cc1C C1(CCNC(C(C)(C)C2(O)CCC2)=O)CCCCN1C(=O)Cc1ccc(O)cc1 c1(C(N2CC(C)(NC(C(C(C)O)N(C)C)=O)C2)=O)c[nH]c2ccc(F)cc2c1=O c1(C2C(OCC)CCN2C(c2cc(C)ns2)=O)cc(C#N)oc1C C(C(=O)NOCCF)(C1CC1)N(C1CCCCC1)C(CN1CCC(C)C1)=O Cc1cc(CNC(=O)CC2CC2CNC(=O)C(C)OCC2CC2)ns1 Cc1cc(CNC2CC(NC(c3cnc(C)o3)=O)C2)cc(C)n1 c1(C(=O)NC2CC(NC(C3N(CCCC)CCCC3)=O)C2)ccc(OC)c(Cl)n1 C(=O)(C(C#N)C(C)C)N1CC(N(C(COc2cc(C)on2)=O)C)C(O)C1 CCCCC(O)C(C)C(=O)NCCOC(C)(C)CNC(C12CCC(C1)OC2)=O c1(OC)c(C(=O)NC2CC2c2cccs2)cnn1-c1ccccc1 C1(NC(C2CCC(CC)O2)=O)CCCCN(C(=O)Cc2nc[nH]n2)C1 c1(C(=O)NC2(CC=C)CCN(C(=O)CC3CCCCO3)C2)ccn2c1CSCC2 C1(CN(C(C2C=CCCC2)=O)CC)CCN(C(C2C(C)C2C)=O)CC1 c1(C(=O)NCC(=C2CN(C(=O)Cc3ccccc3)C2)F)cc2occc2s1 CN1CC(C(N2CCC2CNC(=O)CCCc2cccs2)=O)NC1=O C1(C(=O)NCC2CC(OC)C2)(CC)CCCN1C(=O)Cc1c[nH]nc1O c1(NC(N2CCC(CSC)C2)=O)cccc(C)c1Br C=CCC(C)(CC=C)NC(C1CN(C(=O)CCSCC(C)C)CC1(C)C)=O C1(N(C(=O)C(c2cncn2C)O)C)CCN(C(C2(C)C=CCCC2)=O)CC1 c1(NC(Cn2cc(C(=O)OC)nc2)=O)cncnc1CN(C1CCCC1)C N1(C(CC(=O)NCC)=O)CCCC(NC(C2CC2(F)F)=O)C(F)C1 c1(C(=O)OC)cccc2nc(NC(C3CCC4CC4C3)=O)[nH]c12 N1(C(CC(C)SC)=O)CC2(C1)SCCC2NC(c1nnc(S)n1C)=O c1(C(=O)NC(COC)(C)Cc2ccc(NC(=O)C(C)C)cc2)cc(F)cnc1O c1(C(N2C(C)CC(NC(C=CC=CCC)=O)C2)=O)cncc(N)c1C C1(=CC(=O)NCC(C)OC)CCN(C(=O)CCC2CC2(C)C)CC1 c1(-n2c(CSc3nnnn3C)nc(COC(C)C)n2)ccc(Br)c(F)c1 C1(C(=O)Nc2c(C)cccc2)CN(C(c2c(C)noc2N)=O)CC1(F)F c1(C(N(C2CCN(C(CCOCC)=O)C2)C)=O)ccc(C)c(C)c1Cl CC1(C)COCCC1C(=O)NC1(C)CC(C(=O)NCC2(CO)CCCO2)C1 C1(C2CC2)(NC(c2c(C(=O)O)occ2)=O)CCOC1 c1(C(N2C(C(N(CCOC)C)=O)C3CCC2C3)=O)cc(Cl)cc(Cl)c1O C1(N2CC(C)NC(C)C2)CCN(C(=O)Cc2ccc(Br)cc2Cl)CCC1C CCCCCC(O)C(C)C(=O)N1CC(O)(CNC(C2CCSC2)=O)C1 N1(C(C(c2c(C)nn(C)c2C)C)=O)CCCN(C(=O)C(C)N2CCCC2)CCC1 c1(C(=O)NC2CC(C)(NC(C3(CC)CCC3)=O)C2)cccc(F)c1Br c1(C(CNC(=O)C=CBr)NC(C(CSC)OC)=O)ccccc1F C=CCCCC(C)NC(=O)CC1CCCCC1NC(C1CCC1C#N)=O c1(OC(C)C(=O)NCc2ccc(CNC(=O)C=CC3CC3)cc2)ccc(F)nc1 Cn1ccc2c(C(N3CC(NC(=O)CSc4nncn4C)C(F)C3)=O)ncnc12 Cc1nc(CN(C(=O)C#CCNC(C2CCO2)=O)C)n[nH]1 Cn1c(SCCC(=O)NCCCOCCNC(=O)C(N)=O)nc2ccccc12 Cc1occc(=O)c1OCC(=O)NC1CCC(C)N(C(C2CC2F)=O)C1 c1(C(C(=O)N(CC(C)NC(C2OCCCO2)=O)C)O)cc(F)cc(F)c1 C=CCC(CNC(C1CC(CC)C1)=O)C(=O)NCc1cc(C(C)C)no1 CCC(C)CCCCC(=O)NC(CC1CC1)CC(=O)NCC(C1CCCC1)C N1(C(C(CCC)(C)C)=O)CCC2(CCCC2C(=O)Nc2n[nH]c(C(F)(F)F)n2)C1 CC1=NN(C)C(=O)C1CC(=O)NCC(c1cccc(C(=O)O)c1)O C1(CNC(C2(CO)CC(C)(C)C2)=O)CC2CCC1N2C(=O)C(C1CCCCC1)O C(c1cccc(O)c1)=CC(=O)NC(C1(C(=O)Nc2cnc(CC)nc2)CC1)C C(=O)(C1CCCc2ncnn21)NC1(C)CN(C(c2cccc(F)n2)=O)C1 C(=O)(C(C)(C(C)C)NC(C)=O)N(CCNC(C1CC1C#N)=O)CC C(=O)(CCCC(=O)N1Cc2c[nH]nc2C1)N(C(=O)CCC1CCCCC1)C c1(CNC(C(c2cnn(C)c2)C)=O)c(Br)ccc2ccccc12 C1(CNC(CC)=O)CCC(NC(C2C3CN(C)CC23)=O)CC1 N1(Cc2ccc(N(C)C)cc2O)CCC(F)(F)C(C(=O)Nc2ccnc(Cl)c2)C1 C(=O)(CS(=O)(=O)C1CCCC1)N(CC(C)NC(C1(F)CCCOC1)=O)C N12CCOC(C1)CC(=O)N1CC(CC1C)SCC2=O.CCCCOC c1(C(N2CC(C=C)C(NC(C3C=CCS3)=O)C2)=O)cc2ccccn2c1 c1(C(N(CCNC(=O)C(C(C)C)OCC)CC)=O)cn2cc(Cl)ccc2n1 C1(CNC(c2c(CCNC(CCCCN(C)C)=O)n[nH]c2)=O)OC(=O)NC1(C)C CC1C(NC(C23COC(CCO2)C3)=O)CC2CCC1N2C(=O)CCCN=[N+]=[N-] c1(C(=O)NCCN(C(=O)CC=C(Cl)Cl)CC(C)O)cc(Cl)cc(Cl)c1F Cc1cc(NC(=O)C(=O)NC2CC3CC(C(C)(C)C)CC23)cc2cccnc12 Cc1nn(C)c(C)c1C(=O)NC1CC(F)(CNC(=O)CCc2cncc(O)c2)C1 N1(CCC)CCCC(NC(C2(CO)CCCOC2)=O)C1.C(C)(C)(C)O N1(C(c2cc(C)oc2)=O)CCC(F)(CNC(C2(CO)COC2)=O)CC1 c1(C(=O)NC2C3CN(C(C4CCN(C(C)=O)C4)=O)CC2C3)ccc(C)c(C)c1O N1(C(CCn2ccc(C)n2)=O)CC2CC(O)C1C2NC(c1c[nH]c(=N)o1)=O c1(-c2scc(C(C)C(=O)NC3CC(C)(NC(=O)CCF)C3)n2)ccc(F)cc1 N(C1CCCc2occc21)C(CCN(C(=O)C(C)OCCN(C)C)CC#C)=O c1(C(N2CCN(C(Cc3nnc(C)s3)=O)CC2C)=O)ccc(N)c(N)c1F Cc1cc([N+](=O)[O-])c(F)c(SCCCCC(=O)OC(C)(C)C)c1F c1(C(=O)NC2CN(C(c3csc(C)c3N)=O)CC(C)C2)[nH]nc2c1CCC2(C)C CC1(C)C=C(C(=O)NCC(O)CC(=O)NCc2cccnc2O)C1 O=C(N=c1cc(C2CCOC2)[nH][nH]1)C1CN(C(C2CC(O)C2)=O)CCS1 c1(N2CCC(C)C(NC(c3cc(CF)on3)=O)C2)nc2cccc(F)c2s1 c1(CC)cccnc1C(=O)NCCOCCN(C(=O)CC1(C)CCCO1)C N1(C(CN(C(C)=O)C)=O)CCCCC(N(C(=O)Cc2cc(F)cc(Cl)c2)C)C1 C(C1CCN(C(=O)CCc2ccc[nH]2)CC1)=CC(=O)N(C)CCn1ccnc1 c1(C(=O)NCC(CNC(=O)C(F)(F)CO)CO)ncc(Cl)cc1F N1(C(CC(C)O)=O)CCC2C(C(=O)NCCc3ncc[nH]3)C2C1 c1(C(=O)NC2CC(NC(CS(CC)=O)=O)C2)cc(O)nc(OC)n1 C(CC(C)C)(C(=O)NCc1cc2occc2[nH]1)ONC(=O)C1CC1CCC C1(C(N2CC3C(CNC(Cn4c(C)nc(C)n4)=O)(C3)C2)=O)OCC2CCCC1C2 CC1(C(=O)NC23CC2COC3(C)C)CCN(C(C2CCCC2F)=O)CC1 N1(C(C(C2CCOCC2)OC)=O)CC2(CCC2NC(=O)CCCc2ccsc2)C1 N1(C(C(C#C)(C)C)=O)CC2(NC(C3CCOC3c3nccn3C)=O)CCC1C2 C(=O)(C1=CCc2ccccc21)N(CCCN(C)C(C1CC2CCC1C21CC1)=O)C C(C)(C)(CCC(=O)NC1(C)CCCOC1)SC.c12cccc(n1)Cn1cc-2nn1 c1(C(N(CCCNC(CC(=O)OC)=O)CCO)=O)ccc2ccn(C)c2c1 C(CC(=O)N1CCOC(CCNC(C2CCCN2C)=O)C1)(C(F)(F)F)OC C(CC(=O)N(C)Cc1nncs1)(C(F)(F)F)NC(CC=C)=O c1(OC)cccc2scc(C(=O)NC3(C)CN(C(C4CCN(C(C)C)C4)=O)C3)c12 CC1CN(C(c2cc(O)ccc2F)=O)CCN(C(C2CN3CCN2CC3)=O)C1 Cc1cc(N)c(C(N2CCCC(NC(c3nnn4ccccc34)=O)C2)=O)cc1C c1(NC(C=C)C)[nH]c(=NCC2OCCCO2)nc2c1ncn2C(C)C N1(C(CN(C)CC)=O)CCN(CCN(C)C(c2cnc(SC)[nH]2)=O)CC1 c1(NC(CNC(C(COC)C)=O)C(C)(C)C)ccc(C(F)(F)F)cc1[N+](=O)[O-] C(N=c1[nH]nc(C(N)=O)s1)C1CN(C(C(=C(C)C2CC2)F)=O)CC1C Cn1c(Cl)cnc1NC(N1CC(c2n[nH]c(C(F)(F)F)n2)C1)=O C(C(=O)NC(C)CCCNC(C1(c2ccc(C)nc2)CC1)=O)(C(C)C)NC(C)=O c1(NCC(C)N(C(=O)C(C)CC2CCCCC2)C)nccc(S(C)(=O)=O)n1 C=CC(C)(CCOC)C(=O)N1CCN(C(=O)CC2(CNC(C)=O)CC2)C(C)C1 C(N=c1cc[nH]c(=NCCc2cc(C)n(C)n2)[nH]1)C1(OCC)CCS(=O)(=O)CC1 N1(C(c2c(CC)nns2)=O)CCOC(CCCNC(=O)COC(F)F)C1 N1(C(CS(C)(=O)=O)=O)CCC(O)(CNC(c2ccnc(CO)c2)=O)CC1 C1(C2CCCN(C(=O)Cn3nnc(C)n3)C2)(NC(CC2CC(OCC)C2)=O)CC1 CC1(C(=O)NCCC2CCCN(C(=O)C=Cc3cccs3)C2)CC(C#N)C1 N1(C(Cc2nc(C)sc2C)=O)CC2CCCC2(NC(c2ncccn2)=O)C1 c1(C(=O)NC(C)CCNC(C2(C)CC3(CC3)C2)=O)ccc(N)c2ccccc12 C(CCCCCCCO)=CC(=O)N(CCC(C)NC(c1cn2c(n1)CCC2)=O)C Cc1cccc(SCC(=O)NC2CCCC2NC(C2CC(C#N)C2)=O)c1 c1(C(=O)NC(CN2CCN(C(CC(CC)OC)=O)CC2)C)ccc2ncnn2c1 C1(C(=O)NCC(CO)NC(CC(CC)OC)=O)CCN(C)C(=O)C1 N1(C(C2(C)C=CCCC2)=O)CC2(NC(=O)C3=CCCCO3)CCC1C2 c1(C2C(C(=O)Nc3ncccc3Br)C2)c[nH]ccc1=Nc1ccccc1 c1(C(N(CCCN(C(C(C)n2cccn2)=O)C)C)=O)cc2cc(F)ccc2cn1 N1(C(C(C)OCCOCC)=O)C(C(N2CCC(N(C)CC)C2)=O)CCC12CC2 N1(C(C2CCCN2C2CC2)=O)CCC(F)(F)C(CNC(C23CCC(C2)C3)=O)C1 C(CCCOC)(C(=O)NCC(C)(C)C(C)(C)C)NC(c1[nH]cc(C(C)=O)c1)=O c1(C(N2C3CN(C(c4c(CC)occ4)=O)C(C3)C2)=O)coc2c1CS(=O)(=O)C2 CCC(CO)(C(=O)N1CCC(CCC(=O)NCC(C)C2CC2)C1)OC CC1(C)CCc2onc(C(N3C4CCC3CN(C(=O)C(C)(C)CF)CC4)=O)c2C1 C(c1cnc(O)nc1O)=CC(N1CC2(CCN(C(=O)C(Cl)=CCl)C2)C1)=O C(CCCCCNC(C1C(Cl)(Cl)C12CC2)=O)N(C(=O)C(C)O)C c1(CNC(CCCC(=O)OC)OC)cnc2n1NCCC2 N1(C(C2C(C=C)CC2)=O)CC(CNC(c2cccnc2OCC)=O)CC(C)(C)C1 c1(C(N2CCC(N(CCC)C(C3CC3C)=O)CC2)=O)cc(F)cc2c1CCC2 CC(C)CC(CC(C)C)C(=O)N1CCCC2(NC(C3CCNC3=O)=O)CCCC12 N1(C(=O)OC(C)(C)C)CCCOCC1CCN(C(=O)CC(F)(F)F)CCO C1(C(=O)NC(C)CCNC(=O)C(C(C)C)N(C)C)CNC(=O)CC12CCOC2 CCCCC(C(=O)NC1CC12CCN(C(=O)CN(C)CC)C2)C(C)C CC1CCOCC1C(=O)NCC(CO)NC(c1ccsc1)=O c1(CNC(COCCNC(C2(CC)CC2)=O)=O)cn(C2CCN(C)C2)nn1 c1(CNC(CCOC2CN(C(C3CC(=O)N3)=O)C2)=O)cccc(CO)n1 c1(OC2CN(C(C(CCC)OCC(N)=O)=O)C2)ccc2c(c1)CCC2 N(C1CCCc2ccccc21)C(c1c(Cl)c(OC)cc(OC)c1)=O C(C)(C(C)(C)C(=O)NCC(O)CC1CCC1)NC(CCC#CC)=O C1(NC(C2(C)C(C)C2)=O)CN(C(c2ccc(O)c(CO)c2)=O)CC1C1CC1 N1(C(CC)C)CCN(C(c2ccc(I)s2)C(=O)N)CC1.C(C)(C)(CC)CC(=O)N O=C1CC2CCC2(C(=O)NC2CC3CC(NC(=O)COCC(F)F)C2C3)C1 C(N=c1ccnc(C)[nH]1)C1CCCCN(C(CNS(CC)(=O)=O)=O)C1 c1(OC(C)C)cccc(-c2cn(C3CCCCC3C(F)(F)F)nn2)c1 C1(CNC(CSCC#C)=O)CN(C(=O)COc2cccc(Cl)c2)CCO1 C1(CNC(c2n(CC)nnc2C)=O)CCN(C(=O)CC(CC)C2CC2)C(C2CC2)C1 C1(NC(c2ccns2)=O)CCSC12CN(C(=O)C(F)(F)c1nccs1)C2 c1(NC)cc(C(=O)NCC2CC3(CC(NC(=O)C(C)N(C)C)C3)C2)cc(Cl)n1 N1(C(c2n(CC)ccc2)=O)CC2(CNC(C3(C#N)CCCCC3)=O)CCC1CC2 C(=O)(C1=CCCCC1C)N1CCC(C(F)F)(CNC(C(CC=C)OC)=O)C1 CC1CCc2[nH]c(=NCc3ncc(Cl)n3C)[nH]c(=NCCP(C)(C)=O)c2C1 Cc1cccc(Cl)c1C(N1CCCC1CC(N1CCCC(O)C1C)=O)=O C1(CC(=O)N(CCC)CCN(C)CC2CCOC2)CCN(Cc2ccccc2)C1 C1(COC)(NC(=O)CC(C)(C)O)CCN(C(c2ccnc(C(F)(F)F)n2)=O)CC1 CC1(C(=O)NC2CCOC2)CC12CCN(C(=O)C(c1ccc(O)cc1)=O)CC2 c1(CC(=O)NC(C(C(C)C)NC(=O)CC2CCC2)C)c[nH]c2cnc(Cl)cc12 C1(C2CCN(C(C3CCCS3)=O)C2)(NC(c2c(C)cnnc2)=O)CC1 CCCCC(=O)C(=O)N1CCCC1CCC(N1CCOC(C)C1C)=O C1(C(=O)NC2CN(C(c3cn(CC4CC4)nn3)=O)CC2F)Cc2ccccc2S1 c1(C(N2CCC(c3cnn(C)c3)C2)C(=O)NCCC#N)ccc(CO)o1 CC(CCN(C)C)C(=O)N1CC2C(NC(c3cc(C(C)(C)C)c[nH]3)=O)C2C1 N#Cc1cnc(NCC2CC3CC3C2)s1 C(CC(O)C(=O)NCC(C(C)C)NC(C1CCOC(=O)N1)=O)SC C=CCCCCCCCC(=O)NCC(O)CNC(c1cccn1C)=O C(C(=O)N1CCC(NC(c2cc(Br)c(C)o2)=O)C1C)(C(F)(F)F)OC(C)=O C1(C)(NC(Cc2c(C)non2)=O)CCCN(C(c2ccc(C(=O)OC(C)C)[nH]2)=O)C1 C1(C(N2CC(C(CC)C)C2)=O)CC(NC(=O)Cc2nocc2C)CCO1 C12(NC(CC=C)=O)CCC1CN(C(C1(C)CCC(C)CC1)=O)C2 C1(CNC(C2(C(C)C)CC2)=O)CCN(C(C2(Sc3ccccc3)CC2)=O)CC1C c1(OC)cc(OC)c(CNCC2(C#N)CCOCC2)cc1Br c1(CNC(=NC)NCC(C)(C)CCCO)cccc(S(N)(=O)=O)c1 N1(C(C(c2cn(C)nn2)NC(c2cnc(S)nc2)=O)=O)CC(F)(F)C1C1CC1 CC1OCCN(C(=O)C#CCNC(=O)C2CC2)C1C c1(C(N2CCCN(C(C(CC=C)(C)C)=O)CC2)=O)cnc2nccn2c1 C1(CC)CCC(C(=O)NCC(CNC(c2[nH]ccc2COC)=O)OC)O1 Cc1ccc(C(N2CCCCC2CCNC(C23CCC(C2)C3)=O)=O)cc1O C(=O)(C(F)(F)C(C)(C)O)N1CCCC(C)(CC(=O)N(C)Cc2cn[nH]c2)C1 C#Cc1ccc(C(=O)NCC(C)NC(C2C(C)C2C)=O)cc1C N1(C(CC2(OC)CCC2)=O)CCC2(C1)CN(C(C1CCCCN1C)=O)C2 c1(C(N2CCC(C(N(C3CCN(C)C3)CCC)=O)C2)=O)cccnc1Br C(=O)(CC(=O)NCC(C1CCCC1)NC(=O)CN1CCCC1C)NCC CC1C(C)N(C(C2(n3cccn3)CC2)=O)CCN1C(c1ncnc(O)c1Cl)=O Cc1cc(C(N2CC=C(CNC(=O)CC3CC3C)CC2)=O)sc1C N1(C(C(C)N(C)Cc2ccccc2)=O)CC(NC(=O)CC2CN(C)C2)CC(O)C1 C(=O)(C1=CCCC1C)NC(CN(C(C1(c2cccnc2Cl)CC1)=O)CC)C N(C)(C[Si](C)(C)C)C(C)C.C(CCC(=O)NC)CCCCC1CC(C#N)C1 C1C(C)CC(=O)N1.C1(CC#C)(C(=O)NCCOCCN(C)C)CCCC1 c1(C(N(C(CNC(C2CCN(CCC)CC2)=O)CC)C)=O)cnc2c(c1)CCC2 Cc1ccncc1CCNC(=O)C(C1(C)CC1)NC(C1CC1(F)Cl)=O C(=O)(CCS(N)(=O)=O)NCc1nn(C)c(C(=O)NC(C2CC=CCC2)CO)c1 CCC(C)C(=O)NCC(N1CC=CC1CNC(C1CC(CN(C)C)C1)=O)=O C(=O)(C1Cc2ccc(F)cc21)NC(CNC(c1ccc(O)cc1)=O)C1CC1 C(=O)(C#CC1CCCCO1)N(C(C)C)CCNC(=O)CCC1CCOCC1 N1(CC2ON=C(C)C2)CCC(O)C(C(=O)N(CC(N2CCCCC2)(C)C)C)C1 c1(C(N(CC(CNC(c2c(CC)cno2)=O)O)C)=O)nccc2ccn(C)c12 S(=O)(=O)(c1cnc(NC(c2ccc(OCOC)cn2)C)cc1C)NC(CC)(C)C CN1N=C(C(=O)NC23CCCC2N(C(=O)C=CC2CC2)CCC3)CCC1=O CCCC(C(=O)N1CC(C)(C)C1CC(=O)NCCN(C)OC)N(C)C Cc1cc(C(=O)NCC2(CNC(C3CCS(=O)(=O)N3)=O)CCC2)ccc1C(F)F N1(C(Cc2c(C)non2)=O)CCN(C(=O)CCSCC(C)C)C(C)C1 N1(C(C=C(C)C)=O)CCC(CNC(=O)CN2CCCNC2=O)C12CCC2 N(C(=NCCCCCCOC(C)(C)C)NCc1ccccc1)CC1(C)CCCS1 CS(=O)C1CCC(NC(C2CCC(Oc3cccc(Br)c3)CC2)=O)C1 C1(CNC(c2nc(COC)oc2)=O)CN(C(C2CC3CC3C2)=O)CC1C(F)(F)F C1(C(N2CC(C3CN(C(C(CC=C)CC)=O)C3)C2)=O)Cc2cc(Cl)ccc2O1 c1(NCC(C2CC2)SC)nccc(=NCCCc2ccc(O)nc2)[nH]1 N1(C(c2cc(COC)no2)=O)CCOC(CN(C(=O)C(C)CCOC)C)C1 c1(OC)cc(I)c(C(=O)NCC2(C(N3CCOC(C)C3CO)=O)CC2)cc1OC N1(C(C=CCOCCOC)=O)CC(CNC(=O)C=CCCC(C)C)CC1C CC(C)(CCCN=c1ccc(C#N)n[nH]1)NC(=O)CCC(F)(F)F C=CCC(C(=O)NC1CCC(C)(C)C1)NC(c1sncc1C)=O C12(CNC(Cc3n(C)ccc3)=O)CCN(CC1)CC2.C12CC(C1)NC2=O n1(C2(CC)CC2)cc(C2CC(C(F)(F)F)(NC(C)CN3CCOCC3)C2)cn1 c1(NC2C(NC(Cc3c(C)c(F)ccc3)=O)C2)nc2cc(Br)ccc2o1 N1(C(C2CCCN(C(C3(CC)CC3)=O)CC2)=O)CCCC(C2CCC2)C1 C(=O)(C1CCCc2scnc21)N1C(CNC(c2n[nH]c3cc(O)ccc23)=O)CC1 c1(C(N(C(CC)CNC(c2ccn(C(C)C)n2)=O)C)=O)nc(C)ncc1Cl N1(C(c2c(CNC(C(C=CC)O)=O)n[nH]c2)=O)CC(CC)C(O)C1 CCCCC(C(=O)NCC1CN(C)CCN1C(C1CC2C=CC1CC2)=O)C(C)C CCCS(=O)(=O)C(C)C(=O)NCC1CCCN1C(c1ccc2nn[nH]c2c1O)=O c1(C(N2CCC(C(C)NC(C=Cc3ncc(C)[nH]3)=O)C2)=O)ccc(C)c(CO)c1 CC1=C(C(=O)N(CCCNC(c2cnn(C)c2F)=O)C2CC2)SCCO1 c1(OC)ccc(C(=O)NC2CCC(CNC(C34CCC(C)(C3)OC4)=O)C2)cc1Cl CC1(C)CC2(CN(c3cc(NC(=O)C(O)CC[S+](C)C)ncn3)C2)C1 c1(NC(C2(F)CCN(C(C3C(C#N)CC3)=O)CC2)=O)ccc2ncnn2c1 CC1COCC(C(C)(C)CNC(=O)N(CCC(F)=C(F)F)CCC#N)O1 C(C)(C)(C(=O)N(C)C(C1CCOCC1)C)N(C(C1(CC=C)CCC1)=O)CC.OC CC1C(NC(C2(C)CC=CC2)=O)CCN1C(c1cccc(OCC2CC2)c1)=O O=C(C1=CS(=O)CCC1)NC1(CNC(c2ccnc(Cl)c2O)=O)CCCC1 Cc1cc(C(=O)NC(CC2CC2)C(N2CCCC(C#N)C2)=O)nc(C)c1 C=CC1CN(C(c2cnc(-n3cccn3)cn2)=O)CC1NC(=O)CCC(=O)OCC CCC(C)(C(=O)N1CCC(C)(CNC(=O)Cc2cnc(C)nc2O)CC1)C(N)=O CC1CN(C(C2C3CN(C(=O)CC4CCSC4)CC23)=O)CC(C(N)=O)O1 C1(O)(CNC(C(C)OCCC#C)=O)CCN(C(c2cc(CCC)n(C)n2)=O)CC1 C1(C#N)(C(=O)NC(C)CCNC(c2cc(F)n[nH]2)=O)CC2CCC1C2 CC(C)CC(C(=O)NC(CO)C(C)NC(c1c2c(nn1C)CCC2)=O)C(N)=O N1(C(CC(=O)NCC)=O)CC(CNC(c2coc(Cl)n2)=O)C2CC12 C1(C2CCCCC2)(C(=O)NCCC2CCN(C(C3CC4(CSC4)C3)=O)C2)CC1 c1(C(=O)OC)ccoc1CNC(=O)COCC(=O)OCC(C)COC C1(C2CC2)(NC(C(N)=O)=O)CCN(C(c2cnnc(-c3ccccc3)c2)=O)C1 c1(C(=O)NC(C(C(C)C)NC(c2cnsc2)=O)C)ccc2c(c1)S(=O)(=O)NC2 Cc1cnc(C(N2CC(NC(C3CCCN3N=O)=O)C(F)C2)=O)cc1C#N c1(C(=O)NC(CNC(c2ccc(CC)nc2)=O)C)ccc(F)c(C(F)F)c1 c1(C(N2C(CNC(CCCN(C(C)=O)C)=O)C=CC2)=O)ccnc(C(C)(F)F)c1 O=C1CC(=O)NC(C(=O)NCc2ccoc2C(=O)NCC2CC2C2CCC2)C1 CCCCCCCCC(C)C(=O)OCC1C(C(=O)OC)C1(C)C C1(C(N(CC(CO)(CO)NC(C2CSC2)=O)C)=O)C2CCCCCC12 c1(CC(N2CC(CCn3cc(CSCC)nn3)C(OC)C2)=O)cccc(C#N)c1 CC1CCC(NC(c2cnc(=N)[nH]c2)=O)CN1C(=O)Cc1cccc(F)c1 N1(C(c2c(N)nccn2)=O)CC=C(CCNC(c2csc(Cl)c2Cl)=O)CC1 C(=O)(CC(C)(C)C)NC(C)C(=O)N(C(C)CNC(c1cc(O)n(C)n1)=O)C C(=O)(C(C)C(C)(C)C)N1CC(CNC(c2cc(CCC)c(C)s2)=O)C(C)C1 C1(CC(=O)NC2CCC2NC(c2cc(Cl)cs2)=O)CCCCC1O c1(C(C(C)NC(=O)Cn2cnnn2)NC(C2C(CCC)C2)=O)ccccc1 CS(C)(=O)=NCC(=O)NCC1CCN1C(=O)COCc1ccncc1F C1(CC(=O)Nc2ccc(Br)c(C(=O)O)c2C)(OC)CC2(CCOCC2)C1 CC(C)C(CNC(c1cc(C2CCCN2C)[nH]n1)=O)NC(C1CNC(=O)C1)=O Cc1cn(C(C)C)cc1C(=O)NCC(O)CCNC(=O)CCc1ccn(C)c1 C(CCCCCCCCCO)NC(C1(CNC(c2c(NC)cccc2)=O)CC1)=O N1(C(c2c(C)scn2)=O)Cc2[nH][nH]c(=NC(=O)c3ccc(O)cc3)c2C1 C1(C(N(C)CC2CCN(C(=O)Cc3cccnc3)C2)=O)CCC2(CCCC2)CC1 c1(C(N(CC(CNC(C2CC(OC)C2)=O)C)C)=O)cc2c(Cl)nccc2o1 Cc1ncc2cc(C(=O)N(CC(C)(C)NC(C3C4C5CCC(C5)C34)=O)C)ccn12 C1(NC(C2(C)CC(=C)C2)=O)CCCC(CNC(c2cc(Cl)c(Cl)s2)=O)C1 Cc1ccn(CC(=O)NC(C)CNC(c2cc(-n3ccnc3)cs2)=O)n1 C1(C(N2CC(NC(c3ccnc(C)c3C)=O)C2)=O)CC2CCCC(C1)C2 C1(C(N2C(CCC=C)CCC2)=O)(NC(c2conc2CC)=O)CCCC1C c1(C(=O)NCC(CC)NC(C2CCOC2c2ccnn2C)=O)ccn2ccsc12 Cn1ccn2ncc(C(N3CCN(C(C4C(C5CC5)C4(F)F)=O)C(CO)C3)=O)c12 CCCCC(=O)C(=O)NCc1ccc(CNC(=O)Cc2ccc(C)nc2Cl)c(F)c1 C(=O)(C1=CCCCC1C)N1CC(CC=C)(C(=O)NCC2CC(CO)CO2)C1 Cc1oc(C2CC2)nc1C(=O)NCC1CCCN(C(c2cn(C3CC3)cn2)=O)C1 c1(CC(=O)NC2(CC(=O)OCC)CNC2)c(Cl)c(SCC)nn1C N1(C(c2nc(OC)oc2)=O)CCN(C(C2CCC3(CCC3)C2)=O)C(CO)C1 C12(NC(c3cc(-c4ccc(C)cc4)no3)=O)CCOCC1CN(C(=O)C(N)=O)C2 C1(CCNC(C(C(=C)Cl)(C)C)=O)CN(C(=O)C2=CS(=O)CCC2)CCS1(=O)=O C(CCC(O)C(=O)NC1CC2CC2C1)NC(CN1CC(C)(OC)C1)=O CCCCC(C(=O)NCC(n1cc(CN2CCS(=O)CC2)nn1)C)C(C)C Cc1cccc(C(N2CCC(C(=O)NOCC(O)CO)(CO)C2)=O)c1N CC1CN(c2ncc3ccsc3n2)Cc2ccccc21.C1(CO)CCCCNC1 N1(C(CC2(C(=O)OCC)CCC2)=O)CCOC2C(C(F)(F)F)C12 Cc1cnc(Cl)[nH]c1=NCC1CCC2(CCC2)C1NC(c1ccc(Cl)c(Cl)c1)=O C(CC(C(C)C)NC(c1ccc(C)nn1)=O)N(C(C(CC)N(C)C)=O)C c1(C(N2CC(Cn3cc(-c4c(F)ccc(C)c4)nn3)C2)=O)ccc2nsnc2c1 N1(C(C(C)OCCCC)=O)CCN(C(c2ccc(Cl)cn2)=O)CC1CC(F)F n1(CC)ccnc1C(=O)NCC1CCCN1C(c1ccnn1CC1CC1)=O N12CCCC(CC1)C2=O.C(CC1CO1)OC.C(=O)(C(C)C)N(CC(=O)NCC)C C(C)(CC(C)C#N)(c1n(C(CC)(C)C)nnn1)NCc1cc(C)cnc1F C(=O)(CCCC(=O)N1CC2(CCC2NC(=O)CCN2CCCC2)C1)N(C)C N1(C(CC(CC)C)=O)CCC2(C1)CN(C(c1csc3c1CCCC3)=O)CC(C)O2 n1(CCOC)nc(C(=O)Oc2ccc(F)cc2)nc1-c1ccc(C(C)(F)F)cc1 O=C(C(C1=NOC2CC12)N1CCN(C2CCC2)CC1)N(c1ccoc1)C1CC1 c1(C(CCC)C)nc(-c2nc(-c3ccc(Cl)cc3)sc2C)n(CCS(C)(=O)=O)n1 N1(C(c2cc(CC)[nH]n2)=O)CC(NC(c2ccc(OCC3CC3)cc2)=O)CC1C CC1CC(C)N(C(=O)CCCCCc2ccccc2)CCN1C(c1cncs1)=O c1(C(N2CCCC(C(C)NC(=O)C(c3cccs3)N(C)C)C2)=O)cncc(F)c1C c1(C(=O)OC)cc(C(=O)NC2CN(C(c3nnsc3C)=O)CC2C)ccc1F C1(NC(C=CCN(C)CC)=O)CN(C(=O)C(C)N2CC(C)C2)CC2CC12 c1(N(CCCS(C)(=O)=O)C)cc(Br)ccc1S(=O)(=O)N1CC2C3C=CC(O3)C2C1 N1(C(COCC2C(=O)OCC2)=O)CC2(C1)CN(C(c1cccc(CCO)c1)=O)C2 Cc1cnc(NCC2CCC(O)C2)c(S(=O)(=O)NCc2ncccc2C)c1 c1(CC)ncc2c(n1)CCC(C(=O)NCCCNC(C1CN(CC(C)C)C1)=O)C2 c1(C(=O)NC2(C(N(C3CCOC3)CC#C)=O)CSC2)c[nH]nc1CCC Cn1cnc2cc(C(=O)NC3CC4(C3)CN(C(C3CCCC3(F)F)=O)C4)ccc12 c1(CN(C2CC2)Cc2cnc(C(C)C)nc2)cc(O)nc(=N)[nH]1 C(C(C)CC(=O)NCc1cncnc1)NC(C(C1CC1)OCC)=O CC1CCN(C(c2cncn(C)c2=O)=O)CC1NC(C1(C)CC1)=O C1(CN(C)C(C2(N(C)C)CCCC2)=O)CCN(C(C2CC2Cl)=O)C1 c1(C(N2CCC(N(CC(C)O)C)CC2)C(=O)NCCSC)csc(C#N)c1 N1(C(c2n(CCC)ncc2)=O)CCC(NC(=O)Cc2nocc2C)C1C c1(OC)ccc2c(c1)CCCC2CNC(=O)Cc1ccc(C)c(-c2nn[nH]n2)c1 N#Cc1ccc(C(N2CCC=CC2C(=O)NOCC2CCOC2)=O)cc1 N(C(=NCC(C)c1ccc(F)cc1F)NC1CCCC1)C(CC=C)C N1(Cc2cccc(C(=O)NCCOC)n2)CC(OC)CC12CCC2 CC(C)(Cc1ccccc1)CC(=O)NC1CCCCC1NC(=O)Cc1cccs1 c1(C(N(C2CCCN(C(=O)C=CCF)C2)C)=O)ccc(=NC(=O)OC(C)(C)C)[nH]n1 c1(C(N(C(CCNC(C(C(C)C)C)=O)C)C)=O)cc2cc(N)ccc2[nH]1 c1(C(N(CC(C)NC(=O)COC2CC2)C)=O)cc(F)c(F)cc1N(C)C c1(C(=O)NCC2CCC(NC(CCCCC)=O)CC2)ncc2c(F)cccn12 N1(C(CC(CC)SC)=O)CCN(C(c2cc(C)cc(Cl)c2)=O)CC1C(C)C N1(C(c2ccc(N(C)C)c(F)c2)=O)CCCC2(CCC(NC(=O)C(C)(Cl)Cl)C2)C1 C1(NC(c2n(CCCSCC)nnn2)c2csc(C(C)OC)n2)CC12CCCC2 c1(NC)cnc(C(=O)NCC2CCCC3CC23)cn1.C12(CC1)CCNC2=O C1(NC(c2ccnc(C3CCCC3)n2)=O)C=CCN(C(C2(C(F)(F)F)CCC2)=O)C1 c1(C(=O)NCCNC(CC(C(C)C)O)=O)cc(Cl)c(O)c(Cl)c1 Cc1ccncc1C(c1nnnn1C1CCOC1)NCc1ccc(Br)cc1 C(=O)(C(Cc1ccccc1)N1CCCCC1)N.C1(C(F)(F)F)(C(=O)OCCl)CC(F)C1 N1(C(C2C(C)(C)C2)=O)CC(NC(=O)Cc2ccc(C(F)(F)F)nc2)C(O)C1 N1(C(C(C)N(C(=O)C=Cc2cnccn2)CC)=O)CC2(C1)CN(C)C2 c1(C(C(=O)OCCC2C(C)(C)OCC2)F)ccc(Br)cc1Cl C(=O)(C1=CC2(CN(C(=O)CC3CCC4CC34)C2)OC1)NCC1CC(OC)(CO)C1 C1(C(=O)NC)CCN(C(C2(NC(COCCOCCC=C)=O)CC2)=O)C1 N1(C(c2c(CC)non2)=O)CCC(NC(c2nc(Cl)sc2C)=O)CC1C c1(C(=O)NCc2cc(C(=O)NCCC(=O)N(CC)CC)on2)cnc(S)nc1 N1(C(c2c(OC)csc2)=O)CC2CCC1CN2C(C1(C(F)F)CCCC1)=O C1(CN(C(c2cn[nH]c2)=O)CC)CCN(C(=O)CC2CC3(CC3)CO2)CC1 c1(OC)cn2ncnc2cc1C(=O)NC(C)(Cc1ccc(F)cc1F)C(=O)OC Cc1nc(N2CCN(C(C(=O)NC(C)C)c3cnsc3)CC2)sc1C C1(CNC(COC(C)C)=O)CCCC1C(=O)NCc1cnc(C2CC2)[nH]1 c1(CC)ccc(C(=O)NCC2(CC)CC2NC(=O)COCC2CC2)cc1[N+](=O)[O-] NS(=O)(=O)CCCCCC(=O)NCCC1(NC(C2CCCSC2)=O)CCCC1 C(=O)(CCS(=O)(=O)N(C)C)NCC(C)CN(C)C(c1ccc(C(F)F)cn1)=O C1(C2CCN(CC(=O)NC(=O)C3CC3)CC2)(N(C)Cc2ccccc2F)CC1 C1(C(=O)NC2CCC(CO)C2)(CC)CCN(C(C2CCC(=O)NC2)=O)C1 c1(NCCCCNC(C2CC(C)OC(C)C2)=O)cc2nncn2cn1 Cc1cnn2ccc(C(=O)NC(C)(C)C(C)NC(=O)C=CCN3CCCC3)nc12 CCC(F)(F)CC(=O)NCCc1ccc(CNC(C2CC2(F)Cl)=O)cc1 N1(C(C2C(OC)CCC2)=O)CC(C(=O)NCC(C)(C)CSC)C(C)(C)C1 C(C(COC)CC(=O)NC(C)C(C)C(=O)NCC1CCC(=O)NC1)OC Cc1nc(O)nc(C)c1C(N1CC(NC(=O)C(C)CCN(C)C)C(C)(C)C1)=O C(CNC(c1c(Br)noc1COC)c1nnnn1C1CC1)(C(F)(F)F)OCC C(=O)(CC(O)CCSC)N1C(CN(C2CCCC2)C(COC)=O)CCC1 C(=O)(N=c1[nH]n(C)cc1I)NC(c1ccc(-c2c(NC)cccc2)cc1)=O CC(CC(=O)N(C1CC2CC1N(C(=O)CN1C(=O)CCCC1=O)C2)C)C(F)F Cc1ccnc(C(=O)Nc2cccc(CN3CCN(CC(O)C(F)(F)F)CC3)c2)c1 C1(NC(c2cn(C)nc2)=O)COCCC1C(=O)NC(C1CCC1)C1CCC1 c1(C(N2CC(OC)(CNC(=O)Cc3nonc3C)C2)=O)cncc(F)c1C N1(C(CSCCC)=O)CCC(CO)C(NC(=O)CCc2ncccc2C)C1 C(CCCC(=O)NC1C=CC(C(=O)NCC2CC(C)(C)C2)C1)SC c1(C(N2C3CN(Cc4cc(OC)cc(Br)c4)CC32)=O)cccc2ccncc12 C(=O)(CC(C)C(C)(C)NC(c1ccc(CO)cn1)=O)NCc1n(CC)c(C)nc1 N1(CCOC)CCC(N=c2[nH]c3cc(C)nn3c(=N)[nH]2)C(F)(F)CC1 C1(C(=O)NCC2(NC(c3c(C)cccn3)=O)CCCCC2)NC(=O)OC1(C)C C#CC(C(C)(C)C)NC(C1(N(C)C(c2ccccc2CC#N)=O)CC1)=O C(=O)(C1=NOC2(CCC2)C1)N(C)CC1CN(C(=O)C(F)c2ccsc2)CCO1 C12(CNC(CCC#N)=O)CC(C1)C(NC(=O)CN1CC3C=CC1C3)CO2 C#CCCCC(C)C(=O)NCCNC(C1CN(C(=O)CNC(=O)C2CC2)C1)=O C1(CNC(CCNC(C2CC(OC)C2)=O)=O)CCN(C(C)=O)C1 C1(C(N2CCC(NC(C34OCC(C)(C3)C4)=O)C2)=O)CCC2(CC1)CC2(F)F c1(C(N2CCCC(N(C(c3cnn[nH]3)=O)CC)C2)=O)c(C(F)(F)F)ncn1O N1(C(CCCc2ccc(OC)cc2)=O)CC2(CCN(Cc3cn(C)nn3)CC2)C1 N1(c2scc(-c3ccc(C)cc3C(=O)O)n2)CCC(O)C(C2CC2)(CO)C1 Cc1cccc(C(=O)NC2CCCC2C(=O)NCCc2cnn[nH]2)c1O CC(=O)C(C)CC(C)C(=O)N(CCC(=O)Nc1ccc(C)cc1C)C CC(C)CC(F)(F)C(=O)NCC1CC12CCN(C(C13CC1COC3(C)C)=O)CC2 c1(C(N2CCC(C)(NC(C3N(C(C)C)CCC3)=O)C2)=O)ncn2cc(Cl)ccc12 CCC(C(=O)NC(C)(C)CNC(c1cccc2[nH]ccc12)=O)C(F)(F)F c1(C(N(CCCNC(C2CCC(CC)CC2)=O)CC)=O)ccc2[nH]c(=N)oc2c1 CN1Cc2cc(CC(=O)NCCC3CN(C(C4CCCS4)=O)C3)ccc2C1=O C1(CC(N2CC(C)(C)CC(NC(COCC(C)C)=O)C2)=O)CC2(CCCC2)CO1 c1(CC(=O)OC)ccc(C(N2CC(C)(F)C2)C(=O)NC2CCOC2)cc1 c1(C(N2CCC(O)(CNC(CC(C)C)=O)C2)=O)cc2occc2[nH]1 S(=O)(=O)(c1cc(C(F)(F)F)ccc1Cl)NC(C)C(=O)N(C)CC1CCCCNC1 CC(CC(F)F)C(=O)N(C1CCCCC1NC(C1(C)COC1)=O)C C1(C(=O)NCC=CCNC(C(c2cccc(C)c2)O)=O)CCN(C2CC2)S1(=O)=O C1(CC)CN(C(=O)CC(C)CCOC)CCC1NC(=O)C(C)N1CCCC1 C1(CC)CCC(C(=O)NC(C)CN(C(=O)CC(C)c2cnn(C)c2)C)O1 C(C(=O)N1CCC(C(=O)N(C)CC23CCC(CC2)C3)O1)OCC=C Cc1nc(N(C(C)CNC(C2(C)CC(O)CN2C)=O)C)cc(C(C)C)n1 C1(C(N2CC3C(CC(=O)NCC4(C(=O)OCC)CC4)C3C2)=O)CNC(=O)CC1C C1(CCC)(NC(=O)CCN(C(=O)CCC2CCC2)C(C)C)CCNC1=O N1(C(CCN(C(c2nccnc2C)=O)CC)=O)CC2(CCC2O)C1 N1(C(=O)NCCS(=O)(=O)N(C)C)CCC2C1CCCN2S(=O)(=O)c1nccs1 N1(C(c2cnn(C)c2Cl)=O)CCCN(C(C2C3COCC23)=O)CC1CO N1(C(C(C)OCCCC)=O)CC(CCO)(NC(C2(C(C)C)CC2C(=O)NC)=O)C1 C(=O)(C(C)C(=O)NC(C(=O)NCC(=O)N(C)O)C1CCCC1)OC C1(CC(=O)NC2C(CNC(C#CC(C)C)=O)CCCC2)CCCS(=O)(=O)C1 C(CCC(N)=O)(C(=O)N1CC(NC(=O)CC=C(Cl)Cl)C(N=[N+]=[N-])C1)N(C)C N1(n2cc(C3(O)CN(C(Cn4nnc(C)n4)=O)C3)nn2)CCN(C)CC1C c1(C(=O)O)cccc2c1CN(Cc1ccc(Cl)cc1[N+](=O)[O-])CC2 C1(C(=O)NCCN(CC(C)O)C(c2nn[nH]c2Cl)=O)CC(C)CC(=O)N1 CCCC(C(=O)NCC1(NC(=O)CCN(CC)CC)CCCCC1C)C(C)C N1(Cc2c(C)nc(C)[nH]2)CC2(CCC(NC(c3ccc(O)cc3C)=O)CC2)C1 c1(C(N2CCCC(O)(c3ccccc3)C2)C(=O)NCCC)noc2c1COCC2 c1(C(C(=O)NC(CCOC)CNC(=O)C=CC(=O)N(C)C)=O)ccc(Cl)cc1 C1(NC(Cc2ccc(SC)cc2)=O)CN(C(=O)CN2CCCNC2=O)CCC1C c1(C(=O)OC)ccc(O)cc1CCC(N1CCC(O)(CO)CC1)=O N1(C(c2n(C)ncc2)=O)CC2CN(C(c3cc4sccn4c3)=O)CC12 CCCC(C#N)C(=O)NC1CC(NC(=O)C(c2ccc(F)c(Cl)c2)O)CC1O N1(C(CSCCCC)=O)CC=CC1CNC(=O)C(n1cc(Br)cn1)C C1(C)(C(N(CCCN(C(c2cc(OC)n[nH]2)=O)C)C)=O)CCC(=O)N1 n1(C(C)C)ccc(C(=O)NC2CCC2NC(C2CCS2(=O)=O)=O)n1 N12CSCC1C2=O.c1(C(=O)NCC2C(CSCCC)C2)c[nH]nc1CCC N1(c2nnn(C)n2)Cc2ccccc2C1CNCc1c[nH]ccc1=N C1(C(=O)NCC(C(CC)C)C)(CC)CCN(C(=O)C(C)NC(C)=O)CC1 N1(C(CNC(C(CC)CC)=O)=O)CCN(C(C2CC(=O)N(C)C2)=O)C2CCC12 N12CCCC(CC1)C(=O)OC2=O.N(C(C)C)(CC)CC Brc1cc2n(n1)CCN(Cc1ccccc1C(F)(F)F)C2 Cc1ccc2oc(C(=O)NCC3(C)CCN(C(C4C5CCN4CC5)=O)C3)cc2c1 C(CCN=C(NCc1cscc1C)NC1CCS(=O)(=O)C1)=CC c1(C(=O)NC2CN(C(CCN(C)CC)=O)C2)ccc(OC(F)(F)F)cc1Br CS(=O)(=O)c1ccccc1C(N1CC2CC1CN2S(=O)(=O)c1cnc(Cl)nc1)=O c1(C(=O)NC(CN(C)Cc2nc(CC)on2)C)cc(Br)c(C(C)OC)o1 C1(NC(CC2N(C)C(=O)CC2)=O)CC2CC1N(C(c1occc1Cl)=O)C2 C1(CC)CCN(c2nnc(-c3cnccn3)n2C)CC1 c1(C(=O)NCC2(C)CCN(C(C(C=C)OC)=O)C2)cc2c(nn1)CCC2 CCC(C)C(=O)N(C1CCN(C(=O)C(C)OCCC(C)C)C1)CCO C1(NC(C(C)=C2CC2)=O)CN(C(c2cn(C)c(C(F)F)n2)=O)CCC1C C(C(C(C)C(C)C)NC(c1cnnc(C2CC2)c1)=O)NC(Cn1nnc(C)n1)=O N1(C(C2CC(C)C2(C)C)=O)CCC2C(NC(c3ccc(CO)cn3)=O)C2C1 N1(C(C2N(C)CCC2)=O)CC2(C1)CN(C(C1CC(F)(CO)C1)=O)C2 c1(OCC)ncccc1C(=O)NCC1CCC1NC(=O)CCCOC(C)C C1(O)(C(C)NC(c2ccccn2)=O)CCN(C(=O)Cc2csc3nccn23)CC1 C1(NC(c2c(C)n(C3CC3)cc2)=O)C(C)CCN(C(c2cnnc(Cl)c2)=O)C1C c1(N2CCCC(C)(NC(C(C(C)(C)C)O)=O)C2)c(F)cccc1[N+](=O)[O-] N1(C(CCc2n(C)ncc2)=O)CCC(O)C(NC(c2cc(O)nn2C)=O)C1 N1(C(c2cocn2)=O)CC2CC1CN2C(c1coc(Br)n1)=O N1(C(CC2CCN(C)CC2)=O)CC2CC1CCC2NC(C1CCCC1O)=O C1(C(=O)NCc2nn(C)c(=O)o2)CC(N=[N+]=[N-])CN1C(=O)COCCCF c1(C(N2CC(Nc3nc(C)c(Br)cn3)C(C#N)C2)=O)n[nH]c2ccc(F)cc12 C1(NCC2N(C(=O)OC(C)(C)C)CCC2)(CC2CC2)Cc2ccc(Cl)cc2C1 c1(C(N2C(CCNC(CCC=CC)=O)CCCC2)=O)ccc(C)c(C#N)c1 N1(C(C(C(C)(C)C)O)=O)CC2CCN(C(=O)C3=COCCO3)CC(C2)C1 N1(C(C(CC)C)=O)CC(F)(F)CC1CCNC(c1c(Cl)c(CC)nn1C)=O c1(C(=O)NCC(Cc2ccccc2)N(C)C)cc(Oc2ccccc2)ccn1 C(CCC(C)NC(=O)C(C)CC)NC(C(C)OCCOC)=O c1(C(N2CCCCC(NC(C3CC(F)(F)CS3)=O)C2)=O)ccc2[nH]ccc2n1 N1(C(C(CC)COC)=O)C2CCC1CC(O)(CNC(c1cncn1C(C)C)=O)C2 C1(NC(c2c(OC)cccc2)=O)CCN(C(=O)C(C)C2CCC2)CC1(C)C C1(NC(c2c(C)c[nH]n2)=O)CS(=O)(=O)CC1NC(=O)Cc1ccnc(O)c1 C(=O)(CC(C(F)F)N(C)C)NC(CN(C(=O)CC(F)(F)c1ccccc1)CC)C N1(C(C2CCC(C)(CC)O2)=O)CCN(C(C2CN3CCC2CC3)=O)CC1CCO N1(C(Cc2cc(C)n(C)n2)=O)CCCC2C1CCCN2C(=O)CSC(C)C N1(C(C=CC(C)(C)SC)=O)CC2(C(=O)NC(C)CNC(=O)N(C)C)CC1CO2 C1(C)(CNC(c2ccc(C)o2)=O)CCC(NC(c2csc(-c3ccco3)n2)=O)C1 C12(NC(C(CC)OC)=O)CCOCC1CN(C(c1cn3cnnc3cn1)=O)C2 C(=O)(C(C(=O)N(CC(CC(=O)N(CC(C)(C)COC)C)OC)C)OC)OC c1(NC(=O)NCCC(=O)OC)cnc2[nH]cncc1-2 C1(C(N(CCOCCNC(c2cc(CC)[nH]n2)=O)C)=O)CCCC2(CC2)C1 N1(C(C2N(CC)CCC2)=O)CC2CCCC(C1)N2C(=O)C(=O)OC(C)(C)C Cc1nnccc1C(=O)NC(CNC(C1(CF)CCC1)=O)C(C)C C(CCC(=O)N(CCCNC(C1CC1(C)C(C)C)=O)C1CC1)SC c1(NC)cccc(C(N2CSCC2C(=O)NC(C23CCC(CO2)C3)C)=O)n1 c1(C(=O)NCCCC(C)NC(=O)CN2C(=O)CCC2=O)ccc(S(N)(=O)=O)nc1 C1(CCC)CN(C(C2CC2C)=O)CCN1C(=O)C(C(C)C)Oc1cccc(Cl)c1 c1(C(N2CC(NC(c3cc(C(C)C)[nH]n3)=O)C(O)C2)=O)ncnc2c1CCCC2 N1(C(CC2C(=O)NC(=O)N2)=O)CCN(C(=O)Cc2cc(CO)on2)C2(CCC2)C1 Cc1cccc(-c2nc(-c3nc[nH]n3)nn2CC2CCCO2)n1 c1(C(=O)OC)ccc(=NCCNC(C2(C)CCOCC2)=O)[nH]c1OC c1(C(C(=O)NC(C(C)NC(C2(F)CCC2)=O)CO)(C)C)cc(F)cc(C#N)c1 C1(NCC2CC(C(=O)NC3C(C(=O)OC)CC3)CO2)CCOCC1F C=CC(C)(O)CC(=O)NC1CN(C(c2ccc(C)c(N)c2)=O)CC1C c1(C(=O)NC2CCOC(c3ccncc3)C2)ccc2c(c1)C1(CC2)CC1 C1(N(C(=O)C=Cc2nccs2)C)CN(C(c2ccnc(NC3CC3)c2)=O)CC1F C1(CNC(C(=O)NC(c2ccccc2F)C(C)C)=O)CC2CCC(C1)O2 C(C(C(C)C(C)C)NC(c1c(Cl)nsc1Cl)=O)NC(Cc1ccc(C)cc1)=O C(=O)(CC(C)CCCCCC)NC1C(C(N(CCCC)C2CC2)=O)CCCC1 C1(NC(C(C(CC)C)C)=O)CC1C1CCCN(c2ccnc(C)n2)C1 C(=O)(C1=NNC(=O)C1)N1CCCC(C(C)NC(CCc2ccc(C)cc2)=O)C1 C1(O)(C(N2CCCC(O)(CNC(c3cc(OC)n[nH]3)=O)C2)=O)CCC(C)(C)CC1 Cc1nc2[nH]n(C)c(=O)c2c(C)c1CNC(=O)C(CC(C)C)OC(F)(F)F C1(CC(=O)N(CCCNC(c2c(C)nc(C3CC3)[nH]2)=O)C)CN2CCN1CC2 Cc1coc(C(C)C)c1C(=O)NCC1CC(F)CN1C(=O)CSC1CCCO1 N=S1(=O)CCC(Nc2ncnc(-c3ccc(F)cc3)n2)c2cc(F)ccc21 N1(C(c2c(CC)nn[nH]2)=O)CCC2CCC(C1)N2C(C1CCCN(C(N)=O)C1)=O c1(C(=O)NC(c2ccccc2)C(=O)NC(c2ccccc2)C#C)cscc1Cl c1(C(=O)NCC2N(C(c3ccc(SCC)nc3)=O)CC=C2)ccc2cncn2c1 C(=O)(C(C1=CCCSC1)N1CCCC(c2ccccc2)C1)Nc1n(C)ncc1O c1(N2CCCC(NC(C(=O)NC)=O)C2C)ncnc2c1ncn2CCC(C)(C)CO c1(N2CCC(CC=C)(NC(C3CC4(C3)CC4F)=O)C2)cnc2ccccc2n1 Cc1ccc(S(=O)(=O)N2CCC3CC(CN(C)C)C3C2)cc1Br C1(C(=O)NC(CNC(CC2(C#N)CC2)=O)C2CC2)CCc2nnc(O)n2C1 C(=O)(C(F)CC(CC)CC)NC1N(C(CCCC)=O)CCN(CC)C1 C1(CNC(C(c2ccccc2)C)=O)CN(CCc2ccccc2)CCO1 S(=O)(=O)(c1cnc(N2CCC(C)(CO)C2)cc1C)N1CC(OC)C2(C1)CC2 C1(CNC(Cn2c(C)c(Cl)cn2)=O)CCN(C(C23CC(CN2C2CC2)C3)=O)C1(C)C C1(CNC(c2cc3c(s2)CCC3=O)=O)CCN(C(=O)CC2CCOC2)C12CCC2 C1(C(N(C(CC)C2CC2)C)=O)CC(NC(=O)CC2CC(SC)C2)CCO1 Cc1cccc(C(N2CC(C(=O)Nc3ccnn3C(C)(C)C)C(F)C2)=O)n1 c1(C(N2CC(NC(c3c(C)nccn3)=O)C(C)CC2)=O)cccn2[nH]c(=N)nc12 Cc1ccc(NC(=O)CCCCCc2ccc(I)cc2)cc1O C1(NC(C(CSC)C)=O)CCN(C(c2ccc(CO)cc2F)=O)C12CC2 C1(CCC)(NC(c2cccc(C(C)(C)C)c2)=O)CCN(C(=O)C(O)CC)CC1 C1(C(=O)NCC(C(C)C)NC(C2(CO)CCCC2)=O)CC(=O)N(C)C(=O)N1 c1(C(=O)NCC2(OC)CCOC2)ccnc(CNC(C2CCC(CO)CC2)=O)c1 C1(C(=O)NCC(=C)CC)CC2(CC2)CN1C(c1cc(CO)ccc1O)=O CC1=CCC(C)(C(N2CC3CC(C2)C3NC(C2CCCC3CC23)=O)=O)CC1 C1(CNC(c2cscc2F)=O)CC2(CC2)CN1C(=O)Cn1cccn1 C1(CCNC(C2(CSC)CCC2)=O)CN(C(=O)CCC2CC2(C)C)CCO1 C1(NC(CC2N(C(COC3(C#C)COC3)=O)CC2)=O)CC2CC1CC2(C)O N12CCC(CC1)C(=O)OC(C)C2.N1(C(C2CCC2)=O)CCN(C)CC1 N1(C(CSCCC(C)C)=O)CCN(C(=O)CCN2CCCC2)C(C(C)C)C1 C(=O)(CC(F)(F)CS(C)(=O)=O)N(CCCCCCNC(CCCOCC=C)=O)C C#Cc1cncc(C(=O)NC2(C)CN(C(c3sc(-n4cccc4)nc3C)=O)C2)c1 Cc1nn(C)c(=O)c(C(N2CCC(C)(NC(c3cnc(C(C)O)s3)=O)C2)=O)c1C C1(C(N2C(C(N3CC(CCCCC)C3)=O)CSCC2)=O)CCC=CCCC1 CC1CCCC(C(=O)NCC2COCCN(C(C3CCC(C)(C)CC3)=O)C2)CC1 N1(C(c2ccc(C(=O)OC)cc2)=O)CCN(C(=O)CC2CCCCC2O)C(C)C1 c1(C(N(CC(=O)N(C)Cc2cncnc2)C2CC2)=O)cnc2n1CCC2 C12(C(=O)NCC3CCN(Cc4cccc(C)c4)C3)CCC(C)(C(=O)O1)C2(C)C CC1(C(N2CC(NC(C34CCC(OC)C3C4)=O)C3(CC3)C2)=O)CCCCNC1=O.CCO c1(C(N2C(C)(C)COC(C(=O)O)C2)=O)cnc2ccc(F)cc2c1 N1(C(c2c(OC)ccnc2)=O)CC(CNC(c2coc(N(C)C)n2)=O)CC(C)C1 CCC(C)(CC)C(=O)NC1CC(CC(c2ccccc2)C)C1 C1(CNC(=O)CSCc2cscn2)CCCCN1C(C1CC2CCCC12)=O c1(C(C(C)(C)C)NC2CCC2c2nc[nH]n2)cccc(Cl)c1 N1(C(CCC(=O)OCC)=O)CCN(C(C23CC(C)(C2)OC3C)=O)C2(CCC2)C1 C1(NC(CCC#C)=O)(CO)CCCN(C(c2ccnc(CC(C)C)c2)=O)C1 C(CC(C(=O)NCCCC1CCCN1C(=O)Cn1cncn1)OC)OC C1(NC(c2cc(CC)c(C)s2)=O)CN(C(=O)C(C)CC(C)(C)C)CCC12CCC2 C1(CNC(c2c(C)cc(SC)s2)=O)CN(C(=O)C(C)(C)O)CCCO1 CC1CCN(C(=O)CC2CCC(=O)C2C)CC1NC(=O)Cc1ccsc1 c1(SCC(N2CC(OC)(CNC(C3CCCSC3)=O)C2)=O)ccc([N+](=O)[O-])cc1 C(=O)(C(C)CC(F)(F)F)N(C1CCN(Cc2ccc3ccsc3c2)C1)CC c1(C(=O)NCC(CCCC)NC(C2C=C(C)CS2)=O)ccc(F)nc1C c12ncccc1S(=O)(=O)NC2.Cc1cc(C(c2ccccn2)N(C)C)ccc1F c1(-c2c(OC)c(O)ccc2)ccc2[nH]c(C(=O)NC(CCO)C(C)C)cc2n1 C1(CC)CC(C)CN(C(C2CN(C(=O)C(C)OCC(C)C)CC2OC)=O)C1 c1(NCC(C)(C2CC2)NC(C(n2cc(Cl)cn2)C)=O)cc(=O)n(C)c(O)n1 c1(SC)cc(C(N2CC3CC2C3NC(=O)C2=CCC2)=O)ccc1OC(C)C N1(C(C(CCOC)C)=O)CCC(CNC(c2ccsc2C)=O)C(O)C1 C1(C(N2CC(=CC)C2)=O)CCC2CCC1N2C(=O)CC1(OC)CCC1 N1(C(c2ccc(C#C)nc2)=O)CC2CCN(C(C3CC3(C)C(F)F)=O)C2C1 C=CCCCC(C(=O)NC(c1noc(CC)n1)C)NC(=O)CCC(C)(C)N(C)C c1(C(=O)NC(CC)(CNC(=O)Cc2c[nH]nc2O)CC)cc2ccncc2[nH]1 C1(C2CC2)(OC)CN(C(C2(C)CCCN2C(c2ccoc2)=O)=O)C1 N1(C(C(CC)C)=O)CCN(C2CCCN(C(=O)CCC3CCCOC3)C2)CC1 N1(C(C2C(C(=O)OC)C2)=O)CCCC(CNC(c2occ3c2CCC3)=O)(OC)C1 N1(CC(N2CCC(F)(CNC(C3ON=C(CC)C3)=O)C2)=O)C(=O)CC(C)(C)C1=O n1(CCNC(C(C)=C2CN(C(c3ccsc3)=O)C2)=O)cnnc1O C(=O)(C1=NN(CCO)C(=O)CC1)C(=O)C1=CCCOC1.C1(N)CC2(C1)CC(C)C2 c1(OC)cc(NC(c2cnc(NC(c3ccc(Cl)c(Cl)c3)=O)s2)=O)cc(C)n1 C(C1c2ccsc2CCN1C(=O)COC1CC1)NC(c1c(CC)nc(C)[nH]1)=O c1(C(N(C2CCC(NC(c3cc(C)[nH]n3)=O)C2)C)=O)sc2ccc(F)cc2c1C C1(NC(c2nc(C)sc2)=O)CCN(C(=O)CC2CCCC(C)(C)C2)CC1F N1(C(C(N(CC)C2CCCc3ccccc32)=O)=O)C2CCC1c1ccccc12 N1(Cc2cncc(C)c2)CCN(C(C2CCCO2)=O)CC1C C1(CNC(c2nc(C)[nH]n2)=O)CCC2(CN(C(C3CCCS3(=O)=O)=O)C2)O1 C(=O)(CC(C)C(C)C)N1CCC(OC)(CNC(c2cccc(Cl)c2)=O)C1 CCC(C)CC(C)C(=O)NC(CC)CCC(=O)N1CC(C)(CSC)C1 c1(C(=O)NC(C2CCC(NC(=O)Cn3cncn3)C2)C)ccccn1 c1(C(=O)NC(C2N(C(c3cnc(C(C)C)[nH]3)=O)CCC2)C)nn(C)cc1[N+](=O)[O-] C12(NC(C(CCC)N(C)C)=O)COC(C1)C(NC(c1sc(O)nc1C)=O)C2 CC1CCCC1(C)C(=O)NCC1CCCN1C(c1cc(=O)n(C)o1)=O C1(C(N(C2C(C)CCNCC2)C2CC2C)=O)CCC2(CCC2)CO1 c1(C(=O)NC(C)(CNC(=O)C=Cc2ccco2)CO)ccc(C#N)cn1 C1(C(=O)NCC(C)(C2CC2)OC)CCC(C)CN1C(=O)CC1CC1(C)C CC1(NC(=O)CO)CCN(C(=O)CCCc2nc(-c3ccsc3)no2)CC1 C1(c2cn(CC(F)(F)F)nn2)(OCC2N(C(c3cc(C)[nH]n3)=O)CC2)CCCOC1 c1(C(=O)NCC2(F)CC(NC(CC(=C)C)=O)C2)cc2c(s1)CCC2 Cc1nc(=N)[nH]cc1C(=O)NCC(O)CN(C(=O)C1=CCC1)C c1(CNC(=O)NC2CCN(CCC=C)CC2)ccc(N2CCSCC2)cc1C C1(C(=O)NCc2ccnc(C)n2)(NC(CC2CN(C(C)=O)C2)=O)CCCC1C N1(C(C2C(NC(c3cc(C)sc3C)=O)CCC2)=O)CC2CC(C)C2C1 c1(C(N2CCCC(CN(C)C(C3CCCOC3)=O)C2)=O)ccc2ccoc2c1 c1(C(N(C2CCC(NC(CC(=C=C)C)=O)C2)C)=O)ccc(-n2cccn2)c(C)c1 C1(N(C(C2C(C=C)CC2)=O)C)CCC(NC(c2ccc(C3CCC3)nc2)=O)CC1 C1(CNC(CCc2cnc(C)s2)=O)CN(C(c2n[nH]c(C)c2C)=O)CCCO1 C(C(C)(CC(C)C)NC(c1ccnc(C)c1)=O)NC(C(CC=C)NC(N)=O)=O C1(C(=O)NCc2ccc(CC)o2)CC(C)(C)CCN1C(C1CCCCN1C)=O C1(=O)C(C(N(OC)C)=O)(CCC)NC(=O)NCCC1 Cc1ccccc1C=CC(N1CCCC(CCNC(C2(CO)CCC2)=O)C1)=O CC1CN(C(c2cncc3c2CCC3)=O)CC(C)N(C(c2c(Cl)nsc2Cl)=O)C1 c1(CCN=c2[nH]nc(CCC)s2)ccc2c(c1)CS(=O)(=O)C2 N1(C(CCc2onc(C)n2)=O)CC2(CC2)CC1CNC(C12CC1COC2(C)C)=O c1(C(=O)NCC2CCCN(C(C3CCCOC3)=O)C2)cccc2nc(CO)[nH]c12 C12(C(=O)NC3CCN(CCC)C3)COCC1CN(C(=O)Cc1nocc1C)C2 N1(C(C=CC)=O)CC2CCCC2(NC(c2cccc(Cl)c2Br)=O)C1 c1(OC)c(C(N2CCC(CCCNC(=O)C(C)C3CCC3)CC2)=O)c(C)nn1C c1(C(N(C(C)CCNC(c2cn(C(C)(C)C)cn2)=O)C)=O)cccc(CF)c1 c1(OC)ccc(C(N)CC(=O)N2CCC(CC(=O)N(CC(=O)O)C)C2)cc1 C(=O)(C(F)C(F)(F)F)NC1C=CC(CNC(C(c2ccccc2Cl)(C)OC)=O)C1 N1(C(c2cc[nH]n2)=O)CC2CCN(S(=O)(=O)C(Cl)(Cl)Cl)CC2C1 C1(NC(CS(=O)(=O)NC)=O)CCCN(C(c2cn3ccsc3n2)=O)C1C Cc1cc(NC(c2cnc(=NCCCCO)[nH]c2)=O)cc(C)c1O C1(C(N(CCCNC(c2c(CC)scn2)=O)C)=O)CCN(C)S1(=O)=O S(=O)(=O)(c1ccc([N+](=O)[O-])cc1Cl)NC(CNC(C)CCC1CCCO1)=O C(C1SCCc2ccccc21)C(N1CCCC(c2nnnn2C)(C(=O)OC)C1)=O C(C(CC(=O)N1CC2(C1)CN(C(=O)COC1CC(F)(F)C1)C2)C(F)F)OC c1(C(=O)NCC(CN(C(c2c(C)c(C(F)(F)F)n[nH]2)=O)C)O)ccc(Cl)nc1O c1(C(N2CCCCC(NC(c3c(C)noc3C)=O)C2)=O)cc2n(n1)C(C)CCC2 c1(C(N(CC(O)CNC(=O)C=Cc2ccc[nH]2)C)=O)sccc1S(N)(=O)=O C(C1c2ccsc2CCN1C(=O)C(O)Cn1cncn1)NC(c1cc(O)cs1)=O c1(CC)[nH]nc(Cl)c1C(=O)NCC(C1CCCC1)NC(=O)CC(O)C1CC1 c1(C(=O)NC(c2nc[nH]n2)(C)C)ccc(C(=O)NCCSCCO)nc1 Cc1c(C(N(CCNC(=O)C(F)F)C2CC2)=O)cnn1C1CCCC1 CC(Cc1cnn(C)c1)C(=O)N1CCC(CNC(=O)C(CO)NC(N)=O)C1 C(CC(C)C(=O)NCCCC(C)(C)NC(=O)CSCC(F)(F)F)OC c1(NC(N2CC3CN(C(C4C(C)OCC4)=O)CC3C2)=O)ccc2ccccc2c1 Cc1cnc(Cl)c(S(=O)(=O)Nc2ccc(C(=O)N=c3[nH]oc(C)c3Br)cc2F)c1 c1(CN2CC(NC(C=CCCC)=O)C(OC)C2)c(-n2cccn2)nc(O)nc1C Cc1cccn2cc(C(N3CCCN(C(=O)CC4OCCC4(C)C)C3)=O)nc12 C1(C(N(CC(=O)NC(C)Cc2cn[nH]c2)CC)=O)CCC(=O)NC1 C(CNC(C1CC(C)(C)CO1)=O)(CCC(C)C)NC(Cn1c(C)nc(C)n1)=O C1(C)(C(=O)NCCCCNC(CNC(CC)=O)=O)CCC(C)C1 N1(C(C(CC)n2nccc2C)=O)CCN(C(C)=O)C(C)C1.c1(C(=O)OC)nocc1Cl N12CC3(CCN(CC3)C(=O)C1)C2.N1(CCCCc2n(C)ccc2)C(=O)C=CC1=O C1(CC)CN(C(=O)C(C)n2ccnc2)CCC1NC(c1ncc(Cl)cc1F)=O c1(C(=O)NCC2N(C(CCC)=O)CCC2)cc2c(nc1O)CCC(CC)C2 C(=O)(CCC(CC)NC(=O)CCc1cncc(O)c1)NC1(COC)CC=CC1 c1(C(=O)NCC(C)OC)cccc(CNC(=O)CC2CCCC2)n1 c1(N2CCN(C(=O)OC(C)(C)C)CC(C)(F)C2)n[nH]c2c1CC(C)OC2C Cc1cc(C(N2CCC(CO)(CNC(C3(O)CCOC3)=O)CC2)=O)cc(C)n1 C1(CNC(C(CCN(C)C)O)=O)CN(C(c2ccc(C3CC3)s2)=O)CC(C)(C)C1 Cc1sc(C(N2CCC(C)(NC(=O)C(CC#N)c3ccccc3)C2)=O)nc1O CCC(C)(O)C(=O)NOCc1cn(-c2ccc(C)c(C)c2)nn1 C(=O)(C(O)CC[S+](C)C)NC(C1(O)CCN(C(C=CCCC)=O)CC1)C CC1CCN2CC1CC1(CC1)C2=O.C1(F)(C(=O)NC2CC2)CCC1 C1(CC)CN(C(C2(C)C(C)(C)C2(C)C)=O)CCC1CNC(C1(C)CC=CCC1)=O C(=O)(C(C)(O)C(F)(F)F)NCC(C)NC(c1ccc([N+](=O)[O-])o1)=O N1(C(C=Cc2c(C)coc2C)=O)CC(NC(=O)CCC2CCCO2)CC(F)(F)C1 N1(C(c2c(C)nc(O)s2)=O)CCC2(CC(C(N3CCC(CO)C(C)C3)=O)C2)C1 c1(C(=O)NCCCCNC(CC(C=C)CC)=O)cc(N)c(Br)c(F)c1 C1(C(=O)NCC2(C(F)(F)F)CC2)CCCCCN1C(=O)C(F)CC1CCOC1 C=CCC(C(=O)NC1CN(C(c2ncncc2Br)=O)CC1O)C(C)C c1(C(N(C(C)CNC(=O)CCCc2cncs2)C)=O)cc2ncccn2n1 CC1CC(C)N(C(c2ccns2)=O)CCN1C(=O)CCCc1nccs1 C(C(C)(O)CC(=O)NC(C(=O)N(C)CCN1CCOCC1)C1CCCC1)OC c1(C(=O)OCC)cnn2c1OCC(NC(=O)C(=O)Nc1nc(C(C)(F)F)cs1)C2 C1(C2CC2)(CNC(Cc2c(C)ccc(C)c2)=O)CCN(C(C2COC2)=O)C1 c1(NC(=O)CC2C3CN(C(c4cc(O)cc(O)n4)=O)CC23)ccc(Cl)cc1O N1(C(c2cncc(N3CCC(C)CC3)c2)=O)CC2CC1CN(C(C1CC1F)=O)C2 N1(C(C(C)C2CCC2)=O)CCC(CNC(C2CC2C(F)F)=O)C12CCC2 c1(CC(N2CC3CN(C(=O)Cn4cccn4)C3C2)=O)cc(Br)ncc1Br CCCC(C(=O)NCCC1CCCN(Cc2cn(CC(C)C)nn2)C1)C(C)C c1(OC)ccc(-n2nc(C(C)O)nc2CSc2ccnc(Cl)c2)cn1 c1(N2CCC(CNCc3ccc(N(C)C)cc3)C2)ncnc2c1oc1ccccc21 c1(COC)ccccc1C(=O)NC(C(=O)N(C)Cc1csc(C)n1)C1CC1 C(=O)(C1CCC(=O)c2ccccc21)N(C)CC1CCCN1C(C1CCS1(=O)=O)=O c1(OC)ccc(NC(C)=O)cc1NC(C1CC1C(N1CC2CCC(C1)O2)=O)=O C(=O)(C1Cc2c(Cl)cccc21)N1CCN(C(c2ncc(CC)nc2)=O)C(C)C1 C1(NC(=O)C2CC2)CN(Cn2c(C(=O)C=CCO)ccc2)CCC12CCOC2 C(=O)(C1CS(=O)(=O)c2ccccc21)N(C1CCCN(C(=O)Cc2cscn2)C1)C N1(C(C2C3CC(C)(C3)OC2)=O)CCC(C2CC2)C1CNC(=O)CS(N)(=O)=O c1(C(=O)NCC(C)CN(C)C(c2ccc(=N)[nH]n2)=O)nc(O)nc(O)c1F c1(N2CCCC2)cc(Cl)nc(S(C)(=O)=O)n1.c1(CNC)cnc2n1CCC2 N#Cc1cc(Br)cnc1N1CCC(O)(CNC(=O)CC2COCCO2)C1 C(C(C)(C)C(=O)N1CC(NC(c2cccc(CS(C)=O)c2)=O)C(C)C1)NC(C)=O C(=O)(C(CC(C)C)CC(C)C)N1CCCC(CCNC(C2(CC)COC2)=O)C1 c1(SC)ccccc1CC(=O)N(C1CN(C(C2OCCC2C)=O)CC1F)C N1(C(c2c(CC)n(C)cc2)=O)CCC(NC(c2cc(C)sn2)=O)C(O)C1 N1(C(CCC(=O)NCCCOC)=O)CC2CC(C1)CN(C(C1CCN(C)C1)=O)C2 N1(C(c2cc(OC)ncc2)=O)CCC(C2CCN(C(=O)C=NOC)CC2)C1 CC1CCCN(C(=O)Cc2nc(=N)[nH][nH]2)C1CNC(=O)Cn1ccc([N+](=O)[O-])n1 N1(C(C(CC)O)=O)CCC(CNC(=O)CCc2nnc(C(C)C)o2)C12CC2 CCC(C#N)C(=O)N1CC(NC(c2ccc(SC3CC3)cc2)=O)C(C(F)F)C1 c1(C(=O)NCCC(C)CCNc2cc(OCC#N)ncn2)ccc(F)c(Cl)c1 CCCCC(O)C(C)C(=O)N1CCC(C)(C)C1CC(N1CCC(CCCO)C1)=O c1(C(N2CCN(C(CS(CC)=O)=O)CC(CO)C2)=O)[nH]cc2c(=O)n(C)ccc12 c1(C(=O)NC(C)C(C)(C)NC(=O)CNC(=O)CN(C)C)ccnc2ccnn12 C#Cc1cccc(C(=O)N(C2CN(C(C3CC3F)=O)C2)C)c1 c1(CC(=O)NC2C(CNC(CN(S(C)(=O)=O)C)=O)CCC2)cc2ccccc2s1 C(C(=O)NC1CC(F)(CNC(=O)CC(c2ccccc2F)C)C1)(C(C)(C)C)SC N1(C(C2N(C(C)C)C(=O)CC2)=O)CCC(C2CC2)(NC(=O)CCNC(=O)CO)C1 CCC(O)C(F)(F)C(=O)N1CCC(C(C)(C)NC(=O)CCc2cnccn2)C1 c1(COC(C(C(C)C)OC)=O)c(C(F)F)cccc1F C1(NC(CCCCSC)=O)CC2(C1)CN(C(=O)C(C)Sc1nnnn1C1CC1)C2 Cc1nn(C)c(C)c1CCC(=O)NCC(O)CCNC(C1CC1CC(C)C)=O c1(C(N2CC(NC(C3CCC(NC(C)=O)CC3)=O)C2)=O)cc(C)nc(C(C)(C)C)n1 c1(CN2CC(C(=O)Nc3c(C#C)nccn3)C2)cc(Br)cc(Br)c1O c1(C(N2CCC3C(NC(C(C4CC4)OC)=O)C32)=O)cc(O)nc2[nH]c(=N)ccc12 N1(C(C(=O)OC)C)CCN(CC2CCCO2)CC1.c12ccc([nH]c1=O)COC2=O CCC(C)C(=O)N1CC(SCC(=O)NCCC(C)CO)C1 C(=O)(C1CCCC2(CCCC2)C1)N1CCC(C(=O)NC(C(C)(C)C(N)=O)=O)(CF)C1 C(C(C)(C)C)(C(F)(F)F)NC(N1C(CSC)CCC1)=O C1(CC)CCC(c2nnnn2C(C)C(=O)OC)(NCC2CCCCCO2)CC1 C(=O)(CCC(CF)CF)NC1CCCC(C(N2C(C)(C3CCC3)CCC2)=O)CC1 CN1CCOC(C(=O)NCc2ccnc(C(=O)NCC(C)(C)N(C)C)c2)C1 CCC(C(=O)N(CCNC(=O)Cc1ccccc1)CC)C(C)C c1(C(=O)NCC2(NC(c3cn(CCCF)nn3)=O)CC2)c[nH]c(=O)c2ccnn12 CCC(C(=O)NC1COCC1C(=O)NCC1CCCC12CC2)C(C)C c1(OC)ccc(Cl)c(C(N2CCC3CC2CN3C(=O)CC(C)OC)=O)c1F N1(C(c2cnc(C)o2)=O)CCCC(N=c2cc(Cl)nc(CS(C)(=O)=O)[nH]2)C1 CCCCC(C)(F)C(=O)NC1CCN(C(c2cc(C#N)c[nH]2)=O)CC1 c1(C(N(C(CC)C(N)=O)C)=O)cnc(Cn2cc(-c3nccs3)nn2)nc1O CC1CC(NC(=O)CSc2nncn2C(C)(C)C)CN(CC2(C3CCC3)CC2)C1 N1(C(c2ccc(CC)[nH]2)=O)CC2CCC1C1CN(C(=O)Cc3ccno3)CC21 C1(NC(CC2(C)CC2)=O)CCCN(Cc2nnnn2-c2ccccc2)C1 C1(C(=O)NCCCCOC)CC2CC2N1C(c1ccccc1F)=O c1(CC(=O)O)cccc(C2CC2)c1.n1(C2(C(=O)N)CC2)cc(-c2cn[nH]c2)nn1 CC1CCC(C(=O)N(CCCNC(=O)C(C)(C)c2ncco2)C2CC2)S1 N1(C(Cn2c(C)nnn2)=O)CCC(CC(=O)NC2C=CCCC2)C1(C)C N1(C(C(C)NC(=O)NCC=C)=O)CCNC(=O)C1 C1(NC2(c3n(COCCOCC)nnn3)CCCC2CC)CCC2C=CCC1O2 C1(NC(C(C)NC(C)=O)=O)CCOCC1NC(c1cnon1)=O c1(C(=O)NCC2CCCN(C(c3cccc(C)c3N)=O)C2)cnc2[nH]ccc2n1 C(=O)(C(COC(C)C)NC(=O)Cc1cnc(C)[nH]1)N(CC#C)CC c1(CCNC(c2cc(CCCO)cc(OC)c2OC)=O)ccc2c(c1)CC(C)O2 c12ncc(s1)CCNC(=O)NC2.c1(NCC(CO)C2CC2)ccsc1 CC1(C)COC(C(=O)NCC2C=CCN2C(C2CC(=O)CCO2)=O)CO1 c1(OC)ccc2c(c1)C1=NC(=NC(C)C(c3ccco3)N1)N2.C(CN(C)C)SC C(=O)(C(F)C(C)(F)F)N(CC(C)N(C(C(N1CCOC1=O)C)=O)C)C CC(CC1CCC1)C(=O)N1CCCC1CCNC(C1CN(C(=O)N(C)C)C1)=O c1(C(N2CC(COC)(NC(C3(C)CC3(F)F)=O)C2)=O)[nH]c2ccc(F)cc2c1C c1(C(=O)NCC2CN(Cc3[nH]nc(C(C)O)n3)C2)ccccc1F C1(NC(=O)Nc2c(C(C)C)cccc2F)CCS(=O)(=O)C(C)C1 c1(C(C(=O)NC(CCC=C)C)NC(c2nccnc2CC)=O)c(C)cccc1Br C1(NC2C(C)(C(=O)OCC)COC2)CCC2(CCC2)C1 c1(C(=O)NCC(C)(C2CCC2)NC(C2CCCC2)=O)cnc(O)cc1C(F)(F)F C(=O)(C(O)C(C)(C)C)NC1CC(NC(c2cc(CC)on2)=O)C1(CC)OC C(=O)(CC1=CCCC1)N1C(C(C)NC(c2ccc(CO)cn2)=O)CCC1 C(C(=O)N1CC(O)CO1)C1C(CC(=O)NCCCC2CC=CC2)C1 C(=O)(CN=c1cc(NCC(CO)C(C)C)nc[nH]1)NC(c1ccccn1)C=C C(=O)(CCCCC(=O)Nc1c[nH]nc1C(=O)NCCc1ccncc1)OC C1(C(=O)NCCc2nccc(C)n2)CN(C(=O)C(C)n2cccc2)C(C)(C)C1 C(=O)(CCCC(F)(F)F)N1CCN(C(Cc2ccc(C)cc2)=O)C1 C(C(C)CC(=O)NC1COCC1C(N)=O)NC(=O)NCCOC Cn1ncc(C(=O)NC2COCC2n2cc(CCC3CC3)nn2)c1Cl CC1(CNC(C23CC(CO2)C3)=O)CCN(CCc2cccc(F)c2)CC1 C(=O)(C=C1SCC(=O)N1C)N1CCCN(CCNC(C(C)C(F)(F)F)=O)CC1 O=C(C(O)C(F)(F)c1ccccc1)Nc1ncc(Cl)cn1 C1(C(F)(F)F)(CNC(NC2CCCCC2)=NCC2(C3CCOC3)CC2)CC12CCC2 c1(C(N(C2CN(C(=O)Cc3ccc(O)cn3)CC2O)C)=O)ccc(F)nc1 c1(-c2nc(CC(CN(CCC)C(=O)NCC(F)F)(C)C)on2)ccccc1C S(=O)(=O)(c1ccc(N2CCC(OC(C)(C)C)CC2)cc1Br)N1C(CC)C(C)CC1 CCS(=O)(=O)c1ccc(F)c(C(=O)NC(C)(CNC(=O)C(O)P(C)(C)=O)CO)c1 c1(C(=O)NC(c2cccc(Cl)c2)CNC(C(CC)NC(N)=O)=O)cncc(C)c1 C(CCCCCNC(C12CC(CCO1)C2)=O)NC(=O)C(c1ccc(Cl)cc1)O C1(CCC(N2CC(COC)(CNC(c3scnc3CO)=O)C2)=O)CCCCN1C c1(OC)ccc(NC(N(CCC#N)C2CCC2)=S)c(C)c1 Cc1ccc(CCC(=O)NC(C(=O)N(C)Cc2ccn(C)n2)c2ccco2)o1 C(=O)(C1CCc2c[nH]nc21)N1C2CCC(NC(c3nc(COC)oc3)=O)(C2)C1 Cc1cnn(C)c1C(=O)NC1CCCN(C(C2(C#N)CCCO2)=O)C1 N1(C(c2cc(OC)no2)=O)CCC2CN(C(=O)C(C)Cc3ccco3)CC12 N1(C(=O)CCCC2CCCO2)CCN(c2ccccc2O)CC1 CC12CCC(C(=O)NC3C4CC5C3C5C4C(=O)NC3C4CCCCC34)(CO1)C2 c1(C(N2CCCCC(OC(C)=O)C2)=O)ccc(C)c(C=O)c1.CO C1(C(N2CCCC2CN(C)C(c2csc3nnsc23)=O)=O)(OC)CCCCCC1 CCCC(C(=O)NCCC1(C(=O)N(CC(C)(C)CC)C(C)C)CCC1)NC(N)=O C(CCC)(C(C)(C)C)NC(C1C(CCC)CN(C(c2snnc2CC)=O)C1)=O C#CC1CN(C(C2CCC(C)(CC)O2)=O)CCN1C(=O)CCc1cnc[nH]1 N1(C(CNC(C=CCC)=O)=O)CC(OCC(=O)N(n2cccn2)C)C1 C#Cc1ccc(NC(C2CCC(N(C(C)=O)CC)C2)=O)cn1 C1(CC)C(C(N2CC(CO)C2(C)C)=O)CCN1C(c1cc[nH]c(=N)c1)=O CCS(=O)(=O)C=CC(=O)NC1CCCC1CNC(c1cccc2sncc12)=O c1(C(N2CC(O)(C(C)(C)CNC(=O)Cn3cccn3)C2)=O)ccc(N)c(N)n1 n1(CC(C)=O)cc(C(N2CC(CCCCNC(=O)C3CC3)C2)=O)c2ccccc12 c1(C(=O)NC2CCCN(C(C3(C(C)(C)C)CCCC3)=O)C2)occ2c1CCC2 CC(C(=O)NC(C(=O)NC1C(C)C1C)C(C)(C)O)C(C)(C)C C(=O)(C1=CC2(CCOCC2)C1)N1C(C)CN(C(=O)CN2CCCOC2=O)CC1 C1(CCCC)CN(C(=O)Cc2cncs2)CCN1C(=O)C(C)=CC1CC1 C1(NC(C(C(CC)C)O)=O)CN(C(=O)CC(C)C(=O)OC)Cc2nccn2C1 N1(C(c2ncc(C)o2)C(=O)NCC)CCC2C(O)CCCC2C1 C1(NC(Cc2c(OC)nccc2)=O)CCN(Cc2cc3occc3s2)CC1C C(CO)(C(=O)N1CC(OCCNC(c2cnc(N3CCCC3)o2)=O)C1)N(C)C c1(OC)ccc2c(C(=O)NCC3CCN(C(C4C(C)C4C)=O)CC3O)c[nH]c2c1 n1(CC)ncc(Cl)c1C(c1nnnn1C1CCOC1)NCCCOCCCO C1(C(=O)NC2(CNC(C3CC4CCC3CC4(F)F)=O)CC2)CCC2(CCC2)CO1 C(=O)(C1=CC(C)CC1)Sc1ccc(C(N2CC(N)CC2)=O)o1.N1(OC)CCCC1 C1(C(=O)NCC(CCNC(=O)COC2CCOCC2)O)CCC(C(F)F)CC1 c1(C(CNCCCC(C)c2ccccc2)C2CC2)ccc(C)cc1 N1(C(CC(C)NC(N)=O)=O)CCCN(C(=O)Cn2ncc(O)nc2=O)CCC1 C(=O)(CC(C(F)F)NC(C1(C#N)CC2CC2C1)=O)NCC(C(=O)OC)(C)C N1(C(c2c(C)cn(C)c2)=O)CC(C)CN(C(C2CC(C)OC(C)C2)=O)C(C)C1 c1(N)ccccc1Cl.C12(CCO)CN(C1)C(=O)CCNC2=O.C1(NC(C)=O)CC1C Cc1noc2ncc(C(=O)NCCC(C)NC(C3CCC(O)C3)=O)cc12 C(CCC(=O)NCCC1CC(NC(C2(c3ccccc3)CCC2)=O)C1)OC N1(C(CC(C=C)CC)=O)CC=C(C(=O)NCC(C)C(=O)OC)CC1 C=CCC(CNC(C1CC(=C)C1)=O)NC(=O)CNC(=O)Cn1cncn1 C(=O)(C1CCOc2ccccc21)N1C(CNC(=O)CCc2cccc(O)n2)CC1 Cc1nc(CC(N2CC(NC(=O)CCc3cccn3C)C(C)C2)=O)[nH]c1C C(C(C)C)(C(O)C(=O)Nc1cc(OC)n(C)n1)OC.N1(C(=O)NC)CC(C)C1(C)C Cc1cc(=O)n(CC(=O)N(C)CCNC(=O)C(CCO)N(C)C)c2ccccc12 C1(C(=O)NCCCNC(C2(CC)CC(C)(C)C2)=O)CC(c2ccccc2C)=NO1 N1(C(C=CC=CC)=O)CCC(NC(c2cccn3cnnc23)=O)C(CO)C1 N1(C(C(CC=C)CC)=O)CCC(C)(C)CC1C(N1CCC(F)(CF)C1)=O C1(CNC(CCCn2nc(C)c(Br)c2)=O)CCC2(CCC2)C1CN c1(CC)ncc(C(=O)NC2CC(NC(=O)CN(CCO)CCO)C2)[nH]1 CCC(CC1CCCCC1)C(=O)NCC1CC(NC(=O)CSCCC#N)C1 N(C(=NCCC(C(C)C)N1CCOCC1)NC1CCCC1)CCOCC CCCC(C(=O)NC1CC(C)N(C(c2cnn(CCO)c2)=O)C1)NC(N)=O c1(C(C)NC(=O)C(N2CCC(SCC(N)=O)CC2)=O)cccc(Cl)c1 C1(NC(C2(CSC)CCC2)=O)CC2CC(C1)N(C(=O)COCC1CCCCO1)C2 C(N=c1cc(NCC(CCO)SC)nc(C(F)(F)F)[nH]1)c1c(CC)nn(C)c1 Cc1ncc(C(N2CCC(NC(=O)CC3CCCC34CC4)C(C)C2)=O)c(C)n1 Cc1ccccc1CCC(=O)NCC(F)CNC(=O)C(C)n1cncn1 N1(C(CC)=O)CC(C)(C)OC2(C1)CN(C(=O)C=Cc1cc(CO)cc(C)c1)C2 c1(C(C(=O)N(C)CC2N(C(COC)=O)CCC2)OCCC(C)C)ccc(F)cc1 C(=O)(CS(=O)(=O)C(C)(C)C)N1C2CC(C)CC1CC2 N12CCC(O)C1C2=O.N1(CC(=O)NCC(N2CCCC2CCO)=O)CCCCC1 C1(CNC(C2(C(C)C)CC2)=O)CCN(C(c2ncc(Br)cc2N)=O)C1(C)C c1(C(=O)NC(C(=O)NCCOC(CC)(C)C)CC2CCCC2)ncn(C)c1C C1(NC(=O)CC(c2cccc(Br)c2)n2cc(C3CC3)nn2)(CO)CCSCC1 N1(C(C(CC)C#N)=O)CC2=C(C1)CN(C(c1cnn(CC3CCCC3)c1)=O)C2 c1(N2C(=O)CC(C(=O)NC3CC(c4cn(CC)nn4)C3)C2)cc(F)ccc1F c1(C(C(=O)NC(CNC(C(=C)C)=O)CO)NC(=O)OC(C)(C)C)cc(Cl)n[nH]1 C(CC(=O)NCCOC1CN(C(C2CC2(c2ccccc2)F)=O)C1)(C(F)(F)F)OC c1(C(=O)NCCn2cc(CC(C)(C)O)nn2)ccc([N+](=O)[O-])cc1 C1(NC(CCC=CCC=C)=O)CCN(C(C2CC(=O)N(CCC=C)C2)=O)C1C N1(C(c2c(C(C)C)con2)=O)CCC2CN(C(=O)CCOCC3CC3)C2C1 C1(C(=O)NCCCc2ccco2)CC2CC2N1C(c1ns[nH]c1=O)=O C1(O)(COC)CCCC1NC(=O)CCC1CC(NC(=O)CC2CCC(C)(C)O2)C1 N1(C(c2c(C#N)nc[nH]2)=O)CCC2(C1)CN(C(c1cc(Cl)sc1Cl)=O)C2 C(N=c1[nH]c2c(c(=NC3CN(C)CC3C)[nH]1)CCC2)C1(CC)CCCCC1 C1(C(=O)NCCOC2CCN(C(=O)C(=O)N(C)C)C2)(OC)CCC(C)(C)CC1 C1(C(N(CCN(C(CCCn2c(C)ncc2)=O)C(C)C)C)=O)CC(C)N(C)C1 N1(C(C2(CC#C)CC2)=O)CC(NC(C2CC23CCSCC3)=O)CC(C)C1 c1(CC(=O)NCCCNC(C2(Cc3ccncc3)CC2)=O)c[nH]c2nccc(Cl)c12 CC1(C)CN(C(=O)Cc2cccc(F)c2)C(CNC(C2(C)CC=CCO2)=O)CO1 CN1CC(C)(C(=O)NCCCC(CO)NC(=O)Cc2ccco2)CC1=O N1(C(c2c(C)c(F)cnc2)=O)CCC2CN(C(C3CCCCC3C(N)=O)=O)C2C1 C(N=c1nc(C)cc(C)[nH]1)C1OCCC(OCC)C1 c1(C(=O)Nc2cnco2)ccc(C(=O)N)cc1.C1(NC(=O)OCC)CC(C)(COC)C1 CCC(C)C(C)CCNC(C1(CC)COC1)=O C(=O)(N1CC2COCC2O1)C12CCC(CN(C(=O)C#CC3CCC3)C1)C2 c1(CC(C)C)ccc2cc(C(=O)NC3CC(C)(NC(C4CC(F)C4)=O)C3)[nH]c2c1 c1(C(N2CCC(C(N3CC(NC(=O)OC)C3)=O)C2C)=O)c(Cl)c(C)nn1C c1(-c2ccc(C)o2)ccc(S(=O)(=O)NCC2CCCCO2)cc1C C1(C(N2CC(C)(NC(=O)C(F)CC3CC3)C2)=O)CCCC(C#N)C1 C1(NC(c2cnn(CCC)c2Cl)=O)CC2CC(NC(C3(CC)CCC3)=O)CC12 CC1COCCC1NC(C12CC1CCN2C(c1cnco1)=O)=O CN1N=C(C(=O)NC2CCOCC2C(N2CCC(C(C)(C)C)C2)=O)CCC1=O C(=O)(C1=CCC(C)(C)CC1)NCCC1N(C(C(C(=O)OCC)C2CC2)=O)CCC1 c1(OCC=C)cc(OC)ccc1C(=O)NCCNC(=O)C(C)C1CCC1 Cc1cc(C(N2CC3CN(Cc4cc5sccc5s4)C3C2)=O)cc(C)c1 O=C(C1=CCc2ccccc21)N1CC(CNC(C2CC(O)C2)=O)C2CC12 C1(C(=O)NC(CCCNC(CCOCCCOC)=O)(C)C)CC12CCCOC2 Cc1nc(C(C)C)cc(=NC(CNC(c2c(Cl)nsc2Cl)=O)C(C)C(C)C)[nH]1 C(CC(C(C)C)NC(c1cnn(CC2CCCC2)c1)=O)NC(c1c(C)nsc1)=O C1(C(F)F)(OC)CCN(C(c2cc(Cl)ccc2C)C(=O)NC2CCCC2)CC1 Cc1ccc2[nH]cc(CCC(=O)NCC(O)CN(C(=O)Cc3ccon3)C)c2c1 c1(OCC=C)ccc(C(=O)NC(C)(C)CNC(=O)CCCCN(C)C)cc1 c1(C(N2CC(NC(c3c(CC)onc3C)=O)C(C#N)C2)=O)ccc(Cl)c(C)c1Cl N1(C(Cc2nc(C)[nH]n2)=O)CCC(CO)C(NC(C2CC(N3CC(O)C3)C2)=O)C1 N1(C(C2C(C)C2)=O)CCC(N(C)C(C2(CCc3ccccc3)CC2)=O)C1 CC(C(C)(C)NC(=O)Cn1nnc(-c2ccccc2)n1)NC(C1CCOC1C)=O C1(C)(C(=O)NCc2cc(C)c(C(=O)O)o2)CCCN(CC(O)CC2CCCC2)C1 N1(C(Cn2ccc(C)n2)=O)CCC(C)N(C(=O)C(C)Oc2ccccc2)CC1 CC(CC#N)C(=O)NC1CCCC1O.C1(N(C)CC)CCCC1 C(=O)(CS(=O)(=O)C1CCCC1)N(C(C)CCNC(=O)CCc1ccon1)C c1(C(C)NC(=O)NC2CCN(c3ccccc3)C2)c(F)cc(F)cc1F c1(C(N2CC(C(Cn3cc(CCCC=C)nn3)F)C2)=O)cc(C)sc1S(N)(=O)=O O=C1CC(NC(=NCC2(N(C)C)CCSC2)NC2CCOCC2)CCN1 c1(OC)cc(CN2CCN(C(=O)C(C)OC)C(CC#N)C2)c(C(F)(F)F)cc1Br C1(CC(=O)N(CCCCC)CCO)CC2(CCC2)CO1.C12CC(C1)NOC2=O c1(CC)oc(C(=O)OC(c2ccccc2-n2cccn2)C)cc1C c1(C(N2CC(NC(C3(C)CCN(C)C3)=O)CC2(C)C)=O)cc([N+](=O)[O-])nn1C c1(CC(C)C)ncc(C(=O)N(CC(C)N(C)C(c2cncn2C(F)(F)F)=O)C)s1 CCCC(C(=O)NCC(CNC(=O)C(CC)CC)OC)OC c1(C(=O)NCC(CC=C)NC(=O)C(C)C2CC2)cc(C)nc2c1c(C)nn2C N1(C(=O)C=CCO)CCC2(CCCN(C(=O)CC3CCCCC34CC4)C2)C1 C1(C(NNC(=O)NCCCCN2CCCCC2)=O)CCC2C(C1)C2(F)F C#Cc1nc(C(N2CCC(N(CCOC)C(C3CCC3(C)C)=O)CC2)=O)cs1 CCCC(C(=O)N1CC(CF)C1)NC(C1SCCS1)=O c1(-c2cc(C(=O)NC3CC(NC(CC4N(C)CCC4)=O)C3)on2)ccccc1F N1(C(C2CC(C)SCC2)=O)CCCC2(CCCN2C(c2c[nH]c(=N)o2)=O)C1 N1(C(C(C)O)=O)CC2(C1)CN(C(c1nccn1C)=O)CCO2 C(=O)(C1=C(C)OCCS1)NC1(CC(=O)NC(c2ncc[nH]2)CC)CC1 N1(C(COCC=C)=O)CCCC1(C)C(=O)Nc1ccc[n+]([O-])c1 C1(CNC(C2C(C)(C)CC2)=O)C(C2CC2)CCN1C(C1CC2(CCC2)C1)=O C(C)(CCCN=c1[nH]cc([N+](=O)[O-])cc1CO)NC(c1c(C)ccc(F)c1)=O Cc1cc(C(=O)NCCCOCC(C)(C)NC(=O)CC(C)F)ncc1N C1(C(=O)OCC)CCC1C(=O)OCCC(Cl)=C(C)C Cc1nc(N)c(C(=O)NCC(C)NC(=O)C(=O)NC2CC2)c(O)n1.C(C)(C)N Cc1cc(O)ncc1NC(=O)CC1CC(C)(C)CN1C(=O)CCCN=[N+]=[N-] c1(C(=O)NCC2N(C(COCCCOC)=O)CCC2)cccc(Br)c1O C1(CNC(C2(C#C)CC2)=O)CCCN(C(=O)CN(C)C(=O)OC(C)(C)C)CC1.C(C)(C)O N1(C(c2ccc(N(C)C)nc2)C(=O)NC2CC2)CCC2(CCSC2)C1 C=CC(C)(C)CC(=O)N1CC2CCC1(CNC(C1CCCC(C(N)=O)C1)=O)C2 C1(NC(CS(CC)=O)=O)CCC2(CC1)CN(C(=O)C#CC1(C)COC1)C2 C1(NC(COC2CN(C(c3c(C)cc(F)s3)=O)C2)=O)CN2CCC1(C)CC2 c1(C(N2CC(C(N)=O)(CNC(=O)CC3CC3)C2)=O)cc2cc(Cl)ccc2[nH]1 c1(NC(c2cc(C(=O)OC)on2)=O)sc(SCc2cn(C(C)C)nn2)nc1C C1(CC=C)(NC(C2CC2(C)Br)=O)CCN(C(=O)CCc2ccc(N)cc2)C1 CC1(C)CN(C(=O)CCN2CCCC2)CC1NC(=O)Cc1ccon1 c1(OC(C)C(=O)NC2CC(NC(=O)CC3COC(C)(C)C3)C2)cccc(F)c1 C1(CNC(CCc2c(C(C)=O)c(C)[nH]c2)=O)COCCN(C(=O)C=C(C)C)C1 N1(C(C=C)=O)CCC2(COC(CNC(c3c(C)nn(C)c3C)=O)C2)C1 N1(CCC(=O)NCC2(N(C(CCC3(C)CC3)=O)CC)CCOC2)CCP(C)(=O)CC1 C=CCCCCC(=O)NC(C1CCCN1C(c1cnc(O)c(F)c1)=O)C N1(C(C2(F)CCN(C(c3c(OC)ccc(Cl)c3)=O)C2)=O)CCc2cccnc2C1 c1(NC(C2CCN(c3cc(F)ncn3)C(C3CC3)C2)=O)cccn2ncnc12 CC(CC(=O)N1CCC(OCC(=O)NC2CSC2)C1)n1ccnc1 c1(C(=O)NC2(CN(C(c3c(C)nccn3)=O)C)CC2)c[nH]c2nc(F)ccc12 C1(CNC(c2c[nH]c(=NC)o2)=O)C(C)CCCN1C(c1cccnc1O)=O c1(NC(=O)NCC(c2cccc(OC)c2)O)cc(C)c(F)cc1Cl O(NC(=O)C(C)(C)CCNC(=O)C(O)CN1CCCC1)C(C(C)C)CO C=C1CC2(C1)CC(C(=O)NCC1(O)CCN(C(C3(C(F)(F)CC)CC3)=O)C1)C2 C1(F)(C(=O)NCCNC(CC)=O)CCN(C(c2[nH]c(C)nc2CC)=O)C1 Cc1cc(C=CC(N2CC3CN(C(=O)CCCF)CC3C2)=O)ccc1F c1(NC)nnc(COc2ccccc2)n1CC(C)(C)Cn1cncn1 c1(C(N2CCC(C)OC(C)C2)=O)coc2c1N(C)C(=O)CCC2 NS(=O)(=O)c1ccc(SCC(=O)NC2CCCCC2NC(=O)C2=NOCC2)cc1 C1(C(N(CC(CNC(C2C=C(C)CS2)=O)O)C)=O)CCCC(C)(C)C1 CC(CC(N)=O)C(=O)N1CC(OCCNC(C2CC2c2ccccc2)=O)C1 N1(C(C(COC)(C)C)=O)CC2(NC(c3ccc[n+]([O-])c3)=O)CCCC2(F)C1 c1(C(=O)NC2C(NC(COCc3cccc(C)c3)=O)CC2)cc2n(n1)CCC2 O=C(N=NCC(=O)NCCCOCC(F)(F)F)N=c1cc[nH]cc1 N1(C(c2nnc(C3CC3)s2)C(=O)NCCSC)CCC2(CCCOC2)C1 C(=O)(C(F)CC(CC)CC)NC(CCC=C)C(=O)NCC1(CO)CCC2CC12 C1(C(N(C(C#C)C)C)=O)C=CCN(C(=O)CCc2cccnc2)C1 Cc1ccccc1C(N1CC(NC(=O)Cc2ccccc2C(F)(F)F)C(O)C1)=O C(=O)(CC(C(F)(F)F)OC)N1C(COC)CN(C(c2cocn2)=O)CC1 C(CCCCCCCO)=CC(=O)NCC1N(C(C(CC=CC)C)=O)CCC1 c1(CN(C(C(CC)C2CCCN2)=O)C)ccnc(C)n1 C12CC3CC1N(C3)C(=O)N2C.c1(NC(C2CC2(F)F)=O)cccc(F)c1 C1(C)(NC(C)=O)CCN(C(=O)CC(C)(C)NC2CC(S)C2)C1.C(=O)(C(C)(C)C)N C(C)(CO)(C(C)(C)O)NC(CC1ON=C(CC)C1)=O.C1C(C)CC(=O)N1 C1(C(CC(N2CCCC(c3nc(C)c(C)[nH]3)C2)=O)N)CCC(F)(F)CC1 c1(C(=O)NC(CN(C(=O)CC2CCCS2(=O)=O)CC)C)cccc(Cl)c1 N1(C(c2nnn(C)n2)=O)CCCC2(C1)CN(C(=O)CCCC1CCCO1)C2 C(=O)(CC(O)CC(C)C)NCC1C(C(N2CC(C(C)O)C2)=O)CC1 C1(C(=O)NC2(CNC(C(C)CN(C)C)=O)CC2)CC2CCC(C1)N2C1CC1 n1(C(C)C)nccc1C(=O)NC(CNC(=O)C(c1cnn(C)c1)O)C1CC1 C(=O)(C(F)(F)CN(C)C)NC(C)Cn1cc(CCN(C)C)nn1 C(C(F)C(=O)NCCN1CC(C)(O)C1)C1CN(C(C(C)N(C)C)=O)C1 c1(C(=O)NC(C(C(C)C)C)CNC(=O)CSCC(N)=O)cnc2scnc2c1 C(=O)(CCCC(CC)NC(=O)C=C1CCCC1)N(CCN(CCC)CC)CC c1(OC)ccc(NC(c2ccc(NC(C)=O)cc2)=O)c(NC(=O)C(C)(C)C#N)c1 c1(N2C(CCC(=O)Nc3cnc(C(N)=O)nc3)CCC2)ncnc2cc(I)sc12 N1(C(c2cc(C)c(C3CC3)cc2)=O)CC2CC(NC(=O)C=CC3CC3)CC2C1 c1(C(N2CC(NC(C(C)OC)=O)C(C)(C)C2)=O)cnc2sc(C)c(C)n12 Cc1ccc(C)c(CC(=O)NC2CC(C)N(C(=O)CC3CC4CCC3O4)C2)c1 CC1=C(C(=O)NCC(O)CN(C(=O)CCc2ccc(O)nc2)C)CCS1(=O)=O C1(CC(=O)N(C2C(C)CC2)CC)CCCC1NC(c1nc(Cl)cs1)=O C1(CCNC(C(F)=C(C)C)=O)CCN(C(=O)CCCCCF)CC1(F)F CC1CC(C(N2CCOC(CCNC(=O)CN(C)C(=O)C3CC3)C2)=O)CCN1C c1(OC)ncccc1S(=O)(=O)Nc1nc(-c2ccccc2)cs1 N1(C(COCCOC)=O)CCC2CN(C(c3ccnc(OC)c3)=O)C2C1 N1(C(c2cc(OC)c(C)cc2)=O)CC(NC(=O)C(N)=O)C2(CCOCC2)C1 C=C(CN=c1[nH]c(=NC2CCCN(C(C)=O)C2)c2ncccc2[nH]1)c1ccccc1 c1(CC)ccccc1C(=O)NCCN(C(=O)C(C)OCOC)C(C)C CC(C)(C)CCC(=O)NCC(F)CNC(C1CCCOC1)=O c1(C(=O)NC)nc(Nc2ccc(N(C)C)cc2)c2c(n1)CCC2 c1(OCCCC(=O)N(CC(C)N(C(C2CC(OC)C2)=O)C)C)cc(C)ccc1C c1(C(N2C(C(C)NC(C(C)=CC)=O)CCC2)=O)ccc(C)cc1OC Cc1nc2ccccn2c1CC(=O)NC12CCC(C)(C1)OC2 c1(CC)[nH]c(=N)sc1C(N1CCC(NC(=O)COC(C)CC)CC1)=O c1(CNC(C2CCN(C(C=CC)=O)C2c2ccccc2)=O)ccc(OC)c(C)n1 C#Cc1cc(C(=O)NC(C)CCNC(=O)C(F)(F)C2CCCC2)cc(F)c1 c1(C(=O)NCC2C3CN(C(C(C)(O)C4CC4)=O)CC32)ccc([SH](F)F)cc1 C1(C(N2C(C3CCN(C(C4(C=C)CCC4)=O)C3)CCC2)=O)Cc2cccc(F)c2O1 C1(NC(c2cc(C(C)C)on2)=O)CC2CC1CN(C(c1ccc(O)cc1)=O)C2 c1(C(=O)NCC2C(NC(C(CC)C(C)C)=O)CCC2)sccc1S(N)(=O)=O C1(c2nnnn2C2CC2)(NCC(=O)NC2CC2)CCN(C(c2ccsc2)=O)CC1 N1(C(C(C)OC2CCOC2)=O)CCC2C(CCCN2C(=O)CC=C(Cl)Cl)C1 N1(C(Cc2n[nH]c(=NC)s2)=O)CCC(CNC(=O)CC=C(Cl)Cl)C1(C)C c1(C(=O)NC2CC(O)(CNC(C3N(C)CCC3)=O)C2)ccc(NC(=O)NC)nc1 N1(C(c2nc(C)c(C)[nH]2)=O)CCC(N(C(=O)Cc2cc(Cl)n(C)n2)C)C(C)C1 C1(CC)CCN(C(=O)C=C(C)COC)C1C(N1CC(CC)(CO)C1)=O C1(CCC(=O)OC)CCCN(C(c2ccccc2C(C)C)C(=O)NCC(C)C)C1 C(c1nc2ccccc2[nH]1)=CC(=O)NCC(C)CN(C)C(c1[nH]cnc1C#N)=O N1(c2snc(C)n2)CC2(CN(C(=O)C(F)(F)c3nccs3)CC2CO)C1 c1(CC(=O)NC(CNC(CCOC)=O)C(C)C)ccccc1Br N1(C(C(C=C)CC)=O)CCCC(C(=O)NCCc2nccc(O)n2)CC1 CC1(C#CC(=O)N2CC(C(O)C(=O)NC3CCOC3=O)C2)CCCO1 CC(CNC(=O)C(=C1CCCCC1)F)CC(=O)NCc1nc(N(C)C)no1 CC1CCCN(C(=O)CC2CS(=O)(=O)C2)C1CNC(c1cc(Cl)nc(Cl)c1)=O Cc1cc(CNC(=O)CCC2CC(NC(C3(C)CCC(C)C3)=O)C2)cc(C)n1 CC1(C)CN(C(=O)C=Cc2ccccc2)CC1C(=O)NCCCC(=O)NO c1ccc(Cl)cc1Br.c12[nH]nc(Cl)c1-c1nc-2no1.CC Cc1sc(N)c(C(=O)NC2(C(=O)O)CCCSC2)c1C CC(CN1CCOCC1)C(=O)NCCNC(C1CCN(C(C23CCC2C3)=O)C1)=O CN1CC(NC(=O)CCC(C)(C)NC(=O)CCCN2CCCC2)C2(CC2)C1 c1(CN(C(CCCCC)c2ccc(Cl)cc2)C=O)cnc(Br)c(Br)c1 C(=O)(C(CC#CC)NC(C1CCCOCC1)=O)NC1(C#C)CCOC1 C(CN=c1cc(C)[nH]cc1C(=O)OC)c1nc(C2N(C(=O)OC)CCC2)sc1 N1(C(CCNC(C)=O)=O)CCN(C(C2(C)COCC2(F)F)=O)CC1C Cc1ncc(C#N)cc1NC(=O)C(Cn1cncn1)NC(=O)CC1CCC2CC12 c1(-n2c(CNC(CN(CC(C3CCOC3)OC)C)=O)ccn2)ccc(F)cc1 CC1C(F)C(=O)N1.C(=O)(C(N)=O)N(C)CC(C1CC(N(C(=O)OC(C)(C)C)C)C1)=O c1(C(=O)NC(C2CCCN(C(c3c(C)ocn3)=O)C2)C)cc(Cl)c(N)c(Cl)c1 CC1(C)C(NC=O)CC1CC(=O)N.C12(CNC(=O)Cc3cnns3)CCC(CC1)C2 C1(O)(CN(C)C(c2cc(N(C)C)ccn2)=O)CCN(C(=O)Cc2cccs2)C1 C1(NC(c2c(CC)ccs2)=O)CCSC12CN(C(c1sccc1COC)=O)C2 C(=O)(C(C)(C(C)C)OC)N1CC(CCNC(c2c(CC)n(C)nc2)=O)OCC1 S(=O)(=O)(C1CCOCC1)N1CCC(O)(C(=O)NCCCN2CCCCC2=O)CC1 c1(C(=O)NCC(CC)NC(=O)C=Cc2ncco2)c(C)cccc1Cl C1(NC(c2ccc(F)c(C)c2Br)=O)CCC2(C1)CN(C(c1cc(O)n(C)n1)=O)C2 C1(OC)CCC12CC(C(N1CCC(C)(CNC(c3cc(Cl)cn3C)=O)C1)=O)C2 O(NS(=O)(=O)c1ccc(F)cc1)CC(=O)NC(C)C(C)NC(=O)CC1CCC1 c1(N2CCN(CC(CC(C)Sc3nc(C)c(C)o3)=O)CC2)ccc(F)cc1Cl C(=O)(C(C)(C)C(C)O)N1CC(CC)C(C(=O)NC2CN(C3CC3)CC2C)C1 CC(c1ccccc1F)=CC(N1CC2(CCN(C(c3ccnnc3C)=O)C2)C1)=O CCN(CC(=O)NCC(F)(F)F)N1CCC(CC(=O)OC)C1 CC(C)(CN=c1[nH]nc(-c2ccc3c(c2)CCN3S(C)(=O)=O)o1)CC(F)(F)F N1(C(C(c2c(C)n[nH]c2C)C)=O)CCCN(C(=O)CN(C)C2CC2)C(CO)C1 C1(C(N2CCC(NC(C34CCC(CC3)C4)=O)C(F)C2)=O)CN2CCCC2CO1 C(=O)(CC1=CCN(C)CC1)N1CC(C)N(c2nccn3nc(Br)cc23)CC1 c1(C(C)(C)C)nc(-c2ccnn2CCOC(F)(F)F)cs1 CC1(F)CN(C(=O)Cc2ccc(Cl)c(F)c2)CCN(CCCc2ccccc2)C1 N1(c2cn(CCOC)nc2)C(=S)NC(c2ccnn2CCF)C2=C1C(C)NC2=O Cc1nonc1C(=O)NCc1cc(C(=O)NOCCOCCF)co1 C(C)(CNC(=O)C=CC1CCC1)(C(C)C)NC(C(Cc1c(C)nc[nH]1)O)=O C1(NC(c2ccn(CC(F)(F)F)n2)=O)CCCN(C(=O)CCC(F)(F)F)CC1 CC1CN(C(C2(C(C)(F)F)CC2)=O)CCC1CNC(c1ccncc1O)=O C1(C(N2CC(COC)(CNC(c3cc(F)c[nH]3)=O)C2)=O)CCc2nnc(O)n2C1 C1(NC(c2cn(C3CC3)cn2)=O)CCC2(CCC2)C1.C12CCC(C1)CNC2=O C1(c2nnnn2CCCSC)(NCC2(COC)COC2)CCC(OC)CC1 N1(C(C2CN(S(CC)(=O)=O)C2)=O)CCC(O)(CNC(c2csc(C)c2N)=O)CC1 N1(C(C(C)n2ccnc2)=O)CCC2(CCC2)C(CNC(c2cnn(C)n2)=O)C1 c1(C(C)C)nc(NCc2nnnn2C)cc(N2CCOC(C#N)C2)n1 N1(C(=O)NC2(c3ccn(C)n3)CC2)CC2(CNn3cc([N+](=O)[O-])cn3)CC1CO2 C#CC1(N(CCCCCC)C(=O)C(C)(C)Cl)CCCC1.C1(=O)CO1 c1(C(N2CCC(CC(=O)NCC(C(C)C)OC)C2)=O)cccc(Br)c1F N1(C(c2c(C)nc(CNC(c3ccc(C#N)c(C)n3)=O)o2)=O)CCCCCCC1C N1(C(C(=O)NCCCCNC(C=C(C)C2CC2)=O)C)C(=O)CCC1=O c1(C(=O)NCC2N(C(CCc3onc(C(C)C)n3)=O)CC2)cc(O)nc(O)n1 C1(CCNC(C=COCC)=O)CN(C(=O)C(c2nc(C)cs2)C)CCCO1 C1(CNC(C(CN(C(C2C(CCC)C2)=O)C)C)=O)CCCC12CC2 N1(C(c2cnc(CC(C)(C)C)o2)=O)CCCC(NC(=O)C(C)(O)C2CCC2)CC1 c1(C(=O)NC2CC(C)(NC(=O)CCN3CCC(F)C3)C2)ccc(CO)cn1 Cc1cnc(CNC(C2CCCCCC2NC(=O)COC2CCC2)=O)c(C)c1 CC1CCC=C1C(=O)NCC(C1CCN(C(C2CCCCN2C(C)C)=O)CC1)O Cc1cc(C(N2CC3OC(=O)OC3C2)=O)cc([N+](=O)[O-])c1 N1(C(CN(C(C2(c3ccno3)CC2)=O)CCO)=O)CCN(CC(O)Cl)CC1 C1(C(=O)NCC2C(NC(C3CCCO3)=O)CC2)CC(=O)N(c2cccnc2)C1 C1(C(=O)NC(CC2CC2)C(N2CCN(CCSC)CC2)=O)Cc2ccccc2C1 n1(CC(N2C(C)(CNC(C3CC34CC4)=O)CCC2)=O)cc([N+](=O)[O-])ccc1=O N1(C(CC2N(C)CCC2)=O)CCC(C)(C)CC1C(=O)NCC1CC2(C1)CC(O)C2 c1(C(N2CC(NC(CC(C)(F)F)=O)C(C)(C)C2)=O)cc(F)cc2ccccc12 Cc1ccc(Cl)c(CNCC23CCCC2C3)c1 c1(C(=O)C(F)F)cccc(Sc2ncc(C3CCCC3)o2)c1 N1(C(C(CC)C)=O)CC(NC(=O)COc2cccnc2Cl)CC2(CCOCC2)C1 CCCCC(F)C(=O)NC1CCCCC1NC(c1sc(CO)nc1C)=O Cc1[nH]c(C#N)cc1C(N1CC(C)(C)CC1C(=O)NCC(CO)C(C)C)=O c1(C(N2CC(C(=O)NCC3C4CCC(F)C34)C2)=O)ncc(F)cc1F c1(OCC)nc(N2CCOC(C(=O)OCCO)C2)ncc1C N1(C(C(C)(C)C#N)=O)CCC2C1CCCN2C(c1cccn2ncnc12)=O c1(C(N2CC(CNC(c3snc(C)c3N)=O)OCC2)=O)cccc2[nH]ccc12 N1(C(C(=O)N(CCNC(=O)C(n2cc(Cl)cn2)C)CC)C)C(=O)CCC1=O C1(C(N2CC(NC(=O)CCC3CCC3)C2)=O)CCCCC1n1cc(Br)cn1 c1(C(N(CCCOCCN(C(=O)C2=CCC2)C)C)=O)cc(N)c2ncccc2c1 C12(C(=O)NCC(CCNC(c3ccc(CC)o3)=O)O)CCCN(CC1)S2(=O)=O n1(CC(=O)NC2C(NC(Cc3cccc(C)c3)=O)COC2)ncc2ccccc12 C1(NC(C2C(C)(C)C2NC(=O)Cc2ccccn2)=O)CCCSCC1 Cc1ncc(C(N2CCC2CNC(=O)C(C)CN2CCOCC2)=O)cc1C#N c1(CNC(C(c2cncnc2)C)=O)cc(C(N2CC3(CC3)C2)=O)n[nH]1 C1(C(N2CCCC(N(C(c3sccc3Cl)=O)CC)CC2)=O)CCc2nnnn2C1 N1(C(CC2ON=C(C)C2)=O)CCC=CC1C(=O)NCC(c1ccsc1)O C1(C(=O)NC2CCCC2NC(=O)COCCSC)(CC)CCCC1O C1(O)(CCNC(C2CC(C)(F)C2)=O)CCN(C(C2(C)CCCOC2)=O)CC1 Cc1[nH]ccc1C(=O)NC1CC(OCC(=O)NCCCN2CCCC2C)C1 N1(C(c2cn(CCOC)nc2)=O)CC(NC(c2cn(C(C)C)cn2)=O)C(SC)C1 N1(C(C(C)OCCCC)=O)CC(C2(NC(=O)CCCCNC(C)=O)CC2)C1 c1(C(=O)OCC)cc2c(Nc3csc(CC)n3)coc2cc1CNC(=O)C1CC1 C12CN(C(C)(C)C1)C2=O.C1(NC(=O)NCCCOCC)C2CN(C)CC12 N1(C(C(n2c(C)ccn2)C)=O)CCCCC(NC(=O)CN2CCN(C)CC2)CC1 C(=O)(CCCCCC(C)O)Nc1cn(-c2c(NC(C3CCC3)C)nccn2)nn1 N1(C(=O)OC(C)(C)C)CCCC1(C)C(=O)NCCC=Cc1ccsc1 N1(C(c2cccc(C)c2)=O)CCC(C2CC(NC(c3coc(C(N)=O)c3)=O)C2)C1 c1(N(C)CC)ccc(S(=O)(=O)CC(C)C(=O)OC(c2cc(N(C)C)c[nH]2)=O)cc1 c1(N(CCSc2ncc(CO)s2)OCC)cccc(F)c1 CC(C)CCC(F)C(=O)NC1CCN(C(c2nnsc2N)=O)CC1O C1(NC(c2nc(OCC)oc2)=O)CC2CC1N(C(=O)C(c1nc(C)cs1)C)C2 C1(CN(CC(=O)NCCOC)CC(C)O)CCCC(C)C1 N1(C(c2c(CCC)nco2)=O)CC(NC(C2CC(=O)N(C)C2)=O)C(C)(C)C1 CC(C)(C)C(CC(=O)N1CC2CCCC(C2)C1)n1cc(Cn2cc(Cl)cn2)nn1 c1(C(=O)NCC2CC2CNC(C2CSCCS2)=O)cc(Cl)ccc1C(F)(F)F C(CCCCC(=O)N(C1CN(C(c2cc(CO)n(C)n2)=O)CC12CC2)C)OCC c1(N2CCC(SCC)C2)nc(C)cc(=NC(C)c2ccsc2)[nH]1 c1(CCC(=O)NC2(C)CN(C(C3CCOC3=O)=O)C2)cc(Br)ccc1F c1(CC)nc2ccccc2cc1C(=O)NC1CCC(NC(=O)Cc2csnn2)C1 c1(OC)ccc(C(=O)N(CCCCNC(c2csc(C(C)C)n2)=O)C)c(OC)n1 C1(C(=O)NCC(C)(F)F)(NC(C(C)SC)=O)CCN(C)C1 C1(CC)C(NC(C2(F)CCN(C)C2)=O)CCCN1C(c1csc(C)c1C)=O c1(C(N2CC(CC(=O)NCCC(C)(C)C)OCC2)=O)cccc2c1CCCC2 C(=O)(C(C)(C)CCCNC(=O)CC1CCCC1O)N(C)CC1CCC(=O)NC1 C1(n2cccn2)(CC(=O)NC(C)CF)CCN(C(C2CCCSC2)=O)CC1 c1(CC)noc(C(N2CC(NC(=O)COCCc3ccc(Cl)s3)C2)=O)c1C C1(NC(CNC(CC)=O)=O)CC(=O)N(C2CN(C(=O)CC(C)(C)SC)C2)C1 C1(NC(C2C(C(C)C)N(C(C3CCC(C(C)C)O3)=O)CC2)=O)CC2CCC1CC2 c1(CC(C)(C)NC(=O)NC(c2cnn(CCC)c2)CCC)ccccc1 C(=O)(C(C)CC=C(C)C)NC1(CCNC(CCCSC)=O)CC1 C1(C(=O)NCC2N(Cc3onc(CCOC)n3)CC2)CCCCC1O c1(C(=O)NC2CN(C(CC3CC(=C)C3)=O)C(C)(C)C2)cc(OC)cc2c1OCC2 c1(C(=O)NCC2CCN(C(C(C)(C)C(F)F)=O)CC2O)[nH]nc2ncnc(O)c12 C12(CNC(c3nccc(C)c3)=O)CCCN(C(c3cncc(Br)c3C)=O)C1C2 c1(C(N2CCC(NC(C3(CC)CCCCC3)=O)C2C)=O)nn(C)c2c1CCCC2 C(N=c1cc(C)c(C#N)c[nH]1)C1(F)CC(NC(C2C(C=C(C)C)C2(C)C)=O)C1 CC1CN(C(C2(CCNC(C3(CCCF)CC3)=O)CC2)=O)CCS1=O c1(C(=O)NC(CC(=O)NC(C#C)(C)C)C)ccc(C)n1C Clc1ccc2[nH]cc(CCNCC3CCC34CCC4)c2c1 C(C)(C(C)(C)C(C)(F)F)ON1CC(C)N(Cc2ccc(OC)cc2)CC1C C(=O)(CCS(=O)(=O)N1CCC(c2ccccc2)C(O)C1)NCCOCC Cc1cccc(C=CC(=O)NC2(CNC(c3cc(F)cc(Cl)c3)=O)CCC2)c1 C1(CCNC(C(C=C)O)=O)CCCCN1C(c1ccnc(OCCO)c1)=O C1(C(C)NC(CC(C)C2CC2)=O)CCN(C(c2ccncc2C(F)(F)F)=O)CC1 C(=O)(C1CCCc2nnn(C)c21)NC(C)(C)CNC(=O)C(CO)c1ccsc1 C(=O)(CCN(OC)C(=O)CC1CCCC1(F)F)NC(C=C)C1CC1 C(=O)(CCCCCC(C)O)N1CCC(CCOC)(NC(CCOCCC)=O)C1 C(=O)(CCC(C)(F)F)NC1CCC(CCNC(Cc2cn(C)nc2Cl)=O)C1 C1(CC=C)(NC(C2CC(N(C)C)CCO2)=O)CC2CCC(C1)N2C(=O)CC1(C)CC1 c1(-c2cc(C(N(CCC(C)NC(c3nocc3Cl)=O)C)=O)[nH]c2)ccc(Cl)cc1 C1(OC)(CNC(=O)CC2CC2)CCN(C(=O)CCCc2cnccn2)C1 C1(CC)COC(C)(C)CN1C(C1CN(C(=O)COC2CC2)CCO1)=O N1(C(C(CC)N(C)C)=O)CCN(C(C2C(C)(C)C2(C)C)=O)C2CCC12 CN=c1nc(N2CCC(F)(F)C(CO)C2)[nH]c(=NCc2cn3ccccc3n2)[nH]1 C1(NC(c2c(C)n(CCO)cc2)=O)CCN(C(C2CC2c2cncs2)=O)CC1O N1(CC(=O)NCC2CN(C3CCC3)C2)CCC(O)C2CCCCC12 c1(N(C(=O)CC(=O)OC(F)F)C2CC(N)C2)ccc(N2CC(F)(F)C2)nc1 CC1(O)CCN(C(C2CC(C)N(C(c3cnn4c3CCC4)=O)C2)=O)CC1F CCCC(C(=O)NCC(O)CN(C)C(c1cccc(C(N)=O)n1)=O)OC Cc1cc(C)c(C(N2CCCC2CN(C)C(C2(C)CCCCO2)=O)=O)o1 N1(C(C(C)n2ccnn2)=O)CC(O)CC1C(=O)NCCP(C)(C)=O N1(C(C2(CC#C)CCC2)=O)CCC(C)(CNC(=O)CCn2cccn2)C1 Cc1cc(C(=O)NC2C3CC4C2C4C3C(N2CCCCCC2)=O)cc(O)n1 Cc1nc(N2CCC(C)C2CNC(c2n[nH]c(C)n2)=O)c(F)c(C)n1 N1(C(c2c(CC)nns2)=O)CCC(O)C(NC(=O)CC2CCCOC2)C1 c1(C(=O)NC(C(N2CCC(C(=O)OCC)CC2)=O)C)ccc2c(c1)CCC2 C1(C2CN(C(c3cc(O)ccc3Cl)=O)C2)(NC(CNC(CCCCC)=O)=O)CC1 c1(OC)cc(C(=O)NC(C)CCNC(=O)C(C)SC)ccc1OCC#N c1(C(=O)NC2CCC(C(=O)Nc3c(N(C)C)ccnc3)C2)n[nH]cc1[N+](=O)[O-] Cc1ccccc1S(=O)(=O)C1CCN(N2CCN(Cc3cccnc3)CC2)C1 c1(C(N(C)CC2CN(C(=O)CSc3ccccn3)CCO2)=O)cc(N)cc(Cl)c1 C1(NC(C(C)(C)OC(C)=O)=O)C=CCN(C(=O)C(c2ccnn2C)O)C1 N1(C(c2c(C)nc(O)nc2C)=O)CCC2CC1CN(C(=O)CC(C)P(C)(C)=O)C2 C(=O)(C(C)(C)CC#N)NCC1CC(NC(c2nc(C)n(C)n2)=O)C1(C)C N1(C(c2cnc(CCC)o2)=O)CCN(C(=O)C(C)O)C(c2ccc(F)cc2)C1 N1(C(C2CC3(CC(OC)C3)C2)=O)CCC2(CC(NC(c3ncccn3)=O)C2)C1 N1(C(=O)CC2CN(C(c3cc(O)cc(O)c3)=O)CCO2)CCC2(C1)CC2(F)F C(=O)(C(C)(C)CCOC)NCCCN(C(CCCCOC)=O)C C(=O)(CC(C)(C)C(=O)NCC1CN(C(c2cc(F)c(F)cc2F)=O)CC1O)OC CC1=C(C(=O)NCCC2(CNC(=O)CCn3ccc(C)n3)CC2)CCCC1 O=C1CCC(C(=O)N(CC(=O)NCC2CCCCO2)C2CCC2)C1 C1(C(N(C2CCN(C(C(CC)C(C)C)=O)C2)CC)=O)CCc2c(ncn2C)C1 C#CCC(CC(=O)NCCc1cc(C)nn1C)NC(=O)CC(=O)NC1CC1 CC(C1CCCCC1)=CC(=O)N(CCNC(C1(N2CCCC2)CCC1)=O)C1CC1 Cc1ccc(CCCNC(=O)CC(C)(C)n2cc(CS(C)(=O)=O)nn2)cc1Cl N1(C(c2ccnc(OC)c2F)=O)CC2CN(C(C3(C)CC=CC3)=O)CC2(C)C1 C1(C(=O)NCCCSCC)CC(C)N1C(=O)Cc1cnc(C)s1 N1(C(C2(OCC)CN(C(c3cc(C4CCCCC4)[nH]n3)=O)C2)=O)CC(C)C(C)C1 C(=O)(C(C)CC(C)(C)C)N1C(CNC(c2cnc(NC(C)=O)o2)=O)CC(F)(F)C1 c1(OCc2n(CC(=C)C)nc(-c3cccc(N)n3)n2)cc(F)ccc1F c1(C(=O)NCC(C(=O)OC)O)cc(C(=O)O)cc2nc(C(C)C)[nH]c12 C1(NC(C(CCC)OC)=O)CC2CC(NC(=O)Cc3nc(=N)[nH][nH]3)C1C2 N1(C(COCC)=O)CC2CC1C2CNC(=O)Cc1cccc(OC)c1 c1(C(N2CCCC(C)C2CNC(=O)CC(C)(C)N(C)C)=O)cc2cccnn2c1 Cn1ccc(C(c2nnnn2CCC2(C)CC2)NCCCCO)c1 Cc1cc(CN2CCC(F)(C(=O)NCCCC(F)(F)F)C2)c(C)s1 c1(C(=O)OC)csc(C(=O)NCC(Cc2ccccc2)NC(=O)C(N)=O)c1 CC1(C)COC(CC(=O)NCC2CC(NC(=O)C(C)(C)C3CC3)C(O)C2)C1 C1(O)(C(=O)NCCC=CC)CCN(C(c2cccnc2S)=O)CC1 C#Cc1cnn(CC(=O)NC(CCOCC)C(=O)NC2CCOCC2F)c1 CCC(C(=O)NC1(c2cn(CCN(C)C)nn2)CC(F)(F)C1)C(C)C c1(C(=O)NCC2CN(C(c3ccc(C)nc3)=O)C(C)CC2)cc(C)c(C)nc1O C(C)(CCCCN=c1nc(C)c(C#N)c[nH]1)NC(Cc1c(F)ccc(C)c1)=O c1(C(=O)NC(CN(C(C2CCN(C(C)C)C2)=O)C)C)ccc(OC(F)(F)F)cc1 c1(C(=O)NCC(CNC(Cn2nc(C)c(Cl)c2)=O)O)cc(C)n(C(C)C)c1C Cc1cc(C#N)cc(C(N2CCCN(C(c3nc(C4CC4)cs3)=O)CCC2)=O)n1 c1(C(C(=O)NCC(CC)NC(=O)CN2CCSCC2)C)csc2nc(C)cn12 c1(C(=O)OC)nc(=NC2CC3CN(C(c4cc(Cl)nn4C)=O)CC23)c(F)c(Cl)[nH]1 Cc1cc2nc(C(=O)NCCC(C)NC(=O)CCc3cncn3C)cn2cc1C C1(CC=C)(NC(=O)C(C)=CCNC(=O)C(C)(C)CF)CCCCC1.C(=O)(C)O c1(C(=O)NC(C(=O)NCCC(C)(C)C)CCN(C)C)c[nH]c2cnccc12 c1(CNC(C(C(C)NC(c2c(C)nco2)=O)C)=O)c(F)cccc1F C1(F)(CNC(C2CC(CF)C2)=O)CCCN(C(=O)CCCN2C(=O)CNC2=O)C1 CC1(C)CCc2c(C(=O)NC3(C)CN(C(=O)C4=C(C#N)CCC4)C3)n[nH]c2C1 c1(OC)ccnc(NCC(=O)NCC(C)N(C(C2CC(F)(F)C2)=O)C(C)C)n1 C(=O)(NNc1ccc(S(=O)(=O)C(F)F)cc1)C1CCC(N(C)C)C1 CN1CCC(CC(N2CC(F)CC2C(N2CC(C)(CF)C2)=O)=O)C1=O C1(O)(C(C)NC(c2cnns2)=O)CCN(C(=O)CN2C(C)CCC2C)CC1 C(=O)(C(C)(O)C(F)(F)F)NCCC(C)NC(c1cccc2occc12)=O CC1(C(=O)NCC(O)C(=O)NC2(CO)CCOC2)CC(=O)C1 c1(C(=O)NCC(CC)NC(=O)C(C)(C)C#N)cc(Cl)c(F)cc1Br c1(OCC(=O)N(C2CCN(C(c3cocn3)=O)C2)CC)ccc(Cl)cc1 C(=O)(CCCCC(=O)NC(CCF)C(=O)N1CC(OC)C(F)C1)OC Cc1cc(C)c(C(=O)NCc2ccc(C(=O)NC(C)(C)C(C)O)nc2)o1 C1(OC)CC(c2nncn2C)N(C(=O)CC2(c3ccon3)COC2)C1 C1(C(C)NC(c2ccnc(C(N)=O)c2)=O)CN(C(=O)CC2CCCCC2)CCO1 C(CCC(=O)NC1(C(=O)NC2CCC2N2CCCC2)CCCC1)=C(C)C N1(C(C2C(C)(C(C)C)C2)=O)CC2CC(NC(C34CCCC3C4(F)F)=O)CC2C1 CCC(C)C(C(=O)N1CCCCC(NC(c2cc(Cl)c(Cl)[nH]2)=O)C1)NC(C)=O Cc1ccc(C(=O)NC2CCC2NC(c2cnn(CCO)c2N)=O)cn1 c1(C(C)N(C(=O)CCC2(C(=O)O)CCOCC2)C)ccc(-c2nn[nH]n2)cc1 C(c1cccc(Cl)c1)=CC(=O)NC(CC(C)NC(C1(CCF)CC1)=O)C C(=O)(CCC(F)(F)C(F)F)NC1CC2(CC(CNC(CC(C)SC)=O)C2)C1 Cc1ccc2c(CC(=O)NC3CCCCC3N(C)C(C3CC3C)=O)coc2c1 c1(C(=O)NC(CCOC)CNC(=O)C(C)NC(C)=O)cnn2cccnc12 c1(C(=O)NC2CCC(CNC(C3CCCO3)=O)C2)cnc2ccccn12 N1(C(C(CC)OCC)=O)CC2CCN(C(c3ccc[nH]3)=O)C2C1C C(CC(C)(C)C(=O)N1CC(CO)OCC1C)NC(CCCOCC)=O c1(C(N2CCN(CCF)CC2)=O)ccc(Cl)nc1NCc1cc(O)cc(F)c1 C(=O)(CC(F)F)NC1CC(NC(CC2C(C)C2)=O)C1.C12CC(C1)C(=O)N2CCO C=CCCC(C(=O)N1CCC(COCC)C1)NC(C1CC(C)(C)CN1C)=O C(=O)(CCC(=O)NC)N(CC(C)(C)CNC(C1CCSC(C)C1)=O)CC C1(CNC(C(CCC)CC)=O)CC2(CCN(C(c3c(Cl)cnn3C)=O)CC2)CO1 c1(CNC(C2N(C(CCc3cc(C)ncc3)=O)CCC2O)=O)cccc(C)c1F C1(CNC(C2CC(C(C)C)C2)=O)CN(C(c2cc(N)c(F)cn2)=O)CC(C)(C)C1 CS(C)(=O)=Nc1ccc(C(=O)NC2CCCCN(C(C3CC3(F)F)=O)C2)nc1 C1(C(=O)Nc2ccc(C(=O)NC3CC3)cc2)CC1C1CCCCC1 c1(C(C)NC(=O)CCN(C(=O)C=CC(F)(F)F)CCO)ncoc1C Cn1ncc(Cl)c1C(N1CC(NC(C2CC2F)=O)CC1CO)=O C1(C(=O)NCCC(C)CCO)CCC(C)(C)N(C(=O)CC(C)F)C1 Cc1ccc(CC(=O)NCCN2CCN(C(c3cc(O)no3)=O)CC2)cc1F C1(C(C)NC(C(C2CCCC2)OCC)=O)CCCN1C(=O)CC1(CO)CC1 C1(NC(C(CCC)C)=O)CN(C(c2[nH]ncc2C#N)=O)CCC12CCC2 Nc1ccc(F)c2c1CCN(C(N1CC3CC4C(OC(C)(C)C)C1C3C4)=O)CC2 C1(c2cccc(OC)c2)CN(C(=O)C(=O)Nc2ccc(Cl)cc2OC)C(C)(C)C1 C1(O)(CCNC(=O)OC(C)(C)C)CCCN(c2nccc(-n3ccnc3)n2)C1 N1(CCC)CCCC(CNC(C2C(C)CCN2C(=O)CC2CCCSC2)=O)C1 C1(C(N(C)CC2N(C(C(C(C)C)=O)=O)CCCC2)=O)CC1C1(C)COC1 Cc1cc(F)ncc1NC(C1CC1NCc1cn(C)cn1)=O Cc1cc(CC(N2CC3(C2)CN(C(=O)CC2CC(=O)C2)C3)=O)ccc1CO N1(C(c2ccnc(C)n2)=O)CC2CC(CNC(c3cnsc3)=O)CC1C2 C1(CCCNC(CC=C(C)C)=O)CCCCN1C(=O)CSCc1nc[nH]n1 c1(C(=O)NCC2N(C(C3(N(C)C)CCCC3)=O)CC2)cc(C(F)(F)F)cc(F)c1 C1(C)(C(=O)NC(CC=C)CNC(c2cc(C3CC3)on2)=O)CC(C(F)(F)F)=NO1 CON1CC(C(=O)NC(C(=O)N2CCS(=O)CC2C)C(C)(C)C)CC1=O CCC(C)(C)CN=C(NCC(C1CC1)OC)N(C)Cc1ccco1 C1(OCCNC(c2c(OC)nsc2)=O)CCN(C(=O)C(O)C2(OC)CC2)CC1 c1(NCCNC(N2C(CCC)CCCC2)=O)nc2ccccc2nc1C c1(CC(=O)NCC2CCCN2C(c2n[nH]cc2Cl)=O)c(O)ncnc1O C#Cc1cccc(C(=O)NC2CC(C)CN(C(C3CCCCC3(F)F)=O)C2)c1F C1(C(=O)NCC(=O)N(CC(=O)N(CCOCC#C)C)C)(OC)CCSC1 CC(C)(C(=O)NCC1(CNC(c2cc(Cl)no2)=O)CCC1)C1CCCCC1 c1(CC(=O)NCC(C(C)C)(C)NC(C2CCO2)=O)cc(F)ccc1Br c1(C(C(=O)NCC(CO)NC(C(=O)NCC)=O)(C)C)ccc([N+](=O)[O-])cc1 c1(OCC(C)NC(=O)NCc2ccc(SC)o2)c(C)cc(C)cc1C n1(CC)nnc2c1CCC(C(=O)NC1CC13CC(NC(c1cc(Cl)no1)=O)C3)C2 C=C(C)C1CCC(C)(O)C(NC(c2cnc(C(C)C)n2C)=O)C1 n1(CC(=C)C)nnnc1C(C(C)(C)SCCSC)N(CC(=O)NS(C)(=O)=O)C O=C(CCCCCn1ccnn1)NC1C=CCCC1CO C1(C(N(CCOCCOC)C)=O)C2CC3C(C2NC(C2NC(=O)CC2C)=O)C13 N1(CCNC(c2ccc(OC)cc2)C(=O)NC2CC2)C(=O)c2ccccc2C1=O c12ccc(F)nc1NCC1CCN1C(=O)CS2.c1(CC)ccc(C(F)(F)F)cc1 C12(NC(c3c(C)con3)=O)CCCC1N(C(=O)C(C)OCC1CCCCO1)CC2 Cc1nn(C)c(C)c1NC(C1(CSCCNC(=O)Cc2cn(C)cn2)CC1)=O O(NC(=O)C(C)(CSC)NC(=O)Cc1cnoc1)CC(=C)C c1(CC(N2CCN(C(Cn3cccc(N)c3=O)=O)CC2)=O)ccc2nn[nH]c2c1 N1(C(C(C)OC)=O)CC(N=[N+]=[N-])CC1C(=O)N(C1CC(C)(C)C1)C Cc1cc2c(C(N3CC4CC4(CNC(C4CCCN4C)=O)C3)=O)ccc(C)c2[nH]1 C(=O)(CCCCC#N)N1C(CN(C(C2N(CC(C)C)CCC2)=O)C)CCC1 N1(c2snc(C(C)C)n2)CCN(C)C(CO)C1.C1(C=O)CC2CCC1C2 N1(C(c2n(CCCC)ncc2)=O)CC2CC1CN(C(c1nscc1C)=O)C2 c1(C(C(=O)OC)(C)C)cccc(NC(=O)NC2CSC(C)=N2)c1 C1(CCN(C(C(=O)NC2CCCCC2)C2CC2)C)CC(C)(C)CO1.n12cc(cn1)C2 Cc1nc(F)ccc1CNc1ccc(C(N2CCN(S(C)(=O)=O)CC2)=O)nc1 C1(C(NOCC=CC)=O)CCN(C(c2nc(C3CC3)oc2C)=O)C1C C1(CC)CCCCC1CNC(=O)COC1CC(NC(C2CCOC(CC)C2)=O)C1 N1(C(CN(CCC)C(C2CC2(Cl)Cl)=O)=O)CCC2(C=CCO2)C1 Cc1cccc(C(N2CCN(C)C(CNC(C3(CF)COC3)=O)C2)=O)c1C C(c1ccc(O)c(O)c1)=CC(N1CC(CN(C)C(C2CC3CC2C3)=O)OCC1)=O C#CC1(OCC(N2CCC(CCC(N3CCC3(C)C(C)C)=O)C2)=O)COC1 C1(NC(c2c(C)nsc2C)=O)CN(C(=O)CCCc2ncco2)CCC1C c1(CCNC(COC(C)=O)=O)cccc(C)n1.n12nccc1C=CC2 CN1C(=O)CN(C(=O)C(CC(F)F)NC(=O)Cc2nccn2C)CC1=O C1(C(=O)NC(C=C)(C)CC)C2CCCC2CN1C(=O)C(O)CSC N1(CC(=O)NCCCOC)CCC(NC(=O)COc2ccc(SC)cc2)CC1C N1(C(C2CC(C(C)C)C2)=O)CC(NC(C2(F)CC=CC2)=O)CC2(CCC2)C1 Cc1oc([N+](=O)[O-])cc1C(=O)NC1CC(OC)CN(C(=O)C(C)CC2CC2)C1 c1(CC(N2C(Cc3cn(CCCN(C)C)nn3)COCC2)=O)cc(Cl)ccc1O n1(CC)ccnc1C(C)NC(=O)C(C)NC(=O)C(C1CCCCC1)OC(C)C N1(C(=O)NC2CN(C(=O)OC(C)(C)C)C2(C)C)CCC2CSCC2C1 C(C(CNC(C1(OC)CCCSC1)=O)C(F)(F)F)NC(CC(=O)OCC)=O c1(CNC(CCCNC(N)=O)=O)n[nH]c2c1CN(C(c1cn[nH]c1)=O)CC2 N1(Cc2scc(C(=O)NCc3cc(OC)no3)n2)CCCC(N(C)C)C1C N1(C(CC)=O)CCC2C(C1)NC(=O)CN2C(c1cc([N+](=O)[O-])cnc1C)=O N1(C(C(c2cnn(C)c2)C)=O)CCN(C(=O)CNC(=O)C=CC2CCC2)CC1 C(C1CCCCCC1)=CC(=O)NC1C(NC(C(n2ccc(C)n2)C)=O)CCCC1 N1(C(CCCOC)=O)CCOC2(CCN(C(=O)C(C)C(C)(F)F)C2)C1 c1(SC)nccnc1C(=O)N(C(C)C(=O)O)Cc1cccc(CCC(OC)OC)c1 C1(C(N(C2CCC(CNC(C3CC(C)OC3)=O)CC2)C)=O)CCC2(C1)CC2(F)F n1(CC)ccc(C(N2CCN(C(=O)CNC(C)=O)CC2CC(=O)NC)=O)cc1=O c1(C(N(C(CC(C)c2cccnc2)=O)CC(=O)O)C)cccc(Br)c1 CC(C)(O)C#CC(=O)NC(CCC1CC1)C(=O)NCC1CC2(CC2)C1 N1(C(C=COCC)=O)CCCC(N(C)Cc2csc(-c3ccccc3)n2)C1 O=C1CC2CN(C(=O)C(O)CC3CC(F)(F)C3)C1=CC=CC=C2OCCO c1(C(=O)NC2CN(C(c3ccn(CC(F)F)n3)=O)C2)c[nH]c(-c2ccncc2)n1 CC1(NC(c2cc(C(N)=O)ccn2)=O)CCN(C(C2(S(C)(=O)=O)CC2)=O)CC1 C1(C(=O)NC2(C)C(C)OCC2)CC2(CCN(C(=O)CC(C)(C)O)CC2)C1 N1(C(C(=Cc2ccccc2)CC)=O)CC=C(CCNC(C2CC2F)=O)CC1 c1(CC(=O)NCC(CC)NC(c2cccc(OC)c2)=O)cn2cccc(C)c2n1 C(=O)(CCC(F)(F)F)NCCCCCCNC(Cn1ncc(CC)c1)=O N1(C(CNC(=O)NC)=O)CC(C)N(C(c2ccc(C3CC3C)cc2)=O)CC1C C(C(C)(O)CC(=O)NC1CC(CCNC(C2CCCCCCC2)=O)C1)OC c1(OC)ccc(C(N2CC=CC2CNC(=O)C(C2CCC2)C2CCC2)=O)cc1O C12(CCNC(CC)=O)CCC(C1)N(C(=O)CN1CCCC1CC)C2 CC1(C(=O)NCCCCCNC(=O)CCc2cnoc2)CCC(=O)NC1 C1(NC(C2C(C)(C(C)C)C2)=O)COC2(C1)CN(C(=O)C(C)(C)C(C)(F)F)C2 c1(C(=O)NCC2(CNC(c3cc(CC)no3)=O)CC2(F)F)c(CC)noc1C C1(NC(Cc2nc(C)sc2)=O)CCCC(N(C)C(c2cc(Br)c[nH]2)=O)C1 CC(CNC(C1(C(N)=O)CC1)=O)C(F)C(=O)N=c1ccn(CC2CCC2)[nH]1 c1(C(N2CC(NC(C3(COC)CC3)=O)C3C2C3)=O)cc2n(n1)CCC2 C1(CC(=O)NC2CN(CC)CC2C)C2CCC(C2)N1C(=O)CC(C)n1cccc1 N1(C(C(CC=C(C)C)C)=O)CC2(CC(NC(=O)CC3CC(C)(C)CCO3)C2)C1 c1(C(N(CCNC(CC2CC(=C)C2)=O)C)=O)cc(OC)cc(F)c1 CCCCCCC(C)C(=O)NCCC(O)C(=O)NCc1ncc[nH]1 C(Cc1nn[nH]n1)(C(F)(F)F)NC(c1ccccc1C(=O)C(F)(F)F)=O C=C1CCC(N2CCCC(C(N3CCCC(C(=O)NCCCC)C3)=O)C2)CC1 c1(C(=O)NC2CCC(C)N(C(=O)CN3CCSCC3)C2)ccnc2ncnn12 c1(C(=O)NCCN(CCC)C(C2(C)C=CCCC2)=O)ccc(C)n(C)c1=O CCC(CO)C(=O)N(C1CCN(C(c2ccnn2CC(F)F)=O)CC1)CC1CC1 C=CCN=c1[nH]cc(C(=O)NCCCN(C)C(c2nc(Cl)oc2C)=O)s1 CCC(CC(=O)NCC1(CC(=O)NCC2CC2(F)F)CC1)CC(C)C c1(CC(=O)NC2CN(C)C2)ccc(F)c(C)c1.C1(OC)CC2N(C1)C2=O O=C(CC1CCC(NC(c2cc(C(N)=O)c[nH]2)=O)C1)NOCc1ccccc1 c1(CN2CCCC(C)(C(=O)Nc3cc(C)cc(F)c3)C2)ccc2nccn2c1 Cc1cc(CNC(c2cc(Cl)c[nH]2)=O)oc1C(N1CCC(C(C)O)CC1)=O N1(C(c2cnc(CC)nc2)=O)CCC(C(=O)NCC(C2CCCCC2)C)C12CC2 c1(C(N2CCOC(CCNC(C3(Cl)CC34CCC4)=O)C2)=O)cc2n(n1)CCCN2 C1(CCC)CN(C(C2=CCSC2)=O)CCN1C(c1cnco1)=O c1(OC)nc(C(=O)NC2CCCC(NC(c3ccccc3SC)=O)C2)ncc1F c1(OC)nccc(C(=O)N(CCC(F)(F)F)CCC2CCCNC2)n1 c1(C(=O)NC(CC)(C)CNC(=O)C(C)C2(O)CC2)cc(F)ccc1Cl N1(C(c2ccn(C)c(=O)c2)C(=O)NCCC)CCc2c(cnn(C)c2=O)C1 C(CC1=CCN(C(C2(F)CC=CC2)=O)CC1)NC(C(C=C)(C)O)=O C12(C(=O)NC3(F)CCN(OC)C3)CCC(CC1)CC2.c12csc(c1)C(=O)NC2 N1(C(c2ncn(C(C)C)n2)=O)CCCCCC1CNC(c1n[nH]cc1F)=O CCCC(C(=O)NC(C)CCSC)NC(c1[nH]nnc1C1CC1)=O C(c1ccc(C)o1)=CC(=O)N(C1CCCCC1)CC#C.C12CCN(C1)C2 c1(C(=O)Nc2ccc(NC(C3C(Cl)(C(=O)OC)C3)=O)cc2C)cnn2c1CCCC2 CC(C(C)(C)C)=CC(=O)NCC1CCN(C(=O)C(F)(F)C2CC2)C1 C1(CCC(=O)OCC=CC(=O)NC(CN(CCCC)C)C)CCC(=O)N1 N1(C(c2cnn(C(C)C)c2I)C(=O)NCCC#N)CCCC(C)(O)C1 CCC(CC(=O)N1CCCC1C(C)NC(=O)C=CC(F)(F)F)c1ccccc1 N1(C(c2cc(C)c(C)[nH]2)=O)CCC(O)C(NC(=O)C=C2CN3CCC2CC3)C1 N1(C(c2cc(CCC)[nH]n2)=O)CCCCC1C(=O)NCCCC1(O)CC1 CC(C)CC(CNC(C1CCS(=O)CC1)=O)C(=O)N1CC2(CCOC2)C1 N1(C(C(=O)NC(C(CC)O)C)=O)CCC2(C1)CC2(F)F CC(C(F)C(=O)N1CC(NC(c2n[nH]c3c2CCCC3)=O)C(C)C1)C(F)(F)F C(=O)(C(C)(C)C(O)CC)NC1CC(CNC(C2(C)CC2C(=O)OCC)=O)C1 N1(C(c2c(OC)ccnc2F)=O)CC(CNC(C2CCC2(F)F)=O)OC(C)(C)C1 C1(CCC)CN(C(=O)CNc2nccs2)CCN1C(C1CN(C(C)=O)CCO1)=O c1(NC)cnccc1C(N1CC=CC(NC(=O)CN2CC3CC3C2)C1)=O c1(C(=O)NC(C)(C)CCCNC(=O)Cn2cnc(C(N)=O)n2)ccc(N)cc1F C(=O)(C1=COCCC1)N(C1CC(C(=O)Nc2c(C(C)=O)csc2)C1)C C(=O)(C#CC1CCCC1)NCC(N1CCN(C(C2(C)CNC(=O)C2)=O)CC1)=O N1(C(CC=CC(C)(C)C)=O)CCC(NC(=O)C2=CCSC2)CC1c1ccccc1 CC(C(CO)NC(=O)C(C1CCCCC1)F)NC(C1CCCCC1)=O c1(C(=O)NC(C2CCCCN2C(C2CC2Cl)=O)C)ccc(N2CCCC2)nc1 c1(CC(=O)N(C2CC3C(C2)C3(C)C)C)cc(F)cc2c1OCOC2 CC1CCN(C(=O)C(O)C2CCC2)C1CNC(c1cnccc1Br)=O C(CN=c1[nH]c(=NCC2COCCN2)c2ncccc2[nH]1)c1ncc(C)cc1C c1(CC(=O)NC(C2(O)CN(C(c3n(CCC)ncc3)=O)C2)C)ccc(Cl)c(Cl)c1 C(C)(C)(CC(=O)N1CCC(C(C)(C)NC(=O)CC2CCCCC2C)C1)SC c1(NCC(C(C)(C)C)NC(C(CCC)OC)=O)cc(=O)n(C)c(O)n1 N1(C(C=COOCC)=O)CC(n2cc(-c3cccc(OC)n3)nn2)CCC1(C)C N1(C(=O)CCOCC(F)F)CC(NC(C2(CF)CCC2)=O)C2(CCS(=O)(=O)CC2)C1 CNS(=O)(=O)NCC(=O)NCC(C1CCCC1)NC(=O)CCNC(N)=O C(=O)(CC(CC)CCC)NC1(CC=C)CCN(C(c2cc(Cl)cc(Cl)c2)=O)C1 c1(C(=O)NCCN(C(CC(CC)SC)=O)C2CC2)ccc2ncc(Br)n2c1 c1(C(=O)NC2CCN(C(CC(C(N)=O)NC(C)=O)=O)CC2)cc(C)c(F)cc1F N1(C(c2cn(C)nc2)=O)CCC2CC1CN(C(c1ccc3n[nH]cc3c1Cl)=O)C2 c1(NC)ccc(NC(=O)C(CSC)OC)cc1.N12CCOC(C1)CCC2=O C1(C(=O)NCC(C)CNc2cc(=O)n(C)c(O)n2)CCOC2(CCC2)C1 c1(C(=O)NCCCN(C(c2cnsn2)=O)Cc2ccccc2)cncc(N)c1 N1(C(C2CC(OCC)C2)C(=O)NC(C)CC)CCOC(C(N)=O)C1 c1(CC)nnc(C)cc1C(=O)NCC(C(C)C(C)C)NC(c1cc(C)c(C)[nH]1)=O c1(C(=O)NC2C(C)(CNC(C3C(C)C3)=O)CCC2)noc2c(F)cccc12 N1(C(C=CCCC)=O)CC2CCCC(N=c3[nH]cnc4cnn(C)c34)C2C1 CCN=c1[nH]c(C(=O)NC2CN(C(C3(C#N)CC4(CC4)C3)=O)CC2(C)C)cs1 CC1(C)CCC(CC(N2CC3(NC(=O)CC4(O)CCOC4)CC2C3)=O)C1 C(=O)(C(C)(O)C(F)(F)F)N(CCN1CC1=O)C.C=CCNC(C)=O c1(C(=O)NC(CNC)(C)C)ccc2c(c1)C(=O)CCS2 c1(OC)ncc(C=CC(=O)NCC(C)NC(c2ccc(=O)n(C)c2)=O)cn1 C1(F)(C(=O)NC2C(SC)CN(C(c3cc(C)cnc3N)=O)C2)CC2(CCC2)C1 C(=O)(CC(F)(F)Br)NC(c1ccccc1)C.C12CN(C1)C(=O)C=CCO2 C12(OC)CCC(C(=O)NC(C)(C)CNC(=O)CN=S(C)(C)=O)(CC1)C(=O)C2 Cc1ncc2n1CC(C(N1CCCC1C(C)NC(=O)Cc1nccs1)=O)CC2 C(=O)(CC1=CCN(C)CC1)N.C(=O)(CCC(=O)N1CCCC(CC2CC2)C1)NCC C1(CNC(CN(C(=O)C(C)(C)C2CC2)C)=O)CC1C1CCOCC1 C1(CNC(C(c2ccccc2)SC)=O)CC(NC(C23CC(C)(C2)C3)=O)C12CCC2 CC(C(=O)NCC(C1CCCCC1)NC(=O)C(C)(C)CN1CCN(C)CC1)C(F)F CC1CC=CCC1C(=O)NCC1(CNC(=O)C=CCF)CC(C)(C)C1 c1(CC(=O)NCC(CNC(c2c(C)cc(C)[nH]2)=O)O)cc(F)cc(F)c1 C1(N(C)C(C2(C)CN(C(=O)C=Cc3cocn3)C2)=O)CCCCC1C C1(CCNC(C2N(CC)CC2)=O)CCN(C(C2(OC)CCCC2)=O)CC1 c1(N(C2CCN(C)C2)C2CC2)nnc(C2CCCn3cnnc32)[nH]1.CS C1(N(C(=O)COC2CC(F)(F)C2)C)CN(C(C2CCC3(CC3)C2)=O)CC1O N1(C(CCC=CC)=O)CC(NC(c2onc(Br)c2C)=O)CC12CCCOC2 C1(NC(CSc2n(C)nnn2)=O)CN(C(c2ccon2)=O)C2(CCCCCC2)C1 c1(OC)ccc(NC(C2CCCCC2NC(=O)CN2CCCCC2)=O)cc1F C=CC(CC)CC(=O)N1CCCOC(CNC(c2csc(C(N)=O)n2)=O)C1 c1(C(c2nnnn2C(C2CCCO2)NCC(=O)NC)NC)cccc(C#N)c1 c1(OCC)ccc(C(N2CC3CC2C3NCc2ccc(I)o2)=O)cc1C(=O)O c1(CN2CC3C(NC(=O)CCn4ccnn4)C3C2)cnc2ccccn12 C1(NC(CCCSC)=O)(CNC(c2cc3n(n2)CCCO3)=O)CC2CCC1CC2 C(N=c1nc2scnc2c(NC(c2cccc(C)c2)C)[nH]1)C1CCN(OC(C)C)C1 C1(C(=O)NCC(CNC(c2nn(CC)c(=O)cc2)=O)F)CC12CCCCCC2 CCC(O)CC(=O)N1CCSCC1CCNC(C1CCCCN1C(C)C)=O C(c1cccc(F)c1)=CC(N1C2(CNC(c3cc(OC)ns3)=O)CC(C1)C2)=O C1(CC(=O)N(CCCCCO)CC)CN(C(C2(C(=O)OC)CC2)=O)CC(C)(C)C1 c1(C(N2C(CN(C(=O)C(C)(C)c3cnsc3)C)CCC2)=O)cc2sccc2s1 N1(C(C(N(C(CCC=CCC=C)=O)C)C2CC2)=O)CCCCN(C)CC1 c1(CNC(C2C(CC)C2)=O)nocc1C(=O)N(CCCCOC)C c1(CNC(=O)C(Cc2ccccc2)N2CCOCC2)ccc2oc(Cl)cc2c1 N1(C(C2CC(C)(C)C2)=O)C(CNC(=O)CCn2ccccc2=O)CC2COCC12 CC1=NOC(CC(=O)NCC2CCN2C(c2cocc2C)=O)C1 C1(CNC(=O)NCC2(C(=O)NC)CCCCC2)CC(C)CC(C)C1 C1(C(N(C(C)CNC(C2CC3CC2CC3O)=O)C)=O)CC2(CCCCC2)C1 c1(CN=c2scc(CN(c3cccc4c3OCO4)C)[nH]2)ccc2ccn(C)c2c1 C(=O)(C#CC(=O)N1CC(NC(=O)C(C)(O)c2ccccc2)C(O)C1)N(C)C N1(C(c2cnc(Br)s2)C(=O)NC(C(=O)OC)C)CC2CC1CS2(=O)=O c1(C(C)(C)C)ccc(CNC(=O)C(Br)CC2CC2)nn1 Cc1cc(C)c(C(=O)N(C2CN(C(=O)CC3CCOC3C)C2)C)c(C)c1 CC1(C#N)CCC(NCc2nc(CCC(F)(F)F)n[nH]2)C1 Cc1c(C(=O)NCC2CN(C(C3(CCF)CC3)=O)CC2(C)C)cccc1F c1(CC)c[nH]nc1C(=O)NCCC1(CNC(c2[nH]nnc2C2CC2)=O)CCCC1 N1(C(c2c(OC)csc2)=O)CCCCC1C(C)NC(c1cc(Cl)cn1C)=O C(C)(c1cccc(OC)c1)=CC(=O)N(c1ccccc1)CC N1(C(c2c(C)cc(F)s2)=O)CC2CC(NC(C3CCC4(CC4)C3)=O)C1C2 CC#CC1CN(C(C2COCCC2NC(C2CCC3(CC3)C2)=O)=O)C1 C(c1ccccc1)=C(CC)C(=O)NC1COCC1NC(C1CC(CN(C)C)C1)=O C1(NC(=O)CCc2ncccn2)CCN(C(c2cnc(Cl)c(Cl)c2)=O)CC1F C1(C(N2C(CC(=O)NC(c3ccn(C)n3)CC)CCC2)=O)CC(C(C)C)=NO1 N1(C(c2c(C)nsc2N)=O)C(C)C2CC1C2NC(=O)CC1CC=CC1 C1(CN(C)C(c2cc(Br)c[nH]2)=O)CCCN(C(C2(C)CC=CC2)=O)C1 N1(C(CCCNC(=O)CC2CCC=CCC2)=O)CCC(O)CC12CC2 CC1(CNC(c2ncsc2C(F)(F)F)=O)CCCN1C(C1(C(F)F)CCCO1)=O C1(C)(C(=O)NCC(C)CN(C)C(c2cc(C3CCOC3)[nH]n2)=O)CCCC1 C1(NC(=O)CCOC2CC2)C2CC1N(C(c1ccc(Cn3cc(Cl)cn3)o1)=O)C2 C1(NC(c2cccnn2)=O)(CO)CCCN(C(=O)C(c2cccnc2)O)C1 C1(CCCNC(C2C(CC(C)C)C2)=O)CCCCN1C(C1CN(C(N)=O)C1)=O c1(C(=O)NCC=C2CCN(C(=O)CC3(O)CCCC3)CC2)nc2c(s1)COCC2 c1(C(C)C(N2CCC(C)C2CNC(=O)CN2CCCC2)=O)ccc2c(c1)OCO2 C1CC(NC(=O)CNC(=O)COCCOC)C(C)C2C(C2)C1=O.CO.OC N1(C(C2CCN(C(C(CC(C)C)NC(C)=O)=O)C2(C)C)=O)CCSC2(CCC2)C1 C1(O)(C(C)NC(=O)CCC2CCC2)CCN(C(=O)C=Cc2nc[nH]n2)C1 C1(CC)CN(C(=O)NCC(=O)OCC2CC2)CCN1C(c1[nH]ccc1C)=O c1(OC)c(C(=O)NC2CCN(C(c3cnn(C(C)C)n3)=O)CC2O)occc1=O C12(CNC(C(CC)O)=O)CCC(NC(c3ccnc4ccnn34)=O)(CC1)CO2 N1(C(C2C3CN(C(C4CN(C)C(=O)C4)=O)C2C3)=O)CCC2C(O)CC12 c1(NC(=O)CC2CCC(C(N(CC(C)(C)CO)CC)=O)C2)cc(O)nc(C)n1 c1(C(N(CCNC(Cc2c(C)occ2)=O)CC2CC2)=O)cc(C(F)F)ccn1 CC(C)CC(O)C(=O)NCC(CC1CC1)C(=O)NCC1C(C)C1C c1(OCCC)ccc(C(=O)NCCC2(O)CN(C(c3cccc(N)c3)=O)C2)cc1 n1(CC(=O)NCC(CO)NC(C(C)OCCC=C)=O)cc(C)c(C(F)(F)F)n1 c1(C(=O)NC2C(CNC(=O)CC3CCCO3)C2)cc([N+](=O)[O-])n[nH]1 c1(NC(C(C(C)C)CNC(c2cccc(O)c2F)=O)=O)cc(C#N)ccc1O c1(CC)nc(C)sc1C(N1CCC(C(C)NC(=O)Cn2ccnn2)CC1)=O C1(C(CC)NC(CCC)c2nnnn2-c2cccc(F)c2C)CCC(F)(F)CC1 N1(c2n(CC=C)c(C(C)F)nn2)CC2SCC(C2)C1 N1(C(CCSCCC)=O)CC(C(C)(C)O)(CNC(C2CC2Cl)=O)C1 Cc1ccn(CC(=O)NC2CCN(C(=O)COC3CC(F)(F)C3)C23CC3)c(=O)c1 c1(-c2n(-c3ccn(CC)n3)nc(C(CC)CC)n2)cccc2cnnn12 Fc1ccc2scc(CNC(=NCCC3CCCO3)NCC(Cl)C(F)(F)F)c2c1 c1(NC(c2[nH]cc(C(N)=O)c2)=O)ccc2nc(S)oc2c1 c1(C(c2nn(-c3ccc(C)cc3)c(CCCN(C)C)n2)C)nc2ccccc2[nH]1 C1(C)(OC(CN(CCCCC2CCCO2)CC)=O)CCC(OC(C)=O)C1(C)C c1(CCN(C(C2(C(=O)O)CCC(C(C)(C)C)CC2)=O)CCO)cnc2ccc(F)cn12 C1(C(=O)NCc2cc[nH]c2C(=O)NCC(O)C(F)F)(OC)CCCOC1 C1(NC(C(C)Sc2nncn2C)=O)CN(C(c2cc(C(C)(C)C)on2)=O)CC1O c1(C(N2C(CC(=O)NCCCCCN=[N+]=[N-])CC(F)C2)=O)cccc2ccoc12 CCCC(C)CCN=c1[nH]c(N2CCC3(CC2)CN(C)C3)nc2c1CC(C)CC2 c1(COC)ccc(C(c2nnnn2C2CCCC2)NCC2(C#N)CC2)o1 CC(C)(C#N)CCCC(=O)N1CCC2(CC2)CC1C(N1CCC(CCO)CC1)=O c1(OC)cc(OC)nc(N2CCC(CC#N)C2)n1.C12CCCN(C1)C(=O)C(=O)N2 N1(C(C(=O)NC(C)C)=O)CCC2(CC1)OCCc1cc(Cl)ccc12 c1(OC)cc(C(N2CC(CNC(=O)C(c3ccc(Cl)s3)C)C2)=O)cnc1O C(=O)(N=c1cc(Cl)c(C#N)c[nH]1)C1CC2(C(CNC(=O)OC(C)(C)C)C2)C1 CC1CCC(O)CN1C(=O)CCC1CC(NC(=O)CC2CC(C)(C)CO2)C1 C(C(O)CC(=O)NCCN1CCCCC1=O)NC(CCC1(C)CC1)=O C1(C(=O)NCC(CCC)NC(=O)CC2CCN(C(C)C)CC2)CCS(=O)(=O)N1 C1(=CC(=O)N(C)CC2(NC(C(c3c(C)cccc3)C)=O)CC2)CCC(C)(C)CC1 N(C(=NCC#Cc1cnn(C)c1)NCC(F)F)CCCc1c(C)cccn1 N1(C(CN(C(=O)OC)C)=O)CC2CN(C(=O)C(F)Sc3ccc(F)cc3)CC2C1 C(=O)(C1OCCc2ccccc21)NCc1scc(CNC(c2cc(C)ncn2)=O)n1 NS(=O)(=O)c1sccc1C(=O)NCC1CCCN1C(=O)C1=CCCOCC1 C1(CNC(c2cc(CC)no2)=O)CCCCCN1C(C1CC(C(F)F)C1)=O c1(OC)ccnc(-c2cn(C(C)C(=O)NCCn3cncn3)nn2)c1 Cc1nc(C(=O)NCC(O)CCNC(=O)COc2ccccc2O)c(=O)[nH]c1C n1(CC(=O)NCC(C2CC2)NC(C2CC2F)=O)cncn1 CC1CCOC1CNC(=O)C(C)(C)NC(=O)Cc1cc[nH]n1 C(=O)(CC1=NNC(=O)C1)N(CCCNC(C1CCCNS1(=O)=O)=O)C(C)C c1(C(=O)NC2C(CC)N(C(C3CCSC3)=O)CC2)sccc1S(N)(=O)=O c1(C(N2C3CN(C(C4C(C(C)C)CCO4)=O)CC2C3)=O)cnc2ccoc2c1 C1(OCC)COCCC1NC(C1CCCN1C(=O)CCc1cncnc1)=O C(=O)(CCC(F)(F)Cn1cc(C(C)(C)C(=O)O)nn1)NCCCN(C)C1CC1 N1(C(COC2(C)CCC2)=O)CCn2c(CNC(C3(Cl)CC34CCC4)=O)nnc2C1 C(N=c1[nH]c(=NCCN2CC=CC2)c2ncccc2[nH]1)c1ccc(S(C)=O)cc1 c1(C(N2CCC(NC(c3c(OC)ccs3)=O)C2C(C)C)=O)cc(C)nc(O)c1 c1(C(=O)NCCN(C(=O)CCCS(N)(=O)=O)C)cc([N+](=O)[O-])cn1C c1(C(N2CCN(C(c3cnc(C)[nH]3)=O)C3C2C3)=O)ccc([N+](=O)[O-])c(Cl)c1 N1(C(C2C(COC)C2)=O)CC2(CC(NC(c3cn(C)nc3C3CCCC3)=O)C2)C1 N1(C(C(CCCC)O)=O)CCCC2(CCN(Cc3ccc(S(C)(=O)=O)o3)C2)C1 C1(NC(C=CC)=O)CC(C)CN(C(c2cc(C3CCCC3)n(C)n2)=O)C1 c1(C(C)=O)ccc(O)c(C(N2CC3CC2C3C(N2CC(C)OC(C)C2)=O)=O)c1 c1(OC)cc(C(=O)NC2CCCN(C(c3cccnc3O)=O)C2)sc1Br C(C(F)(C(=O)NCCC1CCCN1C)C(C)C)NC(C1(OC)CCC1)=O C=CCN=c1[nH]cc(C(N2CCC(F)C(NC(C3CC(OC)C3)=O)C2)=O)s1 C1(NC(C(CSC)O)=O)CCC2(CCN(C(c3ccnn3C3CCC3)=O)CC2)C1 N1(C(c2c(C)cn(C)c2)=O)CCCC(C)C1CNc1nnc(C(C)(C)C)o1 C(=O)(CCC(N)=O)N(C1CCN(C(=O)CCc2ccccc2C(N)=O)CC1)C C(CCCCC(=O)N(C1CCCCC1)C)N(C(C(C)=C(CC)C)=O)C N1(C(C2C(CC)N(C(C34CC(C#N)(C3)C4)=O)CC2)=O)CCC(C)(OC)CC1 N1(N(C(C2CC3(CNC3)C2)=O)Cc2ccc(Br)c(Cl)c2)CCCC(F)(F)C1 C(=O)(C(C)CCCC(C)C)N1CCC(COC)(NC(=O)Cc2ncoc2C)CC1 C1(C(=O)NC(C)(CO)C2CCCC2)CCN(C(=O)C=Cc2cocn2)CC1O Cc1ccc(Cl)c2cc(C(=O)NCCn3nccc3Br)[nH]c12 c1(C(N2CCSCC2CCNC(C2CC(N3CCCC3)C2)=O)=O)ccnnc1Cl c1(C(=O)OC)cc2c(NC(C)(C)CNC(=O)CC3CCCCC3C)ncnc2[nH]1 C(C(O)CN=c1ccc2ncc[nH]c-2n1)NC(CC1CCC(C)C1)=O C(=O)(C1CNC(=O)c2ccccc21)NC1CC(O)(CNC(C=CCCC)=O)C1 C1(O)(C(=O)NCc2c(C3CN(C(C)=O)C3)ocn2)CC2CCC1C2 C1(NC(c2cnn(CC)c2C)=O)CC2(C1)CN(C(c1oc(O)nc1C)=O)C2 N1(C(CC(CC)C)=O)CC=C(C(=O)NC(C)(C)C(O)CO)C1 c1(C(=O)NC(C2OCCN(C(CCSCC)=O)C2)C)cc([N+](=O)[O-])ccc1SC C1(NC(CCC(=O)NC)=O)CC2CCC(C1C)N2C(C1(C(F)F)CC1)=O CCC(C)(C)CC(=O)N1CCC(CNC(c2cnc3n2CCS3)=O)(OC)C1 c1(CC(=O)NCC(C(C)(C)C)NC(C2CCCOC2)=O)noc2cc(F)ccc12 Cc1cn2c(n1)CC(C(N1CCN(C3COC(C)(C)OC3)CC1)=O)C2 C1(CC(=O)NCC2CCCN(C(c3cncnc3)=O)C2)Cn2ccnc2NC1=O C1(C(=O)OC)CC(CN)CN(C(=O)COc2cc(C(C)(F)F)ccc2Cl)C1 CN1CC2(CCNCC2)C1.C(=O)(C(F)C1CC(C)C1)NC(=O)CC1(O)CCC1 c1(CC(CNC(c2cccc(F)c2)CC(C)F)O)cccc([N+](=O)[O-])c1 c1(CSCc2ncon2)c(CNCc2ccncc2)sc2ccccc12 C=CC(C)(C)CC(=O)NCC1(CO)CCN(C(c2cc(F)ccc2CC)=O)C1 c1(C(=O)OC)ccc(NC(c2ccccc2)C2CC(=C3CC3)C2)cc1 C(=O)(CCC(CC)NC(C1(C)CCC2CC2C1)=O)NC(C=C)C1CCC1 C1(CC(=O)N(C(C)CCNC(C2(C)CC2)=O)C)(C(=O)OC)CCCCC1 C1(CNC(c2ccc(CN(C)C)o2)=O)COCCN1C(C1CC2CC1C2)=O C1(NC(CCN(C)CC)=O)CN(C(=O)CC2CC(O)C2(C)C)CC(C)(C)C1 C(=O)(CCN=C(NCc1ccc(Br)c(C)c1F)NCC(C)COC)NC C(=O)(C(C)C(F)F)NCCNC(CC1(CN(C)C(C2(OC)CCC2)=O)CC1)=O Cc1ncc2n1CCN(c1nc(N3CC(C(N)=O)CC(C)C3)c3c(n1)CCS3)C2 C1(OC)CC(C(=O)N(C)Cc2ccncc2F)N(C(=O)Cc2cnns2)C1 CN1CCCC(C(C)(C)C(=O)N2CCC2n2cc(C3CCC=CO3)nn2)C1 c1(C(=O)NCC(C)N(C(CC(C(=C)C)OCC)=O)C)cc2n(n1)CCCC2O c1(C(=O)OC)cnc(C(N2CCCCC2C2CCNC2=O)=O)c(Cl)c1 c1(C(=O)NCC(C)NC(=O)C(F)=CC2CC2)ccnc(OCC(F)F)c1 Cc1nc(Cl)c(NC(=O)CC2CCN(Cc3cc(Cl)c(Cl)cc3F)CC2)nc1C C1(NC(c2c(CC)occ2)=O)CCCCC1NC(=O)C(C)(C)n1cnnn1 N1(C(C=CCN(C)CC)=O)CCCCC1.C1(NC(=O)CO)CCC(C(N)=O)CC1 CC1CC(C(=O)NCC23CC(CN2C)C3)CN1C(=O)C=CC1CCCN1C c1(CC)cccnc1C(=O)N(C(CNC(C1C2(CC2)C12CC2)=O)C1CC1)C CC1CCN(C(=O)Cn2cc(CNC(c3cn(C)cc3Cl)=O)nn2)CC(C)O1 C(c1c(Cl)cccc1Cl)=CC(=O)NCCC1CCN(C(=O)COCC2CC2)CC1 C=CCC(C)(CC)C(=O)N1CC2CCC1CN2C(=O)CC1CC(C)=NO1 c1(C(N2C(CN(C)CC3CCCOCC3)CCC2)=O)nc2c(s1)CN(C)CC2 Cn1c(=O)nc(O)c2ccc(C(=O)NCCC(O)CNC(c3cccs3)=O)nc12 c1(OC)ccc2nc(C(=O)N(C)Cc3ccc(C)cn3)ccc2c1Br C(C(F)(C(=O)NC1(C(=O)OC)CC1)C(C)C)NC(c1ccn(C)n1)=O c1(NC(CCN(C(CC(C)=C(C)C)=O)CC2CC2)=O)cccc2c1CCC2 N#Cc1ccc(NC(=O)CCCN2CCC(C3(N)CC3)C2)cc1Cl C1(NC(C=Cc2cncc(OC)c2)=O)CN(C(C2CC=CC2)=O)CCC12CCC2 C1(C(=O)NC2(C)CCN(C(C)=O)CC2)CC2(CCN(C(C3CC3(C)C(F)F)=O)C2)C1 CC(CO)C(=O)NCC#CCNC(c1cc(C2CCCCC2)[nH]n1)=O CC1(CCC(N2CCC23CCC3)=O)CCCN1C(c1scnc1Cl)=O O=C(CN1C(=O)Cc2cc(F)ccc21)Nc1nc2c(Br)cccc2s1 c1(OCC(C2CC(C)C2)=O)ccc2c(c1)CC(=O)N(C)C2 CC(CC(C)(C)C)C(=O)NC1CCCC1CNC(C1COCOC1)=O c1(C(C(=O)NC(CNC(c2ccc(C)[nH]2)=O)(C)C2CC2)C)ccccc1C N1(C(C2CN(C(C)C)C2)=O)CC(O)CC1CNC(=O)Cc1csc(S)n1 c1(C(=O)NCCCC(C)NC(Cc2cccc(C#C)c2)=O)cc(S(C)(=O)=O)co1 c1(C2(C(=O)NC3C(CNC(=O)C(=O)NCc4ccccc4)C3)CC2)cccnc1 Cc1cc(C(N2CC3C(NC(C4CC(C(F)(F)F)C4)=O)C3C2)=O)ccc1F N1(C(C(C2CCN(C(c3ccnc(C)n3)=O)CC2)C)=O)CCCC(C#N)C1 C1(C#CC(=O)NCC2(C)CCC(NC(C3(CF)CCC3)=O)C2)(CC)COC1 C1(NC(C(C)(C)C)=O)CN(C(=O)CSCc2cscn2)Cc2nccn2C1 C(CCCCC(=O)NCC(CC1CC1)C(=O)NCC1CC2(CCC2O)C1)SC c1(OC)ccc(C(=O)NC(CNC(=O)CC2CC(C)C2)C2CCC2)cc1 c1(OC)cccc(C)c1NC(C12CC(CO1)N(C(C1CC3CCC(C1)O3)=O)C2)=O C1(C(=O)NCCN(C(C)C)C)CCCCN1C(c1cccnc1)=O N1(C(c2[nH]c(=N)sc2)=O)CC2CC1CCC2NC(=O)CCc1cnccn1 N1(C(c2n(C=C)ncc2)=O)CC(=O)NCC1C(=O)NCC1CCCO1 c1(CC(=O)NC2COCC2NC(C2(CF)CC2)=O)cnc(C(F)(F)F)s1 N1(C(c2cccc(C(C)C)n2)=O)CC(CNC(=O)C(C)(Cl)Cl)CCC1C C1(C(C)C)CN(C(c2cccc(O)c2Cl)=O)CCN1Cc1ccc(Cl)cc1F c1(CNC(c2cc(Br)n(C)n2)c2n(CCCC)nnn2)cccc(C(N)=O)c1 Cc1nc2ccc(F)cn2c1OCc1ccco1 C(c1cc(F)cc(F)c1)=CC(=O)NC1(C#N)CCN(C(C(C)=O)=O)C1 C(c1scnc1C)=CC(=O)NCCOCCN(C(C1(Cl)C(C(C)=O)C1)=O)C c1(OC)ccc2[nH]c(=NCC=C(C)C)[nH]c(=NCC3CC(CO)CO3)c2c1 Cc1ccn(CC(N2CC(NC(=O)CC3CCC(C)(C)C3)C2)=O)c(=O)c1 c1(OC)ncc(C(=O)N(CCCCN(C)C(c2ccns2)=O)C)s1 c1(CC(=O)NCC(O)CNC(=O)C(c2ccc(Cl)cc2)O)cccc2cn[nH]c12 O=C(CCC(=O)N1CCC(NC(C2CCCCC2C(=O)O)=O)C1)Nc1nccs1 C1(OC)CC(NC(c2occc2C)=O)CN(C(=O)COOSc2cccc(Cl)c2)C1.O c1(C(N2CC(C)C(CNC(c3cc4n(n3)CCC4)=O)C2)=O)cc(O)cc(O)c1 CC(CC(=O)NCc1ccsc1)C(C)(C)NC(=O)COCCF c1(C(N2C3CC(CNC(CCOC)=O)C2CC3)=O)coc2cc(C)ccc12 c1(C(=O)NCc2c(C(=O)NCC3(CO)CC(C)C3)[nH]cc2)ccc(F)cn1 C1(CC(=O)N(C2(Cc3ccc(Cl)cc3)CCC2)CCO)CCC2COCCC2C1 C1(CNC(COC(CC)(C)C)=O)CN(C(c2ccnn2CC(F)F)=O)CCCO1 CC1C(O)CCCN1C(c1nc(C(N2CCC(OCCF)C2)=O)cs1)=O N1(C(c2cc(C(CC)C)no2)=O)CCCC(CN(C)C(c2cnc(SC)s2)=O)C1 C(c1cccc(F)c1)=CC(N1CCC(C)(C=O)C1)=O.CC(O)CO c1(C(N2C(CNC(c3c(C)ccnc3)=O)CCC2)=O)coc2c1C(=O)CCC2 C1(C)(C(=O)NCC2(O)CCCN(C(c3c(CC)nn[nH]3)=O)C2)CCC(F)(F)CC1 CCC(CNC(=O)C(F)CC1CCOC1)(CC)C(=O)NCC1(C)CC2CCC1C2 c1(CNC(C)=O)ccc(C(=O)N(C)CC2CCN(C(C3(F)CCCC3)=O)C2)o1 c1(C(=O)NCC(C2(OC)CCC2)(F)F)c(C)nn(C)c1-n1cccn1 CC(C)CCCCCC(=O)N1CCN(C(=O)C(=O)N=S(C)(C)=O)CC1C(C)C N#Cc1sc(=NC(=O)C2CC(O)CN2)[nH]c1Cl C(CCC(C(=O)NCCC(COC)OC)NC(C1CC2C=CC1O2)=O)OC C1(NC(Cc2ccc(C)nc2Cl)=O)CCN(C(c2cnc[nH]2)=O)CC(C)(C)C1 Cc1cc(C(=O)OCCC23CCCC2C3)c(C)o1 N1(C(c2nnn(CC)c2C)=O)CC2(CO)CC1(C(N1CCC(F)(C(N)=O)C1)=O)C2 CC1c2ccccc2OC1CNC(c1c(O)cc(N)cc1)=O.C1(C=O)CC1 C(=O)(CC(F)(F)C(F)F)NC1CC(C(=O)NC(C(=O)OC)CO)C1(C)C N1(C(c2c(C)cncc2)=O)CCC2CCCC12CNC(c1c(C)cccc1O)=O Cc1cc(C2(C(=O)N(CC(C)NC(C3OCCOC3C)=O)CC)CC2)cc(C)c1 C1(CNC(C2C(C(N)=O)C2)=O)CC2CC2N1C(=O)C(c1ccccn1)O c1(C(=O)NC(C2(O)CN(C(c3cnccn3)=O)C2)C)cc2c(nc1O)CCOC2 CCCC(C)CC(=O)N1CC(C(=O)N(C)Cc2c[nH]nc2C)CCC1C N1(C(C(C)OCC#C)=O)CC2CC(O)C1C2NC(=O)CCCc1sccc1C CCCCC(C)CCC(=O)N1CCC2C1CCN2C(=O)C(c1ccccc1)=O c1(CC(C(=O)NCC2CN(C(C(C=CCCC)O)=O)C2)C)ccccc1C C1(NC(CC=CC=C)=O)C2CCN(C(c3cnc(OC)s3)=O)C12 N1(C(C(CCSC)NC(C)=O)=O)CC2CN(CC3(c4cccc(F)c4)CC3)CC2C1 CC(C)(C)C(C#N)C(=O)NC(C1CCCCC1)C(=O)NCCCCF N#Cc1cc(S(=O)(=O)NC(=O)C2=CS(=O)CCC2)ccc1Br c1(C(=O)NCCCCNC(C(C)CF)=O)cc(N=S(C)(C)=O)ccn1 C(=O)(C(CO)C(F)(F)F)NCC(C)NC(CN(S(CCCC)(=O)=O)C)=O NS(=O)(=O)N1CC(C(=O)NCCC2COCCN2C(c2cn(C(F)F)cn2)=O)C1 c1(COC)ccnc(N(C)CC2(C(N3CC(CC4CC4)C3)=O)COC2)n1 Cc1cccc(F)c1NNC(=O)C1CCCNC1C c1(NCC(C)OC)nc(N2CCn3ncc(SC)c3C2)nc2c1ncn2CO CC#CCC(C(=O)NCCCCNC(C1(C(F)F)CC1)=O)NC(=O)OC(C)(C)C C1(C(N2CC3C(CN(C(=O)CP(C)(C)=O)C)C3C2)=O)(CC)CCNC1=O c1(C(N2CCCC(CNC(CSCC#C)=O)C2)=O)cc(F)cc2cnccc12 c1(C(=O)NCC2(C)CN(C(c3ccc(O)nc3)=O)C2)ccc(C#N)c(C(F)(F)F)c1 N1(C(C(C)CO)=O)CCC2(CCCC2NC(=O)Cc2ccnc(F)c2)CC1 c1(C(N(C)CC2CN(c3nnc(C(N)=O)s3)CCO2)=O)cnc2c(c1)CCCC2 C1(CC(=O)NCCC(C)N(C)Cc2csc(C3CC3)n2)CCCOCC1 C(=O)(C1CCc2ccc(Cl)nc21)NCC(CCNC(COC)=O)O c1(C(N2CCC(NC(CN3C(C)CCC3)=O)C(O)C2)=O)cc2cc(F)ccc2o1 c1(C(=O)NC2CC(NC(c3cn(CC4(CC)COC4)nn3)=O)C2)cc(Cl)c(Cl)s1 C1(C(N(C)CC2CCCN(C(=O)C(F)(F)C(F)F)C2)=O)Cc2ccccc2O1 n1(CCCNC(CC2CCN(CC(C)(C)N(C)C3CC3)C2)=O)cnc2ccccc12 C(=O)(CC(=O)NC(c1ccccc1)C(=O)NCCN(C)C(=O)N(C)C)NCC c1(OC)cc(C(N2CCC3(C2)CN(C(C2C(C)CC2C)=O)C3)=O)ccc1C#N C1(C)(C(N(CCC(=O)OC)CC)=O)C=CCN1C(=O)C(C)CC#N N1(c2nnc(-c3cnc(-c4scc(C)n4)s3)o2)CCCC2(CCCCO2)C1 Cc1nn(C(C)C)c(C)c1C(=O)NCC(C)NC(c1c(Cl)nsc1Cl)=O c1(C(N2CCN(C(c3cc(C)sn3)=O)C(CF)C2)=O)ccc(O)c2ccccc12 N1(C(CCOCCOC)=O)CCC(N=c2nc(C3CCCCC3)[nH]s2)C(C)C1 c1(N(C)C)ncc(C(=O)NCC(O)CNC(=O)C(F)F)o1 Cc1ccc(CC(N2CCN(C(C3CC34CCOCC4)=O)C(C)C2)=O)c(Cl)n1 c1(C(=O)NC(CCNC(CC(=O)OC)=O)C)cc(OC)nc2ccccc12 C1(C(N(CC)CC2CCC2)=O)CC=CCN1C(=O)CC1CCCN1C c1(C(N)=O)cc(=NCC2CCCCC2NC(c2scc3c2OCCO3)=O)[nH]cn1 C1(NC(C2C(NC(CN3CC(C)(OC)C3)=O)C2)=O)C2CN(C)CC12 c1(CNC(=O)NCC(=O)Nc2ncc(C3OCCO3)s2)ccccc1F C#Cc1cccc(C(N2CC=CC(NC(=O)CC3C(C)(C)C3(C)C)C2)=O)c1 N1(C(c2c(C)csc2)=O)CCC(NC(=O)CC(C)(C)O)C(C(N)=O)C1 C1(OC)CCC2(C(=O)NC(C3CCN(C(C4CNC(=O)N4)=O)CC3)CO)CC12 C1(C(C(=O)NC2CC2)N(C2(CC#N)CC2)CCOC)C2CCCC12 c1(C(=O)NCC(C)(C2CC2)NC(=O)COCc2ccccc2F)cc(Cl)c(Cl)s1 c1(-c2c(C)cccc2F)ccc(S(=O)(=O)NC(c2ccc(F)cc2)C(C)C)s1 C1(CNC(C2(SC)CN(C(C3CN(C)CCO3)=O)C2)=O)CC2CCC2C1 c1(C(=O)NC2CC(C)(C(=O)NC(c3nc(C)[nH]n3)CO)C2)cccc(F)c1 C1(C)(C(=O)NC2(C3N(C(CN(CCC)C)=O)CCC3)CC2)CC(OC)CN1C CC1CCN(CC(C)(C)O)CCN1C(c1ccc(C#N)cc1I)=O Cc1cc(C(N2CCSCC2CCNC(=O)CC2CC3(CC3)CO2)=O)c(C)s1 N1(C(CCCOC(C)C)=O)CCCC2(CCN(C(C3CC34CCCC4)=O)C2)C1 C1(CCNC(C(n2cnc(C#N)n2)C)=O)CSCCN1C(=O)CS(C)(=O)=O Cc1nc(CNC(C(CCC2OCCO2)C2CCCCC2)=O)c(C)s1 C1(NCCNC(CC2(COC)CC2)=O)CCN(C)CC1C C1(C(N2CC(O)(CNC(c3onc(C)n3)=O)C2)=O)CCCSC1C CC1CCC(CC(=O)N(C)CC2(CNC(C3(O)CCCC3)=O)CC2)CC1C C(=O)(C(C)CC(C)(C)C)N1CC(COC)N(C(=O)Cc2cncn2C)CC1 N1(C(CSc2n(C(C)C)cnn2)=O)CCC(CNC(=O)CC2CN(C)C2)C1(C)C CC1(C)CCCCC1C(N1CC2C(CC(=O)NC(C)(CO)C(F)(F)F)C2C1)=O N1(C(CCOC(C)C)=O)CC2(C1)CN(C(c1sc3cccnc3c1Cl)=O)CCO2 N1(C(CN(c2cccnc2)C)=O)CCCN(C(=O)CN=S(C)(C)=O)CC1CO C1(NC(c2cnc(Cl)[nH]2)=O)CN(C(C2(CF)CCC2)=O)CCC12CCOCC2 C12CN(C(=O)Cc3ccc(C#N)cc3)CCN1C(=O)N2.C(CCCC1CC1)NC c1(C(=O)NC(CN(C(C2C(C#C)C2)=O)CC)C)cc(-c2ccco2)no1 C12(NC(Cc3cn(CC)nc3)=O)CC1CN(C(=O)CC13CCCC1C3)C2 C#CCC(C)(CC)C(=O)N1CC(NC(=O)CC2CC2)C(c2nccn2C)C1 c1(CC(C(=O)OCC)NC(=O)C(C)CNC(=O)CC)ccc(O)cc1 C(=O)(C1=C2CCCN=C2NN1)N(CCC)CCSCC.c1(C=O)n[nH]cc1C1CCC1 C=C(C)CC(=O)NCCCCNC(C1SCCS1)=O CC1CN(C(c2cc(O)ncn2)=O)CC1(C)C(N1Cc2c[nH]nc2C1)=O C1(NC(C(COCC)C)=O)CC2(CCC(NC(c3cc(CC)no3)=O)CC2)C1 C12(C(N3CC(C)C(CNC(=O)CNC=O)C3)=O)CCCCC1OCC2 c1(N2CCC(CNC(c3c(O)ncc(CC)c3)=O)C2)nc2ccc(O)cc2s1 c1(C(N2CCCC(NC(CN(C3CCC3)C(C)=O)=O)C2)=O)cc2ccsc2s1 C12(N)CCCC1(F)CN(C=O)C2.C(=O)(CCCCCF)C(C1CN2CCN1CC2)=O c1(C(=O)NCC(C)N(C(CC(C)O)=O)C)cccc(O)c1 N1(C(C=CCC)=O)CCCC(CNC(c2ccc(CO)o2)=O)CC1 C1(CN(C)C(c2cccnc2)=O)CN(C(=O)CNCC2CCCS2)CCO1 c1(C(=O)NCC(c2cn(C)nc2)C)cnn2ccc(Cl)c(F)c12 C(=O)(C(C)(C)C(C)(C)O)NCCN(CC(C)O)C(c1n(CC)ncc1)=O Cc1cc(C)c(CSCCCNC(=O)NC2C=CCCC2)cn1 C(CC(C(=O)N1CCC(C(C)NC(=O)CN(C)C)C1)NC(=O)OC(C)(C)C)SC C1(C)(C)CNC(=O)CO1.CCC(=O)NCC(=O)NC(CC1CC1)C1CCC1 Cc1cccc(C(=O)N(C2CCN(C(c3ccsc3C)=O)CC2)C)c1F C(C1OCc2ccccc21)NC1CCCC(CC)N1 C1(C(=O)NC(CC(=O)OCC)C)C(C)OCCN1C(=O)C(C(C)OC)OC c1(CC)ccc(C(=O)NC2CN(C(=O)C(C)(C)SC)CC2OC)cc1Br C(=O)(C(C)(C)CC(C)C)N1CC(CN(C(c2c(CCC)onc2C)=O)C)OCC1 C(c1ccc(C)cc1)=CCC(=O)NCC1(C(=O)OC)CC1.C12CC1C(=O)NC2=O C1(N(C(=O)C(C)n2cccn2)CC)CCCN(C(C2(O)CCOC2)=O)CC1 c1(N2CC3N(C(c4c(C)c(Cl)ccc4)=O)C3C2)ncnc2sc(C(C)(C)C)cc12 C1(NC(C(C)SCCN(C(=O)C(n2cc(C)cn2)C)CC)=O)CCC(=O)N(C)C1 C(C)(C)(C(=O)NCCC(O)CNC(C12CCCC1C2)=O)OC(C)=O c1(C(=O)NCCCN(C(CCC=CC)=O)CCO)cc2cc(F)cc(F)c2o1 C1(C(N(C)Cc2ncc[nH]2)=O)CC(C)(C)CCN1C(c1ccncc1)=O C12(C(=O)NCC3CN(C(c4[nH]cc(C)c4)=O)CC3O)CC(C)(C1)OC2C C(=O)(C1CCCn2nccc21)N1CC(CCNC(c2n(CC)cc(Cl)c2)=O)C1 Cc1oc(Cl)nc1C(=O)NCCCN(CCO)C(c1csc(C(C)OCCO)n1)=O Cc1cc(C)c(C(=O)NCC2(F)CC(CNC(c3c[nH]c(=N)o3)=O)C2)s1 Cc1cnc(C(=O)NCCC2(C(=O)NCC3(O)CC(C)(C)C3)CCC2)cc1C C12CCC(C)(C1(C)C)C(=O)OC2=O.N1(CC)CCC(N=[N+]=[N-])C1 C(=O)(CCC(C)(C)F)NC1(C)CN(C(CC(C)Cc2ccccc2)=O)C1 C1(NC(c2coc(Cl)c2)=O)CC2CC1CN(C(=O)CCc1cccnc1)C2 C(=O)(C#CC1CCCO1)N(C)CC1CCN(C(CC=C)=O)C1 C1(NC(CCNC(COC)=O)=O)CC2CN(C(c3ncc(C)cc3F)=O)CC2C1 N1(C(c2nncc(OC)c2)=O)CCC(C2(NC(=O)Cc3csnn3)CC2)C1 Cn1nccc1Cn1cc(CNC(=O)C(O)CC2CCOCC2)nn1 C1(COC)CN(C(C2CC3(C2)CC(C)C3)=O)CCN1C(C1CCN(C)C1=O)=O c1(C(N2CCN(C(c3c(C)ncn3O)=O)CC2CO)=O)ccc2c(c1)OCCO2 C1(C(=O)NCCOCC(=O)OCC)=CC(C#N)=C(C2=CCN(C)CC2)NN=C1 N1(C(CC(=O)OCC)=O)CCC(CNC(c2ocnc2C(C)C)=O)C(C)C1 N1(C(c2c(C)csn2)=O)CC2(CC2)CC1CNC(c1cc(C(C)(C)C)n[nH]1)=O n1(CC(=O)NC2CC(NC(CN=S(C)(C)=O)=O)C2)ccc2nc(O)nc(O)c12 C12(NC(Cn3c(=O)sc(C)c3C)=O)CC(C)(C1)OC21CCN(C(=O)CCF)CC1 c1(C(=O)NCC(CC)NC(c2c(SCC)cccn2)=O)c(C)oc(C)c1C c1(C(N2C(CNc3nccc(CCCC)n3)CCC2)=O)cnc(O)nc1O C1(CNC(C(C)C(F)F)=O)CC(C)(C)CN1C(=O)CC1CC(=O)C1 C1(N(C(c2ccc(CCC)[nH]2)=O)C)CC2CCC(C1)N2C(c1coc(C)c1)=O C1(NC(=O)CCC=CCBr)CCCC(NC(=O)COc2ccc(F)c(F)c2)CC1 C1(NC(CN(CCCCC)CCOC)C)CN(C)C2(CCCC2)C1 c1(CC(=O)NC2CC(CNC(C)=O)OCC2)ccc2c(c1)CCC2 CCCCC(C(=O)OCC)Nc1ccc(OCC(=O)OC(C)(C)C)cc1.OCC c1(CNC(C2CC3CC3C2)=O)nc(N2CCC(C(C)OCC)C2)cc(C)n1 C(CC(O)C(=O)N(CC(=O)NCC(C#N)CC)C(C)C)SC C(=O)(C(O)CCCNC(C1CC12CCCCC2)=O)N(C)Cc1ncc(C)o1 C12(CNc3c(C)cc(NC(C4(C(=O)N(C)C)CC4)=O)cc3)CCOC1CS(=O)(=O)C2 n1(CC)nnc2c1C(C(=O)NCC1CC1)CN(C(=O)Cc1ccc(C)nc1)C2 C1(C)(CN(CC(C2CCC(C)(C)CC2)C)C=O)CC2(C1)CC2(F)F N1(C(C2(C)N(C(C(CC)=O)=O)CC2)=O)Cc2ccc([N+](=O)[O-])cc2C1 c1(N(C(C(=O)NCCC2CC2)c2cnn[nH]2)C)cccc(CC(N)=O)c1 N1(C(c2cc(C(C)(F)F)on2)=O)CCC(=CCNC(=O)CN2CCSCC2)CC1 C1(CC(=O)NC2CCC(F)C2)(Cn2cnnc2)CCCCC1 C1(NC(=O)CC2CCC(CC(=O)Nc3cccc(CO)c3)C2)CCc2nc[nH]c2C1 c1(N2CCN(C(C=CC=CCC)=O)CC2)cc(=O)n2cc(Cl)ccc2n1 N1(C(c2nc(C)sc2)=O)CC(CNC(=O)C(C)N(C)C2CC2)C(F)(F)C1 c1(C(=O)NCC2C(NC(C(CCSC)OC)=O)CC2)cnn2ccsc12 C12(C(=O)NCCOCCNC(c3c(N)ncc(Br)n3)=O)CCCC(=O)N1CCC2 N1(C(c2c(C)cc(F)s2)=O)CCC(C)(CCNC(=O)CCc2cnc(O)[nH]2)CC1 N1(C(C2C(CC)CN(C(C34CCC(C3)OC4C)=O)C2)=O)C2CCCC1CN(C)C2 C(C(F)C(=O)NCC1(CNC(=O)C(C)SC)CCCC1)N(CC)CC C=CC1(CC(=O)NCCC(C)SC)CN(C(=O)Cc2ccccc2F)C1 N1(C(C(C)Cn2ccnc2)=O)CC(=O)NCC1C(=O)Nc1cccc(F)c1 C1(CCO)(NC(C(C)NC(N)=O)=O)CN(C(=O)CCNC(N)=O)C1 c1(C(N2CCC(O)(CNC(COCCCOC)=O)C2)=O)cnn2c(=N)[nH]cnc12 C1(N(C)C(c2ccc(Br)c(O)n2)=O)CN(C(=O)Cn2ccnn2)CC12CC2 C(C(CC(C)C)NC(C1CN(C(C)C)CCO1)=O)NC(CCc1ccc(C)o1)=O O=C(NNc1ccc(C(F)(F)F)nn1)NC1(c2ccc(C(F)(F)F)cc2)CC1 c1(C(CNC(=O)CC2OCCO2)NC(c2ccc(CC)o2)=O)ccc(C)cc1 C=C1Cn2c(C(=O)NC(CCN(C(=O)C(C)(C)SC)C)C(C)(C)C)nnc2S1 C1(NC(CC2CCC(=O)NC2)=O)(CNC(=O)C=C2CCNC2)CCCCCC1 c1(C(=O)NC(C2CC=CCC2)C(=O)NCC2CC(F)(CF)C2)cnc(Cl)s1 C1(NC(c2ncn(CC)n2)=O)C2CCN(C(c3cncc(N)n3)=O)C12 N1(C(c2cn(C)c(=O)nc2O)=O)C2CCC1C(F)C(NC(=O)CC1(CO)CC1)C2 O=C1NCC2(CCCN(C(C3CC(C(=O)Nc4cnccc4Cl)C3)=O)C2)O1 CC1(C(=O)NC2(C(=O)NCC(O)CF)CCCC2)CCOC1 O=C(C1=CCS(=O)(=O)C1)NCC1CC(NC(C2CC23CCSCC3)=O)C1 C(CC(C)(C)CC(=O)NC(C)(C)CC=CC(=O)NC1(CO)CC(O)C1)OC N1(C(c2occ(C)c2C)=O)CC2CCCN(C(C3CCC(=O)N(C)C3)=O)C2C1 C1(CNC(C(c2cn(C)nc2)O)=O)CN(C(=O)Cc2ccno2)CCO1 c1(C(=O)NCC2C(NC(Cc3c(C)occ3)=O)CCC2)ccc(N)c(F)n1 c1(C(=O)OC)ccc2c(CNCc3ccc(N(C)C)nc3)c[nH]c2c1 CCC(C)(C)CCCC(=O)N1CCCCC1CCNC(=O)CCCF n1(C(C)NC(=O)C=COCc2cccc(F)c2)cnc2cc(Br)ccc2c1=O c1(C(N2CCCC(NC(c3n(C)nc(C)c3F)=O)C2)=O)ccc(C#N)cc1Br c1(COCCC(=O)N(CCCNC(C2C(C)C2)=O)C2CC2)ccc(F)cc1 c1(C(N2CC(C(C)C)N(C(C3C(C)C3(F)F)=O)CC2)=O)ccc2c(c1)CC(C)O2 C(C#Cc1ccccc1)NC(C(=O)OC)CC1CCCC1 Cc1nccc(C(=O)NCCCNC(C2(C3CCCO3)CC2)=O)c1C c1(C(=O)OC)ccc(S(=O)(=O)Nc2ccccc2OCCF)c(C)c1 C1(NC(C(C)SCC)=O)CN(C(C2(C3CCCCO3)CCC2)=O)C2CCCCC12 N1(C(c2nc(C(C)C)sc2)=O)CC(NC(=O)CC2CCOC2C)CCC1C C1(CCNC(CSCC)=O)CN(C(=O)COC2CC2)CCS1(=O)=O c1(C(=O)NC2CC(OC)CN(C(C3CCC(=O)NC3C)=O)C2)cc(C)cc(O)n1 c1(C(=O)NCC2CN(C(c3c(C)con3)=O)CC2C)ccc2c(c1)NCCC2=O Cc1csc(CC(=O)NCCCC(=O)NCC2(C)CCCS2)c1 c1(C(=O)NCC2C(NC(C(C(C)(C)O)F)=O)CC2)cc(N)c(F)cc1F C12(CCNC(c3c(OC)c[nH]n3)=O)CCC1CN(C(c1cc(C3CC3)cs1)=O)C2 CCCC(C(=O)NC(c1ccnn1C)C(=O)NC(C)(COC)C(N)=O)OC CCCC(CCCNC(=O)C(N1CC2(CCOCC2)C1)=O)NC(=O)CC(C)C c1(CNC(c2c(C)noc2C)=O)ccc2c(c1)CN(C(C1(C(N)=O)CCC1)=O)C2 c1(CCCC)cc(C(=O)NC2CC(OCC=C)C2(C)C)c(C)o1 N(C1CCCc2ccc(C(C)(C)C)cc21)C(C=O)=O.c1(CNCC)ncccn1 c1(C(N(C(CC(F)F)C(=O)NC2C(C)CCC2C)C)=O)ccc(=O)n(C)c1 Cc1cc(O)ccc1-c1cnc(C(=O)Nc2ccc(OC(F)F)cc2)cc1C n1(C(C)C)cc(S(=O)(=O)NC2(n3cc(Br)cn3)CC2)nn1 CC1(C)CC(CNC(=O)COCCF)CN1C(=O)C=Cc1ccccc1 C(CCCCN)N(C(C)C)C(C1CC(F)C1)=O.C(=O)(C(C)SC)C(=O)CSC(F)(F)F N1(C(CCCC2CC2)=O)CCCN(C(=O)C(C)(C=C)CCNC(C#C)=O)CCC1 CCC(C)C(O)C(=O)N1CCC2C(NC(=O)CC(Cc3ccccc3)CC)C2C1 N1(C(C(C=CC)O)=O)CCN(C(c2cnc(CC(C)C)[nH]2)=O)CC1C(C)(C)C C1(NC(CS(C)(=O)=O)=O)C(CNC(C2(C(F)(F)F)CCCC2)=O)CCC12CCC2 C1(CCC)CN(C(C2CCC2C)=O)CC1C(=O)NC1CCCC1F N1(C(c2c(C)scn2)=O)C2CCC1C(NC(c1ccc(N(C)C(C)C)cc1)=O)C2 C#Cc1cc(C(=O)NCC2CCC(C(=O)NC3(C)CCCC3CC)O2)ccc1C CCC(C)C(CC(=O)NCC1CCCCO1)NC(=O)Cc1ccn(C)n1 c1(CNC(C=C(C)Cl)=O)ccc(C(C)NC(c2cc(C)no2)=O)cc1 C(CC1C(=O)N1)n1cc(CSCC)nn1.C1(C(=O)O)CC2CCC1C2 N1(C(CC2(OCC)CCC2)=O)CCOCC(NC(=O)C(OC)OCC)C1 N1(C(C(C(=O)OC)OC)=O)CC2(CCC2)CC1CNC(=O)C=Cc1cccnc1 C1(C(N2CCC(NC(=O)NC)C2)=O)CCC2(CC2)N1C(=O)C(c1cncn1C)C C(=O)(CCCCC(N)=O)NC(C(=O)NCC(C)CC1CCCC1)CCN(C)C C1(CC#C)(C(=O)NCCC2(O)CN(C(=O)Cc3ccccn3)C2)CC=CCC1 S(=O)(=O)(c1c[nH]ccc1=NC(C)CCCCCCCO)N1CCC(O)(CC)CC1 c1(C(=O)NC(CN(C(c2c(C(C)C)nns2)=O)C)C)cccc2ncnc(O)c12 Cc1nc(CC(=O)NCCCc2ccn(C)n2)c(Cl)s1 c1(-c2c(F)ccc(C(=O)Nc3cc(OCC)ncc3)n2)ccc2oc(C)nc2c1 C(C(C)CC(F)F)NC(C1(N(C(Cn2c(C)ccn2)=O)C)CC1)=O c1(C(C)O)ccc(C(N2CCCC2CN(C(=O)C(c2ccccc2)F)C)=O)cc1 C1(CCC)CCCC1C(=O)NCCOCCNC(c1nccn1C(C)C)=O C1(C(=O)NCC(CCOC)NC(c2cc(OC)n[nH]2)=O)Cc2cc(C)ccc2S1 O=S(=O)(c1nc(NCCCCl)ccc1Br)NC(c1ccccn1)CN1CCC1 CC1=C(C(=O)NCC(C(C)C)NC(C2CC(F)CN2C)=O)CCC1 C1(C(=O)NCCN(C(C)C)C)CCn2cc(C(F)(F)F)nc2C1 CCCC(C)CCCC(=O)N(C)CCOCCCNC(=O)CCC1CCC1 C1(C(=O)NCC(CNC(Cc2nc(C)oc2)=O)F)CCCS(=O)(=O)C1 C1(NC(c2c(C)c(C3CC3)on2)=O)CC2CC(C1)N(C(=O)C=CC1CCCO1)C2 Cc1cc(O)nnc1C(N1CC(NC(C2CCC(C(N)=O)C2)=O)C(F)C1)=O n1(CC)cc2ccc(C(=O)NC(CN(C(=O)C=C3CCSCC3)C)CC)cc2n1 CC(C)CC(O)C(=O)NC(CC(=O)NCC1CC=CCC1)C(F)F c1(OC)ccc(CC(N2CCOCC2C(N2CC3CC2CN3C)=O)=O)cc1OC C1(C(=O)NC2CC3C(NC(CC4CC(=O)NCC4)=O)C3C2)CCC([N+](=O)[O-])CC1 C1(NC(C=Cc2ccc(C)o2)=O)CC1C1CCN(C(=O)C(O)CC2CC2)CC1 CCC(C(=O)NC(C1(O)CN(C(=O)C=CC(F)(F)F)C1)C)OC1CCCCC1 CN=c1[nH]cc(C(N2CCC(C(C)C(=O)NC3CCC(C)(C)C3)CC2)=O)o1 C(C(C)C(=O)N1CCC1C(=O)NCCCc1nncs1)OC C1(CNC(C(C)C(C)(F)F)=O)CCCC2(CN(C(=O)CCCC#N)C2)O1 C1(CC)CN(C(C2CCC2)=O)CCN1C(C)=O.c1(C(=O)N)ccnc(-n2cccc2)c1 c1(C(N2CCC3(CC2)CC(CO)C3)C(=O)NC2CC2)cc2c(cn1)OCCO2 C12(NC(=O)C=C3CCSCC3)CCCC1N(C(c1ccc(Cl)cc1F)=O)CC2 C1(CNC(C=NOC)=O)CN(C(C2CC(n3ccnn3)C2)=O)CC(C(F)(F)F)O1 N1(C(C(CSC)O)=O)CC(C2(NC(=O)C(c3ccccc3)NC(C)=O)CC2)C1 N1(c2cccc(OC)c2)CCCN(C(c2ccc(F)cc2CN)=O)CC1=O N1(C(c2cc(C)oc2C)=O)CCCN(C(=O)CCCC(C)C)C(C(C)C)C1 O=C(NOC1CCCC1)C1=CC(O)C(NC(c2nsnc2O)=O)C1 c1(C(C)NC(=O)NCC(c2ccccn2)(C)C)ccc(F)c(Cl)c1 C1(C(=O)NC2CC(NC(C3(CN(C)C)CC3)=O)C2)CC12CCC2 N1(C(Cn2ncc(C#C)c2)=O)CCCCC(NC(=O)C(C=C)CC)C1 Cc1ccc(C(=O)NC2CN(C(=O)Cc3ccccc3O)CC2F)cc1Cl N1(C(C(=O)NCC2CCCN(CC)C2)=O)CCN(C(C)C)CC1C N(C1CCCOc2cc(Cl)ccc21)C(C(=O)N(C)CC1CC2CC2C1)=O N1(C(N2CCC3(CC(OC)(OC)C3)CC2)=O)C(CO)CCC1C1CCCO1 C1(CNC(Cc2n[nH]c(=N)s2)=O)Cc2ccccc2CN1C(C1CC2CCC2C1)=O C1(CNc2cc(NCc3c(NC)nccc3)ncn2)CCOC(C)(C)C1 C(c1ccc(O)c(O)c1)=C(C(=O)NCCCC(C)NC(c1n[nH]cc1Cl)=O)C Cc1sc(O)nc1C(=O)NCc1cc(C(=O)NCC2CSCCO2)co1 N1(C(CSCCC#N)=O)CCC(O)C(NC(c2cccc(F)n2)=O)C1 N1(CCn2ncn(CC)c2=O)CCC(=O)N(Cc2ccnn2C)C1=O c1(C(N2C(C(=O)NC3C(CCC)C3)CN(C)CC2)=O)ccc(C#N)c(C)c1 C(=O)(CCCNC(N)=O)NC1(C(=O)NC2(CC(C)C)CC2)CC1 CC(C)(C)CC(C(=O)NCCCC1CC1)NC(=O)CC1CC(C)(C)C(=O)N1 Cc1nn(C)cc1C(=O)NC1CC(C)(NC(c2cncc(C(C)C)c2)=O)C1 C1(NC(c2c(OC)oc(C)n2)=O)CCN(C(=O)CC(=O)NC2CC2)CC1C(C)C c1(N2CC(C(N)=O)OCC2)cccc(S(=O)(=O)NC(Cc2ccsc2)CO)n1 C(=O)(C1CCCc2cccnc21)N(C1CCCCN(C(C2(CCF)CC2)=O)C1)C C(N=C(NCC(C)(C)C)N1CCC1)c1ccc(C)cn1 C12(CNC(c3ccc(O)c(Cl)c3)=O)CCC1CCN2C(=O)C1=CCCC1 N1(C(C(COC)N(C)C)=O)CCC2C(CCCN2C(c2ncc(F)cc2F)=O)C1 C(c1ccc(Cl)cc1)=CC(=O)NC1CN(C(C(c2ccccc2)C)=O)CC1F N1(C(CSc2ccc(OC)cc2)=O)CCN(C(=O)C(O)C(C)C)CC(O)C1 c1(N2CCC(NC(Cc3cc(CC)on3)=O)C(F)C2)ncc([N+](=O)[O-])cc1Cl C(=O)(C1CCCn2cncc21)N1CC2CCN(C(c3cccc(C)c3)=O)C2CC1 CCCCCC(O)C(=O)NCC1(CNC(c2cc(OC)ncn2)=O)CCCC1 C1(c2n(-c3c(C)cccc3)nc(CCC(C)(C)C)n2)CC2CCC1CC2 Cc1c(NC2CCCCCC2F)ncnc1NC1CCN(CCF)C1 Cc1ccc(F)c(C(=O)NC2CCN(C(c3ccc(N)cc3C)=O)C(C)C2)c1 CC(C)C(F)(F)CC(=O)NC1CCC(N(C)C(c2cc3n(n2)CCO3)=O)C1 c1(C(=O)NC2CCCC(CNC(C3CCCCC3)=O)C2)cnc(O)c(Br)c1 C12(NC(=O)NC3CNCC34CS(=O)(=O)C4)CC3CC(C1)CC(CO)(C3)C2 N1(C(CC2N(CC)CCOC2)=O)C2CCC1(CNC(=O)C(C)(Cl)Cl)CC2 C(C(C)(C)CC(=O)NCCCn1ccnc1)NC(C(C(C)C)=O)=O CC1(CNC(=O)CN2C(=O)CCC2=O)CC(F)(F)CN1C(=O)C1=CCCCO1 CCC(O)C(=O)NCCC(C1CC1)NC(=O)C(F)C1CCCC1 CC(F)(F)C(C)(C)C(=O)N1CCCCC1Cc1cn(Cc2ccccc2F)nn1 CC(C)C(O)C(=O)NCCn1cnc(C(=O)NCc2cscn2)c1 c1(C(=O)NC2CN(C(C(CC)SC)=O)CC(C)(C)C2)cc(OC)c(S(N)(=O)=O)s1 N1(C(c2ccc(Cl)c(O)c2)=O)CC2CCC(C1)N(Cc1c[nH]c(Br)c1)C2 N1(C(C2CCN(C(=O)CCOCC3CCC3)CC2)=O)CC(O)CC12CCOC2 N1(C(c2csnn2)=O)CC2(CCN(C(=O)CC3CCCCO3)CC2)C1 C1(N(C(C2ON=C(C)C2)=O)C)CCCN(C(=O)CC#N)C1 C1(NC(CCN(C)CC)=O)CCCCC1NC(c1nccnc1C)=O Cc1ncn(C)c(=O)c1C(N1CCCC(CNC(=O)C(C)c2cccs2)CC1)=O N1(C(C(=O)NCC=C)c2cncs2)CCCC(Cc2ccn(C)c2)C1 C(=O)(C1=C(Cl)CCC(C)C1)NC1(C)CC(NC(CN(C(C(C)C)=O)C)=O)C1 c1(C(N(C)CC2(O)CCN(C(C3(C=C)CCC3)=O)C2)=O)sc2ccccc2c1C c1(C(=O)Nc2c(CC(N3C(C)CCC3)=O)cccc2)cccc(C#N)c1 Cc1nsc(C(=O)C(CCCCCN)=O)c1N.N1(CC(=O)NC)CC=CC1 c1(CN(C(C(CC)C)CO)C(C)=O)ccc(C)cc1C c1(CC(N2C(CNC(CC(C)N(C)C)=O)C=CC2)=O)cccc2cnccc12 c1(-n2ncc(CNC(=O)NCc3ccccc3O)c2)cccc(F)c1 N1(C(CC(C)(C)N(C(=O)C2=C(C)CCC2)CC)=O)CCN2C(=O)NCC2C1 C1(C(C(=O)NCCCCC(=O)NC)(C)C)CCCCN(C(C2CCOC2)=O)C1 c1(OCC(=O)OC)ccc(C(N2CC(CNC(=O)C(O)C3CC3)C(C)C2)=O)cc1 c1(OC)cc(C(=O)NC2CCCC2CNC(=O)CNS(=O)(=O)C2CC2)cc(C)n1 C(C(O)CC(=O)NC1C(C)CCC1C)NC(CC1ON=C(CC)C1)=O C1(C(=O)NCC(C)OC)CCCN1NC(=O)C1COCCN1C(C)=O c1(SC)nc(O)nc(C)c1C(N1C2CCC1CN(C(C1(F)CC1C)=O)C2)=O C(=O)(C1Cc2c(Cl)cccc21)N1C(CN(C(=O)Cn2cnnn2)C)CCC1 N1(C(C(CC)OC)=O)CCCC(C2CCN(C(c3ccncc3F)=O)CC2)C1 c1(C(=O)NC2CN(C(c3c(C)nc(C)[nH]3)=O)CC23CC3)cc2cccc(Cl)c2s1 C1(C(N(CCCC)CC)=O)CC(F)(F)CN1C(C12CCCC(CO1)C2)=O Cc1nc(C(F)(F)F)sc1C(=O)NC12CC1CN(C(C1(CF)CC(F)(F)C1)=O)C2 N1(C(CCCCCN(C(=O)CN2CCCC2=O)C)=O)CCCC2NC(=O)CC12 CCCC(CCCO)C(=O)NC1(CNC(=O)C=C2CCC2)CC1 O=C(C1=CCCCC1)NC1CN(C(=O)CCC2CCCC2)CC1F C12CC(CN1)CC(=O)NC2.c1(NC(C2C(CC)C2)=O)ccc(COC(C)(C)C)[nH]1 N1(C(C(C(C)NC(c2scc(OC)c2)=O)C(C)C)=O)CCN2CC(O)CC2C1 c1(OCCCC)ccc(C(N2CCC(C(=O)NCC3C=CCC3)CC2)=O)c(Cl)c1 C1(OC)(CNC(=O)C2=CCCSC2)CCN(C(c2cc(C)cs2)=O)CC1 C1(NC(=O)NC2CC2C2CC2)(CO)CC2CCC1C2 CN1CC(CNC(C2CC(O)CN2C(c2nn(C)cc2Cl)=O)=O)CC1=O C1(NC(c2cc(OC)cc(Br)c2)=O)CCC2CC1CN2C(=O)CCC(C)C C(=O)(CCCCCCNC(=O)CC1CCCC1(C)C)Nc1c(C)ncnc1 c1(C(=O)NCCC2CCN(C(C3(CCCC)CCC3)=O)C2)c(CO)noc1C C(=O)(C(C(C)C1CC1)N1CCCC1CN(S(C)(=O)=O)C)NCCCCCC CCC(CC)C(C)C(=O)NCC1(CO)CCN(C(C2C(C)(C)C2(F)F)=O)CC1 c1(C(=O)NC2CC(NC(c3nc(CCCC)sc3)=O)CC2O)cc(O)ccc1C N1(C(CCCSC)=O)CC23CCCC2(C1)CN(C(c1nc(C)n(C)n1)=O)C3 C1(NCc2nc(C)nn2C)CCN(C(C2CCCCC2)=O)CC1C C1(CNC(C(C2CCCO2)NC(CCSCCCC)=O)=O)CN(C(C)=O)CCO1 N1(C(C2C(C(C)(C)C)OCC2)=O)CCC2(CC1)CN(C(c1cscn1)=O)CCO2 C1(n2ncc(C(N(C)C)=O)n2)CCN(C(c2cnc(C3CC3)cn2)=O)CC1 C1(CC=C)(C(=O)NC2(C)CCCC2)CN(C(=O)CCCc2ncco2)C1 CCCCC(CC)CC(=O)NCc1cc(C)c(C(=O)N(CC(C)OC)C)o1 C1(C(C)N(C(CN2CC(CC)C2)=O)CC)CCCN1C(c1cnc(C2CC2)[nH]1)=O n1(CC)ncc2c1CC(C(=O)NC1CN(C(C3(OC)CC3)=O)CC1(C)C)CC2 N1(C(CNC(C(CC)C)=O)=O)CCN(C(c2sc(C)nc2C)=O)CC1C1CC1 C#Cc1cc(F)c(C(=O)N(C)CCN(C)C(c2ccc(=NCC)[nH]c2)=O)cc1F C1(CNC(CCOC)=O)(OC)CCN(C(c2csc(C(C)=O)c2)=O)CC1 CCCC(C)CCCC(=O)N(C1CC2CCC(C1)N2C(c1cn(C)[nH]c1=N)=O)C N1(C(C(CCSC)OC)=O)CCC2C(C1)CN2C(=O)CN1CCCCC1 c1(OC)ccccc1C(N1CC(NC(c2coc(Cl)c2)=O)C2CC12)=O CN1CC(C)(C(=O)NNC(c2ccc(Cl)c(Cl)c2)=O)CCC1=O N1(C(C(=O)N(C(C)CNC(=O)CC2CC3CC3C2)CC)=O)CCCC(C)C1 c1(C(=O)NC(CCNC(Cc2cccc(C(=O)OC)n2)=O)C)cncn(C)c1=O c1(N2CC(OC(C)(C)C)CC(OC)C2)nc(C)[nH]c2nccc1-2 CC1(CC(=O)NCCCOC2CC2)CCN(C(c2ccc(F)cc2)=O)C1 CC(CC(C)NC(=O)CC1(CS(C)(=O)=O)CC1)NC(=O)CCCn1cccn1 C(CC1CCCCC1)(C(=O)NCCCN(C(C1CC1C(C)C)=O)C(C)C)OC C1(CNC(C2(n3c(C)cnc3)CC2)=O)CN(C(c2cnc[nH]c2=N)=O)CCC1C N1(C(CSCC#C)=O)CCC(C2CCCN(C(=O)C(c3cnn(C)c3)C)C2)C1 c1(N(CC(N2C(CN(C)C(C3CN(C)C(=O)N3)=O)CCC2)=O)C)ccc(Cl)cn1 c1(C(=O)NCC2C(C)CN(C(=O)Cc3cocn3)C2)c(F)ccc(Cl)c1N c1(CC(N2CCN(C(C(CC=C)(C)C)=O)CC2C)=O)csc2sc(C)cc12 N1(C(C(CC)C2CCOCC2)=O)CCCC(C2CCNC2=O)C1 CN1CCN(C(=O)CC23COC(C2)C3)C(CNC(=O)Cn2nc(Cl)ccc2=O)C1 C(=O)(C(C)(C)C(F)(F)F)NC(C1CCCN1C(C1CCC(F)(F)C1O)=O)C Cc1nc(NCC2CN(C(c3cc(Cl)no3)=O)CCC2C)c(Cl)cc1[N+](=O)[O-] C(c1cccc(Cl)c1)=CC(=O)NC1C(NC(CN(CCC)C)=O)CC1 C1(C(N2CC(CNC(C3(C)CCNC(=O)C3)=O)C(O)C2)=O)CCC(N=[N+]=[N-])CC1 CCS(=O)CCNC(=O)CC1CC1C.C12CC1C(C)NC2=O C=CC(C)(C)CCN=c1[nH]c(=NC2CCC(C)(CN(C)C)CC2)c2ncccc2[nH]1 c1(N2CCC(NC(=O)NC3CS(=O)(=O)C3)CC2)ccc2nncn2n1 C1(OC)CCCC(C(N2CC(C)(NC(=O)C(c3ccc(C)o3)C)C2)=O)C1 NC1CC=C(C(=O)N2CCC(n3cccn3)(Cc3ccccn3)CC2)C1 N1(C(C2C(OC)CCC2)=O)CCCOC(CNC(=O)CCCC2OCCO2)C1 N1(C(C(CCC)CNC(=O)C(C)CO)=O)CCCC(C)(C#N)C1 c1(C(N2CCC(CNC(c3cc(C)ns3)=O)C2)=O)cc2c(C)cccn2n1 C1(N(C(CSCC#C)=O)C)CN(C(=O)C(C2CCCN(C)C2)(C)C)CC1(C)C C1(C(=O)NCC2C(NC(Cc3c(C)nccc3)=O)CC2)Cc2nnc(C)n2C1 CC(C(=O)N(CCCN(C)C(c1noc2c1CCCCC2)=O)C)C(C)S(C)(=O)=O c1(C(N2CC(NC(C3CCCCC3)=O)C3(C2)CC3)=O)cnn2cccc2c1 c1(C(N2CCC(NC(C3ON=C(C(C)C)C3)=O)C2C)=O)c(O)ccc(Cl)c1O c1(OC)cc(C(=O)NCCOCC(=O)NCC2CCCC2CO)on1 N1(CC(=O)NC2C(CC)CN(C(C3CC3(F)F)=O)C2)C(=O)NC(CC)(CC)C1=O c1(CC(N2CCN(C(c3ccc(C#C)cc3)=O)C3C2C3)=O)ccc2c(c1)CCC2 C1(C(N2CCC(CCNC(c3ncc(Cl)s3)=O)C2)=O)CCCCC1(F)F N1(C(CCN(CC(=O)N)C)=O)CCCC(OC(C)=O)C1.C1(O)CCCC1 C(c1ccccc1S(=O)(=O)c1ccoc1)N1C(C)CC(c2ccc(CN)cc2)CC1 Cc1ccc(C(=O)NCCC2CCCN(C(c3cncn(C)c3=O)=O)C2)c(F)c1 C1(C(N(CC#CC)C)=O)CCOCCN1C(=O)CCCC1CC1 c1(C(=O)NCCC(C)(C)NC(c2scnc2C2CC2)=O)ccc(C2CC2)nc1 C(=O)(C(CC(C)C)C(N)=O)N1CC(C=C)C(NC(=O)Cc2cncn2C)C1 CCS(=O)c1ccccc1C(N1CCCC(CNC(=O)CCNC(C)=O)CC1)=O C(C(CC1CC1)C(=O)NCCN1CC=CCC1)NC(C1(C)CC(=C)C1)=O CC1CCN(C(=O)OC(C)(C)C)CC1NCCC(C)(C)N1CCOCC1 C1(C)(NC(c2n(CCC(=O)OCC)nnn2)c2ccn(C)n2)CCCOC1 C1(CNC(C2C(=C)C2)=O)CCC12CCN(C(c1cnn3ccc(C)nc13)=O)CC2 C(C(=O)N(CC(=O)NCC1CCCO1)C1CC1)(C(C)C)OCC N1(C(c2c[nH]c(=NC)s2)=O)CCC(C)(C)C1CC(=O)NC1C(=O)OCC1(C)C C(=O)(C1Cc2c(Cl)cccc21)NC(C)CCN(C)C(c1csc(CO)n1)=O Cc1cccc(CC(=O)NC2(CCNC(C3COC(C)C3)=O)CCC2)c1 c1(CNC(=O)C=Cc2cocn2)cnn2c1CN(c1nccc(CO)n1)CC2 N1(C(C2CCC(=O)C2)=O)CCN(C(=O)Cc2ccsc2Cl)C(c2ncc[nH]2)C1 C1(CC(N2C(C)CCC(NC(CC=C(C)C)=O)C2)=O)CC2(C1)CC1(CCC1)C2 N1(C(CC(C)n2ccnc2)=O)CCOCC1CN(C)C(c1ccncn1)=O C(c1ccc(C)o1)=CC(=O)NC(C1(O)CN(C(C(C2CC2)OC)=O)C1)C C1(NC(=O)NC2CCN(c3ccc(COC)cc3)C2)Cc2ccccc2C1 N1(C(C(CCC)CNC(=O)CP(C)(C)=O)=O)CCn2c(C)cnc2C1 N1(C(C(C)SCCCC)=O)CC(NC(=O)C(c2ccccc2)OCC)CC1CO N(C(=NCc1ccco1)NCC(C1CCN(C)CC1)OC)Cc1n(CC)nnn1 c1(CNC(=O)NN2CCCC(C3CCC3)CC2)cccc2oc3ccccc3c12 c1(CC(=O)NCC2C(CNC(C(CC)C)=O)C2)ccc2c(c1)CCCN2C N1(C(c2c(C)n(C)cn2)=O)CCN(C(=O)Cc2nnc(O)s2)C(CO)C1 CC1OC2(C(=O)NCCCCC(C)NC(=O)C(C)(C)C(N)=O)CCC1CC2 N1(C(=O)OC)CC2CCC1C(C(N1CC3CC(C1)N(C(c1ccsc1)=O)C3)=O)C2 c1(CC(=O)NCC2(NC(Cc3c(C)con3)=O)CC2)ccc(Br)c(F)c1 C(=O)(CCCNC(=O)C[N+](C(=O)C(C1C=CCCC1)(F)C)([O-])NC)NC(C)(C)C CN1CCC(C2(C(=O)NCCCN(C(=O)Cc3ccc(O)c(Cl)c3)C)CC2)CC1 C1(CN(C(C2CCCN2C)=O)CC)CCN(C(C2CCC=CO2)=O)CC1 c1(NC(CC(CC)NC(c2ccc(C)n2C)=O)=O)ccccc1C#N N1(C(C(C(C)C)OC)=O)CC2(CCCC2)C1C(=O)NCC(=O)N1CCCO1 c1(C(=O)NC2(CNC(CC(=O)NC)=O)CCCCCC2)cccc(F)c1C#N N1(C(c2ccc(CC)nc2)=O)CC2(C)CC1(C(=O)NCCOCCCF)C2 c1(CCC)nc(C)c(C(=O)N(CCNC(=O)COC(c2cccc(OOC)c2)C)CC)o1.O c1(C(=O)NC2C(C)N(C(c3cnc4n3CCS4)=O)CC2)cc2c([nH]1)CCC2 c1(C(=O)OCC)n[nH]c(CC)n1.n12nnnc1C(C1CC3CC3C1)NCCC2 C(=O)(C(C)(F)CC1CCCC1)OC(C)(C)C.C12(OCCO1)CCNC2 c1(C(=O)NC2C(C=C)CN(C(=O)C(C)NC(=O)CC)C2)cn(C)c2ncccc12 CCC(F)(F)CC(=O)NC1CC(C(N2CCN(C)CC2)=O)CC1O N1(C(CCC(N)=O)=O)CCC2(C=C(C(=O)N3CCCC(C4CCC4)C3)C2)C1 c1(C(=O)NCCN(C(c2coc(O)n2)=O)CC)c(C(C)=O)[nH]c2ccccc12 C(=O)(C(CNC(C1CCCCC1O)=O)C(C)C)NC1C(C(=O)OC)OCC1 CCC(CC(=O)NC1(CO)CCCN(C(c2ccc(O)nn2)=O)C1)CC(F)(F)F C(C(=O)NNC(=O)CN1CCOCC1=O)c1c(C(=O)OC)ccc(Cl)c1 Cc1cc2ncc(-c3cc(CO)cs3)cn2n1 N1(C(C2CC2Cl)=O)CCCC2(CCN(C(=O)C(F)(F)c3nccs3)CC2)C1 C=Cc1cncc(C(N2CC(NC(C3C(C)C3C)=O)C(C(F)F)C2)=O)c1 c1(CC(C)C)ncc(C(=O)N(C(C)CNC(c2cscc2C2CC2)=O)C)[nH]1 c1(CN(CC(=O)Nc2ccc(OC)cc2)C)cccc(OC)c1F C1(OC(CC(C)(C)C(=O)NCCCn2cc(C(O)C3CC3)nn2)=O)C(F)(F)C12CCC2 N1(C(C2CCC(C(=O)OCC)CC2)=O)CCOCC(NC(=O)C2=CCCS2)C1 CN1C(=O)OCC1C(N1CCC(C)(NC(=O)CSc2nnnn2C2CC2)C1)=O C1(C#CC(=O)NC2(C3CN(C(c4cc(N)cnc4Cl)=O)C3)CC2)(CC)CC1 C#Cc1ccc(C(=O)NCCN2CCN(C(=O)C(C3CCOC3)OC)CC2)nc1 CC1CCCCCN1C(C12CC(NC(C3CCC(C(N)=O)C3)=O)(C1)C2)=O C1(CCC)CCCN(C(c2cc(CNC(c3cncs3)=O)on2)=O)CC1 N1(C(C(C2CCC2)OC)=O)CCC(OCCNC(=O)CCc2nc(C)cs2)C1 c1(C(=O)NCC(C2CCN(C(C(CC)(C)C#N)=O)CC2)C)cnc2ccnn2c1 C1(CC)CN(C(C2(N)CC(C)(C)C2)=O)CC(=O)N1 c1(CC)cnc(C(N2CCC(CC(F)(F)F)C2)C(=O)NCC2CC2)[nH]1 C(C1CCC(C)CC1)=C(C)C(=O)NC1CC2CC1CN2C(C12CC(F)(C1)C2)=O c1(OC)cncc(C=CC(=O)Nc2cccc(C)c2)c1.C1(CN)(CO)COC1 N1(C(c2cc(C(C)=O)no2)=O)CC(CNC(=O)CCC2CC2C)C(C(F)(F)F)C1 C(=O)(CC(c1ccccc1)c1ccccc1)N(CC1CC(=C)C1)CC CCCCC(CC)CC(=O)N1CCC2CCCC12C(=O)N(CCC(C)C)CCO c1(C(=O)NCC(CC(C)C)NC(c2c(CC)scn2)=O)cc(Cl)cc(F)c1N C(C)(C(C)(C)C(=O)N1CC(C#N)C1)NC(C1CC(C#C)(O)C1)=O C1(NC(=O)C(N2CCCC(CO)C2)=O)CC2(CCC2)C12CCC2 C(CCC(=O)N(CCCCCNC(=O)CC1CC(n2cnnc2)C1)C)SC N1(C(CCC=C=C)=O)CC(C2CCCN(C(=O)CC3CCCC(OC)C3)C2)C1 C1(NC(C(C)(C)C(N)=O)=O)CN(C(C2(O)CCOCC2)=O)CC2(CC2)C1 C#Cc1ccc(C(N2C(C(=O)NCc3cc(Br)no3)CCC2C)=O)c(Cl)c1 CC1(C(=O)NCCOC2CCN(C(c3ccnn3C(F)F)=O)CC2)COCCO1 N1(C(C(CC)n2ccnc2)=O)CCC(C(=O)NCc2nccnc2C)CC1(C)C c1(C(=O)NC2CC3CN(C(C(=O)NCCOC)=O)C2C3)cccc(C)c1NC CC1CN(C(=O)C(C)n2cccc2)CC1NC(C1(CCc2ccccc2)CC1)=O C=C1CC2(C1)CC(C(=O)NC1CC3CN(C(=O)C(C)CCC)CC13)C2 N1(C(c2c(C(F)(F)F)nn(C)c2Cl)=O)CCCC2(CCN2C(c2ccno2)=O)C1 C1(CN(C(=O)C(F)(F)c2cnn(C)c2)C)CCCN1C(C1CCCC1C(F)F)=O c1(O)cccc(CN)c1.c1(CNC(N(CCC)C2CC2)=O)ccc(C(C)C)cc1 O=S(=O)(c1cc(F)c(F)c(F)c1)N1CC2CN(Cc3cc(F)c(F)cc3Br)C2C1 C1(NC(CCOC(C)C)=O)CCC(N(C)C(c2nnn(C)c2C(F)F)=O)CC1 CCC(CC(=O)NCC1CCN1C(=O)CCCn1cccc1)C1CCC1 N1(C(C(=O)NCC)=O)CCN(CCN(C)C(c2occc2C2CC2)=O)CC1 c1(OC)cccc(NC(=O)C(N2CCC(CO)(OC)C2)c2ccsc2Cl)c1 c1(COC)ccccc1C(=O)NCC1CCCN(C(C2COC(O)=CO2)=O)C1 N1(C(Cc2cccc(COC)c2)=O)CC2(CCN(C(=O)C(C)(C)CSC)CC2)C1 c1(C(N2CCC(O)(CCNC(c3[nH]cc(CC)c3)=O)C2)=O)cnc2cc[nH]c2c1 C(=O)(CC(c1ccccc1)n1cccc1)NCCCN(C(c1cccs1)=O)CC C1(CNC(CCCC)=O)C2CCCC1N(C(C1CCC(CN(C)C)O1)=O)C2 c1(OC2C(C=C)OCC2)nc2ncccn2n1 c1(NC(=O)Cc2ccc(NC(c3ccccc3)=O)cc2)ncnc2scc(Br)c12 C(=O)(CCC(=O)N1CC(O)CC1C(=O)NCCCS(N)(=O)=O)NC C(=O)(CCCC(C)(C)NC(c1cc(C2CC2)on1)=O)NC(CC)C1CCC1 c1(C(=O)Nc2ccc(Cl)cc2)cn2c(n1)CN(Cc1ccc3nc[nH]c3c1)CC2 c1(C(N(CC(C)NC(c2cnc(CCC)s2)=O)C)=O)cn(CCN(C)C)nc1C c1(OC)ccc(Br)cc1C(N1CCC(CN(C(=O)C(F)C(F)(F)F)C)C1)=O C(=O)(CCC(=O)NN(C)C)NC1CC(NC(C=CC(C)(C)SC)=O)C1(C)C CC1(CNC(C2(CNC(c3nsnc3O)=O)CC3(CC3)C2)=O)CC(F)(F)C1 N1(C(CS(C(C)C)(=O)=O)=O)CCN2CCN(C(=O)Cn3cnnc3O)CC2C1 C1(C)(CC(=O)NCC(C)(C)NC(C2(N(C)C)CCCCC2)=O)CC1(Cl)Cl Cn1ncc2c(O)cc(C(N3CCN(C(=O)CC(C)(F)F)CC3C(F)F)=O)cc12 C1(CC(N2CCC(CNC(CC(COC)C)=O)CC2)=O)CCC2(CC1)COC2 C1(CNC(C2(C=C)CCC2)=O)CN(C(C2(CC(C)C)CCC2)=O)CC1C(F)F N1(C(Cn2nnc(C(C)C)n2)=O)CC(NC(C2CC=CC2)=O)CC2(CCC2)C1 C1(NS(CCCCC)(=O)=O)CC=C(c2ccc(F)cc2)CC1 c1(CC(N2C(C)CCC(NC(C3OCCCO3)=O)C2)=O)noc2cc(F)ccc12 N1(C(CC(=O)OC)=O)CC2(C1)CN(C(=O)Cc1ccccc1)CC2CO c1(C(CC)C(=O)N2CC(C)(c3cn(C4CCOCC4)nn3)C2)ccc(F)cc1 C1(C(N(CC(CCC)O)C)=O)CCC(C)(C)N(C(c2ccc(CO)o2)=O)C1 C(=O)(CC(O)CCSC)N(CC(C)(C)NC(C1N(CCCC)CCCC1)=O)C c1(C(=O)NCc2ncsc2C(=O)NCC(CC)OCC)cc(S(N)(=O)=O)n(C)c1 C1(NC(C2CCC(C)(C)OC2)=O)CCC2CCN(C(=O)C=Cc3cocn3)C1C2 c1(C(=O)NC(CNC(Cn2nc(C)c(Cl)c2)=O)CO)cc2c([nH]1)CCC(C)C2 N1(C(C2C(C)=C2)=O)CCC(C2CC2)C1CNC(=O)C1=CCCOCC1 N1(C(CC2(OC)CC2)=O)CC2(C)CN(C(c3cc4c([nH]3)CCCC4)=O)CC2(C)C1 CCCC(CCCNC(=O)CCC1CCOC1)NC(=O)C(C)(C)C1CCCC1 c1(C(C(=O)NCC)NC(=O)C(C)(CC)OC)c(C)cccc1Br.C=CC(O)COC C1(C(=O)NCCOC2CC2)CCCN(C(C2C=CCS2)=O)C1 C12(CNC(c3nnc4ccccn34)=O)CN(C(C3CC(CF)C3)=O)CC1CCO2 CC1CCC(C(=O)NC(c2ccno2)C)N1C(c1c(Br)cnn1C)=O C(=O)(CCS(C)=O)N(CC(C)(C)CNC(c1csc(C2CCCO2)n1)=O)C CC1CCCCC1CC(=O)N(CCCCN(C(=O)C=Cc1ccc(Cl)s1)C)C C1(CCNC(c2ccc(C)nn2)=O)CN(C(c2c(C)csc2C)=O)CC(C)O1 N1(C(c2cn(CC)nn2)=O)CCC(C)C1CNC(c1cc(C)sc1C)=O N1(C(C(C(CCC)NC(c2cc(O)n(C)n2)=O)O)=O)C2CCC1CC1(C2)N=N1 c1(C(=O)NCC(N2CCN(C(CCC(C)OC)=O)CC2)C)cncc2sccc12 c1(OCC)ccc(-c2nnc(CN3CCCC(CNS(=O)(=O)CC)C3)o2)cc1 Cc1noc(C)c1CC(C)C(=O)NCC1CC(F)CN1C(C1CCCC(O)C1)=O c1(C(N(C)C)=O)[nH]c2ccccc2c1CC(N)=O.C1C(CO)C(=O)C=CC(=O)N1 N1(C(CCC=C)=O)CCCCC(C2CN(C(c3cncc4nc[nH]c34)=O)C2)C1 C12(C(N3CC(C)S(=O)CC3)=O)CCN(C(=O)C(C)NC=O)CCC1C2 c1(C(=O)NCCCN(C)C(c2cc(C(F)F)no2)=O)ncc(Br)cc1F c1(CC(=O)NCC2CCCN(C(C3CC3(F)F)=O)C2)ccc2c(c1)CCCC2 C1(COC(C(C)OC2CN(C)C23CCCCC3)=O)CC2COCC(C1)C2(F)F C=C1CC(C(F)(F)F)(C(=O)NCCN(C)C(c2cscc2CC)=O)C1 C1(C)(C(=O)NCC(CC=C)NC(C)=O)CCCN1C(c1sc(CCC)nc1C)=O C1(C(=O)NCC2N(C(C(CSC)C)=O)CC2)(NC(N)=O)CCCCC1 N1(C(Cc2cccc(OC)c2)=O)CCCCC(N=c2[nH]nc(C(N)=O)s2)C1 c1(N2C(C(CNC(C(C(C)C)N(C)C)=O)(C)C)CCC2)nccc(C#N)n1 N1(C(c2cnc(SC)s2)=O)CCC2(CC1)CC(NC(=O)CCCC1(C)CC1)C2 C(=O)(CCCC(C)(C)CC)N(C1CN(C(c2cc(CCC)oc2C)=O)C1)C N1(C(c2c(C)noc2)=O)CCC2(CCC(CNC(=O)C(O)C(F)(F)F)OC2)CC1 CCCCC(CC)C(=O)N1CC(NC(=O)C(C)(C)C(=O)NC)CC(C)(C)C1 C1(C(=O)NC(C2CC2C(=O)NC2CCCC(SCCF)C2)C)CN(C)CC1(F)F N1(NS(CCCC)(=O)=O)CCCC2C1CCN2C(c1cnc(Br)s1)=O C=CC(C)(CC)C(=O)NC1CCC1NC(c1c[nH]c(-c2ccccc2)c1)=O C1(C(=O)NCC(n2cccn2)C)CN(C(=O)C=Cc2ccncc2)C(C)(C)C1 C(N=c1nc(N2CCC(CCN(C)C)C2)c2[nH]ccc2[nH]1)C1CCCN(CC)C1 CCC(C)CC(C)N(C(=O)CCCNC(=O)CSCCC#N)C C1(NC(C=CCCC=C(C)C)=O)CCCC(NC(=O)C(C)(C)c2ccccc2)C1 N1(C(C2CCCN(CCC)C2)=O)CC2CC(NC(C3CC(O)C3)=O)C(C2)C1 Nc1c(C(=O)NC2CC2NC(c2ccc(Cl)cc2)=O)cnn1-c1ccc(F)cc1 N1(C(C2C(NC(C=Cc3n(C)ncc3)=O)CCO2)=O)CCC(O)C(C)(C)C1 N1(C(c2c(C)cc[nH]2)=O)CC(NC(=O)CCN2CCC(C)CC2)CC1C c1(N(C)C)nc2ccsc2c(=NCCSCc2cn3c(n2)SCC3)[nH]1 N1(C(C(CC#C)O)=O)CCOCC(CNC(C2CC3(CCCO3)C2)=O)C1 N1(C(CCNC)=O)CC(OC)CC(C(=O)Nc2nc(=O)n(C)cn2)C1 c1(OC)cc(C(=O)NCCN(C(=O)C(C)CC2CCCO2)C)sc1Br c1(SCC(N2CC(O)(CN)C2)=O)ccc(OC)c(OC)c1.C(CC(=O)OC=C)=CC=C N1(C(CN2C(=O)NCC2)=O)CCC12CCN(C(c1cc(I)c[nH]1)=O)CC2 c1(CNC(=O)OC(C)(C)C)nnc(SC23CC(c4ccccc4)(C2)C3)s1 C1(CCC)CN(C(=O)Cc2ccc(C)cc2)CCN1C(c1cc(CC)no1)=O c1(CC(N2CCC(NC(c3ccc(C(N)=O)[nH]3)=O)C2)=O)cc(O)nc(O)n1 c1(CC(=O)NCC2CCN(C(=O)CCN3C(=O)C=CC3=O)C2)ccc(F)cn1 N1(C(c2c(CC)nc(=N)[nH]c2)=O)CCCN(C(=O)C(O)C2CCC2)C(C)C1 C1(CN(C)C(C2CCC2C)=O)CCCN1C(=O)C(F)=CC1CC1 N1(C(C(CCC)O)=O)CCC2(CCC(NC(=O)CCC3CCC3)C2)C1 CC(CC(C)NC(c1cocn1)=O)NC(=O)C(F)(F)c1csc(=N)[nH]1 C1(C(=O)Nc2c(CC)nsc2)C(C)CCN1C(=O)CN1CCC(OC)C1 C1(C2N(C(C=CCOC)=O)CCC2)CN(C(=O)CCOC2CCCCC2)CCO1 N1(C(C=CC=CCC)=O)CCCC(C(C)C(N2CCCC2CF)=O)C1 c1(CC(=O)N(C2CC(C#N)C2)CC(=O)NCC(n2ccnn2)C)nncn1C Cn1ccc(C(=O)NC2(C(=O)NCCCS(N)(=O)=O)CCCC2)cc1=O C(CCN=c1[nH]c(=NCc2ccsc2)[nH]c2c1SCC2)c1ncn(C)n1 C12(C(=O)NCC3(C(=O)OC)CC3)CCC(CC1)N(C(C13CCCCC1C3)=O)C2 c1(SC)ccnc(N2CC(C)(NC(=O)C(c3ccccc3)N(C)C)C2)n1 C1(C(=O)NCCOCC(N)=O)CCN(C(=O)CCC2CC2)C12CCC2 C(=O)(C1Cc2ccccc21)NC(C)(C)CC(F)C(=O)NC1CCc2n[nH]cc2C1 CC1CC(CC(=O)NCC(C)NC(C2(CNC(N)=O)CCCCC2)=O)C(C)O1 Cc1ccc(C)c(S(=O)(=O)N(c2cc[nH]c(=NCC3CCCC4(CC4)C3)n2)C)c1 c1(C(=O)NC23C(CN(C(c4ccc(C(C)=O)cc4)=O)C2)C3)ccnc2[nH]ncc12 Cc1ccc(C)c(C(=O)NCC(O)CNC(c2cccc(F)c2C(C)C)=O)c1N N1(C(=O)COCC2CCCO2)CC2=C(C1)CN(C(C1CC13CCSCC3)=O)C2 C(=O)(C1=CC2CCCCCC12)N1CC2CC(NC(=O)CCc3cncnc3)C2C1 N1(C(c2c(C)n(C)nc2)C(=O)NCC2CCCO2)CCC2CCCC12 c1(C(=O)NCCCCNC(C2C(C(=O)OC)C2)=O)ncccc1C(F)F N1(C(CCn2c(C)csc2=O)=O)CCC2CCN(C(=O)Cc3ccsc3)CC2C1 Cc1n[nH]c(C)c1C(=O)NCc1cn(C2CCN(C(=O)C3=CCC3)CC2)nn1 C=CC(C)(CCOC)C(=O)N1CCCC(O)(CCNC(=O)CN2CCSCC2)C1 C1(C(N)=O)(CO)CN(C(C2CCC(NC(=O)C(F)(F)C3CC3)C2)=O)C1 C1(C(N(CCC(=O)NCC2CCCC2O)C)=O)CSCC(=O)N1 C1(CNC(CC2CCN(C)CC2)=O)CCC2CN(C(=O)CNC(N)=O)CC12 CCC(CO)(C(=O)NC1C=CC(C(=O)NCc2ccccc2OC)C1)OC c1(CC(=O)NCCNC(c2[nH]n(C)c(=O)n2)=O)ccn2cncc2c1 N1(C(C2=C(C)CCC2)=O)CC2OCCN(C(c3cc(F)cc(F)c3N)=O)C2C1 CC(C)CC(C(=O)NCc1cc(F)cc(F)c1)N(C(=O)CC(C)N(C)C)C C(=O)(C(C)(C)CN(C)C)NC(CNC(C(C)OCCC=C)=O)CC C1(NC(c2ccc[nH]2)=O)CCN(C(=O)Cc2cnns2)C12CCC2 Cc1ccc(F)c(C(=O)NC(CN=[N+]=[N-])C(=O)NCC2(N(C)C)CC2)n1 C=CCCCCCC(=O)NC1CC(O)CN(C(=O)CCCCCNC(C)=O)C1 C1(C(N(CCNC(C)=O)C)=O)CCCN(C(c2cn(C)nc2C)=O)C1 C1(NC(=O)CSC(F)(F)F)CN(C(C2CC3C=CC2CC3)=O)C2CCCCC12 c1(C(=O)NCCCCCN(C(C(CC=C)C)=O)C)ccc2c(c1)NC(=O)CCC2 C1(CNC(C=CC=CCC)=O)C(C2CC2)CCN1C(c1nccn1CC)=O N1(C(C=CCOC(C)C)=O)CCOC2(CCN(C(=O)CSC3CC3)CC2)C1 c1(C(N2CCCCC(NC(c3cnc[nH]3)=O)C2)=O)coc2c1CCCC2 N1(C(C(=O)NC(C)C)=O)CCN(C(=O)CCc2ccoc2)CCC1C N1(C(c2ccc(O)cc2)=O)C(C(N2CCCC2c2ccc(F)cc2)=O)C2(CC2)C1 C#CC1CCC(C(N2CCCN(C(C3COCCN3C)=O)CC2)=O)CC1 CC(C)S(=O)(=O)CC(=O)NCC1COCC1NC(=O)Cn1ncc2ccccc12 C(=O)(C1CCCc2ncnn21)N1CC(CNC(=O)Cc2ccc(F)cc2)C(O)C1 c1(C(N2CC3C(NC(C(CC(C)C)N(C)C)=O)(C3)C2)=O)cc2n(n1)CCCC2=O C1(C)(CC(=O)NCC(=O)OCCCC)CCCN1C(c1c[nH]nc1CCC)=O CN1CCCC(CCC(=O)N(C2C3CN(C(C4(F)CCC4)=O)CC23)C)C1 C=C(C)CCCC(=O)NC1CCC12CN(C(c1ccc(Cl)cc1C(F)(F)F)=O)C2 C#CCCCCCCCNC(=O)C1=CCCN(C(C2(C#N)CCOC2)=O)C1 N1(C(CNC(N)=O)=O)CC2(CCC2)CC1CNC(=O)Cc1ccc(F)cc1 C1(CNC(c2c(C)scn2)=O)CN(C(=O)CCC(C)C#N)C(C)(C)C1 CC1(NC(c2cn(CCO)nn2)=O)CCN(C(C2(C)CNC(=O)C2)=O)CC1 N1(C(C(CC)OC)=O)CCN(C(=O)CN(C)C(=O)OC(C)(C)C)CC(CO)C1 N1(CC(C)C)CCN(C(=O)CC(N)c2ccccc2)CC1.N12CC(C1)C2=O c1(OC)ccc2c(c1)CCCC2CNC(=O)NC1COc2ccccc2C1 CCC(CC(C)C)C(=O)NCC=CCNC(c1cnc2snnc2c1)=O C1(NC(C2CC(N(C)C)C2)=O)CC2CC1N(C(=O)Cc1ccc(C3CC3)cc1)C2 c1(C(N2CCC3CC3C2)C(=O)OC)ccccc1Cl O=C(CCC(=O)N1CC2CC2C(F)(F)C1)CCC(=O)c1ccccc1 O=C1CC(C(=O)NC2CN(C(C3CC(C(F)(F)F)C3)=O)C2)Oc2ccccc21 c1(OC)nc(C(=O)NC2CCCN(C(C3CC(SC)C3)=O)C2)sc1C C(C(C)CC(=O)NC(C)C(C)C(=O)NC1CC(CCOC)C1)OC N1(C(CNC(CC(C)C)=O)=O)CCCC(C)(C(=O)Nc2ccon2)C1 C1(C(N2C(C(=O)NCCc3ncccn3)CC(OC)C2)=O)CCC(O)CN1C N1(C(C)=O)CC2CC1CN2N1CCCC1CC(=O)N.c1(C=O)c(C)coc1C C(CC(CC)C(=O)NC1CC2(C1)CC2NC(=O)CCc1cncn1C)=CC Cc1c(C(=O)NC2(CO)CN(C(=O)C(C)(O)C3CCC3)C2)ccc2cncn12 c1(C2C(C(=O)NC(C3CCOC3)CNC(c3n[nH]cc3Br)=O)C2)ccccc1 C1(CCC)CN(C(=O)C=CC(C)NC(=O)CC2CC2(C)C)C1 N#Cc1cccc(NC(=O)CNCc2ccccc2Br)c1 Cc1cc(C(=O)NCC(c2ccc(F)cc2)NC(=O)CC(C)(F)F)cn1C C(=O)(CCCC(C)(C)NC(=O)CCc1cccn1C)N(C)Cc1onc(CC)n1 c1(C(N2C(C)CN(C(COCCOCC)=O)CC2C)=O)cncc(S(C)(=O)=O)c1 C1(N(C)C(C)=O)C2CN(C(=O)CCC(=O)NC(Cc3cscn3)C3CC3)CC12 C1(COC)(CNC(C2CCCC2C)=O)CCN(C(C2CC(C)CCO2)=O)C1 C1(C(=O)NC2CN(CCC)C2)CC(C)CCN1C(c1nnn(C)c1C)=O N1(C(c2ccc(C)n(C)c2=O)=O)C2COCC1CC(NC(C1CCCO1)=O)C2 c1(C(N(CCC)CCNC(=O)C(C(C)C)OC)=O)cc(CC)cc(N)c1 c1(CN2CC(C(=O)Nc3ccc(SC)cc3)OCC2)c(Cl)cnc(Cl)c1Cl C(=O)(CC1CCOc2ccccc21)NCCC1CCCN(CCCOCC)C1 c1(CC(=O)NCCNC(C2(OC)CCCC2)=O)ccc2c(c1)CCCC2 C1(CCN=c2ncc(C#C)c[nH]2)NC(=S)N(CCCC)C2=C1C(=O)OC2 C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)NC1CCN(C(C(CCC)N(C)C)=O)C1 C1(C)(NC(CC(=O)OC)=O)CCCCC1C(=O)NCc1cnccc1Cl C1(C(=O)NC2CCN(C(=O)CC3CSCCS3)C23CC3)C2CC3CC(C2)CC1C3 N1(C(c2c(C)nco2)=O)CC(CNC(=O)CN2CCCNC2=O)CC12CCC2 C(C(C)(C)C(=O)NC1CC1CNC(c1cc(C(C)C)oc1C)=O)NC(C)=O c1(CC(=O)NC(CN(C(CCSCCCC)=O)CC)C)ccc(SCC)cc1 N1(C(c2c(-c3c(C)nc(F)cc3)nccn2)=O)CCN2CCNC(=O)C2C1 c1(C(=O)OC)cn(CC(N2CCCC2CCCNC(c2sccc2F)=O)=O)nn1 C1(CC(N2CCC(CC(F)F)C2)=O)CCCCN1C(=O)C=C1CCC1 C1(C(=O)NC(CN(C(=O)C(n2nc(C)cc2C)C)CC)C)CC2(C1)CC(C)(C)C2 C#Cc1ccc(C(=O)N(C2CCN(C(C3CC34CCCOC4)=O)CC2)C)cc1C C(=O)(C1=C(Cl)CCOC1)NCCCCC(=O)N(C1CCN(C)C1)CCO c1(C(=O)NCC(CC)NC(=O)Cc2cc(C)ccc2C)c2c(c[nH]c1=N)CCC2 CC1(C)CCOC(C(=O)NC2(C)CC(C(=O)NCC3CCC=CCC3)C2)C1 C1(S(C)(=O)=O)(C(=O)NCC(CNC(C(CCC)C#N)=O)(C)C)CCOCC1 c1(NC(=O)C(=O)NC2CC2)ccc(=NCCC(F)(F)C2CCNC2)[nH]n1 c1(CCC(=O)NC(COC)CC(=O)O)c(C)nc2ncnn2c1C N1(C(C)C)CCCCC1C(N1CCC(C(C)(C)NC(=O)Cc2nnc(O)s2)C1)=O c1(C(=O)NCC(CO)NC(=O)Cc2cc(-c3ccccc3)on2)ccncc1O N1(C(C(CC=C)N(C)C)=O)CC2CCC1C(NC(c1ccnn1COC)=O)C2 c1(NC(=O)NC(C)Cn2cccn2)ccc(Cl)cc1N(C)C N1(C(c2ncc(N)nc2)=O)CCC(F)(CNC(C2Cc3nccn3C2)=O)CC1 c1(CNC(c2cnc(C)[nH]2)=O)cccc(NC(c2nscc2C)=O)c1 CCC(=O)C(=O)N1CCC(CNC(=O)CCc2nc[nH]n2)C1 C(=O)(C1=NOCC1)N(CC(O)CN(C)C(c1c[nH]nc1C1CCOC1)=O)C CC1(C)CCOC1C(=O)NCC1(C)CCN(C(C2(NC(N)=O)CC2)=O)C1 C1(C(N(CCNC(CCCN(C(C)=O)C)=O)C)=O)CCCCN1C(C)C C1(C)(C(=O)NC(CSCC)C(=O)N(C(C)CC(C)C)C)CCCCCC1 C(=O)(C(CCCC)NC(=O)C(CC)CCOC)NCC(=O)OCCCC c1(SCC2(F)CC(NC(C=CC(C)NC(c3ncn(C)n3)=O)=O)C2)ccccc1 C1(O)(CCN(C)C2CC2)CCCN(C(=O)CSCCO)C1 N1(C(c2c(CSCC)cccc2)=O)CCCC(C)(NC(=O)C(C)n2cccn2)C1 c1(C(N2CCCC(O)(CN(C(=O)CCS(C)=O)C)C2)=O)cc2ccnc(Cl)c2s1 c1(CNC(c2n(CCCOC)nnn2)CC2C=CCC2)ccc(Br)cc1F N1(C(COCC(C)C)=O)CCN(C(C2CN3CCC2CC3)=O)CC(C)(C)C1 c1(NC2CCN(C(=O)NC(COC)C)CC2)nccc(N2CCCC2)n1 N1(C(C=C(C)Cl)=O)CCC2CC(NC(C3SC4C=CC3CC4)=O)CCC2C1 c1(SC)ccc(CN2CCC(NC(c3cc(C)no3)=O)C2)cc1 C1(C(=O)N)CCC2(CCOCC2)CN1.Cn1nc(C(=O)OC)c2cc(Br)ccc12 c1(CC(=O)N(C2CN(C(=O)COC3CCOC3)C2)CC=C(C)C)ccccc1 n1(CC)c(NC(=O)C(N2CCC(NC(C)=O)C2)=O)nc2c1CCOC2 c1(OC)nccnc1C(N1CCC(C(=O)Oc2cnc(Br)cn2)C1)=O C1(NC(=O)C(Cl)=CCl)CCCC12CCN(C(c1cnc3ccncc3c1)=O)CC2 N1(C(CCC(C)SC)=O)CCOC(C(=O)NCCC2(O)CCOC2)CC1 c1(OC)c(C(=O)O)nc2n1CCN(C(=O)CN1CC(=O)N(C)C1=O)C2 C(=O)(C(CCSC)OC)NC(CC)CNC(c1occc1C)=O c1(CNCC(C2C(C)CCCN2C(=O)OC(C)(C)C)C)ccc2ccnn2c1 c1(CC(O)CNC2CCN(c3nnnn3C3CC3)CC2)ccc2c(=O)[nH]ccc2c1 Cc1oc(CNS(C)(=O)=O)cc1C(=O)OC(=O)C(C)O.C12CC(F)(C1)CCNC2=O C1(CC#C)(C(=O)N(CCC(=O)N(C(C)CC)CC)C)CCCN1C(C)=O N1(C(C(=O)NCCSC)C2CC2C(F)F)CC(C(N)=O)S(=O)(=O)C(C)(C)C1 C1(CS(N2CCCC(O)(C3CC3)C2)(=O)=O)CCC2(CCOCC2)CO1 C(=O)(C(C(C)C)N(C)C)N1C(C2(NC(c3c(C)[nH]cc3)=O)CC2)CCC1 Cc1cc(Br)ccc1CCC(=O)NC(C)CN(C)C(c1cccc(Cl)c1N)=O CC1CN(C(=O)CCc2nccn2C)C(C)CN1C(=O)CSCc1ncc[nH]1 CC(C)C1C(=O)N2CCCC2C2C(C2)C(=O)N1.c1(OCCN)ccccc1 C1(CC(=O)NCCOCCNC(=O)C=CC2CC2)COC2CC1C2 C(C)(C)(CC(=O)N1CC(=O)CC1C(=O)NC1CC12CCCC2)OC O(NC(=O)C(C)C(F)(F)F)C(CC(C)C)C(=O)NC(C)(CO)CO CCC(CCC(=O)N(C(CC)C(=O)NC(C1CC1)CC)CC)OC.c1(C)ncc(C)nc1C CN1CCN(C(c2cnn(-c3ccccc3)n2)=O)CC1CNC(C1CC1(C)C)=O C1(C)(C(=O)NCC2C(CNC(CNS(NC)(=O)=O)=O)C2)CC2(CC2)C1 c1(C(=O)NC(CCOC)CNC(=O)C(C)CC2CCCC2)cccc(C)c1F c1(C(=O)NC(C(C)NC(Cn2ccc(C)n2)=O)C)cnc(C(F)(F)F)cc1O c1(C(N(CC(C)CNC(C2CC2[N+](=O)[O-])=O)C)=O)ccncc1Cl C1(C(=O)NC2CCC(NC(C(C=C)(C)O)=O)CC2)CCC2(CC1)NC(=O)NC2=O C1(C(=O)NC2C(SC)CN(C(C3CCC(OC)CC3)=O)C2)CCc2c[nH]nc2C1 c1(C(=O)NCC2(CCNC(CC(C)SC)=O)CC2)occ2c1CCC2 C(=O)(C1=CCCSC1)NC(CCNC(c1c(C)nc(COC)s1)=O)(C)C C(CCC1CCC1)(C(=O)NCCCc1ccccn1)NC(Cc1n(C)nnn1)=O C(=O)(CC(C)C(=O)N1CCN(CCN(C(=O)C(C)(Cl)Cl)C)CC1)OC CCCC(C(=O)NC(C)C=CC(=O)NCc1coc(C)c1)N(C)C c1(C(=O)NC2(CSC)c3nnnn32)cccc(CS(C)(=O)=O)c1.C1(N)CC1.C1CC1 CC(C)(C)C(=O)N(C1CCCCC1)CCN(C(=O)C=Cc1ncco1)CCO c1(C(=O)NC(CC)CN(C(=O)C(O)C2CC2)CC)cccc2nc(O)ccc12 c1(N(CC(COC)(F)F)C)nc(=NC(C)c2ncccn2)[nH]c2c(C)nn(C)c12 C(=O)(C(F)C(F)(F)C(F)(F)F)NCC(CNC(c1c(C)nc(C2CC2)o1)=O)C C(=O)(CCC(=O)N1CCNCC1)NCCSC.C1(C=O)C2CC3C(C2)C13 c1(CN2CC(C)(CC(=O)N(C)CC#N)C2)nnc(C(C)(C)C#N)o1 c1(C(=O)NC(C(C)NC(c2cn(C)cn2)=O)C)cc2ccccc2c(O)n1 c1(C(=O)NCCC(C)NC(=O)Cc2csc(C3CC3)n2)cncc2c1CCC2 c1(CN2CCC(C(=O)NC(c3cccc(C(C)(C)C)n3)C)C2)ncccc1Br c1(CC2(C(=O)NCCC(C)N(C(C3N(CCCC)CC3)=O)C)CC2)ccccc1 N1(C(c2c(C)cc[nH]2)=O)CCN(C(C2CCc3nn[nH]c3C2)=O)C2(CC2)C1 C1(C(N(C2CCCC(C)(C)C2)C)=O)CC2CN(C(=O)CC3CCC(C)(C)O3)CC2C1 C#CCC(C)(C)C(=O)NCC1(CNC(=O)CC2CCCC(C(F)(F)F)C2)CC1 C(=O)(C(C(C)O)N(C)C)NC(CNC(CC1CC(CC)C1)=O)CO Cc1c(F)ccc(C(N2CC(CNC(=O)CCCn3cccn3)C(C)C2)=O)c1N C1(CCCNC(c2cncc(O)c2)=O)CN(C(c2cnccn2)=O)CCO1 c1(NCC(=O)NC2CC(NC(C3(C)C(C(=O)OC)C3)=O)C2)ccc([N+](=O)[O-])o1 C(N=c1[nH]c2c(c(=NCC3CC(N(C)C)C3)[nH]1)SCC2)c1[nH]nc(NC)n1 C1(N(C(=O)CC2(O)CCC2)C)CN(C(c2[nH]ccc2C2CC2)=O)CC1(C)C N1(C(C=C(COC)C)=O)CCC(C(C)CNC(=O)COC2CCC2)CC1 C=CC1OCCCC1C(=O)NC1CCC1NC(=O)Cc1cnccc1C c1(C(C)C)nc2[nH]ccc2c(=NCCCn2cnnc2C)[nH]1 c1(OCC(=O)N(C(C)C)CCC)ccc(C(C)(C)C)cc1OCC(F)F S(=O)(=O)(c1ccc(C(=O)OC)o1)COCC=C.N12CCC(C1)NC(=O)C2C C1(C(=O)NCc2ncc(C)o2)CCC2(CCN(C(c3ccsc3C)=O)CC2)C1 C1(CCNC(C(C)=CC)=O)CCCN(C(=O)C(C(C)C)SC)C1 N1(C(c2n(CC#C)ccc2)=O)CC2(CCN(C(=O)CC(O)C3CCCC3)CC2)C1 CCC(CCC(=O)Nc1cccc(Cl)c1O)NC(C1CC1C1(C)COC1)=O N1(C(Cc2nc(=N)[nH][nH]2)=O)CCOC(C(N2CCCC(C(F)F)C2)=O)C1 c1(OC)cccc(CC2C3CN(C(=O)C(N4CCSCC4)C)CC23)n1 Cc1nccnc1C(=O)NC1C=CCN(C(=O)C(n2ccc(Br)n2)C)C1 C1(C(=O)Nc2cnn(C)c2)(COC)C=CCN1C(C1C=CCCC1)=O c1(CNC(C23CC(NC(c4nc(CC)sc4)=O)(C2)C3)=O)ccc(C(=O)O)cn1 c1(C(N2CCC(CNC(C(n3ccc(C(F)F)n3)C)=O)C2)=O)cnnc(O)c1 c1(OC)ncnc(C)c1C(=O)N(CCCCN(C(=O)CN1CCS(=O)CC1)C)C c1(CC)nc(=N)[nH]cc1C(=O)NCCN(C)C(c1ccncc1Br)=O O=C(C1=CNC2=NCCC2=C1)N1CCC1CNC(c1cn2cc(Cl)cnc2n1)=O N1(C(C(C)=CC)=O)CC(C(C)(C)C)CC(CNC(=O)C(c2cnn(C)c2)C)C1 N1(C(C2(COC)CC=CC2)=O)CC(N(C(=O)CCC(F)F)C)C2(CC2)C1 C1(C(N(CCCC(=O)NC(c2c(C)ccnc2)C)C)=O)CCCC(C#N)C1 C(C(C)(C)C(C)(F)F)NC(c1ccc(CNC(c2c(C)cccc2)=O)cn1)=O c1(OC)c(C(=O)NC(CNC(=O)C(C)c2ccco2)CC(C)C)csc1Cl c1(SCC(=O)NCC(CN(C(c2c(CC)ocn2)=O)C)C)ccc([N+](=O)[O-])cc1 C1(N(C(Cc2c(C)con2)=O)C)CCC(NC(=O)Cn2cc(Cl)cn2)CC1 c1(CCC(=O)NC(C2N(C(C=CC)=O)CCCC2)C)ccc2c(c1)OCCCO2 c1(OC)cc(OCCc2ncccc2SC)ccc1[N+](=O)[O-] C(=O)(C(C)(C)C(N)=O)NCC1(OC)CCN(C(CC(COC)C)=O)C1 c1(C(N2CC(N(C)C)CC(C)(C)C2)C(=O)NCCSC)cc2c(nn1)CCCC2 c1(C(=O)NCC(N(C(c2[nH]cc(C)c2)=O)C)C2CC2)c(S(N)(=O)=O)cnn1C N1(C(C2(OCC)CCCC2)=O)CCC(NC(=O)C#CC2CCC2)CC1C1CC1 c1(C(=O)OC)ccc(O)c(C(=O)N(CCCNC(=O)C(F)C2CCC2)C2CC2)c1 c1(C(=O)NC2CN(C(CCC#C)=O)C(CC)(CC)C2)ccc2c(=O)ccoc2c1 C#CC(C(C)(C)C)NC(=O)C=CC(C)NC(C1CC(=O)CCO1)=O C1(NC(c2ccc([N+](=O)[O-])cn2)=O)CC2CC(C1)CN(C(c1nocc1Cl)=O)C2 C1(NC(=O)Cc2ccc(Cl)cc2)CC(F)CN(Cc2cc([N+](=O)[O-])c[nH]2)C1 N1(C(CCSC)C)CCC1.C1(C=O)(CO)CCSCC1 N1(C(C(C)Oc2ccccc2F)=O)CCCCCC1CNC(C1CC(C)C1)=O N1(C(CCCC)=O)CCCCC(NC(C2CC(CCC)C2)=O)C1 C1(C2CC2)(C(=O)NCCCCCCNC(=O)Cc2cnc[nH]2)CC=CC1 N1(C(C(C)SC)=O)CC(NC(C2CNC(=O)N2)=O)CC12CCCCCC2 c1(C(N2C(CN(C(C(C)(CO)OC)=O)C)CCCC2)=O)ccc(C)cc1SC c1(CCC(=O)NCC2CCC(NC(=O)CC3CCCO3)CC2)cncc(Br)c1 C1(NC(c2ccn(CCNC(C3CCC(N(C)C)C3)=O)c2)=O)CCCC(O)C1 C1(NC(c2c(OC)ccnc2)=O)(CNC(C2CCOC2=O)=O)CC2CCC1CC2 N1(C(=O)NC(c2nc(CC)on2)C)CC2CC(C1)CS(=O)(=O)C2 C12(CNC(c3nc(CC)oc3)=O)CN(C(C3CCOC3C)=O)CC1CCO2 N1(C(C(C(C)C)(C)O)=O)CCCC(C2CCN(C(=O)CN3CCC(C)C3)CC2)C1 c1(NC(=O)NCC2N(C(C3(c4cccc(C)c4)CC3)=O)CC2)cc(C)ncc1C C=CCC(C)C(=O)NC1CN(C(=O)C(C)(C)Cc2cccc(Cl)c2)C1 C12(O)CCN(C1)C(=O)C1(CC1)C(=O)N(C)C2.C1(N)C=CCS1.C1CC1 C1(CN(C(=O)CS(=O)(=O)NC)CC)CCCN(C(C2(C3CCCCO3)CC2)=O)C1 C(c1ccco1)=C(C)C(=O)N(CCO)CC1COC(CN=[N+]=[N-])C1 O=S(=O)(NC1CCCOC1)N1CCCC1.C1(C)CNC1 c12nccc(c1C)NC(=O)C1CC1S2.CCC(CC)NC(N1CCCC1)=O c1(CC(N2CCC(N(C(CCC=C=C)=O)CCO)C2)=O)c(C)cc(C)nc1O Cc1ccc(Cl)c(F)c1C(N1CCCCC(NC(=O)COc2cn[nH]c2)C1)=O Cc1ccc(C(=O)NC(C)CCN(C)C(C2SCCCS2)=O)n1C c1(C(N2CC3C(N(C(C4C(OCC)C4)=O)C)C3C2)=O)c(OC)cc(OC)cc1N C1(OC)CCC(N(C(=O)C(C2CCC2)NC(=O)Cc2ncccc2F)C)CC1 N(C1CCCn2nccc21)C(C1=CCCN(C(C(COC)(C)OC)=O)C1)=O C1(C(NC(C)C2CC2)=O)CN(C)CCN1C(=O)CCCC1CCC1.N1CCOCC1 CC1CCc2nc(C(N3CCC(CCNC(=O)CC(C)(C)F)CC3)=O)cn2C1 C(=O)(CC(F)(F)CC(=O)OC)NC1CC(CNC(C(CC)(C)CC)=O)C1 N(C1CCc2c1ccc(Br)c2F)C(=O)Nc1ccc(C(=O)OCC)cc1 C1(NC(C2CC=CC(NC(c3c(OC)nn(C)c3)=O)C2)=O)CC(C)CCC1O C#CCCCC(=O)N1CC(C(C)NC(c2ccc(NS(=O)(=O)CC)cc2)=O)C1 c1(CC)cc(C2CC2)n(NS(=O)(=O)NC2(COC)COC2)n1 c1(C(=O)NCC2N(C(C(C(C)C)NC(C)=O)=O)CC2)nnc(O)c(Br)c1O C(=O)(C1CCCc2c[nH]nc21)NC(CN(C(c1c(F)cc(CC)cc1F)=O)C)C c1(CC(N2CC(C(C)NC(C3CCNC(=O)C3)=O)C2)=O)ccc2c(c1)CCCS2 C(=O)(C1=CCc2ccccc21)N1C(CNC(CC2(C)CCCC2)=O)C=CC1 C(N=c1nc2c(cnn2C)c(NC(c2ccc(C)nc2)CC)[nH]1)C1(CCC)CC1 CS(=O)C1CN(C(=O)CCCC2CN(C3COC3C3C4CCCC34)C2)C1 c1(C(=O)NCCC(CCNC(C(CC(C)C)O)=O)C)cc(S(N)(=O)=O)co1 C12(C(N(CCC)C)=O)CC(C)(CN1C(=O)C(C)(C)CC1CC1)C2 C(C(=O)NCC1CN(C(C2(O)CCC2)=O)CC1C(F)(F)F)(C(C)C)NC(C)=O Cc1cc(S(N)(=O)=O)cc(Br)c1OC(F)(F)F.c12cccc(c1)OCCN(C)C2 N1(C(C(COCC)(C)C)=O)CCC(NC(=O)Cc2nn(C)cc2Cl)C(C)C1 C1(NC(C2(CC#C)CCCC2)=O)CN(C(C2(C)C=CCC2)=O)CCC1CO C1(NC(CCc2c(OC)cccc2)=O)CCOC2(CCN(C(=O)C(C)C)CC2)C1 NC(=O)CCCC(=O)N1CCC(F)C(NC(=O)C=Cc2cccc(CO)c2)C1 CCCCC(O)C(=O)N1CC(=C(F)CNC(c2cccn2Cc2ccccn2)=O)C1 C1(NC(CCC(C)OC)=O)CCCC2CN(C(c3cnn(C(C)C)n3)=O)CC12 CC(C)(C#N)CCNC(=O)NC1CC1c1ccc(OC(F)F)nc1 C1(C(F)(F)F)(NC(=O)NCc2cc(Cl)ccc2CO)CCCCCC1 C1(C(N2CC3CC2CN3Cc2cc(F)ccc2Cl)=O)CCCC2CCCCC12 C(=O)(N=c1cc(C2(CN(C)C)CC2)o[nH]1)C1(C)N(C)CC(O)C1 N1(C(C(C(C)C)C)=O)CCCC2(CC(NC(=O)CCC3(C)CC3)C2)C1 c1(C(=O)NCCC2(NC(C=CC(C)C)=O)CC2)cc(O)nc2ncccc12 CC1CC(CO)(NC(C2CCC2CNC(=O)CCn2cccn2)=O)C1 C1(NC(c2c(C)nsc2C)=O)CCN(C(=O)C2CC2)CC1C CC(CC(=O)NCCCC1CCN(C(C2CCOC2)=O)CC1)P(C)(C)=O Nc1cc(F)c(CC(=O)NC2CN(C(=O)C(F)C(F)(F)F)C2)cc1F N1(C(C(C)N(C(=O)CCNC(=O)NC)CC)=O)CCC(F)(C#N)C1 C(N=c1cc[nH]c(=NCCCN(C)C)[nH]1)c1ccc(N(C)C)s1 Cc1coc(C(=O)N(CC(C)CNC(=O)CCCc2ccsc2)C)c1 C=CCC(C)(C)C(=O)NC(C)C(C(C)C)NC(c1nccnc1SC)=O C1(CC=C)(C(=O)NCCCCOC(C)=O)CCCN1C(c1ccc(CF)cc1)=O C12(C(N(C3CC3(C)C)C)=O)COC(C1)C(NC(C1(C)CCCC1)=O)C2 c1(C(=O)NC(C(C)C)CNC(C2CC3C(C2)C3(F)F)=O)ccc2[nH]c(=N)oc2c1 c1(C(=O)NC2C3CN(C(C(C)(C(C)C)OC)=O)C(C3)C2)ccc2cccnn12 C(=O)(CC(O)CC(C)(C)C)N1CCC(C(C)C(N2CCN(CCO)C(=O)C2)=O)CC1 C1(C(N2C(C(N3CCC(OC4CC4)C3)=O)CCCC2)=O)CC2CC1CC2O C(=O)(C1CCc2nccn21)NCC(C)(C)NC(c1cccc(C(C)(F)F)n1)=O N1(C(c2c(C)nn(C)c2C)=O)CCC2(CC1)CC2NC(=O)CCc1n[nH]c(=N)s1 c1(C(=O)NC2CCC(NC(C(Br)=C(C)C)=O)CC2)nc2nc(C)cc(C)n2n1 C(=O)(C(COC(C)C)NC(=O)CCC1CC1)N(C)CC1(OC)CCC1 CCC(CC)(C(=O)NCC(F)CNC(c1cc(C)cc(C)n1)=O)c1ccccc1 Cc1cc(F)ncc1C(N1CCC(CN(C)C(c2ccccc2Cl)=O)C1)=O C(=O)(C(O)CCSC)NCC1(NC(c2ccc(COC)[nH]2)=O)CCCC1 C1(OC)CCCC(N=c2cc(C)[nH]c(=NCc3cc(-c4ccccc4)no3)[nH]2)C1 C12(C(N(CCOC)CCOC)=O)CC(CO)(CN1C(c1scnc1C#N)=O)C2 C(CCC(C)C(=O)N1CC(CNC(c2cccn2C(C)C)=O)C(C)C1)OC N1(C(C(COC)O)=O)CC2(CCC(CNC(c3cc4[nH]ccc4s3)=O)O2)C1 CC1(C)Cc2cccc(C(=O)NCCSC)c2O1.c1(C(=O)N)ccn2nccc2c1 CC1CCC(Cc2ccc(SCC(=O)NC(c3ccco3)CC)cc2)CC1 C1(O)(CNC(=O)C=Cc2cc[nH]n2)CCN(C(C2C3CCCC23)=O)CC1 CCCCC(C(=O)NCC1CC2CCC1N2C(=O)CC(C)(C)C)N(C)C C1(CNC(C2CCCOC2)=O)CCCCCN1C(=O)Cc1ccns1 C1(CNC(CCCN(C)C)=O)(NC(=O)C(F)n2ccnc2)CCC(F)(F)CC1 N1(C(CSC(C)C)=O)CC(N(C)C(C2CC3(CC3)CN2C)=O)C(C)(C)C1 CC1CN(C(c2ncccc2Cl)=O)CCCN1C(c1c(F)cc(F)cc1Cl)=O C1(C)(COC)CC(NC(=O)CC2(CO)CC2)CN1C(c1cnoc1C)=O C1(COC)CN(C(=O)CSC)CCN1C(C1CCCNS1(=O)=O)=O c1(N2CC(CC)OCC2)nc(=NCCC2CC(O)C2)[nH]c2cccnc12 CCCCCC(O)CC(=O)NC(C)C=CC(N1CC2(CCC(=O)NC2)C1)=O c1(CC)cccc(NC(C2CN(C(c3ccccc3Cl)=O)CC2C)=O)c1 C(=O)(C(O)CC(C)(C)C)N1C2(C(=O)NCc3ccc(C)c(C)c3)CC2CC1 n1(CCC)nccc1C(=O)NC1CN(C(=O)COCC(F)F)C1 c1(C(=O)NC2CCCCN(C(CCN(CCC)C)=O)C2)cc2cccnc2cn1 CC1CCC(C)N1CC(=O)N(C)CCN(C(=O)C=Cc1cccn1C)C c1(CCCC)ccc(C(=O)NC(CNC(=O)C(Cl)=CCl)CCOC)cc1 C12(NC(C3C(C)(C)OCC3)=O)CCC(NC(=O)C(O)C(F)(F)F)(CC1)C2 c1(C(N2CCN(C(CCCC(C)C)=O)CC2CF)=O)ccc2ncccc2n1 N1(C(CN(CCC)C)=O)CCCC(C2CCN(C(C3(CO)CC3)=O)C2)C1 CC1CN(C(=O)CC2(CO)CCOCC2)CCN1C(C1CC(C2CC2)=NO1)=O c1(CCC(=O)N(C(C)CNC(=O)C(C)n2cccc2)CC)cccc(C)c1 C1(C(N(CC#N)Cc2ccccc2)=O)CCCN(c2ccc(F)cn2)CC1 C12(CCCN)CC(C(=O)NCCc3ccc([N+](=O)[O-])cc3)(C1)C1(CCC1)O2 C1(C(N2CC(C(C)NC(C3CC3CNC(=O)OC)=O)C2)=O)(COC)CCC1 c1(C(=O)NCC2C(CNC(c3cc(C)nnc3)=O)C2)cc(C)c(O)c([N+](=O)[O-])c1 c1(C(=O)NCC2CCN(C(C(C)SCC)=O)C2)cc(OC)nc(F)c1 N1(C(c2cc(CNC(CC(CCOC)(C)C)=O)on2)=O)CCC(C2CCOC2)C1 N1c2ccccc2CCC1C.Cc1cc(C)c(S(=O)(=O)N2CC3COCC3C2)s1 c1(C(N2CC(NC(=O)CC3C=CCC3)CC(C)C2)=O)ccc2c(c1)CCCC2=O c1(C(=O)NC23CN(C(CC4CC(OCC)C4)=O)C(C2)C3)ccnc(Cl)c1OC N1(C(CC2=NOC(C)C2)=O)CCC2C(O)C(C)(C)C12.c1(C(C)OC)nc(C(=O)O)co1 Cc1nc(C(=O)NC2(C(=O)Nc3cccc(CCF)c3)CCCCC2)cc(O)n1 c1(C(N(CCC(C)NC(c2cc(CC)[nH]n2)=O)C)=O)ccc(F)cc1Cl Cc1cc(C(N2CCC(C)C2CNC(=O)CC2CCC2)=O)cc([N+](=O)[O-])c1Cl C(=O)(C1=CCCC1C)N1C(C)(C(N2CC(C#C)(F)C2)=O)CCC1 N1(C(C(C2CCC2)OC)=O)CC2(CCCC2)C1.c1(C2C(=O)N2)cn(C)nn1 c1(C(=O)NCC2CC(C)CN(C(C3CCC3(F)F)=O)C2)ccn2ccnc2c1 c1(C(=O)NCC2CCCC(NC(C=C(C)C3CC3)=O)C2)cccc2nc(O)oc12 Cc1nccc(C(=O)NCC2(NC(=O)C3=CSCCO3)CCOC2)c1C c1(OC)ccccc1C(=O)NC1CCC(CO)CC1.C1(=O)C(CC2CCCC2)N1 CC1(CNC(c2n[nH]c(C3CC3)n2)=O)CCN(C(c2n[nH]cc2F)=O)C1 N1(C(c2c(C(C)=O)coc2)=O)CCC(N(C)C(C2CC(OC(F)F)C2)=O)C(C)C1 c1(N2CC(COC)C(CO)C2)ncc(C)cc1S(=O)(=O)N1CCC(OC2CC2)C1 c1(C(N2CCC(NC(C(=O)NCC3(O)CC(N(C)C)C3)=O)C2)=O)cccnc1Cl CON1CCC(CC(N2CC(O)CC2CNC(=O)C=CCn2cccn2)=O)CC1 c1(C(=O)NC(c2cnn(C)c2)CC)ccc(C2=CCCC2)cc1 C(=O)(C1=NOCC1)NCC(C(=O)NC1COCCC1O)N(C)C C1(C(=O)NC2CC(CNC(COCCN(C)C)=O)C2)C(C#N)C1(C)C Cc1cccc(-c2nnc(CN3CC(NC(c4scc(C)c4C)=O)C3)o2)c1 C#Cc1cc(F)c(C(N2CC3(CNC(c4ccc[nH]4)=O)CCC2C3)=O)cc1F C(=O)(CS(=O)(=O)CCO)NCC1(F)CCC(NC(c2ccc([N+](=O)[O-])s2)=O)C1 CCC(CC)(CC)C(=O)NC1CCCN(C(c2nc(C(C)(C)C)c[nH]2)=O)C1 c1(C(=O)NC(CN(C(c2nc(C(F)(F)F)sc2C)=O)CC)C)cccc(O)c1F c1(CC(=O)Nc2c(C)cnc(C)n2)ccc(F)cc1[N+](=O)[O-] c1(CN(CCCNC(C2C(C(=O)OC)C2)=O)CCN(C)C)ccc(OC)cc1F C1(NC(Cc2c(C)nccc2)=O)CC(C)CN(C(=O)Cc2cncn2C)C1 CCCC(CC(C)C)C(=O)NCC1CC(NC(c2ccc(O)cc2C)=O)C1 Cn1nc(NC(C2(C)CCN2Cc2cc(Br)c(O)c(I)c2)=O)c2cc(I)cnc12 N1(C(Cc2c(C)nc(O)nc2O)=O)CCN(C(c2cccn2C)=O)CC(C)(C)C1 Cc1cn2c(C(=O)NCCCNC(C3CSCN3C(=O)C(C)(C)C)=O)cnc2s1 c1(C(c2n(C(C)C)nnn2)NCCCn2ccnn2)cc(F)ccc1Br C1(C(N(C(C)C(N)=O)C)=O)OCCC1CNC(C1CCN(C)C1)=O C#Cc1ccc(F)c(C(=O)NCC(C)NC(C2CCN(CCO)C(=O)C2)=O)c1 CCC(C(=O)NCC1(F)CCCN(C(=O)C(C)(C)c2ccsc2)C1)C(C)(C)CC C1C(C)C(C)C(=O)N2CCC(C2(C)C)CC(=O)N1.C1(COC)CC(=C2CCC2)C1 N#Cc1ncc(C(=O)NCC2CC2NC(=O)CCC2CC2)s1 c1(C(=O)NCCCOCCCNC(C2C(C)OCC2)=O)ccc(C(N)=O)cc1 c1(SC)cc(C)c(C(=O)Nc2cccc(NC(c3cc(C)nn3C)=O)c2)o1 C(=O)(C1CCCc2ccnn21)N1CC(C)N(C(c2cc(Cl)c(N)c(Cl)c2)=O)CC1 CC(C)CC(C)C(=O)NC1CN(C(c2ccc(F)s2)=O)C1 c1(C(=O)NCC(=O)NC(C(C)NC(C2C=CCCC2)=O)CO)cccc(C(N)=O)c1 c1(CC)noc(CCC(=O)N(CCN(C(C2CC2Cl)=O)CC)CC)n1 CC1CCCC1C(=O)NC1CC(C(=O)NOC2CCC2(C)C)C1 Cc1cc(=NC2CCC(NC(=O)C(C)C(C)(F)F)CC2)[nH]cc1C#N C(=O)(C(CO)C(F)(F)F)NC1C(NC(Cc2cc(CC)nn2C)=O)CCC1 C1(CC(=O)NCC2CC(N(C(=O)C(O)c3ccco3)C)C2)CCC(=O)CC1 N(C(=NCCF)NCC1(CC)CCCCC1)CC1(OCC)CCCC1 c1(CC(=O)NC(CNC(c2ccn(CC)c(=O)c2)=O)C)c(Cl)ccc(O)c1Cl CCC(Cc1ccccc1)CC(=O)NCC(C)NC(c1cnc(SC)cn1)=O.C(C)C N1(C(C(CSC)O)=O)CCC(C2CC(NC(=O)C3=C(Cl)CCC(C)C3)C2)CC1 C1(C(N2CCCC(CN(C(=O)C(O)C(C)C)CC)C2)=O)CCC(O)CN1C O=[N+]([O-])c1ccc(F)cc(N2CC(CO)C(c3c(F)cncc3F)C2)c1=O c1(C(=O)NCC2(CNC(c3csnc3Cl)=O)CC2)cc2cc[nH]c(=O)c2s1 CC1CN(C(=O)C=CCN(C)C(C2(C)CNC(=O)N2)=O)CCCO1 C1(CC(=O)Nc2c(O)ccc(C)n2)C2CCC1CN(C(=O)CCCn1cccc1)C2 C1(NC(C2(OCC)CCC2)=O)CCC(C)N(C(C2CC3(CCC3)C2)=O)C1 c1(CC)cnn2c(N(CC(c3ccc(Br)c(F)c3)C)C)cc(Cl)nc12 Cc1nn(CC2CC2)c(=O)c(-c2nc(-c3ccsc3)nn2C2CCSC2)c1C c1(C(N2CC(N(C(c3c(C)coc3)=O)C)C2)=O)c(C)nc(C)nc1C C(=O)(CCCC(=O)NCC(C)NC(C1CCCN1CC1CC1)=O)OCC C12(CNC(C3CC(CC)C3)=O)CC1CN(C(c1ccc(OC(C)C)nn1)=O)C2 N1(C(C2C(C(N)=O)C2)=O)CCN(C(=O)COCC2CCOC2)C2(CCC2)C1 Cc1cc2occ(CC(=O)NC(CCc3ccccc3)CC(F)(F)F)c2cc1C CC1CC(C)N(C(=O)CCc2cccnc2F)CCN1C(=O)CS.C1CCC1C(C)C Cc1cn(C)nc1C(=O)N(C)CC1(O)CN(C(c2c(C)nsc2NC2CC2)=O)C1 N1(C(CSC)=O)CCOC2CN(C(C3CC4CCC3C43CC3)=O)CC12 Cc1nnc(N2CCC(C)(NC(c3coc(CC4CC4)n3)=O)C2)c(C#N)c1C N1(C(C2CCS(=O)CC2)=O)CC(C2CN(CCF)C2)C1 c1(-c2cc(SC)on2)nc(C(=O)O)nc2c1CC(C)CC2 N1(C(C(OC)OC)=O)CCC1(C)C(N1CCC(c2nc[nH]n2)C1)=O CCC(C)CCC(=O)NCC1(C(N)=O)CN(C(c2cc(C(C)(C)C)on2)=O)C1 C#CC1(C)CCCN(C(=O)C(CCC=C)NC(=O)CC(C)(C)CN(C)C)C1 c1(C(C(C)NC(=O)C(=O)N2CSC2C2CC2)=O)ccc(F)cc1 C(=O)(CC(C)(C)C(=O)NC1CN(C(=O)CC2CCC(=O)NC2)CC(C)(C)C1)OC c1(C(N(C2CCN(C(=O)CCC(C)(C)C)C2)C)=O)cnn2c(=N)[nH]cnc12 Cc1cc(C(=O)NCCC2CCCN2C(c2cc(C)oc2C)=O)cc(Cl)n1 O=C(CN=c1ccc(F)c(Br)[nH]1)NCCCn1cc(CCC2CCCC2)nn1 C12(NC(Cc3cccc(CC)c3)=O)CN(C(=O)C=C(Cl)Cl)CC1CS(=O)(=O)C2 C1(Cn2cc(CN)nn2)CN(C(=O)C(F)C2CCOC2)CCO1 N1(C(COc2cn(C)nc2)=O)CC2CC(CNC(c3coc(C4CC4)n3)=O)CC1C2 c1(C(=O)N)cnn(C)c1C.C12CC(C1)CCNC(=O)CS2.C#CCOCCSC c1(CCC(=O)NC(CC)CNC(C2CC3CC3C2)=O)ccc2c(c1)CCO2 c1(OC)ccc(C(=O)NCCNC(=O)Cc2ccc(CO)c(C)c2)c(N)c1 CC1(C(N2CCC3(CC3CNC(=O)CC3CCC34CCC4)C2)=O)CCC(=O)CC1 c1(CNC(C2OCCN(C(C(C)=CC(C)(C)C)=O)C2)=O)nc(C)cc(C)n1 n1(CC(=O)NC2(CNC(CCCCOCC)=O)CC2)cnc2ccc(C)cc12 c1(C(=O)N)cc(O)nc(O)n1.N1(C(C(C)C#N)=O)CCC(C)(Cc2ccccc2)C1 C(C)(CCC(=O)NC(CCC(=O)N(C)C)c1ccccc1)SC N1(C(C(C)Sc2ccccn2)=O)CCC2(CC1)CC2NC(=O)C(C)(CO)CO c1(OC)ccc2c(C)c(C(N3CCC(C(C)NC(=O)C=C(C)C)C3)=O)[nH]c2c1 c1(CCC(=O)NC2CN(C(C3(CC)CCCCC3)=O)C2)cc(Br)ccc1F CC1=CCC(C)(C(=O)NC2C3CCC(C3)C2CO)CC1 c1(C(N2C(CCNC(C=Cc3nc(C)sc3)=O)CCC2)=O)cn2ccncc2n1 C1(C(=O)NC2CN(C(=O)COC3CCCC3)CC2C2CC2)CC2(CCCC2)CO1 CCC1=C(C(=O)NCCN2CCN(C(=O)CCc3ncc(C)[nH]3)CC2)SCCO1 C1(NC(c2cc(C)sn2)=O)CC2CC(NC(c3ccsc3Br)=O)C2C1 c1(C(=O)NC2C(NC(C3CC(OC)C3)=O)CCCC2)cc(F)cc2c1CCC2 C1(NC(CS(CC)(=O)=O)=O)CCCC2CN(C(C3(C#N)CC(=O)C3)=O)CC12 c1(NC(C2N(C(c3c(OC)ccs3)=O)CCOC2)=O)ccc2c(c1)CCCO2 c1(C(N(CC(CNC(C(CC)NC(N)=O)=O)O)C)=O)csc2c(F)cc(F)cc12 C1(NC(C(C)(C)F)=O)CN(C(c2csc(=N)[nH]2)=O)CC2(CCOCC2)C1 C#CC1(C(=O)N(CC(C)NC(=O)C(C)Oc2ccc(Cl)cc2)C)CCOCC1 C12CC3(CCN(CC3)c3ncnc(Cl)c31)C2.C(C)(C(=O)OC)OCC=C CCC(CC)C(F)C(=O)NC1CC(C(=O)NCCCCCCCO)C1(C)C N1(C(c2cc(C(C)(F)F)on2)=O)CCC2(NC(c3c[nH]cc3Br)=O)CC2C1 O=[N+]([O-])c1cc(Cl)c(Cl)cc1S(=O)(=O)NC1CC2(CCOCC2)CO1 Cn1cc(CNCCc2ncon2)cc1C#N N1(C(c2cnc(C)n2C)C(=O)NCc2ccc(OC)cc2)CC2CSCC2(C)C1 N1(C(=O)NC(CCCC)C(=O)OC)CCC2CCC(C1)N2CC1CCC(CN)C1 C1(CCN(C(C=CCN(C)C)=O)C)CCCCN1C(C1CC2(CSC2)C1)=O C(=O)(C(CC1CC1)C(C)(C)C)NC(C(=O)OC)C1CC1.C1(=O)C(C2CCC2)N1 c1(C(N2CCC(COC(F)F)CC2)=O)cccnc1O N1(C(c2cc(N3CC(C)C=C(C)C3)ncn2)=O)CCC(C2(OC(C)C)CC2)CC1 Cc1cc(C(=O)NO)ccc1C#N.C(=O)(C(C)(C)c1ccccn1)N1CC(C(=O)CN)C1 N1(C(C2N(C(CCC)=O)CC2)=O)CCC(NC(c2cc(CC)on2)=O)(CC)CC1 c1(CCC(=O)NCC2CN(C(=O)CC3CCCOCC3)CCO2)cccc(Cl)c1 C1(C2CCN(C(C3CN4CCCN3CC4)=O)C2)(NC(C(C)CCN(C)C)=O)CC1 C(=O)(C(C)(C)CN(C)C(C1CC1Cl)=O)NCCC1(OC)CCC1 N1(C(C(C(C)C)C#N)=O)C(C(=O)NCC2(C)CSC2)C2CC(O)C1C2 Cc1cnc(C(=O)NCC2CCN2C(=O)CCOc2cc(F)cc(F)c2)c(F)c1 Cc1cc(C)c(C(N2CC(C3(NC(c4ccns4)=O)CC3)C2)=O)c(O)c1 c1(CCC)n[nH]c(=NC2CCCC3CN(C(=O)C(=O)CC(C)C)CC23)s1 C1(NC(CC(C)(C2CCC2)N(C)C)=O)CN(C(=O)CC(C)F)CC1N=[N+]=[N-] C1(C(=O)NCc2n(C)ccc2)CC2(CCC2)CN1C(=O)C1=CCCCC1 C(c1cccnc1)=CC(=O)NC(C)C(=O)N(CCC(=O)NCCOC)CC#C C(=O)(CC1=CCN(C)CC1)N(CC(CNC(C(CC)CC1CCCC1)=O)O)C c1(OC)cccc2c(CC(=O)NCC(F)CNC(=O)C(O)P(C)(C)=O)coc12 c1(CC(=O)NC2C(C)CCN(C(CCCC=C)=O)C2C)ccc2oc(C)nc2c1 N1(C(CSC(C)C)=O)CC(NC(=O)C(C(C)C)N2CCCC2)C(n2ccnn2)C1 c1(C(=O)NC(CNC(C(CC)O)=O)C)ccc(O)cc1-c1ccc(F)cc1 N1(C(C2C(NC(=O)NCC)CCO2)=O)CCc2c(NC(=O)C(F)(F)F)cccc21 CCCC(C)(CC)C(=O)NCC1(NC(C2CC(C)CCO2)=O)CCOC1 N1(C(C(C)NC(N)=O)=O)CC2CCC(CNC(=O)C(C)(F)C(C)(C)F)C2C1 c1(C(C)NC2CC(n3cccn3)C2)nc(=O)o[nH]1 c1(C(N2C(C(=O)Nc3ccc(CC#N)cc3)CC3CC32)=O)c[nH]c2ccccc12 c1(OCC=C)ccc(C(N2CCOC(CNC(C34CC3C4)=O)C2)=O)cc1 N1(C(Cc2c(N)cccc2)=O)CCN(C(=O)C(F)=C2CCC2)CC1C1CC1 C(=O)(CCCC(F)(F)CO)N1C(C(=O)NCCN(C2CCS(=O)(=O)C2)C)CCCCC1 N#Cc1nc(Cl)ccc1NC(C1CC2CC2N1C(c1ccc([N+](=O)[O-])[nH]1)=O)=O CCCCCC(O)CC(=O)N1CC2(CCN2C(=O)COc2cn[nH]c2)C1 Cc1cccc2c1N(Cc1n[nH]c(C)c1Cl)CCC2C C(=O)(C1=CCC(C)CC1)NC(C)CNC(c1c[nH]c(C#N)c1)=O C12(NC(c3cnc(CC)[nH]3)=O)CCCN(C(=O)C(c3ccc(O)cc3)=O)CC1C2 N1(C(C(C2(O)CC(C)(C)C2)C)=O)CCC(C(F)(F)F)C(NC(=O)C=CI)C1 c1(C(C(=O)NCC2(F)CC(NC(CCC#C)=O)C2)C)ccc(F)c(Cl)c1 c1(OC)cc(C(N2CCC(C(=O)NC3CC(C)(C)C3)C2)=O)c(OC)cc1Br c1(C(N(C2CCN(C(C(C(C=C)C)C)=O)CC2)CCC)=O)cnc2ccsc2c1 c1(C(=O)NC2CCCN(C(c3cncc(COC)c3)=O)C2)cccc2nsnc12 C1(CCC)CCCC1NC(=O)NC1CC1(C)CC N1(C(C23N(C(c4c(CC)con4)=O)CCC2C3)=O)CC2(CCCC2)C1 CCC(N=c1[nH]c2c(c(=NCCCn3ccnc3)[nH]1)COCC2)c1ccccc1 Cc1cc(CCCNC(=O)C(c2cnn(C)c2)NC(c2cocc2C)=O)on1 C(=O)(C(CCCC(C)C)N1CCC(C(=O)NCC(F)(F)F)C1)NC C1(C(N2CC3C(CNC(c4n(C)cnc4)=O)C3C2)=O)C2Cc3ccccc3C12 CC1CC(=O)NC(C(=O)NC(c2ccccc2)CNC(=O)CCCN(C)C)C1 C(CC)(C(=O)N(C)CC1CCCN1C(=O)C(c1ccccc1)OCC)=CCCC CCCCC(O)C(=O)N1CC(O)CC1Cn1cc(-c2ccc(C(=O)O)cc2)nn1 C(CC(=O)NOCCC(C)C)C1CC(NC(C(=Cc2cn[nH]c2)C)=O)C1 C1(OC)CN(C(=O)CN2CCCNS2(=O)=O)C(C)(CNC(=O)CC2(OC)CC2)C1 C1(N(c2c(C)c(Cl)ncc2)C(C2CCCS2)=O)COC2(CCNCC2)C1 C(=O)(C1=CCN(C(=O)CCc2nc(O)n[nH]2)CC1)NC(c1ccn(C)c1)C c1(C(N2CCCC(C(=O)NCC3C(C)CCC3)CC2)=O)ccc2cc[nH]c2n1 C=C=C(C)CC(=O)NCC1(F)CC(CNC(=O)CCC(=O)c2ccc(C)s2)C1 C=CCC(CN=c1nc2scnc2c(NCCCCN2CCOC2=O)[nH]1)OCC N1(C(CCC)=O)CCC2(CC1)CN(C(C1(CO)CC(C)(C)C1)=O)C2 N(C(=NCCCCN1CCOC1=O)NCc1ccnc(CN(C)C)c1)C1C(C)C1 c12cnc(c(F)c1Cl)N(C)C2C(=O)NC1CCC1.C1(CC)CCC(NCC)CC1 C1(O)(c2cn(Cc3ccc(OC)cc3)nn2)CCN(C(N2CCCC2=O)=O)CC1 CC(CN=c1[nH]c2c(c(=NC3CC3F)[nH]1)COCC2)Oc1ccccc1F N1(C(CCOC(C)(C)C)=O)CCC(C(C)(C)F)(CNC(=O)NC2CCCC23CC3)C1 N1(C(C(C)C#N)=O)CCCC2CN(C(c3ccc(C4CC4)cc3Cl)=O)CCC12 C1(C(=O)NC(C(C)(C)O)(C)C)CN(C(=O)C=CC(=O)OC(C)(C)C)CC1(F)F Cc1ncnc(C)c1C(=O)NCCNC(=O)C(O)CCn1cncn1 c1(OC2CC(NC(C3CCCO3)=O)C2)ccc(F)cc1.c12occc1CNC2=O C12(C(N3C4CC(NC(COC(C)=O)=O)CC3CC4)=O)CCC(N(C)C)(CC1)CC2 c1(C(=O)NCC(C)N(C)C(C2CCC2C)=O)nc[nH]n1 CC1=C(C(=O)NC2CCC(CC(=O)NCCOC3CC3)CC2)CCC1 c1(C(=O)NC2CCN(C(C3C(=C)C3)=O)C2C)ccc(Cl)c(N2CCCS2(=O)=O)c1 Cc1cc(C(c2nnnn2CC2CC2)NC2CCC3(CC3)C2)ccc1C#N c1(Sc2c(CC)cccn2)ccc2c(c1)CCCC2 c1(C(=O)NC(C)CC(C)NC(=O)COC2(C)CCCC2)ccnc2ncccc12 CC(C)C(C)CC(=O)N1C2CCC1C(CNC(c1ccnn1C1CCCC1)=O)C2 N1(C(c2cccn3ncnc23)=O)CCC2(CCN(C(c3cncs3)=O)C2)C1 C1(C(=O)NC2C(CNC(CCCN(C)C)=O)CC2)CCC(F)(F)CC1 Cc1cc(Cl)nc(N)c1C(=O)NCCCn1cc(CSc2c(Br)nnn2C)nn1 c1(C(N2C(C)CCC(NC(c3ccc[n+]([O-])c3)=O)C2)=O)nnn2c1C(=O)NCC2 N1(C(CC(C=C)(C)C)=O)CCC(CNC(c2cc(SC)oc2C)=O)C(F)(F)CC1 C1(NC(=O)CCC2CC3CCC2C3)CCN(C(=O)CCn2cccn2)CC1F CCCS(=O)(=O)NCC(=O)NC(C1CCCCC1)CNC(=O)CCNS(C)(=O)=O CCCCCCC(F)C(=O)N1CCN(C(c2cc(Cl)c(N)cc2F)=O)C(CC)C1 C1(CNC(c2cc(OC)no2)=O)(OC)CCN(C(C2(C)CCOC2)=O)C1 c1(C(N(CCOCCNC(C2C(C3C(C)C3)C2)=O)C)=O)cc2ccccc2o1 CCC(CC(F)F)C(=O)N1CC(O)(C(C)NC(=O)CC2CC3(CCC3)CO2)C1 c1(-c2scc(CC(=O)NCC3CCCC34CC4)n2)ccccc1Cl C(=O)(C1c2c[nH]nc2CCN1Cc1nn(C)cc1CN)OC c1(C(=O)NCc2scc(CNC(=O)OC(C)(C)C)n2)cc(O)cc(N)c1Cl C1(CNC(C(c2ccccc2)C)=O)CC2CC1CN(C(C13CC(C)(CO1)C3)=O)C2 C1(C(N2CCC(N(c3cc(O)ncn3)CC3CC3)CC2)=O)(CC)CCNC1=O c1(NCC(C(CC)C)O)ccc(S(=O)(=O)N(C)C(C2CCCCCC2)C)cc1Br N1(C(CCCC2C(C)C2)=O)CCCC(CCO)(NC(C2CCCC(O)CC2)=O)C1 C1(NC(CSCC(C)C)=O)CN(C(=O)CCc2ncc(F)cn2)CCC1C C(=O)(CCC(C)(C)C(=O)N1CCN(C(c2cccnc2C(F)(F)F)=O)CC1)OC C1(CC#C)(C(N2CCCC(N(C)C)C2)=O)CCN(C(=O)CCC(C)=O)C1 Cc1cc(F)ccc1C(=O)NC(C)CC(C)NC(c1cc(C2CC2)nnc1O)=O c1(C(N2CCN(C(C3CC3F)=O)CC2)=O)cc2c(cn1)OCCC2 C12(SCC)CCC(NC(c3cc4sccc4cn3)=O)(CC1)CC2 c1(OCC)ccc(C)nc1C(=O)NCCC(C)N(C(=O)C=Cc1cnc[nH]1)C C1(=O)C(CNC(=O)NC)C1=O.C(=O)(C(CC)C1CC1)NCCNCC(C)C.CCOC N(C1CCOc2ccccc21)C(c1nccc(-c2cnc(C(F)(F)F)cn2)n1)=O C(C(C(=O)N1CCCC(O)C1CO)C(C)C)NC(c1c(OC)nsc1)=O CC1CN(C(c2cnc(Cl)cc2Cl)=O)CCN1C(c1cccnc1Cl)=O C(C(C)(C)CNC(=O)CCNC(c1ccccc1)=O)N(C(=O)CC1C=CCC1)CC C1(NC(CC(=C)C)=O)CCSC12CN(C(=O)C(F)=CC1CC1)C2 CCCCC(O)C(=O)NC(C)C(CO)NC(=O)CNC(=O)Cc1ccc(O)cc1 c1(CC)cc(Cl)ccc1C(=O)NCCCCNC(C1OCCC1CC)=O C=CC(C)CC(=O)NCC(C)CNC(=O)CC(=O)N(C)C CCCCC(C)N=c1nc(N2CC(CC)OC(C)(C)C2)c2[nH]ccc2[nH]1 Cc1ncc(C(N2CC(O)(CCNC(=O)CC(F)(F)Cl)C2)=O)n1C C1(C(N2CCCN(CCNC(CCCC(N)=O)=O)CC2)=O)CCn2cnnc2C1 C1(NC(CCCC(=O)NC)=O)CC2CCC(C1)N2C(=O)Cc1cn2ccsc2n1 Cc1ccc(C(=O)NCC(C2CC2)NC(c2cnc(C3CC3)nc2C)=O)cc1N Nc1cc(C(=O)NCC(O)CNC(=O)C(O)C2CCCC2)ccc1Cl C1(C2(O)CN(C(C3(O)COC3)=O)C2)(CNC(C23CCC(CO)(CC2)C3)=O)CC1 CC1CC2CN(C(C3C4CCCCC34)=O)CC2N1C(c1ccc(C(C)(C)C)[nH]1)=O c1(C(=O)NC(C2CC=CCC2)C(=O)NCCCN(C(C)=O)C)cn(C)nc1C C1(CC)(NC(=O)CCC2CCN(C)C2)CCN(C(=O)C(=O)C(C)(C)C)CC1 N1(C(c2cocn2)=O)CCC2(CC1)CC(N1CCC3(CC1)CC(F)C3)C2 c1(CC2(C(=O)NC(C(=O)OC)CSC)CC2(F)F)cc(F)cc(Br)c1 c1(C(N2CC(C)OCC2(C)C)=O)cc2c(-c3cscn3)cncc2s1 c1(C(C)NC(C(C(C)C)S)=O)cccc2cccnc12 N1(C(C(CCC)O)=O)CCC2(CCN(c3nccc(N4CCCC4)n3)C2)C1 C1(NC(C2(CO)CCCC2)=O)C2CCC1CN(Cc1cn3ccccc3n1)C2 C1(NC(C2CC(C)OC2)=O)CC2CCC(C1)N2C(=O)CCc1cn(C)nn1 C(=O)(C1=CS(=O)(=O)CCC1)N(CC(CN(C(=O)CCCC1CCCCC1)C)O)C c1(CC(C)N(C(C(=O)NCC(CSC)OC)=O)C)cccc(F)c1 c1(COC)cc(C(=O)NC(CNC(C2CC2F)=O)C2CCC2)n(C)n1 c1(C(=O)NCCC(C)NC(C2CC2CF)=O)cc(Br)n2ccccc12 Cc1ccccc1-c1cnc(C2(C(N3CCSCC3CO)=O)CC2)o1 C=CCC(C)(C(=O)NCC1CC2(CC2)CN1C(=O)CCN1CCOCC1)N(C)C C1(C(=O)NC2CCC(NC(c3c(CC)nn[nH]3)=O)C2)CC(C2CCC2)C1 N1(C(c2cc(C(=O)OC)n(C)c2)=O)CCn2nc(CNC(=O)CN(C)C)cc2C1 Cc1cc(O)nc(CSc2ccc(C(=O)OC(C)(C)C)c(C)n2)n1 C1(C)(C(N(C(C)CCNC(C2CCCCN2C)=O)C)=O)CCCC(F)(F)C1 c1(C(=O)NCC2OCCN(C(C=CC=CC)=O)C2)ccnc(F)c1F N1(C(C2(COC)CC(=O)C2)=O)CCCC(CC(=O)NCc2cnn(C)c2)C1 Cc1cccc(Cl)c1C(=O)NCC1CCCN1CCCn1cccn1 c1(CC(=O)NC(CC)CN(C(=O)CC2C=CCC2)CC)cccc(C2CC2)c1 N1(C(c2nc(CC)oc2)=O)CC(O)CC1CC(=O)N(C1CCN(C)CC1)CC c1(CCOCC(=O)N(c2ccccc2)C)cc(F)cc2c1OCOC2 C1(C(NOCCCOC)=O)CCC(O)CN1C(=O)C(C#N)C(C)C O=C1CCC2(CN1)CN(C(C1CC(O)C(O)CC1CNC(=O)C1CC1)=O)C2 C12(NC(=O)CNc3nccs3)CCC(C3CC(CC(=O)OC(C)(C)C)C3)(CC1)C2 c1(OC)cc(C#N)ccc1CN1CCC(O)(C(=O)Nc2cc(Cl)cc(C)c2I)C1 C1(C(N(CC(C)N(C)C(c2ccc(Cl)c(F)c2F)=O)C)=O)CC1C1CCCCC1 C12(C(N3CC(NC(C(CC)O)=O)C(C)C3)=O)CCCN1CCC2 C(CC)(C(=O)N(C1CCN(C(c2cc(C(CC)CC)no2)=O)C1)CCO)OCC c1(OC)cc(CO)ccc1C(=O)NC(C)CNC(=O)C(c1ccc(N)cc1)(C)C c1(C(N2CCC(C)(NC(C)=O)C2)C(=O)NC)ccc(C=CC(=O)OC)cc1 C1(CNC(c2cnc(C)s2)=O)CC2(CO1)CN(C(C1(F)CC=CCC1)=O)C2 CN1C(=O)c2ccccc2C1CN1CCCCC1C1(O)CC1 c1(NC(=O)NC(c2ccc(OC)c(Cl)c2)CC(=O)OC)ccc(C(C)=O)c(C)c1 C(N=c1nc2c(ncn2C)c(Nc2nccc(=N)[nH]2)[nH]1)c1scc(N(C)C)n1 N1(C(CC(CC)C2CCC2)=O)CCCC(CC(=O)Nc2cnccc2C)CC1 n1(CC)nc(C)c(C(=O)NC2CC3(C2)CN(C(=O)C(C)C(C)O)C3)c1Cl C(CNC(c1cc(C)ccc1C)=O)(C(C)C(C)C)NC(C1(SC)CC1)=O Cc1ccc2c(n1)CN(C(c1cn(-c3ccccc3)cn1)=O)C2 C1(C(=O)NC2C=CC(CNC(c3c(CC)cco3)=O)C2)CCC(C)=C(C)C1 CCC(C)(C)C(O)C(=O)NC1CN(C(c2cc(C(F)F)ccn2)=O)CC1OC C(=O)(C1=CCCCC1)NC1C(C)(C)C(CC(=O)Nc2ccc(F)nc2)C1 Cc1cc(C(=O)Nc2ccc(NCc3[nH]c(C)cc3C)nc2)ccc1[N+](=O)[O-].CC C1(CC(=O)NCC2(CN(C)C(c3cccnn3)=O)CC2)CC2CC2C1 N1(c2nc(C)on2)CCCC(NC(=O)NCCCc2ccncc2Br)C1=O C=CCC(C(=O)NCC(CC=C)NC(c1cc(C(F)(F)F)nn1C)=O)C(C)C C1(C(N(c2ncc(C)cn2)CC2CCNCC2)=O)CCc2nc[nH]c2C1 N1(C(CN2CCC(C(F)(F)F)(C(N)=O)C2)=O)CCOc2ccc(Br)cc2C1 N1(C(c2cnc(C)o2)=O)CCN(C(C2(C)C=CCC2)=O)CC1CO c1(C(N2CCC(O)(CNC(C3(C)CC3(F)Cl)=O)CC2)=O)ccnc2[nH]cnc12 N1(C(C(CC)O)=O)CCCC2(CCCN(Cc3ccc(Br)cc3F)C2)C1 CN1C(=O)CSC1=CC(=O)NC1CCN(C(c2cnc(S(C)(=O)=O)s2)=O)CC1O C12(NC(C(C)(C)SC)=O)CCCC1N(C(C1CN(C)CCO1)=O)CC2 c1(C(=O)OC)c(C)[nH]c(C(=O)NC2CCC2NC(=O)CCCNC(C)=O)c1C C(=O)(C(C)CCCC(C)C)NCCCN(C(c1n[nH]c(C)c1Br)=O)C c1(C(N2C(CNC(C(C(CC)C)O)=O)CC(F)(F)C2)=O)cc2ccncc2s1 N1(C(C(C)(CSC)NC(COC(CC)C)=O)=O)CCC(C)=C(F)C1 C(CC(F)(F)Cn1cc(-c2cncc(N)c2)nn1)NC(COC)=O N1(C(C2N(Cc3c(C(=O)OC)cc(F)cc3)CCOC2)=O)CC2CCN(C)CC2C1 N1(C(C=CC)=O)CCC(C(=O)NCc2cnn(CCC(F)(F)F)c2)CC1C1CC1 O=C(C(F)CC1CCC1)NC1CCN(C(c2cc(Cn3cccn3)on2)=O)C1 c1(C(N(C)Cc2ccc(CNC(C3CC3(F)Cl)=O)cc2)=O)ccn2ncccc12 CCCCC(CNC(=O)Cc1cn[nH]c1)NC(=O)CC(=O)NCC c1(OC)cc(NC(CC(C)C)C(C)C)cc(F)n1 C1(N(CC2CC2)CC)CCN(CC)C1.C1(CC2CCC2)C(=O)N1 C1(C(=O)NC(CN(C(c2ccccc2)=O)CC)C)(C(=O)NC2CC2F)CCCCC1 c1(C(N(CC(C)O)CCNC(=O)C(F)n2cccn2)=O)cncn1C(F)(F)F c1(C(N)=O)csc(NC(=O)CN2CCOC2=O)n1 c1(C(=O)NC2CN(C(C(CC(C)C)O)=O)CC3C2C3)ccc2c(n1)OCCO2 N1(C(c2cc(OC)no2)=O)CC(NC(c2cccc(CC(C)C)c2)=O)C2CC12 CC(C)(Cl)CC(=O)N1CC(NC(c2ccc(C(F)F)nc2)=O)C(O)C1 C1(SC)CN(C(c2nncn2C2CC2)=O)CC1n1cc(-c2cscn2)nn1 c1(N)ccc(S(=O)(=O)NC(C2CCC2)c2nccs2)cc1Cl.CCC(CC)C1CC1 C(=O)(C(O)C1=CCCCC1)NCCN(C(C(C)n1ccnn1)=O)C c1(CCONC(c2cn(C)nn2)=O)ccccc1Cl.C(C(C)C(=O)OC)OC C(=O)(C1=C(C)OCCS1)NC1CCC(NC(c2cc(CC)c(F)cc2)=O)CC1 N1(C(COC(CC)CC)=O)CC=CC(NC(c2ccn(C(C)C)n2)=O)C1 c1(C(C)C)ccc(F)cc1C(=O)NCC1C=CCN1C(=O)C=CBr N1(C(c2cc(OC)n[nH]2)=O)CCC(CNC(c2cc(O)cs2)=O)CC1 c1(CC(N2C(CC)C(NC(c3ccccc3Cl)=O)CC2)=O)cc2ccccc2o1 N1(C(c2ccnc(-n3cncn3)c2)=O)CCCCCC(NC(C2CC(O)C2)=O)C1 c1(C(N2C(CCC)CN(C(C3CCCCC3O)=O)CC2)=O)cc([N+](=O)[O-])oc1C C#CCC(C)(C(=O)NCC1(C(O)C(C)C)CC1)NC(C1CC2(CCO1)CC2)=O c1(C(N2CC3C(CCNC(C(C)=C(CC)C)=O)(CC3)C2)=O)cnc2ccccn12 c1(C(=O)NC(C(CO)NC(Cc2c(C)n(C)cn2)=O)C)ncc(Cl)cc1F C1(C)(C(N2CC(CC(C)NC(c3cnc(SC)s3)=O)C2)=O)CC(C(C)C)=NO1 c1(C(=O)NCC(C)(C)OCCNC(C2CC(C)OC2)=O)cc(F)ccc1Br Cc1nc(C)c(C(=O)NC2(CNC(C3CC(=O)N(c4cn[nH]c4)C3)=O)CC2)o1 CN1CC(NC(=O)CNC(=O)CC(C)(C)C(F)F)C2(CC2)C1=O C1(CC)CN(C(c2c(C)noc2C(F)F)=O)CCC1NC(=O)CCCSC Fc1cc(Br)cc(F)c1CN(C12CC(C1)NC2)CC=Cc1ccccc1 CN1CCCC(NC(=O)C(F)C2CC(NC(C3CC=CC3)=O)C2)C1=O c1(C(=O)NCCCOCCNC(CC2N(C)CCOC2)=O)occ2c1CCCC2 c1(C(N2CCC3C(NC(=O)CCC(F)(F)F)C3C2)=O)cc2ccccn2n1 c1(C(C(=O)NCCOCC)N(C)CC(c2cnc(CCC)s2)=O)ccc(C)nn1 c1(C(=O)NC(COCC)C(=O)N(C)Cc2noc(C)n2)cccc2c[nH]nc12 C1(N(CCNC(=O)Cc2cncs2)CC)CCN(c2ccccc2F)C1=O O=C(C1=CCCCCC1)NCC1CC(O)CN1C(=O)COCC1CC1 C(CCCC(CO)NC(=O)CN1CC2CC2C1)NC(C1C(C(C)O)C1)=O c1(C(N2C3CC(N=[N+]=[N-])C(C3)C2)=O)cncc2cc(Cl)ccc12 CCC(O)C(C)(C)C(=O)N1CC(C(C)NC(=O)Cn2ncc(O)nc2=O)C1 C1(CC(=O)NCC2CC23CCCC3)C2CCCC2N1C(=O)CC1CCCCO1 c1(NC2CC(C)N(C(C3CC4CCCC4C3)=O)C2)ncnc2ccc(Cl)cc12 C1(OC)CC2(CCC(CN(C(=O)C(=O)NC3NC(=O)NC3=O)C)CC2)C1 CC1(C)C2CC(NC(C3COC4(CCC4)C3)=O)CC12 c1(C(=O)NCCCCCNC(C2(CO)CCC2)=O)ccc(Cl)c(Cl)c1 c1(CN2C(CCC(=O)NCC3CCCCO3)CCC2)cc(Cl)c(Cl)cc1O C(=O)(C(=O)N(C)C)NCCN(C(=O)C(C)n1cnnn1)CCC C1(OC)(OC)CCCN(C(=NCCCF)NCCN2C(=O)CCCC2=O)C1 c1(C(c2nnnn2CCCF)NCC2(CC)CCCCC2)cc(Cl)c(Cl)cc1C CC1CN(C(=O)CC2CCC2)CC(CCNC(c2csc(C(F)(F)F)n2)=O)O1 O(C1CCCc2ccccc21)CC(N1CCN(CCNSC(F)F)CCCC1)=O N1(C(c2cc(OC)ns2)=O)CC2(NC(c3ccc(CO)nc3)=O)CCCC2(F)C1 C1(COC)C=CCCN1C(=O)C(CNC(c1cnnc(O)c1)=O)CC1CC1 N1(C(c2n(CC)ccn2)=O)CCCCC(NC(=O)C=Cc2cncs2)C1 N1(C(C2C(C=CC)CN(C(=O)C3=CCCC3)C2)=O)CCCC2CN(C)CC12 c1(N(C(N2CCC(CCCC)CC2)=O)Cc2ccc(C)cc2)ccc(C)cc1 c1(-n2c(C3CCCCN3)nc(CCCCC)n2)ccc(C(C)OC(C)=O)c(C)c1 c1(C(CNC(=O)NC(c2scc(C(=O)OCC)n2)C)(F)F)c(F)cccc1F c1(OCC(N2CC(C(C)NC(c3ccccc3)=O)C2)=O)cc(Cl)ccc1Cl S(=O)(=O)(c1ccc(Br)cc1NCC1(S(C)(=O)=O)CCC1)NCC(=C)c1ccccc1 C1(OC)CN(C(c2cn(C)cn2)=O)CCC1NC(c1coc(SC)c1)=O CCC(C(=O)N1CCCC1C(=O)N(CCCF)CC1CC1)NC(N)=O Cc1csc2c(C(=O)N(CCCNC(C3CC3C(F)(F)F)=O)C)ncnc12 C1(C(N(CCC(F)(F)F)C(C)C)=O)CCNCCC1C C12(C(N(C)Cc3ccccc3O)=O)COCC1CN(C(C1CCC(F)(F)C1)=O)C2 C1(CC)(NC(=O)CC(CC)SC)CCN(C(=O)Cc2ccccc2F)CC1 C1(C(N(C)CC2(NC(c3ccoc3C(F)(F)F)=O)CC2)=O)CC2C=CC1CC2 C(=O)(C(C)CCC(C)(C)C)NC1C2CN(C(CCOCC#C)=O)C(CC2)C1 CCS(=O)CC(=O)N1CC(F)CC1CC(=O)NCC(F)C1CCC1 c1(C(N2CC(O)CC2CNC(C2COCC2C(F)(F)F)=O)=O)c(F)cccc1F c1(OC)ccoc1CNC1CC1C(=O)NCc1cnc(C)s1 N1(C(CCC=CCC=C)=O)CCN(C(C2(CF)CC2)=O)CC1CC(=O)NC C1(C(=O)NCCCCC#C)CCC(C)(C)N(C(=O)C(C)CO)C1 c1(OC)c(C(=O)NCCCCC(C)NC(C2(C(N)=O)CCC2)=O)nc(O)nc1O C1(NC(C(F)=C(C)C)=O)CN(C(c2ccoc2C(C)C)=O)CCC1F C12(C(=O)NC3CCC(CNC(C4(O)CCC4)=O)CC3)CCOC1CS(=O)(=O)C2 N1(C(C(C)OC2CCCC2)=O)CCC(CCNC(=O)Cn2ccnn2)C1 S(=O)(=O)(c1ccc(OCCCC2(C)CC2)cc1)NC.N12CC(OC)(C1)CC2=O Cc1nn(CC(=O)NCCC(C)NC(C2(c3ccco3)CC2)=O)nc1OC(C)C c1(C(=O)NC(CC)CNC(=O)CCc2ccnc(Br)c2)cnc2n1CCC2 O=C(CC(C(F)(F)F)N1CCOCC1)N1CC(CNC(=O)C(Cl)=CCl)C2(CC2)C1 C1(NC(C2CCC3CC3CC2)=O)CCN(C(=O)CSC2CC2)C12CCC2 C1(C(=O)OC(C)(C)C)CCN(C2CCC(Br)CC2)C2CCCCC12 c1(C(N(CC#C)C)=O)ccc2c(n1)CN(C(=O)CC1CC=CCC1)CC2 C1(CNC(C(C)NC(C)=O)=O)CCN(C(=O)Cc2ccon2)C(C)C1 N(C(=NCC(C)C)NCc1ccc(N2CCOCC2)nc1)C1CC(CC)OCC1 N1(C(C(CCC)OC)=O)CCC2CN(C(c3cnn(CC4CCC4)c3)=O)C2C1 Cc1c(C(N2CCOC(CNC(C3(C)CCCCCC3)=O)C2)=O)cc(N)cc1O C=C1CCC1(C(=O)NC(=O)Cc1cccs1)C(N(CCC(=O)OC)C)=O N1(C(CCSCCCC)=O)CCC(C)(C(=O)NCC2CCCOCC2)CC1 C(=O)(C(F)C(C)CNC(C1C2CCCC12)=O)NC1CCC(OC)C1 N1(C(C2C(C)C2(F)F)=O)CC(CNC(c2cc(C(F)(F)F)ncn2)=O)CC1(C)C N1(C(c2cn(CCC)nc2)=O)CCCC(C2(NC(=O)CSC)CC2)C1 C1(C(N2CCC(CCN(C(C(C)C(C)(F)F)=O)C)CC2)=O)Cc2ccccc2C1 C=CC1CN(C(=O)CC2C=CS(=O)(=O)C2)CC1NC(C1C=CC=CC=C1)=O c1(C(=O)NCC2(C)CCCN2C(=O)C2=CS(=O)CCC2)nccc2c1NCCC2 C1(OC)CC(NC(=O)C(CCSC)NC(C)=O)CN(C(C2(C)CC(C)=NO2)=O)C1 C(=O)(C(O)CC(F)(F)F)NC(C(C)C)CC(=O)NC(CCO)C1CCCC1 N1(CC(=O)NCCN(C(=O)C(c2ccc(F)c(F)c2)O)C)CCP(C)(=O)CC1 c1(C(=O)Nc2cnc(C(F)(F)F)cn2)ccc(I)c(I)c1 C1(C(C)NC(=O)C=CC=C(Cl)Cl)CCN(C(N)=O)C1.c12cn(nn1)CCNC2=O Cc1nc(CCC(=O)NC2CC(CNC(C3(CC(C)C)CC3)=O)C2)oc1C N1(C(CN2CC(C)(OC)C2)=O)CC(CNC(C2(F)CC=CCC2)=O)C(C)C1 c1(C(=O)NCC2(NC(CCCCC(N)=O)=O)CC2)ccc2nnn(O)c2c1 C1(CC(=O)N(C(CC)C2CC2)C)CCCC(N(C(c2ncn(C)n2)=O)CC)C1 c1(OC)nc(C(N2CCCC2CN(C(=O)C(F)=CCCF)C2CC2)=O)cc(O)n1 C(C(=O)N1CCC1CC(=O)N(C(C)C(C)C)C)(C(C)C)OC(C)=O CC(C)C(=O)NC(C(=O)NC1CC(Cn2cccn2)C1)C1CCCC1 C#CC12CCC(C(=O)NCC3(CCNC(=O)C(CC=C)C(C)C)CC3)(CC1)CC2 c1(OC)ccc(OC)c(CC(N2CCC(CNC(=O)CN(C)C(N)=O)C2)=O)c1 Cc1ccc(C(=O)NC2CC(CNC(C3CC3(F)F)=O)C2)cc1N CC1(C)CCCN(C(=O)C(F)C2CCCC2)C1C(=O)NCC1CC(F)(F)C1 c1(CNCC2(CC=C)CC2(F)F)cc(OC)c(-c2nn[nH]n2)cc1F CCC(C#N)(CC)C(=O)NC1CCN(C(=O)Cc2nc(C3CC3)nn2C)CC1C C1(C(=O)OC(C=Cc2c(SC(C)(C)C)[nH]cn2)=O)CCCN(Cc2nnn(C)n2)C1 c1(N2CC(C)C(NC(c3cccc(=O)n3O)=O)C2)ncc2ccsc2n1 CCC(C)C(O)CC(=O)NC(Cn1cccn1)C(=O)NC1CC(O)C1 N1(C(c2c(CC)noc2)=O)CCCCC1C1CCN(C(C2(P(C)(C)=O)CC2)=O)C1 C(C(O)C(=O)NC1(CNC(=O)CCc2cnc(C3CC3)o2)CC1)SC N1(C(C(CC)(C)O)=O)CCCC(F)(CNC(=O)CC2COC3CC2C3)CC1 C(=O)(CC1=CCOCC1)NC(C)C(N1CCC(C)(F)C1)=O c1(CN2C(C(=O)Nc3cnncc3Cl)C=CC2)cnc(Cl)nc1Cl c1(N2CCC(C)(CC)C2)ncc(S(=O)(=O)NC(C2CCCCC2)CO)cc1Cl C1(CC=C)CCCN(C(CCC2CCCC2)C(=O)NCC2CCCO2)C1 CCCCC(C)NC(C1(NC(=O)CC2(O)CCCC2)CC(F)C1)=O c12cccc(c1)C2.C1(CCCC)(C(=O)NC2CC2NC(=O)C=CCF)CCCC1 N1(C(C=C(C)C(F)F)=O)CCC(C)(C)C(CNC(=O)CC2CCOCC2)C1 c1(C(N2CC(CCCCNC(Cc3cc(C)nn3C)=O)C2)=O)ccc(C)c(Br)c1 C#CCCN=C(NCC)N1CCC(S(C)(=O)=O)(C(=O)NC2CCCC(F)C2)CC1 N1(C(CNC(c2cscn2)=O)=O)CC2CC1C2NC(C1CC1c1ccsc1)=O C(=O)(CCCC(C)(C)C)N(CCN(C(=O)CC1CC2CC2C1)C)CCOCCO N1(C(c2ccnc(C)n2)=O)CCC2CCC(C1)N2C(C12CC(C)(C1)OC2(C)C)=O c1(NC(C2C(NC(C(c3ccccc3F)C)=O)CCCC2)=O)cc(F)c(C)cc1Br n1(CC(=O)NCC(C)CNC(C2COC(=O)C2)=O)ccc(=O)c([N+](=O)[O-])c1 c1(CN(C(c2ccccc2OC#N)C)C)ccncc1Cl C1(C(=O)NC(C)Cc2cn[nH]c2)C(C)CCN1C(=O)CC(=O)OC(C)(C)C N1(C(CCCN(C)C)=O)CC2C(CC(=O)Nc3cncc(Br)c3)C2C1 N1(C(C2N(C(C(C)CC3CCC3)=O)CSC2)=O)CC(CO)C(O)C1.n12cc(nn1)C2 c1(OC)ccc(C(=O)NC2CN(c3cc(C(C)(C)C)ncn3)CC2(C)C)c(F)c1 c1(OC)ccc(S(=O)(=O)NCCCC(=O)N(C)C)cc1C(=O)OC(=O)CO Cc1ccncc1C(N1CCCC1C(N1CCC(c2ccccc2)C1)=O)=O.CCO CCCCC(O)CC(=O)N(CCNC(=O)CCc1cc(C(C)=O)c(C)o1)CC c12cccc(c1)N2.c1(C(C)(C)C)cc(C(=O)NCC2(C(=O)N)CC2)n[nH]1.C1(C)CC1 c1(C(N2CCCC(NC(=O)C(F)(F)CC3CCCO3)C2)=O)coc2c1COC2 Cc1ccc(C(=O)NCC2COCC2NC(=O)C(C)(C)C(C)C)cc1C Clc1ccc(C2(c3ccncc3)CC2)cc1.C1(c2nc(C)on2)CC2CC2C1 c1(CCC)cccc(C(N2CCCC(N(C(=O)CC3CC3(C)C)CCF)C2)=O)c1 c1(C(N(C2CC(NC(=O)CC3CCCCC3O)C2)C)=O)cc(F)cc(F)c1O CC(C)CC(CNC(=O)CCC(C)(C)C)C(=O)N1CC(C)(C)CCC1CO C(=O)(C#CC1CC1)NCC(CN(C(CC(C)NC(=O)OCCO)=O)C)O.C(C)(C)(C)O C12CCCN(C1)C(=O)CN2S(C)(=O)=O.C1(C(=O)OC)CCCCN1CC(F)F C(=O)(CC(C)(C)n1ccnn1)N1C(CNC(C2N(CCC)CCC2)=O)CC1 Cc1ccn2c(C(=O)NCC(C(C)(C)C)NC(=O)CC3CC3C(F)(F)F)cnc2c1 c1(C(=O)NCC2CCCN(C(COC(CC)C)=O)C2)cc(O)ccc1C C(=O)(C1=NN(CCO)C(=O)CC1)N1C(C)(COC)CC(NC(=O)C2=NOCC2)C1 C=CC1(CC(N2CCOC(CCO)C2)=O)CN(C(=O)C(=Cc2ccco2)C)C1 C(=O)(C(C)CC(N)=O)N1CCC(C(N(CCC#C)CC)=O)CC1 Cc1cc(CC(C(=O)O)NC(=O)C(=O)NCC2(CCO)CCCC2)cc(C)c1 c1(OC)cc(C#N)ccc1CN1CCCC(C(N2CCCC(O)C2C)=O)CC1 c1(NC(=O)OC(C)(C)C)cnc(F)cc1NCC(=O)NC(c1ccc(Br)cc1)C CC1(CC(=O)NC(CO)CCC2CC2)CCN(C(C2CC(=O)C2)=O)C1 C12(CNC(c3cccc(COC)c3)=O)CCC1CCN2C(c1c(C)cnn1C)=O N1(C(c2c(=N)[nH][nH]c2)=O)CCC(NC(c2cc3n(n2)CCO3)=O)C12CC2 CC(C)C(C#N)C(=O)NC1(CC(N2C(C)CC2(C)C)=O)CCCCC1 C(=O)(NNc1cccc(F)c1Cl)C1CN(C(=O)OC(C)(C)C)C(C)(C)CC1 c1(C(N2CCN(C(C(C)(C)CO)=O)CC2CF)=O)cc2ccc(Cl)cc2c(O)n1 CC1=NN(C)C(=O)C1CC(=O)NC1COCCN(C(=O)CCCCOC(C)C)C1 N1(C(c2cc(C#C)c(C)nc2)=O)CCC(N=c2[nH]ccn3nnnc23)C(C)C1 CC1(O)CCC(NC(c2cc(CCNC(C3CC3(F)F)=O)on2)=O)CC1 Cc1ccc(NC(C2(NC(=O)CCCC#N)CCCC2C)=O)cc1C Cc1conc1CC(=O)NCCC1CN(C(=O)CCN(c2ccncc2)C)C1 c1(N(C)CC2CCN(C(C(CCC)N(C)C)=O)C2)nc(Cl)nc2c1ncn2C C1(C(=O)NCC2(C(N(C3CCCC3)C)=O)CC=CC2)CCOC1(C)C C1(C(=O)NCC2(O)CN(C(c3c(SC)n(C)nc3)=O)C2)C2CCC3C(C2)CC13 C1(CNC(=O)Cn2cc(Br)cn2)CC(NC(=O)CCF)C(O)C1 N1(C(c2c(C)non2)=O)CC(O)CCC1C(N1CC(C(C)C)C1)=O C(=O)(C(F)C(=O)NCC(C)N(C(=O)C(c1c(C)noc1C)C)C)OCC C1(CNC(C2N(C)CCC2)=O)CCCCN1C(c1cc(C(F)(F)F)sn1)=O C=C=CCCC(=O)NC(CNC(=O)CCc1cn(C)nn1)C(C)C N1(C(c2cc(OC)n[nH]2)=O)CCC(CF)(NC(c2ccn(CC(C)C)n2)=O)C1 C1(NC(C(C)CF)=O)C2CC3CN(C(=O)Cn4ncn(C)c4=O)C1C3C2 c1(C(=O)NC2CC(C)N(C(=O)CN3CCCC3)CC2)nccc2[nH]ccc12 CC1CN(C)CC(C(=O)NC23COC(CNC(=O)CSCC4CCCO4)(C2)C3)O1 C=CCCCCCCCC(=O)NCC(CO)NC(=O)C=Cc1ccc(C)cc1 N1(C(C=CCCC=C(C)C)=O)CCC(O)(CCNC(C2(F)CCOCC2)=O)C1 CC(C)CC(C(=O)NC1CC(F)CN(C(c2cccc(F)c2C2CC2)=O)C1)N(C)C c1(C(=O)NCC(C2N(C(c3scc(C)c3)=O)CCC2)(C)C)ccnc(C(F)F)c1 O=S(=O)(c1cc(CNC2CCCCC2)co1)N1CCCC1.c12noc(n1)C2 C(CN=c1nc(N2CC=C(C)CC2)c2ccc(C)cc2[nH]1)C1(C)N=C(C)SC1 N1(C(C2OCCN(C(C3OCCN(CC)C3)=O)C2)=O)CCc2oc(C)nc2C1 C1(C(N2CCN(C(CC)C)CC2)=O)CC2CC1CC2NC(=O)CCc1cnc[nH]1 c1(Cc2nc(C(N3CCC(C4CC4)C3)C(=O)NC(C)C)sc2)ccc(F)cc1F N1(C(C=CCOC)=O)CCC2(CC1)CC(NC(c1cc(C)sc1C)=O)CO2 c1(C(=O)NC(Cc2ccc(CNC(C(CC)C)=O)cc2)C)cc2sccc2n1C CC1(C(=O)NC2CCN(CCCNC(C3CC4CCC3O4)=O)C2)CCCCO1 CC(CN=c1[nH]c(N2CC(F)(F)C(F)(F)C2)nc2c1CCC2)c1ccccc1Br c1(OC)ccc(C)c(C(N2CCC(C)(C(N3CCC(n4ccnc4)C3)=O)C2)=O)c1 N1(C(CC2(COC)CC2)=O)C2CCCC1CN(C(C1CCOC(C(C)C)C1)=O)C2 C1(NC(CCOC(C)=O)=O)C=CCC(C(=O)N(CCN(C)C)C2CC2)C1 C12(C(=O)NCCC(=C)C)CC(CO)(CN1C(=O)C(C)NC(=O)C1CC1)C2 CC(N=c1nc(N(C)Cc2c(Cl)cccc2Cl)c2c(ncn2C)[nH]1)C(F)F C=C(C)C(C)(O)C(=O)N(CCS(=O)(=O)CCCn1cc(C2CCCCO2)nn1)C CCCC(CNC(c1ccc(F)cn1)=O)C(=O)NCC(C)(O)CCO Cc1cn(C)nc1C(=O)NC(CNC(c1cnc(Cl)[nH]1)=O)C(C)(C)C N1(C(CCCc2n[nH]c(=N)s2)=O)CCCN(C(=O)CCNC(N)=O)CC1 c1(OC)ncc(C(N2CCC(C)C2CNC(=O)CNC(=O)C(F)(F)F)=O)nc1C N1(C(c2ccc(C(C)O)cc2)=O)CC(NC(=O)CO)CC(F)C1 C(N=c1[nH]c(=NCCc2nc(Cl)ccc2Cl)c2[nH]ccc2[nH]1)C1N(CC)CC1 CC1(CC(=O)NCC2(NC(c3ncoc3C3CC3)=O)CCCC2)CCCCC1 C(=O)(C(F)C(C)C(F)(F)F)NC1CN(C(c2ccc(NC(C)=O)c(Cl)c2)=O)C1 N1(C(C2COC(=O)O2)=O)CCCN(C(c2cc3ccccc3[nH]2)=O)C(CO)C1 N1(CC(=O)NC2(C)CC(NC(C(CSC)c3ccccc3)=O)C2)CCCNC1=O CC(C)CC(O)CC(=O)N1CCCN(C(c2ccc(-c3ccoc3)cc2)=O)CC1 C(N=c1[nH]cnc2ccc(O)cc12)C1(C)CCN(C(C2CC(CC)OCC2)=O)C1 CS(=O)CCC(=O)N1CCOCC1CNC(=O)C(c1ccccc1F)(F)F Cc1cc(C(=O)NCC2CCN(C(=O)C(C)Cc3ccc(O)cc3)C2)sc1C N1(CC(=O)NCCCCCCN(C)C(c2ccc(F)cc2)=O)CCCCCC1=O c1(C(=O)NCCC(CNC(=O)Cn2cnnc2O)OC)cnn(C)c(=O)c1 c1(C(=O)NCC(O)CNC(C2CCCC2O)=O)c(O)cc(F)cc1F C1(C(N(CCN2CCCC2)Cc2cn(C(C)C(=O)O)nn2)=O)CC2CCC1C2 c1(N(C2CNCCOC2)C(=O)OC(C)(C)C)ccnc(N)n1.CCO N1(C(C2C(CC(C)C)C2)=O)CCC(F)CC1C(=O)NC(C)CC1(O)CCC1 C12CCCN(CC1)c1ccc(cn1)NC2=O.C1(N(CC)CC)CCC1 C#CC1(C(=O)NCCC(C(=O)NC2CCCC2C)OC)CC(=O)C1 C1(CNC(C(F)=C(C)C)=O)CN(C(=O)C=C(C)I)CCC12CCOCC2 c1(C(=O)NC2CCC(CNC(C3CCC(CC)O3)=O)C2)cc(Cl)ncc1F c1(C(N2CCN(C)CC2CNC(c2cc(C#N)c[nH]2)=O)=O)n[nH]c2ccccc12 C1(CNC(CCC(C)SC)=O)CCN(C(c2c(Cl)cncc2Cl)=O)CC1C C(=O)(C(CO)NC(c1ccc(F)s1)=O)N(CC#C)CC1CCOC1 c1(C(C(F)(F)F)NC(C2CCNC2)CC)cc(OC(C)C)ccc1O c1(C(=O)NC(CC)CCC(=O)N2CCSCC2C2CC2)cc2ccccc2o1 C1(CCNC(c2c(C)nc(CO)s2)=O)C(C)CCCN1C(=O)CCNC(=O)CO c1(CC(=O)N(CCOCCCNC(CC(=O)NCC)=O)C)c[nH]c2cccnc12 c1(CC)c[nH]c(C(=O)NCCC2(CNC(c3cncn3C)=O)CC2)n1 C1(C(=O)NC(C)CN(C)C(C2CCCC3CCCN23)=O)CCS(=O)(=O)C1(C)C c1(C(=O)NCC(CC(C)C)NC(c2c(C)cccc2)=O)nc(C)c(N)cc1C N1(C(C2C(C)CC2C)=O)CCC2(C1)CN(C(c1ccc3nc[nH]c3n1)=O)C2 CCCCCC(C(=O)NC1(C)CC1)N1CCC(C)S(=O)(=O)CC1 C1(N(C(C(C)=CC2CC2)=O)C)CN(C(=O)Cc2ccn(-c3ccco3)n2)CC1F Cc1cc(CO)oc1C(=O)NCC1CCN(C(=O)Cc2csc(NC=O)n2)CC1 CONC(=O)C(=O)NCc1cccc(C(=O)N(C2CCCC2)C2CC2)n1 c1(CN2C(C)(C(=O)Nc3ccc(-c4ccccc4)s3)CC2)ccc(F)c(C#N)c1 c1(C(=O)NCC(CNC(c2nc(C)c(C)s2)=O)F)noc2c1CC(C)CC2 N1(c2nnc(CC(C(C)C)(C)O)n2CCC2CC2)CCN2CCCCC1C2 CCC(C)(O)C(=O)NC1CC(NC(c2cncn2-c2ccc(Cl)cc2)=O)C1 N1(C(CNS(CC)(=O)=O)=O)CC2CN(C(C3(F)CCOC3)=O)CCC12 N1(C(CC(=C)Br)=O)CC2CCC(C1)N2C(=O)CN(C)CNC(=O)NC(C)(C)C c1(C(N2CC(NC(CS(CC)(=O)=O)=O)C(SC)C2)=O)cnc(Cl)c(F)c1N C1(CCNC(COCCCC)=O)(CNC(=O)C(C)NS(=O)(=O)CC)CCC1 C1(C(=O)OCC)CC1C(=O)N(CC(C)O)CC1CC1 c1(CC)nn(C)c(N2CCC(CNC(c3cc(C)sc3C)=O)C2)c1[N+](=O)[O-] c1(C(N(CC(C)NC(C(COC)N(C)C)=O)C)=O)cncc(F)c1Cl c1(CC)ccc(C(=O)NC2(CNC(C3CC(O)CN3C)=O)CCCC2)nc1 C(C)(C)(CCCNC(=O)C(n1cc(C2CCCN(C)C2)nn1)C)N(CC)CC C1(C(=O)OC)(CCl)CCCN(Cc2ccc(F)c(Cl)c2)C1 S(=O)(=O)(c1cnc(NC2CCC(CC(C)C)C2)cc1C)NCc1ccc(C)cn1 C1(CC(=O)NC(C2CCCC2N)C)(N(S(C)(=O)=O)C)CCOC1 N1(CC(c2nccs2)=O)C2CCC1(c1cn(-c3ccccc3Cl)nn1)CC2 CC1CN(C(c2ccc(F)cc2)=O)CC1CNC(C1COCCO1)=O N1(C(C(CCC)OC)=O)CCC2C(C(=O)N(C)CCC3CCCC3)C2C1 N1(C(C(CC)OCC)=O)CCN(C(C2CCC(N=[N+]=[N-])C2)=O)CCC1C CC(CCNC(=O)C(O)CNC(=O)C(N1CCOCC1)C)CCO c1(C(N2CC(C)C(NC(=O)C=CCN(C)C)CC2)=O)ccc(F)c(C#N)c1 C1(C)(CNC(Cc2cc(C)on2)=O)CCC(NC(=O)CCc2ncc(C)[nH]2)C1 N1(C(C=CCOC)=O)CCCC(CNC(C2(C(N3CCN(C)CC3)=O)CC2)=O)C1 C1(C(N(CC(C)CNC(=O)CC2CC2)C)=O)CSC(c2ccccc2)=N1 Cc1ccc2ncccc2c1NC(N1CCC(c2nncs2)C1)=O C1(CC(=O)OC)CCC2(CC1)CCN(C(=O)NC1CCCCC1N1CCCC1)C2 N1(C(c2c(OCC)nccc2)=O)CC2(CCC2CNC(=O)Cc2conc2C)C1 c1(C(N2C(C3(NC(CC(C)c4cccnc4)=O)CC3)CCC2)=O)ccc[n+]([O-])c1 C1(N(C)C)CN(CCN2CCCCC2NS(=O)(=O)CCc2ccccc2)C(C)(C)C1 C1(CNC(C(C)NC(C)=O)=O)CN(CC=CCl)CCC1C c1(-c2n(CCC=C)nc(C3CCC3)n2)ccc2[nH]nc(Br)c2n1 Cc1cccc(OC(C)C(=O)NCC2CC2NC(c2cccc(C3CC3)c2)=O)c1 Cn1nc(C(=O)N(CC(=O)NCC23CCN(CC2)CC3)C2CC2)cc1[N+](=O)[O-] C1(CC(=O)NC2C(NC(c3c(CC)nn(C)c3)=O)COC2)SC2=NCCN2C1=O C1(NC(c2n(CC#C)cnn2)=O)CC(O)CN(C(C2(C)CCCCC2)=O)C1 Cc1c(Cl)cccc1S(=O)(=O)N1CC2CC1C2C(=O)Nc1cn[nH]c1 CC(C)CCC(C)N(C)C(C1OCCC1CNC(C1(F)CCOC1)=O)=O N1(C(CC(CC)OC)=O)CCCC(COC)CC1.C12(CCCC1)C(=O)NC2 c1(C(=O)NCC2CN(C(CCCC(C)=O)=O)C2)cnc2[nH]c(O)nc2c1 N1(C(C(C2CC2)OC)=O)CCC(C2CCN(C(=O)C(C)(F)F)C2)C1 N1(C(C(CC)(C)COC)=O)CCOC2(C1)CN(C(=O)C(C)NC(N)=O)C2 c1(C=O)cc(F)cc2cnccc12.C12(C(=O)NCCN)CC3CC1C2C3O N1(C(CC2(C#N)CCC2)=O)CC2(CCC(CNC(C3COCCO3)=O)O2)C1 CC(C(=O)NC1CC(CNC(=O)C=CC(=O)N(C)C)CC1O)C(F)(F)F c1(NCC(c2csc(Cl)c2)N(C)C)ccc(CCCN)cc1 C1(C(=O)NC(C2CC(NC(C=C(CCC)C)=O)C2)C)COCC1(C)C Cc1nn(CC(=O)NCCNC(C2(c3ccc(O)cc3)CC2)=O)cc1Br N1(C(C(n2ccc(C)n2)C)=O)CCCC(O)(CN(C)C(c2ncccc2F)=O)C1 C(=O)(C1=Cc2ccccc2OC1)NC1CCN(C(C(CCCC)CCCC)=O)C1 c1(CCNC(CC2(CC)CC2)=O)ocnc1CNC(C1CC(C2CC2)C1)=O N1(C(C(=O)NCCCF)CC2CCCCO2)CC2COCC2C1 c1(C(N2CCCN(C(CSCCOC)=O)C(CO)C2)=O)c[nH]c2cccc(F)c12 N1(C(C2C(NC(Cc3c(C)n[nH]c3)=O)C2(C)C)=O)CC2OCCN(C)C2C1 N1(Cc2c(OC)cccc2)CCC(NC(=O)Cc2ccncc2)C(F)C1 C(C(C)C(F)C(=O)NCCN(C)C)NC(c1cn(C(C)C)nn1)=O c1(C(=O)NCC=CC)cnc(CNC(c2snnc2C)=O)nc1 c1(C(=O)NC(CCC)CCCNC(C2CCC2OC)=O)ccc(F)c(C)c1F c1(C(N2C(C(=O)Nc3cccc(COC)c3)CC2)=O)cc(O)ccc1C C(=O)(CCC(=O)NN(C)C)N1CC(OC)C(NC(=O)CCCn2cccc2)C1 c1(C(=O)NC(CNC(C2(F)C(C)(C)C2(C)C)=O)C2CC2)cc(C#N)c(N)cc1O N1(C(C(CC=C)CC(C)C)=O)CC23CCCCC2(C1)CN(C(=O)C(C)OC)C3 Cc1nnc(O)c(C(N2CCC(CO)(NC(=O)CC3CC3(C)C)CC2)=O)c1C c1(N(C2CCN(C(C3CC3[N+](=O)[O-])=O)CC2)CC2CC2)ncc(Br)c(O)n1 C1(C(=O)NC2C=CC(CC(=O)NC(c3cccnc3C)C)C2)C2CCC(C2)C1C N1(C(c2nc(CC)oc2)=O)CCC(C)C(CNC(=O)CSc2ccc(Cl)cc2)C1 c1(CC(=O)Nc2cc(NC(N)=O)ncc2)cccc(Br)c1F c1(CNC(CC(C)n2cccc2)=O)cc(C(=O)NC(c2cccnc2)C)ccn1 Cc1coc(C=CC(N2CCCC(N(C(=O)Cn3cccn3)CCF)C2)=O)n1 c1(NC(C2(COC)CC2)=O)nnnn1C(C)(C)C.C1(NCCC(C2CC2)N)(CO)CC1.CO c1(C(N2C3CN(C(C(C(C)C)(O)C)=O)C(CC3)C2)=O)cnc(O)c2cncn12 CC1(C)CC(NC(=O)COC2CCSC2)CN(C(C2CC3(C2)CC(F)(F)C3)=O)C1 C#CC(CNC(=O)C(F)C1CC(NC(=O)Cc2ccc[nH]2)C1)C(C)C C1(F)(CNC(CCC#C)=O)CCN(C(c2ccc(Cl)nc2C(F)F)=O)CC1 C1(NC(c2c(OC)cc(Cl)cc2)=O)CN(C(c2n[nH]c(=N)[nH]2)=O)C2CCCCC12 c1(OC)cc(C(N2CC(CNC(C3CCC3C)=O)C2)=O)c(C)cc1O N1(CC(=O)NC2C3CN(C(C(C)OCC)=O)CC32)C(=O)c2ccc(Br)cc2C1=O N1(CCOC(C2CC3CCC(C2)O3)=O)CCC2(CC1)SCCS2 c1(N(C(C(=O)NC(CC)(C)C)CC2C=CCC2)CCOC)ccc(OC)cc1 c1(OC)ccc(CC(N2CC(CNC(=O)CCC(OC)OC)C(O)C2)=O)nc1 c1(C(N(CC(CN(C(CC(CC)(F)F)=O)C)O)C)=O)ccc(O)cc1[N+](=O)[O-] C1(CNC(=O)OC(C)(C)C)CCn2nnnc2C1.c12cc(cc[n+]1[O-])OC2=O C(C)(CCCCO)NC(CONC(C1CC(OC)(OC)C1)=O)=O c1(NCCCC)ccccc1C(=O)NC1CCN(C(=O)Cc2cn[nH]c2)CC1 N1(C(c2c(C)n[nH]c2)=O)CCOCC(CNC(=O)CCc2cccc(Cl)c2)C1 C(=O)(CC(C)C(F)F)NCC=CCNC(c1occ(C)c1C)=O N1(CC(=O)NC2C(NC(Cc3c(C)n[nH]c3)=O)CC2)C(=O)NC(C)(C2CC2)C1=O CC(C)(C)CC(c1ccccc1)N(CC(=O)N(O)Cc1ccccc1Cl)C1CC1 c1(C(CNC2CC3CN(C(c4ccc(C)o4)=O)C2C3)=O)ccc2occc2c1 c1(C(N2CCC(OC)(CNC(=O)CCc3ncccn3)C2)=O)c[nH]cc(C)c1=O c1(NC(=O)NC)ccccc1CC(=O)NCC1CCC1c1nnc(C(F)(F)F)s1 c1(OCC)ccc(-c2cnc(N3CCC(C(=O)NCC(C)C)CC3)s2)cc1 C1(CC(=O)NCC2C(NC(C(C)n3cccn3)=O)CCCC2)CN2CCC1CC2 N1(C(CC(C=C)CC)=O)CCCCC2(CCN(C(=O)CC(C)(C)C)C2)C1 C1(C(=O)Nc2cccc(NC(N)=O)c2)CN(CC(O)CCC2CC2)CCC1O Cc1csc(C(=O)NCc2noc(-c3ccc(Br)cc3)n2)c1C N1(C(c2c(C)ncs2)=O)CCC(C(N2CC3C(C2)C3(C)C)=O)C(O)C1 Cc1cc(C(N2CCCC2(C)CNC(=O)CN2CCCC2CO)=O)ncc1N C1(C(=O)NC(c2cccc(C)n2)C)CCCCCCN1C(C1CCC2CC12)=O OC1CCN(S(=O)(=O)c2ccc(N3CCCC3)cc2)C12CCSC2 C1(C(=O)OC)CN(C(=O)NCc2cccc(OC3CC3)c2)C1(C)C C(=O)(C1=NOC(C)(C)C1)NCC#CC(=O)NC(CC(=O)OCC)C N1(C(=O)NCc2ccc(C3C(OC)CCO3)o2)CC(=O)NC(=O)C1C c1(C(N(C)CC2CCC(CNC(c3ccco3)=O)CC2)=O)cc2c[nH]cnc-2n1 C1(C(N(CC(C)O)CCNC(c2cncc(C)n2)=O)=O)CCCN2CCCCC12 C1(Nc2ccc(NC(=O)C3CC3)cc2F)C2CCC3(COC(=O)C13)O2 c1(C2C(C(C3CC3)NC(=O)NC(c3ncccn3)C)C2)ccccc1 Cn1cnc2c1CCCC2C(=O)N1CCC(C)(NC(c2cnc(C(F)F)s2)=O)C1 N1(C(Cn2c(C)nc(C)n2)=O)CC2CCCC1C2c1cn(-c2ccn(C)n2)nn1 C(=O)(C1OCC(C)(C)c2ccccc21)N1CC(C(C)C)C1 C#CC1(C(N2CCC(CCCC)C2)=O)CN(C(=O)CCCCC)C1 C1(CNC(=O)Cn2cnnn2)CC2(CCC2)CN1C(C1CCC(CCO)CC1)=O C(CN=C(NCC(c1ccc(F)cc1)(F)F)NC(c1ccc(Br)cc1)C)SC c1(C(=O)NC2CN(C(C3CCC(C)CC3)=O)C(C)C2)cc(N)c(O)c(F)c1 c1(CN2CCC(N3CCOCC3)C2)ccc(CBr)cc1.N12CCC(O)(C1)C2=O C(=O)(CC(CC(C)C)NC(=O)C(O)CN(C)C)NC(C1CCCC1)CC C12(C(=O)NC(CNC(c3c(C)csc3)=O)C)COC(CO)(C1)C2 c1(OC)nc(C)ncc1C(=O)NC1CC(CO)N(C(C2CCC(=O)N2C)=O)C1 Cn1cc2c(CN3CCCC(C(=O)Nc4c[nH]c5ncccc45)C3)cccc2n1 C(CC(=O)N1CCCCC1)(C(F)(F)F)NC(c1c(=NC(CC)C)[nH][nH]c1)=O C(C(CC(C)C)C(=O)N1C(CC)CCC1C)NC(C(CC)N(C)C)=O c1(C(N2CC(C)OCC2)=O)c[nH]c2ccc(-c3cccc(C#N)c3)cc12 Cc1cnc(C(N2CCC2CNC(=O)C=CC2CCCC2)=O)c(F)c1 N1(C(C(CC=C)C(=C)C)=O)CCCC2(CCCN(Cc3ccc(OC)cc3)C2)C1 C12(CCNC(CCNC(N)=O)=O)CCC(C1)N(C(=O)CN1CCCCCC1)C2 N1(C(C=CC)=O)CCC(NC(=O)Cc2ccnn2C(C)C)C(CO)C1 Cc1cc(=NCC(C)(C(C)C)NC(=O)COCc2cccnc2)[nH]c(Cl)n1 c1(C(N(CC(O)CN(C)C(C2C3CCN2CC3)=O)C)=O)cc2cc[nH]c(=O)c2s1 CC1CCN(C(=O)CCC2CC(NC(=O)C(C)(C)C#N)C2)CCS1 C=CCCC(C(=O)OC)NC(C1(C)CN(C(c2ccnnc2)=O)C1)=O N1(C(c2c(C)cns2)=O)CC2(CCCC2NC(c2ccc3ncsc3c2)=O)C1 C(N=c1nc2sccc2c(NCc2ccc3c(n2)OCCO3)[nH]1)c1n(CC)ccn1 c1(C(=O)NCc2scc(C(N(C)Cc3cscn3)=O)c2)cn(C)nc1CO C1(NC(Cc2nc(C)sc2)=O)CC2CN(C(=O)C=C3CN4CCC3CC4)CC12 C(=O)(C#CCCCC1CCCC1)N1C(C2(NC(=O)C=CCNCCO)CC2)CCC1 c1(OC)ccc(C2CC2)c(C(N2CC3CC3(NC(c3csc(O)n3)=O)C2)=O)c1 c1(N(C)CC2CCCN(C(c3cccc(F)c3I)=O)C2)ncnc2c(F)cccc12 C(CC(=O)NC1CCOCC1(C)C)(C(C)OC)NC(COCCCC)=O CCCCC(O)C(=O)NC(CO)CCCCNC(=O)C=C(C)C1CC1 c1(C(=O)NC23CN(C(C4(COC)CCCO4)=O)C(CC2)C3)cnc(O)n(C)c1=O C(C)(C)(CCC(=O)NCC1(C)CCCN1C(c1nc(C(C)C)ncc1Cl)=O)OC C(=O)(CCC(F)(F)F)N1CCC(CNC(C(CC)Cc2ccccc2)=O)CC1 CCC(C)(F)C(=O)N(C)CC1CCCCN1C(=O)C1=COCC1 C1(NC(C2C(C)C2)=O)CN(C(=O)CCn2ccccc2=O)CCC1C(F)(F)F n1(CC(=O)NC2C(NC(c3cnc(C(C)O)s3)=O)CC2)cc2ccccc2n1 c1(-c2nc(CSCCNC(C)=O)on2)cccc(F)c1 N1(CCC(C2CCC2)N(C)C)CC(=O)N(CC(C)(C)C2CC2)C1=O C1(NC(C2(CC)CCCN(C(=O)CC3CCCN3C)C2)=O)CCCCC1N=[N+]=[N-] c1(C(=O)NCC2(CCNC(CCCOCC)=O)CC2)cc2n(n1)CCCC2 N1(C(C(F)OC)=O)CCC(C2(NC(c3ccc(CN(C)C)cc3)=O)CC2)C1 c1(C(=O)NCC(CC=C)NC(c2ccco2)=O)cc(C)c(CO)cn1 N1(C(C2C(Cl)(C(=O)OC)C2)=O)CCN(C(=O)CSc2n[nH]c(=N)s2)CC(C)(C)C1 Cc1ccc(C#N)cc1C(N1CC(N(C(=O)CN2CSCC2=O)C)C1)=O C(CCCCCC(=O)NCC1CC1CO)NC(CS(CC)(=O)=O)=O C1(NC(C2CCN(C)C2=O)=O)CCCCN(C(C2CCCCC2(C)C)=O)C1 C1(C(N(C2CC2(C)C)C)=O)CCC(=O)CC1(C)C N1(C(CS(=O)(=O)NCC)=O)CCC(NC(=O)CN2CCSCC2)C(C)(C)C1 N1(CC(=O)N(C2CCN(C(=O)COc3ccsc3Cl)C2)C)Cc2ccccc2C1 N#CCCCCC(=O)NC(C1CCCCC1)CNC(c1cc(N)ccc1Cl)=O c1(C(N2CCCC(N(C(CCSCC)=O)C)C2)=O)cnc2[nH]cc(C)c2c1 N1(C(C(=O)NC)=O)C(C(=O)NCC2(COC)CCCC2)CC1C c1(C(=O)NCCC2CCCN(C(c3c[nH]nc3C(F)F)=O)C2)c[nH]nc1[N+](=O)[O-] c1(C(=O)OCC)ccnc(SC2OCCC2CN2CCCC2COC)c1 N1(C(c2c(OC)cccc2)=O)CCOC2CN(Cc3c(Br)ccc(F)c3F)CC12 N1(C(CCC(=C)C)=O)CCN(C(c2ccc(-n3ccnc3)nc2)=O)CC12CC2 N1(Cc2cccc(C)c2)CCC(C)(NC(c2sc(-c3cccs3)nc2C)=O)CC1 CS(=O)(=O)c1ccsc1C(=O)NCC(O)CNC(c1cc(N)c(F)cn1)=O C1(NC(c2cccc(CC)c2)=O)(CO)CCN(C(c2cc(Cl)cnc2Cl)=O)CC1 N1(C(C(CNC(c2ccc(Cl)cc2)=O)N(C)C)=O)CCC(O)C(F)(F)C1 C1(CCNC(c2cc(-c3cnccn3)[nH]n2)=O)CN(C(C2CCSC2)=O)CCO1 N1(C(Cc2cn(CC)nn2)=O)CCC2(NC(=O)Nc3ccc(Cl)cc3)CCCC12 CC1CN(C(C2CCSC(C)C2)=O)CCN1Cc1cn(-c2ccccc2)nn1 c1(C(N(C)CC2(O)CN(C(=O)C3=CC(C)(C)C3)C2)=O)cncn(C)c1=O N1(C(=O)CCc2cnccn2)CC2CCC(C1)N(Cc1ccc(Br)nc1)C2 C1(NC(CC(=O)N(C)C)=O)CCCC1(C)CN(C(=O)CNC(C1CCCC1)=O)C c1(C(N2CC(NC(c3c(CC)onc3)=O)C(C)C2)=O)c(F)ccc2nc[nH]c12 c1(C(=O)NC2(CO)CCN(C(C(C)n3cnnn3)=O)C2)cncc2ccsc12 C1(NC(CC(CCC)OC)=O)CCN(C(=O)COCC)CC12CC2 c1(C(=O)NCC2C(NC(CCCOC)=O)C2)cc(Br)c(Cl)cn1 N1(C(C2(C(C)C)CC2)=O)CCC(F)(F)C(CNC(=O)CC2CCC(F)(F)CC2)C1 CC(C)CCCC(C)C(=O)N(CCC(=O)NC1CN2CCCC1C2)CCO C(=O)(C(C(C)C)OC)N(C(CSC)C(=O)N1CCC(Nc2nnc(OC)s2)C1)C c1(OC)cc(CC(N2CCN(C(=O)C(O)CSC)C(C3CCC3)C2)=O)ccc1C CC1(C)CN(C(=O)C=CBr)CCN(C(c2c[nH]c3cc(F)ccc23)=O)C1 c1(C(N(CCCNC(C(C(CC)C)O)=O)CCO)=O)sc2nccn2c1C c1(C(=O)NC(CC)CN(C)C(c2cncn2C)=O)oc2cc(Cl)ccc2c1C CC(C)CC(C)CC(=O)N1CCC(C2CCCN2c2cc(C3CC3)ncn2)C1 CCCCC(=O)OCCOC.C1(CCc2ccccc2)CNC(=O)CNC(=O)N1 Cc1cc(CC(=O)N(C2CN(C(=O)CC3CCOC3=O)CC2(C)C)C)ccc1F c1(CC(C)C)ccccc1C(=O)NCCC1(O)CCN(C(=O)C(C)C(C)C)C1 c1(OC)ccc(C(N(C(=O)C2CC2)C(c2cnc(O)o2)c2ccccc2)=O)cc1 c1(CNCC2(C)CC(c3ccc(Cl)cc3)C2)cccc(C(F)(F)F)c1 C1(NC(c2ccc3c(c2)CC3)=O)CCC2CCN(C(c3ccccc3)=O)C1C2 N1(C(C(COC)OC)=O)CC2CCC(C1CO)N2C(c1ccc(F)cc1F)=O C(N=c1cc[nH]c(-c2ccc3nonc3c2)c1)c1n(C(=O)O)ncc1 C(=O)(C(CNC(=O)CC1COCCOC1)C(C)(C)C)NCc1cc(C)sc1C C(CC(C(=O)N1CCC(CCNC(=O)Cn2ccnn2)C1)NC(N)=O)SC C(C(C)C(=O)NCC1CCN1C(=O)CSc1cnn(C)c1)OC C1(C(=O)NCCCOCCNC(C2CC(C)(F)C2)=O)CC2(C1)CC2(F)F c1(CC)cc(C(N2CC(F)(CNC(C3(CC)CCNC3=O)=O)C2)=O)cc(F)c1 C1(C(=O)NC2CN(C(C)C)CC2C)CCN(C(=O)CC(C)(C)CN(C)C)C1(C)C c1(C(N2CCC(NC(=O)COC3CCCCC3)C(F)C2)=O)ccnc2[nH]nnc12 C(=O)(C(F)C(C)CNC(=O)C(=O)Nc1ccnc(-c2ccccc2)n1)OC c1(CC(C)CO)ccc(CC(=O)NCCN(C(=O)C(O)C2CC2)C2CC2)cc1 N1(C(C=CSC)=O)CC2(CCCC2NC(c2cccc(C(C)(C)C)n2)=O)C1 C(=O)(C1=NN(CC2CC2)C(=O)CC1)NCC1C(NC(C2(C)N(C)CCC2)=O)CC1 N1(C(C=CCC2(NC(C(CCC)C)=O)CCC2)=O)CCc2ccccc2C1 C(c1ccccc1)(C(F)(F)F)=CC(=O)N(CCCN(C)C(C1CC1(C)C)=O)C C#CC1CCN(C(c2cnc(Cl)s2)C(=O)NC2CCCCC2)CC1 C1(CNC(N2CCC(CCF)C2)=O)C2CN(c3nnc(C4(C)CC4)o3)CC12 Cc1cc(Cl)cc(C)c1C(=O)NCC12CC(NC(=O)C(C)CC(F)(F)F)(C1)C2 Cc1cc(CN(C(=O)C(CCF)NC(C2CS(=O)(=O)C2)=O)C)nn1C c1(C(N2CCC(N(C(c3ccc(F)s3)=O)CC)C2)=O)cc(OC)cc2c1CCC2 Cc1cc(C(=O)NNC(=O)C(C)(C)CF)c2cccc(O)c2n1 N1(C(n2cc(-c3cn(C)nc3)nn2)=O)CCN2CCCCC2C1.C12C(C1(F)F)C2 c1(C(=O)NCCC2(NC(CCCS(N)(=O)=O)=O)CC2)cc(=O)n2ccsc2n1 CC(C)CC(O)C(C)C(=O)NC(C(=O)NC1(C)CC(N(C)C)C1)C(C)C N1(Cc2onc(CCC)n2)CCC(NC(=O)CC2CCCCO2)C(O)C1 C1(CNC(C2(C)C(CC)CCC2)=O)CC(C)CN(C(c2ccc(OC)c(Cl)n2)=O)C1 C1(CNC(CCCC#C)=O)CCN(C(c2cc(Cl)c(C)c(Cl)c2)=O)CC1(F)F C1(NC(CNS(CC)(=O)=O)=O)CC12CCC(NC(c1c[nH]cc1C)=O)CC2 c1(C(N2C(CNC(C(C(=C)Cl)(C)C)=O)(COC)CCC2)=O)cc2cnccc2[nH]1 Cc1cccnc1C(=O)NCc1cc(C(=O)NCC(C)(O)C2CCC2)on1 c1(CC(=O)NC(CC)CNC(=O)Cc2ccc(Cl)s2)ccc(Cl)c2cccnc12 c1(NC(C2CC=C(C)CC2)=O)ccc2nc(Nc3c(C(=O)OC)n[nH]c3)sc2c1 Cc1ccc(F)cc1CC(=O)NC1CCN(C(C2CCOC(C)C2)=O)CC1 C(C(C)(C)CCO)NC(C(C1CCCCC1)NC(C(C)N1CCC1)=O)=O C(C)(CC(=O)NCC1CCC1C(=O)NCC1(O)CSC1)SC N1(C(C2C(CC)CCO2)=O)CCC(C2CCN(C(=O)COCCO)C2)C1 N1(C(CN(CC)CC)=O)CCC(CNC(c2cnc(NC(=O)C(F)(F)F)o2)=O)C1 N1(C(c2cc(OC)no2)=O)C2CCC1C(NC(=O)C(C)SCc1ccccc1)C2 C=C(C)C(CC(=O)N1CCN(C(c2cc(OC)ns2)=O)CC1C(C)C)OC C1(CNC(CCCC=C)=O)(OC)CCCN(C(C2CN(C(N)=O)C2)=O)C1 C(=O)(CCS(=O)(=O)CC(C)C)N1CCC(NC(C=C(C)C)=O)C12CC2 CCCCCCCS(=O)(=O)N(C)CC1CCSCC1 c1(C(=O)NCCC(C)NC(C2CN(CCC)C(=O)C2)=O)c(N)ccc(Cl)c1F c1(OC)nc(C(=O)NCCCCC2CCN(C(=O)C=CCF)CC2)cc(O)n1 C1(C(CC)C)CCN(C(=O)C=CCN(C)C(C2CC3C=CC2C3)=O)CC1 N1(C(CC2(OC)CN(C(=O)C(C)(C)SC)C2)=O)CCC(N=[N+]=[N-])CC1 c1(NC(C2C(C(=O)NCC(C(C)C)NC(Cc3nc(C)oc3)=O)C2)=O)ccc(Cl)cc1 N1(C(C2(NC(C(C)N(CC)CC)=O)CC2(C)C)=O)CCN(CC2CC2)CC1 Cc1cnccc1C(=O)N(CC(C)(C)NC(=O)CC1(O)CCOC1)C C#Cc1cc(F)c(C(=O)NCCCCCNC(=O)CCc2nc(C)no2)cc1F c1(N(C)Cc2ncc(F)cc2F)nc2c(c(=NCC(C)c3cccs3)[nH]1)COCC2 c1(NC2CC(C)N(C(c3cc(Cl)on3)=O)C2)c(F)cc([N+](=O)[O-])cc1F C1(CC)CCN(C(c2csc(C)c2)=O)C1CNC(=O)CC(=O)OC(C)(C)C c1(C(=O)O)cccc(CC2CCN2C(=O)Cn2cc(Cc3nn[nH]n3)nn2)c1 c1(C(N2CCC(NC(c3cnc(OC)nc3)=O)C(C)C2)=O)nn(C)cc1[N+](=O)[O-] C(C(C)(C(=O)NOC(c1ccccc1)C)NC(c1[nH]nnc1C)=O)SC c1(C(=O)NC)ccc(NC(c2coc(C(=O)NC3(C)CCC3)c2)=O)cc1 Cc1[nH]c2ccc(C(N3CC=CC3CNC(C3CCCN(C)C3)=O)=O)cc2c1C N1(C(COCCOCC#C)=O)CCC(C)C(N(C)C(c2ccsc2SC)=O)C1 N1(C(C2CCC3(CC3)C2)=O)CCC(C(N2CCC3CC23)=O)C12CC2 C(N=c1nc2c(cnn2C)c(NC2CCC3CC23)[nH]1)c1c(C)cn(C)n1 c1(CSC)ccc(F)cc1CNC(C1(CO)CC(F)(F)C1)=O N1(C(C)=O)CC(O)CC1C(=O)NC(C)(C)C(C)NC(=O)Cc1cnns1 C(c1ccc2c(c1)COCC2)=CC(=O)NC(CC)CN(C)C(c1cnc(S)[nH]1)=O n1(CC)ncc2cc(C(=O)NCC(CNC(=O)CCCOC)CO)cnc12 Cc1cncc(C(=O)NC2CN(C(C3C4CCCC34)=O)CC2C)c1Cl c1(OC)ccc(C(=O)NC2CC2CNC(C2(O)CCOC2)=O)cc1C1CC1 C1(NC(c2cccc(Cl)c2Cl)=O)CN(C(C23CC(F)(C2)C3)=O)CC2(CC2)C1 C1(C(N(C(C(=O)N(CCN=[N+]=[N-])C)(C)C2CC2)C)=O)CCC(C2CC2)C1 n1(CCCC(=O)OCC)c(N(C2CCCSC2)C)nnc1COC c1(-n2c(C(=O)NCC(CNC(C(C)C3CC3)=O)O)cnn2)cccnc1Cl c1(CNc2scc(C(=O)Nc3cc(OC)c(Br)cn3)n2)ccc2nnsc2c1 c1(C(N2C(CCNC(=O)CCN3CCC(O)CC3)CCC2)=O)cc2scnc2[nH]1 C1(C(=O)NC(c2ccc(C)cc2)CNC(C2(C)C=CCC2)=O)CCOC(=O)CC1 CN1N=CC(CC(N2CCC(N(C)C(c3cccc(C(F)(F)F)c3)=O)C2)=O)C1=O c1(C(=O)NC2CCCC(N(C(c3cnc(OC)s3)=O)C)C2)cnc2n1CCCC2 C12(C(N(C)Cc3ccc(CC)o3)=O)CC(CCO1)N(C(c1cn(CC)nn1)=O)C2 C1(NC(C(C)(C)Cl)=O)CCOCC1C(=O)Nc1ncn(-c2ccccc2)n1 N1(C(CSCC)=O)CCN(C(=O)C(C)N(C)C)CC1CCO c1(C(=O)NC(CNC(CNC(CCC)=O)=O)(C)C2CC2)ccnc(F)c1N CN(CC(=O)NCC1CCCC1)N1CCc2[nH]c(=O)c(N)c(C#N)c2C1 CC1C(C(=O)NC2(C(=O)NCC3(F)CCN(C)C3)CCSC2)=NOC1C C1(C(=O)Nc2c(CC)nn(C)c2)CN(C)CCN1C(C1CC1(C)C(F)F)=O C(C(C)(O)CNC(C1(CC(C)C)COC1)=O)NC(C(C)SCC)=O c1(CCC(N2CC(C(C)NC(C(CCC)OC)=O)C2)=O)ccc(C)c(Cl)c1 c1(C(=O)NC2CN(C(c3cncc(OC)c3)=O)C3C2C3)ccc(F)c(F)c1C C1(C(=O)NC(CNC(c2ccc(CN=[N+]=[N-])o2)=O)C2CCC2)(COC)CCCO1 C(=O)(C1=C(Cl)CCCC1)N(C1CCCN(C(=O)C(C)c2ncco2)C1)CC CC1CCC(F)(C(N2CC(O)(CNC(=O)Cc3nc(C4CC4)n[nH]3)C2)=O)CC1 N1(C(CC2CC(OC)C2(C)C)=O)CCOC(C)(CNC(c2ccnc(O)c2)=O)C1 N#Cc1ccccc1NC(C1CN(C(c2ncc(Cl)cc2Br)=O)CCC1O)=O c1(C(=O)NCC(C2CCC2)NC(CCC2N(C)CCC2)=O)ncc2[nH]ncc2n1 C(=O)(C(C)CC(F)F)N1CCC(OC2CN(C(C3C(C)OCC3)=O)C2)CC1 C(=O)(C(Cl)=CCl)NC1C(NC(C(c2ccccc2)OCCC(C)C)=O)CC1 N1(C(c2cn(CCC)nn2)=O)CCC(CNC(=O)CN2CC(C)(C)C2)(COC)C1 c1(C(C)(C)C)n[nH]c(=NC2CN(C(=O)CCC(=O)NCCC#N)CC23CCC3)s1 n1(CC)ncc(Cl)c1C(=O)NCCCN(C(=O)C(C)Sc1nncn1C)C C=CCC(C(=O)NCC1(C(=O)NCCOC(F)F)CCCO1)OC C#Cc1cn(C)nc1C(=O)NC1CN(C(c2nc(O)sc2C)=O)C1 Cn1c(O)nc(N2CCC(C3(NC(=O)CNC(=O)C(F)(F)F)CC3)C2)cc1=O C1(CN(C(=O)C(C)(C)NC(=O)C(F)(F)F)C)CCCS1(=O)=O N1(C(C(C(C)(C)C)=O)=O)CCOCC(C)(CNC(C2CCCCCC(=O)C2)=O)C1 c1(N(C2CCN(C(c3cn[nH]c3)=O)C2)C)nc(Cl)nc2c1S(=O)(=O)CC2 CCC(O)C(C)(C)C(=O)NCC1CN(C(c2cccn3cncc23)=O)CCO1 C=CC1(CC(=O)NCC(=O)NCCC(Cl)Cl)CC1 C#CCCCCC(=O)NC1CC(C)(NC(=O)CNC(c2ccc(F)c(F)c2)=O)C1 N1(C(C(COC)OC)=O)CC=CCC1C(=O)NCc1ccnn1C(C)C c1(C(C)NC(N2CC(=O)N(c3cn[nH]c3)C2)=O)ccc(C(F)(F)F)cc1 CCC(CC(=O)NCC1CN(C(c2cccnn2)=O)C1)SC N1(C(C(CC=C)CC)=O)CC(C)(C)OCC1CNC(c1cc(C)n(C)c(=O)c1)=O Cc1cc(C(N2CC3(COC(=O)C3)C2)C(=O)NCCCF)c2c(c1)CCC2 C(=O)(C1=C(Cl)CCC1)N1C(C2CCN(C(c3nccc(COC)c3)=O)C2)CCC1 c1(C(=O)NCC(CCNC(CCCOC(C)=O)=O)F)ccc2c(c1)OCC(=O)N2 c1(OC)ccc(C)cc1CC(N1CCC(C(=O)NCCc2cccnc2C)C1)=O C12(C(=O)NC(C3CCCC3)CNC(=O)CCC3CC3(Cl)Cl)CCCN1CCC2 c1(C(N(CC(C)N(C(c2c(CC)scc2)=O)C)C)=O)ccc(F)c2cccnc12 C1(CN(C(=O)CCCc2cnn[nH]2)C)CCCC(O)C1.C1CC(=O)NC(=O)N1 CC(C)C(F)(CNC(c1cnn2c1OCC2)=O)C(=O)NC1(C2CCC2)CC1 CCCCC(=O)C(=O)N1CCCC(NC(=O)Cc2ccc(OC)nc2)CC1 C1(C(=O)NCC(N(C(CCCC)=O)C)C2CC2)COCCOC1 C1(O)(CNC(=O)COCC(F)(F)F)CCN(C(=O)CNC(=O)C(F)(F)F)CC1 CCCCC(CC)C(=O)N1CCC(NC(c2c(I)n[nH]c2C)=O)C1 C1(Cn2cc(CN(C)C(N)=O)nn2)CCCCN1C(=O)C(C1CC1)NS(C)(=O)=O C=C1CCC(CNC(=O)CC2CCCN(C(C3CC(C)=NO3)=O)C2)CC1 c1(C(N(C(CC)CC(=O)Nc2cccc(C)c2)C)=O)ncc(F)cc1F CCCC(CC)C(=O)NCCC(O)C(=O)NCCCCCC1CC1 N1(C(c2ccc(C(C)C)cn2)=O)CC2(C1)CN(C(C13CCCCC1C3)=O)C2 C1(NC(c2n(CC)nnc2)=O)CC2CCCC(C1)N2C(=O)CN(C)CCO N1(C(c2scc(OC)c2)=O)CCC(C)C(NC(c2ncoc2C(F)(F)F)=O)C1 c1(CC)ccc(OCC(F)(F)F)c(CC(=O)ONCC2(CN)CC(F)(F)C2)c1 N1(OCc2c(C)cccc2)CCCCCC1.CC(C)C c1(N2CCCC(CNC(CC(CC)C)=O)CC2)ccn2ncc(I)c2n1 c1(CCNC(=O)NC2CC3(CC(C#C)C3)C2)cc(Br)cc2c1OCC2 C=CC1(C(=O)NC(C)CCC(C)C)CCN(C(c2ccncc2C)=O)C1 c1(CC(=O)NC(CCNC(c2c(C)nc(SC)s2)=O)C)cc(C)ccc1F n1(CCNC(C)=O)cc(C(C)(C)N(C(=O)CCc2ccc(C)o2)CCF)nn1 c1(CNC2CCC(C(=O)Nc3c(C(N)=O)scc3)CC2)ccc(Cl)cc1Cl N1(C(c2ccc(C(=O)NC)nc2)=O)CC(NC(=O)CC2CC2C2CC2)CC1(C)C c1(CC(=O)NC(C(=O)NC(C)Cc2cnn[nH]2)CN(C)C)nc(=N)[nH][nH]1 c1(C(=O)NC2CCN(CCNC(C(COC)C)=O)CC2)ncc([N+](=O)[O-])n1C c1(OC)ccc(CCC(N2CCC(F)(C(=O)NC(C)C)C2)=O)cc1 CC1(CNC(=O)Cc2cccnc2Br)CCCN1C(C1CCCN1C1CC1)=O c1(C(N2CCC(C)(NC(C34CCC3C4)=O)C2)=O)ccnc2ccccc12 c1(C(N(C2CCN(C(=O)Cn3cc(CO)nn3)C2)CC)=O)cnc2cc[nH]c2c1 c1(CN2C(C(=O)Nc3ccnc(Br)c3F)CC(O)C2)cc(F)cc(F)c1O c1(C(=O)NC)ccccc1Cn1nc(-c2cccs2)nc1COc1ccsn1 N1(C(C2N(C(C)C)CCC2)=O)CCN(CCN(C)C(C2(C)CCCC2C)=O)CC1 N1(C(c2ncn(C)c2)=O)CCCC(C2CCCN(C(=O)C(O)CC(C)(C)C)C2)C1 C12(NC(c3cc4cccnc4[nH]3)=O)CCCC1CN(C(c1cc(Cl)no1)=O)C2 N1(CC=CC)CCC2(CC1)CC(C(=O)Nc1cccc(CC)c1)CO2 C1(C(=O)NCc2cc(C)oc2)CN(C(=O)CN2C(C)CCCC2C)CCC1(F)F c1(C(N(CC#C)CCF)=O)cnn(CCNC(c2nc(Cl)cs2)=O)c1 CC1(CNC(=O)CC2CC3CCC2C3)CCCN1C(=O)CC1CCC2CC12 S(=O)(=O)(c1ccc(C)c(C)c1)N1CCC(S)C1.c1(OC)ccc(Br)c(NC)n1 Cc1nc(N(C)C)sc1C(=O)Nc1cccc(NC(=O)CSCc2cccs2)c1 c1(NC(N2CC(C)C(O)CC2)=O)nc2nccc(Br)c2o1 C1(C)(SC(CCNC(c2c(C)nccn2)=O)C)CCCCN1C(=O)OC(C)(C)C N1(C(Cn2ncn(C)c2=O)=O)CC(CNC(=O)C=Cc2ccncn2)C(F)(F)C1 C(C(CC1CC1)C(=O)N1CCSCC1C1CC1)OCC(=O)NCC1CCCC1 N1(C(C(C)C)=O)CCC2CN(C(c3cccc(CO)c3)=O)CC12 N12CCC(C1(C)C)C(=O)NOCC1N(C)CCN2C1.Cc1cc(C=O)ccn1 c1(C(CC(=O)N(C2CCN(CC(F)F)CC2)CC)N)ccc(C(F)(F)F)cc1 c1(C(C(=O)NCCC(C)NC(C2COC(C)(C)C2)=O)(C)O)ccccc1F C1(NC(c2n(C)ccc2)=O)COC2(CCN(C(=O)CN(CC(C)(C)C)CCO)C2)C1 C12(NC(N3CCC(O)(C(C)C)C3)=O)CCC(C1)OC2C c1(C(=O)NCC(CNC(C(COC)C)=O)(C)O)nc(OC(C)C)ccc1Cl c1(-n2cc(C(CC)N)nn2)ccccc1CNS(=O)(=O)CC C1(COC)CN(C(=O)C(C2CCC2)NC(=O)C2=COCC2)CCO1 C1(N)(CC)CCCN(C(=O)Cc2ccn(-c3ccc(Br)cc3)n2)C1 C1(C(=O)NC2CCC(CNC(c3cc(C(=O)OC)[nH]c3)=O)C2)CCC(F)(F)CC1 N1(C(c2on(C)c(=O)c2)=O)CCC2(CCOC2)C(CNC(=O)C(C)(C)C(F)F)C1 c1(C(N2CCCN(C(C3(C=C)CC3)=O)CC2C)=O)cc(F)cc2ccoc12 c1(C2(CNC(CC(C)C3CCCO3)=O)CC2)ncccc1[N+](=O)[O-] C(=O)(C1=CCC(F)(F)CC1)NC1CN(C(CCC#C)=O)CC(C)C1 c1(C(=O)NCC2C3CN(C(C4CC(C)(C)OC4)=O)C(C3)C2)ccn2ccnc2n1 c1(CNC(=O)NCCCC(O)CO)cc(F)c(F)cc1I c1(C(=O)OC)nc(NCC2CCCCN2C(c2cnc(C)s2)=O)sc1C Cc1ncc(C(=O)NC(CCC(C)C)C(=O)NCc2nn[nH]n2)cc1C#N N1(C(CC=CC=C)=O)CCCC2(CCC(NC(=O)C(C)(C)C3CC3)C2)C1 C1(N(C(CCc2scc(C)c2)=O)C)CCCCN(C(c2cn(C)c(=O)cn2)=O)C1 C1(CNC(c2cccc(SCC)c2)=O)CN(C(=O)CCCSC2CC2)CCC1C c1(C(=O)NCC2(C)N(C(C3C(C=C)C3)=O)CCC2)cc2n(c1)CCS(=O)(=O)C2 c1(C(=O)NC2C(CNC(C(c3cccc(C)c3)O)=O)C2)cccc2nccn12 c1(NC(C(C)NC2C(CO)C3CCCC23)=O)cc2ccccc2s1 N1(C(CCC(CC)=O)=O)CC2CCC(N(C)C(c3ccc(CC)[nH]3)=O)C2C1 C1(C(N2CC(NC(C(CCCC)F)=O)C(C)(C)C2)=O)CCOC2(CCC2)C1 c1(C(=O)NCC(Cc2ccccc2)CO)cc(Br)cc(F)c1F CC#CC1CCN(C(=O)Nc2ccnn2C)CC1 C#CCC(CC#C)C(=O)N1CC(CNC(=O)CC(CC)C2CCC2)C2(CC2)C1 C1(C(=O)NC(C2CCCC2)CNC(=O)C2=COCC2)CC2OC1C1CC21 N1(C(C(C)C2CCC2)=O)CCC(NC(=O)C(C)(F)F)C(F)C1 C1(CC(N2CC(CC(C#C)C)C2)=O)CCCN(C(=O)C(COC)OC)CC1 C1(NC(c2cc(F)c[nH]2)=O)COCCN(C(C2CCOC2)=O)C1 c1(NC2CCN(C(c3ncc(C)nc3)=O)C(C)C2)ncnc2[nH]ccc12 Cc1cc(NC(=O)CCC2CCCCN(C(c3c[nH]nc3C)=O)C2)cc(C)c1C CC12CC(CC(=O)Nc3ccccc3C3CCNCC3)(CO1)C2 N12C(C3CC(O)C1C3)C2=O.c1(N(C(=O)C2CC2)C)cccc(CC2CCC2)c1 N1(C(=O)C=Cc2ccc(Br)s2)CC2CCCC(C1)N2Cc1cn[nH]c1 C1(C(N(CCCCNC(C(CCCC)F)=O)C)=O)CCc2nncn2C1 C(=O)(CCCCCS(N)(=O)=O)NCC(CNC(C1(C)CCN(C)CC1)=O)CO c1(C(N(C2CC(NC(COCCOCC#C)=O)C2)C)=O)ccnn1CC(F)(F)F c1(CN2CCN(C3CCN(C(c4cc(CC)on4)=O)CC3)C2)ccc(F)c(F)c1 c1(C(N2CC(NC(c3sc(C)c(C)c3C)=O)C(O)C2)=O)nccn2nccc12 C1(OC)CCC12CC(C(=O)NCCCCCCNC(c1onc(C)c1C)=O)C2 N1(CC)CCN(CCC(=O)N(C(C)CNC(=O)C(c2cccs2)SC)C)CC1 CC(CCC(C)(C)C)C(=O)N1CCOC(CC(=O)Nc2cccc(F)c2OC)C1 c1(C(=O)NCCC2CCN(C(c3ccc(C)n3C)=O)C2)cc(Cl)ccc1Cl C1(C(N2CC(c3cn(CC(=O)NCCO)nn3)(F)C2)=O)CC1C1CCCC1 c1(C(N2CCC3(CC2)CC3)C(=O)NC(C(=O)OC)C)cccc(C)c1Br C=CCCC(C)(C)C(c1nnnn1CC1CC1)NC(CC)CCC(F)(F)F Cc1cc(NC(C2CCN(C(c3cnn4ccsc34)=O)CC2)=O)cc(C)c1C C1(CC(N2CCOC(C(=O)NCC3(CF)CC3)C2)=O)(OC)CCCCC1 c1(NC)ccc(SC)cc1.C1(SC)CC(C(=O)N(C2CN(C(=O)C(C)C(N)=O)C2)C)C1 C=CCC(CC(C)C)C(=O)NCC1(F)CCN(C(c2ccc(C)o2)=O)C1 N1(C(C(C)(C)C2CC2)=O)CC(NC(=O)Cn2nc3c(n2)CCCC3)C2(CCC2)C1 c1(C(N2CCCC(CCNC(C3CCCO3)=O)C2)=O)cc2ccc(Br)cc2[nH]1 CCC(C)C(O)C(C)C(=O)N1CCC2(CCC2)C(CNC(=O)CC(CC)SC)C1 Cc1ccc(C(C)C)cc1C(=O)NC1CCC(NC(c2cncnc2)=O)CC1 c1(C(=O)OC)c(NC(C2CCN(C(C3CC3F)=O)C2)C)nnc(C)c1C OC1CCN(CC2CCN(C3CC3)CC2)CC1c1ccccc1 CC(C)(C(=O)N1CCC(NC(=O)CC(=O)NCC2CC2)C1)c1cnc[nH]1 C1(NC(=O)CCCCC2CC2)CCCCCN(C(c2c[nH]nc2C2CC2)=O)C1 C(=O)(N=c1ccn(CCCO)[nH]1)C1(CNC(C(CCC)C#N)=O)CC1 c1(OCCNC(=O)C(=O)NCC2CCOCC2)ccc(Cl)nc1 c1(C(N2CC(N(C(=O)C(F)CC3CCC3)C)C2)=O)c(F)ccc(F)c1O C(=O)(C(=O)N=S(C)(C)=O)NC1C(NC(c2c(OC)cc(F)cc2)=O)C1 C=CC(C)(CC)C(=O)NCCC1(NC(=O)CN2CC3CC3C2)CCC1 c1(C(=O)NCC(=O)NC(C)C(C)NC(c2cn(C)nc2Cl)=O)c(F)cccc1Cl C#CC(C)(C)C(=O)N1CCN(C(C2CC3CCC2C3)C(=O)NC(C)C)CC1 c1(CNc2cn(C)c(C(=O)Nc3csc(Br)c3)c2)c[nH]c2nscc12 Cc1nccnc1C(=O)NC(C)(C)CCNC(=O)CSCc1cccnc1 c1(CNC(C2CCC(NC(C3CCCS3)=O)C2)=O)cccc(F)c1F c1(OC)ccc(F)c(C(=O)NCCC2(O)CN(C(=O)CCCN(C)C)C2)c1N N1(C(C(N2CCC(C)CC2)=O)=O)CCC2CN(Cc3ccc(C(=O)O)s3)CC12 c1(C(=O)NCC(CC(C)C)NC(=O)C(C)(C)CC(F)F)ccc2nc(O)oc2c1 c1(C(=O)OC)c(NC(C2CCN2C(C2(C#N)CC2)=O)=O)sc2c1CCC2 C(C(C(=O)C(C#N)C1CCCC1)c1ccccc1)NC(CC)C1CCC1 C1(O)(CCNC(C(C)(CO)OC)=O)CCCN(C(c2coc(O)n2)=O)C1 C1(N(C(CCN(CCC)C)=O)CCNC(=O)CCNC(N)=O)CCCCC1 c1(C(N2CCC(C)(NC(c3occc3F)=O)C2)=O)ccc([N+](=O)[O-])s1 C(CCCCNC(=O)C(C)(C)c1nncn1C)N(C(CN(C(COC)=O)C)=O)C N1(C(C2CCN(C)C2=O)=O)CC(NC(C2CC(F)(F)C2)=O)CC(F)C1 C(=O)(C(C)C(C)C(C)(C)C)N1CCC(N(C(=O)CCCS(C)(=O)=O)CCC)CC1 c1(N2CC3C(C(=O)NC4CC4c4ccncc4)C3C2)ncnc2sccc12 C(=O)(CCCC(=O)Nc1cc(F)ccc1C(=O)N(C)CCN1CCOCC1)OCC c1(C(=O)NC2CCN(C(C(CC)SC)=O)C23CC3)sc2cncn2c1C CCCC(C(=O)N(CCNC(=O)CCCc1nnc(C)n1C)C(C)C)C(C)C CCCS(=O)(=O)CC(=O)N1CCC(C)C(NC(C2OCC2(C)C)=O)C1C Nc1cc(NC(C2CCCN(C(=O)Cc3ccccc3)C2)=O)ncc1F CCC(N=c1ccnc(N2CCC(OCCO)C2)[nH]1)c1ccc(Cl)cc1 c1(CC(N2CC(C)C(NC(C3(C)CC3C)=O)C2)=O)cc2ccccc2o1 C1(C(=O)NC(C)CC2CC3(CC3)CN2c2ncc(F)cn2)COCC(C)(C)O1 C=CCN(OC)C(=O)CC(C)NC(c1sccc1CC)=O N1(C(CCN(CCCCC)C)=O)CC2(COC(CNC(c3cc(C)cs3)=O)C2)C1 CC(CC1CC1)C(=O)NCC(O)CCNC(=O)C(c1cncn1C)O c1(OCC(N2CC(CCNC(CCNC(C)=O)=O)C(C)C2)=O)cccc(C#N)c1 N1(C(=O)NCc2cncc(CC)c2)CCN(C)CC1CO C1(CC)CN(C(=O)CC2CCC23CCC3)CCN1C(c1cc(C(=O)OC)cs1)=O c1(C(N2CCC(NCCCN(C)C(C3CC3Cl)=O)CC2)=O)cc(F)cnc1O C1(O)(CC(=O)Nc2ccc(F)cc2)CCN(C(=O)Nc2ccccc2CO)CC1 C12=C(C)N=CNC1=NCC1(F)CCN(CC1)C2=O.C1(OC)(CO)CC1 N1(C(C(C(C)(C)C)NC(c2cnn[nH]2)=O)=O)CCC2CC1C(=O)O2 CC1C(C)N(C(c2ccncc2F)=O)CCN1C(=O)Cc1csc(S)n1 c1(C(=O)NC2CCCC2C(=O)OC)ccc(SC)cc1.CCC(CSC)N(C)C N1(C(C(CCCC)C)=O)CC2CCCCC2(CNC(c2ncoc2C2CC2)=O)C1 C1(NC(c2noc(C3CCC3)n2)=O)CC2CN(C(=O)C(F)(F)CC)CC12.C1CO1 Cc1nc(C(C)C)ccc1C(=O)NC(C)CNC(c1cnc(S)n1C)=O c1(CC)ccc(OC)c(C(N2CC(O)CCC2C)C(=O)NC(C)(C)C)c1 N1(C(C(C)Sc2nncn2C)=O)CCC(NC(=O)CC2CC=CCC2)C12CCC2 N1(C(c2nccc(C)c2)=O)C2CCC1CC(NC(c1cccc3nonc13)=O)C2 C(C(CC(C)C)C(=O)NC1CCC2(CCC2)C1)NC(Cc1nc(C)sc1)=O N1(C(C(C)OC(C)C)=O)CCN(C(=O)CN(c2ncccn2)C)CC12CC2 CC1CC(NC(c2cc(C3CCOCC3)[nH]n2)=O)CN1C(c1cccnc1)=O C1(NC(C2CC2F)=O)(CO)CCN(C(C2(n3cnnn3)CCOCC2)=O)C1 Cn1cc(C(N2CC(NC(=O)CCc3cn[nH]c3)C(O)C2)=O)ncc1=O C12(C(=O)NCC3OCCN(C)C3)CCC(CN(C(=O)CC3(O)CCC3)C1)C2 C1(C(N2CCCC(NC(C(C)(C)C3CC3)=O)C2)=O)CC(=O)c2ccccc2C1 N1(C(CCCc2ccc(C)s2)=O)CCCCC(NC(=O)COCC2CC2)CC1 N1(C(C2=C(C)OCCC2)=O)CC2CCC1C1CN(C(c3cc(C)sn3)=O)CC21 c1(C2OCCN(C(C(n3ncc(C)c3)C)=O)C2)nnc2ccccn12 c1(C(N2CCCC(CN(C)C(C3(F)CC=CC3)=O)C2)=O)cc2nc(Cl)ccc2o1 CC(CNC(C1(CO)COC1)=O)(CO)NC(=O)CSCCC(F)(F)F C(=O)(C1=CCC2CCC1N2C(=O)C(CC)N(C)C)N(CC#C)C C1(CC=C)(NC(C(C)OCCC=C)=O)CCN(C(=O)C2=CSCS2)CC1 C1(NC(C2(C)CCC2)=O)CC(C2CCN(C(c3cc4n(c3)CCCC4)=O)CC2)C1 C1(NC(=O)Cc2csc(CO)n2)C2CC(O)C1N(C(=O)C(O)C1=CCCCC1)C2 Cc1cc2c(cc1NC(c1onc(Br)c1C)=O)CCO2 C12(C(=O)NCCn3cc(C(=O)NC4(CCCC)CC4)nn3)CCCC1CCC2 C1(N(C)C(c2cnn(C3CC3)c2Cl)=O)CN(C(C2CCCS2)=O)CC1(C)C C(=O)(C(C)(O)C(C)(C)C)N1CC2CC(NC(c3cn(CC)nn3)=O)C2C1 C1(NC(CSCC#C)=O)CN(C(c2ccc(-c3cccs3)nc2C)=O)CCC1F c12ncn(c(=O)n1CCc1ccc(C)cc1)n2.CCCCOCC C(=O)(CC(C)(C)CNC(C1COCC1C(N)=O)=O)N(CCCC)C1CC1 C1(C2(C)CC2)(C(N2CC(C(C(=O)NC3CCOC3(C)C)OC)C2)=O)CC1 n1(CCC)ncc(C(=O)NC2CCCCC2CNC(=O)C(C)NC(N)=O)c1C CCC(Cc1ccccc1)CC(=O)NCCC(C)N(C(=O)CN(C)C1CC1)C c1(C(=O)NC(CC(C)NC(c2cc(C(F)F)ccn2)=O)C)nnn(C)c1N c1(CC)[nH]nc(Cl)c1C(N1CCC(N(CCO)C(C2CCC(=O)N2C)=O)C1)=O N1(C(C(CN(CC)CC)F)=O)CCC(C)CC1C(N1CCCN(CCO)CC1)=O O(C=CC(=O)NCC1CCCN1C(c1c[nH]nc1C1CCOCC1)=O)CC N1(C(C2N(C(C3(OC)CCOC3)=O)CCC2)=O)CC(C)CC(C)(C)C1 N1(c2ccc(OCC)cc2)CCN(C(F)(F)C(F)(F)F)C(=O)C1 Cc1cc(F)ccc1C(=O)NCC1(O)CCN(C(=O)C2=CCCC2C)CC1 C(=O)(C(CN=[N+]=[N-])NC(=O)C=Cc1ccsc1)N(C)CC1CCN(C)C1 c1(N(CCC#N)C(=O)NC2(C(C(C)C)OCC)CC2)cnc(OCC)cn1 N1(C(c2nccc(OCC)c2)=O)CC2CN(C(=O)CCN3CCOC3=O)CC12 c1(CN2CCCCC2)ccc(F)cc1F.N12CCCC1NC2=O CC1(C)CCN(C(=O)C=CC(c2ccccc2)=O)CC1NC(c1cnns1)=O CC(C)C(F)C(=O)Nc1cccc(NC(=O)CC2CCCN2CCN(C)C)c1 CC(c1ccccc1)=CC(=O)NC1CCN(C(=O)NCC23CC(CO)(CN2C)C3)C1 c1(C(C(=O)NCCN(C(C=CC(CC)=CC)=O)C2CC2)C)cccc(Cl)c1 O=C(C#CC1CCC1)NC1COCC1NC(=O)Cc1ccoc1 c1(CC)cc(C(=O)NC2CCN(C(=O)C=CC3CCC3)C23CC3)ccc1OC c1(OCC(=O)N(C2CC(NC(C(C)C)=O)C2)C(C2CCCO2)=O)cccnc1Cl S(=O)(=O)(CC(=O)NCC1(C)CCCN1C(=O)CSCCC(F)(F)F)NC N#CC1(C(N2CCC(CF)(NC(C34CC(F)(C3)C4)=O)C2)=O)CC2C=CC1C2 C12(NC(c3c(OC)scc3)=O)CCCC1N(C(C1(NC(C)=O)CCCC1)=O)CC2 C1(C(C)NC(C2CCO2)=O)CCN(C(C2CC(N(C)C)C2)=O)CC1 c1(C(=O)NCC(CC)(CC)NC(=O)CC2(C3CC3)CC2)nccn2ccnc12 C1(NC(=O)C(O)C(F)F)CC2CCCC(C1)N2C(c1c(Cl)cnn1C1CC1)=O C=CCCC(C(=O)NCCN(C)OC)NC(c1cnns1)=O C1(C(N2C(CNC(=O)Cc3n[nH]c(O)n3)CCCC2)=O)CC12CCSCC2 C(N=c1[nH]c(=NCc2ccc(N)cc2)[nH]c2ccccc12)C1C(C)C1 C(=O)(C1=C(Cl)CCC1)NC1CCN(C(c2n(COC)ncc2)=O)C1 CC(CO)C(C)N=c1[nH]c(=NCCC2OCCC2(C)C)[nH]c2c1COC2 N1(C(CCCC#C)=O)CCC(CO)C(NC(c2ncn3c2CCC3)=O)C1 c1(NC(=O)CNC(c2cnn(-c3ccccc3)n2)=O)ccccc1F O=C(C1=CC2(CCOC2)C1)N1CC2CCC(C1)N2C(C12COC(F)(F)C(C1)C2)=O N1(C(COC2C(C)C2)=O)C(CC(=O)NC(CC2CCC2)CO)C2CCCC12 c1(C(=O)OC)cc(S(=O)(=O)NCc2nn(C)c(Cl)c2I)sc1C N1(C(C(C)=C2CC2)=O)CC2CC2(CNC(c2cc(-c3ccco3)no2)=O)C1 N1(CC)CC(C(=O)NCC2(O)CCN(C(C3(C(=O)NC4CC4)CC3)=O)C2)CC1=O C1(C(=O)NC(C2CN(C(c3c(C)cc(C)s3)=O)C2)C)CCc2n[nH]cc2C1 C1(C(C(=O)NC2CC(CNC(=O)C(O)C3CCC3)C2)OC)CCC(F)(F)CC1 C(=O)(C1=CC2CCCCC12)NC1C(C)N(C(=O)Cn2ccc(=N)[nH]2)CCC1 CC(C)(CO)C(=O)N1CC(C)(C(=O)NC(C2CC(C)(C)C2)CO)C1 c1(C(=O)NCCCCCNC(C2(CC#C)CCCCC2)=O)c(OC)cccc1Cl C1(NC(C(COCC)C)=O)CC2CC(NC(c3c[nH]c(C(N)=O)c3)=O)CC12 C(CC(=O)NC)(C1CC1)NC(CCN(CCCCC)CC(C)OCCO)=O C1(N(C(c2nccc(CC)c2)=O)C)CCCCN(C(C2CCN(C)C2C)=O)C1 C1(C(C)(C)NC(C(CN(C)C)O)=O)CCN(C(c2c[nH]c(C(N)=O)c2)=O)CC1 c1(OC)cccc(C)c1C(N1CCC(O)(CCNC(C2CCC2(C)C)=O)C1)=O C(=O)(C1OC(=O)c2ccccc21)NCC1CCN(C(C(CCOC)(C)C)=O)C1 N1(C(C2CC(OCC)C2)=O)CCCC1C1CCCN1C(=O)Cc1ccnc(C)n1 Cn1nc(C(=O)NCC(C)(F)CNC(=O)C2=CC3CCC(C2)C3)c2c1CCSC2 C1(C(N(C)C)=O)CCN(C(c2cc(C(C)(C)C)no2)C(=O)NCCO)C1.C1CC1 N1(C(C=CC)=O)CCN(C(=O)CN2CCCCC2=O)CC1C(C)C CC1CN(C(C2CCCN2C)=O)CCC1NC(C1(C(=O)NC2CC2)CCC1)=O C1(NC(C(C(C)C)OC)=O)COCCN(C(=O)Cc2cc(C(C)C)no2)C1 CC(CC(F)(F)F)C(=O)NCC1CC(NC(=O)CCC(F)F)C1 C(=O)(CC1=NN(C)C(=O)C1)NCC(C)C(=O)NC(C)Cc1cccnc1 C1(C(=O)NCC2(F)CC(CNC(c3sccc3F)=O)C2)COC2(CCC2)CO1 c1(CC)c(C(N2CC(CCNC(=O)CC3CCOC3(C)C)C2)=O)nnn1C C1(C(=O)NCc2c(C(=O)NC3C(C)COCC3)cco2)CC2(C1)CC21CC1 N1(CC(C)(O)C(=O)Nc2cccc(C3CC3)c2)Cc2ccccc2C1=O CC(CS(C)(=O)=O)C(=O)N(CC(C)(C)N(C(=O)C(C)Cc1ccccc1F)CC)C CC12CC(CO)(CO1)C2.c12ccc(cc1)CNC2c1nnnn1CC1CCCO1 c1(C(=O)NC2C(CNC(Cc3cnc(C)s3)=O)CC2)cc(N)ccc1[N+](=O)[O-] c1(CNC2C(C(=O)Nc3cnc(CC)nc3)C2)ccc(Br)c(C)n1 CC1CC(NC(=O)C=CCO)CCN1C(C1CC2CCCC12)=O n1(CCCC)nccc1C(=O)NCCOCCNC(=O)CCCN(CCC)C(C)C c1(C(N2CC(O)(CN(C)CC3CCCS3)C2)=O)coc2c(F)cc(F)cc12 N(C(=NCc1cccs1)NC1COC(C(F)F)C1)C(c1cocn1)C C(=O)(CS(=O)(=O)C(C)C)N1C(C)CC(NC(C(CC)NC(N)=O)=O)C1 C(=O)(C(COC)NC(C)=O)N(C(CCNC(CN(CC)CC)=O)C)C c1(C(=O)NCC2CCC(NC(c3nc(Cl)cs3)=O)C2)cc([N+](=O)[O-])n[nH]1 c1(C(N(C2CCN(C(CSC)=O)CC2C)C)=O)cccn2ccnc12 C(=O)(C(=O)NCC(F)(F)F)NCC(CC=C)NC(=O)C(CO)NC(N)=O CN1CC2(CC2)CC1C(=O)NCCCCCCC1CC1.C1(C)(C)C(=O)N1 C1(NC(C(C)NC(C)=O)=O)CN(C(C2(C(F)(F)F)CC(F)(F)C2)=O)CC(C)(C)C1 c1(C(=O)NC2C(C)(C)C(CNC(C3CC=CC3)=O)C2)[nH]c2ccccc2c1Cl N1(C(c2ccc(C(c3nnnn3C3CCCC3)OC)o2)=O)CCCC(OC2CC2)C1 c1(C(N2CCC(NC(C(C)C3CC3)=O)(CF)C2)=O)ccn(C)c(=O)c1 Cc1cccc(C(=O)NCC2(CNC(c3ccc(C)n3C)=O)CC2)c1C(F)(F)F N1(C(C(C)(F)c2ccon2)=O)CC(O)CC1C(=O)NCC1CC1.C1CO1 c1(CNC(=O)NC2C(NC(=O)OC(C)(C)C)CC2)ccccc1S(=O)C(F)(F)F C1(C(=O)NC(c2cccnc2)COC)CC(C)C1(C)C c1(C(=O)NC(CC=C)CNC(=O)CCOCC(F)(F)F)cn(C)nc1OC C1(NC(CCC=CC)=O)CCC2CCN(C(=O)C(C)(C)CC3CC3)C1C2 C1(C(=O)NCC(F)C2CCC2)CN(C(=O)CNC(=O)C2CC2)CC1F CCC(O)C(C)C(=O)NCCOCCN(C(=O)C(C1CC1)SC)C N1(C(CC2CC(=C)C2)=O)CCCCCC(NC(=O)C(C)(O)C2CCC2)C1 c1(C(N(C(CCNC(C(C)OCC#C)=O)C)C)=O)c(O)nc(C)c([N+](=O)[O-])c1C C1(CNC(C(C(=C)Cl)(C)C)=O)CC2(CCC2)CN1C(c1sccc1C1CC1)=O Cn1cnc(C(=O)NC(C(=O)NCC2CC23CCC3)C2CCC2)c1 n1(CC(=O)NC(c2nc(C)sc2C)C)c(F)cc(C(F)(F)F)c1F N1(C(C2C(C)(C)C2)=O)CCCCC(CNC(=O)Cc2cnc(C3CC3)[nH]2)C1 c1(NCc2nccc(C)c2)ccc(C(=O)NC2CC(=O)NC(=O)N2)cc1C c1(C(N2CC3(C(NC(=O)Nc4ccc(C)cc4)C3)C2)=O)cccc(S(C)(=O)=O)c1 N1(C(C(CC)NC(N)=O)=O)CC(NCc2cc(COC)[nH]n2)C(n2cccn2)C1 C1(C(=O)NCC2(CCNC(c3c(C)c[nH]c3)=O)CC2)COc2ccc(F)cc2C1 CC1(C)CCC1C(=O)NCCCCCNC(c1coc(-c2ccsc2)c1)=O CC12CCOC(C(=O)NC3CCN(C(=O)CC4(O)CCOC4)C3)(C1)C2 c1(CCC(=O)NC2C(CNC(C3(NC(CCC)=O)CC3)=O)C2)cccc(C)c1 c1(-n2cc(C3CCCN(Cc4c(C)ccnc4C)C3)nn2)c(F)ccc(N)c1F c1(C(N2CC(N3CCN(Cc4nc(C)oc4)CC3)C2)=O)ccc(F)cc1Cl c1(CC(=O)NCC2C(C)(C)CCN2C(c2cc(Cl)no2)=O)ccc2c[nH]nc2c1 CN1CCN(C(c2cnsn2)=O)CC1CNC(c1coc(Cl)n1)=O C1(C)(CC)CN(C(=O)CCOCC2CC2)CCO1 C(=O)(C1=CCCCC1)NC1CC(CC(=O)N(C2CCC2)C)C1(C)C C(=O)(C(CCC)C(C)C)NC(CCCC)C(=O)NCC1CC2(CCC2)CO1 C12(NC(c3c(C)onc3)=O)CCC(C1)N(C(=O)CC(O)CN(C)C)C2 CCCC(C)(CCC)C(=O)NCC1CC(CNC(C2(CF)CCC2)=O)CO1 C1(NC(C2CC(OCC)C2)=O)C2CN(Cc3ccc(CC)cc3)CC12 c1(C(N2CCCC(CN(C)C(C3(F)CC3)=O)C2)=O)cc(C(F)(F)F)cc(O)c1 c1(NC(C(C2CCN(Cc3c(C)scn3)CC2)C)=O)ccc(O)c(C(F)(F)F)c1 c1(OCc2nc(C3CC3)no2)cc(C(F)(F)F)ccc1F.C1(=O)C(=O)NC(C)N1C N1(C(C(=O)NCCCC)C2CC(CC)C2)Cc2c[nH]nc2C1 n1(CC)cc(C(=O)COCC)cn1.C1(=O)C(C)N1C.C(COC(=O)C1CC1)S C=CCC(C)(C)CC(=O)NC1CC(O)(CNC(=O)CC2COCCO2)C1 C(c1ccc(Br)s1)=CC(=O)N(CCCN(C(C(=O)OC)=O)C)C n1(CC(=O)NC(COC(C)C)C(=O)NC(c2cncn2C)CO)ncn(C)c1=O CCCCC(O)C(=O)NCC1(C)CCN(C(=O)C(c2ccccn2)O)C1 c1(C(CC)N(C(COC(C)(C)C)C(=O)OC(C)(C)C)CC)ccc(C)nc1 c1(N2CC(CNC(C(C(CC)C)C)=O)OCCC2)c(C)c(C)nc2ncnn12 c1(NC(C2CCC(NC(c3c(OCC)scc3)=O)CC2)=O)cccc(C)c1F C(C(CC1CC1)C(=O)Nc1cccc(OC)c1)NC(C1C(C(=O)OCC)C1)=O c1(C(=O)NC2C(CC)CN(C(=O)C(F)(F)CC3CC3)CC2)ccc2c(c1)CCCS2 c1(CC(=O)N(CCCNC(=O)COCC2CCOCC2)CC)ccc(C#N)nc1 c1(C(=O)NCC=CCNC(C(c2ccc(C)nc2)=O)=O)c(Cl)nn(C)c1Cl c1(C(=O)NC2CC(CNC(CN(CC(=O)NC(C)C)C)=O)C2)ccsc1C N1(C(c2c(N(S(C)(=O)=O)C(C)C)occ2)=O)CCOCC1c1cn(CCF)nn1 Cc1cc(N2CCC(NC(=O)CCCn3ccnn3)C(O)C2)nc(CO)n1 N1(C(=O)OC(C)(C)C)CCC(NC(N)=O)CC1.C123CC(C(C1)C2)C(=O)NC3 c1(C(=O)NCCCN(C(c2ccoc2)C)CCc2ccccc2)cc(O)n(C)n1 Cc1c(-c2cn(-c3c[nH]nc3C)nn2)cccc1Br c1(C(C)NC(C2(CNC(=O)C(O)C3CCC3)CC2)=O)ccc(CC(F)(F)F)cc1 c1(C(=O)NCC2(NC(C(CC)F)=O)CC2)ccc(Cl)c2c1OCCO2 C1(CNC(CN(CCC)C)=O)CCCN(C(=O)C2CC2)C1 N1(C(c2ccc(C(=O)OC)[nH]2)=O)CCCOC(CNC(C2CC2(C)C)=O)C1 N1(C(CC(C)C(C)(C)NC(C2CC3CCC3C2)=O)=O)CC2(C)COCC2(C)C1 c1(C(=O)NCC2CCN(C(c3ccc(SC)s3)=O)C2)cccc(C(F)F)c1 C(=O)(C(C)S(C)(=O)=O)N1CC(CNC(c2noc(C)c2Br)=O)C1 C(CN=C(NCC1(CC(C)C)CC1)NC(c1cccs1)C)c1ccn(C(C)C)n1 N(C(=NCC1CC1)NCC1(C)CCCS1)CC1CN(C)C1 Cn1cc(CNC(=O)C(C2CCN(C(=O)C=C3CCC3)C2)F)nn1 c1(N2Cc3n(cc(C)n3)CC2)nc(NC(C)CC(C)(C)CO)c2ncn(C)c2n1 N1(C(CSCCC(C)C)=O)CCN(C(c2ncc(Cl)cc2F)=O)CC(O)C1 C1(CCNC(c2cn(C)nc2)=O)COCCN1C(=O)CCc1ccc(Cl)nc1 c1(CC)c(C(=O)NC(c2ccccc2)C(=O)NCC2CCCO2)cnn1C c1(C(=O)OC)sc2c(c1I)CNC2S(=O)(=O)Oc1ccc(S(C)(=O)=O)cc1 c1(CC(C(=O)NC)N(C2CCC(F)(F)CC2)C)cc(O)ccc1[N+](=O)[O-] Cc1cc(C(=O)NC2(C(=O)NCC3CCCC(CO)C3)CC2C)nc(O)c1 Nc1c(C(=O)NCCC(O)CNC(C2C3CC4C(C3)C24)=O)cnc2ncnn12 c1(C(ONC(=O)Nc2ccnc(CO)c2)CCO)ccc(F)cc1F CN1CCC(C(=O)NC2CCC2CNC(C2(CO)COC2)=O)C1 c12cc(C)ccc1CNC2=O.C1(NC(CSCC)=O)CCCCC1n1cccn1 N(C(=NCCOc1ccccc1)NCC(C)(C)F)C(C=C)C.C1(OC)CCOC1 Cc1cccc2c1CCN(C(=O)CC1CCN(Cc3ccc(Cl)c(CO)c3)C1)C2 Cc1csc(C=CC(=O)NC2CCCC2NC(C2CCCN2C(C)C)=O)n1 c1(OC)ccc(C(=O)NC2C3CC2N(C(c2cc(C)n(C)c2)=O)C3)c(C(F)F)c1 c1(NC(C(C)n2ccnc2)=O)cc(Cl)c2cc[nH]c2c1.C12CN(C1)C2 CC1CCN(CC(N2CC(CNC(c3cn(C4CCOC4)cn3)=O)C2)=O)C1 C(=O)(C1=C(Cl)CCOC1)NCC(C)N(C(CN(CCC)C)=O)CC CC(C)(C)CC(O)CN(C(=O)C=CC(C)(C)NC(=O)C=C)CC.c1scnc1Cl c1(CN2C(C(N(CC(C)C)CCO)=O)CSCC2)c(Cl)cncc1F Cc1cc(C)c(C(=O)NCC(F)CNC(=O)C(C)SCc2ccccc2)[nH]1 C(C1c2ccccc2CN1C(C1CCCC1O)=O)NC(CSCCC)=O CC1CCC(NC(=O)CCSCC(N)=O)CN1C(=O)CN1CCCCC1=O Cc1oncc1C(=O)NC1CC(NC(=O)C(C)(C)Oc2ccccc2)C1 C#CCC(CC(=O)N(CC(=O)OCC)C1CC1)OC.c12cc(no1)NC2=O c1(C(N2C(C)CC(NC(c3ccc(Cl)c(F)c3)=O)C2)=O)cncc2nc(O)[nH]c12 N1(C(C2C(C)=C2)=O)C2CCC1C(C)C(NC(c1cc3c(o1)CCCC3)=O)C2 C#Cc1ccc(CC(N2CCOCC2C2(NC(C3(C4CC4)CC3)=O)CC2)=O)cc1 C#Cc1ccc(F)c(C(=O)NC(C#N)C(N)=O)c1.C12(CCCCC1)C(=O)NC2 Cc1c(C(=O)NCC(C)(C)CNC(=O)C(=O)NCC(F)(F)F)cncc1N C(C(CC1CC1)C(=O)N1CCC(CN(C)C)CC1)NC(COCC#C)=O CCC(CC)(CC)C(=O)N1CCC(CC(=O)NC(CC2CC2)CC2CC2)C1 C1(CC)CCCC1N=c1[nH]c2c(c(=NC3CCCN(C)CC3)[nH]1)COC2 c1(CC)ccc(C(N2CCC(O)(C(C)CNC(=O)C3=CCCC3)C2)=O)cc1F c1(C(N2CC3(OCC(NC(C4(OC)CC4)=O)C3)C2)=O)nccn2nc(C)cc12 C1(c2cccc(C(C3CN(C(c4cncnc4)=O)C3)C)c2)CC2(CC(=O)C2)C1 C(=O)(C1=NOC(C)(C)C1)NCCC1N(C(CCCN(C(C)=O)C)=O)CCCC1C C1(C(N2C(CNC(C3(Cl)C(C)(C)C3)=O)CC2)=O)Cc2ccccc2NC1=O CC(C)C(F)(CNC(C1(F)CCOC1)=O)C(=O)NCCF c1(N(CCN(C)C(c2c(F)ccc(F)c2Cl)=O)C)cc(=O)n2ccccc2n1 C=CC(CCC)CC(=O)NCCN(C(c1sc(CC)nc1C)=O)C1CC1 Cc1[nH]c2ccccc2c1CCC(=O)NCC(C)(C)CNC(=O)C1CC1 CN1CCN(C(c2ccc(Cn3cccn3)o2)=O)CC1 C(=O)(CC(C)(C)C(F)F)N1CC2C(CC(=O)NCC3(C=C)CCC3)C2C1 N1(C(c2cnc(C(C)(C)C)o2)=O)CCOCC1CCNC(=O)CCc1cc[nH]n1 CN1CCCC(F)(C(N2CCC(NC(C3(N4CCCCC4)CC3)=O)CC2)=O)C1 C(C)(C(F)(F)C(F)(F)F)NC(CCC#C)c1ccccc1 c1(CN(C(C2CCN(C(c3nc(=N)[nH][nH]3)=O)C2)=O)CC)ccc(O)cc1 CC1CCC(OCCCCC(=O)N2CC(C)C(O)C2)CC1 N1(C(C(n2ccc(C)n2)C)=O)CCC2(CCC2)C(NC(c2coc(CO)c2)=O)C1 Cc1ccc(C)c(C(=O)NC2(CC(N3CCN(CCC(C)(C)C)CC3)=O)CCC2)c1 C1(F)(CNC(=O)C=C2CCSCC2)CCN(C(=O)CSCc2ncc[nH]2)C1 Cc1c(C(=O)N(CCCNC(C2CCC3(C2)CC3(F)F)=O)C)nn2ccccc12 C(CC1CC1)(C(=O)C(C=CC(CC)C)=O)NC(CC(C)NC)=O.OC CC12CCC(C(=O)NCC3(NC(C4CC4C(F)F)=O)CCCC3)(CC1)CO2 C(C)(N=c1nc(NCC(C)(C)CC(=O)NC)c2c([nH]1)CCS2)c1n(CC)ncc1 N1(Cc2ccc(CC)s2)CCC(O)(C(=O)NC(c2cncnc2)C)C1 c1(C(=O)NCC(C2CCN(C(=O)CC3CC3(C)C)CC2)C)nccc(Cl)c1O C(=O)(C1Cc2ccccc21)N1CCC(O)(CNC(c2n[nH]c3c2CCC3)=O)CC1 C1(CNC(c2n(CC#C)ccc2)=O)COC(C)(C)CN1C(C1CCS(=O)(=O)C1)=O c1(C(=O)NC(CNC(Cc2c(C)ocn2)=O)(C)CO)oc(CO)nc1C N1(C(C(C)OCCC(C)C)=O)CCC2(CC1)C(NC(=O)CSC(=N)N)CS2(=O)=O C1(CC#N)CN(Cc2cc(F)ccc2Br)CCN1C(c1ccc(O)nc1Cl)=O CC1CN(C(C2(C)COC(=O)OC2)=O)CCC1CNC(=O)CCc1cn[nH]c1 CN1CCN(C(n2cc(Br)c(=O)c(I)c2)=O)CC1Cc1ccccc1 N1(C(CCNC(=O)OCC)=O)CCCCC1CNC.C1(C(=O)N)CCC1C(F)(F)F N1(C(C2CCC(NC(c3snc(C)c3N)=O)CC2)=O)CC(C)(C)C2COCC12 c1(C(N(CCOCCNC(CCC(C)CN(C)C)=O)C)=O)cc(F)c(F)cc1O c1(NC(CC)=O)cccc(NC(=O)Nc2c(C3CCOCC3)cnn2C)c1 N1(C(Cn2c(C)cnc2)=O)CC2(CCOCC2)CC1CNC(C1C2COCC12)=O C(=O)(C1Cc2ccccc21)N1C2C(NC(C=C(CC)CC)=O)CC(CC2)C1 c1(C(=O)OCC=C)c(CNC(c2nc(Cc3ccccc3)no2)=O)cnn1C C1(CC)CC(N=c2[nH]c(N3CCC4(CCC(C)CC4)C3)nc3c2CSC3)CCO1 C1(NC(c2cc(C)c(C)[nH]2)=O)CN(C(=O)Cc2ccc(F)cc2C)C2CCCC12 c1(C(=O)NC2CC(N(C(=O)CC3CC4(CC4)CO3)C)C2)ccc2c(c1)NCC2 c1(C(N2CCN(C(C3=NNC(=O)C3)=O)CC2CF)=O)cc2n(c1)CCCNC2=O Cc1cc(C(N2CC3CCC2CN(C(=O)C(C)(C)F)C3)=O)ccc1[N+](=O)[O-] C12(NC(c3n(C)cnc3)=O)CCC1CN(C(=O)CSc1n[nH]c(=N)s1)C2 n1(CC(=O)NC2(CNC(c3cc(C(=O)OC)no3)=O)CCOC2)c(C)ccc1C c1(NC(C(CCNC(C(CSC)O)=O)O)=O)ccc(CO)c(F)c1 c1(C2N(C(C3CCN(C(=O)OC(C)(C)C)CC3)C(=O)NC)CC2)ccc(F)cc1 Cc1nc2cc(C(N3CC(C(C)NC(=O)Cc4cncnc4)C3)=O)[nH]c2s1 C#CC1(NC(=O)CN(C(=O)Cc2ccc(O)nc2)CC)CC2CCCC12 N1(C(C(C2CCCCC2)NC(C(C=C)CC)=O)=O)CC2CC1CN2C c1(C(=O)OC)cc(CNC(=O)C(C)(C)CN(C)CCNC(N)=O)ccc1[N+](=O)[O-] N1(C(C(CCC)NC(N)=O)=O)CCN(C(=O)Cc2nncn2C)CC12CCC2 Cc1cc(C)c(C(=O)NCCCN2CCN(C(=O)CN(C3CCC3)C)CC2)s1 C(CCCCCC(=O)OCC(=O)NC1(c2ccccc2F)CCC1)SC c1(C(N2CCC(CC=C)(NC(=O)CN(C)CCO)C2)=O)ccnc(F)c1N c1(CC(=O)N(C)CC2CCC(=O)N2C)cc(Cl)cc(Cl)c1.C1CC(N)C1 N1(CC(=O)Nc2ccccc2Br)CCN(c2cccc(C(=O)O)c2)CC1 C1(C(=O)NCCCN(C(c2cn(CC(F)F)cn2)=O)CC)CCCCC1F c1(NC(N(c2ccccn2)C)=O)cnccc1NC(=O)Nc1csnc1Br N1(C(=O)Nc2nccc(COC)n2)CCC(CN(C)C)C(O)C1 c1(N2CCC(C(N(C(CC)C)C(C)C)=O)C2)cccc(OC)c1 C1(CNC(C(C)OC)=O)CC(O)CN1C(c1c[nH]c(=N)s1)=O N1(C(c2c(C)nc(CC)o2)=O)CC(NC(=O)CN(C)C2CC2)C(C2CC2)C1 C=CCC(C(=O)NC(C1CCN(C(=O)C(C)OCC)CC1)C)C(C)C c1(N(C)CC2CCCC2)nc(=NCC(F)CO)[nH]c2c1CC(C)CC2 c1(C(=O)NCCC2(OC)CN(C(c3cn(C)cc3C)=O)C2)cc(SC)oc1C Cc1nc(O)c(C(=O)NC(C)CCN(C)C(c2ncoc2C2CC2)=O)nc1C c1(C(=O)NCCCCN(C(CCC(=C)Cl)=O)C)cc2c(s1)CCCCCC2 C(=O)(C(CNC(=O)C(C)CO)CC(C)C)N1C(C#C)CCCC1 N(C(=NCCC1(OCF)CCOC1)NCCF)CCC(CC)Cc1ccc(F)cc1 N1(C(CCC(=O)OCC)=O)CCN(C(C2CCC3CC3CC2)=O)C(C2CCC2)C1 C(=O)(C(O)CC(N)=O)NC1CCN(C(C(C)N(C(=O)CC(F)(F)F)C23CC(C2)C3)=O)C1 c1(OC)cccc(Br)c1C(N1CC2CC(NC(C3CC34CCC4)=O)C1C2)=O C1(CNC(C=C(C)Cl)=O)CCCC(NC(=O)CCc2cnc[nH]2)C1 c1(OC)cccc(F)c1C(=O)NC1CC(N(C)C(c2nc(C)ccc2F)=O)C1 C(CN=c1[nH]nc(C(F)F)s1)N(C(=O)C=CC1(C)CCOCC1)C Cc1cnc2n1CCC(C(=O)NCCN(C(=O)Cn1cncn1)C1CC1)C2 C1(C#N)(C(N2CCC(=CCC(N(CC(=O)NC)C)=O)CC2)=O)CC12CCC2.CCO CS(=O)c1cccc(C(N2CC=CC(NC(=O)C(F)(F)c3csc(Cl)c3)C2)=O)c1 C=CCCCCCC(=O)NC(C)CN(C(C1CC2C=CC1CCC2)=O)CC c1(Cn2c(C(C3(C)CCCC3)NCCSCC(F)(F)F)nnn2)ccc(Cl)cn1 S(=O)(=O)(c1cccc(=NCCc2ncc(Br)cn2)[nH]1)NCC(C)(C)C1CC1 c1(C(=O)Nc2c(C(=O)OC)c(F)ccc2)[nH]nc2c(=O)n(C)cnc12 c1(CN(C(=O)CC=CCNC(=O)CSC2CC2)C(C)C)nccn1C Cc1csc(C(=O)NC2(C(N3CCCC(C(C)(C)O)C3)=O)CC2)c1Cl C1(NC(c2cscc2Br)=O)CN(C(C2CCC(F)(F)C2)=O)CC1O N1(C(C(C2CCOCC2)C)=O)CCC2(CC1)CC2NC(=O)CSc1ccncc1 c1(SC)ccnc(N2CCCCC2)n1.c12cnc(cn1)NCC1CCN(C1)C2=O C1(C(=O)NC(CN(C)C)CO)(CO)CCN(C(=O)CCCCC2CC2)C1 C1(NC(c2c(OCC)cccn2)=O)CN(C(=O)C(F)CC2CCC2)C2CCCC12 C1(NC(C(Cc2cc[nH]n2)NC(c2cc(O)cc(F)c2)=O)=O)COC2(CCC2)C1 CCC(C)CC(C(=O)NCCN1CCCOCC1)NC(=O)COc1ccccc1 Cc1coc(C(N2CCC(F)(CNC(=O)CC3CC(C(F)F)C3)C2)=O)c1C N1(c2ccc(S(=O)(=O)NCC3C(C)(C)C3)cc2Br)CCOC2(CCCS(=O)(=O)C2)C1 c1(CCC(=O)N(C(C)CCNC(c2cnccn2)=O)C)ccccc1[N+](=O)[O-] Cc1nc(C(=O)N(C(C)CNC(c2ccnn2Cc2ccccc2)=O)C)n(C)n1 c1(C(N(C2CCN(C(C3CCNC3=O)=O)CC2)CCC)=O)cc(C(C)C)nn1C C1(CNC(C=CCOC)=O)C2CCCC1N(C(=O)C1=CCCCO1)C2 n1(CC)ccc2cc(CNC3(CO)CCNC3)ccc12 N1(C(C2CC2C(=O)NCC#C)=O)CC(C)(NC(=O)CCC2CCC2)C1 c1(NCC2CN(C(C)C)C2)cc(NC(C2CCCCCC2)C)ncn1 CC1CN(C(c2cccc(Cl)c2)=O)CCC1NC(C1(OCC(F)F)CC1)=O C1(C(=O)NC2COC(=O)C2)(CC)CN(C(C23CCCC2C3)=O)C1 O(C=CC(=O)N(CC(C)N(C)C(C1CC1c1ccsc1)=O)C)CC C1(CC)CN(C(=O)Nc2c(Cl)cccc2Cl)CCN1C(c1cc(Br)cc(Br)c1)=O C#Cc1cccc(C(=O)NCC(CC)NC(C23CCOC(C)(C2)C3)=O)c1Cl C12(NC(c3ccnc(O)c3)=O)CCCC1N(CCN1C(=O)CNC1=O)CC2 C1(C(=O)NCc2c(C)noc2)CC(NC(=O)Cn2nnc(C)n2)C12CCC2 C(=O)(CC1COc2cc(O)ccc21)NCCCN(C(C(C(CC)O)C)=O)C C1(CC)(NC(=O)CC(C)N2CCCC2=O)CCCN(C(=O)C=C(C)C(C)(C)C)C1 CC1CC(C)CN(S(=O)(=O)N2CCC(N(C)C)C2)C1 C1(NC(COCCC)=O)CCOC(C2CCN(C(c3coc(SC)n3)=O)CC2)C1 N1(C(CCc2onc(C)n2)=O)CC(C(=O)NC(CN(C)C)CO)C2(CCC2)C1 c1(C(C)C)ccc(C(=O)NC(CNC(=O)Cc2ccc(O)cc2)C(C)C)cc1F Cc1oc(C#N)cc1C(N1CCCC1(C)C(=O)NC1(C2CCCC2)CC1)=O C1(CNC(c2onc(CC)c2C)=O)C(C)CCCN1C(c1cnc(C(C)C)[nH]1)=O c1(C(N2C(C)CC(NC(c3ccn(C)c3)=O)C2)=O)cc2cnc(Cl)cc2s1.C=O C1(C)(CCC(=O)N(CCC)C)CN(C(=O)C(C)C)C(C)(C)C1 C1(CNC(Cc2cn(C(C)C)nn2)=O)CC(C)(C)CN1C(=O)COC(F)F CN1CCC2CN(C(=O)CCN(C(c3ccc([N+](=O)[O-])o3)=O)C3CC3)CCC12 C1(CC(=O)N(C)Cc2ccc(F)c(F)c2)CN(C(C2COCCO2)=O)C(C)(C)C1 C1(C(=O)NCC2(C)CN(C(=O)CC3=CCCCC3)CCO2)CCn2nncc2C1 C1(NC(=O)C=CC(F)F)CCN(C(=O)CSC2CC2)CC1c1ccccc1 N1(C(c2scc(C)c2C)C(=O)NCCCC)CCS(=O)(=O)C(C)(C)C1 CCC(COC)C(=O)NCC(C)(C)CN(C)C(C1(C2CCCO2)CC1)=O c1(C(N2C(C(=O)NCC3(Cl)CC3)CCC2)=O)cc(C(F)(F)F)ccc1Cl c1(C(N2C(CCNC(c3nc(C)[nH]n3)=O)CCCC2)=O)cc(F)c(F)c(F)c1F N1(C(Cc2c(C)occ2)=O)CCC(C2(O)CN(C(C3CCC(C)CC3)=O)C2)CC1 O=S(=O)(c1ccc(Cl)cc1F)NC12CC(Nc3ncc4ccccc4n3)(C1)C2 n1(C(C)C)ncc(C(=O)NCC2(CCNC(c3cc(C#N)c[nH]3)=O)CC2)c1Cl C(=O)(CCCCCC(C)C)NC(c1cccc(C)c1)CNC(CC1C(CC)C1)=O c1(SCC)ccc(=NC(C)c2ccc(C(F)(F)F)cc2)[nH]c1N1CCN(C=O)CC1 CC1CCC(NC(=O)CCC2CC2)CN1C(C1(C2CCCO2)CCC1)=O N1(C(c2[nH]cc(C)c2)=O)Cc2ccc(C(C)NC(C3CCC(F)C3)=O)cc2C1 Cc1cc(=NC2CC(Oc3ccccc3)C2)[nH]c(=NCCc2ccc(F)cc2)[nH]1 C1(NC(c2cc(C3CC3)cc(C3CC3)c2)=O)CC2CN(c3ncns3)CC2C1 c1(CC(=O)NCC2(O)CC(NC(c3c(C)cn(C)n3)=O)C2)cccc2sccc12 C(=O)(C1=NN(CC)C(=O)CC1)NCCC(C(C)C)NC(CC1CC(CC)C1)=O N1(C(c2cscc2Cl)=O)CCCC2(CCN(C(c3ncncc3Cl)=O)C2)C1 N1(C(c2ccc(C(C)C)cc2)=O)CCCCCC1C(F)F CCC(C)C(O)C(C)C(=O)NC(C1CCCCN1C(c1nnsc1N)=O)C C(=O)(C1=Cc2ccccc2OC1)N1CC(NC(CC(C)C2CCCC2)=O)C1 C(CCN(C)C)(C(=O)NCC1(O)CC1)NC(C(C)SC)=O C1(NC(c2ccc(C(C)C)c(Cl)c2)=O)CC2CCC(C1)N2C(=O)CO.C1(N)CCC1 C1(NC(C2(C)CCCC2)=O)CCN(C(=O)CC2CC(F)(F)C2(F)F)C12CCC2 N1(C(C(C)OCCC=C)=O)CC2CC1(CNC(=O)C=CCCCC)C2 C1(C(=O)N(CC(C)NC(=O)Cc2ccno2)C)(OC)CCC(C)CC1 C12(C(N3CCC(C)C(CNC(=O)CN(C)CCO)C3)=O)CC(C)(C1)OC2C C1(NC(CC2C(C)(C)COC2)=O)CCC2(CC1)CCN(C(=O)CCC1CC1)CC2 c1(C(N2CC3(CCN(C(=O)C(F)C(F)(F)F)C3)C2)=O)c(F)cc(F)c(F)c1F C1(C(F)(F)F)(C(=O)NCC2(OC)CN(C(C3C(C(=O)OC)C3)=O)C2)OC2CCC1C2 C12(C(=O)NC3CN(C(CCc4c(C)noc4Cl)=O)CC3O)CC(CO)(C1)OC2C c1(NC)snc(C)c1C(=O)NCCC1CC(NC(=O)COCC2CCCC2)C1 C#CCC(C)(C)C(=O)N(C)CCC(N)(C)CC.C(=O)(C(C)(C)C1CCCO1)N C1(CN(CC(CC)C)C)CCCN(C(c2cccc(F)n2)=O)C1 Nc1cc(F)c(Cl)cc1C(N1CC2CC(NC(C3CCSC3)=O)CC1C2)=O C(=O)(C(C)(C)CC(F)(F)F)N(CC(C)NC(C12CCC(=O)N1CCS2)=O)C C1(C(=O)NCC2(NC(CC(C)C(F)F)=O)CCCCC2)CC2(C1)NC(=O)NC2=O Cc1nc(C)c(NC(c2cnc(-c3cnn(CCN(C)C)c3)cn2)=O)nc1C C(=O)(C1=CS(=O)CCC1)NC(CN(C(c1n(CC)nc(C)c1)=O)CC)CC CC1(NC(C2CCS(=O)(=O)N2)=O)CCCN(C(C2CCCC2(F)F)=O)C1 N1(C(CNS(CC)(=O)=O)=O)CC2(C1)C(NC(=O)CSC1CC1)CCS2(=O)=O N1(C(c2c[nH]cc2C(F)(F)F)=O)CCN(C(C2CCS2(=O)=O)=O)C2(CCC2)C1 CC1CCC(NC(c2cnsn2)=O)CN1C(c1cc(Cl)nnc1Cl)=O C1(C(N(C2CC(O)C2)C)=O)CCCN(C(=O)C(F)CC2CCOC2)CC1 c1(C(N2CCC(NC(=O)Cc3ccccn3)C(F)C2)=O)c(F)c(F)cc(F)c1F C(C(C)(O)C(=O)NC1CCCC1CC(=O)NCc1cn(C2CC2)cn1)OC NS(=O)(=O)c1ccc(NC(=O)NCC(c2cc(Cl)c(F)cc2F)=O)cn1 O=C1CCC(C(=O)NC2CC(CCCNC(=O)Cc3ccncc3)C2)O1 C(=O)(C(C(C)(C)C)NC(c1n[nH]cc1Cl)=O)NCC(C)Cn1cccn1 C1(C(=O)NC(C(C)NC(C2(C(F)F)CCOCC2)=O)CO)CC2CCCCCC12 c1(CC)cc(F)ccc1C(=O)NC1CCC(C)(CNC(=O)C=CC=C(Cl)Cl)C1 c1(NC(c2nnnn2CC2CCOCC2)(C2CCCO2)C)cccc(F)c1 C1(C(N2CCC(O)(CCNC(c3c(CC)nc[nH]3)=O)C2)=O)CCC(F)(F)CC1 Cc1cc(C)n2cc[nH]c(=NCCCNC3CCCNC3)c12 c1(OC)ccc(C(N2CCC(NC(C3(C)CCCN3C)=O)C(F)C2)=O)nc1OC Cc1nc2ccc(C(N3CC(NC(=O)COCCF)C(C4CC4)C3)=O)cc2s1 CCC(C)CC(C(=O)Nc1cccc(C(N)=O)c1)NC(=O)C(C)N=[N+]=[N-] C#CCCN=C(NCc1c[nH]nc1C)NCC1(CO)CCOC1 CC#CCCCC(=O)N1CC=CC1C(N1CCC(C)=C(C)C1)=O C1(C(=O)OCC)(C(=O)N)CCCCC1.CCC(C(=O)N1CCC1)OC.C(=O)(C1CC1)NC c1(C(N2CC(CNC(c3cnn(C)n3)=O)OCC2)=O)ccc2cc[nH]c2c1F c1(N(CC(=O)N(C2(CNC(C3CCC(=O)N3)=O)CC2)C)C)ccc(Cl)nn1 N1(C(C=CCOCCOC)=O)C(C(=O)NC2C3CN(C)CC23)C2CC(O)C1C2 Cc1cccc(C2CC2NC(=O)NC2CCC(CCOC(C)(C)C(F)(F)F)C2)c1 c1(C(=O)NC2CCCN(c3nc(O)cc(C)n3)C2)c(F)ccc2ccoc12 Nc1c(C(=O)NCC2CCN(C(C3CCC3(F)F)=O)C2)cccc1C(F)(F)F C1(OC)CC2CC(C(=O)OCc3ccc(SC)c(C)c3)CC2C1 C12CCCN(C1)C2=O.C(C)(C)(C(=O)NCC(C1CCC1)OC)NC(=O)NCC=C CCCC(C(=O)N(CC(=O)NCCCS(C)=O)C)OCC N1(CC)C(C)CN(C(C2COC(CNC(c3csnn3)=O)C2)=O)CC1C c1(C(=O)NC2(C)CN(C(C3CC3(C)C(F)F)=O)C2)cc2ccccc2s1 C1(NC(c2cc(C)cc(C)c2)=O)CCN(C(=O)Cc2sc(S)nc2C)CC1(C)C c12nc(cs1)CC(=O)NC(C1CCC1)CNC2=O.c1(C(NC=O)=O)csc(Cl)n1 c1(C(=O)NC(C(CO)NC(CCOC(C)C)=O)C)cccc(C2CC2)n1 C(C(C(=O)NCCn1cc(C(=O)NCc2cc(Cl)no2)nn1)OC)OC c1(C(=O)NCCCc2c(OC)cc(OC)c(OC)c2)ccc2c(n1)OCC(=O)N2 C(CNC(C1CN(C)C(=O)N1)=O)(C(=O)NOCc1ccc(C(N)=O)o1)N(C)C c1(C(=O)NC2CC3CC(NC(c4c(C)con4)=O)CC32)cc(N)c(F)cc1F C1(NC(c2ccc(CCC)[nH]2)=O)CCCC(NC(C2(C#N)CCC2)=O)CC1 C1(O)(C(C)NC(C2(C)CC2F)=O)CN(C(c2csc(CS(C)(=O)=O)n2)=O)C1 CN1N=CC(CC(=O)NCC2CC(F)(CNC(C3CCC(C)CC3)=O)C2)C1=O N1(c2ccc(S(=O)(=O)NC3CCN(C=O)CC3)s2)CCc2ccncc2C1 Cc1ncc(Br)cc1C(=O)NCC1CN(C(c2ccc[nH]2)=O)CCC1C N1(C(=O)CC2C=CCCC2)CCC2(CC1)CN(C(=O)CC1(c3ccccc3)CC1)C2 Cc1cnc(C=CC(=O)NCC2CC(C)N(C(c3ccc(C(C)C)s3)=O)C2)[nH]1 c1(C(N2CC(N(C(c3cc(C(C)=O)on3)=O)C)C2)=O)cc2c(C)nn(C)c2s1 c1(C(=O)NCCCn2cc(CC3(CO)CCC3)nn2)c(F)cc(Cl)cc1F Cc1ncc(C(N2CC(O)(C(F)C(N3CC(O)(C(C)C)C3)=O)C2)=O)n1C C=CC(C)C(=O)N1CCCC1CCCNC(=O)CC1CCOC1=O c1(NC(COC)C(=O)OC)ccc(CNC(=O)CC2CC3(CCC3)C2)nc1 C1(CCO)CCC(N2CCCC2C2CCOC2)O1 C1(NC(C(C)SCCCC)=O)CN(C(c2c[nH]c(=N)nc2O)=O)C2CCCC12 C1(NC(N2C(CNC(C3CCCCC3)=O)CC2)=O)CC2(CCC2)C1.c12cn-1nn2 N1(c2n(CCc3ncc(C)s3)c(C(C)C)nn2)CCC(P(C)(C)=O)C1 C1(NC(C2N(CC(C)C)CC2)=O)CC(F)(CNC(c2cnc[nH]2)=O)C1 C1(C)(C(=O)OC)CC(F)(F)CN1C(c1ccc(Cn2ccnn2)o1)=O CN1C(=O)COCC1CNC(c1coc(CNC(c2csc(Cl)c2)=O)c1)=O N1(C(C(CCC)n2cccc2)=O)CCC(C)C(NC(C2CC3CCC2O3)=O)C1C C1(C(=O)NC2CC(CC)(CC)C2)C2CCN(C(=O)C=CCO)CC12 C1(CC)CC(C)CN(C(C2CCCCCC2NC(=O)CC(C)(C)COC)=O)C1 Cn1cc(C(=O)NCC2(F)CC(CNC(=O)CC3CCCCC3)C2)cc1Br c1(C(=O)Nc2cnn(CC(F)(F)F)c2)ccc(-n2cncc2)cc1 c1(C(=O)NCC2N(C(=O)C(O)CC3CCOCC3)CCC2)ccc(O)nn1.C1(C)CC1 Cc1nc2cc(C(N3CCC(CNC(=O)C4=NNC(=O)C4)C3)=O)cc(Br)c2[nH]1 C#CC(CCC)NC(C12CC(NC(c3cccs3)=O)(C1)C2)=O c1(C(C(N2CCN(C(COCC#C)=O)CC2CF)=O)C)nc2ccccc2s1 c1(CN(c2n(CCCC(F)(F)F)nnn2)C2CCSC2)cc(F)cc(Br)c1 N1(Cc2c(C)csc2)CCC(NC(=O)CCOc2ccccc2Cl)CC1C CC1(C)C(CC(=O)NC2CC2OC2CC2)CCN1C(=O)CC1(C(F)(F)F)CC1 N1(C(C2(CCC=C)CC2)=O)CCC(O)(CCNC(=O)CCC(C)(C)C)C1 c1(C(=O)NCC(CCOC)NC(C23CCC2C3)=O)cccc(-c2ccncc2)c1 C1(N(C(c2c(C(C)C)[nH]cc2)=O)C)C2CN(C(=O)C(C(C)C)OCC(C)C)CC12 c1(SC)cccc(C(=O)NCC2(O)CN(C(C3CCC(C)O3)=O)C2)c1 C1(CNC(COC(CC)C)=O)CCC(N(C)C(C2CCCCC2)=O)CC1 C#CCC(C)(C(=O)N(C)CCc1ccncc1)NC(=O)C(CC)OC C(=O)(CCCCCn1cc(CC2(O)COC2)nn1)NC(c1cc(F)ccc1Cl)C c1(OC)ccc(C2CN(C(=O)CCC3CC3C(=O)OC(C)(C)C)CCO2)nc1C C1(NC(C(C(C)C)F)=O)CC2CN(C(=O)C(C)(C)N(C)C)CC12 CCCC(C)(CC)C(=O)NC1CC2CCC1C(NC(C1(F)CCC1)=O)C2 N1(C(CC(C=C)CC)=O)CCC(NC(c2ncc(C)cc2Br)=O)C(F)(F)CC1 c1(CC)nn(C)cc1C(N1CC(CC(=O)NCC(C)(CC)CC)CC1C)=O C1(C2(NC(=O)Cc3ccns3)CC2)CCCCN1C(C1CCCS1)=O C#CCCCC(c1nnnn1CC(C1CC1)OC)NC1CC1c1ccc(Br)cc1 C1(C(N(CCC(=O)OC)CC=C)=O)CCN(C(=O)C=CC2CC2)CCO1 C1(C(=O)NCC(=O)N(C2CC(=O)NC2=O)C)CCC(C2CC2)C1 C(=O)(C(F)C(C)CNC(=O)CCC(C)(C)OC)N(C(C=C)C)C C1(O)(NC(COCCOCC)=O)CCCN(C(=O)CC2CC(C)(OC)C2)CC1 C1(CNC(C(C)C2CC2)=O)CN(C(c2snnc2C(C)C)=O)CCO1 N1(C(C(=O)NCC=C)c2ccns2)CCC(C(N2CCCC2)=O)C1 N1(C(C(C)OCC=C)=O)CC(OC)CC(NC(c2cc(C)nc(C)c2)=O)C1 N1(C(=O)CCC2CCC2)CCOCC1Cc1cn(CC(F)(F)F)nn1 CC1(C)COCC(C(=O)NCC2(NC(=O)CC34COC(C)(C3)C4)CC2)O1 N1(C(C2=NOC(C)C2)=O)CC(NC(=O)CCN2CCC2)C2(CCS(=O)(=O)CC2)C1 c1(OC)cnc(C(=O)NC(C)CN(C(=O)CCN2CCCC2=O)C)nc1 c1(C(C)C)nn(C)cc1C(=O)NCCCC(C)(C)NC(=O)COc1ccsn1 C1(C(N(CCC(=O)OC)CC2CC2c2ccc(F)cc2)=O)CCCOCC1 C(C(CC(F)(F)F)NC(C1CC(CF)C1)=O)NC(=O)Cc1ccc(Cl)s1 Cc1cccnc1CC(N1CCC(N(C(=O)C(C)Sc2ccc(Cl)cc2)C)C1)=O C(=O)(C1=NNC(=O)C1)NC1CC(O)(CNC(c2cnc(CCCC)s2)=O)C1 C1(C)(CNC(C(CCC2CCC2)NC(C2C(C)C2)=O)=O)CCC(=O)N1C C=CC1(CC(N2CCCCC2CN(C)C(C2OCCOC2C)=O)=O)CCOCC1 C12(NC(C(C(C)C)N(CC)CC)=O)CC3CCC(C1C2)N3C(c1ncn(C)n1)=O c1(C(N2CCOCC(CNC(CC(=C)C)=O)C2)=O)cc2n(n1)CCCNC2=O CCC(CC)C(=O)N1CCC(Cn2nc(C)cc2C)C1.n12cc(nn1)C2 C1(C(=O)NC(CNC(C(C2CC2)OC)=O)(C)C)CCc2c(ncn2C)C1 N1(C(C=CC(CC)C)=O)CCC2(CC1)CCN(C(C1OCC3CCCCC13)=O)C2 N1(C(C2CC(NC(=O)CC3CC(C4CC4)C3)C2)=O)CCN2CC(O)CC2C1 C(=O)(N=c1ccn(-c2ncccc2Cl)[nH]1)C1N(Cc2c(NC)cc(C)cc2)CC1 C1(CNC(c2c(C)nc[nH]2)=O)CC2CC(C1)N(C(C1COCCN1C=O)=O)C2 C1(C(N2C(C(C)NC(=O)CC(C)(C)C)CCC2)=O)COc2ccc(F)cc2C1 N1(C(CCOC(C)C)=O)CCN(C(C2CC2CC(C)C)=O)C(C(F)F)C1 CCC(C)(C(=O)N1CCC(C)(CNC(=O)CCc2ccc(C#N)cc2)C1)C(F)F CC(C)C(C#N)C(=O)N1CCSCC1C(N1CC2(CC(F)C2)C1)=O C1(CC)(NC(=O)CNC(c2cncs2)=O)CCN(C(=O)Cc2ncccn2)CC1 N1(C(CCCOC)=O)CC(NC(=O)C(N2CCCCCC2)C)CCC1C CCC(C(=O)N1CC(C(=O)NCC(C)=C(C)C)C(F)C1)C(C)(C)CC C1(C(=O)NCCCN(C2CC2)CC)CC2(CCCO2)C1.C12=CC=C(C=N1)C2 Cc1cc(C)n2ccc(C(=O)N(CCCNC(=O)Cc3nonc3C)C(C)C)c2n1 N1(C(C2(C=C)CCOCC2)=O)CC2(CC(NC(C3CC3(C)C(F)(F)F)=O)CO2)C1 [N-]=[N+]=Nc1ccccc1C(=O)NCC1CCN(C(C2(N(C)C)CCCCC2)=O)C1 N1(C(CC(C)(C)NC(C2CCC(=C)CC2)=O)=O)CC2CCC=CC12 C1(C(=O)NCC2CC(C(=O)NC(C(=O)OCC)C3CC3)C2)CCC(C)C1 N1(C(C2CC(O)(CC#C)C2)=O)CCN(C(c2cscc2C)=O)CC1 c1(C(=O)NC(C(C)NC(C(C)SC(C)C)=O)(C)C)ccc(C)c(NS(C)(=O)=O)c1 C1(C(=O)NCCC=CC)CNC(=O)CN1C(=O)C=CC1CC1 c1(CC)nn(C)cc1C(=O)NC(C)(CNC(=O)COc1ccsn1)CC N#CC1(C(N2CC(CNC(=O)CC3COCCO3)C(O)C2)=O)CCSCC1 C=CC(C)CC(=O)N1CCOC(CNC(C2(CN3CCCC3)CCCC2)=O)C1 c1(CC(=O)NCC(C(=O)NC)CC2CCOCC2)cccc2nn(C)cc12 C1(NC(=O)CN2C(=O)CCC2=O)CC2(C1)CC(NC(C1CC3C=CC1CC3)=O)C2 c1(C(=O)NCC(C(=O)OC)CC2CCCC2)ccc(OC(F)(F)F)c(F)c1 c1(CC)cccc(C(=O)N(C2CN(C(c3cc(CC(C)C)c[nH]3)=O)CC2O)C)n1 N1(C(C2(CC)CCC2)=O)CCN(C(=O)Cc2ccc(F)cc2F)C2(CC2)C1 C(C(=O)N1CCC(N)N1S(=O)(=O)CCOC)c1cn(CC)nc1 N1(C(C2(c3cc(C)no3)CC2)=O)CCC(NC(=O)CC(O)C(C)C)C(O)C1 N1(C(C=CC=CC)=O)CC(C)(C)C1C1CCN(C(=O)CCc2cnn[nH]2)CC1 C1(CNC(c2c(C)coc2)=O)CC(C)N(C(c2cnc(CC(C)C)[nH]2)=O)C1 c1(C(=O)NCC2CC(OC)CN2C(=O)C=CS(C)=O)coc2cc(F)cc(F)c12 c1(C(N(C)CC2CCCN(C(C3N(CC)CC3)=O)C2)=O)c(Cl)ccc2c[nH]nc12 c1(NC(C2COCCN2C(C2CNC(=O)C2)=O)=O)ccc(C(F)F)cc1.C(CO)S C1(CNC(=O)CCOc2ccccc2)CN(C(c2nc(Cl)cs2)=O)C2CCN1C2 N1(C(CCn2ccc(C)n2)=O)CCC(C)(C)CC1C(=O)N(CC(F)Cl)C C1(CC(=O)NC(C=C)(C)CC)CCCCN1C(c1ccc(C(N)=O)o1)=O C1(C(=O)NCC2(C(N3CC=CCC3)=O)CC2)CC2C=CC1CC2 c1(C(N2C(CCC)CN(C(C3COCOC3)=O)CC2)=O)cc2c(Cl)cccc2s1 c1(C(=O)NCCCC(C)NC(c2cnn(C)n2)=O)cn(C)c(=O)cn1 C1(C)(CC)CCC(C(=O)NCc2ccsc2C(=O)NC2CC3C=CC2O3)O1 c1(OC)cc(=NC(=O)C(C)C2CCN(C(=O)C=CC(F)(F)F)CC2)[nH]n1C C1(CCC)CN(C(c2cc(C)c[nH]2)=O)CCN1C(=O)CC1NC(=O)NC1=O C(c1cncs1)=CC(=O)NC(C(=O)N(CCCN(C)C)CCC)C1(C)CC1 C1(CNC(=O)C=Cc2cncnc2O)(NC(=O)Cc2cc[nH]c2)CC2CCC1C2 O=C(CC(C(F)F)c1ccc(F)cc1Cl)NCC1CN(C(C2COC2)=O)CC1O S(=O)(=O)(c1cccc(=NCCCCCC(C)C)[nH]1)NC(CC(OC)OC)C c1(OC)ccccc1C(=O)NCCN(CCOCCO)C(C1CC1C(F)(F)F)=O c1(C(N2CCC(NC(CS(CCC)(=O)=O)=O)C2)=O)csc2ncnc(O)c12 C1(C(CC)NC(=O)C=CCN(C(=O)CN(C)C)C)CCOC1 C1(C(N2CC(CCC)C2)=O)CCCCC1(C)NC(c1cc(Cl)n(C)n1)=O Cc1cc(NC2CC3CN(C(=O)Cn4c(C)c(C)sc4=O)CC23)n2ncnc2n1 C12(CCNC(C3CSCCN3Cc3cccc(C(F)F)c3)=O)CCCN1CCC2 c1(CNC(C2CCN(C(C(C)OCCCC)=O)C2)=O)cccnc1O CCC(C)(C)C(O)C(=O)N(CCC(=O)N1CC(CO)CC12CCC2)OC C1(C(=O)Nc2cn(CC)c3c2cccc3)CC2CC(F)(F)CC(C1)C2=O C1(NC(c2cn(CC)nc2)=O)CC1C1CCCN(C(c2cocc2C)=O)C1 CC1CN(C(=O)CN(C)C2CC2)CCCN1C(c1cc2n(n1)CCOC2)=O N1(C(C(CC)=CCCC)=O)CCC2CCN(C(c3conc3C)=O)CC12 CC1CN(C(C2(C3CC3)CC2)=O)CC(C)N(C(c2cc3cccnn3c2)=O)C1 C1(CNC(c2n(CC)ccn2)=O)CCN(C(=O)C(C)(C)C#N)CCC1(F)F C1(CNC(=O)CSC(F)(F)F)CCC(NC(c2cn(-c3ccccc3)cn2)=O)C1 CCCC(CC1CCCC1)C(=O)NC1CCN(C(C2(COC)CCC2)=O)CC1F C1(CC(=O)NC(C2CCN(C(c3csc(C4CCCCC4)n3)=O)C2)C)CCCCC1 N1(C(c2ccc(C)nn2)=O)CC2CC1CN2C(C1(CO)CC(F)(F)C1)=O C1(=O)CCN(OC)C(=O)C23CC(C(C)C)(CN12)C3.C(C)(C)(C)OC(=O)OC c1(CC(CNC(C2COCC2c2ccccc2)=O)CO)ccc(F)cc1Cl N1(C(CN(C)CC)=O)CC(NC(=O)CN2CCCCCC2)C(c2ccccc2)C1 C1(NC(C(=C(C)C2CC2)F)=O)CCCCC1CNC(c1cccnc1S)=O C(C(CC1CCCC1)C(=O)NC(c1ncccc1C)C)NC(CSCCOC)=O c1(CC(C)C)ncc(C(=O)NCC(C2CCC2)NC(=O)CCC#N)[nH]1 c1(C(N2CCOC(C#N)C2)C(=O)NCCC)cc(F)c(Cl)cc1F C(C(C)(C)C(=O)NC1CCC(C(=O)NCCN2CCC(CO)C2)C1)N(C)C C1(CNC(=O)CC2CCSCC2)CCN(C(=O)CCCF)CC1C1CC1 CCCCCCC(F)C(=O)NC1CC(CNC(C2CC2CF)=O)C1 C(C)(CCC(F)(F)F)NC(CN(CC(=C)C)C)=O.C(=O)(C=CC=CCC)O C(=O)(C1c2ccccc2CN1S(=O)(=O)C1=COCC1)NC(COC)(C)C O=C1CCC(CC(=O)NC2CCOC2C(=O)NCc2ncsn2)N1 n1(CC(NSc2c3nnn(C)c3ncn2)=O)c(=O)oc2cc(Br)ccc12 N1(C(CC2ON=C(CC)C2)=O)CCN(C(=O)CN2CC3CCC2C3)CC1CO C(CCC(=O)NC1CC1NC(C1CCC1)=O)N(C)C.c1(C)cn(CC2CCCO2)nn1 C#CC1(NC(=O)CC2CCN(C(=O)CC(=O)OCC)C2(C)C)CC2CCCC12 C=CCCC(CC(C)C)C(=O)N1CCC(NC(=O)Cc2ccoc2)C12CC2 c1(CC(C)C)nc(C(=O)N(C2CN(C(=O)Cc3nncs3)C2)C)cs1 C(=O)(C(C)(C)C(=O)NC1CCC1NC(=O)CCCc1ccc(C)c(C)c1)OCC N(C(=NCC(C)Oc1ccccc1Cl)N1CCN(CC#N)CC1)CC N1(C(CNS(CC)(=O)=O)=O)CC2(CC2)CC1CNC(C1CC(OC(F)(F)F)C1)=O N1(C(C2(C)CC2F)=O)CCC2(CC1)CN(C(c1ccc(Br)c(F)c1)=O)C2 C(=O)(C(F)C(C)C)NC(CNC(CSC)Cc1nnc(-c2ccc(C)cc2)o1)C C(=O)(CC(C)(C(F)F)N(C)C)N1CC(C)C(NC(=O)C=Cc2ccncc2)C1 Cn1nc(C2CCC2)cc1C(N1CCC(NC(N2CCCCC2)=O)CC1)=O C1(C)(OCC(=O)OCC(c2ccccc2)C)CC(=O)N(C)C1.C1(=O)CCCN1 c1(-n2c(COC)nc(Cc3n(CCC=C)ncc3)n2)ccc(F)c(Br)c1 N1(C(CN2C(=O)C(C)C(C)C2=O)=O)CC(CO)C2(C1)CN(C(c1ccsn1)=O)C2 c1(CC(=O)NC2(C3CCN(C(=O)CC4=CCCC4)C3)CC2)n[nH]c2ccccc12 Cn1ccc(C(=O)NCC(c2ccccc2)CNC(c2scnc2C(F)F)=O)c1 N1(C(C2(NC(c3c(C)noc3)=O)CCCC2C)=O)C2CCC1CN(C)C2 N1(C(C(C)SC(C)C)=O)CC2CCN(C(c3cnc[nH]3)=O)CC2C1 c1(OC)ccc(F)c(C(=O)NCC2CN(C(=O)CCS(C)=O)C2)c1N Cc1nc2c([nH]1)C(C(=O)NC1(C)CCOC(C)(C)C1)CCC2 c1(C(N(C)CC2CCCN(C(C(C)CCN(C)C)=O)C2)=O)cc(F)c(F)cc1F c1(C(N2CCC(OC(C)C)CC2)C(=O)NCCC)ccc(C)nn1 N1(C(C(C)(C)n2cccn2)=O)CCCC(C)(C(N2CCC(CC(N)=O)C2)=O)C1 CN1CCOC(C(=O)NC2(CNC(C3(C(F)(F)F)CCCC3)=O)CC2)C1 c1(CC)ncc(C(=O)NC2(C(=O)NC(C)Cc3ccco3)CC(CO)C2)o1 N1(CC2(C)CCCOC2)CCCC(F)(F)CC1.c12cccc(c1)NC2=O C1(C(=O)NCC2CC(NC(=O)CCN3CCCCC3=O)C2)CCC=CCCC1 C(=O)(C(C)CC(F)F)N1CCC(C)(CC(=O)NC(C=C)C)C1 C1(C(C)C)Oc2ccc(C(=O)NCc3cn[nH]c3)cc2NC1=O CC(C)(C(=O)NC1CCC(Nc2cn(CCN3CC(O)C3)nc2)C1)C1CCCO1 C1(CCCNC(C2N(C(C)=O)CSC2)=O)CCCN(C(=O)CC2(C)CC2)C1 C(=O)(CS(=O)(=O)CCOC)NCC(CCOC)NC(c1cccc2ccnn12)=O c1(C(N2CC(NC(CCC(N)=O)=O)C(C3CC3)C2)=O)ccc(F)c2c1CCC2 C1(C(=O)NCC(CC(C)C)NC(C2CN3CCCC2C3)=O)CCC(C)(C)OC1 N1(C(CCNS(CC)(=O)=O)=O)CCCCC(NC(=O)CCC(C)(C)N(C)C)C1 C1(NC(CCC(=C)Cl)=O)CC12CCC(NC(c1cc(CCC)oc1C)=O)CC2 C1(CC)CN(C(=O)CCc2ccon2)CCN1C(=O)C(N1CCN(C)CC1)C c1(CCC)nc(-c2cn(C(C)(C)C)nc2Br)n(CCF)n1 C1(CNC(C2C(C)OC(=O)N2)=O)CC2(CCC2)CN1C(c1ccno1)=O C(=O)(C(N)CCS(=O)(=O)C(C)C)NC(C)(C)C=CC(=O)NC(C)C CCCCCCCNC(=O)CC1CCCN(C(C2(C(C)(F)F)CC2)=O)C1 C1(C(=O)NC(CC)CNC(=O)CSc2n[nH]c(=N)s2)CCC(C(N)=O)C1 C(=O)(C1=CCCC1)N1CC(c2ccc(C(=O)OCCn3cc(C4C(C)C4)nn3)o2)C1 C(C)(C)(CC(C)(C)C)NC(CC(C)N(C)C(c1ccc(O)cc1F)=O)=O c1(C(CC)C(=O)NC2CC(N(C(=O)Cc3cnoc3)C)C2)c(C)noc1C C(=O)(C(C(F)(F)F)C(F)(F)F)NCCCOCCNC(C1(CC#C)CCC1)=O c1(C(=O)NC2CCN(C(CCC(C)(C)C#N)=O)C2)cc(O)nc2[nH]c(=N)ccc12 Cc1n[nH]c(C)c1C(N1CCCC(CNC(=O)C=Cc2nccn2C(C)C)C1)=O N1(C(c2cc(C)ns2)=O)CCC=C(C(=O)N2CCC(C(=O)N(C)C)C2)C1 N1(C(C(CC=C)OC)=O)CCCC2(CCCN2C(=O)CC2(OC(C)=O)CCC2)C1 C12(CC(=O)NC3CC3NC(=O)CSc3nnc(S)s3)CCC(CC1)OC2 c1(C(=O)NCC2N(C(C3C(C)OCCO3)=O)CCC2)cccc2ncnn12 c1(C(=O)NCCN(C(C2CC(C)C2(C)C)=O)CC)cccc(CO)n1 C(CN=c1cc(C)nc(C(C)(C)C)[nH]1)OCCNC(c1cc(C)c(Cl)cc1C)=O CCC(C)CC(C)C(=O)N1CCC(N(C)C(C2(CS(C)(=O)=O)COC2)=O)CC1 N1(C(C(C)SCCCC)=O)CC(CNC(c2cc(Cl)no2)=O)C(F)(F)C1 CCC1=C(C(=O)N2CCC(NC(=O)Cc3nonc3C)C23CCC3)CCCO1 c1(C(=O)NC2(C)CCCN(C(=O)COCCF)C2)cc2ccccc2o1 CC12CCC(=O)N1CCN2C(C12OCCCC1C2(F)F)=O CC(C)(C)C(C#N)C(=O)N1CC(C(O)C(N2CCC(F)C2)=O)C1 N1(CCCn2cc(C(CC)N(C)C)nn2)CCCCC1C N1(CCC(=O)NCCCC(=O)OCC)CCN(C(C)C(=O)NC)CC1 CC1(CN)CN(C(c2sc(C(F)(F)F)nc2-c2ccccc2)=O)CC1(F)F c1(NCc2c(C)nc[nH]2)cn(C)c(Nc2ccnn2C)n1 CON=CC(=O)N(C1CCN(C(C2CC2C(=O)NCCO)=O)C1)CCO C1(CCC(=O)N(C(c2ccccc2)CNC(c2cc(Br)no2)=O)C)CCC(=O)N1 C(C(=O)N=c1ccn(CCC(C)C)[nH]1)(C1CC1)NC(CC(C=C)CCC)=O C(N=c1ccnc(C2CCC2)[nH]1)C1C(NC(c2cn(CC)nc2)=O)CCC1 C1(NC(c2nc(N)c(O)cc2)=O)CN(C(=O)C(F)CC2CC2)C2(CCCC2)C1 Cc1cc(COC2C(COCC(=O)N(CC(=O)N(C)C)C)COC2)on1 Cc1cc(C(=O)NC(C)CC(C)NC(C2CCCCO2)=O)nnc1C C(C1C(C(=O)NCCC(C)NC(c2ccc(C(N)=O)[nH]2)=O)C1(C)C)=C(C)C CCC(CC(=O)N1CCC(C(C)C(=O)NCC(C2CCCCC2)O)CC1)C1CC1 c1(OC)ccc2c(c1)CCN2C(c1ccc(C2CC2(F)F)cc1)=O CCCC(CNC(=O)COC(C)(C)C)C(=O)NC(C)Cc1ccnn1C c1(C(C(=O)NC(C)(C)CC)N(C2CCOC2)CC)c(C)nc2sc(C)nn12 C(=O)(C1=CC2(CCOCC2)C1)N1C(CC)C(NC(c2cncnc2C)=O)CC1 C(N=c1[nH]c(=NCCC2CC(=O)N(C)C2)c2ccccc2[nH]1)C1(COC)CC1 c1(C2C(NC(N(C)Cc3ccc(Cl)s3)=O)C2)ccccc1F C(=O)C#CC1CCOC1.C1(c2cn(CC(COCC)(F)F)nn2)COC(C)(C)C1 c1(C(=O)NCC2CCC(NC(c3cnc(CC)s3)=O)CC2)occ2c1CCOC2 c1(NC(=O)NC2CCOC(C(F)(F)F)C2)ccc(F)cc1OC(F)F C1(C2(NC(C=CCN(CC#C)C)=O)CC2)CCCCN1C(c1ccn(C)n1)=O c1(CC)nn(C)c(C(=O)NCC2CC3(C2)CN(C(C2CC(C)C2)=O)C3)c1Cl c1(NC)ncccc1C(=O)NC1CCC1NC(C1CCN(C)C1C)=O N1(C(CSc2ccc(OC)cc2)=O)CCCC(CNC(C2CC2C)=O)CC1 C1(C(=O)NCC2CN(C(=O)CC3CC=CC(C(=O)OC)C3)C2)CC2(CCO1)CC2 C1(C(=O)NC2(C)CCCN(C(C3CC4CCC(C3)C4)=O)C2)Cc2cccnc2C1 C(CCNC(=O)Cc1conc1C)(C(C)C)NC(Cc1cn(CC)nc1)=O c1(C(N(CCCNC(C(CSC)C)=O)C(C)C)=O)c(OC)nsc1OC C1(NC(c2[nH]c(C)c(-c3ccccc3)c2)=O)CCC12CCN(C(=O)C(C)C)CC2 c1(C(=O)NCC=CCC(=O)NC(C(COC)C)C)cc2cccnn2c1 C(c1c(Cl)cccc1Cl)=CC(N1CCC(O)(CNC(C2(C)CCOC2)=O)CC1)=O C(=O)(CC(CNC(=O)CCC1CC(C)C1)OC)N(CCCCOC)C C(=O)(C1=Cc2cc(Br)ccc2OC1)NCC(C)NC(C1(O)CCOC1)=O c1(C(N2CC3(CC)CC2(CNC(C2(CC)CC2)=O)C3)=O)cc2ccccc2cn1 N1(C(C2(C)CC=CC2)=O)C2CCC1CC(C(=O)NCCCC1CC1)C2 N1(C(c2c(CC)n(CC)nn2)=O)CC(NC(C2(C3CC3)CC2)=O)CCC1C Cc1oc(Br)cc1C(=O)NCC(C1CCCCC1)NC(=O)COC1CCC1 c1(C(=O)NC2CCN(C(C3(c4ccccc4)CC3)=O)C2)ccc2nc(O)sc2c1 Cc1cccc(C)c1C(O)C(=O)NCCCC(C)NC(C1CCCCNC1=O)=O CC(C)(CF)C(=O)N1CC(NC(c2cn(CCCF)nn2)=O)C(F)C1 c1(OCC)nc(C)ccc1C(=O)N(C1CCCCC1NC(C1CC1[N+](=O)[O-])=O)C C12(C(=O)OCC)CCN(CC(c3cc(Br)n[nH]3)NC3CC3)CC1C2 C1(NC(c2c(C)nn[nH]2)=O)CCC(C)(CNC(=O)CC2CC=CC2)C1 c1(C(=O)NCC#CCNC(C2CCC(C)C2)=O)cnc2cc(Br)ccn12 Cc1ccc(C)c(-c2nc3sc2c(=O)[nH]3)c1.N1(S(C)(=O)=O)C(C)CCCC1C CC1=NN(C)C(=O)C1CC(N1CC(O)(CNC(=O)CCc2cc(Cl)no2)C1)=O C1(NC(C(CC)OCC)=O)CN(C(=O)CCc2ccnn2C)CCC1F c1(C(N(c2ccc(SC)cc2)CC)=O)cc(Br)c2cn[nH]c2c1 C1(CNC(CNC(CCC)=O)=O)CN(C(=O)CC(=O)OCC)CCC1(F)F C(CCN(C(=O)C(c1ccccc1)SC)C)(C(C)C)NC(CCCC)=O CC1(C)C(NC(C2CCC(=O)N2)=O)CCN1C(c1c[nH]c(=N)o1)=O n1(CC(N2CCCC(CC(OCC)OCC)CC2)=O)ccc2cc(F)ccc12 C1(CC(=O)OCC)CCCCN1C(c1ccc(CC)s1)C(=O)NCCC1(C)CC1 c1(C(N(C(=O)CC(c2ccccc2)N(C)C)C(C)C)C)cn(CC(C)(C)C)nn1 C1(C(=O)Nc2ncc(F)cc2Br)CC(O)CCN1Cc1ccc([N+](=O)[O-])s1 c1(CC(C(=O)N2CCOCC2)Nc2ccccc2)cccc([N+](=O)[O-])c1 C(CNC(=O)CC1C=NN(C)C1=O)(CCCC)NC(CC1(OC)CCC1)=O C(=O)(C(CCOC)NC(c1ccccc1O)=O)NCC1C(CC)C1 C=CC(C)(O)CC(=O)N(CC(C)(C)CNC(C1(C)C=CCCC1)=O)C c1(C(N(C2CN(C(C(C(CC)C)C)=O)C2)C)=O)cc2c(C)cccn2c1 C1(OC)C(OC)CN(C(=O)Cc2cc[nH]c2)C1CNC(=O)CCN1CCCC1=O Cc1cccc(C)c1CNC(C1CCCN1C(=O)Nc1ccc(C#N)cc1)=O CON1CC(C(N2CCCCC2CC(=O)N(C)Cc2cccnc2)=O)CC1=O CCC(CO)(C(=O)N1CCC(CC(N2CC3(C2)CN(CC)C3)=O)C1)OC(C)=O C1(C(N(C(CC#C)C)C)=O)CCN(C(c2ccnnc2)=O)CC1(C)C N1(C(C(C2CC(C)(C)C2)OC)=O)CCN(C(=O)C2=NNC(=O)C2)C(CF)C1 c1(OCC)cccc(C(=O)NC(C2CCCCN2C(c2cn(C)cn2)=O)C)c1 C(=O)(CCCCN=[N+]=[N-])N1C(CC(=O)NC2(COCC)CC2)C2CCCC21 c1(C(N(CC(CNC(C(=O)N(C)C)=O)O)C)=O)nc2c(s1)COCC2 C1(CNC(C(C)(F)c2ccccc2)=O)COCCN(C(=O)CN2CCCC2=O)C1 c1(NC(=O)C(O)CN2CCCCCC2)cccc(CSc2ccccc2)c1 c1(NC(CC(=O)OC)=O)nn(C2CCOCC2)cc1-c1nn[nH]n1 N1(C(C2N(CCC)CCCC2)=O)CC(CNC(C2CCC2)=O)C2(CC2)C1 N1(C(C(=O)NCC(F)F)=O)CCC2(CCN(C(=O)CC3CCCCC3)CC2)C1 c1(C(=O)NC(CNC(c2c(C)ccc(N)c2)=O)(C)C(C)C)ccc(C#N)cc1O C=CCCCC(C1CC1)NC(=O)CCOCCNC(=O)COCc1nc[nH]n1 C(=O)(C1=CCC(F)(F)CC1)NC1C(CC)CN(C(=O)C=Cc2cncs2)CC1 C(C(C)(O)C(=O)NC(C)CCNC(=O)Cc1ccco1)OC c1(C2(C)COC2)ccc(NCCNS(C)(=O)=O)nn1 C(CCC(C)C(C(=O)NCC(C)C)N1CCN(c2cncnc2)CC1)=C(C)C N1(C(C(C(C)C)OC)=O)CC2CCC1C(CNC(C1(C)CC(C)(C)C1)=O)C2 C1(C(=O)NCC2CC(=O)NCC2)C2CCC(C2)C1NC(C12CCCN1CCC2)=O CN1CCCC(CC(N2CCSCC2C(=O)Nc2ccccc2O)=O)C1 C1(C(=O)Nc2ccno2)CN(C(=O)CCC2CCC2)CCN1 Cc1ccc(CC(C)C(=O)NC2CC(CNC(c3cn(C4CC4)cn3)=O)C2)cc1 c1(C(=O)NCCC(C)(C)NC(C2C(CC)CCO2)=O)ccn2nccc2n1 C1(NC(CCC2COC(C)(C)O2)=O)CC12CCC(NC(=O)CCC(F)(F)F)CC2 c1(C(=O)NC2CN(C(=O)CSC3CC3)C2)ccc(-c2coc(O)n2)cc1 CC(F)(F)CCC(C#N)N(C(C1CCC(C(F)F)CC1)=O)CCO c1(CNC(C2C3CN(C(C4C(CC)OCC4)=O)C2C3)=O)ccc(F)c(F)c1 N1(C(c2cnc(CCCC)s2)=O)CCC(O)(CCNC(C2CCCC2)=O)C1 c1(OC)ccccc1NC(N1CCOC(C(=O)Nc2nccs2)C1)=O Cc1cn2c(n1)CCC(C(=O)N(CC(O)CNC(=O)C(C)S(C)(=O)=O)C)C2 N1(C(C(C)OCCC=C)=O)CCN(C(C2CCN2CC)=O)C(CCC)C1 C(=O)(C(CC(F)F)N(C)C(c1ccc(Cl)s1)=O)N1CC(C(C)OC)C1 N1(C(Cc2cc(C)sc2)=O)CCOC2CCN(C(c3ccc([N+](=O)[O-])cc3)=O)CC12 C(CCS(C)=O)NC(C(C)N(C(C1CCNC1=O)=O)C1CC1)=O CS(=O)CC(O)COC(c1ccc(NCC(CO)CO)cc1)=O S(=O)(=O)(c1nn(C)cc1Cl)NCc1cc(N2CCCC(N(C)C)C2)ncc1 CCC(CC(=O)N1CC2CCN(C(=O)CCc3cnc(O)[nH]3)C2C1)C(F)F N1(C(C2ON=C(C)C2)=O)CCC2(CC1)CCN(C(=O)CS(=O)(=O)N(C)C)C2 C1(CNC(C(C(C)OC)NC(C=CCOC)=O)=O)COCC(=O)N1C C1(NC(C2C(CC)C2)=O)CN(C(c2ccc(OC)c(OC)c2)=O)CCC1(C)C N1(C(C(CCOC)C)=O)CCC(NC(=O)C(c2ccccc2OC)C)C1C C=C(C)CC(C(=O)N(C)CC=CC(=O)NCC1CC(=O)NC(C)C1)OC C1(C(=O)NC2(CN(C(C3C(=C)C3)=O)C)CC2)C(F)(F)C12CCC2 C#CCCCC(=O)NCCOCCOCCNC(C1(c2cc(C)on2)CC1)=O N1(C(CCc2cn(C)nc2)=O)CC2(C1)CN(C(C13C=CC(CC1)C3)=O)C2 Cc1cc(NCCN(C)C(=O)NC2CCOC(c3cccnc3)C2)cc(Br)c1 CC1CN(C(c2ncccc2Cl)=O)CC(C)C1NC(=O)CC1CN(C)C1 c1(SC)cccnc1C(=O)NCC1CC(C)N(C(=O)CCSCC(C)C)C1 C1(CC#C)(C(=O)NCCC2CN(C(c3ccn(CCO)c3C)=O)C2)CC=CCC1 C1(CC(=O)NC(C2CCCC2)CNC(C(CC)F)=O)CCN(c2nc(C)ns2)CC1 C(c1c(F)cccc1F)=CC(=O)NCC(N)=O.C12(COC1)C(=O)N(CC)C2 C1(C(C)(C)NC(C2C(C)=C2)=O)CCN(C(c2ccccc2SCCO)=O)CC1 C(=O)(C(O)C(C)c1ccccc1)NCCN(C(c1c(C)ncs1)=O)C c1(CC)occ(C)c1C(=O)NCc1ncccc1C(N1CCCC1C(C)CC)=O c1(NCCC2(OC)CCC2)ccc(S(=O)(=O)N2CC(C)C(F)C2)c(Br)c1 CC1NC(=O)OC12CN(C(C1(F)CCN(C(C3(CO)CCCCO3)=O)CC1)=O)C2 C1(C(C)NC(=O)NCCS(CC(C)C)(=O)=O)COc2ccccc2O1 N1(C(COCCCN=[N+]=[N-])=O)CCCCCC1C(N1CCC(C#N)C1)=O N1(C(c2c(C)nco2)=O)CCC2(NC(c3nn4cccnc4c3Cl)=O)CCCCC12 N1(C(C2CCC(=O)NC2)=O)CCC(C2CN(C(C3CS(=O)(=O)CCO3)=O)C2)CC1 N1(C(c2c(C(=O)OC)[nH]cc2)=O)CCOC(C)(CNC(=O)C(F)=C(C)C2CC2)C1 Cc1cc(C(N2CCC(C(=O)N(CC(C)(C)C)CC(C)C)C2)=O)c(C)cn1 c1(OC)ccc([N+](=O)[O-])c(C(=O)NCc2cc(Br)cnc2F)n1 C1(C(=O)NC2C(C)(C)N(C(c3cc(N)cnc3Cl)=O)CC2)CC2C=CC1C21CC1 c1(C(=O)NC(C23CC(CN2C(=O)OC(C)(C)C)C3)C)c(C)ccc([N+](=O)[O-])c1C C1(C(c2nnnn2Cc2ccc(Br)s2)NC2CCCC2)(OC)CC(C)(C)C1 CC1=NNC(=O)C1C(=O)N(CC(=O)N(C)Cc1ccncc1)C1CC1 c1(OC)ccc(N)c(C(=O)NCC(O)CN(C)C(c2ccc[n+]([O-])c2)=O)c1 C1(CCN(C(CC2(C(=O)OC)CC2)=O)C)CCCCN1C(C1CC2CC2C1)=O C(CC(=C)Cl)(C(=O)NCCC=CCCC)NC(C(C=C)C)=O N1(C(CC2CC(CC)C2)=O)CCC(C)(C)C1CC(=O)NCC(C)(C(C)C)OC N1(C(CCOCCCNC(CC2CCC(C)(C)O2)=O)=O)CC2CCCCCCC12 C1(C(N(c2cccc(NC(C3CCCN3N=O)=O)c2)CC)=O)CCC(C)C(C)C1 S(=O)(=O)(c1ccc2[nH]c(=NC(C)CCC(C)C)sc2c1)NCC1(CCC=C)CC1 C(c1ccc(Br)c(Cl)c1)=CC(N1CCC(c2nc[nH]n2)C1)=O c1(C(N2CCCC2(C)C(C)C)C(=O)NCC=C)n[nH]c(C)c1Cl c1(CC(N2C(C)CC(CNC(C(C)=C3CC3)=O)C2)=O)cnc2ccccc2c1 C1(CC(=O)N(C2CCN(C(=O)C=CC3CCOC3)C2)C)CCCNC1=O Cc1nc2n(n1)CCN(C(=O)CC13CCC1CN(C(=O)C1=CCCC1(C)C)C3)C2 C=C(F)CN=c1[nH]cc(C(=O)N(CC)Cc2cccnc2)s1 c1(C(N2CCN(C(CC(C)F)=O)CC2c2cn[nH]c2)=O)ccc(S(N)(=O)=O)nc1 c1(CNCC(c2ccccc2)(n2cc(CO)nn2)C)ccc(C(F)(F)F)cc1Cl C(C(C)(C(=O)N1CCCc2ccnn21)NC(=O)C=Cc1ccco1)SC C(=O)(C(F)(F)CCn1cc(C(C)O)nn1)NCC1(OCC)CCC1 C1(CN(C)C)COCCN1C(C1CC(F)CN1C(=O)Cc1ccc(Cl)cn1)=O c1(NCCN2C(=O)CNC2=O)nc(=NCc2cncc(F)c2)[nH]c2c1CCCC2 c1(NC(C(=O)NC(c2ccnc(Br)c2)C)=O)cccc(-c2cnn(C)c2)c1 c1(C(N(C2CCN(C(C(C(CC)O)(F)F)=O)C2)C)=O)ccc(O)c2ccccc12 C(=O)(C(O)C(C(C)C)CNC(c1cc(CC)[nH]n1)=O)N1C(CO)CC(OC)C1 O=C1Cc2cc(C(N3CCC4(NC(=O)CC(Cl)Cl)CC4C3)=O)ccc2CN1 C1(C(N(C)CC2CCCN2C(C23CC(O)C2C3)=O)=O)CCC(=O)N1CCC(F)(F)F C(C(C)(C)CNC(C1(N(C(=O)CCC2CC(C)C2)C)CC1)=O)OC C(=O)(CC1OCCc2ccccc21)NCC(C)CNC(=O)CCCC(C)(C)C#N C(N=c1[nH]c(=NCC2CN(C(N)=O)C2)c2ccccc2[nH]1)c1ccc(OC)s1 C(=O)(C1CCCc2nccn21)Nc1c(C)cc(NC(c2cncn2C)=O)cc1 S(=O)(=O)(c1cnn(C)c1)NCC(=O)NCC1OCCN(C(C(C)OCC=C)=O)C1 C(=O)(CS(=O)CC(=O)C(c1ccc(F)cc1)c1nc(C2CC2)no1)OC Cc1nc2c(C(=O)NC3CC(C)N(C(c4cc(C)c(C)o4)=O)C3)cccc2o1 C1(NC(C2CC(NC(CCCCOC)=O)C2(C)C)=O)CCN(C)C1(C)C c1(CC(=O)NCC(C)CNC(c2c[nH][nH]c2=N)=O)ccc([N+](=O)[O-])cc1 c1(CC)ccc(CCC(=O)NCC#CCNC(=O)CSCC(N)=O)cc1 c1(NC(C(N2C(C(=O)OCC)C(=O)NCC2)=O)=O)ccc(OC)c(OCC)c1 Cc1ccc2c(ccn2CCC(N2CC3CCN(C(c4cnc[nH]4)=O)CC23)=O)c1 CN1CCC(C)(C(=O)NCC2CC(F)(CNC(c3cc(CO)[nH]n3)=O)C2)C1=O C1(OC)(CNC(c2cncc(CO)c2)=O)CCCCC1C.C12(CC1)CC(=O)NC2 C12(C(=O)NCC3(O)CN(C(=O)C=CC(F)F)C3)CCC(CC1)O2 c1(NC(=O)CC2CCCN2C=O)cccc(C(F)F)c1.c1(CO)ccccn1 S(=O)(=O)(c1ccc(N2CCOC(C)CC2)c(Cl)c1)N(CC(CC)OC(C)(C)C)C C(=O)(CCCC(=O)c1ccns1)NC1CCN(C(C(C)CBr)=O)C1 CCCC(CCC)C(=O)N1CCC(NC(c2nnc(-c3ccccn3)o2)C)C1 c1(C(N2CCN(C(c3c(C)c(F)ccc3)=O)CC2CO)=O)csc2c(F)cccc12 c1(C(=O)NCC2CN(C(CCCOCCC)=O)CC2O)coc2c(C)cccc12 c1(OC)cc(C(=O)NCC2CC(C(=O)NCc3cc(O)no3)C2)ncn1 CCCCC(CC(=O)NCC1CC(O)C(O)C1)NC(=O)CN(C(=O)COC)C N1(C(CSCCC(C)C)=O)CC2CC(C1)CN(C(C1CCOC1)=O)C2 C(CCCCC(=O)N1CC(NC(=O)COCCCC(C)C)CCC1C)SC C1(NC(Cc2cc(CC)nn2C)=O)CC2CC(C1)N(C(c1cccnc1O)=O)C2 c1(OC)ccnc(F)c1C(=O)N(CC(O)CNC(=O)C(C)NC(C1CCC1)=O)C C1(NC(c2cc(CC)nn2C)=O)CCN(C(C2CC(C#N)C2)=O)CC1(C)C C1(CNC(C(C)C)=O)C=CCN1C(=O)Nc1cc(-c2cnn(C)c2)[nH]n1 C1(NC(C2CCCC(NC(C(C(C)C)O)=O)C2)=O)CCC(O)C(O)C1 CC1CC(C(N2CCOC(c3ccccc3)C2)C(=O)NCC2CC2)CC(C)C1 c1(C(=O)OCC)c[nH]ccc1=NC1(CC)CCCCN(C(c2cnsn2)=O)C1 N1(C(c2c(C)noc2)=O)CCC2(C=C(C(=O)N(CC(C)O)C(C)C)C2)C1 C(CC(=O)NC1CC2(CC2)C1)(C(F)F)NC(C(C)C1(O)CCC1)=O C1(CC(N2CCCC(NC(c3ccn(CCOC)n3)=O)C2)=O)CCOCC1(C)C C(=O)(C1=Cc2cc(F)ccc2OC1)N(C(CNC(C1(C)CC1)=O)C1CC1)C C(=O)(CC(C)(C)C#N)NCCC(=C)CNC(=O)C(C)Cc1cccc(Br)c1 C1(C(=O)NC2CC(CNC(CCN(C)CCO)=O)CC2O)CCc2ncnn2C1 C(CNC(C1CC2CCC1O2)=O)(CC(F)(F)F)NC(c1cc(C(C)C)[nH]n1)=O c1(CCC)cc(C(=O)NC2(CCNC(C3(C(=O)OC)CC3C)=O)CCC2)c(C)o1 N1(C(c2cn(C)nc2SC)=O)CC2CCC1C(C(=O)Nc1c(OC)ccnc1)C2 CC1CC(NC(=O)CCOCCN(C)C)CCN1C(=O)C(C)(C)C1CCCO1 N1(C(C(CSC)OC)=O)C(C(=O)N(C2CC=CC2)C)CCC1C(C)C CCC(F)(F)CC(=O)NCc1cn(C2CCCN(C(C3(C)CC3)=O)C2)nn1 c1(C(N2CCC(NC(c3n(C=C)nnc3)=O)(CC)CC2)=O)ccc2[nH]nc(O)c2c1 CC(C)C(C(=O)N1CC(N(C)C(C2(c3cc[nH]n3)CC2)=O)C1)n1ccnc1 c1(C(C(=O)NC2CCCN(C(c3c(C)nn[nH]3)=O)C2)O)cc(F)cc(F)c1 c1(C(=O)NC(C(c2ccccc2)NC(c2c(C)onc2)=O)C)cc(=O)n(C)cn1 C(=O)(C(O)CC(F)(F)F)N1CC(NC(c2cccnc2OC(F)F)=O)C2(C1)CC2 C1(NC(CC=C)=O)CC2(C1)CN(C(c1cnn(CC3CCCCO3)c1C)=O)C2 c1(NC(C2CCN2C(=O)CCC2CCCC2)=O)cccc(F)c1F C1(CS(=O)(=O)N(CCN(C)C)C)CC2C(C1)C2(F)F C(C(C)C(=O)NC(C)(CNC(=O)CCSc1n[nH]c(C)n1)CO)OC c1(C(=O)NCC(=O)NCC(=O)N(C2CCCC(O)C2)C2CC2)cc(O)cc(F)c1 c1(C(=O)NC2C(CNC(C(COC)C)=O)COC2)nn(C)c2c1CSCC2 N1(C(CCC(=C)Cl)=O)CCC(C)C(NC(=O)C#CC2CC2)C1 C(=O)(C(O)C1=CCCCC1)N1CCC(CCCNC(c2c(C)ocn2)=O)CC1 CS(=O)(=O)c1cc(N2CC3CC(NC(=O)Cn4nnc(C5CC5)n4)CC2C3)ncn1 C1(Cn2cc(C(C(=O)OC)(C)C)nn2)CCCN(C(=O)C(C)CSC(F)(F)F)C1 C1(C(=O)NCCC2CN(C(CCNC(COC)=O)=O)C2)CCC(C)O1 N1(C(C(C2CC2)NC(C2N(C)CC2)=O)=O)Cc2c[nH]nc2C1 CCCCCCCC(F)C(=O)NCCCCN(C(=O)C(O)C(C)CC)C O=C1CC(C(=O)NCC2CN(C(=O)CC3CCCOCC3)CCCO2)CCCN1 c1(SC(c2ccc(Cl)cc2)C)ccc(CN2CC(CS(N)(=O)=O)C2)cc1 c1(C(=O)OC)ccc(NC(=O)CC2CCCN2C(c2ccccc2Cl)=O)cc1 c1(OC)c(Cl)cccc1S(=O)(=O)NCCCC1=CCNCC1 C(=O)(CC(F)(F)C(F)F)N(C(C)C)CCNC(=O)COc1nn(C)cc1Br C1(C)(CC)CN(C(=O)NCc2cn(C)nc2OCn2ccc3ccccc23)CCO1 Cc1[nH]c2ccccc2c1S(=O)(=O)N1CCN(C(=O)CCC(N)C(N)=O)CC1 C1(CNC(CCc2ccn(C)n2)=O)CN(C(C2(C)CNC(=O)C2)=O)CCC1(F)F N1(CCCC)CCCC1CNC(=O)CC1CCCC1NC(C1(N(C)C)CC1)=O N1(CCOC)CCOCC1CSc1ccnn1C.C1(N2C(=O)C2)CCCCC1 Cc1cccc(C(=O)NCC2(NC(c3cc(C#N)cn3C)=O)CCOC2)c1F N1(C(CNS(N)(=O)=O)=O)CCC(C2CC2)C1CNC(c1n[nH]cc1Cl)=O CN1C(=O)CSC1=CC(=O)NCC1CC(NC(=O)COCCc2cccs2)C1 C1(N(C)C(c2ccon2)=O)CN(C(C2CCC3(CCC3)O2)=O)CC12CC2 C1(CNC(c2cnns2)=O)CCCC(NC(=O)C(c2ccc(O)cc2)=O)C1 C1(NC(c2cnnn2C2CC2)=O)CC2CCC1N(C(=O)Cc1cnsc1)C2 Cc1ccc(O)c(S(=O)(=O)NCCOCc2ccc(Cl)c(Cl)c2)c1 C1(CCC=C)CCCN(C(c2nocc2C)C(=O)NCCCOC)C1 N1(C(c2n[nH]c(=N)s2)=O)CC=CC(NC(c2ccc(C(F)(F)F)[nH]2)=O)C1 c1(OCC)ccc(F)c(C(N2CCOC(CNC(=O)CCSC(C)C)C2)=O)c1F O=C1COc2ccc(C(=O)NC3CCCN(C(C4CCO4)=O)CC3)cc2N1 Cc1cc(N2CCCC(CCNC(C3CC(C)C3)=O)C2)n2nc(C)cc2n1 C(=O)(CC(C)CC(C)(C)C)N1CCCC(CCC(=O)Nc2c(C)scc2)C1 c1(NC(C2CCN(C(C3CCCOC3)=O)C2)=O)cccc(O)c1 C1(CC(=O)NCC2CCN2C(C2CCCC23CC3)=O)COc2ccccc2O1 N1(C(C2C(CC)C2)=O)CC2CCCC1C2CNC(c1ccc(C)cc1)=O N1(C(C(C)OCC(C)C)=O)CC2(CCCC2NC(=O)C=Cc2cnn(C)c2)C1 c1(C(N2C(CNC(C(C(=O)OC)C)=O)CCCC2)=O)ccc2sccc2c1 C(C)(CC(N)C(=O)NCc1cnc(N2CCOCC2)nc1C)OC c1(C(N2CC(F)CC(NC(C(CC#C)C3CC3)=O)C2)=O)cc(C)c(F)cc1F c1(OC)ccc2sc(C(N3CC(C(=O)Nc4cc(O)nc(SC)n4)C3)=O)cc2c1 N1(C(c2cccc(C(=O)O)c2)=O)CCC(C(F)(F)F)C2(CCOCC2)C1 c1(C(=O)NCC2CC(NC(C=C(C)Cl)=O)C2)ccc2c(c1)NC(=O)C2(C)C n1(CC(=O)N(C2(CC=C)CCN(C(=O)C=CC=CCC)C2)CC)ccc(O)nc1=O C(=O)(C1=NOC(C)C1)NC1C(CNC(c2c(CC(C)C)n(C)nc2)=O)C1 CCCCCC(O)CC(=O)NCCCC(CCC)NC(=O)CC(C)(C)C c1(OC)ccc(Br)nc1NC(=O)CC1CC2(C1)CN(C(c1nc(C)sc1C)=O)C2 C1(NC(CC(C)SC)=O)CCC2CN(c3cc(Cl)c(O)nn3)CCC2C1 CC#CCCCC(=O)NCC1(COC)CCN(C(=O)C(CO)C(C)C)CC1 c1(-c2n(CC)nc(CS(C)(=O)=O)n2)c(F)ccc2c1OCC2 Cc1cccc(C(=O)N(CCN(C(=O)Cc2nnsc2Cl)C)C(C)C)c1 Cn1nc2ccccc2c1S(=O)(=O)NC(C1CCCOC1C(C)(C)C)=O c1(OC(C)C)ncccc1C(=O)NC(C1CN(C(=O)C(O)C2CCC2)CCO1)C Cc1cc(C)c(C(=O)NC(c2nocc2C(=O)NCCC2CC(O)C2)C)o1 c1(OC)n[nH]cc1C(=O)NC(CN(C)C)C(=O)NCCCn1ccnc1 c1(CC)cscc1C(=O)NCCCC(C)NC(=O)C(n1ccc(C2CC2)n1)C Cc1ccc(F)c(-c2nnc(NC(N3CC(C)C(C)C3C)=O)o2)c1F c1(Cc2cn(CCC(N3CCC(CN=[N+]=[N-])C3)=O)nn2)ccc(Cl)cc1F c1(C(N2C(CNC(C(CC)SC)=O)CC(C)(C)C2)=O)cnc2c(c1)NCC2 c1(C(N2CC(C(C)(C)O)(CNC(COC(CC)C)=O)C2)=O)cc(C)[nH]c1C CN(CC(F)(F)F)N(CC)C(=O)CCc1ccccc1 N1(C(C(C)Cn2cccn2)=O)CCN(C(c2ncccc2O)=O)CC1CC(F)F N1(C(c2scc(C)c2C)=O)CCC2(CCCC2NC(c2ncccc2C)=O)C1 C(C(C)(CC(C)C)NC(C1CC1C(F)(F)F)=O)NC(c1c(C)n(C(C)C)nc1)=O C(CCCCC(=O)N(C)CC1CCN(C(C2C3CC(=O)CC23)=O)C1)SC N1(C(CCN(C(C)=O)C)=O)CCSCC1CCNC(=O)Cc1cscn1 c1(C(C(=O)NCC(CC)NC(=O)Cc2scnc2C)O)ccnn1C N1(C(C2(CC#C)CCOC2)=O)CC(C)(CNC(=O)CSCCCC)CC1(C)C N1(C(c2c(C)nsc2)=O)CCC(NC(c2cc(=O)n(C)s2)=O)C(CO)CC1 CCCCC(O)C(C)C(=O)NCC1CC2CCCC2N1C(c1cnc(C)cn1)=O Cc1c(N)ccc(C(=O)NC2CC(CNC(C3CC4CC3CC4(F)F)=O)C2)c1C N(C1CCc2cc(F)ccc21)C(c1nnnn1CC1CCCO1)CCC O=C1CSc2ccccc2N1CCNS(=O)(=O)c1ccc(CN2CCCC2)cc1 CCCC(CNC(C1CN(CC)CCO1)=O)C(=O)NCC(F)(F)C(=O)OC N1(C(c2c(C)cccc2)=O)CC(CNC(c2cccc(C)c2C)=O)C(C)CC1C CC1CC(N=c2[nH]c(=NCCC3(C)CCC3)[nH]c3c2CCCCC3)CN1C Cc1cnc(C(N2CCC(C)(NC(C3CCCN(C(C)C)C3)=O)C2)=O)cc1C#N Cc1cccnc1C=CC(=O)NCC(C(C)(C)C)NC(=O)C=CS(C)=O c1(C(N2CCC(C(C)NC(COCCC#C)=O)C2)=O)cc(Cl)cc2c1OCC2 CN(C)S(=O)(=O)NCC(N1CC(CCNC(C2(CO)CC2(F)F)=O)C1)=O c1(C(N2C(C)(C)CC(C(=O)NC3CCC=CCC3)C2)=O)ccnc2cc[nH]c12 C1(C(=O)NC(C2CCCN2C(=O)C(=O)C2CC2)C)CCCN(CP(C)(C)=O)C1 c1(C(=O)OC)cc(C)c(C(N2CC3CC3(NC(C3CCCC3)=O)C2)=O)o1 C12(C(N3CCC(C)(C)C3CNC(C3CNC(=O)C3)=O)=O)CC(C)(C1)OC21CCC1 C(=O)(C(CC)(CC)CO)NCc1cncc(C(=O)NC2CCN(CC)CC2C)c1 c1(NC(c2ccc(OC)cc2)c2ccccc2)ncnc2c1cnn2C C1(C(=O)NC2(CC#C)CCC2)COCCN(C(C2C(OC(C)=O)C2C)=O)C1 c1(CNC(CC(C)C2CC2)=O)ccc(CN(C)C(c2cccnn2)=O)cc1 C1(CC(=O)N(C2CCC3(CC2)CC3)C)CC2(CC2)CN1C(=O)CC1CCCO1 c1(C(N(C(C)C(=O)NC(C)(C)CF)CC)=O)cc[nH]c2nccc1-2 C(C(O)C(=O)NC(C)CC(C)NC(c1csnc1C)=O)=CC CCC(C)(CCO)NC(=O)C(C)CNC(=O)Cn1cccn1 CCC(COC)C(=O)NCC(N1CCN(C(C2(C)CC2(F)Cl)=O)CC1)=O N1(C(c2c(C)con2)=O)CCCOC(CNC(c2ccncc2F)=O)C1 C(=O)(C1=C(C)CCNC1)NC(=S)Nc1ccc(OCC(F)(F)F)cc1 N1(C(C2N(C)CCN(C)C2)=O)CCC(C)(C)C(CNC(C2CCCCS2)=O)C1 C(C(COC)CC(=O)NC1(C)CC(C(N2CC(SC)C2)=O)C1)OC C1(COC)CCCN(C(=O)C=CC(C)(C)NC(=O)C(n2ccnc2C)C)C1 c1(C(N2CC3C(CNC(CNC(C)=O)=O)(C3)C2)=O)ccccc1NC1CCC1C C=CCC(CNC(=O)C(C)n1cnnn1)C(=O)NCCCCC1CCCO1 C#Cc1cnn(CC(=O)NC2CC(C)(NC(c3cccc(CC)n3)=O)C2)c1 Cc1cnc(F)cc1NC(=O)COc1ccccc1.C12(CCCC1)CO2 c1(CCC(=O)NC23CC2CN(C(=O)CSc2ccccc2)C3)cc(Br)ccc1F C1(CN(C(=O)C(F)C2CC2)C)CN(C(=O)CNS(N)(=O)=O)CCO1 C(CC(C)C(=O)N(C(C)CCNC(c1cc(C)nn1C(F)F)=O)C)=CC CCCC(C)(C)CC(=O)N(CCN(C(=O)CSc1cccc[n+]1[O-])C)C1CC1 C1(NC(c2c(C)ocn2)=O)CN(C(C2CC3CCCC23)=O)Cc2nccn2C1 c1(OC)cc(OC)c2ccccc2c1.N12CCc3nn(C)cc3C1CNC2=O C(CCC(C)(C)C(=O)Nc1cnn(C)c1Cl)OC C1(CNC(C2C(C(=O)OC)C2)=O)CCN(C(c2cccc(SC)c2)=O)C12CCC2 c1(-n2c(CC(CSC)C)nc(C3CCSC3)n2)cc(C)ccc1C C1(CN(C(=O)Cc2cncn2C2CC2)C)CCCN(C(=O)Cc2csc(S)n2)C1 CCC(CC)C(=O)NCCCN(C(C1(C)CC1(F)F)=O)Cc1ccccc1 C=CCC(C(=O)NC(CC(=O)N1CC(CO)C2(CC2)C1)C(F)(F)F)C(C)C C#CCC(C)C(=O)N1CC2CC2(NC(c2ccc(-c3cccc(F)c3)o2)=O)C1 c1(C(=O)NCCCC2N(C(c3c(N)non3)=O)CCCC2)cc(F)cc(F)c1 CC1CC(NC(=O)Cc2cccc(O)c2F)CCN1C(c1cnc(Cl)s1)=O C(=O)(C1=Cc2ccccc2C1O)N1C(CCNC(c2c(C)occ2)=O)CCC1 CC1(C(=O)NCCNC(C2CN(C(C3CC3(C)C)=O)C2)=O)CCSCC1 CCC1=NOC(C(=O)NC(C)(CSC)C(=O)N(C(C)CN(C)C(C)=O)C)C1 C1(CC)C(NC(=O)Cc2c(C)cnn2C)CCN1C(=O)Cc1ccc(O)nc1 c1(OC)ccc(C(=O)NCCCCc2cn(-c3ccnc(Cl)c3)nn2)nc1 C12CCCCCC1N2.c1(OCCNC(=O)OC(C)(C)C)ccc(Cl)c(Cl)c1 c1(OC)ccc(CCCC(=O)N(CC(O)CNC(=O)Cn2nnnc2C)C)cc1 n1(CC)cc(C(=O)NCCC(C)NC(=O)CCOCC(F)F)nn1 c1(N(CC(C)NC(CC(n2c(CC)ncc2)C)=O)C)nc(Cl)nc2c1cnn2C C1(NC(c2cocn2)=O)COCC1C(=O)NCCCn1ccnc1 Nc1c(C(N2CCCN(C(=O)CC3CCOC3)CC2CO)=O)cccc1[N+](=O)[O-] C1(CC(=O)NCC2CC(NC(C(c3cncn3C)N(C)C)=O)C2)CCC(=O)NC1 CC1Oc2ccc(C(N3CCC(C4CCC4)C3)C(=O)NC3(C)CC3)cc2C1C c1(NCC)ccc(C=CC(=O)NCC(CNC)C)o1.C1(C=O)C2COCC12.C(C)N C=C(C)CN=C(NCCC1CCCO1)N1CCCC(OCCCOC)C1 C1(N(C(C(C)OCC=C)=O)C)CC2CC1N(C(=O)Cc1csnn1)C2 CCC(C)(COC)C(=O)NC1CN(C(=O)C(SC)SC)CC1F c1(C(=O)NCC2(F)CC(CNC(c3c(CC)nn(C)c3)=O)C2)ccc(C)nc1O CC1(C(=O)NC2CCCCN(C(C3CC=CCO3)=O)C2)COC(=O)OC1 C(=O)(CN=c1ccc(Cl)n[nH]1)N(C)CCNC(=O)C(O)CCS(C)=O c1(C(N2CCCC(CN(C(CCC)=O)C)C2)=O)ccc2oc(O)nc2c1 C(C1COCc2ccccc21)Nc1cc(N(N2CCN(C)CC2)C)ncn1.C1(C)CC1 C(=O)(C1Cc2c(Cl)cccc21)NC1(CCNC(CCOC)=O)CC1 Cc1nc(C)c(-c2cn(CCNC(=O)CCOc3ccccc3F)nn2)s1 c1(C(=O)NCC(CNC(CC(C)CN(C)C)=O)O)cnc(O)c2ccccc12 CCC(O)C(C)C(=O)NCCC(C)(C)C(=O)NCCCCC(C)(C)C C1(CCC)CCCN(C(=O)CC2CN(C(=O)C(C)CO)CCC2C)CC1 N1(C(Cc2c(C)occ2)=O)CCCC(C(C)NC(C2CC=CC2)=O)C1 C1(N(C(=O)CCCOc2cccnc2)C)CCCN(C(=O)C(C)(C)CC2CC2)C1 c1(OCCCC(N2CCC(N(C(=O)C(C)C)CCC)CC2)=O)ccc(C)cc1 C1(CS(=O)(=O)NC(C(C)Cc2ccc(Cl)cc2)=O)CCC(F)(F)CC1 c1(C(=O)NC2(CCOC)CCN(C(CCC=CC)=O)C2)cc(C)c(C)c(C)c1 Cc1nn(C)cc1C(C)C(=O)NCC1(O)CCN(C(c2ccc(C(N)=O)o2)=O)C1 c1(CCC(=O)NCCN(C(C2CCN(S(C)(=O)=O)C2)=O)CC)cc(C)cc(C)c1 Cc1ccc2oc(C(N3CC4(CCCCN4C(=O)C4=NNC(=O)C4)C3)=O)cc2c1 c1(SCC(=O)NC(C2CCN(C(C3CC34CCC4)=O)C2)C)nnnn1C C1(NC(CC(COC)C)=O)CC2CCC(C1)N2C(c1ccoc1)=O C(CN(C)C)(C(=O)NCCNC(C1CCC1)=O)N(C)C.C12CN(C1)C(=O)CS2 C1(CCC)CN(C(c2cc(C3(C)CC3)on2)=O)CCN1C(c1cnn(CC)c1)=O C=CC(C(=O)NC(c1ccccc1)C(N1CCC(CCCO)C1)=O)OC c1(NC(C2C(NC(CC(CC)C)=O)C2)=O)nc(C)c(Br)c(C)n1 c1(C(N2CCCCC(NC(=O)C=Cc3cnc[nH]3)C2)=O)cc2c(s1)CCOC2 C1(CC2(CS(C)(=O)=O)CCC2)OCCC1(C)C.C1=CC(=O)NCCCOC1(C)C N1(C(c2ccc(CC)s2)C(=O)NCCCSC)CCc2c(ccnc2Cl)C1 C(=O)(C(C)C(C)COC)NC1(NC(C(CC)C)=O)CN(C(CN(C2CC2)CC)=O)C1 C=CC(CCC)CC(=O)N1CCC(C(C)(C)NC(=O)CCCS(N)(=O)=O)CC1 c1(CNC2(CC(=O)NC3CCC(C)C3)CCCC2)noc2ccc(F)cc12 C(CCC(=O)NCc1ccc(C(=O)NC2(C)CC2(C)C)s1)OC(C)(C)C c1(CCC(=O)NCC=CCNC(CC2CCC(C)(C)O2)=O)nnc(S)nc1O N1(CC(=O)OC(C)(C)C)CCCC(C(=O)NC2(CO)CCC2)C1.c1cncc(O)c1 C=CC(C)(CCOC)C(=O)N1CCC1(C)CC(=O)NC(C1(O)CCCCC1)C c1(C(N2CCN(C(C(=C)F)=O)C(C)C2)=O)nccc2nc[nH]c12 C=C(C)CC(C(=O)NCC(C)(C)F)NC(=O)CC1CC(F)(F)C1 CC(C)CCC(O)C(=O)NCC1(C)CC(NC(c2cnc3[nH]cncc2-3)=O)C1 C(=O)(C1=CC(C)(C)C1)N1C(CNC(CCOc2c(C(C)C)cccc2)=O)C=CC1 CCS(=O)(=O)CC(=O)N(CC(C)(C)CNC(=O)CCCN1CCOC1=O)C N1(C(c2ccc(C)c(O)c2)=O)CCC2(C1)CN(C(c1ccc(C(C)F)cc1)=O)C2 c1(C(N2C(CNC(=O)Cn3nnc(=O)[nH]3)CCC2)=O)cnc2c(c1)NCC2 N1(C(CC=CCC)=O)CC(CC(N2CCCC(O)CC2)=O)C2(CC2)C1 c1(CC(=O)NCC(CNC(c2ncoc2SC(C)C)=O)OC)cnc(C)s1 C(N=c1ccn(C(F)F)[nH]1)(c1c(F)cccc1F)c1n(CC=C)nnn1.C(C)C C1(CNC(C2C(CC)C2)=O)C(O)C(O)CN1C(c1cc(=O)c(OC)c[nH]1)=O C1(O)(C(C)NC(=O)C(N)=O)CCN(C(C2(c3ccc(F)cc3)CC2)=O)C1 c1(C(N(CCCNC(=O)CCc2cnn(C)c2)CC)=O)ccc(C(F)(F)F)n1C c1(NCCn2cncn2)ccc(N(C(=O)CC2CCC3CC23)C2CCC2)nc1 c1(OC)noc(C2CC2)c1C(=O)NC(C)C(C)NC(=O)CCc1ccccc1O C(=O)(C1Cc2ccccc21)N1CC2(OCC(NC(C3=NOC(C)C3)=O)C2)C1 N1(C(C2CC(NC(C3(C)CCNC3=O)=O)C2)=O)CC(CO)C2(CCC2)C1 N1(C(CSCCCC)=O)CCN(C(c2cccnc2C)=O)C(C)C1C C1(NC(C23C(C(=O)OC)(CCC2)C3)=O)CN(C(c2cocc2C)=O)C(C)(C)C1 C1(C(N(C)CCOCCO)=O)CN(C(=O)CC2CCCC(=O)N2)CC1F C1(C)(CNC(C=C(CCC)C)=O)CN(C(C2(C3CCC3)CCC2)=O)CCO1 N1(C(CNS(NC)(=O)=O)=O)CC(CNC(=O)CCc2nc[nH]n2)C2(CCC2)C1 C1(NC(CCSC)=O)CN(C(=O)CCCSc2ccccc2)CC1n1ccnn1 C(Cc1ccco1)(C(=O)NCc1cnns1)NC(C(C)c1ccco1)=O c1(-c2cccc(C(=O)NC(CCC)CCO)c2)n[nH]c2c1CCCC2 C1(C(N(CCCNC(c2c(C)csc2)=O)CCO)=O)CCC(=O)N1C(C)=O CCC(CC(=O)N(C)CC1CCCN1C(c1cc(C)c(F)cn1)=O)CC(C)C c1(OC)ccncc1C(N1CCC(C(F)C(=O)NC2CCC=CCC2)C1)=O C1(CNC(C=CC)=O)(CNC(C2(C3CC3)CCC2)=O)CC12CCC2 Cc1sc2ncnc(N(CCO)CCCC(C)C)c2c1C c1(Cn2c(C(c3ccc(CCF)cc3)NCC(C)CO)nnn2)cccc(F)c1 N1(S(c2cc(COC)c(OC)cc2)(=O)=O)CCCc2c(Cl)cccc21 C(=O)(C1CNC(=O)c2ccnn21)N1CCC(CCNC(Cc2c(C)occ2)=O)C1 c1(NC(C(C2(C)CC2)NC(c2cc(C)no2)=O)=O)cc(Cl)ccc1O C1(NC(CC=CCC)=O)CC12CC(NC(C1(c3cc[nH]n3)CC1)=O)C2 c1(-c2c(C3C(CNC45OCC(C(=O)OCC)(C4)C5)C3)occ2)cn(C)c(=O)cn1 N1(C(CCC=CC)=O)CCCC(C(C)NC(C2(n3cc(Br)cn3)CC2)=O)C1 c1(C(N2CC(CNC(C=CCCC)=O)C(O)C2)=O)cccc(Cl)c1F C(N=c1[nH]c2c(c(=NCCOC3CCC3)[nH]1)COCC2)c1cc(C)nc(O)c1 CC1CC(NC(=O)CCCn2cc(Cc3cc(F)cc(F)c3)nn2)CCCC1 CC1=C(C(=O)N(C)CC2C3CN(C(C4CCNC4=O)=O)CC23)CCO1 N1(C(C2CCN(C)C2)=O)CC2CCC2(CNC(c2ccccc2CC#N)=O)C1 C(=O)(C(C)C(C)CCC)NC1(CC=C)CN(C(c2cnn3ccsc23)=O)C1 C1(CC)C(C(=O)NC(CO)CCCO)CCN1C(c1nc(=N)cc[nH]1)=O c1(C(=O)OC)c(C(N2CCC(NC(=O)C(c3ccc(Cl)s3)C)C2C)=O)noc1C C=C(Cl)CC(C(=O)NC(C)C(C)(C)CO)NC(=O)C(C)n1ccnn1 CC1(C)CC(NC(c2sccc2CC#N)=O)CCN(C(=O)COC(F)(F)F)C1 C(=O)(CN=c1[nH]c2ccccc2s1)NCCCN(C(C(C)OCC)=O)C1CC1 c1(C(=O)NC2CN(C(C(C)SCC)=O)C2)cccc(C(C)(C)C)c1 c12ccc(cc1)C(=O)NC1CN(C1)C(=O)C2.C1(COC(C)C)COC(CF)C1 C1(C(CO)NC(C(C)OCC2CC2)=O)CCN(C(=O)CS(C)(=O)=O)CC1 c1(C(=O)NCCOCCNC(CC2ON=C(CC)C2)=O)cc2c(Cl)ccnc2s1 c1(CC(=O)N(C2CN(C(C3CCSC3)=O)C2)C)cc(F)cc(F)c1 c1(OC)nc(C)c(C(=O)NC2CCC(C)(CNC(C3SCCCS3)=O)C2)s1 c1(OC)cc(C)c(C(=O)NC(CNC(=O)CCn2ccnn2)C2CC2)cn1 N1(C(C2CCC(C)O2)=O)CC=C(CNC(c2cnn(C3CC3)c2Cl)=O)CC1 Cc1nnc(O)c(C(=O)NC2CCC(CNC(=O)CCCCO)C2)c1C N1(C(CC(C)n2ccnc2)=O)CCC(NC(c2ncc(Cl)n2C)=O)C(C(N)=O)C1 C#Cc1cnc(NC(CC(=O)NCCCCCCCC)c2ccccc2)c(C)c1 CC1CN(C(=O)Cc2ccon2)CC2(CCN(C(C3(CF)CC3(F)F)=O)CC2)O1 C1(NC(C(CC)n2ccnc2)=O)CN(C(=O)CO)CC12CCOCC2 C1(CNC(C(P(C)(C)=O)O)=O)CN(C(c2ccc(CCF)cc2)=O)CCC1(F)F C(C)(C)(C(=O)N(CCCNC(c1ccco1)=O)C)NC(=O)OC.C1CC1C(F)(F)F N1(C(Cc2cc(C)on2)=O)CCC2(CC1)CC2C(N1CCC2(CCC2)C1)=O N1(C(c2c(CC)c(C(=O)NC(C)=O)c(C)[nH]2)=O)CC(C)C(C(=O)OC)C(C)C1 C1(NC(C(CC#C)O)=O)CCC2(CC1)CN(C(c1cnc(OC)s1)=O)CCO2 C(=O)(C(C#N)C(C)C)NC1CCCC(C(=O)NCc2cc(CC)on2)C1 CCCC(C(=O)N1CC(O)(CNC(=O)C(C)Oc2ccccc2C#N)C1)C(C)C C#CCCCN(C(=O)C(C)=CCNC(=O)C(C)NC(C)(C)CC)CCOC C(=O)(CCCCCCC(OC)OC)NCC(CC(C)C)NC(C(F)=CC)=O c1(CC2C3CN(C(c4ccc(F)c(CO)c4)=O)C(C3)C2)cc2ccccc2o1 n1(CC)nnc(C)c1CNCC12CCC(NC(=O)OC(C)(C)C)C1C2 C1(NC(c2c[nH]nc2F)=O)CN(C(=O)C=C2CCC2)CC12CC2 c1(N2CCC(C)(NC(C(C)Cn3ccnc3)=O)C2)nccn2nnnc12 CC1CC(C(=O)N(C2CC(C(=O)NC3CN(C(N)=O)C3)C2)C)CO1 c1(OC)ccncc1C(=O)NC1CCCC1CNC(C1CC(n2cnnc2)C1)=O C12(C(N3CCC(CN(C(=O)COC4CC4)C)C3)=O)COCC1C2(F)F C1(CC)C(NC(C2(CC(F)F)CCC2)=O)CCN1C(C1CC(O)CN1C(C)=O)=O N1(C(C(C)SC2CC2)=O)CCCCCC1c1cn(CC2CCC3(CC3)CO2)nn1 C1(CNC(C(C2CCC2)OCC)=O)CC2(CCN(C(C3(C)CSC3)=O)CC2)CO1 CCC(C)(C)C(O)C(=O)NC(C(=O)NC1CNC(=O)C12CC2)C(C)OC C1(CN(C(c2ccc(CC)[nH]2)=O)C)CCN(C(=O)C(F)CC2CC2)CC1 C1(NC(c2cccc(C)c2C)=O)CCC2CN(Cc3nc(=O)n(C)[nH]3)CC2C1 C1(CNC(c2noc3cc(F)ccc23)=O)CC2(CCN(C(=O)CCF)CC2)CO1 c1(C(=O)NC2(C)CN(C(CC(C)c3ccccc3)=O)C2)cc(N(C)C)ccn1 C#Cc1cncc(C(N2CCC(N(C(=O)C(C(C)C)NC(=O)OCC)C)C2)=O)c1 n1(CC(=O)NC2CCC(C)N(C(c3nc(Cl)cs3)=O)C2)c(O)nc2ccccc12 C1(CC#C)(C(=O)N(CCC(C)NC(c2cncn2C(F)(F)F)=O)C)CC=CCC1 C=CC1CCN(C(C(=O)Nc2ccc(OC)cc2)C2(CC(=O)OC)CC2)CC1 N1(C(CCN(CC)CC)=O)CC(NC(=O)C(F)C(C)C)CC1CO Cc1cnc(N2CCC2(C)C(N2CCCC2C(N)=O)=O)nc1C CC1CC(C(N2CCOC(CNC(c3ccncc3)=O)C2)=O)CN1C c1(C(N2CCCC(CCNC(C3(C)CCOC3)=O)C2)=O)c(Cl)ccc2c1OCO2 N1(C(CNS(N)(=O)=O)=O)CC2CCC1C(CNC(c1ccc(Cl)c(Cl)c1O)=O)C2 c1(N2CCCC(NC(c3cc(C)oc3C)=O)(CO)C2)nc(C)nc2scc(C)c12 C1(CCO)(NC2(c3n(CC)nnn3)CC(CC#N)C2)CCSCC1 N1(C(c2cc(OCC)n[nH]2)=O)CCC(C(=O)NCCC2CCCO2)CC1C C(=O)(CCC(C(C)C)NC(C1CSCC(=O)N1)=O)NCCC(C=C)C c1(C(=O)NC2(CC=C)CN(C(=O)Cc3ccsn3)C2)nn(C)nc1C N1(C(c2ccc(SC)s2)=O)C2CCC1CC(C(=O)NC(C)Cc1cnccn1)C2 C1(C(N(CCCn2cc(-c3cccc(CN)c3)nn2)C2CC2)=O)CCCNC1=O C1(C(=O)NCCN(C(=O)CC2CC(O)C23CCC3)CC)C2CC3CC(C2)CC1C3 N1(C(C(C)C)=O)CCOCCC1C(=O)NC(c1ccns1)C CCCC(C(=O)N1CCN(C(C2CCC(=O)N(CC)C2)=O)CC1C)C(C)C c1(C(=O)NC2CC(CNC(C3CC3(F)F)=O)C(O)C2)cc(F)ccc1Cl Cc1cc(C(=O)N(C)CCC2CCCCN2C(=O)C(C)C(F)F)c(N)c(F)c1 CC(C(=O)NC1CN(C(c2csc(-c3ncc[nH]3)n2)=O)CCC1F)C(C)(C)C C(CC(C)C(=O)NC1C2CC1N(C(c1cccc(C3CC3)c1)=O)C2)=CCC NS(=O)(=O)N1CCCCC1C(N1CCCC(NC(c2cnco2)=O)C1)=O Cn1nncc1CCNC(=O)C(C1CCN(C(=O)CC2CC(N(C)C)C2)C1)F c1(SC)cc(CNC(=O)NC2CCC(C)C2)n(C)n1 C1(CC(=O)NCC(CCNC(=O)CC2(OC(C)=O)CC2)OC)CCCCN1C C1(C(=O)O)(C(F)F)CCCN(C(=O)C(C(=O)NC(C(C)C)C)c2ccccc2)C1 C(=O)(C(CCN(C)C)NC(=O)CCc1nccs1)NCCCC1CC(C)C1 CCC(F)(F)C(=O)NCCC1CCCN(c2cc(-c3ccc(F)cc3)ncn2)C1 c1(C(N2CCC(CNC(=O)CCCC(F)F)C2)=O)coc2c(Cl)cccc12 c1(C(N(CCCCC(=O)N(c2cn(CC)nc2)C)C)=O)cc(C#N)oc1C N1(C(c2c(CC)cccn2)=O)CCC(C)C(CNC(=O)C2=C(Cl)CC2)C1 CCC(CC(=O)N(C1CCCCN(C(=O)CS(N)(=O)=O)C1)c1nc(=N)[nH][nH]1)C(F)F CC1=C(C(=O)NC2CN(C(c3oc(C)nc3C)=O)CC2C)CCCO1 C1(C(=O)NC(CNC(CCN2C(C)CCCC2)=O)CO)CC(F)(F)CCC1(C)C N1(C(C2C(C=C)OCC2)=O)CCCCCC1CNC(c1cncc(CC)c1)=O C1(C(N(C)CC2(CNC(Cc3cc(CC)nn3C)=O)CC2)=O)CC2CCC1OC2 C1(NC(c2nc(CCC)oc2)=O)CC2CC(C1)N(C(=O)Cc1c[nH]ccc1=O)C2 c1(OCC)ccccc1C(C)NC(=O)NCCCCc1[nH]c(C)nc1C N1(C(C=CCC)=O)CCOC2(CCCN(C(c3nc(C)oc3OCC)=O)C2)C1 c1(CN(C(=O)C(F)C2CCC2)CCNC(C2(C(C)(F)F)CCC2)=O)ccc(Cl)nc1 N1(C(C(C)(C2CC2)OC)=O)CC(C(=O)NCCN2CCC(C)C2)C(C)(C)C1 C(=O)(C(CO)C(C)(C)C)N(C1CCCN(C(c2cscc2Cl)=O)C1)CC C12(CNC(C#CC(C)C)=O)COCCN1CCN(C(c1nncs1)=O)C2 N1(C(C2CC(CC)N(C(=O)CCC(C)(F)F)CC2)=O)CCOC2CCCC12 CCCCC(C(=O)NC1CCC(N(C)C)C1)NC(=O)Cn1ncn(C)c1=O C1(NC(COCCCCC)=O)CCOCC1C(=O)NC1(C)CC(N(C)C)C1 c1(NC(C2(Cc3ccccc3)CN(Cc3c(C)scn3)C2)=O)ccc(O)c(Cl)c1 CC(CCC(F)(F)F)NC(=NCC1CCCO1)NCC12CCC(CC1)O2 C1(NC(C(Cn2ccc(C)n2)C)=O)CN(C(c2ncsc2C)=O)CC1(C)C c1(CNC(C(C)N2CCC2NC(=O)CN2CCC2)=O)ncnc2[nH]cnc12 C1(C(=O)NC2CCC(NC(C3CN(C(N)=O)C3)=O)C2)CC(=O)NC(=O)N1 N1(C(C(=O)NCCCSC)CC2CCCC2)CCOC2(CCCC2)C1 C1(OC)(CNC(=O)C(C)N2CCC2)CN(C(c2cc(CCCO)on2)=O)C1 C1(NC(c2ccn(CC)c(=O)c2)=O)CN(C(=O)CC2CCCCO2)CC2(CC2)C1 c1(NC(CCNC(CC)CSC)C)cccc(C(=O)NCC)c1 C1(CC=C)(NC(C2(O)CC2(C)C)=O)CCN(C(=O)CC2(C)CCOC2)CC1 N1(C(C(P(C)(C)=O)O)=O)CCCC2(C1)CN(C(=O)CCNC(c1ccsc1)=O)C2 N1(C(c2c(C)ccs2)=O)CCN(C(C2CCCC2C)=O)C2CCCC12 c1(OC)cccc(NCCC(=O)NC(C)C(C)(C)NC(C2CCC(=O)N2)=O)c1 C1(NC(c2ccccn2)=O)CCCC1CNC(C1(O)CCCC1)=O C1(NC(C(CC)N(C)C)=O)CCN(C(c2cc(Cl)c(Cl)s2)=O)CC1F c1(C(=O)NCC2CN(C(C3C(CCOC)C3)=O)C2)cc(S(C)(=O)=O)oc1C C1(NC(=O)NCCSCc2cc(C3CC3)on2)CCCN(C2CCC2)C1 Cc1cc(C(=O)NCC(C)(C(C)C)NC(=O)CSCc2csc(C)n2)cnn1 C12(NC(C(C)C3CC3)=O)CCC1CN(C(c1cc(N(C)C)cc(Br)c1)=O)C2 N1(C(CCC(C)NC(=O)C=C2CCOCC2)=O)CC2NC(=O)OC2C1 C1(CC(=O)NCC2(CNC(c3c(C)n(C)cn3)=O)CCC2)COCC(C)(C)O1 N1(C(=O)Cn2nccn2)CCC(O)(C2CCN(C(c3cccnc3)=O)CC2)C1 N1(C(=O)C(=CC2CCCCC2)F)CCC2(CCN(C(=O)CO)C2)C1 c1(C(N2CCN(C(C3(F)CC=CCC3)=O)CC2)=O)nc2ccccc2s1 C1(C(N2CCN(C(C3=NOC(C)C3)=O)CC2)=O)CN2CCC1(C)CC2 C12(CNC(CC3N(CC)CCOC3)=O)CCCC(CN1C(=O)C1=CCOCC1)C2 c1(OC)cccc2[nH]c(C(N3CCCC3(C)C(N3C4CCC3CC4)=O)=O)cc12 N1(C(CCC(C)=O)=O)CCC2(C1)c1ncn(C)c1CCN2C(=O)CC1=CCCC1 N1(C(Cc2nc(C)[nH]n2)=O)CC(C(=O)NCCCOC(=O)N(C)C)OC(C)C1 C(=O)(C(O)CC(F)(F)F)NC1CCC(NC(c2nc(CC)oc2)=O)C1 N1(C(CC(C(C)C)c2ccon2)=O)CCC2(CC1)CC(C(F)C(=O)O)C2.CCC#N C1(CN(C(C)C)C(C)C)CN(c2cccc(Br)c2)C(=O)O1 c1(C(N(CC)CC2CCCN2C(C2CCC(=O)N2)=O)=O)cccc2sncc12 C(C(C)(F)CNC(c1ccccc1)=O)NC(COC(C)C)=O C(=O)(C(C)C(C)S(C)(=O)=O)NCC1(CNC(C(=Cc2ccc(F)c(F)c2)C)=O)CC1 c1(C(=O)NCC2(OC)CC(F)(F)C2)cc(C(C)C)ccc1OC c1(SCCC)ncccc1CNCC1CC(NCC2CCCC2)CC1O CC1C(C(=O)Nc2ccccc2)CCCN1C(=O)CSCC(c1ccoc1)=O N1(C(C(C)NC(C)(C)C)=O)CC(F)(F)CC1(C)CNC(=O)C(C)n1ccnn1 C1(CNC(=O)OCCCCC)CCCC2(CCC2)O1 CC(CNC(c1cncc(O)c1)=O)CC(=O)NC(C)C(F)(F)F c1(C(=O)NC(C(C)NC(CN(CCCCCC)C)=O)C)ccnc(C(=O)OC)c1 Cc1ccc(F)c(CN2CCN(C(C3CC4(CCC4)C3)=O)C3CC23)c1 Cc1c(Br)sc(C(N2CC(Cn3cc(-c4c[nH]c(C(F)(F)F)c4)nn3)C2)=O)c1C C1(CNC(c2c(C)cc[nH]2)=O)CCCN(C(c2ccc(C3CC3(F)F)cc2)=O)C1 N1(Cc2cccc(CO)n2)CCC(F)CC1.C123CC(C1)(C2)CNC3=O C1(C)(CNC(c2c(SC)cccn2)=O)CCCN(C(c2ccc[n+]([O-])c2)=O)C1 c1(C(=O)NCC(N(C(=O)CC2CC=CC2)C)C2CC2)ccc(C(C)(C)C)cn1 Cc1nc(C)c(CC(=O)NCC2C(C)CCCN2C(c2cnco2)=O)c(O)n1 C1(NC(c2cccnc2O)=O)CCC(C(=O)NCCSc2ccccc2Cl)CC1 C1(C(=O)O)(C(=O)NCC(C2CC=CCC2)N2CCCC2)CCNCC1 c1(C(=O)NCC(C(C)(C)C)NC(CC(C)F)=O)ccc(Br)c(Cl)c1 Cc1ccc(Cl)c(N)c1C(=O)NC(CNC(C1CC1(C)C)=O)C1CC1 C1(NC(C2(CC)N(C(c3cnc(CC)o3)=O)CCC2)=O)CCCCC1(C)C C(=O)(C(C(C)OC)NC(c1ccc(C#N)[nH]1)=O)NCC(COCC)O c1(NC(C2CCCN(c3ncc4[nH]ncc4n3)CC2)=O)cc(Br)cc([N+](=O)[O-])c1 Cc1oc(Cl)nc1C(=O)NCC1(O)CN(C(c2csc(Cc3ccccc3)n2)=O)C1 CC1CN(S(=O)(=O)N2CCN(C(c3ccccc3)=O)CC2)CC(C)N1CC#N c1(-c2cc(C(C)NC(=O)NC3C(COC)CC3)[nH]n2)ccc(F)cc1 c1(C(N2CCC(N(C(=O)C=Cc3cn(C)cn3)C)C2)=O)ccc(N)cc1F C1(C(C)NC(c2ncccc2O)=O)CCN(C(=O)COCC(F)(F)F)CC1 Cc1ccnc(C(=O)NC2CC(CNC(c3ccc(F)s3)=O)C2(C)C)c1N C12(C(=O)NCC3CC(OC)C3(C)C)CCC(NC(=O)CCSC)(CC1)C2 C=Cc1cc(C(=O)NC(C2CN(C(C3C4(CC4)C34CC4)=O)CCO2)C)cc(F)c1 CCC(CC(=O)N1CCOC(CCCNC(c2cccn2C)=O)C1)C(F)F C(=O)(C1=CC2(CCOCC2)C1)N(C)CC1N(C(c2[nH]cc(CC)c2)=O)CCOC1 c1(C(=O)NC(Cn2cccn2)C(=O)NCCc2cscn2)ccnnc1O C1(c2nnnn2C)(NCc2c(C)n[nH]c2C)CCCC(C#N)C1 S(=O)(=O)(c1cccnc1Cl)N1CC2(CCN(C(=O)CC3CCC(F)(F)CC3)C2)C1 C(N=C(NCc1cc(C)on1)N1CCC(O)C(C)C1)c1c(C)n[nH]c1C C(=O)(CCC(C)(F)F)NCC(CCOC)NC(C1CCCCN1C)=O C1(NC(C(C)(C)OC(C)C)=O)CCCN(C(C2(C#N)CC2)=O)CCC1 N1(C(c2nc(C(=O)OC)oc2)=O)CC(NC(=O)C#CC2(C)CC2)CC12CCC2 c1(C(=O)NCC(C)NC(c2nccc(CC)c2)=O)cccc2c1CNC2=O c1(CCC)cc(C(=O)N(CC(O)CNC(c2c(C)n[nH]c2C)=O)C)sc1C c1(CCC(c2n(C(C)C)nnn2)NCC(C)Cn2ccnc2)ccccc1F c1(CC(Cn2c(OC)ccn2)=O)cccc(O)c1 C1(C(N2C(CNC(=O)Cn3ccnn3)CC(F)C2)=O)CC12CCOCC2 c1(CN(C(CC)C(=O)OC)C)c(F)ccc2occc12 CCC(C#N)C(=O)NCC1(F)CC(NC(c2ccc(O)nc2)=O)C1 C12(C(=O)NC3CN(C(C(c4cn(C)nc4)O)=O)CC3F)CCCN(CC1)C2 c1(C(=O)NC2CC(CNC(C3(CC)COC3)=O)C2)cnn2ccc(Br)cc12 N1(C(COC(C)=O)=O)CC(CNC(c2ccnn2C)=O)CC1C.c12cc([nH]n1)C2 N1(C2CC2CC(=O)OCC)CC(CNC(=O)CNC)C1.C(=O)(CNC(C)=O)C(=O)OC C1(C(=O)NCc2cc(C3CC3)n[nH]2)(COC)CN(C(=O)CC(C)c2ccco2)C1 c1(NC(c2n(CC=C)nnn2)CC2CCOCC2)ccc(C2CC2)c(Cl)c1 c1(C(=O)NC2(CNC(C=CC)=O)CCOCC2)cc2ccc(F)cc2o1 N1(C(C(CC=CCC)C)=O)Cc2[nH]nc(C(N3CCC(C)(C4CC4)C3)=O)c2C1 C1(C(=O)NCCCC2(NC(C3CC(OC)C(OC)C3)=O)CC2)CCCCC12CC2 c1(C(N2CCCC(C)(NC(C(CC=C)C)=O)C2)=O)nc2sc(C)cn2c1C CCCCC(CC)C(=O)N1CCC(C2(NC(=O)Cc3sc(O)nc3O)CC2)C1 N1(C(c2c(C)oc(C)c2C)=O)CCC2(CC1)COC(CNC(C1(O)COC1)=O)C2 c1(C(=O)NCC(C2CCCC2)NC(C(C)NC(C)=O)=O)cnc2ccccc2c1 C(CCNC(C1(C)CCCC1)=O)(C(C)C)CNC(C(=O)NCCNC(C)=O)=O C1(CC)CN(C(=O)CCCCCNC(=O)CCc2nccn2C)CC(C)O1 C(N=C(NC1CC1)N1CCCC(C2(C)OCCO2)C1)c1cc(CC)c(O)cc1 N1(C(Cn2ncc(C(=O)OC)c2)=O)CC2CC2(CNC(c2ccc(SC)s2)=O)C1 N1(C(C(C)N(C(C(CSC)C)=O)CCC)=O)CCC(C)(C(=O)OC)CC1 N1(C(c2cc(C(=O)OC)c(CC)o2)C(=O)NCC)CCC(C2(O)CCC2)CC1 C1(C(C)C)CN(C(C2(C)CC2)=O)CCN1C(C1CCC(F)(F)CO1)=O N1(C(c2cc(CNC(CCC(C)(C)C)=O)[nH]n2)=O)CC2CCC(C1)C2C#N C1(C(=O)NCC(C)N(C(c2nnn(CC)c2C)=O)C)CCc2nnc(O)cc2C1 c1(-c2n(-c3cccc(C)c3)nc(CO)n2)cc2c(F)cc(F)c(F)c2[nH]1 N1(C(C=CCN(C)C)=O)CCCC2(C1)CN(C(C1OCC1(C)C)=O)CCO2 c1(OC)ccc(F)c(C(=O)NCC2C=CCN2C(C2CCCS2)=O)c1Cl N1(C(C2(SC)CC2)=O)CC(CNC(=O)CC2CCCC(C)(C)C2)C2(CCC2)C1 O=C(NNc1ccc(Br)c(F)n1)NC1CC(O)C12CCC2 Cc1nc(C)c(C(N2CCC2C(=O)NC(c2ccc(Cl)cc2)C2CC2)=O)s1 c1(N2CCCCC(C)C2)nc(N2CCC(OCCO)C2)nc2ncn(C)c12 C(=O)(CCCCCNC(N)=O)NC(CCCCNC(c1cccc(OC)c1)=O)C C1(CNC(CCSC)=O)CN(C(c2ccc(C3CCC3)nc2)=O)CC(C)(C)O1 C#Cc1cccc(C(N2CC3CC2C3NC(=O)CC(C)C=C)=O)c1Cl Cc1cncc(C(=O)N(CCNC(c2coc(Cl)n2)=O)CC2CC2)n1 c1(C(=O)OC)ccc2occ(CCC(=O)NC(COc3nccs3)CO)c2c1 N1(CCCCOC)CCC(CNC(c2ccn(C(C)C)n2)=O)C1 c1(C(=O)NCCC(C)N(C)C(C2CCCCS2)=O)cncc(Br)c1 C1(CNC(c2c(C)cccc2)=O)CC2(CC(NC(c3cccc(O)n3)=O)C2)C1 N1(C(c2cccc(CNC(C3CCO3)=O)n2)=O)CC(CO)CC12CCC2 c1(CC(=O)NCCCNC(C=C(C)C)=O)csc(-c2cnccn2)n1 c1(OC)cc(OC)c(C(=O)NC2CCC(NC(c3cccnn3)=O)CC2)cc1Br c1(C(N2C(CNC(COC)=O)CC(F)C2)=O)ccc(OC)c(F)c1 Nc1nc(Cl)ccc1C(=O)NCCC(O)CNC(=O)C(F)C(F)(F)F C#Cc1ccccc1CC(=O)NCC(CCOC)NC(=O)CC1(O)CCCC1 C1(CC(=O)NCCCCN(C(C(C)c2ccco2)=O)C)CC(F)(F)C1 C1(NC(c2c(SCC)ccc(Cl)c2)=O)CN(C(=O)CNC(C)=O)CC2CCCC12 c1(C(C)N(C(C)CC(O)C2CC2)C)cccc(Cl)c1 C1(NC(CN(CC)CC)=O)C=CCN(C(=O)CC2(CC)CCC2)C1 N1(S(C)(=O)=O)CCC(CCNC(c2nccc(Oc3ccccc3)n2)=O)CC1 C(CCCCC(=O)NCC1NC(=O)NC1=O)N(C(c1cc(COC)nn1C)=O)C c1(CC(C)C(=O)NC2CC2C(N2CCC(O)C(C)C2)=O)ccc(C#N)cc1 CN=c1[nH]c(C(=O)NCCSCC2CN(c3nnc(O)s3)C2)cs1 C1(C)(CC)CC(NC(=O)Cc2ccccc2)CN1Cc1ccccc1 N1(C(C2CC(OC)C2)=O)CCN(C(c2oc(SC)cc2C)=O)C2CCC12 C1(CN(C)C)COCCN1C(=O)C(c1cccnc1)NC(=O)CCc1cnoc1 c1(CN2C3CC(NC(=O)Cc4ccncc4)CC2CC3)cc2ccncc2[nH]1 CCS(=O)(=O)CC(=O)N(C)CCOCCCN(C(=O)CCc1cnccn1)C C1(C(=O)NCC2CC(NC(C34CC(C#N)(C3)C4)=O)C2)OC2CCC1CC2 C(=O)(CC(F)(F)CS(C)(=O)=O)NCC1(C)CCN(C(C2CCCCC2O)=O)CC1 C12(NC(c3c(C)cccn3)=O)CCCC1N(C(=O)C=Cc1ccc(Cl)nc1)CC2 C(=O)(C1CNC(=O)c2ccnn21)NCC(CCC)NC(c1sccc1OC)=O Cc1cc(S(=O)(=O)N2CCCC(n3cc(CO)nn3)C2)c(C)s1 C1(NC(CCOCCOC)=O)CCC(CNC(=O)CC2(C)CCCC2)CC1 C1(NC(CCCc2onc(CCC)n2)=O)CN(C(=O)COCCCOC)CC1F c1(C(N2CC(O)(CCNC(c3cc(C(CC)C)no3)=O)C2)=O)ccc(Cl)cc1F N1(C(C(CNC(CCOC(C)C)=O)C)=O)CCc2n[nH]cc2C1 c1(C(=O)NC(C2CC(NC(C34CC5CC3C4C5)=O)C2)C)cc(O)n(C)n1 C#CCCN=C(NCc1cccnn1)NCC1CCC12CCCO2 CC1(CNC(=O)CNC(c2ccccc2)=O)CCN(C(=O)Cc2sccc2Cl)C1 C1(C(=O)NC2(C)CSC2)(CC)CCCN1C(=O)CC1CCCNC1=O c1(N(C)Cc2cccnc2)ccc(-c2ccc(CNC(C3(O)CC3)=O)cn2)nc1 N1(C(C(COC)OC)=O)CCCC2CN(C(c3cc(C)c(Br)s3)=O)CC12 CC(CNC(=O)CNC(c1cccnc1)=O)(CO)NC(C1CCCS1)=O C1(C(=O)NC2CC(C(C)C)OC2)(NC(c2cncn2C)=O)CCN(C)C1 C(C(=O)NC1(C)CC(CN2CCCCCC2)C1)(C(C)C)n1ccc(C)c1 c1(C(=O)NCCC2CN(C(=O)CC3CC(F)C3)C2)ccc(F)c(C2CC2)c1 N1(C(c2cc(C)oc2)=O)CC2CCCC(N(C(C3CC3c3cnc[nH]3)=O)CC)C2C1 CCC(C)C(C(=O)N1CCC(C(=O)OC)C1)NC(c1ccc(C)nn1)=O N1(C(CC=C)=O)CCC(N2CCCC(C(=O)NCc3ncnn3CC)C2)CC1 C(=O)(CC(C)CC(=O)NC1CCCC1NC(c1cc2ccncc2[nH]1)=O)OC C1(C(=O)NCC2(O)CN(C(CCN(C)CC)=O)C2)CCOC(=O)N1 N1(C(c2c(OC)cc(Br)cc2)=O)CCC(C)N(C(=O)CC2(C#N)CC2)CC1 N1(C(c2cn(C)nc2Br)=O)CCC2(CC1)CC2(C#N)CO c1(NC(C(C)S(N)(=O)=O)=O)cccc2c1CN(C(=O)OCS(C)(=O)=O)C2 c1(C(N2CC(CC(C(=O)NCc3ocnc3CO)F)C2)=O)ccc(O)cc1O N1(C(c2c(OC)csc2)=O)CCCC(O)(CNC(=O)CNC(C2CCC2)=O)C1 N1(C(CC=CCC)=O)CCC2CCN(C(=O)CCn3cc(Cl)cn3)CC12 c1(C(N2CCCC3(CNC(c4ccnnc4)=O)C2C3)=O)cc(F)c(F)cc1F N1(C(C2(SC)CC2)=O)C(C)CN(C(=O)C(C)(C)C(F)(F)F)CC1C CN1CC(NC(C2C3CN(C(=O)OC(C)(C)C)CC23)=O)Cc2ccccc21 C1(NC(Cc2cc(C)no2)=O)CS(=O)(=O)CC1NC(C1CCC(O)CC1)=O C1(C(=O)NC(CC=C)C(=O)NCCC2CCCN(C)C2)CC(C)CC(C)C1 c1(C2N(C(C34CNC(C(=O)O)(C3)C4)=O)CC2)ccc(F)cc1F CCC(C)C(CC(=O)N(C)CC1(C#N)CC1)NC(=O)C(C(C)C)C(C)C N1(C(COCC(=O)OC)=O)CCN(C(c2cc(C)c[nH]2)=O)C(C)C1 Cc1nnccc1C(=O)NC1(CNC(c2ncc(F)cn2)=O)CCOC1 C(=O)(C(F)C(F)(F)F)NCCC1(CNC(=O)CCC(=O)c2cccs2)CC1 Cc1cc(C(=O)OCC(=O)Nc2nc(-c3cnco3)cs2)n2nccc2n1 c1(C(N(CC(=O)Oc2ccccc2Cl)C)=O)cccc(F)c1 N1(C(CC(CC)O)=O)CCCC(CO)(NC(=O)CCCCN(C)C)C1 c1(NCC(c2ccccc2)CNC=O)ccc(-c2ccccc2)cn1 C1(C(N(C)CC2CCN(C(c3cc(C4CC4)[nH]n3)=O)C2)=O)CCC(F)(F)C1 C1(CNC(c2oc(CC)c(C)c2)=O)CCC2CN(C(C3(C)CCNC3=O)=O)CC12 N1(Cc2cccc(C)c2)CCC(NC(=O)CCCc2nc(C3CC3)no2)CC1C C12(CNC(C3CC(OC)C3)=O)CCC1CN(C(c1cc(C3CC3)n(C)c1C)=O)C2 C1(CC)CC(C)CN(C(=O)CC2(NC(=O)CC(C)NC(N)=O)CCCCC2)C1 CC(CCN=c1[nH]c2ccc(N)cc2s1)NC(=O)CC1CC(C)(C)CO1 C1(C)(CNC(C2(OC)CCCCC2)=O)CN(C(=O)C(O)CCC(C)C)C(C)(C)C1 CC(C)CC(C(=O)N1CC2CCC(C(=O)Nc3cncc(CO)c3)(C2)C1)C(N)=O Cn1ccc(-c2cc(C(=O)NC(C)(C)CNC(C3CC3(C)C(F)F)=O)no2)n1 Cc1ccnn1CC(N1CC(C)(C(=O)Nc2cnn(C(C)(C)C#N)c2)C1)=O c1(C(=O)NCc2cccc(C(C)C)c2)ccc(Br)nc1F.N12CC(C1)CC2=O C12(CCNC(c3nc(C)sc3C)=O)CCC(C1)N(C(C1CC(=C3CC3)C1)=O)C2 C1(N(C(Cc2c(C(C)C)con2)=O)C)CN(C(C2(C)CCCCC2)=O)CC1F Cc1cc(C(=O)N(c2ncc(Br)cn2)C2CCNCC2)nn1-c1ccccc1 C(=O)(C(C)CCCCCC)N(CCC(=O)NCC(=O)NCCC)C N1(C(=O)C=Cc2ccsc2)CCC2C(CCCN2C(=O)CN2CC3C=CC2C3)C1 C=CCC(CC(=O)NCC(C)C(=O)OCC)NC(C1CCCC(=O)C1)=O C=CCC(C(=O)NC1CC(NC(c2ccc(OC(F)F)c(Cl)c2)=O)C1)C(C)(C)C CCC1=C(C(=O)N2CCC2(C)CC(=O)NC2COCCC2(F)F)CCCO1 CCC(CC(=O)NC(C)(C)CCCF)NC(=O)Cc1coc(C)n1 C(=O)(CC(C)C(F)(F)C(F)(F)F)N(C)CC1OCCN(C(c2c(C)[nH]cc2)=O)C1 C=CCCC(CO)NC(c1cnn(CCNC(=O)C(C(C)C)NC(N)=O)c1)=O C12(C(=O)NC3CCN(C(CC4C(OC)CC4)=O)CC3O)CC3CC(C(=O)N1)C2C3 C1(C(N2CC(CNC(c3cnc[nH]3)=O)OCC2)=O)COCCC1(F)F N1(C(c2ccc(C)s2)=O)CCN(C(=O)CCCCC#N)C(C2CCCC2)C1 C=C1CC2(C1)CN(C(C1CC(F)CN1C(C1CC3C=CC1CC3)=O)=O)C2 O=C(O)C(C(O)c1ccc(F)cc1)NCc1ccnc(O)c1 N1(C(C2NC(=O)CC(C)C2)=O)CC2CCN(C(=O)CCP(C)(C)=O)C2C1 C(C(C(=O)NCC(C)(C)CCOC)C(C)C)NC(CC(C=C)CC)=O CCC(COC)C(=O)NCc1ccc(CN(C(=O)CC2CCSC2)C)cc1 Cc1nnccc1C(=O)NC1CCCCC1C(=O)N(C1(CO)CC1)C C(=O)(C1=CS(=O)(=O)CCC1)N1CC(CNC(C(C)(C)Cc2ccc(O)cc2)=O)C1 C(CCc1ccccc1)(C(C)O)NCc1nc(OC(c2scc(C(C)=O)c2)=O)no1 c1(CN(C(c2coc(Cl)c2)=O)CC)cn(CC2(CC(=O)OC)CC2)nn1 C1(CC)CC(O)CN1C(=O)CC(C)(C)N(C)C(C1OCCC1C)=O c1(NC(CC2N(C(CCOCC#C)=O)CCC2)=O)cncc(C)c1 C1(C2CCC2)(C(=O)NCC#CCNC(=O)CCCc2ccsc2)CC1 Cc1cccc(F)c1CC(N1C2CCC1C(NC(=O)Cc1ccno1)C2)=O C1(C(=O)NC(C)CNC(=O)CN2CCN(C)C(=O)C2)CCC2CCCCN12 c1(CC)ncncc1C(N1CC(OC)CC1C(=O)NC(C)CN1CCCCC1)=O CC(C)C(CCC(=O)NC(CC1CCCC1)CO)NC(C1CC2(CC2)C1)=O C1(CNC(Cc2c(C)noc2Cl)=O)COc2ccc(Cl)cc2C1.C12CCN1C2=O C12(NC(c3ccc4cc[nH]c4n3)=O)COCCC1CN(C(=O)C1=CCOC1)C2 CCC1=C(C(=O)NC2CC(F)CN(C(=O)C=C(C)C3CC3)C2)SCCO1 CC#CCC(C(=O)N1CCOC(C)(C2CC2)C1)NC(c1csc(Cl)c1)=O CCC(C)C(O)C(=O)NCC1CCCCN1C(c1cn(CC)nc1C)=O C1(CNC(C2(CC#C)CCCCC2)=O)CC(F)(F)CN1C(=O)C(C)OCC=C c1(C(=O)NC2(CCNC(c3c(SCC)cccn3)=O)CC2)cccn2nnnc12 Cc1cccc2oc(=NCC(O)CNC(C3Cc4cc(F)ccc4O3)=O)[nH]c12 C1(NC(=O)Cc2csc(C3CC3)n2)CC(NC(c2cc(Cl)sc2Cl)=O)C(O)C1 c1(C(C)C)[nH]nc(C(=O)NC(CO)C(C)NC(=O)C2=NOC(C)(C)C2)c1[N+](=O)[O-] c1(C(=O)NC2CCCN(C(c3cccc(OC)c3)=O)C2)cc(C)c(O)c(C)c1 C(=O)(C1=Cc2cccc(Br)c2OC1)NCCC(C)NC(C(CCCC)CC)=O c1(NC2(CC)CCOC2)ccc(S(=O)(=O)NN(C2CCCCCC2)C2CC2)c(Cl)c1 C(N=c1cc(NCC2CC(O)CN2C)nc(C(F)(F)F)[nH]1)C1OCC(C)(C)C1 C12(C(=O)NCCCCN(C(=O)Cc3ccc(Cl)cc3F)C)CC1CCC2(F)F N1(C(C=C(CNC(CNC(=O)OCC=C)=O)C)=O)CCC2(CC1)CC2C#N C1(N2C(=O)C2)CCN(C(c2scc(C)c2Cl)=O)CC1.C(C)(C)(C)SC C1(C(=O)NCCCC(C)(C)NC(C2COC(=O)N2)=O)CC2C=CC1C21CC1 C1(c2n(C)cnc2)NC(=O)CCC1NC(=O)C(F)C(F)(F)F c1(C(=O)NCCC2CCN(C(C3(NC)CC3(F)F)=O)C2)cnc(Cl)cc1Cl N(C1CCCn2nc(C(C)(C)C)cc21)C(COc1n(C)nc(C(F)(F)F)n1)=O c1(C(=O)NCC2C(NC(c3ccc(NC)cc3C)=O)C2)cc2c(nc1O)CCC2 CCCC(C)C(=O)NC(C)(C)CCNC(c1scc(C)c1Cl)=O C#CC1CCN(C(C2(NC(=O)CCc3cncn3C)CCCC2C)=O)CC1 N=c1cc(C(N2CC3C(NC(=O)CC4CCCOC4)C3C2)=O)nc(Cl)[nH]1 c1(C(=O)NCC2N(C(CNC(c3cn(C)nc3)=O)=O)CC2)cc(Cl)cc(Cl)c1 C(=O)(CC(COc1cn(-c2nccc(Cl)c2F)nn1)C(=O)OC)OCC CC1=C(C(=O)NC(C)C(C)C(=O)N(C23CCC(CC2)CC3)C)SCCO1 c12ccnc(c1)NC2=O.C(=O)(CCOCC)N(CCCC)C(C)CC C1(C(N2CC(O)(C(C(=O)NC3(C(F)(F)F)CC3)F)C2)=O)CC2(CC2)CO1 Cc1nc(COc2ccccc2)ncc1C(=O)NCC1CCN1C(=O)C(C)O C1(CC(=O)NC(CC)Cn2cncn2)CN(C)CCN1C(=O)Cc1ccc(C)s1 C(=O)(C(F)CCC(C)(C)C)N1CC(C(C)NC(C2C=CCN2C2CC2)=O)C1 C1(C(=O)NC(CC(=O)OC)(C)c2ccc(Br)cc2)CC12CC(C)(C)C2 CCC(CCc1ccccc1)C(=O)N1CC(NC(C2CCN2CC)=O)(COC)C1 CC1CC=CCC1C(=O)NCC1C=CCN1C(c1ccoc1Br)=O c1(-n2ncc(C(N(CCNC(CCOCC)=O)C)=O)n2)ccc(Cl)cc1 C(=O)(C(O)CCC(C)C)NCC1(COC)CC1.c12ccc(c(Cl)n1)c(=O)[nH]2 C1(OC)CN2CCCC2CC1CNC(=O)NC12CCC(C)(CO1)C2 CN1CCOCC1CCCNC(=O)NCC1CCCC1c1cn(C)nn1 c1(CC)cncc(C(=O)NC(C2CCOC2)CNC(=O)CCCOC)c1 c1(C(N(CC(CNC(C(C2CC(F)(F)C2)OC)=O)C)C)=O)cnn2ccn(C)c12 C(CC(=O)N1CCC(C)C(O)C1)(C(F)(F)F)NC(C1(CC#C)CCCC1)=O c1(C(=O)OC)nccnc1NC(=O)CC1(N)CCC1 c1(C(=O)OC)ccc2c(C(F)(F)F)cc(=O)oc2c1.c12cc(cs1)CC(=O)O2 N1(C(C2CCC(C(CC)(C)C)CC2)=O)CCC2C(C1)NC(=O)CCN2C c1(OC)cc(C(F)(F)F)ccc1NC(C1CN(Cc2cc(Cl)ccc2OC)C1)=O C(CC(=O)N1CCC1C(C)(C)O)(C(F)F)NC(CCNC(COC)=O)=O c1(NC(c2cc(OC)cc(Cl)c2)=O)ncnc2c1nnn2C(C)C Cc1cc(C#N)c(F)cc1NCc1cc(OC(C)(C)C)ccc1C(F)(F)F N1(C(C2(C)N(C(C=C(CC)CC)=O)CCC2)=O)CCC2(CSC2)C1 c1(C(=O)NCCCN(C(=O)C=C2CCCCC2(C)C)C)[nH]nc2c1COC2(C)C C1(C(=O)NCCc2n(CC)cnn2)CC=CCC1NC(=O)C(N1CCOCC1)C c1(C(=O)NC(C2CN(C(=O)CC(O)C3CC3)C2)C)oc2ccccc2c1CS(C)=O N1(CC2CC(SC)C2)C(=O)CCN(CCc2cccc(F)c2C)C1=O C1(OCC)CC2CN(C(=O)C(C)(C)C(C)NC(C3CC(O)C3)=O)CC12 C(CCC(C)C(=O)N(C1CN(C(=O)COCC2CCC2)CC1(C)C)C)OC C(=O)(C1=CC2CCC=CCCC12)NC1CC(NCC#N)C12CCC2 Cc1ccc2c(C(N3CCOC(C(=O)NC4CN(C)C4)C3)=O)cccc2c1 N1(C(C2CC(CC)C2)=O)CCCC(CCNC(=O)C(C)CCOC)C1 C1(NC(CC(COC)C)=O)CC2CN(C(c3ccon3)=O)CC2C1 c1(OCC(N2C3C(NC(C4CCC4)=O)C(C3)C2)=O)ccc(N2CCCCC2)cc1 C(C1CSc2ccccc21)Nc1c(N2CCN(C)CC2)cccc1.CC(F)F C(=O)(C1=NNC(=O)CC1)N(C(CNC(Cc1cc(C)cc(F)c1)=O)C1CC1)C CC1CN(C(c2csc3nccn23)=O)CC(C)C1NC(=O)CCOC1CCCC1 CC(=O)C(C)CC(C)C(=O)N1CC=C(CNC(=O)Cc2ccccc2)CC1 C1(CC(N2CC(OCC(N)=O)C2)=O)CN(C(=O)Cn2cnnc2)C(C)(C)C1 C1(CNC(C2CC2c2ccc(F)cc2)=O)(CO)CCCN(C(=O)C2=CCCC2)C1 N1(CC(=O)NC2(C(N3CC(C(N)=O)C3)=O)CC(F)C2)CCCNC1=O c1(C(N(C)CC2CCCC(NC(CCC(=O)NCC)=O)C2)=O)ccc(Cl)c(C)c1 C1(CC(=O)NC(CC)CNC(=O)CCOC2CCCOC2)CCCCCCC1 n1(CC=C)c(N2CCC(C(OC(C)(C)C)OC)C2)nnc1-c1cnc(C)[nH]1 c1(SC(C)(C)C)nnc(-c2ccccc2Cl)n1Cc1cn(C2CCOCN2)nn1 CCCC(C(=O)NC1CC(SCC(N2CC(F)C2)=O)C1)N(C)C N1(C(C(C)OC)=O)CCC2(C1)CN(C(c1nccc(OC)c1F)=O)CCO2 c1(CC(=O)NC2CN(C(C3CC(c4ccccc4)CO3)=O)C2)ccc(Cl)cn1 C1(NC(C2CCC(OC)C2)=O)CCN(CCNC(c2cc(C(N)=O)[nH]n2)=O)CC1 c1(CN2CCC(CNC(c3cc(C(C)C)on3)=O)CC2)ccc2ncnn2c1 c1(C(N(CC(C)O)CCNC(CC(CC)(F)F)=O)=O)ccc([N+](=O)[O-])cn1 CCCC(C)CC(=O)N(CCNC(c1cn(C)nc1Oc1cccnc1)=O)CC C(CS(=O)(=O)CC(=O)NCC(CC1CC1)C(=O)NCCc1cnccc1C)OC c1(N(C(C)C)C(C2COC(C)C2)=O)nc2ccc(Br)cn2c1Cl C1(CNC(=O)CN2CCCC2)(CC2CCCC2C(=O)NCC2CC2)CCCC1 C1(NC(C(C(CC)C)N2CCC(CNC(C)=O)CC2)=O)CCC2C(CC1)C2(F)F c1(C(=O)NCC(C)(C)CNC(c2cn(C3CCOC3)cn2)=O)cc(Cl)cnn1 N1(C(CC(CC)OC)=O)CCCC2(NC(C3CNC(=O)N3)=O)CCCC12 c1(CNC2CCC(NC(c3cccc(C)c3I)=O)C2)ccc([N+](=O)[O-])cn1 c1(C(N(C(C(=O)NC(c2cc(C)no2)C)(C)C2CC2)C)=O)ccc(O)cn1 c1(C(=O)NC2(C)CCN(C(C3CC4CC3C3CC43)=O)C2)ncnc2ccsc12 c1(C(C(=O)NCC)N(C)Cc2cccc(F)c2)cc(C(C)(C)C)nn1C c1(C(=O)NC2(CC=C)CCN(C(C3(C)CC3Br)=O)C2)nc[nH]c2ncnc1-2 C(C(=O)NCCCC(N1CCC(C)(C(=O)OC)CC1)=O)(c1ccccc1)=CC C1(OC)CC(CC(=O)NC2CC(C)(Nc3ncncc3C)C2)C1(C)C C1(C(=O)NCCC2CCN(C(CCC#C)=O)C2)CCCN(CC)C1 C1(NC(c2cc(CC)n(C)n2)=O)CC2CCC(C1)N2C(=O)CC(C)SC CC(C)C(C(=O)NCCC1CC1)C(C)NC(=O)Cn1[nH]cnc1=N CC(CC(=O)N1CCN(CCNC(C2CN(C)C2)=O)CC1)C(C)(C)C N1(C(c2cnc(C)n2C)=O)CC(NC(C2(C)CCC2)=O)C(C)(C)C1 N1(C(c2cc(CCC)[nH]n2)=O)CC2CCC(C1)N2C(C1(CCF)CCC1)=O C(CCCC(Cc1ccccc1)C(=O)OC)NC(c1ccccc1Cl)C C1(=O)C(C(C)(C)C)OC(C)CC(=O)NCC(OC)CN1.S(C)CC C1(C(N(C)CC2CCCN(C(=O)COCCF)C2)=O)CCCCC(C)(C)C1 C1(COCC)CN(C(=O)C=CC(F)(F)F)CCN1C(=O)CCc1cccc(O)n1 c1(C(=O)NC2CC3(CN(C(C(C4CC(F)(F)C4)OC)=O)C3)C2)ccc(C)c(C)c1N N1(C(c2c(F)cc(C)c(F)c2)=O)CC2CS(=O)(=O)CC2(NC(=O)OC(C)(C)C)C1 S(=O)(=O)(c1cccc(Br)c1F)NC1CN(C(CCNC(C)=O)=O)CC1C Cc1cccc(C)c1CNC(=O)C(N1CCCC1c1ccn(C)n1)=O c1(C(=O)NCCCCNC(=O)Cc2ccc(Cl)cc2)cc2n(n1)CCCC2 CC1(C)CC1C(=O)NCC1(NC(=O)CC23CC(C2)C3)CC1 c1(C(N2CC(N(C(C)=O)C)C(F)C2)=O)cc2c(Br)cccc2cn1 c1(CN2CCC(CC(N3C(C(=O)OC)CCC3)=O)C2)cc(F)cc(C)c1O CCCCCC(O)C(=O)N(C1CN(C(C2(c3cccc(F)c3)CC2)=O)CC1O)C C1(C(=O)NC(CC2CN(C(C3(C=C)CC3)=O)C2)C)COCCC1(F)F C(=O)(C(C)(C)C(=O)NC(c1ccccc1Br)CNC(C1CC(F)C1)=O)N(C)C C1(C(=O)OC)C2C13CC3CNC2=O.c1(SCC(C)C)ccccc1Br C1(NC(C2C(COC)CC2)=O)CCN(C(=O)C(CO)NC(C)=O)C1C c1(OC)cccc(C(=O)NCC2(NC(=O)CCCC(=O)C3CC3)CCC2)c1C C1(N(CC(=O)NC(C)C)C)C2CCNCCC12.c12ccc(cc1)OC2 C1(C(N(CCN(C(=O)Cc2ccccc2[N+](=O)[O-])C)C)=O)CCn2ccnc2C1 c1(C(N2CCC(O)(CN3CCNC3=O)CC2)=O)ccc(F)c(C(F)(F)F)c1 C(=O)(CCCCC(C)=O)NCC(CNC(C(CC)(C)OC)=O)(C)OC N1(C(c2ncn(CC)c2)=O)CCN(C(=O)CC(=O)N(C)C)C2CCCCC12 C1(n2cccn2)(C(=O)NC(C(CCC)C)C)CCN(C(c2cccnc2O)=O)CC1 C1(CCC)CN(C(c2c(C)noc2CC)=O)CC1NC(=O)Cn1cccn1 N1(C(C(C)OC2CCCC2)=O)CCC(C(=O)NCCOCCC2CC2)CC1C N1(C(CC2(OC)CCC2)=O)CC2CCCC2(CNC(c2sccc2F)=O)C1 c1(C(=O)NC(C(C)NC(C(=Cc2ccccc2)C)=O)CO)ccc(F)c(F)c1 c1(C(C)C)cc(NC(=O)CC2CC3(C2)CN(S(=O)(=O)c2cn[nH]c2)C3)ccc1Br N1(C(C(F)=CCC)=O)CC(C2CCCN(C(C3(C4(O)CCOC4)CC3)=O)C2)C1 c1(C2C(C(N3CCN(C4CCCC4O)CC3)=O)C2)c(Cl)cccc1Cl c1(CC(=O)NCC2C(CNC(C3(C)CCC(=O)N3)=O)C2)ccc2nc(O)[nH]c2c1 C(=O)(C1=CC2CCCCC12)Nc1ccc(C(N)=O)c(C(F)F)c1 CC(C)(C(=O)NCC1CN(C(c2ccc(-c3ccccc3)nc2)=O)C1)C(F)(F)F C(=O)(CC(CN(C)C)C(F)F)N1CC(CNC(C(CCC)NC(N)=O)=O)C(C)C1 CS(=O)(=O)CCCN1CCC(SC(F)(F)F)CC1.C1(N)CCOCC1 c1(C(N2CCC(N(C(c3sc(F)cc3C)=O)CC)C2)=O)ncnc2c1CCCC2 c1(C(=O)NC2CC(CCNC(c3cc(CCOC)on3)=O)C2)ncnc(C)c1C C(CCC(C)C)SCC(C)NCCC(=O)OC c1(SC)cc(C(=O)N)ccc1OCC1CC(NC2(CN)CCC2)C1.C(C)(C)(C)CCl C(C1(O)CCc2ccccc21)NCC(c1nc(Br)n2ccsc12)=O n1(CC)c(O)nc2ccc(C(=O)NCC3CC3CNC(c3cnccn3)=O)cc12 c1(N(CCCNC(C)=O)CC)ncnc(Cl)c1C.C(=O)(C(C)(C)CO)NC C1(CNC(=O)C2=CCOCC2)CC12CCN(C(c1ccc(F)c(Cl)c1)=O)CC2 C1(C#N)(C(=O)NCC2C(NC(C3CN(CCC)C(=O)C3)=O)CCC2)CCCCC1 n12nnc(c1C)c(=O)[nH]2.c1(-n2cc(-c3cc(C)no3)nn2)ccc(C(C)C)cc1 CC1(C)CC(CNC(=O)CC2CCCC(NC(C3(CO)CCCO3)=O)C2)CO1 OC1CCC(SCC2CCCC(C(F)(F)F)C2)CC1 c1(CC(C(=O)OC)NCc2cnn[nH]2)cc(F)ccc1Cl C1(NC(C(C)(F)F)=O)COC2(CCN(C(=O)Cc3cncnc3O)C2)C1 CS(=O)(=O)c1cccnc1C(=O)NCCC(O)CNC(c1cccs1)=O N1(C(C2(CCC)CCC2)=O)CC2CC2(NC(=O)C=Cc2ccncc2)C1 C1(C(N2CC(CCCCNC(CS(=O)(=O)NC)=O)C2)=O)CC(C)OC(C)C1 c1(OCC)ccccc1C(N1CCCC1C1(NC(c2nccnc2N)=O)CC1)=O c1(C(CNC(=O)CC2CN3CCN2CC3)O)nc2ccc(Br)cc2[nH]1 N1(C(c2c(CC)noc2)=O)CCCC(N(C)C(c2ccnn2CCF)=O)C1 CC(C)C(C(C)C)C(C(=O)NCCCOC1CC1)N1CCC(O)C(F)(F)C1 c1(CC)nc(C)c(C(=O)NC(C(C2N(Cc3ccccc3O)CCC2)(C)C)=O)o1 c1(CC(=O)NCCC(C)NC(c2ccnn2C2CCOC2)=O)cn(C2CC2)cn1 C1(C(N(CC(C)NC(c2c(F)ccc(Cl)c2F)=O)C)=O)CCCC2(C1)CC2(F)F C1(CNC(c2cccnc2CO)=O)COCCN1C(=O)Cc1ccns1 n1(CCCO)nc(-c2cccc(Br)n2)nc1-c1coc(Cn2ccnn2)c1 CC(C)C(CNC(=O)CCC(C)(C)F)C(=O)NCC1CCC=CO1 c1(C(=O)NC(C2CN(C(C3COC(C)C3)=O)C2)C)ccc(F)nc1 CCS(=O)CC(=O)NCC1(C(F)F)CCN(C(=O)Cn2nnnc2C(C)C)C1 C1(NC(c2cc(C)c(C)s2)=O)CC2(C1)CC(NC(=O)Cc1ccc(O)cc1Cl)C2 C1(CCC)(NC(C2CCC(C(N)=O)C2)=O)CCCN(C(c2ccc(Cl)cc2)=O)C1 N1(c2ccc(C(=O)OC)c(C)n2)CC2CN(C(=O)C3=CS(=O)CCC3)CC2C1 N1(C(C2C3CCC(=O)C23)=O)CCCCC(NC(C2(C3CCCO3)CC2)=O)C1 C1(CCNC(C(C)N(C)C)=O)(CO)CCN(C(=O)C(c2cccc(Cl)c2)N(C)C)C1 N1(CC(=O)NC(C)(CNC(c2nccnc2C(N)=O)=O)C2CC2)CCCNS1(=O)=O C1(NC(CCc2cncc(C)c2)=O)CN(C(c2cnn(CCO)c2)=O)CC12CC2 C1(C2CC2)(C(=O)NCc2ccc(CC)s2)CN(C(=O)Cc2cnns2)C1 C=C1CC(C(=O)NC2(C)CC2C)(CNC(c2cc(C)sn2)=O)C1 CCCCCCC(C)C(=O)NC(C)(CNC(=O)CCC(=O)NC)CC C12(NC(C(N3CC(CC(=O)OCC)C3)=O)=O)CCCN(CC1CO)C2 Cc1cnc(F)c(CN2CC3(CC(CC(=O)NC4CCCCC4)C3)C2)c1 N1(C(C2CCC(C)(C)CO2)=O)CC2CCC(Nc3cc(C(N)=O)ncn3)CC2C1 c1(CC)c(C(=O)NC2CCCC2NC(=O)CN(C)C(N)=O)cnn1C c1(C(=O)NCC2CN(C(c3c(C)ocn3)=O)CC2C)c(O)cc(Cl)cc1F N1(C(COCCC)=O)CC2CCCC(CNC(=O)C(O)C(C)(C)CC)C2C1 Cc1c(C=CC(=O)NC2CN(C(c3coc(CO)c3)=O)CC2(C)C)cnn1C c1(CC(=O)N(CCCC)CC2CCOCC2)cc(C)c(Cl)s1 N1(C(c2ccn(C(C)C)n2)=O)CCCC(C(=O)N(C2CCOC2=O)C)CC1 C1(NC(C2CC(O)CN2C(c2cc(O)cc(F)c2)=O)=O)CCC(O)C(O)C1 Cc1cccnc1CC(=O)NCC1(C)CCC(NC(=O)CC2CCCCC2)C1 Cc1cc(Cl)nc(N)c1C(N1CC2(C1)CN(C(=O)Cc1cc[nH]n1)C2)=O C(CCCCCN=C(NCCF)NC(c1cccs1)C)SC c1(C(=O)NC(CC)CNC(=O)CCc2cccs2)cc(C)c(F)cc1N Cn1nc(C(=O)NCC2CCCN2C(C2(C(F)(F)F)CCCCO2)=O)cc1F N1(C(C(C2CC2)OC)=O)CCC2C(C1)CN2C(=O)COc1ccccc1C(N)=O CCC(CC(C)C)C(=O)N1CCC1Cn1cc(C2(C3CC3)CC2)nn1 C1(NC(CN(CC)CC)=O)CN(C(c2ccc(C(F)(F)F)cc2Cl)=O)CC12CC2 c1(C(C)C)nnsc1C(=O)N(CCNC(=O)CN(C)C(N)=O)CCc1ccccc1 c1(OC)cc(CN2CCCC(C)(CNC(c3cccc(Br)c3)=O)C2)cc(C)c1 CC(C)C(O)CC(=O)N1C2CCC1C(NC(C1CCC(c3ccccc3)C1)=O)C2 C1(C(N2CC(OC)C(F)C2)=O)CCC(C)(C)N(C(=O)CCCCC2CC2)C1 C(=O)(C1=CCS(=O)(=O)C1)NCCN(C(CCNC(=O)C=CCl)=O)C1CCCC1 N1(C(C2CCC(C)(CC)O2)=O)CCCC2(C1)CN(C(=O)CSCC(C)C)C2 N1(C(C(CC)C)=O)CCOC2(CCN(C(c3cnc(SC4CC4)[nH]c3=N)=O)C2)C1 C1(NC(CC(C)N(C(CCC)=O)C)=O)CC2CC3C(C2)C13 C(CC(=O)NOC(CO)C(C)C)OCCN(C(CCOC)=O)C Cc1noc(C)c1CNC(=O)C(C)(C)C1CCCN1C(=O)Cc1ccoc1 C(=O)(C(C(C)(C)C)N(C)C)NCCc1cc(C(N2CCC(C)C2CO)=O)no1 n1(CC(N2CCCC(N3CCN(C(C)=O)CC3)C2)=O)c(C)nc2ccccc12 CC1CN(C(c2ccc(O)c(N)c2)=O)CCC1NC(=O)C(c1cccc(Cl)c1)O C(C(F)(F)F)(C1CC1)NC(=O)NC1CCC(NC(C(O)C2(C)CC2)=O)C1 Cc1ccc(-n2cc(NC(C34CC(n5cc(COC(C)C)nn5)C3C4)=O)nn2)s1 N1(C(c2cn(CCC)nc2)C(=O)N(CCC#N)CC2CCCO2)CCCOCC1 N1(C(C(C)N(CC)CC)=O)CCN(C(c2cnc(C(C)C)nc2C)=O)CC1C C1(C)(CNC(CN(C(C)=O)C)=O)CCCN(C(c2cnccc2C)=O)C1 n1(CC)ccc2c(N3CC(NC(c4ccc(OC)s4)=O)C4(CC4)C3)ncnc12 C12(C(=O)NC(CNC(c3c(C)ncn3C)=O)C(C)C)CCC(=O)N1CCS2 C=CCC(C)(O)C(=O)NCC1CCC(C(=O)NCCc2ccncn2)CC1 N1(C(C2C(NC(c3cccc(F)c3F)=O)CCC2)=O)CCc2c(O)cccc2C1 N1(CC(=O)OC)CCN(C(=O)C(N)C2CC2C(F)(F)F)CC1=O C1(C(=O)NC2CC(CNC(=O)Cc3cc(C4CC4)on3)C2)CC2OC1C1CC21 Cc1c(C(N2CCC3(CC3C(=O)NC(c3nncs3)C)C2)=O)oc2ccccc12 CC1(C)C(C(=O)NCC2C3CN(C(C4CC5(CCOC5)C4)=O)CC23)CCS1(=O)=O CCCC(CC)C(=O)N(C1CCN(C(C2CC(S(C)(=O)=O)C2)=O)C1)CC Cc1c[nH]c(C(=O)NC2CCN(C(c3ccc(F)cc3)=O)C2C(C)C)c1C c1(SC)sccc1C(=O)N(C1CCN(C(=O)CC(=O)N(C)Cc2nccs2)C1)C C1(NC(C2C(C(N)=O)C2)=O)CN(C(c2cocc2C(N)=O)=O)CC1n1ccnn1 Cn1nc(Br)cc1C(=O)NCC(O)CCNC(C1CC=CC1)=O N1(C(CC(CC)SC)=O)CCCN(C(c2ccc(N(C)C)cc2)=O)CC1CO.OC C1(NC(CC(COC)COC)=O)CC2CC(C1)CN(C(=O)C1=C(Cl)CCOC1)C2 c1(C(=O)NC2CCCN(C(C=CSC)=O)C2)coc2c1C(=O)NCCC2 c1(C(N2CCC2(CO)CO)C(=O)NC2(C)CC2)nnn(C(C)(C)C)n1 CCCC(CC)CCC(=O)NC(C)CCN(C(=O)C1=CC(C)(CC)C1)C CCCC(CCCNC(C1CCC(C)(C)OC1)=O)NC(c1ccc(C)c(Cl)c1)=O c1(C(N2CCN(C(c3n(C)ccn3)=O)C3C2C3)=O)ccc(=O)n2c1CCCC2 c1(C(=O)NCCN(CCC)C(c2cn[nH]c2)=O)cccc(N2CCCC2)n1 c1(CC(=O)NC2CC(NC(c3c(C)noc3)=O)C2)cn2ccccc2n1 N1(C(c2c(C)con2)=O)CCC(CN(C(C2(C(C)C)CCC2)=O)C2CC2)CC1 N1(C(C(c2ccccc2)C)=O)CCC(C2CCCN2)CC1.c12scnc1CN2 Cc1ccc(C(=O)NCC(=O)N(C(C)CNC(=O)CC2CCC(=O)O2)C)cc1C CC1(C)CC2CN(C(C3(C)CCCN3C(=O)Cc3ccccc3F)=O)CC12 C(=O)(CCCCCF)NC1CC(NC(c2c(OCC(N)=O)cccc2)=O)CC1O CC1CCCC1(C)CNC(=O)C(c1cccs1)NC(=O)C=Cc1cnn(C)c1 C1(C(=O)NCC2C(NC(c3n(C)ncc3)=O)CCC2)CC2CS(=O)(=O)CC2C1 c1(C(=O)NCC2C(NC(CCCc3nc(C)sc3)=O)CCC2)cn(C)[nH]c1=N C1(C(=O)NCC(C)(C)CSC23CC(C2)C3)CCC(C(=O)OC(C)(C)C)CC1 C(=O)(CCCCCC(C)(C)C)NC(C)CC(C)NC(c1cc(O)cc(O)n1)=O N1(C(CC(C)SC)=O)CCCN(C(c2n[nH]cc2[N+](=O)[O-])=O)CCC1 C(c1cccc(Cl)c1Cl)=CC(N1C2(CN(C(CN(C3CCSC3)C)=O)C2)CC1)=O N1(C(c2ccc(N(C)C)nc2)=O)CCC(CO)C(NC(=O)CCn2ccnn2)C1 c1(C(C)=O)cc(C(N2CCC(N(C)C(c3cnn(C)n3)=O)CC2)=O)c(C)o1 C1(CC)C(C(=O)OC)CCN1C(=O)Nc1cnn(C(C)(C)C)c1 S(=O)(=O)(c1ccc(N2CCC3CCC(C2)N3C)c(Cl)c1)N1C(C)CN(C)CC1C c1(C(=O)NCCC2CC(NC(c3cc(C(N)=O)[nH]c3)=O)C2)ncccc1C(F)F C1(NC(CCc2nc(C)c(C)o2)=O)CC(F)(F)CC1NC(c1cncnc1C)=O S(=O)(=O)(c1cccnc1NCCC1CC(C)(C)CO1)NC(c1nnnn1C)C CC(C)(C(=O)N1CCC(CNC(=O)COCC2CCCO2)C1)n1cncn1 C1(C(N(C2CCCCC2)CCNC(=O)C=Cc2ccccn2)=O)CC2C(C1)C2(F)F C(=O)(C(C)(C)C#N)NCc1ccc(C(=O)NCC(n2ccnn2)C)o1 N1(C(C(n2c(C)ncc2)C)=O)CC(CNC(c2cnc(O)s2)=O)OC(C)(C)C1 C1(CNC(CCCC#C)=O)COCCN(C(=O)CCN2CCCCC2C)C1 C=CCC(CC=C)C(=O)N1CCC(C(=O)N(C)Cc2ccncc2)C(C)(C)C1 C1(CNC(c2ccco2)=O)CN(C(C2CC3C=CCC(C2)C3)=O)CC2(CCC2)O1 C1(C(N2C(C)CCCC2C)=O)COC2(CCN(C(=O)C(C)n3cncn3)CC2)C1 C1(NC(CN(C)C)=O)CN(C(c2cnc[nH]2)=O)CC12COC2 C1(C(=O)NCC(c2ncc[nH]2)C)CC2(CC(NC(=O)C(F)(F)C(C)O)C2)C1 N1(C(c2nc(CC(C)C)sc2)=O)CCCN(C(C2CC3C=CC2C3)=O)C(C)C1 c1(C(N(C(C)CN(C)C(C2(C(F)F)CC2)=O)C)=O)ccnc(O)c1F C=CCCC(C)(C)C(=O)NC(C)(C)CN1CCN(C(C2CC2(C)Br)=O)CC1 CCCC(O)C(=O)N1CCCC1CCC1CCN(C(C2(C(F)F)CC2)=O)CC1 c1(OCC#C)cccc(NC(C2CC2C(=O)NCC2(SC)CCCC2)=O)c1 CC(N=c1[nH]c(=NCCC2CCOC(C)(C)C2)c2c(F)cccc2[nH]1)c1cncs1 CCC(C(=O)N1CCN(C(=O)Cc2ccc(OC)cc2OC(F)F)CC1)C(C)O Cc1cccc(C(N2CCCC2C(C)(C)C(=O)NCCC2(C)N=N2)=O)c1 c1(OC)ccc(Br)c(C(N2CC(CNC(c3nnsc3C)=O)C2)=O)c1C C1(C(=O)NCCc2cccc(OC)c2)CCc2nc(C(F)(F)F)ncc2C1 c1(-n2cc(C(N(C(c3nn(C)cc3N)=O)CC)C)nn2)cccc(OC)c1F Cc1cc(F)c(C(N2CC(NC3CC3)C(O)C2)=O)cc1F.C12CCCN1C2=O C1(C(=O)NC2CCCN(C(c3c(OC)ccnc3)=O)C2C)CCC2CCCCN12 CN1CC=C(CC(=O)NC2CC3CCC2C(NC(c2ncc[nH]c2=O)=O)C3)CC1 c1(OC)cccc(C=CC(=O)NC(C)CCNC(C2CCC(F)(F)C2)=O)c1 n1(C2CCCN(C(C(=O)NCC3CCCCO3)=O)CC2)nc2c(n1)CCCC2 c1(C(=O)NCC2(F)CCC(NC(C3(O)CCOCC3)=O)C2)ccnc2c1CCC2 c1(OC)cccc(NC(=O)C(C)N(C(=O)Cc2ccco2)C(C)C)c1F C1(CN(C(c2cc(CC)on2)=O)C)CN(C(=O)CC2CC(O)C2(C)C)CC12CC2 CC(C)C(C)(F)CNC(=O)C(C)CNC(C1C=CCS1)=O C1(NC(C2CCC(CC)O2)=O)CCN(C(=O)CCC2CC2(Cl)Cl)CC12CCC2 CCCCCC(C)CC(=O)NC1CCCC1CNC(c1scc2c1OCCO2)=O c1(N2C(CN(C(C(CCCCC)O)=O)C)CCC2)ccc2c(n1)CCCC2=O C12(NC(CCCOCC)=O)CCCC1N(C(=O)CC1(C3CC3)CC1)CCC2 Cc1c(C(=O)NC2CCN(C(=O)CC3COC(=O)C3)C2)[nH]c2c1CCCC2 c1(C(=O)NC2C(CC)N(C(C3Cc4ccccc4C3)=O)CC2)cccc(C#N)c1C c1(CC)cc(C(N2CC(CNC(c3cc[nH]c3C3CCC3)=O)CC2C)=O)sc1C c1(C(=O)NC2CC(F)(CNC(c3nc(NCC)oc3)=O)C2)cc(C)nc(C)c1 N1(C(c2c(CC)con2)=O)CC2CC(C)N(C(C3CCCN(C(C)C)C3)=O)C2C1 CC1(C)CN(C(=O)CC2(C)CCC2)CC1NC(=O)Cc1cc(F)ccc1F c1(OC)ccc(CN=C(NCC(c2c(C)noc2C)O)NCC(C)(C)C)cc1Br C1(C(N2CC3C(C(N(C)Cc4cc(C)no4)=O)C3C2)=O)CCCCCN1C N1(C(C(C)OCCN(C)C)=O)CCCCCC1CNC(=O)CCCN(C)C Cc1cc(F)ccc1C(c1nnnn1-c1ccccc1)NCC1CCCCS1 C(=O)(C(CC)C(C)C)NC(C1CCCCC1)C(=O)N(CCC#C)CC C(C(=O)NCC(CO)NC(=O)C=CCOc1ccccc1)(C(C)C)SC Cc1nc(C(=O)NC(C(=O)N2CCCC(C(C)C)C2)C(C)C)c(C)o1 c12cn(nn1)C2.c1(CC(N2C(C(N)=O)CC2)=O)cc(Br)cs1 C1(NC(c2c(COC)cccn2)=O)CN(C(c2cc(Cl)no2)=O)CC2CCCC12 C1(NC(COC2CCN(C(C(CC)C#N)=O)C2)=O)CC2CC1CC21CC1 N1(C(c2c(SC)cnn2C)=O)CC(NC(=O)CC2CC(OC)C2)CC2(CCC2)C1 C(=O)(CC(C)C(C)(C)C)NCC1C2N(C(C(CC)(F)F)=O)C(CC2)C1 O=C1CC(NC(C2(NC(c3cncnc3)=O)CC(CO)C2)=O)CN1 C1(CCC(=O)NC(C2CCCC2)CNC(C2N(C)CC2)=O)CCC(=O)NC1 CC1CN(C(c2cc(Cl)sc2Cl)=O)CCN1C(=O)CCCCF c1(C(=O)NC(CC=C)CNC(=O)C(C)(C)C(C)O)cc2c(nc1O)CCCCC2 c1(C(N2C(CNC(=O)CCCc3cccnc3)CCC2)=O)cccc(F)c1 c1(CC#N)ccccc1C(=O)NCCOC.C1(C=O)CC(C2CC2)C1.C1CCO1 N1(C(C2(CC#C)CCCC2)=O)CC2CC(NC(=O)CCOCC(F)(F)F)C2C1 c1(C(N2CC=C(CNC(c3n(CC)cnn3)=O)CC2)=O)ccc(OC)c(Cl)c1F CC(C)CC(O)C(C)C(=O)N1CC2(CC2)CC1CC(=O)NCC1(F)CCC1 N1(C(C(CN(CC)CC)F)=O)CC2OCC(NC(c3cn(C(C)C)nn3)=O)C2C1 c1(SC)nc(Cl)c(CN2CCN(C(c3cnn(C)c3)=O)C(C)C2)c(Cl)n1 c1(NC(CCCn2c(C)ncc2)=O)cc(F)c(Br)cc1C N1(C(=O)C=Cc2ccc(F)cc2)CCC(NC(C2(N(C)C)CC2)=O)C12CCCC2 c1(OC)ccc(C(=O)NCc2ccc3[nH]c(C)c(C)c3c2)c2[nH]ncc12 c1(OC)cc(C(=O)NCC(C(C)C)NC(c2ncn(C)c2C)=O)ccc1Cl N1(C(c2cc(C)oc2)=O)CC2CCC1C(NC(c1cc([N+](=O)[O-])nn1C)=O)C2 c1(C(=O)NC(C)C(C)C(=O)NCCC(O)C(F)F)cc(C#N)ccc1N N1(C(C2CCC(CNC(C3CC3[N+](=O)[O-])=O)CC2)=O)CCC(CO)C(O)C1 N1(C(C2(CCCC)CC2)=O)CCC(N(C(=O)CN(C2CCC2)C)C)C(C)C1 c1(C(N2C(CN(C(c3c(CC)cno3)=O)C3CC3)CCC2)=O)cnccc1OC C1(C(=O)NC(C)Cn2cncn2)CCCCC1(C)NC(=O)CN1C(=O)CNC1=O N1(C(C(C)OC(C)C)=O)CCc2c(C(N3C4COCC3C4)=O)n[nH]c2C1 C12(CNC(c3cncc(C)c3)=O)CC(NC(C3CCC3(F)F)=O)(C1)C(C)O2 c1(NC(CC(CC)N(C)C(c2cc(COC)on2)=O)=O)cc(C#N)ccc1O c1(OC)cc(CN2CC(F)CC2C(N2CCCC(Br)C2)=O)cc(C(F)(F)F)c1 c1(N2CC(C(C)C)OCC2)nc2cccc(F)c2c(=NCCN2CC3CC3C2)[nH]1 C1(CC)CCC(C)CC1NC(=O)CC1CCN(CC2(C)CCCCC2)C1 c1(C(N2CC3C(CCNC(C(C)OCC)=O)(CC3)C2)=O)c(Cl)ccc(Cl)c1O N1(C(C(C2CC2)SC)=O)CCCC2(CCN(C(C3CCC4(CCC4)CC3)=O)C2)C1 C1(CCC(=O)OC)CCN(C(C)C(=O)NCC(C)C)C1 O=S(=O)(c1cc2sc(=NCCC3CCC3)[nH]c2cc1Cl)NCCc1ccccc1Br N1(C(CCNC(C2CCCO2)=O)=O)CCC(n2cc(CC3(O)CCSC3)nn2)C1 C(=O)(C1=CCCOCC1)NC(COC)C(=O)NCc1nc(C)no1 C1(O)(CC(=O)N(C2CCCN(C(c3nc(C)sc3C)=O)C2)C)COC(C)(C)C1 c1(CC)ncsc1C(=O)NC(CNC(=O)CC1CCC2CC12)C1CC1 C1(C(=O)N(c2ccsc2)CCO)CC(F)(F)CN1CCN1CC(O)C1 c1(-n2cc(CNC(CC)(C)CCO)nn2)cccc(Cl)c1Br c1(C(N(CCN(C)C(=O)OC(C)(C)C)C)=O)ccccc1 N1(CCNC(c2c(CC)con2)=O)CCN(C(=O)CCc2cccc(O)n2)CC1 C(=O)(C(C)(C)C(=O)NC1CCCCC1CNC(c1csc(Cl)c1)=O)NC CC1(C)CN(C(c2n[nH]c(=N)[nH]2)=O)CC1NC(c1ocnc1C(F)F)=O c1(C(=O)NC(CNC(C(C)(C)n2cnnn2)=O)(C)C)cn2ncccc2n1 Cc1ccc(C(=O)NNC(=O)C2CCC(O)C2)cc1-n1ccnn1 C12CCC(CC1)CC(=O)N2.C1(OC)CC(CN(C)CC(=O)CCOC)C1.C1CC1 N1(C(C(=O)NC)C2CCC2CO)CCC(CCO)(CCO)CC1 C(C(=O)NC1CC(C)(NC(=O)CCCn2cccn2)C1)(C(C)(C)C)N(C)C c1(N(CCNC(C2C(CC)CCC2)=O)CC)ncc(O)cn1 c1(C(N(CCN(C)C)C)=O)cccc(NC(=O)C2CC2)c1 C1(NC(C(c2csnn2)N(C(C)CC)CC=C)=O)CCC(F)(F)CC1 C(=O)(C(C)(C)CCCF)NC1CCCC(C(N2CCC(OC)C2C)=O)CC1 c1(C(=O)NC2(C)CCN(C(=O)CC3CCC(C(F)(F)F)O3)C2)cc2scnc2[nH]1 c1(N2C3CC(CN(C(C4C(C)CC5CC5C4)=O)C3)C2)ncnc2cccc(Br)c12 C1(CC(F)F)(C(=O)NCC(CC)NC(=O)CC(C)F)CCOCC1 n1(CC)cc2ccc(C(=O)NC3CN(C(=O)CCSC)CCC3C)cc2n1 n1(CCC)cc(Cl)c(C(=O)NC2CCCC(NC(=O)CC3CCC(=O)N3C)C2)n1 C1(NC(CC(C)OC)=O)CCCC(NC(c2ccncc2-n2cccn2)=O)C1 c1(C(=O)NC2C3CN(C(=O)COCc4ccncc4)CC23)ccn2ccsc12 CC(C)CC(CNC(c1cc(F)ccc1O)=O)C(=O)N1CC(F)C(F)C1 c1(C(N2CCC(N(Cc3ccc(C(=O)O)s3)C3CC3)C2)=O)ccc(F)c(F)c1O N1(C(CNS(C)(=O)=O)=O)CCC2CN(C(c3coc(C(F)F)c3)=O)CC2C1 Cc1ncn(C)c(=O)c1C(=O)NC1CCCC1NC(=O)CCn1ncn(C)c1=O Cc1c(C)cccc1O.N12CCN(CC1)Cc1ccc(o1)C(=O)NC1CN2C1 N1(C(C2(C(C)(F)F)CC2)=O)CCC(N(CCO)C(C2CCCSC2)=O)C1 c1(OCC(=O)NCC(C)NC(=O)C(F)(F)C(O)C2CC2)c(F)cccc1F c1(C(N2CCN(CC(=O)N(CCCO)C3CC3)CC2)=O)cc(F)c(Cl)nc1Cl C1(CNC(COC)=O)(CO)CCCO1.C1C(CC2CC2)N1 c1(OCC(=O)N(CCCn2cc(CC(CSC)O)nn2)C)ccc(F)cc1 n1(CCC)nnnc1C(C1CCCO1)NCC1CCC(=O)N1 C(=O)(N=c1ccn(C2CC2)cc1C)S(c1ccc(CCC)cc1)(=O)=O C1(C(N(CC=C)CC=C)=O)(OC)C=C(c2ccnc(OC)c2)C=N1 n1(C(C)C)ncc(Br)c1C(N1CC2CC1C2NC(=O)C=Cc1ccco1)=O CCC(O)C(F)(F)C(=O)N1CC(NC(c2cc(F)ccc2Cl)=O)CC(C)C1 N1(C(=O)NCC(C)(C)C)CCCC1C1(NC(=O)COC2CC(F)C2)CC1 C1(C)(CNC(COCCCC(C)C)=O)COCCN(C(C2CC(=O)C2)=O)C1 C1(CN2CCC(NC(C)=O)C(F)C2)CCn2cncc2C1.n12nc(c(Cl)c1C(C)C)C2=O c1(C(N(C)CC2CCN(C(C3ON=C(C)C3C)=O)CC2)=O)c(F)cc(Cl)cc1F C1(C(N(C(c2ccncc2)C)C)=O)(CO)CCN(C(c2cnsc2)=O)C1 Cc1cccc(C(=O)NCC(C(C)C)NC(=O)C(C(C)C)n2ccnc2)c1 C1(CCC(=O)N(C2CC(OC)C2)C)CN(C(=O)CN2CCCCC2)CC1C CON=CC(=O)NC(C)CCNC(=O)C=Cc1cscn1 c1(C(=O)NCC2C(Cn3cc(CC(C)C)nn3)C2(F)F)ccc2c(c1)CC(C)O2 Cc1cc2[nH]c(C(N3CCC(CNC(c4cccc(N)c4O)=O)C3)=O)cc2o1 C1(CNC(CN(CC)CC)=O)CCC(NC(=O)C(C)n2cncn2)C1 C(CCCCCC(=O)N1CCC12CCOCC2)NC(c1ncn(C)c1)=O c1(NCC#C)nn[nH]c1C(=O)NCCC(=O)NC(C)C N1(C(CC(CCCC)NC(C2CCOC2C(C)C)=O)=O)CCN2C(=O)NCC2C1 c1(CCC(=O)NCCCNC(C(c2cn(CC)nc2)=O)=O)ccc(Br)cc1 C(=O)(CCCCC(N)=O)N(CCC)CCNC(=O)CSc1cccc(Cl)c1Cl C(=O)(C(CNC(=O)C(N1CCOC1=O)C)N(C)C)N(CCCO)C(C)C Nc1cnc(Cl)cc1C(=O)NCCC1(O)CN(C(=O)CN2CCC2C)C1 C1(C(N2CCCC(CC)(CO)C2)=O)N(C(c2n[nH]cc2Cl)=O)CCCC1(C)C C1(C)(C(=O)NC2CC(NC(C(C=C)c3ccccc3)=O)C2)CCC2CC2C1 CCCCCC(O)C(C)C(=O)NCCC1CCN(C(=O)Cc2cnoc2)CC1 C12(NC(c3c(CC)n(C)nc3)=O)CCCC1N(C(=O)C=C1CCC(C)C1)CCC2 C1(CNC(CCC2CC(NC(C3(CC=C)CC=CC3)=O)C2)=O)CC2(CCCO2)C1 C=CCCCCCC(=O)NC(CN(C(=O)C(c1ccccc1)NC(N)=O)C)CC CC(C)(C)C(C(=O)NC1CCCN(c2cc(F)ncn2)C1)c1ccccc1 c1(C(N2CCCN(C(C(C)n3cncn3)=O)CCC2)=O)coc2cc(O)ccc12 c1(N2C(COC)(CO)CCC2)ccc(S(=O)(=O)N(C)C)cn1.C1(C(=O)N)CC1(F)F N1(C(C(=O)NCC(C)(C)N2CCC2)=O)CC2CCNC(C2)C1 C1(OC)CN(C(=O)CCCn2ccnc2)CC1NC(=O)OC(C)(C)C c1(C(N2C(CC=C)(C(=O)NCC(CC3CC3)OC)CCC2)=O)cc[nH]c(=NC)c1 C1(CNC(c2[nH]cc(C)c2)=O)CN(C(c2n[nH]c3c2COC3)=O)C2CCCCC12 C=CC(CC)CC(=O)N1CC(CCNC(C2CC2c2ccccc2F)=O)C1 Cc1nc(N)c(CC(=O)NC(C(C)NC(c2n[nH]cc2C)=O)C(C)C)c(O)n1 C(C)(C(O)C(=O)NC1CC(F)(CNC(=O)CCN(C2CCCCC2)C)C1)OCC C(CC(C)(C)CC(=O)NCC1CN(C(C2(C)CSC2)=O)CCO1)OC c1(C(=O)NC(CNC(C=COCC)=O)CC(C)C)ccc(F)cc1-c1ccccc1 N1(C(C2(COC)CCCO2)=O)CCC12CN(C(c1cccc(C3CC3)c1)=O)C2 c1(CC)ccc(C)c(C(=O)N(CC(C)NC(c2cc(O)n(CC)n2)=O)C)c1 C(=O)(C(CC=CCl)c1ccccc1)NC1C(NC(c2cnc(C(C)(C)C)[nH]2)=O)C1 C(=O)(C(F)C(C)(F)F)N(C)CC1CCN(C(C2CC(OC3CC3)C2)=O)CC1 c1(C(=O)NCCC(C)N(C(C=C(C)C(F)F)=O)C)ccc2c(c1)C(=O)N(C)C2=O N1(C(=O)OCc2ccccc2)CCC(C2CC(CN3C(=O)CCC3=O)C2)C1 c1(CCN(C(C(C(C)c2ccccc2)N)=O)C)cc(Cl)cc2c1OCOC2 N1(Cc2nc(C(C)C)nn2C)CCC2(CC2C(=O)N(CC)Cc2ccccc2)C1 C(C)(CCC(=O)N(C)CCN(C)C(c1cnn(C)c1-c1ccccc1)=O)OCC c1(C(=O)NC2CC2CNC(c2n[nH]c3c2CCC3)=O)cc2c(s1)CCS(=O)(=O)C2 O=C(C1=CC2CCC(C1)C2)NC(C1CCCCC1)C(=O)N(C1CC1)CC1CCC1 C1(CCC)C(=O)NCCN1C(=O)C(Cc1cccc(F)c1)c1ccccc1 c1(OCCCOC(COCCOC)=O)ccn2ncc(CO)c2c1 C(=O)(CCCCCCCC1CC1)NC1CC(OC(C)(C)C)C12CCC2 C(c1cc[nH]c1)=CC(=O)NCCC(C)N(C(=O)Cc1cncnc1)C N1(C(C(C)(C)F)=O)CCCCC2(CCN(C(=O)CCNS(=O)(=O)C(F)(F)F)C2)C1 c1(C(N2C(C(=O)Nc3cc(OC)n[nH]3)CC2)=O)cc(Br)cc(Br)c1F c1(NC(C(=O)NCC(C2CCOC2)NC(C)=O)=O)ccnc(CN(C)C)c1 S(=O)(=O)(c1ccc(Br)cc1NC(C1CCC1C(N)=O)=O)NC(c1n(CC)ccn1)C N1(C(CC(C)C(F)F)=O)CCC(C(=O)NCc2ccnc(F)c2F)C12CCC2 C1(C(C)C)(C(=O)NCc2nncn2C)CCN(C(=O)CCC2CCC(=O)C2)C1 c1(N(C(=O)C(F)C(=O)O)CCN(C)C)ccc(Cl)c(Cl)c1 CCC(C)C(C(=O)NCCC1CC(NC(c2cccc(F)c2OC)=O)C1)OC Cc1ccc(C(=O)NC2CC3(C2)CN(C(C2CC2c2ccsc2)=O)C3)c(F)c1 N1(C(CCCC#CC)=O)CC2CCC(CNC(c3cccc(F)c3)=O)C2C1 Cc1c(C(=O)NCCC(C)NC(c2ccc([N+](=O)[O-])[nH]2)=O)nn(C)c1N Cc1ccc(NC(N2CCC(N(C)C(c3cccn(C)c3=O)=O)C2)=O)cc1C CC(F)(F)CCC(=O)NC1CCCN(C(=O)C=CCOC(C)(C)C)C1NC(N)=O CC(CO)C(=O)NCC1CCN1C(C1(N2CCCC2)CCC1)=O Cc1c(C(N2CCC(C)(CNC(C3CC3F)=O)C2)=O)ccn1CC1CC1 C1(CNC(C2CC23CCCC3)=O)CCCN(C(C2(C3CC3)CCC2)=O)C1 N1(C(C2N(C(CNC(C)=O)=O)CC2)=O)CCCC(N(c2cc(CO)ncn2)C)C1 C1(C(N(CC(CNC(CC(C)C)=O)C)C)=O)CC2(CCC2)CO1 c1(CNC(N2CC=C(C(F)(F)F)C2)=O)cccc2ccnn12 C(=O)(CC(C)(C)C(F)(F)F)NCC1(F)CC(NC(c2c(OC)cccc2O)=O)C1 c1(C2CNC(=O)C(C)O2)cccc(Cl)c1.c1(CO)nc[nH]n1.C12(CC1)C(=O)NC2 c1(C(=O)NCC(O)COC2CCC(F)(F)CC2)c2c(cc3c1CCC3)CCC2 C1(NC(C=C(CNC(c2c(C(C)C)ocn2)=O)C)=O)CCC2CC2CC1 c1(C(N(CCCCNC(=O)C2=NOCC2)C)=O)nnc(O)nc1O N1(CC(N2CC(N(C(CCC3C(C)C3)=O)C)C2)=O)CCC(CCC=CCl)CC1 c1(OC)ccncc1NC(C12CC1CN(C(C1CC(C)=NO1)=O)C2)=O c1(N(C(C)C(=O)N2CC(n3cc(CNC(=O)C4CC4)nn3)C2)C)cnc(S)n1C C(CCCCC(=O)N1CCN(C(c2ccc(Br)o2)=O)CC1CCO)OC C1(NC(CCOCC)=O)CN(C(C2CCCN2S(C)(=O)=O)=O)CCC1(C)C N1(C(C2NC(=O)OCC2)=O)CCc2ccc(CNC(=O)C(O)C3CC3)cc2CC1 CCC(O)C(C)C(=O)N1CC(C)(C)CC1CNC(C1(C(F)F)CCC(C)CC1)=O CCCCC(C(=O)N1CC2CC2(CNC(c2ccc(C)c(OC)c2)=O)C1)C(C)C C(=O)(C1=CCN(C(c2ccc(F)cn2)=O)CC1)N(C1CCC(C)(C)C1)C S(=O)(=O)(c1ccc(I)cc1)NC1CCN(Cc2cccc(CC(=O)O)c2)CC1F C(=O)(C(CC(C)C)ONC(c1cc(CO)[nH]n1)=O)N(CCC)CC1CC1 C(CCCC(N)=O)NC(c1c(CNC(C2(C(C)(F)F)CC2)=O)c[nH]n1)=O CCC(F)(F)CC(=O)N(CCN(C)C(c1cccn1C1CCCC1)=O)C(C)C c1(OC)cc(C(=O)NCC(C)(C)CNC(C2CC3(CCC3O)C2)=O)cnc1C N1(C(c2c(CC)cncc2)=O)CCC2CN(C(=O)Cc3sc(O)nc3O)C2C1 C(CC(C)N=c1[nH]c2c(F)cccc2o1)NC(c1c(C)nccn1)=O c1(C(N2CCC(NC(C(CC)SC)=O)C2)=O)cc(-c2ccncc2)nn1C N1(CC(C)NC(=O)CC2CCC3CC23)CCN(C(=O)CC2(C)CCCCC2)CC1 N#CC1(CC(=O)NC(CNC(C2CCC3(CCC3)O2)=O)C2CCC2)CCOCC1 N1(C(Cn2ccc(C)n2)=O)C(CC(=O)NC(C)(C)CCN(C)C)C2CCCC12 C1(CN(C(=O)CN(C)C(C)=O)CC)CCCN1C(=O)CCCc1ccccn1 C1(CC(N2C(CNC(CCOCC#C)=O)CCCC2)=O)COCC(C)(C)O1 N1(C(C(C=C)(F)F)=O)CCC2(C1)CN(C(=O)CCCCC)CCO2 Nc1cnccc1C(=O)NC1CCCCC1NC(c1coc(O)n1)=O N1(C(C(CC(C)C)C)=O)CC2CC(O)C1C2NC(c1cc(Br)n(C)n1)=O C1(O)(C(C)C)CCN(C(=O)CSCc2ccc(F)cc2)CC1 C1(C(=O)NC(CNC(CNC(c2ccc(C)s2)=O)=O)C2CC2)CCC=CCCC1 N1(C(c2c(CCC)n(CCO)nc2)=O)CC2CC(C1)N(C(=O)C=C(Cl)Cl)C2 C12(C(=O)NC(CCCNC(c3scc(C)c3)=O)c3ccccc3)CCOCC1C2 C12(NC(C(C)OCCCC)=O)CCC(C1)N(C(=O)CC1(C)CCOCC1)C2 c1(C(N(C)C)C2CC2)cccnc1C(=O)NCC1CC(NC(C2CCCS2)=O)C1 C=CCC(CC(F)F)NC(=O)CN(C(=O)CCn1cccc1)C1CC1 N1(C(c2nc(CNC(C(C)S(C)(=O)=O)=O)oc2)=O)CCCCC(F)(F)C1 C(C)(CCC(=O)NC(C)C(CO)NC(c1conn1)=O)OCC C#CCC(C)(CC)C(=O)NCC(C1CCC1)NC(c1sc(C2CC2)nc1C)=O C(=O)(CC(C(F)(F)F)C1CC1)N(C1CC2CC1N(C(=O)C(C)(C)C(C)(F)F)C2)C CC1CN(C(C2CC(O)C2)=O)CCCN1C(=O)C=Cc1ccc(C(F)(F)F)o1 c1(C(C(=O)Nc2ccccc2C)N(CC#N)CC)cccc(C(F)(F)F)c1F c1(C(N(C2C(N(C(=O)CC3CC4(CC4)C3)C)CCCC2)C)=O)ccc2c(c1)CC2 N1(C(=O)NC(c2ccccc2I)Cc2ncccc2F)CCCCc2ccccc21 C1(CNC(COC(CC)C)=O)CN(C(=O)C(F)(F)CCn2cccn2)CC12CC2 C1(NC(=O)C(F)OC(F)(F)F)CCC(O)CN(C(C2COC(=O)C2)=O)C1 c12cc(ccc1F)NC(=O)NC2.C1(CC)CCCCC1CC12CC(OC)(C1)C2 C1(NC(c2ccc(OCC)c(C)c2)=O)CC2(CCN(C(=O)C=CC(F)(F)F)C2)C1 Cc1nn(C)c(C)c1C(=O)NCC1CC(C(=O)NCCC(C)N(C)C)CO1 c1(C(N(CC(CNC(CC2(C=C)CCC2)=O)C)C)=O)cnc(O)n(C)c1=O CCC(C#N)(CC)C(=O)NC(C1CCN(C(c2c(F)ccc(F)c2O)=O)C1)C Cc1cc(F)ncc1CNc1cnc(Cl)cc1C(=O)Nc1nc(C(N)=O)cn1C C1(CC=C)(NC(=O)C(C)=C(C)CC)CC2CCC(C1)N2C(C1CCC(F)C1)=O CCC(C)C(O)CC(=O)N1CCC(C(=O)NCC(C)(F)C(C)C)C(O)C1 C(=O)(C(O)CCS(C)=O)NCN(CCNC(C1CCN(C(C(C)C)=O)CC1)=O)C(N)=O c1(C(N2CCC(NC(C(CC)=CC)=O)C2C2CC2)=O)ccc2c(n1)CCO2 C1(C(=O)NCCCCCN(C)C(c2cc(O)nc(O)n2)=O)CC(F)(F)C1(F)F c1(C(=O)NC2CCN(C(CN3CC(CC)C3)=O)C2)ccc(OC)nc1OC N1(C(C=CC(CC)=CC)=O)C2CCCC1CN(C(C1CC(OC(F)(F)F)C1)=O)C2 CC(CCC(=O)NCC(C1CC1)Nc1cc(C(F)(F)F)ncn1)N(C)C Cn1ccc(=NCc2cccc(C(=O)N(CCCO)CCN)c2)nc1O c1(C(N2CC=CC(NC(C=C(CC)C)=O)C2)=O)cccc2c1CC(C)(C)C2 CC(C)C(O)(C(=O)N1CC=CC(NC(=O)Cn2ncn(C)c2=O)C1)C(F)(F)F c1(C(=O)NCC2CC3(CC(CN)C3)C2)cc2n(n1)CCNC2=O O=S(=O)(c1ccc2[nH]c(=NCC(Cl)(Cl)Cl)ccc2c1)N1CSCCC1CO N1(C(c2c(C)c(F)ccc2N)=O)CCC2CN(C(=O)CC3CCOC3)CC2CC1 C(=O)(C(C1=CCSC1)N1CC(CCO)OC(C)(C)C1)N(C)CCF C(=O)(CC(C)C(C)(C)NC(=O)CC1CCC2CC12)NC1(CC(C)C)CC1 N1(CC(N2C(C(C)(C)C)C(NC(c3cc(F)cs3)=O)CC2)=O)CCC(=O)NC1=O C(=O)(CC(C)CC(C)C)N1C(C(=O)Nc2cccc(C)c2)CSCC1 C(=O)(CCCC(F)(F)CO)NCc1c(C(=O)NCC(CN(C)C)O)c[nH]n1 N1(C(C2N(CC)CCOC2)=O)CCC=C(C(=O)Nc2cccc3c2CCC3)C1 N1(CC)CCC(O)C(C(=O)NCCOc2ccc(Br)cc2)C1.C1CS(=O)(=O)O1 c1(SCC(=O)CN2CCC(F)(F)C2)nc2ccccc2o1 C(=O)(C1CCCc2scnc21)NCC1(NC(c2cncc(OC)c2)=O)CCCC1 C#Cc1ccc(C(=O)NC2(C)CCCN(C(c3coc(C(F)F)n3)=O)C2)nc1 C1(C(=O)NC2CC(NC(C3CC(CC)C3)=O)C2)Cc2ccc(F)cc2O1 CC1CN(C(c2n[nH]cc2F)=O)CC(C)C1NC(c1cccc(OC(F)F)c1)=O n1(CCC)nccc1S(=O)(=O)N1N=CCC1(C)C n1(CC)cnc2nc(=NCCC3CC4(CCC4)CO3)[nH]c(NCCC(F)(F)Cl)c12 C#CCC(C)(CC)C(=O)N1CC(O)CC1C(=O)N(C1CN(C2CC2)C1)C C1(C(N2CC(O)(CN(C(=O)C=Cc3nccs3)C)C2)=O)CCC2(CCOCC2)C1 CCC(O)C(C)C(=O)Nc1cccc(CNC(=O)C=CCOC)c1 c1(C(N(C)Cc2ccccc2CNC(=O)C2=CSCS2)=O)ccc(=O)n(C)c1 CCCCC(O)C(=O)N1CC2CC2(CNC(=O)C(C)NC(C2CCCC2)=O)C1 c1(C(c2n(CC=C)nnn2)NCC2CC=CCC2)ccnc(C(F)(F)F)c1 CCC(C(=O)N1CC(CNC(=O)CC2CSCCO2)C1)N1CCCC1=O CCCC(C(=O)NC1CCCN(C(=O)Cn2cc(C3CC3)nn2)CCC1)C(C)C C(CC(CC)C(=O)NCCC1CC(NC(c2cnn(C)n2)=O)C1)=CC C1(CNC(c2cn(CCC)nc2)=O)CC2CC1CN2C(=O)C(C)SC(F)(F)F N1(C(C=CC=CC)=O)CC(C)CN(C(=O)CCc2ccccc2Br)C(C)C1 n1(CC(=O)NC(C2CCCCN2C(=O)CCC(=O)OC)C)ccc([N+](=O)[O-])n1 c1(C(N2C(C)C(NC(=O)CSCCC(F)(F)F)CCC2)=O)ccn2nncc2c1 C1(C(=O)NCCC(=C)CNC(c2cccc(OC(C)C)n2)=O)C2CCC(F)(F)C12 C1(CCc2ccccc2)(CO)CCCN(NC(c2c(C)n(CC3CC3)cc2)=O)C1 c1(CC)nc(C(=O)NCCc2n[nH]cc2C(N2CCOCC2C(C)O)=O)c(C)o1 c1(C(N2C(C(N(CC)Cc3cccnc3)=O)CC2)=O)c(Cl)cc(Cl)cc1Cl C12(CCOCC1)OCCC1C(C1)C(=O)NC(CO)C(=O)NC2.CC c1(CN(C)C)ccc(C(=O)NC2CN(C(c3cc(C(F)F)cs3)=O)C2)cn1 N1(C(C=CCN(C(C(CCC)(C)O)=O)C)=O)CC2(CNC(=O)C2)C1 c1(CSC)ccc(C(c2nnnn2C(C)(C)C)NC(c2cn(C)nc2C)C)cn1 C#CC1(C(=O)NCCCN2CCCC2C)CCN(C(c2cc(O)nn2C)=O)C1 CC1CN(C(=O)NCC2CC(CS(N)(=O)=O)C2)CCN1c1cnn(C)c1 c1(CC)sccc1C(N1CC(CCNC(=O)CC2CCOC2)(OC)C1)=O N1(C(C2CC(C)SCC2)=O)CCC(O)(CNC(=O)C2=NOCC2)CC1 CCCC(CCC)=CC(=O)NC(C1CCN(C(c2cncc(N)c2)=O)CC1)(C)C N1(C(C2N(C(CCc3ncn(C)c3)=O)C3(CC2)CC3)=O)CCC2(CC1)CC2C#N N1(C(C(C)N(C)C(C2CCC(F)CC2)=O)=O)CCCCC2(CCC2)C1 C(=O)(C1=NN(C2CC2)C(=O)CC1)NC1CCCN(C(c2c(N)non2)=O)CC1F C12(CNC(Cc3c(C)ccs3)=O)CC1CN(C(=O)CC1CC3C=CC1C3)C2 C1(C(=O)Nc2nc(C(=O)OCC)c(CC)s2)CCC2CCCCC2C1 C(N=c1nc2c(c[nH]1)CCC2)C1C(NC(=O)CCN2CCOCC2)C1 c1(C(=O)NCC(CN(C(C2(COC)CC2)=O)C)O)ccc2nsnc2c1 C(=O)(C(CC)C(=O)N1CC(O)(CCNC(=O)C(C)COC)C1)OCC Cc1cc(Br)cc(Cl)c1C(N1CCC(C)(C(=O)NCc2ccc(Cl)cc2)C1)=O C12(CC(=O)NCC3(O)CCN(C(c4nc(=N)[nH]cc4)=O)C3)CCCN1CCC2 Cc1nc(-c2ccccc2)ccc1C(=O)NCC12CC1CN(C(=O)C(C)O)C2 C(C)(CC(=O)NC1C=CCN(C(=O)CC(F)F)C1)(C(F)(F)F)N(C)C C1(CNC(c2occc2Br)=O)CN(C(c2ccc(Cl)nn2)=O)CCCO1 c1(C(N2CC(CCC)OCC2)C(=O)NCCOCC)ccc2c(c1)C(=O)NCC2 CC1COc2ccc(C(=O)Nc3cn(C4CCCN(C(=O)C5CC5)C4)nn3)cc21 c1(NC(=O)Cc2nc(-c3cnn(C4CCCCO4)c3)cs2)nnc(Cl)cc1Br C(=O)(C(C)C(F)(F)C(F)F)NC1CCCCCN(C(c2cc(CC)c(C)s2)=O)C1 C(CCC(F)(F)C(F)(F)F)NC(C(COC(C)=O)C)=O C(c1cccc(Cl)c1)=C(C)C(=O)NCC12CC1CN(C(=O)C(C)(C)C1CCO1)C2 c1(C(N(CCOCCNC(c2cc(C)no2)=O)C)=O)cccc2oncc12 N1(C(c2nn(C)nc2Br)C(=O)NCC2(CC3CC3)CC2)CCCC(F)(F)CC1 N1(C(c2c(C)nc(CCC)o2)=O)CC(NC(C2CN(C)CCN2C)=O)CC(C)C1 C(=O)(C1=CC2C=CC(C1)C2)N1C(C)CC(NC(CCCCCCC)=O)C1 c1(C(=O)NCc2nc(CNC(=O)COCC3CCCO3)on2)n[nH]c2c1CCC2 C=C1CCN(C(=O)COCCC(C)C)C(C(N2CC3(CC3CC)C2)=O)C1 c1(C(=O)NCc2cc(C(=O)NC(C3CCOC3)(C)C)n[nH]2)cccc2ccoc12 S(=O)(=O)(c1ccccc1F)N1C(Nc2ncnc(N(C)C)c2[N+](=O)[O-])C=CC1 c1(C(N2CCN(CCCc3cccc(C)c3)CC2)COC)cccc([N+](=O)[O-])c1 CN1CCN(Cc2cn(Cc3nc4cc(Br)ccc4s3)nn2)c2ccc(Br)cc21 N1(C(C2(COC)CC=CCC2)=O)CC2(CCN(C(c3ccsc3C(F)F)=O)C2)C1 C1(CNC(C(C)=CC)=O)CCCCN(C(C2CC(CO)N(C)C2)=O)C1 c1(NC(C2C(c3c(OC)ccc4c3CCC4)C2)=O)ccc2c(c1)CCN(C)C2 C1(C)(CC(=O)NC(CC#C)CC)CCN(C(c2cnc(OC)s2)=O)C1 CC1C(=O)N(CC(=O)NC2CCCCN(C(=O)C(C)(O)C3CC3)C2)C(=O)C1C c1(C(C)C)ccsc1C(=O)NC(C1CCN(C(C2(CC(F)F)CC2)=O)C1)C CCC(CC(=O)NC1CC(F)CN(C(c2ccc(C3CC3)o2)=O)C1)C(C)C C1(C(=O)NC2CC(NC(C3CCN(C(C)C)CC3)=O)C2)CC2CCC(C1)S2(F)F CC1CCN(C(=O)C(=O)NCC(C2CCCCN2C(C2(C)COC2)=O)(C)C)CC1 N1(C(c2nccc(C)n2)=O)CCC(NC(c2ncoc2Br)=O)C(C(C)C)C1 S(=O)(=O)(c1ccc(NCC=CCO)cc1Br)NC(C)CCc1ccncc1 C1(CNC(C2CCC(C(C)=O)O2)=O)N(C(c2ccc[nH]2)=O)CCC1(C)C C12(C)CC(CCO1)NC(=O)C1(CCOC1)NC2=O.c1(CC)ccc(O)c(C)c1 CN1CCC(C)(C(=O)NC2CC(C(F)C(=O)Nc3cccnc3)C2)C1=O N1(C(CN(CCOC)C)=O)CCCC(O)(CNC(c2cccc(CO)n2)=O)C1 C(C(O)(CNC(=O)Nc1ccc(C2CCC2)nc1)CO)OC C(=O)(C(C)(C)CN1CCOCC1)NC1C(CNC(C(c2cnn(C)c2)C)=O)CC1 c1(CNCC2N(C(C3CCC(NC(C)=O)CC3)=O)CCCC2)cnc(C)[nH]c1=N C1(CC)CN(C(=O)C2=COCC2)CCN1C(c1nc(C)oc1OCC)=O c1(OC)ccc(C(C)NC(=O)NN2CCOC(c3nccn3C)C2)nc1 Cn1cc(C(c2nnnn2CC(F)F)NCC2(C)CCO2)nn1 c1(NC(C(CN(C(=O)CC2CC2)C)(C)N(C)C)=O)ccccc1CO c1(C2C(C(=O)NC3C(C(=O)NC(c4cnn(C)n4)C)C3)C2)ccc(Br)s1 Cc1cc(C(N2CC(NC(c3ccco3)=O)CC(C)C2)=O)ccc1Cl N1(C(c2c(COC)ccs2)=O)CCN(C(=O)C(n2cnc(C#N)n2)C)CCC1C N1(C(C=CC(=O)N(C)C)=O)CC2CCN(C(c3cc(Cl)ccc3N)=O)CC(C2)C1 C1(CN2C(C(=O)NC3CC(C(N)=O)C3)CCC2)CCS(=O)(=O)CC1 C1(CNC(C(C)(C)OCC)=O)C(CC)CCN1C(c1cc[nH]c1C)=O Cn1nc(C(N2CC3C(C(=O)NN4CCCOCC4)C3C2)=O)ccc1=O c1(C2(C(=O)NCC3(COC)CCCC3)CCCO2)cccc(Br)c1 N1(c2cc(C)nc(C3CC3)n2)CC2CCCC(NC(C3(F)CCOC3)=O)C2C1 C1(NC(c2cnc(CC)[nH]2)=O)CCCCC12CCN(C(=O)COCCOC)C2 C(=O)(CCC(=O)N(C)C)N(c1nnc(C2CCC(=O)CC2)s1)CC CN1CCCc2cc(CC(N3CC(N)C(F)(F)C3)=O)ccc21 c1(C(=O)NCCC2(OC)CN(C(C(CCC)CC)=O)C2)cnn2c1CC(C)CC2 C#CCC(C)(CC)C(=O)NC1CC(NC(=O)CC2(C=C)CCCCC2)CC1O C1(CNC(CC(CNC(C(C)NC(N)=O)=O)O)=O)CCC(C)(C)O1 N1(C(Cn2c(C)csc2=O)=O)CCC2(CC1)CC2NC(C1CCCCN1C)=O CP1(=O)CC(NC(C2(c3ccc(Cl)cc3)CCC2)=O)C(O)C1 N1(C(c2cnc3n2CCC3)=O)CCC2C1CCCN2S(=O)(=O)c1cccnc1 C1(O)(CN(C(=O)C(C2CC2)N(C)C)C)CCN(C(C2Cc3nncn3C2)=O)CC1 c1(C(=O)NCC2(CNC(c3c(CC)noc3)=O)CCCC2)cccc(F)c1OC C12(C(=O)NCCCCC(C)NC(CNC(=O)OC)=O)CCCC1OCC2 C(=O)(C(C)(C)C(C)O)NCC(c1ccccc1)NC(Cc1c(C)noc1)=O C(C(F)(F)CN(C(=O)CN(C(c1sccc1C)=O)CC1CC1)C)OC Cc1cc(C)c2nc(N3CCN(C(c4ccn(C(C)C)n4)=O)CC3)sc2c1 c1(C(N2CCC(O)(C(C)NC(CCC(=C)C)=O)CC2)=O)nccc2ccn(C)c12 N1(C(CN(C)C)=O)CC(C(O)C(=O)NCc2cc[nH]n2)C1 C=C(C)C1OCCCC1C(=O)NCCN(C(=O)C(C)(C)C1CCOC1)C1CC1 N1(C(C2(C#N)CC2C(F)(F)F)=O)CCC2CCC(C1)N2C(=O)C#CC1CC1 C(=O)(C(C)CCCC)NCC(CC=C)NC(=O)CCC(C)CC C(CCCC(C)NC(c1nc(Br)sc1C)=O)NC(C(C)OC)=O c1(C(C)C)cccc(-n2cc(CCCCNC(c3cnc(C4CC4)s3)=O)nn2)c1 c1(C(=O)NCCC(C)CCNC(=O)CNC(N)=O)cc2c(Br)cc(F)cc2[nH]1 CCC(CC)CC(=O)NC(C)(CNC(c1ccnc(O)c1Br)=O)CC C1(CCCC)CN(C(=O)C2=C(Cl)CC2)CCN1C(=O)Cc1nonc1C N1(C(C2C(C)OC(C)C2)=O)CCN(C(=O)CN(C)C)C(CC2CC2)C1 C1(NC(c2ccc(S(C)(=O)=O)o2)c2n(CCSC)nnn2)CS(=O)(=O)N(C)C1(C)C n1(CC)nc(C(N2CC(N(C(=O)C(C)CCOC)C)C2)=O)c(Br)n1 C1(C(=O)NC(C(=O)OCC)CC)C=CCN(C(=O)CNC=O)C1 CC1(C)CN(C(=O)C=Cc2ccccc2)CC1C(=O)NCC1CCCC2(CC2)C1 C(=O)(N=c1ccn(C)[nH]1)C12C(CN(C(CCNC(=O)NC)=O)C1)CC2 CC1(C(=O)NCC(=O)NC2CC2O)CCCN(C(C2CC(C)(C)C2)=O)C1 C(=O)(CCCC(C)NC(c1ccc(C#N)cn1)=O)NC1(c2nc(C)on2)CC1 C1(N(C)C)(CNC(=NCC2CC2)NCC2OCCC2(C)C)CCCCC1 N1(C(c2ncn(CC)n2)=O)CCOCC1CNC(C1CC1F)=O C1(CC(=O)NC2CN(C(c3cc(O)ccc3F)=O)CC2O)CC2CCC1CC2 c1(OC)ccc(C(N2CC(NC(=O)CC3CC=CCN3C)CC2(C)C)=O)nc1Cl CC1CCCC(CONC(C)(C)C)(NC(=O)N(CCCOCCO)C)C1 N1(C(c2cc(OC)cc(C)c2)=O)CCC(C(=O)NCCCP(C)(C)=O)C(C)(C)C1 N1(C(C2C(NC(C(C)Cn3ccnc3)=O)COCC2)=O)CCC(O)CC12CC2 c1(CC)onc(C2CCCOC2)c1C(=O)N(C(C)CNC(C)=O)C N1(C(COCCCC)=O)CC2CCN(C(c3ccncc3C)=O)CC2C1 N1(C(C2CC(C#N)C2)=O)CCN(C(=O)CCc2ccoc2)C(C2CC2)C1 C1(C(N2CCC(c3ccc(C#N)cc3)CC2)=O)Cc2nccnc2C1 C1(CC)CN(C(=O)CC2OCCO2)CC1NC(=O)CCC1C(=O)NN=C1C N1(C(CC2(N(C(n3c(C)nnn3)=O)C)CC2)=O)CCC(N(C)C)CC1 c1(-c2n(CCC(C)C)nc(Cn3cncn3)n2)cc2c(F)cccc2[nH]1 c1(CNC(N2CC(OCOC)C2)=O)sc(Cc2ccccc2)nc1C CCCC(C)(C)CC(=O)N(C(C)C(=O)NCc1nncn1C1CC1)CC C(C)(c1ccccc1C)=CC(=O)NC(C1CCN(C(C(C=CC)O)=O)C1)C N1(C(C(C=CCCC)O)=O)CCCC(C2CN(C(=O)C=CC3CCOC3)C2)C1 c1(Nc2c(CN(CC(CC)(C)OC)C=O)cccc2)ncnc(OC)c1Cl C12(C(=O)NCC=C)CCC(C(=O)Nc3cc(OCC)ncn3)(CC1)CC2 Nc1c(C(N2CCC3(CC2)CC3NC(C2CC(F)C2)=O)=O)cnc(Cl)c1F n1(CCC(=O)NCCN2CCOCC2)cc(CNc2ccccc2)nn1 c1(C(C(N2CCC(C)(CNC(CSCC#C)=O)C2)=O)C)ccc(F)c(F)c1 C1(C(=O)NCC=CC)C2CCN(C(=O)CN3CCCCC3)CC12 c1(CC)ccc(C(N2CCC(CN(C)C(C3CCCC(=O)N3)=O)C2)=O)c(C)n1 Cc1nn(C)c2cc(-c3nc(CCCN(C)C)nn3-c3ccc(Cl)c(F)c3)cnc12 C1(C(=O)NC2CC(CCNC(CCc3cnn(C)n3)=O)C2)CC2CCC1NC2=O C(CCO)(CC(C)C)N.c1(C(N(CC)CC)=O)cc(C2CC2)n(C)n1 C1(OC)CN(C(=O)CCC2CCCC(O)C2)CC1NC(=O)CN(C)C C1(NC(c2nn(C)c(CC(=O)NC)c2)=O)CC2(C1)CC(CF)C2 C1(C(=O)NCC2(O)CC3CCC2O3)CN(C(=O)C=Cc2ccoc2)CC12CC2 c1(CN2C(C(N3CCC(CCCO)CC3)=O)CSCC2)ccc(Cl)c([N+](=O)[O-])c1 c1(CCC(=O)NCC(CC)NC(c2cnnn2CC)=O)ccc(O)nn1 C=CCC(CNC(C1OCCC1C(C)C)=O)C(=O)Nc1cncc(N(C)C)c1 C1(NCC2(O)CN(C(C3C(C(C)C)(CC)C3)=O)C2)CC2CCCCC12 CCCC(C(=O)OC)C(=O)NC1CCCCC1C(N1CCC12CC(O)C2)=O c1(NCc2[nH]cc(C#N)c2)cccc2cnc(Cl)cc12.N12CCCC1C=CC2=O C(=O)(C(CCOC)NC(=O)CC(CC)SC)N(CCCOCC)C C1(NC(C(CC)NC(C)=O)=O)CCCC12CN(C(c1nc(Cl)c(Cl)s1)=O)C2 c1(CC(=O)NC2CC(NCc3ccc(F)cn3)C2)cccc(C(F)(F)F)c1 CS(=O)c1ccc(C(=O)NCC2COCCN2C(=O)CCCN=[N+]=[N-])cc1 C1(C(=O)NCCc2cn(CCCCC)nn2)CCC2C(CC1)C2(F)F c1(C(N(CCCCNC(c2ccn(C)c(=O)c2)=O)C)=O)ccnc2c1nnn2C CC(C)C(CNC(C1(C)CC1(F)Cl)=O)NC(=O)CC1C=CCC1 c1(C(N(CCN(C(=O)CC(F)F)C(C)C)C)=O)cnc(S)n1-c1cnn(C)c1 C1(NC(NCC(=O)NC(C)C)=NCCN2CCCC(C)C2)CCCC2(CC1)CC2 C1(C(=O)NC2(CNC(c3cnc(C(F)(F)F)s3)=O)CC2)CC2CSCC(C1)C2 C(=O)(C1=Cc2ccccc2C1)N1CC(OCC)(CNC(=O)C(C)SC(C)C)C1 N1(C(C(C=C)C)=O)CCC(C(=O)N(C2CCC2O)C)C(C)(C)C1 C1(OC)(CNC2(C(=O)O)CCCO2)CCOC1 N1(C(C2C=C(C)CN2)=O)C(C(=O)O)CC2CCCC12 c1(C(=O)NC2CC(C)N(C(=O)CCCCNC(N)=O)CC2)nnn2c1CCCC2 C#Cc1cc(F)c(C(N2CC(NC(=O)Cc3ccon3)CC(O)C2)=O)c(F)c1 c1(C(C)C)[nH]ccc1C(=O)NC1CC1NC(=O)Cn1cccn1 c1(CN(c2ccc(Cl)o2)C(N(C(C)C(C)C)CC)=O)cccc(F)c1 Cc1nc2c(s1)CCCC2C(=O)NC1CN(C(=O)C(=O)Cc2ccccc2)C1 c1(OC)ccc(C(N2CCOC(CCNC(C3(SC)CC3)=O)C2)=O)c(F)n1 C1(CNC(C(C)C)=O)CN(C(=O)Cc2ccccc2N2CCCC2)C2CC12 N1(C(C(C2CC2)NC(CCOCC(C)(C)C)=O)=O)CCNC(=O)CC1 C1(SC)CC(NC(=O)CNC(=O)COCCF)C1(C)C CCC(C)CC(C)C(=O)N1CCCC1(C)CNC(C1CC1(C)C)=O Cc1cc(C(=O)NCCCC(C)(C)NC(c2cc(CCCO)on2)=O)ccc1Cl C1(NC(c2c(CC)nccc2)=O)CCCN(c2ccc(C(F)(F)F)nn2)CC1 c1(NC(Cc2cccc(C)c2)=O)ccc2c(c1)CN(C(=O)C(O)CC(C)C)CC2 N1(C(C2C(C(=O)OCC)C2)=O)C2CCC1CC(NC(c1csc3nccn13)=O)C2 C1(C(=O)NC2CCOC(C(=O)NCCc3ncccn3)C2)CC2C(C1)C2(F)F CC(C)(COC(=O)CCN(C)CCO)C1CCCC1 C1(CC=C)(C(=O)NC2COCC2CC)CCCN1C(=O)CNC(=O)OCC N1(C(c2ncccn2)C)CCC(NC(=O)CCC2NC(=O)NC2=O)C(C)C1 c1(C(N2C3(CNC(c4cnc(C)[nH]4)=O)CCC3CC2)=O)nn2c(c1C)OCCC2 C(=O)(CCCC(F)F)NCC1(O)CCN(C(C(C)OCCC(C)C)=O)C1 Cn1nncc1C(C)(C)NC(c1cn(CCNC(=O)C(F)n2ccnc2)nn1)=O C=C1CCN(C(=O)C(c2ccnn2C)O)C(C(=O)NCC2(N(C)C)CC2)C1 N1(C(C(=O)NCc2c(C)cc(I)cc2)=O)CCCCC1[Si](C)(C)C c1(CC(=O)NC2C(NC(c3c(C)nc(CC)s3)=O)CC2)ccc(O)c(C)c1 c1(-c2ccccn2)c[nH]c(=NC2CC3CC2C3)o1 c1(C(=O)NC(CNC(c2c(CCC)occ2)=O)(C)C(C)C)cc2ncccc2s1 c1(C(=O)NC2CCN(C(CC(C)OC)=O)C2)ccc(SC)c([N+](=O)[O-])c1 c1(C(=O)NCC(CN(C(C(N2CCSCC2)C)=O)C)O)ccc([N+](=O)[O-])s1 c1(C(=O)NC2CCC(N(C(C3C(C)C3)=O)C)CC2)cc2c[nH]cnc-2n1 C1(CCC)CC(C(=O)NCC2(CO)CCN(C(=O)C(O)C3CCC3)C2)CCO1 N1(C(CCC)=O)CCCC(Oc2ccc(C)cc2)C1.C12C=CCC(C1)NC2=O N1(C(CSC)=O)CCC(O)(C2CCN(C(=O)CC3CCC(C)CO3)CC2)C1 c1(OC)cc(C(=O)NC2CCC(NC(C3CCC34CCCO4)=O)CC2)cc(C)n1 N1(CC(CC2CCCO2)OCC)CCc2nc(Cc3ccc(F)cc3)sc2C1 C(N=c1[nH]c(=NCCC(C)CO)[nH]c2ccc(Cl)cc12)c1c(OCC)cc(Cl)cc1 N1(C(C(C(C)C)(C)O)=O)CCCC2(C1)CN(C(C1CCCCC1)=O)CCO2 c1(CC)cccc(C(=O)NCC2(O)CCCN(C(C3CC(C)(C)CO3)=O)C2)c1O Cc1nc(Cl)ncc1NC(=O)CC1CC(C)(C)CN1C(=O)CC12CCCC1C2 c1(C(=O)OC)ccnc(CNC(C2CCN2C(=O)CC(C)C2CCCCC2)=O)c1 c1(CNC(C2C(NC(C(CCC)OCC)=O)C2(C)C)=O)ccn(C)c(=O)c1 c1(C(=O)NCCCC(C)NC(c2ccc3c(c2)CC3)=O)ccc(C#N)cc1F C1(NC(=O)CC2COCC2O)CCCCC1C(=O)NC1CC2CCCC12 c1(CC(=O)NCC(C(C)(C)C)NC(CC(COC)C)=O)ccc2sccc2c1 c1nc(C(C(=O)NCC2CC2)NCc2ccns2)n[nH]1 c1(CC)ccc(F)cc1NC(C1C2CCC(C2)C1NC(C1CN(C(C)C)C1)=O)=O N1(C(c2cn(C(C)C)nn2)=O)CCCC(C)C1CNC(c1cc(O)cs1)=O CC(C(=O)NO)NC(=O)C(C)CN(C(=O)CCCC(=O)NC1CC1)C C1(C(=O)NC(Cn2cc(CCC(C)=O)nn2)C)CCC(F)(F)CO1 C1(C(=O)NCCC2CCC(C)CC2)CC2(CCN1C(=O)C(=O)C1CCCC1)CC2 Cc1ncsc1C=CC(=O)NCCC1CC(NC(C2CC23CCCC3)=O)C1 c1(C(N2CCC(CCCCNC(CC)=O)CC2)=O)ccc(C#N)c(O)c1 C(=O)(CC(C)(C)C)N(CC(C)NC(c1n[nH]cc1Cl)=O)C C1(C(C)NC(c2nc(CCC)oc2)=O)CCN(C(c2nncs2)=O)CC1 C1(NC(c2c(CC)ccs2)=O)CCCC(NC(c2coc(C(C)OC)n2)=O)CC1 C1(CNC(c2c(C)nc(C)[nH]2)=O)CC2CCC1N(C(c1cccc(O)c1)=O)C2 c1(-c2scc(NC(C3CN(C(C)=O)C3)=O)n2)ccc2c(c1)OCO2 C1(C(N(CC#C)CCO)=O)N(C(=O)C(O)CN2CCCC2)CC12CCCC2 c1(C(=O)NCC(CCOC)NC(c2c(CC)nc(C)[nH]2)=O)cccc(Cl)c1Cl CC(O)C(F)(F)C(=O)N1CC(CCNC(=O)C(F)(F)C(O)C2CC2)C1 C1(C(=O)NCC2(CNC(c3cnc(C)o3)=O)CCCC2)CCn2ccnc2C1 C(=O)(CCCCCCn1cc(C(c2ncc(C(=O)OC)s2)O)nn1)NC N1(C(C2CCC(OCC)CC2)=O)CCN(C(=O)C(=O)NC2CCOC2)CC1C Cc1cc(NC(C2CC2NCc2ccc(CO)cc2)=O)cc(C)c1I C1(COC)(NC(c2cccc(F)c2Cl)=O)CCCN(C(C2CC(CF)C2)=O)C1 Cc1c(F)ccc(-c2cnc(CC(=O)NCCOc3ccccn3)nc2)c1C c1(C(=O)NCC2CCN(C(C3CC(CC)C3)=O)CC2)c(C(C)C)cccc1C C1(CNC(CCC#C)=O)CCCCN1C(=O)CNC(c1ccsc1)=O C1(C(=O)NCC(C)C(=O)N(CCCF)C)CCCOCC1 N1(C(c2ccc(CC)s2)=O)CC2CCOC2(CNC(=O)C=CC(C)CC)C1 C1(C(N2CCC(NC(CC)=O)C2)=O)CN(C(c2sccc2C)=O)CC12CC2 CCCCC(O)CC(=O)N(C(C)CCNC(c1cc(C(=O)C(C)C)c[nH]1)=O)C C1(CNC(=O)C(c2ccccc2)C2CC2)CN(C(=O)CCCC2CC2)CC12CC2 C1(C2CCN(C(C3CSCN3C)=O)CC2)(NC(C(C2CCCOC2)NC)=O)CC1 c1(CN2CCN(c3c(C)ncnc3O)CC2)ccc2c(c1)CN(C)C2 n1(C(C)C)ncc2c(NC3CC(NC(C4(CF)CC4)=O)C3)ncnc12 C1(CC(=O)NCCOC2CCN(C(=O)CC3CCC34CCC4)C2)CC2(CCC2)C1 c1(SC)cc(F)ccc1C(N1CC2(NC(=O)Cc3cncn3C)CCC1C2)=O c1(N(CC(N2CCN(C(=O)C=Cc3ncc[nH]3)CC2)=O)C)ccnc2ccccc12 C(CCC(=O)N(C(C)CO)CCO)(C(C)C)NC(c1cc(OC)ncc1)=O c1(CC(N2C3CN(C(c4[nH]cc(CC)c4)=O)C(C3)C2)=O)ccc2nc(O)[nH]c2c1 CCCC(C)(C)CC(=O)NC1CCC1NC(=O)CCCC1CC1 C(=O)(C1=CCCSC1)N(C1CN(C(=O)Cc2ncncc2Cl)CC1F)C N1(C(C(CC)N(C)C)=O)CCOC(C2CN(C(=O)CC(O)CC)C2)C1 C1(CNC(CN2CC(C)(C)C2)=O)CCCC12CCN(C(C1(CF)CC1)=O)CC2 C1(C(=O)NCc2c(OC)cccn2)CC(C)CN(C(=O)C(c2ccc(C)s2)C)C1 C12(NC(C3=CC(C)(CC)C3)=O)CCCC1(F)CN(C(=O)CNC(=O)NC)C2 c1(C(=O)OC)cc(O)ncc1CNC(c1ccc(CN2CCCC2)cc1)=O c1(C(=O)NC2(C)CN(C(C3C(C)(COC)C3)=O)C2)ccc2occ(C)c2c1 C(=O)(CC(O)CNC(=O)Cc1ccc(O)cn1)NCC(c1nccs1)C c1(CC)nc(C(=O)N(CCNC(C2CCCC2C)=O)CC)co1 N1(C(=O)NCC)CCCCCC1.C12(CC(F)C1)C(=O)OC2 C1(C2(O)CN(C(C3CCCCC3O)=O)C2)(CNC(C2(C#N)CCCOC2)=O)CC1 CC1(C)CCC(C)(NC(=O)CC2CN(C(C3CC(=C4CC4)C3)=O)C(C)(C)C2)CC1 c1(CCC)cc(C(N2CCCC2CNC(=O)CSc2ccncc2)=O)c(C)o1 NC1CCCS(=O)(=O)C1Cc1cccc(CO)c1 N1(C(c2c(OC(C)C)ccc(F)c2)=O)CCN(C(=O)CCC#N)C(C)C1C C1(NC(=O)CSc2cccc[n+]2[O-])CC2(CCCN(C(c3cnc(S)[nH]3)=O)C2)C1 c1(C(=O)NC(C(=O)OC)CC2CCOC2)ccc(N)cc1C(F)F C1(F)(C(N(CCC)CCN(C)C)=O)CN(C(=O)CCc2cnoc2)C1 C(C(C)(C)C(=O)N1CCC(NC(C2CCCO2)=O)C1)N(C)C CCCC(C)(CC)C(=O)N1CCCC(CN=C(NC(C)CC)NC2CCCC2)C1 Cc1ccc(C=CC(N2CC3CC(C2)C3NC(c2nccn2C)=O)=O)c(C)c1 Cc1ccc(CC(N2CC(C)C(O)C2)=O)cc1C.C(C=O)O C1(NC(=O)CC(F)(F)c2ccccc2)CCN(C(=O)C=CC(F)(F)F)C12CC2 C1(C(NOCC(=O)N(CC(C)(C)OCCC)CC)=O)CC12CCCCC2 c1(C(=O)NCCC(C)NC(C2CCC(=O)N2C2CC2)=O)cc([N+](=O)[O-])cnc1N N1(C(C2N(S(C)(=O)=O)CCC2)=O)CC2=C(C1)CN(C(=O)C(C1CCOCC1)F)C2 c1(C(=O)NC(C(C)NC(C=CCC)=O)CO)cc2c(=O)cc[nH]c2s1 c1(C(N(C)CC2C(NC(c3cccc(CC)c3)=O)CCC2)=O)[nH]ccc(=O)c1C C=CC(C)(C)CC(=O)N1CCC(NC(=O)Cc2cnsc2)C1C C1(N(CCOC)Cc2ccc(Br)s2)CCN(c2ccc(OC)cn2)CC1 N1(C=O)C(C(N2CC(C(=O)O)C2)=O)CC1C.C1(CCOCC)(CO)CC1 CC(CC(C)(C)C)C(C(=O)NC1CCOCC1)N1CCCCC1C1CCC1CO C1(CNC(=O)NCC2(c3ccccc3)CC3(CC3)C2)CC(O)C12CCC2 c1(Nc2c(CC(=O)NCc3cc(C#N)sc3)cccc2)cc(Br)cc([N+](=O)[O-])c1 c1(-c2nc(CC(C)OC)nn2CC2CCC2)csc(S(C)(=O)=O)c1 c1(OCC)cccc(=NC(=O)C2CCN(C(=O)CCCCBr)CC2)[nH]1 N12CCCC(C1)OCC2=O.N1(C(=O)Cc2ccco2)CCC(N(C)CCO)C1 c1(OC)cc(CN2CC(O)CC2C(=O)Nc2cccc(Cl)c2O)ccc1C C1(C(=O)NC(C2N(C(c3ccc(C)o3)=O)CCC2)(C)C)CC2(CCCCC2)C1 Cc1c(CC(N2CCC(C)C2CNC(=O)C(c2ccc(F)cc2)O)=O)ncn1C C1(CNC(C2(CC(C)=O)CCCC2)=O)CC(C)N(C(c2cc(C)c(C)o2)=O)C1 C1(NC(CCCOCCC)=O)CCN(C(c2cc(COC)ccn2)=O)CC1C C(CCCC(=O)NC1(CCNC(c2cc(C)cc(Cl)c2)=O)CCC1)(OC)OC C1(C2CC2)(C(=O)NC(c2nccc(O)n2)C)CN(C(c2n[nH]cc2[N+](=O)[O-])=O)C1 c1(C(N(C(C)CCNC(C2CC(C(N)=O)C2)=O)C)=O)ccc(=O)n2c1CCCC2 N1(C(c2c(OCC)ccc(F)c2)=O)CCCCCC(NC(=O)C(C(C)C)SC)C1 C(CC(C)(C)CC(=O)NCC1COCC1NC(C1CC=C(C(C)C)CC1)=O)OC c1(CC)cc(F)ccc1C(=O)NCC1CN(C(C2CC3(CC(N(C)C)C3)C2)=O)C1 c1(OCC)cccc(C(N2CCC(C(=O)NCC(O)CF)(CF)C2)=O)c1 N1(C(C)=O)CC(NC(=O)CCC2CC2(Cl)Cl)C2(CCC2)C1 c1(C(N2CC(N(C(C(COC)C)=O)C)C3(C2)CC3)=O)cc2c(Cl)nccc2s1 C#CC1CC2(CC2)CN1C(C1CC2CCC(C1)N2C(C1CCSCC1)=O)=O C1(NC(CC(C)NC(N)=O)=O)CN(C(=O)CC(C)(C)c2ccccc2)CC1F C1(CNC(C(CCC)CC)=O)CN2CCCCC2CN1C(C1CCCC1)=O C1(NC(C(C)Oc2ccccc2)=O)CC2(NC(c3csnn3)=O)COC1C2 C(=O)(C#CC1(C)COC1)N1CCC(N(C(c2c(CC)n(C)nc2)=O)C)C1 c1(CCNC(C2(N(C(CC3C(C)OCC3)=O)C3CC3)CC2)=O)ccnc(O)c1 c1(C(N2CC3C(CN(C(CN(CCOC)C)=O)C)C3C2)=O)ccn2ccnc2c1 CC1CC(=O)CCC1C(=O)NC1CC(C)N(C(=O)C=CC2CC2)C1 N1(C(c2scc(OC)c2)=O)CC(NC(c2cc(C)nc(O)n2)=O)C2(CC2)C1 Cc1nc(NC2CCN(C(=O)COc3ccsn3)CC2C)c2c(C)csc2n1 C(CCC(C)C(=O)N1CCC(N(C)C)C(C)C1)OC.c12ccnc(c1)C(=O)NC2 C(=O)(CC(O)CC(C)C)N1CCC(COC)(NC(=O)C(C)n2ccnn2)C1 c1(OC)ccc(CC(N2CCC(O)(CN(C)C(c3cc(C)c(Cl)s3)=O)C2)=O)nc1 c1(CN(CC)Cc2nncn2C)nc(-c2ccco2)nn1CCN1CCOCC1 c1(C(=O)NCC(C)CNC(=O)COCC2(F)CC2)ccc(C(C)=O)cc1Br c1(C(=O)NCC(C)N(C)C)ccc(CNC(=O)C(N)=O)o1 C1(NC(C2C(C)OC(C)C2)=O)CC2CCC1N(C(c1cccc3c1OCC3)=O)C2 c1(NC(C2C=CC(NC(c3nc(C)sc3C)=O)C2)=O)ccc2ncnc(O)c2c1 N1(C(C(C)=CCOC(C)(C)C)=O)CSCC1N.CCCC=CCCC Cc1nccc(Cl)c1C(=O)NCC1(CNC(C2CCC(=O)N2)=O)CC12CCC2 c1(C(=O)NC(CC)CNC(=O)C(n2nnnc2C(C)(C)C)C)cnccc1OC Cc1cccc2oc(C(=O)NC3CN(C(=O)CCC4CCC4)C3)cc12 N1CCC2CC2N(C(c2ccc(C)c(F)c2)=O)CC1.c1(CC)cnn(CC)c1 C1(C(=O)NCCCCNC(C(C)NS(C)(=O)=O)=O)CCOC(=O)CC1 c1(Cn2cc(CONC(c3n(C)ccc3)=O)nn2)cc(F)cc([N+](=O)[O-])c1 N1(C(C(CC)(C)F)=O)C2CCC1C(CNC(=O)CCNC(C1CCC1)=O)C2 c1(CC)n[nH]cc1C(=O)NC(Cc1cc[nH]n1)C(=O)NC(C)CCF c1(C(N2CCC(C(C)(C)NC(c3cscc3F)=O)CC2)=O)ccc(S(N)(=O)=O)o1 c1(OC)cc(OC)c(C(C)NC(=O)C(=O)NCCc2nnc(C)s2)cc1C CCCC(CNC(C1CC2CCC(C1)C2)=O)C(=O)NCCCN1CCOCC1 c1(C(N2CCCC(CCNC(c3c(CC)cno3)=O)C2)=O)nccc(C)c1F C(=O)(N=c1[nH][nH]c2nc(C)ccc12)C1CCCN(C(C)=O)CC1 C1(C(N2CCC(CN(C)C(C3CCCC4CC34)=O)CC2)=O)CC2(CCCCC2)C1 c1(C(N(CC(C)NC(C2CC3(CC3)CO2)=O)CC)=O)sc2cncn2c1C c1(C(N2CCC3NCCC23)C(=O)OC)ccc(F)cc1F C1(CCCNC(C(C)(C)c2cscn2)=O)CCN(C(=O)CC2(C#N)CC2)CC1 N1(C(C(c2c(C)cccc2)(C)C)=O)CCC(NC(=O)CC(O)C2CC2)C(C)(C)C1 C1(C)(CN(CC(=O)OC(C)C)C)NC(=O)NC1=O.c12ccc(cc1)[nH]c2=O C(=O)(C1CCCn2nccc21)N1C2(CN(C(=O)OC(C)(C)C)C2)SCCC1 C#CCC(C(=O)NCC1CC1CC(=O)NCC(CO)C(C)C)C1CC1 Cc1cc(C(N2CC(NC(=O)Cn3ncc(Br)n3)C3(CC3)C2)=O)cc(C)c1O N1(C(C(C)Cc2cnc[nH]2)=O)CCCOC(CNC(=O)C(C)(C)N2CCCC2)C1 c1(C(=O)NC23CCN(C(CCCCC)=O)CC2C3)ccc(S(C)=O)cc1 c1(C(=O)NCCC2CC(NC(C(C=CC)O)=O)C2)c(C(F)(F)Cl)n[nH]c1C C(=O)(C1CCOc2ccc(Cl)cc21)NCC(CC(C)C)NC(c1cnc[nH]1)=O c1(C(=O)NCC(C)CN(C(=O)CN2CC3CC3C2)C)coc(C2CC2)n1 N1(C(c2cc(C)c(Br)o2)=O)CC2CC1CN2C(c1ccccc1OC(F)F)=O N1(C(C2N3C(C)CN(CC3)C2)=O)CC2CCCC(C1)N2C(=O)CCC1CC1(Cl)Cl CC(CF)CC(=O)NC1(C(=O)NCC2CCC(NC(c3ccccc3)=O)C2)CC1 c1(-c2nc(-c3ccc(F)cn3)nn2Cc2c(F)cccc2I)ccc2nccn2c1 C1(OC)CN(C(=O)Cc2cc(C(F)(F)F)n[nH]2)CC1NC(=O)CN(C)C c1(OC)ccc(C(=O)NCCN(C)C(C2C(c3ccccc3)C2(F)F)=O)c(F)n1 S(=O)(=O)(c1c[nH]c2cc(Cl)ccc12)N1CC2C(C(=O)NC)C2C1 c1(CN(C(CC)=O)CC(=O)NC(c2ccccc2)(C)C)ccncc1OCC(F)F c1(OCC)ccnc2ccc(NC(C3CC3NC(c3cc(C)cs3)=O)=O)cc12 O=C(C(O)Cc1ccccc1)NC(CCCNC(=O)CC1CC(F)(F)C1)C1CC1 c1(C(N(C2CCCN(C(c3cccc(N)n3)=O)C2)C)=O)ccc2c(c1)CC(=O)N2 c1(C(N2CC(NC(C(CC)NC(C)=O)=O)C(C)CC2)=O)cc(S(C)(=O)=O)co1 C1(CNC(c2c(CC)cns2)=O)N(C(=O)CC2CCCOC2)CCCC1(C)C C(C(CNC(=O)Cc1cscn1)OC)NC(CN(CCOC)C)=O CC(C)CC(C(=O)NC1(C)CCCN(C(C2(C)CCCNS2(=O)=O)=O)C1)C(N)=O N1(C(c2cccc(Cl)c2O)=O)CC2(CCCN(C(c3cnn(CCO)c3)=O)C2)C1 C(=O)(C1=Cc2ccc(Cl)cc2OC1)NC(C)CCCCNC(=O)C1CC1 c1(CNC(C(C)(C)CF)=O)nc(CNC(c2ccc(Cl)cc2N)=O)cc(O)n1 c1(CCC)cc(C(=O)N(C(C)C(=O)N(CCCCO)C)CC)no1 N1(C(Cc2c(C)nc[nH]2)=O)CC(n2cc(C(C)(C)CO)nn2)C(C)C1 C1(NC(COC2CN(C(CC)=O)C2)=O)CCOC2(CCCC2)C1 c1(NC(C(C2CN(C(CCCOCCC)=O)C2)OC)=O)ccc(O)cc1Cl c1(C(=O)NCC2CN(C(C3CCC(F)C3)=O)CCO2)cccc(C#CCO)c1 c1(C(N2CC(CC(=O)Nc3cccnn3)(OC)C2)=O)cccc2c1OCC2 c1(C(N2CC(NC(C(C)(C3CC3)OC)=O)(CO)C2)=O)ccn(C)c(=O)c1.C(C)(C)N N1(C(C(=O)NCCn2ccc(C)n2)=O)CCCc2c(N3CCCC3)cccc21 c1(NC(C(C2CCN(C(C3(Cl)CCC3)=O)CC2)C)=O)ccc2ccncc2c1 c1(C(=O)NC(CN(C)C)C(=O)NCC2(C)CC(O)C2)ccc2c(c1)CC2 c1(C(C)NCCSC)nc(C(C)(C)OC)nn1-c1nccn1C C1(CC(=O)NCC(CNC(CN(CCOC)C)=O)(C)O)N2CCC1CC2 C1(CNC(C(CC)OC)=O)CC2(CCC2)CN1C(c1cc(Br)cn1C)=O CCCCC(C(=O)N(CC(C1CCCC1)O)C)NC(c1cccc(CC#N)c1)=O Cc1cccc(C(N2CCC(CNC(=O)COC3CCCC3)C2)=O)c1I Cc1cc(F)cc(Cl)c1NC(=O)NC1CC1C(N1CC(=O)NC(C)C1)=O c1(C(N2CC(C)(NC(=O)C(F)(F)F)C2)=O)cc(C)n(CCN)n1.CCO Cc1cc2cc(C(NC3CCc4ccc(F)cc43)C3CC3)ccc2n1C C1(F)(CC(=O)NC(C)C)CCN(C(=O)CC2CCOC2)C1 C1(O)(CNC(C(C(C)C)O)=O)CCCN(C(C2CCC(O)CC2)=O)C1 Cc1ccc(NCc2coc(C)n2)c(OC2CCOC2)c1 C(=O)(C1=CCS(=O)(=O)C1)NCCC(C)N(C)C(c1nncn1C)=O Cc1cc(C(=O)NCC2CC(NC(=O)CN(C)C)C2)cc(Cl)c1Br S(=O)(=O)(c1ccccc1[N+](=O)[O-])NC(C1C(C(=C)C)OCCC1)=O N1(C(c2cccc(OC)n2)=O)CCC(C2(O)CN(C(=O)C(C)CN(C)C)C2)CC1 C1(NC(=O)C2=C(Cl)CCC2)CCCCCN(C(=O)Cc2ccc(Br)cc2)C1 C1(c2ccccc2)(C(=O)NC(C)CCCNC(C2CC2F)=O)CCN(C)C1 N1(C(c2c(CCNC(C(CC)CN(C)C)=O)n[nH]c2)=O)CC2CCC(C1)O2 Cc1ccc(C(=O)Nc2cccc(NC(C3(C(F)(F)F)CCC3)=O)c2)cc1 C1(C(N2CCC(C(=O)OC)C2)=O)(NC(=O)C(=O)NC(C)C)CCCC1C CC(CCC(=O)N(CCCNC(c1cc2n(n1)CCC2)=O)C)S(C)(=O)=O N1(C(COCCC)=O)CCOC2(CCN(C(c3nc(C(F)(F)F)cn3C)=O)C2)C1 Cc1ccc(C=CC(=O)NCC2CN(C(c3cnc(C)nc3C(C)C)=O)C2)cc1 c1(C(=O)NCC(C)N(C(c2c(CC)cno2)=O)CC)ccc2ccncc2n1 C1(C)(C(N(CCC)CCNC(=O)Cn2nc(C)c(Cl)c2C)=O)CC(C)OC(C)C1 C1(OCC(C(=O)CNCC(=O)NC2C(C(=O)OC)C2(C)C)=O)CCCN(C(C)=O)C1 Cc1ncc(C=CC(=O)NC2CC(CNC(=O)C=Cc3cncs3)C2)s1 c1(NC(=O)NC(CC)CO)c(Cl)cc(S(=O)(=O)NC(C)(C)C)cc1Cl c1(CC)cc(C(=O)NC2C=CC(CNC(C3CCCS3)=O)C2)ccc1O N1(C(C=CCCC)=O)CCCC2(CC(NC(=O)CC34COC(CF)(C3)C4)CO2)C1 N1(C(Cc2cn(C)nc2)=O)CC2CCCC(NC(C3CSCCS3)=O)C2C1 CC(C)(CNC(c1n[nH]cc1C1CC1)=O)Cn1cc(-c2ccsc2)nn1 C#CCC(CC(F)F)C(=O)NCCCN(C(C1CCC(F)(F)CC1)=O)C1CC1 CC1CCCC(O)(C(=O)N(CCCNC(=O)CCOc2ccccc2F)C)CC1 C(CCCCC)(C(=O)Nc1cccc(Cl)c1C)N1CC(C)CC(CC)C1 Cc1cc2ccnc(NCc3ccc4cccc(Cl)c4n3)c2c(C)n1 c1(C(N2CCC(N(C(=O)CCC(F)F)CC)C2)=O)cc2c(o1)CCCNC2=O C1(CC)C(NC(c2c[nH]nc2-c2ccn(C)n2)=O)CCN1C(=O)Cc1ccco1 CC(C)CCC(C)N(C)C(C1CCN(C(=O)COCC(F)F)C1)=O C1C(C(C)C)C(=O)N1C1CC1.c1(C(CO)NC(COCC(=O)OC)=O)cnn(C)c1 c1(CC(=O)NC2CC(NC(c3cn(CCO)nn3)=O)CC2O)c[nH]ccc1=O C(=O)(C1=C(C)CCCC1)NCCCC(CCC)NC(c1ccc(OC)cn1)=O N1(C(C(C2CC2)SC)=O)CCN(C)CC1C(=O)NOCC1CC(O)C1(C)C N1(C(C2C(C)CC(=O)N2)=O)CCCCC(CNC(=O)CC2(C)OCCO2)C1 c1(CNC(C2N(Cc3ccc(C(=O)OC)cc3)CC(O)C2)=O)cccc(Br)c1Cl c1(C(=O)NC(C2CCN(C(COCCC)=O)C2)C)cc2cccnn2c1 C1(NC(c2c(COC)cco2)=O)CCN(C(c2cc[nH]n2)=O)C1C(C)(C)C c1(C(N2C3CCC(CNC(CC(COC)C)=O)(C3)C2)=O)ccc2c(c1)CCO2 C1(C(F)F)(CNC(CC2N(C)CCC2)=O)CCN(C(C2(C(C)(C)O)CCC2)=O)C1 c1(CN(C(=O)CC2CN(Cc3ccc(Br)cc3)C2)CC)ccc2ncccc2c1 C1(NC(c2cc(COC)sc2)=O)CN(C(=O)CN(C)C)CCC1C.C1C(=O)N1 N1(C(CC(CC)O)=O)CCC2(CNC(c3[nH]c(O)nc3C)=O)CCCC12 C#Cc1ccc(C(=O)NCC2CC23CCN(C(=O)Cc2ccsc2)CC3)c(F)c1 C#CCC(C)(C(=O)N1CCSCCC1C)NC(=O)CC1(C#N)CC1 C(=O)(C1CSc2ccccc21)NCC(CNC(c1nc(C)[nH]n1)=O)(C)O CC1(C)CCC12CCN(C(c1cc(Cl)c(F)cc1F)=O)CC2 C1(C(=O)NC(C2CCCOC2)CC)C=CCN1C(=O)CCCN(C)C c1(SCC(=O)N(CCCNC(C2CCCC2O)=O)C(C)C)ccccc1Cl CN1CC(O)CC1(C)C(=O)NC1CN(C(c2ncn(C)n2)=O)C1 C1(CNC2(O)CCN(C(=O)OC(C)(C)C)C2)CCCCNC1=O c1(C(N2CCC(CNC(Cn3c(C)ncc3)=O)C2)=O)snc2ccccc12 c1(C(=O)NCC(CO)N(C)C)c[nH]c2cccnc12.C12CC(C)(C1)NC2=O C1(CC)CN(C(=O)CCn2cc(-c3ccsc3)nn2)CC(C)S1(=O)=O c1(C(=O)OCC)ccc(CNC(Cc2ccccc2)C(OC(F)F)OCC)cn1 C1(NC(c2cnc(-c3ccccc3)o2)=O)CCC(NC(c2n[nH]cc2Cl)=O)CC1 c1(C(N2CCC(NC(=O)Cn3cc(Cl)cn3)C2C(F)(F)F)=O)cc(F)ccc1F c1(OC)cc(I)c(CSC2CCN(C3CCCCC3c3ccc(Cl)cc3)C2)cc1OC c1(C(N(C)CCOCCNC(=O)CC#N)=O)cncc2sccc12 c1(COC)ccc(C(N2CCCCC2c2nc(=O)o[nH]2)=O)c(OC)c1 Cc1ccc(C(N2C3CCC2C(F)C(NC(C2CC2C)=O)C3)=O)c([N+](=O)[O-])c1 N1(C(C)=O)CCc2sc(C(=O)NC3CCn4nccc4C3)cc2C1 C(C1c2ccsc2CCN1C(c1ncoc1C1CC1)=O)NC(C1(OC)CC1)=O C=CCCC(C(=O)N1CCC(CN=[N+]=[N-])CC1)NC(=O)C(C)CCOC c1(C(=O)NCC(CNC(c2nccc(OC)c2)=O)O)ccc(P(C)(C)=O)o1 c1(C(N2CCCC(CN(C(C(SC)SC)=O)C)C2)=O)cccc(F)c1O C1(CN(C(COC(CC)C)=O)C2CC2)CCCN1C(=O)C(F)n1ccnc1 c1(C(N(C)CC2CCCC(NC(CCSC)=O)C2)=O)cnc2n[nH]c(C)c2c1 N1(C(c2cc(C(=O)OCC)n[nH]2)=O)CC2CCC1C(C(=O)NC1CC(C)C1)C2 c1(OC(C)C(N2CC(NC(=O)CCF)C(c3cncn3C)C2)=O)cccc(N)c1 c1(C(N(CCn2cc(-c3ncn(CC)n3)nn2)CC)=O)cnc2sccc2c1 N1(C(C(C)n2cncn2)=O)C2CCCC1CC(NC(C13CC(CO1)C3)=O)C2 C1(C(=O)NC(CN(C(C2(OC)CC2)=O)C)C)CCCC(C)(C)C1 C12(C(=O)NC(CC(C)NC(C3(O)CCCC3)=O)C)CCCN(CC1)C2 N1(C(CC(CC)C)=O)CCC(C2CCCN(CCC(C)C)C2)C1 C(=O)(C(C)CC(F)F)NC1(CCNC(c2cccc(C(C)=O)c2)=O)CCC1 N1(CC2CN(C(=O)OC(C)(C)C)C3(C2)CCC3)CC(=O)Nc2cc(Br)c(Br)cc21 c1(NC(C(C2CN(C(c3cnc(C)s3)=O)C2)O)=O)c(C(N)=O)cccc1Br Cc1cnc(NC(=O)C(COC(C)(C)C)NC(c2cccc(Cl)c2)C)cc1I CC1=NOC(CC(N2CC(C)(NC(=O)CSc3nncn3C3CC3)C2)=O)C1 c1(CC(N2CCN(C3CCCN(C(C(CC)C)=O)C3)CC2)=O)cnc(Cl)cc1C c1(NC(c2c[nH]nc2CNC(C2CN(C3COC3)C2)=O)=O)cccc(O)c1 c1(C(=O)NC(CNC(CCC(C)SC)=O)(C)C(C)C)cccc2ncnn12 c1(OC)cc(C(=O)NC2CN(C(c3ncccc3F)=O)CC2C)c(Cl)cc1Cl c1(SC(C)(C)C)ccnc(NC(=O)CC2CCN2C(C2(CSC3CC3)CC2)=O)c1 Cc1cc(C(N2CCN(C(C3CC3CC(C)C)=O)CC2C2CC2)=O)c(C)cn1 CC(C)CCCOCC(=O)NC(C1CCN(C(=O)Cc2ccsc2)C1)C N1(Cc2ccc(CN(CCCNC(=O)C(=O)N(C)C)C)o2)CCC(F)C1 C1(NC(CC2C(C)(C)C(NC(=O)Cc3ccco3)C2)=O)CCC(C#N)CC1 N1(C(C2OCCN(C(CSCCCC)=O)C2)=O)CCC(CO)C1(C)C N1(C(C(CC=C)OC)=O)CCCC(F)(CNC(c2cnccc2Br)=O)C1 C12(C(=O)NCC=CCC)CC(CO1)N(C(C1CC13CCCCC3)=O)C2 C1(NC(CCC2CCC(=O)NC2)=O)CCN(C(c2ccc(O)cc2)=O)CC1F C#Cc1ccc(NC(=O)COC2CN(C(c3cc(C)c(C)s3)=O)C2)c(C)c1 c1(CC)[nH]nc(C(N2CC(CNC(=O)CNC(c3cccs3)=O)C(C)C2)=O)c1C C#CCC(C)(C)C(=O)NC(CNC(c1ccc(C2CC2)o1)=O)CCOC c1(C(=O)NCCN(C(C(=O)NCC)=O)CCOC)cc(Cl)c(CC)cc1F N1(C(C(C)(F)F)=O)CCC(NC(=O)CC2CCCC2O)C(F)C1 C1(NC(COCCOC)=O)CCC2(CC1)CN(C(=O)C(F)=C(C)C1CC1)CCO2 c12c(cnn1C)C(=O)NC2.C(=O)(CC(=O)OC)NC1C(CNNc2nccs2)C1.O C(C)(C)(CCO)N(C(=O)CCC1CCC(NC(=O)OC(C)(C)C)C1)C C(=O)(C1=CC(C)(C)C1)NC1C(CNC(c2n(CC)ncc2)=O)COC1 c1(NCC(C)CN(C)C)ccc(S(=O)(=O)NC2C=CC(CO)C2)c(Br)c1 C(=O)(C(C)(C)SC1CCC1)NCC1(CCNC(C(C)N(S(C)(=O)=O)C)=O)CC1 N1(c2cccc(CNCC3CC(OCC)C34CCC4)c2)CCS(=O)(=O)CC1 N1(C(CC(CCC)NC(C2CCCC2F)=O)=O)CCC12CCC(O)CC2 C1(COC)(CNC(=O)CC2CSCCS2)CCCN1c1cccnn1 C(=O)(CC(C)(C)C(=O)OC)NC(c1ccc(CC)cc1)C(=O)NC(CC)C1CC1 c1(C(N(C2CCN(C(C3(COC)CCC3)=O)CC2)CCC)=O)cc(C)sc1C C1(CNC(C2C(C)C2)=O)CN(C(c2ccccc2C(C)(F)F)=O)CCC1(F)F C1(C(=O)NCc2ncn(C)c2)CC2(CCN1C(=O)C=Cc1cscn1)CC2 c1(-c2cnc(OC)c(O)c2)cccc2cc(C(=O)Nc3cc(Cl)cnc3O)sc12 N1(C(C2(CNC(CN(C)C(=O)C3CC3)=O)CC2)=O)CCC2CCN(C)C2C1 N1(C(C(C)C2CCC2)=O)CC(NC(=O)C=Cc2cnn(C)c2)CC12CCCCC2 N1(CC(=O)NC2C(NC(C(C)N(C)CC)=O)C2)C(=O)CC(C)(C)C1=O C1(C(N(C2CCCN(C(=O)CSc3n[nH]c(O)n3)C2)CC)=O)COCCOC1 C=CCC(C)(C)C(=O)N1CCC(C(F)C(=O)N(C)C(C)C)C1 C(=O)(C(O)C(C(C)C)OC)NCC(CC)(C)NC(C1CC(C(C)=O)C1(C)C)=O N1(C(Cc2nnc(C)n2C)=O)CCC2(NC(C3CCC(=O)N(C)C3)=O)CCCC12 Cn1cc2c(C(=O)NCC3CCC3NC(c3ccc(C#N)o3)=O)cccc2n1 C1(CNC(CSCc2nc(C)sc2)=O)CC(C)(C)CN1C(C1COCCO1)=O N1(C(c2nc(Br)cs2)C(=O)NCC)CCc2cccc(Cl)c2C1 n1(CC(=O)NCC(CCNC(=O)C(C)C(C)O)OC)cc(C)c(O)nc1=O c1(C(N2C(CNC(C3CCC(=O)C3)=O)CCCC2)=O)cc2sccc2cn1 c1(C(N(C)CCOCCNC(=O)CC2(C)CC2)=O)nncc2c1CCCC2 C1(C(=O)NC(CCCNC(C(CCC)OC)=O)C)CCc2cncn2C1 C12CCCC1C(=O)NC2.C(C(F)(F)CC1CC1)NC(=O)CSC(F)F c1(C(N2C(C(N(C3C(C)CC3)C)=O)CCC2)=O)cc(O)cc(=O)o1 N1(C(=O)NC2CN(C(C)=O)C2)CCc2ccsc2C1C c1(NC(C2C(CNC(=O)CC3CC3)CCC2)=O)ccc(O)cc1C(=O)O CCN=C(NCc1ccc(Cl)c(Cl)c1)N1CCCC(Cn2ccnn2)C1 N1(C(CCn2c(C(C)C)ncc2)=O)CCCC(C)C1CNC(=O)COCCCF C1(C(=O)NC(C2CCN(C(c3ccc(C(N)=O)s3)=O)C2)C)CC(=O)N(C2CC2)C1 c1(C(N2CCN(S(Cc3ccc(C#N)cc3)(=O)=O)CC2)=O)ccc2nsnc2c1 C1(NC(C2(OC)CC2)=O)CC2CCC1C(NC(=O)CC1=CCOCC1)C2 CC(C)C(O)CNC(=O)C(=O)N(CCc1ccccc1)Cc1cccs1 C(=O)(CC(C(F)F)C(C)(C)C)NC1(c2ccc(-n3c(C)ncc3)nc2)CC1 N1(C(c2c(C)nc(C)[nH]2)=O)CCC2CCC12CNC(=O)CNC(c1ccco1)=O N=c1nc2ccc(C(=O)NC3CCN(C(c4cncc5nc[nH]c45)=O)C3)cn2[nH]1 CCC(C)(CO)C(=O)NC(C)CCNC(c1ccc(Cl)cc1N)=O c1(CS(=O)(=O)N(C)C)ccc(OC2CCN(Cc3ccccc3)C2)cn1 C1(C)(CNC(C(C)c2cncs2)=O)CCCN1C(=O)COc1cccc(F)c1 c1(N)nc2ccccc2s1.C12COCCN1C(=O)COC2.C(CC)(C(=O)NC)=CC Cc1ccc(C(N2CCC(C(C)(C)C(=O)NC(c3nnc(C)o3)C)C2)=O)nn1 c1(C(=O)OC)c(C)ccnc1NC(C)CN(C(=O)CCCc1nc(C)no1)C C(=O)(C#CC1(C)CCCO1)NC1CC2N(C(C3CCC(OC)CC3)=O)C(CC2)C1 c1ccc(C#N)c(I)c1.c1(NC(N(C)C)=O)cccc(NC(C2CC2C)=O)c1 C(=O)(CCCCNC(C1(C)CCC1)=O)NCC1C(N(C)C)COC1 C(C(=O)N1CC(CC(=O)Nn2cc(CO)nn2)(OC)C1)(C(C)C)SCC C(C)(N=c1[nH]c(=NCCCn2cccn2)[nH]c2c1COC2)c1cn(CCOC)nc1 C1(CSCC)CN(C(c2cn(C(C)C)nn2)=O)C(C)(C)C1.C12(CC1)C(=O)N2 n1(C(C)C)ncnc1C(N1CC(F)(CNC(=O)Cc2cnsc2)C1)=O CN(OCC(F)(F)F)C(=O)OCCC(c1nc(C(C)(C)C)cs1)C(=O)O c1(SCCCNC(=O)CCN2C(=O)CCNC2=S)cnc2ccc(F)cc2c1 c1(C(N2CCC3OCCC3C2)C(=O)NC(C(=O)OC)C)ccc(Cl)c(F)c1F c1(OC)cc(C(=O)NC2CCCC2CNC(=O)CC2CCC(C3CC3)O2)ncn1 Cc1cc2[nH]c(C(N3CCC(NC(C4CCC(C)(C)OC4)=O)C(O)C3)=O)cc2o1 CN=c1ccc(C(=O)NC2CC3CCC2N3C(=O)Cc2ccc(Cl)cn2)c[nH]1 C(=O)(C(C)CC(N)=O)N(C1CCN(C(=O)C(C)NC(C)(C)CC)C1)CC c1(C(C)C)ccc2c(C(=O)NCC(CO)C(N3CCC4(CC3)CC4)=O)ncn2c1 c1(C(N2CCC(N3CCC(O)C3)C2)C(=O)NCCC2(C)CC2)cc(F)ccc1F c1(OC)ccc(CN(c2ccc(C3SCCS3)cc2)C(C2CCCCC2)=O)cc1F CC1=C(C(=O)N2CC(NC(C3(C)CCCNC3=O)=O)CC(F)C2)CCCC1 S(=O)(=O)(c1c[nH]c(=NCC2CC(F)C2)cc1C)N(C(C)CO)CC N1(C(C(CNC(=O)CCc2ccoc2)N(C)C)=O)CCOCC1CO c1(NC(C)=O)ccc(Cl)cc1C(=O)NC1CCC(NC(c2occc2Br)=O)CC1 C=CC(C)(O)C(=O)NCCN(C(=O)CCCNC(c1cccs1)=O)CC1CC1 c1(C(=O)OC)ccc(OC)c(NC(C2CC(NC(c3cc(F)ccn3)=O)C2)=O)c1 CC(CNC(c1[nH]nnc1C1CC1)=O)C(=O)NCCc1cc[nH]n1 N1(C(Cc2cnc(C)[nH]2)=O)CC2CCN(C(c3cnc(C4CC4)[nH]3)=O)CC2C1 CN1CCC(C)(C(=O)N(CCCNC(C2CCO2)=O)Cc2ccccc2)CC1 n1(CC)cc([N+](=O)[O-])c(C(=O)N(C(C)CN(C(=O)CC2CN(C)CC2O)C)C)n1 N1(C(c2conc2C2CCNCC2)=O)CCCC(NC(=O)C(F)(F)F)C1 c1(C(=O)NCC(C)N(C(=O)COCC2CCCO2)C)cc[nH]c1C1CC1 C1(NC(c2c(C(=O)OCC)con2)=O)CCN(C(=O)C(=O)C(C)C)CC1O CC1CCN(C(=O)CCn2ccccc2=O)CC1NC(=O)CC(F)(F)F N1(C(CC2CC(=C)C2)=O)C2CC=C(C(=O)NCC(CO)C(F)(F)F)C1CC2 Cc1cc([N+](=O)[O-])ccc1C(=O)CCC(=O)N(CC(C)NC(C1C=C1C)=O)C CC1CN(C(c2c(Br)cnn2C(C)C)=O)CC1C(F)(F)F CC1CCCn2cc(C(=O)NC3(CNC(=O)CCS(N)(=O)=O)CCC3)nc21 C1(C(=O)NCC(Cn2cc(C(C)(C)OC(C)=O)nn2)F)CC(CN)C12CCC2 C1(CNC(c2cc(C)ncc2)=O)CN(C(C2C3CNC(=O)C23)=O)CC(C)(C)O1 S(=O)(=O)(c1ccc(Br)c(F)c1)N1CC2CCN(C(c3c(OCC)ccs3)=O)C2C1 Cc1cc(=NCCC(C)(C)C)[nH]cc1S(=O)(=O)N1CCC(OC(F)F)CC1 C1(C(=O)NC(CN(C(COC)=O)CCCCC(=O)OC(C)(C)C)=O)CC12CC2 c1(C(N2C(C)CC(NC(=O)Cc3cscn3)C2)=O)ccc(O)c(Cl)c1 CC(CC(C)(C)C)C(=O)N1CCCC(C(=O)NCCCCCC2CC2)C1C Cc1nc2n(n1)CC(N=c1cc[nH]c(=NCCN3C(C)CCCC3C)[nH]1)CC2 c1(C(C(=O)NCc2cccs2)N(C)Cc2cnc[nH]2)cnc(-c2ccccc2)s1 N1(C(c2ocnc2C2CC2)=O)CC(C2CCCN(C(c3cnns3)=O)C2)C1 C(CC(=O)NC1CC(CNC(=O)C(N2CCCC2)C2CC2)C1)N(C)CCO Cc1ccc(C=CC(=O)NC2CCC2CNC(=O)Cc2cccnc2C)o1 C1(C(=O)NCCC(CNC(CN(C)C(c2cccs2)=O)=O)O)CC2(CCCC2)CO1 C1(NC(c2c(CC)non2)=O)CCCN(C(=O)C(C)c2cc[nH]n2)C1CC c1(NC(C(c2cccc(OC)c2)C)=O)cnc(Cl)nc1C C(=O)(C(C)(C)C)NCCCCCNC(C1(NS(CC)(=O)=O)CC1)=O N1(C(C(=O)NC2CCC(c3ccccc3F)C2)=O)CCCC2(COCCN2)C1 Cc1cc(C(N2CCCCC2C2(NC(C3CCCC3F)=O)CC2)=O)nc(C)c1 CCCCC(CC)CCC(=O)N1CCC(C)(NC(C2(OC)CC2)=O)C1 C1(C(=O)NC2(CNC(CN(C3CCCC3O)C)=O)CCCC2)CCCC(C)(C)C1 N1(C(Cn2c(C)nnn2)=O)CCN(CC(N)=O)C(=O)C1.C1(N)CCN(C)CC1 CCC(CC)(C(=O)N(CCCCNC(=O)CN1CCOCC1)C(C)C)OC c1(CC)ccc(NC(c2ccco2)COc2ccc(C(F)(F)F)cn2)nc1.SCC C1(C(N2CC(CNC(C3C4CCC3CC4)=O)OCC2)=O)CCC(C2CCC2)CC1 c1(C(=O)NCC(CNC(C2(C)CC(C)C2)=O)F)ccc2c(c1)C(=O)CCO2 C1(OC(C(C)C)C)CCCCN1C(C1CC2CC2N1C(=O)OC(C)(C)C)=O c1(CC(=O)NC(CC(C)NC(c2cnc(CC)s2)=O)C)ccc(C(F)F)cc1 c1(C(N(CCCCN(C(=O)CCOC2CCCOC2)C)C)=O)cccnc1O c1(C(=O)NCCCC(C)NC(CCc2onc(C(C)OC)n2)=O)ncccc1Cl N1(C(CCC=CC)=O)CCC2(CCC(CNC(=O)CC3CCCN(C)C3)O2)CC1 C1(C(=O)NC(CC)CNC(=O)CCc2ccnn2C)CCC(N=[N+]=[N-])CC1 Cc1cc(NC(=O)CCc2ccc(C)s2)ccc1NC(=O)CN1CCOC(C)C1 n1(CC(=O)NC2CN(C(C(C)O)=O)CC(C)(C)C2)c(S)nc2ccccc2c1=O N1(C(C(COC)OC)=O)CCC(CNC(c2cccc(=O)n2O)=O)C1(C)C c1(CCC)ccccc1C(=O)NC1CCC(N(C(=O)CC2CC=CC2)C)CC1 c1(NC(C2C(C(N(CC(CC)O)C)=O)C2(C)C)=O)cccc(C2CC2)n1 C1(CCNC(C2CC2(Cl)Cl)=O)CN(C(c2cccc(=O)o2)=O)CCS1(=O)=O C12(CNC(CCC=CC)=O)CCC1CCN2C(c1cccc(Br)c1N)=O C(C(=O)N1CCC(CNC(=O)CC2CCCSC2)C1)(C(C)(C)C)OC C1(C(N2CCC(NC(=O)CC34CCCN3CCC4)C2)=O)CCc2ccccc2O1 c1(NC(c2ccn(C)c2)C)ncc2n1CCC2 N(C1CSCc2ccccc21)c1cc(NC(CSC)C)nc(C(F)(F)F)n1 C(=O)(C(C(C)(C)C)NC(C1COCC(C)O1)=O)NC(C1CCOC1)C#C N1(C(c2ccc(C(C)(C)C)s2)=O)CC2(C1)CN(C(=O)C(F)n1ccnc1)CCO2 N1(C(c2noc(C3CC3)n2)C(=O)NC(C)C)CCCC1C#N c1(CCCC)ccccc1COC(c1cnc(-c2cnccn2)s1)=O C(C(CNC(c1nn(C)cc1SC)=O)C(F)(F)F)NC(C(C)NC(=O)OCC)=O C1(C(=O)NC(CCCNC(C=CCC)=O)C)CCC(N=c2cncc[nH]2)CC1 O(C=CC(=O)NC1(CNC(=O)C(C)CC)CC1)CC.OCC C(C(C(=O)N1CCC2(CC2)C1)C(C)C)NC(COCCOCC)=O.C(=O)(C1CC1)N Cc1ccc(C(N2CC(O)(C(C)(C)NC(C3CCCOC3)=O)C2)=O)c(F)c1 C1(C(N(C2(CC(=O)NC(C)C)CC2)CCOC)C)CCCO1 c1(C(=O)NCCC(C)NC(c2cn(C)nc2Cl)=O)ccc(P(C)(C)=O)o1 C(=O)(C(C(C)C)N1CCCC1=O)NC1CC(CCNC(CC=C=C)=O)C1 C1(CNC(C=C(C)Cl)=O)CN(C(c2cc(CO)c(C)o2)=O)CC(C)(C)C1 N12CCC(CC1(C)C)NC(=O)NC(C(C)OC)C2.C(C)(C)(C)NC(=O)OC C1(C(N2C(C)C(O)CCC2)=O)C2CCCC1CN(C(c1cc(F)ccc1Br)=O)C2 c1(NC)cnc(C(=O)NCC2CCN(C(C3CCC(OC)C3)=O)CC2)cn1 Cc1ccc(COCC(=O)NC(C)C(C)NC(=O)CC2(C)CC2)cc1 C1(NC(CCn2ccc(C)n2)=O)CCC(C)N(C(=O)COc2cccc(F)c2)C1 N(C1c2ccccc2CC1NC(=O)C(C)N1CCC1)C(C=CC)=O C1(C(=O)NCCCC#C)CN(C(c2nn(C)cc2Br)=O)CC1c1ccsc1 c1(NCC(=O)N(C)C)cccc(C(c2nnnn2C)Sc2ccncc2)c1 c1(C(=O)NCCn2cc(CNC(CC(C=C)C)=O)nn2)cc(Cl)cc2c1OCC2 N1(CC(=O)NCc2scc(C(N)=O)n2)CCCC2(CCCCN2)C1 C1(C(=O)NC2CC(CC)OCC2)CCN(C(C2(CCF)CCC2)=O)C(C)(C)C1 C1(C(N(C(C)C(=O)OC)CC=C)=O)CCCC(NC(c2ccnn2CCC)=O)C1 Cc1nn(C2CCOC2)cc1C(=O)NCC1(F)CN(C(c2cccc(Cl)c2)=O)C1 c1(NC(=O)NCc2cn(-c3nccc(C)c3)nc2)c(F)cccc1Br C1(NC(c2c(CC)c[nH]c2)=O)CCN(C(C2(C)CS(=O)(=O)C2)=O)CC(C)(C)C1 c1(N(C2CC=C(C(=O)OC)C2)C)ccc(S(=N)(=O)C(F)(F)F)cc1 c1(C(=O)NC2COCCN(C(=O)C(C3CC3)C3CC3)C2)cc2c(Cl)nccc2s1 c1(C(=O)NC2C=CC(CNC(C(C)(C)OC)=O)C2)ccc2[nH]ccc2c1 C(=O)(CCCCCN(C)C(c1c[nH]nc1Cl)=O)N(C1CC(O)C1(C)C)C c1(OC)cncc(C(N2CCN(C(C3CC3C(F)F)=O)CC2C)=O)c1C n1(CC)ncc(Br)c1C(=O)NCCCn1cc(Cn2cncn2)nn1 C1(C(N(C(C(=O)NC(c2ccn(C)n2)C)C)C2CC2)=O)CC2C(C1)C2(F)F C1(C(N2CCCC(C(C)=O)C2)=O)CC2CCN(C(=O)CC3CCCOC3)CC12 C(c1cc(C)no1)=CC(=O)NC(C(N1CCC(C(=O)OCC)C1)=O)C1CCCC1 C12(OC)CCC(NC(C3CCCN(C(C(C)OCC4CC4)=O)C3)=O)(CC1)C2 C1(NC(c2c(C)nc(COC)s2)=O)CCCN(C(=O)COCC2CCOC2)CC1 c1(C(=O)NC(C)CNC(=O)CCC2CC2(F)F)cnc2n1C(C)CCC2 C1(OC)CC(C(=O)NCC=CCNC(=O)Cc2cnc(C)[nH]2)C12CCC2 N1(C(C2(CC#C)CCCO2)=O)CCC(NC(=O)CC(C)(C)C(C)=O)C(C)(C)C1 C(CCCCC(=O)N1CC(NC(=O)CCC(=O)N2CCC(O)CC2)CC1C)SC C(=O)(CCCCCN=[N+]=[N-])NC(C(=O)NCCOCCC#C)(C)C1CCC1 C1(C(=O)NCCC(C)NC(c2ccc[nH]2)=O)CCN(S(=O)(=O)N(C)C)C1 CC(C)C(F)(F)CC(=O)N1CCCC1CNC(=O)C(n1ccc(Br)n1)C C#Cc1ccc(C(=O)NC2CCCC(CC(=O)NCC3(CN=[N+]=[N-])CC3)C2)cn1 c1(OC)ccc(F)c2[nH]c(C(=O)NCC(C3CCC(C)CC3)C)cc12 O=S(=O)(c1ccc(OCC2CCCC(c3ccc(F)cc3)C2)cc1)NC1CC1 N1(C(C2OCCN(CC)C2)=O)CCCC2(NC(=O)CC3(OC)CC3)CCCC12 N1(C(c2cnc(C)n2C(F)F)=O)CCCC2CCC12Cc1ccccc1 C(=O)(C1CCCc2ccccc21)N1C(CNC(CC2(NC(C)=O)CC2)=O)CCC1 CC1(C)C(C(=O)NCc2cccs2)CCN1C(=O)CC1CCSCC1 C(=O)(C(F)(F)C(C)O)N1CCC(CC(=O)NCC(COCC)(C)C)CC1 C1(C(N(CC(C)CNC(c2ccn(C(F)F)n2)=O)C)=O)CC2OC(C)(C)OC2C1 O=S(=O)(c1cnc(N2CCCc3ccccc3C2)c(Cl)c1)NC1CCCC1O c1(C(=O)NC(CNC(C(C)NC(C)=O)=O)C(C)C)cc(Cl)ccc1C(C)C C1(CC=C)(NC(=O)CC2CCCCC2O)CCN(C(=O)CNC(=O)CC(C)C)C1 C(CCCCC(=O)N1CC2CC2(NC(C2CCN(C3CC3)C2=O)=O)C1)N(C)C c1(CN(CC2CCN(C(c3c(CC)noc3)=O)C2)CC2CC2)ccccc1C N1(C(C2CCN(C(c3cccc(CC#N)c3)=O)C2)=O)CCC2OCCC2C1 c1(C(=O)NCC(C2CCCC2)NC(C2(CC=C)CC2)=O)c[nH]c2nc(F)ccc12 C1(CNCCC(C)C)(C)CCCC1.C1(SC)CCC1C(=O)N(CCC#N)C1CC1 c1(NCc2ccc(CC)s2)[nH]c(=NC(C)CC2CCCO2)nc2c1cnn2C(C)C C12(C(N3CCCC(NC(C(C)C4=CCCC4)=O)CC3)=O)CCCN1S(=O)(=O)CC2 c1(C(N2CCCN(C(c3nccc(CC)c3)=O)CC2)=O)cccc2c1OCC2 Cc1ncc2n1CCN(C(c1cc(-c3ccccc3Cl)nn1C)=O)C2 N1(C(CCc2ncc(C)[nH]2)=O)CCN(C(=O)Cc2cccc(C(C)C)c2)C2CC12 Cc1nc(C(=O)NC2(CNC(=O)CC3(C)CC3(F)Cl)CCCCC2)c(C)o1 C1(CN(C(C2(CC=C)CCCC2)=O)C)COCCN1C(c1csc(C(F)F)c1)=O c1(C(N2CCC(N(CCC)C(c3ccc(CO)o3)=O)C2)=O)ccc(CC)c(F)c1 c1(C(C(=O)NC2CCC2)N(C(C)Cc2cnn(C)c2)C)ccnc(F)c1 c1(-n2cc(CN(CCCCCN=[N+]=[N-])CC=C)nn2)ccc(Cl)cc1F c1(C2CC2SC)nc2ccccc2s1.C1(C2C(=O)N2CC2CCCO2)CCC(C)C1 C(=O)(CC(C)(C)C)NCC(CC)(C)NC(c1cccn1Cc1cccnc1)=O C1(C(N2CCC(NC(c3c(C)ccs3)=O)(CF)C2)=O)CCCCN(C)C1=O C1(CNC(c2ncn(CC)n2)=O)CC2(CCC2)CN1C(C1(C#N)CCC1)=O c1(CC(N2C(CNC(c3c(Cl)nc(NC)s3)=O)CC2)=O)nn(C)c2ccccc12 c1(OC)ccc(NC(=O)NCc2c(C(=O)O)cccc2F)c(Cl)n1 c1(C(CNC(C(COC)(C)C)=O)NC(C2CCCN(C)C2)=O)cc(F)cc(Cl)c1 c1(C(=O)OCC)sc(CC(C)C)nc1C.c12cccc(c1)C(=O)NC(=O)NC2 C=CCC(CC(=O)N1CCC(C)C1CC)NC(C1CN(C2COC2)C1)=O C#CCC(C)(CNC(C1CC(C)CN1C(=O)CCCCN(C)C)=O)CO c1(C(N(C2CC(NC(c3scc(C)c3)=O)C2)C)=O)ccc(F)cc1OC(F)F CCC(C)(CNC(=O)C(C1CC1)OCC)NC(c1cc(C(C)(F)F)on1)=O C1(C(N(CC(C)NC(c2c(C)nc(N(C)C)s2)=O)C)=O)CCCC(C)(C)CC1 C1(NC(CNC=O)=O)CCN(C(C2(F)CCCC2)=O)CC1F C1(F)(CNC(C2C3CCCC23)=O)CCN(C(=O)CC2COCCO2)CC1 N1(C(C(CCC)NC(C)=O)=O)CC2CCCC2(C(=O)NCC(C)(C)C(C)C)C1 c1(C(N2C3C(C(=O)Nc4cncc(SCC)n4)C(C3)C2)=O)c(C)ccc(Br)c1F N1(CC(C)C)CC(C(=O)NC(CNC(c2ccsn2)=O)CO)CC1=O c1(C(=O)NCCCCCNC(c2n(C)ccc2)=O)c(Cl)csc1Cl c1(C(=O)NC)ccc(C(c2nnnn2C2CCOC2)NCC2CC(F)(F)C2)cc1 c1(CNC(C(C2CCC2)OCC)=O)ccc(F)nc1C.C1C(C)(C)C(=O)N1 CCC(C)(CCNC(c1nccn1C)=O)NC(c1cnn(C(C)C)c1)=O C(=O)(C#CC(C)(C)CNC(=O)C(C(C)OC)N(C)C)N(CCC)CCO Cn1ccc(C(=O)NCC2(C(F)F)CCN(C(=O)CC3(C)CC3)C2)cc1=O C1(C(N2C(C(N(C(C(=O)OC)C)C)=O)CC2C)=O)C2CCC(F)C12 CCC(CC)C(C(=O)NCC1(O)CC(C(=O)NCCC(O)CCO)C1)OC C(C(=O)NCc1cc(C)ns1)(C(C)OC)NC(C1C(=C)C1)=O N1(C(CC(CNC(C(CNC(C)=O)(C)C)=O)C)=O)CCC(F)(C#N)C1 C1(C(=O)NCCCCCCNC(Cc2cc(OC)no2)=O)CCCCNC1=O Cc1ccc(C(C)CC(=O)NC2(CNC(=O)Cc3cnsc3)CCOC2)cc1 C1(N=c2[nH]ccn3nnnc23)(CNC(C2(C)CC2(Cl)Cl)=O)CCOCC1 c1(CC)cc(C(=O)NC2CCCN(C(C3CC3c3ccc(F)cc3)=O)C2)sc1C c1(NC(=O)OC(CCC)C)ccc(C(=O)NCCNC(=O)COCCOC)s1 c1(C(=O)OC)ccc(C(c2c(CC)cccc2)=O)c(F)c1 C(CN=c1[nH]c(=NCC2CSC2)[nH]c2c1CCC2)n1c(CC)ncc1 C1(C(N2CCOC(c3nc[nH]n3)C2)=O)CCOC12CCS(=O)(=O)CC2 C#Cc1ccc(C(N2CCN(CC(=O)NC3(C(N)=O)CCOC3)CC2)=O)c(C)c1 N1(C(c2n(CC)ccc2)=O)C2CCC1C1CC1(NC(=O)C(Br)=C(C)C)C2 C1(C)(CSC)CCN(C(C2(N3CCCCC3)CCCCC2)=O)C1 c1(N2CCC(CCC(C)O)CC2)ncnc2c1ncn2CCC1CCCCCC1 N1(C(CCNC(COC)=O)=O)CCCC1C1(NC(=O)COCC(C)C)CC1 CCCCCCC(=O)Nc1ccc(NC(c2cc3n(n2)CCC3)=O)cn1 CC(C)C(C(=O)NCC1CCN(C(C2(C(C)C)CC2)=O)C1)n1cnnc1 C(=O)(C1=CC2CCC=CCCC12)NCc1ccc(NC(C2CCCC2)=O)nc1 C1(C(N2CCc3ncccc3C2)=O)COC2(CCN(C(C3CC3F)=O)CC2)C1 N1(CC(OCC(C(=O)NCC(CC)(C)N2CCOCC2)COC)=O)CCCCS1(=O)=O C1(CNC(=O)OC(C)(C)C)CCCN(C(C2CC(OC)C2)=O)C1.CCCC1CCC1 c1(NC(C2N(Cc3scc(C)c3)CCOC2)=O)nc2ccc(I)cc2o1 C1(NC(CN(CCC)C)=O)CCCC(NC(c2ccc(=O)n(C(C)C)c2)=O)CC1 C1(CNC(Cc2c(C#C)cccc2)=O)CCCC2(CN(C(=O)C(CC)OC)C2)O1 CCCC(CC)NC(=O)C(C)CN(C(=O)CSC(F)(F)F)C1CC1 CC1C2CCC(C2)C1C(=O)NCC12CCC(C(=O)O)(CO1)C2.C12(OCC3CC3)CCC(C1)C2 C1(NC(C2(C)C(C)(C)C2)=O)CCC(C(=O)NCc2ccccn2)CC1 CCC(C)C(C(=O)NC1CC(=O)N(CCOC)C1)N(C)C(C1CC(=O)C1(C)C)=O C=CC(C)CC(=O)NCCC(C)CCNC(=O)CCS(C)=O c1(C(c2nnnn2-c2ccccc2C)NC2CC(=C)C2)cc(Cl)cc(Cl)c1 S(=O)(=O)(c1ccc(=O)n(C(C)Cc2ccc(C(F)(F)F)nc2)c1)NCC(=O)OC N1(C(c2cc(OC)ns2)=O)CC(NC(C2(F)CC2)=O)CC2(CCC2)C1 C1(NC(C2CC(C)C2)=O)CC2(C1)CC(NC(=O)C=Cc1ccc(O)cc1)C2 C=CCC(C)(CC)C(=O)NCC1CC(C(=O)NCC(C)C(=O)NC)=NO1 C(=O)(C(C(C)CC)N(C(=O)CCN(C)C)C)N(CCC#C)CC C1(CNC(c2ncn(CC)c2)=O)CCCCN(C(c2cn(C)nc2C2CC2)=O)C1 C1(NC(C2(CC)CN(C(C(CC=C)C)=O)C2)=O)CCc2nn[nH]c2C1 c1(CC(=O)NCC2(CNC(C(CCC)OC)=O)CCC2)ccc(Br)c(F)c1 C1(C(=O)NCC2CN(C(CCOC)=O)C2)CCCN(C(C)C)C1 N1(C(C(c2cnn(C)c2)OC)=O)CCC(CCNC(=O)CC2COC(=O)N2)CC1 c1(C(N(C(C)CNC(c2cc(C)nc(O)n2)=O)CC)=O)cnn(C)c1S(N)(=O)=O c1(C(=O)NCCN(CCC)C(c2n[nH]c(C3CC3)c2Cl)=O)cnn(C2CC2)c1C C=C=CCC(=O)N(CCCN(CCO)C(C1CC1c1ccccn1)=O)CC N1(C(C)=O)CCCC2C1CCN2C(C1CCc2nc(O)[nH]c2C1)=O.c1c[nH]c(=N)s1 CCC(C)CCCC(=O)NC1(COC)CCN(C(c2cc(F)c(C)cc2Cl)=O)C1 C(C)(N=c1[nH]c2c(c(=NC3CC(CCF)C3)[nH]1)SCC2)c1ccc(C)s1 c1(CCC(=O)NC2CC(O)(CNC(=O)C=CC(=O)NC3CC3)C2)cccc(Cl)c1 c1(C(=O)OC(c2cc(C)nn2C)C)ccc(F)c(CC#N)c1 c1(C(C(=O)NC2C(CNC(CC=CC=C)=O)C2)(C)C)ccc(CC)cc1 CCCS(=O)(=O)CC(=O)N(C(c1ccc(Br)cc1)(C)CO)C c1(COC)nc(NC(C)Cc2ccc(F)cc2)cc(=NC(COC)C2CC2)[nH]1 c1(C(N(CC)Cc2nccs2)=O)ccc(Br)c2ncccc12 c1(CC(=O)NC(CC)CNC(=O)COc2cn[nH]c2)ccc(Br)c(F)c1 S(=O)(=O)(c1cc2c(cc1Br)COC2)N(C(CN(C)C)(C)C)C C(=O)(C1=NOC2COCC12)NCCn1cc(C(=O)NCc2c(C)nn(C)c2)nn1 CS(=O)(=O)C1(C(=O)NCC2CCCCN2C(=O)CNC(C2CCC2)=O)CCC1 N1(CCC(N2CC(NC(CCC)=O)C2)=O)CCOCC1.C(=O)OC c1cc(O)ncc1F.N1(C(CCOC)=O)CCC(CNC(C2C(C)C2)=O)C1(C)C C1(NC(C(C2CCN(C(C3(Cl)CC3)=O)CC2)C)=O)CC(=O)N(C)C1 Cc1oc(Cl)nc1C(=O)NCCC(C)CCNC(=O)CC(=O)NC1CC1 c1(C(=O)NC2CCC(NC(c3nc(Br)cs3)=O)C2)c(F)cc(Cl)cc1F N1(C(CN(C(=O)C2CC2)CC)=O)CCCC(C(=O)NCC(C)O)C1 N1(C(CN2CCN(C)CC2)=O)CCC(CO)C(NC(C2CCOC(=O)N2)=O)C1 N1(C(C(C)N(C(C2CC(=O)C2)=O)CC)=O)CCSc2ncccc21 CC1(C)CC(CNC(C2CNC(=O)N2)=O)CN1C(=O)CNC(c1ccsc1)=O c1(C(N2CCCC(N(C(=O)CN3CC4CC4C3)C)C2)=O)ccc2snnc2c1 c1(C(N(CC(C)NC(=O)C(C)(C)CCSC)CC)=O)ccc2c(c1)N(C)CC2 C12(C(N(CC(C)N(C(c3cnc(CC)[nH]3)=O)C)C)=O)CCC(CC)(C1)OC2 CC(C)C(C(=O)N1CCC(C(=O)NOCc2ccccc2F)CC1)N(C)C c1(N2C(CNC(C(C)OC)=O)CC(F)C2)ncnn2c(Br)ccc12 N1(C(C2(C)CC(C)C2)=O)CCCC(n2cc(-c3ncccn3)nn2)C1 N1(C(CCC(C)=O)=O)CCN(C)CC1CNC(c1cc(C(C)(C)C)c[nH]1)=O CC1=NC(C)(CNC(C2(C3CCCN3C(=O)COCC(F)F)CC2)=O)CS1 c1(N2CCC(C)(CC)CC2)nc(=NCCc2nccn2C(C)C)[nH]c2c1SCC2 c1(NC)ccc(C(=O)NCCC(O)CNC(C2CCC2(F)F)=O)cc1F C1(CNC(c2csc(-c3cnc[nH]3)n2)=O)CN(c2cnc(F)cn2)CCCO1 c1(C(C(=O)O)NC(=O)CCC2CCCOC2)cccc2c1OCO2 C(C(C(=O)N1CC(SC(F)F)C1)C(C)(C)C)NC(CC(C)C1CCCO1)=O C1(C(=O)NC(C(=O)N(C)CC2CCC2)CC2CCC2)CC(F)C(=O)N1 C(C(C)(C)C)OCC(=O)N(C(CNC(COCCOC)=O)C)N(C)CCO C1(CNC(C(CCSC)NC(c2ccco2)=O)=O)CC2CCC(C1)C2 c1(C(=O)NC2CCCCN(C(C(C)CC(F)F)=O)C2)cc2cnccc2o1 N1(C(C(CC=CC)NC(C2CCCCC2F)=O)=O)CCC2(CC(CO)C2)C1 C1(C(N2CC(CCNC(c3c(C#C)cn(C)n3)=O)C2)=O)CCc2cnc(C)n2C1 c1(NC)cc(OC)ccc1N.c1(C(C)O)cncc(N(CC)Cc2ccncc2)n1 C12(CNC(C3CCCCCCC3)=O)CCCC1CN(C(=O)C(F)CC1CCC1)C2 CCC(C)CCCCC(=O)NCC1N(C(c2cccc(N)c2)=O)CCCC1(C)C C1(NC(c2ncccc2C2CC2)=O)CCN(C(=O)CC2CCCCC2)C1C1CC1 N1(C(Cc2n(C)cnc2)=O)CC2CCC(CNC(C3CC(=C4CCC4)C3)=O)C2C1 c1(C(N2CC(C)C(N(C(=O)C=CC3CCCC3)C)CC2)=O)cccc2c1CCN2 c1(C(=O)NC2CCCCCN(C(C3(CC#C)CC3)=O)C2)nc(C)n2c1CCCC2 N1(C(CC(=C)C)=O)CCC2(CCCN(C(=O)CCOCC(C)C)C2)C1 N(C1C(=O)Nc2cc(Br)ccc21)C(=O)NOC1CCOC1 N1(C(C2COCCN(C(c3cnn(C)n3)=O)C2)=O)CCC(O)CC12CC2 CCC(CC(=O)NC(C1CCCCC1)CNC(=O)C=CBr)CC(F)(F)F CC(C)C(F)C(=O)N(C(C)(C(=O)NC(C1(O)CCC1)C)C1CC1)C c1(C(C(=O)NCCC(=C)CNC(=O)CCC2CC2(F)F)O)cccc(F)c1 N12CC3CN(C3C1)C2=O.c1(OCOC)ccccc1CC(=O)Nc1ccc(C#N)s1 C1(CNC(=O)NC2(CO)CC(OC)C2)CCC2COCCC2O1 C(=O)(CCCCC(=O)N1CCC(O)(CC(N2CCN(CCF)CC2)=O)C1)OC C1(C2CC2)(C(N(CC)Cc2ccncc2)=O)CN(C(c2cc(C(F)F)[nH]n2)=O)C1 c1(C(N2CCC3(CN(C(=O)CC4CSCCS4)C3)C2)=O)cc2n(n1)CCCC2O c1(OC(C)C(=O)N(CCCNC(=O)C(C)c2cc[nH]n2)C)ccccc1F CC(CCCCC#N)(c1nnnn1C1CC1)NC(=O)NCC1CCCC(C)(C)O1 c1(OCC)cc(C(=O)NC(C)CN(C)C(c2ccc(SC)o2)=O)ccc1C c1(C(=O)NCCN(C)C(C2CC=CCC2)=O)c[nH]nc1OCC(F)(F)F N1(C(COC(C2C(c3n(CC)ncc3)N(C)C(=O)C2)=O)=O)CCC(C)CC1CC CCC(C)CCCC(=O)N1CCC(C(O)CN(C(=O)C(O)C(F)(F)F)CC)CC1 N1(c2snc(COC)n2)CCC(C(C)NC(=O)CNC(c2ccncc2)=O)CC1 c1(NC(C2C(NC(c3ccc(SCC)cc3)=O)C2)=O)nc2cc(F)ccn2n1 C(=O)(CCC(CF)CF)N1CC(N(C(Cc2ccc(C)c(C)c2)=O)C)C(F)C1 N#CC1=C(C(=O)N2CCCCCC2C(N2CCC3CCCC3C2)=O)CCC1 N1(C(CC2N(C(C)=O)CSC2)=O)CCC(C)(NC(=O)CC=Cc2ccccc2)C1 CC(C)C(O)C(C)C(=O)N1CCC(O)(CNC(c2ccc(O)nc2Cl)=O)C1 C=C1CCN(C(=O)CN(C)C(=O)C2CC2)C(C(=O)NCCCC2CCC2)C1 C1(C(N2C(CNC(C3C(CC)C3)=O)CC(F)C2)=O)CC(=O)NC(=O)C1 C1(C(N2CC(C)(NC(c3cc(C(C)C)on3)=O)C2)=O)CCc2nnnn2C1 c1(CN2CC(O)C(F)C2)ccc(O)c(CN2C(C)(CC)CCC2)c1 CCC(C(C)(C)C(=O)NOCC(C)CC)NC(c1coc(N(C)C)n1)=O N1(C(c2cnc(OC)nc2)=O)CCC2CCN(C(=O)C=Cc3ccccc3)C2C1 N1(C(c2c(C)onc2Cl)=O)CC(CNC(C2(CO)CCCO2)=O)C(C)(C)C1 C1(CC(=O)NCCC2(CNC(=O)COC3CC(F)(F)C3)CC2)CCC2(CC2)CO1 N1(C(c2cnc(O)n(C)c2=O)=O)CCCC2(NC(=O)CC(O)C3CC3)CCCC12 c1(C(C)C)c(C(=O)NC(C2(O)CN(C(=O)CC(F)(F)F)C2)C)cnc2ncnn12 Cc1cc(=NC(C)C(C)C)[nH]c(N2CCC(N3C4CCCC3CN(C)C4)C2)n1 CCCCCCCC(=O)NC1CCOCC1NC(c1c(SC)nc(O)nc1C)=O n1(C(C(=O)NC(C2N(C(COCCOC)=O)CCC2)C)CC)cnc(C#N)n1 c1(NC)cnc(C(=O)NCC(C)(C)OCC(=O)NCC(C2CCCCC2)C)cn1 CCCC(C(=O)NC1CCC(N(C(=O)C#CC2CC2)C)CC1)N(C)C c1(C(CCCC)=O)ccc(NC(=O)Cc2ocnc2C)o1 Cc1cc(C(=O)NCCC2(NC(C3CS(=O)C3)=O)CCC2)no1 c1(C(N(C)CCNC(c2cc(F)c(F)cc2O)=O)=O)c[nH]c2cc(F)c(F)cc12 C(=O)(C(C)(CC)CC)N1C(CCCNC(c2c(CC)non2)=O)CCCC1 C(=O)(C1CCc2cccnc21)N(C)CC1(CNC(c2cc3n(n2)CCO3)=O)CC1 c1(NC2CC(NC(c3ccc4nc[nH]c4c3)=O)C2)ncc2c(Br)cccc2n1 C1(CC(C(=O)NC2(c3nc(C)on3)CCCC2)N)CC2(CC2)CO1 C(=O)(C1=CCOCC1)NCC(CNC(C(C(C)C)c1ccccc1)=O)CO c1(C(N2CCOC(C3CCOCC3)C2)C(=O)NCC2CC2)n[nH]c2ccccc12 C1(O)(CNC(=O)NC2CCCCO2)CCCN(Cc2ccc(O)nc2)C1 c1(CC)cscc1C(=O)NCCCNC(=O)C(CC)C1CCOCC1 c1(C(N(C(CNC(CCCN(C(C)C)C)=O)C)C2CC2)=O)ncccc1Br Cc1cccc(C(N2CC3(C2)CN(C(c2cc(O)nn2C)=O)C3)=O)c1N C1(OC(C(C)(C(C)C)OC)=O)CCc2cc(Br)ccc2C1 c1(C(=O)NCCN(C)C(N)=O)ccc(N)cc1.C1(CC(=O)NCS(C)(=O)=O)CCCO1 CC(C)C(C#N)C(=O)N1CCOCC1CC(=O)NCC1SCCS1 N1(C(C)=O)CC2CC(NC(c3cc(Cl)sc3Cl)=O)C1C2 c1(CNC(c2nnnn2CCC)(CSCCC)C)csc(-c2ccco2)n1 c1(-c2nc(C(=O)Nc3cc(OC)c(Cl)cc3)sc2)ccc2sc(C)nc2c1 C1(NC(c2c(CC)scc2)=O)CC2CC(NC(c3cn(C)cn3)=O)C2C1 C=CCC(C)(C)C(=O)NCC1CC1CNC(=O)Cc1cc(C2CC2)on1 c1(C(N2CC(CC)C(NC(=O)C(C)(F)F)CC2)=O)ccc2sccc2c1 N1(C(C2CC(=C)C2)=O)CCC(F)(C(=O)Nc2cc(C)on2)C1 Cc1oc(C2CC2)nc1C(N1CC(O)CC1CNC(=O)CNC=O)=O CCC(C)(CC)C(=O)NCc1cc(O)nc(CNC(=O)Cc2cc(C)no2)n1 c1(CC(=O)NC(C)CNC(c2ccc(C#N)[nH]2)=O)ccc2c[nH]nc2c1 C1(C(N2C(CN(C(C(COC)N(C)C)=O)C)CCCC2)=O)CCC(O)CN1C Cn1cc(C(=O)NCc2ocnc2-c2nn[nH]n2)nc1O c1(C(=O)NC2C(CNC(C(C)CC3CCCC3)=O)C2)cc2cc(Cl)ccc2o1 c1(CNC2CCC(NC(c3c(C)n(C)nc3)=O)C2)ccncc1[N+](=O)[O-] N1(C(C2(C)CCN(C)C2)=O)CCCC(C2CN(C(c3ccnc(Cl)c3F)=O)C2)C1 N1(C(C(C)C2CCC2)=O)CCC(C(=O)NC(CCO)C2CCC2)C1(C)C c1(C(N2C(C)(C(=O)Nc3cccc(F)c3O)CC2)=O)cnc2c(F)cccc2c1 c1(C(=O)OCCN2CCCC2)noc2ncccc12 C1(CNC(CC2CC(SC)C2)=O)(COC)CC12CCC2.c1(C(=O)CN)ccnnc1S C(=O)(C1=NOC(C)C1)NCc1cc(C(N2C(CC)CC(C)C2)=O)on1 Cc1n[nH]c(C)c1CCC(=O)NC1CCN(CCCNC(=O)CNC=O)CC1 CCC(C)CC(C)C(=O)N1CCC2(C1)CN(C(=O)CC1CC(OC)C1)C2 C(C(=O)N1CCCC(O)(CN(C)C(c2n[nH]c3c2CCC3)=O)C1)(C(C)(C)C)OC CC1(C)CCCC(CC(=O)NCC(=C2CN(C(c3cnnc(O)c3)=O)C2)F)O1 N(C(=NCCC1CCS(=O)(=O)CC1)NC1CC1)CC(C)(C)CO C(=O)(C=CS(C)=O)NCC(CNC(c1ncc(Br)cn1)=O)OC C(CCCCCC(=O)NCC1COC(C)(C)C1)NC(c1c(CC)cno1)=O c1(C(=O)NC(CCN(C(C2N(CC)CCOC2)=O)C)C(C)C)cc(O)cc(Cl)c1 C(CCCC(=O)NCC1CC(C(N2CCC2(C)CCO)=O)CO1)N(C)C C1(CC(=O)NCc2cnnn2C2CC2)COCCN1C(c1cc(C2CC2)no1)=O CC1CC2(CCN(C(C3CCCCCC(=O)C3)=O)CC2)CN1C(=O)CC1CC1 c1(CC(C(=O)NCCCC(C)NC(C2(CC)CC2)=O)C)cccc(F)c1 N1(C(c2c(C)c[nH]c2)=O)CC2CCC(CNC(=O)C(O)C3CCCC3)(C2)C1 O=C(CN=c1cc[nH]cc1)NCC1CN(C(c2ccc(F)s2)=O)CC12CC2 C1(C(=O)NCC(NOCC)=O)(NC(=O)CN(C2CCC2)C)CCCCC1 c1(C(C(=O)OCCCOC(=O)NC)O)cccc(Cl)c1 N1(CC2C(CC(N3C4(C(C)(C)C)CCCC43)=O)C2)CCCC2NC(=O)CC12 Cc1nn(C)c(C)c1C(N1CCCCC(NC(c2c(F)cncc2Br)=O)C1)=O C1(OCCNC(C2CC(F)(CO)C2)=O)CCN(C(=O)CCn2ccnc2)C1 C1(N(C)C(C2C3COCC23)=O)CN(C(=O)C2CC2)CC(C)(C)C1 c1(CC)cnc(Cl)nc1N(CCCNC(C1CN2CCC1CC2)=O)C c1(C(=O)NCC2CN(C(=O)C(Cl)=CCl)CC2O)cc(F)cc(F)c1 CS(C)(=O)=NC(=O)C(=O)NC1CCCC1NC(=O)C(O)CCc1ccccc1 C1(NCC2CC(C(F)F)(OC)C2)CC(C23CC(C2)C3)CN1 c1(C(=O)NC2CCCN(c3snc(CC)n3)C2C)csc2c(F)cccc12 N1(C(C(C)OC(C)(C)C)=O)CCC2(CC1)CC(C)N(C(=O)C=CS(C)=O)C2 c1(C(=O)NCC(CN(C(=O)COC(F)F)C)O)cc2c(Br)ccc(F)c2[nH]1 c1(C(=O)NC(C(=O)NC2CN(C(=O)OC)C2)CC2CC2)n[nH]c(C)c1Cl N1(C(C2(C#N)CC23CCCC3)=O)CCCC2(CCCN2C(=O)CCCC(F)F)C1 c1(C(N2CCC(C)C2CNC(c2cc(Cl)ccn2)=O)=O)cccc(Cl)c1N CC1=NN(C)C(=O)C1CC(=O)NC1CC2(C1)CN(C(c1csc(CO)n1)=O)C2 O=C1CC2C(=O)NC1=C(F)C=CC=C2NCCCCNC(=O)C(F)(F)C(F)F c1(C(=O)OC)ccc(C(N2CC(C)(NC(=O)Cc3ccc(C(N)=O)s3)C2)=O)s1 C1(C)(CNC(Cc2c(C)cco2)=O)CCCN1C(=O)CCN(S(C)(=O)=O)C C1(C(N2CC(CN(C)C(c3ccnn3C)=O)C2)=O)CCCC1c1ccccc1 C(CNC(c1[nH]c(C)nc1C)=O)(CC)(CC)NC(C(C)NC(COC)=O)=O N1(C(CSCC(C)C)=O)CCCC(N(C(=O)C(C)(C)C2CCCC2)C)CC1 c1(C(C)C)ccccc1CC(=O)NCC(O)CCNC(=O)C(C)OCC1CC1 C12(C(=O)NCC(CC(=O)N(CC(C)O)C(C)C)O)CCCC1C2(F)F c1(C(=O)NC(C(C)NC(C(CC)CCOC)=O)CO)cccc2c(C#N)c[nH]c12 c1(SCC(C)CO)ccc(NC(=O)NC)cc1.c1(-c2nccs2)ccccc1Cl c1(NC(C2C3CN(C(C4CCC(O)CC4)=O)C2C3)=O)ccc(Cl)cc1[N+](=O)[O-] N1(C(c2cc(CNC(COCCCC)=O)sc2)=O)CC(C)(C)C1C(C)C C1(=O)NNC(=O)c2cn(nn2)C2CCC12.c1(CN(C(C)=O)CC)ccccc1 C1(CNC(C(C)SC)=O)CN(C(=O)CCCSc2ccc(F)cc2)CCC1CO N1(C(c2c(CC)occ2)=O)CCN(C(c2ccc(Br)c(N)n2)=O)CC1CC CC(C)(C(=O)NC1CCCC1CNC(c1cc(Br)co1)=O)c1cccs1 c1(C(=O)NCC(CC=C)NC(C23CC2COC3(C)C)=O)cc([N+](=O)[O-])cn1C C(=O)(CCCCC(C)C)NCC1CCN(C(CC(C)(C)OC)=O)CC1C Cc1nn(C)c(C(=O)NC(CNC(c2cnn[nH]2)=O)CO)c1-c1ccccc1 N1(C(c2c(C)oc(Cl)n2)=O)CCN(C(=O)C(F)CC2CCOCC2)C(C(C)C)C1 c1(C(N(CCC(=O)NCC(O)CC(C)C)C(C)C)=O)ccc2occc2c1 c1(C(=O)NCC(CNC(c2n(CC)cc(Cl)c2)=O)(C)C)cc(F)ccc1N N1(C(C(C)NC=O)=O)C2CCC1CC(CNC(=O)CCCC1CCCC1)C2 c1(C(=O)NC2CCC(CNC(c3c(C)nccc3)=O)C2)cnc2c(c1)CCCC2 N1(C(c2c(N)nccc2)=O)CCCC2(NC(c3cc(Cl)no3)=O)CCCC12 Cc1nn(C)c(F)c1C(=O)NCC(C1CCCCC1)NC(=O)C(F)=CCCF c1(CC(=O)NC(c2ccccc2)CNC(CN(C(N)=O)CCF)=O)cccc(F)c1 c1(CC(C)C)cc(=NC(=O)C(=O)N2CCCC(CNC(N)=O)C2)[nH][nH]1 C1(NC(c2c(F)cc(F)cc2F)=O)CC2CC1CN(C(=O)C(O)C(F)(F)F)C2 c1(C(N(CC(CN(C(=O)CSC(F)F)C)O)C)=O)cnc2ncc(Cl)cn12 C1(CNC(C=CC)=O)CN(C(c2cccc(-n3[nH]nnc3=N)c2)=O)CC12CCC2 C(=O)(CC(C(F)(F)F)c1nccn1C)NCC#CCNC(C(CC(C)C)O)=O N1(C(c2nc(OCC)oc2)=O)CC2(CCC(CNC(=O)C(O)CSC)O2)C1 N1(C(C(=O)NCC2(c3ccccc3)CCOC2)=O)CCCCc2cc(Br)ccc21 N1(C(C(C)OC)=O)C2CCC(C2)C1CC(=O)NCC(F)F CN1CCC(C(=O)NC2CC(NC(C3(c4ccccc4)CC3(F)F)=O)C2)C1=O c1(SCCNC(C2N(C(CCCC=C)=O)CCSC2)=O)cccc2ccccc12 c1(C(N(CCCCNC(c2c(CC)n(C)nc2)=O)C)=O)ccc(OC)nc1F c1(C(N2CCC(CCNC(C(C)C(C)(C)C)=O)CC2)=O)cc(F)c(F)c(C#N)c1 c1(C(N(CCNC(C(C)(CO)OC)=O)C)=O)cc2ccncc2[nH]1 C1(C(=O)NCC(C)NC(=O)C2CC2)CCN(CCO)C(=O)C1 C(=O)(C1Cc2ccccc21)N1Cc2c(ccc(C(=O)N(C3CCCC3)CCO)c2)C1 Cc1n[nH]c2cnc(C(N3CCCN(CCNC(=O)CC(C)F)CC3)=O)cc12 C(=O)(C(CC)(CC)CO)NCC1N(C(c2c(CC)occ2)=O)CC(F)C1 C(=O)(C(C)(C)C(C)C)N1CC(CCNC(c2cc(CC)n(C)n2)=O)OCC1 Cc1ccc([N+](=O)[O-])c(C(=O)NCCCCNC(=O)C(C)N(CC(F)(F)F)C)c1 C(CC1=CCN(C(=O)CC(C)F)CC1)NC(c1cc(C)c(C)nn1)=O c1(C(N2C(CCNC(COC)=O)COCC2)=O)ccc(S(C)(=O)=O)[nH]1 CC(C)CC(C(=O)NCC1CC(F)(CNC(=O)CN2C(=O)CCC2=O)C1)C(C)C N1(C(C(Cn2cccn2)NC(C2N(S(C)(=O)=O)CC2)=O)=O)CC2CC1CC2O C(C(F)(F)C(F)(F)F)OCCC(=O)NCC(C1CC1)NC(C1(C)CC1)=O CC(C)=C=CC(=O)N1CCC(OCCNC(C2CCCC2C)=O)C1 C1(C(=O)NCC2N(C(c3occ(C)c3C)=O)CCCC2)CCS(=O)(=O)C12CCC2 O=[N+]([O-])c1n[nH]c(=NC(CC2CCCC2)CC2CCC2)cc1O C1(CN(C(=O)C=NOC)CC)(CNC(C2CC23CCC3)=O)CCCC1 c1(C(=O)NC2C(CNC(C3CN(C)C3)=O)CC2)cn(C)nc1C1CCOC1 N1(C(c2c(CC)nns2)=O)CC2CCCC2(NC(=O)CCc2csc(C)n2)C1 c1(OC)ccc(Br)cc1C(=O)NC1CCC1CNC(=O)CCC(C)(C)C C1(=CC(=O)NC(C2(O)CCN(C(CS(CC)=O)=O)C2)C)CC2CCC(C1)N2C C(C(=O)NNC(=O)CNC1(NC(C2CCCN2C(C)=O)=O)CCOCC1)=COC CCC(C)(CC)C(=O)N(CCN(C)C(c1c[nH]c(C(N)=O)c1)=O)C(C)C N1(C(COC(CC)C)=O)CCC(CNC(c2sc(C(F)(F)F)nc2C)=O)(OC)C1 C(=O)(C1=C(Cl)CCC1)N(CCN(C(=O)CC(C)Cc1ccc(Cl)cc1)CC)CC c1(CC(=O)NCC(CNC(C(C)Oc2cccnc2)=O)CO)ncn2c1CCC2 NS(=O)(=O)c1ccc(CC(=O)NC23CCN(C(=O)CC4(CO)CC4)CC2C3)s1 N1(CSCC2(C)N(c3ccc(C)cc3)C(=O)CNC2CC)CCSC(C)C1C CC1=C(C(=O)NC2CCCCC2NC(=O)C(=Cc2cn(C)cn2)F)CCO1 CC1OCCC1C1CC1NC(C1Cc2ccccc2C1)=O C1(NC(CSC(C)C)=O)CN(C(c2csc(Cl)c2)=O)CCC1O Cc1cc(F)ncc1-c1cn(C2CCC(C(=O)NC3(C)CC(C(=O)O)C3)C2)nn1 C1(C(C)(C)C)COCCC1NC(=O)CNC(=O)CCC1CC1 C1(C(F)(F)F)(C(=O)NC2CCC(NC(C)=O)CC2)CC2CCC1C2 CCC(CC(=O)N1CCC2(CC(NC(=O)CSc3nccn3C)C2)C1)C(C)C C=CCC(C(=O)N1CCC(N2CCN(C(C3(O)COC3)=O)CC2)C1)NC(C)=O C1(CNC(C=COCC)=O)(NC(c2cnn(C)c2SC)=O)CCCCC1C c1(C(=O)NC2(CN(C(=O)C=CC(=O)N(C)C)C)CC2)cnn(C)n1 O=C(C1=C(Cl)CCC1)NCCC1CCCN1C(=O)C(c1ccc(Br)cc1)O C12=CC(=O)N(CC1)CC2.C1(C(=O)NCC2(C(=O)OCC)CC2)CC(=O)CS1 N1(C(C2C(COC)C2)=O)CC2CC(NC(c3cccc4cc[nH]c34)=O)CC1C2 c1(-c2scc(C(=O)NCC(CN(C(CSCC=C)=O)C)O)n2)ccc(F)cc1 CCC(CNC(C1CNC(=O)CN1C(=O)C1=CCCC1C)=O)C(C)(F)F C1(CNC(c2cncc(F)c2)=O)CC2(CCC2)CN1C(c1cc(Cl)nnc1O)=O C1(C(=O)NC(C)CCO)C2C3CC4C1C2C34C(N1CCOC(CO)CC1)=O C1(NC(CCOC)=O)CC(CNC(=O)CCC2CCCCO2)C(O)C1 CN1CC2(CCN2C(C2(C)CCCN2C(C2CCCC2F)=O)=O)C1 C(C(CNC(c1cccc(CO)c1)=O)S(C)(=O)=O)NC(c1c(C)cns1)=O N1(C(C(C(CC)C)O)=O)CCN2CCN(C(c3cccc4nsnc34)=O)CC2C1 Cc1sc(=O)n(CC(=O)NCC2C3CCC(C3)N2C(=O)Cn2nccc2N)c1C C1(NS(CC)(=O)=O)CCCC(C(N2CCC(N(C(=O)C(F)F)CC3CC3)C2)=O)C1 c1(CC)cccc(C(N2CCC(C)C2C(=O)NCC2(N(C)C)CC2)=O)c1 c1(C(N(CCOC)CCNC(=O)CN(C(=O)C(C)C)C)=O)cc(F)c[nH]1 C(CC(O)C(=O)NCCC(O)C(F)F)NC(C(C)(C)n1cnnn1)=O C(=O)(C(C#N)C(C)C)NCCN(C(c1oc(C)c(Br)c1)=O)C(C)C CCC(O)C(C)C(=O)NCC1CC(NC(=O)C2=C(Cl)CCC2)C1 c1(C(N2C(CCNC(=O)C(F)C3CC3)CCC2)=O)ccc(O)c([N+](=O)[O-])c1 c1(N2CCC(NC(c3cn(CC)nn3)=O)C(F)C2)ncc(Cl)cc1[N+](=O)[O-] Cn1ccc(=O)cc1C(N1CC2CCC2(C(=O)NCc2cccnc2)C1)=O C(=O)(CCC1=NNC(=O)CC1)N1CCCC2(CN(C(c3c(CC)[nH]cc3)=O)C2)C1 c1(CC(=O)N(CCCNC(=O)CSc2cn[nH]c2)C)cnc2cccnn12 C(c1cccc(O)c1)=CC(N1CC(O)(C(C)NC(C2CCC=CCC2)=O)C1)=O c1(Nc2ccc(CC(=O)O)cc2)ccc(F)c(Cl)c1F N1(C(C(C=C)O)=O)CCCC(C(=O)NCC(C)(CNC(=O)OC(C)(C)C)OC)C1 CS(=O)(=O)CCCCCN=c1[nH]c(NCC2CCOC2Cl)nc2ccsc12 c1(N(C)Cc2ccc(OC)nc2F)ccc(C)c(C#N)c1 N1(C(c2c(C)onc2)=O)CCOCC(CNC(=O)Cc2ccccc2)C1 Cc1cc(C(=O)NC2CCCN(C(C3CC4CC4C3)=O)CC2)nc2[nH]nc(O)c12 C1(C(=O)NC(CCC)C)CN(C(=O)Cn2ccccc2=O)CC1(C)C N1(C(COC2(C)CCCC2)=O)CCC(O)(CNC(C23CC(C#N)(C2)C3)=O)CC1 N1(C(c2n(CC)c(O)nc2)=O)CCC2CN(C(=O)Cc3cscc3Br)CC12 N1(C(CCc2c(C)noc2)=O)CCC2(CNC(=O)COC3CCC3)CCCC12 C(=O)(CC(C(F)F)NC(c1sccc1CO)=O)Nc1ccc(OC)cc1 C1(NC(C2(C)CSC2)=O)CCCCN(C(=O)CCCNS(C)(=O)=O)C1 c1(C(=O)NCC2(C)CCN(C(C(C)(C)CC#N)=O)C2)cccc2c1CCN2 CCC(C(=O)N1CCC1CNC(=O)CCOc1ccc(C)cc1)C(C)C c1(NC(c2ccc(OCC(=O)C3CC3)cc2)=O)c[nH]c2ccccc12 c1(NC(c2cccc(NCC3CCCC(C)CC3)c2)=O)c(Br)cccc1[N+](=O)[O-] c1(OC)cc(C(=O)N(C)CC2CCCN2C(C2CCSC2)=O)cnc1O Cc1nc2c(O)cc(C(=O)NCCN(C(C3CC3F)=O)C(C)C)cc2n1C N1(CCNC(=O)Cc2cccnc2)CCC(NC(=O)CC2CC(F)C2)CC1 c1(NC(C(c2ccc(O)cc2)C)=O)cccc(NC(c2ccnc(Cl)c2)=O)c1 CCCCCCCCCC(O)C(=O)NCCCN(C(=O)CNC(=O)CN(C)C)C Cn1cnc2cccc(C(N3CCC(C)(C)C3CNC(c3nccs3)=O)=O)c12 C1(CC(N2CC(CCC)C2)=O)CN(C(=O)Cc2scnc2C)CC12CC2 C1(CCOC)COCCN1C(c1cccc(C(C2CCCC2)=O)c1)=O c1(CN2CCN(c3c(C#N)ccnn3)C3C2C3)cn2cccc(C(F)(F)F)c2n1 C=CCC(C(=O)N1CCCC1C(C)NC(=O)C(C)(C)n1ccnn1)NC(C)=O C(=O)(C(F)(F)CC(C)C)NC(CN(C(C12CC(OC)C1C2)=O)CC)C CCC(C)(CNC(c1cnn(CC2CCC2)c1)=O)NC(c1ccc(CO)o1)=O CC12CCN(C(C3CC3C3CCCO3)=O)C1CN(C(=O)Cc1c[nH]c(=N)[nH]1)C2 N1(CC(=O)N(CC)CC)CC(NC(=O)Cc2ccc(C(N)=O)s2)CCC1C Cc1cc(C(N2CCCC(CN3CCCC3)C2)=O)ccc1-n1cncn1 Cc1ccc(-n2nc(Cc3ccccc3Br)nc2-c2[nH]c(COC)nc2C)cc1 c1(CNC(CC(CNC(C(C)OCC#C)=O)(C)C)=O)ccc2ncnn2c1 Cc1ccc(CNC(=O)CNC(=O)CNC(=O)Cc2nccs2)n1C N1(C(=O)NCC(CCC)OCC)CCC(CC#N)CC1.C1(CSC)(O)CCCCC1 C(C)(C)(C(=O)NNC(=O)CC(O)Cn1nnc(-c2cn(C3CCC3)nn2)n1)OC C1(C(=O)NC(C)(C)CCNC(=O)C(C)(C)F)CC2CCCN2C(=O)N1 Cc1cc(C(N2CCC(NC(C34CC(O)C3C4)=O)C23CC3)=O)cc(C)n1 c1(-c2scc(C(=O)NC3C(CNC(c4c(CC)ccs4)=O)C3)n2)ncccc1F CON1CCC(C(N2CC3(CC(CC(=O)Nc4ccc(F)c(C)c4)C3)C2)=O)CC1 CN1CCCC1C=CC(=O)NCCCCCCNC(=O)Cc1ccc(O)nc1 S(=O)(=O)(c1ccc(-c2cncnc2)c(C)c1)NCCN(CCC)CC N1(C(C2C(C)C2)=O)CC2(CC(NC(=O)C(O)CCCc3ccccc3)CO2)C1 CC(C(=O)N1CCOC(CN(C)C(c2ccn(CCF)n2)=O)C1)C(F)F c1(C(=O)NCC2(F)CN(C(=O)CC3CCCO3)C2)ccc2[nH]ccc2c1F c1(CC(N2CCC(N(C)C(C3CCOC(=O)N3)=O)C2)=O)csc2cccc(F)c12 c1(C(N2CCN(C(c3c(C)nsc3)=O)CC2CO)=O)ccc2cnsc2c1 c1(C(=O)NCC(=O)N(CCC#C)C)cc(CC#C)ccn1.C1(=O)CCOCCN1C N1(C(CCCCC=C)=O)C2CC=C(C(=O)NOC3CCOCC3)C1CC2 c1(C(=O)NC(C)(CNC(=O)C(F)n2cccn2)CO)occ2c1CCOC2 CC1(NC(=O)Cn2c(O)nnc2O)CCCCC1C(=O)NCc1nc(CO)n[nH]1 c1(CC)occ(C)c1C(N1C(C(=O)NCC(O)CCC2CC2)CCC1C(C)C)=O CCCCCC(O)CC(=O)NCCCN(C)C(c1c(Cl)c(CC)nn1C)=O N1(C(C(CCCC)O)=O)CC(NC(=O)C=Cc2ccc(SC)s2)CCC(O)C1 C1(C)(CN(C(c2cnc(C(C)C)[nH]2)=O)C)CCCC1NC(=O)CCn1cnnn1 C1(C(=O)NCC(CC)C#N)CC12CC(NC(=O)CCOCCOC)C2 N1(C(COc2cn(C)nc2)=O)CC2CCN(C(=O)CC3CCC(O)C3)CC12 CC(CC(F)(F)F)C(=O)NC1CC2CCC1CN2C(C1CC2CC1CC2O)=O C1(C(N2CCC(CCC(=O)NCC(CCOC)(C)O)CC2)=O)CCC2(CCC2)C1 c1(NC(=O)OC(C)(C)C)ccc2[nH]c(CNC3CSCCS3)cc2c1 C(=O)(CC(C)(C)CNC(C1(CSC)CC(=O)C1)=O)NC(C(CC)C)CN(C)C N1(C(CC)=O)CCC(C(C)C(=O)NCc2cc(C)c(C(N)=O)o2)CC1 N1(C(=O)OCC)CCN(C(c2cccc(C)c2)C(=O)NCc2ccco2)CC1 c1(C(N(CCNC(c2ccc(C)cc2)=O)CC)=O)ccc2c(c1)NC(=O)C2 Cc1ccc(CN2CCC(NCc3ccc(OC(F)(F)F)nc3)C2)c(C)c1 c1(C(N2C(CNC(C(CCC=C)(F)F)=O)CCC2)=O)ccc2c(c1)NC(=O)CN2 C1(NC(CC2(C)CCCCC2)=O)CC2CC1CN(C(=O)C(C)(Cl)Cl)C2 N1(C(C(C)Sc2nncn2C)=O)CC2CC(NC(c3coc(C#N)c3)=O)CC1C2 C#CCC(C)(C)C(=O)NC(C)CCCNC(=O)C(C)(Cl)Cl CC1CN(C)C(C)CC1NC(=O)CC(CNC(c1coc2c1COC2)=O)C1CC1 C12(C(N3CCCC(OCC#C)C3)=O)CC(CO)(CN1C(=O)C#CC(C)(C)O)C2 C1(C(C(=O)N(C)CCOCCNC(c2ccc(Cl)nc2)=O)O)CCCCCCC1 N#Cc1ccc(NC(C2CC23CCN(Cc2cccc(F)c2I)CC3)=O)c(F)c1 Cc1ccc(CC(CNC(=O)NC(C2CCN(c3ccncc3)C2)=O)CO)cc1 c1(C(=O)NCC2CCN(C(C3(O)CCOC3)=O)C2)cc2c(F)cccc2s1 C(C(N=[N+]=[N-])C(=O)N1CCN(C(c2c[nH]cc2C)=O)C(C)C1)OCC C1(CNC(CCOC)=O)CCCC2CN(C(C34CCC(CC3)C4)=O)CC12 C1(NC(C2C(CC)C2)=O)(CNC(C2CC2c2ccccc2F)=O)CCOCC1 C1(C(N2CCC(CC)C2)=O)CCCCC1(C)C.C12(CCCCC1)CNC(=O)N2 C1(C(=O)NC2CC(C)(NC(c3cnc(Cl)s3)=O)C2)CN2CCCN1CC2 c1(C(=O)NC2CN(C(C=CC(=O)N(C)C)=O)CC2C)cc2c(c([N+](=O)[O-])c1)OCO2 CC(C(=O)N(CCCCNC(=O)CCOCC1CC1)C)c1ccsn1 c1(C(N2CCN(CCNC(C(C)(C)OC)=O)CC2)=O)sc2nccn2c1C N1(CCC#C)CCC(CC(=O)NCC(C)(O)CNC(C2CC(O)C2)=O)CC1 N1(C(c2cc(C)sc2C)=O)CCc2ccc(CC(N3CCOC(C)C3)=O)cc2C1 C1(C(=O)NCCNC(C(C)NC(C)=O)=O)(OC(c2nn[nH]n2)C)CCOC1 Cc1cn2nccc2c(NCC(c2ccccc2)N2CCCC2)n1 C(=O)(CS(=O)(=O)C(C)C)NC1CC(NC(CCc2ccc(OC)cc2F)=O)C1 c1(O)cnc2cc(Br)ccc2c1.c1(C(=O)OC)nc(C2CN(C(=O)NC)C2)no1 N1(C(c2c(OC)c(F)c(C)cc2)C(=O)NC2CC2)CCc2ccc(C#N)cc2C1 Cc1ccoc1C(=O)NCC(C)(C1CCC1)NC(c1cnn(CC(F)(F)F)c1)=O C(CCC(C)(C)C(=O)NC(CO)C(C)O)NC(c1n(CC)nc(C)c1)=O N1(C(C2C=CCN(C(c3cnc(O)o3)=O)C2)=O)CC(F)(F)CC1CO C(=O)(CCC(O)C(C)(C)C)NCC(CN(C(c1c(OC)ccc(F)c1)=O)C)C c1(OC)ccc(Cl)cc1CC(N1CC2CC1C2CNC(=O)C=Cc1nccs1)=O CC1CC(C(=O)NCCCOCCNC(=O)C2=C(Cl)CC2)C1(C)C C(C)(C(=O)N1CC(C)(NC(C2CC2C(C)(F)F)=O)C1)(C(C)C)OC S(=O)(=O)(c1cccs1)N1C(C)(C(=O)Nc2ccccc2I)CCC1 c1(C(=O)NCC(C2CCC2)NC(=O)CC2CCSC2)cscc1Cl N1(C(Cc2c(C)ccs2)=O)CCC2(CCN(C(c3cc(CF)on3)=O)CC2)C1 CCC(C)(CNC(=O)CC(C)(C)NC(=O)C(C)N=[N+]=[N-])CC Cc1nnn(C)c1C(=O)NCC1CCC(NC(=O)C=C2CCC(C)C2)C1 CCC(C)CC(=O)C(=O)N1CC2CC(C(N3CC(C)CCC3CC)=O)(C2)C1 c1(N(CCOC)C)ccc(Br)c(S(=O)(=O)N2CC3OCCOC3C2)n1 CC1=C(C(=O)NCC2CC(NC(c3cc(C(N)=O)ccn3)=O)C2(C)C)CCC1 C1(C(C(=O)NC2CC(=C)C2)N(CCC(=O)NC2CC(F)(F)C2)C)OCCC1(C)C C1(NC(C(c2n(C)ncc2)(F)F)=O)CCCCN(C(=O)CCc2nc[nH]n2)C1 N1(C(CSC(C)C)=O)CCCN(C(c2cc(F)c(F)cc2C(F)(F)F)=O)CC1C C(CN=c1[nH]c(=NCCC2CSCCO2)[nH]c2c1CSC2)(N(C)C)C1CC1 c1(OC(C(=O)NCCC2CC(NC(c3n(CC)ccc3)=O)C2)C)cccc(F)c1 C=CC1CN(C(=O)CCOCC)CC1NC(C1(C)CC2CCC1O2)=O N1(C(c2c(OC)ccs2)=O)CCC(C(C)CNC(=O)C(C)(CO)OC)CC1 CCCCCC(CC)C(=O)N1CC=CC(C(=O)NC(C)Cc2ccco2)C1 c1(C(N(CCN(C(C(=O)NC(CC)C)C)C)C)=O)cccc(-c2cnccn2)c1 C=CC(C)(C)CC(c1nnnn1C(C)(C)CC)NCC12CCC1CCO2 c1(C(N(C(C)C(=O)NCCc2ncnn2C)CC)=O)n[nH]cc1NC C1(CC)CN2CCC1NC2=O.c1(C(=O)OC(C)(C)C)cccc(C(=O)O)c1OC c1(NC(C(c2ccco2)NC(c2cc(C)ncc2)=O)=O)c(C)cc(C)nc1C c1(C(=O)NC(c2cn(C)nn2)C(=O)NC(c2onc(C)n2)(C)C)noc(=O)n1C C1(CCCC)CN(c2nncn2C2CC2)CCN1 C1(C(=O)NCC(CC)(CC)NC(C(CCC)=CCC)=O)CCC2(CCC2)O1 C1(NC(C(c2ccoc2)NC(C2N(C)CC(F)C2)=O)=O)CC2(CCOC2)C1 C1(C(N2CCC(=C)CC2)=O)CC(F)(F)CN1Cc1ncn(C)n1 C1(NCC(=O)NC2(CNC(=O)Cc3nccs3)CC2)CCn2cncc2C1 C12(NC(c3cncc(C)c3)=O)CCN(C(=O)CCN3CCC(C)CC3)CC1C2 n1(NCC(CCCC)N(C(C)C)C)ccc(O)nc1=O.C(=O)(CNC=O)N C12(C(N)=O)CCCC1(C(N1CC(O)(CNC(c3cc(Cl)no3)=O)C1)=O)C2 O=C(C(F)CC1CCCC1)NC1COCC1C(=O)NCC1CCCOC1 Cc1c(NCC2CC2C)ncnc1NC1CC(=O)NC(=O)C1 Cc1cc(C(=O)NCCCN(C(=O)CP(C)(C)=O)C2CCCC2)n(C(F)F)n1 N1(C(C2(CC#C)CCCCO2)=O)CC2(CCCN(C(=O)C=CCC)C2)C1 C1(NC(c2ccc(CCC)[nH]2)=O)CCC2(CC1)CC(NC(c1ccc(Cl)o1)=O)C2 c1(NC(C(CC#CC)NC(c2cc(C)c[nH]2)=O)=O)cccc2ccoc12 Cc1no[nH]c1=NC(=O)CC1CCCN1C(=O)CCc1c(C)[nH]c2ccccc12 N1(C(C(CSC)O)=O)CCCC(C2CCCN2C(=O)CCC2CCCCO2)C1 C1(NC(C(CC)n2ccnc2)=O)CN(C(=O)CNS(C)(=O)=O)CC2(CC2)C1 c1(OC)ccccc1CC(=O)NCC(C)N(C)C(c1ccc(C(N)=O)cc1)=O c1(C(=O)NC2CC(NC(c3c(C4C(C(=O)OC)C4)noc3)=O)C2)ccc(C)cc1 N1(Cc2ccc(C(C)(C)C)nn2)CCC(O)C(O)C1.c12cccc(c1)C(=O)N2 c1(C(N2C(CNC(C(C)N(CCC)CCC)=O)CC2)=O)cocc1C.C(=O)OC CC1=NS(=O)(=O)NC(C)=C1CCC(=O)NCC1CC(NC(=O)C(F)F)C(O)C1 c1(C(=O)NC2C(C)N(c3ncnc(Cl)c3C#N)CC2)cccc2c1NC(=O)CC2 CN1CCC2CC1CN2C(=O)CC(c1ccccc1F)c1ccccc1 N1(C(CNC(CN(C2CCC2)C)=O)=O)CCC(NC(N)=O)C(C)(C)C1 C(C)(C)(CC(=O)N(C1CN(C)C1)C)NC(c1c(OC)csc1)=O N1(C(CC2C(C)C2)=O)CC2CCC(C1)N2C(c1cc(=O)cc[nH]1)=O N1(CCNC(C2C(CC)CCC2)=O)CCCN(C(=O)C(C)(C)C#N)CC1 c1(CC)nc(C(=O)NC(C2CCCCC2)C(=O)NCCCC2CCOC2)cs1 C(CC(C)C)(C(=O)NCCc1cn[nH]c1)NC(C1CCC(C)(CC)O1)=O c1(N2CCC(C)(CNC(C(CC)OCC)=O)C2)ncc2cccnc2n1 N1(C(COC(CC)CC)=O)CC2(CCN(C(=O)CNC(C)=O)CC2)C1C(C)C Cc1nc(C(=O)NCCN(C(c2ccnc(C(F)F)c2)=O)C2CC2)c(C)o1 N1(C(c2c(CC)nns2)=O)C(C(=O)NCc2cncc(F)c2)CCC1C c1(C(=O)NC(C2C(C(=O)NCCCC(=C)C)C2)C)cc2n(n1)CCO2 C(=O)(C(C)C(C)C)NCCCN(C(c1cc(OC)no1)=O)Cc1ccccc1 c1(C(N2CC=CC2)=O)ccc(C(=O)NCC(C(=O)NCCOC)N(C)C)[nH]1.CC C(=O)(C(O)COCC(=O)O)NCC1CC(NC(C(C)=CC)=O)C1.c1(S)ccccc1 C1(NC(c2c(C)nn(C)c2)=O)CC2CC1CN2C(c1nc(C(C)C)oc1C)=O c1(C(=O)NC(CC=C)CNC(c2ccc(SC)s2)=O)cc2sc(Cl)cc2[nH]1 CCC(O)CC(=O)NC(C)CNC(=O)C(c1cccc(C)c1)=O Cc1ccc(C=CCC(=O)NCC2CCN(C(c3c[nH]c(C)c3)=O)C2(C)C)cc1 C12(C(=O)NC3(C)CSC3)CC1CN(C(c1ccc(CO)nc1)=O)C2 Cc1n[nH]cc1CC(=O)NC(CC1CC1)C(=O)N1CCC(N2CCCCC2)C1 N1(C(C2(NC(c3ccn(CC)c3C)=O)CCOCC2)=O)CCC2CC1C(=O)O2 c1(CNC(C(c2cnn(C)c2)NC(C2CC(SC)C2)=O)=O)cncc(Cl)c1 C(=O)(C(C)(F)C(=O)NCC1CCCC1NC(c1ccc(C)cc1)=O)OCC c1(C(C(=O)NCCC)N(C)Cc2ccco2)cc(-c2ccccc2)no1 C1(c2nc(-c3cn(C4(C(F)F)CC4)nn3)no2)COC2CN(C(N)=O)CC12 N1(CCNC(c2c(C(C)(C)C)ncs2)=O)CCC(NC(c2cscc2Cl)=O)CC1 Cc1ccc(CC(=O)NC2(CN(C)C(C3CC(=O)NC3(C)C)=O)CC2)c(F)c1 N1(C(C2C(C=C)C2)=O)CCC(COC)(NC(=O)COc2c(C)occc2=O)CC1 N1(C(C(C)C2CCCC2)=O)CCCCC2C1CCCN2C(=O)CS(N)(=O)=O C(=O)(C1CCc2cc(Cl)ccc21)N(CCNC(C(CSC)O)=O)CCOCCO C=CCCCCn1cc(C2(O)CC(CNS(N)(=O)=O)C2)nn1 C(=O)(C(CC(=C)C)NC(=O)C=CC(C)(C)SC)NC(C#C)CC1CCC1 C1(NCc2c(C)ncs2)CC2CC(C1)N(Cc1ccccn1)C2 N1(C(C(=O)NCCC)CCC2(C#N)CC2)CCOC(C)(C(C)(C)C)C1 C1(N(C(c2c(OC)scc2)=O)C)CCCN(C(c2ccc(C)cc2F)=O)CC1 N1(C(=O)NCC#C)CC2CCC(C1)N2C C1(CC(=O)NCCCC(C)NC(C(CC)C)=O)CC2(C1)CC1(CCC1)C2 C(C(C(=O)NC1(C2CC2)CCCO1)N(C)C)NC(CCSCC(C)C)=O N1(C(=O)C=Cc2cocn2)CCC2CCCC12C(=O)NCCC(O)C(F)F Cc1cnc(N2CCC(C(C)NC(=O)C(F)CC3CCCC3)C2)nc1C CC1CCCC1(C)NC1(c2nnnn2CC2CCOCC2)CCN(C)C1 c1(-n2ccc(C(=O)NC3CC(NC(CC4(OC)CC4)=O)C3)n2)ccc(F)cc1 c1(OC)cccc(C=CC(=O)NCC2(NC(=O)C(C)n3cccc3)CC2)c1 N1(C(C(C2CCCO2)OC)=O)C2CCC(C(=O)NCc3cc(C)c(C)s3)C1CC2 c1(NCC)ccc(I)cc1[N+](=O)[O-].c1(CN2C(=O)C3CCCC3C2)ccccc1C c1(C(=O)NCC2N(C(C3CCC(C)O3)=O)CC2)ccc(Cl)cc1[N+](=O)[O-] N1(C(COCCC#C)=O)CC(C)C(C)(NC(=O)COC2CC(C)C2)C1 c1(NC(C2C(O)CCN(Cc3scc(C)n3)C2)=O)cc2c(cn1)OCCC2 C1(CNC(C=C(C)C(F)F)=O)CCN(C(=O)CCc2cnc[nH]2)CC1C n1(C2(C(N(CC)CC3CC3F)=O)CC2)cc(Br)nn1.C12CC1NC2=O.NCC CC1CN(C(=O)CC2CCCNC(=O)C2)CCN1C(C1CC12CCCC2)=O C1(C(=O)NC2C(N(C)C)COC2)CC2CCC1N2C(c1ccccc1C1CC1)=O C1(C(=O)NCCCOCCN(C(CCn2ccc(C)n2)=O)C)CCC(O)CC1 C1(NC(C2CCN(C(C)=O)CC2)=O)C2CCC1CN(C(=O)CCC(C)(C)F)C2 C(=O)(CCCCC(=O)N1CCC(CN(C(=O)C(C)CC(C)C)C)CC1)NC C(=O)(C(C)C(F)(F)C(F)F)N1CCN(C(c2[nH]cc(C)c2C)=O)C(CC2CC2)C1 c1(C(=O)NC(c2cc(OC)cc(OC)c2)C2CC2)c(C#N)cnn1-c1ccccc1 O=S(=O)(c1ccc(F)c(F)c1)N1CCc2cccc(-c3ccc(F)nc3F)c2C1 N1(C(c2cc(C)oc2)=O)CCC(C)(C)C(NC(c2ccc(C)c(C)n2)=O)C1 n1(CC)ncc(C(N2CCN(C(c3sc(OC)nc3C)=O)CC2)=O)c1C c1(OC)ccccc1NC(=O)C(c1nccs1)N(C)N(C)C.c1(COC)cncs1 C1(CCNC(C2C(C)CCC2)=O)CCCN(C(=O)CCc2cc(Cl)no2)C1 N1(C(c2c(Cl)ncc(C)c2)=O)CCC2CN(C(=O)C=CCBr)CC12 N1(CCC2(C(=O)OC)CCCCC2)C(=O)CN(CC2CC3CCC2CC3)C1=O C1(CC(=O)NCC2(N(C)C)CCC2)(CNC(=O)CSC(F)(F)F)CCCC1 c1(C(=O)NCC(CNC(CC(CCCC)O)=O)C)ccc2c(c1)N(C)C(=O)CC2 C1(NC(C(CC)OCC)=O)CN(C(=O)C(=O)Nc2ncc[nH]2)CC2(CC2)C1 N1(C(C(C)C2CCC2)=O)CCCN(C(C2CCS(=O)(=O)CC2)=O)C(C)C1 c1(CN(C(=O)C(=O)NC2CC23CCNC3)C)ccc(F)c2ccccc12 C1(CNC(C(CNC(C(C)NC(C)=O)=O)CC2CC2)=O)CC2CCCC2C1 C(CS(=O)(=O)Cc1ccc(F)cc1)NC(N1CCN(CCN2CCCC2)CC1)=O N1(C(c2ccnc(Cl)c2F)C(=O)NC2(C)CC2)C2CCC1CC1(C2)N=N1 N1(C(CC(C)(C)OC)=O)CCC2(CCCCN(C(C3CCCC3)=O)C2)C1 CC1(C(=O)NCCC2(O)CCN(C(C3(CO)CCC3)=O)C2)CC=CCO1 C(=O)(C1=COCC1)NCCC(Cc1ccccc1)NC(Cc1c(C)occ1)=O N1(C(CC2CCC(C)C2)=O)CC2(CNC(c3cc[nH]n3)=O)CC1CCO2 c1(C(C)C(N2CCOC(CN(C(=O)CC3CC3)C)C2)=O)ccc(F)c(F)c1 CCCCCCCC(=O)NC1CN(Cc2cccc(I)c2F)C1 N1(c2ncc(C(=O)OCC)s2)CC2CCCC(NC(=O)Cc3csc(S)n3)C2C1 C1(C(N(CC(CO)(CO)NC(c2cc(C(N)=O)n[nH]2)=O)C)=O)CCCNS1(=O)=O c1(C(=O)OC)ccc(C(N2CCC(NC(c3cc(Cl)c(C)cn3)=O)C2)=O)c(F)c1 C(=O)(C(C)(C)C(=O)N(C)C)NCCC(C)CN(C(=O)CC(C)CF)C CC1(C)CC(C(=O)NCc2cccs2)N(C(C2CCC3(CC3)C2)=O)C1 C(CCC(=O)NC(CNC(=O)COCC1CCCCO1)C1CCC1)OC(C)=O C(CCN(C)C(C1CN(C2CCOCC2)C1)=O)(C(C)C)NC(C(C)=CC=CC)=O c1(C(=O)NCC2(O)CN(C(C3C(C(=O)OC)C3)=O)C2)cccc(C2(F)COC2)c1 CC(C)(C)CCC(=O)NC1CC(NC(=O)CC2CC(O)C2(C)C)C(O)C1 N1(C(C(C)=O)=O)CCC(F)(CNC(c2cnc(O)c(Br)c2)=O)CC1 CC1COCCC1N(C)C(c1cc(CCNC(=O)CCc2cnoc2)on1)=O C1(C(=O)NCC2(C(=O)NCCC(C(C)C)O)CC2)CC2CCC(C1)O2 C1(CNC(c2nc(C)oc2)=O)CN(C(=O)CCN2CCC(F)C2)CC(C)(C)O1 CCCCC(O)C(C)C(=O)NCC1(O)CN(C(c2ccccc2OCCC)=O)C1 c1(CCCC)nc(C)c(C(=O)NCC(C)(C)CN(C)C(c2cnc(O)n2C)=O)s1 C1(NC(C(C=C)C)=O)(CF)CCN(C(=O)CCc2cccnc2)C1 N1(C(Cc2c(C)cccn2)=O)CC2CC1CCC2NC(c1c(C)nn(C)c1Cl)=O Cc1noc2nc(C(=O)NCCC3CN(C(=O)C(F)(F)c4nccs4)C3)ccc12 N1(C(C2C3(CN(C(C(C)Cn4cncn4)=O)C3)C2)=O)CCc2ccc(F)cc2C1 c1(C(=O)NC2CCN(c3cc(C)ncn3)CC2F)cnn2ccn(C)c12 C1(NC(C2ON=C(C)C2)=O)CN(C(c2ccnc(C3CC3)n2)=O)CC1(C)C Cc1ccc2oc(C(=O)NCC(C)N(C(=O)C(c3cccnc3)C)C)cc2n1 c1(C(=O)NCCN(C(C2CN(CC)C(=O)N2)=O)C(C)C)ccc2c(c1)NC(=O)C2 O=C1CCC(C(N2CC=CC2CNC(c2ccc(-c3csnn3)cc2)=O)=O)CN1 c1(NC2(COCC)CCCNC2)cc(C(N)=O)c2n1CCCC2 CN1CCC(NC(C2(n3cc(C(N4CCOCC4)=O)nn3)CC2)=O)C1=O n1(CC)nnc2c1CCC(C(=O)NCCNC(=O)CCC(C)c1ccccc1)C2 N1(C(C2(OC)CCOCC2)=O)CC(CNC(c2ncsc2C)=O)OC2(CCC2)C1 n1(CCC)ncnc1C(c1nnnn1CCC)NCC1(CO)CC1 N1(C(C=CC)=O)CC(C(=O)N(c2ncc(CC)cn2)C)CC(C)C1.C(C)(C)(C)OC=O c1(OC(C2(C3CC3)CCOCC2)=O)ccc(CN(C)CC)c(CN(C)C)c1 c1(C(N2CCC(CNC(C(C(C)C)O)=O)C2)=O)cn2c(n1)CCC2 C=CCC(C(=O)N1CCN(CCCCNC(c2cscn2)=O)CC1)OC c1(C(=O)NC2CC3(C(NC(=O)CCF)C3)C2)cnc2c(=O)[nH]cc(CCO)c2c1 N#Cc1ccc(NC(c2sc(-c3ccc(F)cc3O)nc2C)=O)cc1Cl N1(C(CC=C=C)=O)CCCC(C(C)N(C(=O)CCCOCC=CCC)CC)C1 O=S(=O)(c1ccnn1C1COC1)NCc1ccc(Cl)cc1N1CCSCC1 N1(C(C(CNC(=O)OC(C)(C)C)O)=O)CC(NC(c2cccnc2)=O)C(F)(F)C1 C(c1ccc(C(=O)CCCC(C)C)nc1)=C(C)C.C1(C(=O)OC)CC1CO c1(OC)ccc(CN2CCC(CC(=O)NC(c3ccc(Br)cc3)CO)C2)cc1Cl c1(C(=O)NCC#CCNC(c2ccc(OC)s2)=O)cccc2cccnc12 Cc1cc2c(C(N3CC4CC(CNC(C5CCN(C)C5)=O)C4C3)=O)nccn2n1 c1(C(=O)NCCSCC(=O)NC(COC)CCO)ccc(C)c(C#N)c1 C(C)(N=c1[nH]c(Cl)ncc1Br)c1c(C)nc(C)s1 c1(C(=O)NCC2C(CNC(C3C(C)OC(C)C3)=O)C2)nn(C)cc1[N+](=O)[O-] C1(C(=O)NC(C(=O)N(C(C)C2CC2)C)(C)C2CC2)C2CC(=O)CC12 c1(C(=O)NC2CCC(NC(C=C(C)CN3CCOCC3)=O)C2)ncc[nH]c1=O c1(C(=O)NC(CC)(COC)c2cccs2)cc(-c2ccn(C)n2)nc2onc(C)c12 CC1=C(C(=O)NCC2(CC(=O)NC3CCC(C4CC4)CC3)CC2)COCC1 N1(C(c2n(C)ncn2)=O)CC2(CC(NC(=O)Cc3noc4ccccc34)CO2)C1 C1(CCC)CN(C(=O)C(O)C2CC2)CCN1C(C1CN(C2CCC2)C1)=O Cc1cc(C(=O)NC2CN(C(C3CCN(C)C(=O)C3)=O)CC2C)c(N)c(C)c1 c1(C(=O)NC2C(NC(c3cc(SC)c(N)cc3)=O)C2)c(C)sc2ccccc12 CC(C)(C)C(=O)OCC(NC(NCC#C)=S)N1CCCC1 C(=O)(C1OC(=O)c2c(F)cccc21)NCCN(C(=O)C1=CCC(C)(C)CC1)C c1(CNC(=O)C(=O)Nc2cccc(C(=O)NC(C)C)c2)cc2ncccc2s1 N1(C(C(C)Sc2ccccc2)=O)CC2CC2(CNC(=O)Cn2cccn2)C1 C(=O)(C1CCCc2nn[nH]c21)NC1CC(CCNC(c2c(OC)cncc2)=O)C1 CS(=O)(=O)C1CC(C(=O)NCC2(O)CCN(C(C3CC(C#N)C3)=O)CC2)C1 C12(NC(c3cc[nH]n3)=O)CCC(CC1)N(C(=O)C(CC(F)F)C1CCC1)C2 c1(C(Cc2ncco2)N)ccc(Cl)c(Cl)c1.OC(CCc1ccsc1)C1CCCC1 C1(NC(CC(COC)(C)C)=O)CC2CCCC2N1C(C1(CCC(F)(F)F)CC1)=O C(=O)(CC(C)CC(F)(F)F)NCCC1OCCN(C(c2c(OC)n[nH]c2)=O)C1 C1(C(N2CC(NC(C3CC4CC4C3)=O)C(F)C2)=O)(OC)CCCCCC1 N1(C(c2ccc(OCC)cc2)=O)C2CCC1CC(NC(C1(C)CC(C)C1)=O)C2 c1(OCC(C)C)ccc(C(N2CCC(N(C(=O)COCC3CC3)C)CC2)=O)cc1 N1(C(C2CCN(C(CC)=O)C2)=O)CCN(C(C2C3CCCC23)=O)CC12CCC2 c1(N(C)C)ccc(F)c(C(=O)NC2CCN(Cc3cc(-c4ccns4)on3)C2)c1 C(C(C(=O)NCC1COCCO1)NC(=O)C=CCF)OC C(C)(C(=O)NCCOCCN(C)C(C1(F)COC1)=O)SC Cc1ccc(C(=O)NCCCCC(C)NC(C23CC(CN2C2CC2)C3)=O)c(Cl)c1 c1(C(=O)Nc2cn(C)c(CNCc3ccc(CBr)s3)c2)cc(F)ccc1[N+](=O)[O-] C(=O)(C1=NOC(C)(C)C1)NCC1N(C(c2n(C)cnc2)=O)CC1 C(N=c1cc(NCC2C=CCC2)nc(C)[nH]1)c1ccc(OC)cc1Br c1(C(N2CCCC(N(C(=O)CC(C)O)CC)C2)=O)cc2c(C)cc(OC)cc2[nH]1 C1(CC)CCN(C(=O)CC2CCCN2C(=O)C(C)c2ccco2)CC1 C(=O)(CCCC(=O)N(C)C)N(CCC(c1cccs1)NC(C12CCC1CC2)=O)C N1(CC(=O)NC)CC2CC2C1.C1(c2ccccc2)CCCC1.C12(CC1)CCNC2=O C1(C(=O)NC2CCCC(CO)C2)CN(C(c2cc(O)nc(O)n2)=O)CC1(F)F CCCCCCCCC(=O)NC1COC2(C1)CN(C(C1(C)CC(F)C1)=O)C2 C#CCCCCCCC(=O)NC1CN(C(C2CC(N3CCCC3)C2)=O)CCC1C c1(C(=O)OCC(N2C(C(N)=O)CCCC2)=O)nnc2ccccc2n1 c1(CC(N2CC(C(C)NC(C(CO)OC)=O)C2)=O)cc(C)cc(F)c1 C(=O)(C(C)(C)C(C)C)N1CCC(C(C)NC(C(CC)CN(C)C)=O)CC1 CC1(CC(=O)NCC(=O)CCCF)CCCC1C(=O)O C1(C(CNC(c2cc(C(C)=O)on2)=O)F)CCN(C(=O)C#CC2CC2)CC1 C(=O)(CC(O)CC(C)(C)C)NCC(CC)(CC)NC(C12COCC1C2)=O N1(C(c2ccc(O)cc2F)=O)CC2CCCN(C(c3ccn(CCF)n3)=O)C2C1 C1(NC(C(CC)(F)F)=O)CC2CC(NC(=O)CC(C)c3ccncc3)CC2C1 C1(CCNC(C2(C)C(C)C2)=O)CCCN(C(C2COCCN2C)=O)C1 Cc1cnc(C)c(C(=O)NC2CCOCC2NC(=O)C2=CCCSC2)c1 C1(C(=O)NC2(CCNC(C(C)C(C)(C)C)=O)CCOCC2)CCn2ncnc2C1 c1(CC(C)NC(c2cnc(C3CCOC3)s2)=O)cn(C)cn1 c1(C(=O)NCC(C)NC(=O)C(O)CN(C)C)ccc(N2CCNC2=O)cn1 C1(CC(=O)NC2CC3CN(C(=O)CC4(CO)COC4)CC23)CC2(CCC2)CO1 CCCC(CC1CCCC1)C(=O)N(CCCN(C(=O)CC1CCCO1)C)C S(=O)(=O)(c1cnoc1C(C)C)NCCCc1ccc(C)c(F)c1 CC(CCCNC(=O)C(N)=O)NC(c1conc1C1CCCO1)=O CC1=NNC(=O)C1CC(=O)N(C)CC1(O)CCN(C(c2cnns2)=O)C1 C=CCC(C)(CC=C)n1ccnc1-c1ccc(-c2cc(C)ccc2C)cc1.C(C)C Cc1nc(C)cc(=NC(C)CN(C)C(c2c(F)c(C(F)(F)F)nn2CF)=O)[nH]1 c1(C(N2C(CNC(c3nc(C)oc3C)=O)CCC2)=O)cccc2c(C)ccnc12 N1(C(Cc2c(C)scc2)=O)CCC(C(=O)NC2C(C)C2(C)C)C12CC2 N1(C(c2cc(C(C)=O)sc2)=O)CC2CC(NC(=O)CN(C)C)C(C2)C1 N1(CCC)CCC(C(=O)NCC=CCNC(=O)C(c2ccccc2)F)CC1 Cc1cc2c(C(=O)NCC3CC4CN(C(c5csc(O)n5)=O)CC34)nccn2n1 c1(NC(C=C2CCN(CC=CC)C2)=O)cnc(OC)c(Br)c1C(=O)OC C1(CNC(C(=CC2CCCC2)C)=O)CCCCN1c1nccc(CSC)n1 C1(NC(c2ccc(SC)s2)=O)CC(F)CN(C(=O)Cc2cc(C)cc(C)c2)C1 N1(C(C2C(C)CCO2)=O)CC(=O)CC1C(=O)NCCCC(F)(F)F C12(NC(=O)CCC3CCCCO3)CCC(CNC(c3c[nH]c(=S)cn3)=O)(C1)OC2 CCCC(CCC)C(=O)N1CCC(NC(=O)C(C2CC2)OC2CC2)C1 N1(CC(N)=O)CCCC(C)(C(=O)N(CCc2ccn(C(C)C)c2)CCCl)C1 C1(C#N)(C(=O)NC2(c3ccccc3)CN(C(C3C(OC)CC3)=O)C2)CC=CC1 c1(C(N2C(CCNC(=O)C#CC3CCC3)CCC2)=O)ccnc2ccc(Cl)cc12 C1(CCCC)CN(C(=O)Cc2cnsc2)CCN1C(=O)C(C1CCCCC1)C c1(C(N(CCOCCNC(Cn2nnc(C)n2)=O)C)=O)cnc(S)n1C c1(C(=O)OCC)c(N(CCNC(C2C3COCC23)=O)CC)nnc(C)c1C c1(OC)cccc(C(=O)NC2CCC(NCc3c(Br)ccnc3Cl)C2)c1Cl c1(C(N2CC(N(C(c3nn(CC)c(C)c3)=O)C)C2)=O)cc2n(n1)CCCC2=O c1(NC(C(Cc2cccs2)NC(=O)OC(C)(C)C)=O)coc2cc(O)ccc12 c1(OCC(N2C(NC(N3CCCC3)=O)CCCC2)=O)c[nH]c2ccc(Br)cc12 C(CCN=C(NC1CCOCC1)N(C)Cc1ccc(C#N)o1)NC C12(n3cc(CNC4C(N)CCC4)nn3)CC3CC(C1)CC(F)(C3)C2 c1(Nc2cnn(CCCC)c2C2CC2)cc(F)cc(C)c1O c1(N2CC3CN(C(C)=O)CC3C2)ncccc1S(=O)(=O)NCCCNC(=O)C1CC1 c1(NCC(CC=C)(C)C)ccc(S(=O)(=O)NC2C(C)C2C)c(Br)c1 N1(C(C2(C)COC(=O)C2)=O)CC2CC(NC(=O)CCSc3ccccn3)C1C2 CC1CCN(C(c2cc(Br)c(F)cn2)C(=O)NC2CCCC2)CC1C c1(OC)ccc(C(=O)NC2C3CN(C(=O)C(C)C)CC23)cc1[N+](=O)[O-] C1(OCC(=O)NCC2(F)CC(NC(C=CC)=O)C2)CCCC(C)C1 c1(C(=O)NCCN(C(=O)C(C)C(F)(F)C(F)F)CC)csc2c(OC)cccc12 CN(S(N)(=O)=O)CCCC(COCC(F)(F)F)NC(=O)CC(=O)OC(C)(C)C C1(C2CC2)(COC)CN(C(=O)C(=O)NCC(c2ccccc2)C(C)C)C1 C#CC1(F)CCN(C(C(=O)NCC2CC2)c2ccon2)CC1 CCC(CC)CCCC(=O)NCCN(C1CCCC1)C(c1cc(C(C)C)n[nH]1)=O O=C1CC2(CCN(CCNC(=O)C=C3CCCCC3)CC2)C1 C1(O)(C(C)NC(=O)C=Cc2ccccn2)CCCN(C(C2CC2c2ccco2)=O)C1 C(CC(C)(O)C(=O)Oc1ccccc1)N(C)C.n12cc(nn1)CC1CN(C1)C2=O C1(CNC(C=C(CCC)C)=O)CC2CCC1N2C(C1(OC)CCS(=O)(=O)C1)=O Cc1ncnc(C(=O)NC2(C(N3CC(O)(CO)C3)=O)CC(O)C2)c1C c1(CNC(C2CCN(C(C)C)C2c2ccccc2)=O)nc2ccc(C#N)cc2o1 C(CCCC(=O)N1CCN(C2CCCN(C(=O)C(C)CSC)C2)CC1)SC C1(C(=O)NC(CNC(c2c(CC)ccs2)=O)CO)CCc2c[nH]nc2C1 c1(C(N(C)CC2CCCN(C(C3C(OC)CC3)=O)C2)=O)cc2sccc2cn1 N1(C(CCCOCCOC)=O)CC2(CC(CNC(C3CC4CCCC4C3)=O)C2)C1 N1(C(C2CCN(C(C)=O)CC2)=O)CC2CC1CN(C(=O)CNS(=O)(=O)N(C)C)C2 C(=O)(CC(C)CC(=O)NC(C)(C)Cc1nn[nH]n1)OC C1(C)(NC(c2ccccc2)=O)CC=CCC1.CC(C)(CN1CC1=O)c1cscn1 C1(CN(C(=O)C(C)OC2CCCCC2)CC)CCN(C(c2nn[nH]c2Cl)=O)C1 Cc1ccc(CC(=O)NC2(C)CCCN(C(C3CCO3)=O)C2)cc1[N+](=O)[O-] CC1(C)CC2(CC2C(=O)NC2CC(F)(CNC(c3cc(Cl)ncc3N)=O)C2)C1 c1(C(CC)CC)[nH]c(C(=O)NCCn2cc(-c3ccc(Cl)cc3)nn2)nc1CC CC(C)CC(C)(CNC(=O)Cc1cccc(C#N)c1)NC(c1cn(C)nc1Cl)=O CC1CC(NC(=O)C=Cc2ccncn2)CN(C(=O)C(c2ccc(F)cc2)O)C1 C1(CNC(c2c(C)nc[nH]2)=O)CN(C(=O)C=C2CCC2)CCC1(C)C N1(C(C(C)(C)C2CCOC2)=O)CCC(O)(CCNC(=O)COC2COC2)CC1 c1(OC)ccc(C)cc1C(N1CCC(O)(CN(C)C(C2CC(OC)C2)=O)CC1)=O C(=O)(C(CC(F)F)N(C)C(C1CC(C)CO1)=O)N1CCC(C(CC)C)CC1 O=C(CC(=O)NCC(C1CCCC1)SCC1CC1)NCC(=O)NC1CC2CC2C1 c1(C(=O)NC(CNC(c2ccc(Br)o2)=O)C2CC2)ccnc2ccnn12 Cc1cccc(CC(=O)N(C2CCCC2)CCNC(C2C(C)CC2C)=O)c1C c1(N2CC(CC(C)NC(c3ccc(Cl)o3)=O)C2)ncc([N+](=O)[O-])cn1 C1(CCNC(C(C=C)C)=O)CC(OC)CN1C(c1cc(C)c(C)s1)=O c12ccc3c(ncn3c1)NC2=O.C(C(C)(C)C)NC(C=CC=CC)=O c1(OC)ccc(CC(=O)NC2CC(F)(CNC(=O)CN3CCCCC3C)C2)cc1 c1(-n2ncc(C(N3CC(OCCNC(C(CC)O)=O)C3)=O)n2)cccc(Cl)c1 C(=O)(CCC(=O)NCC1CC1CNC(c1cc(Cl)ns1)=O)N(CC)CC CCCC(C)CCN=c1[nH]c(=NC(C)c2ccc(CC)s2)[nH]c2ccsc12 N1(C(CN(C)CC)=O)CC(C(=O)Nc2c(C)cc(Br)cc2F)CC2OCCC12 c1(SCC(N2C3CN(C(C4CC(OC)C4)=O)C(C3)C2)=O)ncnc2[nH]cnc12 c1(CNCc2nc(-c3c(O)ncc(Br)c3)sc2)cnn2c1CCCC2 C(=O)(C1CCc2ccc(Cl)nc21)N1CC(N(C(CCOCC#C)=O)C)C(O)C1 Cc1cccnc1CNC(C1CCC(NC(C2CCC2)=O)C1)=O O=C(CS(=O)(=O)C1CCCC1)NCCCC1CCCCN1C(c1ccc(Cl)[nH]1)=O CC1(C(=O)NCC(CNC(c2ccoc2Cl)=O)CO)CCC(F)(F)CC1 Cc1cc(Cl)ncc1CNC(C1(c2cccc(OC(F)F)c2)CC1)=O c1(CC(N2C(C)CC(NC(C3CC3(C)C)=O)C2)=O)ccc2ocnc2c1 CCCCS(=O)(=O)CC(=O)N1CC(NC(c2ccc(CCOC)cc2)=O)C(F)C1 CN1CC=C(C(=O)N2CCC(C3CC3)(CNC(c3ccc([N+](=O)[O-])cc3)=O)C2)C1 c1(OC)cc2c(cc1OC)CCN(c1cc(=O)c(O)nn1-c1ccccc1)CC2 c1(C(=O)NC(C)CC(C)NC(c2cc[nH]c2C2CC2)=O)c(F)ccc2occc12 C1(C(N(C)OCc2ccccc2)=O)CC12CCN(C(=O)C=Cc1ccncn1)C2 N1(C(C2(C)CCC(C)C2)=O)CCC(CO)(NC(=O)CCC2CCCCO2)CC1 C1(NC(C2C3CCC(C3)N2C(C2CC2Cl)=O)=O)CCCC(F)(F)C1 c1(C(=O)NCC2(C)CN(C(c3csnn3)=O)CCO2)cnc2n1CCOC2 C(CCCC(F)(F)F)NC(C)C(C)(C)c1cn(CC)nn1.C(=O)C(F)F c1(CC(N2CCC(CNC(C(CC=C)OC)=O)C2)=O)ccc(F)cc1C CC1CC2(CCN(C(=O)CNC=O)CC2)CN1C(=O)CC(C)(C)CN(C)C c1(OC)cc(C(=O)N(CCC(=O)NC(C)Cc2ccccc2F)C)ccc1Cl c1(NC(CN(C(COC)(C)C)Cc2nc(C)no2)=O)ccc([N+](=O)[O-])cc1 C12(NC(C=CC=CCC)=O)CCCC1N(C(c1ccnc(OC)c1Br)=O)CCC2 C(CN=c1[nH]c2c(c(=NCCCn3cnnn3)[nH]1)CC(C)CC2)N1CC=C(C)C1 C12(CNC(c3nccc(COC)c3)=O)CC(CO1)N(C(=O)CC1CC3CC3C1)C2 C1(C(=O)NCC(CC(C)C)(C)NC(=O)CCNS(C)(=O)=O)CCCCN(C)C1=O CC1CC(C(=O)NC(C)(C)CN(C(=O)Cc2cn(CCO)nn2)C)C(C)O1 C1(C(=O)NC(CCCC)CC)CC12CCN(C(=O)C(C)(C)C1CCOC1)CC2 N1(C(C2(CCC)CC2)=O)CCOC2(CCCN(C(C3CC3F)=O)C2)C1 CC1CC(NC(=O)C(=O)Nc2ncc[nH]2)CN1C(c1cc(Cl)ccn1)=O N1(C(Cn2cnc(=N)[nH]2)=O)CCOC2(CCC(NC(C3CC=CCC3)=O)CC2)C1 N1(C(CC(CC)N(C)C(c2cncc(OC)n2)=O)=O)CCC(C)(C2CC2)C1 CON1CC(C(=O)NCCCN(C(=O)CCn2cc(C)cn2)CCO)CC1=O C1(CC(N2CC(CCC=C)(C(N3CCC3C(N)=O)=O)C2)=O)COCC(C)O1 C(=O)(CC(C)(C)O)NCCOCCCNC(C(c1nc(C)sc1)=O)=O CC1(CC(=O)NCCCO)CCN(C(=O)CCc2ccccc2O)C1 CC1=C(C(=O)NCCCCCC(=O)NC(C)CCO)COCC1 c1(CC(=O)N(CC(C)NC(C)=O)CC)cc2cccnc2nc1C C1(C(=O)NCCC(CNC(=O)Cc2cccc(O)c2)O)Cc2c[nH]cc2S1(=O)=O Cc1cc(-c2nc(C(N3CC(=O)NCC3C(=O)O)=O)cs2)cc(C)c1 C(C(CC(C)C)NC(c1cc(-c2ccccn2)ns1)=O)NC(C(C)(C)OC)=O N1(C(CSCC)=O)CCC(C(C)(C)C)(CNC(C2C(CC(F)(F)F)C2(C)C)=O)C1 N1(C(C(CC)n2cncn2)=O)CCC(C)(CCNC(C2CC(CC)=NO2)=O)CC1 C1(NC(c2cc(C)ncc2)=O)CC2CC1CN(C(c1cc(C)c(Br)o1)=O)C2 c1(NC(C2CCC(=O)N2)=O)cccc(-n2cc(C(=O)O)nn2)c1 C1(CNC(=O)NC(C)CCc2ccccn2)CCC(N(C)C)CC1 O=C(C#CC1CCCC1)NCC1CC2(CC2)CN1C(c1cccc(CO)c1)=O C1(C)(C(=O)NCC2C(NC(C(C)c3ccsc3)=O)C2)CCCNC1=O Cc1cnc(N2CCCC(CNC(=O)C(C)(O)C3CCC3)CC2)nc1C C(=O)(CCCC(C)CC)N1CCCCC(NC(CCCC)=O)C1 N1(C(C(CNC(c2ncc(CC)cn2)=O)(C)C)=O)CCCN(CC)CC1 c1(C(C)O)ccc(S(=O)(=O)N2CC(NCC3CCCO3)CC(C(C)C)C2)cc1 CC1(C)CN(C(=O)CC2C=CC(NC(C3(CO)CC3)=O)C2)CCO1 CC1=NOC(CC(=O)NC(CNC(=O)CCC2CCCOC2)C2CC2)C1 C1(C(=O)NC2CC(NC(COc3ccn(C)n3)=O)CC2O)CC(=O)NC(=O)C1 C12(C(N3CC(F)(CNC(C4(COC)CCCCO4)=O)C3)=O)CCC(C)(C1)OC2 c1(CC(=O)NC(C(=O)NCCc2cscn2)C2CC2)cncnc1 N=c1cc[nH]c(=NCCCC2CCCCO2)[nH]1 c1(C(C)=O)ccc(C=CC(=O)NC2CN(C(=O)Cc3n[nH]c(C)n3)CC2C)o1 CC(CN(C)C)CCC(=O)NC(C1(O)CCN(C(=O)C2=CCCCO2)CC1)C C1(NC(=O)CCCOc2ccc(F)cc2)CCN(C(=O)C(F)OCF)CC(O)C1 Cc1ccc(OCC(=O)NCCC2(NC(c3c[nH]nn3)=O)CC2)cc1 C(c1cc(C)cc(C)c1)=CC(=O)NC1C(NC(C2(OC(C)=O)CC2)=O)COC1 Cc1nc(NCCCOCCNC(C2CC3CCCC23)=O)cc(C#N)n1 c1(C(=O)NCCC(C)NC(=O)C2=CCOCC2)ccc2cnccc2n1 C1(C(=O)NC(C#C)CC)CCN(C(c2cnc(C)cc2C)=O)C12CC2 C(C(C)(C)C(=O)NCC(C)N(C)C(C1CC(=O)N(C)C1)=O)OC(C)C C1(NC(c2nc(C(C)OC)sc2)=O)CC2CC(NC(=O)C(C)(C)C(N)=O)C1C2 N1(C(c2ncc(Br)s2)C(=O)NCCCOC)CCS(=O)(=O)CC(C)C1 N1(C(c2cccc(CSC)c2)=O)CCN(C(=O)C(C)n2cccn2)CC1C N1(C(CCC)=O)CCC(C(=O)Nc2cccc(NC(C3CCC(O)C3)=O)c2)CC1 C(=O)(C1=C(C)CC(C)(C)CC1)NCC1N(C(c2c(OC)ccc(F)c2)=O)CC1 N#Cc1cnn(CC(N2CCCOC(CNC(=O)CCn3ccnn3)C2)=O)c1N c1(CCC(=O)NCC(C)N(C(=O)CCSC(F)(F)F)C)nnc(C(F)F)o1 c1(CCC)cnc(N(C(C2CNCC(O)C2)=O)C(c2ccnc(F)c2)C)nc1 c1(C(N2CCC(CN=c3[nH]nc(C4CC4)s3)(C)C2)=O)ccc(F)c2ccccc12 CC(C)(CC(=O)N1CC=C(C(=O)NCC(C)(CO)CO)C1)C(F)F C1(NC(CCCCC#C)=O)CN(C(=O)C(n2nccc2C)C)C2CCCC12 C1(C(N(CCCCC=C)C)=O)CC(=C)CCN1C(=O)C(C)OCCOC(C)=O CC1CCc2nc(C(c3cccnc3OC(F)F)NC(=O)NC3CCC3)sc2C1 CC1(C)CCC(O)(C(=O)NC2CN(C(=O)CC(C)(C(F)F)N(C)C)CC2O)CC1 C(=O)(CCC1=CCCCC1)N1CC2CC(NC(C34OCC(CC)(C3)C4)=O)CC2C1 Cn1c(C(N2CC3C(NC(=O)CC4(n5cncn5)CC4)C3C2)=O)ccc1[N+](=O)[O-] CC1CC(CNC(=O)CONC(C2CC(=O)C23CCC3)=O)CC(=O)N1 C(=O)(C(CC)C(=O)NCCCOCCN(C(=O)COCCF)C)OCC.CCS C#CC1CCCC(CNC(=O)C(CC=CC)NC(=O)Cc2ccc(F)cc2)C1 C1(NC(C2(C(=O)OCC)CC2)=O)CCC(NC(c2cncc(C)n2)=O)CC1 C1(C(N2CCOC(C3CN(C(c4ccc[n+]([O-])c4)=O)C3)C2)=O)CC(C2CC2)=NO1 c1(C(N2CCC(C(C)(C)NC(C(C)=C(CC)C)=O)C2)=O)ccnc(C)n1 n1(CCCC(N2CCCC(F)(CNC(CC(C)F)=O)C2)=O)cnc2ccccc12 C(=O)(CC(CC=C)NC(c1ccccc1CC#N)=O)NCCCC=C c1(C(=O)NC2C(C(=O)NCc3cn(CC)nc3)CCC2)ccc(C)n1C CN=c1cc(C(=O)NC(CC(C)C)C(=O)NCC(O)CC(C)C)cc[nH]1 CCC(CC(=O)NC1CN(C(c2ccc(C(C)C)c(C)c2)=O)CC1(C)C)C(F)F c1(C(=O)NC2C(CNC(=O)CC(=O)Nc3nccs3)C2)cc2n(c1)CCSC2 C(=O)(C(C)(C)CS(N)(=O)=O)NC(C)C(N1CCC(c2ccco2)C1)=O C1(C(=O)NCC(CC)NC(=O)CCOCCOC)CCC(C(N)=O)C1 C1(NC(CSCCCC)=O)CCN(c2nc(CC)nc(C)c2OC)CC1(C)C c1(C(N(CCC(O)CO)C)=O)ccc(N)c(F)c1F Cc1nc(C(N2CC(CCNC(=O)Cc3ccccc3Br)C2)=O)nn1C OCCC(N=c1nc(N2CCCc3c[nH]nc3C2)c2c([nH]1)CCS2)C1CCC1 c1(C(N(CCNC(C2(OCC)CCCC2)=O)CC)=O)ccc(Cl)c(F)c1O C(=O)(CC(F)(F)C(F)F)N1CCCC(CN(C(=O)CCN(S(C)(=O)=O)C)C)C1 CC(C)C(F)(F)CC(=O)NC1CC(CO)N(C(=O)CCn2cccc2)C1 Cc1[nH]c(=N)nc(O)c1CCC(=O)NC(C)CNC(c1cc2ccncc2o1)=O C1(C(=O)NCC2(N(C)C)CC2)(COC)C=CCN1C(c1cc(=N)[nH][nH]1)=O Cc1cc(C(=O)N(CC(=O)NC2CCSC2)C)cnc1O c1(C(C)C)cnc(C(N2CCC(C(C)(C)O)C2)=O)s1 N1(C(C(C)OC(C)(C)C)=O)CCN(C(C2CC=CCC2C)=O)CC(C)(F)C1 N1(C(C(F)=CC)=O)CCC(O)(C(C)NC(=O)C(C)Oc2cc(Cl)cc(Cl)c2)CC1 c1(C(=O)NCC2(OC)CN(C(C(CC)C(F)(F)F)=O)C2)c[nH]c(=N)c2[nH]ccc12 c1(C(C(=O)NC2CCCCC2)N(C)CC2CCSC2)cnc(Cl)cc1 CCC(CC)CCC(=O)NCCC1CCCN(C(c2cc(CO)[nH]n2)=O)CC1 c1(C(N2CC(O)(CN(C(=O)CCOCC3CCC3)C)C2)=O)ccc(C(F)F)cn1 c1(C(=O)NC2CCN(C(=O)Cc3csc(Cl)c3)CC2CO)cnc2n1CCOC2 C(=O)(C(C(=O)N1CCC(Cc2ocnc2C(=O)OC)C1)n1cccn1)OC N1(CC(=O)NCC(=C)CCNC(=O)C2=CC(C)(C)C2)C(=O)NC(C)(C2CC2)C1=O CCCN=C(NCC1CC12CC2)NCCOc1ccccn1 C(=O)(C(C)C(O)C(C)CC)N1CCC(CCNC(COCCC#C)=O)CC1C N1(C(c2nc(OC)oc2)=O)CCC(CNC(=O)C(C)c2ccsn2)C(F)(F)C1 Cc1ncc(C(=O)NCC2(CNC(c3n[nH]c(C)c3O)=O)CCOCC2)cn1 N1(C(CN(C)C)=O)CC(F)(F)CC1CCNC(C1CC(O)C1)=O N(C(=NCCCOC)N1CCCC(C(F)(F)F)CC1)C1CC(OCOC)C1 C#CCCCCCCCNC(C1CC(CCNC(=O)CC(C)C(F)F)C1)=O N1(C(c2c(C)cccn2)=O)CCCC2(NC(=O)CCOCCOCCO)CC2C1 C1(O)(CCNC(=O)Cc2nc[nH]n2)CCN(C(=O)C2=CCOC2)C1 C(CCCC(=O)NCc1cc(C(=O)NC2CCCC2O)ccn1)OC CN1CC(NC(=O)C(F)C2CC(CNC(=O)CC3CCOCC3)C2)C2(CC2)C1 c1(CCC(=O)NC2(C)CCN(C(c3c(C)coc3)=O)C2)ccc(F)cc1Cl N1(C(=O)NC)CCC(C(=O)NCC(C)CN(C)C(C2CCCO2)=O)C1 C(=O)(C1CCCn2cnnc21)N1CC(=O)N(Cc2ccn3cnc(C)c3c2)C1=O C1(CNC(c2c(F)cccc2F)=O)CN(C(c2cccs2)=O)CC12CC2 c1(C(C)O)ncc(C(=O)NC(CNC(=O)CC2(CO)CC2)CO)s1 N1(C(CC2C(C)(C)C(NC(=O)Cc3cccnc3F)C2)=O)CCOC2COCC12 CC1(C)CCC=C1C(=O)NC1CN(C(c2cc(Br)sc2Cl)=O)CC12CC2 c1(-n2c(-c3sc(C)nc3C)nc(CCOC)n2)ccc(Br)cc1C CCC(CC)C(C)C(=O)N(C1(C(=O)NCCCN2CCC2)CCOCC1)C C1(C(N2CC(C)(O)C2)=O)CCN(C(C2CN(C(N)=O)C2)=O)C12CC2 C1(C#N)(C(=O)NCCn2cc(C(N(C(C#C)C)C)=O)nc2)CCCOC1 C1(NC(C(C)C2(O)CCC2)=O)CCN(C(c2cc(C3CC3)n(C)n2)=O)CC1 c1(OCC)oc(C)nc1C(N1CC(CO)(NC(=O)CCCN2CCCC2)C1)=O c1(CC)noc(C(N2CC(NC(c3ncsc3Br)=O)C(C)C2)=O)c1C C1(N(C)C(C2(c3ccccc3Cl)CC2)=O)CN(C(=O)C(F)C2CC2)CC1O CCCC(F)C(=O)NCC1CCCCN1C(c1cncc(NC)c1)=O c1(C(=O)NCC(N(C(=O)CC2(CO)CC2)C)C2CC2)cnc2c[nH]nc2c1 C1(C)(NC(C(COC)(F)F)=O)CCCN(C(=O)CN2CCC(=O)NC2=O)C1 c1(C(N(C)CC2CCCN2C(=O)CCOC2CCC2)=O)c(Cl)ccc(O)c1Cl CCCCC(CC)C(=O)NC1CC=C(C(=O)NCCCCCCO)C1 C1(C(N(C(C)C)CCNC(c2ccc(C(N)=O)[nH]2)=O)=O)CC2CCC1C2 N1(C(c2c(SC)n(C)nc2)=O)CCN(C(=O)Cn2cncc2C)C(C)C1C C1(O)(CC)CCN(C(=O)C(CNC(=O)CCS(C)(=O)=O)CC2CC2)CC1 C(=O)(CS(=O)CC)NC(C(C)NC(c1c(CCC)nco1)=O)(C)C CC1(C)CC(NC(C2CN(C(c3ccc(Cl)o3)=O)CC2(F)F)=O)C2(CCC2)C1 N(C(=NCC1CCC1)N1CCC(C)(C(N)=O)C1)Cc1c(OC)nc(C(C)C)cc1 CC1CN(C(=O)Cc2ccc(I)cc2)CC1n1cc(-c2cccs2)nn1 c1(OCCC(N2CC3C(NC(CN(C)C4CC4)=O)(C3)C2)=O)ccccc1C#N N1(CC(=O)N(C2CN(C(c3ccc(OC)o3)=O)CC2O)CC)CCN(C)C(=O)C1 C1(CC(=O)NCC(CC)N(C(c2c(C)cc(CC)o2)=O)C)OCCCC1(C)C c1(C(=O)Nc2cccc(CNC(=O)CSC(F)F)c2)cc2c(nn1)CCOC2 n1(CC(N2CCCC(C(C)NC(CC(CC)CC)=O)C2)=O)nc2c(n1)CCCC2 CN(CCS(=O)(=O)N=c1cc[nH]cc1)C(=O)Cn1cc(CO)nn1 CC(C(=O)N(C)CCn1ccnc1)NC(=O)C(F)n1ccnc1 C#CCCCCCC(=O)NCCOCCCN(C(=O)C(N1CCCC(C)C1)=O)C c1(C(=O)NCC2CC(NC(c3cnn(CC)n3)=O)C2)c(C)cc(Cl)cc1C c1(C(=O)NCC2(CNC(C3CCCS3)=O)CCC2)cnc2cc(Br)ccn12 c1(C(=O)OC)ccc(S(=O)(=O)Nc2cccc(Cl)c2C)cc1[N+](=O)[O-] Fc1cc(Br)c2cc(CNCCOc3ccccc3F)[nH]c2c1 Cc1ccc(C(=O)NC2CC(O)(CNC(C3CC3c3ccc(F)nc3)=O)C2)nn1 c1(CC)cc(C(N2CCC(O)(CN(C(=O)CC3CC(CC)C3)C)C2)=O)cc(N)c1 CC12CC(NC(c3cccc(Cl)c3Cl)c3ccccc3)(C1)C1(CNC1)O2 c1(C(=O)NCC2N(C(c3ccc(C#N)[nH]3)=O)CCC2)cnc(O)c(F)c1 N1(C(CCC(=O)N(C)C)=O)CCCN(CCNC(c2ccc(Cl)[nH]2)=O)CC1 N1(C(C2N(CCC)CCC2)=O)CCC(C(=O)NCc2nnnn2CC)C1C Cn1cnc2c(C(=O)NC(C)(C)CNC(C34CCCCC3C4(F)F)=O)cccc12 c1(C(N2CC3C(CNC(C=C(C)C)=O)C3C2)=O)ccc(N)c2cnccc12 C(CCC(C)C)(C(=O)NCc1sccc1C)NC(Cc1c(C)n[nH]c1)=O C1(NC(CCCOC(C)C)=O)CN(C(=O)Cc2nnc(O)s2)CCC1O C1(CC(=O)NC(CSC)C(C)(C)C)CN(C(C)=O)C2(CCC2)CO1 N=c1nc2scnn2c(=S)n1CCS(=O)(=O)C(F)F C1(C(C(=O)N(CCOC)CCC2CCN(CC(F)F)C2)OC)CCOCC1 C1(OC)(CNC(=O)Cc2cn(CO)nn2)CCN(C(c2ccc(SC)cn2)=O)C1 CCCC(O)(CCC)CC(=O)NCC1(C)CN(C(=O)CSC)CCO1 C1(NC(C=C(C)C(C)(C)C)=O)COCCC1C(N1CCCC(C(C)C)C1)=O n1(CC(=O)NC2CCCC2NC(C2CCCN2CC(F)F)=O)cnccc1=O c1(NC(CC2N(Cc3cc(C)[nH]c3C)CCC2)=O)ccc2n[nH]cc2c1 C1(NC(Cc2c(C)noc2Cl)=O)CN(C(c2cc(O)nn2C)=O)CCC1CO C12(C(=O)N(C(C)Cc3ccc(O)cc3)C3CC3)C3CC1C1C(C(CC=C)=O)C3C21 C12CCN(CC1F)C2=O.C1(CC(N)=O)(NC(C(C)OCC2CC2)=O)CCCC1 C(=O)(C1CCCc2scnc21)N(CCCNC(c1nccc(OC)c1)=O)C(C)C C1(C(=O)NC(C)CC(C)NC(C2(C)CC2)=O)CC2(CCCCC2)C1 N1(C(=O)NC2(c3c(C)cno3)CC2)CCC2(C(C3CCC(F)C3)=O)CCCC12 N1(C(c2n(CC)cc(Cl)c2)=O)CCCC2(CCN(C(c3ccccc3O)=O)C2)C1 c1(C(C)(C)NC(C(c2ccccc2Br)NC(=O)OCC)=O)ccnc(O)c1 N1(C(COCCOCC)=O)CCC(C)(C)CC1C(N1CCN(C)C(C)C1)=O C(CC(C(=O)NCC(C)(O)CCO)NC(=O)CC1CCC(=O)NC1)OC Cc1cn2c(CCC(=O)NC3(C)CCN(C(C4CCC45CCC5)=O)C3)csc2n1 CCCCCCC(CC)NC(c1c(OC(F)(F)F)cccc1Br)=O N1(C(C(C)CO)=O)CC2CC2(CNC(=O)C(F)=CCCF)C1 N1(C(COC(CC)C)=O)CC(C2CN(C(C3(CO)CCC3)=O)C2)C1 c1(C(=O)OC)ncc(F)cc1NC(C1CC(O)CCN1C(c1nc(Br)cs1)=O)=O C1(NC(CCCC2(C)N=N2)=O)CCN(C(C23CSC(C2)C3)=O)C1(C)C c1(CNC(C2COCCN(CC(C(=O)OC)(C)C)C2)=O)ccc(C)c(Cl)c1F c1(NC(C2N(C)CCN(C(=O)CN3CC4CC4C3)C2)=O)cccc2c1OCO2 N1(C(C)=O)CC2CC(C(=O)N(CC(C3CCC3)OC)C)C(C2)C1.C12CC1C(=O)N2 N1(C(CCc2cc(C)no2)=O)CC2(CC2)CC1CNC(C1CC(C)(C)CN1C)=O c1(C(=O)NC2CN(C(=O)OCC)C(=O)C2)cc(OC)ncc1-c1cccc(Br)c1 N1(C(COCCOCC#C)=O)C2CCC1CC(N(C(=O)C(O)c1ccsc1)C)C2 c1(C2N(CC(N(OCC(=O)OC)C)=O)CCC2)cccc(C)n1 c1(C(N(C2CN(C(c3cnc(C(C)C)s3)=O)C2)C)=O)ccccc1F C#Cc1ccc(CC(=O)NCCCN(C(C2CCCCNC2=O)=O)CC)cc1 c1(CN(CCC(c2ccccc2)O)C)cc2ccncc2s1 N1(C(CSC)=O)CC(C(=O)NC(C)Cc2cnn(C)c2)CC1(C)C C1(=O)C(C)(O)CO1.c1(C(C(C)Oc2ccccc2)=O)ccccc1F c1(CNCc2c(C)cc(O)cc2)cccc2c(C3=CC(=O)CC(C)(C)C3)cccc12 C1(CC)CN(C(=O)CC(Cl)Cl)CCC1NC(=O)CC1=CCCC1 c1(C2(NC(=O)N(C)Cc3ccsc3Br)C(CC)C2)c(F)cccc1F c1(CNC(N2CCN(c3c(Cl)cccc3Cl)CC2)=O)cccc(F)c1F C(CCCCCC(=O)NC1C2CCC1N(C(=O)C(C)(Cl)Cl)C2)N(C(C)=O)C c1(C(N2CCCC2c2cc(Br)cs2)=O)coc(Cl)n1 n1(CCC)ccc(CNC(C(F)(F)F)C2CC2)c1 C1(C)(COC)CC(NC(=O)CC(C)(C)O)CN1C(c1coc(C(C)C)n1)=O C(=O)(C1CCCc2sccc21)N1C(CNC(CN(CC)CC)=O)(COC)CCC1 C1(CNC(C)=O)CCN(S(=O)(=O)N(C)N(C)C(=O)OC(C)(C)C)CC1 c1(C(N(c2cc(OC)ncn2)CC2CNCCO2)=O)c(F)ccc(Br)c1Cl c1(OC)cccc(NC(C(c2cccc(OC)c2)N(CCOC)CC#N)=O)c1F c1(C(=O)NC(C2CCCN2C(=O)CCOCC2CC2)C)ncccc1F CC(CC(=O)N1CC(F)(F)CC1CNS(=O)(=O)CCC1CCOCC1)CC(C)(C)C c1(C(=O)N(CCN(C2CCCC2)C(CNS(CC)(=O)=O)=O)CCCC)c[nH]cc(C)c1=O C1(CNC(c2ccn(CC)n2)=O)CCC(C)N(C(c2cc(C(F)(F)F)no2)=O)C1 CC1CCC(NC(=O)C(C)N(C(=O)C(O)CC2CCCC2)C2CCC2)C1 N12CC3C(C3C1)C2=O.c1(CCCNC2CCN(C)C2)cccc(F)c1 N1(C(c2ccn(CCNC(CCCCCC#C)=O)c2)=O)CC2CN(C)CC2(C)C1 Cc1c(C(=O)NCC23CC(NC(=O)CN4CCCCC4)(CO2)C3)nn(C)c1N c1(OCCOC)cccc(C=CC(=O)NC2CN(C(C3C=C3C)=O)CC2SC)c1 Cn1cc(C(N2C(C(=O)NC(CC3CCCC3)CO)CCC23CC3)=O)ncc1=O C12(C(=O)OCC)CC(C(F)F)CC1CN(C(=O)NC1CN(Cc3ccco3)C1)C2 n1(CC(=O)NCC(C2N(C(CC(C)F)=O)CCCC2)(C)C)cc(Cl)c(O)nc1=O Cc1nnsc1C(=O)NC(C1(CNC(c2cccnn2)=O)CC1)C C12(C(N(CC(CNC(c3c(C)cno3)=O)O)C)=O)CCC(CC1)C(C)O2 Cc1cc(C(=O)Nc2ccc(-c3ccccc3)s2)cs1.C12(CC)CN(C1)C2=O.CC CCCCCCC(C)CC(=O)N(CC(C)NC(c1ccc(Cl)nc1Cl)=O)C N1(C(CCC=C)=O)CCN(C(C2CCCCN2C(C)=O)=O)C(CC(F)F)C1 N1(C(C(C)NS(CCCC)(=O)=O)=O)C2CCC(C2)C1CNC(=O)COC1CC1 N1(C(c2ccc(C#N)cn2)=O)CCC2(CCCN(C(=O)Cc3cnsc3)C2)C1 N1(C2CCCN(C)C2=O)CCC2(CCC2)C(NC(c2ccncc2)=O)C1 C#Cc1ccc(C(=O)NCCC(C)N(C)C(C2(CSC)CC2)=O)cc1Cl [SH](=O)(=O)C1CC2(CC2c2onc(-c3cc(OC)c(Br)cc3)n2)C1.C(=O)O C(CCCC(=O)NC1CN(C(=O)CN2CCCS2(=O)=O)CC1C)N(C(C)C)C C1(CNC(CC2N(C(Cc3cc(OC)no3)=O)CCC2)=O)NC(=O)OC1(C)C c1(C(=O)NC(CC(=O)OC)C)cc(C)c(-c2c[nH]c(=N)c(C)c2)cn1 C1(NC(CN(C(C(C)C)C)C(C)Cc2cccs2)=O)OCCC1(C)C c1(CC)ccc(O)c(C(=O)NC2CC(C)CN(C(c3cc([N+](=O)[O-])c[nH]3)=O)C2)c1 OC1COc2c(-n3nc(-c4ncccn4)nc3C3COC4(COC4)C3)cnn2C1 Cc1cccc(C(=O)NC2C3CC(NC(C4CN(C)C(=O)N4)=O)CC23)c1 C1(NC(c2ncc(C)c(Cl)c2)=O)CCOC12CCN(C(C1CSCCS1)=O)CC2 C(=O)(CCCC(F)(F)CO)N1CCC(N(C(C2CC3(C2)CC3F)=O)CC)CC1 c1(C(=O)NC2CC(NC(CNC(=O)OC)=O)CC2O)csc2ccncc12 C12(CCCC1)CCC(=O)N2C1CC1.C1(CC(=O)C(c2cnsc2)C)OCCCO1 c1(C(=O)NCC2CC(C)(C)CN2C(C2CCCS2(=O)=O)=O)nc2ncccn2n1 CN1CCC(C)(C(N2CCC(O)(CNC(=O)Cc3nncs3)CC2)=O)C1=O N1(C(CCC(C)(C)NC(C(C)OCCC(C)C)=O)=O)CC2(CO)CCC1CC2 C1(C(N(CC)CC)=O)COCCC1NC(=O)CN(C(=O)COc1cnn(C)c1)C CC1CC(C(N2CCC(F)(CNC(=O)CCc3cncn3C)CC2)=O)CCN1C c1(C(=O)NC2CCCC(NC(C3(C=C)CC3)=O)C2)[nH]c(C)c(C(C)=O)c1C CC1CC(C(=O)NCCC2CCCOC2)N1C(c1cn(C)nn1)=O c1(OCC)ccc(Cl)c(C(N2CCN(C(c3nccn3C)=O)C(CO)C2)=O)n1 Cc1cc(C(c2nnnn2Cc2ccc(F)cc2)NCC(C)(C)F)c(C)s1 C1(C#N)(C(=O)NC2CC(NC(c3ccc(COC)cn3)=O)C(O)C2)CCCOC1 C(=O)(CS(=O)(=O)CCOC)N(C1CCN(C(c2ncc(F)cn2)=O)C1)CCC CCCCC(C)C(=O)NCC(O)CNC(C1(c2ccc(O)nc2)CCC1)=O C12(CNC(c3cc(SC)c(O)cc3)=O)CN(C(C3CNC(=O)N3)=O)CC(F)(C1)C2 C(=O)(C(C(C)CC1CCCC1)NC1COC1)Nc1cccc(OC)c1 N1(C(c2c(CC)scc2)=O)CC(NC(=O)CN2CCCC2CO)CC12CCCC2 CS(=O)(=O)c1cccc(C(=O)Nc2cccc(CN3CCNCC3)c2)c1F CC1CN(C(c2n[nH]cc2C2CCC2)=O)CCN(C(=O)CCC(C)(C)C)C1 C(=O)(C(CCCC#N)COC(=O)C(C)Cc1cnco1)OCC C(=O)(CC1C(=O)Nc2ccc(C)cc21)N1CC(NC(C=C(C)C)=O)CC1(C)C c1(C2(C(=O)NC3C(CNC(C(F)=CCC)=O)CC3)CCC2)ccccc1Br c1(C(N2C(CCNC(CCN(CC)CC)=O)COCC2)=O)cccc(O)c1F Cc1cccc2cc(C(=O)NC3(CCNC(=O)C(O)C4CCCC4)CCC3)oc12 c1(OC)c(F)c(C(N2CCC(C(=O)NCc3ncccn3)C2)=O)cc(F)c1F C1(C(N2CC(C(C)NC(=O)CCCc3nncn3C)C2)=O)CCS(=O)(=O)C1 C=CC1(NC(c2nnnn2CCOC(C)(C)C)C2CC2)CCCCC1 c1(C(N2CC(CNC(C(C)C=Cc3ccccc3)=O)C2)C)c(F)cccc1F c1(CCC)cc(C(=O)NC2(CCNC(=O)C(C)CC3CCC3)CC2)n(C)n1 c1(C(N2CCN(C3CN(C(c4ccsn4)=O)C3)CC2)=O)n[nH]c2c1CCCC2 C(CC(C(=O)N1CCOCC1CO)NC(=O)C(C)OCCOCC)=CC N1(C(C(CC)OCC)=O)CCC2(CC1)CC(CNC(C1CC(CC)(CC)C1)=O)C2 C1(NC(C(C)NC(CC)=O)=O)CCC2(CC1)CC2NC(=O)CCOC c1(CC(=O)NC2CN(C(C(F)OC)=O)CC2C)c(C)cc(Br)cc1C C1(C(N(CCOCCCN(C(=O)CCCN2CCCC2)C)C)=O)CCC2CC12 C1(NC(C(C)OCC=C)=O)CCN(C(=O)Cc2ccc(Cl)c(C)c2)CC1O c1(C(=O)NCC2C(NC(C3C(C)C3)=O)CCC2)cccc2cnccc12 C1(C(N2C(C(C)(C)C)C(NC(=O)CCCC3CC3)CC2)=O)CC2CC(O)C(C1)C2 c1(C(=O)NC2CN(C(C3(O)CCC(C)CC3)=O)CC(C)C2)cc2cccnn2c1 c1(C(N(C(CC)C)CC)=O)cc(CNC(c2ccc(CO)nc2)=O)nn1C N1(C(c2c(C)nc(C)o2)=O)CCC(C)N(C(=O)CN2CCSCC2)CC1 C1(CCC)C(=O)NCCN1C(=O)C(C1CC(OC)C1)N(CC)CC C1(C(=O)NCC2(C)CC(O)C2)(CC)CCN(C(=O)CC2CCOCC2)C1 CC(C)CC(C)C(c1nnnn1CCC1CC1)NCCCc1ncn(C)n1 N1(C(c2[nH]c(CC)c(Cl)n2)=O)CCC2(CC1)C(OC)CC2NC(=O)C=CCO N1(C(CC2CC(OC)C2)=O)C2CCC1CN(C(c1conc1C1CCCC1)=O)C2 O=C(C1=CCCCO1)NCC(CC(=O)N1CCC1CN=[N+]=[N-])C1CCC1 C1(CNC(COCC#C)=O)CN(C(=O)Cc2cccc(C(F)(F)F)c2)CC1O CC1=C(C(=O)N(C2CCOCC2)Cc2cc(N)c(F)cn2)CCC1 N1(C(C2C(CNC(CC(=O)OCC)=O)OCC2)=O)CCN(C)CC1C N1(C(C(CC)O)=O)CCCN(C(=O)COCc2ccnn2C)CC1 C1(C(=O)NC(C)CC(F)(F)F)(OC)CCN(C(C2CC2C(N)=O)=O)C1 Cc1ccc(C=CC(N2CCC(NC(c3cnn(C)c3C)=O)C(O)C2)=O)cc1C CCCC(CCC)CC(=O)N1CC(O)CCC1C(=O)NCCOCCO C1(CNC(CC=CC(C)(C)C)=O)CC(NC(=O)CC(=O)N(C)C)C12CCC2 N1(C(C(CC=CC)NC(=O)C(C)NC(N)=O)=O)CC2CCC2(CO)C1 C(=O)(CCCC(C)=O)NCCCCC(C)NC(CCC(=C)Cl)=O CC1CN(C(=O)CC2CN(C)C2)CCC1N(C)C(c1cn(CC(F)F)cn1)=O N1(C(C(C)(C)CO)=O)CC2(C1)SCCC2NC(=O)CSCc1cscn1 C12(NC(c3[nH]c4cc(C)sc4c3)=O)CCOCC1CN(C(C1(C)CC=CC1)=O)C2 N1(C(Cc2c(C(C)C)con2)=O)CCC2(C1)CN(C(=O)Cc1ccnnc1O)C2 CC1CC(NC(=O)C(=O)NCC(F)(F)F)CN1C(=O)CC=C(Cl)Cl C#CCC(C(=O)N(C)CC1CCN(C(=O)COc2cccnc2)C1)C1CC1 C(C(C)(COC)C(=O)NC(CC(=O)N1CCS(=O)CC1C)C(C)C)OC C1(S(C)(=O)=O)(C(=O)NCC(C)N(C(=O)C(C(C)(C)C)NC(N)=O)CC)CCCC1 CCCCCCCC(=O)N1CC2CC1C2NC(c1csc(C(C)OC)n1)=O C1(C(=O)NC2C(CNC(C3C(OCC)CC3)=O)CCC2)CC1C1CCC1 C(=O)(C(CC(CC)CC)N1CCOCC1(C)C)NCC(=C)C c1(N2CCC(SC)CC2)ccc(S(=O)(=O)NN(C2CCCCCCC2)C)c(Br)c1 C(=O)(C1=C(F)CN(C(=O)C=Cc2cnccn2)CC1)N1CCC(C(C)C)CC1 C(CC1CCCC1)(C(=O)NCC(C)CNC(C1CN(C(N)=O)C1)=O)OC c1(C(N2CCCC(CN(C(C(CC(C)C)F)=O)C)C2)=O)cccn2[nH]c(=N)nc12 C1(CC)CN(C(=O)Nc2oc(C)nc2-c2noc(C(C)(C)C)n2)CCC1(F)F C1(O)(CN(C)C(C2CCOC2)=O)CCN(C(=O)CSCc2csc(=N)[nH]2)CC1 C1(C)(C(N2CCC(N(C(C(C)OCCCC)=O)C)CC2)=O)CCCCNC1=O Cc1cccc(C(N2CCC(C)(C)C2CNC(=O)Cc2ccn(C(C)C)n2)=O)c1Cl N1(C(C(C2CCOCC2)OC)=O)CC2C(CNC(c3cccn3C3CC3)=O)C2C1 C1(NC(CCC2C(C)C2)=O)CC(O)CN(C(c2cnc(OCC3CC3)cn2)=O)C1 N1(C(c2c(C)c[nH]c2)=O)CC2CCC(C1)N2C(=O)CSc1cccs1 C1(CCC)CN(C)CCC1C(=O)Nc1ccc(Cl)c(F)c1 N1(C(c2cncc(N)c2)=O)CC2(CCN(C(=O)CC3CCC4(CC4)CO3)C2)C1 c1(C(=O)NC2CC(NC(c3cc(CC)cc(C)c3)=O)C2)c(C)cc(C)cc1C N1(C(C(c2c(C)nn(C)c2)O)=O)CCC(NC(=O)C(C)N(C)C)CC1C C1(NC(=O)C(F)=CCCF)CN(C(=O)CCC2CCCCC2)CCC1CO C(=O)(C(C)C(O)C(C)C)NCC1ON=C(C(=O)NCc2ccc(COC)cc2)C1 c1(C(=O)NCC#CCNC(c2nc(C)oc2)=O)cc2cccc(Br)c2s1 C1(F)(C(N(CCC(=O)NCc2nc(C(C)C)n[nH]2)CC)=O)CC=CCC1 CCCCC(C(=O)NCC(C1CC1)NC(=O)Cn1nc(C)oc1=O)NC(N)=O c1(CC(=O)NC(CC)CNC(c2ncc[nH]2)=O)n[nH]c(=N)s1 c1(CNC(CN(C(=O)CCC2OCCO2)C(C)C)=O)ccn(C2CC2)n1 c1(C(C)NC(c2cnc(C)n2C)c2n(CCCOC)nnn2)ccc(OC)cc1 C(=O)(C(C)C(C)NC(C1(CNC(=O)CC2CCC(C)CO2)CC=CC1)=O)OC c1(C(=O)OC)ccc(CNC(c2cnn(C)c2Br)c2nnnn2C2CC2)c(Br)c1 C#CCCC(O)C(=O)N1CCC(C(C)(C)NC(=O)CNc2ccc(Cl)cc2)CC1 c1(C(N2CCC(O)(CCNC(CCOCC)=O)C2)=O)cccc(F)c1CC N1(C(CC)C)CCN(C(=O)CC2CC2CNC(=O)C2=CCSC2)CC1 C1(C(=O)NCC(C)NC(=O)CSc2nnc(S)s2)CCN(C)C(C)C1 N1(C(C2N(C(C(C)C)=O)CCCC2)=O)C2CCC1CN(C(=O)C1=COCC1)C2 C(=O)(C(CNC(C1(F)CCCC1)=O)CC1CC1)NCC(C)(C)OC Cc1cnc(C(N2CCN(C(=O)C(C)(F)F)CC2CC(F)F)=O)cc1Cl C1(CC(=O)OC)CC(C)N1C(=O)C(C)CN(C(=O)Cc1ccsc1)C Cc1ccc(-n2cc(C3(C)CCN(C(=O)Cc4nnc(C)o4)C3)nn2)cc1C CCCC(C)C(=O)NCc1ccc(C(=O)NCc2c(C)noc2C)cn1 C1(C(N(CCN(C(=O)CC2CC3(CC3)CO2)CC)CC)=O)CCCC12CC2 C(=O)(C(C1CC1)OCC1CC1C)NC.C(=O)(C(C)=CCN)C(=O)CNC(=O)N C1(C)(C(N(CCCC)CCCC)=O)CN(C(c2nc(C)sc2C)=O)C(C)(C)C1 C(=O)(C1=CCC(NC(=O)CCCC2CC2)C1)NC(CC)Cn1cncn1 N1(C(C2CCC(CNC(=O)CC(C3CC3)C3CC3)O2)=O)CCOC2CCCCC12 c1(OCC)cccc(C(C)(C)C)c1O.C123C(C4CC1C2C4)NC3 n1(-c2n(CC)ccn2)nc(C(F)F)nc1-c1cc(C2CCOC2)c[nH]1 c1(C(N2CC(n3cc(C4CCC4)nn3)C2)=O)ccc(O)c([N+](=O)[O-])c1 CC1CC2(CCCCN2C(=O)OC(C)(C)C)O1.C1(C)CCN(C)CCN(C)N1 N1(C(CSc2c(C)ccc(C)c2)=O)C2CCC1CN(C(=O)CCS(C)=O)C2 c1(OC)ccc(CCC(=O)NC2CC2NC(c2cn(C)nc2Br)=O)cc1 C(#Cc1ccccc1)CN=C(NCC1CCCS1)NCC1CCCSC1 C(=O)(C#CC1(C)CCCO1)NC1C(C(=O)NC(CC=C)CC(F)F)CC1 Cc1cc(C(=O)N(CC(=O)NC(C2(O)CCCCC2)C)C2CC2)cnn1 N(C(=NCCOC(F)(F)F)NCCN1CCCS1(=O)=O)CCOCC=C c1(CNC(C2C(NC(c3c(C(C)C)ocn3)=O)COC2)=O)ccc(O)nc1 N(C(=NCCCF)NCC(C)C(F)(F)F)CCc1ncc(C)nc1 C#Cc1ccc(C(N2CCC(=C)CC2C(N2CCC(F)(C(N)=O)C2)=O)=O)c(C)c1 C#Cc1cc(NC(=O)CCCCCNC(c2c(C)cnn2CC)=O)cc(F)c1 c1(OC)nscc1CN1CC(c2c(C(=O)O)con2)C1.C1(=O)C(C)OCCN1.OC C1(CNC(c2c(C(=O)OC)coc2)=O)CN(C(c2csc(Cl)c2)=O)C2(CCC2)C1 N1(C(CS(C)(=O)=O)=O)Cc2ccccc2CC1CC(=O)Nc1ccc(C#N)nc1 C1(NC(c2n(CCC)ncc2)=O)CCC2(CCCN2C(=O)C=CS(C)=O)CC1 CC1(C)CC(NC(=O)Cc2csc(-c3ccoc3)n2)CN(C(=O)CC=C(Cl)Cl)C1 c12cc3c(s1)CCC(C3)C(=O)N(CCC)CCNC2=O.C1(C)(CC)CC2CC2C1 c1(OC)cc(C(=O)NC2CCCC2NC(c2cc(O)nn2C)=O)cc(Cl)c1O c1(C(=O)NC(C)CCCNC(=O)CNC(=O)C(F)(F)F)ccc(Cl)cc1O N1(C(C)=O)CCCC1C(=O)NCCN(CC(F)F)C.C12(CC1)C(=O)N2 CN1CC(OCc2ccccc2)C2(CN(S(=O)(=O)N=S(C)(C)=O)C2)C1 C1(NCC)CCN(C(=O)C(c2ccccc2)NC(=O)CN(C)C)C1.C(C)(C)(C)S Cn1ncc2c(NCC3COCC3F)nc(N3CCC(F)(F)C(C#N)C3)nc12 C1(CN(C(C2CC(C)C2)=O)C)CCCN1C(=O)CC(C)c1ccccc1 C=CCCCCC(=O)NCC(O)CC(=O)N(C1CC1)CC1CC1 C(=O)(C(C)C(F)(F)F)NC1CC(CC(=O)N(C(CC#C)C)C)C1 n1(CC(=O)NC(C)CN(C)C(C2CC3CC3C2)=O)c(=O)n(C)c2ccccc12 Cc1cnc(C(N2CCOC(CNC(c3cnc(O)s3)=O)C2)=O)c(F)c1 C(=O)(C(C(=O)OC(C)(C)C)C(C)C)N(C1CN(C(=O)CCC(N)=O)CC1C)CC C1(NC(C2N(C)C(=O)OC2)=O)CN(C(=O)Cc2ccc(F)cn2)CC(C)(C)C1 C1(NC(C(C)(C)CCNC(c2nncs2)=O)=O)CC12CCCCCC2 n1(CC(C)C)[nH]c(CC(=O)N(C)CCN(C)C(c2cc(Cl)on2)=O)cc1=O C1(C(=O)NCC(C2CC2)NC(c2ccn(CC)n2)=O)(OC(C2CC2)=O)CCCOC1 N=c1[nH]cncc1NC(C1(C(C)(C)C)CCN(NC(=O)CC2CCC3CC23)C1)=O C(C(C)(C)C#CC(=O)N1CC=CC1CF)NC(c1nc(C)sc1)=O Cc1cccc2c(C(=O)NC3CCN(C(c4n[nH]c5c4CCOC5)=O)C3)csc12 Cc1ccc2c(c1)N(C1CC3CC1CN3C(=O)OC(C)(C)C)CC2 N1(C(C(n2cc(C3CCOC3)cn2)=O)=O)CCCC(CNCCN2CC=CC2)C1 N1(C(c2c(CC)ocn2)=O)CC(NC(C2CCCCC2CC)=O)C(SC2CC2)C1 CCC1=C(C(=O)N2CCC3CC3(NC(=O)CC(COC)COC)CC2)SCCO1 C(=O)(C(F)C(=O)NC(CCN(C)C)C(=O)NCCOC(CC)C(=O)NC)OCC c1(C(C(=O)NC(CC)C)N(C2CCS(=O)(=O)C2)C)ccc(F)c(F)c1Br C1(N)CCCCN(N2CCP(C)(=O)CC2)C1.C1(O)(CNC(CC)=O)CCOCC1 c1(C(C(=O)NC(CC)CNC(C2CCC(=O)N2C)=O)(F)F)cccc(Cl)c1 N1(C(C2C(C=C)OCCC2)=O)CC(CNC(c2conc2CC)=O)C2(CCC2)C1 N1(C(c2c(OC)c(C)sc2)=O)CCC12CN(C(=O)C(C)Cc1ccccc1C)C2 c1(C(N2CCCC(CC)(NC(=O)CNC(C)=O)C2)=O)nccc2c(C)cccc12 c1(C(=O)NCC2N(C(c3cc(C)n(C)c3C)=O)C3C(C2)C3)cnc2ccncc2c1 C(=O)(C1=CCCCC1)NCC1C(C(F)(F)F)CN(C(C(CC)C#N)=O)C1 c1(NC(c2c(C)n(-c3ccc(Cl)c(F)c3)nc2)=O)sc2ncccc2c1N C(C(=O)N1OC2CCC1C2)C12C(CN(C(COCCCC)=O)C1)CC2 c1(C2(NCC(c3n[nH]c(=N)s3)=O)CC(OC(=O)CC(F)(F)F)C2)ccc(F)cc1 C1(NC(CSC(C)(C)C)=O)CC(CNC(=O)CCc2cscn2)CC1O c1(C(N2C(C3CCN(C(C(CC)OC)=O)CC3)CCC2)=O)ncn2c1COCC2 C12(N(C)C(C3CC3c3ccco3)=O)CC(C1)N(C(C1CCCN1N=O)=O)C2 Cc1cc(C(=O)NC(C(=O)NCCc2csc(C)n2)C(C)(C)O)cc(C)n1 Cc1c(Br)sc(NC(C2CCCCN2Cc2ccccc2)C)c1C c1(C2(O)CN(C(=O)NC(c3nc(C(F)(F)F)n[nH]3)(C)C)C2)cccc(Cl)n1 C(CCNC(=O)C(c1ccccc1)C)(C(=O)NCC(n1cncn1)O)OC C1(OCC)CCN(C(=O)Nc2ccc(CC(C)C)cc2)CC1C N1(C(C2(OCC)CCC2)=O)CCn2nc(C)c(CNC(=O)C(C)SC)c2C1 C1(CC2CCN(C(C(c3cccnc3)NC(C)=O)=O)C2C)CN2CCN1CC2 c1(OCC(=O)NC2CN(C(C(CCCC)CC)=O)C2)ccc2c(c1)CCCC2 C1(OC)CN(C(c2cccn2C)=O)CC1NC(=O)CCC(c1ccccc1)N(C)C c1(NC(C2CCC(CNCc3cn(C)nn3)CC2)=O)ccc(Br)c(I)c1 C(C(COC)C(=O)N(CC(C)C(=O)N(C1CCSC1)C)C)OC C1(CNC(=NCC)NCc2ccc(P(C)(C)=O)cn2)CC2CCC(C1)S2(=O)=O CC(N=c1cc(C(F)(F)F)nc(Cl)[nH]1)C1CCN(CCC2=CCCCC2)CC1 CC(C)(CCNC(=O)CC1OCCCO1)C(=O)N1CCCC(OC2CC2)C1 N1(C(c2cccnn2)C(=O)Nc2ccccc2Cl)CCC(CO)C(F)(F)C1 N1(C(C2(C#C)CCN(C(=O)CC3(C4CC4)CC3)CC2)=O)CCCN(CC)C(=O)C1 N1(C(c2cc(C(C)(C)C)nn2C)=O)CCN(C(=O)CC2CCCCO2)CC1CF c1(C(N2CCC(C)(CNC(c3ccnc(O)c3F)=O)C2)=O)n[nH]c2c1CCOC2 C1(CC(=O)NCCC(C)NC(c2ccnn3ccnc23)=O)CCn2cncc2C1 C1(C)(CC)C=C(C(=O)NCC2CN(C(=O)CC3(OCC)CCCCC3)CCO2)C1 c1(-c2cn(C3CC(CO)OC3)nn2)ccc(Cl)c(OC(F)F)n1 c1(-n2c(CC3COC(=O)C3)nc(CCCOC(C)C)n2)ccc(Br)c(F)c1 C1(C(=O)NCC(F)(F)C(N)=O)(CC)CCCN(C(=O)CC2CC2)C1 c1(C(=O)NCC(C(C)C)NC(c2ccsn2)=O)cnc2c(Br)cccn12 CCC(O)C(C)C(=O)NCCCCCC(=O)N(C1CCCC1)C C12CCCN(CCC1)C2.CCC(C(=O)NCC=CC(=O)NC)N(c1cc(Cl)no1)CC CC(CNC(C1CC=CC(NC(C2(C)CCCCO2)=O)C1)=O)S(N)(=O)=O C1(NC(CN(C2CC2)CC)=O)CN(C(c2nn(C)cc2C)=O)CC1(C)C S(=O)(=O)(CCC(=O)N(CCCNC(C1CCCC(C)CC1)=O)C1CC1)NC C(=O)(C(C)(CC)C(=O)N1CC(NC(=O)CNC(=O)C2CC2)C(O)C1)OCC CC1(C)CCCC(CC(N2CCCC(O)(CCNC(c3cnc(O)s3)=O)C2)=O)C1 C1(C(C)(C)C)(CO)CCN(C(=O)NC2CC(N3CCC(F)CC3)C2)C1 S(=O)(=O)(c1cccnc1)Nc1c(C(=O)OC)ccc(Br)c1.N12CCCCC1CC2=O c1(C(=O)NC2CC(C)(C)N(C(=O)CCC3CC3)C2)c(F)ccc(F)c1F c1(C(=O)NCC2N(C(CC3CCN(C)C3)=O)CCOC2)ccc2c(cnn2C)c1 CC1CN(C(c2ccc3c[nH]nc3c2)=O)CCCN1C(C1CCOC1=O)=O Cc1cc(C(=O)NC(C(=O)NCC(C)CF)C2CCOC2)n(C)n1 C1(NC(C)=O)CCCCCC1NC(c1cc(C)ns1)=O.C12CCN(C1)C2=O C(CCN=C(NCc1cccc2cc[nH]c12)NCC(c1cc(C)oc1C)O)SC c1(C(=O)NCC2C(NC(=O)Cc3ccncn3)CCC2)ccc(F)cc1[N+](=O)[O-] C1(OC(N(C(=O)C(C2CC2)C2CC2)C2C(C)C2)=O)CC(N2CCCC2)C1 C(C(C)C(C)C(=O)N1CCN(CCN(C)C(c2ccc(F)cn2)=O)CC1)OC CCCC(CC(C)C)C(=O)N1CC2(CCC(CNC(C3CCCOC3)=O)O2)C1 c1(C(=O)NCC2CC(NC(C(C(C)C)C)=O)CC2O)ccc(F)cc1[N+](=O)[O-] N1(CC(=O)NCC2CCCC(C)C2)CCc2c(Cn3nccn3)cccc2C1 CN1CC=C(C(=O)NC2CCN(C(=O)CC3CC4CCC3O4)C(C(N)=O)C2)C1 c1(C(c2n(CCC)nnn2)NC(C)Cn2ccnc2C)c(F)cccc1F CCC(Cc1cccc(C)c1)C(=O)NC1(CNC(C2CCC2OC)=O)CCCC1 N1(C(=O)NC(c2c[nH]ccc2=N)C)CC(NCc2ccc(CO)cc2)CC(C)C1 C1(C(=O)NC(c2nccc(O)n2)C)CN(C(C2(C#N)CCCO2)=O)CC1(C)C c1(C(=O)NC2(CO)CN(C(c3c(CCC)occ3)=O)C2)ccccc1P(C)(C)=O C1(C(N(CC=C)CC)=O)CCN(C(=O)C=CCCC(C)C)C1C C1(CC(C)C)(C(=O)NC2CCCC2CNC(=O)Cn2cncn2)CNC(=O)C1 c1(CCC(=O)NC(CC(C)NC(CC2(OC)CC2)=O)C)cccc(Br)c1 Cc1cc(C#N)c[nH]c1=NCC1(NC(=O)CCc2cccc(Cl)c2)CCC1 N1(C(C(C2N(C(C(C=C)OC)=O)CCC2)(C)C)=O)CC(=O)NC(CC)C1 C1(CC(=O)N(C)C)CCCN(CC(N)=O)CC1.c12ccc(cc1)CS2 C1(COC)CN(C(=O)CC2(O)CCCN(C)C2)CCN1C(=O)CCCNC(C)=O CCC(C)(C)C(=O)C(=O)N1CC2C=CC1C(C(=O)NC1CCC1C)C2 Cc1ccc(C(N2CC(C3CC3C(=O)N3CCCO3)C2)=O)c(O)n1 Cc1ccc(CC(N2CC(CNC(c3csnn3)=O)C(C)C2)=O)cc1C CC1CC2(CCN(C(C3C4CC5C(C4)C35)=O)CC2)CN1C(=O)Cn1ncnn1 C12(NC(CC(C=C)C)=O)CC(CNC(C3(C)CC(NC(C)(C)C)C3)=O)(C1)OC2C C1(C(=O)NC2C(NC(c3cccc(CC#N)c3)=O)COCC2)CCC(F)(F)CC1 N12CCC(C1)CC(=O)N(C)C(c1ccccc1)C2.C(CC(N)=O)SCC(=O)OC Cc1[nH]ccc(=NC(=O)c2ncncc2-c2cccc3ccnn23)c1F c1(C(CC)O)nc(C2CC(C(C)(C)C)CCO2)n(CCOc2ccccn2)n1 CCCCC(F)C(=O)NCC1CC2(CC2)CN1C(c1ncc(C(F)F)s1)=O N1(C(=O)C=Cc2cnc[nH]2)CC2CC1CCC2NC(=O)CC1CCOCC1 C1(C)(C(=O)NCC(C2CCCC2)NC(CC(=O)OC)=O)CC2CC2C1 CC1(C(c2nnnn2C2CCOCC2)NCC2CC(F)CN2)CCCOC1 Cn1ccnc1C1CCCC1C(N1CC(C(N)=O)(CNC(c2cc(F)n[nH]2)=O)C1)=O Cc1ccc(Br)c(C(=O)NC(C(C)NC(c2c[nH]nc2C)=O)C(C)C)n1 C12(C(=O)NCCNC(c3ccc(C(C)C)cn3)=O)CCCCC1OCC2 C(CC(C)CCNC(c1cncc(-n2ccnn2)c1)=O)NC(COCCOC)=O CS(=O)c1cccc(C(N2CC3C(NC(=O)C=Cc4ccncn4)C3C2)=O)c1 c1(C(=O)NC(CNC(C(CC(C)C)(F)F)=O)CO)cnn2c(Cl)cccc12 Cc1nc(=NC2CCC3CN(C(c4ccnn4CCF)=O)CC23)s[nH]1 C(C(C(=O)NCC(C)(C)NC(C1(OC)CC1)=O)n1cccn1)COCC Cc1ccc(C)c(CN2CC3(CN(C(c4ccc(CO)o4)=O)C3)C2)c1 C(=O)(C(F)(F)C(C)(C)O)NC1CCC(CCNC(C(C(=C)C)(C)C)=O)C1 C=C(C)C(O)CC(=O)NC1CCC(C)N(C(=O)Cc2sccc2C)C1 N1(C(C2CCCN(C)C2)=O)CCCN(CCNC(=O)CC(C)(F)F)CC1 N1(C(c2cnn(C)c2N)=O)CCN(c2cc(NCCOC(C)C)ncn2)CC1 N1(C(c2c(CCC)n(CC)nn2)=O)CCCC(C)(CNC(=O)C(C)(C)CCC)C1 C(N=c1[nH]c(Cl)ncc1F)C1CCN(C(=O)C=CCn2cncn2)C1 c1(CNCC2(F)CCN(C(=O)CCC3CCCC3)CC2)c[nH]c2ncccc12 C1(NC(Cc2ccc(C)cc2)=O)CCSC12CN(C(c1cnc(S)[nH]1)=O)C2 N1(C(c2c(C)nc(O)cc2)=O)CCC(C)(C)C(C(=O)NOC(C)(C)CO)C1 CN1CCOC(C(=O)NCC2CN(C(c3ccn(C(F)F)n3)=O)CCO2)C1 Cc1cccc(-c2nc(C(=O)NC3COCC3NC(=O)C(N)=O)cs2)c1 C1(C(=O)OC)CC(F)CN(C(C2(OC)CCCCC2)=O)C1 C12(NC(C(CN(C(COCC(N3CCOCC3)C)=O)C)C)=O)CCC(CC1)CC2 Cc1cnnc(O)c1C(=O)NC1CCOC(C(=O)NC2CC(C)(C(N)=O)C2)C1 C1(CNC(CC(CC)C)=O)CN(C(c2cc(C)c(CO)cn2)=O)CC(C)(C)O1 N1(C(CCN(C)C)=O)CCCC1CNC(C1CCOC1)=O c1(C(=O)NCC2CCCC3(CN(C(C4CC4F)=O)C3)O2)cc2nc[nH]c2cc1F C1(CNC(c2c(CC)con2)=O)CC(C(F)(F)F)CN1C(=O)C(F)COCC C1(CNC(C2(C#N)CCC2)=O)CC2(CC(NC(C3C4CCCC34)=O)C2)C1 C1(C(=O)NC2C(NC(=O)CC3CCSCC3)COC2)Cc2ccccc2NC1=O C1(N(C(c2n(CC)ncc2)=O)C)C2CN(Cc3ccccn3)CC12 c1(C(N2C3C(C(=O)Nc4c(I)ccc(C)n4)C(C3)C2)=O)ccc(F)c(F)c1Cl N1(C(=O)Cc2ccc(O)c(Cl)c2)CCC(NC(C(C)NS(CC)(=O)=O)=O)CC1C C1(C(C)NC(=O)Cn2cnc(C(F)(F)F)n2)CN(C(=O)C(O)C2CC2)CCO1 C(=O)(C1=NN2CCC(C)N=C2N1)NCCNC(Cc1c(CC)n(CSC)nc1)=O C1(NC(c2cnc(C)s2)=O)C2CC3CN(C(c4ccccc4Cl)=O)C1C3C2 C1(C(N2CCN(C(CNS(N)(=O)=O)=O)C(CF)C2)=O)COc2ccccc2O1 N1(C(=O)CSC2CC2)CC2(SC)CCC1C2.c1(OC)ccc(N)cc1.C1(=O)C(OC)N1 C1(C(=O)NC2C(NC(CCC(C)OC)=O)COCC2)CC2(CCC2)CO1 C1(CNC(C(C)=C(CC)C)=O)CCCCC1NC(c1ccccc1OCCF)=O C1(N(C(C23CCC(C2)C3)=O)CC)CCCN(C(C2OCCC2C(F)(F)F)=O)C1 c1(C(N2CCN(c3cccs3)CC2)C(=O)NCC=C)ccc(CC)c(F)c1 C1(C=O)CC1C1CCCC1.C12(O)CN(C1)C2=O.C1(OC)C(C(=O)NC2(C)CC2)C1C c1(SC(c2noc(-c3c[nH]nc3-c3cccc(OC)c3)n2)CC)c(Cl)cccc1Cl C=CCC(C)(C)CC(=O)N(c1ccc(C)cc1)CCC(C)Cc1cnn(C)c1 Cc1cc(C(N2CC(CNC(=O)CCCC(C)C)C(F)(F)C2)=O)c(Cl)cc1F C1(C(=O)NCCC(C)CO)CC2CCC(C1)N2C(C1CC1C(=O)N(C)C)=O C1(C(=O)NCc2nc(CNC(C(CC)O)=O)sc2)CCC(=O)N1C N1(C(c2c(CC)c[nH]n2)=O)CC2CCC1CN2C(c1cnc(CCOC)[nH]1)=O C=CC1CCCC(N=c2ccnc(NCc3ccccc3C3CC3)[nH]2)C1 CC(CC(=O)NCC1CCN1C(=O)CNc1ccccn1)N(C)C C(=O)(C(O)CC(N)=O)N1CCC(c2n(CC)nnn2)(C(=O)OCC)C1 C12(NC(CCCC(=O)NC)=O)CCCC1N(C(c1ccnc(S)c1)=O)CC2 Cc1ccc(F)cc1CCNC(=O)NCCN1CCN(c2ccnc(C)n2)CC1 Cc1cn(-c2ccccc2Cl)nc1C(=O)N(CCN(C)C)Cc1ccc(Cl)cc1 N1(C(c2c(CC)nc[nH]2)=O)CC2CCCC(C1)N2C(=O)C(C)OC Cc1c(C(=O)NCC(CC(C)C)NC(C2(C)CCCO2)=O)sc2ccc(Cl)cc12 Cc1noc(Cl)c1CC(=O)NC12COC(CNC(=O)CC(F)(F)F)(C1)C2 c1(C(N2CC(F)(C(=O)NCC(C(=O)NC)C)C2)=O)ccc(C)c(C)c1 C1(CSC)CCN(C(C2CC(NC(=O)CC3COCCO3)C2)=O)C1 N1(C(=O)NC2(C)CCN(CC(=O)OCC)C2)CCOC(CC)(CC)C1 N1(C(c2cccc(S(=O)(=O)N3CCCC(O)C3)c2)=O)CCC(CO)c2ccccc21 N1(C(c2nccc(OC)c2F)=O)CCCC12CCN(C(=O)C=C=C(C)C)C2 C1(CC)CC(C(N2CC(C)(C)C2COC)=O)CCN1C(c1cnn2c1OCC2)=O c1(C(=O)NCC(C)(F)CNC(C2CCCCCCC2)=O)cnc2ncccn12 c1(C(=O)NC2CCCN(C(Cc3c(OC)csc3)=O)C2)cc2ccccn2c1 C=CC(F)(F)C(=O)N1CCC(N(C(c2c(Cl)n[nH]c2C)=O)CC)C1 CC1CCCCCN1CC(=O)Nc1ccc(OC(CNC(C)(C)C)=O)cc1 c1(SCCOC(C2CC(C(F)(F)F)CO2)=O)ncc(C(F)(F)F)o1 N1(CC(=O)NC(C)CCNC(=O)CC2CCCN(C)C2)CCN(C)C(=O)C1 C1(C(=O)NC(C)CNC(C23CC(F)CC(F)(C2)C3)=O)Cc2cc(Cl)ccc2O1 c1(C(N2CCC(NC(C3CCCCO3)=O)C2)=O)cnc2c(c1)CCCC2 N1(C(C2(C(OCC)N)CC2)=O)CC2(CCC(Oc3ncnc4[nH]cc(I)c34)C2)C1.CC c1(C(N(CCCNC(C2CCCSC2C)=O)CC)=O)ccc2c(c1)CCCC2=O N1(C(c2n(CCC)nc(C)c2Cl)C(=O)NC2CCCC2)CCCC2CC1C2(C)C NC1(C(=O)NCc2cn(CCO)nn2)CCC2CCCC12 c1(C(c2n(C(C(=O)OC)C)nnn2)NCCCCC2CC2)ccc(C#N)nc1 N1(C(COCCC)=O)CC2CCCC2(Nc2ncnc3c2CCO3)C1 N1(C(c2cnc(-c3ccccc3)[nH]2)C(=O)NCCCSC)CCOCC1C#N c1(CCCC=C(C)C)cccc(NC(=O)C(C)CF)c1.C12CCCC1C(=O)NC2 C(C(C)C(=O)NC1CC(C(C)O)C1)NC(C(C)OCCCC)=O c1(C(=O)NCC(CNC(=O)CCC(=O)c2cccs2)F)cncc(F)c1Cl CC1CCC(C)(C(=O)NCCCCC(=O)N2CC(C(C)(C)C#N)C2)C1 c1(C(N(CC(C)CNC(c2cscc2Cl)=O)C)=O)ccc(N)c2ncccc12 N1(CC(C)C)CCCC(C(=O)N(C2CCCN(C(C3(C(C)(C)O)CC3)=O)C2)C)C1 N1(C(=O)OC(C)(C)C)CCCOC(CNC(C2(C(=O)O)CC(O)C2)=O)C1 N#Cc1cnn(CCNC(C2CN(C(C3CC4C=CC3O4)=O)CCO2)=O)c1 CCC(C)(COC)C(=O)NCC(C)C(F)C(=O)NCC(O)C(=O)OC C(=O)(CCCN=[N+]=[N-])N1CC(C(C)NC(CCc2cccc(OC)c2)=O)OCC1 C1(C)(C(=O)NC(C2CC(NC(c3ccc(OC)s3)=O)C2)C)CCCOC1 c1(C(=O)NCc2cc(C(=O)NC3(C)CCCC3O)n[nH]2)cc2ncccc2[nH]1 Cc1ccc(CN(C2CC(C(F)(F)F)C2)C(=O)C2CC2)c(C(=O)OC(C)(C)C)c1 C12(C(N3CC(Cn4cc(CCNC(C)=O)nn4)OCC3)=O)CC1COC2(C)C C1(C(C)NS(=O)(=O)Cc2ccc(Br)cc2)CN(Cc2ccncc2)CCC1C c1(C(C(=O)NCCCOCC)NC(CCC(=C)C)=O)cc(C(F)(F)F)ccc1F N1(C(C(CC)COC(C)=O)=O)CC2CC(C(C)C)C1C2 N1(C(c2c(C)scc2)=O)CCC(CC(C)NC(C2CCOC2C)=O)CC1 CCCCCCC(C)NC(C1(F)CCCN(C(C2(O)CCCCCC2)=O)C1)=O c1(C(=O)Nc2c(C(N3C4C(C(=O)OC)C(C4)C3)=O)nc[nH]2)c(F)cc(Br)cc1F CC1(P(C)(C)=O)CCCN1Cc1ccc(-c2nn[nH]n2)s1 Cc1cc(Br)ccc1C(N1CCOC(CC(=O)NCC2(C)COC2)C1)=O C(CNC(=O)C(F)OC(F)(F)F)(CCOC)NC(CCN(CCCCC)C)=O C=CCCC(CO)NC(c1cnn(CCNC(=O)CCC2CCC(C)O2)c1)=O c1(OC)ncc(Cl)cc1NC(N1CCC1C1CCCOC1)=O CCC(C)(C#N)C(=O)NCC1C2CN(C(=O)Cc3ccc(OC)cc3C)CC12 N1(CC(C)=CC)CCN(C2CC2)C(C)C1.C(c1ccccc1)=C(C(=O)OC(CC)=O)C CC1Cc2c[nH]nc2C(C(=O)NCCCCNC(c2cc[nH]c(=N)c2)=O)C1 Cc1ccc(F)cc1C(C)NC1COC(c2ccccc2)C1 Cc1c(OCc2ccccc2)cccc1C(N1CSCC1C(N)=O)=O N1(C(CC(=C=C)C)=O)CC2(CCN(C(c3c(OC)ncnc3OCC)=O)CC2)C1 CCC(C)(C#N)C(=O)N1CCC(O)C(N(C(=O)Cc2ncn3c2CCC3)C)C1 n1(C(C)C)cc(C2CC2C(N2CCC2(C)C)=O)cn1 Cc1nc(NC(N2CCC(n3cnc(C(N)=O)n3)C2)=O)nn1-c1nc[nH]n1 CCC(F)(F)CC(=O)NC1CC(C(=O)NCC(C2CC(C)(C)C2)O)C12CCC2 N1(C(C(C)CN(C(=O)C(c2ccn(C)c2)C)C)=O)CCC12CCCOCC2 c1(Cn2cc(CC3CCN(C(=O)Cc4nc(CO)n[nH]4)C3)nn2)ccccc1F N1(C(C(CSC)O)=O)CCCC(CN(C)C(c2cc(C)sc2C)=O)C1 Cc1cnc2nc(C(=O)NC(C3CCOC3)CNC(=O)CC(F)(F)F)nn2c1 C(C(C)(O)CC(=O)NC1CCCC1NC(=O)C(c1ccc(F)cc1)O)OC c1(CC(=O)NCC2CC(NC(C(CC)OC)=O)C2)cccc2sccc12 n1(C(=O)N)nc(C)oc1=O.CCCC(CCC)NC(=O)CCOC(C)C N1(C(c2cc(CC)n(C)n2)=O)CCCC(F)(C(=O)NC2CN(C)NC2=O)C1 c1(C(N2CCC(O)(CCNC(c3c(C)coc3)=O)C2)=O)cnc2[nH]ccc2n1 C(C)(C)(CCC(=O)NC1CCC1(C)C)NC(C(c1ccn(C)n1)C)=O N(C1CC(NC(C)=O)c2ncc(Br)cc21)c1c(F)cc(C(=O)OCC)cc1Br c1(C(=O)NC2CCN(c3cc(OC)ncn3)C2)ccc([N+](=O)[O-])cc1C c1(C(=O)NC(C(=O)N(C)CC2(OC)CCC2)C)conc1C Cc1ncnc(C(=O)NC2C3CCC2N(C(=O)C(C)OCC2CCCO2)C3)c1C C(=O)(CCCC(N)=O)N(CCCCN(C)C(C1CN(C(=O)OC(C)(C)C)C1)=O)C C1(NC(CC(C(F)F)NC(CCC(N)=O)=O)=O)CC12CCCCCC2 N1(C(=O)NCC2N(C(C)C)C(=O)CC2)CCc2ccccc21.C(C(O)CC(F)(F)F)S c1(C(=O)OC)nc(N2CCN(C)CC2CNC(C2CCC(C)(C)O2)=O)ncc1Cl Cc1ccc2c(CC(=O)NCCC(C)(C)NC(c3coc(CO)c3)=O)c[nH]c2c1 c1(N2C(CC)CN(Cc3ccc(C)s3)CC2)ncc2[nH]ncc2n1 Cc1nc(C(=O)NC(C2CN(C(=O)CC(C)(C)CN(C)C)C2)C)c(=O)[nH]c1C C1(C(N)=O)(CNC(C2CC(F)(F)C2)=O)CN(C(=O)CC2CCOC2=O)C1 C#CCCCCCC(=O)NC1CCC1NC(c1coc(-c2ccsc2)c1)=O N1(C(C=Cc2ncc(C)[nH]2)=O)CC2CC(C1)N(C(=O)COc1ccccc1F)C2 Cc1nc(N2CC3CC2CN3C(c2cccc(C(C)C)n2)=O)c2c(n1)CCC2 c1(CC)cc(C(=O)N(C2CCN(C(C3CCS(=O)(=O)N3)=O)C2)C)ccc1C c1(OC)ccc(Cl)c(CN2CC(F)(F)CC2C(=O)Nc2cccc(O)c2)c1F CC1(O)CCN(C(=O)CC2CN(C=O)C2)CC1O.C12CCN(CC1)C2(C)C.C1CC1 C(=O)(C(F)(CNC(=O)C1=CCC(C)CC1)C(C)C)Nc1cn(CCC#C)nc1 C(=O)(C(C)CC(=O)NCC1CC1CC(=O)NC(c1c(C)n[nH]c1C)C)OC c1(C(=O)NC(C(=O)N(C)Cc2nnc(C)s2)CN(C)C)cccc2c[nH]nc12 C1(NC(CN2CC(=O)NC2=O)=O)C2CCC1N(C(c1ncc(C(F)F)s1)=O)C2 Cc1ccc(C(N2CCOCC(NC(c3cc(C(C)C)[nH]n3)=O)C2)=O)c(C)n1 c1(C(=O)NCCC(CNC(C(CCCC)O)=O)O)cccc2oc(=N)[nH]c12 N1(C(C(C)=CC2CC2)=O)CC(CNC(c2oc(CO)cc2C)=O)C(C)C1 c1(C(N2C3CC(NC(C=CCC)=O)C2CC3)=O)c[nH]c2ccc([N+](=O)[O-])cc12 c1(C(=O)NCCCN(c2cn(CCO)nn2)C)cccc2ncnc(O)c12 c1(CC(=O)NCc2ccc(C(C)C)cc2)cccc(Br)c1F C#Cc1cc(C(N2CC(CNC(=O)CSc3cccc[n+]3[O-])C2)=O)cc(Cl)c1 C1(CNC(C(=O)NCc2ccnc(C(F)F)c2)=O)CC2(CCCCC2)C(=O)O1 Cc1cc(Cl)cc(C(=O)NCC2CN(C(=O)Cc3nc[nH]n3)C(C)(C)C2)c1O N1(C(CC(C)(C)C)=O)CCC2(CNC(C3CC3C(F)(F)F)=O)CCCC12 N1(Cc2cccc(C(C)C)c2)CCN(C(=O)C(C)(C)CCl)C2(CC2)C1 C#CC1CN(C(C2CC(=C3CC3)C2)=O)CCN1C(c1cccc(CC)c1)=O C1(NC(C(COC)OC)=O)CN(C(c2ccc(Cl)c(C)c2O)=O)CC(C)(C)C1 c1(C2C(C(N3CC(CC(C)NC(CC(C)(C)OC)=O)C3)=O)C2)c(Cl)cccc1Cl CCCCC(CN=c1[nH]c2cc(Br)cnc2s1)NC(=O)C(C)C1CCCO1 C=CCC(C)(C)C(=O)N1CCC(C(=O)NC(c2nncs2)C)C(C)C1 c1(C(N2C3C(NC(C(CC)n4cccn4)=O)CC(C3)C2)=O)cc2n(n1)CCCCO2 N1(C(C(C)OCCCC)=O)CCOCC1C(=O)NC(C)CC(=O)OCC C(=O)(C1=C(C#N)CCC1)N1C(CCC(=O)NCC2(N(C)C)CCCC2)CCCC1 C1(C2CCN(C(C3CC3Br)=O)CC2)(NC(C)=O)CC1 c1(C(N2CC(CC)CC(C)C2)C(=O)NCCCC)ccc2n[nH]cc2c1 c1(C(=O)NCC2CCCC2N)ccccc1[N+](=O)[O-].C12(NC(=O)C3CC3)CCC1CC2 c1(C(=O)NCC2(NC(CC3C(C)=NOC3=O)=O)CC2)ccc2nc(CO)[nH]c2c1 N1(CC(c2ccc(C(C)C)cc2)O)CCC2(CCCCCC2)CC1 C12CCCN1C(=O)c1csc(n1)NC1C(C1)NC2=O.c1(SC)ccccc1 c1(-c2cn(CCC(=O)OCCCCC(C)N(C(C)=O)C)nn2)ccc(C)cc1Cl C1(CC=C)(NC(C2(CCCF)CC2)=O)CCN(C(=O)CCc2nccs2)C1 Cc1cnccc1-c1cn(C2CC(C(=O)NC3(C(=O)N(C)C)CC3)C2)nn1 C(=O)(C1CCCn2nccc21)NC(C)CCCCNC(C1(O)COC1)=O N1(C(c2c(OC)c(C)cs2)=O)CCCC(C2CN(C(=O)CSC3CCCO3)C2)C1 C1(F)(CNC(C(F)=CCC)=O)CC(NC(=O)Cn2ncc(Br)n2)C1 C1(NC(c2occ(C)c2)=O)CN(C(=O)C(C)OC(C)(C)C)CC12CCOCC2 N1(C(C(C)=O)=O)CCC(C2CC2)C1CNC(c1nc(C)no1)=O c1(C(=O)NCC23C(CN(C(c4cn(C)nc4)=O)C2)C3)cc(F)c([N+](=O)[O-])c(F)c1 C(CC(C)(O)C(=O)N1CC(CCNC(=O)CN(C)S(N)(=O)=O)C(C)C1)OC N1(C(c2ccncn2)=O)CCCCC(N2CCOC(c3ccc(Cl)cc3)C2)C1=O C1(C(N2CCC(C)(CNC(=O)CCC3CC3(F)F)C2)=O)CCCCC(=O)C1 c1(C(=O)NC(CC)CN(C(=O)CCC(C)C)C)ccc(Br)cc1OC N1(C(Cc2ccn(C)n2)=O)CCCC2(CCN(c3nc(Cl)c(C#N)s3)CC2)C1 C(c1ccco1)=C(C)C(=O)N(C1CCN(C(C2CCCN2C(=O)C2CC2)=O)C1)C CCCCS(=O)(=O)CC(=O)NC1CN(C(=O)C(C)(C)NC(C)=O)CC1C c1(C(=O)NC2CC(C)N(C(=O)Cc3cccnc3Br)C2)ccc2c(c1)CCN2 c1(OC)cccc2scc(C(N3CC4CC3CC4CNC(=O)COC3CC3)=O)c12 C(=O)(C1=C(C)S(=O)(=O)CC1)NCC1(CNC(C=CCC)=O)CC12CCC2 CC(C(=O)NNC(=O)CSc1ccc(Cl)cc1)c1nc2ccccc2[nH]1 N1(C(CCN(C(CCC)C)C)=O)CCCCC1CNC(=O)C(CCO)N(C)C C1(C(=O)NCC2C(NC(Cc3ccc(C#N)cc3)=O)C2)CCOCC12CCCC2 C(=O)(CC(O)CCCC)N1CC2C(NC(c3c(SCC)oc(C)c3)=O)C2C1 C1(CCCNC(=O)CCC2CCCO2)CCN(C(=O)CC2CC(CF)C2)CC1 c1(CCC)nc(C(=O)N(C(C)C(=O)NC(CO)C(C)O)C)co1 CC1CC(NC(=O)N(C(c2cccc(F)c2)C)C2CC2)CN1C1CC1 C(C)(C(C(=O)N1CCCC1C(C)(C)C(=O)N1CCC(CN(C)C)C1)N(C)C)OC C1(CCSC)CCN(C(C2(CCNC(c3coc(C(F)F)c3)=O)CC2)=O)CC1 C(c1cnc(O)nc1C)=CCC1ON=C(C)C1 C(=O)(CC(O)(C(F)(F)F)C1CC1)NCCC1C(C)CCCN1C(=O)COCCF c1(CNC(C2C(C(N3CCC(CC(=O)OC)CC3)=O)C2)=O)ccc(F)c(F)c1 c1(C(=O)NC2C(CNC(C(C=C)(C)C)=O)CC2)cc2oc(Br)cc2[nH]1 O(P(=O)(CNCC(C)(CO)NC(=O)OC(C)(C)C)OCC1CC1)CC Cn1nc(C(F)F)cc1C(N1CCC(C(C)(C)CNC(=O)CC2CC2(Cl)Cl)CC1)=O C=C(C)C(CC(=O)N1CC2(NC(=O)CCc3nnnn3C)CCC1C2)OCC c1(C(C)C)cc(=NCC2CC(NC(=O)COC3CCOC(C(C)C)C3)C2)[nH]cn1 N1(C(=O)CN(C2CC2)CC2CCCCO2)CCN(C(=O)CC23CCCC2C3)CC1 CC1CC(NC(C2(C(=O)OC(C)(C)C)CC2)=O)CN1C(C1C2COCC12)=O c1(NC(N2CCC(c3scc(C)n3)C2)=O)ccc2c(C)[nH]nc2c1 CC1CN(C(=O)CC2CCCC3CC23)CC(C(N2CCCC3CC23)=O)O1 C1(CN(C(c2ccc(Cl)n2C)C(=O)NCCCSCC)C)CCc2nccn2C1 CN1CCN(CC(N2CCC(CNC(C3CCCC3O)=O)CC2)=O)CC1 N1(C(C(C)=C2CCCC2)=O)CCC(C)(CNC(c2coc(C(C)(C)C)n2)=O)CC1 n1(CC(=O)NCC2COCCN2C(=O)CSC2CC2)cnc2c1CCCC2 N1(C(c2c(C)cnnc2O)=O)CCN(C(c2cc(C#N)c[nH]2)=O)C(C)CC1C c1(C(N(CC(C)(C)CNC(c2cc(OC)ncn2)=O)CC)=O)cc(Cl)ccc1C c1(C(N(CCCN(C(=O)COCC2CCCO2)C)C)=O)scnc1C1CC1 C1(CCCCNC(C(CC)OCC)=O)CCN(C(=O)C=CC2CCCC2)CC1 c1(NC)ccc(C(N2CCCN(C(c3snc(Cl)c3Cl)=O)CC2)=O)cc1F c1(C(N2CCCC(C)(NC(c3c(CC)noc3C)=O)C2)=O)cccc2nonc12 C12(C(=O)NCC3(C(N)=O)CC3)CC1CCN2C(c1cc(C(F)F)no1)=O C(=O)(CCCC(F)(F)F)N(C)CC1N(C(C(c2ccccc2)OC)=O)CCCC1 C1(NC(COCCCC)=O)CCN(C(=O)C(N2CCC(C)C2)=O)CCC1(F)F C(=O)(C1COc2ccccc21)N1CCN(C(COCCC)=O)CC(O)C1 C(CCCCC(=O)NC1CC(C(N2CCC=C(F)C2)=O)C1)OCC c1(C(=O)NC(CCCC)CNC(=O)CN2CCCC2C)cc2ccnc(Cl)c2[nH]1 n1(CC(=O)OC)cccc1C(=O)NC1COCC1Nc1ccccc1 C1(CC(=O)N(CC(C)(C)NC(c2ccc(=O)oc2)=O)C)CCC(F)(F)CO1 C1(C(C(=O)N(C(COC)COC)C)F)CCN(C(=O)CNS(N)(=O)=O)C1 N1(C(C(C(CC)O)(C)C)=O)CCC(C2(NC(c3cocc3C)=O)CCC2)CC1 Cc1nsc(N)c1C(N1CCC(C(C)NC(=O)CC2CCC(C)(C)O2)CC1)=O N1(C(C(=O)N(CCc2ccccc2)CC)=O)CCCC(CO)C1 CC1(C)CCC(C(=O)NCCC2(O)CCN(C(=O)C=Cc3cn[nH]c3)CC2)CO1 C12(C(N(CCCC)CC)=O)CC1CCN2C(=O)CCn1cccc1 C12CCN(CC1C)CC1(CCCC1)N2.C(C)(C)(C(=O)OC)OC C(CCCCC(=O)NCCCOCCNC(C1CCC12CCC2)=O)OC c1(CCC(=O)NC2CCN(C(COC)=O)C2)nc2ccccc2[nH]1 c1(CC)cccc(NC)n1.C12CC(C(O)C1)NC(=O)NC2 N1(S(CC(=O)OC)(=O)=O)C2CCC1CN(C(C13CC(C1)C3)=O)C2 c1(NC(CC(=O)Nc2c(CC)nc[nH]2)=O)ccc(C)c(C)c1.C1(C)C(=O)O1 C1(NC(CCCC#C)=O)CS(=O)(=O)CC1NC(=O)Cc1nnc(C)o1 C1(CNC(=O)Cc2cscn2)CCN(C(=O)C=CC2CCCCCC2)CC1(F)F C123CC(CN(C1)C(=O)CCc1cn(nn1)C2)C3.Cc1nn(C(C)C)c(=S)n1C N1(C(C(CCC)O)=O)CCCC2(CC(C(=O)NCc3cccc(C)c3C)=NO2)C1 C#CCCCCCC(=O)N(CCCO)CCCC.C1C(OC)C(=O)N1 C(=O)(C1=CCC(F)(F)CC1)NC1CCCC(CNC(C2CN(CC)C(=O)C2)=O)C1 CCC(C)CCCCC(=O)NCC1CCC(F)(CNC(C2(C(C)C)CC2)=O)CC1 n1(CC(=O)NC(CCCCNC(C=CC=CCC)=O)C)ccc2c(C)cccc12 c1(N2CC(OC)C(NC(=O)OC(C)(C)C)CC2)cc(C)[nH]c(=NCC(F)CO)n1 c1(C(=O)NCC(C(C)C)NC(c2c(OC)cccc2Cl)=O)cc2c(ncn2C)s1 Cc1ccc(C)c(N(CCC#N)C(N2CCN(c3nc(C)cs3)CC2)=O)c1 C1(NC(c2cccc(OCC)c2)=O)CC(F)CN(C(=O)CCCSC)C1 c1(SC)cccc(C)c1CO.n12ccnc1NC(=O)NCC2 c1(SC)cccc(-c2cccc(C3CC3C(=O)NCc3cccs3)c2)c1 c1(C(=O)NC(C)CNC(c2cccn2Cc2cccnc2)=O)nc(=N)cc[nH]1 C(CCCCC(=O)N1CCSCC1CCNC(=O)CCC(C)(C)C)OC c1(C(N2CCC(C(F)C(=O)NC3CC(F)C3)C2)=O)ccnnc1O n1(CC(=O)NCCCN(C)C(C2CC(=O)N2)=O)c(-c2cccs2)csc1=O N1(C(c2n(CC#C)ccc2)=O)CCN(C)C(CNC(c2ccc(=O)n(O)c2)=O)C1 N1(C(C(=O)NC)C2CCSC2)CCOCC2(COCCN2C)C1 C1(C(=O)NCC(CNC(CSc2cccc(OC)c2)=O)CO)COCCC1(F)F c1(CC(=O)NC(CC2CN(C(c3c(C(C)=O)coc3)=O)C2)C)ccc(C)cc1 CC1CCN(C(=O)CCC2CCN(C(c3cocc3C(N)=O)=O)C2)CC12CCC2 N(C1CCCc2cnn(C(C)C)c21)C(COc1ccc(NC(C)=O)cc1)=O C(=O)(CC(CC)C(C)C)NCCN(CCC)C(c1cc(C)oc1C)=O Cc1cc(=N)[nH]cc1C(N1CC=C(CNC(=O)C#CC(C)C)CC1)=O CC(C)(C)C(CC(=O)NC(CNC(c1ccc(C(F)F)c(N)c1)=O)CO)C(F)F c1(C(=O)NC(C(=O)N(C(COC)C)C)Cc2cnn(C)c2O)ccc(=O)n(C)n1 c1(CNC(C2N(C(CC3CC(=O)C3)=O)CC2)=O)cccc(Cl)c1 c1(CN2C(C(=O)Nc3cncc(C(=O)OC)n3)C(O)CC2)c(C)nn(C)c1Cl N1(C(C(C)S(C)(=O)=O)=O)CCN(C(c2cnc(C3CC3)[nH]c2=N)=O)C2(CC2)C1 C(C)(CC(C)NC(=O)C(F)F)NC(C=CCOC)=O C1(CNC(N2CCC2C2CCOCC2)=O)CCC(F)(F)C1 c1(-c2cn(CC(=O)OCC)nn2)ccc2c(c1)CCN(C(c1cc(C)ns1)=O)C2 c1(NC(Cc2ccc(SC)cc2)=O)cc(S(=O)(=O)NC(C)=O)ccc1C C=C1CCC(C(=O)NC2(C(N3CCC(O)(C(F)F)C3)=O)CC(O)C2)CC1 CC1C(NC(=O)Cn2nnc(=O)[nH]2)CC2CCC1N2C(C1(F)CCC(=O)CC1)=O C=CCCCCCCCCC(=O)NCC(C)(C)CNC(C1CCCC(F)(F)C1)=O CCC(C(=O)NCCC(=O)N(C)C1CC1)N(C)C(C1CCC(=O)O1)=O c1(Nc2ccc(NC(C)=O)nc2)ncnc2c1S(=N)(=O)CCC2 c1(OC)cc(N)c(F)cc1C(=O)NC1CC(NC(c2ocnc2C(F)(F)F)=O)C1 C1(C(=O)NCC=CCNC(C2(CCC)CCC2)=O)CCCOCC1 C(CCCC(CO)NC(C1(C)CCCC1)=O)NC(C1(CCCC)CCC1)=O n1(CCN(C)C)cc(C(=O)NC(C)(COc2ccccc2)C(=O)O)c2ccccc12 C1(NC(CCC)=O)CCCCC1N(C(=O)COc1ccc(C2CC2)cc1)C N1(C(C(CC)(CC)CC)=O)CCC2(CC1)CC(N1CC(F)C(F)C1)CO2 N1(C(C(C)CN2CCOCC2)=O)CC(CNC(=O)C(F)=C2CCCC2)C(C)(C)C1 CCC(C)(O)C(=O)NC1CC(C(=O)N(C)CC2CCOC2)CC1O C1(NC(C23CCC(OC)C2C3)=O)CCC(CNC(C2(C)CC3CC3C2)=O)CC1 C1(CNC(c2cc(F)n[nH]2)=O)CCN(c2nnc(C(F)F)s2)CCC1(F)F Cc1cccc(C(=O)C=CC(=O)NCC2(NC(c3cocc3C)=O)CCCCC2)c1 c1(CC)ccc(OCCCC(=O)OCC2CCCN(C(=O)CC(C)C#N)C2)cc1 c1(SC)nc(O)c(C(N2CC(NC(C3(CCOC)CC3)=O)C(C)C2)=O)cc1C#N CC(C)C(C)(CNC(=O)C(c1ncccc1F)(F)F)NC(=O)C(O)CNC(N)=O N1(C(C=CCC)=O)CC2(C(=O)N(CCNC(C3CCCCO3)=O)C3CC3)CCC1C2 N1(C(c2c(C)cno2)=O)CC(CNC(=O)CCC2CC2C)CC1(C)C c1(OC)ccc(CC(=O)N(C)CCNC(=O)CNC(c2ccccc2)=O)cn1 c1(OCC)ccc(C(N2CCCCC(NC(C3CC(O)C3)=O)C2)=O)cc1Cl C1(c2ccccc2)(NC(CCSC)=O)CCN(C(=O)CCC2CCN(C)C2)C1 Cc1ccc(NC(C2CCN(C(c3ncn(C)c3C)=O)C2C)=O)c(C)c1O c1(NC(N2CC(C(=O)NC(C)C(=O)OC(C)(C)C)C2)=O)ccc(Br)cc1Cl c1(CC(=O)N(c2ccccc2)CC2CCCC2)csc(Cl)c1Cl N1(C(c2cncc(C)c2)=O)CC2ON=C(CNC(c3cnc(C(C)C)s3)=O)C2C1 n1(CC)cnc2[nH]c(=NCCS(=O)(=O)CC)[nH]c(=NC3CCCc4cnccc43)c12 CCC(CC)C(=O)N1CC(=O)CC1C(=O)NCCOC1CC1 C12(C(=O)NC3(CN(C(C(C)Cn4ccnc4)=O)C)CC3)CC3CC(CC1C3)C2 C1(C)(NC(CCNC(=O)OC)=O)CCCCC1C(=O)NCC1CCCC1O N1(C(CCC(C)=O)=O)C(C(=O)N(C(C)CC(F)(F)F)C)CC2CC12 C1(C)(CNC(C2(CCNC(C(N3CCOCC3)C)=O)CC2)=O)CC2CCC1C2 C1(C(=O)NC2CC3CC(NC(c4ccn(CC)n4)=O)C2C3)CC2(CCOCC2)C1 N1(C(C2CCCN(CC)C2)=O)CC(NC(C2CSC2)=O)CC12CCC2 CCC(CC)CC(F)C(=O)N1CCCC1(C)C(=O)Nc1cccn2ncnc12 N1(C(c2c(Cl)cn(C)n2)=O)CCC(CO)C(NC(=O)C(F)CC2CCCC2)C1 c1(C(=O)NCCN(CC(C)O)C(c2c(C)csn2)=O)nc(C)c(C)[nH]c1=O c1(OC)cncc(C(N2CCC(CCN(C(=O)CN(C)CCOC)C)CC2)=O)n1 C(CC(=O)NC1COCC1C)(CC(C)C)NC(c1c(C)cc(CC)o1)=O CS(=O)(=O)c1ccc2c(c1)C(NC(NC1CCCc3ccoc31)=O)CO2 c1(C(N(CCn2cc(CC(C(=O)OC)C)nn2)C)=O)cnc(O)c(Br)c1 N12CC3(C1)CN(C3)C(=O)C1(CC)CC(C1)C2=O.c1(CC)cc(OC)ccc1Cl C1(C(N(C)Cc2nccs2)=O)CC2CCC1N(C(=O)C(c1ccc(Cl)cc1)=O)C2 C(=O)(CS(=O)(=O)CCCc1ccccc1)N(CCN(C)C(C12COCC1C2)=O)C CCCCC(O)CC(=O)N(C)CC1CCN(C(c2cccc3occc23)=O)C1 C(=O)(CCCCCC(C)O)NCC(CNC(C(c1ccccc1Cl)OC)=O)(C)C c1(C(N2C(C(=O)NCC3(OCC)CCC3)CC2C)=O)cc(C)cc(C)c1 c1(NCCOCCOCCOC)nccc(=NCc2nc(C)ccc2Cl)[nH]1 C(=O)(C(C(C)NC(=O)Cc1ccnn1C)C(C)C)N(C(CCCC)C)C c1(C(=O)NCC2N(C(C(C)S(N)(=O)=O)=O)CCC2)ccc(Cl)c(F)c1N c1(N2CC(C)C(Nc3ncc(C(C)(C)O)cn3)C2)ncc(S(C)(=O)=O)cc1Cl Nc1c(Cl)cnc(C(=O)NCCCCNC(C2CCOC2C2CC2)=O)c1Cl N1(C(C2CC(C#N)C2)=O)CC2(C1)CN(C(c1cc3occc3[nH]1)=O)CC2CO CCCCC(O)C(C)C(=O)N1CCC(C(C)C(=O)NCCc2nc(C)no2)CC1 c1(C(N2CCC(N(CCC)C(c3ns[nH]c3=O)=O)C2)=O)cc(S(N)(=O)=O)cn1C c1(CNC2CC(NC(c3cc(O)cc(Cl)c3)=O)C2)cccc2ccoc12 c1(C(=O)NC2CCC(NC(COCCC=C)=O)C2)cc2cc(C)ccc2o1 c1(C(=O)NCC(C(C)(C)C)NC(=O)C=Cc2cccc(F)c2)ccc(N)c(F)c1 C1(C(=O)NCC2(CNC(C=CC)=O)CCC2)CCN(CC(C)C)CC1 c1(C(N2CC(F)CC(C(N(C(C)C)C)=O)C2)=O)ccc(F)c([N+](=O)[O-])c1 Cc1cc(C(=O)NC2(CCNC(=O)Cc3nnc(C)o3)CC2)c2n[nH]cc2c1 C(c1cncnc1O)=CC(=O)NC1(C)CCN(C(C(C)CN2CCOCC2)=O)C1 Nc1cncc(C(=O)NCC2CC(O)CN2C(C2CC2Cl)=O)n1 N1(C(C)=O)CCC(C)N(C(=O)CCCn2c(-c3cccc(C)c3)nnc2S)CC1 N1(CC)CCn2nccc2C1C(=O)O.c12cccc(c1)N(CC)C2=O C(CCCC(=O)NCC1CCC(NC(C2CC3CCC2O3)=O)C1)(OC)OC C1(C(=O)NCCC(=O)NCCN(C(=O)Cc2cc[nH]c2)C)CCCC1O C1(CNC(C2(OC)CCOC2)=O)CCN(C(c2ccc(F)c(SC)c2)=O)C(C)C1 N1(CC(=O)N(C2CCCN(c3cc(C4CC4)ncn3)C2)C)CCCCCC1=O C(=O)(C(C(C)NC(c1cc2ccccc2[nH]1)=O)C(C)C)N(C(CC(C)C)C)C Cc1sc(NC(=O)CCc2ccco2)nc1-c1cccc(Cl)c1 CN1CC(C(=O)NCCN(C(c2cc(CS(C)(=O)=O)on2)=O)C2CC2)CC1=O CC(C)CCCCCC(=O)NCC(CO)Nc1ncc(C#N)cc1Cl c1(NC(CCc2ccc(C)nc2)=O)ccc(NC(=O)CC2(C)CC2)c(C)c1 CC1CCCC(CNC(=O)CC(O)CNC(=O)CN(CC(C)(C)C)C)C1 c1(C(=O)NC(CC)(CNC(c2scnc2C)=O)CC)sc(N=S(C)(C)=O)nc1C c1(C(=O)NCCN(C(Cc2c(C)nsc2)=O)C(C)C)ccc2cnc(C)n2c1 N1(C(C(C=CC)O)=O)C(CNC(=O)COc2cccc(OC)c2)CC2COCC12 C1(NC(CC2C(C)(C)C2)=O)CN(C(=O)C=Cc2nccs2)CC1N=[N+]=[N-] Cc1c(N)ccc(C(N2CCC3(C2)CN(C(=O)C(C)(F)C(F)(F)F)C3)=O)c1C C(CC(C(=O)N1CC(CCCCNC(C2CC(CCO)C2)=O)C1)NC=O)SC c1(CC)c(C(=O)NC2(CNC(C3CCCC3SC)=O)CC2)cccc1F C(CC1CC1)(C(=O)NOCCN(C)C)NC(CN(C(C)=O)C)=O CCC(C)C(C(=O)N(C1CCN(C(c2[nH]cnc2C)=O)CC1)CC1CC1)OC c1(C(N2CCN(C(=O)CC3CCOCC3)C3C2C3)=O)ccc(I)cc1[N+](=O)[O-] C(=O)(C(CCCC(N)=O)OC)N1CC(NC(CCOCCOCC)=O)C(F)C1 N1(C(C(C)NS(CC)(=O)=O)=O)C2CCC1C(CNC(=O)CC1CCCCC1C)C2 CC1CN(C(c2c[nH]c3ccccc23)=O)CCN(C(c2coc(C(F)F)c2)=O)C1 N1(C(C(C)NC(C)=O)=O)CCN(C(c2cscc2C2CC2)=O)C(CO)C1 N1(C(c2cc(C)cc(Cl)c2)=O)C2CCC1C(C)C(NC(C13CC(C)(CO1)C3)=O)C2 c1(OC)cc(C(N2CCN(C(=O)C(C)(C)c3cscn3)CC2C)=O)cc(N)c1 C(=O)(C(C)(O)CC(C)C)NC1(C)CCN(C(C2(COC)C=CCC2)=O)CC1 c1(C(N2CC(N(C(c3ccc(CC(C)C)o3)=O)C)C2)=O)c[nH]c2cccc(Cl)c12 c1(CC)nc(C)c(C(N2CCC(C)(NC(C3C(C#N)C3(C)C)=O)CC2)=O)c(C)n1 CC1CC(CNC(C2CC2CNC(=O)CC2CCC2)=O)C1 C1(NC(C2C(=C)CC2)=O)CN(C(C2CC2(C)C)=O)CC1(C)C c1(CN(CC(N2CCC(CNC(=O)C(O)CF)CC2)=O)C)ccc(F)c(Cl)c1 C1(CNC(CC(C)O)=O)CCN(C(C23CCC(CO)(CC2)C3)=O)C12CCC2 C(=O)(C1=CCCCCC1)NC(c1cccc(F)c1)CC(=O)OCC C1(O)(CCNC(c2ncn(C)c2)=O)CCCN(C(=O)CCn2ccnn2)C1 CCC(C)C(C(=O)NCCc1cc(C)on1)N(C)C(c1cncc(C)c1)=O N1(C(CC2(CCC#C)N=N2)=O)CC=C(CC(=O)c2ccccc2)CC1 c1(-c2nc(CC(C)OC)nn2CC2CCOC2)cnn2c1CCCC2 c1(C(N2CCCN(C(C3N(CC)CCOC3)=O)CC2)=O)c(C)ncn(C)c1=O C(=O)(CC(COC)COC)NC(CN(C(=O)CC1CCCC1)CC)C C1(NC(C2(Oc3ccc(Cl)cc3Cl)CC2)=O)CN(C(=O)C2=CCC2)CCC12CCC2 S(=O)(=O)(c1cnc(NCC(CO)C(C)C)c(Cl)c1)NCc1cnn(CC)c1C c1(C2C(C(=O)NCC3C(NC(c4c(C)noc4)=O)COC3)C2)ccncc1F C#CCCC(O)C(=O)NCC1CCN(C(C2CC(OC(F)(F)F)C2)=O)C1 C#CC1COCCN1C(C1CC2(CC2)CN1C(=O)Cc1ncn(C)c1C)=O C12(C(=O)NC3CC4CC3N(C(C3CCCOC3)=O)C4)CC3CC(C1)CC(O)(C3)C2 C(CCCC(=O)N1CCCC1C(=O)N(CCCc1nccs1)CCO)N(C)C c1(OC)ccc(Br)c(NC(C2C(O)CCN2c2ncnc3cc(I)sc23)=O)c1F C1(C(=O)NC(C(=O)OCC)Cc2cncn2C)CSC(C)(C)C(=O)N1 C(N=c1[nH]c(=NCC2CC(C)CC(C)C2)c2cccc(F)c2[nH]1)c1c(C)noc1 C(=O)(CCCCCN(C)C(C12CSCC1C2)=O)NC(C#C)(C)CC c1(OC)ccccc1C(O)CNC(=O)N(CCCn1nccn1)C1CC1 CC1C(=O)Nc2ccccc2N1C(c1ccccc1CNC1=NCCC1)=O C(=O)(CCC(F)(F)Cc1ccccc1)NC(C)(C)C1CC1 N1(C(c2cc(CC)no2)=O)CC2CC1CN2C(c1cn(C)nc1-c1ccoc1)=O c1(OCC)cc(Cl)ccc1C(=O)NCc1ncc(-c2ccc(N)cn2)cn1 c1(C(C(=O)NC2(C)CC(NC(c3cccnc3O)=O)C2)O)ccc(F)c(Cl)c1 C1(NC(c2cnn3ccsc23)=O)CCC2(CCN(C(=O)CCc3csnn3)C2)C1 Cc1ncc(C(=O)NCc2cn(CCNC(=O)C(c3ccc(Br)s3)O)nn2)cn1 N1(C(C(CC)=CCCC)=O)CC(CO)C2(C1)CN(C(c1ccc(F)c(N)c1)=O)C2 C1(C(=O)NCCOC)Cc2cc(O)ccc2CN1C(C1(c2ccn(C)n2)CC1)=O C(=O)(C(C)(CO)NC(=O)CN1CCNC1=O)NC(CC(=O)OCC)C c1(NC(C(c2ccc(Cl)cc2)CC)=O)c(N)cccc1[N+](=O)[O-] C1(C2C(C(=O)NC3CC(C#N)C3)CCO2)CCN(C(=O)CSc2nncs2)CC1 c1(C(N2C(CN(C(=O)COC(F)F)CC)CCC2)=O)cc(C)c(O)c(N)c1 N1(C(c2cccc(N(C)C)n2)=O)CCCC2CC(NC(=O)CC3CCC3)CCC12 Cc1cc(Br)ccc1CNC(C1CCC(n2cc(CCN(C)C)nn2)C1)=O C1(C(=O)NCC(CN(C(C(N2CCOCC2=O)C)=O)C)C)CN2CCN1CC2C CC(C)(CCC(=O)N1CC(NC(=O)C=CCOC2CCOCC2)C1)[N+](=O)[O-] C1(CNC(c2cncnc2)=O)CC2(CC2)CN1c1cc(C2CC2)ncn1 CC(C)(CC#N)C(=O)NCCC1CSCCN1C(=O)Cc1cccc(N)c1 N1(C(CC2CN(C)C2)=O)CCN(c2ncc(C(=O)O)cn2)CC1 N1(C(c2c(OC)scc2)=O)CCN(C(=O)COCc2nnc(C)s2)C2(CC2)C1 C1(C(C)(C)C)CN(C(=O)Cc2cccc(Cl)c2)CCN1C(C1CC1F)=O c1(NC2(CC(C)C)CC2)cc(S(=O)(=O)N2CCC3(CCC(C)C3)C2)c(Br)cn1 c1(C(N2CCC(NC(COCCOCC)=O)CC2)=O)sccc1S(=O)(=O)CC N1(C(c2c(OC)scc2)=O)CC2(CCN(C(=O)CCCn3cccn3)CC2)C1 c1(C(=O)NC2CC(CNC(c3ccc(OC)o3)=O)C2)oc(CC2CC2)nc1C c1(C(C(=O)NCCC(O)C2CCC2)NC(CCSC)=O)ccnn1C CC(CNC(=O)CC1CC=CC1)CNC(C1CCO1)=O C(=O)(C1CCc2cccc(F)c21)NC(C1CN(C(C(CCC)(C)O)=O)C1)C C1(NC(c2n[nH]c(C)c2C)=O)CCN(C(C2CCC(C)C(C)C2)=O)CC12CCC2 CC(C)(C)CC(O)C(=O)Nc1cccc(CNC(C2SC3=NCCN3C2=O)=O)c1 N1(C(CC(=O)NC2CC2)=O)CCC2(CC1)C(NC(c1cc(Cl)on1)=O)CS2(=O)=O C1(CC(=O)NC2CCCCC2NC(c2cnc(C3CC3)s2)=O)CC2(CCC2)CO1 C1(C)(NC(C2(CNC(c3ncccc3F)=O)CC(=C)C2)=O)CCC(=O)NC1=O C1(C(=O)NC2(CF)CCN(c3c(C(C)=O)cccn3)C2)CC(=O)NC1(C)C N1(C(C2(F)CCCCC2)=O)CCC(c2n[nH]c(CNC(C3(Cl)CC3)=O)n2)CC1 S(=O)(=O)(c1cccnc1Cl)N1CC(CC(=O)NCc2ccc(F)c(Br)c2)OCC1 N1(C(COC(C)=O)=O)CCCC(NC(=O)Cc2cccnc2F)C1C C1(C(N(C)CC2(F)CCC(NC(c3csc(Cl)n3)=O)C2)=O)CCCC1(C)C Cc1csc(C=CC(=O)NCCCCC(C)NC(C2CC2(c2ccccc2)F)=O)n1 CC1CCC(C)N1CC(=O)NCC1(C(=O)NCC2N(C(N)=O)CC2)CC1 CC#CCC(C(=O)NCC(CNC(=O)CC(=O)OC(C)(C)C)(C)O)NC(C)C N1(C(=O)NC(C)Cc2cncs2)CCCCC1c1nccn1C N1(C(C(C)OCC(C)C)=O)CC2(CCCC2NC(c2ccc3c(c2)CCC3)=O)C1 CC1CCOC(C(=O)N(C(C)(C)CC(=O)N2CCCC2C)C)C1 C(=O)(CCCCC(N)=O)NCC(=O)NCC(C)C1CCC1 O=C(N=c1[nH][nH]cc1C1CC1)N1CCCC1c1cncc(Br)c1.C1CCC1 c1(CN2C(CC(=O)NCC(F)F)COCC2)ccnc(F)c1F c1(C(N2CCC(NC(C=CCOC)=O)C2C2CC2)=O)ccc(Cl)c(Cl)c1C c1(C(=O)NC2(COC)CN(C(C34CCC(CC3)OC4)=O)C2)cc(SC)ccc1F c1(C(N(C2CN(C(c3cnc(OC)nc3)=O)C2)C)=O)cccc2c(C)ccnc12 c1(CC)nc(C)n(C)c1C(=O)NCCC1(NC(c2cccnc2C)=O)CC1 C(=O)(CC(C)C(C)(C)C)N1CC(C)N(C(=O)CCCn2ccccc2=O)CC1 c1(NC)ccccc1C(=O)NC(Cc1cn[nH]c1)C(=O)NCCC(C)O C1(C(=O)NCC2CCC(CNC(C3CCCC(=O)O3)=O)CC2)COC2(CCC2)C1 CCCC(C)(C)C(=O)NCCCCC1CN(C(c2ccc(Br)cn2)=O)C1 C1(CNC(=O)NC(C2CCN(CC3CCCC3)CC2)C)CC2(CCC2)C1 C1(C(N(C(C(C)C)C)C2CC2)=O)(NC(c2ncc[nH]2)=O)CC(F)C1 Cc1ccc(C(=O)NCC2CC(O)CN2C(=O)Cc2cn[nH]c2)c(Cl)n1 C(=O)(CCCC(C)NC(=O)CS(=O)(=O)NC)NCCC(CC)CO CC12CN(C(C3CCC(=O)N3)=O)C(C(=O)NC34CC3COC4(C)C)(C1)C2 N1(C(c2c(OC)cc(N)c(F)c2)=O)Cc2ccccc2C(NC(=O)C=CBr)C1 c1(CC(=O)NC(C2CCCN2C(=O)CC2CCNC(=O)C2)C)cccc(F)c1 c1(SCC(=O)NCC(c2ccccc2)NC(C2C(CC)C2)=O)cnn(C)c1 C1(NC(C=CC(C)C)=O)CC(C(=O)NCCCCc2cnc[nH]2)C1 C12(CNC(C3(CC(C)C)CC3)=O)CC1CN(C(=O)CCN(c1ccccc1)C)C2 N1(C(=O)Cc2ccc(F)c(F)c2)CCC2(CCCC2N2CCCC(F)(F)C2)CC1 C1(C(N(C)OC(C(=O)NCc2ccccc2)=O)=O)CC1C1CCOC1 Cc1cc([N+](=O)[O-])cnc1NC(c1ccc(OC(F)(F)F)c(Cl)c1)=O CC1CN(C(c2cc(OC(F)F)cc(Br)c2)=O)CCN1C(=O)C(O)C(F)F C(=O)(C(C(C)C)C1CCC1)N1C(C(C)NC(c2cn(CC)nc2)=O)CCC1 c1(C(=O)NC2C(NC(C3(C)CC3)=O)CCCC2)nc(O)nc(O)c1F CC1C=C(C(=O)N2CCOC(Cn3cc(C4C5CCCOC45)nn3)C2)C1 C1(C(c2nnnn2C)(C)NCC2CCS(=O)(=O)C2)(OCC)CCSCC1 O=C1CC(CC(=O)N2CC3(CCC(C(=O)Nc4nnco4)O3)C2)c2ccccc21 N1(C(c2cc(CC)nn2C)=O)CCN(C(C2CC2OC(C)=O)=O)C(C)C1 c1(OCC)nc(N2CC(NC(c3coc(C)n3)=O)C(n3ccnn3)C2)cc(C)n1 c1(CCCC)ccc(C(=O)NCC2CC2NC(C2(C3(C)CC3)CC2)=O)cc1 N1(C(c2cccc(C)c2C)=O)CCC2(CCCN2C(C2CC2F)=O)CC1 CN1CC(O)CCC1C(=O)NC1CCC(NC(=O)CCN2C(=O)CCC2=O)C1 C1(C(=O)NCC(C)(C)OCCO)C2CC(O)C(C2)N1C(=O)Cc1ccc[nH]1 c1(C(N2CCC(O)(CN(C(CC(=O)NCC)=O)C)C2)=O)cc2c(Cl)cccc2s1 Cc1cc(C(N2CCOCC(NC(=O)CC3CCCCN3C)C2)=O)c(C)nc1C N1(C(C2CC(C#N)C2)=O)CCC2(CCCCC2NC(c2cc3cscc3s2)=O)C1 C(C1=CCSC1(C)C)NC(c1n(CCOC)nnn1)(C)CCSC N1(C(c2c(SC)snn2)=O)CCOCC1CCNC(=O)Cc1ccn(C)n1 C#CCC(C)(C(=O)N1CCSC2CCC12)NC(c1nc(CC)oc1C)=O C1(NC(C=CSC)=O)CN(C(C2CCCC(=O)N2)=O)CCC1C C1(C(=O)NC)CN(C(=O)C(CCN(C)C)N(C)C(=O)OC(C)(C)C)CCS1 CC(CC(=O)NCCC(O)CNC(=O)CSS(C)(=O)=O)C1CC1 C(=O)(C(C)S(C)(=O)=O)NC1C(C)N(C(=O)CC2CCC3CC3C2)CC1 c1(CC(=O)N(C2CCN(c3nc(C)ns3)C2)CCOC)ccc(O)c(C)c1 Cc1nn(C)c(C(=O)N(CCNC(C2CCCN(CC(F)F)C2)=O)C2CC2)c1Cl c1(OC)c(NC(=O)CCOCCN(C)C(c2ccc(C)c(O)n2)=O)cccc1F C1(=O)CCCN=C2N=C(C3=C(N2)CCOC3)N1C.c1(CNC)nc(=N)[nH][nH]1 C(=O)(C1=CC2(CCOCC2)C1)NC1C(C)(C)CN(C(c2cc(C(F)F)[nH]n2)=O)C1 c1(C(N2CC(OC)C(NC(=O)CN3CCC(O)CC3)C2)=O)cccc(N=[N+]=[N-])c1 C1(OC)(OC)CC(C2CCN(CCC3(C#N)CC3)C2)C1 C(=O)(C1=NOC(C)C1C)NC(CC#C)C(=O)NC1(C)CCC(O)CC1 c1(C(N(C2CCN(C(CCC#CC)=O)C2)CCO)=O)cc(C)c(C)nc1C Cc1cnn(CCC(=O)NC2(CN(C)C(C3CC3c3ccsc3)=O)CC2)c1 c1(C(F)(F)F)nccc(N(C2CCN(Cc3cnoc3)C2)C2CCCC2)n1 N#Cc1cccc(S(=O)(=O)NC2CN(Cc3cccnc3Cl)C2)c1 c1(CC)ccc2occ(C(=O)NC3CN(C(C4CC5(CCC5)C4)=O)C3)c2c1 Cc1cc(N2CCN(C(c3ccc(F)cc3F)C)CC2)ncc1C#N c1(C(=O)OC)ccc(C=CC(N2CC(NC(c3cnc(S)[nH]3)=O)C(F)C2)=O)o1 N12CCCC1C1CCCN1C(=O)C(=O)N2.C1(O)COC2(CCCC2)C1.CC(C)(C)O C(=O)(CCC(C)(F)F)NC(C(N1C(C=C)CC1)=O)Cc1ccco1 C(=O)(C1Cc2c(Cl)cccc21)NC(CNc1cc(CC)nc(C)n1)C1CC1 C1C(C)(C)CNC(=O)C(C)OCC2C(C2)C(=O)N1C.C1(C2(OC)CC2)CCCO1 c1(CNC(c2nnnn2C)C2(CC=C)CCC2)n[nH]c(C)c1C C(C)(CCC(C)(C)C)(c1n(CC)nnn1)NC(C)CC(C)(C)OC O=C(CC(C(F)(F)F)NC(=O)Cc1cnoc1)NC1CN2CCCC1C2 c1(CNC(C(c2ccc(Cl)s2)N(CC(=O)OC)C)=O)ccccc1 C1(C(N2C(C)CN(C(=O)C(C)(C)c3cncnc3)CC2)=O)CCn2ccnc2C1 c1(C(N2CC(NC(c3cn(C)nc3)=O)C(F)C2)=O)cc(C#N)ccc1[N+](=O)[O-] C=CC1(C(=O)NCCCCS(C)=O)CCN(C(C2CC=CC2)=O)C1 CC1(C)CCc2[nH]c(C(N3CC(O)(CNC(c4csc(C#N)c4)=O)C3)=O)cc2C1 c1(C(=O)NC2CN(C(c3cc(F)cc(Cl)c3)=O)CCC2F)ccnn2ccnc12 CC1CCN(C(C2COC(C)C2)=O)CCN1C(c1ccc2nn[nH]c2n1)=O C(=O)(C1=Cc2ccccc2C1O)N1C(CNC(c2c(C=C)cnn2C)=O)CC1 c1(CN)cccc([N+](=O)[O-])c1.C=C1CCN(C(=O)C(O)CCCC)C(C=O)C1 C#Cc1ccc(C(=O)NCCC2CCCN(C(=O)C3=NOCC3)C2)nc1 c1(C(N2CC(C)(CC(=O)OCC)C2)=O)ccc2ccc(F)c(F)c2n1 N1(C(c2c(CCC)nns2)=O)CC2CCCC2(NC(c2cnsc2)=O)C1 c1(C(=O)NC2CN(C(C(CC(C)C)(F)F)=O)CC2O)ccc2c(c1)CC(C)(C)C2 C(=O)(C1=CCC(C)(C)CC1)NC(C(=O)NCC(C(C)O)O)Cc1ccoc1 CC1CCC(CCNC(=O)CC2CC(NC(c3ccc(CO)s3)=O)C2)CC1 N1(C(C(=O)OCC)C2CC2c2ccnn2C)CCOC(C#N)C1.C1(=O)CCCN1 C#CC1(C(=O)NCCCCS(C)=O)CCN(C(c2c[nH][nH]c2=N)=O)CC1 N1(C(CN(C(=O)OCC)C)=O)CCCC(N(C)Cc2ncsc2Br)C1 C1(NC(CC2(NC(C(=Cc3ccco3)C)=O)CCC2)=O)CCC(=O)NC1C C1(OCCC)CCN(N2CCN(C)C(C(F)F)C2)C1 c1(N2CCC(CCOC)C2)cc(S(=O)(=O)N2CCC(SC)C2)ccc1C#N C1(C2CC2)(NC(C(=O)N(CC=C)C(C)C)=O)CCNC1 c1(C(=O)OC)cc(Br)c(O)c(Br)c1.C12CN(S(=O)(=O)CCCCl)CCN1C2 C#CC1(NC(=O)CN(C(=O)C(C)(F)F)C2CCCC2)CCCOC1 Cc1ncc(S(N)(=O)=O)cc1C(N1CCC2(NC(=O)Cc3cscn3)CC2C1)=O N1(C(C(N2CCOCC2)C)=O)CCC(NC(c2cccc(NC)n2)=O)C1C(C)C N1(C(c2cc(OC)c(F)cc2N)=O)CCC2(CNC(=O)OC2)C1 N1(C(C=CCC)=O)CC2(CCCCN(C(c3ccc(CO)cn3)=O)C2)C1 C1(NC(C(CC)OCC)=O)CCN(C(c2cccc(C)c2F)=O)CCC1(F)F c1(OC)ccc(C)cc1NC(=O)CC1(N(C(C2CC2(Cl)C(=O)O)=O)CC)CCC1 C1(O)(C(N2CC(OC)C(NC(=O)C=C(Cl)Cl)C2)=O)CCC(C)(C)CC1 c1(C(=O)NCC2C(CNC(c3c(C)ccs3)=O)C2)c[nH]c2ccncc2c1=O C1(CNC(c2cn(C)nn2)=O)CC(O)CN1C(=O)CCN1CCCC1 CCCCC(C)(F)C(=O)N1CC2(NC(c3ccc(OC)c(Cl)c3)=O)CCC1C2 c1(C(=O)NC(CN(C(c2n(CCC)ncc2)=O)CC)C)cccc(F)c1F N1(C(c2nc(C)c(Br)cn2)=O)CCC2(CCCN(C(=O)Cc3ccccc3)C2)C1 c1(CC(N2CCC(O)(C(C)NC(C=C(CCC)C)=O)C2)=O)nc2ncccn2n1 C1(C(=O)NCC2(C(N)=O)CN(C(=O)CC3CC4CC4C3)C2)(COC)CC=CCC1 C12(NC(CCC(=C)Cl)=O)CC(CNC(=O)C(C)OCC3CCCO3)(C1)OC2(C)C c1(C(=O)NCC2(NC(C(C)SCCCC)=O)CCOC2)cc(N)c(C)cc1C Cc1[nH]nc(Cl)c1C(=O)NCC(C)NC(C1CCOC(C(C)C)C1)=O Cc1onc2ccc(C(N3CCCC(NC(=O)CC4COCCOC4)C3)=O)cc12 N1(C(C2CC(C)(CC)C2)=O)CCC(CC(C)NC(=O)CSCc2cscn2)CC1 C(CCOCC1CCCO1)(C(=O)NOCCF)NC(c1ccc(C#N)[nH]1)=O C1(CCC)(NC(C2CCCCO2)=O)CCCN(C(c2[nH]cnc2C)=O)C1 O(S(=O)(=O)c1ccc(Cl)cc1F)c1cc(Cl)ccc1F.c1(C(C)=O)ccc(O)cc1C n1(CC)ccc(CC(=O)NCCCC2CCCN2C(c2cnc(C(C)C)s2)=O)n1 C1(CNC(C(C)N(C(CCN(C)CC)=O)C2CC2)=O)CC2C=CC1O2 N1(C(C(n2ncc(C)c2)C)=O)CCCC(C(=O)NC(c2ncccc2F)C)CC1 c1(C(=O)NCC(CCNC(c2coc(C3CC3)n2)=O)O)cc2c(s1)CCCC2 O=C1NC(=O)N2CCN(C(c3ccc(F)cc3Br)C(=O)NC3CCCC3)CC12 C1(NC(C(C)OCCC=C)=O)CCOCC1NC(=O)CCc1cc(C)nn1C C(=O)(CC(=O)NCCN(C(C1CC(OC)C1)=O)C1CC1)NCC#C N1(C(Cc2c(C)n[nH]c2)=O)CCC2(CCCN(C(C3CCCCC(F)C3)=O)C2)C1 c1(C(=O)NCC(C(C)C)NC(C2C(OC)CCCC2)=O)cnn2ccccc12 C(=O)(CCCC(C)S(C)(=O)=O)N1CC2CC(CN(C(CS(=O)(=O)NCC)=O)C2)C1 CCC(CCC(=O)NC1CC12CCN(C(c1cc(COC)[nH]n1)=O)C2)OC c1(CC)ncc(C(=O)N(C2CCN(Cc3nnnn3-c3ccccc3)C2)C)o1 C1(O)(CNC(CCN(CCCCC)C(C)C)=O)CC(NC(C2CC2F)=O)C1 Cc1[nH]cc(C(=O)NCCC2CC(NC(=O)C3=COCCC3)C2)c(=O)c1Cl C1(CN(C(=O)CCCC#N)C)COCCN1C(c1scnc1C(F)(F)F)=O c1(C(=O)NC2CC(C(=O)O)C2)ccc2c(n1)COCC2 CC1CCC(NC(=O)CCC(C)(C)C)CN1C(c1cncc(-n2cccn2)n1)=O O=C(CCS(=O)(=O)c1ccccc1)N1CCC2(CC1)CCN(C(C1CC1F)=O)C2 C=Cn1ncc(C(N2CCC(CC=C)(C(N3CC(CC)(OC)C3)=O)C2)=O)c1N N1(C(C2C3CN(C(C4CCC5(CCCC5)C4)=O)CC32)=O)CCc2c(O)noc2C1 Cc1ccc2c(c1)CC(C(N1CCN(C(c3cc(F)ccc3O)=O)CC1)=O)S2 C(=O)(C1=CCS(=O)(=O)C1)N1CC(Cc2nc(C(C)OCC(CC)CC(C)C)on2)OCC1 C1(CNC(=O)Cn2cnnc2)CN(C(=O)CC2CCCC2)CC12CC2 c1(C(=O)NC(C2CN(C(c3ccc(S(C)(=O)=O)[nH]3)=O)C2)C)cccc2nccn12 c1(OC)ccc(Cl)c(C)c1C(N1CCC(CNC(=O)CS(C)(=O)=O)C(O)C1)=O Cc1ccc(C(N2CCC2)=O)cc1.N12CCOC(C1)C(=O)N(CC(C)C)CC2=O Cc1csc2c(N3C4CCC3CC(NC(C3CCC(C)O3)=O)C4)ncnc12 C1(C)(COC)CCCN1C(=O)CCCn1cc(-c2nc(C)c(C)[nH]2)nn1 c1(C(=O)NC2CCN(S(CC)(=O)=O)C2)oc(CNC(=O)NC)nc1C CC1(C)C2CC(C(N3CC(NC(c4ccc(C(N)=O)o4)=O)C(O)C3)=O)CC12 C1(CC)CN(C(=O)C(C)CC2CCC2)CC1NC(c1coc(C(C)C)n1)=O C#CCC(C)(C(=O)NCc1ccncc1F)NC(c1ccc(C)[nH]1)=O C(=O)(C(C(C)(C)C)N(C)C)NC1C(C)CN(C(=O)COCc2ccnn2C)C1 Cc1cn2c(n1)CN(C(=O)CCCNC(=O)CC1CCCNC1=O)CC2 CCCCS(=O)(=O)CC(=O)NC12COC(C1)C(NC(=O)C(F)(F)C(O)C1CC1)C2 N1(C(C2CCCC(OC)C2)=O)CC2(CCN(C(c3ccnc(Cl)c3)=O)CC2)C1 c1(C(C(=O)NCCC2CCN(C(C(COC)OC)=O)C2)(F)F)ccc(Cl)c(Cl)c1 c1(CN2CCC(C)(C(=O)NCCC(=O)NC)C2)n[nH]c2ccccc12 CC(C(F)C=O)C(F)(F)F.C1(C)(COC)CCN(C(=O)C(F)(F)C2CCOCC2)C1 CN1CCC(C(=O)NC2CCC(CCNC(C3(C)CC(=O)C3)=O)C2)C1 N1(C(CC2CC(C)(C)OC2)=O)CCOC2(C1)CN(C(=O)Cn1ccc(=N)[nH]1)C2 c1(NC(N(C2CCC(OCC)C2)C)=O)c(C)cc(Cl)cc1C C(=O)(C(CCCOC)NC(=O)C=C1CCOCC1)NCC(CC)O N1(C(C(C)CC2CC2)=O)CC2CCCC(C1)N2C(=O)CC1CCCC(C2CC2)O1 CC1CN(CCOCCOC(c2cccc(Sc3ccccc3)c2)=O)CCO1 c1(CNC(N2C(CN(C(=O)OC(C)(C)C)CC)CCC2)=O)cncc(Cl)n1 n1(CC)ncc(C(=O)NCC(=O)NC2CCC(C(=O)NCC(C)(C)O)C2)c1C N1(C(C(C2CCC2)OCC)=O)CC2CC1CN(C(c1csc(C)c1)=O)C2 c1(C(=O)NC2C(C)N(C(c3nncs3)=O)CC2)ccccc1C#N C1(F)(CNC(C2(C(C)C)CCCO2)=O)CCN(C(c2cccc(N)c2)=O)CC1 C(=O)(CCCC(F)(F)Br)N1CC(O)(CNC(CCC(=C)C)=O)C1 C12(C(N(C3(C#C)CC3)C)=O)CCCC1CN(C(c1ccc(SCC)cc1Cl)=O)C2 N1(C(CC(C)c2ccccc2)=O)CCC(NC(c2c(Cl)cncc2Cl)=O)C(F)C1 C(CC(C)(C)C(=O)N1CC(CNC(C2(CO)CCCC2)=O)CC1(C)C)OC N1(C(CCOC)=O)CCC2(CCCC(CNC(=O)C(O)C3CC3)O2)CC1 N1(C(C(C)=C(C)C)=O)CCCOC(CNC(=O)CCNc2ccc(N)cc2)C1 Cc1ccc(S(N)(=O)=O)cc1C(=O)N(CCC(F)(F)Cn1cc(C2CC2)nn1)CC c1(OC(C)C)nccc(C(N2CCN(C(C3CC(=O)N(C)C3)=O)CC2)=O)c1F C(=O)(C1CCCc2c[nH]nc21)NC1C2CN(C(C(C(C)C)F)=O)C1C2 c1(C(=O)NCC(CC)NC(c2cn(CC)nc2C)=O)cccc2c1oc(=O)n2C C(=O)(CCCC(CC)NC(c1cnc(=N)[nH]c1)=O)NC(CCC=C)CO N1(C(C(C2CC2)SC)=O)CCN(C(=O)CC(C)c2cnn(C)c2)C(C(C)C)C1 c1(OC)cccc2c(CNC(C3CC3CC3CC3)=O)coc12.C1(=O)C=CCN1 CC1CN(C)CCC1NC(=O)C(C(C)(C)O)NC(C1CCC(CO)CC1)=O CC1CN(C(c2ccc(CNC(c3ccc(F)cc3)=O)cc2)=O)CCCO1 Cc1ncncc1C(=O)NC(C)C(c1ccccc1)NC(=O)CN(C)C(N)=O C1(C)(C(=O)NC2CCCC(C(N3CCC(OC)CC3)=O)C2)CCCCCC1 C(=O)(C(C)CCCC(C)C)NC(CCC(=O)NCCC(C)N(CCC)C)C c1(C(=O)OCC)cncc(C=CC(=O)NCC2CCC2NC(C2CSC2)=O)c1 N1(C(c2n(C(C)C)cnc2)=O)CCCC12CCCN(C(=O)CCN1CCC1)C2 N1(C(COCC)=O)CCN(C(=O)COc2ccc(COC)cc2)CC1CC(F)F Cc1cc(=NC2CN(C(C3(O)CCC3)=O)Cc3ccccc32)[nH]c(S(C)(=O)=O)n1 N1(C(c2cccnn2)=O)CC2(CCC(NC(C3(CSC)CCOCC3)=O)CC2)C1 C(C(O)CC(=O)N(CC(c1ccccc1)O)C)N(C)C.C1CO1.C1CO1 c1(C(=O)NC2(CNC(c3ncccc3F)=O)CCCC2)[nH]cc2c1CCC2 C(C(C)(C)C(F)(F)CC)N(C(CCc1cccc(C#C)c1)=O)C(C)C N1(C(C2(SC)CN(C(=O)CC3(O)CCOC3)C2)=O)CCOC(CCF)C1 Cn1ncc(C(=O)NC(CC2CCCC2)C(=O)N2CC(CF)C2)c1N c1(SCC(=O)NC23CN(C(CN(C)C4CC4)=O)C(C2)C3)ncnc2[nH]cnc12 c1(C(=O)NC2C(NC(CC3(C(=O)OC)CCC3)=O)CCC2)nccc(C(F)F)n1 C(C)(C)(CCC(=O)NCCCC1(NC(=O)CC(C)c2ccccc2)CC1)OC c1(C(=O)NC2(C)CCN(C(c3nccs3)=O)C2)ccccc1[N+](=O)[O-] N1(C(C(C)OCCCC)=O)CCCCC(C(=O)NC2(c3cc[nH]n3)CC2)C1 C#CCC(CC(F)F)C(=O)N(C)Cc1cn(C(=O)NC2CC(NC(C)C)C2)nn1 C1(NC(c2cccc(C)c2F)=O)CCC2CN(C(=O)CC3CC=CC3)CC2C1 C(CCCCCC(=O)N1CCC(N2CCC2)C1)NC(c1cc(C)nc(O)c1)=O N1(C(C2(CNC(c3[nH]cc(C(C)=O)c3)=O)CC2)=O)CCn2c(C)nnc2C1 N1(C(c2cscn2)C)CCC(=O)N(CC2CC3C=CC2C3)C1=O c1(N2CCC(NC(=O)CCc3cnn[nH]3)C2)nc2cccc(F)c2o1 C1(CNC(CC)=O)CCN(C(C2(C)CCNC2=O)=O)CC1C.C(C)(C)(C)OC(=O)N C1(C)(CNC(c2n(C)cnc2)=O)CN(C(c2cnn(C)c2N)=O)C(C)(C)C1 C1(C(N2CCC(CCNC(C3(CC=C)COC3)=O)CC2)=O)Cc2nccn2C1 CON1CCC(N=c2ncnc3[nH][nH]cc2-3)C1 Cc1cc(C(N2CCCC(c3cncn3C)C2)=O)c(C)cc1Cl O=C(C1CCCc2nn[nH]c21)N1CCN(C(c2c[nH]ccc2=O)=O)C(CF)C1 c1(C(=O)NCC2(F)CCN(C(=O)CC3CSCCS3)C2)cnn2c1OCC2 Cc1cccc(C(CNC(=O)OC(C)(C)C)C(=O)Nc2nnnn2C2CC2)c1 c1(C(=O)NCC2CC(NC(Cc3c(C)nc(SCC)s3)=O)C2)c(C)ccnc1C Cc1nc2c(s1)C(N(C)C(C(=O)NC1CCCC1)C1CCC1)CCC2 CC(Cc1ccccc1)C(=O)N1CC(CCO)(NC(=O)CNc2ncccn2)C1 c1(C(C)NC(C2(CCC=C)CN(C(=O)C(C)NC(C)=O)C2)=O)ccnc(F)c1 C1(C(CN(C(C)=O)C2CC2)(C)C)CCCN1C(=O)CC1(C)CC1 c1(CCCC(=O)NC(C2CCN(C(=O)C=CBr)CC2)C)ccccc1N Cc1ccnnc1C(=O)N(C)CCN1CCN(C(C2CN(C)CCO2)=O)CC1 C12(C(NOCCOCC#C)=O)CCN(C(=O)C(C(C)C)C3CCC3)CCC1C2 c1(CNC2CC(NC(c3ccc(C)nc3)=O)C23CCC3)ccc2n[nH]cc2c1 C#CCCN=C(NCC1CC1c1cccc(F)c1)NC1CCC(C(N)=O)CC1 C1(C(N(CCCCC(=O)NCC(CC)(C)OC)C)=O)CCc2nnnn2C1 CC(C)C(C(=O)NC1CCCN(C(=O)CNC(=O)NC2CC2)C1)C1CCC1 CCC(C#N)(CC)C(=O)NCC(F)CNC(c1cccc2nn[nH]c12)=O C1(NC(c2cnc(CC)s2)=O)C(CNC(=O)Cc2nonc2C)CCC12CCC2 C1(C(=O)NC(C)C(=O)N(C(C(N)=O)C2CC2)C)CC(N=[N+]=[N-])C1 N1(C(C(C(C)C)OCC)=O)CC2CC(C1)C2NC(c1cncc(F)c1C)=O C(N=c1[nH]c(C)nc(C)c1C)C1C2CN(C(COc3ccc(CC)cc3)=O)CC21 C(N=c1nc2sccc2c(N(C)Cc2c(F)cccc2Cl)[nH]1)c1nc(CC)sc1 n1(CC)c(C)nn(CC(N2CC(CNC(=O)C=C(C)Cl)C(O)C2)=O)c1=O c1(OC)cc(C)nc(N2CCCC(CNC(=O)CCC(C)(F)F)C2)n1 c1(C(C(=O)N(C)Cc2cccnc2)(C)N)cccc(Cl)c1 C(Cn1cncn1)(C(=O)NC(C)CN1CCCCC1)NC(C=CC)=O c1(N(CC(=O)OC)C)ccc(NS(C)(=O)=O)cc1.c12nsc(n1)N(C)C2 c1(N(c2cccc(C)c2)C(=O)CN2CCC3(CC2)CNC3)c[nH]c2cc(C#N)ccc12 c1(C(=O)NCCC2(NC(C(CC)N(C)C)=O)CC2)cccc2nncn12 Cc1cccc(C)c1C(O)C(=O)NCCOC1CN(C(=O)CC2CC(=O)C2)C1 CC1CN(C(=O)CSc2ccncc2)CCC1CNC(c1cc(Cl)cnc1O)=O N1(C(C(C)N(C(C)=O)C)=O)CC(C)C(C)(C(=O)NC2CCCC2)C1 N1(C(c2cc(C(C)C)[nH]n2)=O)CC2(CC(CC(N3CC(O)(C(C)C)C3)=O)C2)C1 C(=O)(C(C1=NOC2CC12)N1CC(O)C(F)C1)NCc1c(C)cccc1 C1(OC)CC(CC(=O)OC2CCC(C)CC2)N(C(=O)NC(C)(C)C)C1 Cc1nsc(N2CCC(F)(CNC(=O)C3=NOC(C)C3)CC2)c1C#N Cc1csc(C(C(=O)NC2CCCC2)N(CCC2=CCCC2)C)c1C c1(C(=O)Nc2ccc(-c3c(C)nc(F)cc3)cc2F)cc(F)c(F)c(Cl)c1 N1(C(=O)C2CC2)CC2CC2(C)C1.c1(C(=O)NC2(n3cncn3)CC2)ccccc1F c1(C(N2C(CN(C(C3CCC(C)(CC)O3)=O)C)CCC2)=O)ccsc1S(C)(=O)=O c1(OC)ccc(CCC(=O)N(CC(C)NC(=O)CC2CC=CCC2)C)cn1 C12C3CN(CC13)C(=O)c1cnc(s1)C(=O)N2.CC1(c2cccs2)CSC1 N1(C(C2(C)N(C(CC(CC)C)=O)CCC2)=O)CCCC(OC)CC1 Cc1nc[nH]c1C(=O)NCC1CCC(NC(=O)CCc2ccc[nH]2)C1 c1(C(=O)NCC2CN(C(C(CC)C)=O)CC2(C)C)ccc(Cl)c(S(C)(=O)=O)c1 N1(C(c2nnn(C)n2)=O)CCN(C(c2ccc([N+](=O)[O-])[nH]2)=O)C2CC12 N1(C(=O)OC(CCCCN(C(CCOC(C)=O)=O)C)=O)CC(C)=CC(C)C1 CC1C2CCC(C2)C1C(=O)N(CC(C)C(=O)N(CCO)C1CC1)C C1(OC)CN(C(=O)C(=O)Nc2cn(C)nc2C(F)(F)F)CC1CN(C)C C1(C(N2CC(C(CC)CC)C2)=O)CN(C(C2CCOCC2)=O)CC1C CC1OC2(CNC(C3C=CC=CC=C3)=O)CC1(NC(=O)CN1CCC(C)(O)C1)C2 N1(C(C(COC)C)=O)CCC2(CCCC2NC(=O)C=CCCC=C(C)C)CC1 Cc1nc(CCC(=O)NCCN(C(=O)CNC(c2ccc(Cl)cc2)=O)C)[nH]c1C C1(C2CC2)(OC)CN(C(C2(CNC(=O)CC3C(C)(C)C3(C)C)CCCO2)=O)C1 N1(CC)CCC(C(N2CCCC2C(C)(C)C(=O)N2CCC2C(C)C)=O)CC1 CC(C)(C#N)CC(=O)N1CCC(O)(CNC(=O)CNC(C2CCOCC2)=O)C1 c1(C(=O)OC)cc(F)ccc1NC(C1CCC(NC(=O)C2=COCC2)CC1)=O C(C(F)(C(=O)NC1CC(C#N)C1)C(C)C)NC(C1=C(C)CCC1)=O Cc1[nH]ccc1C(N1C(C(N2CC(OCC(N)=O)C2)=O)CC1C)=O C(CCC(C)C)(C(=O)NC1CN(CC(F)F)C1)NC(CC(CC)C1CCC1)=O Cc1cc(C(=O)NC2CCC3CCN(C(=O)Cn4cnnn4)C2C3)n2ncnc2n1 c1(C(=O)Nc2cccc(NC(c3n(CC)ncn3)=O)c2)c[nH]cc(Cl)c1=O c1(C(=O)NCC2N(C(C(C)(C3CC3)OC)=O)CCC2)c(F)cccc1Cl c1(CN2CC(NC(=O)NCCCN3CCC3)C2)csc2ccc(F)cc12 O=C(C1Cc2ccc(Cl)cc21)NC1CCN(C(=O)CC2CCCC2)CC12CCC2 CC1C(CNC(c2c(C3CC3)cnn2C)=O)CCCN1C(=O)CCCC1CC1 c1(CC(n2cc(CN(O)C(=O)C3CC3)nn2)C)ccccc1 n1(CC)cc(NC(=O)C(C2CCN(C(c3nnsc3N)=O)C2)F)c(C#N)n1 C(=O)(C1=CCC(C)(C)CC1)NCCC(C)NC(c1cc(OC)cc(F)c1)=O c1(OC)cc(C(=O)NCC2C3CN(Cc4c(C)cccc4O)CC23)cc(Cl)c1 c1(C(N2C3CN(C(C(COC)C)=O)C(C3)C2)=O)cnn2cc(C)cnc12 c1(OCC(=O)NC(CNC(CCCOC)=O)(C)CO)ccc(C)cc1OC CON(CCC(=O)N1CC(O)(C2CC2)C1)C(=O)Cn1[nH]cnc1=N c1(OC)ccc2c(c1)CCCC2C(=O)N(C(C)CNC(=O)Cc1cc[nH]c1)C CC(C(C)C(=O)N1CC(C)(NC(c2cn(CCCF)nn2)=O)C1)S(C)(=O)=O C1(CC(=O)N(CCn2ncc(C)c2)C)CCCN(C(c2occc2C2CC2)=O)C1 c1(CN2CC(SC)C2)ccc(I)c(CC(=O)N(C2CCN2)CCC)c1 c1(C(=O)NCC(C2CC2)NC(C(C)SC)=O)ccc2cccc(O)c2c1 N1(C(c2cncc(CC)c2)=O)CC2CN(C(=O)CC3(OC)CCCC3)CC2C1 Cc1cc(C(=O)C(=O)NCC(C)NC(C2(C#N)CCCC2)=O)ccc1F c1(OC(C)C)ccc(C(=O)NCCCCCNC(=O)CC23COCC(C2)C3)cn1 C1(C(N2CCCC(c3cc(OC)c(F)cc3)CC2)=O)COc2ccccc2O1 CCC(CNC(=O)CN(C)C(c1ccoc1)=O)(CC)NC(c1ccsc1C#N)=O c1(C(=O)NC(CNC(CCC=CC(C)C)=O)(C)C2CC2)cc2n(n1)CCNS2(=O)=O c1(C(=O)NCC(CCCC)NC(C2CN(C(C)C)C2)=O)cc(C)ccc1[N+](=O)[O-] N1(Cc2cccc(OCC(=O)O)c2)CCC2C1CCCN2C=O.C1(C(=O)O)CCC1 c1(OC)ccc2[nH]c(C(N3CCCC(N(C)C(c4ccoc4C)=O)C3)=O)cc2c1 N1(C(CCC=CC(C)C)=O)CCC2(CC1)CC(CNC(c1c[nH]ccc1=O)=O)C2 n1(CC(C(=O)CCCC(=O)NCCC(C)NC)=O)nc(O)ccc1=O CC1CN(C(c2cccnc2O)=O)CCN1S(=O)(=O)Cc1ccc(Cl)cc1 S(=O)(=O)(c1cccnc1)NCCC(=O)NC1(C)CCN(C(=O)C=CC2CCC2)C1 c1(OC)cccc(C#N)c1SC1CCC(C)C1 N1(C(N(CC(C)SC)C)=O)CCc2c(C)cc(C)cc2C1 c1(OC)ccc(CN2CC(N(C)C(c3ccc(SC)cn3)=O)C(C#N)C2)cc1O C1(CCNC(CCN(C)C)=O)CCCCN1C(c1cn(CCO)nn1)=O C1(C(=O)NC(C)CO)CN(C(c2ccc(I)c(F)c2)=O)CC(F)(F)C1 c1(C(=O)NCCNC(C2CC2c2cncs2)=O)ccc2cccnc2c1 c1(C(N(C(C)CNC(C2CC2C)=O)C)=O)ccc(Cl)nc1N(C)C C1(CN(C(C(C)OCC(C)C)=O)C)CN(C(C2CC(C#N)C2)=O)CCO1 CC1(C)COC(C(=O)NCCCCNC(C2CC2c2ccccc2)=O)CO1 C1(CNC(C2C(=C)C2)=O)CC2(CC2)CN1C(=O)C=Cc1ncc[nH]1 N1(C(C(C=C)OC)=O)CCC(F)(F)C(CNC(c2c(C)noc2C)=O)C1 C1(NC(c2c(C)noc2)=O)CCS(=O)(=O)C12CN(C(=O)C(C1CCC(=O)N1)C)C2 Cc1nc(N2CC(C)(NC(=O)CCNC(=O)CC(C)C)C2)c2cc[nH]c2n1 c1(C(C(=O)N(CC#C)Cc2ccccc2)N)ccc(OC(F)(F)F)cc1 N1(C(C2CCC(CC)O2)=O)CCN(C(=O)Cn2cc(C#N)cn2)CC(O)C1 C1(CNC(c2cccc(NS(N)(=O)=O)c2)=O)CC2COCC2N1C(=O)C=CBr N1(C(CSC(C)C)=O)CCC(CCC(=O)N(CCC(N)=O)C)C1 N1(C(C(C)(C)OC)=O)CCC(C)C(NC(c2ccc(SC)cc2Cl)=O)C1 C1(C)(CNC(C2(SC)CCC2)=O)CCCN1C(c1cn(C(C)C)cn1)=O C1(N(C(=O)CN2CCC(C(N)=O)CC2)C)CC2CCC(C1)N2C(=O)CCC#N c1(OC)ccccc1CN(CC(c1nnn(C)n1)O)Cc1cccs1 C1(NC(C(C=C)OC)=O)CC=C(C(=O)NC2CC(C)(OC)C2(C)C)C1 n1(C(CC)C)nnnc1C(c1cnco1)NCCc1nc(CC)no1 N1(C(c2ccn(-c3ccc(Cl)cc3)n2)=O)CCC2(CCCNC2=O)CC1 N1(C(C(=O)NC(C)CC)C2(CC)CC2)CCCN(N2CCOCC2)CC1 c1(OC)ccc(C(N2CCCC2(C)C(=O)NCCCc2cccnc2)=O)c(O)c1 c1(-n2ccc(C(=O)O)n2)cccc(OC2CC2(F)F)c1 c1(C(N2CCC23CCCC3)=O)ccn2c(C(F)(F)F)nnc2c1 C1(C(=O)OC)CC2C=CC1N(C(=O)Nc1cccn1-c1ccc(Br)cc1F)C2 c1(C(N2CCCC(CNC(CC(C)C3CC3)=O)C2)=O)coc2c1C(=O)NCCC2 N1(C(C2C(C)(COC)C2)=O)CCCCC12CN(C(=O)Cc1cccc(C)c1C)C2 Cc1ccc([N+](=O)[O-])cc1C(=O)N(C1C2CC3C(=O)OC1C3O2)C1CC1 C(=O)(C(=O)C(C)(C)C)NC(C)CCC(=O)N1CCOCC1CCO c1(CC)ccccc1-c1nc(-c2ccc(CC)cc2)n(CC)n1 N1(C(c2n(CC)nnc2)=O)CC2(CCCN(C(=O)C(C)CS(C)(=O)=O)C2)C1 N1(C(=O)OC(C)(C)C)CCCc2cccc(OCC(C)(C)C(C)(F)F)c21 N1(C(C(C)SC)=O)CCCC1(C)CNC(C1CCC(C(C)(C)O)CC1)=O c1(NC(=O)NC2(c3ccccc3)CCC2)c(Cl)cc(Br)cc1Br C(=O)(CC(F)(F)C(F)F)NCCC1N(C(CCc2c(C)cccc2)=O)CCCC1 C1(CC(=O)N(C(CNC(c2coc(CO)c2)=O)CO)C)SC2=NCCN2C1=O N1(C(Cn2ccc(C)n2)=O)CC2(C1)C(NC(C1CC1F)=O)CCS2(=O)=O c1(CC)cc(C(=O)NC2CN(C(=O)CC(C)OC)CC2(C)C)ccc1Cl Cc1cccc2nc(N(C3CN(C(=O)C(C)(O)C(C)C)C3)C)sc12 C#Cc1ccc(C(N2CCC(CO)C(NC(=O)CC(C)C(F)F)C2)=O)cc1C C1(NC(=O)CCc2ccon2)C=CC(CNC(C2CC=CCC2)=O)C1 N1(C(Cc2c(C)cccn2)=O)CC(NC(c2cnn(C)c2Br)=O)CC(O)C1 C1(C(N(C(C)CN(C(=O)Cn2cccc2)C)C)=O)OCCC1C C1(NC(c2c(C)oc(SC(F)(F)F)c2)=O)CCN(C(C2CC(F)(F)C2)=O)C12CC2 C1(C2CC2)(NC(C2C(CC)CCC2)=O)CCN(C(c2cccc(C(C)C)c2)=O)C1 n1(CC(=O)OCC)cc(C(=O)NC2COCC2NC(C2CCC2)=O)nn1 C1(CC(=O)NC23CC(NC(c4cscc4F)=O)(C2)C3)CCCC1(F)F c1(C(=O)NC(C(=O)NCC(O)C(F)(F)F)C2CC2)cnnc(O)c1 C1(C(N2CCC(OC(C)C)C2)=O)CC12CCC(F)(F)CC2 C(=O)(C1CC(=O)Nc2ccccc21)N1CCN(CC#C)CC1 N1(C(CC2(C=C)CCC2)=O)CCN(C(=O)CNC(c2ccc(F)cc2F)=O)C2CC12 c1(CNC(C2CCCCCC2)=O)ncccc1C(=O)NC1CCCC(O)C1 CN1C(=O)C(=O)N(CC(=O)NC2CCC(CNC(C3CCC(=O)N3)=O)C2)C1=O C(=O)(C(Cc1cnc[nH]1)NC(=O)CC1(C)CCC1)NC(C#C)Cn1cccn1 CCC(C)CC(C(=O)Nc1cc(C)cc(C)c1C)NC(=O)Cc1cncs1 C(=O)(CS(=O)(=O)C(C)C)N1C(CNC(COCCCC(C)C)=O)CC2(CCC2)C1 c1(NC(C2CN(C(CCc3c(OC)cccc3)=O)C2)=O)cc(Br)ncc1[N+](=O)[O-] C(=O)(C1CCCCc2ccccc21)NC12CCC(CNC(CC=C)=O)(CC1)OC2 C1(CCOC)(C(N2CC(NC(C3(C4CC4)CCCO3)=O)C(O)C2)=O)SCCCS1 c1(C(=O)NCC2(COC)CCCN2C(=O)C(C)CC2CC2)cc2cccn2cn1 C1(CNC(c2n(CC)cnc2)=O)CC2CCC(C1)N2C(c1ccc(=O)n(C)n1)=O c1(OC)c(Cl)cc(Cl)c(OC)c1C(N1CCN(C(C2(Br)CC2)=O)CC1C)=O S(=O)(=O)(c1ccc(Cl)s1)N1CC(CC(N2CCCC3(COC3)C2)=O)OCC1 CCC(C)(C)C(=O)C(=O)N1CCC(CC(=O)NC(c2ccn(C)n2)(C)C)CC1 C(=O)(C(C)(C)CC(C)C)N1CCC(C(C)(C)NC(C2N(C(C)=O)CC(O)C2)=O)C1 c1(C(N(C(C)CN(C(=O)C=CC2CCCO2)C)C)=O)ccc(F)c(S(C)(=O)=O)c1 Cc1cc(=NCCCCNC(=O)CC2CCC(C(F)(F)F)O2)[nH]cc1C#N CC1COc2c(C(N3CC(O)(CCNC(=O)C(F)(F)CC4CC4)C3)=O)cccc21 C=CC(C)(O)CC(=O)NC(C(=O)N(c1ccc(OC)cc1)C)C(C)(C)C c1(CCC(=O)NCC2C(NC(C=C(C)C)=O)CCCC2)cccc2cnccc12 n1(CCOC(C2CCC(C(=O)OC(C)(C)C)C2)=O)c2ccccc2c2ccccc12 CON(CCC(=O)NC1(CCO)CCOC1)C(=O)C(C)CCC(C)(C)C C1(CNC(=O)Nc2ccc(OC(C)(C)C)cc2F)COc2ccccc2O1 N1(C(C(OC)OC)=O)CC(C)N(C(=O)CCc2cc(Cl)cc(Cl)c2)CC1C c1(C(=O)N(CCN2CCCC2)C2CC2)cccc[n+]1[O-].C12(CC1)C(=O)N2 c1(CC(=O)NC(CCCNC(C2C(CC)C2)=O)(C)C)c(F)cccc1F CC(CC(F)(F)F)N(C(=O)CCC1CCN(C(C2(C)CC(C)(C)C2)=O)CC1)C c1(C(N(CC(=O)NC(CCC)CO)C(C)C)=O)nnc(S)n1C n1(CC)ncc(C(N2CCC(N3CCN(C(=O)CP(C)(C)=O)CC3)CC2)=O)c1Cl CCCC(C(=O)NCCC(F)(F)C(C)C)C(C)C.c1(Cc2nnn[nH]2)ncccc1Br N(C1CN(C(C2CCC(F)(F)C2)=O)Cc2ccccc21)C(=O)CC1CC1 c1(C2CC(C(N(CCCNC(=O)C(C)C#N)C(C)C)=O)C2)ccc(F)cc1 c1(C(=O)NC2(CCNC(c3cn(CCOC)nc3)=O)CCC2)nc(C)ncc1Cl Cc1[nH]nc2c1CC(C(N1CCN(C(c3cnc(O)nc3O)=O)CC1C)=O)CC2 N1(C(C(F)OC)=O)CCCC2(CNC(=O)CCSC)CCCC12 Cc1ccccc1CCNC(N1CCOC(c2cccc(Br)c2)C1)=O C1(NC(CC=C)=O)CCN(C(c2ccc(-c3cn[nH]c3)c(Cl)c2)=O)CC1(C)C CC1CCOCC1C(=O)NCCCCCN(C(=O)C(N)=O)C CCCC(C(=O)N(C1CCC1)CCN(C)C)NC(c1ccsc1C#N)=O N1(C(CCC=CCC=C)=O)C(C(=O)NCCC2CCCN2C)CCC12CC2 c1(C(N2CCC(N(C)C(C3CC(O)C3)=O)C2)=O)ccc(=O)n2c1CCC2 N1(C(c2n[nH]c(CC)c2Br)=O)CCC(NC(=O)CC2CCOC2)C(C)(C)C1 N1(C(C(C)C(C)(F)F)=O)CCCc2ccccc21.c1(C(NO)=O)cc(=O)n(C)c(=O)o1 Cc1nc(C(=O)N(C2CN(C(=O)C(C)NC(c3ccccc3)=O)C2)C)n(C)n1 C12(C(=O)NC(c3noc(C)n3)CC)CC(C)(CN1C(=O)CN1CCC(=O)CC1)C2 n1(CC)ccc(CC(=O)NCC2CCCC2C(=O)NCC2CC(OC)C2)n1 c1(NCc2c(C)nccc2)[nH]cnc2nc(Br)cc1-2.N12CCC3(CC1)CC3C2=O C(=O)(CCCCC(=O)NC1CCC(C)N(C(C2CC2C(C)O)=O)C1)NC c1(CC)nccn1C(C)CC(=O)NC(C)CC1CN(C(=O)C(C)C2CC2)C1 C1(CNC(c2n(C)nc(C(C)(C)C)c2)=O)CN(C(C2CCCC2O)=O)CC1(F)F C1(CNC(c2cn(CC(=O)NC)nn2)=O)CCCCCN1C(C1C2CCCC12)=O CCCC(C)CC(=O)NCC(=C)CCNC(=O)C(C)OCCOC C1(CN=C(NCC2C(C)C2C)NC2CC2)CC2CCC1CC2 N1(C(C2CCC(OC)C2)=O)CC(=O)NCC1C(=O)NCC1(CCO)CC1 c1(C(=O)NC2CC(CNC(CC(OCC)OCC)=O)C2)cnc(C(F)F)cc1C c1(OC)cccc(CC(=O)NC(C)C(C)NC(C)=O)c1C.c12cc(ncn1)OC2 C1(C(F)(F)F)(OCC)CN(C(=O)Nc2coc(CC)n2)C1 C(c1ccccc1C#N)=CC(=O)NC1CC(C)CN(C(=O)C=CC2CCCO2)C1 N1(C(C(=O)NC(CN(CC)CC)C)=O)Cc2ccc(C)c(Br)c2C1 c1(C(=O)NC2C(C)CN(C(C3CC(C(F)(F)F)C3)=O)C2)ccc(=O)n(CCO)c1 c1(N(C(=O)NC(C)CS(C)=O)C)ccnc(O)c1 C1(C(=O)Nc2cccc(CNC(C34COC(CF)(C3)C4)=O)c2)CCC2(CCC2)O1 C1(NC(=O)CCC(F)F)CC(F)CN(C(c2cn(C3CCOC3)nn2)=O)C1 c1(C(N(CCNC(CN2C(C)CC2)=O)C)=O)nnn(-c2ccccc2)c1C(F)F C12(CNC(COC(CC)C)=O)CC(CN1C(c1cc[nH]c1C(C)C)=O)C2 CN1CC=C(CC(=O)N2CC(NC(=O)CC3CCSCC3)C(C)(C)C2)CC1 C(=O)(C(C#N)C(C)(C)C)N(CCNC(C1CCCC12CC2)=O)CC c1(C(C(=O)NCCCC)N(CCCO)C2CC2)cccc(OCC)c1 C1(C(=O)OC)CC(C)CN(N2CC(C(C(=O)NC3CC3)OC)C2)C1.C(=O)C=CC1CC1 N1(C(C)=O)CCC(Nc2cccc(F)c2[N+](=O)[O-])c2cc(F)ccc21 C1(n2c(-c3cc(F)c(F)cc3OC)nc(CCCC)n2)CCc2nc(C)nn2C1 C(CNC(C1(O)CC1)=O)(CC(=O)NC(c1cnc(C)s1)C)OC C1(C(=O)NCCC(C(=O)OC)C)N(C(c2csnn2)=O)CCCC1(C)C C(=O)(CC(C(F)F)n1cccn1)NC(CNC(Cc1n(C)cnc1)=O)C1CCC1 N1(C(C(CC)OCC)=O)CCN(C(C2CC(C(F)(F)F)C2)=O)C(C)C1 c1(NC2CCc3n(CC)ncc3C2)[nH]c(=NC2CCSC2)nc2scnc12 C1(CCNC(c2cccc(CC)n2)=O)CN(C(C2CC2C2CC2)=O)CCS1(=O)=O C(=O)(C1CC(=O)Nc2cc(F)ccc21)OCCCC(=O)OC(C)C1CC1 C(c1ccc(Cl)cc1F)=CC(=O)NC1(CCNC(C(CC)(C)CC)=O)CCC1 N1(C(CCSCCC)=O)CC2CS(=O)(=O)CC2(CNC(c2nnn(C)n2)=O)C1 c1(C(C)CNC(=O)C(=O)N2CC(n3ccnc3)C2)ccccc1 c1(C(=O)NC2C3CN(C(c4cnc(OC)s4)=O)C2C3)ncc(N)cc1C Cc1nc(CNC(C2(NC(C3CC3C(N)=O)=O)CC2C)=O)no1 C1(CN(C(=O)CCn2ccnc2)CC)CCCCN1C(=O)Cn1cnnc1 CC(C)CC(C(=O)NC1CC(CN(C)C)C1)NC(=O)C(C)(C)C C1(C(=O)NCCC(C)N(C)C)CC12CCN(C(C1(C)CC3CC3C1)=O)CC2 c1(SC)ccc(C)c(C(=O)N(C(C)CCNC(C2(CO)CCCO2)=O)C)c1 c1(C(=O)NC2C(NC(COCC=C)=O)CCCC2)cnc2sc(C)cn2c1=O C1(C)(NC(c2scc(C)c2)=O)CCN(C(C2CCCC2C(C)C)=O)CC1 C(=O)(C(C)Cc1ccco1)N(CCCCNC(C1CC(C)C1)=O)C C#Cc1cncc(C(N2C3CCC2C(CNC(=O)CC2(C)CCC2)C3)=O)c1 C=CC1CN(C(c2csc(-c3ccoc3)n2)=O)CC1NC(C1(C)COCCO1)=O c1(C(=O)OC)cc2ccc1-2.c1(C2CNC2)cccc(C(C)C)c1 c1(C(=O)NC2C(NC(CCC=C=C)=O)CCOC2)cccn(C(C)(C)C)c1=O C(C(F)(C(=O)N(CC(C)(C)COC)C)C(C)C)NC(c1c(C)cc(CC)o1)=O CCC(CC)OCC(=O)NCC(C)CNC(C1CC(OC(F)F)C1)=O C1(C(=O)NC(C2CCCC2)C#C)(COC)CCCN1C(=O)Cc1cc[nH]c1 C12(CNC(C3(N(C)C)CCC3)=O)CC(CO1)N(C(C1CCCS1)=O)C2 C1(N(C(C=C(C)C(C)C)=O)CC2CCCC2)CCC(NC(c2cnoc2C)=O)C1 N1(C(C=CCOC)=O)CCC2(CC2NC(=O)Cc2ccn(C(C)C)n2)C1 N1(C(C2N(C(C)=O)CCC2)=O)C2CCC1(CNC(=O)C=Cc1ccc(C)s1)CC2 c1(C(=O)NCC#CCNC(c2cnc(C(C)(C)C)s2)=O)cscc1C#N c1(C(=O)NC2C(C)CN(C(C3(C#N)CC=CC3)=O)CC2)ccn2c1CCCC2 Cc1cccc(C(N2CCCC2CN(C)C(C2CC3CC2CO3)=O)=O)c1C Cc1cc(C(F)(F)F)c(-c2nccnc2C(=O)Nc2cccc(C)c2I)cc1C C(=O)(C1=COCCC1)NC1CC2(C(NC(=O)Cc3cc(C4CC4)on3)C2)C1 c1(C(N(CC(C)NC(=O)CCN(CC(F)(F)F)CC)CC)=O)ccc(OC)cc1 C(=O)(C1=CCN(C(=O)CCCOC)C1)N(CC(COC)O)C C=C(C)CCC(=O)N1CC(F)CC1CN(C(=O)C(C(C)C)c1ccn(C)n1)C c1(C(=O)NC2CC(CNC(C(CC)SC)=O)C(O)C2)c(C)cc(C#N)cc1C C(CCC(C)C)(C(=O)NC1CC(CSCC2CC2)C1)NC(CN(CC)CC)=O c1(C(=O)NC(CCCNC(CCC(=O)NCC)=O)C)ccc(C#N)c(OCC)c1 Cc1c(C(=O)NCC(O)CCNC(=O)CC2CC(C)C2)nnn1-c1ccccc1 C1(NC(COC(C)C)=O)CC2CC1N(C(=O)Cc1cccnc1)C2 c1(C(N(C)C)=O)ccc2cnccc2c1.C12CC(C1)NC(=O)CS2 C1(N2CCC(OC)C2)CC2CC1CN2C(=O)C(C)(C)CF C(=O)(C1CCC(=O)c2cccn21)N1CCC(NC(c2n(CC)ncn2)=O)C1 O=C(CC1NC(=O)c2ccccc21)NCC1(O)CCN(C(c2coc(Br)c2)=O)C1 c1(Cc2nn(OC)c(Br)c2)ccc(C)c(-n2cc(CN(O)C(=O)N(C)C)nn2)c1 c1(C(=O)NC(C(C)NC(C(CC=C)CC)=O)(C)C)ccc2c(c1)NCC2 c1(CC)nc(C)n(C)c1C(=O)NCC1CN(C(=O)CCC2(C#N)CCC2)CC1C C(=O)(C(C)(C)F)N(CCOC1CN(C(C(C)N(C(C)=O)C)=O)C1)CC1CC1.CN c1(CNC(N2CCCN(S(C)(=O)=O)CC2)=O)ccc2c(Br)cccc2c1 c1(CN=C(NC(CC)C)NCC(C)(C)OC(C)C)ccc2c(c1)CCCS2 C1(C(N(CCN(C(=O)C(c2ccccc2Cl)O)C)C)=O)CCOCC12CCCC2 C1(NC(c2nccc(CC)c2)=O)CN(C(=O)CCc2ccc(C)s2)CC1(C)C C1(C(N(CC(CC)(F)F)C)=O)CC2(CC(NC(C3(NC(C)C)CC3)=O)C2)C1 CC1CN(C(C2CCC(F)(F)C2O)=O)C(C)CN1C(=O)C=CC(C)(C)C N(C(=NCCCCl)NC1CCCN(C(C)=O)C1)CC(C(=O)NCC)(C)C Cc1cc(C(N2CCC3C(NC(=O)C(N4CCSCC4)C)C23)=O)cc(C(F)F)c1 c1(CC(N2CC3(CC(NC(CSCC(=O)OC)=O)C3)C2)=O)nc2ncccn2n1 C(=O)(CC(C)C(=O)OC)NCCCCn1cc(CCCN(C(C)=O)C)nn1 CN1CCCCc2ccc(NC(=O)Nc3cnn(-c4ccccc4Cl)c3)cc21 C=CCCC(CO)NC(=O)C(C)OC1=CCCC1.c1(CNC)ccccc1 C=C(C)C(CC(=O)Nc1ccc(NC(=O)C(F)CC)c(F)c1)OCC CC1CN(C(=O)OC(C)(C)C)CC(C)S1.c12c(ncn1C1CC1)NC2=O c1(NC(c2c(CC)ncn2C)=O)cc(C(F)(F)F)cc(SC)c1 CC1C(NC(=O)CSc2cnn(C)c2)CCN1C(C1CC2CC2C1)=O Cc1nc(COC2C(CNC(CSC3CCCC3)=O)C2)cs1.C12CCN1C2=O N1(C(C(C)SC)=O)CC2(CCN2C(c2cnn(C)n2)=O)C1 C=CCCC(C(=O)NCC1(CC2CC2)CC1)NC(=O)CC1CN2CCC1CC2 C1(C(=O)Nc2ccc(C)nc2Br)CC12CCN(S(=O)(=O)CCBr)CC2 Cc1nc(NC(c2cccc(-c3cnn(CCO)c3)c2F)=O)cnc1C#N c1(CC)c(C(=O)NC(C)(C)CCCNC(c2nc(C3CC3)sc2C)=O)ccn1C C=CC1(C(=O)NC2CC2NC(c2cc(CC)ccn2)=O)CCCCC1 CCCCC(CNC(=O)CCCF)NC(C1(C2CC2)CCCO1)=O c1(C(N2CC=CC2CNC(C2CC(O)C2)=O)=O)cc(Br)c2nccn2c1 C1(OC)CC2(C1)CC(NC(=O)NCC1CCCC(=O)N1C(=O)OC)C2 CC(CN=c1ccnc(NCC2CSCCS2)[nH]1)n1cccn1 C1(C(=O)NCc2cccc(F)n2)(OC)CCN(C(=O)CC(Cl)Cl)C1 CCC(O)C(C)C(=O)N(CCCNC(=O)CCn1cc([N+](=O)[O-])cn1)CC Cc1conc1C(=O)N(CCC(C)NC(c1ccoc1C1CC1)=O)C N1(C(C2(OC(C)=O)CC2)=O)CCC(C(=O)NCc2nn(C)c(=O)o2)C(C)(C)C1 N1(C(C(C)n2cncn2)=O)CC2(C1)SCCC2NC(=O)Cn1ccc(C2CC2)n1 CCC(CC)C(C)C(=O)NC1(C(=O)NCCCN2CCC2)CCC(C)(C)C1 N1(C(c2n(CC)nnc2)=O)CC2(C1)CN(C(c1cc(-c3csc(C)n3)c[nH]1)=O)C2 CCC(CC)CC(=O)NC(CC(=O)N(C)Cc1c(C)noc1C)C(F)F C1(CC)CN(C(=O)CSc2nnnn2C)CCC1NC(=O)CC1CCC(C)CC1 c1(C(N(C)CC2CCCN(C(=O)C(C)(C)C)C2)=O)ccc([N+](=O)[O-])cc1Cl N1(C(CCC(C)OCC)=O)CCN(C(=O)C(C)(F)F)CC1C1CC1 C#Cc1cn(C)nc1C(N1CC(CCNC(c2ccc(F)cc2O)=O)C1)=O C(=O)(NN1C(=O)NC2(CCCCC2)C1=O)Nc1c(C(C)(C)C)cccc1 c1(C(=O)NC2(CNC(C(C)OCC(F)(F)F)=O)CC2)cc(Cl)c(N)c(Cl)c1 N1(C(C2C(C)=C2)=O)CCC2(CCCN(C(c3cc4cccnc4cc3N)=O)C2)C1 N1(C(CCc2ccc(C)o2)=O)CC2(CC(NC(c3ccc(Cl)c(C)c3)=O)CO2)C1 c1(C(N(C2CCN(C(c3coc(Cl)c3)=O)C2)C)=O)cc2n(n1)CCCC2O N1(C(c2cc(COCCOC)on2)=O)CC2(CCCC2NC(=O)C=CBr)C1 c1(C(N2CC(n3cc(CCCC)nn3)C(O)C2)=O)ccc2c(c1F)CCC2 Cc1cc(CNC(c2csc(Cl)n2)=O)oc1C(=O)Nc1cccc(O)c1 c1(CC(C(=O)NC(C)CCCNC(c2ncncc2Cl)=O)O)c(F)cccc1Cl O=C(CCC(CF)CF)NCC1(O)CN(C(c2ccnn2CC2CC2)=O)C1 CC(C)CC(O)C(C)C(=O)N(CCN(CCS)CC)C.C(C(C)S(C)(=O)=O)C1CC1 C(=O)(CCCC(CC)NC(=O)CNC(=O)C(C)(C)C)NCCS(CC)=O c1(N(C)CC2CCC(=O)N2)nc(N2CCC(C(F)(F)F)CC2)nc2c1ncn2C Cc1ccc(C(=O)NC2CCN(C(C34CC(C3)S(=O)(=O)C4)=O)C(C)C2)cc1C CCCC(C(O)C(=O)NCCc1cccs1)NC(=O)Cn1ncn(C)c1=O C(=O)(C1=NOC(C)C1)NC1C(NC(C(c2ccc(CC)s2)=O)=O)C1 c1(C)ccc(Cl)cc1Cl.C1(OCCNC(c2ccco2)=O)CN(C(=O)CO)C1 S(=O)(=O)(c1ccc(NCc2ccncc2Cl)c(Cl)c1)N(C1CC(C)N(C)CC1)C c1(OC)ncnc(C(=O)NCCN(CCOC)C(c2cncc(C#N)c2)=O)c1F c1(C(=O)NC2(C)CCCN(C(C3CN4CCC3CC4)=O)C2)cccc([N+](=O)[O-])c1 C1(CC)CCC(C(=O)NC2CN(c3ccnc(-c4ccccc4)n3)CC2F)CC1 Cc1cccc2c1N(C)C(=O)C2NC(=O)C(=O)C1(C(=O)O)CCC1 C1(C2CCN(C(C3CCCN3C(C)C)=O)CC2)(NC(CS(=O)(=O)NC)=O)CC1 O=C(C1COc2ccccc21)NC1C=CCN(C(C2CCC(O)CC2)=O)C1 C(=O)(CC(C)(C)C(=O)NC1CCCC1(C)CNC(=O)CC1CCC1)OCC C1(CNC(Cc2c(C(N)=O)cccc2)=O)CC2(CC2)CN1C(C1CCSCC1)=O c1(OC)ccc2c(c1)N(C(=O)COC(C)(C)C)CC(C)(C)O2.C1C(C)NC(=O)N1 CN1CCn2ncc(C(=O)NCC(F)CNC(c3ccc([N+](=O)[O-])cn3)=O)c2C1 C=CC1CN(C(C2CCNC(=O)C2)=O)CC1NC(C1(COCC)CC1)=O c1(N(CC(N2CCCC2)C)C)ccc2cc(S(=O)(=O)NCC3CC3)ccc2n1 C(CN=c1nc(-c2ccc(C)cc2)[nH]s1)=CCNC(C(C1CCCC1)OC)=O CC(C)(CC(=O)N1CCN(C(c2ocnc2C2CC2)=O)C2CC12)C(F)(F)F C(CCCCCC(=O)NC1(C)CCN(C(=O)Cc2cc(C)no2)C1)SC c1(C2CC(c3n(CC)nnn3)(NCSc3nccc(C)n3)C2)ccc(Cl)cc1C N1(C(c2cc(Cl)ccc2F)C(=O)NCCC2CC2)CCCc2[nH]ccc2C1 c1(C(N2CC(OC)C(NC(=O)C(F)F)C2)=O)nc(C)n2ccccc12 N1(C(c2ccc(SC)cc2)=O)CC(NC(=O)C(C)Cn2cccn2)C(C)(C)C1 c1(CSCCc2nnc(C(=O)OC)s2)coc2c(Cl)cc(Cl)cc12 N1(C(C2N=C(C)SC2)=O)CCCC(C(=O)NCc2ccc(N3CCCC3)nc2)C1 N1(C(CC2(C)N(C(c3ccc(CC)[nH]3)=O)CC2)=O)CCCC2(CCOC2)C1 C(=O)(C(O)CCCNC(=O)C(c1cccn1C)=O)NCCCCC1C(C)C1 Cn1cc(NC2CCCC(CO)C2)cc1C(c1ccccc1)=O C(=O)(C(C)(O)CNC(C1(C)CN(C(=O)CCN(C)CCO)C1)=O)OC O(NC(=O)C1=NOC(COc2cc(F)cc(F)c2)C1)C(C(C)C)COC(F)(F)F C1(CC(=O)NC(CCC=C)C2CC2)C2CCCC2N1C(=O)CC1CSCCO1 N1(C(c2ccc(SCC)cc2)=O)CC2CC(C)N(C(=O)C(C)(F)C(C)(C)F)C2C1 C=CC(C)(CCOC)C(=O)N1Cc2occ(C(=O)NCC3(CO)CC=CC3)c2C1 c1(C(N2CCC(CC=C)(NC(c3ccco3)=O)C2)=O)cc(F)ccc1Br C#Cc1cn(C)nc1C(=O)NCC1(O)CN(C(C2CCC2C)=O)C1 CC1(CNC(c2cnc(C3CCC3)s2)=O)COCCN(C(c2csc(=N)[nH]2)=O)C1 c1(CCC(=O)NCCNC(c2n(C)cc(C(N)=O)c2)=O)ccc2[nH]ccc2c1 c1(C2C(C(N(CCCNC(C=C(C)C)=O)C)=O)C2)cccc(C)c1 Cc1nc(N2CCC(C(C)NC(=O)CC3CC3(C)C)C2)cc(Cl)n1 c1(NC)ccc(Cl)c(C(N2CC(C3CN(C(=O)CCOC)CCO3)C2)=O)c1 C1(NC(C2CC(C)(C)C2)=O)CCCCCC1CNC(=O)COC1(C)CCC1 Cc1cc2c(cc1C(N1CCC3(CC1)CC3NC(c1occc1Cl)=O)=O)OCO2 c1(N2CCC(C)(NC(C3CC3(F)F)=O)C2)ncnc2scc(Br)c12 C#Cc1c[nH]nc1C(=O)NCCN(C(C1CCN1S(C)(=O)=O)=O)C1CC1 C(=O)(N=c1ccn(C2CN(c3ncccn3)C2)[nH]1)c1ncc(-c2c(C)ncs2)nc1 C(=O)(C(Cc1ccccc1)CC)N(CC(CC)NC(C1(c2cccs2)CC1)=O)C c1(C(=O)NC(C2CCN(c3ncccc3[N+](=O)[O-])CC2)C)cc(F)c(F)c(F)c1 N1(C(c2cnc(Cl)s2)CC)CCN(C(c2ccc(F)cc2)CO)CC1 c1(NC(=O)NC2(Cc3ccnc(Cl)c3)CCC2)ccc(Cl)cc1Cl N#Cc1cc(C(=O)NC2COCCN(Cc3c[nH]c(Br)c3)C2)ccc1Cl c1(OC)cc(N)c(C(N2CCC(C(C)C(N)=O)CC2)=O)cc1OC C1(C(=O)OCc2ccns2)CCCN1C(c1cc[nH]n1)=O c1(NC(CC2CC(NCc3ccc(C(C)=O)o3)C2)=O)nccnc1Cl c1(C(N(CCCCN(C(=O)C(C2CCCO2)C2CC2)C)C)=O)ccnc(F)c1F C1(CCOC)(NC(c2cnc(O)cc2C)=O)CCN(C(=O)C(COC)SC)CC1 c1(C(=O)NC2CCCC(CNC(CCC=CC)=O)C2)ccc(OC)c(F)c1N Cc1cncc(C)c1C(=O)N(CC(C)C(=O)NCC(N1CCCCC1)=O)C CCCC(CNC(c1cc(Br)sc1C)=O)C(=O)NC1CC(=O)N(C)C1=O N1(C(C)=O)CC(C)(C(=O)NC(C)(C)C(=O)NCCCCC(C)C)C1 c1(OC)cc(F)c(C(N2CCC(C(C)NC(c3nnn(C)n3)=O)CC2)=O)c(Cl)c1 N1(C(C(C)Sc2cccs2)=O)CC2CN(C(=O)C(Cl)Cl)CC12.C1C(=O)N1 C1(CNC(C(C)=C2CCCC2)=O)C2CN(C(C3(C)CCCCO3)=O)CC12 c1(C(C(=O)NCCC)N(c2ccccc2)CCN(C)C)nc(C(C)C)cs1 C(CNCCCn1ccnc1C)(CC(C)C)OC C=CCCC(C(=O)NC1CC(CC)C1)NC(C1CC(F)C(=O)N1)=O c1(CNC(CSSC)=O)ccnc(N2CCN(C(C3CCCC(=O)N3)=O)CC2)c1 N1(C(c2cnc(CC)s2)=O)CCC(N(CCOC)C(c2cc(C3CC3)on2)=O)CC1 C1(C(N(C)CC2(C)CCC2)=O)CCCN(Cc2ccc(CC#N)cc2)C1 C1(C(=O)NCC2CCCN(C(CS(=O)(=O)NCC)=O)C2)CNC(=O)CC1(C)C Cc1nc2cc(C(N3CCCCC(NC(c4sncc4C)=O)C3)=O)cc(O)c2o1 C(CC(=O)N(CC(F)(F)F)CC(C1CCCC1)O)OCCCOC.C1(=O)C(C)N1 Cc1ccc(Br)c(CNC2(CC(=O)Nc3cnc(Br)c(F)c3)CCC2)c1F c1(CNC(C(N2CCOCC(C(=O)N(C)C)C2)C(C)C)=O)ccnc2ccnn12 C1(CNC(=NCCC)NCC(c2cnn(C)c2)C)CC2(CO1)CC(OC)(OC)C2 c1(C(N2CCC(C(CC)C)C2)=O)cccnc1CNC(C1CC(=O)C1)=O C12(C(=O)NC(CC)(C3CCC3)C3CC3)CCCC1CN(C(=O)Cc1ccns1)C2 C(=O)(CCCC(F)(F)CO)N1CCCC(N(C(COCC)=O)C)CC1 C1(CCOC)CN(C(=O)COCCOCCNC(c2ncc[nH]2)=O)CC(C)O1 C1(NC(c2n(CCC)nc(C)c2)=O)CN(C(=O)C(C)=CC2CC2)CC2CCCC12 c1(-n2cc(CN(C(C3CCC3)C)CC)nn2)cccc2n[nH]cc12 c1(C(=O)NCC2N(C(CCCSC)=O)CCOC2)ccc(C(F)F)cc1F c1(C(=O)NC(CNC(c2nc(CC)oc2)=O)(C)C2CC2)cnn2ncccc12 C1(N(CCN2C(=O)CCC2)C(c2cncc(C3CC3)c2)=O)CC2(CCNCC2)C1 N1(C(COCCCC#C)=O)CCC(NC(c2c[nH]c(=N)s2)=O)CC1C Cc1sc(C(N2CC(NC(C3(CF)COC3)=O)CC(O)C2)=O)cc1[N+](=O)[O-] c1(CC(=O)NC(CNC(c2nc(C)n(C)c2C)=O)C(C)C)ccc(F)c(Cl)c1F N1(C(c2c(C)cccc2)=O)CCCCCC(NC(c2ccncc2F)=O)C1 N1(C(=O)C=Cc2cccnc2)CCC(N=c2nn[nH]n2Cc2ccccc2)C1 CCC(CNC(c1cc(Cl)cs1)=O)(CC)C(=O)NC(c1ccccc1)C C1(NC(C(c2ccc(C)cc2)C)=O)CN(C(=O)CNC=O)CC(F)(F)C1 Cc1cc(C)c(C(=O)NC(C)CC(C)NC(C23CC2COC3(C)C)=O)c(N)c1 c1(C(N2CCN(C(c3c(CC)c[nH]c3)=O)C3C2C3)=O)nn2ccccc2c1Br c1(OC)ccc(F)c(CNc2cnc(F)cc2C(=O)Nc2cc(Cl)nc(Cl)c2)c1 O=C(C(CCC1CC1)NC(C1CC1C(F)(F)F)=O)NCC1CC1(F)Cl C1(CNC(C2CC(NC(c3n(C)ncc3)=O)C(O)C2)=O)CC2C(C1)C2(F)F c1(SC)ccccc1CC(=O)N(C1CCCC(N(C)C(c2ccc(Cl)o2)=O)C1)C c1(C(=O)N(C(C(CC)NC(=O)OC(C)(C)C)C)CCO)cnc2cc(C)ccc2c1 C1(NC(c2ccc(Oc3ccc(C)cc3)cc2)=O)C2C=CC(C2)C1S(C)(=O)=O c1(C(=O)NCCCN(CCC)C(C2CC(=O)CS2)=O)cnc2n1CCC2 Cc1cc2sc(C(N3CCC4(C3)CN(C(c3cc(=N)[nH]c(Cl)n3)=O)C4)=O)cc2s1 N1(C(c2cc(C(F)(F)F)ccn2)C(=O)NCCC#N)CCCC2(CCC2)C1 c1(C(c2n(C(C)(C)C)nnn2)NC(N2CC(c3ccon3)C2)=O)cccc(Br)c1Cl c1(C(N(C2CCN(C(c3nc(=N)cc[nH]3)=O)C2)CC)=O)cc([N+](=O)[O-])oc1C C(N=c1[nH]n(C)c2cccnc12)c1cccc(-c2ccc(OC)cc2)n1 C1(CC(N2CC(C)C(NC(=O)Cn3ccc(Br)n3)C2)=O)CCC(C)(C)CC1 c1(C(N(C(C2(O)CC2)=O)CC)C)c(F)cccc1F.C1(C(F)(F)F)(C)N=N1 c1(CN2CC(C)(C(N(C3CCS(=O)(=O)C3)CCCC)=O)C2)cc(F)c(O)cc1F C1(C)(C(=O)NCC(CCCC)NC(=O)C(=O)NC(C)C)CCN(C)C1=O C12(C(N(CCN(C)C)C)=O)CCCC1CCN2C(c1nnc(S)n1C)=O C1(C(N(CCNC(CC2(C=C)CC2)=O)CCC)=O)CCc2ccc(F)cc2C1 c1(NC(c2scc(CNC(C3C(C)C3C)=O)c2)=O)cccc(CN(C)C)c1 C(=O)(CC(C)CF)NC(C)CCNC(c1ccc(C(N)=O)o1)=O N1(C(C2CC(C)(C)OCC2)=O)CCC2(CCC2NC(=O)Cn2ccnn2)CC1 c1(CC)ncnc(CC)c1C(N1CCC(CN(C(=O)Cn2nnc(=N)[nH]2)C)C1)=O CC(C)C(CCN(C)C(c1cc(Br)co1)=O)NC(=O)C(C)(C)c1nncn1C CC(C)(CN=c1ccc(S(=O)(=O)N2CCCSC2)c[nH]1)SC(F)(F)F C1(C(=O)NCCC(C)(C)F)CCCCN(C(=O)C2=C(Cl)CC2)C1 n1(CC)nc(C)c(C(N2CC(C(N3CCC(C)(C)C3)=O)CC(C)C2)=O)c1C c1(CC)oc2ccccc2c1C(=O)N(C)CCNC(c1ccnc(O)c1)=O C1(F)(CNC(C2(OC)CCC2)=O)CCCN(C(=O)C(F)C(C)(C)O)C1 C1(C(=O)NCC(C)CNC(C23C4CC(CC24)C3(F)F)=O)CCC2C(C1)C2(F)F c1(C(N(C(CNC(C=CCOC)=O)CC)C)=O)ccc(OC(C)(C)C)cn1 Cc1nc(C#N)cc(=NCC(CNC(C2CC23CC(C)(C)C3)=O)C(F)(F)F)[nH]1 C1(OC)CCCCN(CCN(c2ccccc2)C(=O)N(CC(O)C(F)(F)F)C)C1=O c1(C(=O)NC(CNC(c2cc(C(N)=O)[nH]n2)=O)C2CC2)cc2c(nn1)CCOC2 N1(C(C2=CC(C)(C)C2)=O)CCC2CC1CN(C(C1CCC(C)(C)OC1)=O)C2 C(=O)(C1=C(Cl)CCC1)N1CC(CNC(c2cc(-c3ccco3)[nH]n2)=O)C(O)C1 c1(CC(=O)NC2CC23CCN(C(C2CCCCC2)=O)CC3)noc2ccccc12 C(CC(C(C)(C)C)NC(=O)CNC(=O)CN(C)C)N(C(C(CC)(F)F)=O)C C1(NC(=O)Cc2cccc(C(F)F)c2)CN(C(=O)C(O)C2CC2)CC12CCC2 Cc1nn(C)c(N)c1C(=O)NCC1CC(C)N(C(=O)Cn2cc[n+](C)c2)C1 c1(C(N2CCC(n3cc(CCCSCC)nn3)CC2)=O)ccnc(OC)c1Br C(=O)(C(F)CC(C)(C)C)NCC(C1CCOC1)NC(c1cncc(CC)c1)=O Cc1cc(C(=O)NCC(O)CN(C)C(C2CCC(=O)N2)=O)ccc1Br c1(C(C)C)ccc(N)c(C(=O)NC2CN(C(=O)CN(C3CCSC3)C)CC2C)c1 c1(SC)cccc(-c2nc(C(=O)NCc3ccc[nH]3)c(C)s2)c1F N1(CSCc2cn(C3CC(CNC(CCCCSC)=O)C3)nn2)CCC(C#N)CC1 C1(CC#C)(C(N2CC3CC3(NC(c3cc(C4CC4)on3)=O)C2)=O)CC=CCC1 c1(C(=O)NC(C2CCCN(C(c3ncccc3Br)=O)C2)C)cc(I)c(F)cc1F C(=O)(CCCC(C)(C)C#N)N(CCNC(c1cn2c(n1)CC(C)CC2)=O)C(C)C c1(C(N2CC3CC(NC(c4nc(C)[nH]n4)=O)CC3C2)=O)cc2c(s1)CC(C)(C)C2 C1(C(=O)NCC(C(C)C)NC(=O)COCCOc2ccccc2)C2CCCCC12 c1(C(N2CCC(C(C(=O)NC3(CC)CCOCC3)C)C2)=O)cccc(O)c1F c1(OCCCC)ccc(CNC(C2C=CCN2CC)=O)cc1OC.C(COC)O C1(NC(c2cc(CC)on2)=O)C2CC1CN(C(C1CCC(F)C1)=O)C2 N1(C(Cc2ccc(C)s2)=O)CCCCC1CNC(c1cn(C(C)C)cc1C)=O C(=O)(C(C)CC(=O)NCC(C)(C1CC1)NC(c1cnc(CC(C)(C)C)s1)=O)OC N1(C(C2C(CNC(c3cc(C)on3)=O)CCC2)=O)CC2COCC2C1 c1(C(=O)NC2(CNC(CC3(C)CC3(F)Cl)=O)CCCC2)ccc2[nH]c(=N)[nH]c2c1 C1(CCNC(=O)CC2CC3CC3C2)COCCN1C(=O)CCN1CCCCC1=O N1(C(c2ccc(CC)s2)=O)CCC(NC(=O)Cc2cccnc2Br)C(O)C1 N1(Cc2cn(C(C)C)nc2)CCC(C(=O)Nc2sccc2CC#N)C(C)(C)C1 c1(OC)ccc(C(C(=O)NC(C)C)N(C)Cc2ncsc2C)cc1Cl N1(C(C2C(NC(c3ccc(N(C)C)nn3)=O)C2)=O)CC2CCC1CC2 c1(CNCC23C(CN(C(=O)Nc4cccc(C)c4)C2)C3)cc(Br)c(O)cc1O C=C(C)CC(C(=O)N1CCC1COC)NC(C1CC2CCC1CC2)=O Cc1nc(C(=O)NC(C2CCCN2C(C2CCC3(CC3)C2)=O)C)c(C)o1 C(CCCCC(=O)N1CCCC1N(C)C(c1cc(=O)cc[nH]1)=O)N(C)C C(=O)(CCCC(=O)N1CCC(COC)(NC(c2ccc(C(C)=O)[nH]2)=O)C1)NCC C1(C(N2CC(NC(Cn3nc(C)oc3=O)=O)C(C)C2)=O)CC2C=CCC(C1)C2 C#CCC(CC#C)C(=O)NCCOC1CN(C(C2CC(C3CC3)=NO2)=O)C1 c1(CC(=O)NCCOCCN(C(CSC)=O)C)cnn(C)c1 C(=O)(C1CC(=O)c2ccccc21)NCC#CC(N1CCC(C)(C#N)C1)=O N1(C(C(C)OCC=C)=O)CC(C(=O)Nc2cnccc2SC)CC1(C)C C1(C(=O)OC)(C(=O)NCC2CC2C2CC2)CCCN(C(=O)OC(C)(C)C)C1 c12nc(C)[nH]c1C(=O)NC1CN(C1)C2=O.c1(CC)ccc(OC2CCOC2)cc1 N1(C(C2C(C)(C(C)C)C2)=O)CCC2C(C1)CN2C(C1CC(OCC2CC2)C1)=O c1(C(=O)NCC2=CCN(CC(=O)NCC#C)CC2)ccc2c(c1)C(=O)NCCO2 C1(C(=O)N(CC(F)(F)F)Cc2cccnc2)C2CN(C(c3ccccc3)=O)CC12 c1(C(C)C(=O)NCC2CCN(C(=O)COC3CCOC3)C2)cccc(F)c1 CCCCCCC(=O)NCCCN(C(=O)CC1CCCC(C)(C)O1)C(C)C C12(C(N(CCN(C(c3ccc(C)o3)=O)CC)CC)=O)CC3CC1C2C3O c1(CCC)nsc(N2CCC(CNC(=O)C=CCOC3CCOCC3)C2)n1 c1(CNC(C2C3CC2N(C(C2CCCC(C(F)(F)F)C2)=O)C3)=O)ccncc1F C1(CNC(COCCCC#C)=O)CCC(C)(C(=O)N(CCCC=C)C)O1 N1(C(CCC2C(C)(C)C2)=O)CCCC1CCNC(=O)CSCC1CCCCO1 C#CCC(C)(C(=O)NCc1ncnn1CC)NC(=O)C1CC1 c1(OC)ccc(F)cc1C(N1CC(O)(CNC(=O)Cc2nncn2C)C1)=O Cc1nc2sccn2c(=O)c1CCN=C(NCC(C)CCC#N)NC(C)C Cc1cc(Br)sc1C(N1CCOCC1CNC(C1CCC1)=O)=O c1(C(N2CCN(CCNC(C(CC)C)=O)CC2)=O)cc(F)cc(Br)c1F c1(CC)cc(C(N2CCCCC2C(C)NC(c2nc(C)sc2C)=O)=O)cc(N)c1 C(=O)(C(CO)C(C)(C)C)N1C(CC(=O)N(C)CCc2ccccn2)CC(F)C1 Cc1cccc2c(CC(N3CCC3CNC(C3CN4CCN3CC4)=O)=O)c[nH]c12 c1(SC)cccnc1C(=O)NCc1ccc(CNC(C)C)o1 c1(C(N2CCCC(N3CCNCC3=O)C2)=O)nc2cccnn2c1Br CC1CC2CN(C(C3CCCN3C)=O)CC2N1C(=O)CCCC(N)=O N(C1COCc2ccoc21)C(C(N1C(c2cn(C)nc2)COCC1)=O)=O N12CCCC(O)(CC1)C2=O.C(=O)(CCOC1COC1)NCC(C)N(CC)CC C(C(=O)NCC1(CC(N2CC(F)(C#N)C2)=O)CC1)(C(C)C)SCC Cc1csc(C=CC(N2CCCC(CCNC(=O)CCCn3ccnc3)C2)=O)n1 c1(C(=O)NCCC(CCNC(C(C)(C)OC)=O)C)cnn2c1CCCC2 C1(NC(C2N(C)CC(F)C2)=O)CC2CC1CN(C(C1(Br)CC1)=O)C2 CC(=O)CCCC(C)C(=O)N1CCCC(N(C(=O)C(C)CO)C)CC1 CCCCC(F)C(=O)NCCC(C)N(C)C(C1CC1C(C)(F)F)=O Cc1cc(O)ccc1C(=O)NCCCCCC(=O)N1CCSCC1 C(=O)(C(C)(O)Cc1ccccc1)NC1CC(C(=O)NCC2(CC)CCC2)C1 C1(C)(C(N2CC(C)(NC(CCC=CC(C)C)=O)C2)=O)CCCCC1(F)F c1(C(N2CC(C)C(NC(c3cnc4[nH]nnc4c3)=O)C2)=O)c(N)cc(Cl)cc1F CC1(C)OCCN2C(=O)N(CCc3cccc(F)c3F)CC12 CCCC(CC(C)C)C(=O)NCC1(CCNC(=O)C(C)(CC)CC(F)F)CC1 N12CC3(CC3C1=O)C2.N1(C(C2C(NC(=O)OC(C)(C)C)C2)=O)CCCC1 c1(C(=O)NCCNC(=O)CSc2cn[nH]c2)ccc([N+](=O)[O-])nc1 c1(CC(N2CCC(C)(NC(C3CCCCN3N=O)=O)C2)=O)n[nH]c2ccccc12 CC1=CC(C(=O)NCC2CC(C(=O)NCC(C)C#N)CO2)SC1 c1(CN(C(c2ccccc2)C(=O)OC)C(c2ccccc2Cl)C)cnc(S)n1C N1(C(C2(CC)CCOC2)=O)CCN(CC2(NC(C3CCC=CCC3)=O)CC2)CC1 C(=O)(CCC(=O)C(C)(C)C)NCC=CCC(NOCCCC)=O c1(CC)ncc(C(=O)NC(CNC(=O)C(C(C)C)NC(C)=O)(CC)CC)cn1 c1(C(=O)NCC2OCCN(C(C(CC)F)=O)C2)cc(Cl)ncc1F CN=c1nc(C(N2CC3CCC3(CCNC(C3CC4(CC4)C3)=O)C2)=O)cc(C)[nH]1 c1(CNC(C(=O)NCCCCn2cnnc2)=O)cccnc1 N1(C(CCOCC(C)C)=O)CCC2(CCC(NC(=O)C3=CCC(C)CC3)C2)C1 c1(C(c2nnnn2CCC2CC2)NC(=O)CCCNC(CC)C)c(Cl)cncc1Br N1(C(c2cc(C(C)=O)ncc2)=O)CCCC(C)(C(N2CCC3CC3C2)=O)C1 C(=O)(CCN(C)C(=O)NCCS)OC(C)(C)C.C1C(C)(C)N1.CC(C)O C(=O)(C1=C(Cl)CCC(C)C1)NC(CN(C(c1cn(C)c(=O)nc1O)=O)CC)C c1(C(=O)NCCCCC2N(C(CC)=O)CC(C(F)(F)F)OC2)cc([N+](=O)[O-])cn1C S(=O)(=O)(c1ccc(NCc2cccc(OC3CC3)c2)cc1Br)NS(C)(=O)=O C1(C(=O)NCCn2cc(CCC3CCCCC3)nn2)CCc2ccccc2C1O N1(C(CCc2ccc(C)cc2)=O)CCC(CNC(C23COCC2C3)=O)C(F)(F)C1 C1(N(C(c2cnc(C3CC3)nc2)=O)CC)CCCN(C(=O)Cc2cc[nH]c2)CC1 C(=O)(C(C)(C)C1=CCN(C(=O)CC2CCC(C)CC2)C1)NCC1CC(C)OCC1 c1(C(=O)NC(C)CNC(C2(c3cc[nH]n3)CC2)=O)ncccc1Br N1(C(CCOCCC)=O)CCCC(CN(C)C(c2nccc(C)n2)=O)C1 c1(CC)ccc(C(C)C(N2CCC(F)(CNC(c3ccc(F)o3)=O)C2)=O)cc1 CCCCC(CC)CCNC(C1(NC(c2ccc([N+](=O)[O-])o2)=O)CC1)=O N=c1cc(-c2cn(CC3CC(CNC(=O)CC=C(Cl)Cl)C3)nn2)cc[nH]1 N1(C(C)=O)CCCC1CN(C(c1cnn(C(C)(C)C)c1)=O)C.C1(C(=O)N)(CO)CCC1.C c1(NS(N2CC(C)C(C(=O)N(C)C)C2)(=O)=O)nnc2ccc(C(F)(F)F)cn12 c1(C(=O)NC(CNC(C2(C(C)C)CC2)=O)C2CC2)ccc(CO)cc1.C1C(=O)N1 Cc1nn(C)c(C)c1CCC(=O)N(CC(O)CNC(c1ccc(Cl)cc1)=O)C CC1CCCCN1CC(N1CC(C)(NC(=O)CNC(=O)C2CC2)C1)=O C(=O)(C(COC(C)(C)C)CC(C)C)Nc1c(C(=O)OCC)ccc(Cl)n1 C1(C(=O)NCC(CNC(C(C)N(C(C)=O)C)=O)C)CCCN1S(C)(=O)=O C(=O)(CC=C(Cl)Cl)NC12CC(C(=O)OC)(C1)C2.C12(C)CCN1C2=O c1(CCC)cc(C(=O)NCC2(N)CC2)cc(O)n1.C1(CC(=O)C=O)CCCCC1F c1(C(=O)NC2CCN(C(c3n(C)ncc3C#N)=O)CC2O)ccsc1S(N)(=O)=O c1(C(=O)NC23CC(CNC(C(CC)(C)O)=O)(OC2)C3)cc(Cl)cnc1OC c12ccc(cc1)C(=O)NCc1ccn-2n1.Cn1ccc(-n2cnc(C(F)F)c2)n1 n1(CC(=O)NCCCN(C(COCCC)=O)C(C)C)ncc(Br)c1C C(CCc1ccccc1Br)(C(C)(C)C)NC(C(C)NC(=O)C(F)(F)F)=O C(=O)(C(O)CCCNC(c1c(C#N)cnn1C)=O)Nc1ccc(C(C)=O)cc1 C1(CC(N2CC(CNC(c3on(C)c(=O)c3)=O)OCC2)=O)CCn2cncc2C1 Cc1ccc2c(c1)CN(C(=O)C(=O)NC1CC(CC(=O)O)C1)CC(C)O2 CC(C(C)C(=O)NCC1CC(CF)C1)NC(c1[nH]nnc1C1CC1)=O C1(NC(c2cnc(CC)s2)=O)CC2CCC1(Nc1ncc(Cl)cn1)C2 C(=O)(C1CCCc2ccccc21)NC1CCC(CNC(C=C(CC)CC)=O)C1 C(C)(C(C)(C)CO)N(C)C.c12cc(on1)CNC(=O)CCN(C(C)C)C2=O c1(CN2CCC(O)(C(N3CCC(CO)CC3)=O)CC2)cccc2c1CCNC2 C12(NC(c3cn(C(C)(C)C)nn3)=O)CCN(C(=O)COCCN(C)C)CC1C2 CC(CCO)C(=O)N1CCC(O)(C(C)NC(=O)C(c2ccc(N)cc2)(C)C)C1 O=C(O)C(CNCc1cnn(C2(SCCCl)CCC2)c1)Cc1ccccc1 C1(NC(CCOC)=O)CC2CC(C1)N(C(C1(OC)CCCCCC1)=O)C2 C1(CNC(=O)CC2CCC(C(N3CCC(CC)C3)=O)CC2)CC2CCC(C1)N2 c1(COCC(N2CC3C(CNC(c4cnns4)=O)C3C2)=O)ccc(F)cc1F C1(c2n(C(CC)C)nnn2)(NCc2ccc(CO)o2)CCC(SC)CC1 c1(N(C(=O)Nc2c(C)c3cnccn3c2C)CC)cc(C)cc(S(N)(=O)=O)c1 C1(NC(c2c(CC)scn2)=O)CCC2CCN(C(c3ccc(O)c(Cl)n3)=O)C1C2 C(=O)(C1=CC2CCC1C2)NCC1(NC(C2CN(C(N)=O)C2)=O)CCOCC1 N1(C(C2(CC)CCCOC2)=O)CCC(CO)C(NC(=O)CCCN(C)C)C1 C1(CNC(C2(C)ON=C(C)C2)=O)CN(C(=O)CN(C)S(N)(=O)=O)CC(C)(C)O1 N1(C(c2n(C=C)ncc2)=O)CC2(CC(NC(=O)CC(C3CC3)C3CC3)CO2)C1 C1(C(N2CC(NC(Cc3c(CC)cccc3)=O)C2)=O)CCc2nc(O)[nH]c2C1 n1(CC(=O)NC(C2N(C(COCC)=O)CCC2)C2CC2)c(=O)n(C)c2ccccc12 c1(C2C(C(=O)NC(CCNC(CC=CC)=O)(C)C)C2)cccc(CC(F)(F)F)c1 CC1CCC(NC(c2ccc(C#N)o2)=O)CN1C(C1CCC(=O)O1)=O c1(C(=O)NC2C=CC(SC)C2)cc(C(=O)N(CC(=O)NC2CC2)C2CC2)on1 C#CCC(CC#C)C(=O)N1CC(C(N)=O)(CNC(=O)C(F)(F)c2nc(C)cs2)C1 C(=O)(C1=CCC(C)(C)CC1)NC1CC(NC(=O)COC2C(CN=[N+]=[N-])CCC2)C1 CC(CCCCNC(C1CCC1C)=O)NC(=O)C(O)Cc1cnc[nH]1 Cc1cc2[nH]c(C(N3CCCCC(NC(c4cnc(Cl)c(Cl)c4)=O)C3)=O)cc2o1 C(c1cccc(F)c1F)=CC(N1CC(F)CC(NC(C2(C#C)CCC2)=O)C1)=O c1(C(=O)NC2C(O)CCN(CCCC)C2)cccc2nc(O)oc12 Cc1ccncc1CNC(=O)CC1CCC(NC(=O)CC#N)C1 C(=O)(C(O)CC[S+](C)C)NC(CCCC)CNC(c1c[nH]c(C)cc1=O)=O N1(C(CC)=O)CCN(C(c2ccc(CSC3CCCOC3)nc2)=O)CC1 c1(CC)cccc(C)c1C(=O)NC(C)C(C)NC(c1ncc[nH]c1=O)=O c1(C(=O)NC(C)CCNC(=O)C(C)n2cncn2)cc(N)nc(Cl)c1 c1(C(N2C(CO)CC(NC(C(n3ccc(C)n3)C)=O)C2)=O)ccc(O)c(N)n1 C(=O)(C1COc2ccc(F)cc21)N1CCCC(NC(=O)COc2ccsc2)C1 C=CCC(CNC(=O)CCc1nc(O)n[nH]1)C(=O)NCCCC1CCC1 C1(CC(=O)NCc2ccc(NC(C)=O)s2)CSc2ccccc2NC1=O N1(C(c2[nH]c(=N)sc2)=O)CCC2CCN(C(c3ccn4c(O)nnc4c3)=O)CC12 C1(C(=O)NC2C(C)CN(C(c3ccc(N)c(Cl)n3)=O)CC2)CC2(C1)CC(F)(F)C2 C1(CNC(CCC=C)=O)CCC2(CO1)CC(NC(c1cn(C)nc1OCC)=O)C2 CC1CC2CN(C(=O)CC3COC(C)(C)C3)CC2N1C(C1CC2(CCC2)C1)=O Cc1ccsc1C=CC(N1CC(CCNC(c2ccnn2C)=O)C(C)C1)=O c1(OC)ccc(C2CCCCC2C(=O)Nc2cc(C3CC3)nn2C)cc1 O=S(=O)(c1cn[nH]c1)NCC1CCCN1C1CCCC1 CC(C(=O)N(C1CCC(NC(c2cscc2F)=O)CC1)C)C(C)S(C)(=O)=O c1(CC(=O)NCC2(F)CC(NC(c3c(C)nsc3N)=O)C2)nc2ccccc2s1 c1(CNC(CC2C(C)C2)=O)cc(C(=O)N(C)C2CC2)co1.C1C(=O)N1C1CC1 Cn1nc(C(=O)NCC(O)CNC(c2cc(Cl)ns2)=O)cc1[N+](=O)[O-] C1(NC(C=C(CC)C)=O)CC(NC(=O)CCc2nc[nH]n2)CC1O C1(C(N(C(C)CNC(=O)C(CO)N(C)C)C)=O)CCc2c(ncn2C)C1 c1(C(=O)NC(CC)CNC(=O)CC2CC(F)(F)C2)cccc(-n2cc(C)cn2)c1 Cc1ccccc1C=CC(N1CCC1CNC(C1CC1c1ccccc1)=O)=O Cc1cccc(COC(C)C(=O)NCC2CCN2C(=O)CC(F)(F)Cl)c1 Cn1nnnc1C(CC1(C)CC1)NC1CCOC1 N1(C(=O)CCOc2cccnc2)CCC2(CC1)OCCO2 Cc1ncncc1C(=O)N(C1CCCC1C)C1CC1.N12CCC(C1)C2=O c1(C(=O)NC2CCN(C(CC(=O)NC)=O)C23CCC3)cccc2cccnc12 C1(NC(=O)COCCO)CC2CN(C(c3ccc(-n4ccnc4)nc3)=O)CC12 N1(C(C2(O)CC2)=O)CC2CN(Cc3cc(Cl)c(Cl)cc3F)CC2C1 c1(NC(N(C2CCOC2)CCCC)=O)ccsc1OC N1(C(=O)C=CCO)CCN(C(=O)C(O)Cc2cnc[nH]2)C(c2ccc(F)cc2)C1 N1(C(CSc2cccc(C)c2)=O)CC(NC(=O)CC(C)C(F)F)CCC(O)C1 N1(C(c2cccc(OC)c2Br)C(=O)NC2COC2)Cc2cnc(C(C)C)nc2C1 c1(SC)cccc(C(C(=O)O)NC2CC(CO)C2)c1 N1(C(c2[nH]cc(CN(C)C)c2)=O)C2CCC1CN(C(=O)CN1CC3CC3C1)C2 C1(CC(=O)NCC2CCCN2C(C2CC2c2cccc(F)n2)=O)NC(=O)NC1=O c1(C(=O)NCC2(C)C(NC(CNC(CC)=O)=O)CCC2)ccc2ncccc2n1 C=C(F)C1(CC(=O)NC2(CNC(=O)Cc3cnsc3)CCCCC2)CCOCC1 N1(C(CCC(=O)NCC)=O)CCCC2CN(C(=O)CC3CC4CC4C3)CC12 Cc1ncc(CO)c(NC(=O)CNC(=O)C(F)(F)CN2CCNCC2)c1O Cc1c(C(=O)NC2CCC3CC2CN3C(=O)C(F)F)oc2ccc(Br)cc12 N1(C(C(=O)Nc2n(C)ncc2Cl)C2CCC2)CCC(c2ccccc2)(CO)CC1 S(=O)(=O)(c1cc(Br)cnc1N)N1CCCC(c2onc(C(C)C)n2)C1 c1(CC)onc(C)c1C(N1CC(C(C)(C)O)(CNC(=O)C(C)NC(=O)NC)C1)=O C(CCSC)(C(=O)NC1(C)CCN(C(=O)C2CC2)C1)NC(C)=O.c1cccnc1SC C(=O)(CC(C)CC(C)(C)C)NC1(CNC(C(Cc2c(C)cccc2)C)=O)CCC1 C1(CNC(C2(C)CN(C)C(=O)C2)=O)CN(C(c2nocc2Br)=O)CC(C)(C)C1 c1(CC)cc(C(=O)NCCOC2CCN(C(=O)Cn3ncn(C)c3=O)C2)nn1C C1(N(C(=O)C=CC2CCCO2)C)CCN(C(=O)CSc2n[nH]c(O)n2)CC1 N1(C(C(C=C)CC)=O)CC(CNC(c2ocnc2C)=O)C2(CCC2)C1 CCC(O)CC(=O)N1CC(N(C)C(c2cccnc2C(F)(F)F)=O)C(O)C1 C12(CC(=O)NC3(C#C)CCOC3)CCCC1CCN2C(c1cc(OC)no1)=O C=CCC(CNC(C1CC(=C2CC2)C1)=O)NC(C1(SC)CC1)=O c1(CC)nc(=NCCC2CCC(NC(=O)C=CC3CCCC3)C2)[nH]c(C)c1F C(CC(C(=O)NC)NC(C1(C(=O)NCCc2ccc(F)nc2)CC1)=O)SC C1(NC(=O)C2=COCCO2)CC2CCC1N(C(=O)CC1CCCOC1)C2 N(C1CCOc2ccc(Cl)cc21)Cc1cc(C)on1.c12csc(n1)NC2=O c1(NCC(=O)NC(CC)CNC(=O)CCNC(=O)C=CCl)cccc(OC)c1 C1(N(C(c2c(C)noc2C)=O)CCC2CCOCC2)CCNCCC1C c1(CC2C(C(N(CCCC)Cc3ccoc3Cl)=O)C2)ccc(Cl)cc1 CCCCC(C)(F)C(=O)NC1CCCN(c2ncccc2C(=O)C(F)(F)F)CC1 Cc1noc(C)c1C(C)(C)C(=O)N1CC(C(C)NC(=O)C(C)C2CCCO2)C1 n1(CC(=O)NC2CC(C)(NC(CN3C(C)CC3)=O)C2)ncccc1=O C1(OC(=O)CC(O)C(C)C)CCCCCC1C(=O)OCc1c(OC)cccc1 C12(CNC(CNC(C)=O)=O)CCC(C1)N(C(=O)C(C)(C)C1CCCC1)C2 C1(CNC(C2(SCC)CC2)=O)(NC(=O)Cn2nccn2)CCCCC1 c1(C(=O)NC2C(NC(CCNC(C(C)(C)C)=O)=O)CCCC2)nccc(Cl)c1F C#CCC(C)(CC)C(=O)N1CC(C(=O)N(C)OCC(F)(F)F)C2(CC2)C1 C(CC1=CCN(C(c2nncs2)=O)CC1)NC(c1cn(CCO)nn1)=O N1(C(c2ccc(CN(C)C)o2)=O)CC(NC(c2ccncc2F)=O)CC(C)(C)C1 N1(C(C(n2cnc(C#N)n2)CC)=O)CC(NC(c2c[nH]nc2F)=O)C2(CCC2)C1 C(CNC(c1cn(CC)nn1)=O)(C(C)(C)C)NC(c1c(CCC)nns1)=O n1(CCCCOC)cc(CCC2CCCN2C(=O)C(O)CN2CCOCC2)nn1 S(=O)(=O)(c1cnc(NCc2ccsc2Br)c(Cl)c1)NCCC(C)(C)OC N1(C(=O)NC2CC(C(=O)NC(CCOC)(C)C)(CC)C2)CCCCCC1 CCC(C)(C)C(O)C(=O)NC(C)(CNC(c1cnnc(C)c1C)=O)C1CC1 c1(CCNC(=O)CC2COCCN2C(C2C3COCC23)=O)cccc(Cl)c1Cl N1(C(CCCOCCOC)=O)CCCN(C(c2c(Cl)cncc2Cl)=O)CCC1 CC1CC(C(=O)NC(C)(C)CC2CCC2)CN(C(C2C=CCS2)=O)C1 Cc1cnc(C(=O)NC(C)C(C)NC(=O)C(c2ccccc2C)(F)F)cc1C#N C1(C(=O)NCC#CCNC(c2nn(C)c(C(F)F)c2)=O)CC2(C1)CC1(CCC1)C2 N1(C(CN2C(C)CCC2)=O)CCCOC(CNC(C2(C3CCC3)CCC2)=O)C1 N1(C(CC2CC(=O)NC2)=O)CC2(CCCN(C(c3scc4c3CCCC4)=O)C2)C1 c1(-c2nc(CC(CC)C)nn2CC(C)C2CC2)nc2ccccn2c1F Cc1c[nH]cc(C(=O)NCC(C)(CC(C)C)NC(c2ccc(C#N)o2)=O)c1=O c1(OC)cc(C(=O)NC(CNC(C2SC3C=CC2CC3)=O)CO)cc(OC)c1C C1(CNC(c2ccc(N(C)C)nc2)=O)CN(C(=O)C2=CSCCO2)CC(C)(C)C1 c1(C(=O)OCC)c(C)[nH]c(C(=O)Nc2onc(C)c2C)c1C.N12C(CC3CC13)C2 c1(C(=O)NC(CC)CNC(=O)Cc2cc(C)no2)cn(C)c(=O)cc1OC N1(C(C2C(C)(C)CCO2)=O)CCCCCC1C(=O)NCCC1(O)CCC1 Cn1ncc2c(NC3CCOC3c3ccnn3C3CCC3)nncc12 CCC(C#N)C(=O)NC(C1CCN(C(c2n[nH]c(C3CC3)n2)=O)CC1)C N1(C(CCN(CC)CC)=O)CCC(NC(C2CC(F)(CO)C2)=O)C(CO)C1 C=CC1CCN(C(C2CN(C(C3(CO)CCC3)=O)CC(C)O2)=O)CC1 C1(N(C(=O)CCNC(=O)CO)C)CCCCN(C(=O)CC2(C)CCOC2)C1 N1(C(CC(CCC)C)=O)CC2CCC1CN2c1nc(C2CC2)nc(C)c1OC c1(CCC(N2C(C)CC(NC(CC(=C=C)C)=O)C2)=O)ccc(C)cc1Br N1(C(c2ccc(O)nc2)=O)CCC2(C1)CN(C(c1cc(-c3ccco3)on1)=O)C2 C(=O)(C(C(C)(C)C)SC)NCC(CNC(c1cc(OC)ns1)=O)OC C12(CNC(C(C3CCOCC3)OC)=O)CC1CN(C(c1nc(=N)cc[nH]1)=O)C2 Cc1cc(C(=O)NCC2(C)CCC(NC(c3cc(N(C)C)ccn3)=O)C2)cnn1 c1(OC)cc(C)c(Cl)cc1S(=O)(=O)N1CCN(C(=O)C(C)(C)CCl)C(C#N)C1 C12(C(=O)NCC(CCOC)O)CC(CO)(CN1C(C1CC(C)C1)=O)C2 C(CC(C(=O)N(C1CC(F)(F)C1)C)NC(C1CCC1C)=O)OC N1(C(C(COC)COC)=O)CC(C(=O)NC2C(O)CC2O)CC(C)(C)C1 c1(N2C(CNC(=O)C(O)C3CCC3)CC3COCC32)nc2ccc(Br)cc2s1 N1(Cc2ccccc2)CCC2CC2C1.N12CCCC1NC(=O)CNC2=O C1(C(N(C)CC2(O)CCN(C(c3cc(OC)n[nH]3)=O)C2)=O)CC(C(C)C)=NO1 C1(NC(c2c(CNC(c3c(C(C)C)onc3)=O)c[nH]n2)=O)CCCC2(CC1)CC2 CCC(CC(=O)NC1C=CC(CO)C1)N(C(=O)CNC(=O)CN(C)C)C c1(OC)nc(=NC2CC(NC(C3CC4C(C3)C4(F)F)=O)C2)nc(OC)[nH]1 CC(C)C(C(=O)NCC1(F)CCN(C(c2ccc(=O)oc2)=O)C1)c1cnn(C)c1 c1(C(N(CCCCNC(=O)CC2CCC2)C)=O)c(F)cc(F)c(F)c1F c1(C(=O)NCC2N(C(COCc3onc(C)n3)=O)CC2)ccc(S(=O)CC#N)cc1 C1(CNC(CN(CCC#C)C)=O)CCCC2(CN(C(=O)C(C)CS(C)(=O)=O)C2)O1 NS(=O)(=O)c1cccc(CNC(C2CSCCN2Cc2nccs2)=O)c1 C1(CN(C(=O)CCC2CCCOC2)CC)COCCN1C(=O)CCSC N1(C(C(c2cccc(Cl)c2)OC)=O)CCC2C(NC(=O)C(C)O)C2C1 C(=O)(C(Cc1cccc(Cl)c1)CCCO)NC(CCC)C1CCC1 Cc1nc(NC(C2CC(NC(c3c(Cl)cccc3Br)=O)C2)=O)ccc1Br C12(CNC(c3c(COC)non3)=O)CC1CN(C(=O)CNC(=O)CC(C)(C)C)C2 N1(C(C(C)OC)=O)CCN(C(=O)COC2(C)CCC2)CC1c1cn[nH]c1 C1(CC=CNC(c2ccc(C3C(C)C3)o2)=O)COCCN1C(=O)C(C)n1cccn1 C1(NC(C(CC)C#N)=O)C2CCCN(C(c3cnnn3C)=O)C2C1(C)C N1(C(CC=C)=O)CCCCC2(CCN(C(=O)CC(C)CCC)C2)C1 c1(OC)ccc(NCC)cc1OC.C12CCC(C1)C(=O)N2.C(=O)(C(C)=C(C)C)NC C1(CNC(c2c(CNC(c3c(C)nsc3)=O)cc[nH]2)=O)CC(=O)N(C)C1 CC(C)CCC(=O)NC1(CO)CN(C(=O)C(N2C(C)CCC2C)C)C1 c1(CNC(CC2(OC)CN(C(=O)CC3(C#N)CC3)C2)=O)nn(C)cc1C C1(C(=O)NC2C(C)CN(C(c3cn(C)[nH]c3=N)=O)C2)CCn2ccnc2C1 C1(O)(CC(=O)NC(C2CN(C(=O)CN3CCC(CO)CC3)C2)(C)C)CCCCC1 c1(C(=O)NCC2CCN(C(=O)C(=O)Cc3ccccc3)C2)ccn2nnnc2c1 C(=O)(CC(C)C(C)C(C)C)NCC1CCC(C)(Nc2nc(C)nc(C)c2F)CC1 Cc1cccc(CN2CCOC(CC(=O)Nc3ccccc3CC#N)C2)c1O C(CCC(C(=O)N1CCC1)N1CCCCC1C(N1CCOCC1)=O)OC.C(=O)OC C(=O)(C1CCCc2c[nH]nc21)NCCN(C(C1(c2cccnc2Cl)CC1)=O)CC c1(C(=O)NCC(O)CCNC(=O)C(O)c2ccsc2)cccc2nc(CO)[nH]c12 CC1CN(C(C2CCC(C)CC2)=O)CCC1NC(=O)COC(F)F c1(C(N2CCC(NC(C(CC)NC(N)=O)=O)C2C)=O)ccc2c(c1)COCO2 C(=O)(CCCN(C)N=O)N1CC(C(=O)NCC#CCOC)C2(C1)CC2 N1(C(C2(CC(C)C)CCNC2)=O)CC(C#N)C2(CCOCC2)C1 c1(C(N2CC(C(C)NC(c3cnc(SC)nc3O)=O)C2)=O)cc2nc[nH]c2cn1 c1(CC(C(=O)NC2CC(CNC(c3c(C)snn3)=O)C2)C)c(C)n[nH]c1C c1(C(N2CCN(C(C(COCC)(C)C)=O)CC(O)C2)=O)ccc2sc(C)nc2c1 c1(C(=O)NC23CC(NC(C(C)SC(C)C)=O)(C2)C3)ccc2c(c1)C(=O)N(C)C2=O C(C)(CCCCNC(c1nccc(C)n1)=O)NC(c1cc(CCOC)on1)=O N1(C(C(C(C)C)OC)=O)CCN(C(C2C=C(C)CS2)=O)CC12CC2 C1(C(=O)NCC(CNC(C2(C(N)=O)CCC2)=O)O)CC12CCOCC2 C12(NC(CC(C)(C)C3CC3)=O)CC3CC(C1)CC(NC(=O)C(O)C1CCC1)(C3)C2 N1(C(c2c(CC)c(C)ccc2)=O)CCN(C(C2CCC(CC)CC2)=O)C2CCC12 N1(C(C2C(CC)N(C(C3CC4CCCC4C3)=O)CC2)=O)CCC2(C=CCO2)C1 CCCC(CC(C)C)C(=O)NCCCN(C)C(c1c(C2CC2)cccc1F)=O C(CC(O)C(=O)NC1CCC(NC(=O)CC2(C)CCOC2)CC1)SC C(C(C)(O)CC(=O)NC1CC(CNC(=O)Cc2cc(Cl)n(C)n2)C1)OC C1(C(=O)NC2CC(C)CN(C(c3cnncc3O)=O)C2)CC12CCC1(CC1)CC2 C=C(C)CC(C(=O)NCC1CCCC2(CC2)C1)NC(C1COC(=O)N1)=O CON(C)S(=O)(=O)c1ccc(C(=O)N(C2(C)CCS(=O)(=O)C2)C2CCCC2)cc1 c1(CC(=O)N(C)CC2CCN(C(C3CC3COC)=O)C2)ccc(C(N)=O)cc1 O=S1(=O)CCC(n2nc(-c3cscn3)nc2C23CC(C2)C3)C1 C(c1c(C)noc1C)=CCc1cccc(OS(CC2C(C(C)C)CCO2)(=O)=O)c1 C1(C)(CC(=O)N(CC(=O)NCC2(CCOC)CCC2)CC(C)C)CCCO1 C1(C(N(OC)C)=O)CCCC1.N12CC(C1)OC2=O c1(Cn2cc(C(CCC)NC(=O)Cc3sncc3Br)nn2)ccccc1[N+](=O)[O-] c1(NC(C2CC2CN2CCCC(CO)C2)=O)cccc(S(=O)(=O)N2CCCC2)c1 CC(C)CC(C)(C)C(=O)N1CC2CC(CNC(=O)C(C)N(C)C)C2C1 CC(C(=O)N(CCCNC(C1(c2cccc(F)c2)CCCCC1)=O)C)S(C)(=O)=O C(=O)(C1=C(Cl)CCC(C)C1)N1C2CC(CN(C(CSC(C)C)=O)C2)C1 N1(C(c2cc(CC)c[nH]2)=O)CCC(CO)(COC)C1.C12(CC=C)CC(C1)NC2=O C1(NC(C(CC)C)=O)CCN(C(C2(C(F)F)CCCC2)=O)CC1O C1(CCO)(NC(=O)C(=O)NC2CCCC2)CN(C(=O)Cc2ncc(Cl)s2)C1 Cc1cc(C(N2CC3(C2)CN(C(=O)Cc2ccsc2)CCO3)=O)c2n[nH]cc2c1 C1(C(=O)NCc2nc(CNC(C(COC)OC)=O)sc2)CCC(F)(F)CO1 C(C(C(=O)N(CC(C)(C)CNC(=O)C=C(C)Cl)C)N(C)C)OC C(=O)(CC(C(F)(F)F)n1ccnc1)N1CCCC(CNC(CC(C)N(C)C)=O)C1 c1(C(=O)OC)cc(Cc2ccccc2)cc(F)c1.C12CN(CCC1CN(C)C)C2 C=CC1(C(=O)NCCC2CCCC2(C)C)CCN(C(c2ccncc2C)=O)C1 CC(C)C(O)C(C)C(=O)N1CCCN(C(C2CCn3nccc3C2)=O)C(C)C1 N1(C(c2[nH]cc(C)c2)=O)CCCC(N(C)C(c2ccc(C3(O)COC3)cc2)=O)C1 Cn1c(O)nc2c(C(N3CCCC3CNC(c3ncncc3F)=O)=O)cccc12 C(=O)(C1=NNC(=O)CC1)NC(C)CCC1C(c2c(C)cc(Cl)cc2)C1 c1(C(=O)NC2CCC2NC(c2ocnc2C(F)F)=O)cnc(C2CCC2)nc1O Cc1cc(C(=O)NC(C2CCCN2C(C2CCCCNC2=O)=O)C)ncc1Cl C(=O)(CCCCCCSC)N1C(C(NOCC(=C)Cl)=O)C(CC)CC1 C1(CNC(COC)=O)CC(NC(c2cnoc2C)=O)C(O)C1.c12ccc(cc1)[nH]2 C1(CC(N2C(CNC(C=C(C)Cl)=O)CCCC2)=O)CCCC(C)(C)O1 Cc1ccc(C=CC(=O)N(C)CC2CCCN2C(C2CC3(C2)CC(O)C3)=O)cn1 Cc1c(O)ccc(C(N2CCCN(C(c3occ4c3CCOC4)=O)CC2)=O)c1C C(=O)(C1CCCc2nnn(C)c21)NCCC1(NC(C2ON=C(C(C)C)C2)=O)CC1 C(C)(C)(C(F)(F)F)OCC(=O)NCCCCNC(C1C(C(C)C)CCO1)=O c1(C(=O)NCC2(O)CCN(C(C3CC(=O)N3)=O)C2)ccc(C#N)cc1 c1(C(N2CCCC(C(=O)NCC3CC[Si](C)(C)C3)C2)=O)ccc(F)cc1I c1(C(=O)OC)cccnc1NC1CCOCC1C N1(C(=O)CCCOc2ccc(O)cc2)CCC(OCc2ccccc2)C12CC2 Cc1cnc(F)c(C(=O)N(c2nccc(C)n2)CC2CNC2)c1 CC(O)C(C(=O)NC1CCC1CNC(c1ccsc1Cl)=O)N(C)C N1(C(C(C)N2CCC2)=O)CCC(O)(CNC(C23CC(O)C2C3)=O)CC1 C(C)(C)(CC(=O)NCC1(C)CCN(C)C1)N(C(C(OC)OC)=O)C N1(C(CCCNC)=O)CCn2ncc(-c3c(C)ccnc3F)c2C1 c1(SCC(N2CCN(c3cccc(OCC)c3)CC2)=O)ncnc2[nH]cnc12 N1(C(=O)NC(c2ccc(OC(C)(C)C)cc2)(C)C)CCC2CCC(O)C1C2 C(=O)(C(O)CC(N)=O)N1CCC(CCCCNC(CC2(C)CCOC2)=O)CC1 c1(OC)nc2cc(Br)ccc2cc1C(=O)NCCCOc1ccc(F)cc1 C#Cc1ccc(C(N2CCCCC(C(=O)NC3CCC(O)C3)C2)=O)nc1 c1(-n2ncc(C(=O)NC3C(NC(C(C)=C(C)C)=O)CCC3)c2)ccc(Cl)cc1 C(=O)(C1CCCc2c(O)cccc21)N(C)CC1N(C(C(F)OC)=O)CC(F)C1 c1(CN2CC(N(C)C)C(C)(C)C2)cccnc1S(C)(=O)=O C1(C)(CC(CNCC(c2ccc(Cl)cc2)N(C)C)O)NC(=O)NC1=O N1(C(c2cn(CC)nn2)=O)CCN(C(=O)C(O)CSC)CC1c1ccccc1 CC(C)C1=NOC(C)(C(=O)N=c2[nH]nc(-c3ccccn3)s2)C1 c1(NC(C(N2CC(C(C)C)C2)=O)=O)csc(CCc2ccccc2)n1.C1CO1 C1(NC(CC2(C)CC2(Cl)Cl)=O)CC2CC1N(C(=O)C(O)CC1CCCCC1)C2 C1(NC(c2c(O)ccc(CC)c2)=O)CN(C(=O)C(C)(O)C(C)(C)C)CC12CCC2 C1(CC(N2CCC(CN(C(=O)CSc3cccs3)C)C2)=O)CCC2(CCC2)O1 C(=O)(C(CCF)NC(=O)CC1OCCCO1)N(CC(F)Cl)C C1(C2CCCO2)(C(=O)NCC(CNC(C(c2cn(C)nc2)=O)=O)(C)F)CCCO1 c1(C(N(C(CNC(C(C(C)C)NC(N)=O)=O)C)C)=O)ccc2ccoc2c1 C1(C(C)=O)CC1(Cl)C(=O)NCC1CC1CC(N1CC(n2cnnc2)C1)=O N1(NC(C(N2CCCC(NC(C)=O)C2)c2nc(Br)cn2C)=O)CC(C)OC(C)C1 c1(C(=O)NC2CC2NC(C2CCSCC2)=O)coc2ccc(F)cc12 N1(c2ccc(C#N)nn2)CCC2(CCCC2NC(=O)CCN2CCCCC2)CC1 C1(CNC(c2ccc(C(C)(C)C)cc2)C(C)C)CN(C)CCO1 c1(CNC(c2n(CCCC(=O)OCC)nnn2)C(C)C)cccc2c1nnn2C c1(OC)cc(CCNCc2cc(F)nc(F)c2)cc(F)c1F c1(C(=O)NCC2CN(c3ccncn3)CCO2)n[nH]c2ccc(F)cc12 C1(C)(COC)CC(NC(=O)C(F)=CCCF)CN1C(=O)C=Cc1c[nH]cn1 N1(C(C(=O)NCC)=O)CC2(CCCN(C(=O)Cn3cnc(Br)n3)C2)C1 C=CCC(CC=C)C(=O)N(C1(CCC)CCN(C(c2nc(C)no2)=O)CC1)CC c1(C(N2C(CCNC(=O)COC3CCC3)CC(OC)C2)=O)c(C)ncn1OC C1(CC(C)C)CCC(CNC(=O)CCCN(C(=O)CCOCC(F)F)C)CC1 CN1CCN(C(c2ccnc(C(N)=O)c2)=O)C(CNC(C2CC(F)C(=O)N2)=O)C1 C#Cc1nccnc1NC(=O)CN(C(C1CC1C(=O)OC)=O)C1CC1 c1(C(=O)NC2CCN(C(c3cnc(C)o3)=O)C(C)C2)ccc2c(c1)ncn2C Cn1ncc(C(=O)NC2CCC2CNC(=O)C(C2CCOCC2)F)c1C1CC1 C(=O)(C1=CCCCC1)N1CC(=C(CNC(CC2C(C)C2)=O)F)C1 CCCC(C(=O)NC1CC2(C1)CC2C(=O)NCC1(CN(C)C)CC1)C(C)C c1(CC(N2C(C3(NC(C(C=C)O)=O)CC3)CCC2)=O)cccc(S(=O)(=O)CC)c1 C#Cc1cc(F)c(C(N2CCN(C(=O)CC(C)(C)C#N)CC(C)(C)C2)=O)c(F)c1 CCCC(C)(O)CC(=O)NC1CCN(C2CCN(C(c3ncccc3O)=O)C2)CC1 C1(NC(C2CC23CCCC3)=O)CN(C(C23CCC(F)(CC2)C3)=O)CC12CC2 n1(CC(=O)NC(C(=O)NCCSC)Cc2nn[nH]n2)c(C)ccc1C c1(CCC)ccc(N)c(C(=O)NCC2CN(C(=O)C(C)(C)C(N)=O)CCC2C)c1 N1(C(C2(CCOC)CC2)=O)CC2COCCC2(NC(c2cc(Cl)cnn2)=O)C1 CCC(C)C(C(=O)NCC(C)N(C)C(c1ccn2ccsc12)=O)OC c1(C(=O)NC(CCNC(C(C(CC)O)C)=O)C)cc2cc(N)ccc2[nH]1 CC(C)CCC(C(=O)NC1CCC(=O)NC1=O)NC(C1CN(C)C1)=O O=S(=O)(C1CN(CC(c2ccncc2Br)O)C1)N1CCCC1 N#Cc1[nH]nc2ccc(NC(=O)CC3CCCN3Cc3ccc(C(N)=O)[nH]3)cc12 c1(C(=O)NC2CN(CCN3CCNC3=O)C2)ccc(N2CCOCC2)cc1 C1(C)(CNC(c2ccc(OC)nc2OC)=O)CC(F)(F)CN1C(=O)CNC(N)=O Cc1n[nH]c(C)c1C(C)C(N1CCCCC1c1cccc(O)c1)=O N1(C(C2C(C=C)OCC2)=O)CC(NC(c2cnc(C(C)(C)CF)o2)=O)CC(F)C1 C1(C)(CCNC(COCc2ncc(C)o2)=O)CCN(C(C2CC2C(F)(F)F)=O)C1 Cc1nc(CC2CC2)sc1C(=O)NCC1C2CN(C(c3[nH]cnc3C#N)=O)CC12 N1(CCCC(=O)N(C(C)CNC(C2CC(C)(C)C2)=O)CC)C(=O)CNC1=O Cc1oc(CNC(C2CCOC(C3CC3)C2)=O)nc1C(=O)NC1CC(S)C1.C(C)C CCCC(C)(C)C(=O)NC1CCCN(C(=O)CC(C)CC)CC1 C1(CNC(CN(C2CCSC2)C)=O)CCC(NC(C2(Cl)CC2(C)C)=O)C1 C1(NC(CC2CCC(C)(C)CC2)=O)CC1C1CCCN(C(=O)CC2(CO)CC2)C1 N1(CC=C)CCCC(N(C)Cc2c(-c3c(C)n[nH]c3C)cnn2C)CC1 c1(C(=O)OC)ccc(O)c(NC(C23CC2CN(Cc2ncc(Br)cc2F)C3)=O)c1 c1(C(=O)NCC(CC2CC2)C(=O)NCC2=CCCC2)c[nH]c2cnccc12 N1(C(C=C(C)c2cccs2)=O)CCCCC(NC(=O)C(N2CCSCC2)C)C1 c1(C(N2CCC(N3CCN(C(C4(C#C)CCC4)=O)CC3)C2)=O)cc(C)cc(F)c1 C12CCC(C1)NC2=O.C1(C2(C)N=N2)CCCC1NC(C1CC(C)(F)C1)=O C1(C(=O)NC2CCC(CNC(C3CC3C(F)F)=O)CC2)CCC2CC2CC1 C1(C(=O)NC(C(=O)NCCCc2cccs2)C2CCC2)C2CCC(F)C12 N12CC(CC(F)(F)C1)C(=O)N(CC)CC=CCC(=O)Oc1ccsc1C2.OC N1(C(c2cc(CC)ncc2)=O)CCN(C(=O)C(CC(C)C)NC(C)=O)CC1CF C1(C)(CNC(C(C)(C)NC(C(C)NC(N)=O)=O)=O)CCCCO1 C1(NC(CC2C(C)(C)C2)=O)CN(C(c2ccnc(S)c2)=O)CC1CO c1(C(=O)NC(CNC(c2nc(CCC)sc2)=O)CO)cc(C)nc2[nH]nc(C)c12 C1(NC(c2c(C)oc(Br)c2)=O)CN(C(=O)C=Cc2ccc[nH]2)CC12CCC2 C(C(COC)CC(=O)NCC(C(F)(F)F)c1ccon1)OCCC N1(C(c2nc(C)sc2)=O)CCC(=O)NC2CN(C(C3CC(C(F)F)C3)=O)CCC12 CC(C)(C)C(C#N)C(=O)NCC(c1ccccc1)NC(C12CCC(N=[N+]=[N-])C1C2)=O c1(OC)ncc(S(=O)(=O)NC(Cc2ccccc2Cl)C(=O)O)cn1 C(=O)(C(CC1CC1)NC(c1csnn1)=O)NC(c1cn[nH]c1)C c1(CC(N2CC(C(CNC(N)=O)NC(COCC(C)C)=O)C2)=O)cc(F)cc(Cl)c1 c1(CCC)cccc(C(=O)NC2CC23CC(NC(C2CC2COC)=O)C3)c1 CC(C)C(O)C(C)C(=O)NCC1CCCC1C(=O)N(CC(C)O)CC1CC1 N12CCN(N3CC(CO)(C3)c3c(C)c1ncn3)CC2.N(C)C N1(C(COC(C)=O)=O)CCC2(CC1)CC2(CO)C(N1CC(=O)NC(C(=O)O)C1)=O N1(C(c2nc(NC(C)=O)sc2)=O)CC2CC1CCN2C(=O)CC1(C)CCCC1 N1(C(c2ccc(CC)cc2)C(=O)NC(C)(C)CC)CCCC2(CC(=O)N(C)C2)C1 C1(NC(N)=O)CCC2(CC2)N1C(c1ccoc1)=O.CC(C)(C)O c1(N2CCN(C(=O)CCC(F)(F)F)CC2)cc(C2=CCCS2(=O)=O)ccc1 c1(CNC(C2C(C(=O)OCC)C23CC3(F)F)=O)ccc(C)c(F)c1F N1(C(C(C(C)(C)O)F)=O)CCN(C(c2coc(Br)c2)=O)C2CCCC12 N1(C(CC(C)n2ccnc2)=O)C2CCC(C2)C1C(=O)NCC(C)(O)C(F)F O=C1CCN(CC2CCCS2)C(=O)N1Cc1csc(-c2ccccn2)n1 Cc1n[nH]c(C)c1S(=O)(=O)NC1CCN(C(=O)C(CO)c2ccccc2)CC1F C1(CC#C)CCCCN1C(C1CC12CCOC2)C(=O)NC1CCCC1 C1(C(=O)N(CC(F)F)CCO)CCN(C(=O)c2c[nH]ccc2=O)O1 C=CCC(C(=O)N1CCC(NC(=O)C(C)SC)C1C)c1ccccc1 C1(CC)C(C(=O)NCCCN(C(C)CO)CC)CCN1C(=O)CC1(OC)CC1 n1(CCNC(=O)NCC2CC(n3ccnn3)C2)cc(Cl)cn1 c1(COC)nn(C)cc1C(=O)NC1CC(CNC(C2CC(n3cccn3)C2)=O)C1 CCC(C)(CCNC(C1CN(C(C)=O)C1)=O)NC(C1CCCSC1C)=O C1(C(N2CCN(C3CCC3)CC2)=O)N(C(=O)Cc2cncnc2)CC12CCCC2 C1(C(N2CCC(COC)(NC(c3cc(C)sc3C)=O)C2)=O)OC2CCC1CC2 c1(C(=O)NCC(C)CNC(C2(c3ncccc3F)CCC2)=O)cc(Cl)cnn1 c1(NC(C(=O)NCCCC)C(C)C)ncnc(OC)c1Br CC1(NC(=O)CC2CSCCS2)CCC(NC(=O)CN2CCCC2)CC1 Cc1cccc(C(=O)NC(C)C=CC(=O)NCC2(F)CC(O)C2)c1C N1(C(c2cc(C(=O)OC)oc2C)=O)CCC(O)(CNC(=O)CN2CCC2C)CC1 C1(OC)CN(C(C2(C(F)(F)F)CC=CCO2)=O)CC1NC(=O)C1=CCOC1 N1(C(c2cc(CNC(=O)C=Cc3cnccn3)ncc2)=O)CCCC(O)CC1 c1(CC(C)C)ncc(C(=O)NC(C)CCNC(=O)CCc2nc(C3CC3)no2)[nH]1 C(=O)(C1CCc2c[nH]nc21)N1CCC(CN(C(C(CSC)O)=O)C2CC2)CC1 N1(C(Cc2c(C)ncs2)=O)CCCCC(NC(c2nc(C)ns2)=O)C1 C12(CNC(C(C3CC3)SC)=O)CC(NC(C3CCC(C)S3)=O)(CCO1)C2 CC(N=c1[nH]c(N2Cc3ccccc3C(F)(F)C2)nc2ccccc12)c1ccns1 N1(CCC(N2CCC(NC(C3(C(C)C)COC3)=O)C2)=O)CCCC(N(C)C)C1 C1(C(C)C)CCC(C(N2CC(C)(C)C2c2cn(Cc3cnn(C)c3)nn2)=O)CC1 N1(C(=O)C(F)OC(F)(F)F)CCC2CCCC(C1)N2C(=O)CN1CCS(=O)CC1 c1(C(N2CCCC(C(N3C(COCC)CCC3)=O)C2)=O)c[nH]c(C)cc1=O CC1(CC(=O)NCC2(C)CCCN2C(=O)CCn2cc(N)cn2)CC(F)(F)C1 C1(CC(N2C(C3(NC(=O)CCC4CCC4)CC3)CCC2)=O)CCN(C2CC2)C1=O C1(CCC)CN(C(=O)CS(=O)(=O)NC)CCN1C(=O)CN1C(=O)CN(C)C1=O c1(CNC(c2ccc(C)o2)=O)ccc(C(=O)NCCNS(N)(=O)=O)nc1 n1(CC)cnc2nc(=NC3CCCC(C)(C)C3)[nH]c(NCCCCCCSC)c12 C(N=c1cc(Cl)c(O)n[nH]1)C12CC(NC(c3c(F)cc(C)c(F)c3)=O)(C1)C(C)O2 C1(CC=C)(NC(=O)CC(C)OC)CCN(c2ccnc(C3CCC3)n2)C1 C(=O)(CC1=CCOCC1)NC(C(C)(C)NC(c1c(C(C)C)noc1)=O)C N1(C(CCCNC(C)=O)=O)CC2(CCC2)CC1CNC(C1(C)CCC(O)CC1)=O c1(OC)cncc(C(=O)NC2(CN(C)C(C3CCOC(=O)N3)=O)CC2)c1 c1(C(=O)NC2CC(C(=O)NC3CN(C(=O)NC)C3)C2)ccc(OC)nn1 C1(OC)CN(C(=O)Cn2nccn2)C(C)(CNC(=O)CSc2ccc(F)cc2F)C1 Cc1cc2c(cc1C(N1CCC3(NC(=O)CCF)CCCC13)=O)CCN2 c1(NC(CN2CCC(NC(=O)CC(O)c3ccco3)CC2)=O)c(O)ncnc1O N1(C(=O)Cc2cnn(C(F)F)c2)CCN(C(c2cnccn2)=O)CC1 CCC(CCC(=O)N1CC(C(C)OC)C1)NC(=O)CCCc1ccc(C)cc1 CC1(C)C2CC1C(=O)N2.c1(C(N2CC(n3ccnc3)C2)=O)ccc(F)cn1 C(=O)(CS(=O)c1ccc(Cl)cc1)NC1CC(CNC(C(=C(C)C2CC2)F)=O)C1 C1(C(N2C3C(NC(c4cccc(F)c4O)=O)C(C3)C2)=O)CC2(CCOCC2)CO1 N1(C(CCC#C)=O)Cc2ccccc2OC2(C1)CN(C(=O)Cc1ccc(C)o1)C2 N1(c2snc(CCOC)n2)C2CCC1CC(NC(=O)CCC1CCC(C)O1)C2 c1(CCCC(N2CC(F)(CNC(c3occ(C)c3)=O)C2)=O)ccc(O)cc1 C1(CNC(C2C(C)C2)=O)CCCCCN1C(C1CCCC1F)=O C1(C(=O)NCC2(C)N(C(C(C=C)O)=O)CC(F)(F)C2)COc2ccccc2O1 CC(CNC(C1CCC(=O)C1)=O)CC(=O)N1CCC1 c1(C(=O)NCC(CC=C)NC(c2c(C)nn(CC)c2C)=O)sc2cncn2c1C N1(C(C(C=C)C)=O)CCCC2C(NC(=O)CC3CCCC(C)O3)C(C)(C)C12 CC1CC(C(=O)NCc2cncc(F)c2)CN(C(C2CC3(C2)CC(O)C3)=O)C1 Cc1ccc(SCc2ccc(=N)[nH]c2)cc1.c1(C(N(C)C=O)C)cncs1 O=C(CC1(c2ccncc2F)CCNCC1)NN1C(=O)NC2CCC1C2 c1(C(=O)NCc2c(C(=O)NCCC3=CCCCC3)nco2)cnn2ccccc12 C(=O)(C(C)CC(=O)N1CCN(C(C2CC2OC)=O)CC1)NCC N1(C(Cn2ccc(C(=O)OC)n2)=O)CC2(CCN2C(C2(C)CCCO2)=O)C1 C(CC(F)F)(C(=O)N1CC(O)CO1)NC(C(CC1CN(C(N)=O)C1)F)=O N1(C(C(N2CCSCC2)C)=O)CCN(C(c2cc(Cl)ns2)=O)CC1C1CC1 C1(C(=O)N(CCO)CCO)CCC2(CN(C(c3ccnc(O)c3)=O)C2)O1 CC(C)CC(C)(CNC(C1(F)CCOCC1)=O)NC(=O)CN1CC2CC2C1 N1(C(C2(CC#C)CC2)=O)CC2CCCC(NC(=O)CC3CCCCC3(C)C)(C2)C1 c1(C(=O)OC)cnccc1C(=O)NC1C(C(=O)NC2CC2C)C1.OC C1(NC(=O)CC2CC(NC(C3CC3(F)Cl)=O)C2)CCCC(O)C1 c1(C(=O)NC2CC(C)(NC(CCCC#C)=O)C2)cc(F)c(CC)cc1F C(=O)(CC1c2ccccc2C(=O)N1C)N1C(CC=C)CCCC1 C1(NC(CCCC=C)=O)CCN(C(=O)Cc2csc3nccn23)CC1O c1(C(=O)NC2(CCOC)CCOC2)cccc(C(=O)OC)c1N c1(CN2C(CCC)CCOCC2)c(N(C)C)ccc(Br)c1F CC1(C)CCN(C(=O)CC2CCCS2(=O)=O)CC1CNC(=O)CN=S(C)(C)=O C12(C(=O)NC(c3cccs3)CC)CCC(CC1)N(C(C1CC1C(C)C)=O)C2 Cc1nn(C)c2c(N(C)Cc3cccc(Cl)c3)nc(=NCc3ccc(Br)s3)[nH]c12 C(=O)(C(C(C)NC(c1cn(C)c(=O)cn1)=O)C(C)C)NCc1c(C)c(O)ccc1 C1(OC)(CNC(C2CCC2)=O)CC(NC2C(C(=O)NCc3csc(Cl)c3)C2C)C1 N1(C(C(CC#C)(C)C)=O)CCCN(C(c2ccc(C3CC3)cc2OC)=O)CCC1 CCCC(C(O)C(=O)N1CCC(C)(O)C1)NC(C1C2CCCC12)=O C12(C(=O)NC(C)C(=O)OC(C3CCN(CC)CC3)C)CC(C)(C1)OC2C CC1OC(C)Cc2c(C(=O)N(C)CCNC(C3CCC(=O)NC3)=O)n[nH]c21 c1(C(=O)NC(C)C(CO)NC(C2(C)CCC(=O)NC2)=O)cc([N+](=O)[O-])cn1C C1(C(=O)NC(C2CCCCC2)C#C)CCC(CNC(c2coc(C)c2)=O)C1 N1(C(c2cc(C(=O)OC)[nH]c2)=O)CCSC2(CCCC2)C1 c1(C(=O)NCC2(O)CCN(C(C(CC)SC)=O)CC2)ccc([N+](=O)[O-])nc1 C1(NC(c2cc(CO)[nH]n2)=O)CCN(C(C2CN3CCC2CC3)=O)CCC1CO C1(C(=O)OC)CCN(C(=O)NC2CC(c3cccc(Cl)c3)C2)CC1O C1(NC(Cc2cc(C)no2)=O)CCCCC1CNC(c1ncnn1C(C)C)=O c1(C(N2CCOC(c3nc(C)cs3)C2)C(=O)NCC)nn(C)c(C)c1Br CCCCC(O)C(=O)N1CC(OC)CC1C(=O)Nc1ncc(I)cc1Br CCC(CC)C(F)C(=O)N1CC=CC(NC(c2cncc(F)c2)=O)C1 N1(C(CCC2CC(OC)C2)=O)CCC(CCC(=O)NCC(c2cccs2)C)C1 CN1C(=O)NCC1C(=O)NC(C)(CNC(=O)CS(=O)(=O)N1CCCC1)C1CC1 C(CN=c1nc(N2CCCC3(CC2)CC3)c2c([nH]1)CSC2)c1ccccn1 C1(C(=O)OCC)Cc2cccc(F)c2N(C(c2nc3c(OC)cccc3s2)=O)C1 C#CCCCC(=O)N(C)CCOCCN(C)C(c1cc(C)cs1)=O C(=O)(C1=NOC(CNC(c2ccccc2C2CCC2)=O)C1)NC1N(CC)CCC1 C1(NC(COCc2cc(C)no2)=O)CC(NC(c2ccc(F)cc2)=O)C1(C)C N1(C(=O)Nc2cn(C3CC(NC(C4CC5C=CC4C5)=O)C3)nn2)CCC(F)(CF)C1 N1(C(C2C(COC)C2)=O)CCC(C)C(CNC(c2csc(-c3cnc[nH]3)n2)=O)C1 C#CC1(NC(=O)CC(C(C)(C)C)NC(=O)C=Cc2ccc(C)o2)CCC(C)CC1 c1(OC)cc(Br)ccc1C(N1CC(F)(F)CC1C(=O)NCC1CNC(=O)CO1)=O Cc1ccc(C(N2CCC2CNC(c2ccc(Cl)o2)=O)=O)cn1 c1(CC(C)NC(=O)CNC(=O)C(N)=O)ccc(CNC(=O)Cn2ccnn2)cc1 C(=O)(C1=C(C#N)CCC1)NCC(C(=O)NC1(C)C(C)CCC1)N(C)C N#Cc1nc(=NC2CC(NC(c3cnc4n3CCC4)=O)C23CCC3)cc[nH]1 c12cc(ccc1C#N)S(=O)(=O)NN2.C1(F)(CCN(CC)CC)CCC1 C1(C(=O)NC(c2ccncn2)C)CCN(C(=O)CCCC2CCCC2)O1 C(=O)(C1CN(C)C(=O)c2ccccc21)NC(c1ccc(OC)cc1)C N1(C(c2nc(CCOCC)oc2)=O)CCC(CC(C)NC(=O)C(C)C2CC2)CC1 c1(C(=O)NCCN(C(=O)COC2CCOC2)CC2CC2)ccnc2ncnn12 C(=O)(CC1=NNC(=O)C1)NCCNC(C1CCCN(C(C2CC=C(C)CC2)=O)C1)=O C1(C(C)C)COCCN1C(c1cncc(C2CC2)c1)=O.c12cc([nH]n1)CNC2=O Cc1nc2cccnn2c1C(=O)NC1CN(C(=O)CC2CSC2)CCC1C CS(=O)(=O)c1cc(C(N2CC(NC(=O)Cc3cn[nH]c3)C2)=O)ccc1F C(=O)(C(=O)C(C)(C)C)NCC(C(C)C)NC(C1CC(=O)NC1(C)C)=O c1(C(C)C)ccc(C(=O)NCC2CCC(NC(=O)C(F)(F)c3cnnn3C)C2)o1 N1(C(c2cc(C)oc2C)=O)CCN(C(=O)CCc2nc(=N)[nH][nH]2)CC(CO)C1 C1(NC(CN2CCC(C)C2)=O)CC1C1CCN(C(=O)C(C)(C)C(C)(C)O)CC1 c1(C(N(C2CCN(C(=O)COC3CCCOC3)CC2)CC)=O)nc(C)sc1C C1(C)(CNC(C(C)=C(C)C)=O)CN(C(=O)CC2CC3(CC3)C2)C(C)(C)C1 c1(C2c3nnnn3N2)cccnc1OCc1cccs1.C1=CC(OCCO)CC1 CC1(C)CCN(C(C23CSCC2C3)=O)C1C(=O)NC1CC2(CC2)C1 c1(CC(=O)NCCC2CCC(NC(c3ccccc3)=O)C2)ccc2c[nH]nc2c1 C(=O)(CCC1=NNC(=O)CC1)N(C)CC1CCCCN1C(=O)CCC(N)=O CC(C(=O)N(C)CCc1nn[nH]n1)N(C(=O)C(C)N1CCCC1)C C1(CCCSC)(C(=O)NC2CCCC2CNC(=O)CC2CCOC2=O)CCCC1 C(C)(C(C(=O)NCCC(C)N(C)C)C(C)C)NC(CC(COC)(C)C)=O c1(CC)ccc(NC(=O)NC)c(F)c1.N12CC(O)CC1C2 c1(CC(=O)NCC2(O)CCN(C(Cc3n(C)nnc3)=O)C2)cc(Cl)cc(Cl)c1 c1(C(C(=O)NCC(CCOC)NC(c2coc(C(N)=O)c2)=O)O)ccccc1Cl CCC(C(=O)N1CCOC(C(=O)NC2CC3(CCCCO3)C2)CC1)C(C)(C)CC c1(C(=O)NC(C(=O)NC(CSCC)CO)C(C)(C)O)cccc2ccnn12 n1(Cc2cc(C)on2)nnc(C(=O)NC(C)(CNC(=O)C(C)O)C2CC2)c1C C(c1ccc(OC)cc1C)=CC(=O)NC1CCC(C)(NC(C(CC)F)=O)CC1 C1(C(=O)NC2C(NC(=O)CC3(CO)CC3)CC2)CC12CCC2 CCC(CC(=O)NCCNC(=O)CSC(F)F)N(C(=O)C(C)C)C C1(Cc2cn(CC3CN(C(C4NC(=O)C(F)C4)=O)C3)nn2)(CO)CC(F)(F)C1 C(=O)(C(C)(C)CCCNC(=O)CCC(C)(C)C)N1CCC(N(C)CC)CC1.O(N)CC N1(C(c2ccc(CN)cc2)=O)CCn2ccnc2C1 C1(COC)(NC(C2C(C)C2(F)F)=O)CCN(C(=O)CCc2csc(C)n2)C1 Cc1nc(C)c(C(=O)NC2CCN(C(C3(CN(C)C)CC3)=O)CCC2CO)nc1C Cc1cc(NC(=O)C(CN(C)C)NC(=O)C(C)O)c(F)cc1F C1(C(=O)NC(CC=C)CO)CN(C(c2cc(C)co2)=O)CC12CCC2 N1(C(C2C(CNC(=O)CN3CCOC3=O)CCC2)=O)Cc2cccnc2C1 C(CCC(=O)NC1(CCCCNC(=O)CCOC(C)=O)CC1)C1C(C)C1 C(CC)(C(=O)N1CCCC1C(C)(C)C(=O)N1CC(O)(C(F)F)C1)=CCCC C1(c2n(CC(=C)C)nnn2)(NCC(c2ccc(F)cc2)CO)CCN(C)C1 N1(C(C(C=C)O)=O)CCN(C(=O)CCn2nc(C)cc2C)C(C2CCCC2)C1 N1(C(c2cc(OC)n(C)n2)=O)CCN(C(c2sc(=N)[nH]c2C)=O)CC1CO CON=Cc1ccc(C(=O)NCCCCNC(C2CCC3CCC23)=O)cc1 c1(NC(C(=O)NC2CC(SC)C2)=O)nc2c(s1)CC(C)CC2 N1(CC(=O)N(C(C)C)CCNC(=O)CC2C(C)C2(F)F)CCC(CO)CC1 N1(C(=O)CCC2CCCN(C(c3cc(=O)cc[nH]3)=O)C2)CCN2CC(F)CC2C1 N1(C(C(C)n2cncn2)=O)CC(NC(=O)CCc2ccccc2)C2(COC2)C1 C1(C)(COC)CN(C(C2CC=CC2)=O)C1.c12cc(no1)CNC2=O c1(C(=O)NCC(C)CN(C)C(c2ccsn2)=O)sc(N2CCCC2)nc1Cl C1(N(C(C=CC(C)C)=O)CCO)CCN(C(=O)CCc2ccccn2)C1 n1(CC(=O)NCC(CO)NC(c2cc(C)sc2)=O)nc(C2CC2)cc1C(F)F Cc1coc(C(C)C)c1C(=O)NC1CC(F)(CNC(C2CCN(C)C2=O)=O)C1 c1(SCC)ccc(C(=O)NCC(CC)NC(c2[nH]cnc2C#N)=O)cn1 CCCC(C(=O)NCC1CC(F)(F)CO1)NC(c1c[nH]c(C)c1)=O c1(C(=O)NC(CC)(C)CNC(C2(CF)CC2)=O)cc(C)c(C)cc1Cl N1(C(C2C(C)CC2)=O)CCC(C2CCN(C(c3ccc(C4CC4)cc3)=O)C2)CC1 c1(COC)ccc([N+](=O)[O-])cc1C(=O)NC12CC(CNC(C3(CO)CC3)=O)(C1)C2 C(C(C(=O)N1CCC1C(=O)N(CC)CC)NC(=O)C(CC)NC(C)=O)CC c1(CC)ccc(NC(=O)CC(C)CNC(=O)OC(C)(C)C)cc1COC C(CN(C(=O)CN1CCS(=O)CC1)C)(CO)(CO)NC(C1CCN(C(C)=O)C1)=O c1(C(N(CCCNC(c2cc[nH]c2)=O)CC)=O)cccc(OC(F)(F)F)n1 c1(CC)nn(C)c(CC(=O)NCC2(NC(=O)CCCc3csc(C)n3)CC2)c1Cl N1(C(c2n(C(CC)CC)ncc2)=O)CCC(N(C(=O)C(C)NC(=O)NC)CC)C1 C1(C(N2C(C(C)NC(C3(C=C)CCC3)=O)CCC2)=O)CC(C2CC2)=NO1 CS(=O)(=O)c1ccccc1-n1nc(CCC(N)=O)nc1-c1cnc(C2CC2)s1 C1(COC)(CNC(=O)Cc2n[nH]c(=N)s2)CCCN1C(c1ccn(C(C)C)n1)=O C(=O)(CC(C(N)=O)c1cnc[nH]1)N(CCCNC(CSC)=O)C O=C(NNc1ccc(F)c(F)c1F)N(c1ccncn1)C1CCCC1 C(=O)(C(C(F)(F)F)C(F)(F)F)N1C(C)CC(NC(c2cc(OC)n[nH]2)=O)C1 c1(C(=O)NC2CCCN(C(C(C(C)O)N(C)C)=O)C2)ccc(N)cc1Br n1(CC(N2CC3CC(NC(C(CC)N(C)C)=O)C3C2)=O)c(C)cc(O)cc1=O C(=O)(C1=CC2CC(C1)CC2O)N1CC(NC(=O)Cn2cccn2)C1 CON(C)CCCNC(C1(C)CC(NC(c2nccnc2C)=O)C1)=O C1(C(=O)NC(CN(C)C(C2CCCOC2)=O)(C)C)CC2(CCC(CN)OC2)C1 C1(NC(Cc2ccc(CC)cc2)=O)CC2CC1N(C(C1CNC(=O)C1)=O)C2 c1(C(N2CC3C(NC(CC4(NC(C)=O)CC4)=O)C(C3)C2)=O)cc(Cl)c(N)cc1F C(C(COC)CC(=O)N1CCC(C(=O)NCC2CCC3(CC3)C2)C(C)C1)OC Cc1ccc2oc(C(=O)NC3CCCN(C(C4CC5CCC4O5)=O)CC3)cc2c1 C1(CNC(CC=C(C)C)=O)CN(C(=O)CCc2c(C)noc2Cl)C(C)(C)C1 c1(C(=O)NCC2(C)N(C(c3c(CCC)[nH]cc3)=O)CCC2)ccc(C)nc1N Cc1ccnc(-c2cn(CC(C)NC(c3ccc(Cl)s3)=O)nn2)c1 C1(CN(CC(=O)O)CC=C)CC2C=CC1O2 c1(CCC)nc(C(=O)N(C(C)C(=O)N(C)CC2CC(O)C2)CC)cs1 C=Cn1nccc1C(N1CCC(C(=O)NC(C)CCCOC)(OC)C1)=O C1(=CCNC(c2ccncc2F)=O)CCN(C(=O)CCC2CCCC(O)C2)CC1 C(=O)(CCCN(C(=O)C(c1sccc1C)N)C)OC c1(C(=O)NCCC(C)(C)CNC(C2(CF)CC2(F)F)=O)ccc(Cl)cc1O c1(OCCCC)c(-c2cscc2C(=O)Nc2ccc(F)cc2Cl)cccc1F c1(-c2cn(CC3CN(C(C4(OCC)COC4)=O)C3)nn2)cccc(F)n1 c1(CCCN(C(C2CCCC2O)=O)CC)ccc(C)s1 C1(COC)(CNC(C2CC2c2cncn2C)=O)CCCN1C(c1cscn1)=O C(=O)(C(C)CC(=O)NCCCCCCNC(c1nccnc1C(F)(F)F)=O)OC C1(CNC(C2CCCC3(CC3)C2)=O)CCCCN(C(=O)C2CC2)C1 C1(NC(C2CCCOC2)=O)CCN(C(c2ccn3nncc3c2)=O)CCC1CO C=CCC(C(=O)NCC(C)NC(c1ccc(SC)s1)=O)OC C1(CNC(C2(C)CC(=C)C2)=O)COCC2(CCN(C(=O)C(C#N)C(C)C)CC2)O1 C1(CCC)CN(C(C2CCC(=O)NC2)=O)CCN1C(=O)Cc1ccc(Cl)nc1 C1(CNC(c2nn(C)c(C(N)=O)c2)=O)CC12CCN(C(C1CCCCS1)=O)CC2 c1(C2CC2)ccccc1C(=O)NC1(NCC2(CCOCCC)CC2)CCC1 c1(C(=O)NC2CCN(C(c3ccc(CC)o3)=O)C2)cnc(OC)nc1C Cc1ccnn1C(C)C(=O)NC(CNC(c1cccn1C)=O)C1CCC1 N1(C(c2c(CC)n[nH]c2)=O)CC(NC(C2CCC3CC2CO3)=O)CCC1C c12cccc(c1)-c1c[nH]nc1C(=O)NC2.c1(C(CNCC)O)ccccc1 c1(CC)cccc(OCC(N2CCCC(C(=O)Nc3ccccc3)C2)=O)c1 c1(C(=O)NC(CNC(c2c(C(C)C)nns2)=O)C2CCC2)ccc(N)c(Cl)c1O C1(NC(CCNC(N)=O)=O)CCCC(NC(C2CCC(C(N)=O)C2)=O)C1 C#Cc1cccc(NC(=O)CC2CCN2C(C2CCC(C)(C)OC2)=O)c1 Cc1ccc(CCC(=O)NCC2CCCN(C(C3CC=CCC3)=O)C2)cn1 C(Cc1cnc[nH]1)(C(=O)NOCCOC)NC(CCN(CCCCC)C1CC1)=O N1(C(C(CC2CCCC2)OC)=O)CCC(F)(CNC(C2CCCN(C)C2)=O)CC1 c1(N2CC3C(CNC(=O)C=Cc4ccco4)C3C2)cccc(F)c1[N+](=O)[O-] C(=O)(C(F)CC(C)(C)NC(C1C(C)(C)C1(F)F)=O)NCCc1ncc(C)nc1 c1(C(=O)NCC(C)NC(C2C(COC)(COC)C2)=O)cc2n(n1)CCC2 C(=O)(C(C)P(C)(C)=O)N(CC)CC1CCCN(C(c2snnc2C2CC2)=O)C1 CC1(C)CC(NC(c2cnc(-c3ccccn3)s2)=O)CCN(c2nnco2)C1 N1(C(c2ccc(CC)cc2N)=O)CCN(C(c2cccnc2C)=O)C2CCC12 C1(OC)CCCC1N=c1cc[nH]c(=NCC(=O)NC2CC2)[nH]1 c1(C(N2CCCN(C(c3c(CC)occ3)=O)CC2)=O)cccn2ncnc12 C(=O)(C(C#N)CC1CC1)NCC(C)(C1CC1)NC(=O)Cn1ncnn1 c1(OC)cccc(NC(C2CC(NC(=O)Cc3cncs3)C2)=O)c1OC N1(C(CCc2cc(C)nc(C)c2)C(=O)NCCC2CC2)CCC(C)C2(CCC2)C1 N1(C(c2scc(C#N)c2)=O)CCC(C2CCN(C(C3(CF)CC3(F)F)=O)CC2)C1 Cn1ncc(C)c1NC(=O)NC1CC(Nc2cccc(C(N)=O)c2)C1 c1(C(=O)NC2(CC=C)CN(C(=O)CCCC(C)=O)C2)ccc(C)c(S(C)(=O)=O)c1 C(C)(CC(=O)N1CCC(NC(=O)Cc2ccsc2Br)C1)OC C1(C(=O)NCCN(C(C2CCN(C)CC2)=O)CCOCCO)CCOC(C)(C)C1 c1(CC(=O)N(CC(CNC(C(=C(C)C2CC2)F)=O)(C)C)C)cc(Cl)cc(Cl)c1 C12(CNC(C3(C(=O)NC(C#C)CC4CCCO4)CC=CC3)=O)CCC(OC)C1C2 Cc1nn(C)c(C(=O)N(CCNC(=O)Cc2cnc[nH]2)C2CC2)c1Br C(CN=c1[nH]c(C(F)(F)F)nc2c1CC(C)CC2)c1c(C)noc1C C(c1ccc(F)cc1)=CC(=O)NC(CNC(C1(C#C)CCCC1)=O)CO N1(C(CCSCC)=O)CCOCCC1C(=O)NCCn1ccnc1C c1(C(=O)NC(CC)CN(C(=O)C2=CCN(C)C2)CC)cc(Cl)cc(Cl)c1[N+](=O)[O-] Cc1cc(C(=O)NC2CCCN(C(c3cc(C(F)F)cc(F)c3)=O)C2)ncc1F Cc1oc(-c2ccccc2)nc1C(=O)NCC(C)NC(=O)CC1COCC1O Cn1ccnc1C(=O)NCCCN(C(=O)CCCN1CCCCC1)CC1CCCC1 C1(C(c2n(C)ccn2)N2CCCC2CC(=O)NCCCCCO)CCC(=O)NC1=O c1(C(=O)NC2C(C(N3CC(SCC)C3)=O)COCC2)cccc(C#N)c1C Cc1cccc(C(=O)NCC2CCC(C(=O)NC3CCCSC3)CC2)n1 c1(CC(=O)OCC)cc(C(=O)NC2(CNC(c3ccc[nH]3)=O)CCC2)cs1 N1(C(CS(CC)=O)=O)CCC2(C1)CN(C(C1CC1(Cl)Cl)=O)CCO2 N1(C(c2c(C)ncc(C)c2)=O)CC2CCN(C(=O)COCC3(F)CC3)CCC2C1 C=CCCCCCCC(=O)N1CC2CC1CN(C(c1cc(Cl)c(Cl)cc1N)=O)C2 c1(C(N2CCC(CNC(=O)CC3CCCCC3)(CO)C2)=O)cnn2c1OCCC2 N(C(=NCc1cn(C)nn1)N1CCC(OC(C)(C)C)C(C)C1)CCOC c1(C(=O)NCC(CC)(CC)NC(C2CCCSC2C)=O)cc(O)cc(F)c1F C(=O)(C(C)(F)C(C)(C)F)N(CCC(C)NC(C1(C2CC2)CC1)=O)C Cc1cc(C(N2CC3CC2CN3C(c2cccnc2SC(F)F)=O)=O)cc(N)c1 Cc1ccc(SC(C)C(=O)N(C)CC2CN(C(c3nocc3C)=O)C2)cc1 c1(C(=O)OC)cn2ccccc2n1.C1C(O)C(=O)OCC2CC2C(C(=O)OC)N1 Cc1cc(C(N2CCN(C(C3C(C)C3C)=O)CC2)=O)c2c(C)n[nH]c2n1 C(C(C)(C)CC(=O)N1CC(C(=O)NCC(C)CC(C)C)CCC1C)OC CC1=C(C(=O)N(C2CCN(C(C3CCCN3N=O)=O)C2)CCO)C(=O)OC1(C)C C1(NC(c2cnccc2Cl)=O)CN(C(c2cc(C3CCC3)on2)=O)CCC1CO Cc1ccnc(C(N2CCC(NC(=O)C(n3ccc(C4CC4)n3)C)C2)=O)n1 C#CCC(CC(F)F)C(=O)NC(C)(CNC(C1CCCN(C(C)=O)C1)=O)CO c1(C(C(=O)N2CC(CNC(Cc3cnc(C)[nH]3)=O)C2)(C)O)ccc(F)cc1 c1(CNC(c2cc(C)nn2C)C)cc2c(O)cccc2nc1O CCCC(C(=O)NCC1(CO)CCCN(C(=O)CC2(CO)CCC2)C1)C(C)C n1(CC)cc(C(=O)NC2C3CCN(C(=O)CCc4nc(C5CC5)no4)C23)c(C)n1 C1(C(=O)NC(C#C)(C)C)CC(F)CN1C(C1CC(=O)CS1)=O C(=O)(CCS(C)(=O)=O)N(CC(CN(C(C1(CC)CCCCC1)=O)C)O)C N1(C(C(CC)(C)F)=O)CC2CCC1C(CNC(C1CC(=O)N(CC(C)C)C1)=O)C2 c1(CNC(C(CC=C)C)=O)ccc(CNC(=O)CCOCC2CCCO2)c(F)c1 C(=O)(C(CC=CCl)c1ccccc1)NC1CC(NC(c2ccc(C(C)C)o2)=O)C1 c1(-n2c(CCC=C(CC)CC)nc(-c3occc3C)n2)cc(Cl)ccc1C N#Cc1cccc(C(=O)NCC(=O)NC2CCCCC2CN(C(=O)CCF)CC)c1 c1(NC(C)C(=O)NC2CCN(C(C3(F)CCCC3)=O)CC2F)ccc(Cl)cc1Cl N1(C(c2ncsc2Br)=O)CC2CCCC(C1)N2C(C1CCCO1)=O C(=O)(C1CCCn2ccnc21)NCC(CNC(c1nccc(OC)c1F)=O)(C)C Cc1ccccc1NC(=O)C(c1csc(Br)n1)N(C)C(c1ccco1)C C1(N(C(=O)Cc2csc(S)n2)C)CN(C(=O)CCCF)CC1F C1(CC)CCC(CNC(C2CCC(NCc3cnn(C)c3C)C2)=O)CC1 c1(C(CC)C)nc(N2CC(OCCNC(=O)CCCc3nc(C)no3)C2)cc(C)n1 C1(C(N(CCCCCC)C)=O)CC(NC(=O)C(C2CC2)SC)CCO1 N1(C(c2c(C)nn(C)c2)=O)CCC(O)(C(C)NC(c2cc(C3CC3)on2)=O)CC1 CON1CC(C(=O)NC2CCCC(NC(C3OCCCO3)=O)C2)CC1=O C1(CNC(CNC(CCCCC)=O)=O)C(C2CC2)CCN1c1ncc(C)c(O)n1 c1(OC)nc(N2CC(NC(=O)CC3CC4CCC3O4)C3(CC3)C2)ncc1C c1(C(N2CC(CN(C(=O)C(O)C3CC3)C)C2)=O)cn2ccccc2n1 c1(C(=O)NCC(CO)NC(=O)Cc2c[nH]nc2O)c[nH]c2cnccc12 C1(C(N(CCCOC)C)=O)CC(C)CN(C(=O)Cn2cc(C#N)cn2)C1 N1(C(C(C)OCC2CC2)=O)CC2CC(C(=O)NCC3C(C)(C)C3(C)C)(C2)C1 N1(C(c2nc(N(C)C)oc2)=O)CC2CC2(NC(C2CC(CC(C)(C)C)C2)=O)C1 c1(CNc2cn(C)c(C(=O)NCCF)n2)cccc(C(F)(F)F)c1Cl Cc1noc(NC(=O)NC2CCC(OC(F)(F)F)CC2)c1Cl C12(NC(c3c(Cl)n[nH]c3C3CC3)=O)CCN(C(c3c(O)cccc3F)=O)CC1C2 CC1CC(NC(c2cccc(N)c2)=O)CCN1C(=O)CC1(C)CC1(Cl)Cl C1(NC(COC(C)C)=O)CCC(C)N(C(=O)COc2ccc(C(F)(F)F)cn2)C1 N1(C(=O)C=Cc2ccco2)CC2CC(C1)C(CO)C2NC(C(CC)(C)C(N)=O)=O c1(OC)ccc(C(=O)NCC2(NC(=O)Cc3ccno3)CCOC2)c(OC)c1 C(=O)(CCCC(N)=O)NCC(CNC(=O)CCc1nnc(SC(C)C)o1)OC N1(C(CSc2n(C)cnn2)=O)CCN(C(c2nc[nH]n2)=O)C(CO)C1 Cc1cn2c(C(=O)NCCn3cc(-c4cccc(N(C)C)c4)nn3)cnc2s1 C1(C(N(CCNC(c2c(C(C)C)n(C)nc2)=O)C2CC2)=O)CC2C=CC1CC2 Cc1cccc(C(N2CC(NCc3n[nH]cc3Cl)C3(CC3)C2)=O)c1O C1(C(N2CCCC(OC(C)C)C2)=O)COCCN(C(=O)C2=COCC2)C1 C1(C(N2CCN(C(c3c(C)cc(F)cn3)=O)CC2CF)=O)CCC2CC1C2(C)C c1(C(C(=O)NC2C(CC)OCC2)C)ccc(Br)cc1F c1(C(=O)NCC(C2CC2)NC(=O)C(O)CC(F)(F)F)ccc2c(c1)CCCS2 CC12COCC1(C)CN(C(C1CCCN1C(c1cc(C#N)cs1)=O)=O)C2 Cc1cc(C)n(CC(=O)NCC(C(C)C)NC(=O)Cc2ccc(F)cn2)c(=O)n1 C(=O)(CC(=O)NC1CC1)NC(C1CCN(C(=O)C=CC2CCOC2)C1)C C1(NC(COCCNC(CCc2nc(=N)[nH][nH]2)=O)=O)CCC2(CCCC2)C1 C1(C(=O)NCCCc2ccncc2)C2CN(CC3COCCO3)CC12 C1(CN(C(c2ccn(C)n2)=O)CC)CN(C(=O)CCc2conc2C)CC1(C)C n1(CCN(C(=O)C(=O)NC2CCC(SC)C2)CCO)c(=O)n(C)c2ccccc12 c1(C(N2CC(O)(CNC(CC(C)C)=O)C2)=O)ccc(Br)c2ncccc12 N1(C(Cc2ccc(C)nc2)=O)CC(CNC(C2(F)CCCC2)=O)CCC1C c1(C(=O)NC(CC(C)C)C(=O)NC2CCc3nncn3C2)cc2cccnc2[nH]1 c1(CSC)ccc(C(N2CCCC2C(C)(C)NC(=O)C=CI)=O)o1 C1(NC(C(CC)OCC)=O)CN(C(c2coc(COC)c2)=O)CC1C(F)(F)F Nc1ccc(F)c(C(=O)NC2CCC(NC(C3CCCN3C3CCCC3)=O)C2)c1 C=CCC(CC)N=c1[nH]c(N2CCN(C3COCC3O)CC2)nc2c1COC2 C(C(C(C)(C)C)NC(=O)CC1CC1)NC(C(C1CCCCCC1)C)=O Cc1nc(C=CC(=O)NCC23CC2CN(C(c2ccncc2CO)=O)C3)[nH]c1C C1(CNC(COCCOC)=O)CC2(CCN(C(=O)CCc3cc[nH]n3)C2)CO1 c1(C(N(C)CCN(C)C(C23CCC(C2)C3)=O)=O)cn(C)nc1-c1cccs1 c1(OC)cccc(C(=O)N(CCNC(=O)COc2cccc(C)c2)C2CC2)c1F Cc1ncnc(C(=O)N(C(C)CNC(=O)CSCC2CCCO2)CC)c1C C1(CC)(NC(=O)CC=Cc2ccccc2)CCN(C(C2CCOC2=O)=O)CC1 c1(C(c2nc(Br)cn2OC)N(CCCC)C(C2CC2)C2CC2)ccc(C)c(C)c1 O=S(=O)(C1Cc2ccccc2C1)N1c2ccc(Br)cc2CCC1C(F)F C1(C)(NC(CN(C2CCCC3CC23)C)=O)CN(C(=O)C=CC=C(Cl)Cl)CCO1 c1(C(=O)NCC2N(C(C(Br)=C(C)C)=O)CC2)ccccc1C1CC1(F)F C(=O)(CCC(F)(F)F)NCC(=O)NC(=O)NC.C1(=O)CN(CC)CCCN1 C1(CC2(CC(=O)NC3CC(CNC(=O)CCC(F)(F)F)C3)CC2)CCOCC1 c1(C(N(CC)Cc2nccc3c2NCCC3)=O)cc(O)c2cnn(C)c2c1 N1(C(COCCC)=O)CCN(C(C2CCCC3(CC3)C2)=O)CCC1C O(C=CC(=O)NCCc1ocnc1CNC(=O)C(C)(O)c1ccccn1)CC Cc1cc2c(C(=O)NCC3C(C)CCN3C(=O)COC3CCCC3)cccc2[nH]1 CC(O)C(C)(C)C(=O)NC1CC(CCNC(=O)COc2cc(F)cc(F)c2)C1 C1(NC(c2c(C)ocn2)=O)C2CC1N(C(C1(C)COC(=O)N1)=O)C2 C(Cc1ccoc1)(C(=O)NCC=CC(F)(F)F)NC(c1csnn1)=O CCC(CNC(=O)C(CCSC)OC)(CC)NC(=O)Cc1n[nH]c(C)n1 C1(CNC(C(CSC)C)=O)CCCCN1C(=O)CC[SH](C1CCCO1)CCO CC1CN(C(C2(C)CCN(C(C3CCC(=O)N(C)C3)=O)CC2)=O)c2cccnc21 CC(C)C(F)(F)CCNC(=O)C(C1CC1)N(C(=O)CCCN=[N+]=[N-])C N1(CC)CCCN(C(c2ccnc(C)c2)C(=O)NCC2CC2)CC1=O C1(NC(C(=O)N(C(c2cccc(Cl)c2)COC)C)=O)CCOC2(CCC2)C1 N1(C(CC2N(C(c3ncn(CC)c3)=O)CCCC2)=O)CC2CCCC2C1 CCC(C)CCCCC(=O)NC(C1(C(=O)Nc2c(C)cccc2O)CC1)C Cc1nc(N2CCCC2CN(C)C(C2CCCCC(F)(F)C2)=O)ncc1[N+](=O)[O-] N1(C(C(C=C)O)=O)C2CC1CN(C(=O)CC(C)NC(N)=O)C2 C1(C(N2C(CC(=O)Nc3cccc(CO)c3)CCCC2)=O)CCCNC1=O C1(CC(N)=O)(NC(CCCCOC)=O)CCN(C(c2ccc(CO)cc2F)=O)CC1 C1(C(=O)NOCCn2cncn2)C(C2CC2)CCN1C(C1CC2CCCCN2C1)=O Cc1c(F)cc(C(=O)NC2CN(C(=O)CC3OCCC3(C)C)CC2C)c(F)c1N C1(CC)(CC)NC(=O)N(CC(N2CC(NC(=O)CSCC)C3(CCC3)C2)=O)C1=O n1(C2CCN(C(Cc3ccc(N)cn3)=O)C2)c(O)nc2ccccc12 c1(C(COCCOCc2ccccc2)NC(=O)OC(C)(C)C)ccc(F)cc1F C1(CCN=C(NCc2n(C)c(=O)on2)NC2CCC2)Cc2ccccc2C1 N1(C(C2OCCN(C(C)C)C2)=O)CCCC(NC(=O)CCC(C)(F)F)C1C C1(CC(=O)Nc2cncc(OC)c2)C2CCC(C2)N1C(C1COCC(C)O1)=O C(=O)(CCCC(=O)N1CCN(C(=O)C(F)=C2CCCC2)CC1C1CCC1)OC c1(-c2n(CCC)ncc2)cnn2cc(C(=O)Nc3cnn(C)n3)cnc12 c1(-n2cc(CNC(=O)Cc3ccsc3Br)nn2)ccc(Br)cc1 C=CCC(CC(C)C)C(=O)NCC(C)(C)CC1CN(C(c2cc(N)cc(N)c2)=O)C1 Cc1c(CNC(=O)COC(C)(C)CNC(=O)C(F)n2cccn2)cccc1F C12(C(=O)NC3C(NC(=O)Cn4cnnn4)COC3)CCC(C(F)(F)F)(CC1)CC2 C1(O)(C(CC)NC(C(=O)NCC(CCO)c2cncn2C)=O)CCCCC1 N1(C(CC=C)=O)CCCCC1CNC(=O)CCNC(c1ncc[nH]c1=O)=O C1(O)(CNC(C(C)(c2ccccc2)N(C)C)=O)CCN(C(C2CCOC2)=O)CC1 c1(CC(=O)NC(CO)C(c2cccc(Br)c2)O)c[nH]c2cccnc12 c1(C(=O)NC2CCN(C(CC#C)=O)CC2O)ccc2nc(Cl)ccc2c1 S(=O)(=O)(c1ccc(C)c(C)c1)N(C(CCC)CO)C N1(C(C2(C(C)C)CCOCC2)=O)CCCN(C(c2cc(Cl)cnn2)=O)CC1 CC1CCc2nc(C(N3CCN(C(=O)CC4CCSC4)CC3C)=O)cn2C1 C1(CNC(C2N(C(=O)OCC)CSC2)=O)(NC(C)=O)CCCOC1 C1(C(=O)NCCNC(c2cc(Cl)c(C(F)F)cc2F)=O)CN2CCCCC2CO1 C#CCCCCCC(=O)N1CCC2CN(C(=O)Cc3cc(F)ccc3OC)CC12 CC(C)C(C(=O)NC1COCCC1NC(=O)C(C)N(C)C)OCC1CC1 CCCCCCC(=O)NC1CS(=O)(=O)CC1NC(c1cnn(CC)c1C)=O C1(CC)(CO)CCN(C(C2CC(CNC(=O)CCCC#N)C2)=O)CC1 CC1CCCCNOCCC=C(C(=O)C(C)(C)CNC(=O)C(F)(F)F)C(=O)N1 N1(C(C2CCC=CO2)C(=O)Nc2ccc(OC)cc2)CC(OC)CCC1C CC1CC(C(=O)NC2CCCCC2C(=O)NC(c2ccc(O)cc2)C)CC(=O)N1 Cc1ccc(C(=O)NCC(CC(C)C)NC(C2CC3CCCCC23)=O)c(F)c1F C(=O)(CC(C(F)(F)F)NC(C1CC(CC)C1)=O)N(CCC)Cc1ccco1 C1(CCNC(c2coc(-c3ccccc3)n2)=O)CCN(C(=O)COCC(F)F)C1 N1(C(=O)CN2C(=O)CCC2=O)CCCC2C1CCN2C(c1ccnn1CCF)=O c1(CC(=O)NCC(C)(C)CNC(c2ccc(O)nc2)=O)ccc2c(c1)NC(=O)C2 C1(C(=O)NC2(CC(N)=O)CC2)(NC(C2CCC2(F)F)=O)CC(O)C1 CCC(CC(=O)NCCc1cc(C)[nH]n1)NC(=O)CC1CCSCC1 C(C(O)C(F)(F)F)OC.C1(COC(=O)CC2(CN)CC2)SCC=C1C Cc1nn(CC(=O)NC2CCCC2NC(C2(c3ccc(O)cc3)CC2)=O)cc1Cl c1(C(N2CC(CCNC(C3(CC)CCC3)=O)C2)=O)ccc2c(c1)CCN2 C1(O)(C(C)NC(c2c(OC)c[nH]n2)=O)CCN(C(C2CCC(CO)CC2)=O)CC1 c1(C(=O)NCC2(C(N)=O)CN(C(C34CC(CO3)C4)=O)C2)nc[nH]c2nccc1-2 Cc1nc(C(C)C)nc(O)c1C(=O)NC(C)CN(C)C(C1(CF)CC1(F)F)=O c1(-n2c(CCCOCCOC)nc(-c3ccnc(Cl)c3)n2)ccc2nncn2n1 CS(=O)(=O)c1ccccc1NC(C1CCN1Cc1cccc(Cl)c1C(=O)O)=O Cc1cccnc1C(=O)NCC1CC1NC(c1cccc(C(F)(F)F)c1)=O C1(C(=O)NC(C2CN(C(=O)Cn3ccc(O)nc3=O)C2)C)CCn2nncc2C1 N1(C(C=C(C)c2cccnc2)=O)CCC2CC2(NC(=O)CS(N)(=O)=O)CC1 C1(NC(=O)C=C(Cl)Cl)CCCC2CN(C(C3CCCC4CCCN34)=O)CC12 C1(CC=C)(NC(c2cc(O)cs2)=O)CCN(C(=O)CC(C)(F)F)C1 N1(C(=O)NC(c2cccc(C)c2)C2CC2)CCCc2nc[nH]c2C1 N1(C(c2cc(C)on2)=O)CC2(C=C(C(=O)NC3CCOC(C(C)C)C3)CO2)C1 Nc1cc(C(N2CCC(NC(=O)C(=O)NC3CC3)C(O)C2)=O)cc(O)c1Cl C1(C(=O)NC2(C=C)CCC2)CC12CCN(C(C1CC(=O)C13CCC3)=O)C2 C(=O)(C(C)(F)C(C)(C)F)NC1CN(C(c2c(C)nn(C3CCC3)c2)=O)CC1(C)C CC1(NC(c2cn(C3CC3)cn2)=O)CCN(C(=O)Cc2ccccc2Cl)CC1 N1(C(C(C(=O)NC)(C)C)=O)CCC2(CC1)CC(C)N(C(=O)C=CC=C(Cl)Cl)C2 c1(C(C)NC(C2CC(O)(c3ccccc3)C2)=O)cc2cnccc2o1 c1(C(C)=O)cn(C)nc1C(=O)NC1CC(NC(c2ccnc(C(F)F)c2)=O)C1 Cc1ccc(I)c(C(=O)NCCC2CCCN(c3nc(C)cc(C)n3)C2)c1 C=CC(C)(C)CC(=O)NCC1C(C)CCCN1C(=O)Cc1cn(C2CC2)cn1 CCC(CCC(=O)NCCCC(C)NC(C12CC(C)(CCO1)C2)=O)OC C1(NC(=O)CC2CC=CCC2)CCOCC1NC(=O)C(O)(C1CC1)C1CC1 c1(C(N2CC=C(C(=O)N(C3CCCOC3)CC)C2)=O)cccn2nccc12 C(C(C)(C(C)C)NC(C1CCCN1C=O)=O)NC(C=CC(=O)OCC)=O C(C(O)C(=O)N(C)CCNC(=O)C(C)C)NC(C(C)OC)=O O=C1CCC(C(=O)N2CCC(CCNC(=O)C(c3cccc(F)c3)CO)C2)=NN1 C(=O)(C1=Cc2ccccc2C1C)NCCN(C(C(CC)CC1CCCC1)=O)C c1(CC)nn(C)c(C(=O)NCC2CN(C(c3ccc(OC)nc3)=O)C2)c1Cl C1(NC(Cc2nc(C(C)(C)C)sc2)=O)CCCC12CCN(Cc1ccccc1)CC2 c1(C(N2CC(O)(CNC(CC(=C)C)=O)C2)=O)cc2ccc(C)cc2o1 c1(NC(c2n(CC(=C)C)nnn2)c2ccsc2C)ccc2ncccc2c1 c1(OC)cc(OC)c(F)c(C(=O)NC(C2(O)CN(C(c3cn[nH]c3)=O)C2)C)c1 c1(C(=O)NCC(N(C(=O)C(F)n2cccn2)C)C2CC2)cc(Cl)on1 c1(OC)cc[n+]([O-])c(C(N2CCN(C(c3conc3C)=O)C(C3CC3)C2)=O)c1 C(=O)(C(n1nnnc1C)=C(C)C(=O)N1CC(C2(C(=O)OC)N=N2)C1)OC N1(C(C2N(CCCC)CCCC2)=O)CCCN(C(=O)Cc2cnsc2)C(CO)C1 C=CCC(CNC(c1ccc(C)[nH]1)=O)C(=O)NCC(COC)C(C)C c1(C(N2CCC(C(=O)NCC(C)C(F)(F)F)C2)=O)coc2ccccc12 CCCC(O)CC(=O)NC(CNC(=O)C(F)(F)c1csc(=N)[nH]1)CCOC C12(C(=O)Nc3cnn(CC(F)F)c3)CCCC1CN(C(=O)COCC1CCC1)C2 N1(C(C(CCC)C#N)=O)CC(C2CCCN(C(c3ccnc4[nH]cnc34)=O)C2)C1 C(=O)(C(O)C1=CCCCC1)NCc1scc(C(=O)NC2C3(CC(OC)C3)C2)c1 n1(CCCC)nc(C(N2CCCC2C(C)(C)CNC(=O)CCOC)=O)ccc1=O C(=O)(CS(=O)(=O)CC(F)(F)F)N(C(C)C)CCNC(C1CC1c1cnn(C)c1)=O C1(CNC(Cc2ccc(C)cc2Cl)=O)CCC2(CCC2)C1NC(=O)CC(C)(C)C CC1(C)CC(NC(C2CC2F)=O)CN1C(=O)C(C)(F)c1ccon1 c1(CCC(N2C(CNC(CSCC#C)=O)CC2)=O)cc(Br)ccc1F C(=O)(C(C(C)C)NC(C1CCCC1)=O)NCCN(C(=O)C(C)C(C)O)CCOC C1(CO)(NC(=O)Nc2cncc(OCCC)c2)CCc2cc(Br)ccc21 c1(C(C)(C)C)ccc(C2CC2c2nc(C34CCCC3C4)n(-c3cccnc3)n2)cc1 CC1C(NC(c2ncoc2-c2ccon2)=O)CCCN1C(c1ccc(F)nc1)=O Cc1cc(NC(=O)NCCCC(F)F)c(OC(F)(F)F)cc1C(F)(F)F C1(O)(C(C)OCc2onc(COC)n2)CCN(C(=O)C2=CCCCC2)CC1 Cc1ccc(Cl)c(C(=O)NC2CCN(C(C3NC(=O)OC3(C)C)=O)C2)c1O C1(C2CCN(C(=O)CCC3CC3)C2)(NC(=O)CC2CCOC2)CC1 C1(NC(C(COC)C)=O)CCCN(C(=O)CCc2ccsc2Cl)CC1 c1(C(=O)NCc2c(C(=O)NCC(C(C)(C)C)OCC)occ2)nnc(O)cc1O c1(NC)nc(C)ccc1C(N1CCC(NC(c2ccccc2OCCF)=O)C1)=O C(=O)(C1COc2ccc(F)cc21)NC(C(C)NC(CN(C)CC)=O)CO C1(CN(C(=O)C(C2CCCO2)C2CC2)C)CCCCN1C(=O)COc1ccsn1 C(=O)(CC(C)COC)NCCC(C)N(C(c1ncc(C(F)F)s1)=O)CC C=C1CC(C(N2CC(CF)C2)=O)(CNC(=O)C(c2ccnn2C)O)C1 N1(C(C=C(C)Cl)=O)CC2CC(C)N(C(=O)C3=CCCCCCC3)C2C1 N1(C(c2c(CCC)nns2)=O)Cc2ccc(CNC(C3CC(OC)C3)=O)cc2C1 C(=O)(CCC(=O)NN(C)C)NC1(C(C)C)CCCN(C(=O)CCC(CF)CF)C1 n1(CC(=O)NC(C)(C)CNC(=O)CN2CCCC2CO)cnc2c1CCCC2 N1(C(C(=C(C)C2CC2)F)=O)CCCC(C2CCCCN2C(=O)C2CC2)C1 N1(C(CC=C(C)C)=O)CCCN(C(=O)CN2CCC(C)C2)CC1CO C1(NC(c2cc(C)sc2)=O)CC12CCN(C(c1cc3c(o1)CCCC3)=O)CC2 C(=O)(CCCS(C)(=O)=O)NCC1C(NC(C(C(C)C)OCC(C)C)=O)CCC1 C(=O)(C(C(=O)OCc1ccc(C(=O)OC(C)C#N)cc1)C(C)C)OCC Cc1nc(NC(=O)COC(c2ccccn2)C)c(COC)n1C.c12nc(n[nH]1)C2 c1(CC(=O)NCC2CCCN(C(C(CCN(C)C)O)=O)C2)cccc2sccc12 C1(C(N2CCC(C(C)NC(=O)C(C)(F)F)C2)=O)CCC2(CC1)CC(=O)C2 CC(=O)CCCC(=O)N(C(C)C(N1CC(CO)CC(C)C1)=O)C1CC1 c1(CC)nc[nH]c(=NCC(C)(C)NC(C23CCCC2C3(F)F)=O)c1F C1(C(N2CCCC(NC(C3(C(=O)NCCCC)CC3)=O)C2)=O)CCCC12CCC2 CC(CN(C)C)CCC(=O)N1CC(O)C(O)C1CN(C)C.C12CC(C1)NC2=O c1(C(=O)NC(C(C)C)CNC(=O)Cn2nccn2)ccc(S(N)(=O)=O)cc1N N1(C(C(CC2CCOCC2)NC(C2CC3CCC3C2)=O)=O)CCC2CCC(C1)S2 C1(CC=C)(NC(=O)Cc2cc(SC)on2)CCN(C(=O)C(O)CCSC)C1 C1(NC(c2c(OCC)ccs2)=O)CCCN(C(c2csc(-c3nc[nH]n3)n2)=O)C1 c1(N(C2C3CNCC23)C(c2cc(OC)c(F)cc2)=O)ncnc2c1CCC2 CC1CC(=O)NCC1C(N1CC(O)(C(F)C(=O)NC2CCC2)C1)=O.C1CO1 c1(C(N2CC(CCO)(NC(Cc3cnc(C)[nH]3)=O)C2)=O)cccc(C(F)F)c1 c1(C(N2CCN(CCSc3nc(C)nc(Cl)c3)CC2)=O)ccn2c(O)nnc2c1 c1(C(=O)NCCNC(c2cncc(-n3ccnc3)n2)=O)ccc2nsnc2c1 N1(C(C(CC)OC(C)=O)=O)CCCN(C(=O)OC(C)(C)C)CC1 c1(OC)cc(C(=O)N(CC(=O)NCCOC2CC2(F)F)CCO)[nH]n1 Cn1ccnc1CC(=O)NCCCCCNC(=O)CC1CC(n2cnnc2)C1 c1(C(=O)OC)ccc2c(c1)OC(C)CN2n1nnnc1C12CCC(C1)C2OC C(COC)(C(=O)NOCCC(C)O)NC(C(C)NC(CCOC)=O)=O c1(CNC2CCCN(C(=O)OCC)C2)ccc(Br)cc1Cl C1(C(=O)NCC(C)OCC=C)CC2(CC(NC(C3(Cl)CCC3)=O)C2)C1 Cc1cc(C)c(C(N2CCC3(CCOC3)C2)C(=O)NCCOCC2CC2)cc1C C(CCNC(=O)Cc1c(Cl)cnn1C)(C(C)C)NC(C1(CCOC)CCC1)=O c1(C(CNC(C(CCC)=CCC)=O)NC(C2COC(=O)O2)=O)ccc(F)cc1F O=C(C1=C(F)CN(C(C23COCC2C3)=O)CC1)N1CCN(C2CCC2)CC1 C1(CNC(c2cc(C(C)C)no2)=O)Cc2ccccc2CN1C(=O)CC(C)N(C)C CN1CCC(C)(C(N2CC3CC2C3C(=O)NCCC(C)(C)O)=O)CC1 N1(C(c2c(C(C)C)con2)=O)CCCC(NC(C2CCCCO2)=O)CCC1 CCCCC(O)CCC(=O)NCC(C)(C1CCC1)NC(=O)CC(C)(O)C(F)(F)F c1(C(C(=O)NCC2CCOC2)N(CC(=O)NC)C)cnc(C)nc1 N1(C(C2(C)CCC2)=O)CC(CO)C2(C1)CN(C(=O)Cn1cnnn1)C2 N1(C(c2ccc(CCCC)o2)=O)CC(C)(C)CC1CNC(c1ncsc1OC)=O N1(C(c2c(C)nc(C)nc2C)=O)CCC(NC(=O)COCC(C)C)CC(C)(C)C1 c1(OC)ccc(N=c2[nH]c(Cn3cccn3)nc3ccc(Cl)cc23)cc1 C1(NC(C(C2CC2)OC)=O)CC=C(C(=O)N(C)CC2(C)CCCC2)C1 C(=O)(C(CCSC)NC(C1COC(=O)N1C)=O)NCC(=O)OCCCC C1(C(CNC(CCNC(=O)OC(C)(C)C)C)OC(CCCC)=O)CCCCC1 C1(C)(C(N2CC(CN(C(c3c(C)cc[nH]3)=O)C)OCC2)=O)CCCCNC1=O Cc1nn(CC(N2CCOCC2CNC(c2cc(F)cs2)=O)=O)c(C)c1Cl c1(C(=O)NC2C(C(N3C(C(N)=O)CCCC3)=O)CCC2)ccc(O)cc1O N1(C(C(COC)OC)=O)CCCC(C(=O)NCC2CCOC2C)C1 CC1CCCN(C(c2ncccc2N)=O)C1CC(=O)NCc1ncccc1CO CCC(CNC(=O)C(C)C1CCC1)(CC)NC(c1cc(C2(C)CC2)on1)=O N1(C(c2c(CC)nns2)=O)CCCCC1CNC(c1cc(=N)[nH][nH]1)=O N1(C(c2c(C)c(CSC(C)C)ccc2)=O)CCOCC(C)(NC(C2CCC2)=O)C1 N#Cc1ccc(NC(C2CC2NC(c2ccc(F)c(F)c2Br)=O)=O)c(C#N)c1 Cc1cc(C(N2CCC(C(C)NC(c3nocc3C)=O)C2)=O)c(N)s1 n1(CC)nc(C(=O)NCCOCCCN(C(=O)C=CC2CCCN2C)C)cc1C C1(NC(C(F)=CCC)=O)CCC(C)N(C(c2ccnc(OCC)c2F)=O)C1 c1(C(=O)NCCC(C)N(C(CCC(C)CN(C)C)=O)C)cc2cc[nH]c(=O)c2s1 CN1C(=O)CCCc2occ(C(=O)NCCC(C)(C)NC(c3cscn3)=O)c21 c1(C(C)(C)C)ccc(F)nc1NC(=O)CC1CN(Cc2cccc(Cl)c2F)C1 C12(NC(CCSCC)=O)CC(C1)N(C(=O)CCOCCOC)C2 C(=O)(CC1=CCOCC1)NC1C(C2CN(C(C=CC(C)(C)C)=O)C2)CCCC1 c1(-c2ncc(C(=O)NC3(C)CC(NC(CCC4C(C)C4)=O)C3)s2)cccc(F)c1 C1(C(N2CC(F)(CNC(C3CCCCO3)=O)C2)=O)Cc2cc(Cl)ccc2O1 Cn1cc(Cl)c(CC(=O)NC(CNC(c2ccc[n+]([O-])c2)=O)CO)n1 C(c1ccc(O)cc1)=CC(=O)NC1C2CN(C(C=C3CCC(C)CC3)=O)C1C2 NC1COc2c(C(=O)NC3(C(N)=O)CC4CCC3C4)cnn2C1 c1(C(=O)NCCCN(C(C2CCCN(C(C)=O)C2)=O)C)cncc(Cl)c1C N1(C(c2c(C)cns2)=O)C(C)CN(C(C2(C(F)F)CCCCC2)=O)CC1C C(=O)(C1CCCc2scnc21)N1C(CNC(C2CCOCC2)=O)CC1 c1(C(C(=O)NCCCN(C)C(C2(C(N)=O)CC2)=O)(F)F)cccc2ccccc12 C1(C(=O)NCCCCC)CCN(C(c2occ3c2CCC3)=O)CC1(C)C C(C)(CNC(=O)CN(C1CCC1)C)(CC(C)C)NC(CCn1c(CC)ncc1)=O c1(C(N(C2CCN(C(c3cnc[nH]c3=N)=O)C2)CC)=O)[nH]c(C)cc1C c1(SC)cc(C(=O)N(C)CC2(O)CCN(C(c3[nH]c(C)nc3C)=O)C2)ccc1F N1(C(=O)CCCc2ncco2)CCC2(CCN(C(c3cnsc3)=O)C2)C1 C(C)(C)(CCC(=O)N(C)OCC#N)Nc1ccnc(NC(C(CCC)C#N)=O)n1 C1(C)(C(=O)NCC(CNC(=O)Cc2ccc(Br)nc2)OC)CCN(C)C1=O c1(OC)ccc(Cl)c(C(=O)NC(C)C(C(C)C)NC(c2nncs2)=O)c1 c1(CCC(N2CC3C(NC(C(C)(O)C4CC4)=O)(C3)C2)=O)ccc(Cl)c(F)c1 C(=O)(CC1OCc2ncccc21)NCCNC(c1cnc(C(C)(C)C)s1)=O C1(NC(C2CC(OCC)C2)=O)CN(C(=O)C2=COCCO2)CCC1(C)C c1(OC)ccc(C(N2CCOC(CCNC(=O)Cc3cnccn3)C2)=O)cc1 Cc1cc(CC(=O)NCC2(Nc3ccnc(C(C)(C)C#N)c3)CCCC2)sc1Br C1CCCC2(C1)CC2(F)F.CC(CO)C(=O)N1CC(O)(c2cn(C)nn2)C1 C(CCN=C(NCC1(OC)CCCCC1)N1CCCC(C(O)C(F)(F)F)C1)OC C#CC1CCCC1NC(=O)C(C1(O)CN(C(=O)CCOC2CCC2)C1)F C1(N(C(C(CC)F)=O)CC)CCCN(C(=O)CCCCF)C1 CC1CN(C(C2CN(C)CCO2)=O)CC(C)N(C(C2CCCCC2O)=O)C1 c1(NC)ccc(CCC(N2CCNC(=O)C2C(=O)NC)=O)cc1Cl c1(C(N2CCC(CNC(CC(C)SC)=O)C2)=O)ccc([N+](=O)[O-])c(C)n1 c1(C(COC(CC(C)(C)SC(C)=O)=O)=O)c[nH]nc1S(N)(=O)=O C(=O)(CC(C(C)C)C(C)C)N1CCN(CCCNC(C2C(OC)CCC2)=O)CC1 CC1CN(C(C2CCN(C(C3(N(C)C)CCOCC3)=O)CC2O)=O)CCN1C c1(OC)cncc(C=CC(=O)NCC2C=CC(NC(C3(F)CC=CCC3)=O)C2)c1 C1(NC(c2ccc(COC)s2)=O)CCCCC1C(N1CC(OC(=N)O)C1)=O C1(C(N(c2cccnc2)C)=O)CN(C(=O)Cc2cncnc2)CC1F C(C1OCc2ccccc21)NC(=NCCCC)NCC1(F)CCOC1 Cc1ccnc(O)c1C(N1CC(CC(=O)NCCc2cccc(O)c2)C(C)C1)=O C(=O)(CCCCCNC(=O)C=CCOCCOC)NCCC(CCC)C1CC1 c1(C(N2CC(CCNC(COCC)=O)OC(C)C2)=O)nccn2ccnc12 CN1CCCC(C(N2C(C(N3CCCC3(C)C)=O)CC3CC23)=O)C1 C1(O)(C(=O)NCCC(C(=O)NCC#CCC)O)CCC(C)CC1 C1(CC=C)(NC(c2nn(C)c(Cl)c2Cl)=O)CCN(C(=O)Cc2nncs2)CC1 C1(C(=O)NCC2C(NC(C(COC)O)=O)COC2)(COC)CCOCC1 C1(NC(C)=O)CC2C(NC(=O)CCn3cncn3)C2C1 N1(C(CN2C(C)CCC2)=O)CCC2(CC1)CC2NC(c1cc2nc[nH]c2cn1)=O C(CCNC(c1ccc(C(C)(C)C)cc1)=O)(C(C)C)NC(C1C(OC)C1)=O CC1CN(C(c2sc(F)cc2Br)=O)CC1CCNC(=O)CC1CC1 C(=O)(C1=NOC(C)(C)C1)NCC(c1ccc(C)cc1)NC(c1cncnc1)=O c1(C(=O)NC(CN(C)C)C(=O)NCc2nnnn2C2CC2)cccc(F)c1O C(=O)(C1=NOC(C)(C)C1)NC1CCCC(NC(C(CCC#C)O)=O)C1 C1(NC(c2nc(C)n(C)n2)=O)CN(C(C2CC3(CC(=O)N3)C2)=O)C2CCCCC12 C(C)(C(CC(=O)NCC(c1ccnn1C)O)NC(=O)CN1CCCCC1=O)OC c1(CNC(C2CC3CCC3C2)c2n(CCCC)nnn2)cccc(SCC)c1 C=CC1CN(C(c2c(C)coc2C)=O)CC1NC(=O)C(C(C)OC)N(C)C CC1=C(C(=O)NCCC2CCC(NC(C3CCN(C(N)=O)CC3)=O)C2)CCO1 C1(CC(=O)N(C2(CNC(C3CSCCS3)=O)CC2)C)CC2(CC2)C1 Cc1c(C(=O)CNC2CCCC(C)C2)cccc1O c1(C(N(C(C)CNC(=O)COCC2CC2)C)=O)cc2ccc(F)cc2o1 C1(CC)CCC(CNC(c2[nH]ccc2CNC(=O)C(C2CCCCC2)F)=O)O1 c1(C(=O)NCC2OCC(CNC(=O)C=CSc3nc[nH]n3)C2)cc(Cl)ccc1O C(=O)(CS(C)(=O)=O)NCCCCNC(c1cc(NC(=O)OC(C)(C)C)n[nH]1)=O Cc1nn(C)cc1CCNC(=O)CCC1CCC(NC(=O)COC2CCOC2)C1 C1(n2cc(NCc3n(CC)ccn3)nn2)CCN(Cc2ccncc2C)CC1 C1(C(N2C3C(NC(C4C(C)(C)CCO4)=O)C(C3)C2)=O)CC2CCC(C1)C2 C(CC(=O)NCC1CC(=O)N(C)C1)(C(F)(F)F)NC(c1c(CC)con1)=O N1(C(=O)NC2N(C(=O)OC)CCCC2)CC2(C)CC1CC(C)(C)C2 CC1CCC(C)N1CC(=O)NCC1(O)CCN(C(c2csnn2)=O)C1 C1(CCOC)(NC(c2occ(C)c2C)=O)CCN(C(=O)C=CC(=O)N(C)C)C1 c1(C(N2C3C(NC(CNC(C)=O)=O)(CCC3)CC2)=O)[nH]c2cc(F)ccc2c1C Cc1scc(C(=O)NC2CCN(C(c3cccc(CO)c3)=O)C2C)c1C C1(C(=O)NCC2N(C(C=CC=CC)=O)CCN(C)C2)CCC2(C1)CC2(F)F CC(C)CC(CCO)NC(=O)C(O)C1CN(C(C23CCCC2C3)=O)C1 C(=O)(CCCCC1CC1)NCCN(C(C(C)Cc1ccncc1)=O)C1CC1 c1(C(N2CC(O)(CNC(COCCCC)=O)C2)=O)ccn2nncc2c1 c1(C(N(C2(C#N)CCNC2)c2ncncc2I)=O)cc([N+](=O)[O-])ccc1Cl C1(CC(C)(C)C)CN(C(=O)CCn2ccnc2)CCN1C(c1c[nH]c(C#N)c1)=O c1(OC)ccc(CC(=O)NC2CN(C(c3ccccc3)=O)CC2C(=O)O)nc1 N1(C(c2cc(-c3ccn(C)n3)on2)=O)CC2(CCCCN2C(=O)CCCF)C1 C1(CNC(c2n[nH]c(CC)c2Cl)=O)N(C(C2C=CCS2)=O)CCCC1(C)C CCCN=C(NCCC1(C)CC1(F)Cl)NC1CCN(C(C)C)CC1 c1(C(=O)NC2CN(C(c3c(OCC)scc3)=O)C(C)CC2)cccc2c1NCC2 C(C#Cc1cccc(C)c1)OC(CC(CC)SC)=O c1(N2C(CNCc3ccc(CCC)cc3)CCCC2)ccc(C)cc1F N1(C(C2CCC(CCC(C)C)CC2)=O)CCC(O)(CNC(=O)C=CCF)CC1 c1(OC)cccc(C2C(=O)N2)c1.C12(C(=O)NCCSC)CC(F)(CO1)C2 c1(OC)ccc(NC(=O)C(O)C2CN(C(c3cc(C)sn3)=O)C2)c(O)c1 C(=O)(CC(N=c1[nH]c(NCCCNC)nc(=N)[nH]1)c1ccccc1)NC.SC C1(C(=O)NCC(O)C(=O)N2CCC(F)C2)CC12CCCCC2 c1(C(N(C)CC2OCCN(C(CCC=C)=O)C2)=O)ccn2ccnc2n1 Cc1onc(-c2cccc(Cl)c2)c1C(=O)NCCC(C)NC(=O)CCOC1CC1 N1(C(C=CC=CCC)=O)CCC2CCC(C1)N2C(c1cnc(OC)c(C)c1)=O c1(C(N2CC(O)(CNc3cc(SC)ncn3)C2)=O)cccc([N+](=O)[O-])c1 C1(C(N2C(C)CN(C(=O)CCc3ncco3)CCC2)=O)CC2(CO1)CC(F)(F)C2 C12(NC(Cc3ncc(C)s3)=O)CCCC1N(C(=O)Cc1ccc3c[nH]nc3c1)CC2 c1(C(=O)NC2C(NC(C3N(C=O)CCC3)=O)C2)ccc2ncnc(O)c2c1 C(=O)(C1=C(C)OCC1)NCC1CCN(C(C2C(OC)(OC)CC2)=O)CC1 CCCCC(C)(F)C(=O)NC(CO)C(C)NC(c1cc(C)nn1CCC)=O CC1CN(C(=O)CCCc2ncco2)CCCN1C(c1ccsn1)=O c1(OC)cc(C)c(C(N2CC(NC(=O)CCC=CC(C)C)C(O)C2)=O)cn1 C12(C(NOCC(=O)N(C)C)=O)CCN(C(C3CCC(F)(F)C3)=O)CCC1C2 n1(CCC)nc(C)c(C(N2CCOCC(CNC(C3CCC3CF)=O)C2)=O)c1C C(CC(=O)NC1CN(C)CC1(C)C)(C(F)F)NC(C1(NC(C)=O)CCCC1)=O C1(C(NCP(C)(C)=O)=O)(NC(C2CC(SC)C2)=O)CCC(C)(C)C1 CCC(C)CC(=O)C(=O)NC(C1CCCC1)CNC(c1ccccc1F)=O c1(NC(C)C(=O)N(c2ccccn2)C(=O)C2CC2)nc(C2OCCO2)cs1 N1(C(C(=CC2CCCC2)C)=O)CC=C(C(=O)N2CC(F)(F)C2C2CC2)C1 c1(C(C(=O)NC(CCNC(C=C(C)Cl)=O)C)(C)F)ccccc1F Cc1c(C#N)c(N2CCCC(Cc3ccccn3)C2)nc2ccccc12 c1(CNC(C2C(NC(Cc3cccc(OCC)c3)=O)C2)=O)ccn(C)c(=O)c1 c1(C(C(C)C)=O)ccc(C(N(C)Cc2cn(CCCNC(N)=O)nn2)=O)cc1 C1(C(=O)NC(C2CCCCC2)C)(OC)CCN(C(=O)CC(O)CN(C)C)C1 C(=O)(CC(C(C)C)NC(=O)CC1CCCC(=O)C1)NC(CSC)C N1(C(CN(C(C(C)C)=O)C)=O)CCCC2(NC(c3c[nH]nc3C3CC3)=O)CC2C1 C(CNC(c1c(C)ncnc1C)=O)(C(C)C(C)C)NC(c1c(C)sc(Cl)n1)=O N#Cc1c(NC(c2n[nH]cc2NC(c2c(Cl)cc(Cl)cc2Cl)=O)=O)cccc1Br c1(CN(CC(=O)NCC(CNC(C2C3COCC23)=O)CO)C)ccc(F)cc1 C1(NC(CC(C=C)CC)=O)CCC2(CC1)CN(C(=O)CCCS(C)(=O)=O)CCO2 C1(C(=O)NCC2CC(NC(CC3N(CC)C(=O)CC3)=O)C2)CC(=O)NC1(C)C c1(C(=O)NC2C(NC(CC(=C=C)C)=O)CCC2)ccc(S(=O)(=O)N(C)C2CC2)cc1 C1(Cc2ccoc2)C(=O)N1.C1(C(=O)OC)CC1(Cl)C(=O)NC(C(=O)OC)C1(C)CC1 c1(OC(C)C)cccc(C(=O)NCC2CCC(NC(=O)CN(C)S(N)(=O)=O)C2)n1 c1(C(C(=O)NCCN(C(=O)CCn2c(C)csc2=O)CC)(F)F)ncccc1F C1(NC(C(=O)NC(c2cn3ccsc3n2)C)=O)CCc2c[nH]nc2C1 N1(C(c2c(C(=O)OC)csc2)=O)CC(CNC(C2CN(C)CCO2)=O)C(C)C1 CCCC(C(=O)NC)NC(=O)CC1CCC(NC(C2CC2Cl)=O)C1 N1(C(C(C)OCCC=C)=O)CCC(CC)(NC(c2cnc(O)nc2O)=O)CC1 N1(C(C(C)NC(=O)NC)=O)CC2(CC(NC(=O)CCC(C)C)c3nccn32)C1 C#Cc1ccc(C(=O)NC2CC2)c(F)c1.N12CCCCC1CCNC(=O)CC2=O N1(CC(=O)OCc2ccsc2)CCCCC1C(C1CCC1)O C1(CC)CN(C(=O)Cc2cccc(F)c2O)CCN1C(=O)Cc1cnc(C)[nH]1 CC1CN(C(C2CC(O)CN2C)=O)CC1CNC(C1SCCS1)=O C1(CC(=O)NC)CN(C(c2ccon2)=O)CCN1C(c1ccnn1CC(C)C)=O n1(CCCCNc2c(OC)cc(F)c(Br)c2)c(C)nc2ccccc12 C(=O)(C(C(C)CC)N1CCC(=C)CC1)NCCCC c1(NC(C(C2CC2)NC(C(C)OCC#C)=O)=O)cccc(CO)c1C c1(CSc2nnc(SCC34OC(C)(C)C(C3)C4)o2)nc2ccccc2[nH]1 c1(C(=O)NCC(CNC(c2cc(C)c(O)cc2)=O)F)coc2c1C(=O)CCC2 C1(C(N(C)CCNC(c2csnn2)=O)=O)OCC2CCCC12 c1(C(N2CCC(C)(NC(C3CCCS3)=O)CC2)=O)c(Br)ccc2ccccc12 c1(C(N(CCCNC(C(C)SC)=O)C(C)C)=O)ccc(Br)o1.C1C(=O)N1 c1(C(=O)NC(CNC(CC2C(C)CCCC2)=O)C)ncnc2ccsc12 c1(C(C(C)(C)NC(=O)NCc2c(OC)nsc2)O)ccc(F)cc1C N1(C(CNS(CC)(=O)=O)=O)CCCC(C2CCN(C(c3cc(C)nn3C)=O)C2)C1 c1(CNc2cc(C(N3CCCC(Br)C3)=O)ncc2)cccc2ccnn12 N1(C(COCCCC)=O)CCC(C2CC2)(CNC(=O)C(c2ccccc2Cl)O)C1 c1(C(=O)NCC2N(C(C(CSC)(C)C)=O)CCC2)ccc(O)nc1Cl n1(CC)ncc(C(=O)N(C(C)CN(C)C(c2ccccn2)=O)C)c1Br c1(C(N2C(CNC(C(CC=CC)C)=O)CC(F)(F)C2)=O)ccc2nnnn2c1 N1(C(CCOCCCOC)=O)CC(O)CC1CNC(c1ccncc1OC)=O CCCCCCCCCC(=O)N(C)CC1CCN(C(c2cnn(C)c2F)=O)C1 C1(C(=O)NC2C(CNC(CCCOC)=O)C2)CC2C(C1)C2(F)F N1(C(c2ncc(OC)cc2F)=O)CCC2(NC(=O)C=C(C)C(F)F)CCCCC12 N1(C(CC(CC)CN(C)C)=O)CCOCC12COCCN(C(=O)CNC=O)C2 C1(CNC(N(C)CC2CCCCC2)=O)CCCC1(C)C C1(O)(CN(C(=O)CCCNS(C)(=O)=O)C)CN(C(=O)CCc2cn[nH]c2)C1 C(CCC)(CCCNC(=O)CNC(c1ccccn1)=O)NC(c1c[nH]c(=NC)s1)=O CC(C)CCCCC(=O)NCCCC(=O)Nc1ccsc1C c1(C(=O)OCC(c2ccc(C(=O)OC)s2)=O)ccc(S(N)(=O)=O)c(Cl)c1 C(C(=O)N=c1ccn(CC(N)=O)[nH]1)=CCNC1CC(C(C)C)OCC1 C12(CNC(=O)CC3CCSCC3)CCCCC1N(C(C1(CO)CCCO1)=O)CC2 C12(CC(=O)NCC3CCN(C(CCC4N(C)CCC4)=O)CC3)CCC(CC1)OC2 N1(C(CCN(C(CCC#CC)=O)CC2CC2)=O)CC(C)SC(C)C1 C(=O)(C(CNC(=O)C(C)n1ccnc1)(CC)CC)N(CCCC(=O)OC)C N1(C(C2CN(C(C)C)C2)=O)CC2(C)CN(C(C3CCCCC3(F)F)=O)CC2(C)C1 CC(=O)CC(C)(C)CC(=O)NCC1CCCCC1NC(C1CCCC(F)C1)=O c1(C(C(=O)NCCC(=O)N(C2CCCC2)C)F)ccc(F)c(Cl)c1 N1(C(C#CC2(CC)COC2)=O)CC2CN(C(C3CCS3(=O)=O)=O)CC(C1)O2 C1(CNC(c2csc(-c3ccccn3)n2)=O)CCN(Cc2cccnc2)CC1(F)F C(c1ccc(Cl)cc1F)=CC(=O)NC1CC(NC(C2(COC)CCCC2)=O)C1 c1(C(=O)NCCN(C(=O)C=CC(F)(F)F)CC)cnnc(O)c1 c1(-c2cn(CC3C=C(C)CS3)nn2)cccc(Br)c1.C12CC(O)(C1)CN2 CN1CCN(C(C2CCCCC2)C(=O)NCCc2ccc(OC(F)(F)F)cc2)CC1 Cc1ccc(C(=O)NCCCOCCCNC(=O)CC2CCCO2)cn1 Cc1cc(O)nc(C)c1C(N1CC2CN(C(=O)CCNC(N)=O)CC2C1)=O C(CCCCC(=O)c1nccn1C1C(=O)NCCCN1)OC c1(NC(C)(CNC(=O)C=CCF)Cn2cccn2)ncnc2cc(Br)ccc12 N1(C(C(C)N2CCC2)=O)CC2CN(C(c3cc(N)nc(Cl)c3)=O)CC2C1 O=S(=O)(c1cccc(C(F)F)c1)NCCC1CC2(CCC2)CO1 C1(NC(COC(C)(C)CNC(c2ccc(C#N)[nH]2)=O)=O)CCCC1N=[N+]=[N-] C1(C(=O)NC2(CC(N)=O)CCC2)(COC)C=CCN1C(C1CCC(=O)NC1)=O c1(C(=O)NC2CC(=O)N(C3CCCC3)C2)ccc(Br)nc1Cl CC1(C)CC(C(=O)NC2CCCSC2)CN(C(c2cc[nH]n2)=O)C1 CCC(C)(C)C(O)C(=O)N1CCOCC1CNC(=O)CC1(O)CC1 C1(C(N)=O)CN(C(=O)CN2CCC(OC(C3CCCCO3)=O)CC2)CCC1(F)F Cc1[nH]c2ccccc2c1C(N1CCC(C)(C(=O)NCCC(C)(C)O)C1)=O NS(=O)(=O)CCC(=O)NCc1cc(O)nc(CNC(C2C3CCC(=O)C23)=O)n1 c1(CC(=O)NC(CCNC(CCCC(=O)NCC)=O)(C)C)ccc(C)c(F)c1F C(=O)(CCS(N)(=O)=O)N1CC(C)(NC(=O)CC2CCCC3CC23)C1 C(C#CC(=O)NOCC=CCl)NC(C(C)(C)O)=O c1(-c2nc(COCC)nn2CC2CCC2)sc2nc(C)nc(N)c2c1C c1(N(C)C)ncccc1NC(C1CCCN(C(=O)C(C2CC2)C2CC2)C1)=O c1(CC)ccc(C(N2CCOC(C)(c3nn[nH]n3)C2)=O)c(Br)c1 N1(C(C(c2ccccc2)SC)=O)CCOCC(C(=O)NCCCC(F)F)C1 c1(NC(CNC(=O)NCCCC)=O)nc2ccc(S(C)(=O)=O)cc2s1 c1(C(N2C(C(C)NC(c3ccc(C)cc3)=O)CCC2)=O)cc2occc2s1 c1(OC)cnc(C(=O)NC2C=CCN(C(c3csc(C4CC4)n3)=O)C2)cn1 Cc1nc(=NC(=O)N2CCC3(CC2)N=N3)n(-c2cccnc2)[nH]1 c1(NC(CNCCC)=O)ccc2c(cnn2CC2CC2)c1 C1(CC(=O)NC(COCC)C(=O)NCC2CC(C)(C)C2)CCCC(=O)N1 c1(CNC2(c3nnnn3C)CC(COCCOC)C2)cc(C)c(Br)cc1C CC(C)C(C(=O)OC(C)(C)C)N1CCN(C(=O)NC2(C)CC(N(C)C)C2(C)C)CC1 c1(COC)ccc(CNC(c2nc(C(C)C)ns2)c2nnnn2C(C)(C)CC)o1 N1(C(c2cnc(C(C)O)s2)=O)CCC2CCN(NC(c3nnc(C)s3)=O)CC2C1 C1(NC(COCCOC)=O)CN(C(c2cccc(Cl)c2C)=O)CC2CC12 c1(C(=O)NC23CCN(C(COC)=O)CC2C3)ccn2cnnc2c1 C(=O)(C1Cc2ccc(F)cc21)NCCN(C(c1c(C)cno1)=O)CC1CC1 CCCC(C)CC(=O)N1CCOCC1(C)c1cn(Cc2cnn(C)c2)nn1.CC Cn1ncc2c(C(=O)O)ccnc12.C12C(CC1O)NC(=O)c1cnn2c1 C(CC(=O)N1CC(n2cc(CC(C)C)nn2)CO1)N(CCCCCC)C C(=O)(C1=C(Cl)CC1)N(C)CCCOCCCN(C(C(C)OC1CCOC1)=O)C C12(C(=O)OC)CCCN(CC3COCCN(C)C3)CC1C2 N1(CCc2c(C)nn(C)c2)CCN(C)CCC1C(C)C c1(OC)ccc(C(=O)NC2CCCCC2NC(=O)COCC2CCCCC2)cn1 C1(C2CCN(C)CC2)(C(=O)NCC2C(NC(c3ccc(OC)nn3)=O)C2)CC1 C1(CC)CN(C(c2cccc(=S)n2O)=O)CCN1C(c1cccc(Cl)c1)=O C12(CNC(c3c(OC)nsc3)=O)CCCCC1N(C(c1ccc(CO)o1)=O)CC2 c1(NC(c2nc(C)on2)(C)C)cc(Oc2ccccc2)ccc1[N+](=O)[O-] c1(CC(=O)N(C)CC2(CNC(C(C)=CC)=O)CC2)c(C)nn(C)c1C CC1(C(N2CC3C(NC(C4CCCCO4)=O)C3C2)=O)CCC12CCC2 c1(C(N2CC(NC(c3c(COC)ccs3)=O)C(OC)C2)=O)cc(OC)ncc1F N1(C(C=C(C)c2ccco2)=O)CCN(C(c2csc(C(F)F)c2)=O)C(CF)C1 c1(C(C)C)nocc1C(=O)N(CC(C)O)CCNC(=O)CCNC(=O)C(C)(C)C C(C(C)(C)C)OCC(=O)NCC1(CN(C)C(C2(F)CC2)=O)CC1 Cc1cc(C(=O)N(CCCCCC(=O)NCCC2CC(C)(C)CO2)C)cnc1C c1(NC(C2N(C(=O)C(O)CC(C)C)CCC(CC)C2)=O)cnn2c1CCCC2 N1(C(C)=O)CS(=O)(=O)CC1C(=O)N(C)CCNC(c1c(C)nn(C(C)C)c1C)=O C(=O)(C1=C(Cl)CCCC1)NC(CNC(c1cc(C)c(C)s1)=O)C(C)(C)C N1(C(CC(C=C)CCC)=O)CCC(C2CC(NC(=O)Cc3ccon3)C2)CC1 C1(NC(=O)C=CC2CCOCC2)CCC12CCCN(C(c1coc(CO)c1)=O)C2 c1(OC)cncnc1C(=O)NCC1(NC(=O)C(C)c2ccco2)CC1 CC1C=C(C(=O)N2CCC(C(C)(C)NC(=O)Cn3nnc(=O)[nH]3)C2)CC1 c1(C(=O)NCC(C)(CO)NC(C2C(CC)C2)=O)nccc2cc[nH]c12 c1(OC)ccc(CCC(=O)NCCn2cnc(C)c2C)cc1N C(=O)(CC(C(C)C)NC(c1ccc(CO)cn1)=O)N1CCC(C#C)C1 c1(C(=O)NC(C2(O)CCN(C(C(CC=C)(F)F)=O)CC2)C)ncnc2c1CCC2 Cc1ccc(N)cc1C(N1CCN(C(c2ccc(=O)n(C)c2)=O)C(CCO)C1)=O CCCC(C(=O)OC)NC(C1CCCN1C(=O)Nc1ccc(CC)cc1)=O N1(C(C(C)OCc2ccccc2)=O)CCC2(CCN(C(=O)CC(F)(F)F)C2)C1 c1(CC)nc(C)n(C)c1C(=O)NCC1CC(OC)CN1C(c1cc(CC)[nH]n1)=O CC1CC(NC(C2(N(C)C)CC2)=O)CCN1C(c1cccc(CN=[N+]=[N-])c1)=O C(=O)(C1Cc2ccccc21)NCC(C)CNC(=O)Cn1cnnc1 CC1(C)C(=O)CC1NC1CCN(C(C2(COc3ncccn3)CC2)=O)C1 N1(C(C(N2CCOC2=O)C)=O)CCCCC1CCCC1CCCN1C(=O)C1CC1 C1(NC(c2c(C)nn(C)c2Cl)=O)CN(C(c2ccn(C)c2)=O)CC2CCCC12 c1(C(=O)NCC2CC(F)CN2C(c2nocc2Cl)=O)ncnc2[nH]cnc12 CCC(CS(C)(=O)=O)NC(c1cccn1C)c1nnnn1C1CCCC1.C1CN1 c1(C(CNC(C2(C)CC(C)C2)=O)NC(C(CC)NC(N)=O)=O)ccccc1F N1(C(c2c(C)coc2C)=O)CC(C)(C)CC1CC(=O)NC(c1c(C)n[nH]c1C)C N1(C(c2c(CC)nccc2)=O)CCC(C2CCCN(C(=O)CC=C(C)C)C2)C1 Cc1cc(C(C23CC2CCN3C(=O)OC2CC(C)C2)=O)cc(C)c1.C(C)(C)(C)O c1(C(=O)NCCCCCN(C(C2(OCC)CCC2)=O)C)cc(C)nnc1O Cc1ccc(C)c(C(=O)NCCC2CCN(C(C3CC(=C4CC4)C3)=O)CC2)c1N c1(C(N2CCC(C(C)NC(=O)Cc3cocn3)C2)=O)cnccc1Cl C12(CNC(COCCNC(c3ccc(C(C)=O)o3)=O)=O)COC(C1)C(O)C2 C(CC(C)C)(C(=O)NCC1(F)CC(NC(=O)Cc2cccnc2)C1)OC CCCCC(F)(F)C(=O)NCC(F)CNC(=O)CCNC(=O)CO C1(NC(C2(C)CC2(F)F)=O)CCC2(CC1)CN(C(=O)CCc1n[nH]c(=N)s1)C2 C1(NC(c2c(C)ocn2)=O)CC(CNC(c2cc(C(C)(C)C)on2)=O)C1(C)C c1(C2N(CC(=C)C(C)(C)C)CCC2)ccc(F)cc1OC c1(CO)cn(CCC(=O)NC(c2c[nH]c(C(N)=O)c2)=O)nn1.C(CCSCC)N(C)C N1(c2ccnc(C)n2)CCC2(CCC(C(=O)NCCn3cc(CO)nn3)CC2)CC1 c1(CC(=O)NC2C(NC(c3n(CC)ncc3)=O)C2)cc(=O)n(CC(C)C)[nH]1 c1(CNC(C2CCCN2C)=O)cccc(N)n1.Cn1ccc(SCC(=O)OC)n1 CCC(CNC(C1CC1C1CCCCO1)=O)(CC)NC(c1ccc(CSC)o1)=O CCC(C)CC(C)C(=O)NCC1CCC(CN(C)C(c2c(C)ncn2C)=O)CC1 c1(-n2c(C3CC4CC34)ncn2)cc(-n2cnnn2)ccc1F.c1cn[nH]c1 n1(CC(CC(=O)OC)C)c(-c2cccc(SC)c2)csc1=Nc1ccnc(Cl)c1 C1(C(CNC(c2cnc(C)o2)=O)F)CCN(C(=O)CC2C=NN(C)C2=O)CC1 Cc1ccc(NC(C2(OCC(=O)NCC3CCCO3)CC2C)=O)c(F)c1 c1(CC(N2C(CNC(c3c(C)csc3)=O)C=CC2)=O)cc(F)ccc1F N1(C(C2(F)CCOC2)=O)CCC2(CC1)CC(N(CCO)Cc1ccccn1)CO2 C1(NC(c2ccc(OCC)c(Cl)c2)=O)C2CCN(C(=O)CCC(C)=O)CCC12 C1(NC(c2cnc(OC)s2)=O)COCCN(C(=O)C(N2CCC(C)CC2)=O)C1 Cc1ccc(F)cc1C(=O)NCC1CC(NC(C2(C)CCOC2C)=O)C1 CC(C)CC(C(=O)NC(C)C(C)(C)C(=O)NC1CC(n2cncn2)C1)C(N)=O c1(C(C)C)ncc(C(=O)NCC2(NC(=O)CCCN(C)C)CCCC2)n1C N1(C(C)=O)CCCC(CC(N2CC(N(C(=O)CCn3ccnn3)C)C2)=O)C1.C1CC1 C(=O)(C1COc2ccccc21)NC1C(NC(Cc2nnc(C)s2)=O)CCC1 c1(C(=O)NC(CNC(C=CC=CC)=O)CC(F)(F)F)cc(S(N)(=O)=O)co1 c1(C(N2CCC(NC(C3N(CCC)CCC3)=O)CC2C)=O)cc2c(ccn2C)[nH]1 c1(NC(C(N(C(=O)CC2CCCSC2)C)C2CC2)=O)ccc2ccoc2c1 N1(C(C(CC=CC)C)=O)CC(OC)CC(NC(=O)CN2CCCC2)C1 c1(C(=O)NC2CCCC(NC(c3sc(CC)c(C)c3)=O)C2)cnc2[nH]cncc1-2 N1(C(c2c(C)cc(C)nc2)=O)CCCN(C(=O)CCc2cccnc2C)C(C)C1 C(=O)(C1=NOC(C)(C)C1)N(CC(C)NC(C12COCC(C1)C2)=O)C N1(C(C(C(C)C)O)=O)CC2CC(NC(=O)CC3CCC(C)C(C)C3)CC1C2 c1(SCC(N2CC(CC(=O)N(C(C)C(N)=O)C)C2)=O)ccc(Cl)cc1Cl c1(C(=O)NC2C3(CN(C(C4C(CC)OCC4)=O)C3)CC2)cnc2ccccc2n1 N1(C(CC(=O)NCC)=O)CCN(C(=O)C(S(C)(=O)=O)C2CC2)CC1CC c1(CC(=O)NCCN(C(C)C)C(c2cscn2)=O)cn2cc(F)ccc2n1 O=C(C#CC1CCOCC1)NC1CCC(CCNC(=O)C(C2CCOCC2)F)C1 C1(C(=O)NCCCNC(c2cc(C)n(C3CCOCC3)n2)=O)CN2CCN1CC2 C1(CN2CCC(OC3C(C)CCCC3)C2)CC2CCC1CC2 n1(CC)cnc(C(=O)NCCCCNC(=O)C(C)C2CCOC2)n1 N1(C(C=C(CC)c2cccs2)=O)CCCCC(CNC(=O)CCC2CC2)C1 C1(C(N2C(C(C)NC(c3c(C)n[nH]c3)=O)CCC2)=O)CCCN(S(N)(=O)=O)C1 C1(C)(C(=O)NCC2(CCC)CCC2)CCN(C(=O)NCc2ncc[nH]2)C1 CCC(CCC(=O)N1CC(C)C1(C)C)NC(=O)CCCCOCC S(=O)(=O)(C1CCOCC1)N(C1CCNCC12CC2)C(c1cc(OC)ncc1)=O c1(C(=O)NCC(=C)CCNC(=O)C(c2ccccc2)C)c(C)nn2c1OCCC2 c1(C(=O)NCCOCCNC(c2cc(C)on2)=O)nn(C)c2c1CSCC2 C(=O)(CC(C)(C)CC(F)F)NCC(CNC(C1(C)ON=C(C)C1)=O)C(F)(F)F c1(C(N2CC(C(N)=O)(CNC(COC(CC)C)=O)C2)=O)cc(C)c(C)[nH]1 N1(CC)CCCN(C(=O)C(CNC(c2cc(C(N)=O)c[nH]2)=O)N(C)C)CC1=O C1(CNC(Cn2c(C)ccn2)=O)CN(C(=O)CC(C)C2CCCC2)CCO1 N1(C(C2CC(C)(F)C2)=O)CCC(NC(=O)CCN2CCCCC2)C12CCC2 C1(NC(CCNS(CC)(=O)=O)=O)CCCCC1C(=O)N(C)Cc1occc1C C1(CNC(C=C(C)C)=O)CCN(C(=O)CC2CSC2)CC1C c1(COC(CC(CN(C)C)C(F)F)=O)nc2cccc(C(F)(F)F)c2[nH]1 C1(C(=O)NC(CCOC)CNC(=O)CN2CC(C)(C)C2)CSCC(=O)N1 C(=O)(C#CC1CCCCC1)N1CC(CC)N(C(c2cccc(CCO)c2)=O)CC1 N1(C(CCc2c(C)cccc2)=O)CCCN(C2CC2)C(c2cn[nH]c2)C1 C1(CN(C(C(COCC)O)=O)CC)CCN(C(=O)C2=CCSC2)CC1 C1(C(=O)Nc2ccsn2)C=CCN(C(=O)COC2CCCOC2)C1 c1(C(C)C)cccc(C(N2CCCC(CN(C(=O)C(C)c3ncco3)C)C2)=O)c1 c1(CN(C(C=CC(CC)C)=O)C)nc(C)ns1.C1C(=O)N1CC c1(C(=O)NC23CC(C(=O)NC(c4cn(C)nn4)C)(C2)C3)scc(C)c1C C1(NC(=O)CC2(O)CCOCC2)CCC2(CCC2)CC1.C12(CC=CC1)C(=O)NC2 C1(C(=O)NCCOCCOC)CN(C(=O)CC2CCCC3CC23)CC1(C)C c1([SH](CCC(c2nn[nH]n2)C(=O)CC2CCCCO2)C)cnn2c1CCC2 CS(=O)(=O)C(Cc1ccccc1)C(=O)NC(CNC(c1cnc(O)s1)=O)CO C1(CC(=O)N(CCCC)CCCO)CC(F)CN1C(C12CSCC1C2)=O c1(C(N2CCC(OCCNC(C(C)SC)=O)C2)=O)cc(C)c(Cl)s1 S(=O)(=O)(c1cc(Br)c(F)cc1Cl)N(C)Cc1c(Br)cnn1C c1(C(=O)NC2(CC)CCCN(C(=O)C=C(C)C)C2)cc(N)c(Cl)c(O)c1 c1(NCCC2(OC)CN(C(c3cnnn3C)=O)C2)ncc(Br)cc1C#N c1(C(N2CC3C(CNC(c4n(C)nc(C)c4Cl)=O)C3C2)=O)cnc2c[nH]nc2c1 c1(C2CC(CC)C2)cn(CC(C)(C)CNC(=O)C(C)OC(=O)CO)nn1 C#Cc1cccc(C(=O)N(C2CCCCN(C(=O)C(C)SCC)C2)C)c1F c1(C(=O)NCCCCc2cnc[nH]2)cnc2sccn12.C12(CC1)C(=O)NC2 C1(C(=O)NCCNC(c2c(C(C)C)nns2)=O)CS(=O)(=O)CC12CC2 c1(C(=O)NCC2CC(NC(CC3(COC)CCCC3)=O)C2)ccn2ncnc2c1 C(=O)(C(C)(C)c1cn(C(C)CSCCO)nn1)NCC(C)C1CCC1 C1(C(N2CC(C(C)NC(c3c(C)nc(CC)s3)=O)C2)=O)COC2COCC12 CC(C)(CNC(c1ccoc1)=O)CC(=O)NC1CC1(C)C CC1CC=C(C(=O)NC2COCCN(C(c3cc(CN(C)C)c[nH]3)=O)C2)CC1 C1(OC)CC(NC(c2cc(C)cc(Br)c2)=O)CN(C(=O)C(C)(C)C2CC2)C1 CC1CC(CNC(=O)C(O)Cc2cnc[nH]2)CN(C(C2(C)CCCN(C)C2)=O)C1 c1(C(=O)NCCC(C)(C)NC(c2cn(C3CC3)cn2)=O)csc(C#N)c1 C(=O)(CC(C)(C)C)N(C12CC(F)(C1)C2)CCCOC(C(C1CCCCCC1)C)=O c1(C(=O)NCC2(C)N(C(c3cnc(CCC)s3)=O)CCC2)c(F)ccc(N)c1F C1(C(=O)NCC(=O)NCCC)CCN(C(C2CCC2OC)=O)C12CCC2 C1(COC)CN(C(c2cccc(F)c2Cl)=O)CCN1C(c1cscc1Cl)=O C(CCCCC(=O)NCC(C)CNC(C1(S(N)(=O)=O)CC1)=O)OCC C12(C(=O)N)CCC(OC)C1C2.C1(C)(C(=O)OCC)CN(C2C(C(=O)NC)C2)C1 c1(COC(C2CC2NC(C)(C)C)=O)cc(CO)c(C(=O)NC2CC3OCCC23)[nH]1 C1(C(=O)NCC(C)OCC=C)CN(C(=O)CN2CCNC(=O)C2)CC1C1CC1 N1(C(C2N(C(C)=O)CC=C2)=O)CCC2(CC1)CC2NC(=O)CN(C)C(N)=O C12CCN(CC1C)C2=O.c1(NC(c2cc(C(=O)OC)no2)=O)cn(C)nc1SC c1(CN(C(=O)C(CO)NC(C2CC(C)(F)C2)=O)C)cnn(C)c1O C1(NC(C(CCF)NC(=O)CN2CC3CC3C2)=O)CCOC12CCCC2 N1(C(CC2CCN(C)C2)=O)CCC2CN(C(=O)C(N)=O)CC2C1 C1(NC(c2ccoc2Cl)=O)C2CN(C(C3CC(CCO)C3)=O)CC12 C1(NCCC2(CS(C)(=O)=O)CC2)CN(CCF)CCO1 N1(C(C2C(=C)C2)=O)CCC2CCC(NC(=O)C(C)N(C)C)C1C2 CC1(C)C(NC(c2ccc(C3CC3)o2)=O)CC1C(N1CCC(CCF)CC1)=O C1(CC(=O)NCC(C(C)C)NC(=O)CN2CCCCCC2)CC2(CCC2)CCO1 c1(NC(C(=O)NC(CC)C(N)=O)=O)cc2c(cc1Cc1ccccn1)OCCO2 N1(C(c2c[nH]c(=NCC)s2)=O)CC2CN(C(=O)CN(C)C)CC2C1 c1(C(N(C(CNC(CCCC(=O)OC)=O)C)C)=O)cn(C)c2ccc(F)cc12 N1(C(CCC#C)=O)CC2CC(NC(c3sc(CCOCC)nc3C)=O)CC1C2 C1(C(=O)NC(C(N2CCN(C(=O)NC)CC2)=O)CCF)Cc2nccn2C1 n1(CC)nc(C)c(CC(N2CCC(O)(C(C)NC(c3cnc[nH]3)=O)CC2)=O)c1C c1(CNC(C2(CC)CCN(C(c3coc(C(N)=O)c3)=O)C2)=O)c(C)nn(C)c1C c1(C(=O)NCC(CC)NC(c2cnn(C)c2Cl)=O)c(C)sc2ccc(F)cc12 C1(NC(c2ncnc(C)c2C)=O)CN(C(C2CCC(C)CC2)=O)C2(CCOC2)C1 N1(CC(=O)NC2CC(NC(CC(=O)NCC#C)=O)C2)CCSC2CCCCC12 CN1CCC2CN(C(c3ccc(-c4cc[nH]n4)s3)=O)CC2C1 c1(C(=O)NCCCC(C)(C)NC(C(C)SC(C)C)=O)ccc(=N)[nH]c1Cl c1(C(N2C(C)CN(c3ccnc4ccnn34)CC2)=O)cccc2c1nnn2C c1(C(=O)OCC2N(C)C(=O)C2)c(C#N)sc2ncccc12 c1(C(N2CCN(C(C(C(C)C)(C)C)=O)CC2C)=O)cccc(S(=O)(=O)C(F)F)c1 N1(C(C(C(C)C)OC)=O)CCC2(CC1)CN(C(=O)CCCCCSC)C2C(C)C CC#CCCCC(=O)N1CCOC(CNC(=O)C(C)Oc2cc(F)cc(F)c2)C1 C(CN=C(NCCOc1ccc(Cl)c(F)c1)NCC1CCN(C)C1(F)F)OC Cc1nc2c(s1)CN(C(=O)NC(c1cc(F)c(F)c(F)c1)C)CC2 c1(C(=O)NCC(CNC(C(C(C)C)SC)=O)(C)O)cc(N)c(Cl)cc1C C1(C(=O)NCCCNC(=O)C=Cc2ccco2)CCCCN1C(C1CCO1)=O c1(C(=O)NC2CC(CNC(CNC(N)=O)=O)C(O)C2)cc(C(C)C)nc(O)c1 c1(OCC(N2CC(F)(CNC(C(C(C)O)(F)F)=O)C2)=O)ccc2c(c1)OCCO2 C1(C(N2CCC(C(C)NC(=O)C=Cc3ncc[nH]3)CC2)=O)CCCCC1(C)C c1(C(=O)NC(C2CCCCC2)CNC(CCOC)=O)n[nH]c2ccc(Br)cc12 c1(C(=O)NCC(C)(CNC(=O)C(C)Cn2ccnc2)OC)c(C)ccnc1O c1(C(=O)NC(C(CO)NC(CCCOC(C)=O)=O)C)cnnc(C2CC2)c1 C#CC1(C(=O)Nc2ccc(O)c(F)c2)CCN(C(=O)CC2(CSC)CC2)C1 C(=O)(C1=Cc2ccccc2C1)NC(c1cc(OC)c(OC)cc1)C.C1C(=O)O1 c1(C(=O)NC2C3N(C(COCCC)=O)CC(CC3)C2)ccc2c(c1)C(=O)CCN2 c1(CC)ccc(O)c(C(N2CC3CC(C2)N3C(=O)C(C)O)=O)c1 C(=O)(CCCCC(F)F)NC(C1CCN(C(CCC(=C)Br)=O)C1)C Cc1c(C(=O)NC2CN(C(=O)C=Cc3cocn3)CC2C)cc(F)cc1Br C#Cc1ccc(CCC(=O)NCC2(C)CN(C(=O)CCC3CCC3)CCO2)cc1 C1(NC(C2(C)CCCC2)=O)CC2CCC(C1)N2C(C1(F)CCCC1)=O C1(NCCC2CCOC2)C=CC(CC(=O)N(C(C2C(C(N)=O)C2)=O)C2CC2)C1 C(=O)(C1CNC(=O)c2ccnn21)NCCN(C(c1cc(C)c(C)[nH]1)=O)C CC1CCC(CC(N2CC(CC(=O)N(CC(F)Cl)C)C(C)C2)=O)OC1 c1(C(=O)NCC2C(CC(=O)NC(CCOC)C)C2)ncncc1Cl c1(C(=O)NC(C2(O)CN(C(C3CC(OC)C3)=O)C2)C)cc2c(C)ccc(F)c2[nH]1 Cc1n[nH]cc1C(c1nnnn1C1(C)CC1)NCCC1CCOC1 C1(CC=C)CCCN(C(=O)CCCC2(NC(C3(F)CC=CCC3)=O)CCC2)C1 O=C(CS(=O)(=O)CCCc1ccccc1)NC1C(C2CC2)C1(F)F C1(NC(CC(=O)NC)=O)CC1C1CCN(C(c2ccc(OC)cc2F)=O)CC1 c1(CN2C3CN(C(CCC4CCC(C)CC4)=O)CC32)c(Cl)ccnc1Br N1(C(c2ncc(P(C)(C)=O)cn2)=O)Cc2c(O)n[nH]c2C(F)(F)C1 Cc1ccc(Br)c2[nH]c(C(=O)NC3COC4(C3)CN(C(C3CCO3)=O)C4)cc12 C1(CC)(CC)CCCN(C(=O)C(C)(C)CNC(=O)C(CO)OC)C1 C(CCSC)(C(=O)NCC1(OCC)CC1)NC(C=CCCC)=O CCCC(CC)CCC(=O)NC1CN(C(c2ccc(F)c(F)c2N)=O)CC1CC c1(C(=O)NCCCN(C(CC(=O)OC)=O)C2CC2)ccc(C2=CCCC2)cc1 c1(C(=O)NC2(C)CC(NC(c3cc(CCC)[nH]n3)=O)C2)ccc(C)c(C)c1N N1(C(C2C(C)=CC(Cl)=CC2)=O)CCC(NC(c2cc(=N)[nH]c(=N)[nH]2)=O)CC1C c1(CN(C2CC(=O)N(C3CC3)C2)CC#C)cccc(Cl)c1Cl Cc1nc(C)c(F)c(=NCC2CC(C)N(C(c3ccc(CO)c(F)c3)=O)C2)[nH]1 C(=O)(CCCCCN=C(NC1CCC1)NC(C1COC1)C)OC(C)C c1(Cc2nc(C3ON=C(CC)C3)on2)ccc2c(ccn2C)c1 C(=O)(C(C(C)C)NS(=O)(=O)C(F)F)N1CC(CCO)(NC(C=CC)=O)C1 C#Cc1cccc(C(=O)NC2(CC(N3CCC(C)C3(C)C)=O)CCC2)c1 C(=O)(C(O)Cc1cnn(C)c1)NCC#CCNC(C(C)NC(=O)OCC)=O c1(OC)cccc(OC)c1CC(N1CCCC(NC(c2ncoc2CN)=O)C1)=O N1(C(C2(C)CCCS2)=O)CCC(NCc2c(C(F)(F)F)nc(C)[nH]2)C(CO)CC1 Cc1cc(N2CC3CN(C(c4nc(Cl)sc4C)=O)CC3C2)c(C#N)cc1[N+](=O)[O-] Clc1cnc(C(c2nnnn2C2CC2)NCc2cnc(-c3ccccc3)[nH]2)s1 CCC(O)C(=O)N1CC(OCCNC(=O)Cn2cc(Br)nn2)C1 C(C1CN(C(c2c(C#N)ncn2C)=O)CC1C(N1CC=CCC1)=O)=CC c1(C(N2CCCCC(CNC(c3c(C)scn3)=O)C2)=O)csc2c1CCCC2 CS(=O)c1ccc(C(=O)NC2CCC2NC(c2ccncc2Br)=O)cc1 c12nc(nn1C1CCC1)-c1cccc(c1)C2.CC(C)(C(F)F)N1CCCC1 Cn1cc([N+](=O)[O-])c(C(=O)NC2CCC(F)(CNC(=O)C(F)CC3CCC3)C2)n1 N1(C(CC2C(C)(C)OCC2)=O)CC(NC(c2cscc2Cl)=O)CC1(C)C N1(CC(CC)C)CCC(NC(c2cc3c(Cl)cncc3s2)=O)CC(C)(C)C1 Cc1ccc(CC(=O)NCCC2(C(=O)NC3CCCSC3)CCC2)o1 C1(NC(C(C)NS(CC)(=O)=O)=O)(CO)CCCN(C(=O)CNS(=O)(=O)N(C)C)C1 N1(C(c2c(C(C)C)noc2)=O)CCC(C)N(C(c2cc(N)cc(N)c2)=O)CC1 c1(C(N2C(C(=O)NCC3CCCC(OC)C3)CCC2)=O)cc(C)cc(O)c1 CCC(CCN)C(=O)NCC(c1cnc[nH]1)C c1(C(=O)NCCNC(C(C)(C)C)c2nnnn2C2CCOCC2)cc(F)c(F)cc1 C1(NC(C(CNC(c2cc(COC)[nH]n2)=O)N(C)C)=O)CCCC(OC)C1 c1(NC(=O)Cc2noc(Cc3ccc(F)cc3)n2)cccc2nc(O)ccc12 N1(C(c2c(C)nc(CC)s2)=O)CCCC2(CCN(C(=O)C(F)CC(C)C)C2)C1 c1(C(N2CCC(NC(c3cccc4cncn34)=O)C2)=O)ccc([N+](=O)[O-])cc1Cl c1(C(N(CCCNC(C(C=CC)O)=O)CC)=O)c(C)nsc1N CCCC(C)(O)C(=O)NCC1(F)CCC(NC(c2cc(O)nc(C3CC3)n2)=O)C1 c1(C(=O)NC2CN(C(C3(F)C(C)C3)=O)C2)cccc2cc(O)ccc12 C(=O)(C#CC1CCC(=O)CC1)C(=O)C1=CCCC(C)(C)C1.CC1CC(C=O)CCN1 CC1(C)CC(C(=O)NC2C3CC4C2C4C3C(=O)NC2CCOC2=O)CCO1 N1(C(C(=O)NCCN(C(=O)C=C2CC2)CC)C)C(=O)c2ccccc2C1=O c1(CC)cc([N+](=O)[O-])ccc1C(=O)NC(C)CN(C)C(C1(F)CCCOC1)=O C#CCC(C)(C(=O)NC1COC2(CCC2)C1)NC(c1ccn(C)c1C)=O C(=O)(CCN=[N+]=[N-])NCC1CC(O)(CNC(C(C)NC=O)=O)C1 Nc1cc2c(cc1C(=O)N(CCNC(=O)CCc1ccc(Cl)s1)C1CC1)CCC2 C(=O)(C1=CCS(=O)(=O)C1)NC1CCCC(NC(CCS(N)(=O)=O)=O)C1 N#Cc1nc[nH]c1C(N1CCCCC1C1CCN(C(c2csc(S)n2)=O)CC1)=O c1(C(N2C(CNC(CC(CC)SC)=O)CC2)=O)ccc(OC(C)C)cc1F Cc1c(C(=O)NC2CCCN(C(c3cn(C4CCC4)nn3)=O)C2)nnn1C(C)C CC1(C)C2CC(C(=O)NC3COCC3NC(C3CCN(CC(F)F)CC3)=O)CC12 c1(C2CCN(C(c3c(Br)noc3)c3ccccc3)CC2)nc2ccc(F)cc2s1 c1(C(C(=O)NCC(C)C)N(CCCc2ccco2)C)sc(=O)n(C)c1Cl C1(C(N(C2CCCCC2)CCNC(C2C(F)(F)C23CC3)=O)=O)CC1C1CCC1 C(C)(CCCCNC(c1cc(CO)[nH]n1)=O)NC(=O)NCC(=O)N.C(C(C)(C)C)OC C1(CC(=O)NCCC2CCCN2C(C2COCCO2)=O)CCCC2(CCC2)O1 c1(N(C)C)ccc(C(N2CCC(C3CCCN3C(=O)C=CC3CCC3)C2)=O)nc1 c1(C(=O)NC2(C3N(C(C=CCC)=O)CCCC3)CC2)cc(COC)cc(F)c1 N1(CC(=O)NCC2CC(O)(CNC(=O)CC3CC3)C2)CCCNS1(=O)=O C(C)(C)(CCC(=O)NCC=CCNC(=O)CCCCc1cnn[nH]1)OC C1(CNC(C(c2cncc(F)c2)C)=O)CN(C(=O)CC(C)(C)C#N)CCCO1 c1(OCC)cc(C(N2CC(CCNC(C3CC3(C)C)=O)C2)=O)[nH]n1 CC12CN(CC3CCCCO3)CC1(C)CN(CCC1CC(F)(F)C1)C2 c1(C(N2CC(C=C)C(NC(=O)Cc3cncnc3)C2)=O)sc([N+](=O)[O-])cc1Cl c1(CC(=O)NC2CCC(=O)NC2)cc(Cl)ccc1Br.c12ccc(cn1)c(=O)n2C1CC1 c1(C(N2CCC(C)N(C(=O)CCC3CC3)CC2)=O)cccc(S(=O)(=O)C2CC2)c1 n1(CC=C)ccnc1C(=O)NC(C)C(C)(C)OC(F)F N1(C(C(N2CCN(CCC3CC3)CC2)=O)=O)CC(CO)CC12CCC2 N1(C(C2N(C(CC(C(=C)C)OCC)=O)CC2)=O)CCN2C(=O)CCC2C1.C(=O)N C1(CC)COCCN(C(c2cccnc2CNC(c2c(CO)noc2C)=O)=O)C1 NC(=O)CCC(=O)N1CCN(C2CCNC2=O)CC1.C(=O)(CCC1CCCO1)N1CCC1 C(=O)(C(C(C)(C)C)C1CCCC1)NC(C1CN(C(=O)CC2CC2(C)C)C1)C C(=O)(C(C)(CO)NC(=O)C(C1CCCCC1)O)N(CCN(CC)CC)C CC(C)C(C)(O)C(=O)N(C1CCN(C(c2ccnnc2)=O)C1)CCCCl N1(C(C2(C)CNC(=O)C2)=O)CCN(C(c2cc(C(F)(F)F)cs2)=O)CC(O)C1 c1(CC(=O)NC2(CF)CCN(C(C(C)OCC=C)=O)C2)noc2ccccc12 C1(C(=O)NCC(CNC(c2cc(C)c(C)s2)=O)CO)CC2CCCC2C1 C1(C(C)C)CN(C(c2cnnn2C)=O)CCN1C(c1ccc(C(=O)N(C)C)[nH]1)=O c1(NC(=O)NCCS(CC)=O)ccc2c(c1)nc(O)n2CC1CC1 C(=O)(CC=C(Cl)Cl)N(CCC(=O)NCCCc1n(C)ncn1)CCO c1(OC2CC(CCn3cc(-c4nccc(OC)c4)nn3)C2)ncc2n1CCCC2 Cc1nc(=NC2(CO)CCCN(C(=O)OC(C)(C)C)C2)[nH]n1C C(=O)(C1=CCC(NC(=O)Cc2cccc(C#N)c2)C1)NC(C)CCCCO CC(CCC(=O)OC(C)(C)C)N=c1[nH]n2cc(C(C)(C)C)nc2s1 N1(C(C(CC)C)=O)CC2(C1)CN(C(=O)CC1CCC(C(F)(F)F)O1)C2 c1(C(N2C(CNC(C(C)CC3CCCO3)=O)CC2)=O)cccc2nsnc12 N1(C(C2C(CC)CCCC2)=O)CC2CN(C(=O)Cc3cccc(C)c3)CC(C1)O2 C(CC(=O)NC(C)CN1CCCC1=O)(C(F)F)NC(C1(CCCC)CCC1)=O C1(N(C(Cc2c(C)cccn2)=O)C)CN(C(=O)CSCCC(C)C)CC12CC2 Cc1cccc(OCc2nc(-c3cncc(C(N)=O)c3)n(-c3cnn(C)c3)n2)c1 CP(C)(=O)c1ccc(C(=O)NCC2CCCC2NC(C2CCCCCC2)=O)o1 C1(NC(C2N(C(C)=O)CCC2)=O)CCN(C(c2cc(Cl)c[nH]2)=O)CC1(C)C c1(C(=O)NC2CCCN(C(c3c(C)ccc(C)n3)=O)C2)cccn2nnnc12 c1(C(N2CCN(C(CNC(=O)OCC)=O)CC2CF)=O)ccc2c(c1)CNC2=O C1(C(=O)NCCN(C(c2c(SC)csc2)=O)Cc2ccccc2)CCN(C)C(=O)C1 C(=O)(C(CO)C(F)(F)F)N1C(C(=O)NCC(CCC)(C)C)CC1C C1(C(N(C2C(C)C2)C)=O)COCCN(C(=O)CCC2CCCCCC2)C1 C=CC1CN(C(=O)COCC)CC1NC(c1ccc(N2CCCCC2)cn1)=O c1(C(N2CCC3C(C2)CN3C(=O)NCCOC)=O)c(F)ccc(Cl)c1F C1(NC(C2(OC)CC2)=O)CCCC1C(=O)NCC1(CC2CC2)CC1 C1(CNC(C(C)NS(CC)(=O)=O)=O)CN(C(=O)Cn2cc(Cl)cn2)CC(C)(C)O1 c1(CNC2C(C(=O)Nc3ccc(C(=O)OC)o3)C2)nc(Cl)ccc1Cl CCC1=NOC(C(=O)NC2CCCCC2CC(=O)NCC2(COC)CCC2)C1 c1(N2CC(O)(CNC(C3CC(N=[N+]=[N-])C3)=O)C2)nc(Cl)nc2sccc12 C1(C(N(C(CN(C(c2c(CC)ocn2)=O)C)C)C)=O)CNC(=O)CC1(C)C C(=O)(C1NCCc2c(C)cccc21)NCC1=C(C)OCCS1 c1(CCC(=O)NCCN(C(C(F)OC)=O)C(C)C)cc(F)cc(F)c1 Cc1cc(=O)cc(CNC(C2(CCNC(c3cc(CO)oc3C)=O)CCC2)=O)[nH]1 N1(C(c2nc(C(C)NC(=O)CC3CCCC3O)oc2)=O)CC2C(C1)C2(C)C C(=O)(CC(C)(C)CN)NCC=C(C)C.C(=O)(C(=O)N(C)C)NCC c1(OC)noc(C)c1C(=O)NCC(C)NC(C1CCCS1)=O C(=O)(CCCCC(F)F)NC(CCNC(C(CC)(C)OC)=O)C Cn1ncc2ccc(NC(=O)N(c3ccccc3)CCC#N)cc12.C1C(=O)N1 C(=O)(CCCS(C)(=O)=O)NCC(C)NC(C=Cc1nc(C)c(C)[nH]1)=O C1(NC(CNS(CCCC)(=O)=O)=O)CCN(C(=O)CC2CC(C)C2)CC1O C1(c2nnnn2C2CCC2)(NC2(CC)COC2)CC2CC(OC)CC12 c1(NC(C2N(S(CCCC)(=O)=O)CCC2O)=O)cc(F)c(Br)cc1[N+](=O)[O-] C(C(CC(=O)N1CCC(OCCF)C1)NC(c1cc(C(C)=O)on1)=O)OC N1(C(C(=Cc2cccnc2)C)=O)CCC(C(=O)NC(c2ccco2)C)C(C)(C)C1 c1(SCC(=O)NCC2N(C(CCC=C)=O)CC(O)C2)ccc(C#N)cc1 Cc1cc(Cl)ccc1OCC(=O)NCC(CO)NC(c1csc([N+](=O)[O-])c1)=O N1(C(Cc2cnc(C)s2)=O)CC(NC(=O)C(C)Cc2cccnc2)C2CCCC12 c1(C(=O)NCC(O)CNc2ncc(I)cn2)cccc(O)n1 C12(NC(CS(N)(=O)=O)=O)COC(C1)C(NC(=O)CC1CCS(=O)(=O)C1)C2 CS(=O)(=O)c1ccc(C(=O)NCC2CC2CNC(c2cc3sccc3[nH]2)=O)o1 N1(C(c2c(C)ccnn2)=O)CCN(C(=O)CSC2CCS(=O)(=O)C2)CC1C C1(C(N2CC(C(=O)NCCSC(C)(C)C)(OC)C2)=O)CC2CC(=O)C1O2 C1(CN(C(C2N(CC)CCC2)=O)C)CN(C(c2c[nH]c(=N)s2)=O)CCO1 Cc1conc1CC(=O)NC(C)CC(C)NC(=O)C(C#N)=CC1CC1 c1(C(=O)NC(CN(C(c2c(Cl)cc(C)s2)=O)C)C)cc(F)c(C(F)F)cc1F c1(C2C(CN(C)C(C3(C)CC3(C)C)=O)C2)cccc(Br)c1.C12CC(C1)CNC2=O C1(NC(C2CCN(C(C(=O)NCC)=O)C2CC)=O)CC2CCC1CC2 N1(C(c2cc(C(C)=O)oc2C)=O)C(CNC(c2cc(C)ns2)=O)CC2COCC12 Cc1ccc2cc(C(=O)NCC3(F)CN(C(=O)CC4COCCO4)C3)ccc2c1 C1(CNC(C2(C(=O)NC)CCC2)=O)(OC)CCN(C(=O)C(C)CC2CCC2)C1 N1(C(Cc2ccc(CC)cc2)=O)CCCC2CN(C(=O)CC3(C)CCCC3)CC12 c1(C(=O)NCC2(F)CC(CNC(c3ccncc3)=O)C2)ccc(Cl)cc1Cl N1(C(CCOCC#C)=O)CC(CNC(=O)C(c2cncn2C)O)C(C(F)(F)F)C1 C(CC(C)(C)C(=O)N1CCC(C(C)CNC(C2(C(F)F)CCC2)=O)CC1)OC C1(F)(C(=O)NCCC2N(C(C(c3cn(C)nc3)=O)=O)CCSC2)C(C)(C)C1(C)C Cc1ccc2nc(C)cc(C(N3CCC(NC(c4ccsc4)=O)C3)=O)c2c1 c1(OC(C)=O)ncc(F)c(N(C(C2CCCN2)=O)Cc2ccccc2F)n1 N1(C(CNC=O)=O)CCCC2(CCCN2C(=O)CN2CC=CC2)C1 N1(C(Cc2c(C)cc(C)s2)=O)CC(C2CCCCN(C(c3cnoc3)=O)C2)C1 CC1=C(C(=O)N2CC(O)(CN(C)C(c3cc(C(C)C)no3)=O)C2)CCC(C)(C)C1 C1(C(C)C)CC(C(=O)NC2CCN(C(c3ccsn3)=O)C2C)CCO1 CC1(C(=O)NC2CC2NC(=O)CSCCN(C)C)CCc2ccccc2C1 c1(NC(C2CC2C(=O)NC2(CC(F)F)CC2)=O)cc(F)cnc1Cl C1(CN2C(=O)OCC2)CCN(CC(=O)NC=O)CC1 Cc1nc(CCC(N2CCCC2C(C)NC(C2(S(N)(=O)=O)CC2)=O)=O)oc1C N1(Cc2nc(CCC)on2)CC2CN(C(C3CCCNS3(=O)=O)=O)CC2C1 C1(CN(C(=O)CC2CC3(CC3)C2)C)COCCN1C(=O)C(F)C1CCC1 N1(C(Cn2cccc(C)c2=O)=O)C2CCC1CN(C(C1CCCC1C)=O)CC2 C1(CC)C(C(=O)N(C(C)C(C)(C)C)C)CCCN1C(=O)C(N)=O C(=O)(C1CCNc2c(C)cccc21)N(CCNC(C(CCCCCC)CC)=O)C N1(c2n(C)nnn2)CCCOC(CNC(c2nnn(C(C)(C)C)n2)(C)C2CC2)C1 Cc1cc(F)cc(C)c1C(=O)NC1CC(CNC(=O)CC2CCC(C)C2)C1 N1(C(c2c(OC)csc2)=O)CCC(NC(c2ccnn2C(C)(C)C)=O)C(CO)C1 C1(C(=O)NCC2(CC)CC2)C(C)CN1C(=O)C(O)CSC C1(CC)CCC(C(=O)O)CN1C(=O)C(C)OC1CCC(F)(F)CC1 N1(C(C(CC=C)C)=O)CCCC(C)(NC(c2ccc(C3CC3)s2)=O)C1 Cc1ccc(Br)c(C(=O)NCC(C)CNC(=O)CC2C(C)(C)C2(C)C)c1N c1(C(=O)NCCCN(C(=O)C=C2CCC(C)CC2)CC)ccc(Br)nc1N C1(CC(=O)N(C)CC2CC2(F)F)C2CCCC2N1C(c1cc2occc2[nH]1)=O C1(C(=O)OCC)(NC(=O)NC2CC(C(C)(C)C)C(O)C2O)CC(C)CC(C)C1 CC1CC(NC(c2cn(-c3cnn(C)c3)cn2)=O)CN(C(=O)CCCC(F)F)C1 C1(C(=O)NCCOCC)(CCNC(C2CC2F)=O)CCC(=O)N1 c1(C(=O)NC2(C(=O)NCCCP(C)(C)=O)CCC2)cnn2c1OCC2 c1(C(=O)OCCOC(F)F)nncc2ccccc12 C1(C(=O)NC(C=C)C2CCC2)CC(C)CN(C(=O)C(=CCCCCC)C)C1 c1(C(=O)NCC2CN(C(c3cncc(C)n3)=O)C3CC23)ccn2nccc2c1 CN1CCC(OCC(N2CCC2CN2CCSCC2)=O)CC1.C1(=O)C(F)(F)N1 c1(C(N2CC3CN(c4nc(OC)c(Br)cn4)CC32)=O)ccc2cccnc2n1 C1(C(=O)NC2CCN(Cc3ccc(C)o3)C2)NC(=O)OC1(C)C.N12CCCC1C2 C1(CCN(C)C(c2ccc(F)cc2)=O)CCN(C(=O)Cn2c(O)nnc2O)CC1 C1(C(N2CC(O)(C(C)NC(c3cn(C)cn3)=O)C2)=O)CCCC1S(C)(=O)=O C1(CC(=O)NC(C2CCCN(Cc3cnc(Br)s3)C2)C)CCCCN1C C1(CNC(Cn2c(C)ncc2)=O)CN(C(=O)COC(F)(F)F)CC1(F)F Cc1cc(F)cc(C(=O)NCCC2(C)CCN(C(c3cncc(F)c3)=O)C2)c1N N1(C(C(CCOC)OC)=O)CCN(C(C2CCN(OC)CC2)=O)CC(C)(C)C1 C1(NC(c2ccoc2)=O)C=CCC(C(=O)N)C1.N1(CCC2CC2)CC=CC1 C(C1CCCC1)=CC(C(=O)CC1(N(C)C)CCC1)=O.CC(C)CNCCO N#CC1CCCN(C(=O)CCCNC(c2csnc2Cl)=O)C1 c1(C(N(CC(C)(C)CNC(c2cnn(C3CC3)c2)=O)CC)=O)c(C)cccc1C N1(C(C(CSC)C)=O)CC2N(C(C34CC5CC3C4C5)=O)CCC2(C)C1 c1(C(N(CCNC(c2sccc2C(=O)OC)=O)CC)=O)cn2cc(C)c(C)cc2n1 CCCCCCC(C)C(=O)NC1CCC(NC(C2CCC(C(C)(C)C)CC2)=O)C1 C(=O)(C#CC1CCCCC1)NCC(CNC(C(c1ccc(C)cc1)=O)=O)F C(=O)(C(O)C(C)CC)NCC(CC)(CC)NC(c1c(CC)n(C)nc1)=O C(C(C)(C)C(=O)NCCc1ocnc1C(=O)NCC1(C)CCCC1O)N(C)C c1(C(=O)NC(CC)CNC(c2cnn(C)c2SC)=O)cc2c(s1)CN(C)CC2 C12(COC)CC(NC(=O)CC3(OC)CCCC3)(CN1C(c1cn[nH]c1)=O)C2 n1(CC)nc(C(=O)NCC23CC(CN2C(=O)CC2CC24CC4)C3)cc1C c1(C(=O)NC2C(CNC(=O)CN3C(=O)CNC3=O)CCC2)ccn2ccsc12 N1(C(=O)NCCn2ccc([N+](=O)[O-])n2)CCC2(CC1)CC(N1CCOCC1)CO2 C12(COC)CC(NC(C3CC3C(C)NC(=O)CC3CCN(C)C3=O)=O)(CO1)C2 C=CCC(C)(CC)C(=O)N1CC2CC2C1 C(=O)(C#CC1CCCCC1)NC(COC)C(=O)N1CC(C)(C)C1 C1(N(C(c2c(C)cc(C)o2)=O)C)CCN(C(c2cnccc2C(F)F)=O)CC1C CCCC(CCCO)C(=O)N1CCOCC1CNC(C12CC(CC(F)F)(C1)C2)=O C12(C(N3CC(N(C)C)C3)=O)CC1CN(C(c1ccc(=O)oc1)=O)C2 c1(C(N(CC(C)N(C(Cc2cc(C)no2)=O)C)C)=O)cc(F)cc(Br)c1O C12(CNC(CC(C)(C)C(F)F)=O)CCCC1N(C(=O)CC1CC(=O)C1)CCC2 N1(C(CC)=O)C2CCC1CC(CNC(c1cncn1-c1ccncc1)=O)C2 C=C(C)CCCC(=O)NC(C)(CNC(=O)C(C)C=Cc1ccccc1)C1CC1 N1(CCN(C(c2ccccn2)=O)C)CCCOC1=O.C1(C(C)C(=O)O)CCOCC1 Cc1nn(CC(C)C)c(Cl)c1CN(C(Cc1cccs1)=O)Cc1ccco1 N1(C(=O)NCCCCc2scc(C)n2)CCOC2(CCCOC2)C1 c1(OC)cc2c(cc1C(=O)NC(C)CNC(c1nccc(SC)n1)=O)CCC2 N1(C(C2CN(C(C)C)C2)=O)CC2CCC1CN2C(C12CCC(CC1)C(C)O2)=O c1(NC(C2CCCOC2C)=O)cc(S(N)(=O)=O)c[nH]1.C12(CC=C)CN(C1)C2=O C1(N(C)C(c2cc(C(F)F)[nH]n2)=O)CN(C(C2CCCN2C)=O)CC1O c1(OC(CC)C(=O)NCC2CCN(C(C)=O)C2)ccccc1Cl Cc1ccncc1CC(=O)N(CCC(C(C)C)NC(=O)C(C)(C)O)C c1(C(C(=O)NC2CCN(C(=O)CN3CCCC3)C2)(F)F)ccccc1Cl c1(CCC)cc(C(=O)NC(C)(CNC(=O)CC2CCC(C3CC3)O2)C2CC2)no1 c1(C(=O)NCCC2(NC(C3OCCC(C)C3)=O)CC2)cc(F)c(C(F)F)c(F)c1 C1(CC)(OC)CCN(C(c2[nH]nnc2C)c2nnnn2C2CCCC2)C1 N1(C(c2c(C)nnn2C)=O)CC2CCC1CN2C(C1CCCCC1C1CC1)=O O=S(=O)(c1cccnc1NC1C=CCCCC1)NCCS(=O)(=O)CC1CC1 C(=O)(C1=CSCCO1)N1CCC(N(CCC)C(c2c[nH]nc2F)=O)C1 c1(C(N2CCC(C(C)NC(C3CCCCS3(=O)=O)=O)C2)=O)noc2c1COCC2 c1(NC(C2CN(c3cc(C)nc(C)n3)CC23CCC3)=O)ccc2c(c1)CCC2 C1(C(C(=O)NC(CC)C)N(C2CCCOC2)C2CC2)C2CCCCC12 N1(C(c2ccccn2)CC)CCC(O)(CC(=O)OC)C1 C1(NC(C(C)N(C)C(=O)OC(C)(C)C)=O)CCC(NCC2CC2)CC1CCC#N c1(C(=O)N(C2C3CNCC23)C(c2ncncc2F)=O)cc(F)cc2[nH]ccc12 C1=CC(=O)C(=O)Cc2scc1c2.C1(N)C=CCN(C(=O)CO)C1.N1(C(C)=O)CCCC1 N1(C(CSC)=O)CC(Nc2ccnc(CO)n2)CCC1C C(=O)(CC(C)(C)c1cccs1)NCC1CCC(NC(c2cnc(C(C)O)s2)=O)C1 N1(C(=O)OC(C)(C)C)CC(NC(=O)NCC2CC=CCC2)COCC1(C)C C1(C(=O)NCCCCNC(=O)CCNC(C2CCCCC2)=O)CCC12CCCO2 c1(C(=O)NCC2(OC)CN(C(C(CC(C)C)N(C)C)=O)C2)ccc2sncc2c1 C1(CN(C(c2c(CC)nn[nH]2)=O)CC)CCCCN1C(C1CC12CCC2)=O c1(-c2ccc(NC(c3c(OC)ccc(O)c3)=O)nc2)cc(C)c(N(C)C)cc1C CCCCCCCCCC(=O)N1CCC(CNC(c2c(C)cc(C)oc2=O)=O)C1 C=CC1(C(=O)NC2CCC(CC(N3CC4CC3CS4)=O)C2)CCCC1 C1(NC(CCCCC#C)=O)CCCOC12CCN(C(C1CCC(C)(C)O1)=O)CC2 N1(CC)CCC(Oc2nc(C(N3CCCC3C=CC(=O)OC)=O)no2)CC1 CC1CN(C(=O)COC2CCCOC2)CC(C)N(C(=O)C=Cc2ccoc2)C1 c1(C(N(C)CC2(O)CN(C(C3(C(C)C)CCC3)=O)C2)=O)cc(O)c2ccsc2c1 c1(C(N2CCCC(NC(c3c(C)onc3)=O)C2C)=O)cc2n(n1)CCOC2 n1(CC(=O)NC2CC(CC(N3CC4CCCCC4C3)=O)C2)ccc2ccccc12 C1(NC(C2CC2c2cnc[nH]2)=O)CCCN(C(c2cscn2)=O)C1 S(=O)(=O)(c1ccc(Cl)cc1F)N(CC)C.Cc1ccc(I)c(C)c1NC(=O)CSC c1(-c2nc(CCCOC)nn2C2CCS(=O)(=O)C2)occ2c1CCOC2 c1(OC)cscc1C(N1CC(OCCC(=O)NCCC2CCCC2)C1)=O c1(C(N2CCC(NC(C3(CC)CCOC3)=O)C(O)C2)=O)c(Cl)cnc(OC)c1Cl Cc1noc(C2CC2)c1C(=O)NCc1ccc(CNC(=O)CNC=O)cc1 c1(CC(=O)NC2(CNC(C(C)(C)C3CCCO3)=O)CC2)cccc(F)c1 c1(OC)ccccc1C(=O)NC(C)C(C1CCCCC1)NC(c1cc(Cl)no1)=O C(CCC(C)(C)CO)NC(=O)CN(C)C(C)C.CC(=NOCC#N)C=O c1(C(N2CCC(O)(C(C)CNC(=O)Cc3cnccn3)C2)=O)c(N)cccc1Cl C1(C(=O)NCC2CCC2)CC2CCCCC2N1C(c1cnc(C(F)(F)F)cn1)=O C1(C(=O)NC(C)CC2CN(C(=O)CSCCN(C)C)C2)CCCCC1C CCCC(C(O)C(=O)NNC(=O)CCC1CCCCC1)NC(=O)OC(C)(C)C.CC CC1=C(C(=O)NC(C)CCCNC(c2ncn(C)n2)=O)C(C)(C)CCC1 Cn1cnc2sc(C(=O)NC3CN(C(=O)CCC4CC4)CCC3(C)C)cc12 C1(NC(CC)=O)CCCN(N2CCC3CNC(=O)C3C2)C1 c1(NC(=O)NC(C2CCN(C(=O)OC(C)(C)C)CC2)C)cccc(NS(N)(=O)=O)n1 CC(N=[N+]=[N-])C(=O)NCC1CN(C(c2[nH]nnc2C2CC2)=O)CC1C C=CCC(CNC(=O)C=Cc1ccco1)C(=O)N1CC(CC)C1 CC1(C2CCN(C(C3(NC(C4CC5(CCO4)CC5)=O)CC3(C)C)=O)C2)CC1 c1(C(C)C)cc(C(=O)NCc2cc(C(=O)NCCn3ccnn3)co2)n[nH]1 c1(-n2cc(CC3CN(C(C4CCN(C)CC4)=O)C3)nn2)cc(F)cc([N+](=O)[O-])c1 N1(C(C2C(OCC)C2)=O)CCN(C2CCN(C(=O)CC3C(=O)ON=C3C)C2)CC1 c1(C(N2CC(OC)(CNC(=O)CN3CCCC3C)C2)=O)cn(C)c(O)n1 C1(C(N2CC(C)OC(C)C2)=O)(OC)COCC1(C)C.c12cccnc1C(=O)N2 C(N=c1nc(NCc2cnccc2C)c2c([nH]1)c(C)nn2C)C1CC(CC)C1 CCC(C)(CC(=O)N(C)CCOCCNC(=O)Cc1cncnc1O)C(=O)OC n1(CC)ccnc1C(=O)NC(C)C(C)NC(=O)C(C1CCC1)OC c1(C(N(C2CCN(C(c3ccc(SC)o3)=O)C2)CC)=O)cc(C2CC2)ccc1Cl C1(C(N2CC(C)(C(=O)Nc3ccnc(OC(F)F)c3)C2)=O)CC2(C1)CN(C1CC1)C2 C1(CNC(CCCCC#C)=O)CCCCN(C(=O)COc2ccc(Cl)nc2)CC1 C(=O)(C(F)(F)C(C)(C)C)N1CCC(CNC(c2ccc(OC)c(Cl)c2)=O)C(C)C1 C(=O)(C(CCCOC)NC(c1cnn(C)c1Cl)=O)N1CCN(CCC#C)CC1 c1(C(=O)NCCN(C(C2C(CC)CCC2)=O)C(C)C)cc2cccc(O)c2[nH]1 C(=O)(C1CCCc2nncn21)N1C(CCNC(C(C(C)O)C)=O)CSCC1 CC(C(=O)N1CCCCC1CCCNC(c1cn(CCO)nn1)=O)CS(C)(=O)=O c1(C(N2C(CN(C(=O)C(F)n3cccn3)C)CCC2)=O)n[nH]c2c1CCC2 C12=NC(Cl)=CC(=NC1=O)N2.c1(C(C)OC)cc(F)cc(F)c1 N1(C(c2c(C)snc2)=O)CCCC(NC(c2conc2C2CCC2)=O)C1 C1(CCC(=O)N(CCO)CC)CC2(C1)CN(C(=O)Cc1cccnc1C)C2 n1(CC(=O)NC2C(C)CN(C(c3cnc(O)s3)=O)C2)cccc(O)c1=O C1(NC(C(C)N(CC)CC)=O)(CO)CCCN(C(c2[nH]nnc2C2CC2)=O)C1 C(C(C)(C)C#CC(=O)NC(C)CCN(C)C)NC(COC)=O n1(CC(=O)NCC2N(C(CC(C=C)C)=O)CCCC2)ccc(C)cc1=O c1(NC(C(=O)OCC)Cc2cccnc2F)ncnc2cc(Br)sc12 c12ccccc1C(=O)C(C)N2.C1(C(C)C)C(=O)N1.C1(OC)CCCCC1 C1(C(=O)NC2C=CC(CNC(=O)CSCc3ccc(Cl)s3)C2)CC2CCC(C1)O2 C1(C(=O)NC2C(NC(=O)CCc3cccnc3)CCC2)CCc2nnnn2C1 CC1(C)CCCC(C(=O)NCCC2CCCN2C(=O)C(=O)NCCC(N)=O)CC1 CN1C(=O)OCC1C(=O)NCC1(CNC(c2cc(C#N)c[nH]2)=O)CCCCC1 c1(OC)cnncc1C(=O)N(C1(C(=O)NOCCC2CC2)CCC1)C1CC1 C1(NC(CCCNC(C)=O)=O)CC2CC1N(C(c1cc(C)c(C)s1)=O)C2 N1(C(CC2CC(NC(CNC(C(C)(C)C)=O)=O)C2(C)C)=O)CC(F)(F)C(F)(F)C1 C12(n3cc(C(N4CC5CCC4C5)=O)nn3)CCC(NCCC3(C)CC3)(CC1)C2 C(=O)(C(CCC)N(C)C)NC1(CCC(=O)NC2CC(C(C)C)OC2)CCC1 C1(C(=O)NC(COC)CO)C=CC(NC(=O)CCc2cscn2)C1 C(=O)(C(C)(C)CC(=O)OC)N(CCCNC(c1cccc(CC)c1C)=O)CC C1(NC(N2CC(COC(C)C)C2c2cccnc2)=O)CC2(CO1)CC(F)(F)C2 Cc1cc(CC(=O)N(C2CN(C(C3CCCOC3)=O)C2)C)no1 Cc1[nH]c(C(=O)NCC23CC(CO2)N(C(C2CCS(=O)(=O)C2)=O)C3)c(C)c1C C(=O)(C1CSc2ccccc21)NCCN(C(=O)C(O)Cc1ccccc1)CC C(CC(=O)NCC1OCC2CCC1C2)(C(C)(C)C)NC(C(C)n1cncn1)=O Cc1c(C(N2CCN(C(c3ccc(N4CCCC4)nc3)=O)CC2)=O)cnn1C Cc1ccccc1COCC(N1CC(NC(=O)COCC(F)F)CC1C)=O CCC(C)C(C(=O)NCCC1(O)CCC1)NC(=O)CC1CCSC1 C1(NC(CC(C)(C)C)=O)CCCC12CN(C(c1cc(C3CCC3)on1)=O)C2 C(=O)(CC(O)CNC(=O)C(F)C1CC(NC(=O)CC=C(C)C)C1)OC n1(C(C)C)nccc1CC(=O)NCC1(NC(=O)Cn2cc[nH]c2=N)CCCC1 c1(C(N(CCOCCN(C(C(C=C)CC)=O)C)C)=O)cccc(F)c1CC C(=O)(C(CC(C)C)NC(=O)C(c1cnc(Cl)n1C)N1CCC(CCOC)C1)OC C1(C)(CNC(C(C)Oc2ccccc2)=O)CCCN(c2ncns2)C1 C1(C(N(C(C)CNC(=O)C=C(Cl)Cl)CC)=O)CC(=O)C1C Cc1ccc(C#N)cc1N(C1CCS(=O)(=O)C1)C(C1(C)Cc2ccccc2N1)=O Cc1c(F)ccc(C(N2CCC(C(C)C(=O)NC3C=CCCCC3)CC2)=O)c1F c1(CC(=O)NCC(CC=C)NC(c2ocnc2C)=O)ccc(Cl)c(C)c1 C(=O)(CCCCN(c1ccco1)C)N(C(CC)CC)C C1(CC(=O)OCC)CN(C(c2csc(=N)[nH]2)=O)CCN1C(c1ccc(F)cc1)=O c1(C(N2CCC(N(CCC)C(C3CCC3C)=O)C2)=O)cc(CC)n(C)n1 Cc1cc(OC(F)F)cc(C)c1C(=O)NCC1CC(C2CCC2)C1 c1(C(=O)NCC2CCCN2C(c2c(Cl)n[nH]c2C2CC2)=O)ccccc1F C1(NC(C2COCCO2)=O)CN(C(=O)CSc2nncs2)CC2CC12 C(CC(C)(C)CNC(=O)C(C)(C)Cc1cnn[nH]1)NC(C(C)OCOC)=O N1(C(C2(C(=O)NC)CC2)=O)CCCCC2(CCN(C(C3(Cl)CC3C(C)=O)=O)C2)C1 c1(OCC(=O)NC2CN(C(c3cnc(C)n3C(F)F)=O)C2)nc(O)nc(O)n1 Cc1cc(C(=O)NOCC(N2CC(O)(C3(C)CC3)C2)=O)sn1 C1(OC)CC(NC(c2cnoc2C(C)C)=O)CN(C(=O)C(=C2CCCCC2)F)C1 C1(NC(c2nc(COCC)sc2)=O)CN(C(c2cc(OC)ncn2)=O)CC1(C)C N1(C(c2ccc(C)nc2O)=O)CCC2CCN(C(c3cccc(CO)c3)=O)C2C1 c1(C(=O)NC2CCCCN(C(CCC=C(C)C)=O)C2)cc2cccc(O)c2n1C N1(C(CNC(C(C)=C(CC)C)=O)=O)CC(C)(SC2(C(=O)NC)CCC2)C1 N1(C(C2N(C(C(C)NC(CC)=O)=O)CC=CC2)=O)CCN2CC(C)CC2C1 CC1CCC(NC(=O)CC2CCC(C3CC3)O2)CN1CCc1cc(Cl)nc(=N)[nH]1 n1(CCNC(=O)CC2CC2)cc(C(=O)NC(CO)C2(O)CC2)nn1.c1nc[nH]n1 N#Cc1cc(F)cc(F)c1NC(C1CCN1C(=O)Cc1ccccc1[N+](=O)[O-])=O C1(CNC(Cc2c(C)nn(C)c2)=O)COCCN(C(C2CCC(=O)N(C)C2)=O)C1 C1(NC(C(COC)(C)C)=O)CS(=O)(=O)CC1N=c1ccc2c([nH]1)CCCC2=O C1(CC)CN(C(c2n[nH]c(C3CC3)n2)=O)CCC1NC(c1nnnn1C)=O C(=O)(CCCC(CC)NC(=O)C(O)COC)N(CCCC)CCO C12(CC(=O)N(CCNC(CC3CCCC(OC)C3)=O)C)CCC(CC1)C2(C)C c1(C(N2C(C(N3C4CCC3COC4)=O)CC3CC32)=O)cccn2ccnc12 Cc1sc(O)nc1C(=O)N(CC(C)C(=O)NCC(CC1CC1)CO)C C1(NC(C2N(C)CCCC2)=O)CC2CCC1CC2NC(C1CC1(C)C(F)(F)F)=O N1(C(C(C)CN(C)C)=O)CCCCCC1CNC(c1ccc(N(C)C)cc1)=O CCC(CC(=O)NCC1CC2CC2N1C(c1ccc(C#N)[nH]1)=O)CC(F)(F)F N1(C(c2c(OCC)nccc2)=O)CCN(C(c2cncc(Cl)c2Cl)=O)CC1C S(=O)(=O)(c1ccc(C)s1)NCC(=O)N(CCCNC(CCC)=O)C c1(C(N(CCCNC(C2(CC)CCC2)=O)C)=O)cc(-c2ccco2)on1 c1(C(C)C(=O)NC2(CNC(C3CC(Cl)(Cl)C3)=O)CC2)ccc(F)cc1 C1(C(=O)NCc2cc(C(=O)NC3(C#C)CC3)n[nH]2)CCCN(C)C1 Cc1ccc(C(=O)NCCOC2CCN(C(c3c(C)csc3Cl)=O)CC2)nc1F Cc1nsc2ncc(C(N3CCN(C4CCN(C(=O)CC(C)F)C4)CC3)=O)cc12 Cc1cc(NC(C2CCCC2CNC(=O)C(O)CC(C)C)=O)cc(C)c1 C(=O)(CS(=O)(=O)C(C)C)NC(CC)CNC(c1coc(C(C)OC)n1)=O C(=O)(C=C1SCC(=O)N1C)NC1C(OC)CN(C(C2CC3(C2)CC32CC2)=O)C1 c1(OC)ccc(CC(=O)NC23CC2CN(C(c2ccccc2CSC)=O)C3)cn1 CC1(C)CC(C)(NC(=O)C(C2CC2)NC(=O)CCC2(C)N=N2)C1 C1(C#N)(CCOC)CN(C(C2COCCC2C)=O)C1 c1(C(=O)NC(c2ccccc2)C(=O)NCC(C)(C)N(C)C)ncccc1N c1(C(=O)NCCN(C(=O)C(C2(O)CCCC2)F)CC)cc(C(C)C)[nH]n1 N1(C(COCCOC)=O)CCN(C(C2OCC2(C)C)=O)CC1C(F)F c1(OC)ccccc1CNC(C)Cc1nc(COCCCC#N)no1 C1(CCC(=O)N(CC(=C)C)CC)CCCN(C(=O)C=Cc2cnn(C)c2)C1 CC1CN(C(C2(CCO)CC2)=O)CC1CNC(=O)C(c1cccc(F)c1)(C)C CCS(=O)CC(=O)NC1CC(NC(c2ccccc2Cl)=O)C1 C1(NC(c2c(OC)csc2)=O)(CNC(c2ccn3ccsc23)=O)CCCCC1C c1(C(=O)NCC2N(C(C3OCC(C)C3)=O)CC(F)(F)C2)ccc2oc(=O)oc2c1 C1(CC(N2CCC(N(C(c3nc(C)oc3)=O)C)C2)=O)NC(=O)NC1=O CCN=c1[nH]cc(C(=O)NCC2CC(NC(=O)Cc3ccns3)C2(C)C)s1 N1(CC)C(=O)CCC1C(=O)N(C)CC1(O)CN(C(c2nn(C)cc2SC)=O)C1 C1(C(=O)NC2C(OC(C)(C)C)CC2)CCCCC1NC(c1cocn1)=O Cc1cccc(C(N2CCC(N(CCO)C(c3nccc(Cl)c3F)=O)C2)=O)c1F C1(CC(=O)NC(C)C(=O)NCC2C=CCC2)CN(C(C2CC23CC3)=O)CCO1 Cc1nnc2n1CCCC2C(=O)NCC1CN(C(C2(F)CCOCC2)=O)CCO1 C(=O)(CC1=CCCCC1)N1CCC(OCC(=O)NC(C=C)C(F)(F)F)C1 N1(C(=O)NC2C(C)(C)COCC2)CCC(S(=O)(=O)c2ccc(Br)cc2)CC1 C12(NC(C=COCC)=O)CCCCCC1N(C(c1cc3nc[nH]c3cn1)=O)CC2 c1(C(N2CC(OC)CC(NC(CC(=O)OC)=O)C2)=O)n[nH]c2c1CCCC2 C(C(O)CC(=O)C(=O)CCc1cnn(C)c1)N(C(C1(CCC)CC1)=O)C1CC1 N1(c2ncc(C)c(C)n2)CC2CCC1C1CN(C(=O)CCc3cn(C)nn3)CC21 C1(NCCC(CC)CO)CCC2(CC1)CCN(C(=O)C(C)CC(=O)OC)C2 N1(C(C2C3CCCC2CC3)=O)CCc2ccc(Br)cc2C1C(F)(F)F N1(C(c2ccc(C#N)cn2)=O)C2CCC1CN(C(=O)CCCC#N)CC2 Cc1cc(F)oc1C(N1CCC(C(C)C(=O)N(C)C(C)C)CC1)=O c1(-c2ccc(CN3CCC(O)CC3)cc2)ccc(C(F)(F)F)c2ccncc12 C(CN=c1cccc(S(=O)(=O)NC(CO)CC(C)(C)C)[nH]1)Oc1c(OC)cccc1 N1(C(c2n(CCC)cnc2)C(=O)NC(C)CC)CC(CO)OC(C)C1 c1(C(F)F)cccc(NC(C2COCCO2)C2CC2)c1O C1(CCNC(CC(C)(C)O)=O)CN(C(=O)CCCC2CCC2)CCCO1 Nc1c(C(N2CC=CC(NC(C3CCCS(=O)(=O)C3)=O)C2)=O)sc2nccnc12 N1(C(Cc2cnc(OC)c(Cl)c2)=O)CC2CN(C(=O)COCC3CCC3)CC2C1 c1(C(=O)NC(C2CCN(C(=O)CN3CC4CC4C3)C2)C)c[nH]c2cc(N)ccc12 C(=O)(C(C)C(CC)CC)N(C)Cc1cccc(CNC(CSCC=C)=O)c1 N1(C(c2n(C)ccn2)=O)CCC(OC2CN(C(=O)CC3(CN(C)C)CC3)C2)CC1 O=C(C(CC(Cl)Cl)C(F)(F)F)n1cc(CCC(F)=C(F)F)nn1 C12(NC(c3cc[nH]c3)=O)CC(C1)N(C(c1cccc(OC(F)(F)F)c1)=O)C2 C1(NC(Cc2cn(C)nn2)=O)CCN(C(c2ccc(O)cn2)=O)C1C(C)(C)C CCCCCCC(C)NC(=O)C(C1CC1)NC(=O)COCCSC Cc1ncc(C=CC(=O)N(CC(C)CNC(C2COCCO2)=O)C)s1 c1(CNC2CCCC(C(=O)NCCCOCCCCC)C2)ccc(C#N)cc1Br c1(OC)c(Cl)cc(C(N2CC(NC(=O)CCN(C)CCO)CC2C)=O)nc1Cl c1(C(C(=O)NCC2CCCO2)N(C)Cc2ccccc2)csc2c(Br)cccc12 C(=O)(CCCCCNC(c1c[nH]nc1C)=O)N1CCCC(CC)C1 C1(NC(Cc2cnc(C)s2)=O)CC2CN(C(C3CC4CCC3O4)=O)CCN2C1=O c1(C(C)C)ncsc1C(=O)N(CC(C)(C)CNC(=O)CSC(F)(F)F)C CC1=NNC(=O)C1CCC(=O)NC1CC(C(C)NC(=O)C(C)(C)CO)C1 C1(CNC(c2cnc(COC)s2)=O)CN(C(C2CCC(C)=C(C)C2)=O)CC12CC2 CC(CC(N)=O)C(=O)NCC1(C)CCCN(C(=O)Cc2cc(F)ccc2F)C1 Cc1cc(=O)n(CCC(=O)NCC2CCN(C(C3CC(C)OC(C)C3)=O)C2)cn1 Cn1c(CCC(=O)NCC2CCN(C(C3CC4CCC3C4)=O)CC2)nnc1S Cc1cc(C2CC2)ccc1C(=O)NNC(=O)NCCC(C)(C)O N1(C(C(C=C)O)=O)CCCCC2C1CCCN2C(c1cnn2c1CCC2)=O CCC(CC)(C(N)=O)NC(C1CC(C)(NC(C23CCC(OC)C2C3)=O)C1)=O C1(C(N(C(CC)C(=O)NCC2(O)CCOCC2)C)=O)CC12CCCCC2 C1(C(=O)N(CCO)CC#N)CCN(SCl)CC1.CC(C)(C)SCC(=O)N1CC1 CC1=NN(C)C(=O)C1CC(=O)NCC1(F)CCCN(C(C2COC(=O)N2)=O)C1 CC(CC(C)(C)C)C(=O)N(C1(C(=O)NCC2(C)CCC(O)CC2)CC1)C CC1CN(C(C2CCCO2)=O)CC(C)N(C(=O)C=CC2CCCCC2)C1 C1(NC(N2CCCC(N(c3[nH]c(=N)sc3)CCO)C2)=O)CC2CCCC(C1)C2 CC1(C)CC(CNC(c2nc(Cl)sc2Cl)=O)N(c2ccnc(CO)n2)C1 CC1(CC(N2CC3C(C(N)=O)C3C2)=O)CCN(C(C2CC3(CC3)CO2)=O)C1 C(C(C)(C)COC(C)(C)C)(c1ccc(Br)cc1)N(C(C)C)Cc1c(C)nc[nH]1 Cc1ccc(C(=O)NC2(C(N3CC(O)CCC3C)=O)CCOCC2)cc1C C1(CNC(c2cnc(C3CC3)[nH]2)=O)(CO)CCN(C(c2ccsn2)=O)CC1 N1(CC(c2c(C)ccc(F)c2)=O)CC2(CNC(=O)OC2)C1.C1C(=O)N1C(C)C c1(OC)cc(CC(N2CCCC(CNC(C3C4CCC(=O)C34)=O)C2)=O)ccn1 c1(CC)ccc(C(=O)NC2(CCNC(=O)CCc3ccccc3F)CCC2)nc1 c1(OC(C(=O)N(CCNC(C2CC(OC)C2)=O)C)C)ccccc1Cl N1(C(C2C(CNC(=O)CCC3CCCO3)C2)=O)CCC2(CCCCC2)C1 C1(C(N2CCC(N(CCO)C(C3CCCSC3)=O)CC2)=O)CCCCCCC1 n1(C(CC)C)c(SCC=O)nnc1-c1cccc(N)c1.C1(=O)CC(=O)CCN1CC.OC C1(C2(O)CN(C(=O)C(C3CCCC3)OCC)C2)(CNC(C(C=C)(C)O)=O)CC1 c1(C(N(C2CCN(C(=O)CC3COC(C)(C)CO3)C2)C)=O)cccc2ccoc12 N1(C(C=CCOC)=O)CCN(C(C2C(C)C2C)=O)C(c2ccc(CC)cc2)C1 c1(CNC(c2cc(SC)oc2C)=O)ccc2c(c1)CCC2NC(C1(O)CCC1)=O C(=O)(CC(O)Cc1ccccc1)NC(CNC(C1N(CC)CCC1)=O)CCOC c1(-n2cc(CNC(C(C)(O)CCc3ccccc3)=O)nn2)cnc2c[nH]nc2c1 c1(NCC2CCN(C(CC3(OC)CCC3)=O)CC2O)ncccc1S(C)(=O)=O C(CCCCC(=O)NC(C)(C)CNC(c1cc(C)on1)=O)SC Cc1cc(C(N2CC3(CC(C(=O)NC(C)C4CC4)C3)C2)=O)c2c(C)n[nH]c2n1 Cn1ncc(C(N2CCCC2(C)CNC(=O)CC2CC23CC3)=O)c1N N1(C(CC(CC)NC(=O)Cc2cnsc2)=O)CC2CC=CC1C2 N1(C(c2c(O)ccc(CC)c2)=O)C2CCC1CC(NC(=O)CC1(CO)CC1)C2 c1(C(=O)NC(C(N2CC(CCC)C2)=O)c2ccco2)nscc1C Cc1cnc(C(C)NC(=O)C(=O)N(C)CC2CCSC2)o1 C(=O)(C(F)CC1CCC1)NC(C1(CNC(C2CC2(C)C)=O)CC1)C c1(C(N2C(CNC(C3CCC3C(F)F)=O)CC(F)C2)=O)cc(Cl)nnc1O C1(OC)(CNC(=O)COCC2CCCO2)CCN(C(C2C=CC2C(=O)OC)=O)C1 CCCCCCC(=O)NC1(CNC(=O)CC2CCC2C(=O)OC)CC1 C(N=c1[nH]c(=NC2CCCS(=O)(=O)C2)c2c(ncn2C)[nH]1)c1ccc(C)cn1 CC(C)CCC(=O)C(=O)NCC(C(=O)NC(c1ccnn1C)CO)N(C)C N#Cc1cc(F)cc(C#N)c1OCc1noc(C(F)F)n1 N1(C(CN(CCC)C)=O)CCC(C(=O)N(C)CC2CN(C)C2)C(C)C1 N1(C(CC(=O)N(CCC(=O)NC)CC)=O)CCC2(CCCO2)CC1 S(=O)(=O)(c1c[nH]c2nccc(Cl)c12)NC(Cc1cccc(C)c1)C(=O)O CC(C)(CC(F)C(=O)NCC1CCC2(CC2)CO1)NC(c1coc2c1COC2)=O N1(CCS(CC)(=O)=O)CCC(=O)N(CC2CCN(CC(C)C)C2)C1=O Cc1cc(C2CC2)cnc1C(=O)NCCC(C)N(C)C(c1ccc(Cl)cc1C)=O C1(NC(CC(C)NC(N)=O)=O)CCN(C(c2cccc(CCO)c2)=O)CC1O CC1(C)CCN(C(c2cc3ncccc3s2)=O)CC1NC(C12CC(CCO1)C2)=O C1(C(N(C(C)CCNC(=O)CC2CCC2)C)=O)CN(S(=O)(=O)N(C)C)CCO1 Nc1cc(Cl)ccc1NC(C1CN(S(=O)(=O)C(F)(F)F)C1)=O C1(NC(c2ccc(OC)nc2)=O)CN(C(c2ccoc2C(C)C)=O)CCC1CO C(=O)(C(C)C(C)C)NCCCN(C(=O)CC1CCCCN1C)CCC CC1(C)CCC(C(=O)NCC(O)CNC(c2cc(N)ccc2Br)=O)OC1 C12(C(=O)NCC(c3ccccc3)N(C(CCCC#C)=O)C)CCCC1CCC2 N1(CC2(Cn3c(C)ncc3)CCOCC2)CCCC2(c3ccccc3)CC2C1 CCCC(C)CC(=O)NCC1CCN(C(c2cc(C(F)F)ccc2C)=O)CC1 C1(NC(C(C)=C(CC)C)=O)CCN(C(=O)CSCC(c2ccccc2)=O)CC1C c1(NCCCC(N)=O)nc(N2CCN(C3CCC3)CC2)nc2sccc12 C1(NC(CCCN(C(C)=O)C)=O)C(C)CN(C(c2cc(C)c(C)cn2)=O)CC1C CCCCC(CC)C(=O)N1CC(OCC)C(NC(c2c(Cl)cncc2Cl)=O)C1 C(C(=O)NNc1cc(C(=O)N(c2ccccc2)CCO)ccc1Cl)(C(C)C)OC C1(NC(c2c(C)ocn2)=O)CC2(C(=O)NCCCc3ccsc3)COC1C2 C1(CN(C)C(C2Cc3ncccc3C2)=O)CN(C(=O)CNC=O)CC12CC2 c1(CC)cc(N)c(C(=O)NCC2CCC2NC(=O)C(O)CC(N)=O)cc1F C1(CN(C(=O)CC2CCSCC2)C)CC(F)CN1C(C1CC=CCO1)=O c1(C(N2CCC(C(C(C)C)NC(=O)C(C)C(F)F)CC2)=O)nccc2cc[nH]c12 CC1(C(=O)NCC2CC(NC(=O)Cc3ccc(Cl)s3)C2)CCCOC1 C#CCC(O)C(=O)NC(CCC1CC1)C(=O)NC1(c2cccs2)CC1 C1(NC(COC(C)=O)=O)CCN(C(c2cc(C3CC3)cnc2Cl)=O)CC1CO N1(C(=O)NCC2(C)CCC2)CC(CO)(CO)C1(F)F C(=O)(C1COc2ccccc21)N1CCC(NC(C=Cc2n(C)ncc2)=O)C(F)C1 c1(C(N2CCCC(CCNC(c3nn[nH]c3Cl)=O)C2)=O)cc2cc(F)ccc2[nH]1 N1(C(c2n(C=C)ncc2)=O)CC(NC(c2cc(O)cs2)=O)C2(CC2)C1 C=CC(C)(CC)C(=O)N(C)CC1(O)CCN(C(c2csc(COC)c2)=O)C1 C(=O)(N=c1[nH][nH]c(C)c1C)C1N(C(c2c(OC)ccnc2F)=O)CC(F)C1 C1(O)(CN(C(=O)CCCNC(N)=O)C)CCCN(C(C2CCC3(CC3)C2)=O)C1 C1(NC(C(CC=C)C)=O)CN(C(=O)CCc2cc(C)on2)CC2(CC2)C1 C(N=c1[nH]nc(CC(C)C)n1C)c1nc(COC)c(C)s1 c1(N(C(C)C2CC2)C(c2cccnc2Cl)=O)ccnc(N2CCOCC2)n1 c1(C(N2CC3C(C2)N3C(C2(C3CC3)CCOCC2)=O)=O)ccc2c(c1)CCNC2 n1(CC(=O)NCC2N(C(C(C)C(F)(F)F)=O)CC3CC32)sc(=O)c2ccccc12 N1(C(C2CCOCC2)=O)CCCC(C2CCN(C(C3(O)COC3)=O)C2)C1 C12(NC(C3CCN(C4CCN(C(C(CC)O)=O)CC4)CC3)=O)CCCN(CC1)C2 CC1CCN(C(c2nccc(Cl)c2O)=O)CC1CNC(=O)C(O)C1CCC1 S(=O)(=O)(c1ccncc1)NCC1(O)CCCN(Cc2cc(OC)cc(F)c2)C1 N1(C(CCCCN(C)C(C2(CO)CC2)=O)=O)CCC(F)C(O)C1 CC(C)CCCC(C)C(=O)N1CCC(NC(=O)CSC(C)(C)C)C(O)C1 c1(C(N2CC3C(CNC(C(CO)NC(N)=O)=O)(C3)C2)=O)ccc(Cl)c(Cl)c1 c1(C(=O)NC2CN(C(c3n(C)c(=O)ccc3)=O)CC(O)C2)cc(Cl)c(N)c(Cl)c1 Cc1csc2ncc(C(N3CCCCC3CNC(=O)C(C)(C)C3CCC3)=O)n12 C(=O)(N=c1[nH]c(Cl)ncc1O)C1N(Cc2ncc(C)nc2)C2CCC1C2 CCC(CC)C(=O)N(C1CN(C(C2(C#N)CCC2)=O)CC1O)C c1(C(=O)NCC(C2CCC2)NC(c2cc(C(N)=O)oc2)=O)ccc2nncn2c1 c1(NC)ccc(C(=O)NC2CCC(NC(=O)CC3(O)CCCOC3)C2)cc1F N1(C(C(CCC)=CCC)=O)CCC2CCN(C(=O)Cc3ncncc3Cl)CC12 C1(NC(CC(=O)NC2CC2)=O)CC2CCCC(C1)N2C(c1ccon1)=O C12(NC(=O)NCCNC(C(c3ccccc3)N(C(C)=O)C)=O)CC(C)(C1)C2 C(=O)(CCCC(=O)N(C(C)CC(=O)NCC1CCCNC1=O)C)OCC C1(CNC(CC2CC(C)(C)C2)=O)CCCCCN1C(C1CCCOCC1)=O Cc1ccc(NC(=O)CC2(C)CCN2C(C2CCC(=O)NC2)=O)c(C)c1 c1(NCc2nnc(C)o2)nccc(=NC(C)c2c(F)cccc2Br)[nH]1 c1(SCC)ccc(OC)c(-c2ccc(Nc3cn(C)cn3)nc2)c1 Cc1oc(CNC(=O)COC2CC2)nc1C(=O)Nc1cnn(CCO)c1 C(=O)(C1=C(CCl)N(CC)C(=S)NC1c1nc(-c2ncccn2)no1)OCC N1(C(C2(CC)CCOC2)=O)CC2(CCN(C(c3csc(C)c3N)=O)C2)C1 C1(CCC(=O)NC(C(=O)N(CCCN(C)C)C)C2CCOC2)CCC(=O)C1 CC1=C(C)CC(C)(C(=O)NCCC2CN(C(c3c[nH]c(C#N)c3)=O)C2)CC1 N1(C(CC(=C)C)=O)CCN(C(C2(NC(N)=O)CCCCC2)=O)CC1C1CCC1 C1(O)(CN(C(c2c(CCCC)ocn2)=O)C)CCCN(C(=O)C(F)CC)C1 O=C1CCC(C(=O)NCc2ncc(C(=O)N(CCCCO)CCO)cn2)CN1 N1(CC(C)NC(=O)CC2(C)CCN2C(=O)CCN2CCOC2=O)CCOCC1 C1(COCCN(C(=O)Cn2cc(C(F)(F)F)nn2)C)CCCC(CN)C1 CCC(C)C(CNC(=O)CCN(C(=O)CC1CC(=O)NC1=O)C(C)C)CO c1(C(=O)NC(c2ccc(C)cc2)CNC(=O)CC(F)(F)F)c(C)ccnc1C N1(C(c2c(C(C)C)noc2)=O)CCC(C(=O)NCC2CCC(F)C2)CC1 Nc1cc(Cl)nc(Cl)c1C(N1CCOC(CNC(C2CCCCCC2)=O)C1)=O c1(CC(N2CC3(CN(C(=O)CSCC4CCCO4)C3)C2)=O)nc2c([nH]1)CCCC2 c1(NC(C2N(C(c3scc(C)c3Cl)=O)CC(C)C2)=O)ccc2ncn(C)c2c1 n1(CC(C)C)cc(Cc2cc(C(=O)Cc3ccccc3)co2)nn1.C(=O)O C1(CNC(C2C(C(C)C)(CC)C2)=O)CCN(C(C2CC3CC3C2)=O)C1(C)C C1(NC(C2(CC=C)CC2)=O)CC1C1CCCN(C(=O)COc2cncc(C)n2)C1 C1(NC(CCCN(C)C)=O)CC2CC1CN(C(=O)CC1SC3=NCCN3C1=O)C2 c1(SCc2cc(Cl)cc(C)n2)ccc(S(C)(=O)=O)cn1 c1(C(=O)NC2CCC(NC(=O)CCC3CCCO3)CC2)cnn2c1CC(F)(F)C2 C(=O)(C1=CCCCC1)NC(C(=O)NCCC1CCCN(C)C1)CC1CCOCC1 c1(C(=O)NC2COCC2NC(c2cn(CC(F)F)cn2)=O)cc2ncccn2n1 c1(CC(=O)NCC23CC2CN(C(=O)C(F)C(F)(F)F)C3)cccc2ccsc12 C(CCC(=O)NNc1cc(Cl)ccn1)NC(C1(NC(=O)OC(C)(C)C)COC1)=O CC1CN(C(c2nscc2Br)=O)CC1NC(c1cccc(Cl)c1)=O O=C(CCC(=O)c1cccs1)Nc1ccc(Cn2ccnc2)nc1 C=CC(CC)CC(=O)NC(CNC(=O)CCc1cc(C)on1)CO Cc1ccc2c(c1)CCCN2C1CCN(C(=O)C(F)(F)F)C(C)(C)C1 C1(NC(C2OCCN(C)C2)=O)CC2CCC(C1)N2C(=O)CCn1ccnn1 c1(C(N2CCC(C3=NOCC3)C2)C(=O)NCCC2CC2)cccc2cnccc12 N1(C(c2nc(C)sc2C)=O)C(C(=O)NCC2(CO)CC(F)(F)C2)CCC12CC2 Cc1cc(OCC(N2CCN(C3CCCN(C)C3)C(=O)C2)=O)cc(C)c1 Nc1c(C)cc(CNCC(c2ccc(Br)cc2)F)cc1[N+](=O)[O-] c1(C(C)(C)C)cc(=NCCOCCNC(=O)Cc2cccc(Cl)c2F)[nH]c(Cl)n1 CN1CCC(C(=O)NC2CC2C(=O)NC(c2ccccc2)CO)C1 c1(N2CC3OCC(NC(C4C=CCCC4)=O)C3C2)ccc([N+](=O)[O-])cc1Cl CC1(C)CC(C(=O)NC2CN(C(=O)C(C)(F)C(F)(F)F)C2)CC(C)(C)O1 C#Cc1cnc(C(=O)NC2(C(=O)NCCC(C)SC)CCSC2)c(C)c1 c1(C(=O)NCC(C)(C)NC(c2ccc(F)cc2F)=O)c[nH]cc(Br)c1=N c1(NCC(CNC(Cc2nc(CC)sc2)=O)O)nc(C(F)(F)F)cc(C)n1 N1(C(CNC(C)C)=O)CC2CC1CC2NC(c1ccccc1C(F)(F)F)=O N1(C(C2C(C)(C)C2)=O)CCC2CCC(NC(c3conc3C(F)(F)F)=O)C12 c1(OCC(N2CCC(NC(C(C)=C3CCCC3)=O)C2)=O)cc(C)ccc1Cl N1(C(C(C)OCC#C)=O)CC(CO)C2(C1)CN(C(c1ccn3cncc3c1)=O)C2 CCCC(C(=O)NOCCC(F)F)NC(=O)C=CC(=O)N(C)C Cc1nc(C(=O)NCC2CCN2C(c2ccc3c(n2)CCO3)=O)ccc1C#N C1(F)(CNC(CC2C(CC)C2)=O)CCN(C(=O)CCC(=O)c2ccc[nH]2)C1 c1(-c2ccc(C(N(C(CCC(=C)Br)=O)CC)=O)o2)ccc2c(c1)OCO2 N1(C2CCN(C(CC=C)=O)C2)CCC(NC(=O)C=Cc2nccs2)CC1 c1(C(N2C(C(=O)Nc3ncc(O)cc3Cl)CC(C)C2)=O)ccc2cnccc2c1 N1(C(C2CN(C)C2)=O)C2CCC1C(CO)N(C(c1ccc(C3CCOC3)s1)=O)C2 C1(NC(C2(C=C)CCOCC2)=O)CCC2(CC1)CN(C(=O)CCCCCCC)C2 C1(CC)CN(C(=O)C(F)=C(C)C)CCN1C(=O)N=CC1CCC(C)(C)C1 N1(C(c2c(Cl)cn(CC)n2)=O)CCN(C(C2CC2F)=O)C2COCC12 N1(C(c2c(C)sc(O)n2)=O)CCC2CCN(C(C3CN(C)CC(C)O3)=O)CC12 C1(C(=O)NC(CC=C)(C)C)(CC=C)CN(C(=O)CCCNC(C)=O)C1 C(C)(C(C)(C)C(=O)N1CC2(CC2C(=O)OC)C1)NC(c1c(C)snc1)=O Cc1cc(C(=O)NC2CC(NC(c3cnn(C(C)C)n3)=O)C2)c2c(n1)CCCC2 c1(OC)ccc(NC(C2CCN2C(c2ccc(CO)cc2OC)=O)=O)c(OC)n1 c1(C(N2C3CN(C(CCc4ccc(C)s4)=O)CC32)=O)cccc(F)c1C c1(C(=O)NCCCC2(NC(C(C)SC(C)C)=O)CC2)cc(C2CC2)nnc1O N1(C(=O)C(F)CC2CNC2)CCCC(CC2CC2)CC1 Cc1cc(C(N2CCN(C(=O)CC3CCNC(=O)C3)CC2CF)=O)nc(O)c1 c1(OC)cccc(CN2CCCCC2=O)c1.n1(CC(=O)NCCOC)cc(CN)nn1 C1(CNC(CC(C=C)C)=O)CN(C(C2CN3CCN2CC3)=O)C2(CCC2)C1 N1(C(CC(C)OC)=O)CC2(C1)CCCN(C(c1cnc(Cl)cc1N)=O)CC2CO CN(C1CCCc2nc[nH]c21)CCn1cnc2c1CCCC2 c1(OC)ccc(-n2cc(C3C(C)CCN3C(=O)C(F)(F)C3CC3)nn2)c(F)c1 c1(CN2C(CNC(C(C)Cc3ccccn3)=O)CC2)cc(Cl)ccc1F c1(CC(N2C(C)(CC)CC(NC(C3OCCO3)=O)C2)=O)cccc2ccncc12 c1(C(=O)NCC#CC(=O)OC)cnn2c(C(F)(F)F)cc(C)nc12 CC(=O)CCCCCCC(=O)N1CCCC(CNC(=O)C(C)C2CCC2)C1 n1(C(CC)(C)C)nnnc1C(CC)NC(c1ncc[nH]1)C1(c2cccs2)CC1 C(C)(CNC(=O)Cc1sc(C2CC2)nc1C)(C(C)C)NC(C1C(C=C)C1)=O C(CC(=O)N(CC(=O)NC(C)CO)C)OCC CC1CCN(C(C2(C3CCCO3)CC2)=O)C(C)C1NC(c1ccc(O)nc1)=O C1(C(=O)NCCCN(S(C)(=O)=O)C)CC12CCN(C(C1(CO)CC(C)(C)C1)=O)C2 N1(C(C(C)OC)=O)CCC(C(=O)NC2(CO)CCCCC2)C(O)C1 C1(C(N(C)CC2(CO)CCCO2)=O)CCC2(CCC2)CO1.C12CC(C1)NC(=O)C2 C1(S(C)(=O)=O)(C(=O)NCC2N(C(c3cc(SC)oc3)=O)CC=C2)CCC1 N1(C(Cc2cnn(C)n2)=O)CC2CC(NC(c3cc(F)c(F)c(F)c3)=O)CC2C1 C1(NC(c2sccc2Cl)=O)CC2CN(C(=O)CC3Cc4ccccc4N3)CC2C1 c1(C(=O)NCCCCC2CN(C(c3n(C)nnc3)=O)C2)ccc(C2CC2)cc1 C(c1cccc(F)c1)=CC(=O)NCC1CC2(CC2)CN1C(=O)C(O)C(F)F c1(CNC(N2CC(NC(=O)CCC=CBr)C2)=O)ccc(Br)cc1O S(=O)(=O)(c1ccc(CNC(c2cnc(C)nc2OC)=O)s1)NC c1(C(=O)NC2CC3CC(NC(=O)Cc4ccon4)CC32)ncc2n1CCCC2 c1(C(=O)NCc2cnc(CC)[nH]2)ccc(N)c(Cl)c1 c1(CC)ccc(=NCc2ccc(OC(=O)NCC)cc2)[nH]c1 c1(C(N2CCC(C(C)NC(c3coc(C(F)F)n3)=O)CC2)=O)cc(F)ccc1F N1(C(COCC#C)=O)Cc2n[nH]cc2C1C(=O)NCCN1CCC2CC12 N1(C(Cn2ccc(C)n2)=O)CCOCC1CNC(=O)CCc1cnn[nH]1 N1(C(c2occc2Br)=O)CCC2(CCCC2C(N2CC3CCC(C2)O3)=O)C1 C1(n2cc(CCCC)nn2)CC2CCC1(NC(=O)C=CCF)C2 S(=O)(=O)(c1cccc(Br)c1)NC(C1CCC(C)(C)CC1)C c1(C(=O)NCC2(NC(C3CC(C)SCC3)=O)CC2)cc(F)c2cn[nH]c2c1 c1(NC(C2C(NC(C3(CCCC)CC3)=O)CCO2)=O)ccc2nc[nH]c2c1 C(=O)(C1=CCCOC1)NC1(CCNC(C(c2cccc(F)c2)C)=O)CCC1 N#Cc1ccc(CNC(=O)C=C2CCN(C(c3sccc3F)=O)CC2)cc1 C1(CNC(CCn2c(C)nc(C)n2)=O)CN(C(C2CCCOC2)=O)CC1(F)F C12(C(=O)NCCCC)CC(CO)(CN1C(C1(C)CCCCC1)=O)C2 c1(CN(C(=O)Cn2cccn2)C)cccc(-c2cccnc2)c1F C#Cc1ccc(CN(C(C(CC(C)C)ONC(=O)C2(CO)CC2)=O)C)nc1 CCC(C)C(C)C(=O)NCCCCCCN(C(=O)CCc1ncco1)C C(=O)(C1COc2ccccc21)N1CCN(C2CC3(OC(C)C(=O)O3)C2)CC1 c1(C(=O)NCC(CNC(c2ccccc2)=O)F)cnc(O)n(C2CC2)c1=O c1(C2N(C(=O)NCC3CCCCO3)CCC2)cccc(Br)c1 Cc1ccc(Cl)c(F)c1C(=O)NC(C)CCNC(C1(O)CCSCC1)=O C1(CNC(C=C(CC)C)=O)COC(COC(C)(C)CNC(=O)C(C)(C)C)C1 C1(C(=O)NC(c2ccc(F)c(F)c2)CC(F)(F)F)CNC2CCCCC2C1 Cc1cc(F)cc(Br)c1C(N1CC(CNC(=O)C(C)n2ccnn2)C1)=O C1(C)(CC(=O)NCC(CNC(CC(C)N(C)C)=O)CO)CCOCC1 c1(C(=O)NCC2N(C(C3(C)CC4(CC4)C3)=O)CC2)cnc2ccsc2c1 C1(NC(c2c(CC)nn[nH]2)=O)CC2CC(NC(=O)CN3C(C)CCC3C)CC12 C(=O)(CC(C)C(F)F)NCNC(C(C1CCC(C(F)(F)F)CC1)N1CC(OC)C1)=O N1(C(CCC(C)C)=O)CCc2cc(F)ccc21.c1(-n2ccnn2)cnccc1C C12(NC(CN=S(C)(C)=O)=O)CCCC1CN(C(c1cc3ncccc3[nH]1)=O)C2 CCC(C)(CC)C(=O)NC1C=CCN(C(=O)CCc2ccc[nH]2)C1 Cc1ccoc1NC(=O)C(=O)NC(C)(CNC(C1COCCO1)=O)Cn1cccn1 C(CC(=O)N1CCCC1CC(C)C)(C(F)F)NC(c1ccc(CC)[nH]1)=O C1(CC(=O)NC(C2CC(NC(C(C)SC(F)(F)F)=O)C2)C)CCC2(CC1)CC2 C1(OC)CC(CNC(c2cncc(F)c2)=O)N(C(c2ccnc(S)c2)=O)C1 c1(NC(N(C)C(c2ccccc2)c2ncc[nH]2)=O)ncc(I)c2c(Br)cn(C)c12 c1(C(=O)NCCCN(C(=O)CC2CCC(C)(C)CC2)CC)ccc2sncc2c1 C=Cn1nncc1C(=O)NC(C)C(C)C(=O)N1CC(O)CC1CO C1(NC(=NC)NCC(c2ccc(C)c(C)c2Cl)OC)CCn2ccnc2C1 C1(CCC(=O)N(CC#C)CC2CC2)CCCCN1C(c1nccn1CC)=O c1(CN2CCN(CC(=O)OC)CC2)ccc2[nH]c(C)c(C)c2c1 c1(C(=O)NC2CC(c3ccccc3)(CNC(C)=O)C2)cn2ccc(CO)cc2n1 CC1(C(N2CCCC(NC(c3ccc(C#N)o3)=O)CC2)=O)CC2CCC1C2 C(C(O)CC(=O)NCCc1ccncn1)NC(C(C)N1CCCC1)=O N1(S(=O)(=O)CCCCl)CC2CCC1CN2Cc1ncccc1C(=O)O c1(C(=O)NC(CC(C)C)CNC(C2COCC2(C)C)=O)ncn2c1CCCCC2 c1(C(=O)NC(C)CCNC(c2cnn(C3CC3(F)F)c2)=O)ccncc1Cl CCC(C(=O)NCCCN(C)C(C1CCOC1C1CC1)=O)N(C)C1CC1 N1(C(Cc2c(C)ncs2)=O)CCC(F)(CNC(=O)C(N)=O)C1 C12(C(=O)NCC3(CCNC(COCCCC)=O)CC3)CCC(O)(CC1)CC2.COC CC(C)(CC#N)NC(c1conc1CNC(c1ccsc1)=O)=O O=C(O)CCCNC(c1cnc(C2CCC2)s1)c1nnnn1C1CCOC1 C1(C(=O)NC(C2CC(F)CN2C(=O)Cc2ccoc2)C)CCC(C)(C)CC1 c1(OCC(=O)NC(CC)CNC(C2(CCN(C)C)CC2)=O)ccc(C)cc1C N1(C(c2cc(C)no2)=O)CC(C2(NC(c3cc(Cl)ccc3N)=O)CC2)C1 C#Cc1cccc(C(N2CC(NC(=O)CCNC(=O)OC)CC(O)C2)=O)c1F n1(CCC(=O)NCC(CN(C(=O)CN(C)C2CC2)C)(C)C)cnc2ccccc12 C1(CNC(c2c(Cl)ncc(C)c2)=O)CCC2CN(C(=O)CC(C)(F)F)CCC2C1 c1(C(=O)OC)ccc(Cl)c(OCCNC(=O)Nc2nccn2-c2ccccc2)c1 c1(C(=O)NC(C(C)NC(c2nc(COCC)sc2)=O)C)cnc2ccnn2c1C C(=O)(C(C)S(C)(=O)=O)N1CC(C)C(CCNC(c2ccc(=N)[nH]c2)=O)C1 C1(C(=O)NCCN=[N+]=[N-])CCOCC1NC(C1(O)CC1)=O c1(OCC(=O)NC2OCC(CNC(CCC(=O)NC)=O)C2)cc(F)cc(Cl)c1 N1(C(C(C)NC(C)=O)=O)CC(=O)NCC1C(=O)NC(c1ncnn1C)C N1(C(C(CCC)NC(=O)NCCC(=O)OC(C)(C)C)=O)CCCC(O)C1CC C(C(CC(=O)NC1(C(C)C)CC1)OC)NC(CCN(C)CC)=O CC(C)CCCCCC(=O)N1CC2(C1)CN(C(=O)Cc1ccsc1)C2 Nc1cc(C(N2CC(NC(=O)CC(=O)NCC3CC3)C2)=O)ccc1S(N)(=O)=O C1(NC(C2N(C(C3(C(=O)OC)CC3)=O)CCCC2)=O)COCCN(C)C1 CCCCC(C)(F)C(=O)N1CC(OC)C(NC(c2ncoc2Br)=O)C1 C(=O)(CCCC(C)(F)F)NC(C1CCCC1)CNC(C(COC)OC)=O CCC(C(=O)NCC(F)CNC(=O)CSSC(F)F)NC(=O)OC(C)(C)C c1(NC(C23C(CN(c4cc(COC)ncn4)C2)C3)=O)ccc(C(F)(F)F)c(F)c1 CCC(C)CCC(=O)NC(CO)CCCNC(c1nc(Cl)ccc1N)=O C1(C(=O)NC2C(NC(CC3CN(C)C3)=O)COC2)CCC(F)(F)CO1 c1(C(=O)NC(CNC(C(C)NC(c2ccco2)=O)=O)C)ncncc1Br C(=O)(CC(C)CNC(c1cc(C2CC2)[nH]n1)=O)N(CC)Cc1ccncc1 C12(CNC(C(=O)NCC)=O)CC1CN(C(=O)C(c1ccccc1C)(C)C)C2 C1(C(=O)NCC(CCOC)NC(C(CC#C)C)=O)CC2CCCC(C1)C2 C(CCCCC(=O)NC(C)CCCNC(=O)C(C1CC(F)(F)C1)O)SC C(CC(C)(C)CC=O)OC.C1(NC=O)CCC(Cn2cc(CN)nn2)C1 c1(C(=O)NC2CCN(C(C(C)Cc3ccc(F)cc3)=O)C2)cccc2ccoc12 C1(NC(c2c(C)nsc2)=O)CC2CCC(C1)N2C(=O)CCCc1nccs1 CC1(C)NC(=O)N(CC(=O)NC2(C)CCCN(c3nnn(O)n3)C2)C1=O c1(CNc2cccc(NCc3c(O)nccc3)c2)ccn2ccnc2c1 c1(NC(CNC(=NC)NCCSc2ccco2)=O)ccc(Cl)cc1 c1(OC)ccnc(C(=O)N(CC(C)CNC(=O)CCN2CCOCC2=O)C)c1F C1(C(=O)NCC2CN(C(=O)C=Cc3cccnc3)C3CC23)(COC)CCCCC1 C1(CC)CCN(C(=NCC(C2CC2)OCc2cc(C)no2)NC(C)C)C1 c1(C(=O)NCC2(F)CC(NC(C(C)C3CCCC3)=O)C2)cccc2c1CCO2 c1(C(N2CCN(C(c3ccncn3)=O)CC2CO)=O)cccc2cncn12 CC1CCC(N)(C(N2CCCC2c2nccs2)=O)C1 C=CCC(CC=C)C(=O)NC(C)CN(C)C(C1CCC(NC(C)=O)CC1)=O C1(C(=O)NCCC(=O)NC2CCCC(NC(CSC)=O)C2)CCc2n[nH]cc2C1 C12(CNCC3CCN(CC(C)C)C3)CCC1CCCN2 C1C(N2CCCC2CC(=O)OCC)C(=O)N1.C1(CC)CC(SC)C1 c1(CNC(C2CC=CCC2NCCN2CCCC2)=O)nc2ccccc2[nH]1 CC#CCCCC(=O)NC(c1cccnc1)CCC1CCC1 CCCC(C(=O)NC1CN(C(c2ccc(F)s2)=O)CC1c1cnn(C)c1)C(C)C c1(CC)c[nH]c(C(=O)NCC2CCCC2NC(c2cc(C(N)=O)c[nH]2)=O)c1 c1(C(=O)NC2CCC2NC(C2CCOC2)=O)cc([N+](=O)[O-])c2nsnc2c1 C(=O)(CCS(N)(=O)=O)N1CCC(CC(=O)N(C2CCCOC2)CC)(OC)C1 c1(NC(c2cc(C)n(-c3ccc(Cl)cc3)n2)=O)cc(NC(N)=O)ccc1F N1(C(C(=O)Cc2ccc(O)cc2)=O)CC2CN(C(C3CCCC34CC4)=O)CC2C1 Cc1cc(C(c2nnnn2C(C)C)NC(C)C(c2ccccc2)C)cc2ccoc12 N1(Cc2cc(OC)no2)CCC(NC(c2cccc(-n3cccn3)c2)=O)C(C)(C)C1 C(=O)(CC(O)C(C)CC)N(C1CCN(C(c2cnc(OC)nc2)=O)CC1)CCC CN1CCCCC(C(=O)N(C)CC2CCCC2NC(=O)CC(F)(F)C(F)F)C1=O c1(CC)[nH]nc(C(N2CCC2C(N2CCN(c3ncccn3)CC2)=O)=O)c1F c1(C(N2CCCC(NC(c3cc(CC)ncn3)=O)C2)=O)ncc([N+](=O)[O-])cc1C C1(CN(C(=O)NC2(Cc3ccccc3F)CC2)CC)CCN(S(=O)(=O)CC)CC1 N1(C(C(C)(C)CCCO)=O)CCC2(C1)CN(C(C1(C)CCCCO1)=O)CCO2 C1(CNC(C=CCC)=O)CCOC1C(=O)NC1CCC(C(F)(F)F)C1 C(=O)(C(C)(F)C(=O)NCC(F)CNC(c1c(Cl)cccc1Br)=O)OC CC(C)CC(C)(C)C(=O)NCCOC1CN(C(C2CCCOCC2)=O)C1 c1(-c2n(CC)nc(C)c2)ccc2[nH]cc(C(N3CCN(C(C)=O)CC3)=O)c2c1 c1(OCCCC)ccc(NC(=O)NCC2CC(OC)C2(C)C)cc1 C1(NC(CN(CCC#C)C)=O)CCCC(CN(C(=O)Cc2cscn2)C)C1 N1(C(C(C)n2cnnn2)=O)CCC(NC(=O)C2=CCCC2)CC1C c1(C(N(CC(C)CNC(c2ccn(CCC(F)(F)F)n2)=O)C)=O)ccc(Cl)cn1 c1(NC(C2(NC(C3=C(C)OCC3)=O)CCSC2)=O)cccn2nccc12 CC12CCC(C(N3CCN(CCNC(C4CCCC(=O)N4)=O)CC3)=O)(CO1)C2 C#CC1CCCN(C(C2CC2C(=O)OC)=O)C1.c12nc(cc(O)n1)NC2 Cc1ccc(C(N2CC(N(C(=O)C3=CC(C)(C)C3)C)C(F)C2)=O)nc1C c1(NC(C)=O)ccccc1C(=O)N(SC(CCCCNC(c1cscn1)=O)C)CC C#CCC(CC#C)C(=O)NC1CC2CCC(C1)N2C(c1ccc2nn[nH]c2c1)=O CCCCC(CC)CC(C(=O)Nc1ccccc1OC)N(C)CC1CCCSC1 c1(C(=O)NCC2CC2CNC(C2C3CCC2CC3)=O)ncnc(O)c1Br C1(CNC(CSC(C)C)=O)CN(C(C2(C)COC(=O)C2)=O)CCO1 CC(=O)CCCC(=O)NCCN(C1CCCCCC1)C(C1CC2(CC(=O)N2)C1)=O c1(C(=O)NCCN2CC(CC(=O)NCCCO)C2)ccc2ocnc2c1 C(=O)(CCCC(F)(F)F)N1CC(NC(=O)C(=Cc2c[nH]cn2)F)C(O)C1 Cc1ccc(C2CC2C(=O)NC2(CNC(c3cnc(C)s3)=O)CC2)c(C)c1 C1(C(N2C3CC(CN(C(Cc4ccc(C)o4)=O)C3)C2)=O)CCc2cnn(C)c2C1 c1(CCNC(=O)Nc2nc(C)c(C#N)s2)ccc([N+](=O)[O-])cc1Br C12(CNC(CC3(N(C)C)CC3)=O)CCC(NC(=O)C(O)C(F)(F)F)(CC1)C2 N1(C(c2cnc(C)[nH]2)=O)CCC(C)C(NC(C23C4CC(CC24)C3(F)F)=O)C1C CC#CCN=c1[nH]c2c(c(=NC(Cc3ccccc3)CCO)[nH]1)COCC2 C1(N(C)C(C2CC(O)C2)=O)CCCC(NC(c2cc(-c3ccco3)no2)=O)C1 c1(C(=O)NCC(C)OC)ccc(CO)cc1.C1(=O)C(C)OCCN1.C1(NC)CC1 c1(C(N(C2CCN(C(c3ccc(C)s3)=O)C2)CCO)=O)cccc2[nH]ncc12 C(=O)(C1=CS(=O)(=O)CCC1)NCC(C)NC(=O)CC1CCC1(C)C N#CCCCC(=O)N1CCCC1C=CC(=O)NC1(c2nn[nH]n2)CC1 CCCCCCCC(O)CC(=O)N1CCC(O)C(O)C1 N1(C(C(CSC)O)=O)CC2CC1CN2C(c1nc(-c2cnn(C)c2)oc1C)=O C12(CNC(CCOC)=O)CC(NC(C3(CO)CC3(F)F)=O)C(CO1)C2 N1(CC(=O)N(C(=O)C(N)Cc2cccs2)CCSC)CCN(C)CC1.CC c1(NC(C2C(O)CCN2Cc2ccc(F)c(O)c2)=O)c(O)cccc1O N1(C(c2c(C)cn(C)n2)=O)CCC(C(=O)NCC(C)(O)C(F)F)CC1C(C)C N1(C(c2c(N)sc(C)c2C)=O)CCCC2(CC(NC(C3CC3C(F)F)=O)C2)C1 C(C1(C)COC1)=CC(=O)NCCCN(C(C1(OC)CCC1)=O)CC C(=O)(CCCCCCC(=O)NC1(CNC(=O)Cc2ccoc2)CCOCC1)OC N1(C(C2(CCC=C)CCCC2)=O)CC2CC(NC(=O)CS(=O)(=O)CC)CC1C2 N(C1CCc2c(Br)ccc(Cl)c21)CCC1N(C(=O)OC(C)(C)C)CCCC1 CC1CN(C(=O)CN2CC(=O)NC2=O)CCC1N=c1ccnc(C2CCCC2)[nH]1 N1(C(c2sccc2Br)C(=O)NCCC2CC2)CCCC2(CC(O)C2)C1 CCC(C)C(C)C(=O)NC1(CNC(=O)Cc2cc(C)cc(Br)c2)CCC1 C12CCN(C1)C(=O)N2.C(=O)(CC(C)C)N(CC(=O)OCC)CCC c1(CC(N2CCC(CCNC(=O)C(O)C3CC3)C2)=O)c[nH]c2ccccc2c1=O N1(CC(N2CC(O)(CCNC(C(C)C(F)(F)F)=O)C2)=O)Cc2ccccc2C1 n1(CC(=O)NCCC(C)NC(=O)CCc2ccc(O)nc2)ncc2cccnc12 C1(O)(CN(C)C(C2(C3CCCO3)CC2)=O)CCN(C(c2cnn(CCO)c2)=O)C1 c1(CC)c(C(=O)NCC2(F)CC(NC(c3cc(C)nn3CC)=O)C2)cnn1C c1(CC(N2C3C(NC(C(C)SC(C)C)=O)C(C3)C2)=O)ccc2[nH]ccc2c1 N1(C(c2c3ccc(OC)cc3[nH]n2)=O)CCC2CN(C(=O)C(C)N(C)C)CC2C1 C#CCC(CC(F)F)C(=O)N1CCC(C)(CCNC(=O)CCCn2cncn2)C1 C(C(C)(C)C(=O)NC(C)CNC(=O)C(C(C)C)SCc1ccccc1)SC c1(CC(=O)NC2C3(CCN(C(CSCCC#N)=O)C3)C2)ccc2cccnc2c1 c1(N(C2CCN(C(c3ccc(=O)oc3)=O)C2)C)nc2cc(F)ccc2o1 C1(NC(c2cc(O)ncn2)=O)CN(C(c2scc3c2CCCC3)=O)CC2(CC2)C1 C12(CNC(c3cnc(C)[nH]3)c3nnnn3C3CCCCC3)CC(C)(CCO1)C2 CC1CCN(C(c2cc3n(n2)CCC3)=O)C(CNC(=O)CCS(C)=O)C1 Cc1ccc(C(=O)NCCN(C(=O)C(C)N2CC(C)C2)C2CC2)c(Cl)c1Cl Cc1cc(Br)ccc1C(C)NC(=O)C(=O)NC1CNCCC1C c12cc(C)ccc1c2=O.c1(C(N(CC(=O)NC)CC#C)=O)cc(OC)no1.OCC C1(C(=O)NCC(C)CN(C)C)CN(C(=O)CCCNC(=O)CO)CCC1(C)C CCC(CC)C(CCNC(=O)C(N1CCN(C)C(COC)C1)=O)OC c1(C(=O)NC2(CNC(=O)C=Cc3nccs3)CCCC2)ccc2c(c1)CC2 CC1(C)CC(NC(=O)CN2OC(C)(C)CC2=O)CN(C(=O)CC#N)C1 c1(C(=O)NCC2(F)CC(NC(C(CCSC)O)=O)C2)cccc2c1OC(C)C2 N1(C(c2cc(CSCC)on2)=O)CCN(C(c2ccc(Cl)o2)=O)CC12CCC2 c1(C)ccccc1OC.c1(OC)cccc(NC(=O)NC2(CNc3ccns3)CC2)c1 C(=O)(CCC(C)(C)F)NC(C(=O)NCCC1(COC)CC1)CCC1CCC1 CC1(CNC(N2CC(Cn3cccn3)C2)=O)CCOC1C1CC1 CCC1=C(C(=O)NCC(C2CC2)NC(C2CC(C)(C)CO2)=O)CCCO1 C1(NC(c2c(CC)nccn2)=O)CCC2(CCN(C(=O)Cc3nncn3C)C2)C1 c1(C(=O)NCCC2CC(NC(c3ccc(C#C)nc3)=O)C2)ccn2cnnc2c1 c1(C(CNC(C(CC)C)=O)NC(=O)CC(=O)N(C)C)cccc(C)c1 Cc1cnc(NCc2nonc2C)c(S(=O)(=O)NC2CCCC(C)(C)C2)c1 C(=O)(C(C(C)CC)NC(c1cn(C)c(=O)n1C)=O)NC(CC(=O)OCC)C N1(C(CCC2(C)N=N2)=O)CC2CC2C1C(N1CCC(NC(=O)C2CC2)C1)=O O=C(C#CC1CCCO1)NCC1=CCN(C(c2ccc(O)cc2F)=O)CC1 c1(C(N(C)CC2CCCC(NC(C(F)=CCC)=O)C2)=O)cc(F)c(F)cc1O c1(C(=O)NC2C3(NC(CC=CC)=O)CCC(C2)C3)cc(Cl)c(F)cc1O C(=O)(C(F)C(=O)NCCCNC(=O)COC1CCOCC1)OCC C1(C(C)(C)C)CN(C(c2cn(C3CC3)nn2)C(=O)NCC2(C)CC2)CC12CC2 C1(C(=O)NCC2(NC(CC(C(C)C)O)=O)CC2)Oc2ccccc2OC1C C(=O)(C1=NOC2(CCOC2)C1)N1C(C)CN(C(=O)COC2CCOCC2)CC1 N1(C(CN(C(C)C)C)=O)CC2(NC(=O)C(C)C3CC3)CCC1CC2 CC1=C(C(=O)N2CCN(C(=O)CCc3c(C)noc3C)CC3CC23)CCCC1 C(=O)(C1CCCc2nccn21)NCC1=CCN(C(C2CCCN(C(C)=O)C2)=O)CC1 C1(CNCC(=O)OC(c2cn(CCOCC)nc2)=O)CN2CCC1C2.C C(CCCCCN=[N+]=[N-])NC(C(CCOCCO)NC(Cc1c(C)ncs1)=O)=O c1(C2C(C(=O)NCC(C)NC(=O)C(C)N3CC(C)C3)CCC2)cc(Cl)cc(Cl)c1 C1(N(C(=O)Cc2ccccc2F)C)CN(C(C2(C(C)(C)C)CCC2)=O)CC12CC2 N1(C(C2C(C)C2)=O)CCOCC1CNCc1ccnn1CC(=O)O C=C(C)CCC(=O)NCCCOC1CCN(C(c2c(C)csc2Cl)=O)CC1 CN1C(=O)NCC1CNC1CC(C(=O)Nc2cccn2-c2ccccc2)C1 c1(-n2ncc(NC(=O)NC(c3cnc(Cl)s3)CC)c2)cccc(O)c1 S(=O)(=O)(c1cc(NC2CCCC2)ccc1C)NC(C(c1ccc(F)cc1)OC)C C1(NC(C2ON=C(CC)C2)=O)CCN(C(=O)Cc2ccc(Cl)s2)CC1CO N1(C(c2c(Cl)c(C)n(C)n2)C(=O)NCc2cccs2)CCC2CN(C)CC12 N1(C(C(=Cc2cnc[nH]2)C)=O)CCC(CN(C)C(C2CCC(C)O2)=O)CC1 CCC1=NOC(C(=O)NCc2c[nH]nc2C(=O)NC(c2cnn[nH]2)(C)C)C1 c1(C(=O)NCC(CNC(C(C)CC(N)=O)=O)C)ccc(O)c2ncccc12 CC1(C)C2CCC1(CC(N1CCOC3CCC13)C(=O)NC1CC1)CC2 C(=O)(C#CC1(CC)CC1)N1C(C(CNC(CC(=C)C)=O)(C)C)CCC1 N(C(=NCCCCCCO)NCC1CCCO1)C1C(C(C)(C)O)C1 c1(C(=O)NC2CCN(C(c3cccnc3Cl)=O)CC2F)cnc2cc[nH]c2c1 Cc1nc2c(NC3CCC3NC(=O)CCN(CC(F)(F)F)C)ncnc2s1 c1(C2(C(=O)NC3CC(CNC(C(CC=C)NC(C)=O)=O)C3)CC2)ccc(C)cc1F C#Cc1cnn(CC(N2CCN(CCNCC3CC(CF)C3)CC2)=O)c1.C(NC)C Cc1nc(C)n(O)c1C(=O)NCC1(O)CCN(C(c2cn(C)ccc2=O)=O)C1 C1(NC(C(SC)SC)=O)CCN(C(c2ccc(NC(C)=O)cc2Cl)=O)CC1CO c1(C(N2CC(=CC)C2)=O)ccoc1CNC(=O)C(C)C1CC1 N1(C(C(CC)OC)=O)CCC2(CCC(NC(c3ccc(CO)o3)=O)C2)CC1 Cc1nnc(CC(=O)NC(C2CN(C(=O)C(C)(C)C3CCCO3)C2)C)s1 N1(C(c2cnc(SC)nc2)=O)CCCC(C(N2CCCC(C(N)=O)C2)=O)CC1 c1(NC(CCC=C)C)ncc(C)cc1S(=O)(=O)NCc1snnc1C C1(CNC(CC2CC(C)C2)=O)(CNC(=O)CCc2cccn2C)CCOCC1 N1(C(C2N(C(CC(C)(C)O)=O)CCSC2)=O)CCCC(O)(C(N)=O)C1 N1(C(CC2CC(SC)C2)=O)CCCN(CCNC(=O)C(F)CC2CCCC2)CC1 C(=O)(C1CCSc2ccccc21)N1C(C)CN(C(c2cc[n+]([O-])cc2)=O)CC1 N1(C(C2CCc3nncn3C2)=O)Cc2c(Br)cccc2C2(CCC2)C1 N1(C(COCC(=O)NC)=O)CC2CC1C2C(=O)N(C1CCOC1C)C N1(C(C2(CC=C)COC2)=O)CCCCC(CNC(=O)CCN(CC(F)(F)F)C)C1 c1(SC)nc(=NC2CCN(C(=O)CCN(C)C)CC23CCC3)c(C#N)c[nH]1 Cc1ccc(C)c(C(=O)NC2CC3c4ccccc4C23)n1 n1(CCOC)c(O)nc(NC2CC(CCNC(c3cscc3OC)=O)C2)cc1=O CC(C)CCC(F)C(=O)NC1CCCC1NC(c1ccc2c[nH]nc2n1)=O C1(CNC(C(CC)(C)C)=O)N(C(c2cnc3n2CCS3)=O)CCC1(C)C CCC(C(=O)NCC1CN(C(=O)C(N2CCC(C)C2)c2cccs2)C1)n1cncn1 c1(CC(=O)NCC(C)N(C)C(c2ccnc(S)c2)=O)nc2ncccn2n1 S(=O)(=O)(c1ccc(C(=O)NC2CC2CNC(C2CC3(CSC3)C2)=O)cc1)NC CCC(C)(C)CCCC(=O)NC1CN(C(c2cc3cncc(C)c3s2)=O)CC1O c1(N(C)C)ccc(C(N2CCC(N3CCCNC3=O)CC2)C(=O)NC2CC2)cn1 CCCC(C(=O)N1CC(NC(C2CC(CC3CC3)C2)=O)C(O)C1)OC N1(C(=O)OC(C)(C)C)CCCC(O)(C(N2CCC(OCS(=O)(=O)C3CC3)C2)=O)C1 C=CCC(C)C(=O)NC(C)(CNC(c1onc(N(C)C)c1Br)=O)CO N1(C(C2CCN(CC)C2)=O)CCN(C)C(C(N2CCC(COC(C)=O)C2)=O)C1 Cn1nnc2c1CCC(C(=O)NCC1(C)CN(C(c3n[nH]cc3Cl)=O)CCO1)C2 C12(CCCC(=O)NCC3(C(C)NC(=O)C4=CCCC4)CC3)CC3CC(CC(C3)C1)C2 c1(OC)cccc(CC(=O)NC(CNC(=O)CCCc2cccs2)C(C)C)c1Cl CCCC(F)(F)C(=O)N1CC(CNC(C2CC2(C)CC)=O)(OC)C1 N1(C(C2C(OCC)C2)=O)CCC(C2(NC(C3CCOC3)=O)CC2)CC1 c1(C2(C(=O)NCC3C(NC(CC(=C)C)=O)CC3)CC2)ccc(C(F)(F)F)cc1 N1(C(C(C)c2ncco2)=O)CC(NC(C2(C(C)(C)C)CCCCC2)=O)CC1(C)C C(=O)(C(F)(F)C(F)(F)F)NCC1(O)CCN(C(C23CC(CC(F)F)(CO2)C3)=O)C1 C1(C(N2CCC(C(C)NC(c3cnc4n3CCC4)=O)C2)=O)CCCCC1C1CC1 c1(OC)ccc(C)c(NC(c2sccc2CNC(C2C3CC4C(C3)C24)=O)=O)c1 CCCCCC(C)CC(=O)N(CCC(=O)NC(CN1CCCC1)CO)CC C(CO)(CCCCNC(c1ncc(C)cc1OC)=O)NC(CSCCOC)=O c1(OC)ccc(C=CC(=O)NC2CC(NC(C3COCCC3C)=O)C2)nc1 CCCC(CC)C(=O)NCCCNC(C12CC(F)(C1)C2)=O CC(C)(CNC(=O)CC1CC2(CC2)CO1)CC(=O)N1CC=CC1C(N)=O Cc1cc(NC(c2ccc(Br)cc2CN2CCCC2)=O)c(Cl)cc1Cl c1(C(=O)NC2C(CNC(CCOCC)=O)COC2)ccccc1CC1CCC1 CC1CN(C(c2cccc(N)c2)=O)CCCN1C(C1CCCC1C)=O c1(CC(=O)NCC2CC2CNC(=O)COC2CCCC2)cnc2n1CCOC2 c1(OC)cc(C)c2cc(C(=O)OCCC3(C)CCN(C(=O)C(C)O)C3)[nH]c2c1 C(=O)(C1Cc2ccc(F)cc21)NCC1CC(NC(=O)CCn2cccnc2=O)C1 c12ccc(o1)C=CC(=O)NCC1CC1NC2=O.c1(NCC2C(C)C2)n[nH]c(O)n1 Cc1cc(F)ccc1C(c1nnnn1CC(F)F)NCCC(C1CC1)C1CC1 C(CCC(C)CC(=O)N(CC(=O)NC1CN(c2ncccn2)C1)C1CC1)=C(CC)C CCS(=O)(=O)c1ccc(CC(=O)N(C)CC2CCCN2S(C)(=O)=O)cc1 N1(Cc2cccc(OC)n2)CC2CC1CN2C(c1cc(Br)ccc1Cl)=O C1(NC(c2cncc(C)n2)=O)CCSC12CN(C(c1conc1C1CCC1)=O)C2 CCC(CC)CCCC(=O)N1CC(NC(=O)C(Cl)=CCl)CC1(CC)CC C(C)(C)(C(C)NC(=O)CCOCCN(C(=O)CC12CCCC1C2)C)OC c1(C(=O)NC(CC)(CNC(C2C3CCCC23)=O)CC)[nH]c2ccc(F)cc2c1Cl CCC(CC)CCCC(=O)NCC#CCNC(C1CC2(C1)CC(CO)C2)=O C1(C(=O)NCc2c(C(=O)NC(CCC=C)C)con2)CCCC(=O)N1C c1(C(C(=O)NCSc2ccccc2)NC(C)(C)CC(C)C(C)(C)C)csc(C)c1C c1(C(=O)NCC(CN(C)C(C2(C#N)CCCO2)=O)O)cc[n+]([O-])cc1 C1(NC(=O)Cc2ccccn2)CN(C(c2cnc3[nH]ncc3c2)=O)CCC1(F)F c1(C(N2CC3C(CNC(=O)CC4CCC(O)C4)(CC3)C2)=O)n[nH]c2ccccc12 CCCCC(O)C(=O)NC1(c2ccccc2)CN(C(=O)C(F)CCC)C1 Cc1cc(O)c(F)cc1NC(c1ccc(CNC(c2cncnc2)=O)o1)=O n1(CC(=O)NCC2CCN2C(=O)Cn2cc(C3CC3)nn2)cc(Br)cn1 N1(C(=O)NC(C)CCN)CCN(CCOc2cccc(Cl)c2)CC1 C(c1cnc(C(C)(C)C)s1)=CC(=O)NC1C(NC(c2cnc(CC)[nH]2)=O)CCC1 c1(OC)cc(C(N)=O)ccc1F.c12ccnc(c1)Oc1ccc(cc1)NC2 CCCCC(C(=O)NCCCN(C(c1ccncc1N)=O)C1CC1)N(C)C C(=O)(CCCCC(N)=O)NC1(C)CCN(C(C2C(c3ccccc3)C2(F)F)=O)C1 c1(C(=O)NCC(C)NC(C2CC2C(F)F)=O)c(O)ccc(F)c1Br c1(C(N(CCC(C)NC(C(CC)OC)=O)C)=O)ccc([N+](=O)[O-])cc1 C1(C(N(CCCC(=O)NCC(c2ccccc2)F)CC)=O)CN2CCC1CC2 C1(C2CC(C)OC2=O)(c2nn[nH]n2)CCCCC1.c1(C(C)C)cscc1 N1(C(C2CCC(COC)C2)=O)CCC2(C1)CN(C(=O)C=Cc1ccn(C)c1)C2 Cc1cc(C(=O)NCC(C(C)C)NC(=O)C(O)C2CCCC2)c2occc2c1 CCCC(CCCNC(c1ccnc(SC)c1)=O)NC(C1(C(=O)OC)CC1(C)C)=O C1(CC(=O)N(CC)Cc2ccccn2)C2CCCC2N1C(C1CC2(CCO1)CC2)=O C1(OC)CCC2(C(=O)NC3CC(NC(c4csc(NC=O)n4)=O)C3(C)C)CCC12 c1(C(N2C(CNC(CC(CC)C)=O)CCC2)=O)cc(OC)c2ncccc2c1 Cc1ccc2c(c1)CC(C(=O)NCCCN(C)C(c1cnc3[nH]cncc1-3)=O)S2 N1(C(C(C)CO)=O)CCC(O)(CCNC(C2CC=CC(O)C2)=O)CC1 c1(N(C)Cc2cn(CC)nc2)cccc(S(=O)(=O)N2CCOC(CC(N)=O)C2)n1 Cc1c(C(N2CCC(CO)(NC(c3cccc(=O)o3)=O)C2)=O)cnn1C1CCC1 c1(OCC)nccc(C(=O)NCc2c(OC(N3CCC(O)C3)=O)cccc2)c1Cl Cn1ncc([N+](=O)[O-])c1C(N1CC(NC(=O)CCn2cncn2)CC(C)(C)C1)=O Cc1nn(C)c(Cl)c1C=CC(=O)NCC1COC(CNC(=O)C=CCO)C1 N1(C(CS(CC)(=O)=O)=O)CCCC2(CCN(C(C3CCCC3S(C)(=O)=O)=O)C2)C1 N1(C(C2C(CCC)CN(C(C3(CC)CCCC3)=O)C2)=O)CCC(O)C(C)(C)C1 c1(NC(C2CN(Cc3cscn3)CCC2O)=O)cccc2cccnc12 C1(CNC(COCCSC)=O)CC(C)(C)CN1C(=O)CC1CCNC(=O)C1 c1(C(C)C(=O)NC(C)(C)CNC(C2(n3cccn3)CC2)=O)ccn(C)c1 C12C(C3CC3)CCN1C2=O.c1(CNC(Cc2cn(CC)nc2)=O)cncc(C)c1 C1(C2CCCC2)(CC(=O)NC(C2(O)CCCCC2)c2ccc(Cl)s2)CC1 N1(C(C2CC2C(=O)NCCN(C)C(=O)OC(C)(C)C)=O)CCC2(CC1)CC(O)C2 C(=O)(CCCCN1CCOCC1)NCC1C(CNC(c2cc(COC)[nH]n2)=O)C1 C1(NC(=O)C(F)C2CCOC2)(CO)CCCN(C(=O)C(F)OC(F)(F)F)C1 c1(C(N2CCN(C(c3cc(C)nnc3)=O)C(C)C2C)=O)csc2c(F)cccc12 c1(CC(=O)NCCCCC(C)NC(C=CC=CC)=O)c(C)oc2ccccc12 c1(CCC(=O)NCC2C(CNC(CC(CC)O)=O)CCC2)nc2ncccn2n1 C1(NC(C(C(C)C)O)=O)CN(C(c2ccnc(C(F)F)c2)=O)CC1(C)C CC1(C)C(CC(=O)NC2CCCCCC2)CCN1C(=O)CC1CCCO1 CC1C(=O)Nc2cccnc2N1C(=O)C(n1cc(-c2ccnc(F)c2)nn1)C1CC1 N#Cc1c(Cl)nsc1NCCC1CCCN(C(=O)CCCc2ccsc2)C1 c1(OC)cc(C(N2CC(CNC(C3(C)CC3)=O)C(C)C2)=O)ccn1 S(=O)(=O)(c1ccncc1C)CCN(CC#C)CCC1CCOCC1 CCCC(CNC(=O)Cc1ncn(C)c1C)C(=O)NCCOc1cccnc1 c1(CN(C2CCN(CC)C2)C)nc2c(n1C)CCCC2 c1(OCC2CCN(C(C(=O)NCC)=O)C2)ccccc1C1(C)CC1 CCC(C)(C)CC(=O)N1CC(NC(C2C3CCCC23)=O)CC1C C1(NC(C(CCNC(C(C)n2cncn2)=O)O)=O)CCC(=O)NC1=O C1(C(=O)NC2CC(CNC(COCCC#C)=O)C2)OCCC1(C)C C(C(C)(C)CC(C)O)NC(c1c(C)cnn1C)c1n(CCCOC)nnn1 CCCCN(CN1CCCS1(=O)=O)N1CCCC(OCCCOC)C1 CC(C)C1=NOC(C(N2CCC(C)(CNC(=O)Cc3cncn3C3CC3)C2)=O)C1 CC(F)(F)CCC(=O)N1CCC(NC(c2cnc(C3CC3)cn2)=O)C(O)C1 C(C(C)(C)C(C)(C)C)NC(CN(C(C1(C)C(C)C1)=O)CCO)=O Cc1n[nH]c(C)c1CCCNC(=O)C(CNC(C1CCCC1F)=O)CC1CC1 c1(CC)cc[nH]c1C(=O)NC(C(=O)NC1CC(N(C)C)C1)C1(C)CC1 [N-]=[N+]=NC1(C(N2C3CCC2COC3)=O)CCN(C(=O)CC2CC3(CC3)CO2)C1 c1(C(=O)NCC(C)N(C)C(c2ccccn2)=O)ccc2cnsc2c1 C1(NC(CN(C(C)=O)C)=O)CN(C(c2cn(C(C)C#N)nc2C)=O)CC1O Cc1cc(C)c(CNC2(NC(=O)CN3CC(C)(C)C3)CC2)c(O)n1 C(=O)(C#CC(C)(C)O)N1C2C(NC(C(C)OCC3CCCCO3)=O)C(C2)C1 C(=O)(CCCN(C)N=O)NC(CC)CNC(c1cccc(N2CCOCC2)n1)=O c1(CCC(=O)NC(CCCC)CNC(=O)COCCOC)cc(F)cc(F)c1 C1(CCC)(C(=O)N(C2(CC(=O)NOCC)CC2)CC2CC2)CC(=O)C1 Cc1ccc(Cl)cc1NC(=O)NC12CC(C(=O)NC3CC(CO)C3)(C1)C2 Cc1cnn(C)c1CC(=O)N(C1CCN(C(=O)COCC2CCCCO2)CC1)C C(=O)(C1CC(=O)N(C)c2ccccc21)NCC1CC(NC(CCCCCOC)=O)C1 CC1(C)OCCC1NC(=O)C(=O)NC1CCCN(Cc2cncnc2)C1 c1(C(N(CCN(C(c2c(C)n(CCO)cc2)=O)C)C(C)C)=O)cn(C)ccc1=O C(=O)(C(C)(C)C1CCN(C(c2ncoc2C)=O)C1)NCCOCC(=O)NC c1(C(N(C)CC2CN(C(C(CC(=C)C)OC)=O)C2)=O)cc(C)n(NC(N)=O)c1C Cc1cc(N2CC(=C(F)CNC(C3CCCC34CCC4)=O)C2)nc(Cl)n1 CCCCCCC(C(=O)Nc1cccc(Cl)c1C)N1CCC1(C)C Cc1cc(C(=O)NCC2(CCNC(c3c(Br)nnn3C)=O)CC2)c(C)n1C c1(C(N2CCCCC(NC(C3=NOC(C)C3)=O)C2)=O)ccc2[nH]ccc2c1 C1(CNC(CC2(OC)CC2)=O)CCC(C)CN1C(=O)CCCc1cccc(Cl)n1 C1(C(N2CCC(COC)(NC(=O)CCSC(F)(F)F)C2)=O)CC2OC1C1CC21 c1(OC)ccc2[nH]c(=NC3CCCC(NC(=O)CC(O)C4CCCC4)C3)oc2c1 c1(C(N(CC(CO)(CO)NC(C(CN(C)C)O)=O)C)=O)c[nH]c2cccnc12 C1(OC)(CNC(C2(C)CCCOC2)=O)CCN(C(=O)CCc2nccs2)C1 C(=O)(C1=C(Cl)CCC1)Oc1cccc(CC(=O)NC(=O)C(F)(F)F)c1 C(=O)(C(O)CC(F)(F)F)NC1C(C(=O)NCCC(C)(C)C(F)F)CC=CC1 C(=O)(C1CCc2cc(F)ccc21)NCC1(O)CCCN(C(C2(C#C)CCC2)=O)C1 CC1CN(C(c2ccc(N)cc2Cl)=O)CCN1C(C1(C)CCNC(=O)C1)=O N1(C(=O)C=CCNC(C2CC(F)C2)=O)CC2(CCCC2)C1 N#Cc1cc(F)ccc1NC(C12CC1CN(C(c1cc(O)c(O)c(Cl)c1)=O)C2)=O CC1CC(NC(c2ccsc2)=O)CCN1Cc1ccccc1F c1(C(=O)Nc2ccn(CC3CNC3)n2)ccc(-n2cccn2)cc1Cl N1(C(C=Cc2ccc(Nc3cccc(C(C)=O)c3)cc2)=O)CC2(CCCNC2)C1 N1(C(C(n2cnc(C#N)n2)C)=O)CCCCC12CN(C(=O)C(C)n1ccnn1)C2 N1(C(C2CC(C)OC2)=O)CC2CC1CN(C(=O)COc1cccnc1)C2 C1(CNC(COCC(=O)OC)=O)CC(O)C(O)CC1C(=O)N(CC(F)(F)Cl)C c1(C(=O)NC(C(CO)NC(c2cc(CC)c(C)cc2)=O)C)ccc2nccn2c1 Cc1cccc(C(=O)NC2CCC23CN(C(C2COCCO2)=O)C3)c1Cl CC1CN(C(C2(S(N)(=O)=O)CC2)=O)CCN1C(C1SCCCS1)=O C1(C(=O)NC(CN(C(Cc2n(C(C)C)cnn2)=O)C)C)CCN(C(C)C)CC1 CC1(C)CN(C(=O)C=Cc2ccc[nH]2)CCN(C(C2CC3(C2)CC(C)(C)C3)=O)C1 C1(O)(CNC(CCSCC(C)C)=O)CCN(C(C2(CCF)CC2)=O)C1 C1(c2cn(CCC(=O)N3CC(C4COCCO4)C3)nn2)CCC(F)(F)CC1 C1(NC(C2(C)CCCN2Cc2cccc(Br)c2O)=O)CCCC2CCCCC12 C(=O)(C(C(C)(F)F)c1ccccc1)NC(CC)CNC(=O)CCNC(=O)OC c1(C(C)NC(C=CCNC(c2cc(CC)sn2)=O)=O)ncccc1C C1(CNC(c2cn(C3CC3)nn2)=O)CC(F)CN1C(C1CCOC1C1CC1)=O CC1(CC(=O)NCC2(O)CCN(C(=O)CSc3ccccc3Cl)C2)CCOCC1 c1(C(=O)NCCCCCN(C)C(C2C(C)(C)C2(C)C)=O)cccc(N)c1F N1(C(C(CN(C)C)(C)C)=O)CCCC(N(C(=O)Cn2nnc(C3CC3)n2)C)CC1 Cn1c(=O)n(CC(=O)NC2CC(F)CN(C(=O)C(N)=O)C2)c2ccccc12 N1(C(C(C)S(N)(=O)=O)=O)CCCC12CCN(C(C1CCC3(CC1)CC3(F)F)=O)C2 C(=O)(C(CCN(C)C)NC(c1cc(C)on1)=O)NCCc1cc(C)no1 N1(CC(N2CC3C(CNC(c4c(C)nco4)=O)(C3)C2)=O)CCC(=O)NC1=O N1(C(C2(C)CCCO2)=O)CCC(CO)C(NC(c2cc3sccc3s2)=O)C1 Cc1nn(CC(N2CCC(CC(=O)NCc3cn(C4CC4)nn3)CC2)=O)c(=O)o1 c1(C(=O)Nc2cccc(NC(Cn3c(C)ccn3)=O)c2)cc(Cl)c(N)cc1F N12CC3CCN(CC3C1)Cc1cc(cc(Br)c1)C2=O.N(CCO)(CC)CC C12(C(N3CC(CCC)N(C(c4cncc(C)n4)=O)CC3)=O)CCCC1CC(=O)C2 C(c1cccc(F)c1)=CC(=O)NC(C)CC1CN(C(=O)C=Cc2cn(C)cn2)C1 C(=O)(C(F)(CNC(C1COC(=O)N1C)=O)C(C)C)NCCSCCOC C1(NC(CC2(C)CCCCC2)=O)CCN(c2ccnc(CO)n2)CC1O N1(C(c2c(F)ccc(C)c2)=O)CCC2CC1CN2C(c1cccc(F)c1)=O c1(CNC(C2(C)CC(=C)C2)=O)ccc2c(c1)CCC2NC(=O)CCCC(C)(F)F Nc1ccc(C(=O)NC2CCC2NC(C2CCC2n2ccnc2)=O)nc1 C=C(C)CCCC(=O)NCC1(F)CC(NC(c2onc(OC)c2Br)=O)C1 C1(C(N2C(C(N(C3CC(CO)C3)C)=O)CSCC2)=O)CCC2(CC1)CC2 CCC(C)(C)C(=O)C(=O)NCC#CC(N1CC(C2CC2)C1C1CC1)=O C(=O)(C(F)(F)C1=CCOCC1)NC1C(CNC(=O)C2=NOCC2)CCCC1 N1(C(c2ccoc2)=O)CC2(C(=O)NCCCc3ncco3)CC1CO2 N1(C(C2(CCCC)CC2)=O)C(C(N2CC3CCC3(C)C2)=O)CC2CCCC12 C1(NC(COCCCC)=O)CC2CCC1(NC(c1ccc(O)cc1)=O)C2 C1(CC(=O)NCCOC(CNC(CCn2ccc(C)n2)=O)(C)C)CCCCC1O C1(CCC)CCC(C(=O)NCC2CC(NC(=O)CN3CCCC3CC)C2)CC1 CC1CC(NC(c2ccc(Cn3ccnn3)o2)=O)CN1C(=O)CC(F)(F)F C1(C(N2C(CNC(c3[nH]n(C)c(=O)n3)=O)CC2)=O)CCc2ncc(Br)n2C1 c1(C(=O)NCC2N(C(C(c3ccccc3F)C)=O)CC(F)C2)ccc(=O)n(C)n1 C12(C(N(C3CCCCC3)C)=O)CCN(C(c3ccncc3Cl)=O)CC1C2 C(=O)(CC(C)C(C)C(C)C)N(C1CCN(c2ncnc(C(C)(C)C)n2)C1)CC.C1(C)CC1 c1(C(=O)NC2CC(C)N(C(c3ccc(=O)oc3)=O)C2)cc(F)c2c(c1)CCC2 C12COCCN1C2.C1(C(=O)Nc2ncc(CO)o2)CCN(c2ccccn2)CC1 c1(C(=O)NC(C2CCN(C(=O)Cc3nccn3C)C2)C)ccc(=O)oc1 N1(C(CC2CC(=C)C2)=O)CCCC2CN(C(c3ccc(C(C)C)o3)=O)CCC12 N1(C(c2c(CC)con2)=O)CCC(CNC(c2ccc(CC)c(F)c2)=O)C(C)C1 C(=O)(C1=C(C)OCCC1)N1CCC(O)C1.CCC(C)CONC=O C(=O)(CCCC(C)C)N(CCC(C(C)C)NC(c1oc(C)c(CO)c1)=O)C C1(NC(C2CCCCO2)=O)CC2CN(C(C34CCCC(CO3)C4)=O)CC2C1 c1(CS(N)(=O)=O)ccc(C(=O)NC2CCC(NC(C3C4(CC4)C34CC4)=O)CC2)cc1 N1(c2nc(N3CCCN(CC)CC3)c3c(n2)CCS3)CC2C3CCC(CC3)C2C1 N1(C(CSCCC)=O)CC2CCC1C(CNC(=O)C(N1CCCC(C)C1)=O)C2 C(=O)(CC(C)(O)COC)N1C(C(=O)N(C)Cc2n[nH]c(C)n2)(CC)CCC1 N12CC3(CCOCC3)C1c1cn(nn1)CCC2.C1(C(=O)OCF)CC2(CCCC2)C1 C(C(C)(C)CN(C(=O)Cc1ccnn1C(C)C)C1CC1)NC(CN(C(=O)OC)C)=O C(=O)(C1=NNC(=O)C1)NC1C(NC(c2n(C)nc(C3CCCC3)c2)=O)CC1 c1(CC)cc(N)ccc1C(N1CCC(CCCNC(=O)C2=CC(C)(C)C2)CC1)=O Cc1cc(F)cc(C)c1C(=O)NC1CCN(Cc2ccc(F)cc2Cl)CC1F CCCC(C(=O)NC(CC1CC1)C(=O)NC(C)(C)C(F)(F)F)C(C)C N1(C(CCN(CCC)C)=O)CCOCC1CC(=O)NCC1CC12CC2 c1(C(=O)NC(=O)CC2(CC(C)C)CC2)cnn(CCN(C)C)c1 N1(C(c2cccc(CC)c2F)=O)CC2CC(NC(C3(F)CC=CCC3)=O)C(C2)C1 C(CC(=O)Nn1cnnc1C)N(C(c1ncnc(C)c1C)=O)CCO c1(C(=O)NCC(C)(C2CC2)NC(=O)COC2CCCOC2)cccnc1N C1(c2ccc(OC)cc2)CCN(C(=O)NC(C)C(C)SC)CC1SC CC1CC(C(=O)NC2(CNC(C3(CO)CCCC3)=O)CC2)CCS1(=O)=O c1(CNC(=O)NCC2(CC)CCOC2)ccc2[nH]nc(Cl)c2c1 C1(NC(C(C)=CC)=O)CCC12CCN(C(=O)C(C)COC)CC2 c1(C(=O)NCCC2CCN(C(C)=O)C(CN)C2)ccnc2[nH]cnc12 c1(C(=O)NC(c2nc3ccccc3[nH]2)(C)C)cc(Cl)cc2c1NCCC2 c1(CCC(=O)NCC2C(C)CN(C(c3ccsn3)=O)CC2)cc(F)c(F)c(F)c1 N1(C(CCC(=C)C)=O)CCC(CNC(C2(C(F)F)CCCO2)=O)C12CC2 Cc1cc(NC(=O)CC(C(F)(F)F)N(C)C)cc(Cl)c1O N1(CC(=O)N(C(CC)=O)C)CCC(C(=O)NNC(=O)OCc2ccccc2)CC1 C1(C(=O)NCC2CN(C(C)=O)C2)(OC)CCN(C(c2cnsn2)=O)C1 CCC(CCC(=O)NCC=CCNC(c1nc(C(F)(F)F)ccc1N)=O)OC C1(NC(C2N(CC)CCOC2)=O)CCCN(C(=O)C(C2CCCCC2)O)CCC1 CC1(C)CC(CNC(=O)CNC(c2ccsc2)=O)N(C(=O)C=C(Cl)Cl)C1 C1(CC(=O)NC2CCCC(C(N)=O)C2)CC2(C1)CN(Cc1ccccc1)C2 C(C)(CCC(=O)N(CC(C)C)C)NC(C(C)NC(CC)(C)C)=O C1(NC(c2c(OC)n[nH]c2)=O)CCC2(CC1)CC2NC(C1CCC(C)(C)OC1)=O N1(Cc2cc(C)ncc2)CCC(O)(C(N2CCC(CO)CC2)=O)CC1 N12CCC(CC1)CN2C.C1(SCC)CCN(C(C2CC(N(C)C)C2)=O)CC1.C1(C=O)CCC1 C1(C(=O)NC2(CNc3nccc(C)n3)CCCCC2)CC2CCCCCCC12 C1(NC(c2ccc(C(F)F)o2)=O)CC12CCN(C(=O)CC1=CCCC1)CC2 N1(C(C(=O)Nc2ccc(I)c(Br)n2)=O)CC(C2CC2)C(F)(CO)C1 C1(C(N2CC(CN(C(=O)CN(C3CCCC3)C)C)C2)=O)CCCC(C)(C)C1 N1(C(C(C)OCCCC)=O)CCC2CN(C(=O)CCC3CCCCC3)CC12 CC(C(=O)N1CCC(CO)(NC(c2cnc(-c3cccs3)s2)=O)C1)C(C)(C)C C(c1ccc(F)c(F)c1)=CC(N1CC2CCC1CN2C(c1cc(Cl)c(Cl)s1)=O)=O N1(C(C2(C(=O)NC)CC2)=O)CCCCC(NC(c2cc(F)ccc2C)=O)CC1 c1(S)cc(F)ccc1F.CC1(NC(=O)CCN(C)C)CNC(=O)C1C1CC1.C1CC1 N1(C(c2ccc(C(C)=O)o2)=O)CC2CCC1C2NC(c1ncccc1F)=O C1(NC(CCCC(CC)C)=O)CS(=O)(=O)C2CN(C(=O)C3=COCCC3)CC12 C1(NC(c2ccc(C(N)=O)[nH]2)=O)CCN(C(=O)CCNC(N)=O)CCC1CO N1(C(CC=CCNC(Cc2cc(C)n(C)n2)=O)=O)CCN(C)C2CC12 C1(C2CCOCC2)(C(=O)NCC2N(C(CC(C)SC)=O)CCOC2)CCOCC1 C1(NC(Cn2c(C)nnn2)=O)CN(C(=O)C(O)CCN(C)C)C(C)(C)C1 c1(N2CCC(C(C)NC(c3csc(CO)n3)=O)CC2)cc(=O)n(C)cn1 N1(C(C2C3CN(C(CCc4ncn(C)c4)=O)C2C3)=O)CCCC12CCNC2=O C(=O)(CS(=O)(=O)C1CC1)N1CCC(F)(CNC(CCC2C(C)C2)=O)C1 C1(C(N2CC3CC2C3C(=O)NCc2cccs2)=O)(CC)CC(C)(C)C1 CN1CCCCC1CC(=O)NC1(C(=O)NC2COC(=O)C2)CC(O)C1 N1(C(CN(CCC)C)=O)CC2CC(NC(c3cn(CC(O)CC)nn3)=O)CC1C2 c1(OC)cscc1C(c1nnnn1Cc1nnn(C)n1)NC(C)C1CC1 C1(C(=O)NCC=CCNC(c2ccc(C3(C)COC3)o2)=O)CC1C1CCCC1 N1(C(c2ncc(C)cc2F)=O)C2CCC1CC(CNC(C1(CC3CC3)CC1)=O)C2 C1(CN(C(=O)Cc2cn[nH]c2)C)CC(F)CN1C(=O)CCOCC(F)(F)F c1(C(N2C(C)C(NC(C3(C)CCCC3(F)F)=O)CC2)=O)cnc(S(C)(=O)=O)s1 CCCCCCC(C)C(=O)N1CC2CC(C1)CN(C(=O)C(O)CC[S+](C)C)C2 C1(C(=O)NC2CC(NC(c3[nH]cc(C(C)=O)c3)=O)C2)CC2(C1)CC2F C(=O)(CC(C)CC)NC(CC)CNC(C1CCN(c2ccnc(Cl)n2)CC1)=O c1(-c2cnc(NC(C(=O)OCC)C)nc2)ccc(F)c2cccnc12 c1(C(=O)NC(CC=C)CNC(=O)C(COC)OC)cc2cc(Cl)ccc2n1C C1(NC(C(CC)NC(N)=O)=O)CC2CC1CN(C(c1cc[nH]c(=N)c1N)=O)C2 C1(C)(C(=O)NCCC(CC)(C)O)CCCN(C(=O)CCCC2CCCC2)C1 c1(OC)c(C(=O)NC(C)C(C)NC(c2cn(C)cc2C)=O)ccnc1Cl CC(O)(CNC(=O)CCCNC(N)=O)CNC(=O)NC1(C#N)CC1 Cc1ccc(Cl)c(C(=O)NC2CC2CNC(c2cn(C3CC3)nc2C)=O)c1 c1(CC(=O)NCC(=O)NC(CCCC)CNC(N)=O)cccc2c1OCO2 C1(C(C)C)CN(C(=O)CSc2ccccn2)CCN1C(=O)C(F)n1cccn1 c1(OC)cc(C(=O)NCC2CN(C(C3CC3F)=O)CCCO2)c(F)c(Cl)c1 C1(C(N(CC(C)O)CCOC)=O)CCOCC1NC(=O)CN1CC=CC1 C(=O)(CCS(N)(=O)=O)NCc1c(C(=O)NC(c2ccncc2)C)[nH]cc1 c12c(cnc(C)c1O)-c1onc(n1)-c1cnc(nc1)CS2.N1(CC)CCCCC1 C1(C(=O)NC(C2(C(N(C3CN(C(C)C)C3)C)=O)CC2)C)CC2C=CC1O2 C#CC1(C(=O)NCCC(C)(C)NC(=O)Cc2cscc2Br)CCCC1 CC1CN(C(c2cc(Br)ncc2F)C(=O)NC)CC2(CCOCC2)O1 c1(C(=O)NCCCCC(C)NC(=O)CCc2nc[nH]n2)cnc2[nH]nnc2c1 c1(C(N2CCC(CC)C2CNC(c2ncn(C)c2C)=O)=O)cc(N)c(F)cc1C N1(C(Cn2ccc(C)n2)=O)CCCC2(NC(c3ccc(CN(C)C)[nH]3)=O)CC2C1 c1(OC)ccc(C(c2cccnc2)NC(=O)CN(c2ncc(C)s2)C)cc1 CN1C(=O)c2ccccc2C1CC(=O)N1CCCC1CNC(c1n[nH]cc1Cl)=O C(=O)(CC1=CCCCC1)N1CC(CCC)C(NC(=O)C(O)CCn2cncn2)C1 c1(CC)ccc(O)c(NC(=O)C(=O)Nc2ccc(CC3CC(C)C3)c(OC)c2)c1 c1(C(=O)OC)nnc(C(C)NC(=O)NC2CC(OC(C)(C)C)C2)n1-c1ccccc1 c1(C(N(CCOCC#C)C(C)C)=O)cscc1Br C1(C)(NC(c2c(C)con2)=O)CCCN(C(c2cc(O)nn2C)=O)C1 CS(=O)(=O)c1ccc(C(=O)NC23CC(C2)N(C(c2ccc4c(c2)CCO4)=O)C3)o1 c1(C(C)=O)nc(N2CC(CC(C)NC(c3csc(Cl)c3)=O)C2)c(F)c(Cl)n1 CCCC(C(=O)NC)NC(=O)C(CO)NC(=O)CC1CC2(CCC2)C1 C(=O)(CCC(O)C(C)(C)C)N1CC(NC(CC2C(C)CCC2)=O)CC2(C1)CC2 C1(CC)CCC(C(=O)NC2CN(C(C3(CO)CC3)=O)CC2OC)CC1 N1(C(C=CC)=O)CCCC(C2CCN(C(=O)CSCC(F)(F)F)C2)C1 C(C(C(F)(F)F)N1CCN(C(C2CCCC2)=O)CC1)NC(c1nc(C)oc1)=O C1(C(N2CC3C(CNC(c4cc(F)ccc4Cl)=O)(C3)C2)=O)CC2CCC(C1)C2 N1(C(=O)NCCC(=C)Cc2ccccc2)CCC2(CCC(=O)NC2)CC1 C(CC(C)(C)CC(=O)NC(C1CCN(C(=O)CNC(=O)CN(C)C)C1)(C)C)OC C(=O)(C1CCCc2n[nH]cc21)NC1(C)CC(NC(c2ccoc2)=O)C1 c1(CC)cc(NC(=O)CCC2CCN(C(c3[nH]ccc3C)=O)C2)ccc1F C(CCN(C)C(C1CC12CCCCC2)=O)(C(C)(C)C)NC(C(CC)CC)=O C1(COC)(CNC(c2cnnn2C)=O)CCCN1C(=O)CC1CCOC1C C1(NC(C(C(CC)C)O)=O)CC2(CCN(C(c3nocc3C)=O)C2)C1 N1(C(CC2(NC(c3c(CC)ocn3)=O)CC2)=O)CC(O)CC1(C)C N1(C(C2(CC)CC2)=O)CCN(C(C2CC3CC3C2)=O)C(CO)C1 c1(C(N2CCC(N(C(C(C)=C3CCCC3)=O)C)C2)=O)ccn2ncc(C)c2n1 C12(C(=O)NC(COC)CCOC)CCC(NC(=O)C(C)=CC(C)(C)C)(CC1)C2 Cc1nc(O)ccc1C(N1CCC(C(C)C(=O)NC(c2cnn[nH]2)(C)C)C1)=O C1(CNC(CC(C)C(F)F)=O)C(C2CC2)CCN1C(c1cc([N+](=O)[O-])cn1C)=O C(CC#CC)(C(=O)Nn1cncn1)NC(CCC#C)=O N1(C(C(C)C2CCCOC2)C(=O)NC2COC2)CC2CCC(C1)N2C CCC(C)(CCC(C)C)C(=O)NC1(CO)CCN(C(c2ccc(Cl)c(O)c2)=O)C1 N1(C(CN2CC(C)(OC)C2)=O)C2CCC1CC(NC(C1(C)CCC(=O)N1)=O)C2 C(C(CC1CC1)C(=O)NCC1CC1(C)C)NC(COC(CC)(C)C)=O N1(C(c2c(C)ccnn2)=O)C(CNC(=O)CC2CCCCN2C)CC2CCCC12 N1(C(C2C(C)(C)CCCO2)=O)CC2(CCCC2)C1C(=O)NC1(C)CCC2(CC2)C1 CCS(=O)(=O)C=CC(=O)N1CCC(CNC(=O)C(C)(C)NC(=O)C=CBr)C(C)C1 C1(C(=O)NC2CC2NC(C2(S(C)(=O)=O)CCC2)=O)(COC)CCCNS1(=O)=O C1(C(=O)NCC23CC2CN(C(c2cnn(C)c2C(C)C)=O)C3)(CC)CCNC1=O c1(C(=O)NCCC(C)(C)NC(C2CC2C2CCCO2)=O)cccnc1N C(=O)(C(C)(C)CC(=O)N1C(CNC(=O)C(C)(C)C)CC2CC12)OC c1(C(=O)NCC(C2CC2)NC(C(C)(C)OC(C)=O)=O)cccc2c1OCC2C C1(CC(=O)NC2CCC(CCNC(c3c(C)n(C)nc3)=O)C2)CC2(CCO1)CC2 CCC(C(=O)NCC1CCC(C)CN1C(C1CN(CC(C)C)C1)=O)C(F)(F)F CC1(C)CNCCC1C(N)=O.c12cccc(c1)-c1noc(n1)CC(=O)N2 C1(NC(C2(F)C(C)OCC2)=O)CCCCN(C(C2CN(CC(F)(F)F)C2)=O)C1 C(=O)(C(C)(C)CC(F)F)NCCN(C1CCCC1)C(C1(C=C)CCC1)=O CN1CC(C)(C(=O)NC2CCC2CNC(C2CC(O)C2)=O)CC1=O c1(C(N2C(C)C(NC(=O)C(C)(C)C)CCC2)=O)ccc2c(c1)CCCCS2 c1(C(=O)NCC(C)(C2CC2)NC(C(CC)OC)=O)ccc2occ(C)c2c1 Cc1oc(Br)cc1C(N1CCC(C(F)CNC(C2CC=CCO2)=O)CC1)=O c1(NC(C(N2CCC(OC)C(C)C2)=O)=O)cc(C)c(C)cc1C c1(C(=O)OC)cc(C(=O)NC(CO)C(C)NC(=O)C=CCF)c(F)cn1 c1(C(=O)NC2C(CNC(C3(C=C)CC3)=O)CCC2)cnn(CC)c1C C(=O)(CCCCC(C)(C)OC)N1C(C(C)(C)NC(c2c(CC)con2)=O)CCC1 C(N=C(NCC(F)F)N1CCC2C(C1)NC(=O)N2C)c1c(OC)nccn1 N#Cc1cncc(C(N2CCC(C(=O)NC3CC4C(C3)C4(F)F)C2)=O)c1 C(C(C)C)(C(O)C(=O)NC1(C)CCN(C(=O)C(C(C)C)C(C)C)C1)OC c1(C(=O)NC2(CO)CCN(CC)CC2)c(-c2ccnc(COC)c2)cc(F)cc1F c1(C(=O)NC2CC(C)N(C(=O)C(=Cc3cccnc3)F)C2)ccnc2ccsc12 c1(OCC)ccc2ccccc2c1-c1ccc2[nH]c(C(=O)NCC(N)=O)cc2c1 N1(C(c2c(C)n(C)cn2)=O)CCC(O)(CNC(C2CCCC(C)O2)=O)CC1 C(=O)(CCC(=O)NCCC1CCC(NC(=O)C(C)C(=O)OC(C)(C)C)C1)NCC Cn1ccc2ccnc(C(=O)NCC3CC(NC(=O)CNS(C)(=O)=O)C(O)C3)c12 C1(CNC(c2ncn(C)n2)=O)CC2CCC1N(C(=O)COCc1cccnc1)C2 C(C)(CNC(c1nscc1C)=O)(CC(C)C)NC(c1ccc(COC)o1)=O N#Cc1cc(S(=O)(=O)NC2C3CCCC23)ccc1NCC1(CO)CC=CC1 c1(C(=O)NC23CCC(CN(C(CC(COC)C)=O)C2)C3)ccc(Cl)c([N+](=O)[O-])c1 CC(F)CC(=O)NCC1(O)CC(NC(c2c[nH]c(C(F)(F)F)c2)=O)C1 c1(C(=O)NC(C2CCCC2)CNCC=C(C)C)c[n+]([O-])c(C)cn1 C12(CNc3cccc(CNC(c4n(C)ncc4)=O)c3)CNCC(=O)N1CCOC2 N1(C(CN(C)C(N)=O)=O)CC2(C1)CN(C(=O)COC(C)(C)C(F)(F)F)C2 C(CCCCC(=O)N1CC(NC(=O)CNC(c2cccs2)=O)CC(O)C1)SC C1(CC(=O)NCC(C)(C2CC2)NC(c2cc(Cl)cnn2)=O)CCCC(C2CC2)O1 N1(C(C(C)(C(C)C)OC)=O)CC(C(=O)NCC(C)F)CC(C)(C)C1 c1(C(=O)NC2C(CN(C(C3C(C(C)O)C3)=O)C)CCC2)nn(C)cc1Cl N1(C(C(CCCC)C)=O)CCC2(C1)CN(C(C1CC1c1cnc[nH]1)=O)CCO2 N1(C(C=CC=CCC)=O)CCN(C(=O)Cc2cc(C)cc(C)c2)CC1CF C(=O)(C1CCc2cc(F)ccc21)N1CCC(C(=O)Nc2cccnc2[N+](=O)[O-])C1 N1(C(C2CN(C(C)=O)C2)=O)CCC(C)C(CNC(c2cscc2Cl)=O)C1 c1(CN(C)C(C2(CF)CCC2)=O)cnn2c1CN(C(c1[nH]ncc1C#N)=O)CC2 c1(OC)cc(SC)ccc1C(N1CC2CC2(C(=O)Nc2ncc(C#N)s2)C1)=O N1(C(C(C)N2CCCC2)=O)CC(N(C(c2nncs2)C)C2CC2)C2(CC2)C1 Cc1ccc2c(C(=O)NCC(C3CC3)NC(=O)Cn3cccc3)ccnc2c1C CCC(C)CC(=O)NCc1cc(C(=O)NC2C3CCCC23)ccn1 c1(CC)cc(C(N2CC3CC2(CNC(C2CCCN2C(N)=O)=O)C3)=O)cc(O)n1 C(=O)(C(O)(C(F)(F)F)C1CC1)N1CCC(N(C(C(C)OCC=C)=O)CCO)CC1 c1(CCC(=O)NCC2(F)CC(CNC(C)=O)C2)cncnc1O c1(CN(C)CCc2ccccc2)cc(Br)cn1C.C1C(CN)CN1 C12(C(N(C)CCNC(C3CCS(=O)(=O)CC3)=O)=O)CCC(C)(CC1)OC2 N1(C(c2c(C)con2)C(c2ccccc2)=O)CCN(C2CCS(=O)(=O)C2)CC1 C(=O)(C=CS(C)=O)N1CC(N(C(c2c(C)nns2)=O)C)C1 C(CC(O)C(=O)NCc1cccc(O)n1)NC(C)=O C1(NC(=O)C2CC2)CN(C(C2CC(C(F)F)C2)=O)CC12CCOCC2 c1(NCC)cncc(C(N2CC(CNC(C3CC(OC)C3)=O)CC2C)=O)c1 c1(C(C)C)c(N(C2CCNC(=O)C2)C(C2CCCC2)=O)ncnc1Cl c1(C(=O)NC(c2cn(-c3cccc(C)c3)nn2)(C)C)ccnn2ccnc12 c1(OC)cc(C(=O)NC23CC(CNC(c4cc(F)cnc4O)=O)(C2)C3)cc(O)c1 c1(NC(CNC(c2c(OC)cccc2)=O)C2CC2)ncnc2c(Br)nn(C)c12 c1(OC)cc2ccc(C(=O)NC3CC3NC(=O)CCN3CCC3)nc2cc1F CC1CC2(CCO1)CC2C(=O)NCC12CCCC1N(C(=O)CC(F)(F)F)CC2 CCC(C(=O)N1CC(c2ccncn2)C1)N(C(=O)C(C)CC1CCCC1)C N1(C(C(C(=O)OCC)F)=O)CCC(NC(C2CC2CCOC)=O)C(OC)C1 c1(CC(C(=O)NC(C(C)O)CO)NC(=O)CCc2cnco2)ccccc1Br c1(CN2CCC(NC(=O)OC(C)(C)C)(CO)CC2)c(F)ccc(Cl)c1F C(=O)(C(CC(=C)C)OC)NC1CCC(C(N(CC=C)CC2CC2)=O)C1 N1(C(C(C)OC2CCOCC2)=O)CCC(NC(c2cc(O)ccc2F)=O)C(O)C1 c1(C(N2CC(O)(CN(C(C(C)O)=O)C)C2)=O)ccc(Br)c(F)c1F C1(CC(=O)NC(C)(C)C(=O)NCCC2CCC3CC23)CCCCC1O c1(C(=O)NC2CC(NC(CCC(C)SC)=O)C2)cc(C)nc(C(F)F)n1 CC(N=c1nc(N2CCNC(=O)CC2)c2ccccc2[nH]1)c1cccc(Br)n1 N1(C(CONC(c2nc(=N)[nH][nH]2)=O)=O)CCc2nnnn2CC1 c1(NC(C2N(C(c3cc(C(C)(C)C)n[nH]3)=O)CCC(O)C2)=O)ncc(I)cc1I n1(CC(N2CC(NC(c3ccc[n+]([O-])c3)=O)C3C2C3)=O)ccc2cc(F)ccc12 CC(C)(C)CC(O)CC(=O)N1CCCC1C(=O)NCc1c(F)cccc1F C1(NC(C2OCCN(C(C(C(CC)O)C)=O)CC2)=O)CCC(=O)NC1(C)C c1(OC)cc(C(=O)NC2CN(C(=O)C(c3ccccc3)C)CC2F)ncn1 C(=O)(C1=CCCCCC1)NC1C(C(=O)NCc2c(C)n(C)nc2)COCC1 C1(c2nnc(C)o2)CCCCCN1C(c1cnn(C)c1)C(=O)NCC(F)F C1(NC(CC(CC)C2CC2)=O)CCCN(C(=O)C(C#N)=CC2CC2)CC1 Cc1nn(C)c(C)c1CNC1CCCC(C(N2C(C)CCCC2C)=O)C1 c1(C(N2CC(CN(C(C(C)SC)=O)C)OCC2)=O)cnc2ccnn2c1 C(=O)(C(C)S(N)(=O)=O)NC(C1N(C(c2cc(C(=O)OC)oc2C)=O)CCC1)C C1(NC(c2c(OC)nccn2)=O)CN(C(=O)Cc2ccc(O)cn2)CC12CCC2 CC(C)C(C(=O)NCC1CCCN1C(c1ccn(C2CC2)n1)=O)c1cccnc1 O=C(CCCCc1ccc(F)cc1)NC1CCN(c2ccccn2)C1 Cc1nc(Br)ccc1C(N1CCOCC1)=O.c12ccc(cc1)CN(C)C2 N1(C(C2=C(C)CC2)=O)CCC2(CCN(C(c3ncc(N)cc3C)=O)CC2)C1 C(CCCC(=O)NC(C(=O)NCc1ncc(C)o1)C1CC1)OCC C1(COC)(NC(=O)C(C(C)(C)C)SC)CCCN(C(c2cc(F)c[nH]2)=O)C1 N1(C(C2CCC(NC(c3ccoc3Cl)=O)C2)=O)CCC(O)(CO)C1 N(C1CN(C(=O)CN=S(C)(C)=O)Cc2ccccc21)C(c1cc(C)c(C)[nH]1)=O CCC(C)C(CC(=O)NC1CCn2nccc2C1)NC(c1cc(C)cc(C)c1)=O C1(NC(c2ncn(C)c2)=O)C2CCC1N(C(c1cc(F)n[nH]1)=O)C2 C(=O)(CCC(=O)NCC(CC)N(C(C1(C#N)CC1(C)C)=O)CC)N(CC)CC c1(OCCC)ccc(C(=O)NCCCC(C)(C)NC(c2cnn[nH]2)=O)cc1OC N1(C(c2cnc(C)[nH]c2=N)=O)CCC2CC2(C(=O)N(C)CC2(O)CN(C)C2)CC1 C(=O)(C(C)(CC)CCCCCC)NCC=C1CCN(C(C2C(C=C)CC2)=O)CC1 N1(C(C2CCC(CNC(CC(C)N(C)C)=O)C2)=O)CC(CO)CC1(C)C c1(C(=O)NCC(CN(C(=O)C=CCF)C)O)ccc(Oc2ccc(F)cc2)nc1 Cc1cc(Br)cn2c(C(N3CCC3CC(=O)O)=O)cnc12 C(=O)(C(C)(O)C(F)(F)F)N(C(CNC(C(c1ccc(F)cc1)CC)=O)C1CC1)C Cc1cnc(Cl)nc1N1C2CCC1C(CNC(=O)CC1CCC(=O)N1)C2 c1(C(=O)NCC(C2CCCC2)NC(CC(C=C)CC)=O)ccc2cccnn12 N1(C(CCC(CC)C)=O)CCC(C2(NC(=O)C(COC)N(C)C)CC2)CC1 CCC(C)(COC)CNC(=O)C(C(C)O)NC(=O)CCn1ccnc1 C1(C)(NC(CCSc2ccc(C)cc2)=O)CCCN(C(C2(C(F)F)CCC2)=O)C1 c1(C(=O)NC2CCC(N(C)C(c3ccncc3Cl)=O)C2)ccnc2ncsc12 C1(C(=O)NCC(C)NC(=O)CN2C(=O)C(=O)N(C)C2=O)CCC2(CC1)CC2(F)F N1(C(C2(C)CCCOC2)=O)CC2(CCC2)CC1CNC(c1ncc[nH]c1=O)=O c1(CC(=O)NCC2CC(NC(C(c3nc(C)sc3)=O)=O)C2)ccc(C)cc1F CC1(C)CN(C(=O)C2=C(Cl)CC2)CCC1NC(=O)C(C)(C)c1cnco1 CC1(C)C(NC(C2CC2F)=O)C2CCCN(C(C3CCCN3)=O)C12 C1(Nc2ncnc3onc(C)c32)CC2(CO1)CN(C(=O)CCC(C)C)C2C(C)C C1(CNc2ncnc(C(C)(C)C)n2)C(C)CCCN1C(C1CCC(F)C1)=O C1(C(=O)NC2CN(C(C#CC(C)(C)O)=O)CC(F)C2)CC2CCC1CC2(F)F CCCC(C)(CC)C(=O)N1CC2C(CNC(=O)C(F)(F)C(O)CC)C2C1 C1(NC(c2n(C(C)C)ncc2)=O)CCCC(N(C(=O)C=Cc2cc[nH]n2)C)C1 Cc1noc(C)c1CC(=O)NCC(C1CCCN1C(c1ccc(C)n1C)=O)(C)C O=C(NNC(=O)c1cccc(-c2ccccc2)c1)NCC(CO)C1CCOC1 C(=O)(C(C)C(O)C(C)C)N1C(C(N(C(C)C(=O)OC)CC)=O)CC2CC21 CC1CC(O)CN(C(C2CC(NC(c3c[n+]([O-])c(C)cn3)=O)C(O)C2)=O)C1 C12(C(N3CCCC(NC(CNC(=O)C4CC4)=O)CC3)=O)CCC(=O)N1CCS2 c1(NC(CC2CN(C(CNC(=O)OC)=O)C2)C)c(OC)c(Cl)cc(Cl)c1OC CC1CN(C(c2cc(F)n(C)n2)=O)CCCN1C(=O)CC1CCCCC12CC2 c1(C(=O)NC2(CNC(CC(CC)OC)=O)CCOC2)cc(Cl)ccc1N c1(CC(=O)NC)ccc(C(=O)NC2CN(C(=O)OC)C2)cc1 c1(C(=O)NCC23C(CN(C(CC(=O)OCC)=O)C2)C3)ccnc2[nH]cnc12 c1(-n2ncc(CCNC3CCC(CCC(=O)OC(C)(C)C)C3)c2)cccc(Cl)c1 Cc1nccnc1-c1cn(C2CCCC2NC(=O)CC2(N(C)C)CC2)nn1 N1(C(C)NC(=O)NC2CCN(C(CSc3cccc(C)c3)=O)C2)CCCNS1(=O)=O c1(SCC)cccnc1C(N1CCC(C(C)NC(C2CCCC(C)C2)=O)CC1)=O N1(C(c2c(Cl)cn(CC)n2)=O)CCCC(C2(NC(C3(O)CC3)=O)CC2)C1 C1(CNC(c2ccc(OC(C)C)cc2)C)CCCC2(CCOCC2)O1 n1(COC)nnc(C(=O)NC(COC(F)F)(C)C(C)C)c1N.C1(=O)CC2(CC2)CN1 N1(C(c2nc(C)sc2C)=O)CCC2C(CCN2Cc2ncc(C(F)(F)F)[nH]2)C1 N1(C(C=CCOCCOC)=O)CC=CC(NC(c2ccncc2)=O)C1 c1(CC)cc2c(N3CCCC(n4nc(C)nc4C)C3)ncnc2s1 N=c1[nH]ccc(C(=O)NC2C3CC(NC(C4CC(=C5CCC5)C4)=O)CC23)c1Cl.C=O N1(C(C(F)=CCC)=O)CCC(NC(=O)CC2CC3(CCC3)CCO2)C(C)(C)C1 c1(OCCCOC)ccc(SC(c2cc(C)n(C)c2)c2nnnn2C)cc1 N1(c2c(C)nc(C(N)=O)cc2)CCC=C(C(=O)Nc2cnc(Cl)c(C)c2C)C1 Nc1ccc(-c2cn(C3CCCC3NC(c3cnncc3O)=O)nn2)cc1F CC(CN(C)C)CC(=O)N1CC=CC(C(N2CC(O)(CCO)C2)=O)C1 C1(CCNC(C(C)(C)N(C)C)=O)CN(C(=O)C=Cc2cocn2)CCS1(=O)=O N1(C(C2C(C(C)=O)C2)=O)CCC(C)C(NC(=O)CC2(O)CCOC2)C1C n1(CCCCNC(N2CC(N3CCCC3CO)C2)=O)cc(-c2ccc(Cl)s2)nn1 c1(CNC(C(C)(C)OCC)c2nnnn2C)nnn(C)c1C c1(C(N2CCC(CCF)CC2)=O)ccc(O)c(Cl)n1.c12cn(nn1)CCCOC2 C1(C)(C(N2CC(OC)C2)=O)CN(C(c2nc(Cl)cs2)=O)CC1C C1(F)(C(=O)NCC(=Cc2ccccc2)C)CCCN(C(C2CCCCC2)=O)C1 Cc1csc(=O)n1CCCCNC(C1CCC12CCC2)=O c1(CC(C)C)nccc(C(=O)NC(C2CCCN2C(=O)CO)(C)C)n1 C1(NC(=O)Cc2cnns2)CCN(C(=O)C(Cl)=CCl)CC1F C1(NC(c2c(CC)nco2)=O)CN(C(C2CCOC2(C)C)=O)CC2(CC2)C1 C(N=c1[nH]cnc2c(Br)nn(C)c12)C1N(C(C2C(=C)CC2)=O)CCC1 N1(C(C(C)CO)=O)CCc2ccccc2C1CNC(=O)C(c1cnn(C)c1)O CC1(C)CN(C(=O)CCS(C)(=O)=O)CCC1C(=O)NC1CCC(=O)NC1=O c1(C(N(CCN(C(c2nccc(OC)c2N)=O)C)C)=O)nccc2cnn(C)c12 c1(C(=O)NCC2C(CNC(Cc3cc(C)on3)=O)C2)cc2ccccc2nc1O C(=O)(C1COCc2ccccc21)NCC1OCCN(C(CCC=C)=O)C1 CC1(CNC(C2CCCC(CC(F)(F)F)C2)=O)CCN(C(C2(C(N)=O)CC2)=O)CC1 C(c1ccccc1Cl)=C(C)C(=O)NCC(O)CN(C(=O)C(C)(O)C(C)C)C C1(C(=O)NCCCC(C)NC(c2c(OC)nsc2OC)=O)CCCCC(=O)C1 C(=O)(C(Cc1cnc[nH]1)NC(=O)CCCSC)NCC(COC)O c1(OCC)ccc(N2CCN(CCC(C)(C)CNC(=O)OC(C)(C)C)CC2)c(F)c1 c1(C(=O)NC2C3CN(C(c4c(C)nn(C)c4C)=O)CC32)coc2c1CS(=O)(=O)C2 N1(C(Cc2ccc(C(C)=O)cc2)=O)CC=C(CNC(C2C(C)(C)C2(C)C)=O)CC1 C1(NC(c2c(C#N)cn[nH]2)=O)CCCCN(C(c2cc(C(F)F)cs2)=O)C1 C1(CNC(CCC=CC)=O)CN(C(c2cc(C)ccc2O)=O)CCC12CCC2 C(=O)(CC(C)C(=O)NCC1CCCN(C(=O)CC2CC(C)(C)CCO2)C1)OCC C1(NC(=O)NCCC(C)(C)c2ccccc2)CCCCC1CC1CC2CC1C2 CCC(C)(CCC(C)C)C(=O)NC1CCN(C(=O)C(CCC#N)C2CC2)CC1F C1(O)(CNC(=O)C2=CCCO2)CCN(C(=O)CC2(C(O)C(F)(F)F)CCC2)CC1 Cc1c[nH]nc1C(=O)NCCOC1CCN(C(=O)CCc2ccon2)C1 c1(C(N2CC(NC(c3n(CCC)nc(C)c3)=O)C2)=O)ccc2c(c1)C(=O)NC2 C(=O)(CC1=CCCCC1)NCC(C)(CO)NC(=O)CCC(=O)c1ccccc1 C(=O)(C1=CCCOC1)NCC(CC=C)NC(c1ccc(SC)cc1)=O N1(C(C(C)(O)C2CC2)=O)CCOC2(C1)CN(C(c1ccnc(C3CC3)c1)=O)C2 CC(C(O)C(F)F)NC(C1(NC(=O)CC(C)c2ccco2)CC(C(N)=O)C1)=O C(=O)(CCS(C)=O)NC1C(NC(c2ccc(C(C)(C)C)[nH]2)=O)CCC1 c1(C(=O)NC(C)CNC(C2CCC(F)(F)CC2)=O)cc(N=S(C)(C)=O)ccn1 C(Cc1ccc(Cl)cc1)(CC(=O)NC1CC(F)(F)C1)NC(C(C)O)=O Cc1cnn2ccc(C(N3CC(NC(=O)CCc4ccc(F)cc4F)C3)=O)nc12 C1(C(=O)Nc2nc(COC)oc2)CC(C)CN(C(=O)CC2CCCC2)C1 CCC(CC(=O)N1CC2CC1(CNC(c1cc(C)nn1C)=O)C2)C1CC1 c1(OC)cc(OC)c2cc(C(=O)NC3(CF)CCN(C(=O)CSC)C3)[nH]c2c1 N1(C(C2(CC)CCOC2)=O)CC2CC(C1)CN(C(c1nc3c(s1)COCC3)=O)C2 CCC(CCC(=O)N1C2CCC(C2)C1CC(N1CC2CC1CC2CF)=O)OC CC1CN(C(C2CN3CCC2C3)=O)CC(C(N2CCC(CC(F)F)C2)=O)O1 C(=O)(C#CC(C)(C)CNC(c1ccn(CCC)n1)=O)N1CCC(O)(CC#C)CC1 C1(C(=O)NC2CN(CCC)C(=O)C2)CCN(C(=O)CC2(CO)CC2)CC1(C)C C1(CNC(C(CC)F)=O)CC2(CCOCC2)CN1C(c1cc(Br)ccc1C)=O C(=O)(CCC(C)C#N)NCC(CC)NC(c1cnc(-c2cccnc2)s1)=O c1(OC)cc(C(N2CCC(C)(NC(c3cnc(C(N)=O)cn3)=O)C2)=O)cc(C)n1 N1(C(C(=O)NCC(F)F)CC2C=CCC2)CCCCC1c1ccc(F)cc1 c1(CCCC)ncoc1C(=O)N(CCCNC(=O)CC1CCC(C(F)(F)F)O1)CC c12ncccc1C(=O)N(C1(C(N(C)C)=O)CC1)CCN2.C(CCF)O.C(=O)C1CC1 CC(F)(F)CCC(=O)NCc1cc(C(=O)NCc2c(F)cccc2F)ccn1 c1(-c2ccc(C(C)=O)o2)ccc(C)nc1C C(=O)(CC1=CCN(C)CC1)NC1(CN(C(c2cnc(C)[nH]2)=O)C)CC1 c1(C(N2C(C(C)NC(=O)C#CC(C)(C)O)CCCC2)=O)ccc(S(N)(=O)=O)s1 N1(C(Cc2sc(C)c(C(C)C)n2)=O)CC2(CCCC2)C1CNC(=O)CCC(C)C C(=O)(CCC(C)(F)F)NCC(CCNC(CCCc1ccc(C)cc1)=O)O c1(CN(CC(=O)NC(C)CCCNC(C23CC(C)C2C3)=O)CC)cccc(Cl)c1 C(=O)(CC(C)C(C)(C)C)N(CCNC(C(C1CCC(C)(C)CC1)C)=O)CC1CC1 C12(CCNC(COc3c(C)cccc3)=O)CCC(C1)N(C(c1ccnn1C)=O)C2 C1(CCNC(=O)Cc2ccc(F)cn2)CC(F)(F)CN1C(c1cnns1)=O CN1CC(NC(c2cn(CNC(C3(n4nccn4)CC3)=O)cn2)=O)CC12CCC2 C1(CNC(C2CC2F)=O)C2CN(C(c3ccn(CCF)n3)=O)CC12 C1(C)(COC)CCN(C(C2CC(O)CN2C(=O)CC2OCCC2(C)C)=O)C1 c1(C(=O)NC(C2CCCN(C(=O)COCC3CC3)C2)C)cc(F)c2cc[nH]c2c1 N1(C(CCCC#C)=O)CC=C(CNC(=O)CCc2cnc(C)nc2O)CC1 C1(NC(C2(C)CCN(C(c3c(C)nc(C)s3)=O)C2)=O)CN(C)C(=O)C12CC2 C12(CN(C(=O)NC(CC(C)C)CN3CCOCC3)C3CC3)CCCC1C2(F)F c1(C(=O)NCC(C2CCC2)NC(c2ccnc(OC)n2)=O)ncc(C#N)cc1C CC1(C)CC(NC(C2(c3cccc(Cl)n3)CC2)=O)CN(C(=O)CCCN=[N+]=[N-])C1 C(=O)(C1CCCc2scnc21)NCC1N(C)CCN(C(C2=C(C)OCC2)=O)C1 N1(C(C(=CC2CCCC2)C)=O)CC2CCC(C1)N2C(=O)C(C(C)C)n1cccc1 O=C1CC(C(N2CC(C(=O)NCCNC(=O)CC3CCNC3=O)C2)=O)CN1 CCC(C)(C)C(O)C(=O)N(C)CC1CN(C(c2[nH]nnc2C)=O)CCO1 c1(C(N2CC(CNC(CC(C=C)C)=O)OCC2)=O)cncc(O)c1Cl N1(C(C2CCN(OC)CC2)=O)CC23CCCCC2(C1)CN(C(c1ccco1)=O)C3 C1(C)(C(=O)NCCCN(C(=O)CP(C)(C)=O)CC)CC=CCC1 N1(C(C2(CC)CCCC2O)=O)CC2C=CC1C(C(=O)NCC#CC(F)(F)F)C2 c1(CCCC)ncccc1F.N1(C(N(CC(=O)N)CCC)=O)CC2CC2C1 c1(C(=O)NC(CC)CNC(=O)C=C(Cl)Cl)ncnc(OC)c1F C(CC(=O)NCC1CCCC(O)C1)(C(F)(F)F)NC(c1c(C)n(C)nn1)=O Cc1cn(C)nc1C(N1CCC(C)(CNC(=O)C(O)C(C)C)C1)=O c1(C(=O)NC(CNC(CN(C2CCCCC2)C)=O)C2CC2)ccc(F)cc1O c1(C(N2CC(OC)(CNC(=O)CC3CC(C)=NO3)C2)=O)cccc2[nH]nc(O)c12 c1(CC(=O)N(C2CCC(n3cc(C(C=C)(C)O)nn3)CC2)C)nn(C)c(C)c1Cl c1(N(CC(=O)N(C(CNC(C(C2CC(F)(F)C2)OC)=O)C)C)C)ccnc(Cl)n1 n1(CC)ncc2cc(C(=O)NCC3C=CCN3C(C3CCCN3CC)=O)cnc12 C1(C(=O)NC(C)C(C)O)(NC(C(SC)SC)=O)CCC(C)(C)C1 C1(CCNC(CCC)=O)CN(C(C2(C)COC2)=O)CC(C)O1 C(CC(O)CNC(=O)CCC=C(C)C)NC(C(C1CCC1)OC)=O c1(OC)ccnc(C(N2CCC(Br)C2)C(=O)NC2CCCCC2)n1 c1(C(=O)NC(CC=C)C2CC2)cnc(CNC(C2COC(C)C2)=O)nc1 C(CNC(=O)Cc1cncc(Br)c1)(C(C)(C)C)NC(C(=O)NCCOC)=O c1(C(N2CCC(C)(NC(C3CCCN(CC)C3)=O)C2)=O)cnc2ccnn2c1O c1(C(=O)NCC(CNC(C#CC2(CC)COC2)=O)(C)O)ccc2sc(O)nc2c1 C1(CNC(c2c(N(C)C)cncc2)=O)CN(C(c2cc(Cl)cn2C)=O)CC12CC2 CC1CN(C(=O)Cn2cncn2)CC1NC(c1ccc(O)c(C(C)(C)C)c1)=O c1(C(C2CCCCC2)NC(=O)NC2(CCOC)CC2)cc(F)c(F)cc1Cl c1(CC)nc(=NC(=O)N2CCN(CCCN3CCc4ccccc43)CC2)n(C)[nH]1 C1(CNC(CCN(C(CCC)C)C)=O)CCCC(c2ncccc2Cl)C1 c1(-c2cn(CC3CN(C(c4nc(CC)oc4)=O)C(CO)C3)nn2)nccc(C)n1 Cc1c(C(=O)NCC2CCCC2NC(C2CC3C=CC2O3)=O)ccn1C1CC1 C1(CNC(c2cnn(-c3ccccc3)c2F)=O)C2CN(C(C3CC(O)C3)=O)CC12 N1(C(COC)=O)CCC2CC2(NC(c2cc3ccncc3s2)=O)CC1 c1(C(=O)OCC)cc(C(N2CC3CC2C3NC(=O)CC2CC(C)(C)C2)=O)[nH]c1C Cc1nc2ccc(C(=O)NCC(CO)NC(C3C=CCC3)=O)cc2s1 N1(C(C2CC(CCNC(C3C(CC)CCC3)=O)C2)=O)CCCC2(CC1)CC2 N1(C(=O)NCc2ccc(SC(C)C)o2)CC(N(C)C)C2(CC2)C1 N12CC(C3CCCN(C3)CC1=O)C2.CCC(CC)C(=O)NC1CCC(OC)C1 C=CCC(CNC(=O)C(C)COC)C(=O)N1CCC(C)(F)CC1 N1(C(=O)CN2CCC2)CC(C(=O)Nc2cccc(C(N)=O)c2)C2(CCOCC2)C1 c1(N2CC(C)OCC2)ccncc1S(=O)(=O)NC(=O)NC1CCC(CO)C1 C1(C(=O)NC2(C(=O)NC)CC2)CC2(CCN(C(C3CC3C(=O)NC(C)C)=O)CC2)C1 Cc1cccc(CCC(=O)NC(C2CCNCC2)C(N)=O)c1 C1(C)(C(=O)NCCCN2CCN(C(C(C)(C)O)=O)CC2)C2CCC(C2)C1(C)C N1(C(c2cc(C(C)=O)oc2)=O)CC2C(N(C(=O)C(c3ccc(F)cc3)C)C)C2C1 c1(C(=O)NCC(CNC(c2cnn(CCF)c2)=O)CO)cnn2c1CCCC2 C12(C(=O)NCCC3(O)CN(C(Cn4ccc(C)n4)=O)C3)CC(CO1)C2(C)C Cc1oc(Br)cc1C(N1CCC(C(C)NC(=O)C(F)=CC2CC2)CC1)=O CCC(CC)CC(F)C(=O)N1CC(C(=O)NCc2cccc(Cl)n2)(SC)C1 C(=O)(CCCC(=O)NC(C)(C)C(C)NC(=O)CC1OCCC1(C)C)NC(C)C c1(OC)ccc(NC(=O)CCC(C)(C)NC(=O)CC2C(=O)NN=C2C)cc1C C1(NC(C(CCC)OCC)=O)CC2CCC1CN(C(=O)Cc1ccsc1)C2 C(=O)(C1=CC2CC(C1)CC2O)NCC1(NC(CCCC)=O)CCC1 c1(C(=O)NCC(CC)NC(C2CC23CCCC3)=O)cc(N)cc(O)c1 C(N=c1[nH]cnc(NCCN2CCNC2=O)c1C)C1CCC(OC)CC1 Cc1noc(C)c1C(C)C(N1CCCC1c1ccccc1Cl)=O c1(C(N2C(CNC(c3c(C(C)C)onc3)=O)C(C)CC2)=O)cnc2n1CCC2 c1(OC)cc(C)sc1C(=O)NC(C)CCN(C(=O)CSc1nccs1)C c1(C(c2nnnn2Cc2cccs2)NC2(C)COC2)cc(Br)ccn1 C1(NC(C(F)=CC)=O)(COC)CCN(C(c2ccccc2)=O)C1 CC1CN(C(=O)OC(C)(C)C)CC(C)N1C(=O)Nc1n[nH]c2c1CCC2 N1(C(Cn2c(C)ccn2)=O)CC(C(=O)N(CCN2CCCC2)CC#N)CC(F)(F)C1 C1(NC(C=CCC)=O)CN(C(=O)CC(C)n2cc(Br)cn2)CC1OC c1(CCC(=O)NC2CC(N(C)C(C3C4CCCC34)=O)C2)cccc(C(N)=O)c1 C1(NC(C(C2CCC2)OCC)=O)CN(C(=O)Cc2cnn(C)c2C)CC1C C(c1ccc(F)c(C)c1)=CC(=O)NCCC(C)(C)NC(C(C(C=C)C)C)=O N1(C(c2cccc(OC)n2)C(=O)NC2COC2)CCSCC(CO)C1 c1(C(N2CC3CCN(C(=O)Cn4cccn4)C3C2)=O)cc(Cl)cc2ccncc12 C1(NC(CSC)=O)CCC2(CCCN(C(c3ccc(C#N)c(O)c3)=O)C2)C1 C(c1sccc1Br)=CC(=O)NC(Cc1n(C)ccn1)C(F)F C12(CC)CC(NC(=O)CC(C)NC(=O)C(CCSC)NC=O)(CO1)C2 CCC(CC)C(=O)NC12CC(CNC(c3cnc(C)[nH]3)=O)(C1)C2 N1(C(=O)N(O)Cc2cn(C3COCC3O)nn2)CCCCC1c1ccc(Cl)nc1 c1(NCC(=O)NCCCOCC)cc(NC(C)=O)ccn1 CC1CN(C(C2CC(C)OC2C)=O)CC1NC(c1ncnn1C)=O Cc1cc(C(=O)NON2CCCC(n3nccn3)C2)c[nH]c1=N C1(CNC(C(C)=C2CC2)=O)(NC(c2cc(F)cc(F)c2)=O)CC2CCC1C2 C(=O)(C1CCCc2ncnn21)NC1CN(C(c2ncn(CC)n2)=O)CC1O C1(NC(COCC(=O)OCC)=O)CC(O)CN(C(=O)CCCOCCOC)C1 N1(C(c2nc(OCC)oc2)=O)CCC(CO)C(NC(=O)C(C)=C2CCCC2)C1 C(C(C)C)(C(O)C(=O)NC1CC2CCC(C1)N2C(C1CCC1C(C)(C)C)=O)OC C(=O)(CC(C)(C)C(F)F)NC1(C(N2CC(C(=O)OCC)C2)=O)CC1(C)C N1(C(CSCC#C)=O)CCC2CN(C(c3cn(CC)nn3)=O)C2C1 C(=O)(C1=NOC(C)C1)NCC(CO)NC(c1c(-c2c(OC)cccc2)nsc1)=O c1(CN2CCC(CNC(=O)NC3C(C)CCCC3)CC2)cc2ccc(Cl)cc2[nH]1 Cn1nc(C(=O)NC2CC(CNC(=O)Cc3ccon3)CC2O)cc1O N1(C(C(C=C)C)=O)CC2(C(=O)NCc3cnc(C)[nH]3)CC1CO2 Cc1nc2ccc(C(N3CCOCC(CNC(=O)C(O)C4CC4)C3)=O)cc2o1 N1(C(CC(c2ccccc2Cl)C)=O)CC(CNC(C2(F)CC2)=O)CC12CCC2 N1(C(c2c(CC)noc2)C(=O)NC(c2ccccc2)C)CC(C)C(C)C1C C1(C2CC2)(CNC(C2(C)CCNC2=O)=O)CCN(C(C2CCC=CO2)=O)C1 C12CCOC3(CCN(CC3)c3nnc(n3CCSC)OOC1)C2.COCC N1(C(C(OC)OC)=O)CCCCC1C(=O)NCC1(C)CCC1 c1(C(N(C)CC2CC(F)CN2C(=O)COCC2(F)CC2)=O)ccn(C)c(=O)c1 C1(C(F)F)(NC(C2CN(C3CCC3)C2)=O)CCCN(C(c2cccnc2)=O)C1 c1(CN2CCC(C(N3CCC4(CCOC4)C3)=O)C(O)C2)ccc2occc2c1 C(=O)(C(CC(F)F)N(C(=O)CCC1(C)CC1)C)NCC(c1cncnc1)C c1(C(N2C(C)C(NC(=O)CC3C=CCC3)C(C)CC2)=O)cnn2c1C(=O)NCC2 CCCS(=O)(=O)C(C)C(=O)N1CCC(NC(=O)Cc2ccc(S(N)(=O)=O)cc2)C1 c1(C(=O)NC2(C)CCN(C(c3nccc4nn[nH]c34)=O)C2)cccc2[nH]ccc12 N1(C(C(CCC)NC(=O)Cc2ccc(F)cc2)=O)CC2(CCC(=O)O2)C1 N1(C(c2c(C)ocn2)=O)CCCC2(NC(=O)C(O)CCn3cncn3)CCCC12 c1(C(=O)NCC2(C)CCN(C(c3ncc[nH]c3=O)=O)C2)cc(=N)[nH]c(=N)[nH]1 Cn1cc(NC(=O)CC2CCCCC2NC(c2sccc2F)=O)c(O)n1 CC1CN(C(c2csc(CO)n2)=O)C(C)CN1C(c1nocc1Br)=O c1(C(C)(C)C)n[nH]cc1S(=O)(=O)NC1CCC=CCCC1 C1(NC(c2ccsn2)=O)CCCCC12CCN(C(=O)C(F)(F)C(F)(F)F)CC2 N1(C(c2ccc(C)cc2)=O)CCCN(C(C2(F)CCS(=O)(=O)C2)=O)CC1C Cc1ccc(O)c(CC(=O)NC2(C)CCN(C(C3(c4cc[nH]n4)CC3)=O)CC2)c1 C(=O)(C(C#N)C(C)C)N(C(CN(C(C1(OC)CCCCC1)=O)C)C)C C=CCCC(C(=O)NC(C1CCCC1)CO)NC(=O)C(C(C)C)SC CC1(C)CCC(C)(C)N(C(CCCCCO)C(=O)NC2CC(F)(F)C2)C1 C1(C(=O)NCC(CC)(CC)NC(=O)C(C)C2CC2)CCCCC(=O)N1 Cc1ccc(S(C)(=N)=O)cc1CNC(c1c[nH]c2ccccc12)=O Cc1cc(C(=O)N(C(C)CNC(c2ncccc2Br)=O)C)ncc1F c1(OCCCC(=O)NC(C)CN(C(=O)CCc2cc(Cl)no2)C)ccc(F)cc1 c1(C(N2CC(CN(C(C3(CCC=C)CC3)=O)C)OCC2)=O)csc(S(N)(=O)=O)c1 c1(COCc2onc(CC(=O)OCC)n2)ccc2c(OC)n(C)nc2c1 C1(C(C(C)Oc2c(CCC=C)cccc2)=O)CCS(=O)(=O)CC1.C1(=O)CO1 c1(C(=O)NC2CN(C(c3c(CC)[nH]nc3Cl)=O)CC(O)C2)ccc(F)c(C#N)c1 C#CCCC(C(=O)NC(C)CC1=CCCCC1)NC(C1CC12CCCCC2)=O c1(CCCC(=O)NC(CNC(c2ccc(Br)cc2)=O)CO)ccc(F)cc1 CCCCCCCCNCc1ccoc1 Cc1c(C(N2CC3CCC(C2)C3C#N)=O)oc2ccc(Br)cc12 N1(C(C)=O)CCCC1C(=O)NC1CCCC1CSc1nncn1C(C)C C1(NC(c2n(C(C)C)nnn2)c2ccsc2Br)CCC2(CCCC2)CC1 C1(NC(c2cc(C)c(C)[nH]2)=O)COCCN(C(c2ccc(Cl)c(C(F)F)c2)=O)C1 C(=O)(C1=Cc2cccc(Br)c2OC1)N1C(CNC(C(C)=CC)=O)C(CC)CC1 c1(C(N2CC(C)C(NC(=O)CCC3CCCCC3)C2)=O)ccc(Br)c(F)c1 C1(N(C)C(c2ccoc2)=O)CN(C(C2(C)CCCS2)=O)CC1F CC1=C(C(=O)NCC2(C)CN(C(c3ccc(Cl)c(F)c3)=O)CC2C)CCC1 c1(C(=O)NC(CCNC(c2c(C)oc(Cl)n2)=O)C)c(C)nn2c1CCCC2 C1(C(N(C)CC2N(C(c3cc(C)[nH]c3)=O)CCOC2)=O)CCOC(=O)CC1 C=CC(CCC)CC(=O)N(C1CCN(C(c2cn(C)cn2)=O)C1)CCO N1(C(c2ccc(C)o2)=O)CC2CCC2(CCNC(c2c(C)cnn2C)=O)C1 c1(C(C(=O)NCCC#N)N(C2CCCC2)CCF)csc(-c2cccs2)n1 C1(NC(=O)C=CC2CC2)CCN(C2CCCC2)CC1 C(=O)(C(C)(C)CCC(=O)NCC1(F)CC(NC(=O)CCC(C)CN(C)C)C1)OC c1(C(N2CC(NC(C3(CC4CC4)CC3)=O)C2)=O)cc2ccc(F)cc2nc1O N1(CCCc2onc(C)n2)CCOCC(NC(=O)CC2CCCS2(=O)=O)C1 CN1C(=O)CC(CNC(c2cc(-c3cccs3)on2)=O)C1=O Cc1nc(C(=O)NC2CC(CC(=O)NCC(C)(C)C(C)(C)O)C2)cc(O)n1 Cc1ccc(S(=O)(=O)N2CCOC(C(=O)NC(CO)C(C)O)C2)c(F)c1 N1(C(c2c(C(C)C)cccc2)=O)CCC2(CCCC2C(=O)NCCCCCO)C1 Cn1ncc2c1CCCC2NC(=O)C(=O)NC1COc2ccc(F)cc2C1 CN1C(=O)CC(NC(=O)NC2(c3ncco3)CCC2)C1c1ccccc1 c1(OC)cccc([N+](=O)[O-])c1C(N1CC2C(C1)N2C(=O)C(C(C)O)N(C)C)=O CCC(CC)CC(F)C(=O)N1CCN(C)C(C(=O)NC(c2cc(C)no2)(C)C)C1 C1(C(=O)NC(C(C)C)CNC(c2ccnn2CC#N)=O)CCC2CCC1O2 N1(C(C2COCOC2)=O)CC2CCCC(O)C2C1.C=C1CC(C(=O)N)(CO)C1 C(=O)(CCC(C)(F)F)NCCCC1N(C(c2c(C)ncs2)=O)CCCC1 c1(C(=O)NC(c2ccnn2C)C(=O)Nc2c(CC)csc2)cccc(OC)c1 C1(C(C)C)CC(C(N2CCCC(CN3CCC(CO)CC3)C2)=O)CCO1 C12(NC(c3cnc(CNC(CC(C)(C)C4CC4)=O)nc3)=O)CCC(CC1)CC2 Cc1c(C(=O)NCCC2CN(C(=O)CCC3CCCOC3)C2)nn2c1CCCC2 CC1(C(=O)NC2CCCC(CNC(c3coc(Br)n3)=O)C2)CCCCO1 C1(OC)CC(CNC(=O)C(C)CSC)N(C(=O)Cc2[nH]cnc2C)C1 c1(CCC)ccc(C(=O)NCC2(CNC(c3ccc(C(C)=O)[nH]3)=O)CCC2)[nH]1 C(=O)(CC(C)CC(C)C)NC(COCC)C(=O)N(C)Cc1cnn(CC)c1 CCC(C(=O)NC(c1ccc(C)s1)C)NC(c1ocnc1C(C)C)=O N1(C(c2cc3cc(c2)C(=O)N3)=O)Cc2cncnc2C1.CN(C)CCN(C)C C(C(C)(C(C)C)NC(=O)COC1CCCOC1)NC(CCn1ccc(C)n1)=O CCCCCC(O)CC(=O)NC(CNC(=O)Cc1cncnc1)C1CCC1 C1(C(=O)NC(C)(C)CCNC(c2sccc2C(F)F)=O)CC2CCC(C1)C2O c1(OCC)ccc(C(=O)NC2CCN(C(=O)C(C)CCO)C2(C)C)cc1C C1(CN(C)CC2CC2CO)CCN(C(=O)CCc2cc[nH]n2)CC1 N1(C(c2cn(CC)nn2)=O)CCCC(C2(NC(=O)CCC=CC(C)C)CC2)C1 CCCCC(O)C(=O)N1CCSCC1CCNC(c1cccnc1NC(C)C)=O N1(C(c2c(NCc3cc(C)[nH]n3)ccs2)=O)CCN2CCCC2C1 CC1(NC(=O)CC2CC3CCC2CC3)CCCN(C(c2cncnc2)=O)C1 c12ccc(nc1)OC1CCN(C1)C2=O.C(C)(CC(=O)NCCNC(C)C)OC c1(C(=O)NCC(C)N(C(=O)CCc2cccc(O)c2)CC)cccc2c1CCC2 C1(CNC(c2nc(COC)sc2)=O)(NC(c2cn(C)nn2)=O)CC2CCC1C2 C1(CNC(CN(CC)CC)=O)COCCN(C(=O)C2CC2)C1.C(C)SCC CCC(CCc1ccccc1)C(=O)NC(C)(C)CN(C)C(C1(C)CC1)=O c1(C(=O)NC(C)CC(C)NC(C2CN3CCN2CC3)=O)cncc(P(C)(C)=O)c1 N1(C(CC(=O)NCC)=O)CC2CC1CC2CNC(=O)CCC(=O)NC1CCCC1 c1(N(c2ncccn2)CC)nccnc1C Cc1ccc(C(C2CCOC2)NC(=O)CSC(F)(F)F)cc1.C12CCCN1C2 C1(CC)CCN2C(C1)C2=O.C(C(C)CC(=O)NCC(C)(C)CN(C)C)OC N1(C(CC(COC(C)=O)(C)C)=O)CCN(C(C2CC3(CC3)CO2)=O)CC(C)C1 c1(C(=O)NC(COC)C2(C)CC2)ccc(F)cc1CSc1ccccc1 N(C1CCOCc2c(Br)cncc21)C(=O)NC1(N)CCC1 CC1CCCn2c(C(N3CCCC(N(C)C(C4(F)CCCC4)=O)C3)=O)cnc21 c1(C(=O)OC)c[nH]c(=NCCCC(C)NC(=O)C2=C(C)CCCC2)c(C)n1 CC1CCCc2ncc(C(=O)NC(C)(C)C(C)NC(=O)CCN3CCCC3=O)n21 N1(C(C(CC)OC)=O)CCOC2CCN(C(c3ocnc3C3CC3)=O)CC12 C(=O)(C1=NN(C2CC2)C(=O)CC1)NC1C(CC)N(C(=O)C2=CS(=O)CCC2)CC1 C1(CC(=O)N(CCCN(C)C)CCNC(=O)C(C)(C)C2(O)CCC2)(OC)CCCC1 C1(NC(c2c(OC)n(C)nc2)=O)CCN(C(=O)Cc2cn(C)cn2)CC(C)(C)C1 C1(CNC(c2c(CC)cno2)=O)CCN(C(=O)C(C2CCCC2)OC)CC1 N1(C(C2CCC(=O)N2)=O)CCC(CO)(CNC(C2(C(F)(F)F)CCC2)=O)C1 N1(C(c2snc(C)n2)=O)CCCC12CCN(C(c1n[nH]c(C3CC3)c1Cl)=O)C2 N1(C(c2c(C)cc(CNC(c3ccsc3C#N)=O)o2)=O)CCC(C)(C2CC2)C1 c1(CNC(N2CCN(C(C)(C)C)CC2)=O)csc2cc(Br)ccc12 c1(C(N(CCN(C(c2cc(C(C)C)nn2C)=O)C)C)=O)ccc2c(c1)OCCO2 c1(NC(CC)CCCO)ncc(S(=O)(=O)NCCc2nccn2CC)cc1Cl c1(OC)ccc(S(=O)(=O)N2CC3(CCN3C(=O)C(n3nc(C)cc3C)C)C2)cn1 C1(O)(CNC(C2CC(C(N)=O)C2)=O)CCCN(C(c2ncccn2)=O)C1 c1(C(=O)OC(C)C(=O)Nc2ccccc2)cccc2c1OC(C)(C)CC2 C(CC(=O)NCC1COCC(C)O1)(C(C)C)NC(C=Cc1cc(C)no1)=O N1(C(CCN(CCC)C)=O)CC(NC(C2(C)CC3CC3C2)=O)C(C)(C)C1 CCC(O)C(F)(F)C(=O)N(CC(N1CC(O)CC1(C)CO)=O)CC1CC1 c1(C(=O)NC2CCCN(C(CC=C)=O)C2C)ccc(SCC)c([N+](=O)[O-])c1 C1(NC(=O)CCOCC2CCC2)CCCC1NC(c1sccc1Cl)=O C1(CNC(CC(C)NC(N)=O)=O)C2CN(C(=O)C(CCc3ccco3)N(C)C)CC12 CC(CNC(c1csc(CS(C)(=O)=O)n1)=O)(CO)NC(c1coc(C2CC2)n1)=O c1(CNC(=O)CNC(C2CC2NC(c2ccnc(O)c2)=O)=O)cccc(F)c1Cl c1(C(=O)NC(C2CN(C(C3CCOC(=O)CC3)=O)CCO2)C)cc2n(n1)CCO2 C(=O)(C1CC(=O)c2ccccc21)N1CCN(C(c2cnc(O)cc2O)=O)CCC1 N1(CCCNC(C(CSC)O)=O)CCN(C(C2CCC2(C)C)=O)CC1 c1(C(N2CCC(F)(CC(=O)NCCCc3n(C)ncn3)C2)=O)ccnc(O)c1F C1(NC(=O)NC)CC2(C1)CC2C(=O)N(C1N(C(C)=O)CCC1)CCO.C(C)(C)N C1(F)(CNC(c2c(C)coc2)=O)CCN(C(=O)CC(C)(C)C)C1 c1(C(N2CC3C(NC(c4ccn(C)n4)=O)(CCC3)C2)=O)csc2ncnc(O)c12 n1(C(c2n(CC(=O)OCC)nnn2)NCC(F)C2CCC2)cc2ncccc2n1 C(C)(CCC(C)(C)C)NC(c1ccc(CNC(C(C(C)C)SCC)=O)s1)=O c1(C(N2C(C)CC(NC(c3ccn(CC)n3)=O)C2)=O)cc(F)cc(Br)c1F C=CCC(CC=C)C(=O)NCC(CO)NC(c1ccn(C)c(=O)c1O)=O C12(C(N3CCN(C(c4c(CC)nnc(C)c4)=O)CC3C)=O)CCC(CC1(F)F)C2 CCC(C)CC(=O)C(=O)N1CC(C(O)C(N2CC3CC3(C(=O)NC)C2)=O)C1 C1(C(=O)NCCCCC2CCN(C(C(CCC)OC)=O)CC2)Cc2nncn2C1 Cc1cc(C(c2nnnn2CCCF)NCCOC2CCOC2)[nH]c1C C=CCC(C(=O)NCc1csc(CNC(C2CCN2S(C)(=O)=O)=O)n1)C(C)C C(=O)(CC(C)CNC(c1nc(=N)[nH][nH]1)=O)N(C1CCCCCC1)CC Cc1cccc2nc(C(N3CCC(C)N(C(=O)C(C)CF)CC3)=O)cn12 C1(C(=O)NCC2(C(N(C(CC(=O)OC)C)C)=O)CC2)CC(C)(C)CN1C C1(NC(C2(C(N)=O)CCC2)=O)COCC1C(=O)NCC(Cl)=CCl n1(CC(=O)NC(CNC(c2cnn(CCOC)c2C)=O)C)cnc([N+](=O)[O-])c1 N(C1CCCc2cc(SC)ccc21)C(C(CC#C)NC(C)C)=O N1(C(C2C(C)(C)CN(C(c3c[nH]c(=O)cn3)=O)C2)=O)CCC(C2CC2)CC1 N1(C(c2c(COC)ocn2)=O)CC2CCC1CN2C(=O)Cc1ccc(F)cc1Cl c1(C(=O)NCC(CC=C)NC(c2ccccc2SC)=O)cncc(C(F)(F)F)n1 Cc1cc(NCC(F)C2CCC2)c(S(N)(=O)=O)c(F)c1 CCCCCCCCN(C(=O)C(CNC(c1ccc(C)cc1C)=O)C(C)C)C c1(C(=O)N(c2ccc(Br)cc2)CC2CC2)c[nH]c2cc(F)c(F)cc2c1=O C1(NC(c2cccc(C(C)=O)n2)=O)CN(C(=O)CCNC(C)=O)CCC12CCC2 C(C1CCCCC1)=C(C(=O)N(C1CCN(C(=O)CCNC(C2CC2C)=O)C1)CC)F N1(C(C(C)C)=O)CC2CN(C(=O)C=Cc3cncs3)CCC2(CO)C1 N1(C(=O)NC(CCOC)CF)CCOc2cc(F)cnc21 N1(C(C(CSC)C)=O)CCC2(NC(=O)C=Cc3c[nH]nc3C)CCCC12 C1(NC(CCCC)=O)CC(O)CN(C(C2C=CC=CC=C2)=O)C1 c1(C(N2CCC3(NC(C(=O)N(C)C)=O)C(CC2)C3)=O)cc(F)cc([N+](=O)[O-])c1 C1(NC(c2c(CC)con2)=O)CC(O)CN(C(=O)C=CCF)C1 c1(C(=O)NCC(CCNC(C(C2CC2)SC)=O)O)cc2n(n1)CC(C)(C)CO2 C(C(C)CC(=O)NCCCc1cc(C)no1)NC(c1ccn(CC)n1)=O C1(C)(C(=O)NCCCCC2CN(C(C3CCN(CC)C3)=O)C2)CC2CC2C1 c1(C(C)OC)cc(Cl)n[nH]c1=NC(=O)c1cccc(CNC(C)=O)c1 C(=O)(C1=CS(=O)CCC1)N1C2(CNC(C(c3ccc(CC)cc3)C)=O)CC(C1)C2 N1(C(C(C)(Cl)Cl)=O)CCC2(CC(NC(=O)CC3CCCCC3O)C2)C1 N#Cc1ccc(N2CCC23CN(C(C2CC4(CC(=O)C4)C2)=O)C3)cn1 C#CCC(CC(=O)NCC1(C)CCCS1)NC(C1CC(C)(C)CO1)=O c1(C(N2CCCC2CNc2cccc(O)n2)=O)ccc(Cl)nc1C(F)(F)F N=c1nc(CN(C2CCNC2)CCF)[nH]c(=N)[nH]1 c1(C(=O)NC2CC(F)(CNC(C3CC(OCC)C3)=O)C2)ccc(OC)c(F)c1F C1(NC(=O)CC=C(Cl)Cl)CC(NC(c2csc3cncn23)=O)C12CCC2 c1(C(=O)NCC(C)(C)NC(CCCCOC)=O)c(Cl)cnc(OC)c1Cl Cc1csc(C=CC(=O)NCCOCCOCCNC(=O)Cc2cnco2)n1 C=CCC(CCCCC)C(=O)NCC(N1CCN(C(=O)Cc2ccns2)CC1)=O n1(CCC(=O)NCC(C2CCN(C(C(CC)O)=O)CC2)F)cc[nH]c(=O)c1=O N1(C(C(COC)O)=O)CCN(C2CCCN(C(C3(C)CCCC3)=O)C2)C(=O)C1 N1(C(c2c(OC)ccc(CC)c2)=O)CC2CCCN(C(=O)C(O)CC(F)F)C2C1 C12(NC(c3c(C(C)C)nns3)=O)CCC(CC1NC(=O)CCCNC(N)=O)C2 C1(C(N(CC=C)CC)=O)CCCC1NC(=O)COCCOC Cc1ncc(C(=O)NC2CC(OCC(=O)N(CCCC(C)O)C)C2)c(=N)[nH]1 C1(NC2(CO)CC(OC)C2(C)C)CSC(c2ccccc2)=N1 c1(CN(C)C(C2C=CCN2C(=O)C2=CCCC2)=O)cc(Cl)ccn1 N1(C(C(C)N(C(=O)CC2CCC2)CC)=O)CCC(SC)CC1 CON=Cc1ccc(C(N2CC(CNC(=O)C(=O)NC(C)C)C(C)C2)=O)cc1 C1(CNC(CCSCC(C)C)=O)(OC)CCCN(C(=O)CCC2CCOC2)C1 C#Cc1cnn(C)c1C(N1CC2CC2(NC(=O)C(C2CCCCC2)OC)C1)=O N1(C(=O)NCn2ccccc2=O)CC(NC(c2ccc(I)c(Cl)c2)=O)C2(CC2)C1 C1(C2CCCOC2)(NC(c2cccnc2O)c2n(C(C)(C)C)nnn2)CC1 CCN=c1[nH]cc(C(=O)NCC(c2ccccc2)NC(c2csc(C)n2)=O)s1 c1(OC)cc(C(N2CCCC(CCNC(c3coc(Cl)n3)=O)C2)=O)c(Cl)cn1 C1(C(=O)OC2CC3(CCOC3)C2)COCCN(C(c2ccccc2)=O)C1 N(C(=NCCOC(C)C)NCc1ccnc(OC)c1)Cc1c(CC)cccc1.SCC C(=O)(CC(C)(C)OCCNC(C1CC1(C)C(C)C)=O)N(CC#C)C Clc1c(CN2CCC3CCC23)sc2ccccc12 Cc1ccc(C(N2CCCC(C(C)C(=O)NC(C)C3CC3)C2)=O)nc1 C12(C(=O)NCCN(C(C(=O)Nc3ccccc3)=O)C3CC3)CCCC1OCC2 c1(NC(Cc2cccc(C(C)C)c2)=O)ncnc2c1nc1n2CCOC1 c1(C(N(C2CC(NC(CC3(COC)CC3)=O)C2)C)=O)cc2c(F)c(C)ccc2[nH]1 N1(C(C=C(C)C2CC2)=O)CCC(NC(c2n[nH]c3c2CC2CC32)=O)C(F)(F)CC1 C1(CC(=O)N(C2CC(O)C2(C)C)CC)CCN(C(=O)C(C)=CCSC)CC1 C(=O)(C1=NOC(C)C1C)NC1(CC=C)CCN(C(c2c(F)ccc(F)c2N)=O)C1 Cc1cc(C(=O)NC2CC2NC(c2cnc(OC(C)C)s2)=O)c2occc2c1 C#Cc1cncc(C(=O)NCCCCC(C)NC(=O)Cc2conc2C)c1 N1(CCNC(C(C)N(C(=O)C(C)N2CC(C)C2)CC)=O)CCCC1=O C12(NC(c3n(C(C)C)cnn3)=O)CCN(C(=O)COCC3CC3)CCC1C2 C12(C(N3CCCC(C)(NC(C(C)OCC(C)C)=O)C3)=O)C3C4C1C1C2C3C41C CC1CN(C(=O)CC2CC(O)C2(C)C)CCN1C(=O)Cc1cnnn1C c1(C(=O)NCC2(OCC)CN(C(C3CC(C)OC3=O)=O)C2)[nH]c(C)cc1C c1(C(=O)NC(CC=C)CNC(c2csc(C(C)OC)n2)=O)ccccc1SCC c1(C(=O)NCC2CC(C)(F)C2)cncc(-c2ccc(C(=O)NCCF)nc2)c1 C1(NC(C(N2CC(NC(C(C3CCCC3)CC)=O)C2)=O)=O)CC2CC(CO)C1C2 C1(COC)(NC(=O)C(C2CC2)N(C(=O)CCc2ccn(C)n2)C)CCOC1 CCC(C)(C)CC(=O)N1CCC(CCNC(=O)Cn2nc(C(F)(F)F)cc2C)C1 C1(C)(C(=O)NC2(CC)CCCN(C(=O)CSC)C2)CCCC(F)(F)C1 c1(C(=O)Nc2cc(C)c(F)cc2F)cn2cc(-c3ccc(C#N)s3)ccc2n1 C(c1nc(C)c(C)[nH]1)=CC(=O)NC(CC)CN(C(=O)C1=COCC1)C C1(CNC(C(CC(C)C)C)=O)COC(C)(C)CN1C(c1ccc(F)cn1)=O N1(C(C2CC(C#C)(O)C2)=O)CC2(CCCC(CNC(=O)C(C3CC3)C3CC3)O2)C1 c1(C(N(C(C(=O)NCCCOCC)=O)C)C)ccc(C)nc1C CCCC(C)(O)CC(=O)NCC1(CNC(c2cnc(OC)c(C)c2)=O)CC1 C1(NCCC#N)CCc2n[nH]c(C)c2C1.c12cc(nc(C(C)C)n1)N1CCN2CC1 C1(C(N(C2CC(=C)C2)C2CCC2)=O)CC12CCN(C(=O)C(C#N)CCC)C2 C1(CN(C(c2ccccc2Cl)=O)CC)CCCCN1C(=O)CCOC1CCC1 N1(C(CC(C=C)CCC)=O)CC(C2CCCN(C(=O)Cc3cn(C)nc3C)C2)C1 N1(C(CN(CC)CC)=O)CCCC2(NC(=O)CCNC(C)=O)CCCC12 CC1(C)CC(=O)OC1CNC(=O)C(C)(C)C1CCN(C(c2ccc(O)cc2)=O)C1 C1(NC(C(=O)NC2CC2)=O)CN(C(c2cc[n+]([O-])cc2)=O)CCC1C(F)(F)F C(c1ccccc1)=CC(=O)NC(CNC(=O)CN(C1CCC1)C)C1CCC1 C1(F)(C(N(C)CC2N(C(C3C(C)C3C)=O)CCOC2)=O)CC2(CCC2)C1 C1(C(=O)NC2CCN(C(c3c(CC)oc(C)c3)=O)C2CC)CCCCC1C#N C1(O)(CNC(C2CCN(C(CC3(COC)CC3)=O)C2)=O)CC(C)(C)C1 CC(C)C(C(=O)Nc1ccccc1)Sc1ccccc1Cl Cn1ncnc1CCNCC(N1CCC(NC(=O)CNC(=O)CNC(N)=O)C1)=O C(=O)(C1=C(Cl)CCC1)NC1CC(NC(C2C3CC(=O)CC32)=O)C(O)C1 N1(C(C)=O)CCC(O)C1.c1(C(=O)NC)ccon1.C12CCC1CNC2=O N12CC(C3(CC3)C1)CC2=O.Cn1cncc1CC(=O)NC1CCOC1C(C)(C)C N1(C(c2c(C)ncnc2)=O)CC2CC3CC2C1C3NC(C1CCOCC1)=O C(=O)(C1CNC(=O)c2ccnn21)NC(CC)CN(C(=O)CCC(=O)NC)CC c1(C(=O)NC2CC(NC(=O)C(CC(F)F)C3CCC3)C2)coc2c(Cl)cccc12 C(=O)(C(=O)N=c1cc(C)o[nH]1)NC1CC(CCNC(C23CC(SCC)(C2)C3)=O)C1 C1(C(N(CC(F)C2CCC2)C(C)C)=O)(NC(=O)Cn2cnnn2)CCSC1 c1(C(=O)NC2CC3CN(C(CCC(=C)Cl)=O)C2C3)cc2occc2n1C c1(CC(N2C(C)(CNC(C3C(C)CCC3)=O)CCC2)=O)ccc(F)c(Cl)c1 C(C(CNC(=O)Cc1nc[nH]n1)NC(=O)CCc1cocn1)OC N1(C(C(CC)OC)=O)CCC2(CCN(C(c3ccnc(OCCO)c3)=O)C2)C1 O=C1COC2(CN1)CN(S(=O)(=O)c1ccc(NCC(Cl)(Cl)Cl)c(Br)c1)C2 CC1CCSCCN1C(=O)CC1(CNC(=O)C=C2CCOCC2)CC1 N1(C(=O)Cc2cc[nH]n2)CCC2CN(C(C3CC(F)(F)CS3)=O)C2C1 c1(NC(=O)C(F)(F)CC2CCOCC2)cc(N2CCNCC2)ccc1F CC1=C(C(=O)NCC2CCCCC2C(N2CCCC2C2CCCC2)=O)CCCO1 c1(C(=O)NCC2C=CCN2C(c2coc(Cl)c2)=O)ccc2nccnc2n1 c1(N2CCC(C(C)NC(c3cc(Cl)cc(Cl)c3)=O)CC2)ncnc2ncn(C)c12 N1(CC)CCOCC1CC(=O)NC(C)(C)CCNC(=O)Cn1cc(Cl)cn1 N1(C(COCCC)=O)C2CCC(C2)C1CNC(=O)C(=Cc1ccc(Cl)cc1)C c1(C(CN(C(=O)NC(CC=C)C)C)(C)O)cccc(Br)c1 C=CC1CN(C(=O)Cc2cnccc2C)CC1NC(c1sccc1CO)=O CC(C)C(O)CC(=O)NC1(CN(C)C(c2ccc(-c3ccccn3)s2)=O)CC1 c1(CN2CC(C#N)C(NC(=O)CS(N)(=O)=O)C2)c(Cl)ccc(Br)c1F C(=O)(CS(=O)(=O)CC(C)C)NCC(C)NC(c1ccc(OC(F)(F)F)cc1F)=O c1(C(N2CC3CN(Cc4cnc(Cl)cc4F)C3C2)=O)c(F)cccc1I C1(O)(C(C)NC(CC2CC(SC)C2)=O)CCN(C(=O)C2=CSCS2)CC1 CCCC(C(=O)NC1CN(C(C2(C)CCC(=O)C2)=O)C1)C(C)C c1(C(C)C)ccoc1C(=O)NC(Cc1cn[nH]c1)C(=O)NCc1cncs1 Cc1cncc(CCC(=O)N2CC(c3ocnc3CNC(=O)CCC(F)F)C2)c1 C1(=CC(=O)NC(CCOC)CNC(c2cc(F)c[nH]2)=O)CCC(C)CC1 c1(C(=O)NCc2n[nH]cc2Cl)snc(-c2ccccc2)c1Br C1(C)(CC)CCCN(C(=O)CC2CCCCN2C(c2csc(C)c2)=O)C1 c1(C(=O)NC2CC3CC(C2)N(C(c2ccc(O)nc2)=O)C3)cc2cnccc2[nH]1 Cc1cc(C)c(C(N2CC(NC(C3(C)CC3(F)F)=O)C(C)C2)=O)[nH]1 c1(C(=O)NC2(C(=O)NCCCN(CC)CC)CC2(C)C)nnn(C)c1C C(C(C)(C)OC)NC(CC1(COC)CC1)=O.C1(N=[N+]=[N-])(C(=O)NC)CC1 N1(C(CC2N(C(C(C)NC=O)=O)C3CCC2C3)=O)CCC2(CCCC2)CC1 CC1CCC(NC(=O)CCCCN2CCOCC2)CN1C(c1ccon1)=O Cc1cc(C)c(C=CC(=O)NC2CCN(C(=O)Cc3c[nH]nc3C)C2C)c(C)c1 C(CCF)(C(=O)NC1CC(n2ccnc2)C1)NC(C(C)OCCN(C)C)=O C1(NC(C(CCC)c2ccc(C(F)(F)F)cc2)=O)CN(C)S(=O)(=O)C1 N1(C(CC(COC)C)=O)CC2CCCC(C1)N2C(c1ccc(C)cc1F)=O Cc1cc(OCc2scc(C(=O)Nc3ccc(Cl)cc3Cl)n2)ccc1Br c1(CNC(C2(C)CCC(=O)C2)=O)nc(CNC(c2csc(Cl)c2)=O)cc(O)n1 C1(CN)CC2(CCN(C(=O)CC3CCC(O)C3)CC2)C1.C1CCCNC(=O)N1C c1(C(=O)NC(C2CCCN2C(=O)C(F)=C(C)C2CC2)C)cccc(C2CC2)c1 c1(NC(=O)NC(C(CC)C)CO)c(O)ncnc1C N1(CC(C(C)=O)C)Cc2ccccc2Sc2ccccc21 CN1CCC(C(N2CCCC2CC(=O)NCC2CNC(=O)O2)=O)CC1 C1(C(=O)NCC(CCOC)O)CC2(CCN1C(C1CC3CC3C1)=O)CC2 C(C(CC(F)(F)F)NC(=O)C(=O)N(CC(C)O)C)OC C1(C(C)(C)O)CCC(C(=O)NCC(C2CCCC2)NC(=O)C(Cl)=CCl)CC1 c1(C(=O)NCCC2(OC)CN(C(C3CCCCCC3)=O)C2)cnn2c1CCCC2 N1(CCC(=O)NCC2CCCC(NC(c3cccnc3)=O)C2)CCCS1(=O)=O Cc1cnc(N2CCCC2)nc1SCc1nc(-c2ccco2)cs1 N1(C(=O)CN2CCc3ccccc32)CCN(C(=O)Cn2cccc2)CC(O)C1 C12(C(=O)NC3CCC(NC(c4csc(C(F)(F)F)n4)=O)C3)CCCC1C2(F)F C(=O)(CC(C(F)(F)F)NC(c1ncc[nH]1)=O)NCC(CC=C)(C)CO N1(CCNC(c2ccsn2)=O)CCN(C(C2(C3CCCCO3)CCC2)=O)CC1 N1(C(CC(C(F)F)NC(C(CCC)(C)O)=O)=O)CCOC(C)(C)C1C c1(OC)c(F)cc(S(=O)(=O)N2CCC3C2CCCN3c2ccnc(SC)n2)cc1Cl c1(CNC(C(c2ccc(OC)nn2)N(C(C=C)C2CC2)C)=O)ccccc1Br n1(CC(=O)NCC2C(NC(c3cn(C)nc3)=O)C2)nc(O)ccc1=O C1(CCC)CC(C(=O)NCC2CCCN2c2nccc(CO)n2)CCO1 c1(C(N2CC(C(C)C)N(C(C3COC(=O)O3)=O)CC2)=O)nn(C)cc1[N+](=O)[O-] c1(C(=O)NC(C)CNC(=O)C2=CSCCO2)cc2ncccc2cc1Cl C12CC3CC(CC3C1)N2.Nc1cc(C(=O)NOC(c2ccccn2)=O)ccc1Cl N1(CC(=O)NCCCC2CCCC2)CC(C(=O)O)(CO)C1 CC(C)CC(C(=O)NC1CN(C(C2CCC(C)(C)OC2)=O)C1)c1ccccc1 C1(OC)C(NC(=O)CCC2(C)CN(C(=O)CC3(O)CCCOC3)C2)CC12CCC2 c1(C(N2CC(COC)(NC(c3ccc(N(C)C)nc3)=O)C2)=O)ccc(F)c(Cl)c1 c1(C(=O)NCC2CC(NC(COC)=O)C2)sc2ccc(F)cc2c1C c1(C(C)C)nccc(N2CC=CC(NC(=O)COCCCN(C)C)C2)n1 C(=O)(C(C)(O)C(C)(C)C)NC(C)C(C)NC(c1cc(C(C)(C)C)no1)=O C(C(CC(C)C)C(=O)NCC1CCN1C(c1cc(Br)ccn1)=O)OC N1(C(C(C=C)O)=O)CC(CNC(c2cc3oc(C)cc3[nH]2)=O)CC(C)(C)C1 c1(C(C(=O)NCC(CNC(CCNC(C)=O)=O)C)(C)C)cccc(F)c1 N1(C(C(CC)(F)C(=O)N2CCCC2)=O)CCC2(CCC2)C(C(F)(F)F)C1 c1(C(=O)OC(c2nc(C)[nH]n2)C)ccc(C)c(C)c1N N1(C(c2n(CC)nnc2)C(=O)NC2COC2)CC2CCCN2CC1C CC(O)C(C)(C)C(=O)NCc1cc(C(=O)NOC2CCCC2)on1 C(=O)(C1=COCCC1)NCC1(C(C)NC(CC(C)c2cccnc2)=O)CC1 CCC(O)(C(=O)NC1CCCC1NC(c1cnn(CC)c1)=O)c1ccc(Cl)cc1 CC1CCCN(C(=O)C(C)(C)C)C1CNCc1ccc(-c2ccccc2)cc1 C1(CC(=O)NCC(C)NC(C2CC2c2nccn2C)=O)CCC(=O)O1 N1(C(CCC(=C)Cl)=O)C2CCCC1CC(NC(=O)CSc1cccc(C)c1)C2 c1(NC(C(C)NS(CC)(=O)=O)=O)cc2cnc(C)nc2nc1O c1(C(N2CC(NC(C(n3cc(C)nc3)(C)C)=O)C2)=O)ccnc(Cl)c1Cl CCCCCC(O)CC(=O)NCC1C=CCN1C(=O)Cc1ccc(NCC)cc1 C1(CCC)CN(C(=O)C(C)(C)CCSC)CCN1C(=O)Cc1ccc(Cl)nc1F C(CC(C)(C)C)(C(=O)NOCC1CC1)N1C(C)CN(C(=O)CNC(N)=O)CC1 c1(C(C(=O)NCCCC)N(C2CC2)C(C)C)cnccc1C C1(NC(CCc2ccc(C)cc2)=O)CCCN(C(C2C3C4CCC(C4)C23)=O)C1C C1(CNC(c2c(C)noc2)=O)C2CC1N(C(C1CCC1c1ccc(F)cc1)=O)C2 C(C)(C(=O)NCCOCCNC(=O)C(C)c1cc[nH]n1)OCC(C)C C1(CN(C(=O)COCC(=O)NCC)CC)CCCCN1C(=O)C(C)C.Cc1ncc[nH]1 C1(CNC(Cn2nnc(C)n2)=O)C(C2CC2)CCN1C(C1CCC=CCC1)=O CC(O)(CC(F)F)C(=O)N(C)CCOCCN(C(c1cccc[n+]1[O-])=O)C1CC1 c1(C(N2CC(NC(C(C)(C)N3CCCC3)=O)C(O)C2)=O)ccc2cccnc2c1 C1(CC)CCCC2CC12.C(=O)(C(C)CC=CC(C(C(CC)=CCCC)=O)=O)N Cc1cc(Cl)cc(C(=O)NC2CC(NC(=O)CN3CCOC3=O)C2)c1C c1(C(N2CC(CCNC(C3OCCC(C)C3)=O)OCC2)=O)ccc2nn[nH]c2c1 C1(COC)CN(C(C2CCN(C(C)=O)C2)=O)CCN1C(c1ocnc1C)=O c1(C(=O)NCCCOCCN(C(C(CC)C(C)O)=O)C)cc2cc(Cl)cnc2o1 C(=O)(C1=CCCCO1)NC1CC(C)N(C(c2cccc(Cl)c2C(F)(F)F)=O)C1 N1(C(Cn2c(C)ccn2)=O)CC2CCC1CN2C(=O)CCCC#N O=C(C1=CCCOC1)N1CC(C2CN(C(c3sc(Br)cc3F)=O)CCO2)C1 c1(C(=O)NC)cncc(C=CC(C)NCC=CCl)c1 c1(OC)ccc(F)c(C(=O)NCCCCC(C)NC(C2CCCC2(F)F)=O)c1N N1(C(C(CCCCC)O)=O)CCCC2(CNC(C3(Br)CC3)=O)CCCC12 N1(C(C2CN(C(C3CC(F)(F)C3)=O)CC23CC3)=O)CCCC(C2CC2)C1 C1(CNC(Cc2cn(CC)nn2)=O)C(C)CCN1C(=O)C(C)c1cccs1 C1(CC)(CO)CCN(C(=O)CSCC(F)F)C1.C12(CC1)C(=O)NC2 C1(CC)CCN(C(c2csc(C#N)c2)=O)C1CNC(C12CCCC1C2)=O C(=O)(C(C)C(C)c1ccccc1Cl)NCCN(C(=O)CCN1CCC1)CCC C(=O)(CCCN=c1nccc[nH]1)N1CC(O)(CNC(C(CC(CC)C)C)=O)C1 N1(C(c2c[nH]c(=NC)o2)=O)CCC2(CC1)CC2CNC(=O)CCC(C)(C)F c1(COCC)nc(Oc2c(NN3CCC=C(Br)C3)ccc(NC)c2)cc(O)n1 C1(C(=O)NC2(C)CCN(C(CC3C(OC)CC3)=O)C2)CCN(OC)CC1 C1(C)(CC)CC(C(N2CCCCC2)=O)CN1C(=O)CC(C)(C)C N1(C(C2(COC)CC2)=O)CC(NC(c2ccc(CO)cc2)=O)CC1(C)C c1(C(N2CCC(NC(C(CC)F)=O)C(C)(C)C2)=O)ccc2nc(CC)cn2c1 C(=O)(C#CC1CCCO1)N1CCC(CCNC(c2cc3n(n2)CCOC3)=O)CC1 N12CC3CCC(CC3C1)NCC2=O.c1(OC)cccc(NC(=O)COC2CC2)c1 CCC(C)CC(=O)C(=O)N1CCOC(CC(=O)NCC(C2CCC2)OC)C1 N1(C(C(C)(C)C(F)F)=O)CC2CN(C(=O)CC3CCCCC3O)CC2C1 N1(C(C)C(=O)NC(c2ccc(Cl)c(F)c2)C)CCC(O)(C(F)(F)F)CC1 C1(O)(CNC(CNC(C)=O)=O)CCN(C(=O)C=Cc2nnn(C)n2)C1 N1(C(C2CCCC(OC)C2)=O)CCC(C)(NC(c2n[nH]c(C)c2N)=O)CC1 C(CCC(C)C)(C(=O)NCCn1nncc1C)NC(C1N(CC)CCCC1)=O CC1CCn2c(C(=O)NC(c3cccc4ccccc34)CO)cnc2C1 C1(C(N2CC(O)(CCNC(CC3(OC)CCCC3)=O)C2)=O)CC(C2CC2)=NO1 c1(C(=O)NCC23CCC(NC(C(C)C(F)(F)F)=O)(C2)CO3)ccc2n[nH]cc2c1 C1(CNC(C#CC(C)C)=O)CC(O)C(O)CC1C(=O)Nc1cnc(O)c(F)c1 N1(C(C(C)SCC)=O)CCCC2(CNC(c3cccc(C)c3)=O)CCCC12 C1(CC#C)(C(N2CC(N(C)CC)C2)=O)CCN(C(C2CCCCS2)=O)C1 Cc1c(C(=O)NC2CCN(C(=O)C(C)(C)O)CC2C)sc2ccc(Cl)cc12 c1(SC)cc(=NC(=O)C23CC2CCN3C(c2ccc(Cl)cc2)=O)[nH]n1C CCCCC(CNC(=O)CCCCC1CC1)NC(c1nnc(C(C)C)s1)=O S(=O)(=O)(c1c[nH]c(C(=O)NCC(F)CNC(c2cc(O)n(C)n2)=O)c1)NC c1(C2CCCN(C(CC=C)=O)C2)nc2ccccc2o1 C1(CC(=O)NCC2(CNC(CCS(C)=O)=O)CCCC2)Cc2ccccc2O1 C(C(C)CCC)(N1CCN(CCn2cnnc2CC)CC1)c1n(CC=C)nnn1 C(CCCC(=O)N(C1(CC(N2CCC2c2ccccc2)=O)CC1)C)N(C)C CC1COc2c(C(=O)NC3(CNC(=O)Cc4nccn4C)CCOC3)cccc21 Cc1cnn(C)c1C(=O)NCCC1CSCCN1C(C1(CCS(N)(=O)=O)CCC1)=O C#CC1CC2CCC1N(C(=O)COC1CCN(C(=O)CCCCC)C1)C2 N1(C(CN(CCC)C)=O)CCN(CC2CCN(C(=O)CC3CC=CC3)CC2)CC1 C(C)(CC(=O)N(C1CCN(C(=O)CCc2nc(=N)[nH][nH]2)C1)CCO)=C(C)C c1(CC(=O)NC(C)C(=O)NC2CC(O)C2(C)C)cccc(Br)c1 c1(C(=O)NCCCCCNC(c2c(NC)cc(Cl)cc2)=O)cnn2ncccc12 N#Cc1sc(=NCC2CC3CCC2N(C(c2ccns2)=O)C3)[nH]c1Cl CC1(C)COC(CC(N2CCN(C3(C)CC3)CC2)=O)C1 C(=O)(C(C)CCC(C)(C)C)NC(CCOC)C(=O)N1CCC(CC(C)C)CC1 c1(C(N2C(CNC(C3N(C)CCC3)=O)CCC2)=O)cccc2ccnn12 N1(C(c2ccc(OCCOC)nc2)=O)CCC(C2CCN(CC(N)=O)C2)CC1 c1(CC(=O)NCC(CN(C(C(CC2CCC2)OC)=O)C)(C)C)c(C)nn(C)c1C C(=O)(C(CC(F)F)N(C)C(C1CC2(C1)CC21CC1)=O)NC(COC)CCO C(c1ccc(Cl)cc1F)=CC(=O)NC1C(CNC(C(C2CCC2)OCC)=O)C1 Cn1cc2c(n1)C(C(=O)N1CCCC1(C)Cn1cnc3ccccc13)CCC2 C(C(=O)NCC(C)(C)CN(C)C(C1CCCCS1)=O)(C(C)C)N(CC)CC CC1CC(c2nc(-c3ccsc3)nn2CCCO)CCS1(=O)=O Oc1cc(-c2ccncc2F)ccc1-c1nccn1-c1ccc(I)cc1O N1(C(C(C)Cc2cccc(F)c2)=O)CCC(NC(=O)CCCCCF)C12CCC2 c1(NC(=O)NC2(C(=O)OC)CC(O)C2)ccc(S(N)(=O)=O)cc1[N+](=O)[O-] CCCC(C(O)C(=O)NCc1cnc(C)n1CC)NC(=O)CCOC c1(C(N2C(Cn3cc(C(C)OCC)nn3)CC2)=O)ccc2c(c1)OCO2 Cc1c(CN2CCOCC2C(=O)Nc2cc(F)cc(Br)c2)[nH]c2ccccc12 N1(C(CCC(C)SC)=O)CCC2(C)CN(C(C3CC3C(N)=O)=O)CC12 c1(C(N2CC(C)(NC(=O)CC3CCCC34CC4)C2)=O)nc2cnccc2s1 N1(C(C(C=C)C)=O)CCN(CCNC(=O)C(C)C2CCCC2)CC1 c1(COCC)cccc(C(=O)N(CCNC(C2COCCN2C)=O)CC2CC2)c1 CCCCC(O)CCC(=O)NCC1CC2CCC1N2C(=O)COC1CCN(C)CC1 CCCCCCCC(C)CNCC1CNC(=O)CO1 C1(CCC)(NC(C2C=CC2C(=O)OC)=O)CCCN(C(=O)CNC2CCCC2)C1 C(=O)(C1CCc2ccc(OC)cc21)N(CCNC(=O)C1=CCC1)CC N1(C(c2ncn(C(C)C)c2)=O)CCOC2(CCN(C(=O)Cc3cc[nH]c3)CC2)C1 C1(CC(=O)NC2CC(C)(NC(c3ncc(F)cc3F)=O)C2)CCC(=O)NC1=O C(C(CC)CC)(c1nnnn1CC1CCOCC1)N(CC(=O)NCCCC)CC Cc1c(NC(c2nnnn2C2CCOC2)C2(c3ccon3)CC2)sc2nccn12 C1(C(=O)NC2CCC(NC(c3cc(Cl)sc3Cl)=O)C2)CC2(CCC2)CO1 N1(C(C)(C)C)CCC(NC(c2cc(-c3ccccc3)c[nH]2)=O)C1=O c1(C(=O)OC)cc(C(=O)NC2(C(N3CC(SC4CC4)C3)=O)CC2)n2c1COCC2 N1(C(C#CC(C)C)=O)CC2(C(=O)NC3C=CCCC3)CC1CCO2 CC(C)(CCC(=O)NC1CC(NC(c2cnc(C(F)(F)F)s2)=O)C1)[N+](=O)[O-] c1(OC(CC)C)cc(C(=O)N(C)CCN(C)C(c2cc[nH]c2C)=O)ccn1 C=Cn1nccc1-c1nc(C(C)OCc2ccccc2)nn1CCCC c1(C(=O)NCCC(=C)CNC(c2ccc3c(c2)CC3)=O)cc(=O)c(OC)c[nH]1 C(=O)(C(C)(CSC)NC(c1cccc(COC)n1)=O)NCC(CC)CO C=CCC(CC(C)C)C(=O)N1CC2CC(NC(=O)CNC(=O)CCC)CC1C2 c1(CC(=O)NC2(CC(=O)N(CC(COCC)O)C)CC2)cc(C)[nH]n1 c1(C(N2CCC(C#C)(O)C2)C(=O)NCC=C)ccc2c(C)[nH]nc2c1 CCC(CNC(=O)C(C)Cc1ccc(C)cc1)(CC)NC(C1CC(N(C)C)C1)=O N1(C(C(C2CCCC2)NC(C(C)C2CCC2)=O)=O)CCC(F)(C#N)C1 N1(C(CNC(C)=O)=O)CC(C(=O)NCc2ccc(N3CCCC3)nc2)C2CC12 C1(NC(C=CC=CCC)=O)CCCCN(C(=O)Cc2ccc(NC(C)=O)cc2)C1 N1(SCOC(Cc2cc(C)[nH]n2)=O)CCOCCC1CC(c1ccncc1)O Cc1c(CC(=O)NCC2CCN2C(=O)COC2CCCCO2)cnn1C N1(C(c2cc(CCOC)on2)=O)CCC(CC(C)C)(CO)C1 C1(CN(C(C(CC)=CC)=O)CC)CCCCN1C(C1CC=CCO1)=O c1(Cc2scc(NC(c3cn(Cc4ccc(F)cc4)nn3)=O)n2)cc(F)cc(Br)c1 C1(C(=O)NCCN(C2CC2)CC)CCN(C(c2cn(C)nc2OC)=O)CC1(C)C c1(C(=O)NC(CCC)CNC(=O)Cc2ccn(C)n2)nccc2cc[nH]c12 C1(=O)C2=CCCN(C2)C2(C(N(CC)OC)=O)CCC(C2)O1.C(C)(C)(C)OC C(=O)(N=c1ccn(CCF)[nH]1)C1OCCN(C(C(C)NC=O)=O)C1 C1(C(=O)NC(C#C)CC(C)C)C2CC3C(C2NC(c2cnn(CCO)c2)=O)C13 N1(C(C(C)c2cccs2)=O)CCOCC(C(=O)NCCCP(C)(C)=O)C1 C#CC(CC)(CC)NC(=O)C(C)CN(C)C(c1cccc[n+]1[O-])=O c1(OC)ccc(C(=O)NCC2(NC(=O)C3=CCC(C)(C)CC3)CC2)c2ccsc12 N1(C(c2ccnc(OC)n2)=O)CCOC2CN(C(c3ccc(C)c(C)n3)=O)CC12 N1(C(C2CCC3(CC3)C2)C(=O)NC)CCC(C(F)(F)F)C1(C)C N1(C(c2oc(CC)c(C)c2)=O)CCCC2C1CCCN2C(=O)CN(C)C(C)=O c1(-c2c(C)nc(Cl)nc2)nc(C2COc3ccccc32)nn1CC1CCCCO1 c12noc(n1)C1=C(F)CN(CC1)C2.n1(C(c2ccccc2)=O)c(=O)sc2cccc(Cl)c12 N1(C(c2n(C)c(S)nc2)=O)CCCC(C2CN(C(=O)C=CC3CCCO3)C2)C1 C1(OC)CC2CCC1CC2C(=O)NCC1CCN1C(=O)C(C)C(O)C(C)C C(Cc1cnc[nH]1)(C(=O)NC1CCCC1N(C)C)NC(COCCN(C)C)=O C1(C(=O)NCCN(C)C(c2cccc3cnsc23)=O)C2CCC1(C)C2(C)C CCC1=C(C(=O)N2C3CN(C(=O)C(C)=C4CCC4)CC23)CCCO1 C=C(C)CCC(C)NC(=O)C(C)=CCNC(c1cncc(O)c1)=O c1(C(=O)NC2CN(C(c3cc(CC)n(C)n3)=O)C3C2C3)n[nH]c2cc(C)ccc12 c1(CCC(=O)N(C2CCN(C(=O)CCCC(C)=O)C2)CC)cnc2n1CCCC2 CC1CN(C(=O)COC2CC(F)(F)C2)CCC1NC(C12CCC(CC1F)C2)=O C1(NC(C2(N(C)C(C3CCC(F)CC3)=O)CC2)=O)CN2CCC1(F)CC2 c1(C(=O)NCC2CCCCN2C(C2CC2c2ccccn2)=O)occ2c1CCOC2 n1(CC(=O)NCC(C)NC(=O)C(C(C)O)N(C)C)cccc(C(N)=O)c1=O C1(C(=O)NCC(C)(C)NC(c2cccnn2)=O)CC2C(C1)C2(C)C c1(C(=O)NC2(C)CCCN(C(=O)C(C3CCCCC3)F)C2)cc2c([nH]1)CCCC2 c1(CNC(N2CC(CO)C2)=O)ccnc2[nH]ccc12 Cc1nccnc1C(=O)NNC(=O)NCC1(CO)CC1(F)F.C(C)(C)(C)OC(=O)N N(C(=NCCCF)N(C)Cc1cccc(F)c1)Cc1ccc(COCC)cc1 N1(C(CC(COC)C)=O)CCCCC(NC(=O)COc2cccc(OC)c2)CC1 C1(CNC(C(c2nccc(C)c2)(C)C)=O)CN(C(=O)C2=NOC(C)C2)C(C)(C)C1 N1(C(CC#N)=O)CC(NC(c2cccn(-c3ccccc3)c2=O)=O)C(C#N)C1 C(C1CCOC1)=CC(=O)NC1CC(F)(CNC(=O)C(O)Cn2cncn2)C1 Cc1ccc(C(=O)N(C(CNC(c2ccc(Cl)nc2)=O)C2CC2)C)cc1CO c1(C(=O)NC2(C)CC(NC(=O)C(C#N)C(C)(C)C)C2)ccc2nc[nH]c2n1 C1(C)(C(=O)NC2(C(=O)NC3(c4ncc(C)o4)CC3)CC(O)C2)CCCC1O Cc1cc(CN2CC3CC2CN3C(C2CCCS2)=O)ccc1[N+](=O)[O-] N1(CC)CCOCC1C(=O)N(CC(C)N(C)C(c1csnc1Br)=O)C c1(NC(c2c(C)nc(CNC(C3C(C)(COC)C3)=O)o2)=O)ccc(F)cc1O n1(CC(=O)N(CCC)CCNC(=O)CC2CCOC2)nnc(-c2ccsc2)n1 CC(C)(C)CC(F)C(=O)N1CC(C2(NC(c3cc(C(N)=O)co3)=O)CC2)C1 C(CC(C)(C)C)(C(=O)NC(c1nn(C)cc1O)C)NC(C(c1ccnn1C)C)=O C(=O)(CCCCCN=[N+]=[N-])NC1C(NC(CC2(O)CCCN(C)C2)=O)CC1 N1(C(CN(C(C)=O)C)=O)CCC2CCN(C(=O)Cc3cnn(C)n3)C2C1 C1(NC(=O)CCCn2ccnc2)CC2(C1)CC2N=c1[nH]nc(C(F)(F)F)s1 Cc1nc(NCC2CC3(C2)CC(O)C3)cc(=NC(C)c2nccc(O)n2)[nH]1 C1(C(C)C)CN(C(=O)CC2CCCC23CC3)CCN1C(c1ccc(=O)n(C)n1)=O C(=O)(C1CC(O)c2ccccc21)NC1CN(C(c2cc(OC)ns2)=O)CC1(C)C Cc1nnccc1C(=O)NC1CCCC1NC(C1NC(=O)OC1C)=O C1(C(N(C(CCNC(CC=CC=C)=O)C)C)=O)CCCCC(=O)N1 CC1(C)CCCN(C(=O)C2=COCCC2)C1C(=O)NC1CCn2nnnc2C1 c1(NC(=O)NC2CC2C(=O)Nc2ccc(I)cc2)ccc(Br)c(Cl)c1F c1(CCC(N2CCC(N(C(C3CC3C)=O)CC)C2)=O)cccc(C)c1 c1(C(=O)NCC(CC)NC(C2(C)CC(O)CN2C)=O)c(C(F)F)nn(C)c1C c1(OC)ccc(C(N2CCN(C(C3C=CCC3)=O)C(C)C2)=O)nc1Br c1(C(=O)NC2CCN(Cc3cn(C(C)C(=O)O)nn3)C2)cc2cc(Cl)sc2[nH]1 N1(C(c2c(CC)ocn2)=O)CCC2CCCC12C(=O)NCCS(C)(=O)=O CC(O)C(C(=O)NCC(=O)Nc1ccc(CCF)cc1)NC(C1CC1CO)=O Cc1nn(C)cc1CCC(=O)N1CCC1CNC(c1cc(C2CC2)n(C)n1)=O C1(SCC)CCC(C(=O)NCCN(C)C(c2c(Br)noc2C)=O)CC1 CC1CC2(CC(C(N3CCN(C(=O)CC4COCC4O)C(CO)C3)=O)C2)C1 C12(CS(=O)(=O)NC3CC(COC)C3)CN(Cc3c(F)cccc3Cl)CC1CCO2 CCCCC(CC(=O)Nc1ccc(O)c(Cl)c1)NC(=O)C=C(C)c1ccco1 N1(C(CC=C=C)=O)CCC2(CC1)CN(C(c1ccc(C)cc1)=O)C2 C(=O)(CN=S(C)(C)=O)NCCCC(C)NC(C(C)CO)=O N1(C(c2ccc(OC)c(Cl)c2Cl)=O)CC2CCCN(C(c3ccsc3)=O)C2C1 c1(C(N(CCNC(C2CC(C)(C)CN2C)=O)CC)=O)cc2c(nc(C)n2C)s1 c1(CNC(=O)NC(c2nc(=O)o[nH]2)C)csc(Br)c1Br CN1CC2(CCC2)CCC1NC1CCN(c2nc(O)n[nH]2)CC1 c1(C(N2CC3C(NC(CNC(=O)OC)=O)(CCC3)C2)=O)[nH]c2ccccc2c1Cl C1(NC(=O)CC2CCCC2)CCN(C(C2(F)C3CCCC23)=O)CC1 N1(C(C(C)C(=O)OC(C)(C)C)=O)CC2(CCN2C(=O)Cc2ccc(F)cc2)C1 C(=O)(CCCC(C)(C)C)N(C)CC1(NC(c2ccccc2C2CC2(F)F)=O)CC1 CC1(CNC(C2CC3CCCC3C2)=O)CCN(C(=O)CN2CCCCC2=O)CC1 N=c1cc(-c2cn(CCO)nn2)cc[nH]1.C1(N)CCN(C(C2CS(=O)(=O)C2)=O)C1 Cc1cc(=NC(=O)N2CCC(O)C2C)[nH]n1-c1ccccc1OC(F)(F)F CC1CN(C(C2(c3cccs3)CCC2)=O)CCN1C(c1ccc(O)c(F)c1)=O N1(C(=O)NC(C(c2ccc(F)cc2)C)C)CCn2c(nc3ccccc23)C1 N1(C(C(C)C(C)(F)F)=O)CC2(CCCN(C(c3cccc(C(F)F)c3Cl)=O)C2)C1 c1(C(C(=O)NCCC2CC2)N(c2ccc(F)cc2F)CC)ccc(C)c(I)c1 C(=O)(CCC(=O)N(C)C)N1CCC(CCC(=O)NC(C)C2CC2)C1 CC1(C)CC(CNC(=O)CCNC(=O)CO)CN(C(=O)CCn2cc(Cl)cn2)C1 C1(C(=O)NCC2OCCN(C(c3c(SC)csc3)=O)C2)CCC(S(N)(=O)=O)CC1 C1(NC(c2c(C)cccc2)=O)CCCN(C(=O)CCc2cnn[nH]2)C1C C1(C2CCC2)(CNC(C2=C(C)OCC2)=O)CCN(C(c2cc(N)ccn2)=O)CC1 N1(C(c2csc(C)c2C)=O)CC2CC1CN(C(c1cccc(CN(C)C)c1)=O)C2 C(=O)(CC1CCCc2ccccc21)NC1(C)CCN(C(C(C(CC)C)O)=O)CC1 CCC(C(C)C)(c1nnnn1CC1CC1)NC(c1ncc(Br)cn1)C C#CCC(CC#C)C(=O)NCC(CO)NC(c1cccc(C(=O)OC(C)(C)C)c1)=O N1(C(=O)OC(C)(C)C)CCOC(CCCCCOc2c(C)ccc(Cl)c2)CC1 C1(NC(C(CCCC)C(C)C)=O)CCS(=O)(=O)C12CN(C(=O)C1=CCOCC1)C2 C1(C(=O)Nc2cccc(N(C)C)c2)CC2(CCC2)CN1C(=O)Cc1cc[nH]n1 N1(C(c2ccc(C)s2)=O)CCN(C(=O)CCC2CC2(F)F)C2CS(=O)(=O)CC12 C(C1CCCN1CCSC(C)(C)C)=CC(=O)NC1CCOC(=O)N1 C1(CC(=O)N(CC(CNC(c2nn(CC)c(O)c2)=O)C)C)CC2CCC1CC2 CC(CC(=O)N(C)CCN(C)C(c1cc2c[nH]cnc-2n1)=O)CC(F)(F)F C(=O)(CCCCCO)N1CC(CNC(Cc2cccc(OC(C)C)c2)=O)OCC1 N1(C(CCCCC)=O)C2CCC1CN(C(=O)C(C)Cn1cccn1)C2 C(=O)(C(C(CC)CC)C1CC1)OC(CC#C)CC#C Cn1ccc(C(=O)NCC2(C)CC(NC(=O)C=Cc3nccs3)C2)c1C1CCC1 N1(C(CC(C)OC)=O)CCC2(CC1)CC2NC(c1c(NC(C)=O)c[nH]c1C)=O C(=O)(C1=CCC(C)(C)CC1)N1CC(NC(c2c(C)c[nH]n2)=O)C(C2CC2)C1 N1(CC(C)NC(=O)CCC(=O)N(C)C)CC=C(CCc2nc(C)sc2)CC1 CCC(C#N)(CC)C(=O)N1CCOC(C(=O)NC(C)C(=O)OC)C1 c1(C(=O)NC(CC(C)NC(c2ccn(CC)n2)=O)C)cc(C(C)C)ccc1N N1(C(c2c(-c3cn(C)nc3)c[nH]c2)=O)CCCC2(CC2C(=O)O)C1 C(C)(N=c1[nH]c(=NC(C)c2cnsc2)[nH]c2c1SCC2)c1cn(CC)nc1 CC1c2ccc(Cl)c(Cl)c2CCN1C(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 C1(CNC(C2CCC(NC(C3C(OC(C)=O)C3)=O)C2)=O)(CO)CCN(C)C1 C(=O)(C1=C(C)S(=O)(=O)CC1)N1CC(CNC(C2(C#C)CCCC2)=O)C(C(F)F)C1 CC1C(C(=O)NC2CC(CCC(N3CCNC(=O)C3CCO)=O)C2)=NOC1C Cc1nscc1C(=O)N(C)CC1(NC(=O)COC(F)F)CC1 C1(N(C(C2(CSC)CC2)=O)C2CC2)CCN(C(=O)C(C)CSC(F)(F)F)C1 CCC(CC)C(C)C(=O)N1CC(CNC(c2nnn(C)c2C)=O)CC1(C)C C1(C(=O)NCCC(C)OC)CCCN(C(=O)CCc2nc(O)n[nH]2)C1C N1(C(CC(C)(O)C(=O)O)=O)CCc2ccncc2C1.C12CCCC1C(=O)N2 N1(C(CN(C(C)=O)C)=O)CC2CCCC(NC(c3ccc(CN(C)C)o3)=O)C2C1 c1(C(=O)NC2C(CNC(C3(OC)CCS(=O)(=O)C3)=O)C2)cc2c([nH]1)CCCC2 C1(C(=O)NCC(C2CCC2)NC(CN(C)C(C2CCCC2)=O)=O)CC12CC2 c1(CC2CCN(C(c3cnc(C)s3)C(=O)NC(C)C)C2)cccc(Cl)c1 N1(C(c2cc(C(C)=O)no2)=O)CC(C)N(C(c2cnc3nccn3c2)=O)CC1C c1(C(=O)NCCCCn2cc(-c3nc(C4CC4)cs3)nn2)nc(O)[nH]c(=O)n1 Cc1cc(O)nc(CNC(=O)CC2N(C(c3ccncc3O)=O)CCC2(C)C)n1 C=C(Cl)CCC(=O)N1CCC(CCNC(C2CCCCN2C(C)C)=O)C1 Cc1nccc(N(c2cnc(C3CCNCC3)nc2)C(=O)C(Cl)(Cl)Cl)n1 C(=O)(CCC(=O)NCC(C1CC1)NC(c1ccccc1C)=O)N(CC)CC N1(CC)CCN(C(=O)CC(C(F)F)NC(=O)C(CC)n2cncn2)CC1=O C1(CC(=O)NCCN(C)C(C2(C)CCOCC2)=O)CCCC(F)(F)C1 C1(CNC(c2c(CNC(CCOC(C)C)=O)c[nH]n2)=O)C(C)(C)C1(F)F C(c1ccccc1Cl)=C(C(=O)NC1CC(CCNC(CCCC=C)=O)C1)C C1(C(=O)NCC2N(CC)CCC2)CC(C)=CCN1C(c1csc(Cl)c1)=O C(CC(=O)NCCCCN=[N+]=[N-])N(C(=O)COCC1CC1)CC.OC c1(C(c2nnnn2C2CCCCC2)NCCc2n(C)cnn2)ccc(Cl)o1 N1(C(c2c(N)ncc(Br)c2)=O)CCCCC2(C1)CN(C(=O)Cc1cnoc1)C2 C1(NC(CC2CCC(C)C2)=O)CCC2CN(c3ccnc(Cl)n3)CC2C1 c1(C(=O)NC2CC(NC(C3(C)CCCO3)=O)C2)coc2ccccc12 C12(CCNC(COC)=O)CCC1CN(C(c1cc(C)c(Br)cn1)=O)C2 c1(CNCC(CO)Cc2ccccc2I)c[nH]c2cc(Cl)cc(Cl)c12 N1(C(C2(C)CCOC2)=O)CCCC2(CCN(C(C3CC(CF)C3)=O)CC2)C1 C(=O)(C1=C(C)N(C)c2nnnn2C1)NC(C(=O)OC)C(C(C)C)OC c1(C(=O)NC2C(CNC(C(OC)OC)=O)CCC2)ccc2cnc(C)n2c1 N1(C(c2c(C)cco2)=O)CC(NC(C2(N(C)C)CC2)=O)C(CO)C1 C(CCCCC(=O)N1CC(NC(c2cn(CCF)nn2)=O)C(SC)C1)OCC C1(Nc2ccc(C(F)(F)F)cn2)CC2C3CCC(C3)C12 c1(NC2(c3n(C(CC)(C)C)nnn3)CCOC(C)C2)ccc2c(c1)OCCCO2 Cc1ccccc1CC(N1CCOC(CNC(C2CCCO2)=O)C1)=O Cc1ccc(CN=C(NCC(F)F)NC2CCOC(C)C2)cn1 c1(C(=O)NC2C(C)(C)N(C(c3coc(Cl)c3)=O)CC2)cnc2sccn2c1=O C123CC4CC(CC(C4)C1NC2)C3.c1(CNC(CC)=O)ccc(C#N)cc1 C(C(C)N=c1cccc(S(=O)(=O)NCCc2ccnc(Br)c2)[nH]1)OCCOC C(=O)(C(C)(C)C)N(C)CCOCCCN(C)C(C1CCN1C1CCCC1)=O C1(CC(=O)NCc2cc(C(N(C3CCC3(C)C)C)=O)no2)CC2(CCC2)C1 C1(CC)CN(C(=O)CC2CC(N(C)C)C2)CCC1NC(c1ccn(C)c(=O)c1)=O c1(C(=O)NCC(C)N(C(C(c2ccc(C)s2)C)=O)C)cccc2nc(O)n(C)c12 C1(NC(c2c(C)cc[nH]2)=O)CC12CCN(C(=O)C=Cc1cccc(F)c1F)CC2 c1(CC(=O)NCC2CN(C(c3nc(C)[nH]n3)=O)CC23CC3)ccc([N+](=O)[O-])cc1 C=C(C)CC(C(=O)NCCNC(=O)C(C)(C)C)NC(c1cc(OC)ccn1)=O C(=O)(CC(C)C1CCC1)NC(c1csc(CO)n1)C.C(CCN(C)C(N)=O)OC=O N1(C(CC=CCC)=O)CC(C(N2CC(OC)C(OC)C2)=O)C(F)(F)C1 c1(C(=O)NCC2C(NC(c3cncc(C)c3)=O)C2)cnc(C2CC2)nc1C C1(NC(Cc2ccc(C)nc2)=O)CC2CC1N(C(c1cc(Br)nn1C)=O)C2 N1(C(c2nc(C)c(C)s2)=O)CCN(C(c2cccnc2Cl)=O)CC1C c1(C(=O)NC(CCOC)CNC(C2CC3CC2CO3)=O)ccc(C)cc1F N1(C(C2CC(C)SCC2)=O)C2CCCC1CC(NC(c1ccn(CCF)n1)=O)C2 C1(NC(=O)CCNC(=O)COC2CCC2)CCCCC(=O)N1 C1(O)(CN(C)C(c2ccnc(O)c2F)=O)CCCN(C(=O)CS(N)(=O)=O)C1 CC1CC2(CCN(C(C3CC3F)=O)CC2)CN1C(C1CCC2(CC2)C1)=O c1(N(C(=O)C(C)N(C(C2C=CCN2)=O)C2CC2)C(C)C)ccccc1 c1(OC)ccc(Cl)c(C(=O)NC23CCC2CN(C(=O)CCS(N)(=O)=O)C3)n1 c1(C(=O)NC2C(CNC(Cc3n[nH]c(=NC)s3)=O)C2)cc(S(N)(=O)=O)cnc1C N1(C(CC(=O)NCC)=O)CCC(CCN(C)C(C2CC2(F)F)=O)CC1 Cc1ccc(-c2cn(CCCCCCNC(=O)CC(O)c3cccs3)nn2)cc1 N1(C(C(C)N(C(C)=O)C)=O)CCN(C(=O)C(C)(F)F)CC1c1cccc(Cl)c1 c1(C(N2C(C)CC(NC(COCC#C)=O)C2)=O)c(C)ccc2cccnc12 c1(C(=O)NC(C2CN(C(c3cnc(C4CCC4)[nH]3)=O)C2)C)cc(Cl)nnc1Cl N1(C(C2N(C(C(C)=CCC)=O)CSC2)=O)CC(CN(C)CC)C2(CC2)C1 c1(C(=O)NCCC(C)N(C(=O)C=Cc2ccc[nH]2)C)cnnn1C c1(-c2c(C)noc2C)ccc2ncc(C(=O)Nc3cccc4c3cnn4C)n2c1 C1(NC(CSCC=C)=O)CN(C(=O)C(c2ccc(C)cc2)(C)C)CCC1C(F)(F)F C1(C)(CNC(C(C2CCCCC2)C)=O)CC(F)(F)CN1C(=O)C(F)CC1CCC1 c1(CNC(=O)C(=O)NC2CCCNCC2)c[nH]c2ccc(F)cc12 CCS(=O)CC(=O)NCCC1(NC(=O)C(O)C2CC2)CC1 c1(C(=O)NC2C(NC(C(C)CSc3ccccc3)=O)CC2)n[nH]c2c1COCC2 c1(C(=O)NC2C3(CC(NC(c4n[nH]c(C)c4F)=O)C3)C2)ccn2ccnc2c1 c1(C(=O)NC(CN(C(C(C)C2CC2)=O)C)C)c(F)cc(O)cc1F C=C1Cn2c(C(N3CCC4CN(C(C5CC5(F)F)=O)C4C3)=O)nnc2S1 Cc1ccc(C(N2CC(N(C(=O)CCCN3CCCC3)C)C3(CC3)C2)=O)nc1O C(c1cncnc1O)=CC(=O)NCC1C(CC)CCN1C(C1CCSC1)=O N#CC1=C(C(=O)N2CCCC3(NC(C4CN(CC(F)(F)F)C4)=O)CC3C2)CCC1 C(c1cccnc1C)=CC(N1CC2C(CNC(CC=C(C)C)=O)C2C1)=O C(=O)(CCCN(C(c1nonc1N)=O)C(C)C)NC1CC(OC)C1 c1(C(=O)NC2CCC(NC(Cc3c(OC)n(C)nc3)=O)C2)c(C)ccc(C)c1N C(CC(C)C)(C(=O)NOCCC(F)F)N(C(c1c(N)ccc(C)c1)=O)C C1(C(N2C(C(=O)NC)CC2)=O)C=CCCN1C(C1CCCN1C=O)=O N1(Cc2ccc(OC)nn2)CCC2C(CCN2C(=O)CCCn2ccnc2C)C1 CC1=C(C(=O)N2CC(CNC(C34CC(C(=O)OC)(C3)C4)=O)C3(CC3)C2)SCCO1 N1(C(CCN(CC)CC2CC2)=O)CC(NC(=O)CC2COC3CC2C3)C(C)(C)C1 N1(C(c2c(-n3cccc3)cc(C)s2)=O)CC(NC(C2(O)CC2)=O)CC(O)C1 O=C1NC(C(N2CCC(Cc3ccc(O)cc3)CC2)=O)C2CCCC12 c1(C(N2CC(NC(C3CCC(C(=O)OC)C3)=O)C2)=O)ccc(F)c(S(C)(=O)=O)c1 C#CCCCCCCC(=O)NC1C(C(=O)NCc2ncccn2)C1(C)C CC1CN(C(C2CC23CCN(C(C2(CO)CCCC2)=O)C3)=O)CC1N=[N+]=[N-] C1(C(C)NC(Cn2cc(C(C)=O)nn2)=O)CCCN(C(C2CCCCCC2)=O)C1 C1(NS(CCC)(=O)=O)CCCN(Cc2nc(C(C)O)nn2-c2cccnc2)C1 N1(C(c2c(CC)nn[nH]2)=O)CCOCC1CNC(C1(C(F)F)CCCCC1)=O c1(-c2n(-c3ccc(C)cc3)ncn2)cc2cccc(O)c2nc1C.CCCCC C1(CNC(C2C(CC)C2)=O)CN(C(c2ccsc2Cl)=O)CCN1C O=C(C(F)CC1CN(C(=O)Cn2cnnc2O)C1)NCC1CCOC1=O CC1OCCN(C(C2C(COC)C2(C)C)=O)C1C(N1CCC1(C)C(N)=O)=O C1(NC(C2(CC#C)CCCCC2)=O)CN(C(c2occc2Br)=O)C2CCCCC12 O=C1NCCc2occ(C(=O)NCCc3cn(-c4ccc(Cl)cc4F)nn3)c21 N1(C(Cn2nc(C)oc2=O)=O)CCN(C(c2sc(C)nc2C)=O)C(C)C1 C=CCC(CC(F)F)NC(=O)CC1CN(C(C2(CO)CCC2)=O)CC1C C1(C(N2C(C(C)C)CN(C(=O)CC3CS(=O)(=O)C3)CC2)=O)CC2CCC(C1)N2C N1(C(CCSc2n(C)nnn2)=O)CCCN(C(c2sccc2C2CC2)=O)CC1 Cc1ccc(C)c(NC(C2(N(C(=O)CN(C(=O)C(C)C)C)C)CCCC2C)=O)c1 C(CNC(=O)CN1CCOCC1=O)(CC(=O)NCC(C)Cn1ccnc1)OC c1(C(=O)NC(C(C(C)C)NC(CC=CC)=O)c2ccccc2)ncnc(C)c1C C1(CC(=O)NCC2CC2CNC(=O)CN2CC(CF)C2)CCOCC1 S(=O)(=O)(c1ccc(F)cc1)N(CC(N1CC(O)(C(C)NC(=O)CN(C)C)C1)=O)C C1(C(N2C(C(=O)NCC(=C)C(F)(F)F)(CC)CCC2)=O)CCC2(CC1)CC2 C(=O)(C(C)CCC(C)(C)C)NCC1(C(=O)NC(CC#C)CO)CC12CCC2 c1(OC)ccc(C2(NCc3nnnn3C3CC(C)N(C(C)C)C3=O)CC2)cc1F N1(C(CCSCCCC)=O)CCC2CCN(C(c3ccncc3F)=O)C2C1 c1(C(=O)OCC)ccc(NC(c2csc(=NCc3cncc(C)c3)[nH]2)=O)c(I)c1 N1(C(C)=O)CCCC(O)(C(N2CCCC(NC(=O)CCn3ccnc3C)C2)=O)C1 CCC1=NOC(CNC(=O)CCCN(C)C(c2ccnn2C)=O)C1 c1(OCC)cccc2c(CN3CC4(F)CC3C4)ccnc12 N1(C(c2cc(C(C)=O)cn2C)=O)CC2CN(C(=O)Cc3ccoc3)CCC2(CO)C1 C=C(Cl)C(C)(C)C(=O)NCC1(CNC(c2ccc(C(C)=O)cc2)=O)CC(F)(F)C1 C(=O)(CCCCC(C)(C)C)N1C2CC(C(NOCCCOC)=O)C1CC2 N1(c2ccnc(C)n2)CC2CCC1C(NC(c1cn(C)ccc1=O)=O)C2 N1(C(CC2CCN(C)C2)=O)CC2(CCN(C(C3CCCC(N(C)C)C3)=O)C2)C1 c1(OC)cnc(C(N2CCCCC2c2n[nH]cc2NC(=O)C(C)C)=O)c(OC)n1 c1(C(=O)NC(C2CCN(C(=O)Cc3cncs3)CC2)C)cnc(Cl)c(F)c1N C(CC(=O)NC1CC(CNC(C23CCC2C3)=O)C1)OC c1(C(N2CCC(CNC(c3c(C)cc(O)nn3)=O)C2)=O)cc[nH]c2nccc1-2 c1(C(=O)NCCC2(C(=O)NC3CCC(SC)C3)CC2)cccc2occc12 C(CN=c1cc(C)nc(S(C)(=O)=O)[nH]1)C1CCN(C(C=CCOC)=O)CC1 C(=O)(C(C)C(F)(F)C(F)F)NC1C(NC(C=Cc2cc(C#C)c(C)cc2)=O)C1 N1(N(C(C2(N)CC(C(F)(F)F)C2)=O)C)CCC2(C1)CC(F)(F)C2 c1(C(=O)NCC(C)N(C(c2cc[nH]c2)=O)CC)csc(C(C)(F)F)n1 CCCCCCCCC(=O)NC1C2CC1N(C(c1cnn3c1CCC3)=O)C2 N1(CC(=O)NCC(C)CN(C)C(C2(C)CCNC2=O)=O)CCCCCCC1=O C1(NC(c2cc(C)no2)=O)CC2CCC(C1)N2C(c1cncnc1C1CC1)=O c1(C(=O)NCC(C)N(C(CC(C)(C)SC)=O)C)cc2ccc(O)cc2[nH]1 CC(C)CCCCCNC(=O)CC1CCCC(NC(=O)CC#N)C1 C(=O)(CN=c1cc[nH]cc1)NCCCNC(CCC(C)NC(N)=O)=O c1(C(=O)NCC(C(C)C(C)C)NC(CCN(C)CC)=O)cc(C)cc2ccoc12 c1(C(C(=O)NCC(C)NC(C2(CC(N3CCCC3)=O)CCC2)=O)C)cnn(C)c1 C1(CNC(C2C(NC(C=CCCC)=O)COC2)=O)CC[Si](C)(C)C1 C(C(C(=O)NC1CCC(CCNC(c2ncsc2C)=O)C1)NC(C)=O)OC C1(CC)CCCN(C(=O)C(F)C(C)(C)O)C1C(=O)NC(c1nc(C)oc1C)C c1(C(=O)NCC(CCCC)NC(=O)C=Cc2ccc(F)cc2)cc(C#N)[nH]c1C N1(C(CCC(C)OC)=O)CCCC2(NC(c3n[nH]cc3Br)=O)CC2C1 CC1CCCC1(C)C(N1CCN(CCNC(C2CC(F)(F)C2)=O)CC1)=O N(C1CCCn2nccc21)C(CC(C(F)F)NC(CCC=C)=O)=O CN1CCC(C(=O)NC2CC(n3cc(-c4cnn(C)c4)nn3)C2)S1(=O)=O c1(NC(C)=O)cc(C(N2CCCC2C(C)NC(=O)C(C)CC(C)C)=O)ccc1C c1(NC(CN(CC(=O)NCCC)C)=O)ccc(Br)c(F)c1 N1(C(c2c(C)[nH]cc2)=O)CC2(NC(C3CC=CCC3)=O)CCCC2(F)C1 N1(C(c2cnc(OC)s2)=O)CC(CNC(c2cc(C)oc2C)=O)CCC1C C1(C(C(=O)N(C)Cc2ccn(CC)n2)C)CCN(C(=O)CN2CCC(C)C2)CC1 C1(NC(CCC=C)=O)CCC12CCN(C(c1ccc(NC(C)=O)cn1)=O)CC2 N1(C(C(C)(C)NC(c2ccc(C#N)o2)=O)=O)CC2CC=CC1C2 C1(C(=O)NCC2(C)CC(NC(=O)CCc3ncccn3)C2)(CO)CCCCC1 C(c1cccc(Cl)c1)=CC(=O)NCC(=C)CCNC(C1(C(N)=O)CCC1)=O C1(C(=O)NC(C(C)NC(c2c(COC)ccs2)=O)C)CCNC(=O)C1 Cc1ccc(C=CCC(=O)NC(C)C(C(C)C)NC(c2ccc(Cl)cn2)=O)cc1 c1(OC)cc(CNC(=O)NC2CCN(CCc3ccc(CO)cc3)CC2)ccn1 c1(CN2C(C(=O)NCC(O)CO)CC(OC)C2)cc(Cl)ccc1C N1(C(c2cc(I)cs2)C(=O)NC)CCOC(CO)CC1.c1(OC)ccc(C2CC2)cc1 C1(CNC(C2(NC(C3CC4(CSC4)C3)=O)CC(O)C2)=O)CC2CCC1CC2 CC1(C)CN(C(c2cnn[nH]2)=O)C(CNC(C2(C#N)CC23CCC3)=O)CO1 C1(NC(=O)Cc2ccc(C(N)=O)cc2)CCCCN(C(C2CCCS2)=O)CC1 c1(C(C)C)ccc(C(C)CC(=O)NCCCCOc2ccc(Br)cc2)cc1 c1(C(N2CCN(C(C3ON=C(CC)C3)=O)C3C2C3)=O)cc(Cl)c(O)cc1C Cc1cc(C(=O)NCC2CC2CC(=O)NC2CC(=O)N(C)C2=O)ccc1F c1(C(=O)NCc2ccc(-c3ccc(F)cc3F)o2)c[nH]c2ccncc2c1=O c1(CNc2cccc(-c3ccc(F)nc3)n2)cccc2ccoc12 C1(CN(C(=O)CCCN(C(=O)CC2CCC2)C)C)CCCC(O)C1 C(=O)(N=c1[nH]nc(Cl)cc1Br)C1N(Cc2c(CC)cccn2)CC(F)C1 C1(NC(c2ccn(C(C)C)c(=O)c2)=O)CC2CCC(C1)N2C(c1ccoc1Cl)=O CC1(C)CC(NC(c2ccc(Br)cc2)=O)CCN(C(=O)CCCCCF)C1 C1(CNC(c2cccc(Cl)c2)=O)COCCN1C(c1nc(C(F)(F)F)cs1)=O C#CCCC(O)CCNC(=O)CC(C)CNC(c1cc(Cl)n[nH]1)=O c1(NCC(CC)CC)cc(C)c(S(=O)(=O)NCCCOCC(=O)OC)cn1 C(=O)(CCCCCCCCCO)NCC1CCC(NC(CN(C)C)=O)C1 CCC(O)C(C)C(=O)N1CCC2(C1)CC2.c1(C(=O)OC)cnn(CC)c1C C(C(CNC(C12CC(NC(C)(C)C)(CO1)C2)=O)C(F)(F)F)NC(C(C)C(F)F)=O C1(CC(=O)NCC#CCNC(c2cc(OC)no2)=O)CC(N(C)C)C1(C)C C1(C)(CNC(CC(C)(C)C)=O)CCCN(C(C2C(C3CC3)C2(F)F)=O)C1 Cc1cc(C)nc(SCC(N2CC(C)(NC(=O)C=CC(=O)NC3CC3)C2)=O)n1 c1(C(C(=O)NCC(CNC(c2ccc(F)s2)=O)CO)OC)ccccc1O Cc1ccn2cc(C(N3CCCC(C)(CNC(=O)C(C)C(F)(F)F)C3)=O)nc2c1 c1(C(=O)Nc2cccc(C(=O)OC)c2)cc(I)cc(I)c1 c1(C(=O)NCC(CN(C)C(c2cn(C(F)F)cn2)=O)O)ccc(O)c(N)n1 CCC(CC)C(C(=O)NCCN(C)C(c1csc(C(F)(F)F)c1)=O)OC C(=O)(CCCC(F)(F)CO)NC(CNC(c1nccc(C)c1N)=O)(C)C(C)C CC(CC(=O)NCCCN1CCN(C(C2CC2C)=O)CC1)CC(F)(F)F c1(C(=O)NC2C(CNC(CSCCC)=O)C2)ccc(C(F)(F)C(F)(F)F)nc1 Cn1cc(NC(=O)NCC2(n3nccn3)CC2)c2ccccc12 n1(CC(=O)NC2CCCC2NC(=O)CC2CCCC2O)cnccc1=O C(=O)(C(CC(C)C)OC)NCC1(O)CCN(C(CCN(CCC)C)=O)C1 N1(C(Cc2c(C)n[nH]c2)=O)CCC2(COC(CNC(C3CCN3C)=O)C2)C1 C(C1CCCN1C(C1CCOC1(C)C)=O)=CC(=O)N(C)CC1CSCCO1 C1(CNC(c2c(C)snc2)=O)CN(C(c2[nH]c(C3CC3)nc2C)=O)CC12CC2 CC1OC2CCC1(C(N1CC(C(=O)NCC3CCNC(=O)C3)CCC1C)=O)C2 N1(C(C(C)c2ccsn2)=O)CCC(F)C(NC(c2conc2C2CCC2)=O)C1 O=C1CCc2nc(C(=O)NCC=CCNC(=O)CN3CCC3)ccc21 CN1CCC(C)(C(=O)NCC(C2CC2)N(C(=O)CC2CC=CCN2C)C)CC1 C1(C(C)NC(=O)CCC2CC2(Cl)Cl)CN(C(=O)CCc2cn(C)cn2)CCO1 c1(C(c2nnnn2C2CCC2)Nc2ccc(CS(C)=O)cc2)c(Br)c(Br)nn1C N1(C(c2n(C(C)C)cnc2)=O)CCOC(c2ccc(-c3nn[nH]n3)cc2)C1 C12(NC(C3COC4COCC34)=O)CCCN(C(=O)C=Cc3cocn3)CC1C2 N1(C(c2ccncc2C(F)(F)F)=O)CCCC(CO)(Nc2nc(Cl)ncc2Br)C1 Cc1cc(Cl)cc(C(=O)NCCCC(C)NC(=O)CC2CCCC2O)c1O N1(C(C2OCCN(C(C)C)C2)=O)CCCC2(NC(=O)C(C)O)CCCC12 c1(CC(N2C(C(=O)NC)CCC2)=O)cccc(C)c1F C1(CNC(C(CC)CO)=O)CCCN(C(c2nn(C)cc2C(=O)OC)=O)CC1 C1(C(=O)NC(C)(CNC(=O)CCn2cc(Cl)cn2)C2CC2)CC2CCC1CC2 c1(CC(N2CCCCC2C2CCCN2C(=O)CSC2CC2)=O)ccc(F)nc1 c1(C2C(NC(=O)NCC(CN(C)C)(C)C)C2)ccc(CN)cc1.S(=O)(=O)(C(F)(F)F)N c1(NC(C23C(CN(C(c4c(C(C)C)ccs4)=O)C2)C3)=O)cnc2c(c1)CC(=O)N2 c1(SC)c(C(N2CC(F)(CNC(C3CCCC(F)C3)=O)C2)=O)cnn1C Cc1sc(-c2ccc(-c3cc[nH]n3)cc2)nc1C(=O)N(CC)Cc1cccc(F)c1 c1(CC)ccc(C(C)C(N2CC(O)(CN(C(=O)CNS(C)(=O)=O)C)C2)=O)cc1 c1(N(CCCNC(C2CCC3CC23)=O)C)cc(N(C)C)ncn1 N1(C(C(C)CO)=O)Cc2[nH]nc(CNC(C3(C(C)C)CNC(=O)C3)=O)c2C1 C1(c2nnnn2-c2ccccc2)(NC(CCC)C)CCC(C(C)C(=O)OC)CC1 c1(CC)ccccc1CC(N1CCC(OCCNC(c2cc(C)[nH]n2)=O)CC1)=O C1(C(N2CCCC(NC(=O)CC(F)(F)C(F)F)C2)=O)Cc2cc(Cl)ccc2O1 C(C(C)(C)C(=O)N(C)CC1CCN(C(=O)CNc2cccnc2)C1)OC(C)C CCCCC(CC)CC(=O)NC1CC(CNC(C2CCCN(C(C)C)C2)=O)C1 c1(C(C)O)cncc(C(=O)NCC(C2CCCC2)NC(c2ccon2)=O)c1 C1(N(C(Cc2cnc(C)s2)=O)C)CCC(CNC(C2CCSCC2)=O)CC1 C(CC(C)C(F)(F)F)NC(C(C1CN(C(Cc2ccc(C)o2)=O)C1)O)=O c1(C(N(CC(C)NC(=O)C=Cc2ccc(O)cc2)C)=O)cccc2c1CCCC2 C1(C)(CNC(c2cnc(CC)s2)=O)CCCN(C(=O)Cc2csc(C)n2)C1 c12cc(CO)nc(n1)N1CCC(C1)CN2.O=C1OCC(CO)C1c1ccccc1 CCC(CC)CCCC(=O)NC1(CNC(c2cnc(Cl)cc2N)=O)CC1 c1(C(=O)NC2C(CNC(CCSC)=O)CCC2)ccc2c(c1)CN(C)C2 c1(C(=O)NCC(=O)NC(CNC(C2(C3CC3)CC2)=O)C2CC2)ccnc(CO)c1.CO C1(NC(C=C(CNC(C2(CC)CC(=O)C2)=O)C)=O)CCOC(C)(CC)C1 C1(NC(c2c(CC)noc2)=O)CN(C(c2csc(C3CC3)n2)=O)CC(C)(C)C1 CCCCCCC(C)C(=O)N1CCC(CN(c2cc(F)ncc2F)C)C1 N1(C(C2CCN(C(CC)=O)C2)=O)CCCC(C)(O)CC1 Cc1cc(CC(=O)NC(C)CC(C)NC(=O)C=Cc2ccc(F)nc2)cc(C)c1 C1(NC(CSCC=C)=O)C=CCC(C(=O)NC(c2ncc[nH]2)C2CCC2)C1 c1(C(=O)NCC(C)NC(=O)C=CCN(CC(F)(F)F)C)nc(Cl)c(=O)[nH]c1N CCCC(C)(C)N(C1C2C(=O)C(COCCOC1CCOC)CN2)C C1(NC(COCC(C)C)=O)COC2(C1)CN(C(c1cnc3[nH]ncc3c1)=O)C2 C(=O)(C(F)CCC(C)C)N(CC(N1CCCC(C)(CC)C1)=O)CC(C)C Cc1onc(C2CC2)c1C(N1CC(NC(c2ocnc2-c2ccccc2)=O)C1)=O CCCC(C)(CC)C(=O)N1CC(C(=O)Nc2cnn(C)c2)CC12CCC2 C12(C(=O)NC3C(NC(CC4(C)CC4)=O)C3)CCC(C(F)(F)F)(CC1)C2 c1(C(=O)NC(C2C(C(=O)NC(C3CCOCC3)C)C2)C)cc(C#N)cn1C C(=O)(CCCCCCn1cc(CCCC(C)O)nn1)NCCCNS(CC)(=O)=O N1(C(C)=O)CCCC(CN2CCCC(C)C2)C1 N1(C(Cn2ncn(C)c2=O)=O)CCC2(CCCN2C(C23CCC2C3)=O)C1 Cc1cccc(Br)c1CN1CC(O)CC1C(=O)NCC(C)(O)CO c1(SCCNC(N2CCC(CN=[N+]=[N-])C2)=O)ccccc1[N+](=O)[O-] CC1CN(C(c2csc(Cl)n2)=O)C(C)CN1C(c1ccc(F)c(C(F)F)n1)=O c1(C(N2CCC(C(C)NC(c3csc(O)n3)=O)CC2)=O)cc(=O)cc(Cl)[nH]1 N1(C(c2ccc(C)s2)=O)CCC(C2CCCN(C(=O)C(O)C3CC3)C2)C1 Cc1cncc(C)c1C(=O)NC(C)CC(C)NC(=O)CCc1ccc(F)nc1 c1(NC(C(C2CCCN(C(c3c(CC)n[nH]c3)=O)C2)C)=O)ccccc1N=[N+]=[N-] Cn1cnc(CCC(=O)NCC(CNC(=O)CC2CC23CC3)CO)c1 c1(CC(=O)NC2(C)CCN(C(CCOCCCC)=O)C2)cccc2nsnc12 c1(NC(C2CCC(C(=O)O)CC2)=O)c(Cl)cc(CN2CCOCC2CO)cc1Br C1(NC(c2c(CC)con2)=O)CCCC(C(N2CC(C)(CO)C2)=O)C1 c1(OC)ccc(C)cc1CC(N1CCC(CNC(C2COC(C)C2)=O)C(C)C1)=O c1(CN2CCN(C)CC2)ccc(NC(=O)NCCOc2cccc(F)c2)cc1Cl c1(C(=O)NCC2N(C(C3C(C)C3)=O)CC=C2)cccc(N2CCCC2=O)c1 CC1(CNC(C2(CO)CC2(F)F)=O)COCCN(C(=O)CCF)C1 CN1CCc2nc(NC(C3CSCCN3C(=O)NC3CC=CCC3)=O)sc2C1 c1(OC)ccc2c(C(=O)NC3CCC(NC(=O)CC4CCOC4)CC3)cnn2c1 c1(C(=O)NCCC2(C(=O)NCc3ncn(C)n3)CCCC2)cnn2c1OCC2 c1(C(=O)NC(C2CCCC2)CNC(c2n(CCCC)ncc2)=O)cc(F)n(C)n1 c1(OC)cc(C(=O)NC2CN(C(c3cc(C#N)c[nH]3)=O)CC2F)cc(F)c1F c1(C(=O)NCC(CNC(C2(SC)CC2)=O)CO)cccnc1-c1ccncc1 O=Cc1csc(-c2ccnc(NCC(F)(F)F)c2)c1.c12ccc(cc1)COC2 CC(CC(C)(C)C)C(=O)N1CC2(CC2)CC1CNC(=O)C(C)(F)F N1(C(c2c(C)sc(O)n2)=O)CCC(C(=O)NCC2C3CCCOC23)C(C)(C)C1 Cc1nc2cc(C(=O)NCCOCCNC(=O)C(O)CC(C)(C)C)ccc2s1 Cc1ccc(C=CC(N2CC(CNC(C3CC3(F)F)=O)C(F)(F)C2)=O)nc1 Cc1cccc(O)c1C(=O)NC1CN(C(C2(C)CCN(C)C2)=O)CC1C N1(CC)Cc2nnc(-c3ccccc3)n2C(C)C1.c12cc(C(C)NC)ccc1O2 C1(NC(C2(C(C)=O)CC2)=O)CC(CNC(C2(CO)CCCO2)=O)C1(C)C n1(CC)cc(Br)c(C(=O)NC2CC(NC(C3(N=[N+]=[N-])CC3)=O)CC2O)n1 N1(C(C2(C(N)=O)CCC2)=O)CCCC12CCN(C(=O)CN1CCCC1=O)CC2 N1(C(CCCC(C)=O)=O)CC2(C1)OC1(C)CC2(NC(=O)CN2CCC(C)CC2)C1 C1(F)(CNC(C2N(C(CCCOC)=O)CC=C2)=O)CCOCC1 N1(C(C(CC)(CC)CC)=O)CC2CCCC(C1)N2C(=O)Cc1ccc(F)cc1 Cc1cccc2c1C(C)CC2CC(=O)N1CC(C)OC(C)C1 C(CC)(C(=O)NCC(c1ccccc1)CNC(c1cc(Br)c[nH]1)=O)OCC C1(CNC(CC(CC)CN(C)C)=O)CCN(C(=O)CCOC(C)=O)CC1(F)F N#Cc1cc(C(N2CCC(N(CCO)C(c3scnc3Cl)=O)C2)=O)co1 C(CC(C)C(=O)N(CC(C)NC(=O)C(C(C)C)NS(=O)(=O)C1CC1)C)OC Nc1nc2ncccc2cc1C(=O)NC1CCCN(C(C2CCNC(=O)C2)=O)C1 c1(CCC)nnc(S)n1CC(=O)N(C1CSCC1=O)CC CC(C)CC(O)C(=O)OC(C)C(=O)NCc1nc2c(s1)CCC2 CCC(C)CCCC(O)CC(=O)N1CCN(CC(F)F)CC1 N1(C(C(CC(C)C)F)=O)CCOC2(CCC(NC(=O)C=C3CCN(C)C3)CC2)C1 CC(F)(F)C(C)(C)CC(=O)NC1CN(C(=O)Cn2nnc(=O)[nH]2)CCC1CO C1(C(=O)NCCCC(C)NC(C2C(CC)C2)=O)CCN(CC2CC2)CC1 CC(C(F)C(=O)NCC12CN(C(c3cc(C#N)c[nH]3)=O)CC1CCO2)C(F)(F)F N1(C(C=CC)=O)CCCC(O)(CNC(=O)CN(C2CCSC2)C)CC1 C1(C(=O)NC(CC)Cn2cncn2)COCCC1NC(=O)CCOCC1CC1 C1(C(C)NC(CSC)=O)CCN(C(c2nnc(O)s2)=O)C1 c1(C(=O)NC2CCC2)ccnnc1.C12CCC1C(=O)NCCN(C1CC1)C2=O c1(C(=O)OC)cnn(CC(=O)NC2COCC2NC(C2CCCOC2)=O)c1N C1(COC)CN(C(=O)C2=CCCCC2)CCN1C(C1CCC1)=O C1(C(N2CCC(OCCNC(C(C)CC3CC3)=O)CC2)=O)CC2(COC(=O)N2)C1 CCCCC(CNC(=O)CC1CC(O)CN1C(c1ccncc1NC)=O)CCC N1(C(C2(C)C(CC)CCC2)=O)CC2(CCN(C(=O)Cc3cccnc3)CC2)C1 N1(C(CC=C=C)=O)CCOC2(CCN(C(=O)COc3ccc(Cl)nc3)C2)C1 S(=O)(=O)(c1ccc(Br)c(NC(=O)CS(=O)(=O)CCO)c1)NC(C)C c1(C(N2C(CNC(C3CCc4nncn4C3)=O)CC2)=O)ccc2snnc2c1 c1(OCC(=O)NC2C(NC(CCC=C)=O)CS(=O)(=O)C2)ncnc2ccccc12 Cc1cccc(Br)c1C(C(=O)N(C1CN(C)C1)C)NC(c1sccc1C#N)=O c1(C(=O)NCC2COCC2O)cnc(-c2cccc(O)c2)cn1 CC1C2CC(C2NC(c2cccc(=O)n2C)=O)N1C(c1cc[nH]c1)=O c1(NC(C(c2ccoc2)NC(=O)C2=NOCC2)=O)ccc(F)cc1O C1(CNC(C(CC=C)OC)=O)(CO)CCN(C(=O)C(C2CCCCCC2)O)CC1 c1(CC(N2C(CN(C(C(CC)C)=O)CC)CCC2)=O)ccc(C#N)cc1C C1(CNC(=O)Cc2nc[nH]n2)CCN(C(C2CCCC2)=O)CC1(F)F C(CCCCC(=O)N1CC(F)CC1C(=O)NC1(CO)CC=CC1)N(C)C N1(CC(=O)NC2(C)C=CCC2)C2CCC1COC2.c12ccc(o1)c(=O)[nH]2 C(=O)(C1=CSCCO1)NC1C(NC(=O)COC(F)F)CCCC1 c1(C(=O)NCC(C2CC2)NC(c2cn(C3CC3)nn2)=O)cc(C2CC2)cc(F)c1 C(=O)(C(F)(F)CO)NC1CC(C(C)NC(CC=C)=O)C1 C1(C)(SCC)CCC(NC(c2cccc(NS(C)=O)c2)=O)CC1.C1C(=O)N1 c1(CSCC(=O)NC2CCC(NC(CS(=O)(=O)NC)=O)C2)nn(C)c(=O)n(C)c1=O N1(C(CCSC)=O)CC(C(=O)NCCn2nc(C)nc2C)C2(CCC2)C1 N1(C(c2cc(C3CCOCC3)[nH]n2)=O)CC(NC(C2(CO)CCC2)=O)CC(F)C1 N1(Cc2ccc(OCC)cc2Cl)c2ccccc2SC(C)C1C c1(OCC)cc2ccccc2cc1C(=O)NC(C)(C)CNC(c1occc1F)=O c1(OCc2nn(C)c(C(F)(F)F)n2)ccc(C(=O)O)c(Cl)c1 CCS(=O)(=O)CCCCCNC(c1cscc1F)c1nnnn1Cc1ccccc1 c1(C(=O)OC)cc(CC(N2CCC(CN(C)C(C3CC(N(C)C)C3)=O)C2)=O)cs1 C1(C(=O)NCC2CCC(NC(c3c(CC)non3)=O)CC2)CC2CCCC2C1 C1(NC(=O)NC)CCC(NC(C(CO)C(=O)CSC(C)C)=O)C1 c1(OC)ncccc1NCc1ccnc(Br)c1 N1(C(c2cc(N)c(Cl)c(O)n2)=O)CCC2(NC(c3ccc(Cl)o3)=O)CCCC12 C1(NC(Cc2cc(C(=O)OC)sc2)=O)CCN(C(=O)C=Cc2nc(C)co2)CC1C N1(C(COC)=O)CCC(C)(NC(=O)C=Cc2cocn2)CC1 C(=O)(C(O)C(C)(C)CC)NCC1N(C(c2c(CC)nc[nH]2)=O)CCN(C)C1 CC1CN2CC(C)CN12.c1(C=O)cccnc1S.C(=O)CCCS Cc1cccc(CC(=O)NC2CCOC(CNC(c3ccnnc3)=O)C2)c1Cl C(=O)(C(O)C1=CCCCC1)N1CCN(C)CC1C(=O)NC1CN(C2CCC2)C1 C(=O)(CC1=CCN(C(c2cnn(C)c(=O)c2)=O)CC1)NC(CC)C(F)(F)F c1(-c2cc(C(N3CC(NC(CCc4cn(C)nc4)=O)C3)=O)n[nH]2)ccc(Cl)cc1 C1(NC(CC2(OC)CCC2)=O)CCC(CNC(c2cnc(O)o2)=O)C1 c1(OC)cccc([N+](=O)[O-])c1C(N1CC2CN(C(c3ccnc(O)c3)=O)C2C1)=O N1(C(CCSCC)=O)CCOC(C(=O)NCC2CC(CC)=NO2)C1 C1(CNC(C(=O)NCC)=O)CN(C(c2cnc(C(F)(F)F)cc2O)=O)CCC1C C1(C)(CC)CCC(C(N2CC(=C(F)CNC(=O)CC3CCOC3)C2)=O)O1 N12C(=S)NC(C3=C1CCN(CC)C3=O)c1cc(CC)cc2n1.OC c1(C(=O)NC(CNC(C(COC)O)=O)C(C)C)cc(Br)cnc1S O=C1C(NC(=O)NCC(O)C(F)(F)c2ccccc2)CCN1C1CCCCC1 CN1CC2CCN(C(C3CCCCC3CNC(=O)CC3CC(=O)C3)=O)CC2C1 CC1CN(C(=O)CC2CCCN2C(=O)C(F)=CC2CC2)C(C)CO1 N1(C(c2ccc(CC(C)C)s2)=O)CCN(C(c2ccccc2)=O)C2CCCC12 C1(CNC(CCCC2C(C)C2)=O)CCCCN1C(C1CC1c1ccccc1)=O N1(CC#C)CCN(C(=O)C(Cn2cccn2)NC(=O)Cn2ncnn2)CC1=O c1(SC(C)C(=O)NCCCNC(c2cc(-c3cccs3)on2)=O)ccc(F)cc1 CCCC(C(=O)NC(C)CCCNC(=O)Cc1cn(C)nc1C)C(C)C CCCC(C(=O)NCc1nccn1C)N(CC(F)F)CCOC N1(C(C(C)OCC)=O)CC2(CNC(=O)CC(C)CC)CC1CO2 N1(C(C(C2CCN(C(C3CC4CCC3C4)=O)CC2)C)=O)CCc2nc[nH]c2C1 c1(C(N2CC3C(Nc4nccc(I)n4)C3C2)=O)ccc2ncc(Br)n2c1 CCCCCCC(CC)NC(C1CC2CC2N1C(c1cc2ccoc2cn1)=O)=O N1(C(CCCC#N)=O)CCN(C(C2CC2CF)=O)C(c2cc(F)ccc2F)C1 c1(CC)cc(C(=O)NC2CCC(NC(=O)CC3CCC(=O)NC3)CC2)c(C)o1 c1(C(=O)NCCC(C)NC(CCCC(=O)NC)=O)cc(F)cc(N)c1F c1(C(c2n(CC(=C)C)nnn2)NCc2cc(C(N)=O)cs2)ccc(F)c(F)c1Br O=C(C#CC1CCCO1)NCC1CN(C(=O)CC(F)(F)F)CCCO1 C(=O)(C1=CCCC1C)NC1c2ccccc2OCC(=O)NC1.C(CN(C)C)OC C1(NC(Cc2ccc(C)nc2)=O)CCCCN(c2ncc(Br)c(O)n2)C1 c1(CNC(C2(SC)CC2)=O)ccc(CNC(=O)C(C)(O)C(C)C)c(F)c1 c1(CC)cc(C(=O)NCC(CO)NC(c2c(C)cccc2C)=O)cn(C)c1=O C1(CC)CN(C(c2ncc(Cl)cc2Br)=O)CCN1C(c1[nH]nnc1C)=O CC1CCC2(CO1)CN(C(=O)C(O)CCNC(C1CCCCN1C(C)C)=O)C2 c1(C(N(CC(C)O)CCNC(c2c(SCC)nccn2)=O)=O)ccnc(O)c1F c1(C(N2CCC(NC(c3cn(CCC)nc3)=O)(COC)C2)=O)nccc(N)c1Cl O=C1CC2C(C(=O)NC3(C(=O)NCC4(O)CCC4)CSC3)C2C1 CC1CCN(C(=O)Cn2cc(F)ccc2=O)C(CNC(C2(C)CCNC2=O)=O)C1 C1(C(N(C)CC2(NC(C(C)CC3CCCO3)=O)CC2)=O)COCCOC1 CC(C)CC(CNC(C1(CF)CCN(C(C2CCCC(O)C2)=O)C1)=O)CO C(=O)(CC(C)(C)CNC(C1CC1c1ccco1)=O)N1C(CCN(C)C)CCC1 c1(CC)cnoc1C(=O)NCC(C)(Cn1cccn1)NC(=O)CCOCC(C)C C(=O)(C1CC(=O)Nc2ccccc21)N1CC(C)N(Cc2cnn(C)c2)CC1 C1(NCc2cccc(C)c2F)CN(C(c2ccc(OC)nc2)=O)CCC1F C1(NC(C(=O)NCC)=O)CC2CC1CN(C(c1[nH]ccc1COC)=O)C2 Cn1c(O)ncc(C(=O)NC2CC(NC(C3(C(C)(C)O)CCC3)=O)C2)c1=O C(c1ccc(S(C)(=O)=O)o1)=CC(N1C2CCC(NC(C(C)NC(C)=O)=O)(C2)C1)=O C1(N(C(=O)C=CC(F)(F)F)C)CC2CCC(C1)N2C(C1CCNC1=O)=O N1(c2nnn(C)n2)CCC(O)(CNC(=O)C(Cc2ccccc2)C2CC2)CC1 CC1CN(C(C2CCC(=O)NC2)=O)CC1CNC(C1(C(F)(F)F)CCCCC1)=O C#CC1CCCC(NC(C23CC(CO2)N(C(=O)C(CC)OCC)C3)=O)C1 C1(OC)CC(CNC(c2cnn(CCO)c2)=O)N(C(=O)CC2CCCCO2)C1 CC1C(C(=O)N2CCCC(CNC(c3ncn4ccccc34)=O)C2)=NOC1C N1(C(=O)CCBr)CC(CNC(CCC(=O)N(C)C)=O)CCC1C c1(C(N2CC(O)(C(C)NC(=O)CC3CCCCC3F)C2)=O)cn2c(n1)COCC2 c1(NC(c2cc(SC)cc(C)c2)=O)cccc(Br)c1[N+](=O)[O-] Cc1nc2c(C(=O)NC(C)CNC(=O)CCCOc3cccnc3)ccnc2[nH]1 N1(C(c2c(C)nn(C)n2)=O)CC2CCC(CNC(C3OCCC3(C)C)=O)C2C1 CC(=O)CCCC(=O)N1CCC(C(C)NC(C2CN(C3CCCCC3)C2)=O)CC1 N1(C(CC(=O)OCC)=O)CCCC1(C)C(=O)N(c1cccc(CCO)c1)C1CC1 c1(C(=O)NC2CCN(C(C3CC(O)C3)=O)C2)cc(F)c(Cl)c(Cl)c1 n1(CC(=O)NC2CC(CNC(C3(C)N(C)CCC3)=O)C2)cnc([N+](=O)[O-])n1 c12cccc(n1)CNC(=O)N2.c1(COC(C)C)nnc(-c2cccs2)o1 N12CCC3CC(C3C1)C2=O.C1(OC)CC(CN(C)CC2CCN(C)CC2)C1(C)C S(=O)(=O)(c1cc(C)cnc1N1CC2CCC2C1)NC(C1CCCC1)COC C(C)(C(C(C)C)NC(c1cnc(C2CC2)o1)=O)NC(COCc1cc(C)no1)=O C(=O)(C(CC)C(C)C)N1CCN(CC2(NC(CCCC)=O)CC2)CC1 C12(NC(C3C(C(C)(C)C)CC3)=O)CCCC1(F)CN(C(=O)CCC1CCC1)C2 C1(CNC(c2cc(CC)c(C)s2)=O)CN(C(C2CCC(N=[N+]=[N-])C2)=O)CCC1C Cc1cocc1C(N1CC(NC(=O)CNC(=O)Cc2cccnc2)C1)=O c1(C(C(=O)NC)N(CC(C)COCC)CCC)ccnn1C1CC1 N1(C(C2CN(C(C)=O)C2)=O)CC(O)(CNC(=O)CCC2CCCCO2)C1 N1(C(Cn2c(C)c(Cl)cn2)=O)CCC(NC(=O)CCOCC2CCC2)C(C)(C)C1 C(=O)(CC1=Cc2ccccc2C1)NCC1(NC(C2CCCCC(=O)N2)=O)CCC1 Cc1ccc(CNC(=NCCc2nccnc2C)NCCF)c(Br)c1 C1(CC)(NC(=O)CCN2CCC2)CCCN(C(=O)COCc2cccc(Cl)c2)C1 c1(C(N2C(CCNC(C3OCC(C)C3)=O)CCC2)=O)cccc2c1OCCO2 C1(CNC(C2CC3C=CC2C3)=O)C2CN(C(=O)CN3CCC(F)CC3)CC12 c1(C(=O)NCCC2N(C(C=CCOCC)=O)CCC2)ccc(CCO)cc1 C1(C(=O)Nc2ccns2)CC12CCN(Cc1ccc(C(F)(F)F)c(Cl)c1)C2 N1(C(C2C(OCC)C2)=O)CCC2CCC(C1)N2C(=O)CCSc1cncnc1 c1(CC(CC)NC(=O)CSC2CCCC2)ccc(Br)cc1 C1(C(N2CCN(CCC#C)CC2)=O)CCN(C(=O)CSc2nc[nH]n2)C12CC2 C1(C(N(CC(=O)NCC2(SC)CC2)CC)=O)CCN(C(c2cscn2)=O)CC1 c1(C(=O)NCC2(F)CC(CNC(C(C)S(N)(=O)=O)=O)C2)cc2c(cc1Cl)NCC2 N1(C(CSCC(C)C)=O)CC2CC(C1)C2NC(=O)CCc1ccc(F)cc1 N1(C(=O)NCC=C)CC2OCCCC2(C(=O)O)C1 C1(C2CCCO2)(NCCC(C=C)C)CCN(C)C1.O=CNCC1CC1 c1(C(=O)NCC(C)CNC(c2cccc(C3CCOC3)c2)=O)ncnc(O)c1F c1(C(=O)Nc2ncc(OC)cn2)cccc(S(=O)(=O)N2CCN(C)CC2)c1 C1(NC(c2ccnc(C)c2N)=O)CC2CC(C1)N(C(c1cnc(Cl)[nH]1)=O)C2 c1(CC(=O)NCC(N(C(CNC(CCC)=O)=O)C)C2CC2)c(F)cccc1F C(CC(C(=O)N(C(C)CC(N)=O)C)NC(=O)Cc1csc(C)c1)OC N1(C(C2N(C(C)C)CCC2)=O)CCC(C)(C)C(C(=O)N2OC3CCC2C3)C1 c1(C(N2CC(CC(=O)NCC3(CCO)CC3)(OC)C2)=O)cnc(O)c(F)c1 c1(CC)nc(C(=O)NCC(C(C)C)NC(C2C3CCC2CC3)=O)c(Br)s1 Cc1ccc(C)n1-c1sccc1C(c1nnnn1C)NCC1(CO)CCOCC1 c1(CC(=O)N(CCNC(C(F)=C(C)C)=O)C2CC2)cn2ccsc2n1 CCCCCCC(O)CCC(=O)N(C)CCOCCNC(c1ncccc1C)=O C1(CC=C)(NC(c2cscc2OC)=O)CCN(C(c2cc(OC)cs2)=O)C1 C1(CN(C(c2ccc(C)cc2)=O)C)CN(C(c2ncncc2C#N)=O)CC12CC2 C(=O)(C(CCOC1CCCCC1)N1CC(O)CC1c1ccccc1F)OCC=C C(CC)(CCCC(=O)NCC1(C)CC1(F)F)NC(C1(CC#C)CCC1)=O CC(C)(C(=O)NCC1CCN1C(=O)CSC(F)(F)F)C1CCCO1 C1(NC(C=C(CC)CC)=O)CCCN(C(=O)Cc2ccc(C#N)cc2)C1C CC1CCCN(C(=O)C(Cn2cccn2)NC(=O)Cc2cnoc2)C1 c1(C(=O)NC2CCCN(C(c3c[nH]nc3F)=O)C2)cccc([N+](=O)[O-])c1Cl C(CC)(C(=O)NCC=CC(=O)NC1CC(C(=O)NC)C1)OCC C(C)(N=c1[nH]c(=NCCC(F)(F)F)[nH]c2ccsc12)c1ccc(OCCCCC)o1 C1(NC(C2(CC)CCC2)=O)CN(C(C2CCCC(=O)N2C)=O)CC1N=[N+]=[N-] c1(C(N2CCCC(NC(C(F)(F)C3(OC)CC3)=O)C2C)=O)cnn2cccnc12 Cc1ccc(SC(C)C(=O)NCCN(C(=O)COCC2CCCO2)C)cc1 c1(C(N(CCNC(CC2(C(C)=O)CCCC2)=O)C2CC2)=O)cccc(C)c1 Cc1c(Cl)ccc(C(=O)NCC(O)CN(C(=O)C=CCCC(C)C)C)c1O c1(C(CCO)N(C(CCN(CC=C)CC=C)=O)CCCC)ccccc1OC C(c1nc(C)co1)=CC(=O)NCCCCN(C(CCc1cc(C)on1)=O)C C1(C(=O)NC23CC(CNC(c4cc(SC)oc4)=O)(C2)C3)CN2CCC1CC2 c1(OC)cccc2[nH]cc(C(=O)NCCCNC(=O)CC(F)F)c12 c1(CN2CCC(CC)(NC(C3(CO)CCC3)=O)CC2)ccc(C#N)c(F)c1 c1(C(=O)NC2C(CC)N(C(c3ccc(Cl)cn3)=O)CCC2)ccn2ccnc2c1 C(=O)(C(C)(CC)OC)NC(C1N(C(c2cn(CCCC)nc2)=O)CCC1)C C(CC(C)C(=O)NCCC(C)N(C(=O)CCn1ncn(C)c1=O)C)OC CC(C)C(C)CC(=O)N1CC(NC(=O)CC(=O)N(C)C)CCC1C c1(C(=O)NC(CN(C(C(CC)c2cccnc2)=O)CC)C)snc(C)c1N N1(C(CCC(C)OCC)=O)CCOC(C)C1C(=O)NCC1CC(=O)N(C)C1=O N1(C(C(C)CCO)=O)CCC2(CC1)OCCCC2NC(=O)C(C)(C)C1CCCC1 C(=O)(C(C)(C)C(=O)OC)NC1CCC(C(N(C(C(=O)OCC)C)C2CC2)=O)C1 C(CN=C(NCC(=O)NC(C)(C)C)N1CCC(OC2(C)CCOCC2)C1)SC C=CCCCC(C(=O)NCc1ncc(CO)[nH]1)NC(c1cc(O)n(CC)n1)=O Cn1nc(-c2cn(C3COCC3O)nn2)c2cc(C(=O)NOC3CCCC3)sc12 c1(C(=O)NCC2(C)CCC(NC(CC3CC(OC)C3)=O)C2)ccc(C)c(F)c1 N1(CC(=O)NCC(CNC(CCOC)=O)F)CC(=O)N(C)C1=O C(=O)(CC(O)C(C)C)N1C(CCNC(c2[nH]cc(C)c2)=O)COCC1 C1(NCC(COC)C(=O)OC(C)(C)CSC)CCCCN(C(=O)OC(C)(C)C)C1 C(=O)(C1c2ccccc2C2CC1C2)N1CCC(C)(CS(=O)(=O)C(=O)NC(C)(C)C)C1 N1(C(C=C(C)c2ccco2)=O)CCCC(F)(CNC(=O)CC2CCCN(C)C2)C1 c1(C(=O)NCCCCNC(C2C3CCC(=O)C23)=O)cc(OC(F)F)ccc1F C1(NC(c2cc(C)on2)=O)CCN(C)C12CCCN(C(=O)C(C)OCC(C)C)C2 C12C(CC(=O)NOCCC(F)(F)F)CCCN1CCONC2=O.CC.CC c1(C(N2CCC(C)(CNC(C(C)(C)SC)=O)C2)=O)c(F)cncc1Cl C(=O)(C(O)CC[S+](C)C)NC(C1CN(C(=O)CCCNC(N)=O)CCO1)C C1(CNC(Cc2c(C)ocn2)=O)COCCN1C(=O)CC1CCC(=O)NC1 C1(CC#C)(C(=O)NC2CN(C(c3ncoc3C3CC3)=O)CC2C)CCCCO1 Cc1cc(C(=O)NC2CC(C)CN(C(c3cnccc3C)=O)C2)nc(O)n1 C1(NC(C(COC)C)=O)CCC(CNC(c2cccc(Cl)c2)=O)CC1 C1(NC(c2n[nH]c3ccccc23)=O)CN(C(=O)C=CBr)C2(CCCCC2)C1 C1(C(=O)N(C)CCc2cccnc2)(CC)CCCN(C(=O)C(C)CCOC)C1 C1(C2CC2)C(=O)N1.C(C(N)=O)(N(C(C1(OC)CC1)=O)C)C1CC1 c1(CC(=O)NC2CCCCN(Cc3ccnc(F)c3)C2)n[nH]c2ccc(Br)cc12 C1(CC)(OC)CCCN(C(=O)CNC2CC2)C1.C12CCCN1C2=O.CC N1(C(CCC(=O)SC)=O)CCCC(NC(c2csc(CO)n2)=O)C(F)C1 C1(C(=O)NC(C)C(C)(C)OC(=O)N(C)C)CCCCN1C(=O)C#CC1CC1 C#Cc1ccc(C(N2CC(CC(=O)NCc3[nH]c(C)nc3C)CC2C)=O)o1 c1(C(N(CCC)CCNC(=O)CSc2ccc(Cl)s2)=O)c(C)cccc1Cl N1(C(C2CCCN(C)C2)=O)CCN(C(c2cnc[nH]2)=O)C(CO)C1 N1(C(CCCC=C)=O)CC(NC(=O)Cc2c(C)cc(C)nc2O)CCC(O)C1 c1(-c2cc(OC)c(F)c(F)c2)cc(S(=O)(=O)NC2CCNCC2)c(C)cc1C CC(C)C(C(=O)N1CCC(c2cn(-c3cc(Br)ccc3F)nn2)CC1C)C(C)C c1(NC)ccc(Cl)c(C(=O)NC2CCC2CNC(c2ccc(N)cc2F)=O)c1 Nc1cc(F)ccc1NC(=O)C1=NNC(C(F)(F)F)C1.N12CC3CC1C3C2=O Cc1ccnnc1C(=O)NC1CCC(NC(C2(C)CCC(C)C2)=O)CC1 Cc1cccc([N+](=O)[O-])c1S(=O)(=O)N1CCN(CC(c2ccc(Cl)cc2)O)CC1 C1(C(=O)NC(CCSC)C(=O)NC2CN(C)CC2C)CCC2CC1CO2 C(=O)(CCC(C)(C)[N+](=O)[O-])N1CC(CNC(C2(C(C)C)CCOCC2)=O)C1 c1(CC)cc(C(N2CCC(N3CCC(O)C3)C2)=O)ccc1F.C(=O)C(F)(F)CC C(CS(=O)(=O)CC(=O)NCCC(C)(C)C(N1CC2C=CCC(C2)C1)=O)OC C=CC(CCC)CC(=O)NC(CCC(C)C)C(=O)NCC(O)(CC)CC c1(SCC(=O)NC2C(NC(=O)Cc3cccnc3)CCC2)cccc(C(F)F)c1 C1(C(=O)NC(C(=O)OCC)CO)CC12CCN(Cc1ccc(Cl)c(Br)c1)CC2 C=CCC(C)C(=O)NCCCCCCNC(c1cccc(C(C)(C)C)n1)=O C1(C(=O)NCC2(C)CCCC2)CN(C(=O)CC(=O)OCc2ccccc2)C(C)(C)C1 c1(C(C)C)cnn(C)c1C(=O)NOCC(=O)NCC1CC1C(F)(F)F C1(C)(CC(=O)NCC(C)SC)CCN(C(=O)CC2(C#N)CC2)C1 C1(NC(CSC)=O)CCOCC1NC(=O)CC1CCN(C)C1 NS(=O)(=O)CCCC(=O)NC1CCOC(CNC(=O)COc2ccccc2)C1 c1(C(=O)NCCC2CCN(C(c3ccn(C)c3)=O)CC2)cc(F)cc2nn[nH]c12 CC1CC2(CC(C(N3CCC(C(N4CC5CC5C5CC45)=O)C3)=O)C2)C1 C1(NCCN(C(C(CC)NC(C)=O)=O)CCCC)CN(C)CC1O N1(C(CCOCCC)=O)CCN(C(=O)C(C2CCCC2)OC)C2CCC12 N1(C(C23C(CN(C(C4C(C)CC4)=O)C2)C3)=O)CCC(C)(C#N)C1 c1(C(=O)NC(C2CCCN2C(c2csnc2Cl)=O)C)cc(Cl)cn1C c1(C(N2C(CN(C(=O)CC3CC(=O)NC3=O)CC)CCC2)=O)cc(C)ccc1Cl CC1(NC(=O)CC2CCCN2C(=O)CN=[N+]=[N-])CCCC1(F)F c1(NC(C2N(C(c3cnc(C)o3)=O)C(C)C2)=O)nc2ccc(C#N)cc2[nH]1 Cc1nc(C(N2CCC(CNC(c3ncoc3-c3cccs3)=O)C2)=O)n(C)n1 C(=O)(C1COc2cc(C)c(C)cc21)NC1CCN(C(c2cn(CC)nn2)=O)C1 Cn1cc2cccc(C(=O)NC3CCCC3NC(C3(C)CCOC3)=O)c2n1 N#Cc1ccc(NC(=O)CCCCC2CC2)c(O)c1.C12CC(CCO1)NC2=O C(=O)(CCCCCF)NC(N1CCC(C(c2ccc(C)cc2)C2CCCN2)CC1)=O C1(C2CCCC2)(C(=O)OCc2cccc(OC)n2)CCCCC1 C1(NC(CC(C)n2cc(Br)cn2)=O)C=CNCCCC1 C(C(C(=O)N1CC(c2ccccc2)C1)c1occ(CO)n1)OCC=C.N(CC)CC c1(NCC(CNC(c2coc(CO)c2)=O)O)ncnc2sc3ccccc3c12 C1(CNC(COCCOCC)=O)CC(CNC(C2CCC(C(N)=O)C2)=O)CO1.OC CC1CC(NC(=O)C=CC(=O)O)CN1C(=O)CSC(C)(C)C.C(C(F)(F)F)SCO N1(CC(C)C)CCCC(C(=O)NCC2(CNC(c3nnn(C)n3)=O)CCCC2)C1 C(c1ccco1)=C(C)C(=O)NCC(C)(C)CNC(c1ccc(-c2cccs2)[nH]1)=O c1(CN(CC(c2cccnc2)N(C)C)C)cnc(-c2ccccc2)nc1 N12CCC(CC1)C2.C1(CC(=O)N(CC(C)CC2CCC2)C)CCC(=O)N1 N1(C(c2cc(CNC(C(CC)OC)=O)[nH]n2)=O)CCN(C)C(C(C)C)C1 c1(C(=O)NCC23C(CN(C(=O)OC(C)(C)C)C2)CC3)ccc2c(c1)CCCO2 c1(CN2CC(C(=O)Nc3cccnc3)C(O)CC2)cnc2c(F)c(F)ccc2c1 c1(C(=O)NC(CC)CN(C(=O)CCOCC(C)C)CC)ccc(C)cc1C1CC1 C1(C)(CNC(C(c2cnn(C)c2)NC)=O)C=CCCC1 C12(NC(CCCOCCOC)=O)CCC(CC1NC(c1cncc(CO)c1)=O)C2 N1(C(=O)CCc2cnn[nH]2)CCCC(F)(C(=O)NC2CC3CC(O)C2C3)C1 C1(C(N2CC(F)(CNC(C(C)n3cccc3)=O)C2)=O)CCn2nncc2C1 C1(N(C(=O)COCCF)CCO)CCN(C2CCN(C(C3(F)CCC3)=O)C2)CC1 C(=O)(C1SCCc2ccccc21)NCCN(C(=O)CC(C)n1ccnc1)C(C)C c1(CC(=O)N(CC(CN(C(C2(C)CCN(C)C2)=O)C)O)C)ccc2c(c1)CC2 C1(C(C)(C)Nc2ccccn2)CCN(C(C2C(C)C2)=O)CC1.C1CC(=O)N1 c1(SCC(N2CCC(N(C(=O)C(C)OCCC(C)C)CC)C2)=O)cccc(F)c1 c1(CC(=O)NC2COCCN(C(=O)Cc3cccnc3)C2)cc(Cl)cnc1O c1(N(C2CCCOC2)C)nnc(C2CCCCO2)n1CCC#N N1(CC)CCN(C(C2CN(C(c3cc(C)ncc3C)=O)C(C)(C)C2)=O)C(C)C1 c1(C(NC(=NCC(C)C)NCCF)C)c(F)cc(NC(C2CCN(C)C2)=O)cc1F N1(C(c2nccc(OC)c2F)=O)CCOC2(C1)CN(C(C1CCC(=O)N1C)=O)C2 C(=O)(CC(C)CC(F)(F)F)NC(CC)CN(C)C(c1cc(F)c[nH]1)=O c1(C(N(C2CCN(C(C3CC(=C)C3)=O)C2)C)=O)coc2ccc(F)cc12 c1(C(=O)NC(C(=O)NCC(C)NC(=O)OC)(C)C)cc(C)c(C)cn1 CN1N=C(CC(=O)N2CC3CCC2CN3C(c2cnn(CC3CC3)c2)=O)CC1=O C1(NC(=O)CC2(O)CCCCC2)CCCN(Cc2ccccc2)CC1 c1(C(=O)NCC(=C2CN(C(C3CC(C)OCC3)=O)C2)F)ccn2c(O)nnc2c1 O=C1CC(CC(=O)NC2C3CN(C(C4(CO)CCCC4)=O)CC23)=NN1 c1(C(=O)NC2CCCC(N(C)C(c3cccc(N)n3)=O)C2)ccn2cnnc2c1 N1(c2ccc(C#N)nn2)CCC(NC(c2ccc(NC=O)cc2)=O)C(F)(F)CC1 N1(C(C=NOC)=O)CCC(C2CCN(C(=O)Cn3ccc(C)n3)C2)C1 C1(CC=C)(C(N2CC3CC2CC3CC)=O)CCN(C(=O)CC(C)=C(C)C)CC1 CN1CC(C(N2CCC(NC(=O)C=Cc3ccnn3C)C2)=O)CC1=O c1(NCC(c2c(OCC)cccc2)O)cc(=NC2CCOCC2F)[nH]c(CC)n1 N1(C(C=CC)=O)CCC(CO)C(NC(=O)CCN2CCCC2=O)C1 C1(CCC)(NC(c2ncc(F)cn2)=O)CCN(C(c2cnc(C(C)O)s2)=O)CC1 C12(C(=O)NCC(C(C)C)O)CCN(C(C3CC4(CCC4)C3)=O)CCC1C2 c1(CC)cc(Cl)ccc1C(N1CCC(NC(c2ccc(C#N)o2)=O)C1)=O c1(CC)c(NC(CNC(c2cc(C)cc(Cl)c2)=O)C(C)C(C)C)ncnc1Cl CC(C)C(C#N)C(=O)NCC1CCCC(CNC(=O)C(C(C)C)N(C)C)C1 c1(CC(N2CCC(CNC(c3cccc(CC)c3)=O)C2)=O)csc([N+](=O)[O-])c1 c1(C(N2CCC(N(C(CSCC=C)=O)C)C2)=O)c(C)cc(C)c(Br)c1C c1(C(=O)NC2CN(C(c3cnn(C(C)C)n3)=O)CC2C)cnc2[nH]c(O)nc2c1 N1(C(COC(C)(C)C)=O)CCC(F)(F)C(NC(c2cnn3ccccc23)=O)C1 S(=O)(=O)(c1ccc(Br)c(Cl)c1)NC1CC(C)CN(C(C2CCOCC2)=O)C1 C1(C2CN(C(=O)CN(C)C)C2)(NC(COc2ccc(C)cc2)=O)CC1 c1(C(N2CC(N(C(=O)C(=O)NC3CC3)C)C(F)C2)=O)cccc(O)c1F C1(C)(CNC(CCCC#CC)=O)COCCN(C(=O)CC2CCC(OC)CC2)C1 c1(OC)cccc(OCCC(=O)N(CC(C)NC(=O)COCCSC)C)c1 CC1CCC(NC(=O)C(F)Cc2ccccc2)CN1C(c1ccc(O)c(Cl)n1)=O c1(OCC)cncc(C(N2CC(O)(C(C)NC(=O)C(C)NC(C)=O)C2)=O)c1 N1(C(C(C(C)C)OCC)=O)CC(NC(=O)CCC[N+](=O)[O-])CC(C)C1 c1(CCC)n[nH]cc1C(=O)NC1CC(NC(=O)CSc2nnc(S)s2)C1 c1(OCC)cccc(CC(=O)NCCC(C(C)C)NC(=O)Cc2cn(C)cn2)n1 C1(C(=O)NCC(CO)N(C)C)CCC(NC(C2CC2(F)Cl)=O)C1 c1(C(=O)NCCC(N)=O)ccc2[nH]c(NC(=O)C(c3ccccc3)=O)cc2c1 Cc1ncnc(C(N2CC(C)(C(=O)Nc3c[nH]ccc3=O)C2)=O)c1C N1(C(C(CCC)C)=O)CCC(F)(F)C(CNC(=O)C(c2ccccc2)O)C1 Cc1cc(C(=O)NC(C)(C)CNC(C2CC(OC(C)(C)C)C2)=O)nc(N(C)C)n1 CC(C)C(CNC(c1cnn(C(F)F)c1)=O)N=c1nc(CC2CC2)[nH]s1 c1(C(N(C)CC2CCC(NC(C(CSC)O)=O)CC2)=O)cc(Cl)ccc1F CC(C)CC(C)C(=O)NCC(c1ccccc1)N(C)C(c1ccc(C#N)cn1)=O C1(NC(Cc2ccc(OC)cc2)=O)CC2CCC1N2C(=O)Cn1cccc1 n1(C(N(C2CCN(C(=O)C(C)OCCC(C)C)C2)CC)=O)cnc2c1CCCC2 C(=O)(C1CCCc2ccccc21)NC1CCN(C(C(C)OCC#C)=O)C1C N1(CCC(=O)NCC2(C)CCN(C(C(CC)O)=O)CC2)C(=O)NC(C)(C)C1=O Cc1oc(C#N)cc1C(=O)NCC(C)(C)CCNC(c1ccc(F)c(Cl)c1)=O C(=O)NNc1cc(F)cc(Br)c1.CN1CC(O)CC1 CC1(NCc2cccnc2)CCN(C(=O)Cc2c[nH]c(Br)c2)CC1 c1(CCN(C(=O)Cc2ccns2)C)ccc(C2CC2)cc1F.C12(CC1)CC(=O)N2 C12(NC(=O)CCNC(c3ccc(F)cc3)=O)CCC1CN(C(C1CC1F)=O)C2 C1(C(C)NC(c2c(C)ccs2)=O)CCCN(C(c2cn(CCC(C)C)nn2)=O)C1 C=C(C)C(O)CC(=O)NCC1CCN1C(c1cc(Oc2ccccc2Cl)ccn1)=O c1(OC)ccc(C(N2CCCCC2CF)C(=O)NC2(CSC)CC2)c(Cl)c1 c1(OC)ccc(C(=O)NC23CCC(C(=O)Nc4c(C)ncn4C)(CC2)C3)c(Cl)n1 S(=O)(=O)(c1cccnc1)NC(=O)CCc1ccccc1O C(CC(C)(C)COC)NC(c1c(CCC)nco1)=O.N12CCC1(C)C2=O.CCO C1(CNC(CC(C=C)C)=O)CCC2(CC1)CCN(C(=O)CCF)CC2 c1(C(N2C3CC(NC(CC(C)C)=O)C(C3)C2)=O)cc2n(n1)CCCC2 N1(C(C2C(C)C2)=O)C2CCC1CN(C(=O)CSCC(N)=O)CC2 C12(NC3CCCN(C(CSCc4scc(C)c4)=O)C3)CCC(CC(N)=O)(CC1)C2 c1(-c2cc(C(=O)NC3CN(C(C4(SC)CC4)=O)CC3O)no2)ccc(F)cc1C C1(NC(CC=CC)=O)CN(C(=O)C(c2ccncc2C)C)CC2(CC2)C1 C(=O)(C1=CCCOCC1)N1CC2C(N(C)C(C3CCC4(CC3)N=N4)=O)C2C1 N1(C(Cc2cccc(N)c2N)=O)CC2CC(NC(C3CCS(=O)(=O)C3)=O)CC2C1 c1(C(N(C2CN(C(C3(COC)CC3)=O)CC2C)C)=O)ncc(F)cc1N CN1CCN(CC(=O)NC2(C3CN(C(c4cc(CCO)on4)=O)C3)CC2)CC1=O C=CCCCC(C(=O)N1CCOC(CN(C)C)C1)NC(c1csc(CO)n1)=O c1(CC(=O)NCC2CC(NC(=O)C(c3ccccc3)O)C2)cccc(Cl)c1F C1(OC)CC(CNC(c2ncc(C(F)F)s2)=O)N(C(=O)Cc2cncn2C)C1 N1(C(C2C3CCCC23)C(=O)NCc2nnn(C)n2)CCC2CCC(C1)S2(=O)=O Cc1csc2ccc(C(=O)NNC(=O)CC(=O)CN=c3cc[nH]cc3)cc12 C1(CCCC)CN(C(C2CCC(C(F)(F)F)O2)=O)CCN1C(C12CCC(C1)C2)=O c1(SCC(N2CC(=C(CNC(C3CCCSC3)=O)F)C2)=O)nc2ccccc2s1 CC(C)(C)CC(CNC(C1CC1c1cccs1)=O)C(=O)N1CCSCC1 CN=c1[nH]c(=NCCCCNC(C)C)[nH]c(=NC2CCC3(C2)CC3(F)F)[nH]1 N1(C(C(c2cccc(Cl)c2)C)=O)CC(CNC(=O)C(C)(F)F)C(F)(F)C1.C(CO)O c1(OC(C)C)c(C(=O)NCC(C)(C)NC(=O)C(C)C2CCCO2)cccc1N c1(C(N(CCC)CCNC(C2(OC)CCC2)=O)=O)cc(C)nnc1O CC(CC(=O)NCC1C2CC(F)C(C2)C1(C)C)C(C)(C)C C12(c3cn(-c4c(OC)ccs4)nn3)CC(CN1C(C1(c3c[nH]cc3C)CC1)=O)C2 N1(C(C2OCC(C)(C)C2)=O)CCN(C(c2ncc(F)cn2)=O)CC(O)C1 N1(C(C(CC=C)OC)=O)CC(CNC(c2ncccc2SCC)=O)CC1(C)C c1(C(=O)NCC(C(C)C)NC(CC(CC)C)=O)ccc(Br)cc1-n1cncn1 c1(OC)c(C(N2CC(NC(C3C(F)(F)C34CC4)=O)CC2CO)=O)cc(F)cc1F n1(CC)ncc2c(NC(C3C(CNC(=O)NC)C3)=O)cccc12 CC(C(=O)N1CC(C(=O)NCCNC(=O)C2CC2)C1)C1(O)CCC1 c12ccc(C)n3cc1nc23.Cc1cc(NC=O)ncc1C#N.CO C1(CNc2cc(NC(CCSCC)=O)ncn2)CCCC(C(F)(F)F)C1 N1(C(c2[nH]n(C)c(=O)n2)=O)CCC(NC(=O)Cc2ccc(F)cn2)C1(C)C C(=O)(C(C)CCC(C)C)NCCN(C(=O)C(CCCC)N(C)C)CC.CCCO CCC(C#N)C(=O)N1CCC(C(=O)Nc2ccsc2)(SC)C1 CCCC(CC)CCC(=O)NC(Cc1cnc[nH]1)C(=O)NOCCCN(C)C C12(NC(C3(NC(=O)CCC4CC4(F)F)CSC3)=O)CC(F)(C1)C2 c1(OC)c(C(N2CC3C(C(=O)NCC4CCC(F)C4)C3C2)=O)cccc1[N+](=O)[O-] c1(C(N2CCC(C)CC2)=O)n[nH]c2c1CCN(C(c1ccc3sccc3c1)=O)C2 C1(NC(=O)Cn2ccnn2)CCCCC1NC(C1(c2ccc(F)cc2)CCC1)=O c1(C(=O)NC2C(CNC(CCC3(C)CC3)=O)CCC2)cc(N)ccc1C(F)(F)F c1(C(=O)NC2CCCC(CNC(CCCC=C)=O)C2)cc(F)c(F)c(N)c1Cl N1(C(c2ccc(C#C)cc2)=O)CCCN(C(=O)C(C)C#N)C(CCC)C1 c1(C(N2C(CN(C)C(C3(CC4CC4)CC3)=O)CCC2)=O)cc2n(n1)CCC2 C1(NC(C(CC)SC)=O)CC2(C1)CC(NC(=O)CC1CCCN1C)C2 n1(CC)cnc2nc(=NC(C)CCC(C)C)[nH]c(NCC3(CF)CCC3)c12 N1(C(C(=O)N(C(C)C)CCO)=O)CCCNCCC1C c1(C(N2C(CC)CCCC2)C(=O)NCC(F)F)cnc2onc(C)c2c1 C(=O)(CC(C)C(C)(C)NC(c1cnn(C2CC2)c1)=O)NC(C#C)CC1CCC1 c1(C(=O)NC2CC(C)(NC(c3csc([N+](=O)[O-])c3)=O)C2)ccc2nccn2c1 c1(C(=O)NC2CCC(C)N(C(=O)CP(C)(C)=O)C2)cc2ccccc2nn1 C1(C(=O)NCCNC(C2CCCN(C(=O)OC(C)(C)C)C2)=O)CCC12CCNCC2 c1(COC)cccc(NC(C2CCC(CNC(C3(C4CC4)CC3)=O)O2)=O)c1 N1(C(C=C(C)C)=O)CCN(C(C2CCCCC2O)=O)CC1c1ccccc1 Cc1cccc(-c2cncc(C3CCN3)c2)c1.n1(CCCS)cnc(C#N)n1 N1(C(c2scc(NC(=O)CC3CCSCC3)n2)=O)CCc2ccc(Br)cc2C1 c1(CC)cc(NC(=S)NCC)cc(OCc2cc(Br)ccc2F)c1 c1(-n2cc(CCC(=O)OCC)nn2)ccc2nc(OCC(=O)O)oc2c1 c1(C(=O)NCC2N(C(CC(C=C)CC)=O)CCC2)c(OC)ccc2c1CCC2 C(CC1CC1)(CCNC(=O)OC(C)(C)C)Oc1csnc1-c1cnc[nH]1 c1(C(N2CCC(NC(C3(O)CN4CCC3CC4)=O)C2)=O)ccc(F)c2ccsc12 CN1CC=C(CC(=O)N2CCC(C(F)C(=O)NCCc3nc(O)n[nH]3)C2)CC1 c1(NC(CC)CC(F)(F)F)ccc(S(=O)(=O)NCC(O)CC2CCC2)cc1Br C(CCCC(C)NC(=O)CC(C)(C)C1CC1)NC(C(C)OC1CCCC1)=O C1(N(C(=O)Cc2cncs2)C)CCC(NC(c2ccc(-c3ccco3)[nH]2)=O)CC1 C(=O)(C1=CC(C)(C)C1)N(CC(C)NC(c1ccc(CN2CCSCC2)cc1)=O)C C=CCC(C)(C)CC(=O)NC1CC1CNC(c1ccc(F)c(C(F)(F)F)c1F)=O CS(C)(=O)=NCC(=O)NCC1CN(C(C)(C)C)CCO1.C12CC(C1(C)C)C2 C1(C(=O)NC(C=CC(=O)N(CC(=O)OC)C)C)OCCC1C(C)C C(=O)(C(C)(C)CC(=O)N1CCCN(C(=O)COc2cccc(Cl)c2)CC1)OCC Cc1cc(C)c(CC(=O)N(C)CC2CN(C(C3CCC34CCCO4)=O)C2)c(C)c1 C1(CN(C)C(C2CCCN(C(=O)C(F)(F)CO)C2)=O)CCCN(C(N)=O)C1 CS(=O)(=O)c1ccsc1C(=O)Nc1ncc(Br)cc1C(=O)O C12(CNC(C3N(C(=O)OC)CCC3)=O)CC1CN(C(C1(C)CSC1)=O)C2 c1(C(=O)NCC2(O)CC(OC)(OC)C2)cc(F)cc(F)c1 N1(C(c2c(C)nco2)=O)CCSCC1C(=O)NCC1COCCO1 CCCC(C(O)C(=O)NCCC#CCO)NC(=O)C(C)NC(C)=O C1(NC(CC2ON=C(CC)C2)=O)CCCN(C(=O)C=Cc2cncc(F)c2)CC1 C(CCCC(=O)N1CCCC1CCNC(c1c(C)cccc1F)=O)(OC)OC C12(CNC(C(CC)O)=O)CCCC(CN1C(c1ccc(=O)n(CC3CC3)c1)=O)C2 N1(C(CC)=O)CCC2(C1)CN(C(C1CCC(O)CN1C)=O)C2 n1(CC)ncc(C(=O)NC2CC(CNC(=O)C(C)(C)C3CCCO3)C2)c1Cl C1(C(N2CC3C(NC(C4(CSC)CCC4)=O)C3C2)=O)CCn2nccc2C1 c1(C(N2CCCC(O)(CNC(C(CCC)C)=O)C2)=O)ccc(C)c(F)c1F N1(C(C2(COC)CC(=C)C2)=O)CCOCC(NC(C(C)(C)C(C)(C)O)=O)C1 Cc1ncnc(C)c1C(=O)NCC(O)CNC(=O)C(N1CCCCC1)C N1(C(CCC(C)C)C(=O)NCC(C)C)CCCC2(CCCO2)C1 N1(C(Cn2ccc(C)n2)=O)CCC(O)(CN(C(=O)CN2CCC2C)C)C1 N1(C(CCCC2(NC(C(CSC)O)=O)CCC2)=O)CCC2(CCCOC2)C1 C1(CNC(c2cn(C(F)(F)CO)nn2)=O)(NC(c2cc(Cl)no2)=O)CCCC1 c1(C(C(=O)OCC)N(C(C(=O)OCC)C)C)ccnc(OC(F)F)c1 c1(C(=O)NCC(CC)(CC)NCC(C)CS(C)(=O)=O)cnc2sc(C)cn12 N1(C(C=CCCC)=O)CC(NC(c2ccco2)=O)CC12CCCC2 N1(C(CCCNC(COCCCC)=O)=O)CCc2cccc(C)c21 c1(C(=O)OCc2cccc(CC)c2)ccc(C(F)(F)F)nc1N c1(C2(C(=O)NC3C(CNC(c4cc(O)ncn4)=O)CC3)CC2)ccc(F)cc1 c1(C(=O)NCC(C)CNC(c2ccnc(C(=O)N(C)C)c2)=O)ccc(Cl)c(O)c1 c1(C(=O)NC2(C(=O)NC3C(OC(C)=O)C3)CC2C)ccn(C(C)(C)C)c1 N1(C(C(C)OC)=O)CCN(C(=O)CCc2cccc(F)c2Br)CC1CO S(=O)(=O)(c1cccc2scnc12)Nc1onc(C)n1.c12n[nH]cc1N2 C(=O)(C(C)S(C)(=O)=O)N1CCC(F)(CNC(COCCCCCC)=O)C1 C12(C(=O)Nc3cn(C)nc3)CC1CN(C(c1ccccc1C(C)(C)C)=O)C2 c1(C(=O)NCC(CC)NC(c2ccc(-c3ccc(Cl)cc3)s2)=O)ccc(O)nc1 CC1CC(NC(=O)CCc2cccc(O)c2)CN1C(=O)CCOC1COC1 N1(C(C2(C#N)CC2)=O)CC2C(CNC(c3ccc(C(F)(F)C(F)(F)F)s3)=O)C2C1 C(=O)(CCC(C)N(C)C)NCC1N(C(=O)NCc2nc(CC)sc2)CC=C1 N1(c2snc(C)n2)CC2CCC1CN2C(C1CCCCC1C1CC1)=O Cc1ccc(CCC(=O)N2CCC2C(=O)NC2CCCC(=O)N2)c(C)c1 N1(C(C2C(C(C)C)N(C(=O)CCC3CCCCC3)CC2)=O)CC2(C1)CC(C)(O)C2 c1(C(N(CC(C)NC(=O)Cc2nc([N+](=O)[O-])n[nH]2)CC)=O)ccn2nccc2c1 C12(NC(c3cnc(CC)s3)=O)CN(C(C3(C)CCOCC3)=O)CC1CS(=O)(=O)C2 c1(C(N2C(C(C)(C)NC(=O)CCCCCl)CCC2)=O)cc2cc(Br)cnc2s1 C=CC1CCCN1C(C1CCOC1CNC(=O)CC(C)C)=O C1(C2(O)CN(C(=O)CSC3CC3)C2)(CNC(c2c(OC)c(F)ncc2)=O)CC1 c1(NC(CC)CC#N)ncnc(N2CCC(NS(=O)(=O)CC)CC2)c1C N1(C(CSCCOC)=O)CCC(NC(c2ccncc2OC)=O)C(O)C1 C1(CNC(C2(CC)CCCC2)=O)CCN(C(=O)CC2CCC(=O)N2)CC1C CC1(C)CCc2[nH]c(C(N3CC4C(NC(C5CC(=O)N(O)C5)=O)C4C3)=O)cc2C1 c1(C(N2C(C(=O)NCc3cnc(CC)s3)CSC2)=O)nccnc1C(N)=O C1(CNC(c2c(C)n(C)cn2)=O)CN(C(C2(C)CC=CC2)=O)CC(C)(C)O1 n1(CC)ncc(CNC2CCC(N)C2)c1C C(C(O)C(F)(F)F)NC(c1c(CNC(CC2(C=C)CCC2)=O)ccs1)=O C1(C(N2CC(NC(c3c(CC)cccc3)=O)C(OC)C2)=O)COC2(CCC2)C1 Cc1cnnc(O)c1C(N1CC2CC(C1)C2NC(C1CCCN1C=O)=O)=O Cc1cc(F)c(CN2CC3(CC(C(=O)NCCNCCO)C3)C2)c(Br)c1 C1(O)(CNC(C2CC(O)C2)=O)CCN(C(c2ccc(Cc3ccccc3)o2)=O)C1 c1(NC(C2C(C(=O)NCc3c(C)c(F)ccc3)C2)=O)nc(Cl)c(C)c(Cl)n1 N1(C(c2nccc(CC)c2)=O)CC(NC(C23CC(CNC2=O)C3)=O)CC(C)C1 C(c1ccccc1Br)=CC(=O)NCC(CC=C)NC(c1nc(C)sc1C)=O c1(C(N(CC=C)CC=C)=O)ccc(=N)[nH]c1.C1CC(=O)N1CCOC Cc1nc(C(=O)O)c(C)n1C1CC1NCc1nnc(-c2cccc(Cl)c2F)o1 C1(C(N2CCCC(CC)(CC)C2)=O)COCCN(C(=O)C(C)(C)CN(C)C)C1 c1(C(=O)NC2CN(C(C3C(C(=O)OC(C)(C)C)C3)=O)C2)cc2ccccc2o1 CCC(O)C(=O)NCCCCCNC(=O)CCNC(=O)C(C)(C)C CC(Cc1cccc(Cl)c1)N=c1ccnc(NCc2csc(-c3ccco3)n2)[nH]1 C(=O)(C(C)(CC)C(N)=O)NCC(CC=C)NC(=O)COC(F)(F)F c1(CN2C3CN(Cc4ccc(OCC)cc4)C(C3)C2)ncc(C#N)c(OC)n1 c1(OCC(c2nnnn2CSC2CCSC2)Nc2nnc(C)s2)ccccc1F N1(C(C2(OCC)CC2)=O)CCC(F)(CNC(c2cccc(C(C)C)n2)=O)C1 C1(C(C)NC(=O)CN(n2cncn2)C)CCN(C(=O)Cn2cccn2)CC1 C1(c2nc(-c3ncccn3)no2)(OC)CCN(C(c2ccccc2)C)CC1 N#Cc1cc(NC2CN(C(c3cnsc3)=O)CC2C(F)(F)F)c([N+](=O)[O-])cc1F C(=O)(C(F)(F)C(O)CC)NCC1OCCN(C(C(CCC)N(C)C)=O)C1 CCC(CN(C)C)CC(=O)NC1CC(NC(=O)Cc2cc(OC)ccc2OC)C1 N1(C(c2c(CC)nc[nH]2)=O)CC2CC(NC(C3CCC(C)NC3=O)=O)CC2C1 c1(OC)cc(C(N2C3CCC2CC(CNC(=O)C(C)CF)C3)=O)c(OC)cc1Cl C1(CNC(c2c(OC)ccs2)=O)CN(C(=O)C(c2ccccn2)C)CCO1 c1(N(C)C)ccc(C(=O)N(C2CN(C(c3cccn3C)=O)CC2F)C)cc1 C1(C(=O)NCCCN(C(CC2(OCC)CC2)=O)C2CC2)(CC)COC1 CC1CC(CNC(c2[nH]c(=N)sc2C(F)(F)F)=O)CN1C(=O)C=CI C#Cc1cccc(CC(=O)NCC2CC(C(=O)NCC=CCOCC)=NO2)c1 CN1CCC(C(=O)NC2(C)CN(C(=O)C3=NOC(C)(C)C3)C2)c2ccccc21 O=C(CC(Cc1cccs1)C(=O)O)Nc1ccc(OCC(F)(F)F)cc1 C1(c2n(CCC)nnn2)(NCC(=O)OCc2ccccc2)CC2COC1C2 c1(CC(=O)NC2C(NC(CCOCC)=O)CS(=O)(=O)C2)ccc(Cl)c([N+](=O)[O-])c1 c1(C(N2CC(NC(C(CC)=CC)=O)C(C)C2)=O)ccc2cncn2c1 c1(C(=O)NCC2OCCN(C(c3cc(C)oc3)=O)C2)cc(O)c2sccc2c1 C1(C(=O)NCCCC(C)NC(CC(COC)C)=O)CCCC(C)CC1 C1(NC(c2cncc(SC)c2)=O)C(C)CN(C(=O)Cn2ncccc2=O)CC1C c1(CC(=O)N(CCC(=O)NCC(C2CCC2)OC)C2CC2)cn(C)cn1 N1(C(c2cc(OC)cc(C)c2)=O)CC2(CCC(CNC(C3C(C)C3C)=O)O2)C1 N(C1CCCc2nc(C)sc21)Cc1ccc(N(c2ccccc2)CC)cc1 c1(OC)cc(F)c(C(N2CCC(C3CCCCN3C(=O)C=CCF)C2)=O)c(F)c1 C(=O)(C(C(C)(C)C)NC(=O)CC1CCC(C)(C)C1)NCc1c(C)con1 c1(OCC(=O)NC(C)(CNC(c2cc(F)c[nH]2)=O)C2CCC2)ccc(F)c(F)c1 C12CCCN(C1)CC1CC21.CC(C)C=CCNC(=O)NC(C)(C)C C(=O)(C(F)(F)C(F)F)NC1CC2(C(NC(c3nccc(N)c3)=O)C2)C1 C(=O)(C(C)C(C)n1cccn1)NC(COC)CNC(=O)Cc1ccccc1 Cn1cnc2c(C(=O)NC3CCCC3NC(C3(CC4CC4)CC3)=O)cccc12 c1(C(N2CC(CNC(C3(OC)CCCC3)=O)C(O)C2)=O)ccc2c(c1)COCC2 CC(C)CCC(=O)NC1CC(O)(CNC(c2ccccc2-c2cncnc2)=O)C1 CC1CCN(C(=O)C(O)Cc2cn(CCN3CC(C)(C)C3)nn2)C1C1CC1 c1(N(C2CNCC2O)C(C=C(C)C)=O)ncnc2ncc(Br)cc12 c1(CC)noc(CC)c1CC(=O)NCC1CC1NC(c1c(C)noc1N)=O CC(C)(CN=c1[nH]c(=NCCN2CC=CC2)[nH]c2c1CSC2)C(N)=O N1(C(COC)=O)CCC(CNC(c2ccc(N3CCNS3(=O)=O)cc2)=O)C(C)C1 c1(OC)nccc(I)c1CN1CCOC(CC(=O)NCC2(C(F)(F)F)CC2)C1 c1(C(=O)NCc2cccc(CNC(C)=O)c2)c(C)sc(C)c1C C(=O)(C(O)C(C(C)C)OC)NCCN(CCOC)Cc1ccc(C)c(O)n1 C#Cc1ccc(C(=O)NC(CNC(C2CC(C3CC3)=NO2)=O)CO)cc1 Cc1cc(C#N)ccc1C(N1CC(CNC(C2(C)CC2C)=O)C(O)C1)=O N1(C(C(C)CC2CCC2)=O)CCC(NC(=O)COC2CCC(F)(F)CC2)C(O)C1 c1(C(=O)NC(C)CCNC(=O)Cc2ccnc(F)c2F)cc2ccccc2o1 c1(NC(C2SCCN(S(CCC)(=O)=O)C2)=O)ccc(OC)c(S(N)(=O)=O)c1 CC1CN(C(c2csc(CNC(C3CC(C(C)C)=NO3)=O)c2)=O)C(C)(C)C1 C1(C(N2CCN(CC(=O)NC(C)CO)CC2)=O)(OC)CC(C)(C)C1 C=CCC(C(=O)N(CCCNC(C1CC(=C2CCC2)C1)=O)CC)C(C)C CC1CCN(C(=O)C(F)OC(F)(F)F)CC1NC(=O)C(Cc1cccs1)N(C)C C(C(O)CC(=O)N(C)CC1CCCO1)NC(C(C)c1cc[nH]n1)=O CN1CCC(C(=O)NC2CC2NC(c2cccc(F)c2Br)=O)CC1=O N1(C(C(C2CC2)OC)=O)CC(NC(=O)CCC2CCC2)CC12CCCC2 C=CC(C)(O)C(=O)NC(C)CN(C)C(c1nnn(Cc2ccccc2)c1CC)=O C1(CC=C)(NC(=O)COC2CC=CC2)CCN(C(C2(CF)CC2)=O)CC1 c1(Cc2cc(OC)ns2)nc(-c2ccc(C)cc2)nn1C(C1CCOCC1)C c1(-c2scc(CN3CCC(C#N)C3)n2)nc2ccccc2o1 Cc1ccc(-c2ccccc2C(=O)NCC(C)N(C)C(C2CC23CCC3)=O)cc1 Cc1cc(C(=O)NCC(c2cccc(C)c2)NC(C2CNC(=O)N2)=O)cc(N)c1 CC(CC(=O)NCCOCc1ccccc1Br)CC(C)(C)C N1(C(c2c(C)n(C3CC3)cc2)=O)C2CCC1CC(NC(C1CC1F)=O)C2 C1(O)(CN(C)C(C2(C)C(C)(C)C2(C)C)=O)CCCN(C(C2(C)CCCN2C)=O)C1 N1(C(c2ncn(C(C)C)c2)=O)CC2CCN(C(C34CCC3C4)=O)CC12 c1(C(=O)NCCC(C)NC(CCOCC)=O)c(C)ncn(C)c1=O N1(CC2N(C(=O)Nc3ccccc3CO)CCCC2)CCOC(CF)C1 C(CCC(=O)NC1(C(=O)NC)CCC1)C1C(C)C1.C1(CN)CCCCO1 Cc1cc(C(=O)NC23CCC(CC2)N(C(=O)CC24CC(C2)C4)C3)n2ncnc2n1 c1(OC)ccc2c(c1)C(N(C)S(=O)(=O)Cc1cc(C)no1)CC2 c1(C(=O)NC2CC(CNC(CCn3c(C)ncc3)=O)C2)cc2n(n1)CCCC2O C12(NC(C3C(NC(C4C(C)(C)OCC4)=O)CCO3)=O)CCC(CC1O)C2 c1(CC)cccc(C)c1NC(=O)C(c1cccc(Br)n1)N1CCCC(CCF)C1 N1(C(c2c(C)nco2)=O)CCC(C2CC2)(CNC(=O)C=CC(F)(F)F)C1 N1(c2nc(C)c(C)nn2)CCCC(C2CC2NC(c2cnn(C3CC3)c2)=O)C1 Cn1nc(C2CC2)cc1C(N1CC(CNC(=O)Cn2cnnc2)C2CC12)=O CCC(C)(CC)C(=O)NCc1ccccc1CN(C)C(C1CCC12CCC2)=O C(=O)(C1=CCCN(C(C2CCC(N(C)C)C2)=O)C1)Nc1cc(C)cc(C)c1 c1(N2CC(C(C)NC(c3cc(C)ns3)=O)OCC2)ncc([N+](=O)[O-])cn1 c1(C(=O)N(CCNC(C23CCCC2CC3)=O)C2CC2)ccc(F)c(O)c1 N1(C(C2CN(C(c3cc(C)c(C)nc3)=O)CC2(C)C)=O)CC2COC(=O)C2C1 N1(C(C(C)Cc2cnc[nH]2)=O)CC2CCC(NC(=O)C(C)C(C)(C)C)CC2C1 C1(C(=O)NCc2cc(C)nc(C)c2)CC(N=[N+]=[N-])CN1C(c1ccc[nH]1)=O C12(NC(CCC(CC)CC)=O)CC(C)(C1)OC21CN(C(c2cccnc2O)=O)C1 n1(Cc2occc2)ccc(=NC(C)(c2nnnn2-c2ccccc2)C2CC2)[nH]1 N1(C(C(C)(C2CC2)OC)=O)CCOC(C(=O)NCc2cncs2)C1 CCC(C)C(=O)C(=O)NCC(CC1CCCC1)C(=O)NCCCC(CC)CC C1(C(CNC(=O)C(C)Oc2ccccc2Cl)NC(COC)=O)CCCCNC1=O C1(C(N(C)CC2(NC(c3cnn(C)c3)=O)CC2)=O)CC2COCC12 c1(OC)nccc(C)c1C(=O)NCCCOCCCNC(c1cncnc1)=O CC(O)(CN=c1ccn2cccc2[nH]1)c1cc(Cl)cc(Cl)c1 c1(C(=O)NCCN(C)C(C2CCS(=O)(=O)C2)=O)cc2c(=O)n(C)c(=O)n(C)c2s1 C(C(C(=O)NCC1CC2CCC1O2)C(C)(C)C)NC(C(C)CC1CC1)=O c1(C(=O)NC(CC)CNC(c2cc(O)no2)=O)ccc2ncnn2c1 C12(C(N3C(C)(C)CC(CNC(C4CC5(CCC5)C4)=O)C3)=O)CCC(C)(CC1)CO2 Cc1nc(C)c(CNC(=O)CCC2CCN(C(=O)C(C3CCOCC3)C)C2)[nH]1 N1(C(c2ccc3nccnc3n2)=O)C2CCC1C1CC1(CC(=O)NCC(N)=O)C2 C(=O)(CCCC(=O)NCC1CCCCN(C(C2(C)CCCN2C)=O)C1)NCCC c1(CC)ccc(C(N2CCC(CNC(C3(C(F)F)CCCO3)=O)C2)=O)s1 N1(C(C2CCSC2)=O)CC2CCC(C1CO)N2C(c1sccc1CO)=O Cc1cc(C(C)(C)C(=O)N2CCC(C3CCCN3C(=O)C3CC3)C2)ccc1Br C1(NC(CC2(C=C)CN(C(=O)CCCC(=O)C3CC3)C2)=O)CC1C1CCCC1 c1(CC)c(C(=O)NCC(O)C(=O)N2CC(C)(C(F)(F)F)C2)nnn1C C1(F)(C(N2CCC(C(C)(C)NC(c3ccon3)=O)C2)=O)CCCCC1 n1(CCCC)cc(C(=O)NCCOC2CCN(C(=O)Cc3cncn3C)C2)nn1 C1(C)(C(N(C)CCNC(=O)CCCCCC2CC2)=O)CCCNS1(=O)=O c1(CNC2CC3C(N)C3C2)cccn2cncc12 C(CCC(=O)NCC(C1CCCC1)NC(C1CC(CF)C1)=O)NC(N)=O c1(NC(CCOCCNC(CC(CCC)C)=O)=O)cccc(N=[N+]=[N-])c1 C(=O)(CCC1=CCCCC1)N1CC(CCC)N(C(=O)C(F)CC2CC2)CC1 C(=O)(C(C)(F)CC1CCCC1)N(CCCNC(=O)C=Cc1ccco1)C c1(CCC(N2CC(c3cn(C(C)CO)nn3)(C)C2)=O)ccncc1Br C1(C(C)N(C(C)(C)C)C(C2CC(C#N)C2)=O)CCCN(C(c2ccc(O)nn2)=O)C1 c1(C(=O)NCC2(CNC(c3c(CC)nns3)=O)CCC2)nc(C(C)C)oc1C C1(C(N2CCC(CC(N3CCC(C4CCCO4)CC3)=O)C2)=O)CC(=O)C12CCC2 C1(C(=O)NCC(CC)(C)NC(c2cccnc2O)=O)CCn2c(C)cnc2C1 N#Cc1c[nH]c(C(=O)NCC(O)CNC(=O)CN2CCOCC2)c1 N12CC3CC1CCC3CCCNC(=O)CONC2=O.Cc1nc(C(C)(C)C)cs1 c1(C(N2C3C(NC(c4nnn(C)n4)=O)CC(C3)C2)=O)c[nH]c2cccc(C#N)c12 c1(N2CC(C(=O)NC(C)C(F)(F)F)CC(F)(F)C2)ncnc2cccc(F)c12 C1(N)CN2CCC1CC2.C1(C)CCN(C(N(C)C(C23CCC2C3)=O)=O)CC1 c1(NC(C(C)C)C)cncc(C=CC(=O)OC(C)(C)C)c1 C1(C(=O)NCCCN(C(Cn2c(CCC)nnc2S)=O)CC)CCN(C)C(=O)C1 N1(C(C(CN(C)C)O)=O)CCCCC(N(C(=O)Cc2ccc(F)cc2)C)C1 C=CC1(CC(N2CC(OCCO)C2)=O)CN(C(C2(C(C)=O)CC2)=O)C1 c1(C(N2C(C)(C(N3CC4(C3)CC4(F)F)=O)CC2)=O)cccc2ncsc12 c1(C(=O)NC2(CNC(c3ccc(C)nc3)=O)CCCC2)ccnc(C)c1O Cc1c(C(=O)NCC(C)(C)NC(=O)C(F)Cc2ccccc2)cnn1CC(C)C Cc1ccc(C(=O)NCC2CC2CNC(c2cnn(CCO)c2C)=O)nc1C C(=O)(C(C)(C)CC(F)F)NC1CCCCN(c2c(C(=O)OC)c(Cl)ncn2)C1 c1(C(=O)NC(CCCNC(c2cnc(CCC)s2)=O)C)nnn(C)c1C C1(C(N2CC(C)(CC(=O)N(CCN(C)C)CC)C2)=O)CC(=O)N1c1ccccc1 c1(NC2CC(n3cc(C(N4CCCC4)=O)nn3)C2)cc(O)ncn1 c1(C(N2CC(NC(CC3CC(OC)C3)=O)C(C)(C)C2)=O)ccc2cnccc2c1 c1(N2CC(OC)(CNC(=O)CCn3cc(Cl)cn3)C2)ccccc1[N+](=O)[O-] N1(C(CCS(C)(=O)=O)=O)CC2CN(c3ccnc(CCN4CCOCC4)n3)CC2C1 C(=O)(CC1=NN(C)C(=O)C1)N1C(C)CC(NC(CCC)=O)C1 C(=O)(CCCCCN(C)C(c1c[nH]c2ccncc12)=O)NCc1n(CC)ncc1 C(CC(C(=O)NCCOCCC(C)C)NC(=O)CC(CC)C1CC1)=CC c1(CNC(C(=O)OC)CN(C)C)ccccc1C.C(C)(C)O n1(CC)ccnc1C(N1CCCC1C1(NC(c2csc(C(F)(F)F)n2)=O)CC1)=O c1(CC(N2CC(O)(CNC(C3(C)CCCOC3)=O)C2)=O)coc2ccccc12 C1(C)(CC)CN(CC(=O)NC2CC(O)C2N(C)C(C)Cc2nc(=N)[nH][nH]2)CCO1 Cc1c(C(=O)NC(C)CCS(C)=O)sc2ccccc12 C(=O)(N=c1ccc(C)n[nH]1)C1N(Cc2ccc(C(=O)OCC)[nH]2)CCC1 c1(C(N2CCC(NC(CCCC(C)O)=O)C(C)C2)=O)cc2cccnc2[nH]1 c1(-n2c(C)cc(C(=O)NCCC(C)NC(C(CC)SC)=O)n2)ccc(Cl)c(Cl)c1 c1(N2CCCC(NC(C3CCCC(C)C3)=O)(CO)C2)ncc([N+](=O)[O-])cc1Cl C1(NC(C(C2CC2)OC)=O)C2CC(O)C1N(C(=O)CCc1ccc(F)c(F)c1)C2 CC1=C(C(=O)NCC2CCC(CNC(=O)CC34CCCN3CCC4)CC2)CCC1 n1(CCSC)c(C)cc(C(=O)NC(c2ccccc2)C2CC2)c1C.C12CN(C1)C2C1CC1 CC(C)C(C)(C)C(=O)NC1CCN(C(=O)CCOc2ccc(F)cc2)CC1C c1(C(N(C)Cc2cn(Cc3cccc(Cl)c3)nn2)=O)cc(C#N)ccc1Cl NC(CCS(N)(=O)=O)C(=O)NC1C(c2ccccc2)C1(F)F C1(C(N(C)C(C2CC2)C2CC2)=O)C2CN(CC#CC3CC3)CC12 C(CNC(=O)CCCC#N)(CC(F)(F)F)NC(Cc1cccc(CC)c1)=O c1(C(N2C3CN(Cc4c(OC)ncnc4OC)CC32)=O)cccn2c(O)nnc12 C1(C(=O)NCCOC)CN(C(=O)C(C)CC(C)C)CC1(C)C C(C)(C)(CCNC(C1CCC(C(N)=O)C1)=O)NC(CC1CC(C)C1)=O CC1CC(NC(=O)C=CC2CCOCC2)CN(C(=O)CCN2CCCC2)C1 C(=O)(C(C)(C)CN(C)C)NC(C)CC1CN(C(=O)Cc2ccc(C3CC3)o2)C1 N1(C(C2=C(C)CCC2)=O)CCC(NC(c2nc(C)cc(O)n2)=O)C2(CCC2)C1 Cc1oc(C(C)C)nc1C(=O)NCC(C(N1C(C(=O)OC(C)(C)C)CCC1)=O)O CCC(CC)C(C(=O)NC(C)C(C)NC(c1ncncc1C#N)=O)OC C1(NC(=O)CSC(F)F)CN(C(c2c[nH]nc2-n2ccnn2)=O)CC1F C(=O)(C(C)CC(=O)N(CC(C)N(C)C(c1cccc(C(C)C)c1F)=O)C)OC N1(C(c2cccc(O)c2)=O)CC2CCC(C1)N2C(=O)C(c1ccc(F)cc1F)O n1(CC(N2CC(NC(C3CC(OC)C3)=O)C(OC)C2)=O)cc2ncccc2n1 C(=O)(CCCCCCS(N)(=O)=O)NCC1(F)CC(CNC(C2(C(=O)NC)CC2)=O)C1 C=CCC(CNC(c1cc(Cl)no1)=O)C(=O)NC(C)CCC1CCCC1 N1(C(c2nc(C#C)sc2)=O)CCN(C(=O)Cc2nc(C)sc2C)CC(O)C1 C1(CNC(c2cc(Cl)ccn2)=O)CC(F)CN1C(c1cc(C2CC2)[nH]n1)=O n1(CC(=O)NCC2CCN(C(C3(OC)CCOC3)=O)C2)cnc([N+](=O)[O-])n1 c1(Cc2scc(C(N3CC4CC4C3)C(=O)NC(CC)C)n2)ccc(F)cc1 c1(OCCC)ccc(C(C(=O)NC2CCCC2)N(C(C)CC(C)(C)O)C)cc1 C1(CC)CCCCC1C(=O)N(C)CCNC(C1(Br)CC1)=O N1(C(C=CC)=O)CC(OC)C(C(=O)NCC=CBr)C1 n1(CC(CC)O)cc(C(=O)NCC2C=CCN2C(C2CC(C(F)F)C2)=O)nn1 CC1CCC(C(=O)N(C(=O)CCCn2cc(CNc3nccs3)nn2)C)CC1 N1(C(C2CC3CCC2CC3)=O)CCC2(CCCN2C(C2CCCCC2O)=O)C1 C(C(C)(C(=O)N1CC(C(C(=O)NC2CCC2C(N)=O)OC)C1)OC)OC N1(CC(=O)NCCN(C(=O)C(C2CCCO2)C2CC2)C(C)C)CCCC1=O N1(C(c2c(C)non2)=O)CCC(O)CC1C(=O)NC(c1ccc(O)cc1)C c1(CC(=O)N(CC2CCN(C(C(CC)O)=O)CC2)CC)ccc(Cl)cc1F C(CC(F)F)NC(=O)NC(c1cc[nH]n1)C c1(C(=O)NCCN(C(=O)Cn2cccn2)CC)cc(C)cc(Cl)c1N C1(NC(C2C(C)CCN2C(C2CC(C)N(C)C2)=O)=O)CCCCCC1F C1(NC(Cc2nc(C)[nH]n2)=O)CCN(C(=O)Cc2nc(C(C)C)c(C)s2)CC1C N1(C(C)=O)Cc2ccccc2CC1C(=O)NCC1C=CCN1C(=O)CC(C)(C)O S(=O)(=O)(CCCCCl)N.CC1CN(CCC(C)F)CCS1 c1(CN2C(C(=O)Nc3ncccc3[N+](=O)[O-])CC(F)C2)c[nH]c2ccc(Br)cc12 c1(C(=O)NC2(CNC(CC3C(=O)NCCC3)=O)CC2)ccc2c(c1)C(=O)NC2=O c1(CNC(C2C(C)(CC)C2)=O)ccc(CCNC(c2cc(Cl)n[nH]2)=O)cc1 c1(C(N(C)CC2CCN(C(C(C)n3cncn3)=O)C2)=O)cc(Cl)c(F)cc1Cl CC(C)CC(C)(O)CNC(C1CCCC(N)CC1)=O CC(CC=Cc1ccccc1)C(=O)NC1CCCCN1CCOCCO c1(C2CCCN(C(C34C(C(=O)OC)CC(C3)C4)=O)C2)ccc(F)c(F)c1 C1(CC(=O)NC2CCC(NC(CC(C)CN(C)C)=O)CC2)Cc2ccccc2O1 C1(C)(NC(C2N(C(C3C(C(C)C)CCC3)=O)CC=CC2)=O)CCCC1(C)C c1(COC)ccoc1C(=O)NCCOCCCN(C(=O)C(N1CCNC1=O)C)C C(=O)(C1=CCCCO1)NC(C(C)NC(C1(c2cc(Br)ccn2)CC1)=O)C c1(NC(=O)CC2CCN(C(C3CCCCC3)=O)C2)cc(Cl)ncc1Cl CC(CS(C)(=O)=O)C(=O)NC1CN(C(c2cnc(C(F)(F)F)nc2)=O)C1 c1(C(N)=O)cc(C(=O)NCC2(NC(c3csc(C(N)=O)c3)=O)CCOC2)[nH]n1 C1(C(=O)NC2CCN(C(Cc3c(C)nc(C)s3)=O)C2)CC2C=CC1C21CC1 N1(C(Cc2nc(C)oc2)=O)CCC(NC(=O)C(CO)c2ccccc2)CC1C N1(C(CC(CN(C)C)O)=O)CC2CC(N(C(=O)CNc3ccc(Cl)cc3)C)C1C2 N1(C(CC2ON=C(CC)C2)=O)CC(C)N(C(c2c[nH]nc2C2CC2)=O)C(C)C1 C12(C(N(CCC(N)=O)C)=O)CCC(CN(C(c3cnn(C4CC4)c3)=O)C1)C2 C#Cc1ccc(C(=O)NCCC2COCCN2C(=O)C(C)C2CCC2)c(F)c1 C12(C(N(C)CCNC(c3cc(C(F)(F)F)on3)=O)=O)CC=CC(C1)OC2 C1(C(C)NC(c2cnc(O)s2)=O)CCN(C(=O)Cc2ncc(Cl)s2)CC1 CC1CC(NC(=O)CC2CCCC23CC3)CN1C(C1CCS(=O)(=O)C1)=O C1(C(C)C)CCC(c2ccccc2)CC1.C1(C)(C)C(C)NC(=O)C(=O)N1 C1(NC(C(=O)NC(C)C)=O)CCCN(C(c2cc(C(N)=O)n(C)n2)=O)C1 Cc1cc(C(=O)NC2(C)CC(NC(=O)CC3(C)CCCC3)C2)sc1C c1(CC(N2CC(C)C(NC(=O)C=CBr)C(C)C2)=O)ccc2ccccc2c1 C1(C(N(CC(CNC(c2c(C)c[nH]n2)=O)(C)C)C)=O)CCCC(=O)N1 c1(OC)ccc(C(=O)NC2CN(C(=O)C(C)(C)O)C2)c(OC)n1 C1(C(N2CC=CC(NC(c3cccc(C)c3)=O)C2)=O)CC(C)CCC1C(C)C c1(NC(C(C2CCN(Cc3nccs3)CC2)C)=O)cc(Br)c(O)cc1Br N1(C(C2CC(CC3CC3)C2)=O)CCC2CCCC12C(N1CCCC(F)C1)=O N1(Cc2c[nH]c(=N)o2)CCC(CC(=O)N2CCC2)CC1 CC12CCN(C(=O)CSCc3ccncc3)C1CN(C(C1CCCCC1)=O)C2 N1(C(C(C)SCC)=O)CCC2CCC(C1)N2C(c1cnc(C(C)C)nc1)=O c1(CNC(C2(CNC(c3cnc(SC)s3)=O)CC2)=O)ccccc1C(N)=O n1(CC(=O)NC2CCN(C(c3c(C)ccnc3)=O)C2)[nH]cc2c(=O)ncnc1-2 C1(C(=O)NCC23CN(C(CSCC(C)=O)=O)C(C2)CO3)CC2(CC(C)=NO2)C1 C(=O)(C1CCC(=O)Nc2ccccc21)NC1C(NC(C2(CC#C)CC2)=O)CCC1 c1(Cn2cc(-c3cnc(CC)o3)nn2)cc(F)c(Br)cc1F Cc1ccnc(CNC(C2CCCCN2C(=O)CCN2CCN(C)CC2)=O)n1 C(=O)(C1=CC2CCC(C1)C2)N(CC(CN(C(C1(OCC)CCC1)=O)C)O)C N1(C(c2c(C)nsc2)=O)CC2CCC1C2NC(C1CCCN1c1nccs1)=O c1(C(C(=O)NC(C(=O)OC)C)N(C2CN(C(C)=O)C2)C)cccc(F)c1Br C1(NC(C2CC(CCC(=O)O)C2)=O)C2Cc3cc(Cl)ccc3C12 CC1CN(C(c2cn(C)nn2)=O)CCN(C(C2CCCCO2)=O)C1 CC1(C)COC(CC(=O)NC(C(=O)NCCCN2CCCC2)C2(C)CC2)C1 C(CCCC(=O)NC1CCCC1NC(c1ccns1)=O)N(C)Cc1ccccc1 c1(CC(N2CC(CNC(CCCCC)=O)C3C2C3)=O)cc(Cl)cc2c1OCC2 CC1(CNC(=O)CNc2ncccn2)CCN(C(c2cnc3n2CCS3)=O)CC1 c1(C(=O)NC2CC(CNC(c3cc(C4CC4)[nH]n3)=O)C2)cc2c(s1)CCCC2 CC1CCC(CC(N2CC(O)(C(F)C(=O)N(C)CC3CC3)C2)=O)OC1 c1(OCC)ccc(OC)cc1.c1(C(C(=O)O)NC(=O)OC(C)(C)C)ccc(C)cc1 C1(CNC(c2sccc2CN)=O)CC2CCC(C1)O2.C12C=CC(C1)NC2=O N1(C(=O)CC2CCCCN2C(c2cn3c(n2)CCC3)=O)CC2(CCCCC2)C1 C1(NC(C(CC#C)C)=O)CN(C(=O)CSC)CCC1CO CC1(C)CC(CNC(c2cocn2)=O)N(C(c2ccc(O)c(Cl)c2)=O)C1 C1(CNC(C(CC#C)C)=O)CC2CCC(C1)N2C(c1coc(C2CCC2)n1)=O CC(C)CCC(F)C(=O)N1CCCC(CNC(=O)CC2C=CCC2)C1 C1(C(=O)N(C)CC2(O)CN(C(=O)CC3CC=CC3)C2)(OC)CCCOC1 C1(C)(C(=O)NC2(C3N(C(Cc4c(C)ocn4)=O)CCC3)CC2)CCCNC1=O C(=O)(C(C(C1CC1)OC)N(C1CCCN(C(C)=O)C1)C)NCCCC C1(CCOC)CN(C(C2CC2C)=O)CCN1C(C12COCC(C1)C2)=O N1(C(C(CCC)OC)=O)CCOC(C)(CNC(c2cccc(F)c2OC)=O)C1 C(C)(C(=O)NCC1CC2CCC1N2C(c1cc(Cl)on1)=O)(C(C)C)NC(C)=O C1(CNC(c2cccc(OC)c2N)=O)CN(C(=O)CO)CC(C)(C)O1 C1(NC(C(CC)=CC)=O)CN(C(=O)CSCC)CC12CCOCC2 c1(-c2cn(C(C)C(=O)NCCC3CCCN3C)nn2)nn(C)cc1S(N)(=O)=O C=C(C)C(O)CC(=O)N(C)CCN(C(=O)CCc1ccc(C)o1)C C12(NC(=O)CSc3n[nH]c(O)n3)CCCC1N(C(=O)CCn1ccnc1)CC2 C(=O)(N=c1c(Cl)c[nH]cc1I)C1CN(Cc2c(C)ccc(Br)c2)CC(F)C1 C#CCC(C)(CNC(=O)COC1CN(C(C2(O)CC2)=O)C1)CO.C(C)(=O)NC N1(C(C2C(C)C2)=O)CCCC(NC(c2ccn(C3CCCC3)n2)=O)CC1 Cc1cc(NC(=O)C(N2CC(Cc3ccccc3)CC(C)C2)C)ccc1F C1(NC(C(COCC)C)=O)CN(C(c2c(C)nn(C)c2Cl)=O)CC(C)(C)C1 C12(C(N3C(CNC(C4CCN(C)C4)=O)CCC3)=O)CC(C)(CCO1)C2 C(=O)(C(=O)N=c1cc(C)o[nH]1)NCCCN(C(CC(CCCC)O)=O)C c1(NC(C2C(NC(=O)NCC)C2)=O)cc(Cl)nn2c(C)nnc12.C1(=O)CCCO1 C1(NC(C2N(C)C(=O)CC2)=O)CC2CN(C(=O)CC3CCCNC(=O)C3)CC2C1 c1(C(=O)NC2(CNC(=O)CCc3ncc[nH]3)CCC2)cc2c(s1)CCCNC2=O c1(C(N(C)CC2CCN(C(=O)C(O)CC3CC3)C2)=O)ccc2c(c1)COC2=O Cc1nc(CO)ncc1C(N1CCCC1CCNC(C1(C)CCSCC1)=O)=O C(=O)(C(C)(C)CS(N)(=O)=O)NCC1(OC)CN(C(=O)C(F)F)C1 Cc1ccc2c(=NCCc3ccc(N)cc3)[nH]c(=NCC(C)(C)CCO)[nH]c2c1 CC(C)CC(C(=O)N1CCC(n2cc(Cn3cccc3)nn2)C1)n1ccnc1 c1(C(=O)CC(=O)C(CC2CCCC2)N2CCOCC2)cc(C(F)(F)F)c(O)nn1 O=C(CCc1ccc2c(c1)CCCC2)N1CCCc2ccnn21 N1(C(c2ccnc(OC)n2)=O)C2CCCC1CC(CNC(=O)C(=O)N(C)C)C2 C1(=O)C(CCF)N1.c1(C(=O)NC2CC(OCC)C2)c[nH]cc1CC c1(CNC(CC2CCN(C(c3c(CN)ccs3)=O)C2)=O)ccc(O)cn1 c1(C(=O)NC2C(CNC(CC(CC)(C)C)=O)C2)cc(C)c2c(c1)CCCN2 c1(OC)c(NC(c2csc(Cl)c2Cl)c2nnnn2CC2CCCO2)cccc1Cl c1(N(C)C)ccc(F)c(C(=O)NCC23N(C(=O)CO)CC(C2)C3)c1 C1(C(N(C2CCN(C(c3cccc(F)c3)=O)CC2)CC#C)=O)CCC12CCC2 C1(N(C(C)C(=O)NCC(F)F)CCC)CC2CCC1CC2 N1(C(Cc2cn(C(C)C)nc2O)=O)CCC(C)C(CNC(=O)CSC(C)(C)C)C1 c1(C(=O)NCC(CO)NC(c2cccn(C)c2=O)=O)ccc2c(c1)CC(C)(C)O2 C#Cc1cc(C(=O)NCC(CO)NC(c2cc(CC3CCC3)c[nH]2)=O)cc(Cl)c1 N1(C(CSCC=C)=O)CC2C(NC(c3ccn(-c4ccccc4)n3)=O)C2C1 c1(CC(=O)NCC2(F)CC(NC(C34CCCC3C4)=O)C2)cccc(Cl)c1F.C1CC1 C12(C(=O)OC)COC(C(=O)NCC3(NC(C4CCCC4O)=O)CC3)(C1)C2 c1(NC(=O)NC23CC(COC4C(C)CCCC4)(C2)C3)cccc2oncc12 C1(NC(C2CCOCC2)=O)(CO)CCCN(C(=O)CCc2ncccn2)C1 C=CC(C)(CC)C(=O)NCC(C1CC1)NC(C1(COC)CC1)=O N1(C(C(COC)OC)=O)CC(CNC(c2coc(CC3CC3)n2)=O)CC(C)C1 Cc1cccc(C(=O)NCC2CN(C(=O)C(C)C)CCC2C)c1F CCC(C)(CO)C(=O)N1CC(NC(=O)C(c2ccccc2)F)C1 Cc1c(C(=O)N=c2cc(-c3cccc(F)c3)o[nH]2)ccc([N+](=O)[O-])c1O Cc1ccccc1N(C(C1CCCN(C(=O)Cc2ncccn2)C1)=O)C(C)C C(C1CN(C(C2CCC23CCC3)=O)Cc2ccccc21)NC(=O)Cc1cn[nH]c1 C1(CNC(C(C)NC(=O)C(C)(C)C)=O)CN(C(c2nc(Cl)cs2)=O)CC1(C)C c1(C(=O)NCC23CC2CN(C(c2ncoc2C2CC2)=O)C3)ccnc2[nH]ncc12 c1(C(=O)NCCC(=C)CNC(=O)CCC2CC2)cncc2ncn(C)c12 c1(C(N2CC3C(N(C)C)C3C2)C(=O)NCCCC)cccc(OC(F)(F)F)c1 c1(CCOC)cc(CN2CC(O)C(C3CC3)C2)c2cc(CO)[nH]c2c1 c1(C(=O)NC(C=CC(N2CC(C(=O)NC)OCC2)=O)C)ccc(C)cc1O c1(NC(C(c2scc(C)n2)C)=O)ccn2ncnc2c1 c1(NC(=O)NC2COC(C3CC3)C2)cc(C(F)(F)F)cc(Br)c1 N1(C(C2=CC(C)(C)C2)=O)CCC2(NC(=O)CSC(=N)N)CCCC12 C=CCC(C)C(=O)NC(COC)CC(=O)N(CC(F)F)CCOC NS(=O)(=O)N1CC(C(N2CC3CC3(NC(C3CCC4(CC4)C3)=O)C2)=O)C1 CC(C)CC(CNC(=O)C(c1ccnn1C)O)C(=O)N1CCC(C)(C2CC2)C1 c1(C(N2C(C3(NC(=O)CCn4ccnc4)CC3)CCC2)=O)cccc(CCO)c1 N1(C(c2cnc(C(C)C)s2)C(=O)NCCOC)CC(C)OC(C)C1 N1(C(CC(=O)NC)=O)CCC(NC(=O)C=Cc2ccc(C(N)=O)o2)C(C)C1 c1(CC(=O)NC2CCCN(C(c3cn(CC)nn3)=O)C2)ccc2c(c1)COCC2 C1(NC(C(C)O)=O)CN(S(=O)(=O)C2CC2)CC12CC2 CON(CCC(=O)Nc1cc(C2CC2)cc(C)c1)C(=O)C(C)N=[N+]=[N-] C1(NC(C=CC(C)C)=O)CN(C(c2ccncc2[N+](=O)[O-])=O)CC(F)(F)C1 C1(C(N(CC(CC)(F)F)C)=O)CC(F)(F)CN1C(=O)CC1CCOC1(C)C c1(CC)cc(C(N2CCC(NC(=O)Cc3ccc(Cl)cc3F)C2)=O)cn(C)c1=O c1(CC)occc1C(=O)N(C)CCOCCNC(C1COC(C)C1)=O N1(C2CC3CN(C(c4c(C)cno4)=O)C2C3)CCN2CCCC2C1 c1(NC(Cc2n(C)cnc2)=O)cccc(NC(=O)CSCC(=O)N(C)C)c1 c1(C(=O)NC2C(C)CN(C(c3cc4nc[nH]c4cn3)=O)C2)ccc(C#N)nc1O c1(-c2cn(CCN(c3n(C(C)C)ccc3)C)nn2)cccc2[nH]ncc12 Cc1cc(C(N2CC3CC(C2)C3NC(=O)CC2(O)CCOCC2)=O)nnc1C Cc1csc(C=CC(=O)NC2CN(C(c3c(C)[nH][nH]c3=N)=O)CC2C)n1 c1(C(N2CCC(CNC(C3(CCC)CC3)=O)(CO)C2)=O)cc2cccnn2n1 N1(C(c2cnn(C(C)C)c2Cl)=O)CCC(N(C)C(c2ccc(Cl)s2)=O)C(C)C1 C1(C(C)NC(c2cnc(SC)s2)=O)CCCN(C(=O)CCn2cnnn2)C1 c1(C(C)C(=O)NC2CCCC2NC(=O)C(C)NS(C)(=O)=O)ccc(F)cc1 c1(OC)ccccc1-c1oncc1C(=O)N(CC(O)COc1ccccc1)C(C)C CCC(C)CC(C(=O)NCCC#CCO)NC(=O)COC1(C)CCC1 c1(C(=O)NC(CN(C(COC(CC)C)=O)C)C)cc(Cl)cnn1 c1(C(=O)NCC(C(=O)NC2C(C#C)CCC2)C)ccc(C)c(O)n1 C1(C(=O)NC2CC3(CC3)C2)CCCN(C(c2nc[nH]n2)=O)CC1 c1(C(CNC(C2(C)CC2(F)F)=O)NC(CCCOC(C)C)=O)ccccc1F N1(C(c2c(C)nc(CO)s2)=O)CC2CCN(C(c3cnc(Cl)c(F)c3N)=O)C2C1 Cc1nc2cccc(C(=O)NCC3(C)CCCN(C(=O)C(C)NC(N)=O)C3)c2[nH]1 C(CN=c1ccnc(Cl)[nH]1)C1CCN(C(c2n(C)c(O)nc2)=O)C1 c1(C(=O)NC(C(C)NC(=O)Cc2sc(O)nc2O)C)cc(Br)ccc1F C1(NC(CCC=CC)=O)CN(C(c2nc(Br)sc2C)=O)CC1(C)C C1(C(=O)NC(CC)CN2CCCC2)C(C2CC2)CCN1C(=O)CNC(=O)NC C1(C(=O)NC2(SC)CC2)CC2(CC2)CN1C(C1CCN(c2ccncn2)C1)=O C1(=CC(=O)NCC2C(CNC(CC(CC)OC)=O)C2)CCCCCC1(F)F CC1CCC(NC(c2cc(F)cc(F)c2)=O)CN1Cc1cccc(I)c1 C=CC1(C(=O)NC(COC)CCO)CCN(C(=O)CC23CCCC2C3)CC1 C(C(CC(=O)N1CCC(N(C(=O)C2=CCCOCC2)C)CC1)C(F)(F)F)N(C)C N1(C(c2ccc(N(C)C)cn2)=O)CC2CC(CNC(c3cc(N)ccn3)=O)C2C1 c1(C(=O)NC(C(C)NC(CSCCCC)=O)C(C)C)coc(=O)c2ccccc12 Nc1cc(F)cc(C(=O)NCC2CCCN(C(C3(Br)CC3)=O)C2)c1F C(CC(C)N=c1nc[nH]c2[nH]c(C(C)=O)cc12)NC(CCSCCCC)=O CCC(F)C(=O)NCCCCC1CN(C(=O)Cc2ccsc2C)C1 C1(C(=O)OC)N(C(c2cc(-c3nn[nH]n3)[nH]c2C)=O)CCCC1(C)C C1(CNC(=O)CCc2ccon2)CCCC1NC(C1CCOCC1)=O CCC(C)C(=O)NCC(=O)N(C)CCOCCC(N1CCCC1C(C)C)=O N1(C(C2C(CCC)C2)=O)CC2CC1C2NC(=O)CCc1cn(C)nc1C C(=O)(C1=CCC2CCC1N2C(C1CC2CC(=O)C1C2)=O)N1C(C)(C(F)F)CCC1 C(CCC(C)CC(=O)N1CCN(C(C2C=CCC=C2C)=O)CC12CC2)=C(C)C C(=O)(C1CCc2ccccc21)N(C(C(=O)NCC(COC)C)CC(C)C)C C1(C(=O)NCC(C#C)OC)CN(C)CCN1C(=O)CCN1CCCC1=O N1(c2nccc(NC(c3cnccn3)C)n2)CC(C)OC(C)C1 C1(C2CC2)(CNC(c2c(C)onc2O)=O)CCN(C(c2cncc(N(C)C)c2)=O)C1 Cc1cc(Br)c(C(=O)NCCCC(C)NC(=O)CCCC#N)cc1C c1(C(=O)NCC2N(C(c3n(C)cnc3)=O)CC(O)C2O)cnn2c(=O)cc[nH]c12 C(=O)(C(C)(C)CCC#N)NCC1(O)CCCN(C(CCNS(CC)(=O)=O)=O)C1 C1(NC23CCC(CNC(=O)OC(C)(C)C)(OC2)C3)CC2(CCC2)CCO1 C(=O)(C(C)C(C)NC(C1(C)CC1)=O)N(C(C)CO)CCOC c1(CNC(C2CC(NC(c3ccc(O)cc3)=O)C2)=O)cncc(F)c1 C#CC1(NC(=O)COCCOCC)CCOC1.C(C(=O)OC)NC(=O)CC C=CC(CCC)CC(=O)NCC1C=CCN1C(c1nnn(C)n1)=O c1(C(=O)NCC2CCN(C(c3n(C)nc(Cl)c3)=O)C2)cc(Cl)c(F)cc1Cl C1(NC(c2ccc(OCC)cc2)=O)CN(C(c2c(OC)noc2C)=O)CC1(F)F CC1CCC(C)(C=CC(N2CCN(C(=O)CNC(N)=O)CC2)=O)C1(C)C c1(C(=O)NCc2ccc(N3CCCCCC3)cc2)nc(Br)ccc1Br CC(CC(NC(=O)OC(C)(C)C)NCC1CCC1)C(=O)NCC1(CO)CCCC1 C(=O)(CCCC(=O)NC1COCC1C(N1CC2CC2C2CC12)=O)OC C1(NC(=O)C(=C2CCCCC2)F)CC12CCN(C(c1cc(O)nc(O)n1)=O)C2 C(=O)(CCCn1cncn1)N(C(C)C(=O)NCCN(CC)CC)CCC CC(CC(=O)N(C)CCC1CCCN1C)C(C)(C)NC(C1CC(=O)OC1(C)C)=O c1(C(N2CCC(NC(C(CCC)(C)C)=O)C2CC)=O)ccc2c[nH]nc2c1 c1(C(=O)NC(C2COCCN2C(=O)CC2CN(C)C2)C)cccc(C=C(F)F)c1 C1(C(=O)NCc2c(CC)c[nH]n2)CC(C)CN1C(=O)Cc1ccnn1C C1(CC)CN(C(=O)C(F)(F)C2(OC)CCCC2)CCC1NC(=O)CC(C)(C)CC C(=O)(CC(C)(C(F)(F)F)N(C)C)NC1CCC(NC(C(C=C)(C)C)=O)C1 C1(CCC)(C(=O)NCC(C)(O)CNC(c2sccc2C(=O)OC)=O)CCNC1=O C(CCCC(CO)NC(c1cnn2c1CCC2)=O)NC(C1(CC#C)CCCC1)=O CC1(C(=O)N2CC3CCC2C(CO)C3)CCc2cc(Br)ccc21 c1(NC(C(CCOCC)NC(c2ccc[nH]2)=O)=O)cc(Cl)ccc1C c1(OCC)cnc(C(=O)NCC(C2CC2)NC(c2cc(CC)oc2C)=O)c(Cl)c1 N1(C(CC2CCC=CO2)=O)CCC(C)(NC(c2c(C(=O)OC)cccc2)=O)CC1 C(=O)(C#CC1CCCO1)NCC(C)N(C(C(c1cccc(C)c1)=O)=O)C c1(C2C(C(c3ccc(Cl)cc3)NC3CC(NCCCC)C3)C2)ccc(F)cc1 c1(OCC(=O)N(CC(CNC(C2C(C(=O)OC)CC2)=O)O)C)ccc(Cl)cn1 C(=O)(C1=CCCC(C)(C)C1)N1CCN(C(C(C)N=[N+]=[N-])=O)C(C2CCCC2)C1 Cc1cc(O)nc(CNC(=O)CC2(CNC(C3CCCC(=O)N3C)=O)CC2)n1 CC(C)C(F)C(=O)NCC1CN(C(c2cncc(-n3cc(Br)cn3)c2)=O)CC1C Cn1cc2c(CNC(c3csc(Br)c3Cl)=O)cccc2n1 N1(C(C2OCCN(CC)C2)=O)CCC(CNC(=O)CC(C)(C)C(F)F)C12CCC2 CCC(CC(=O)NCCC(C)(C)NC(c1cc(F)n(C)n1)=O)C1CCC1 CC1CCN(C(c2cnn(-c3nccs3)c2)=O)CC1CNC(c1cc(Cl)no1)=O C1(CNC(=O)C2=CCCS2)CC2CCCC(C1)N2C(=O)CC1CCS(=O)(=O)C1 C(=O)(CC1COc2ccccc21)N1CC(CN(C(CCC(=C)Cl)=O)C)OCC1 c1(C(=O)NCCNC(CC2(C)CC2F)=O)ccccc1NC1CCCCC1 C1(CNC(=O)C(Cl)=CCl)CN(C(=O)CCN2CCOC2=O)CC(C(F)(F)F)O1 N1(C(C(C2CCOCC2)OC)=O)CCCC(CNC(=O)C=CBr)CC1 C(N=c1[nH]c(N2CCCC(n3ccnn3)C2)nc2c1CCC2)C1C=CCC1 C(=O)(C(C)(CC#C)NC(=O)C(CCOC)OCC)NC(C#C)CC1CCCC1 c1(C(=O)NCC2CC(CNC(=O)C3=CCSC3)C2)cc([N+](=O)[O-])c[nH]1 C1(NC(C2(C)CCSCC2)=O)C2CCCC1CC(NC(C1CCC(F)(F)C1)=O)C2 S(=O)(=O)(c1ccc(Br)cc1)C(=O)NC1C(C)N(C(=O)NCCCl)CCC1 C1(NC(Cc2c(C)nccc2)=O)C2Cc3ccc(Br)cc3C12 CC1CCN(C(c2ccoc2)=O)CC1NC(C1(Cc2ccccc2)CC1)=O C1(CNC(c2ncn(C)n2)=O)CC2CCC(C1)N2C(=O)CC1CCC2(CCC2)O1 C1(C(=O)NC2(C3CN(C(=O)CC4CCC4)C3)CC2)C(CN)CCC12CCC2 C(=O)(C(c1cccs1)=Cc1cccs1)NCC1CN(C(C(C)c2ccco2)=O)C1 N=c1[nH]ccc(C(=O)NC2CN(C(c3c[nH]c4cc(Cl)ccc34)=O)C2)c1[N+](=O)[O-] N1(C(C(c2ccncc2)C)=O)CC2CN(C3CCCc4ccc(F)cc43)CC2(C)C1 C1(CNC(C(C2CCOCC2)OC)=O)CCCN1C(C1CC1(C)C)=O N1(C(Cc2ncn(C)c2)=O)CC2CC2(CNC(c2ccnc(C(F)F)c2)=O)C1 CC1(CCC(=O)N2CC(F)C2)CCCN1C(c1cc(=N)[nH][nH]1)=O C(c1ccsc1Br)=CC(=O)NCCNC(C1COCCO1)=O c1(CC(N2CCCC(NC(CN(C)C3CC3)=O)C2)=O)cc(O)nc(O)n1 c1(C(=O)NC(C(C(C)C)NC(Cc2nc(COC)sc2)=O)C)nc(OC)ccc1Cl N1(c2ncc(C(C)C)cn2)CC2CCC(C1)C2NC(c1ccc(Br)s1)=O Cc1c(C#N)nn(C(C)(C)C)c1NC(=O)Nc1cncc(C2CC2)c1 CCC(C)(C)CC(c1nnnn1CC1CCCO1)Nc1ccc(F)cc1 N1(C(C)=O)CCCCC1C(N1CC(C)(N(C(=O)CCc2cccs2)CCO)C1)=O N12CCOC(C1)C(=O)N1CCCC1C2.C(=O)(C(F)=C1CCCC1)N(C1CC1)CC C1(CNC(c2n(CC)cnn2)=O)(NC(c2n[nH]cc2Br)=O)CCCCCC1 C1(C(=O)NCC(C(=O)OC)OC)CC2CC1CN(C(=O)COC(C)C)C2 CC(C)C(C(=O)N(CCC(C(C)C)NC(=O)CN(C)C1CC1)C)C1CCCCC1 C1(NC(C=Cc2ccc(C)o2)=O)CC2CCC(C1)N2C(C1CCCC12CC2)=O CC#CCCCCNC(=O)CC(C)CNC(C1CCNC1=O)=O C1(O)(CNC(Cc2c(C)con2)=O)CC2CCC(C1)N2C(=O)CCP(C)(C)=O CC1OCCCC1C(=O)NC1CC(CCNC(c2nc(C3CC3)cs2)=O)C1 C1(C(=O)NC2C3CN(C(c4c(C)[nH]nc4CO)=O)CC32)CCOCC1(C)C c1(OC)nccc(SC)c1-c1ccc(C(=O)Nc2cc(F)cc(Br)n2)nc1 n1(CC(=O)OCC(C)CNC(=O)OC(C)(C)C)cnc(C(F)(F)F)n1 C#Cc1cccc(C(=O)NC2CN(C(=O)Cc3ccc(Cl)cn3)CCC2F)c1 c1(OC)ccc(Cl)c(C(F)F)c1.c12cccc(c1)NCc1cc(no1)CC(=O)N2 C12(CNC(c3cccs3)=O)CCC1CN(C(c1cccc(-c3cc[nH]n3)c1)=O)C2 C1(CC(=O)NCC2CCC(NC(CNS(NC)(=O)=O)=O)C2)CC2CCC1O2 N1(C(C(CC)SC)=O)CCC(CC)(Nc2nc(C#N)c(Cl)s2)CC1 C1(NC(C2(NC(=O)OC(C)(C)C)CC2(C)C)=O)CCOC(C)(C)OC1 N12CCC(C(F)(F)C1)CN1CC(C1)C2=O.c1(C(=O)O)cccc(F)c1Cl C(=O)(C(O)P(C)(C)=O)NCC(CN(C(C(CC)N(C)C)=O)C)(C)C N1(C(c2cccc(CC)c2)=O)CCN(C)CC1C(N1CCN(C(C)C)C(=O)C1)=O c1(OCC)cc(C(=O)NCC2(CO)CCN(C(C3(C)CC(F)C3)=O)C2)ccn1 Cn1ccnc1CCC(=O)N1CCC1CNC(c1csc(-c2cnc[nH]2)n1)=O c1(C(=O)OCC)[nH]c2ccccc2c1NC(=O)NC1CCC(C)(CN)C1 c1(C(=O)NC(CCCC)CNC(c2cn(CC)nn2)=O)cccc(C2CC2)c1Cl N1(C(C=CCN(CC)CC)=O)CCC(C(=O)Nc2ncsc2C)C1 C(C)(CCC(=O)NCC1CCN1C(c1c(C(F)(F)F)noc1C)=O)OCC N1(C(Cc2nc(C)sc2)=O)CCN(C(C2CC(n3ccnn3)C2)=O)CCC1C N1(C(c2c(C)cc(N)cn2)=O)c2cccn2C(C)CC1C N1(CCNC(C2N(Cc3ncc(OC)nc3)CCC2)=O)Cc2ccccc2C1=O C1(N(C(=O)CCCNS(C)(=O)=O)CC#C)CCCN(C(=O)OC(C)(C)C)C1 C1(CO)CC2CN(C(C3(NC(=O)CC=C(Cl)Cl)CCCCC3)=O)CC12 c1(CCC(=O)NCC#CCNC(CCSCCC)=O)ccc(C)cc1C N1(C(C(CNC(C)=O)(C)C)=O)CCOCC(CNC(=O)C(F)=CC2CC2)C1 C(=O)(N=c1c(Br)c[nH]cc1I)c1c(NC(c2ccc(OC)c(F)c2)=O)c[nH]n1 c1(CC(=O)NC2CCN(C(C3C4CCCCC34)=O)CC2)ccc2c(c1)COC2 C1(C(=O)Nc2c(C)c(CO)ccc2)COC2CN(C(=O)C(C)Br)CC12 C12(CNC(C(C)(C)O)=O)CC1CN(C(C1CCCN(C(=O)N(C)C)C1)=O)C2 c1(C(=O)NCCC2CC(OC)CN2C(=O)C=C(C)C)c[nH]c2ncccc12 CCC1=NOC(CC(N2CC(O)(CN(C(=O)C=C(C3CC3)C3CC3)C)C2)=O)C1 CN1CC=CCC1CC(=O)NCC(O)C(=O)NCc1cnns1 C1(C(=O)NCCC2(COC)CC2)C2CN(C(C3CCC4CC34)=O)CC12 N1(C(C(CNC(C(C(=O)OCC)F)=O)C(C)(C)C)=O)CCc2ccc(F)cc21 c1(OCC(=O)NC(C)C(C)(C)NC(c2cccc(O)n2)=O)ccc(F)nc1 Cc1cncc(F)c1C(=O)NCCCCC(C)NC(C12CCC(C1)C2)=O C(CC(C)(C)CNC(=O)Cc1ccccc1Cl)NC(C1CN(C(C)=O)C1)=O c1(C(N2CC(CNC(c3onc(C)n3)=O)OCCC2)=O)nccc2ccsc12 Cc1ccc(C(CNC(c2ccsc2C)=O)NC(c2c(C)n[nH]c2C)=O)cc1 c1(C(N2CCN(C(C=CC)=O)C(C(C)C)C2)=O)ccc(Cl)c2c1OCCO2 c1(OCCCC)ccc(C(N2CCN(C(=O)C=CC(C)C)CC2)=O)cc1 C12(CCOC1)C(=O)NCCO2.n1(CC(=O)N(CCCOC)C)cncn1.C(C)O C1(NC(c2cnc(C#N)s2)=O)CN(C(c2cnnc(O)c2)=O)CC12CCOCC2 C1(NC(C=CCCC)=O)CC2CN(C(=O)Cc3cc(OC)no3)CC12 N1(C(C(CCC)C)=O)CCCC1(C)c1cn(-c2cccnc2)nn1 C(CN=c1nc(N2CCOCC2)cc[nH]1)C1CC(NCC2OCC(C)C2)C1 Cc1c(C(=O)N(C)CCNC(C2NC(=O)CC2c2ccc(F)cc2)=O)ccn1C C1(CNC(CCC(=C)Cl)=O)CN(C(c2cc(C)sn2)=O)CC(C)(C)C1 C1(C(=O)NC2CCC(C(N3C(C(N)=O)CCC3)=O)CC2)CC2(CC(=O)C2)C1 Cc1[nH]nc(Cl)c1C(=O)N(C)CC1CCCN(C(c2cc(C3CC3)ccn2)=O)C1 C(=O)(C1=C(C)CCCC1(C)C)N1CC2CN(C(C(C(CC)(C)C)=O)=O)CC2C1 C1(CC(=O)NC2(C(N(C)Cc3cnn[nH]3)=O)CCSC2)CCCC2CC12 CC(C)CC(C(=O)N(C)CC1CCN(C(C23CCC(CC2)O3)=O)C1)N(C)C c1(C(N2CC3CC(C)C3C2)C(=O)NCCCSC)cc2cccnc2s1 S(=O)(=O)(c1cc(N(C)CCO)ccc1Cl)N1CCC(CCn2cncn2)CC1 Cc1cc(C(N2CCC2CNC(c2cccnc2F)=O)=O)n(C(F)F)n1 C1(C(N2CC(OCCNC(C(COC)OC)=O)C2)=O)Cc2cccc(F)c2O1 C1(NC(c2noc(C)c2C)=O)C2CCC1N(C(=O)Cc1cccnc1Cl)C2 CC1CN2CCCC2CN1C(C12CC(C)(CN1C(=O)CN1CCOCC1)C2)=O C(=O)(CCC(C)NC(=O)OC(C)(C)C)NC(C1(O)CCC1)C CC(F)(F)CC(=O)NCc1cn(CCN(C(c2occc2Cl)=O)C2CC2)nn1 N1(C(COCCOCC#C)=O)CCC(CNC(=O)C(C)n2cncn2)C12CC2 C1(CNC(c2cscc2C(F)F)=O)CCN(C(=O)C=C(Cl)Cl)CC1 N1(C(Cc2c(C)noc2)=O)CC(C)CN(C(c2n[nH]cc2Cl)=O)CC1C C(CC(C(=O)NCCOc1cccc(CC)c1)NC(=O)C=CCF)OCC C1(CCNC(c2c(C)csc2)=O)CN(C(=O)CCc2nccs2)CCCO1 C1(CCC)CN(C(=O)CC(C)(C)CC)CCN1C(=O)CSc1ccc(C)cc1 c1(OC)cc(NC(c2cnccc2NC(c2cc(I)ccc2Cl)=O)=O)c(Br)cn1 c1(N(CCN(C(C2C(C)(C(C)C)C2)=O)C)C)ccc(C#N)c(C(F)(F)F)n1 CN1C(=O)c2ccc(C(=O)NCC3(NC(C4CC45CC5)=O)CCCC3)cc2C1=O c1(OCC(=O)CCC)ccc(Cl)c(C(=O)N(c2ccc(Cl)cc2)C2CC2)c1N N1(C(c2cccc(C)c2)=O)CC(C)N(C(=O)CC2CCCOC2)CC1C C=CCCC(F)(F)C(=O)NCC12CCC(CC1)N2C(c1ccn(C2CCC2)n1)=O CC1CCN(C(=O)CCSC(F)(F)F)CC1NC(c1ccccc1F)=O c1(CC)conc1CC(=O)NCC1CC(F)(CNC(=O)C(F)=C)C1.C(C)(C)=C C(=O)(C#CC1CCC1)N1C(C(C)NC(c2cccc(NC(C)C)c2)=O)CCCC1 c1(C(N(C2CCN(Cc3c(OC)cccc3)C2)C)=O)cc2nccnc2cc1F N#Cc1ccc(F)c(NC(C2CCN(C(C3C=CCC3)=O)C23CCC3)=O)c1 c1(OCCCn2cc(NC(C3C(CSCC)CC3)=O)nn2)ccn2cnnc2c1 C1(C(=O)NC2(CC(=O)NCC(CCC)OC)CCC2)COCCC1C C1(C)(CC)C=C(C(=O)NC(c2ccccc2)C(N2CCCCC2)=O)C1 N1(C(CCC=CCC=C)=O)CCC(O)(C2(NC(c3ccnnc3C)=O)CC2)CC1 c1(C(N2CC(CC=C)(NC(=O)CC3CCCOC3)C2)=O)cccc(Br)c1 c1(C(N2CC(C(=O)Nc3c(C#N)n[nH]c3)NCC2)=O)ccnc(Cl)c1Cl c1(C(=O)NC2C=CCN(C(c3c(C)cc(F)s3)=O)C2)c2ccccc2nn1C c1(COC)cncc(C(=O)N(C2CN(C(=O)Cn3ccsc3=N)C2)C)c1 n1(CC)cc(C(N2CCC(O)(CNC(C3ON=C(C)C3C)=O)C2)=O)c(C)n1 c1(C(=O)NCC2(O)CC(NC(c3c(C)csc3)=O)C2)cc2c(F)ccc(F)c2s1 Cc1cc2ccc(C(=O)NC3CN(C(=O)C(C)P(C)(C)=O)CC3F)cn2c1 c1(C2(C(=O)NCCCCc3cn(CCOC(C)=O)nn3)CC2)ccc(Cl)cc1F CCCC(C(=O)N(CC(C)C)C)NCCOC.C(=O)CCC(=O)N(C)C Cc1nc(N)cnc1C(N1CCCC(NC(=O)Cc2csnn2)CC1)=O O=C1CC(N=c2ccnc(-c3cccc(Cl)c3)[nH]2)C2CCCN12 c1(OC)ccc(Cl)cc1C(F)(F)C(=O)N(CC(O)CN(C)C(C1C(C)C1C)=O)C C(=O)(CC(C)CNC(C1(O)CCSC1)=O)N(C)Cc1c(C)cco1 C1(NC(c2ncc(Cl)s2)=O)CC12CCN(C(=O)C(O)Cc1ccccc1)CC2 CCC(C)C(O)C(=O)N1CCC(Cn2cc(C(c3ccccc3Cl)(C)C)nn2)C1 Cc1cc2c(C(=O)NCC3CC3NC(c3cc4occc4[nH]3)=O)ccc(C)c2[nH]1 C1(C(N(CC(C)C)CC(C)C)=O)CCCCC1(C)NC(c1ccc(F)cc1F)=O C1(=CCNC(C2CCCOC2)=O)CCN(C(c2ccno2)=O)CC1 Cc1c(Br)ccnc1C(N1CCCCC1C1CCN(C(c2cocn2)=O)C1)=O C12(NC(C(Br)=C(C)C)=O)CCCCC1CN(C(=O)C=CS(C)(=O)=O)C2 c1(SC)cc(C)c(C(=O)N(C)CC2CCCN2C(=O)C=Cc2cnc[nH]2)s1 c1(C(NCCC(n2cc(-c3cnc4n3CCC4)nn2)OC)=O)cc(F)c(C)cc1F C1(N(C(C2C(CCC)C2)=O)C)CCC(N(C(=O)C=COCC)CC)CC1 C(=O)(C(F)(CNC(=O)CP(C)(C)=O)C(C)C)NCC1CCN(CC)CC1 C1(C(N(C)CC2CCN(C(C(C)=C3CC3)=O)CC2)=O)C2CCC3(COC(=O)C13)O2 N1(C(C2N(C(CC)=O)CCCC2)=O)CC2CC(C1)CN(C(C1CCN1CC)=O)C2 c1(OC)cc(OC)nc(C(=O)NC2CC(NC(=O)C(C)(C)CO)CC2O)n1 Cc1ccc2c(c1)SC(C(N1CC3CN(C(=O)CCOC4CC4)CC3(C)C1)=O)C2 C1(C(=O)NC2(C)CCN(C(C(C(C)C)NS(N)(=O)=O)=O)C2)CC(S(C)(=O)=O)C1 C1(CC(=O)NC(c2nccs2)(C)C)CC(F)CN1C(=O)CCC1CC1 CCC(C)(C)C(=O)C(=O)N1CC=CC1(C(=O)NC(C(N)=O)C1CCCC1)COC Cc1cnccc1C(=O)NC1(CNC(=O)CC2C=CCC2)CCCCC1 c1(C(=O)NC2(C(N)=O)CC2)cc(F)cc([N+](=O)[O-])c1.C1(CO)CC(=O)N1 c1(C(=O)NCCCNC(c2ccc(CC)cn2)=O)cc2c(s1)CCC(C)C2 C12(C(=O)NCCCC(C)(C)C)CC(CO1)N(C(=O)CC1COCCO1)C2 C(c1cnc(C)nc1O)=CC(N1CC(CNC(C2C(C(=O)OC)C2)=O)C1)=O C12(CNC(c3c(Cl)cn(C)n3)=O)COCCN1C(=O)CN(C(=O)CC1CC1)C2 C1(CNC(=O)CCc2ccsc2)CCCN1C(c1csc(C(F)(F)F)n1)=O Cc1cccc2c1CN(C(C1(NC(c3ccn(C(F)F)n3)=O)CC(F)C1)=O)C2 C(=O)(C(CO)C(C)(C)C)N1C(CNC(c2cc(C)[nH]c2C)=O)CCC1 C1(CCNC(C(C)SCC)=O)CN(C(c2c(Cl)csc2Cl)=O)CCO1 C1(C2CCN(C(=O)CC3(O)CCCN(C)C3)CC2)(NC(C=CCC)=O)CCC1 c1(C(=O)NC2C(NC(CCCNC(=O)NCC#C)=O)C2)nccc(NC)c1O CC(C)(F)C(C)(F)C(=O)N1CCC(O)(CNC(=O)CCSc2cccc(Cl)c2)C1 C12CN(CCC1)C(=O)CS2.C1(CC)CCCCO1.C(=O)(CN)NC(=O)C1CC1 c1(CNC(=O)OC(C)(C)C)ccc(C(=O)NC2CC(C(=O)OC)C2)nc1C c1(C(=O)OC)cc(C)cc(-c2ccc(C(=O)N(C)C(C)C)cc2F)c1F N1(C(c2c(C)nns2)=O)CCN(C(c2cnsc2)=O)CC1CC(C)(C)C C1(C)(COC)CC(NC(=O)CCC2CC(C)C2)CN1C(=O)Cn1nnnc1C c1(C(N(CC(CC)NC(C2(CO)CCCC2)=O)C)=O)cnn(CC2CCCO2)c1 C1(CN(C(CC(CC)SC)=O)C)CCN(C(=O)OC(C)(C)C)C12COC2 N1(C(C(=Cc2ccccc2)C)=O)CCCC(CC(N2CC(SC(F)F)C2)=O)CC1 c1(CC)cc(N)ccc1C(=O)NC(C)(CNC(=O)CCN1CCN(C)CC1)CO C1(NC(COC(C)C)=O)CCN(C(C2CC(F)(F)CS2)=O)CC1F C(=O)(CCCCN=[N+]=[N-])N1CCCC(C(=O)NC(C#C)(C)C)C1C C(=O)(CC(C)C(F)(F)F)NCCCCN(C(c1c(O)ncc(SCC)c1)=O)C C(CC(=O)N1CCCC(NC(=O)CCSc2nnnn2C)C1)(C(F)(F)F)OC C1(CNC(C2=C(C)CC2)=O)CC(C(=O)NCc2c(C)cccc2C)=NO1 CN1CCCCC(NC(C2CCCN(C)C2)=O)C1=O C1(NC(c2cn(CCC)nn2)=O)CC2CCC(C1)N2C(=O)C(c1cccnc1)O N1(C(Cc2c(C(C)C)con2)=O)C2CCC1CN(C(=O)C=CC1CCCC1)CC2 C(=O)(C1=CCC(C)CC1)N1CCN(C(c2c(CC)onc2C)=O)CC1CC(F)F C(=O)(C1=CS(=O)CCC1)N1CC(CNC(c2cccc(C)c2O)=O)OCC1 C1(c2cn(CC)nc2)OCCCC1CNC(=O)NCCC1OCCC1C C1(O)(CC(=O)NCC2N(C(c3c(CC)c(C)sc3)=O)CC=C2)COC(C)(C)C1 N1(C(Cc2c(C(C)C)con2)=O)CCCC(NC(c2cc(C(F)F)nn2C)=O)C1 c1(CCC(N2C(CCNC(C(C)C)=O)CCCC2)=O)cccc(F)c1Cl c1(C(N2CCN(C(c3n(C)ncc3Cl)=O)C(CF)C2)=O)cccc(O)c1[N+](=O)[O-] c1(C(=O)NC(c2cn(C)nn2)C(=O)N(C)Cc2ccn(CC)n2)cc(C)n(C)c1 n1(COCC)nnc(C(N2CC=CC(NC(=O)C(C)(C)OC)C2)=O)c1N C(CCCC(F)(F)F)n1nnnc1.CCC(C)(C)CCN1CC(c2cncn2C)OC1=O c1(NC(COCC=C)=O)ccc(NC(c2cc(C)n(CC)n2)=O)c(C)c1 C1(N)CC2CC(N)C1C2.C1(CC(=O)C(N)=O)CCN1C(=O)CCC1CCOC1 c1(C(=O)NCC(C)CNC(=O)C(F)n2ccnc2)cnn2c1CCC2 c1(C(N2CCC(CNC(C34COCC3C4)=O)C2)=O)cc2ccc(Br)nc2[nH]1 C1(C(N2CCC(NC(CC(C)C)=O)(CO)C2)=O)CC(F)C(=O)N1C c1(OC)ccc(CN2CCCC(C)(C(N3CCOCC3)=O)C2)c(Cl)n1 C(=O)(CCC(=O)NC1CC(C)N(C(=O)CCCN2C(=O)CCC2=O)C1)OC Cc1cc(C(=O)NC2CC(C)(CNC(=O)C(C3CC(F)(F)C3)O)C2)c(C)[nH]1 c1(OC)ccccc1C(O)CN1CCCC1Cc1c(C)noc1C N1(C(C(=O)Nc2c(OC)cccc2)c2nccs2)CCC(N=[N+]=[N-])CC1 C12(C(=O)NC(C)C=CC(N3CC(N4CCC4)C3)=O)CCN(CC1)C2 C1(NC(CCCCC=C)=O)CN(C(c2coc(CO)c2)=O)C2(CCCCC2)C1 c1(C(c2n(CC=C)nnn2)NC2CC(CCF)C2)ccc(CC)cc1 CC(=O)CC(C)(C)CC(=O)N1CC(CNC(c2cncc(C)c2)=O)CC1C Cn1cc(C(N2CCN(C(c3cnsc3)=O)CC2)=O)nc1-c1ccccn1 c1(CN(C(=O)C(c2ccc(Cl)s2)=O)C(C)=O)cncc2nc[nH]c12 O=C(C1=CCC1)NC(c1ccccc1)C(=O)Nc1cncnc1 C(C)(CNC(=O)C(C)(C)c1cscn1)(CC(C)C)NC(Cc1c(C)cccn1)=O Cc1cc(C(=O)NC(CNC(=O)C=C2CCCCC2)C(C)C(C)C)ncc1C#N C(=O)(C(F)(F)CCn1cccn1)N1CC(CN(C(=O)C(O)C2CC2)C)OCC1 Cc1occc(=O)c1OCC(=O)NCc1ccc(CNC(C2CC2CF)=O)cc1 CC1CN(C(=O)C=Cc2ccn(C)c2)CCN1C(c1cc(C2CC2)no1)=O CC1(C)CC(CO)CN(C(=O)CC2(C)CCN(C(=O)CCOCC(F)F)C2)C1 CC(C)C(C)C(C)CC(=O)N1CCCC(NC(c2cc(CF)on2)=O)CC1 N1(C(c2ccc(CSCCC)o2)=O)CCC(C)(C)C(CO)C1.C1(C(=O)N)CCCS1 c1(C(=O)NC2CCC(NC(C(N3CCSCC3)C)=O)C2)cc2cccnc2s1 N1(C(C2(CCC(=O)OCC)CCOCC2)=O)CCC(NC(=O)C(C)(C)F)C(F)C1 C1(C(N(C)N2c3noc2n3)=O)CCN(C(=O)Cc2ccon2)CC1.C1CC1.NC=O c1(CC)scnc1C(=O)NC(CNC(=O)C(C)(C)c1cnn(C)c1)C(C)C c1(C(C(=O)N(CC(CC)NC(C2CCSC2)=O)C)(C)C)cccc(F)c1 N1(C(C=CC(=O)OCC)=O)CC(O)(CNC(C2OCCC2C(C)C)=O)C1 C1(CC)CN(C(C2(C)COC(C)(C)OC2)=O)CCN1C(C1CC2CCC1CC2)=O C12(C(=O)NCCCC(=O)OCC)CCC1CCCN2 C1(CNC(=O)Cn2nccn2)CCCC2CN(C(=O)CCCCC3CC3)CC12 C1(N(C)C(c2csnn2)=O)CN(C(=O)CCCC2CCCO2)CC1(C)C C(CO)(C(=O)N1CCCC1CN(C(=O)C(=O)NCC(F)F)C)OC C1(C(=O)NC2(CF)CCN(C(C3C(COC)C3)=O)C2)CCS(=O)(=O)C1(C)C CC(C)CC(C)CC(=O)NCC1(F)CCCN(C(c2ccnn2C)=O)C1 c1(C(N2CCC(NC(C3(F)CC3)=O)C2)=O)ccc(-c2ccncc2)s1 C#CC1(C(N2CCC(O)(CNC(=O)C(c3ccn(C)n3)C)C2)=O)CCCC1 Cn1c(C(=O)NC2CCC2CNC(c2cc(C3CC3)ncn2)=O)cc2occc12 N1(CCCNC(C2CC2CNC(C2(CCCC)CC2)=O)=O)CCOC1=O N1(C(C2CCC(C)C2)=O)CCC(C(C)C(=O)NCc2cc(C(C)C)no2)CC1 C(=O)(C1=C(Cl)CCOC1)NC1CC(C)CN(C(c2cccc3cncn23)=O)C1 N1(C(C(C)N(C)Cc2ccccc2)=O)CC2CC(C1)N(C(C1C3COCC13)=O)C2 N1(C(C(C)Oc2ccccc2)=O)CC2C(C1)C2(C)C c1(CC)cccc(NC(C2(CO)CC2(F)F)=O)c1.C1C(C)(CO)NC(=O)CO1 N1(C(C2(COCC)CC2)=O)CCC2CCN(C(C3CCCOCC3)=O)CC12 c1(CCC(=O)OC(C)(C)C)cncc(NC(c2cnc(C3CCCN3)s2)=O)c1 C(=O)(C(F)C(F)(F)F)NC1CCC(CCNC(c2c(CC)nc(C)s2)=O)C1 N1(C(CC(CC)CN(C)C)=O)CC2(CCN(C(=O)CCSc3nccn3C)C2)C1 N1(C(C(=O)NCCNC(C)=O)=O)CCC(CN(C(=O)CNc2ncnn2C)C)C1 C=C1CCC(C(=O)NCC2CCCC(CNC(=O)C=CC3CCC3)C2)CC1 c1(NC(c2n(C)nc(CNC(=O)OC(C)(C)C)c2)=O)ccc(Cl)cc1F C1(NC(c2c(CC)nc[nH]2)=O)CCC(F)(CNC(=O)CCc2cncnc2)C1 CC1C2CC(C2NC(c2ccc(C(C)(C)C)o2)=O)N1C(c1ccc(=N)[nH]c1)=O C1(NC(CC)=O)CCC2CN(C(c3cn(CC)cn3)=O)CCC2C1 CC1(NC(=O)C2=COCC2)CCCN(C(C2(C3CCCCO3)CC2)=O)C1 CC1(NC(=O)CCC2CCC2)CCCCC1C(=O)NCc1nnc(O)o1 Cc1ncn(C)c1C(=O)NCC(C1CCOC1)NC(c1cscn1)=O c1(C(=O)OC)ccc(C(=O)NCC2(F)CN(C(c3cc(C)nn3C)=O)C2)c(C)c1 C1(C(N2CCC(N(CCC(C)C)CCO)CC2)=O)CCC2(CC1)CC2(F)F C1(C(=O)NCC(CO)NC(CCCc2onc(CCC)n2)=O)CCCCN1CC S(=O)(=O)(c1ccc(F)c(Cl)c1)N1C2CN(Cc3nccc(SC)n3)CC21 O=C(CS(=O)(=O)C1CCCC1)NC1CCCC1CNc1ncnc2scnc12 N1(C(c2ccc(C)nc2)=O)CCC2C1CCN2C(=O)CCCc1ccncc1 C1(C(=O)NCCOCCOCCNC(=O)CCn2cccn2)CC2CCC1(O)C2 c1(OC)nccc(=NC2CCN(C(=O)CCN(S(C)(=O)=O)C)CC2CO)[nH]1 C1(C2CC2)(C(N2CCN(c3ccc(Cl)cc3)CC2)=O)CCNC1 c1(C(=O)NCC(COCC)NC(=O)CC2CCOC2)cc(O)nc2c1CCCC2 c1(CC)cccnc1C(N1CC(NC(=O)COCCCC(C)C)C2CC12)=O c1(CC)cc(C(=O)NC2CN(C(=O)CNS(=O)(=O)N(C)C)C2)oc1CC c1(C(=O)NCC2(C)N(C(CC3C=NN(C)C3=O)=O)CCC2)cc2cccnn2n1 C(C)(CCN=c1nc[nH]s1)NC(C=Cc1c(OC)cccc1)=O N1(C(c2n(CC)ccn2)=O)CC2CC(C1)N(C(=O)CCC(F)(F)F)C2 c1(C(=O)NC(CCC)(CC)CCC)cc(S(N)(=O)=O)ccc1Cl N(C(=NCC1CC1)N1CCC(C)(C2CC2)CC1)C(C#C)C C1(NC(C2(c3cc[nH]n3)CC2)=O)CCN(C(=O)CC2CCC2)CC1F CC1Cc2cc(F)ccc2CN1Cc1cc([N+](=O)[O-])ccc1Br C(=O)(C(C)C(=O)OC)NC1C(NC(C2(CC)CCC2)=O)COC1 CC1CC2CN(C(=O)CN3CC4CC4C3)CC2N1C(=O)Cc1cscn1 C1(NC(COCC)=O)CCCC12CCN(C(=O)Cc1ccc(CO)c(C)c1)C2 N1(C(CCC=C)=O)CC2CCC1C(NC(c1sc(-c3cnn(C)c3)nc1C)=O)C2 c1(C(N(CC(=O)NCC(=O)NCCCC2CCCCO2)C)=O)ccc(CO)o1 c1(CC)nnc(C)cc1C(=O)NC(C)(C)C(C)NC(=O)C(C)SC(F)(F)F CCCCCCC(C)(CC)C(=O)NC1CN(C(=O)C=CCN(C)CC)CC1C C(=O)(C(O)CCC(C)C)N1C(C(=O)NC(CSC)(C)CO)CC(F)(F)C1 C(=O)(CCCCCCNC(c1cncc(C)c1)=O)NCc1cc(C)cc(C)c1C N1(C(c2cc(COC)c(F)cc2)C(=O)NCCSC2CC2)CC2CC(C1)N(C)C2 Cc1cc(C(=O)N(C)CCOCCN(C)C(C2CC3(CCC3)C2)=O)cc(C)n1 C1(CNC(CCC=C=C)=O)CCN(C(C2CCCNC2=O)=O)C1(C)C Cc1oc(=O)oc1-c1nc(-c2ccc(N(C)C)cc2)nn1C1CC2CCC1C2 c1(CC)nnc2cc(NCC3CN(C(=O)Cc4ccccc4Cl)CCO3)ncn12 CN1CC(O)CC1CNC(=O)C(=O)Nc1ccc(Oc2ccccc2)cc1 C1(C)(CNC(C2CCN(CC(C)C)C2)=O)CCCN(CC2CCCO2)C1 N1(Cc2ncc(C)c(Br)c2)CC2CC(CN(C(=O)CNS(C)(=O)=O)C2)C1 C1(NC(C(CC2CCC2)NC(C)=O)=O)CN(C(=O)C(C)CC2CC2)CC12CCCC2 C1(NC(CC(=C)C)=O)CN(C(c2cccnc2C)=O)CC1CC c1(C(N2CCC(C)(O)C2)=O)ccc2c(c1)CN(C(c1cc(F)ccc1I)=O)C2 CC1CCC(Cl)=C(C(=O)NCCCN(C)C(C2CCCCC2C2CC2)=O)C1 c1(-c2n[nH]c3c2CN(C(C(CC)C)=O)C3)ccc2ncccc2c1.CC(C(=O)O)=CC=C O=C(N=c1[nH][nH]c2cccnc12)C1CCN1Cc1nc2ccc(Br)cc2s1 N12CC3C(=O)CCC3(C1)CNC2=O.CC(CCNC(=O)OC(C)(C)C)O c1(CC)oc(C)cc1C(=O)NCc1cncc(C(=O)NC2CC3(CCC3)C2)c1 CC(C)C(C(C)C)NC(c1c(CNC(=O)CC2CCOC2=O)nnn1C)=O CCCC(C)CC(=O)N1CC2CCC2(CC(=O)NCC2CC3(CCC3)C2)C1 C(C1=CCN(C(C2CCCN2C2CC2)=O)CC1)NC(=O)CC1CCCC12CC2 C1(C(=O)NCC(C)(C)NC(C=C(CCC)C)=O)CCCN1C(=O)OCC C1(CNC(CCCOC)=O)(CO)CC12CCN(C(=O)CN1CCCC1C)CC2 C(=O)(C(C)C(F)(F)F)NC1C(CNC(c2ccc(OCC(C)C)nc2)=O)C1 CC(C)C(C(=O)N1CC2C(C(=O)NCC(=O)NC3CCCC3)C2C1)C(C)C c1(CN2CC(CC(=O)Nc3c(C)nc(Cl)cc3)C2)ccc(Cl)c(Cl)c1F N1(CC2C(=O)CCC2)CCC(=O)N(Cc2cc(Cl)cc(Br)c2)C1=O C1(CNC(CN(C)C)=O)CN(C(C2(CO)CCCCC2)=O)CC1O n1(C(C)C)cc(C(N2CCC(N(C(C)(C)C)C(=O)Cc3ccno3)C2)=O)cn1 c1(CC(N2CCCCC(N(C(CC(C)OC)=O)C)C2)=O)cn2cc(F)ccc2n1 c1(C(N2CCCCC2CO)=O)cc2nc(-c3ccsc3CSC3CC3)ccc2[nH]1 N1(C(c2ccc(N)cn2)=O)CCN(C(C2CCC(F)(F)C2)=O)CC1CF C(=O)(C(F)C(=O)N(CC(O)CNC(=O)CC1CC2CCC1O2)C)OCC Cc1c(C(=O)NC2(C(=O)NCC3(CC4CCC4)CC3)CCC2)c[nH]c1C#N C1(Nc2cc(OC)nc(SC)n2)CCCCCN(C(=O)CC(C)O)C1 c1(N(C2CCCN(C(Cc3scc(C)c3)=O)C2)C)c(C)c(C)nc2ncnn12 c1(CC)cc(C(=O)NCCC(C)NC(=O)C=CC(C)CC)n[nH]1 CC(C#N)C(=O)N(CCCOCCNC(c1ccc(-c2cccs2)s1)=O)C C1(C2CN(C(c3ccc(F)cc3Br)=O)C2)(NC(Cc2c(C)ocn2)=O)CC1 c1(C(=O)NCC(C2CC2)NC(C(CC#C)(C)C)=O)nc2ccccc2cc1Cl CC1(C)CCOC1C(=O)NC1CCN(C(c2ccccc2C2CCCC2)=O)C1 c1(N(C)C)nc(C2CCCN2CC2C3CCCC23)nc2ccccc12 C(=O)(C(=O)N=S(C)(C)=O)NCC(CNC(CCc1ccc(OCC)cc1)=O)CO C(=O)(CCCC(F)(F)F)NC1(C)CCN(C(=O)Cc2nc(F)c(F)cc2F)C1 c1(C(=O)NCC2C(NC(C(C)(C)CC3CC3)=O)CCC2)cc(N)c(F)cc1F C(C(=O)N1CC2CC2(CNC(=O)COc2cccc(F)c2)C1)(C(C)C)SC Cc1ncc(NC(=O)C(CC(C)C)NC(=O)CN2CCCC2=O)cc1C#N Cc1n[nH]c(C)c1CCC(=O)NCC1(F)CN(C(C2COC(=O)O2)=O)C1 C1(N(CC(=O)NC2CC2(Cl)Cl)C)CCCN(C(=O)CSCc2ccccc2)CC1 CCC(CCC(=O)NCCCN(CCO)C(c1cc(OC)n(C)n1)=O)OC(C)C N1(C(C2CC(OC)C2)=O)CCOC(CNC(C2CC(=O)N(C3CCCC3)C2)=O)C1 C1(NC(CCC)=O)CCN(C(c2ccc(-c3ccco3)[nH]2)=O)CC12CCC2 C(CC(C)(C)CC(=O)N1CC(C)(C)CC1CNC(=O)CCOCC1CC1)OC N1(c2c(C#N)c(Cl)ns2)CC2(CN(C(c3nocc3C(F)(F)F)=O)CCO2)C1 C(c1ccc(C2CC2)cc1)=CC(=O)NC(C(C)C)(C)CNC(=O)C(F)CC1CC1 c1(C(=O)NC(=O)OC(C)(C)C)cc(=NC(=O)C2CC2c2nc[nH]n2)[nH][nH]1 C1(C(N(C2CCN(C(C3CC=CCC3C)=O)CC2)C)=O)CC(=O)N(C)C1 C(=O)(C(C)CC(N)=O)NC(CNC(C(Cc1ccccc1)NC(C)=O)=O)C1CC1 Cc1ncn(C)c(=O)c1C(N1CCC(N(C(=O)C(O)c2cnc[nH]2)C)C1)=O C1(C(N2C3C(CNC(c4cccn4C4CC4)=O)C(C3)C2)=O)CC1C1CCCC1 c1(C(=O)NCC2CCN(C(=O)CN3CCS(=O)CC3)C2)ccc2n[nH]cc2n1 c1(CCNC(CCNC(C(c2ccnn2C)C)=O)=O)ccncn1 C(=O)(CC(C)C(F)F)NCCCC1N(C(CCCn2c(C)ncc2)=O)CCC1 CCCCCC(C)(C)C(=O)N1CCC(CCNC(=O)CN2CCCCS2(=O)=O)C1 N1(CC)CCOCC1C(N1CCCCC1C(=O)NCCC1CCSC1)=O C(=O)(CCC(CF)CF)N(CCC(=O)N(CC#C)C)CC#C C1(C(=O)NCC(C)(C2CCC2)NC(C2CCCS2)=O)CC2C=CC1CC2 CC1(C)C(NC(=O)CC2CCCCC23CC3)CCN1C(=O)CCc1cc(Cl)no1 C(=O)(C(C)(CO)NC(=O)CN1CCNC(=O)C1)N1C(C=C)CC1 N12CCN(CC1)CCCNC(=O)C2.C1(OC(=O)C=CCC2CCC2)CCOC1 N1(C(c2cnc(OC)c(Cl)c2)=O)CC2CCCC1(CNC(=O)C=C(C)C1CC1)C2 Cc1sc(C)c(CNCc2ccnn2CC(F)F)c1Br c1(CC(N2C(CN(C(c3cc(CC)n[nH]3)=O)C3CC3)CCC2)=O)ccccc1O Cc1ccc(S(=O)(=O)NC(COC(F)(F)F)C(=O)OC(CO)C(=O)O)cc1 c1(C(N2CC(CNC(c3nncs3)=O)C2)=O)cnc2c(Br)cccn12 CC1CCC(C(C)(O)CN(C(N2CC(c3ccnc(O)c3)C2)=O)C2CC2)CC1 C(=O)(CCC(O)COCC)Nc1c(CCC)nco1 c1(OC)cc(F)ccc1CNC1CC(NC(=O)Cc2ccccc2C(F)(F)F)C1 C1(C)(CC(=O)N(CCNC(C)=O)C)CCN1C(c1[nH]ccc1C)=O C(=O)(C(F)C(C)(C)O)NCC(CC)NC(=O)C(c1ccc(OC)cc1C)C c1(OC)ccc(C(C)NC(=O)NCC(=O)NC(C)C)cc1F C(CCC(C)C(=O)NC1CCC(CC(=O)NCC2CC(C)(C)C2)C1)OC C(=O)(CC(C)(O)C(F)(F)F)N(CCNC(CCN(C(CC)CC)C)=O)C C=CCC(CNC(=O)Cc1cnn(C2CC2)c1)OCCOC(C)=O.C1(=O)C(C)N1 c1(C(=O)NCC=C2CCN(C(c3cc(C)nnc3)=O)CC2)cn2cccnc2n1 CCC(CC(=O)N(C)CC1CCCN1C(C1CCCN1C(C)C)=O)CC(F)(F)F C1(NC(c2nc(C)c(C)s2)=O)CCN(C(c2cc3[nH]ccc3s2)=O)CC1C CC1(C)CCCN(C(C2CN3CCC2C3)=O)C1C(=O)NCCN1CCC(CO)C1 c1(C(N(CC=C)C)=O)ccc2c(n1)CN(C(C1Cc3ccccc3C1)=O)CC2 C=CCC(C)C(=O)N1CCC(CC(=O)Nc2ccnc(OCC)c2)C1 CCC(C(=O)N(C)CC1CCN(C(=O)CCN(C)CCO)C1)C(F)(F)F C1(C(=O)NC2C3CN(C(C45CCOC4CCOC5)=O)CC23)CC2CCCCN2C1 CN(C)S(=O)(=O)N1CCCC1c1nc(-c2ccc(Br)cc2)nn1C1CCSC1 O=C1Cc2cc(S(=O)(=O)NCC3CC(C(=O)Nc4ccc(Cl)nc4Br)C3)ccc2N1 c1(C(=O)NCCOCC#C)ccc2ncc(-c3cccc(F)c3C)n2c1 C1(N(C(CCNC(C)=O)=O)C)CC2CCC(C1)N2C(=O)CCc1csc(=N)[nH]1 CC1CCCn2cc(C(=O)NC3CC(CNC(C4CCCCS4)=O)C3)nc21 Cn1cccc(C(=O)NC(C)(C)CCC(=O)NCC2(C)CCOC2)c1=O N1(C(C2C(C(C)O)C2)=O)CCOC2(CCN(C(C3CCCC34CC4)=O)CC2)C1 CC1(C)CCN(CC(=O)NCCCCC(=O)N2C(CO)CC2CO)C1 CCCCC1C(=O)N1.c12ccc(c(C)c1)COC2=O.c1(CC)nn[nH]n1 c1(OC)cc(F)c(-c2cn(CC(F)CCNC(C3(C)COCCO3)=O)nn2)c(F)c1 N1(C(c2cnc(OC)c(-c3sccc3C)c2)=O)Cc2ccc(Cl)cc2C(C)C1 C(=O)(C1CCc2scnc21)N1C2CC(NC(=O)CCCC3CCCC3)(C2)C1 Cc1cn(C)nc1C(=O)NCC(C)(C1CC1)NC(=O)C(N1CCCC(C)C1)=O C12(CNC(C(=O)NC3CC4(CC(OC)C4)C3)=O)CCC(C)(CC1)CO2 N1(C(c2c(C)ocn2)=O)CCCC(C2CCN(C(C3CC(=O)N(C)C3)=O)CC2)C1 Cc1ccn2nc(C(=O)NCC3(O)CCC(C)C3)nc2n1 c1(NC(C(CCOC)NC(=O)COCCC(C)C)=O)ccc2[nH]nc(Cl)c2c1 N1(C(C)C)C(=O)COCC1C(=O)NCC1(O)CCN(C(=O)Cn2cnnc2)CC1 C1(C(=O)NCC2CC(C)N(C(C3(C)CCC(=O)N3)=O)C2)CC2CCC1C21CC1 c1(C(=O)NC(CNC(C(C)OC)=O)C(C)C)cccnc1Oc1ccccc1 N#Cc1cnc(NCC2CC(NC(C3CC3F)=O)C2)cn1 c1(CNC(=O)NCC2(C(N)=O)CC(F)(F)C2)ccc(OC2CC2)cc1F C1(NC(C(CC)(C)C)=O)CCN(C(c2cn(-c3cccc(C)c3)nn2)=O)CC1F C1(C(N(CCOC)CCNC(c2cc(Cl)cn2CC)=O)=O)CCC2CC2CC1 C(=O)(C(C)(C)CCF)N(C1CCN(C(=O)CCCOC(C)(C)C)C1)CCC C1(CC)(CNC(=O)CC2(O)COC(C)(C)C2)CCN(C(c2csnc2Cl)=O)CC1 C1(C(=O)OC)CC(C(=O)NC23CCC(CC2)N(C(C2CCO2)=O)C3)C12CCCC2 C(=O)(CCC(=O)NCC1CCC1C(=O)NC1(CCO)CCOC1)NCC Cc1ncc(N)cc1C(=O)NC(C(C)NC(=O)Cc1ccc(F)c(F)c1)C(C)C C1(O)(C(C)NC(=O)Cn2cc(CO)nn2)CCN(C(=O)CC(=O)N(C)C)CC1 CC1(C)CCC(C(N2CCC2CNC(c2cc(-c3cccnc3)on2)=O)=O)C1 N#Cc1cc(F)ccc1-n1cc(CS(=O)(=O)Cc2ccc3c(c2)CNC3)nn1 C1(NC(C=CCC)=O)C(C)(C)CN(C(C23OCCCC2C3(F)F)=O)CC1(C)C c1(N2CCC(CCNC(C3C(c4cc(C)no4)C3)=O)C2)nc2cccc(F)c2o1 C(=O)(C1=CCCC1)NCC1N(C(CC2NC(=O)OC2)=O)CC1 Cc1oc(C(C)C)nc1C(=O)N(C(CNC(c1ccncc1)=O)C1CC1)C c1(CC(C)C)cc(C(=O)NCCC(C)NC(=O)CC2COCC2O)n(C)n1 C1(NC(C(=O)N(C)CC2CCCS(=O)(=O)C2)=O)C2Cc3ccccc3C12 C1(NC(CCC=C)=O)CCOC(C(=O)NCc2cc(C)ncn2)C1 C1(CNC(c2ccc(C)c(CO)c2)=O)COC(C)(C)CN1C(=O)C=CC(C)C c1(CN(C(C(CC2CN(C(C3C(CC)C3)=O)C2)F)=O)CC)ccc(C)nc1 CC1C(C(=O)NCCCCCCN)CCCN1C(c1cc[n+]([O-])cc1)=O C(C1COC(C)(C)O1)=CC(=O)NCC(C)NC(=O)CC1CC(F)C1 c1(C(C)OC)nc(CC(=O)NCc2ccsc2C(=O)NCC2CCCOC2)cs1 c1(C(N2C(CNC(c3c(OC)oc(C)n3)=O)CC2)=O)cc(S(N)(=O)=O)c(C)o1 N1(C(C(CCC)OC)=O)CC2(C1)SCCC2NC(=O)CC1=CCOCC1 C(=O)(C1=NOCC1)NC(C1CCN(C(c2c[nH]nc2-c2ccoc2)=O)CC1)(C)C CC(C)CC(O)C(=O)NC1COCC1NC(c1cnc(Cl)c(N)c1)=O c1(C(=O)NCN(C(=O)C(F)OC(F)(F)F)Cc2ncoc2C2(C)CC2)ncccc1F N1(C(CSCCCC)=O)CCC(C(=O)N(C2CCSC2)C)(C(C)C)C1 C(=O)(CCC(C)(C)F)NCC(CO)NC(Cc1cc(C)on1)=O N1(C(C(C)(C)C2CCOCC2)=O)CCC(C)(CNC(=O)CC2CCOCO2)C1 N1(C(Cc2cc(C(C)=O)sc2)=O)CC(NC(C2CC2F)=O)CC(O)C1 C1(NC(C(C)Cn2cccn2)=O)CCCN(C(=O)COc2ccsn2)C1 c1(C(N2CC(NC(C(CC)F)=O)C(SC)C2)=O)cc2ccc(C)cc2[nH]1 c1(OC)cc(C(N2CCC(C(C)C(=O)NCc3nccnc3SC)C2)=O)cc(Cl)c1 Cc1cc(OCC(N2CC(NC(C3(C)C=CCC3)=O)CCC2C)=O)cc(C)c1Cl C#Cc1ccc(CNC(=O)C(CO)NC(=O)CCc2cc(C)on2)cc1 CCCC(C(=O)NCC1C(C)CCN1C(=O)Cc1cc(C2CC2)no1)S(N)(=O)=O CC(c1cnn(C)c1)=CC(=O)NC12CCC1CN(C(=O)COC1CCCC1)C2 N1(C(CN(C(CONCC)=O)C)=O)CCN(C(c2ccn(CC)c2C)=O)CC1CO.O.C C(=O)(C(C(C)C)c1cccnc1)N1CC(C(C)NC(Cc2nc(CC)sc2)=O)C1 c1(C(=O)OC)cc(NCCC2CCC(NC(c3ccccc3Br)=O)C2)ncn1 C(=O)(C#CC1(C)CC1)N1CCC(NC(c2ncn(C(C)C)c2)=O)C1C Cc1cccc(C(C)(C)CNC(C(COC(C)(C)C)C(=O)O)=O)n1 C(=O)(CCC(=O)NC1CCN(C(=O)CC(C)OC)C1C)NC C12(C(=O)NCCNC(=O)C3CC3)CCC(C(=O)O)(CC1)CC2.c1cc(Br)cnc1O C1(C(N2CCN(C(c3ccsc3)CC)CC2)C(=O)NCC)CC2(CC(OC)C2)C1 CON(CCC(=O)N1CCOCC1C)C(=O)C1CC(=O)C1(C)C c1(C(N(CCCNC(=O)CC(C)c2ccco2)CCC)=O)ncc(F)cc1F Cc1cc(C(c2nnnn2C2COC2)NCc2cc(C)[nH]n2)c(F)c(Br)c1 c1(C(=O)NCC(CN(C(C(CC)C(C)C)=O)C)C)cc(Br)n2ccccc12 CCC(C)(C)C(C)CC(=O)NCC1(CCNC(=O)C(C)CN2CCCCC2)CC1 C1(C(=O)NC(CC(C)NC(c2c(C)c(C3CC3)on2)=O)C)CCC(N=[N+]=[N-])C1 c1(C(N2CCC(NC(Cc3nc(C)oc3)=O)C2)=O)ccc(OC(C)C)cc1Cl c1(OCC)ccc(NCC2CCCCN2S(C)(=O)=O)cc1 c1(C(CC)=O)cc(C(=O)NCC2(NC(=O)CCSC)CCCCC2C)ccc1F N1(C(CC=C=C)=O)CC2ON=C(CNC(c3ccc4oc(C)nc4c3)=O)C2C1 C1(C(=O)NCC(CNC(c2cc(O)cs2)=O)O)OCCC1C(=O)O CCC(C)(O)C(=O)NC(CNC(c1ccsc1OC)=O)CO N1(C(C(C=C)(C)O)=O)CC(CC(=O)NCc2nc(C)sc2C)CC1(C)C CC1(C)CCN(C(=O)CCCC#N)C1C(N1CC(F)(C2CC2)C1)=O c1(OC)cc2c(cc1C(N1CCC(CCNC(=O)C3=NNC(=O)C3)C1)=O)CCC2 C1(NC(C2CC(SC)C2)=O)CN(C(=O)CCc2cnc(C)s2)CCC12CCC2 C1(NC(C2N(C)C(=O)NC2)=O)CCCN(C(C2CCCC(=O)N2)=O)CC1 N1(C(c2ccn(C(C)C)c2)C(=O)NCCOC)CCCC2CCC(C)CC12 N1(C(C2(CC)COC2)=O)CCCC(C(N2CCCCC2CCCO)=O)C1 CCC(C)(C)C(=O)C(=O)N1CC(C(C)C(=O)NOCCOCc2ccccc2)C1 c1(C(=O)NCCN(C(=O)C(F)n2cccn2)C2CCCC2)cc([N+](=O)[O-])ccn1 C1(CNC(C(C)OCCC=C)=O)CN(C)CCN1C(=O)CSc1cccs1.COC CC1(C)CC(NC(C2CCNC2=O)=O)CCN(C(c2nc(Cl)ccc2N)=O)C1 c1(CN2CC3CN(C(CCC(C)C)=O)CC32)ncn2ccccc12 c1(NCCC(C)=CC(=O)NC2CCC2CNC(=O)CN(C)C2CC2)ccccc1 C1(F)(CNC(C2C(C)(C)C2(C)C)=O)CCCN(C(C2CCCCC23CC3)=O)C1 C1(C(=O)NCCOC2CCN(C(=O)C)CC2)(OC)CCC(C)(C)CC1.C(C)(=O)O N1(C(c2c(CC)cno2)=O)CCC2(CCCN(C(=O)C=CC3CCCO3)C2)C1 CC(C)C(C)C(CNC(C1CCCC2CC12)=O)N=c1[nH]c(Cl)ncc1[N+](=O)[O-] C1=CC(=O)NC(C(=O)NCCOCC(F)F)C1.C1(=CC)CCC1OC C1(C(=O)NC(C2CCOCC2)C#C)CCN(C(=O)CC2CCOCC2)O1 C1(CNC(CC)=O)CCN(C(C2CCCCC2(C)C)=O)C12CC2 C(c1ccccc1Cl)=CC(=O)NC1CCN(C(C=CCCC(C)C)=O)C1 N1(C(CCCc2n(C)cnn2)=O)CCCC(N(CCF)C(c2cnsc2)=O)C1 Cc1ccc(C)n1CC(=O)OC(c1cccnc1)C c1(C(N(C(C)CNC(=O)CCc2nncs2)C)=O)ncc(C#N)cc1Cl C(=O)(C1=C(Cl)CCCC1)NC(C(C)(C)NC(c1ccc(C)cc1Cl)=O)C C1(C(C)NC(CC(=O)OCC)=O)CN(C(C2C=C2C)=O)CCO1 c1(OC)cc(C(=O)Nc2cccc(NC(C34CC(C(F)F)(C3)C4)=O)c2)cc(C)c1 C1(C)(NC(C=C2CCC(C)CC2)=O)CCCN(c2nnnn2C)C1 N1(C(CC(COC)NC(C2(C)CCCN2C)=O)=O)CC(C)C(C)C1C C1(CNC(CCCOC)=O)CC(NC(=O)COC2CCCC2)CCO1 n1(CC(N2CC(NC(C(C)=CC)=O)C3C2C3)=O)ncc(C#N)c1N C1(C(=O)Nc2ncc(C)nc2C)CCCC12CCN(Cc1scnc1C)C2 C1(C)(CNC(CCCOCC=C)=O)CC(F)(F)CN1C(=O)CN1CC(=O)NC1=O C12CCN(CC1)C(=O)C(=O)N2.c1(NC(CC(C)F)=O)ccc(OC(F)F)cc1 N1(C(C(C=C)(C)O)=O)CCc2c(c(CNC(=O)C3=NOC(C)(C)C3)nn2C)C1 c1(C(N2CCC(NC(C=CC(N)=O)=O)C23CCC3)=O)ccc2c(c1)NC(=O)NC2 Cc1cc(C)nc(NC(C(C)NC(C2CC3CCCC23)=O)C(C)C)n1 c1(C(N2CC(C)C(CNC(c3cc[nH]n3)=O)CC2)=O)ccc(O)c(F)c1F c1(C(N2CCCC(NC(=O)CCCCCF)CC2)C)ccc(Cl)c(Cl)c1 C1(NC(C(CCC)C)=O)CCN(C(c2c(F)cc(Cl)cc2F)=O)CCC1(F)F Cn1cc(C(=O)NC(C)(C)C(=O)NCC(F)CNC(=O)C(F)=CCCF)cn1 c1(CC(N2CCN(C(CSCC(C)C)=O)CC2)=O)cc(F)cc(F)c1 N1(C(CSC(C)C)=O)CC2ON=C(CNC(c3cc4occc4s3)=O)C2C1 C1(C)(CNC(CN(C2CCC2)C)=O)CN(C(=O)C(O)CC(F)(F)F)C(C)(C)C1 C(CCN=C(NCCc1ccc(C#N)s1)NCCC1(C)CC1(Cl)Cl)SC C(=O)(C1=CCOCC1)NC(CSC)(C)C(=O)NCC(C)(O)C1CC1 Nc1ccnn1CC(=O)NC1(CNC(=O)CC2CCCO2)CCCC1 CN1CC2(CCN(C(c3ccc(C(F)C(F)(F)F)cc3)=O)C2)OCC1=O Cc1nc(C)n(C2CCN(CC(C)(C)[N+](=O)[O-])C2)n1.C(C(C(=O)NCS)N(C)C)N C(=O)(C1=CC2CC=CCC12)N1CCC(CNC(c2c(C)[nH]c(C)c2C)=O)CC1 N1(C(c2c(C)scc2)=O)CCC(CNC(C2(C(F)(F)F)CC2)=O)C(O)C1 N1(c2nn(CC)c(C3CC3)c2)CCC2(CCCC2C(=O)OC)CC1 N1(C(C(COC)OCC)=O)CCC2(CC1)CC2NC(C)=O.C1(=O)CCN1.C(C)(C)(C)NC N1(C(CC2C(C)OCC2)=O)CC2CC2(C(=O)NC2CC(CO)N(C)C2)C1 c1(C(N2CCN(C(C(C(C)N(CC)CC)O)=O)CC2)=O)ccc2c(c1)OCO2 C1(CNC(c2cc(CC)no2)=O)CC(O)CN1C(=O)Cc1c(Cl)cnn1C N1(C(=O)OC)CC2C=CC1C(C(=O)NCC=CCNC(c1ccc(C)s1)=O)C2 c1(NC(c2csc(O)n2)=O)cc(Br)cnc1C1CC1.C12CCCCC1CNC2=O c1(NC(C)=O)ccc(I)c(C(=O)NCCC(O)C(F)(F)F)c1 CCC(C)CC(C(=O)NOCCCF)NC(=O)CCc1cccn1C N1(C(C(CCC)OC)=O)CC2CCC2(CC(=O)Nc2ccc(F)cc2)C1 N1(C(c2[nH]c(=N)sc2C(F)(F)F)=O)CCN(C(=O)CCCCCF)C2COCC12 c1(CC)nc(N2CCC(NC(=O)CCS(N)(=O)=O)C(C)C2)c(F)c(Cl)n1 c1(CNC(c2ccncn2)CF)cc(Cl)sc1Cl c1(OC)ccc(C(=O)NCCC2CN(C(=O)Cc3ccsn3)CC(C)O2)c(Cl)n1 C12(C#CC(=O)O1)CC2.C(C(=O)O)(C(C)C)ONC(CCOC(C)=O)=O C(=O)(CCCCN(C)C)NCc1n(CC)ncc1.C12CN(C1)C(C)C(=O)N2 c1(C2C(C(=O)NC3CC(n4cc(C(C)(C)CO)nn4)C3)CC2)ccc(F)cc1 Cc1cc(C(=O)NCC(C)(CO)NC(c2c(F)cccc2F)=O)cc([N+](=O)[O-])c1 C1(C)(NC(CCOCCOC)=O)CCCC1CNC(C1CCC1C(N)=O)=O N1(C(Cc2cc(C)no2)=O)CCn2nc(C3CCC3)nc2C1.C1CO1 N1(C(C2C(OC(C)(C)C)C2)=O)CC(Cc2n[nH]c3c2COC3(C)C)CCC1(C)C N1(C(C2C(=C)CC2)=O)CCCC(NC(C2(O)COC2)=O)C1C N1(C(Cc2c(C)nc(C(C)(C)C)s2)=O)CC2CC(NC(c3cnc[nH]3)=O)C(C2)C1 CC1CCOC(C(N2CCC(C(C)C(N3CCC(N4CCC4)C3)=O)CC2)=O)C1 c1(C(N(C)CC)=O)ccccc1C(=O)NCC1(NC(C2CC(C)OC2=O)=O)CCC1 c1(C(=O)NCNC)cc(Br)cc(S(N)(=O)=O)c1C c1(C(N2CCC(C)N(C(C3CC3(Cl)Cl)=O)CC2)=O)cc(F)cc2nn(C)cc12 Cc1ncc(N)cc1C(=O)NC(C)CN(C(=O)C(c1c(C)noc1C)C)C CCCCC(C(=O)OCC)NC(c1ccc(C2SCCS2)cc1)=O Cc1cccc(F)c1CC(=O)NC1CCCC1CNC(c1[nH]c(O)nc1C)=O N#Cc1cccc(NC(C2C3CN(C(C4(Br)CC4)=O)CC23)=O)n1 c1(C(N2C(C)C2(C)C)C(=O)NCCN2CCOCC2)ccc(F)cc1Cl N1(C(C(CCOC)NC(=O)C=Cc2ccncn2)=O)CCC2(C=CCO2)CC1 C12CS(=O)(=O)CC1NC(=O)C=CC(=O)N2.c1(C(=O)SC2CC2)ccoc1C1CC1 CC(C)(C)CCC(F)C(=O)NCC(CN=[N+]=[N-])C(=O)N1CC2CCCC2C1 C12(CNC(=O)C=CC3CC3)CC3CC(CC(C3)C1NC(C1(CCF)CC1)=O)C2 C(C(O)C(F)(F)F)NC(C1CCCN1C(=O)CCNc1ccc(Br)s1)=O Cc1nc(-c2cn(CC(=O)NCC3(C)CCCO3)nn2)sc1C Cc1nc(N(C)C)ncc1C(=O)NCCSC(CC1CCOC1=O)CO.C(C)=O c1(C(N(C(CN(C(c2c(C)ncs2)=O)C)C)C)=O)cncc2sccc12 C(=O)(CC(C)CC(C)(C)C)NCC(C)NC(CCc1ccc(OC)cn1)=O C(=O)(C1=CCCCCC1)N1CC(NC(c2ccc(C(F)F)c(Cl)c2)=O)CC(C)C1 c1(C(=O)NC2(CC3CCC3)CC2)csc2c1CCNC2 Cc1ccccc1C1(C)CC1C(=O)NCc1ccc(OC(C)(C)C)cn1 C(C)(C)(CCCNC(c1ccnc(C)n1)=O)NC(Cn1ncc(CC)c1)=O c1(C(=O)NC(CNC(c2cncc(CC)c2)=O)(C)C(C)C)nsc2ccccc12 C1(CC#C)(C(N2CCC(CO)(NC(=O)C(O)C3CC3)C2)=O)CCCCC1 c1(CCC(=O)NC(CN(C)C(C2CC3CCC2C3)=O)(C)C)ccccc1Cl CS(=O)c1ccccc1C(=O)NCCC1(O)CN(C(=O)C=CS(C)=O)C1 c1(C(=O)NCCC2CCC(NC(=O)C=C3CCCC3)C2)c(F)cc(O)cc1F c1(C(=O)NCC2C(C)CCN2C(C2(CF)CC2)=O)ccc(N2CCCC2)c(F)c1 c1(NC2CN(C(N3CCC(F)(C(=O)NC)C3)=O)C2)cc2ccc(F)cc2s1 c1(C(=O)NC(CC#C)C(=O)NC(CCOC)C(C)C)ccc(F)c(C)c1 c1(C(=O)NCC(CC(C)C)CO)n[nH]c2c1CN(C(=O)Cn1cccn1)C2 C(C)(C(C(C)C)NC(=O)C(C#N)=CC1CC1)NC(c1c(C)csc1)=O C(=O)(C1=CCc2ccccc21)NC(CC)CNC(=O)C(c1cccc(C)c1)O N1(C(C)C)CCCC(C(=O)Nc2cc(O)ncn2)C1.C12CCC(CC1)N2C CS(=O)C=CC(=O)NCCCC1CCN(C(C23CC(C#N)(C2)C3)=O)CC1 Cn1cc(S(N)(=O)=O)c(C(=O)NCC23CCC2CN(C(C2(C)C=CCC2)=O)C3)n1 CCS(=O)(=O)CC(=O)N1CCCCC1CN(C(c1cn(C)[nH]c1=N)=O)C1CC1 C1(CN(C)C(c2cc(F)c[nH]2)=O)CCCN1C(C1CN(c2nncs2)C1)=O c1(C(=O)NCC#CCNC(c2ncc[nH]c2=O)=O)[nH]cc2c1CCS2(=O)=O c1(NC(C2C(C)S(=O)(=O)CC2)=O)ccc(F)c2ccccc12 C#Cc1cc(C(=O)NCC2CN(C(c3c(C)csc3Cl)=O)CC2O)cc(F)c1 C(CCCCNC(=O)NCC1(c2ccccc2)CC1)OC N1(CCC)CCCC1C(=O)NCC(C)(C)CC1CN(C(c2ccc(Cl)o2)=O)C1 c1(OCCC(=O)NC2C(CNC(C(C)CC3CC3)=O)C2)ccc(Cl)cc1 C(CC(F)F)(C(=O)NCC1Cc2nccn2C1)N(C(=O)CSC(F)F)C C1(Cc2n(CCCOC)nnn2)(NC(c2ccc(F)nc2F)=O)CCCCC1C c1(C(=O)NC2CCOC2)ccccc1CCCN1CCCOC1.SC c1(COC)csc(C(=O)N(CC(C)O)CCNC(C2CCC(OC)C2)=O)c1 CN1C(=O)C(C)(C)c2cc(C(N3CCCC(O)C3)=O)ccc21 C1(O)(CNC(C(C)(N(C(C(CC)OC)=O)C)C2CC2)=O)CCN(C)C1 c1(C(N2CC(CNC(C=CCCC)=O)C(C)C2)=O)cc(C)sc1S(N)(=O)=O N1(C(c2ccc(C)o2)=O)CCCCC1CC(=O)NCCc1[nH]cnc1C c1(OCC)ncccc1NC(=O)C(C)NC(=O)C(CC1CC1)OC N1(C(Cc2ccc(OC(C)C)cc2)=O)CC(NC(=O)CCF)CC12CCCOC2 c1(C(=O)NC(C(C)NC(=O)CN2CCOCC2)CO)nnc2ccccc2n1 N1(C(CCNC(=O)NC)=O)CC2(C1)CN(C(=O)Cc1ccnc(F)c1F)C2 C1(C(N2C3(CNC(C(C)OCCC(C)C)=O)CC(C2)C3)=O)OCCN(C)C1=O c1(C(N(C2CN(C(=O)CSCC(N)=O)CC2F)C)=O)cc(C2CC2)ccn1 C1(C)(NC(C=CCN(CC)CC)=O)CN(C(c2cnsn2)=O)C1 c1(SC)cn(C)nc1C(=O)NCC(O)CNC(=O)C(C)(O)C1CC1 CCC(C)C(O)C(C)C(=O)N(C(C)Cn1cc(CCN2CCCC2=O)nn1)CC C1(CC(=O)NC2(CC(C)C)CC2)CCCN(C(=O)CCC2CCCN(C)C2)C1 CC1CN(C(=O)CC2CCCSC2)C1C(=O)N(C)CC1(O)CCOC1 c1(C(N(C(CNC(CCC(C)SC)=O)C)C)=O)cccc2ncnn12 C(CCCC#N)(c1nnnn1CC1CCC1)NC(CC)=O.C1(CNC2CC2)CC1 CCC(CC)C(F)C(=O)N1CC(C)N(C(C2SCCS2)=O)CC1C c1(NC(C)=O)cc2ccccc2cc1C(N1CCC(N)C1C)=O Cc1ccc(C(=O)NC(C2CCN(C(=O)CSCc3csc(C)n3)C2)C)nc1F c1(CC)cccc([N+](=O)[O-])c1.c12oncc1C(c1nnnn1C1CCC1)NC2 c1(CNCc2cc(C(=O)OC)c(C#N)cc2)cccc2nc[nH]c12 C1(C(=O)NCC(C(C)C)(C)NC(=O)Cc2csc(=N)[nH]2)CC2(CCC2)CO1 C1(CCC(=O)N(CCCCN(C(C(C)NC(C)=O)=O)C)C)CCC(=O)C1 CC(C(=O)NC1CC(CNC(=O)COC(F)F)C1)C1CCCO1 c1(-n2c(-c3cccn3C(F)F)nc(-c3scc(C)n3)n2)cccc2cnccc12 Cc1csc2ncc(C(=O)NC3(CNC(c4cncn4C)=O)CC3)c(=O)n12 C12(NC(C3(NC(=O)CCN(C)CCO)C(C)C3)=O)CCC(CC1)OC2 n1(CC(=O)NCC(CC=C)NC(=O)CC2CN3CCC2CC3)cc([N+](=O)[O-])cn1 C1(C(=O)NC2CC(F)(CNC(=O)CN3C(=O)CCC3=O)C2)CC2CCC1CC2 CC(C)C(C)C(C)CC(=O)N1CCOCC(NC(=O)CCCCn2ccnn2)C1 Cc1c(C(N2CCCC(O)(CNC(c3cncs3)=O)C2)=O)nn2ccccc12 C(C(CNC(c1ncccc1O)=O)C(F)(F)F)NC(c1c(C(C)C)noc1)=O N1(C(c2nc(C)sc2C)=O)CC(NC(C23CCCCC2C3)=O)C2CCCCC12 C1(CC=C)(NC(c2cncc(Cl)c2Cl)=O)CCN(C(=O)C(F)=C(C)C2CC2)CC1 c1(C(=O)NCC2C(NC(C(C)Cc3ccco3)=O)C2)ccc2nsnc2c1 N1(C(C2CC(NC(C(C)CN(C)C)=O)C2(C)C)=O)CCC(C)(C)C(CO)C1 C(C(=O)N1CCC(C(=O)NCC(=O)NC)O1)C1N(CC)CC1 C1(CC)CCCC1C(=O)N(C)CCN(C(=O)Cn1cc(C(C)O)nn1)C C=CC(CCC)CC(=O)NC1(CC=CC(N(C)CP(C)(C)=O)=O)CCC1 C(C(=O)N(CCCF)CC#N)(C(C)SCC1CC1)N(CCC#N)C.c1ccccc1 c1(N(C)C)ccc(C(=O)NC2CCCC2CNC(C2CC(C)(C)C2)=O)cc1 C(=O)(C1CCc2ccccc21)NC(CCOC)C(=O)NC(C1CCC1)C1CCC1 CN1CCCCC(C(=O)NCc2cnc(-c3ccccc3Cl)nc2)C1=O C(C(C)(C)CC(=O)N(C)CC1(O)CCCN(C(=O)Cn2cnnc2O)C1)N(C)C N1(C(C2(C(=O)OC)CC2)=O)CC2CC(NC(=O)CC3CCCC(C)C3)C2C1 C=C1CC(C(=O)NC(CC(=O)OC)C2CC2)(COC)C1.C(CC(=O)OC)N c1(C(=O)NCC2CCCC(CNC(CCOCCC)=O)C2)cnc(SC)nc1O N1(C(C(=O)NCCOC)=O)CCC(CNC(=O)CC(C)C)(OC)CC1 C#CC1CCCN(CC2C(C(=O)NCc3cc(N4CCCCC4)ccn3)C2)C1 c1(C(=O)NC2C3(CC(NC(CC(C)CF)=O)C3)C2)cccc(C=C(F)F)c1 C(C)(CN=c1[nH]c(C)nc(C)c1C)(C(C)C)NCC(=O)Nc1cccc(C#C)c1 C(=O)(C1CCC2(CC1)CC2N)NC1(C(=O)OCC)C2CCCCC12 C1(C(=O)NC(CO)C2CC2)(OC)CCN(C(=O)CN2CCOC2=O)C1 N1(C(C2CNC(=O)CN2C(c2cnn(C(F)F)c2)=O)=O)CC2C=CCC(C2)C1 c1(OCC)cccc2scc(C(=O)NC3(C)CN(C(=O)CN4CC5CC5C4)C3)c12 c1(NC(c2ccc(CNC(C3(CC)CC3)=O)cc2)C)nc(Br)c(Br)cc1Br C1(NC(c2ccc(Cl)s2)=O)CCN(C(=O)CC(C2CC2)C2CC2)C(C2CC2)C1 C1(C(=O)Nc2cnc(C)c(Cl)c2)(CC)CCN(C(=O)CC2CCC2)CC1 N1(C(CSCc2[nH]c(=N)sc2)=O)CC2CC(C1)N(C(c1ncc(C(F)F)s1)=O)C2 C1(NC(=O)OC(C)(C)C)CCCC1(C)CNC(c1ncncc1Br)=O CS(=O)(=O)CCCCN=C(NCc1cccc(F)c1)NC1CSC1 CCC(C(=O)NC(C)CNC(c1cc(C(F)(F)F)c[nH]1)=O)NC1CCCCC1 N1(C(C2N(C(CCC#C)=O)CC(=C)C2)=O)CCC(C)(C#N)CC1 C1(NC(C2C(C)C2)=O)COC2(CNC(=O)CCC(=O)c3ccccc3N)CC1C2 O=C(CCC(F)(F)Cn1cnc2ccccc12)NCCC1CCCC2CCCN12 C(N=c1[nH]c2c(c(=NCCCCCCO)[nH]1)CCCC2)c1c(C(C)C)noc1 Cc1cc2[nH]c(C(N3CC4CC(NC(C5CC(F)C5)=O)C4C3)=O)cc2s1 CCCCC(O)C(=O)NCC(C)(CC)NC(c1cccc(-n2cc(C)cn2)c1)=O c1(NC(C(C2CCN(C(c3cccc(Cl)c3)=O)CC2)C)=O)ccccc1CO N1(C(C2CC(CCC)C2)=O)CC2CC1CC2CF.C(C(CC)OC)N C(=O)(C(O)C(O)C(C)C)NCCN(c1c(OCC)ccc(C(C)(C)C)c1)C c1(C(=O)OC(C)(C)C)ncccc1C(=O)CN1CC1.S(=O)(=O)(CC1CC1CF)N C12(NC(c3cc(C)nn3C3CCC3)=O)CCC1CN(C(c1cc(Cl)cnn1)=O)C2 CN1CCC2(CCCN(C(=O)C(=O)NC3CN(C)C4(CCC4)C3)C2)C1=O CC1CCC(=CC(=O)NCC2CCCCC2NC(=O)CCCC2CCCO2)CC1 C1(C2CC2)(C(N(CCNC(c2c(C)nc(-c3ccsc3)s2)=O)C2CC2)=O)CC=CC1 CC1CCCN(Cc2cc(C(=O)NCC(C)NC(C3CC4CC4C3)=O)n[nH]2)C1 Cc1nn(CC(F)F)cc1C(N1CC(CNC(C2CCSC2)=O)C(O)C1)=O N1(C(c2nccc(CC)c2)=O)CCC(C)N(C(=O)C(c2cncnc2)C)CC1 CCC(C)(C(=O)N1C2CCC1CN(C(=O)C(F)=C1CCCC1)C2)C(F)F C1(NC(CCOC)=O)CC(F)CN(C(=O)COC)C1.c12ccccc1NC2=O N1(C(CC(=O)Nc2c(OC)ccc(CC)c2)C)CCN2C(=O)N(C(C)C)CC2C1 Cn1nc(C(=O)NC2CC(CNCc3ccncc3)C2)c(C(F)(F)F)c1Cl C1(NC(C(CC)CO)=O)CCC2CCN(C(=O)C(c3ccc(F)cc3)=O)C1C2 N1(CC(c2cc(C)nn2C(F)F)=O)CCN(C)C(c2ncc[nH]2)C1 C1(NC(=O)Cc2cc[nH]c2)CC2CC(NC(C3(CO)CC3(F)F)=O)CC2C1 CCC(C)(C)C(O)C(=O)N1CCC2(CC1)CC2C(=O)NC1CC2CCCC2C1 CC1Cc2cc(S(=O)(=O)NCCCC#N)ccc2O1 Cc1cnc(C(=O)NCC2CC2CNC(C2(CCO)CC2)=O)nc1 C(=O)(CCC(=O)N(C)C)NCC(CCNC(Cc1cn(C(C)C)nc1)=O)O.C1(C)CC1 C1(CNC(c2cccc(CC)n2)=O)CCN(C(c2cccc(=O)n2C)=O)C12CC2 N1(C(C2(OC)CCC(C)C2)=O)C2CCC(C(N3CC(C)CC3(C)C)=O)C1CC2 CC(C)C1=NOC(C(=O)NC(CCN(C)C)C(=O)NC2C(C)OCC2C)C1 C1(NC(C2CN(CCC)C(=O)C2)=O)CN(C(c2cnc(C)[nH]2)=O)CCC12CCC2 S(=O)(=O)(c1c[nH]c(=NCCOC2CC2)cc1C)N1CCC(N(CC)CC)CC1 N1(CC)CCC(C(=O)NCC2COCCN2C(=O)C(N2CCCC2CC)=O)CC1 C1(OCCNC(C2(CCOC)CCC2)=O)CCN(C(=O)CC2CC2(C)C)C1 C1(F)(CC(=O)NC2CON(CC)C2=O)CCN(C(C2(CC)CCCO2)=O)CC1 N1(C(C2C(=C)CC2)=O)CC(C)OC2(CCN(C(C3CC(C)(C)C3)=O)CC2)C1 c1(CC)ccncc1NC(C1(COCC)CC1)=O.C12CC(C)N(C1)C(=O)C2 C1(CNC(C(CCCOC)C)=O)CC2COCC2N1C(=O)C(C(C)C)SC C(=O)(C(C)(F)C(C)(C)F)NC(CC1CCC(C)(C)O1)C(N1CCC2(CCC2)C1)=O c1(C(C)C)ncsc1C(=O)N(C)CCN(C)C(C1(c2cnn(C)c2)CCCO1)=O N#Cc1cc[nH]c(=NC2CC(CNC(=O)C(F)(F)F)C2)c1Br N1(C(C2C=CC(NC(C(C)OCCN(C)C)=O)C2)=O)CC=CC(O)C1 c1(C(=O)NC(CN(C(c2c(CCC)n(C)nc2)=O)CC)C)c[nH]c2cccnc12 N1(C(C(C(C)C)O)=O)CC2(C1)C(NC(c1ccc3scnc3c1)=O)CCS2(=O)=O N1(C(CC(C)(C)O)=O)CC2CCOCC2(NC(C2C=CC=CC=C2)=O)C1 C#CCCCC(C)C(=O)NCCCNC(c1ccc(Br)s1)=O N1(C(CN(C2CCCN2C)C)=O)CCC2(C1)CN(C(=O)C(O)C(F)(F)F)C2 CCC(O)CC(=O)N1CC(=O)CC1C(N1CCC(F)CC1)=O C1(CNC(CCC2C(C)C2)=O)CN(C(=O)CSCC#N)CCC1(F)F N1(C(CCC(=O)N(C(C)C)C)=O)CCOC2(C1)CN(C(c1cnnn1C1CC1)=O)C2 C(=O)(N=c1nc(-c2ccccn2)[nH][nH]1)NC1C(C(=O)OC)C(O)C1 c1(C(=O)NCC2CN(C(C3CCCC(O)C3)=O)CCO2)cnc2cccnn12 C(=O)(C1=C(F)CN(C(=O)C(O)C2CC2)CC1)N(C)CCC1CCCCC1 c1(C(=O)NCC(CO)NC(Cc2c(C(C)C)con2)=O)nn(C)cc1SC C1(NC(c2cncc(COC)c2)=O)CC2CC(C1)N(C(=O)C(C)(C)C1CCC1)C2 N1(C(C#C)C)CCN(C(C2(C)CC2)=O)CC1.C1(C(=O)N)CCC(O)C1 N1(C(c2cncc(CC)c2)=O)CC2CCCC2(C(=O)Nc2cnn(C(F)F)c2)C1 c1(C(N(CCNC(C(C=CC)O)=O)Cc2ccccc2)=O)occ2c1CCOC2 c1(CCC)nc(C(=O)NC23CC(NC(C4CC4c4cnnn4C)=O)(C2)C3)co1 c1(CNC(c2c(OC)ccc(Cl)c2)=O)ccc(S(=O)(=O)NC2CNC2)cc1 C(c1ccccc1)=CCC(=O)NC(C)CN(C)C(c1cc(C2CC2)ns1)=O CC12CCC(C(=O)NC3CCCCC3CC(=O)N(CC3CC3)CC3CC3)(CO1)C2 N1(C(CC=CC=C)=O)CCC(C2CC(NC(C3CCC(=O)N3CC)=O)C2)CC1 CCC(O)C(C)C(=O)NC1CC2(NC(=O)CC3CC(OC)C3)COC1C2 c1(C(N2C(C3(NC(CC4(CSC)CC4)=O)CC3)CCC2)=O)cccn2[nH]c(=N)nc12 Cc1c(C(=O)NCC(C)(C2CC2)NC(=O)Cn2cnc(=N)[nH]2)cnn1C1CC1 CCCCC(C)C(=O)NC1C(F)CN(C(C2(Oc3ccccc3)CC2)=O)CC1C C(CCCC(=O)N1CCCCC1CN(C(=O)C(F)CC1CCOC1)C)SC c1(OCC=C)ccc(CC(=O)NC(C)(C)CN(C(=O)C2=CCSC2)C)cc1 C1(NC(=O)CC2OCCO2)CN(C(C2CCSCC2)=O)CC12CCC2 CC#CCC(C(=O)NCc1cc(COC)no1)NC(=O)C(CC)OCC Cc1cc(N2CCCC(C)(NC(c3cc4n(n3)CCC4)=O)C2)n2ncnc2n1 N1(C(c2ccc(Br)cc2)=O)CCC(CN2CCC(c3ncccn3)CC2)C(O)C1 N1(C(C2(SCC)CC2)=O)CC(NC(c2cc(Br)cnc2O)=O)CC(C)(C)C1 C(=O)(C(CC)n1ccnc1)NCC(CC)NC(c1ccc(C(C)(C)C)[nH]1)=O CC1CC(C(=O)NC2CCCC2CNC(=O)Cc2cnn(C)c2)=NO1 O=CN1CCCC1C(N1CCCC1C1CCN(C(=O)COc2ccccc2)C1)=O CC(C)(C)CC(=O)N1CC(O)(CCNC(C2CC(N3CC(O)C3)C2)=O)C1 CC1(C)CCC(CNC(C2CC2CF)=O)N(C(=O)C(F)(F)C2CC2)C1 c1(C(=O)NC(CCCNC(Cc2onc(CCCCC)n2)=O)C)sc(F)cc1C c1(CN(C(c2c(F)cc(I)cc2F)=O)Cc2ccn(C)n2)ccc(F)c(F)c1O CS(=O)(=O)c1cnn(CC(N)=O)c1.c12ccc([nH]1)C(=O)NC(C)CNC2=O C(=O)(CCCCC(F)(F)F)N1CCN(C(C2CCOC2)=O)CC1CF CC1CC(=O)NC(C(N2C3CCC2CC3)=O)C1.C1(C2CC2)C(=O)N1 C12(C(=O)NC3(Cn4cc(CN5CCCC5)nn4)CC3)COCC1C2(F)F C(=O)(C(C)(C)CCNC(=O)C(C)S(N)(=O)=O)NCCc1ccc(C)nc1 C(=O)(C(c1ccccc1)=CC(C)(C)C)N1CCN(C(C2C(C)C2)=O)CC1CO CC1(C)CCC(CCNC(c2c[nH]nc2CCNC(=O)CC2CC2)=O)O1 CN=c1ccc(C(=O)NC23CC(CNC(=O)Cc4ccsc4C)(C2)C3)c[nH]1 N1(C(Cn2nnc(C)n2)=O)CCCC(F)(CNC(=O)Cc2nc[nH]n2)C1 C(=O)(C(CO)C(C)(C)C)N(CCNC(C(CC)(C)COC)=O)C c1(C(C)=O)ncc(C(=O)NCCN(C)C(c2cnc(-c3ccccn3)s2)=O)s1 O=C1NC(=O)C(CCNC(=O)OCc2cn(CCCO)nn2)N1 N1(CC(O)Cn2cc(Br)cn2)CCCc2cc(Br)c(Cl)cc21 c1(OC)cccc(OC)c1CNC(C1CCC(C)NC1=O)=O C1(C#N)(C(=O)NC(CNC(c2ncc(C)cn2)=O)CO)CC2(CC2)C1 N1(C(Cc2n[nH]c(=NC)s2)=O)CCCN(C(C2(Cl)CC2C(C)=O)=O)CC1C(C)C Cc1c(C(=O)NC2CC(C)N(C(=O)CN(C)C3CC3)C2)[nH]c2c(Cl)cccc12 c1(C(=O)NC2CC(NC(c3ccn[nH]3)=O)C2)cc2ccccc2c(=O)o1 C(C(=O)N(C1CCCCCC1)CCNC(=O)C(F)CC1CCC1)(C(C)C)SCC C1(C(=O)NCC2CC(C)N(C(=O)CN3CCOCC3=O)C2)COCCN1C=O Cc1cc(C(=O)NC(C)CCNC(=O)CN2CCCCC2)c2c(C)n[nH]c2n1 Cc1ncc(F)c(NC(C2CC23CCN(Cc2c(Cl)ccc(Br)c2F)C3)=O)n1 C1(C(=O)NCCC(C)CCNC(=O)C=CBr)SC2C=CC1CC2 Cc1cc(N)n2ncc(C(=O)NCC3CC(NC(=O)Cc4ccc(Cl)s4)C3)c2n1 N1(C(CC(C)OC)=O)CC(CNC(c2cc(C)oc2C)=O)C2CCCCC12 c1(C(=O)NC(C(C(C)C)NC(=O)Cn2cncn2)C)cc([N+](=O)[O-])nn1C C1(C(F)(F)F)(NC(c2cncc(SC)c2)=O)CC2CCC1CC2 C1(NC(c2c(C(C)C)cccc2)=O)Cc2ccccc2C1NC(=O)C(C)C1CC1 N1(C(N2CC3N(C(c4ccccc4)=O)C(C3)C2)=O)CCC2CCCCC2C1 c1(C(N2CC(NC(c3c[nH]nc3-c3ccco3)=O)C2)=O)csc(O)n1 CCC1=C(C(=O)NCC2CCN2C(c2ccc(C3=CCCC3)cc2)=O)CCCO1 c1(C(=O)NC2C3CCN(C(=O)Cc4cccc(O)c4)C23)ncn2c1COCC2 C1(C(=O)NCc2cncc(C(=O)NCC(CC)C)c2)CC2CC1CC2=O CCCC(C(O)C(=O)N1CCCC1(C)CO)NC(=O)COC(=O)CO N1(C(C(CC=C)(C)N(C)C)=O)C2CCCC1CC(n1cc(CCOC)nn1)C2 c1(C(N2C(CCNC(C3CCN(C)C(=O)C3)=O)CCC2)=O)cc(F)c(N)cc1F C(=O)(CCCCCC(C)O)NCCC(C)NC(c1cnc(C2CC2)nc1)=O N1(C(C(C)SC)=O)CCC2(CC1)CN(C(C1CCN(S(C)(=O)=O)C1)=O)C2 c1(C(N2CC(C)C(CNC(=O)C(C)(Cl)Cl)CC2)=O)cnc2ccoc2c1 N1(C(c2ncc(OC)cn2)=O)CCC(NC(C2CCCN2C=O)=O)C12CCC2 C1(CNC(C2CC(=O)NC2)=O)CCN(C(C2CC(CCO)C2)=O)CC1(F)F C1(C(=O)OC)CCCN(C(=O)NC(c2cccc(C)c2)CC)CC1 c1(C(=O)NC2(CCNC(C3(C(=O)NC)CC3)=O)CC2)ccc(CSC)o1 N1(C(C(CO)NC(C(COC)(C)OC)=O)=O)CCC2(CNC(=O)O2)C1 n1(CC(=O)NC2CC3(CCCCCC3)C2)c(=O)sc2ccccc12 N1(C(c2c(CC)nccc2)=O)CC2(C1)OC(=O)Nc1cc(Cl)ccc12 N1(C(C(c2ccccc2)OC(C)=O)=O)CCCC2(C1)CN(C(=O)CC=C(C)C)C2 c1(CC(=O)NCC(CNC(C2C(SC)CCC2)=O)(C)O)cnc(C(F)(F)F)cn1 N1(C(C(C)N(C(CC(CC)SC)=O)C2CC2)=O)CC2OCC(CO)C2C1 C1(CCC(=O)NCCCC(C)NC(c2ccnc(Cl)c2)=O)NC(=O)NC1=O C#Cc1cc(F)c(C(=O)NCCN(C(=O)CC2CCCN(C)C2)C2CC2)c(F)c1 c1(C(N2CC(NC(C3CSC3)=O)C3(C2)CC3)=O)ccc2c(n1)COCC2 c1(NC(C(C)C)C)ccc(S(=O)(=O)NCC(O)C(C)C)cc1F Cc1ccc(C(=O)NC2CN(C(=O)COc3cc(Cl)ccc3Cl)C2)nc1C CCCC(C(O)C(=O)NC(C)CCCO)NC(c1cc(C)n(CC)n1)=O Fc1ccc(CNCc2cc(-c3cccc(Br)c3)no2)cc1N1CCOCC1 N1(Cc2ccc(C)c(O)c2)CC2OCCN(C(=O)Cc3cc(Br)cs3)C2C1 Cc1nc(C(=O)NCCC(C)NC(c2onc3c2CCCC3)=O)c2ccccn12 c1(OCC)cc(CN2CCN(c3ccc(F)nn3)CC2)cc(F)c1OCC Cc1cc(=NCC#Cc2ccccn2)[nH]cc1S(=O)(=O)NC1CC(C2CC2)C1 c1(C(=O)NC(C(=O)NCc2n(CC)ncn2)Cn2cccn2)nc(C)ccc1C C1(NC(CC#N)=O)CN(Cc2cccc(Cl)c2F)CC1C#N O=S(=O)(c1ccc(Br)cc1NCCCCCCF)N1CCOC(CCF)C1 c1(CC)nc(C(=O)NC(C)Cc2ccc(CNC(C3CC=CC3)=O)cc2)c(C)o1 C1(NC(CN(CCC)C(c2ocnc2C2CC2)=O)=O)CCCC1C(C)(C)C Cc1ccc(NC(=O)CC(=O)NCC(C)(C)N(C)C(c2nc(Cl)sc2C)=O)cc1 N1(C(C(CCC)NC(N)=O)=O)CCC2(CC1)CC(NC(c1cnc(C)[nH]1)=O)CO2 N1(C(C2(OC)CCN(C(c3cnc(C)nc3C)=O)C2)=O)CCC(C)OC(C)C1 c1(C(N2CC(C)C(NCc3cc(Br)cc(F)c3F)C2)=O)ccc(Br)c(O)c1Br c1(OC)cnc(OC)c(COCc2cc(OCc3cc(C)nn3C)cc(F)c2)c1 CN1N=C(C(=O)NC2CCC(C)(CNC(=O)CCC=CC(C)C)C2)CCC1=O CCCCC(CCC)NC(C1OCCC1NC(=O)Cc1cnnn1C)=O c1(C(N2CC(NC(C3(C(C)C)CC3)=O)C(O)C2)=O)ccc(S(N)(=O)=O)cc1 c1(NCC(C)CO)ncc(S(=O)(=O)NCCC2C=CCC2)cc1Cl CC(CCC(=O)NCCNC(=O)C(C)(C)CO)c1ccccc1.C1(=O)CCN1 N1(C(c2cnc(O)o2)=O)CCN(C(=O)CCn2ccnn2)C2CS(=O)(=O)CC12 CC12CC(C(N3CCCCC3CNC(=O)CCCC3CCC3)=O)(C1)C1(COC1)O2 c1(CC(=O)NC2(CNC(CCCCC#C)=O)CCOCC2)ncnc2sccc12 c1(C(=O)NCC2CC(NC(c3c(OC)n[nH]c3)=O)C2)cccc(S(C)(=O)=O)c1F N1(C(C(C)NC(=O)OC)=O)CC2CN(C(=O)CSc3ncccn3)CC2C1 N1(C(CC(=O)OCC)=O)CC2CCC(C1)C(NC(=O)C(C1CC1)N(C)C)C2 Cc1cc(C(N2CCCC2CCNC(=O)CSC(F)(F)F)=O)c(F)cc1N C1(NCC)CC(NC(=O)CNC(=O)CC(F)(F)F)C1(C)C c1(C(N2CC(C(C)NC(C3C(CCC)C3)=O)C2)=O)ccc(C)c(Br)c1N N1(C(C2=CCC(C)CC2)=O)CCC2(CCCN2C(c2c[nH]ccc2=O)=O)C1 C(=O)(C1=NOC(C(C)(C)C)C1)N(C1CCN(C(=O)CCn2ccnn2)C1)C C(CCCC(C)NC(c1ccc(CO)cn1)=O)NC(C(C)OCCC(C)C)=O C12(C)CCN(CC1)OC(=O)NCCOC(=O)N2.C(C)(C)(C)NCC CCCCCC(=O)NC1CCC1NC(c1cn(C(C)C)nn1)=O N1(C(Cn2nc(C)c(Br)c2)=O)CCC2(CCCC2NC(=O)C2=CCC2)C1 c1(CC(=O)N(CC(C)N(C(=O)C=C(Cl)Cl)C)C)sc(O)nc1O c1(C(N(C)CC2N(C(C(COC)O)=O)CCCC2)=O)cnc(O)c(C)c1 c1(C(=O)NC(C)CC2CN(C(C3(C)CCN(C)C3=O)=O)C2)cc2cccnn2c1 C1(C(=O)NC2(C#C)CC(=O)C2)CC(C(=O)NC2CC(OCC)C2)=NO1 C(=O)(C1COc2ccccc21)NCCCCCCN(C)C(C1CCCCCC1)=O O=S(=O)(c1c[nH]ccc1=NCc1cc(Br)no1)NC1CC2(C1)C(F)(F)C21CCC1 CCCN(OC)C(=O)C(C1CC1)N(C)C(c1cn2ncccc2n1)=O C=C(C)C1OCCCC1C(=O)NC(c1ccc(Cl)cc1)c1cnccn1 c1(OC)ccc(C(N2CCCC2CCCNC(C2(C)CC2)=O)=O)cc1OC Cc1cc([N+](=O)[O-])c[nH]c1=NCC1CCC(NC(c2ccn3nccc3n2)=O)C1 C1(CC(N2CC=CC(NC(C#CC(C)C)=O)C2)=O)CCOC(C)(C)C1 N1(C(=O)NCC2CC2Cc2ccccc2)CC2CC3CC(C2)CC1C3 CC1CC2CN(c3nccc4[nH]nc(C(=O)O)c34)CCN2C1=O c1(C(C(=O)NC(C2CCCCN2)C(C)(C)C)(C)C)ccc2ccn(CCO)c2c1 C1(CNC(C(C)(F)F)=O)CCCC(NC(c2ccc(NS(C)(=O)=O)nc2)=O)C1 C1(O)(CC(=O)NCC(=O)N(CCCN(C(=O)Cc2ccco2)C)C)CCCNC1 c1(OCCNC(=O)NC2COCC2N2CCCCC2)ccc(Cl)c(Cl)c1 C(=O)(C1CC(C)Cc2c[nH]nc21)NCC(CN(C(=O)CC1CC=CC1)CC)(C)C CCC(CC)CC(F)C(=O)NC(CNC(C1CCC=CCC1)=O)CC N1(C(c2cccc(CC)c2)=O)CCN(Cc2cnc(C)[nH]2)C(C)C1 CC(F)(F)C(C(=O)NC1CC1NC(c1c(Cl)cccc1Cl)=O)c1ccccc1 c1(C(=O)NC23CCCN(C(C4(O)CC4)=O)CC2C3)cc2cnccc2cc1F CC1CCN2CCN(C(C3CC4CCCC4N3)=O)CC2C1 C1(NC(c2c(Cl)cc(C)s2)=O)C(C)CCN(C(c2cc(N)cnc2C)=O)C1C N1(C(C(c2cn(C)nc2)O)=O)CC2(C1)C(NC(C13CC(F)(C1)C3)=O)CCS2(=O)=O C1(CN(C(c2cccc(C)c2)=O)C)CN(C(c2nc(C)nn2C)=O)CC12CC2 C12CC(C1(C)C)C(=O)O2.c1(C(C)(F)F)nc(-c2cnn(C)c2)cs1 C#Cc1ccc(C(N2CCN(C(=O)C(O)CCCC)CC2)=O)c(F)c1Cl CONC(=O)CC(C(C)OC)NC(C1CC2(C1)CC21CC1)=O c1(C(N(CCCS)C2CC2)=O)cnc2sccn12.C(CCC(=O)NCCO)NC(N)=O C1(CNC(c2nc(C(C)=O)sc2)=O)CCCCN(C(C2(C)C=CCCC2)=O)C1 c1(C(=O)NCCC(CNC(CC(=C)C)=O)O)cc(F)cc(Cl)c1N C#CC1(C(=O)N(C2CCOCC2)C2CC2)CCN(C(C2CCC2C)=O)C1 C1(n2cc(-c3cc(C(C)=O)c(C)o3)nn2)CN(C(=O)C=CC(=O)N(C)C)CC1C c1(OC)ccc(F)c(S(=O)(=O)NC(=O)NCC2CCCCN(C)C2)c1F c1(CCC(=O)NCCC(C)NC(c2cc(C)[nH]n2)=O)c(F)cc(Br)cc1F C1(NC(C2C(=C)C2)=O)CC2CCC(C1)N2C(=O)COC1(C)CCCC1 N1(C(C(OCC)CC)=O)CCC(CNC(=O)Cn2cccnc2=O)(OC)C1.C1CS1 Cn1nc2ccccc2c1S(=O)(=O)N1CCN(c2nccc(Br)n2)C2CC12 CCC(O)C(C)C(=O)N1CCC(C)(CNC(c2cc(C3CC3)no2)=O)C1 N1(C(Cc2scc(C)c2)=O)CC2CCC(NC(c3cnc(O)n3C)=O)CC2C1 C1(NC(CC(COC)(C)O)=O)CCC2(CC1)CC2NC(c1cnn[nH]1)=O C1(C(=O)NC(CC(C)C)c2ccccc2)CC(C)CN1C(C1CC1F)=O C(=O)(CCCC(=O)NC1COCCC1NC(c1ccc(F)s1)=O)OCC c1(C(=O)NC2(CC=C)CN(C(C3CC34CCCC4)=O)C2)noc(C)c1[N+](=O)[O-] Nc1ccc(C(N2CC(O)CC2C(N2CCCC2CC2CC2)=O)=O)nc1 c1(NC(=O)C=Cc2cc(Cl)ccc2Cl)nc2cc(F)cc(F)c2s1 Cc1cccc(C(=O)NC2COCC2NC(c2nocc2C)=O)c1 C1(NC(C2C(C)(C)C2)=O)CCN(C(c2cc(C(N)=O)c[nH]2)=O)C1C1CC1 C1(C(=O)NCC(COC)NC(=O)CSc2c(C)n[nH]c2C)Cc2nccnc2C1 C12(CC(=O)NCC3(F)CCCN(C(=O)CC4CC4)C3)CC3CC(C1)CC(O)(C3)C2 c1(C(=O)OC)ccc(OC)cc1.C1(NC(=O)CCS)CCCC1NC(C1CCCO1)=O CCC(C)(C)NC(=O)COCC1CC1.c1(C(N2CCCOCC(=O)N2)=O)ccco1 c1(C(=O)NC2CCN(C(C(C(CC)O)C)=O)C23CCC3)[nH]c2ccccc2c1C n1(CC(=O)NC(C2CCCN(C(C3(OCC)CC3)=O)C2)C)cnc2c1CCCC2 C(=O)(C(C)(O)CC(C)C)N1CC(CCNC(c2ccc(SC)s2)=O)C(C)C1 C(C1CCCN1C(c1ccsn1)=O)=CC(=O)NCCCN1C(C)CCC1 CC(C)C(F)(CNC(=O)CCC1CCCOC1)C(=O)N(CC(N)=O)C c1(C(=O)NCC2CCCCN(C(c3nnn(C)c3N)=O)C2)cn(C)c(=O)nc1O c1(C(=O)OC)ccc(C(N2CCC(CCNC(C3CCC3OC)=O)C2)=O)cc1 C1(CNC(=O)Cc2cc[nH]c2)CC2CCC1N(C(c1ccnc3ncnn13)=O)C2 N1(C(CNC(C2CC(SC)C2)=O)=O)CCC(CC2CCCCC2)CC1 CC1CCN(C(C2C3CC4C(C3)C24)=O)C(C)C1NC(c1sc2cncn2c1C)=O C1(C(N2C(CNC(c3ccn(CCCC)n3)=O)CC2)=O)CCOC2(CCCC2)C1 C(C(CC(C)C)NC(c1cn(C)nc1O)=O)NC(C1C(OCC)CC1)=O C(=O)(C(F)(F)C(F)(F)F)N(C)CC1(NC(c2cc(COC)[nH]n2)=O)CC1 C1(CCOC)CN(C(=O)Cc2ccns2)CCN1C(c1onc(C)c1C)=O n1(CC(=O)N(C(C)CNC(=O)C(C)n2ccnc2)CC)ncn2cccc2c1=O CC(CC(F)(F)F)C(=O)NC(c1ccccc1)C(=O)N1CC(CN=[N+]=[N-])C1 Cc1cc(NC(=O)C=CCN(C)C(C2CCC(C)C2)=O)cc(C)c1C CC12CN(C(c3cc[n+]([O-])cc3)=O)CC1CN(C(C1CCCO1)=O)C2 CC(C)(C)CCCCC(=O)NC1CCC(NC(c2cnc3n2CCS3)=O)CC1 c1(N(CC(=C)Br)C)nc(N(C)Cc2ccc(F)cc2)nc2c1COC2 C1(CNC(C=C(CC)CC)=O)CC2(CO1)CN(c1ncc3ccnc-3[nH]1)C2 S(=O)(=O)(c1ccc(NCc2nn(C)cc2C)c(Br)c1)NCC1(C=C)CCC1 C(=O)(CC(C)(C)CC(F)F)N1CCCC(NC(c2cnc(OC)c(Cl)c2)=O)C1 N1(C(C(CCSC)NC(c2cccc(OC)n2)=O)=O)CC2(CCNC2=O)C1 Cc1nn(C)cc1C(=O)NCCCN(C)C(c1csc(C#N)c1)=O c1(C(=O)NCC(CNC(CCc2ccc(C)o2)=O)C)cnn2cccc2c1 Cc1nccc(C(N2CC(CNC(c3c(C)cnn3C)=O)C3CC23)=O)n1 C1(N(C)CC2(C)CCC2)CCN(C(=O)C(=O)NCC(F)Br)CC1 C(CC(C)(C)C)(C(=O)NC1CC2CC2C1)NC(c1nn(CC)c(C)c1)=O C(=O)(CCC(F)(F)F)N1CCC(CN(C(=O)C(c2ccccc2)=O)C)CC1 N1(C(c2c(CNC(C3CCN(C)C3)=O)nccc2)=O)CCC2CCC(C1)N2C c1(C(=O)NC2C(CNC(c3c(N(C)C)nccc3)=O)CCC2)cccc(F)c1Cl c1(NC(C(CCC)C)c2nnnn2C)ccc(N(C)C)c(F)c1 c1(N2CCCC(COC)C2)nc2cccnc2c(=NCCCc2n[nH]c(=N)s2)[nH]1 CCCC(CCC)CC(=O)N1C2CCC1C1CC1(NC(c1sccc1Cl)=O)C2 CC1Cc2cc(CC(N3CCCCC3CCNC(=O)C=CC3CC3)=O)ccc2O1 C1(C(=O)NCCC2CN(C(C(C(CC)O)(F)F)=O)C2)CCc2ncccc2C1 c1(C(N(CC)CC2CCCN(C(=O)CC3CC3C)C2)=O)cc(F)c(Cl)cc1F CC(C)C(C)C(C)CC(=O)N(C(C)CNC(c1c[nH]c2ncccc12)=O)C c1(C(C)C)noc(CNC(=O)CC2CCCN2C(=O)CCCNC(N)=O)n1 c1(C(=O)NCCNC(c2cc(C(N)=O)[nH]n2)=O)ccccc1OC(F)(F)F C(=O)(C1=C(C)OCC1)NCC(C1N(C(CCC(C)=O)=O)CCC1)(C)C C1(CC#C)(NC(c2ccc(C#N)cc2)=O)CCN(C(=O)CSCCOC)CC1 C(CCCCCF)NC(C1(CCNC(Cc2ccc(C)s2)=O)CCC1)=O C1(N(CCNC(C2CC2F)=O)C(C2CC=CCC2)=O)CCCCCC1 CC1CCNCCC1N(C(=O)CCN(C)C)CCO N1(C(CC2N(C(c3c(C)[nH]cc3)=O)CC(O)C2)=O)CCCC(C)(C#N)C1 S(=O)(=O)(c1ccc([N+](=O)[O-])cc1F)N1CC(C(=O)O)C2(C1)CC2 c1(C(=O)NCC2N(C(c3scc(C)c3Cl)=O)CCCC2C)cccc2sncc12 C(=O)(C(C(C)CCCC)N1CCN(Cc2ccc(F)cc2)CC1)NCCCC N1(CCOC(C2(c3ccccn3)CC2)=O)CCC(n2cccn2)CC1 c1(NC(C2(C)CCCN2Cc2ccc(F)cc2F)=O)cnc(Cl)c(Br)c1 C(=O)(C1=NNC(=O)CC1)N1CCCC(NC(C2(CC#C)CCCCC2)=O)C1 Cc1cc(CNC(=O)CC2CCN2C(c2cn(CCO)nn2)=O)cc(C)c1 C1(NC(c2n(C)c(=O)ccc2)=O)CC2CCC(C1)N2C(C1(C)CS(=O)(=O)C1)=O C(CC(=O)N1CCC(NC(=O)CC=C(C)C)C1CC1CC1)(C(C)C)OCC C1(C(=O)NC2(CC=C)CCN(C(C3CCC4(CCC4)O3)=O)C2)CCCS(=O)(=O)C1 C1(CNC(C=CC(C)(C)NC(CC(CC)C)=O)=O)CCCN(C)C1=O c1(NC(C2CC(O)CCN2C(=O)Cc2cc[nH]n2)=O)c(Br)cc(F)c(F)c1F CC1=NOC(C(N2CC(NC(c3c(-c4cccs4)noc3C)=O)C2)=O)C1C c1(C(N2CCN(C(C(C)(C)N3CCCC3)=O)CC2)=O)cc(F)cc(S(N)(=O)=O)c1 CCC(C)CC(C(=O)N1CC2CC2C1)NC(c1cc(C)[nH]c1C)=O CCC(C)CCC(=O)N1CC(=O)CC1C(=O)Nc1ccccc1CCO c1(N(C(c2cn(C(c3cccc(C)c3)C)nn2)C)C)ccnc(C)c1O C1(CNC(C(C)OCC#C)=O)CC2CCC(C1)N2c1ccc(CCC(C)C)nn1 C1(O)(CNC(CC2CC(CC)C2)=O)CCN(C(=O)CC2CCSC2)CC1 N1(C(C2C(C)C2)=O)CC2CC1C2NC(=O)Cc1ccccc1C(F)(F)F N1(C(CCC2CCC(C)O2)=O)CC2CC1(CNC(=O)COC(F)(F)F)C2 C1(CCC=C)(C(=O)Nc2c[nH]nc2OC)CN(C(=O)C(N2CCOCC2)C)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])N(C1(C)C(C)OCC1)C(C1CCN(C(N)=O)CC1)=O C12(NC(Cn3c(=N)nc[nH]3)=O)CCC1CN(C(c1sccc1Cl)=O)C2 c1(NC(=O)C(=O)NC2CC3CNC2C3)cc(Br)ccc1[N+](=O)[O-] C(CN=C(NCc1c(O)cccc1F)NCC1CCCO1)OCC=C C1(C(C)(C)C)CCCCC1OC(=O)COC(=O)C(=O)NC1(CO)CCC1.C(C(F)F)N.CC C1(C(N2CCCC(N(C(=O)CNC=O)C)C2)=O)CN(C)C(=O)CCO1 CC1=NN(C)C(=O)C1CC(=O)NC1CCCC(NC(=O)CN2CC(F)(F)C2)C1 CCC(C)C(C)C(=O)NCC1(C)CCCN1C(c1cc(C)cs1)=O C1(CN(C(C=CCN(C)CC)=O)C)C2CN(C(=O)C(c3ccc(C)cc3)C)CC12 N1(C(CCOCCCNC(c2c(NC)nccc2)=O)=O)CCCC2CC1C2(C)C C=CCC(F)(F)C(C)(C)C(=O)N1CC(CCN=c2[nH]ccc(C)c2Br)C1 N1(C(COC(C2CN(C)C2)=O)=O)CC1(C)C(=O)Nc1ccsc1 C(=O)(C(C(C)O)NC(N)=O)NCC(C)C(=O)NCCOCCNC(C)=O c1(C(=O)NC(C)CC(C)NC(C2CC(C3CC3)=NO2)=O)nc2ccccn2c1F c1(C(=O)NC2CCN(C(C3CC4(CC4)C3)=O)CC2)ccc2nn[nH]c2n1 N1(C(COCCOC(C)=O)=O)CCC2C(N(C)C(c3cc(C4CC4)on3)=O)C12 C1(CNC(CCC#C)=O)CC2CCCC2N1C(C1CC1c1ccncc1)=O c1(C(=O)NCC2CCN(C(C(C)O)=O)C2)cc2nn[nH]c2cc1F C(C)(C)(CC(=O)NCCC1CC2CCC1C2)NC(c1c(CC)c[nH]c1)=O C#CC(CNC(=O)C(C)N(C)C(c1ncc[nH]1)=O)CC c1(CC)ccc(O)c(C(=O)NC2CC2CNC(c2ccc(C(C)C)nc2O)=O)c1 C(=O)(C(C)(C)CN1C(=O)CCC1=O)N(CCCCN(C)C(C1CC(C)(C)O1)=O)C n1(CC)nnc(Br)c1CNC(=O)CCn1cc(CCN(C)C)nn1 c1(COCC(=O)NC2CC(NC(C(c3cnn(C)c3)OC)=O)C2)nnc(S)n1C N1(C(CSC(=N)N)=O)CCn2c(C(=O)NCc3ccc(F)cc3)cnc2C1 C1(CC(=O)NC(CC(C)C)CNC(C2C3COCC23)=O)CC2(CCO1)CC2 c1(SC)cn(C)nc1C(=O)NCC12CC1CN(C(c1cnoc1C)=O)C2 CCCCC(O)CC(=O)N1CCN(C(c2ccnc(O)c2)=O)CC1CCO N1(C(C2C(C)(C)C2NC(=O)CC2(O)CCOC2)=O)CCN2CCC1CC2 CC(CCO)(c1cccs1)NCCC(=O)N1CCCC1 C1(NC(c2c(CC)[nH]cc2)=O)CC(C(=O)NCC(C)(C)C)C1(C)C Cc1nc(C(=O)NCC(CO)(CO)N(C(=O)C(F)CC=C(Cl)Cl)C)c(C)n1C C(CCCCCNC(=O)OC(C)(C)C)N(C(=O)C(=O)NN1CCCCC1=O)C C1(CC(=O)N(C2CC(N)C2)C)CC(OC(F)F)C1 CCC(CC(=O)N1CC(N(C)C(c2cncc(CO)c2)=O)C1)CC(F)(F)F C(CCCCN(C)C(C1CCN1C)=O)NC(C(C)SC)=O C=CC(C)(CCOC)C(=O)NCc1cc(C(N2CC3(CCOCC3)C2)=O)co1 C(=O)(CC(P(C)(C)=O)c1ccoc1)NC(C)CCNC(=O)CN(C)C(N)=O C1(F)(CNC(C2(C(C)C)COC2)=O)CC(CNC(C2CNC(=O)C2)=O)C1 c1(C(N(C2CCN(C(=O)C3CC3)CC2)C)=O)cc2nccnc2cc1F CC1(C)CCC(C(=O)NCC23CC2CN(C(C2CN(C4CCOCC4)C2)=O)C3)C1 c1(OC)cc(S(=O)(=O)NCC(c2ccc(Cl)c(Cl)c2)O)sn1 C1(n2cc(C3CCCN(c4snc(C(=O)OC)n4)C3)nn2)CCC2(CCCC2)C1 C1(C(N(CC(CC)(C)OC)C)=O)C2CN(C(c3cc(C#N)c[nH]3)=O)CC12 C(C(C)(O)CC(=O)NC12CC(CNC(c3c[nH]c(=O)cn3)=O)(C1)C2)OC C(=O)(C1CCCc2c1ncn2C)NCc1c(Cl)cc(C)nc1 n1(CC)cc(NC(=O)C(=O)NCCNS(=O)(=O)N(C)C)c(C#N)n1 C12(C(=O)NC3CCN(C(c4c(CC)sc(=N)[nH]4)=O)CC3)CC(C)(CCO1)C2 N1(C(c2c(C)snc2)=O)CCCC2CN(C(c3n[nH]cc3C3CC3)=O)CCCC12 c1(C(N(C(=O)CC2CCCC(C)O2)CCCC)=O)c(-c2ccccn2)noc1C Cc1cc(C(=O)NC2CC2CNC(c2cccc(N)c2C)=O)ccc1S(C)(=O)=O C1(N=[N+]=[N-])(C(=O)NCC2C(C)(C)CN(C(=O)OC(C)(C)C)C2)CCOCC1 c1(C(=O)NCCOC2CCN(C(C3C(C(=O)OC)C3)=O)C2)cncc(F)c1Cl Cc1coc(C)c1C(=O)NCC1CCCN1C(c1csc(S)c1)=O C1(CNC(C(C(C)C)NC(=O)CCCN(C)C)=O)CCCC(C)(C)C1 C(=O)(CC(C(F)(F)F)OC(=O)CCC(=O)O)NCc1ccccc1.CC1C(C)N1 CCCC(C)CC(=O)NCc1ccc(C(=O)NCCn2cccn2)o1 C(CNC(=O)C(CC1CC1)NC(=O)C(C)Cn1ccnc1)(C(F)(F)F)OC N1(C(C(C2CC=CCC2)NC(c2nc(C)oc2C)=O)=O)CCN(C)CC(O)C1 N1(C(CC2CC(OC)C2)=O)CC(C(N2CCC(OCC(C)C)C2)=O)C(F)(F)C1 c1(OC)cccc(NC(=O)CSc2cccs2)c1.C1CC(=O)N(C)C2CC(C2)S1 C(=O)(CCCC(=O)N1CC2CC2(CNC(c2cncc(C(N)=O)c2)=O)C1)NCC c1(CNC(Cc2nc(=N)[nH][nH]2)=O)cccc(CNC(c2cc(CCO)on2)=O)c1 CC1CCCCC1(C)C(=O)NCCN1CCC(NC(C2(C=C)CCC2)=O)CC1 C1(CN(C(=O)Cn2nnc(=N)[nH]2)CC)CCCN1C(=O)CCN1CCCC1 c1(CNC(C=C(C)C(F)F)=O)cc2n(n1)CCN(C(=O)C(c1ccccc1)C)C2 N1(C(c2nc(COC)sc2)=O)CC(NC(c2cc(-c3ccco3)c[nH]2)=O)C(C)C1 C1(C(N(C(CC(C)C)C)C)=O)CCCCC1(C)NC(C1CCC1C(N)=O)=O C12(C)CCN(CC1)C(=O)C1CC(C)CN1C2=O.c1(COC)cccc(O)c1Cl c1(CN2CC3CN(C)CC3C2)cccc2c1CCN(C(=O)C(S)C(C)C)C2 CC(CC#N)C(=O)N1CCC(NC(c2ocnc2C2CC2)=O)C1 C=C(F)C1(CC(N2CCOCC2CC(=O)NCC2CC2C(C)C)=O)CCC1 N1(C(C2CCN(C(CN(C(C(C)C)=O)C)=O)C2)=O)CC2CCN(C)C2C1 N1(c2nc(C(C)=O)c(C)s2)CC2CCCC1C2CNC(c1cccc(C)n1)=O C(=O)(CC(O)CCCC)NC(C(=O)NCCCCC(=O)OCC=C)CCCC C1(CNC(C(CC)SC)=O)CCC(NC(=O)Cc2coc(C(F)F)n2)CC1 N1(C(CN(C)CC)=O)CCN(C(=O)C(C)CC2CCC2)C(c2ccc(F)cc2)C1 N#Cc1cc2c(nc1N1CC3CCCC(NC(=O)C4CC4)C3C1)CCOC2 C1(NC(C2CC(=O)N(O)C2)=O)CCN(C(C2CC23CCOCC3)=O)CCC1CO c1(C(=O)NC2CN(C(C3C(C(=O)OC)C3)=O)CC2F)ccc2nncn2c1 C#Cc1cccc(C(=O)NC(C(=O)NC2(C)CC2)c2ccoc2)c1 C1(CNC(C2C(C=C)CC2)=O)CN(C(c2cc(Br)c(C)cn2)=O)C2(CCC2)C1 N1(C(C=CC(CC)C)=O)CCCN(C(c2cnn(C(C)(C)C)c2)=O)C(C(C)C)C1 CCC(C)CCC(=O)NC(C1CN(C(c2cnc(SC)[nH]2)=O)CCO1)C C#Cc1ccc(C(=O)NC(C2CN(C(C3CC(C#N)(OC)C3)=O)C2)C)c(F)c1 CC1=C(C)CN(C(c2cn(Cc3ccccc3)cn2)=O)CC1 c1(N2CCN(C(CCC(=O)Nc3cn(C)nc3)=O)CC2)ccc(F)c2c1CCCC2 N1(C(C2(c3c(C)cno3)CC2)=O)CCC(O)(CNC(C2CC(C(C)C)C2)=O)C1 C12CCCCN1C(=O)NC2.Cc1ncc(CC2CSCCO2)s1 c1(C(N2CCCC(CN(C)C(c3cnon3)=O)C2)=O)cc(C(F)(F)F)ncc1Br C1(C(N(CCCNC(c2n(CC)ncc2Cl)=O)C(C)C)=O)CC(=O)NC(C)C1 Cc1ccc(C(=O)NC(C)C(C)NC(=O)CC2C=CCC2)cc1C#N c1(CNC(C2CCCCC2NCc2nc(CO)cs2)=O)ccncc1C(F)(F)F C12(CNC(C(F)=CCC)=O)CC(CC)(CN1C(C1CC1)=O)C2.c1(C(N)=O)ccccc1 C1(CN(CCNS(=O)(=O)Cc2ccccc2Br)CC)Cc2ccccc2C1 CCC(Cc1ccccc1)C(=O)N1CCCC1CNC(=O)C(C)(C)CF C(CN=C(NCC(c1cccs1)O)NCc1c[n+]([O-])c(C)cn1)OCC N1(C(CCc2c(OC)ccc(Br)c2)=O)CC(NC(=O)C=C(C)C)CC(F)(F)C1 C1(C(N(CCn2cccc2)CC)=O)(CF)CCN(C(=O)CCCC#N)C1 N1(C(COCCCC(C)C)=O)CC2CCCC(NC(c3n[nH]cc3Cl)=O)C2C1 CC1CC(C)(C(=O)NC2CCN(C(c3cc(C(F)F)n(C)n3)=O)C2C)CC(C)O1 c1(SC)ccsc1C(=O)NC(c1cnn(-c2ccccc2)n1)C c1(CC)cc(C)nc(N2CCC(OCCNC(=O)C(CO)NC(=O)C(C)C)C2)n1 C1(C)(C(=O)NCCN(C(c2csc(-c3cn[nH]c3)n2)=O)CC)CC1(F)Cl N1(C(c2c(C)onc2C2CC2)=O)CCC(CNC(c2cc(C#N)cs2)=O)C(C)C1 C1(C(N2CCC(C)(C(N3CC(O)(CO)C3)=O)C2)=O)CCc2n[nH]cc2C1 N1(C(C(C)(F)F)=O)CCC2CC2(NC(C2CN(CP(C)(C)=O)C2)=O)CC1 c1(C(N(CC(CC)NC(c2cnc3n2CCC3)=O)CC)=O)cc([N+](=O)[O-])oc1C N1(C(c2c(N)cc(F)c([N+](=O)[O-])c2)=O)CCCC(N=c2cc[nH]cc2)CC1 N1(c2ccnc(C)n2)CCCC(C)(C)C1CNC(=O)C(C)Oc1ccccc1 CC1CCCC(OCC(N2CC(CCNC(=O)Cn3ncn(C)c3=O)C2)=O)C1 C1(CNC(c2ccc(C)o2)=O)COCCN1C(c1cn(CC2CCCO2)nn1)=O C=CC1(C(=O)NCc2cnc(F)cc2C)CCN(C(=O)C=CCN2CCC2)CC1 C(CNC(=O)C(C)Oc1ccccc1F)(CC(C)C)NC(C1(COC)CCC1)=O C(=O)(CC1OB(O)c2ccccc21)N(C(=O)CC(C)(C1CCC1)C1(N)CC1)C C(=O)(C(C)(C)C(=O)OC)NC(C(C(=O)Nc1cccc(CC)c1)C)C N1(C(CC(=C)C)=O)CCC2C(C1)NC(=O)CN2C(=O)C(C)OC1CCCCCC1 C#CC1(C(=O)NCC(C2CC2)N(C(=O)CCc2ncc[nH]2)C)CCC1 n1(CC(=O)NCC(n2cnnc2O)(C)C)cc(C(c2ccns2)C2CC2)nn1 N1(C(c2cc(OC)c(O)c(N)c2)=O)CC(NC(=O)C(C)CO)Cc2ccccc21 C1(NC(CC(c2ccc(C)cc2)C)=O)CC2(C1)CN(C(=O)CCCC(C)C)C2 N1(C(C(CSC)OC)=O)CC2(CC(C(N3CC(C)C3(C)C)=O)CO2)C1 c1(C(=O)NCCCC2CCN(C(=O)C(Cl)=CCl)CC2)cc2c(nn1)CCC2 n1(CCC)cc(Cl)c(C(=O)NCC2CCN(C(=O)COc3ccccc3F)C2)n1 c1(-n2cc(CN(C(c3ccc(CC)cn3)=O)C)nn2)ccc2c(c1)CCC2 N1(C(c2ccc(CNC(C3C4CCCOC34)=O)s2)=O)CC2CCOC2C1 C12(C(=O)NCC3CCN(C(CN(c4nccs4)C)=O)C3)CC(CCO1)C2 N1(C(C(=O)NC(C)C(=O)OCC)=O)CCN(C(=O)NCC)CC1C C12(CNC(COCC=C)=O)CCCC1CCN2C(=O)CCOc1ccccc1C N1(C(C(C)C(F)F)=O)CCC2(C)CN(C(=O)CC(C)N(C)C)CC12 Cc1ccc(CCC(=O)NC2CC3(C2)CN(C(=O)CCNS(C)(=O)=O)C3)c(C)c1 Cc1nc(CC(=O)N(CC(C)CNC(=O)CN(C)C(=O)C2CC2)C)cs1 Cc1nn(C)c(C(=O)NCCC2CN(C(c3ccc(NC=O)cc3)=O)C2)c1Cl C(CN=c1[nH]c(=NCc2n[nH]cc2Br)c2sccc2[nH]1)n1c(C)ncc1 N1(C(=O)Cc2cccnc2F)CC(O)CC2CCCCC12 N1(C(C=CC)=O)CCCCCC(NC(c2cc(C3CC3)oc2C2CC2)=O)C1 N1(C(c2cc(C)nn2C)=O)CCC2(CC(C(=O)N3CCN(C)CC3CO)=NO2)C1 CC1CC(CNC(=O)COc2ccccc2Br)CN1C(=O)CCCC1(C)N=N1 Cc1nc2cncc(C(=O)NC3COCCN(C(C4CN(C)C4)=O)C3)c2[nH]1 c1(C(N2C(CNC(=O)C3=CCCS3)CC(OC)C2)=O)noc2c1CCCC2 c1(C2(C(=O)NCCCCCCC)CCC2)cccc(C2=CCN(C)C2)c1 CC12CC3(C1)C1(CN(C1)C3=O)O2.C(C)(C)(C)OC(=O)NCC#N.C1(O)(CO)CC1 CC#CC1CCN(C(=O)CCN(CCCO)C(c2c[nH]c(=NC)s2)=O)CC1 c1(C(=O)NCC2CN(C(CCNC(C)=O)=O)CC2C)[nH]nc2c1COC2(C)C c1(OC)cc(C)c(C)cc1-c1ccnc(CC(=O)Nc2cccc(CF)c2)c1 N1(C(C2(CSC)CC2)=O)CCCC(CCC(=O)NCCC2CC(C)(C)CO2)C1 Cc1onc(-c2ccncc2)c1C(=O)NCC(C)N(C)C(C1CCCC1(F)F)=O Cc1c(C(N2CCC(C(C(C)C)NC(=O)C(O)CF)CC2)=O)ncn1C O=C(O)C(CNC(=O)C(F)(F)C1(O)CCCC1)Cc1cccc(Cl)c1 C1(CC)C(NC(c2cncc(C)n2)=O)CCCN1C(=O)C(C)CC1CCCC1 N1(C(C(CC)C2CCC(=O)N2)=O)C2CCC1CN(C(C1(CCF)CC1)=O)CC2 C=CC1(CC(=O)NC(C)C(C)NC(c2cc(C)c(C)nn2)=O)CCCCC1 CC1(CNC(C23CC(C2)C3)=O)CCCN(C(c2ncc(Cl)cc2F)=O)C1 C#CC1CC2(CC2)CN1C(=O)CN(C(=O)C=CC=CCC)C1CCC1 O(NC(=O)C(C)n1cc(CC2CC2)nn1)CC1CCC(=C)C1 c1(CC)cc(CC)nc(N2CC(CO)(NC(=O)CCc3ccc(F)c(Cl)c3)C2)n1 C1(NC(COCCC)=O)CCC(C)(C)CC1CNC(=O)CCCc1ccccn1 Cc1ccc(NCCC(=O)N(C(=O)C(C)(O)C(C)O)C2CCOCC2)c(F)c1 O=C(C#CC1CCCC1)NC1(CNC(c2cccc(-c3ccoc3)c2)=O)CCC1 C1(NCCCC2C(C)C2)CC2(CCN2)C1(C)C C1(CNC(=O)C(F)=C2CCC2)C(C2CC2)CCN1C(=O)C(O)CC(F)(F)F C1(C(=O)NCc2cc(O)cc(O)c2)CCN(CCOc2cccc(Cl)c2)CC1O CC1C(NC(=O)C(=O)N(C)C)CCCN1C(c1ncc(Br)cn1)=O Cc1cc(C(=O)NCCCC(C)NC(=O)C(C)n2ccnn2)n[nH]1 C12(O)CCN(CC1)C2=O.C=CCCCN(C)CC1CC1(C)C N1(C(COCC(=O)OC)=O)CC2(CCCCN(C(=O)CSC(F)F)C2)C1 C1(CCNC(c2c(C(C)C)n[nH]c2)=O)CSCCN1C(C1CCCC12CC2)=O N1(C(c2cccc(C)c2C)=O)CCC(F)(F)C(NC(c2ncsc2C)=O)C1 S(=O)(=O)(c1cc(C)c(Cl)cc1F)NC1C2CN(C(C(CSC)(C)C)=O)C(C2)C1 C1(NC(CC2CC(C(=O)OC)C2)=O)CCN(C2CC2)C1=O.C12CC1C(=O)N2 CC(C)(C)C(C#N)C(=O)N1CCCC(F)(CO)C1.C12C3CC4C(C3)C14C(=O)NO2 CC(O)(CC(=O)NC1CC(NC(=O)CCC(N)=O)C1)c1ccccc1 c1(NCc2cc(C)[nH]n2)[nH]c(=NCC2(C)CC2Br)nc2c1ncn2C c1(CNC(Cc2nc(C)oc2)=O)nc(C)c(C(=O)N(C)CC2(O)CCC2)o1 C12(CNC(c3ccc(C(C)C)o3)=O)CC(CO1)N(C(=O)CSCCC#N)C2 N1(C(C2N(CC)CC2)=O)CCCCC(NC(=O)COC(C)(C)C)CC1 C(=O)(CCC(=O)C(C)(C)C)NC1CC(CN=c2cc(C)nc[nH]2)(F)C1 C(=O)(C1CCCc2n[nH]cc21)NC1C2N(C(c3c(C)c(Cl)ccc3)=O)C(CC2)C1 c1(COC)noc(COC(=O)C(c2ccc(Br)s2)N2CCOCC2)n1 N1(C(C(CC)NC(C)=O)=O)CCN(C(=O)C(F)CC2CCOC2)C(CO)C1 N(C(=NCCSCC1(c2ccc(Cl)cc2)CCC1)N)C1C(C)C1 CCC(C)(C)CC(=O)N(C(C)C(=O)N(CCCCCO)C)CC C1CCc2nnc(C)n2C1.C1(NC(c2c(CC)nn[nH]2)=O)(CO)COCCC1C C=CCCCCCC(=O)NC1(C(=O)Nc2ccc(C)c(CSC)c2)CCC1 CC1(C(=O)NCC2(NC(=O)CCS(C)(=O)=O)CC2)OCCc2ccccc21 N1(C(C=C(C)Cl)=O)CC(NC(C2CCCC2O)=O)Cc2ccccc21 C=CCC(C)(CNC(c1sccc1CNC(=O)CCCOCCC)=O)CO N1(C(C)=O)c2ccccc2CC1C(=O)NCC(C)NC(C1CCC2(CCC2)C1)=O C(CCC(C)C(=O)NCCCCCC(=O)NCCN(C(C)C)C1CC1)OC Cc1cccc(C(N2CCC(C)C2CNC(=O)Cc2scnc2C)=O)c1[N+](=O)[O-] CC1(C)CCN(C(=O)Cc2cncnc2)C1C(=O)NCC=CBr C1(c2c(C)ccnc2)NC(=S)N(CCO)C(C2CC2C)=C1C(=O)NC1CC1 CC1Cn2nccc2CN1C(=O)COC1CCN(C(C2(C#N)CCCOC2)=O)C1 C1(C(=O)NCCCN(C(=O)CS(=O)(=O)N(C)C)C)CC12CCC1(CC2)OCCO1 C1(C(=O)NCCCC2CCCO2)CCCN(Cc2n[nH]cc2Br)C1 CCC(C)S(=O)(=O)Oc1ccc(OCCC#N)cc1 C1(N(C(C=CC=CC)=O)C)CN(C(=O)Cc2sc(CC)nc2C)CC1O CN1CCC(C2CCCN(C(c3cn(CC4N=N4)nn3)=O)C2)CC1 O=C(C#CC1CCCC1)NC1CN(C(c2csc(-c3cnc[nH]3)n2)=O)CCC1F C12CCCN(C1)CC(=O)NC2.c1(C(N2CC(CC)C2)=O)cnnn1C1CC1 c1(C(=O)NCC(C)=CC(=O)N(C)CC2CN(C)CCO2)cnncc1O N1(C(c2c(C)cc[nH]2)=O)CCC(CCNC(=O)CC2CCCO2)C(F)(F)C1 C1(CNC(C2CC(F)C(=O)N2)=O)CCC(NC(C23CC(CO2)C3)=O)CC1 CC(O)(CC(=O)NCc1cccc(CNC(C2CCCCS2)=O)c1)C(F)(F)F CC1(CNC(c2csc(CC(F)(F)F)n2)=O)CCCN1C(=O)CN1CCSCC1 C(=O)(C(C)(C)CC(F)(F)F)NCC(C)(C(C)C)NC(C(CO)OC)=O C1(O)(C(C)NC(=O)Cn2cnnc2O)CCN(C(c2cc(Br)ccn2)=O)C1 CS(=O)(=O)c1ccc(NCC2CCC(CC(N3CCC(Br)CC3)=O)CC2)cc1Br C1(NC(C2CC(C)C2)=O)COCC1CNC(C1CC(n2ccnc2)C1)=O Cc1cc(=NC2CCN(C(c3cc(Cl)on3)=O)CC2C)[nH]cc1C#N c1(CCNC(c2n(CC)nnn2)c2csc(Cl)c2)ccc2c(c1)OCCCO2 c1(OC)ccc(C(=O)NCC=CCNC(c2coc(C)c2)=O)c(Br)c1F N12CC=C(C(=O)NC(CC(=C)C)C1=O)CC2.C(C(CC)C(C)(F)F)NC(=O)CCC c1(OC)ccc(Cl)c(NC(C2CC2CNC(=O)CN2CCN(N(C)C)CC2)=O)c1 C1(NC(c2occ(C)c2)=O)CN(C(c2ccncc2C)=O)CC12CCOCC2 CC1CN(C(c2ccccc2F)=O)CC1NC(=O)C(c1cccnc1)O C1(CC(=O)NCC2C(CC)C2)COCCN1C(C1CC(F)C(=O)N1)=O c1(CC)ccc(C(=O)NCC2CCCCCN2C(=O)CC(O)C(C)C)c(F)c1 C(=O)(C(C)C(F)F)NCCN(C)CCOC(C(COC)C)=O C1(NC(C(c2cccnc2)OC)=O)CCC(C)(NC(=O)C(F)CC2CCC2)CC1 c1(OC)cc(C(=O)NC(c2ccc(Cl)cc2)CNC(=O)C(=O)NC2CC2)n(C)n1 N1(C(c2ccc(C)o2)=O)CCC(C2CCOCC2)(CNC(c2cncn2C)=O)C1 C(c1c(F)cccc1F)=CC(=O)NC1CN(C(C23CCCC2C3)=O)CC1O C1(C(=O)NCc2ccc(C(=O)NCC(C)OC)cn2)CCCC(C)(C)C1 CCCCC(O)CCC(=O)N1CCCCC1CNC(c1ccc(COC)o1)=O Nc1cc(C(N2CC3(C2)CN(C(C2COC2)=O)C3)=O)cc(Cl)n1 C1(NC(c2nccc(CC)c2)=O)CN(C(=O)C(CO)N(C)C)CC1(C)C c1(C(N2CC(C(C(=O)N(C(c3ccccn3)C)C)O)C2)=O)cc(=O)cc(Cl)[nH]1 C1(N(C(C2C(CC)C2)=O)CCO)CCN(C(c2cc(C)c[nH]2)=O)C1 Cc1nnc2n[nH]c(NC(C3(F)CCCOC3)=O)c2c1C c1(C(N2C(CCNC(c3csc(F)c3)=O)COCC2)=O)cc2cccn2c(O)n1 c1(CC)cnc(O)c(C(=O)NC(C)CN2CCN(C(=O)C(F)C(C)(F)F)CC2)c1 Cc1ccc(O)c(CNC(=O)C(F)C2CC(NC(c3cccc(CO)c3)=O)C2)n1 C(C(C)(C(C)C)NC(c1n[nH]c(C2CC2)c1Cl)=O)NC(CNC(C)=O)=O C1(C(N(C2CCN(C(C=C(CC)CC)=O)C2)CCC)=O)(CCOC)CCOCC1 C1(CN(C(C)(CO)CO)C(=O)Cc2ccccc2)CCOC(c2cccnc2)C1 N#Cc1ccc(N)c(C(N2CC(C3(NC(=O)Cc4ccccc4F)CC3)C2)=O)c1 CC1CN(C(=O)Cc2cccc(F)c2F)C(C)CN1C(c1cccs1)=O Cc1cc(C(=O)CN2CC3C(CNC(C4CCC4)=O)C3C2)cc(C)n1 c1(CC(=O)NCCCCC(C)NC(C2CC(CN(C)C)C2)=O)nc([N+](=O)[O-])n[nH]1 N1(CC=CCNC(C=CC=CCC)=O)CCC(N2CCCC2)C1 C1(NC(C2CCN(C(CC)=O)C2)=O)CN(C(C2(N=[N+]=[N-])CC2)=O)CC1F Nc1nc(Cl)cc(Cl)c1C(=O)NCC1CN(C(C2(n3ccnn3)CC2)=O)C1 c1(CCC)cc(C(=O)NCC2CC(NC(=O)C(CC)N(C3CCCC3)C)C2)n[nH]1 C1(CC(N2CC(C)N(C(c3cnc[nH]c3=N)=O)CC2)=O)CC2(CCC2)CCO1 c12ccc(c(F)c1)NC(=O)N2.Cc1cn(C)nc1CN1CCOCC1 c1(CC)ccc(-n2nc(-c3cncc(F)c3)nc2C2CCCN2C2CC2)cc1 C12(CNC(C3CC(SC)C3)=O)CCCC1N(C(c1cc(C3CC3)ns1)=O)CCC2 CC(O)C(C(=O)NCCC(C)(C)NC(=O)CO)NC(c1cccs1)=O n1(CC(=O)NCC(C2CC2)NC(c2cc(C)[nH]n2)=O)cc(Br)c(O)nc1=O c1(NC(CC=CCNC(C(C2CCC2)OCC)=O)=O)ccccc1O N1(C(C(CC)OC)=O)CC2(CO)CC2(CO)C1.C(CCCO)N(C(C)=O)CC N1(C(=O)N(CCC(c2ccc(F)cc2)O)CC2CCCO2)CCC2CCC(C1)S2 C1(C(=O)OC(C)(C)C)CN(C(=O)OCc2ncccc2Br)C2COCC2O1 C#CCCCCCC(=O)NCC1CC2CC2N1C(=O)CS(=O)CC c1(C(=O)OC)cc2c(nc1N1CC(C)(NC(C3CCCSS3)=O)C1)CCC2 Cc1nc2ccc(C(=O)N(CC(C)NC(=O)C(C)(C)c3cnsc3)C)cc2s1 Cc1c(C(N2CCCC(CNC(=O)CC(=O)N(C)C)C2)=O)cccc1CO C1(OCC(N2C(C)CCCC2)=O)CCN(C(=O)CCc2ccoc2)C1(C)C c1(OC)cncc(CNC(=O)C(CC2CC2)NC(=O)CC23CCC(CC2)C3)n1 Cc1ccc(C(=O)NCCC(C)CCNC(=O)CCOC(C)C)c(Br)c1 C1(CCNC(CC)CCCO)CCC2(CCOCC2)CO1 c1(NC(CC(CC)CC)C(=O)NC)cc(C#N)cc(S(C)(=O)=O)c1 N1(C(C(C(C)O)C)=O)CCC2(CC1)OCCC2NC(c1ccc(CO)c(Cl)c1)=O C(C(C)CC(=O)N1CCC(N2CCCC2)C1)NC(CN(CCC)C)=O c1(CC(=O)NC2C(CNC(c3c(N)ccc(C)c3)=O)CC2)cccc2ccnn12 C12(CNC(CC(C=C)(C)C)=O)CCCC1N(c1ncnc3c1ncn3C)CCC2 C1(CNC(C(C)SC)=O)CCC2CN(C(c3cc(C)oc3C)=O)CCC2C1 N1(C(CC(CC)C)=O)CCC2(CNC(=O)CCSC(F)(F)F)CCCCC12 Cc1nc2ccc(C(=O)NCC3(F)CC(CNC(C4(C)CC=CC4)=O)C3)cn2n1 Cc1cc(C(=O)NC2(CNC(c3n[nH]c4ccccc34)=O)CC2)c(Cl)cc1N c1(C(N2CCC(C)(CNC(C(C(C)C)OC)=O)C2)=O)ccnc2ccc(F)cc12 c1(NC(C)=O)ccc2cc(-c3noc(C4CCC(O)C4)n3)ccc2c1 C(C(CC(C)C)C(=O)NCC1CC(NC(=O)CCc2nc(C3CC3)no2)C1)OC C(=O)(CC1=CCCCC1)NCC1C(CNC(CC2CCC(C)(C)O2)=O)C1 N1(C(C(c2ccnn2C)NC(c2c(OC)ccs2)=O)=O)CC2(C1)CC(C)(F)C2 C(=O)(C1Cc2ccccc21)N1CC(CNC(=O)C2=CCCOC2)C1 C(=O)(C(CC(C)C)C(N)=O)N(CCCOCCNC(c1cccc(C)n1)=O)C S(=O)(=O)(c1cccc(Cl)c1)N1CCC(NC(=O)OC(C)(C)C)C2(C1)CCC2 Cc1c(C(=O)NC2CCN(C(=O)C(C)c3ccco3)CC2C)cc(O)cc1N Cc1cc(=O)c(C(=O)NC2CN(C(c3ccncc3)=O)CC2O)cn1C C1(C(N2CCCCC(NC(c3c(C#N)cn[nH]3)=O)C2)=O)CC2(CCCCC2)CO1 C1(CNC(c2ncccc2F)=O)CC(C(F)(F)F)CN1C(=O)C(c1ccccc1)F CN1N=C(C(=O)NC2CC(CCNC(C3CC(=O)N(C4CC4)C3)=O)C2)CCC1=O Cc1cc(CC(N2CCN(C(=O)Cc3cnoc3)CC2CF)=O)c(C)n1C1CC1 C1(CNC(CCCCOC)=O)CC2(CCC2)CN1C(c1ccc(C#N)c(Cl)c1)=O C(=O)(C(C(C)C)NC(C1C=CCCN1C(C1CC1(Cl)Cl)=O)=O)NC Cc1nc2cc(CNC(N(CC(C)(C)CN)C(=O)O)=O)ccc2o1 CCC(CC(=O)NCc1ncc(C(=O)NCCCC2(O)CCC2)cn1)C1CC1 c1(C(N2Cc3cccc(C)c3C2)C(=O)NCCCC)n[nH]c2ccc(Br)cc12 N1(C(c2cc(CNC(C(CC)NC(N)=O)=O)oc2)=O)CC2CCC1C(O)C2O CC1NC(=O)OC12CN(C(=O)CC1CC(O)CN1C(=O)Cc1cccnc1Cl)C2 Cc1cc(F)ccc1-n1cc(O)c(C(=O)NCC2CCN(C(=O)C(C)CO)C2)n1 N1(C(C(F)=C(C)C)=O)CCOCC1c1ccc(C(=O)NCC(C)F)n1C N12CCN(C(=O)C1)C2=O.C(C)(CSc1ccccc1)(CC1CCC1)OC N1(C(CC2(COC)CC2)=O)CCCC(C(C)C(=O)NCC(C2CCCCC2)C)C1 c1(NC(C(C)(C)C(N)=O)=O)cccc(S(=O)(=O)N=c2cc[nH]cc2Cl)c1 c1(OC)c(C(N2CCC(O)(CCNC(C3CC4CC3CO4)=O)C2)=O)ncnc1C c1(OC)nn(C)cc1C(N1CCC(O)C1C(=O)NC1(C)CCC(C)C1)=O C1(NC(c2ccc(N(C)C)cc2)=O)CC2CCC1N(C(=O)C(F)(F)C1CC1)C2 N1(C(C(CCC=C)NC(CCC=C=C)=O)=O)CCC(O)C(C)(O)C1 CCCC(C(=O)NCC1(CN(C(=O)C(C(C)C)c2cc(C)no2)C)CC1)C(C)C C(C1=CCSC1(C)C)(c1nnnn1CC1CC2(CC2)C1)NC1(C(=O)NCC)CC1 N12C3CCC1CC(C3)CNC(=O)CCCC2=O.c1(NC(C)=O)cncc(C2CC2)c1 N1(C(CNC(C)=O)=O)CCOCC(C)(CNC(C2(CF)CCC2)=O)C1 c1(C(=O)NCC(C)CN(C(=O)CN(C2CCC2)C)C)cc(F)cnc1Cl c1(C(=O)NCC(CC)NC(c2snnc2C(C)C)=O)ccc(C)s1 c1(SC)ccc(C(=O)NCC2CN(C(=O)Cc3csc(C)c3)CCO2)c(Cl)c1 C1(CNC(C(CCC)O)=O)CN(C(=O)C(c2csc(=N)[nH]2)=O)CCC1(F)F c1(OC)ccc(C(C)C(N2CCCC(CCNC(C3CCOCC3)=O)C2)=O)cc1 N1(C(c2cn(CC=C)nc2)=O)CC(CNC(c2n[nH]cc2CC)=O)C(F)(F)C1 C(=O)(C(C)CC1CCCC1)N(CCNCC=C)CC.C1(C)C(=O)N1 c1(NC(CC2CN(C(=O)Nc3c(C#N)cccc3)C2)=O)cnc2ccccc2c1Cl C(=O)(CC(C)C(F)(F)F)NC1C2CN(C(c3c(OCCC)cccc3)=O)CC1C2 Cc1cnc(C(=O)NCC(C)(C)C(=O)Nc2cncc(C3CC3)c2)c(C)c1 O=C1CCC(c2nnc(CN)n2C)CCO1.C1(N2CCCC2)CC2(CCCCO2)C1 N1(C(CN(C(=O)C(C(C)C)SC)CCOC)=O)CCOC(C2(C)N=N2)C1 C1(NC(CCOCCC)=O)CCCN(C(c2ccncc2C(=O)OC)=O)C1 c1(C(=O)NCC(C2N(C(c3scc(C)c3)=O)CCC2)(C)C)cc2sccc2n1C C(=O)(C(C)C(C)COC)NC(CCC)C(=O)N1CC(OCC(F)F)C1 C(CC(C)(C)CNC(=O)CSCc1ccncc1)NC(C(C)CF)=O C1(C)(N(C)CC)CCN(C(=O)CN(C(=O)C(C)c2ccsc2)C2CC2)C1 c1(OC)cn(C)c(C(N2CCC2CNC(=O)Cc2csc3ccccc23)=O)cc1=O CCCC(CNC(c1ccc(CO)s1)=O)C(=O)NC1(CCC)CCOC1 c1(C(=O)NC2CN(C(c3noc(CC)c3C)=O)CC2C)cnc(C)c(N)c1 C1(C(N2C(C)CN(C(=O)CC3(N(C)C)COC3)CC2)=O)CCc2nncn2CC1 C(C(F)(F)CN=c1[nH]c(=N)[nH]c(=NC(CC2CC2)c2ccc(F)cc2C)[nH]1)OC Cc1ccc2c(c1)CCC(C(=O)OC1CCCC(C(F)(F)F)C1)O2 CCC(CCC(=O)Nc1cccc(F)c1F)NC(=O)Cn1nc(C)oc1=O Cc1nc(C(N2CCC(C(F)CNC(=O)COCCN(C)C)CC2)=O)sc1C CCC(C)CC(=O)NC1CCC(NC(=O)Cc2sc(C3CCC3)nc2C)C1 N1(C(C2CC(CCNC(=O)CC3CCCC(O)C3)C2)=O)CCC=CCCC1 C1(NC(CSCC(C)=O)=O)CN(C(=O)C(C2CC2)C2CC2)CC1O c1(OC)cc(N)ccc1C(N1CCC1C(C)(C)C)=O c1(NC(COC(C2C(CC(C)C)OCCC2)=O)=O)ccc(O)cc1F Cc1cc(F)c(CN2CCN(c3cc(N4CC(F)C4)ncn3)CC2)c(F)c1 c1(C(=O)NC2CC(F)(CNC(C3=C(C)OCC3)=O)C2)cc2c(=O)[nH]ccn2c1 C1(C(=O)NC2(CC=C)CN(C(=O)CC3CCCOC3)C2)(OC(C)C)CCCOC1 C1(CNC(C2C(C=C)C2)=O)CCN(C(=O)C2=CCCCC2)C1(C)C c1(CC(N2CC(CNC(C(CO)OC)=O)C(N(C)C)C2)=O)cc(C)ccc1C CC1CN(C(=O)C=Cc2cscn2)CC1(C)C(=O)NCC1CNC1 c1(C(=O)NC2CC(F)(CNC(C(CN(C)C)O)=O)C2)ccc(N)cc1Cl c1(C(c2nnnn2Cc2cccs2)NC(C)COC2CC2)cc2ccccc2o1 C(=O)(CCCCN1CCOCC1)N1CCC(C(C)NC(c2cc(OC)n[nH]2)=O)C1 c1(C(=O)NCC2C(C)CN(C(=O)CSC(F)F)C2)cc(F)cc(Br)c1 N1(C(c2ccnc(OC)n2)C(=O)NCCSC)CCc2c(cccc2[N+](=O)[O-])C1 C1(N(C(C2CCN(CC)C2)=O)C)CN(C(c2cn(CCF)nn2)=O)CC1(C)C C(N=c1cc(Cl)nc[nH]1)C1CN(C(Cc2ncc(CC)[nH]2)=O)C(C)C1 N1(C(C)=O)CCCCC1CC(=O)N(C1CC(NC(=O)CSC2CC2)C1)C C1(C(C(=O)NCC(CCOC)NC(C2(C#N)CCC2)=O)C)CCN(C(C)=O)CC1 c1(C(N2CC(CNC(c3c(C)occ3)=O)C(F)(F)C2)=O)cc([N+](=O)[O-])cnc1N c1(C(=O)NCCNC(C=C(C)CS)=O)c[nH]c2nccc-2c1.N1(C2CC2)CC=CC1 C1(CC)C(C(=O)N(CC(C)(C)NC(=O)C=CBr)C)CCN1C CC1CN(C(=O)C=CCN2CCCC2)CC1(C)C(N1CCOC(C#N)C1)=O C1(CCOC)(NC(CCCOC(C)C)=O)CCN(C(=O)C(C)(C)SC(F)(F)F)C1 Cc1csc(C(N2CCN(C3(C)COC3)CC2)=O)c1Br c1(C(=O)NC2C(C)(C)CN(C(c3ncc(Cl)cc3Cl)=O)C2)cn2ccccc2n1 Cc1ccc(CNC(C2CCOC2)C#N)cc1Br c1(C(=O)NC2(C)CC(NC(C3CCCS3(=O)=O)=O)C2)cccc2c1OCCC2 C1(C(=O)NC)(NC(c2cccnc2)C2CCOC2)CCCCC1 CC(C)(C)CCCCNC(=O)C1=CCN(C(c2ccncc2Cl)=O)C1 CN1CCN(C(C23CCC(CC2)C3)=O)C(CNC(C2CC3CC2C3)=O)C1 c1(C(=O)NCC(CN(C(=O)C(C)N(C)C)CC)(C)C)cn2c(n1)SCC2 c1(NC(C2N(C(C(C)C)=O)C3C(C2)C3)=O)cc(O)nc(Cl)n1 Cc1c(C(=O)NCc2csc(CNC(=O)CCSc3ccccc3)n2)cccc1Cl Cc1scc(C(=O)NC(C)CC(C)NC(C2CCC2C(C)(C)C)=O)c1C N1(C(C2CC(CNC(CCC(C)OCC)=O)OC2)=O)CCC2(CC1)N=N2 C1(CCC(C)C)C(=O)N1.c1(N2CCC(CC)CC2)cc(C)nc(SC)n1 c1(C(N2C(C(C)NC(COCCC)=O)CCC2)=O)cc(F)c(F)cc1C(F)(F)F C12(CNC(COC(C(C)OCC(C)C)=O)=O)CC3CC(CC(C3)C1)C2 N1(C(CC=CC)=O)CC23CCCC2(C1)CN(C(=O)C(=O)N=S(C)(C)=O)C3 C1(O)(CNC(c2cncnc2C2CC2)=O)CCN(C(c2coc(O)n2)=O)C1 N1(C(C(C=C)O)=O)CCOC2CCN(C(c3ccccc3NC(=O)OC)=O)CC12 C=CC1CN(C(=O)CC(C)(C)C2CC2)CC1NC(=O)COC(C)CC C1(N(C(=O)CCC=C(C)C)CCC)CCN(C(=O)C(O)C2CCCC2)CC1 c1(CNC2CC(C(F)C(=O)OCOC)C2)cc(OC)ccc1C.C1(F)(CC)CCOC1 C1(C)(NC(c2c(CNC(C(c3ccnn3C)C)=O)scc2)=O)CC2CCC1C2 N1(CC(=O)N(C(CNC(C=Cc2ccc(C)o2)=O)C2CC2)C)CCCNS1(=O)=O C1(CC#C)(C(=O)NCC#CC(N2CCOC(CC3CC3)C2)=O)CCCCC1 CCC(C)(CO)C(=O)NCC1CCCN1C(c1ccc(N)c(Cl)c1)=O S(=O)(=O)(c1cccc2cnc(Cl)cc12)N(C1CCCN(C)C1)C c1(OC)cc(C)c(C(=O)NCC(C2CCOC2)NC(C2(C3CC3)CC2)=O)c(F)c1 C1(NC(c2ncn(C(C)C)c2)=O)CCC(C)(CNC(c2nn(C)cc2Cl)=O)C1 C1(CCC)CN(C(=O)Cn2ncccc2=O)CC1NC(=O)C(=O)NCC1CC1 CC#CCC(CO)NC(=O)COCCC(n1cc(CC(O)C(C)C)nn1)OC C1(F)(C(=O)NCC(CNC(C2CC(CF)C2)=O)OC)CCC(F)(F)CC1 CCCCCC(C(=O)NCC(CNC(c1csc2ccncc12)=O)OC)C(C)C C(=O)(C(CNC(C12CCCN1CCC2)=O)CC(C)C)NC(C(=O)NCC)C S(=O)(=O)(c1cccnc1Cl)NC1CCC(CNC(C(C)(C)O)=O)CC1 C(C(O)C(=O)NCCOC1CCN(C(=O)Cc2ccn(C(C)C)n2)C1)=CCCC N1(C(CC)=O)CCCCC1Cn1cc(CCONC(c2cc(Cl)n(C)n2)=O)nn1 C(=O)(C(F)CC(CC)CC)N1C(CC)C(C(=O)NCc2[nH]nnc2C)CC1 CCC(CC(=O)N(CC(C)CNC(=O)CC(C)F)C)CC(C)C C1(NC(=O)NC(C)C(=O)NCc2n[nH]c(-c3ccccc3)n2)CCOCC1 C1(NC(c2c(C)cco2)=O)CC2CC1N(C(c1cnc(C(F)(F)F)s1)=O)C2 N1(C(COC2CC(NC(CC(C)N(C)C)=O)C2)=O)CC2CC(C1)N(C)C2 Cc1nc(C(N2CC(CNC(=O)CSC(F)(F)F)C3CC23)=O)cc(O)n1 c1(C(C)C)nnc(C=CC(=O)NCC(C)(O)CNC(=O)CCc2nccn2C)o1 N1(C(C(c2ccccc2)OC)=O)CCC2(C1)CN(C(c1nn[nH]c1Cl)=O)C2 c1(C(=O)NC2CCC(NC(=O)COC3CC3)CC2)nnn2c1C(=O)NCC2 C12(NC(C(N3CCC(OC(C)C)C3)=O)=O)CCOCC1C2 c1(C(N2C(C(=O)NC(C)CC)CC(=C)C2)=O)c(C)ccc(I)c1C c1(NC(=O)C(C)C(=O)OCc2nc(CC)sc2)cc(Cl)nc(Cl)c1 C1(NC(COCCN(C)C)=O)CC1C1CCCN(C(C2(CO)CCOCC2)=O)C1 C(=O)(C(C)CC(=O)c1ccccc1F)NCC1CN(C(CSCCC)=O)C(C)C1 CCC(O)(CN(C)C(C1CC2CC2N1C(=O)COCc1nc[nH]n1)=O)CC C1(C(C(=O)N(C2CCCC2)CC(=O)OC)C)CN(C(=O)CC(C)(C)C)CCO1 C1(C(N2CC(NC(C3CCCCC3C(F)(F)F)=O)C2)=O)Cc2ccccc2N1 C1(CNC(=O)OC(C)(C)C)CC2(C1)CN(N1CCCC3(C1)CCOCC3)C2 C1(C(=O)NCC(C)(C2CC2)NC(C2CCCC(OC)C2)=O)CCC(=O)N(C)C1 Cc1cccc(C(=O)NCc2ccoc2C(=O)NCC=C(Cl)Cl)c1O C(C(=O)N1CCN(C2CCCN(C(=O)C=C(C)C(C)C)C2)CC1)(C(C)C)SC C=CC(COC)N=c1nc2c(cnn2C)c(NCCN2CC3CCCC3C2)[nH]1 c1(CC)nccnc1C(N1CCN(C(C)CNC(C2CCC(=O)C2)=O)CC1)=O C1(C(C(=O)OOC(F)F)N(N2CCCC2)CCCC2CC2)CCC(OCC)CC1 C(CC(C)(C)C(=O)N1CC(CC(F)C(=O)N(C)CCC2CCOCC2)C1)OC C1(C(=O)NC(C2CC(NC(c3cc(OC)no3)=O)C2)C)CCCSC1C c1(C(c2n(CC)nnn2)NC(C)CCCOC)ccc([N+](=O)[O-])c(C)c1 C(=O)(C(C)CC(F)(F)F)NCC1CCC(NC(C(N2CCCCC2)C)=O)CC1 Cc1ncc(C#N)cc1NC(=O)CC1CCCCN1 C1(NC(c2nc(C)sc2C)=O)CCN(C(=O)CSCC(N)=O)C(C)C1 N1(C(CCc2ccc(OC)c(OC)c2)=O)CCC2(CC1)CC2C(=O)NCC(C)C C(=O)(C(C)S(N)(=O)=O)N(CCNC(c1nc(C)c(C)s1)=O)C C1(C(=O)NCc2ccn(C3COC3)n2)(CNC(c2cnc(O)o2)=O)CCCC1 CCCCC(C)CCC(=O)NC1CCC1NC(=O)CCCCCCSC C1(NC(C=CC)=O)CC2CN(C(C3(c4ccc(OC)cc4)CC3)=O)CC2C1 C=C(C)CC(C(=O)NCC1CC1CC(=O)NCCN(CCO)C(C)C)OC c1(CN(CC(C)(C)C)C(c2cc(C)on2)=O)ccc(N2CCOCC2)c(C)c1 N1(C(c2c(C)csc2)C(=O)NCc2ccco2)CCC2(CC1)COC(C)(C)OC2 CCCC(CNC(=O)CCc1cnco1)C(=O)NC1C2CCCCCC12 C1(C(=O)NCC(CC)NC(c2ncn(C(=O)OC)n2)=O)C=CCCC1 C(=O)(C#CC1CC1)NC(c1ccc(F)cc1)CNC(CC=CC=C)=O C#CCCCCC(=O)N1CCC(NC(=O)Cc2ccccc2)C(C)C1 c1(C(=O)NC2C(CNC(C3CCC(=O)O3)=O)CC2)ccc2occc2n1 C1(N(C(=O)C(O)CC2CCCC2)C)CCC(NC(=O)C=Cc2ccco2)CC1 C(=O)(CCC(C)CC)N1CCC(CC2N(C(CCC(=C)Cl)=O)CCC2)CC1 O(N=C1CCCCCC1)CCN(C(C(=O)NC)=O)CCNC(=O)C1CC1 C1(OC)CC(C(=O)NNC(=O)C2(C)CCCOC2)C1(C)C C1(=O)C(C)(CC)N1CCCNC(=O)OC(C)(C)C.C1(C(=O)OC)CCC1CN.N(C)C c1(CN2CCC(c3ncc(COC)[nH]3)CC2)ccc2c(n1)CCC2 c1(OC)cccc(NC(=O)CNCCCN2CCCC2C(=O)N(C)C)c1 C(C)(C(F)(F)C(F)(F)F)=CC(=O)NC1CCN(C(COCC(=O)OC)=O)CC1O N1(C(c2ccc(C(C)=O)cc2F)=O)CC2(C1)SCCC2NC(=O)CCF c1(C(N2C(C)CC(NC(=O)CNC(N)=O)CC2)=O)nn(C)cc1[N+](=O)[O-] C1(C2CCCOC2)(NC(C23CC(CN(C(CCC(=O)NC)=O)C2)C3)=O)CC1 c1(NC(=O)CCC(=O)N2CSCCSC2)ncc2c(n1)CCNC2 C=CCC(C)C(=O)NC(CO)C(C)NC(C1CCN(CC(F)F)CC1)=O N1(C(C2(C(C)NC(C3(CC(=O)OC)CC3)=O)CC2)=O)CCCC(C(N)=O)C1C C=C=CCC(=O)NC(C1(O)CN(C(=O)C(c2cncn2C)O)C1)C C1(CNC(C2(CSC)CCC2)=O)CCN(C(C2CSC2)=O)CC1(F)F C1(NCCCNC(C2OCCN(C(C)C)C2)=O)CCC(F)(F)CC1 C(=O)(C(F)C(=O)N(C(C1CC(N)C1)=O)C1CC1)OCC.C12CCCC1C2 C(=O)(CC(C)(C)C(F)(F)F)NC1CCCC(CNC(C2(C(C)C)COC2)=O)C1 C(=O)(C1c2c[nH]nc2CCC1C)NC1(C(=O)Nc2c(C)ccc(Cl)c2)CC1(C)C C12(C(=O)NC(C(C)NC(=O)C(O)C3CCCC3)CO)CCCN1CCC2 c1(N(C)CC2(SC)CCC2)nc(N2CCC3(CCCO3)C2)c2c(n1)CSC2 CCC(CCC(=O)NC1CC2(CNC2)C1)N(C1CCOC(C)(C)C1)C1CC1 C(CCC(O)C(=O)NCc1cnn(CCO)c1)NC(=O)CCCF CC(C(C)(C)C)=CC(=O)NC1CCC1C(=O)NC1(CC2CC2)CC1 c1(C(=O)NCC(C2C(CC)C2)NC(C(CC=C)C)=O)cc2sc(C)nc2[nH]1 O=C(N=c1ccn(-c2ccc(F)cc2)[nH]1)NCC(c1ccc(F)cc1F)O CCCC(CCC)CC(=O)NC(C)CN(C(=O)C=CC1CCCCC1)CC Cc1ccc(F)c(NC(=O)C(=O)N(C)Cc2cn(-c3ccc(F)c(Br)c3)nn2)c1 C1(NC(C(CC)F)=O)(CO)CCCN(C(c2cc(C)nc(C(F)(F)F)n2)=O)C1 C(=O)(CCCCCN(C)C(C1COCCO1)=O)N1C(CO)CC(OC)C1 N1(C(=O)C=CCN2Cc3ccccc3C2=O)CCCc2c1ccc(Br)c2C c1(C(=O)OC)ccc(C=CC(=O)N(C)CC2CN(C(C3CCCS3)=O)CCO2)o1 O=C(C1=CSCCO1)NCCC1CCCN(C(c2ccc(Cl)[nH]2)=O)C1 N1(C(CCSC)=O)CC2CC(CNC(=O)COc3ccc(Cl)c(C)c3)CC1C2 c1(NC(C2CCN(Cc3c(OC)cccc3)C2)=O)ccc2ncnn2c1 N1(C(C2(CC(C)C)CC2)=O)CC2CC(C(=O)NCCCC3CCOC3)C(C2)C1 c1(CCC(N2CCC(N(C(=O)CCF)CC)C2)=O)ccc(Cl)cc1Cl Nc1ccc(C(=O)NCC(CNC(C2(n3nccn3)CC2)=O)CO)cc1Cl c1(OC)cccnc1C(F)(F)C(=O)OC(c1cccnc1-n1cncn1)=O c1(NS(CC)(=O)=O)cncc(C(=O)NCC2CCN2C(C2C=CS(=O)(=O)C2)=O)c1 c1(C(CC)NC(=O)NC(c2ccc(OC)s2)C)cccc(C)n1 N1(C(CC2CCC(NC(CC=CC)=O)C2)=O)CCC(O)(c2ccccc2C)CC1 C1(O)(CCNC(c2c(C)nc(C)s2)=O)CCCN(C(C2CC(C)N(C)C2)=O)C1 C(C1CCCC1)=C(C)C(=O)NCCC1(CNC(c2cc(CO)[nH]n2)=O)CC1 C1(CNC(C2C(C)CCC2)=O)CC2(CO1)CN(C(=O)Cc1ccc(Cl)nc1)C2 c1(C(N2CCC(CNC(C3(CO)CCC3)=O)C2)=O)csc2cccnc12 C=C1CCN(C(=O)C(C2CCCCCC2)F)C(C(=O)NCC=C2CCSCC2)C1 C1(NC(CC2C(OCC)COCC2)=O)CCCN(C(=O)Cn2cc(C)cn2)CC1 O(NC(=O)COC)CC(=O)N(C(CC)C)CC(C)C Cc1cc(C)c(C(=O)NCCCOCCCNC(C2CN(C)C2)=O)c(C)n1 c1(C(=O)NC(CN(C(c2csc(S)n2)=O)CC)C)cc(Cl)ccc1C(C)C c1(C(=O)NC2CN(C(C(CC)C(C)C)=O)CC2C)c[nH]c2cccc(Cl)c12 c1(CCCC(=O)N(CC(C)(C)CNC(C2CC=CC2)=O)C)cccc(C(F)(F)F)c1 C1(C(=O)NC2(CCOC)CCN(C(=O)NC(C)(C)C)C2)CC2(CC(OC)C2)C1 N1(C(CNC(C)=O)=O)CC2CC2C1C(=O)NC(C(C)(C)O)C1CC1 C1(C(=O)Nc2cn(C)nc2)CN(C(c2ccccc2C#N)=O)CCC1O N1(C(Cc2cccc(C)c2Cl)=O)CCCC2(NC(c3cccc(Cl)n3)=O)CC2C1 CCC(CC)(CCNC(C1CC2(CC(=O)N2)C1)=O)NC(c1cc(C(C)C)[nH]n1)=O c1(-c2cc(C(C)C)no2)nc(CN(C)C)nn1C(C)C1CC1 N1(C(C(CN(C)C)N(C)C)=O)CC(C(=O)NC(c2ccccc2)CO)C(F)(F)C1 CCC(C)(C)C(O)C(=O)NCC(C)(C)CCNC(=O)CCC(F)(F)F Cc1ncnc(C)c1CC(N1CCC(C(C)NC(=O)C=CC2CCOCC2)C1)=O c1(CC(N2CC(O)CC(NC(=O)CC3(CO)CC3)C2)=O)ccc2c(c1)CCCS2 c1(OC)cc(O)ncc1C(=O)NC1CC1NC(c1cccnc1C)=O c1(C(N2CCC(CNC(c3c(C)ncnc3)=O)C2)=O)ncncc1C#N N1(C(Cc2c(C)nc(C)s2)=O)CCn2ncc(CNC(=O)Cn3ncnn3)c2C1 Cc1c(C(=O)NC2(C(=O)N(CCO)CC3CC3)CCN(C)C2)cccc1F c1(SC(C(=O)NC2C(NC(c3n(CC)nnc3)=O)COC2)C)ccc(F)c(F)c1 N1(C(C2C(C(C)C)OCC2)=O)CC2CCCC2(NC(C2CN3CCC2CC3)=O)C1 C1(c2n(C(CC)(C)C)nnn2)(Nc2cccnc2OC)CCCC(OC)C1 CC1CCN(C(=O)CC(F)(F)Cl)CC1CNC(=O)CCc1cccnc1Cl C1(C(=O)NC2CCC2NC(c2cc(Cl)ccn2)=O)(OC)CS(=O)(=O)C1 Cc1ccc(-c2noc(C(C)CCC3CCCOC3)n2)cc1Cl N1(C(c2cc(OCC)no2)=O)CCC(C(C)CNC(C2COC(=O)N2)=O)CC1 C1(C(N2CC(C(C)NC(C3(C(F)F)CC3)=O)C2)=O)CC(C)(C)CO1 c1(OC)nc(Cl)ccc1C(N1CCN(C(c2ccc(C(F)F)cn2)=O)C2CC12)=O Cc1cc(C(=O)NC2CCN(C(=O)C3=NOC(C)C3)CC2O)cc(F)c1 C12(NC(C3CCN(c4nc(CC)nc(C)c4)C3)=O)C3C4C1C1C2C3C41C(=O)OC C12=CCNC(=O)N(C1)C2=O.C1(C)CCNC(=O)N1.C(C)(C)(C)OC.C(C)(C)S N1(C(CCSCC)=O)CC2CC(NC(c3ccc(N(C)C(C)C)cc3)=O)C2C1 C1(c2n(C)ccn2)CN(C(C2(C)CCCOC2)=O)CC1NC(=O)C(Cl)=CCl CC1CN(C(=O)CCOC2CCOCC2)CC(C)CN1C(=O)C(F)C(F)(F)F C(=O)(C(C)(C)CC(F)(F)F)N(C1CC(NC(=O)C(c2cccn2C)=O)C1)C C#CCCN=C(NCC(C)(C)C(F)(F)F)NCC1CC(O)C12CCC2 N1(C(C2N(C(C(CC(=C)C)OC)=O)CC2)=O)CC2CCCC(C1)N2C C1(NC(C2(COC)CCOCC2)=O)CCN(c2ncc(Cl)cn2)CC(C)(C)C1 C1(CC(=O)NCC2CN(CCC)C2)CCCN1C(=O)CCc1cc(C)no1 N1(C(Cc2ccn(C)n2)=O)CCC(NC(=O)Cn2nccn2)C12CCCC2 C(=O)(CC(C)(O)C(F)(F)F)NCCN(C(c1c(C)cccc1Cl)=O)CC1CC1 C=CC(Cc1nc(-c2ccc(SC)cc2)nn1C(CC)CC)CCC CCCCCCC(O)CCC(=O)N(CC(C)NC(c1ccn(CC)c1C)=O)C C(=O)(C1=CCC(C(F)(F)F)OC1)NCCCC(C)(C)NC(=O)CC1CC2CC2C1 C1(NC(C=CCCC)=O)CCC2CN(C(C3(F)CCS(=O)(=O)C3)=O)CCC2C1 c1(C(=O)OCC2CC2C(F)F)cc(O)nc(Cl)n1 C1(C(=O)NC(C(N2CC(C#CC)C2)=O)c2cccs2)CCC(=O)N(C)C1 C1(CCNC(C(=O)NC(C)C)=O)CCCN(C(=O)CCN2CCC(F)C2)C1 C1(N(CCOC)CC)CCN(C(=O)C(Cl)=CCl)CC1.C1(C=O)CCOC1 N1(C(c2nc(C)oc2C)=O)CCC2(CC1)CCN(C(=O)COc1ccccn1)C2 N1(C(C(CC)F)=O)CCCC(NC(=O)C(C)(C)NC(=O)COC(C)(C)C)C1 C=CCN=C(NCC1(C)CCC1)N1CCC(OCC(=O)NC)CC1 C(CN=c1nc2n([nH]1)CCCC2)N(C)C(C1CCN(Cc2ccccc2)C1)=O C1(COC)(NC(c2[nH]nnc2C)=O)CCN(C(c2cc[nH]c2)=O)CC1 N1(C(c2c(C(C)C)con2)=O)CC2OCC(NC(C3(Br)CC3)=O)C2C1 N1(C(C=CC)=O)CCC(C(C)(O)CN(C(=O)CCc2ccc(C(C)=O)[nH]2)CC)CC1 N1(C(c2n(CC)ccc2)=O)CCCC(N(C)C(c2sc(C(C)C)nc2C)=O)C1 N1(C(COCC#C)=O)CCC(N(C)C(C2CC(c3ncc[nH]3)C2)=O)C1 Nc1cc(Cl)cc(Cl)c1C(=O)NC1CCN(C(C2CC3C=CC2C3)=O)CC1 Cc1c(CCC(=O)NC(C)C(=O)Nc2cccc(OC(C)C)c2)sc2ccccc12 C(=O)(CCCC(C)(C)NC(C1CC(F)CN1C)=O)NC1C2(CC(OCC)C2)C1 c1(N2CCC(C)C2)cc(C(=O)NC2CC(NC(=O)C=CC3CCC3)C2)ccn1 Cc1ccc(C2(C(N3CCOCC(NC(=O)C(O)C(C)(C)C)C3)=O)CC2)c(C)c1 c1(OC(CC)C)cc(NC2CC2C(=O)NCC23CCCC2C3(F)F)nc(C)n1 C(F)(C(=O)Nn1cccn1)C1N(C(CCC=CC(C)C)=O)C2C1CCC2 N1(C(C(c2c(C)cccc2Br)NC(CCC=C)=O)=O)CCOCCC1C c1(NC(C2(OC)CCN(C(=O)C3=CCCCC3)C2)=O)cnc(C)c(C)c1 C1(OCC)(CNC(C2(CCNC(=O)CCOC)CC2)=O)CCCCCC1 c1(OC)noc(C(=O)NCC2(C)CCCN2C(=O)C(C)C2CC2)c1Br S(=O)(=O)(c1cccc(C)n1)N1CC2C(N(C(c3cccnc3)=O)CC)C(CC2)C1 C1(C(=O)NCC2(CO)CCN(C(C3CC(F)C3)=O)C2)OCC2COCCC12 C1(N(CC#C)C(C2CCCC2C)=O)CCN(C(c2ccc(Cl)o2)=O)CC1 C1(SC)CN(C(c2cccc(C)c2)=O)CC1NC(=O)C(C1(O)CCCCC1)(F)F c1(C(N2CCCCC(CNC(CC3C(C)(C)C3)=O)C2)=O)c(F)ccc(N)c1F c1(C(=O)NC(CCCC)CNC(=O)C(C)(C)COCC)ncc([N+](=O)[O-])n1C N1(C(c2cnc(C)n2C)=O)CCC2(CCCC2NC(=O)COC2CCC2)C1 c1(NC(N(CCC#C)CCOC)=O)csc(C)c1CSC c1(CC(=O)NC2CCC2C(F)(F)F)cnn(CCNC(=O)CC2CC3CC3C2)c1 c1(C(=O)N(c2ccnc(Br)n2)CC2(O)CNC2)cc(Br)cc(F)c1F C1(COC)(CNC(=O)CCCN(C)C)CCCN(C(=O)CNC(=O)CN(C)C)C1 C12(C(N3CCC(OC)(CNC(=O)Cn4cc(Cl)cn4)C3)=O)CC1COC21CCC1 C1(C(=O)NC(CC(C)NC(C23CC(C)(C2)C3)=O)C)CC(=O)OC1(C)C c1(C(N2CC(CCNC(CC3C(C)CC3)=O)C2)=O)csc(C(C)(C)C)c1 c1(NC(CC(C)Oc2ccccc2)=O)cc2c3c(c1)CCC(=O)N3CCC2 Cc1ccc(-c2cn(CC3OCCC3C(=O)NC(C)(C)C(C)O)nn2)cc1 CC1C(=O)Nc2ncccc2N1C(C1CC2(C1)C(C(=O)O)C21CCC1)=O Cc1ccc(C(N2CCCC(O)(CN(C)C(C3CC3CF)=O)C2)=O)c(F)c1C N1(C(c2cnc(C#N)s2)=O)CCC(NC(c2ccc(NC=O)cc2)=O)C(CO)C1 N1(C(C2C(=C)CC2)=O)CC(C)(C)CCC1CNC(c1ccc(C(C)C)c(C)c1)=O C1(CNC(c2n[nH]c(C)c2O)=O)N(C(=O)CC2CC=CCN2C)CCCC1(C)C C1(CNC(CC2CCC(C)(C)CO2)=O)CCCCC1N=c1[nH]c2cc(Cl)ccc2s1 C1(C(N2CCCC(OCCOC)C2)=O)Cc2cccc(Cl)c2C(=O)O1 c1(N(C)CC2CC2)ccc(S(=O)(=O)NCC2COC(C)(C)CN2)cc1Br CCC(CC)CCC(=O)NC1(CCCNC(C2CCCSC2)=O)CC1 N1(C(COCCOC)=O)CC(CNC(=O)CNc2ccccc2C)CCC1C C(C)(C)(CC(C)NC(C1(C)CN(C(c2ccn(C)n2)=O)C1)=O)OC C#CC1(C)CCN(C(C2CCC(C3CC3)N2C(=O)C=Cc2cocn2)=O)CC1 c1(C(=O)NC)cc2c(s1)C1(CCN(C(c3cc[nH]n3)C)CC1)OCC2 CC1CCN(C(=O)C=CC(C)(C)C)CCN1C(=O)COCCO CCCN=C(NCCC(C)(C)COC)NCc1cc(Cl)ccc1O c1(NC(C2CCN(C(c3cncc(Br)c3)=O)C2)=O)ccc(Br)cc1[N+](=O)[O-] N1(C(CC2C(SC)CCC2)=O)CCC(C)(Cn2cc(Cc3ccccc3)nn2)C1 C=C(C)CC(C(=O)N1CC(CCCCNC(C2COCC2O)=O)C1)NC(C)=O C1(CNC(c2onc(OCC)n2)=O)(NC(c2sccc2OC)=O)CCCCC1 C(C1=NOC2CN(C(c3cnc(O)cc3O)=O)CC12)NC(c1ccc(F)nc1)=O N1(C(CC(CC#C)NC(c2cc[nH]c(=NC)c2)=O)=O)CCCC(C)(C)C1C C1(NC(CCN(CCCCOC)C)=O)CCN(C(c2c[nH]cc2C2CC2)=O)C1 N1(C(CN(C)C(=O)C2CC2)=O)CC2CCCC1(CNC(c1ccoc1Cl)=O)C2 C=C(C)CCC(=O)NC(C1(O)CCN(C(c2ccc(NC3CC3)nc2)=O)C1)C c1(C(N2CCCC(C3CCCN3C(c3ncc(F)cn3)=O)C2)=O)nc(Cl)c(Cl)s1 c1(OC)ccc(C(=O)NC(CNC(=O)CC2CCCCO2)C(C)(C)C)nc1 c1(C(=O)NC2C(CNC(CC(C)c3cnn(C)c3)=O)CC2)cc2cnccc2o1 C(CC1=CCN(C(=O)CSc2c(C)n[nH]c2C)CC1)NC(C(C=C=C)C)=O C1(NC(C(C2CC2)SC)=O)CC2CC1N(C(c1cnc(C3CCOCC3)s1)=O)C2 C1(OC)CC(NC(=O)CSc2nc[nH]n2)CN(C(C23CC4CC2C3C4O)=O)C1 CCC(CC(=O)NCC1CCCO1)C1CCC1.C1(C(=O)NC)(NS(C)(=O)=O)CC1 N1(C(CCOCC#C)=O)CCC2(CCCC2N2Cc3ccccc3C2)CC1 c1(NC(C2(C)CCCN(C(CSCC=C)=O)C2)=O)cc(C)c(O)c(C)c1 c1(C(=O)NC(CNC(C=C(C)C(C)C)=O)C(C)C)ccc(Cl)c(C)c1O CC1OC2(CO)CC1(NC(=O)NCC1CCCC1(C)c1ccccc1)C2 C(CC)(CC)(CCNC(=O)C=Cc1cnc[nH]1)NC(C1CC(CCC)C1)=O N1(C(C=CC2(C)CCOCC2)=O)CCC2(CC1)CC(NC(=O)C1=CCC1)CCO2 c1(-c2cnc(C3CN(C(=O)CCc4nc(O)n[nH]4)C3)o2)ccc2c(c1)OCO2 c1(NC(C#CCNC(c2cc(CC)nn2C)=O)=O)cc(C)c(F)cc1C N1(C(CCOCCOCC)=O)C2CCC(NC(C3(OC(C)=O)CC3)=O)C1CC2 C1(CCC(=O)NCCCN2CCC2)CCCCN1C(=O)C(F)(F)F c1(C(C)NC(=O)NCC(c2cncn2C)O)ccccc1N1CCCC1 Nc1cc(C(=O)NCC2(NC(C3CC4(CC4)CO3)=O)CCOCC2)c(F)cc1F N(C1CCCn2cnnc21)c1c(C)c(N2CCCC(C)CC2)ncn1 C(CS(=O)(=O)C1CC1)NC(C1CC(C)(O)C1)C N1(C(Cc2c(C)n(C)cn2)=O)CC2(C=C(C(=O)N3CC=C(CO)CC3)CO2)C1 C(C(C)(C)C#CC(=O)NCc1cnsc1)NC(C=CC1N(C)CCC1)=O C1(OC)CN(C(=O)C(C)O)CCC1NC(C1CC(n2cnnc2)C1)=O C1(C(N2C(C(C)NC(=O)Cc3cc(C(F)F)no3)CCC2)=O)C(C)(C)C1(C)C C(CN=c1[nH]c(=NCc2ncccc2N(C)C)c(C)c(C)[nH]1)c1ncc(C)o1 CCC(C)CC(=O)C(=O)NCC1(CC(=O)N(C)Cc2c[nH]nc2C)CC1 N1(C(CCSC)=O)CC2CCN(C(c3cn(C(F)(F)CO)nn3)=O)C2C1 O(N1CCC(CC(=O)NCC2CN(C(=O)Cc3nocc3C)CCO2)CC1)CC c1(C(=O)NC2CC3CN(C(C(CC)OC(C)C)=O)C2C3)[nH]c2ccccc2c1Cl C=CCCC(C(=O)NCCCC(=C)Cl)NC(C1CC(C(C)C)C1)=O C1(C(=O)OC)(NC(=O)OC(C)(C)C)CCCN(C(=O)COC(F)(F)CF)C1 c1(-c2c(C)cc(O)cc2)nc2c(s1)CCN(Cc1cccc(N3CCCC3)c1)C2 CC(C(=O)NCC1CCN(C(c2cnn(CC3CC3)c2)=O)C1(C)C)C(F)(F)F c1(CN(C2(C(=O)OC)CC2)C)cccc(C2(C)CC2(F)F)c1 C1(C(=O)NCC2CCCC(F)C2)(NC(C2CS(=O)C2)=O)CCOCC1 C12(C(N3CCCC(NC(c4cnc(C(C)(F)F)s4)=O)C3)=O)CC1COC2(C)C O(NC(=O)C1=CCC(NC(C23CCN(CC2)CC3)=O)C1)CCC=C N1(C(c2ccn(C(C)C)n2)=O)CC2CCN(S(=O)(=O)c3cnn(C)c3)C2C1 c1(C(=O)NC2(CNC(C3CC(O)C(F)C3)=O)CCC2)n[nH]c2c1CCCCC2 C#Cc1ccc(C(=O)NC2CN(C(=O)Cc3ccsc3Cl)CCC2CO)c(F)c1 Cn1nc(CNC(C2(NC(=O)CN3CCNC3=O)CSC2)=O)oc1=O C(C)(C)(CCC(=O)NCC(C)(C)OCCNC(C1(C)CC1F)=O)OC N1(C(C(C)C#N)=O)CCC(C)(NC(=O)C(CO)c2ccccc2)CC1 C(C(C)(C)CC(=O)N1CCN(C(c2ccc(Cl)[nH]2)=O)C(CCO)C1)OC(C)=O CCCCC(C)(F)C(=O)N1CCCOC(CNC(c2cccc(C3CC3)c2)=O)C1 c1(NC(C(CNC(c2cnc(C)nc2)=O)OC)=O)cnc2[nH]ncc2c1 C(O)(C(=O)N1CCCc2nccn21)C1CN(C(C2N(C)CCOC2)=O)C1 C#Cc1ccc(OCC(=O)NCCCCCNC(=O)CCC(=C)Cl)cc1 C1(NC(C(Br)=C(C)C)=O)C2CC1N(C(C1(OC(C)=O)CCOCC1)=O)C2 c1(CN(C(=O)C)C)cccc2ncccc12.c1(CC)cccnc1.N1COCC1=O C1(C(N)=O)C2CCC(C2)N1C(=O)CN1CCN(C(c2ccoc2Cl)=O)CC1 C(=O)(C1=NN(C)C(=O)CC1)NC(CCCC(=O)Nc1c(C)cc(F)nc1)C C1(C(=O)NC2CCC(F)(F)C2)CCCCCN1CC1COCCN1CC1CCCC1 C1(CC(=O)NC(C2(O)CN(C(=O)CN(C)C3CC3)C2)C)CCC(=O)N1 Cc1cc(C)n(CCC(=O)NCCN(C(c2cnc(C(C)O)s2)=O)C(C)C)n1 c1(C(N(CCCN(C(Cc2ccn(CC)n2)=O)C)C)=O)cccc(C(C)(F)F)n1 c1(C(N(C2CCN(C(=O)CS(N)(=O)=O)C2)CCC)=O)ccc(C#N)c(C)n1 c1(C(C(=O)NC2COC2)N(CC(=O)OC)C)ccc2c(c1)CC(C)(C)O2 O=C(CS(=O)(=O)C1CCCC1)NC1COCCC1NC(C1(CCF)CC1)=O c1(OC)ncc(CN(C(c2nc(Cl)cs2)C(=O)NCCCF)C)cc1C c1(C(=O)NCC(CC)NC(C2(CC)CCC2)=O)csc(Cc2ccccn2)n1 c1(C(=O)NCC(C)(CO)NC(c2cn[nH]c2)=O)ccc(CCF)cc1 C=C(Br)CC(C)(C)C(=O)N1C2CCC1CC(NC(c1ccc(N)c(F)c1)=O)C2 C1(CNC(C2C(OC)CCCC2)=O)CC(N=c2ccc3nnnn3[nH]2)C1 C1(NC(C(C)C)=O)CCN(CCCc2ccccc2)CC1C C#CCC(C)(C(=O)N1CCCC(NC(C)=O)CC1)NC(c1cccc(O)c1)=O N#Cc1ccc(=NCC2(O)CCN(C(C3CC4CCCCN4C3)=O)CC2)[nH]n1 c1(N(C(CCSCC(=O)OC)=O)C)cc(Br)ccc1[N+](=O)[O-] C1(NC(CC=C)=O)CC2CCC1C(NC(C1(O)CCCC(C)CC1)=O)C2 C1(C(=O)NC(C(=O)NCc2cc(C)ncc2)CCF)Cc2ccccc2C1 C1(NC(C2CC(OC)(OC)C2)=O)CC(NC(c2cccc(CC#N)c2)=O)C(O)C1 c1(C2(NC3CCCN(C(C4(SC)CC4)=O)C3)CCCC2)ccc(F)cc1F Cc1cc(CN(C(=O)C(CN(C)C)NC(=O)Cc2ccc[nH]2)C)no1 C(=O)(C(C)(C)C1=CCN(C(=O)CC(C)(C)C(C)(C)C)C1)NC1(CC)CCOC1 c1(CC)nc(O)c(C(N2CC3CC2C3CNC(c2ccsc2C)=O)=O)cc1C N1(C(C(n2cc(C3(C(=O)O)CCCCC3)nn2)C)=O)CCC(C2CC2(F)F)CC1 C(C(N=[N+]=[N-])C(=O)N1CCCC(C(=O)NCc2ncnn2C(C)C)C1)OCC C(=O)(C(C)CC(F)(F)F)N1CCC(C(=O)NCC(C)(C)CO)(SC)C1 C(c1ccncn1)=CC(=O)NCCCCC1CN(C(c2ccco2)=O)C1 c1(C(N(CCC)CCNC(=O)Cc2ccc(C)c(Cl)c2)=O)cccc2c1CCC2 C(CN=C(NCC1(N2CCCC2)CCCC1)NC1CCCC1)OCCC=C C(CC(O)CC(=O)NN1C(C)CCCC1C)c1ccc(C)cc1 C(CO)(CCCNC(=O)C1=NOCC1)NC(C=CCN(C)CC)=O CC1CCC(NC(=O)COc2ccccc2)CN1C(C1CC1(F)F)=O C1(C(=O)NCCNC(c2c(CC)c[nH]n2)=O)CC(c2ccncc2)=NO1 C12(C(=O)NC3C(O)CCN(C(C(CC)CC)=O)C3)CC3CC(C)(C1)CC(F)(C3)C2 Cc1ccc(CN2CCCC2CC(=O)NC(c2ccco2)CO)cn1 Cc1ccnc(C(N2CCC(F)C(NC(=O)C(C)(C)CC#N)C2)=O)c1Br N1(C(Cc2cc(C)[nH]n2)=O)CC(C(=O)NCC2CCC(C3CC3)O2)CCC1C N1(C(CCCOCC=C)=O)CCC2(CCN(C(C3(N(C)C)CC3)=O)CC2)C1 C(=O)(C(C)C(F)(F)F)NC12CN(C(C3(C)CC(OC)(OC)C3)=O)C(C1)C2 C1(CNC(C(C2CN(C(=O)Cn3ncccc3=O)C2)OC)=O)CCC(C)(C)O1 CN1CC(C)(C(N2CC(O)CC2CNC(=O)CC2(C)CCCC2)=O)CCC1=O n1(CC)nc(C)c(CC(N2CCOC(CNC(C3CC4CC4C3)=O)C2)=O)c1C C1(C)(C(N(CC#C)C)=O)CC(O)CN1C(c1ccc(NC)cc1)=O CC1=C(C(=O)N2CCN(C(=O)CCc3ccoc3)CC2C)CCCC1 C1(CC(=O)NC2(CF)CCN(C(c3cocn3)=O)C2)CCCC1(F)F c1(C(=O)NCC(CN(C(=O)CC(C)(C)OC)CC)(C)C)c(F)ccc(C)c1F N1(C(C(CC)CCOC)=O)CCC(C2(NC(c3cncc(Cl)n3)=O)CCC2)CC1 c1(NC(C(CC)N(C(C2CCC(C)C2)C=O)CCC)=O)cccc(Cl)c1C C1(C2CN(C(=O)C=C3CCC3)C2)(NC(c2cccc(C)n2)=O)CC1 C1(CNC(C(C)(C)N2CCOCC2)=O)CCCN(C(c2ccoc2)=O)C1 NS(=O)(=O)CC(=O)NC1COCC1NC(=O)C(C1CC(F)(F)C1)N1CCCC1 C1(CC(C)NC(C(C)CC2CC2)=O)CCN(C(C23CC(C)(CO2)C3)=O)CC1 C1(n2cc(C(C)(C)SC)nn2)CN(C(c2scnc2C(F)F)=O)CC1C1CC1 C1(NC(c2c(CC)sc(=N)[nH]2)=O)COCCN(C(c2oncc2C)=O)C1 N1(C(c2[nH]c(=NCC)sc2)=O)CC2CN(C(=O)C(n3nccc3C)C)CC2(C)C1 C(=O)(C(C)CC(C)(C)C)N1CCC(OCC(=O)N(C)Cc2c(C)ccs2)C1 c1(CNC(C(n2ccc(C)n2)C)=O)nnn(C)c1C(=O)NCC(C)OCCO N1(C(C2OCC(C)(C)OC2)=O)CCOC2C1CCN(C(=O)CCn1ccnc1)C2 c1nccc2c(Br)cccc12.N1(C(C)C)CCC(N(C)C)C1 C1(C(=O)NCC2CN(C(c3ccoc3)=O)CCO2)CCC2CCCCN12 C1(CNC(C=CC(C)C)=O)CCC2(CCN(C(=O)CN=S(C)(C)=O)CC2)O1 c1(C(=O)NCC2CCN(C(C3(C4CCC4)CC3)=O)C2)cc2nc[nH]c2cn1 N1(C(CCCC#C)=O)CC2(NC(c3cc(=O)c(OC)co3)=O)CCC1CC2 C1(NC(c2cc(C)sc2)=O)CC12CCN(C(c1cc(-c3cccs3)[nH]n1)=O)CC2 C(=O)(NN1CCCC1C(=O)NCC1CCNC(=O)C1)c1nc(=N)[nH]cc1 CC1(C)CC(NC(C2CC(F)C2)=O)CN1C(C1CCC1)=O C(C)(CNC(=O)CCc1ccccn1)(C(C)C)NC(c1c(OC)csc1)=O Cc1nsc(N2CCC(C(C)(C)NC(c3cn(CCO)nn3)=O)CC2)c1C#N CC1CCC(CCC(=O)N2CCC2CNC(=O)CNS(N)(=O)=O)O1 c1(C(=O)Nc2cn(C(C(N3CC(C#N)(SC)C3)=O)C)nn2)ccc(C#N)c(C)c1 C1(C(N2C(CC)CC2)=O)CN(C(=O)CCc2ccccn2)Cc2nccn2C1 CCC(CC)(CO)C(=O)N1CC(CC(C)NC(C2CCCC2SC)=O)C1 c1(SC(C(=O)OCC(=O)OCC)c2nc[nH]n2)nncn1CCc1ccccc1 CC(C)(C)C(CN=c1ccnc(Cl)[nH]1)NC(C1CC(F)C1)=O N1(C(CC2(N(C)C)CC2)=O)CC2(C1)SCCC2NC(C1CC2C=CC1CC2)=O C1(C(=O)OC)CC(C)N1C(=O)C(c1cn(C)nn1)NC(=O)C=Cc1cc[nH]n1 c1(C(N(CCCN(C)C(c2scnc2C2CC2)=O)C)=O)cccc2ccoc12 c1(CC(N2CC(NC(=O)CCCn3ccnc3)C(F)C2)=O)c(F)cccc1Cl C1(CNC(COC2CN(C(C)=O)C2)=O)CCCN(C(C2CC(C)(C)CO2)=O)C1 N1(C(CC(=C)C)=O)CCCC(CO)(NC(=O)COc2ccc(C(F)(F)F)nc2)C1 Cn1nc2c(c1NCC(=O)NCc1ccc(S(C)(=O)=O)cc1)CCCC2 c1(CC)cc(C(=O)NC(CNC(C2(F)CC2c2ccccc2)=O)CC)n(C)n1 C1(NC(=O)OC(C)(C)C)CN(c2ncc3ccccn23)CC2(CC2)C1 c1(OC)c(Cl)cc(C(=O)N(C)CC2CCCN2C(c2cnncc2C)=O)nc1Cl c1(C(=O)OCC)cc(CN(c2cc(SC)ncn2)C2CCC(N)C2)ccn1 CC1(C)CC(C(=O)NC2CCC(=O)NC2)CN1C(c1cn[nH]c1)=O C1(C(=O)NCC=NOC)CCCN1NC(=O)C1(CO)CC1 CC1CN(C(c2cnc(C3CC3)nc2)=O)CC1CCNC(c1cc(C#N)c[nH]1)=O N1(C(c2cnc(CC)[nH]2)=O)CC(CN(C)C(C2CC(=O)N(C)C2)=O)C2(CC2)C1 C(=O)(C(O)CCC(C)C)NC1CCN(C(c2c(C)ccc(SC)c2)=O)C1 C1(C(N(CCCNC(CCc2nc(C)sc2)=O)C(C)C)=O)CC2CCCC2C1 Cc1c(Br)ccc(C(=O)Nc2nc(CC(=O)Nc3nccnc3Cl)cs2)c1C c1(CC)cccc(-c2cn(CC(C)NC(C3CCOC3C)=O)nn2)c1 c12ccc(cc1)C(=O)NCCN2CCO.C1(CC(=O)NS(C)(=O)=O)CCCSC1 C(=O)(C(O)CC(C)(C)C)N(CC(CNC(C(C)(C)N(C)C)=O)O)C.CC(=O)O N1(C(CCC(=O)c2cccnc2)=O)CC2(CCN(C(C3CC3C3CC3)=O)C2)C1 C(=O)(C(C)CC(C)C(C)=O)NC(c1nc(C(=O)NC(C)CC2CC2)co1)C c1(SCC(=O)NC(C2CN(C(C(C=CC)O)=O)C2)C)cc(F)ccc1F CCCC(CO)NC(C1CC(C)(NC(c2c[nH]nc2OC)=O)C1)=O N1(C(C)C)CC(C(=O)N(C)CC2(NC(c3cncs3)=O)CC2)CC1=O N1(C(C2CC(C)NC(=O)C2)=O)CC2CCN(C(c3ccc4ccsc4c3)=O)CC12 C1(CCO)CN(CC)CCCO1.c1(CC(O)OC)cn(CCC(=O)NCC)nn1 N1(C(C2(C)N(C)CCC2)=O)CCCC2CN(C(c3ccnnc3O)=O)CC12 N1(C(CC(c2cccs2)O)=O)CCC2(C1)CN(C(=O)CCN1CCCCC1)C2 N1(C(C(CC)n2cncn2)=O)CCN(C(=O)C=CCN(CC)CC)C(CO)C1 c1(C(=O)NC(CC)(C)CNC(=O)C(F)OC(F)(F)F)cc(F)cc(N)c1F N1(C(C2C(C)(C)COCC2)=O)CCCC12CCN(C(c1ncccc1Cl)=O)C2 n1(CC)ncc(C(=O)NC2CC(NC(=O)C(C)CCOC)C2)c1Br CC1(C#N)CN(C(=O)CCC2CCCN(C(C3(C)CCCO3)=O)C2)C1 N1(C(CC(CC)C)=O)CC2(COC(CNC(c3nnn(C(C)C)c3C)=O)C2)C1 c1(C(=O)NC(CNC(c2cc(C)c(O)nc2)=O)C)ccc2nccn2c1 C(=O)(C(F)C(C)(C)O)NC1C(NC(Cc2cccc(COC)c2)=O)CCCC1 C1(C(N(C2CCCN(C(=O)C(C)=C3CC3)C2)CC)=O)CC2CCC(C1)C2O C1(C(C)(C)NC(C=CSC)=O)CCN(C(c2coc(O)n2)=O)CC1 CCCCC(C(=O)NCC(CC)(CC)NC(=O)Cc1cccs1)NC(N)=O C(CC(=O)Nc1ccc(F)c(C)c1)(C(C)C)NC(c1ncn(CC)n1)=O c1(C(=O)NCCCN(C(c2cn(CC=C)nc2)=O)C2CC2)ccc2c(c1)CC2 C1(C(N2CCN(C(C(C)=C3CCC3)=O)CC23CC3)=O)CCn2c(cnc2C)C1 c1(OC)cc(OC)c(C(N2CCC(CNC(=O)C(C)C(F)F)C2)=O)cc1OC C1(C(N2CC(NC(C(C)=CC)=O)CC(C)(C)C2)=O)CCc2c(n[nH]c2C)C1 C(=O)(C1=CS(=O)CCC1)N1CC(CCC)OCC1 c1(C(=O)NCCN(C(c2ncn(C(C)(C)C)n2)=O)CC2CC2)ccc(CF)cc1 C(CC(C)C(=O)N(CC(O)CN(C)C(C1CC(=O)C1(C)C)=O)C)OC c12cc(OC)c(O)c(c1)CN(CCCO)C1CN(C1)C2=O.CCC(=O)OC c1(OC(C(=O)NCCN(C(CCOCC#C)=O)CC)C)ccc(COC)cc1 Clc1ccc2c(c1)CN(Cc1cccc3ccccc13)C2 N1(C(C2N(CC)CCC2)=O)CCC2C(CCN2C(c2ccc(F)cc2)=O)C1 c1(COC)ccc(C(=O)N(CC(C)NC(=O)C(C#N)c2ccccc2)C)[nH]1 c1(NC(C2N(C(c3cnn(C)n3)=O)CCOC2)=O)cccc2c1CCO2 c1(CC)cc(F)ccc1C(=O)N(C1CCC(NC(=O)C2=CC(C)(C)C2)CC1)C N1(C(C2C(CC(C)C)C2)=O)CC(CNC(=O)CCC(=O)c2cnn(C)c2)C(C)C1 C1(C(N(C)Cc2cc(C)on2)=O)CCCCN(C(c2cnc[nH]c2=N)=O)C1 CCC(N=c1[nH]c2c(c(=NC(C)C)[nH]1)COC2)C1CCCOC1 N1(C(COCCCC(C)C)=O)CC(NC(C2(CCN(C)C)CC2)=O)C2CC12 Cc1cc(=NCC2(C)CCCN(C(c3csc4cccnc34)=O)C2)[nH]c(C)n1 c1(OC)nc(Cl)ccc1CONC(C1CC2C=CC1O2)=O c1(NS(C)(=O)=O)cccc(C(=O)NC2CN(C(=O)Cn3cnnc3)C2)n1 Cc1nsc(C)c1C(=O)NCC1CC1NC(c1ccnc(-n2ccnc2)c1)=O c1(C(=O)NC2CCN(C(CCC3N(C)CCCC3)=O)C2)cnc2c(c1)CCCO2 C1(C(C)C)N(C(c2ccc(C#N)[nH]2)=O)CC12CCN(C(=O)C(F)C1CCC1)CC2 C(CCN=c1[nH]cnc2ccc(O)cc12)NC(c1cc2c([nH]1)CCC2)=O c1(SC)ccc(C(=O)NCCC2CN(C(=O)Cc3cc[nH]n3)CC2C)c(Cl)c1 C1(CNC(C(CC=C)OC)=O)CCN(C(C2COCCN2C)=O)CC1(F)F c1(OCC(=O)NC2(CNC(CCC(=O)N(C)C)=O)CC2)cc(C)ccc1C(F)F.C C12(C(=O)NC3CC(CNC(COCCCCC)=O)C3)CCCN(CC1)C2 C1(NC(c2ncc(Cl)s2)=O)CCN(C(C2(c3ccc(F)cn3)CC2)=O)C12CCC2 C#Cc1cncc(C(=O)NC2CCCC(NC(c3cc(C4CC4)n(C)n3)=O)C2)c1 CC1(C)CCCOC1CNC(C12CC(F)C1C2)=O CC(C)(C)CC(O)C(=O)NCC(C)(C)NC(=O)CCOc1ccccc1 Cc1[nH]c(C)c(C(N2CCCC2CCC(N2CC(F)C(F)C2)=O)=O)c1C CC(C)CCCC(=O)NCC1COCCN1C(=O)CCc1ccc(O)c(Cl)c1 CCC(CC(=O)N1CC(NC(C)=O)C(n2cc(-c3n[nH]c(C)c3C)nn2)C1)SC CCC(CCN(C)CC1(O)CC2CCC1O2)C(=O)OCC(F)(F)C(F)F C1(NC(C2(NC(C(C(C)C)O)=O)CCN(C)C2)=O)CC2(COCCO2)C1 C1(N(C(c2ncn(C)n2)=O)CC)CCN(C(=O)CCC2CCC(C)O2)CC1 CC1C(NC(=O)C(C)(C)c2cccs2)CCCN1C(c1csc(C2CC2)n1)=O c1(NC(c2c(CC)c(F)ccc2)=O)cnc2cccnc2c1 C1(C(N2CCC(N(C(c3c(C)ccnn3)=O)C)CC2)=O)CN2CCC1(C)C2 N1(C(C2(C)CCCCC2)=O)CC(NC(=O)COCC2CCC2)CC(O)C1 O=C1CS(=O)(=O)CC(C(=O)NC2CC3(CCN(C(c4cncs4)=O)C3)C2)N1 N1(C(CNC(N)=O)=O)CC(NC(c2c[nH]nc2-c2ccco2)=O)C(O)C1 c1(C(=O)Nc2ccc(-c3ccncc3)cc2)cccc2ncnc(O)c12 C(=O)(CC(C)CC(F)(F)F)NCC1N(C(C(C(C)C)F)=O)CCC1 N1(C(C2OCCN(C(c3c(C)ccc(O)c3)=O)CC2)=O)CC2(CNC(=O)N2)C1 C1(C(=O)NC2CCCC(C)CC2)CN(CCNS(C)(=O)=O)CC(C)(C)O1 C1(C(=O)NCC2CN(C(c3[nH]cc(CC)c3)=O)C2)CCCCC(F)(F)C1 c1(NCC2(CCC=C)CC2)ccc(S(=O)(=O)NC2CCN(C)C2)cc1Cl c1(C(N(CC(C(=O)NC(c2cnn[nH]2)C)(C)C)C)=O)cn(C)c(=O)cn1 CC1CN(C(=O)OC(C)(C)C)CCCN1C(C1CCN(c2nc(=N)[nH][nH]2)C1)=O c1(NCCOCCC)ncnc(NCCN2CCCCCC2=O)c1C N1(C(c2c(CC)ccs2)=O)CC2CN(C(c3cc(F)cc(F)c3O)=O)CCC12 O=C(CCCNC(C12COCC1C2)=O)NCc1ocnc1C1CC1 Cc1ncn2ccc(C(N3CCC(N(CCO)C(C4CC=CC4)=O)CC3)=O)cc12 N1(C(CC2(O)CCCN(C)C2)=O)CCC(C2CCN(C(c3ccsn3)=O)C2)CC1 c1(C(N2C3CN(C(=O)CC4CCCC4)C(C3)C2)=O)onc2ccccc12 c1(NC(C=COc2ccc(OCC)cc2)=O)ccc(C(F)(F)F)cc1OC c1(C(=O)NCC(CNC(c2cc(C3CC3)ccc2F)=O)CO)cc(O)nc(Cl)c1 c1(N2CCN(C(C3C(C)OCCC3)=O)CC2C)cc(C(C)=O)c([N+](=O)[O-])cn1 CC1C(NC(C2Cc3ccccc3O2)=O)CC2CCC1N2c1ncc(Cl)cn1 c1(C(N(CC(C)(C)NC(C(C)=C2CC2)=O)C)=O)cc(S(=O)(=O)CC#N)ccc1F C1(CC)CN(C(C2C3(CC3)C23CC3)=O)CCC1NC(c1cscc1Br)=O n1(CC(N2CC(F)(C(=O)NC(CC#C)CO)C2)=O)cccnc1=O C12(NC(CC3(OC)CN(C(=O)C(C)CC(F)(F)F)C3)=O)CC1COC21CCC1 c1(C(=O)NC(C(C)(C)C)CNC(=O)C=Cc2cnc[nH]2)ccc(C#N)cc1[N+](=O)[O-] Cc1noc(C)c1C(N1CCC(CF)(NC(=O)CC(=O)NCC2CC2)C1)=O c1(O)ccccc1F.C1(C(N2CC(CC3CCN(C)C3)C2)=O)(OCC)CCCC1 CC(C)C(C)C(CNC(c1cc(Br)ccc1Cl)=O)NC(C12CCC(C1)C2)=O CC1CC(C)OC1C(N1CC(C(C)NC(=O)CCC2(C)N=N2)C1)=O CCC(C)(CNC(=O)C=Cc1nccs1)C(=O)NCc1cc(C)c(C)o1 c1(NC(CC2C(NC(c3c(CC)csc3)=O)CCC2)=O)c(O)n[nH]c1C C1(NC(C(C)c2ccsc2)=O)CC(F)CN(C(=O)C=C2CCN(C)C2)C1 C(CCC(=O)NCC1=NOC(C)C1)(C(C)C)NC(c1c(C)coc1)=O c1(OC)ncc(C)c(C(=O)NCC2CCN(C(=O)CCn3ccnc3C)C2)c1Cl C1(CC(=O)OC(C)C(=O)N(C)C)CCCN(C(=O)NC(C)(C)C)CC1 N1(C(C=CC(=O)N(C)C)=O)CCN(C(c2cnc(O)o2)=O)CC1c1ccccn1 c1(C(=O)NCC(=C)CCNC(C2CC3COCC3C2)=O)ccc2ncsc2c1 C1(CC(=O)OCC)(CNC(N2CC(C3CCCO3)C2)=O)CCCCO1 N1(C(Cc2cccc(OC)c2)=O)CCC(C2CN(C(c3cccnc3O)=O)C2)C1 Cc1nn(CC(N2CC(NC(=O)Cc3occc3C(=O)O)CC2C)=O)cc1Cl N1(C(C(C)SCC)=O)CC(NC(c2cc(N)ccc2Cl)=O)CC12CCCC2 N1(C(C(C(C)(C)C)N2CCNC2=O)=O)CC(N=c2[nH]nc(C3CC3)s2)C(C)(C)C1 C1(NC(C2NC(=O)OC2)=O)COCCN(C(=O)C=Cc2cncc(O)c2)C1 C(=O)(C1=CC2CCC(C1)C2)N1CCC(NC(c2cc(F)ccc2F)=O)(CF)C1 C1(C2N3CC(C)N(CC3)C2)CCC2(CC1)CCN(NC=O)CC2.c1(C)ccnn1C CS(=O)(=NC(=O)COCCCC#CCO)C1CCC1C CCC(C)C(C)C(=O)NCCN(C(=O)Cc1ccccc1CC#N)CCOC C(=O)(C(C)(C)C(=O)NCC1C2CN(C(=O)C(C)(C)c3ccno3)CC12)NC N1(C(=O)NCc2cc[nH]n2)C2CCC1CC2 c1(CNC(C2OCCN(C(c3cc(CC)[nH]n3)=O)C2)=O)cccc(C#N)c1 C(=O)(C1=CCCC(C)(C)C1)N1CC(CN(C(c2c(CC)scc2)=O)C)OCC1 C1(C(=O)NCC(CC)NC(=O)C2=NOC(C)C2)CC(=O)N(OC)C1 CCCC(CC)CCC(=O)NC(CN(C)C)C(=O)NC1CC(CC)C1 N1(C(C2(COC)CC2)=O)CCOC2(CCC(NC(=O)Nc3ccccc3)CC2)C1 CC(C(=O)N1CCC(NC(=O)CC(C)(C)C2CC2)C(C(N)=O)C1)S(N)(=O)=O CCCC(CC(=O)NC(c1ccnn1CC)C)NC(C1CC12CCCCC2)=O CC(CC(=O)NCc1cn(C2CN(C(=O)CCC3(C)CC3)C2)nn1)C(F)F C1(NC(c2c(C)cccc2F)=O)CN(C(c2sccc2Cl)=O)C2(CCCOC2)C1 CC(C)CC(CN(C)C)NC(c1cc(C2CC2)on1)=O.C12(CCC1)CC(=O)N2 C#CCCCCC(=O)NC1CC(O)C1CC(=O)NCCn1ccnc1 c1(C(C)=O)cc(C(=O)N(C2CC(NC(c3ccc(C(F)F)o3)=O)C2)C)no1 C(=O)(C(C(C)C)NC(N)=O)N(CCC(=O)NCC(C)OCC=C)CC C1(ON)CC2CCCC2(NC(=O)C=CC(c2cccnc2)=O)C1 C1(CN(C(C=CCOC)=O)C)C2CN(C(=O)C(N3CCCCC3)C)CC12 C1(C(=O)NC(COC)CO)CCN(C(=O)CCn2ccnn2)CC1(C)C C1(C)(C(=O)NCC2CC(C(C)C)C2)CN(C(c2cnn(C)c2)=O)CC1C C1(CNC(C(N2CCOCC2)C)=O)COC(CNC(=O)CSc2cn[nH]c2)C1 C(=O)(C=CS(C)=O)N(CCCNC(C(C)N(C(C)(C)C)S(C)(=O)=O)=O)C c1(CC(=O)NCC2CN(C(=O)C(C3CCCCCC3)F)CC2O)ccc(O)cc1 C(CC(C)C)(C(=O)NCc1ccsc1C(=O)NCc1cncn1C)OC Cc1cc(Cl)c(CN2CCC(C(=O)Nc3cccc4[nH]ncc34)C(O)C2)c(Cl)c1 c1(CC)noc(C)c1C(=O)NCC1(NC(=O)CCc2cncnc2)CCOC1 c1(C(=O)NC)ccc(O)cc1.C1(=O)CC(C2CCC2)N1C(C)C n1(CC)nc(C(=O)NCC(CC)NC(=O)CCCCc2cccc(O)c2)cc1C C(C(=O)N1CCC(c2ccccc2)(NC(c2cscn2)=O)C1)(C(C)C)SC C(CCCCCNC(c1cc(C2CCC2)[nH]n1)=O)C(c1cccn1C1CC1)=O N1(C(c2c(OC)nc(C)s2)=O)CC(NC(=O)CCC(C)(C)C)C(F)(F)C1 N1(C(c2c(C)ccc(C)c2)=O)CCN(C(=O)C(c2ccc(F)cc2)C)CCC1C C1(C(N(CC)CC2CCCO2)=O)COC2(C1)CN(C(=O)CCOCC1CC1)C2 C(=O)(CCCCF)N(C1CCN(C(C(C)n2ccnc2)=O)C1)C c1(C(=O)NCC2CCN(C(=O)CN3CCSCC3)C2)cccn2c(O)nnc12 N1(C(C2N(C(C(NOC)=O)=O)CC2C)=O)CCC(O)CC(C)C1 N1(C(=O)NCCc2cnc(OCC)s2)CC2CCCC1(CO)C2 C1(CC)COCCN(C(=O)C(c2cccs2)NC(=O)C(O)CCN(C)C)C1 C(CCCCC(=O)N1CCCC(CCC(=O)NCCC(F)(F)F)C1)OC C1(C(=O)NCC(C(C)(C)C)NC(CCCC)=O)CCc2nnc(C)n2C1 n1(CC)cc([N+](=O)[O-])c(C(N2CCN(C(=O)CN3CCCC3C)C3(CC3)C2)=O)n1 C(=O)(C(O)C(F)(F)F)N1C(CNC(CCN2CCC(C(N)=O)CC2)=O)CCCC1 c1(CN2CC(N(C(c3ccc(C(=O)NC)cc3F)=O)C)C2)cc(C#N)ccc1O c1(-c2c(C#N)cccc2)cnc2cc(C(=O)NC(CO)C(F)(F)F)[nH]c2c1 c1(NC(NCS(CC)(=O)=O)=O)c(C)ccc2cc(C)ccc12 c1(OC)c(C(=O)NC(C)CNC(=O)CC(C)F)sc(Cl)c1Cl N1(C(C2CC2CC2CCCO2)=O)CCC(c2ccc(Br)cn2)CC1 c1(C(=O)NCCC2N(C(CC#N)=O)CCCC2)cc2cc(Cl)cnc2[nH]1 C1(C(=O)NCC(COC)O)CCN(C(=O)CO)CC1c1ccccc1 C1(CNC(C2C3CCN2CC3)=O)CC(F)CN1C(=O)CC1CCCC1 S(=O)(=O)(c1ccc(O)cc1)N1CC2N(C(c3cc(Br)ccc3Cl)=O)C2C1 c1(C(N2CC(C)C(NC(c3nc(Cl)ccc3Cl)=O)C2)=O)cc2n(n1)C(C)CCC2 C(C(CC(=O)N1CC2(CC(NC(=O)C(C)(C)CN(C)C)CO2)C1)C(F)F)N(C)C C12(CNC(c3ccc(OC)nc3Cl)=O)CCCCC1CN(C(=O)C(C)OC)C2 C1(CNC(C(C)(C)F)=O)CN(c2ncnc3c2CCO3)CCC1(F)F c1(C(N2CC(NC(C(CCC)NC(C)=O)=O)C(C)C2)=O)ccc2sccc2c1 c1(C(=O)OC)c[nH]c2ccccc12.c12cc(O)ncc1C(=O)N2C1CC1 C(=O)(CC(C)CCC=C(C)C)NC1CCC(CNC(C(C2CCC2)OC)=O)CC1 Cc1cc(Cl)nc(Cl)c1C(=O)NC1CCC2(C1)CN(C(c1ncc(Cl)cc1Br)=O)C2 C#Cc1ccc(C(N2CC(F)(F)CC2CCNC(C2(C(F)F)CC2)=O)=O)cc1Cl N1(C(c2cccc(C#C)c2)C(=O)NCCCC)C2CCCC1CC(O)C2 C12CC3(C1)CC3C(=O)N2.N1(C(CCSC)=O)CC(C)(C(N)=O)C1 c1(OCC=C)ccc(S(N)(=O)=O)cc1C(=O)NC1CCN(C(C2(Cl)CC2)=O)C1 c1(C(N(CC(C)NC(c2cnn(C)n2)=O)CC)=O)sc(C(C)(C)C)nc1C C1(CNC(C(C)(C)OCC)=O)CC2CCCC2N1C(c1csc(C2CC2)n1)=O CON(CC1CSc2ccccc21)C(=O)c1cccc(S(C)(=O)=O)c1F C1(CC)CN(C(c2c(C)ncn2O)=O)CC1c1cnn(C)c1 CCCCC(O)CCC(=O)NC(C1CCN(C(=O)C(c2ccccc2)C)CC1)C C(N=c1[nH]c2ccc(O)cc2s1)C1(F)CC(NC(=O)CCCC2CC2)C1 Cc1cc(C)c(C(=O)NC(C)C(C)NC(c2cc(C(C)(C)O)ccn2)=O)cn1 N1(C(c2n(CC=C)ccc2)=O)CCC(O)(CNC(c2cnc(OC)s2)=O)C1 CCC1=C(C(=O)N2CCN(C)C(CNC(=O)CC3CSCCS3)C2)CCCO1 c1(-c2cn(C3CCCN(C(C(C(CC)O)C)=O)C3)nn2)c(F)cc(N)cc1F C1(NC(CCN(C(=O)CC2(O)CCC2)CC#C)=O)CC2(CCCC2)C1 O=C(C(F)C1=CCCCC1)NS(=O)(=O)C1(c2cn(CCOC3CC3)nn2)CC1 c1(C(=O)NCCN(CCC)C(c2[nH]ccc2C)=O)cnncc1OC N1(C(c2cc(C(C)=O)[nH]n2)=O)CC2C(C(=O)NC(C)C(=O)NC(N)=O)C2C1 CCC(CC(=O)N1CC2C(CC(=O)NCCc3nncs3)C2C1)OC C12(CCCCC1)CC(=O)N2.c1(C(C)(C)NC(C)=O)cn(CCC(F)(F)Cl)nn1 CC1(C2CC2NC(C2COCC2n2ccnn2)=O)CCCC1 CC1CCC(CNC(c2nncs2)=O)N(C(C2CC3(CC3)C2)=O)C1 Cc1ccc(C(=O)NC(C(=O)NCCn2ncnn2)C(C)C)cc1 CC(C)CC(C)C(=O)NC1CCCC1NC(=O)CN1CCCC1CO C(C)(CC(C)C(F)F)NC(c1cc(CNC(C=CCC)=O)on1)=O CC(CS(=O)(=O)NC1CCCc2occc21)N=c1nc2sccc2c(N(C)C)[nH]1 C1(CC(N)=O)CCCC12CCN(Cc1nn[nH]n1)CC2 N(C1CCc2cc(Cl)ccc21)c1[nH]c(=NCc2cc(F)c(F)cc2F)cc(C)n1 C1(OCc2cn(CC3N(C(CCC=C)=O)CC3)nn2)CCCCC1=O C(CC(C)C)(C(=O)NC1COCC1NC(c1cc(C)c[nH]1)=O)NC(C)=O C(N=c1[nH]nc(CO)s1)C12OCC(NC(CCCSC)=O)(C1)C2 c1(C(=O)NCC(=O)NC(c2cnsc2)C)cnn(C(F)F)c1 C1(NC(c2c(C(C)NC(COCC)=O)noc2)=O)CCn2ccnc2C1 C1(C(N2C(CNC(CCCN(C(C)=O)C)=O)C(C)CC2)=O)CC2(CCO1)CC2 CC1C(C)N(C(c2cc3cc(Cl)cnc3[nH]2)=O)CCS1(=O)=O N1(C(CC2CC(C(=O)OC)C2)=O)CC(CNC(C2CC=CCO2)=O)C(O)C1 C(C(C)(C)C(C)(C)C)SC.C12(CN(C(C3CCC(F)C3)=O)C1)C(=O)N2 N1(C(C2N(CC)CCC2)=O)CC2OCC(NC(=O)CN3CCCCC3)C2C1 Cc1cccc2c(C(N3CCN(C(c4nc(=N)cc[nH]4)=O)C(C)C3C)=O)coc12 c1(N(C(C#C)C)C)nnc(-c2ncoc2C)n1CCC1CCOC1 c1(C(N2CCC(CNC(COC)=O)(OC)C2)=O)ccc(C)c(Cl)c1 c1(C(=O)OC)ncnc2c1cnn2C1(NC2CC(F)C2)CCCC1 C1(CC=C)(NC(c2nc(C)ncc2Cl)=O)CCN(C(=O)CS(N)(=O)=O)CC1 c12cnc(nc1)CNC(=O)N2.N1(C(=O)NC)CC(C(c2ccccc2)=O)CO1.O CC1CCN(C(=O)C=CC2CCCC2)CC1NC(C1CCC(=O)N1C)=O CN1N=C(C(=O)N2CCC(CCCCNC(C3CC3C3CC3)=O)CC2)CCC1=O N1(Cc2c(OC)ncc(Br)c2)CCC2(CC1)CC2NC(c1ccc(C)c(Br)c1)=O C1(C)(CC(=O)NCC2C(NC(CC3CC(OC)C3)=O)C2)CC1(Cl)Cl C1(CNC(C(CC)(CC)CC)=O)CCCC2CN(C(C3CCN(C)C3C)=O)CC12 c1(OCC(=O)NC2CC(C)OC(C)C2)ccc(S(N)(=O)=O)cc1F N1(C(C)=O)CCNC2(CCC2)C1.C(=O)(C(N)C(C)CC)OCCc1ccccc1 c1(CNC(c2cc(C)ncc2)=O)nc2c(s1)CCN(C(C1CC3C=CC1O3)=O)C2 c1(C(=O)NC2CC(OC)CN(C(=O)C(C)(C)C(C)O)C2)cc(C)cc([N+](=O)[O-])c1 CC(CC(=O)N1CC2C(CNC(c3cnn(CC(F)F)c3)=O)C2C1)C(F)F C1(N2CCC(N(C(c3cccc(Cl)c3C)=O)CC)C2)CC2CCCCC2NC1=O c1(CCNC(=NCCCC)NC2CC23CC3(F)F)cc(F)cc2c1OCOC2 c1(C(N2CC3=C(CN(C(C4CCCC(=O)O4)=O)C3)C2)=O)cc2ccc(O)nc2s1 C12(C(N3C(C)(CNC(CCC#CC)=O)CCC3)=O)CC(CO)(C1)OC2(C)C C12(NC(c3c(Cl)cnc(C)n3)=O)CCCCC1CN(C(C1CC=CC1)=O)C2 C1(OC)COCC1n1cc(CNC(=O)CNC(C2CC2(F)F)=O)nn1 N1(C(C=CC=CC)=O)CCCC2(CCN(c3[nH]cnc4nc(Br)cc3-4)CC2)C1 Cc1c(C(=O)N(C)CC2COCCN2C(=O)C(C)C(F)(F)F)sc2ccsc12 C1(F)(CNC(c2cnn(CC)n2)=O)CCCN(C(C2COCC2(C)C)=O)C1 N1(C(CC(CC)C)=O)CC2CC(NC(c3cnc4sccc4c3)=O)CC2C1 c1(C(N2CC(NC(C=CS(C)=O)=O)C(C(F)F)C2)=O)ccc(F)c(C(F)F)n1 N1(C(C(CCC)NC(c2ncn(CC)n2)=O)=O)CCC2(C=CCO2)CC1 CC12CCC(C(=O)NCC3CCN3C(c3ccc(CO)cc3)=O)(CC1)C2 N1(C(CC=CC=C)=O)CC2CN(C(=O)Nc3ccc(SC(F)(F)F)cc3)CC2C1 c1(C(N2CC(C)(C(=O)Nc3ccc(OC)cc3)C2)=O)cnc2c(C)cc(C)cn12 c1(C(=O)NC(CC(C)NC(CCCNC(=O)OC)=O)C)[nH]ccc(=O)c1C C(CCC(=O)NC1CC(O)C1O)(C(C)C)NC(C1(CC)COC1)=O CCC(CNC(c1ccc(F)cn1)=O)(CC)NC(=O)Cc1cn(C2CC2)cn1 C(=O)(C1CCCc2ccnn21)NC1(CCCCNC(=O)C2=CCCSC2)CC1 Cc1cc(C(=O)N(CCCSc2ccccc2F)C)ccn1 CC1(C)C(CO)OCCN1C(=O)NC1C2CC(=O)CC12 N1(CC)CCOCC1C(=O)NCCC1CC(NC(=O)Cc2ccnn2C(C)C)C1 C1(C(=O)NC2(C)CCN(C(CC3(COC)CC3)=O)CC2)CCn2ccnc2C1 C1(CNC(C(C)OCC=C)=O)CCCCCN1C(=O)CC(C1CCC1)C1CCC1 C1(F)(CNC(C(N2CCN(C)CC2)C)=O)CC(N=c2[nH]nc(C(C)(C)C)s2)C1 N1(C(c2c(C)nccn2)=O)CCC(C(=O)NCC(O)(C2CC2)C2CC2)CC1(C)C Cc1ccnc(Cl)c1C(=O)Nc1ccc(-n2cccc2)c(Cl)c1 C#CC1(N(C)C)CN(C(=O)C(C)c2cc[nH]n2)C1.C(=O)(CO)N c1(C(N2CCC(C)C(CNC(=O)C(C)(F)F)C2)=O)cnc2c(c1)NC(=O)CS2 N1(C(CC2(COC)CC2)=O)CCN(C(=O)CN(C)C(C)C)CC(C)(F)C1 O=C(C1=CC2(CCOCC2)C1)OC1COCCOC1 N1(C(c2ncc(OC)nc2)=O)CC(=O)NCC1C(=O)NC(C)Cn1cnnc1 C(C1CCCN1C(C1CCC1)=O)=CC(=O)NC(C(C)C)C1CC1 Cc1cc2cccc(NC(C3CCOC4(CCOCC4)C3)=O)c2cn1 C(=O)(CC(C)CC(C)C)N1CC(OCCC(=O)NCC=CC(CC)C)C1 C1(C(N2CC(F)(CNC(=O)CN3CCSCC3)C2)=O)CCCc2ccccc2C1 N1(C(=O)CCC2CC2)CC2CCC1C2NC(C12CC3CC1C2C3)=O C1(CC)CCCN(C(c2cnc(OC)s2)=O)C1C(=O)NC1CCC(C(N)=O)C1 c1(C(=O)NC(C2CCN(C(c3cc(F)c[nH]3)=O)C2)C)cc(Cl)cc(Cl)c1N C(=O)(C(F)C(F)(F)F)NCCC1(CNC(C2CCCC2O)=O)CC1 O=C(CS(=O)(=O)C1CC1)NC1CCCC1NC(C1CCN1Cc1ccccc1)=O c1(CC)ccc(NC(=O)C(C)(C)CNC(c2cnns2)=O)c(C)n1 Cc1cc(F)ccc1CC(=O)NC1(Cn2cc(CCC(C)O)nn2)CC1 C12(C(=O)NCCC(C)N(C(C3C(C)(C(C)C)C3)=O)C)CCCC(CO1)C2 S(=O)(=O)(c1ccc(Cl)nc1C)Nc1c2ccc(C)cc2no1 CCC(CC(=O)N1C(C(=O)NCCCOCC(F)F)CC1C)CC(C)C CS(=O)(=O)CCCC(=O)NC1CCCN(C(=O)C(F)(F)c2cnccn2)CC1F c1(C(=O)NCC2(OC)CN(C(C3CCC3F)=O)C2)cncc(Cl)c1Cl C1(C)(OC)CN(C(c2coc(CNC(C(C)OCCCC)=O)n2)=O)C1 N1(C(C2C=CCN2C(c2csnn2)=O)=O)CCOC2COCC12 c1(CN2CC(N(C)C(c3ccc(Cl)c(CO)c3)=O)C2)cc(Br)cc([N+](=O)[O-])c1O C1(NC(c2c(CC)nn[nH]2)=O)CN(C(=O)C(C)(O)C(C)C)CC(C)(C)C1 C(C)(N=c1[nH]c2c(c(=NCC3CCCC(F)(F)C3)[nH]1)COC2)C1(COC)CCC1 c1(C(=O)NCCOCCN(C(CC2(CS(C)(=O)=O)CC2)=O)C)ccc(Cl)nc1O CCC(C)(C)C(=O)NCc1csc(C(=O)N(C)CC2(N(C)C)CC2)c1 C1(C(=O)NC2CC2F)CC1(F)Cl c1(C(N2CC(CC)N(C(C3CC(C)(C)CO3)=O)CC2)=O)ccc2c(c1)ncn2C c1(C(=O)NC2CN(C(C=C(C)Cl)=O)CC2O)cc(C)cnc1C C1(CC(=O)NC2(C(=O)NCCC(C)OCC)CC2)COCCO1 C=CCCCC(=O)N1CCCC(n2cc(-c3cnsc3)nn2)C1 C1(NC(C2(C)CCCOC2)=O)CCC2CC1CN2C(c1cc(N)cc(F)c1)=O N1(C(C=CC)=O)CSCC1C(=O)N(C)Cc1cnco1 c1(C(N2C(CNC(C(C(C)C)OC)=O)CCC2)=O)oc2c(C)ccc(C)c2c1C CCCCCCCCC(=O)N1CC(O)CC1(C)C(N1CC(C#N)(COC)C1)=O N1(C(C(C)(C)c2cc[nH]n2)=O)CCC(CO)C(NC(c2cccc(Cl)c2)=O)C1 c1(OC)cc(OC)c(C(=O)NCC2(F)CN(C(C3CC=CCO3)=O)C2)c(OC)c1 CC1Cc2cc(C(N3CCC(NC(=O)C4=NOCC4)CC(O)C3)=O)ccc2O1 C(=O)(CCCCC(F)(F)F)N1CC(N(C(=O)COC2CCOC2)C)CC12CCC2 C(=O)(C(F)C(F)(F)F)N1CC(CCCCNC(Cc2cc(CC)nn2C)=O)C1 N1(C(C2CC(F)CN(Cc3nccs3)C2)=O)CCc2c(F)cccc2C1 c1(C(CNC(c2cnn(C3CCC3)c2)=O)NC(C(C)SC)=O)cccc(C)c1 CCC(C)C(O)C(=O)NCCCC1CCCN1C(=O)Cc1ccc(O)c(O)c1 c1(C(CNC(CC2C(C)OCC2)=O)NC(c2cnsc2)=O)ccccc1F Cc1ccc(C(N2CC3CC2CC3NC(=O)CCCn2cccn2)=O)cc1O N1(C(CCC(C)SC)=O)CC2OCCN(C(c3ccc(CO)nc3)=O)C2C1 N1(C(C(C(=O)OCC)(C)CC)=O)CCCC2(C1)CN(C(=O)C=CCOC)C2 N12CC3(C1)CN(C3)C(=O)C=CCCC=C2.c1(CC)ncccc1C(=O)OC c1(C(=O)Nc2n(C)ncc2I)ccc2c(C(N3CCOC4CC34)=O)n[nH]c2c1 C(=O)(C1CCCc2ccccc21)NCCN(C(CC(C=C)CC)=O)CC1CC1 C1(C(N(CCC)CCC)=O)CN(C(=O)C(c2cnn(C)c2)=O)CC(C)(C)C1 N1(C(C2(C)CC2(F)Cl)=O)CCOC(CNC(C2CC2c2ccccc2)=O)C1 c1(CNC(c2c(Cl)cc(N(c3nc(C)ncc3F)C)nc2)=O)n[nH]c2c1CCCC2 N#Cc1ccc(C(N2CC3(C2)SCCC3NC(=O)CCSC(F)(F)F)=O)c(F)c1 CC1CC(N=c2[nH]nco2)CN1C(=O)C1CCCc2nncn21 Cc1cc(NC(c2cc(S(C)(=O)=O)c(Cl)cc2Cl)=O)nc2ccccc12 CCS(=O)c1ccc(-c2cccc3[nH]nc(C(=O)Nc4cncs4)c23)cc1 N1(CC(=O)NCCN(C(=O)C(O)C2CC2)CCC)CCS(=O)CC1 C(c1cc(F)c(O)c(F)c1)=CC(=O)NC1C(C(=O)O)C2CCCCC12 c1(C(=O)NCC(C2CCN(C(CC3ON=C(C)C3)=O)CC2)O)cc(C)cc(Cl)n1 N1(C(CCC#N)=O)CCC(NC(=O)C(C2(O)CCCC2)F)C(C(N)=O)C1 c1(C(=O)NC23CC(NC(C(=O)N(C)C)=O)(C2)C3)ccc2c(c1)nc(C)n2C1CC1 C1(NC(CC2(COCC)CC2)=O)CN(C(c2cncnc2)=O)C2(CCCC2)C1 N1(C(=O)NC2(C(=O)O)CC(C#C)C2)C(C)CC(C)CC1C CC1(NC(c2cnc(Cl)cn2)=O)CCCN(c2cc(Cl)nc(C(F)(F)F)n2)C1 Cc1n[nH]c(C)c1CC(=O)N(C1CCOC1)C1(C(=O)NC2CC2)CC1 N1(C(C2(CC)CCC(O)CC2)=O)CC2CCCC2(NC(=O)CS(N)(=O)=O)C1 c1(N2CCC=C(F)C2)nc(N2CCOc3ncccc3C2)c2c(n1)CSC2 C1(NC(=O)CN2CCCC2CO)CCCCN(C(=O)CC2=CCCCC2)CC1 CC(C(C)C(=O)NCC1(C(=O)O)CCCC1)S(C)(=O)=O c1(C(=O)NCC2(CCNC(c3cnc(OC)s3)=O)CC2)csc2c(O)ccnc12 CC1(C)CCC(C(=O)NC2CC(CF)C2)CN1C(C1(O)CCCC1)=O C1(NC(C(C)Oc2ccccc2F)=O)CN(C(=O)CCC(N)=O)C(C)(C)C1 C1(C(=O)NCCC2CCCC2)CCCCN(C(=O)CCC2CCC2)CC1 n1(CC)cc(NC(=O)C(COC)NC(=O)CCN=[N+]=[N-])ccc1=O c1(C(N2CCCC(C(N3CCN(C(=O)C4CC4)CC3)=O)C2)=O)cnnc(Cl)c1 N1(CC(=O)NCC2(OC)CN(C(=O)CCc3ccccc3C)C2)CCCC(O)C1 N1(C(C(CC)(F)F)=O)CC2(CNC(C3CCN(C)C3C)=O)CC2(C(F)(F)F)C1 C(=O)(CS(=O)(=O)c1ccccc1Cl)NC1(CO)CCCN(C(CC2C(C)C2)=O)C1 Cc1cc(C(=O)NC2CCN(C(=O)CC(=O)N(C)C)CC2O)c2ccccc2n1 c1(COC(=O)C(C(=O)NC2CC2)NC(=O)OC(C)(C)C)cc(Cl)cc(Br)c1F C(=O)(CCC(C)CN(C)C)N1CC(CCNC(COCC(C)C)=O)C(F)C1 C(C(C)(C(=O)NC(C1CC(NC(c2cccnc2O)=O)C1)C)OC)OC C1(NC(CNC(CC)=O)=O)CCC(CC(=O)NCC2(C)CCN(C)C2)CC1 c1(C(=O)Nc2cnc(F)cc2C(=O)Nc2cc(F)c(Cl)cn2)cnn2ccccc12 C(=O)(CCCCC#N)NCC(CC(=O)NCCN1CCC(OC)C1)C C12(C(N(CC(CNC(C=C(C)C(C)C)=O)O)C)=O)CC(C)C1C2 c1(OCC(=O)N(CCNC(C(C)Cn2cccn2)=O)C)cnc2ccccc2c1 CC1(NC(c2ccnnc2S)=O)CCCN(C(=O)C(O)CC2CC2)C1 N1(C(=O)NCC(C)N(C)C)CCCCC1C1CCCN1C(=O)NC(C)(C)C N1(C(CC2(COC)CC2)=O)CC(N(C)C(C2COCCN2C(C)=O)=O)C(F)C1 c1(C(N2CCC(OCC)C2)C(=O)NCCC2CC2)ccc(C(F)(F)F)cc1C C1(CCC)(NC(C2CC(C)N(C)C2)=O)CCCN(C(c2c(C)noc2N)=O)C1 c1(NCCNCCNC(CC2CCCC(OC)C2)=O)c(C)nc2n1CCCC2 c1(COC)ccc(C(N2CC(F)CC2C(=O)NCCC2CCO2)=O)c(C)c1 C1(CNC(=O)Cc2cnccn2)CCN(C(C2CNC(=O)N2)=O)CC1(F)F C1(NC(=O)CN2CCCC2)CC2CCC1(CNC(c1ccc(O)cc1Cl)=O)C2 c1(CCNc2nc(C)c(N3CCOCC3)cc2)c(F)ccc(Cl)c1F C1(C(=O)NCC(CN(C(CCc2ccc(C(=O)OC)[nH]2)=O)C)C)CC2C=CC1C2 N1(C(C(c2ccnn2C)C)=O)CCC2CN(C(c3nnc(O)cc3O)=O)CC2C1 C(C(C(=O)NCC1CCCSC1)NC(C)=O)NC(=O)CC1(N(C)C)CCC1 C(C(=O)N(C)C)(C(C)C)NC(C1C(OC)CC1)=O.C1(CNC=O)(ON)CN(C)C1 c1(C(N2CC(NC(CCc3cnn(C)n3)=O)(CO)C2)=O)cccc2oncc12 Cc1ncnc(N2CCOCC(CNC(C3(O)CC3)=O)C2)c1C#N C1(NC(C2CC(=C)C2)=O)CC2(CCC(CNC(C3CCCNS3(=O)=O)=O)CC2)C1 N1(C(c2c(SC)nn(C)c2)=O)CCN(C(C2CCCCO2)=O)CCC1C Cc1ccc(C(=O)NCC2(C(=O)NCC3(C)CCN(C)C3)CC2)n1C C1(C(=O)NC2(CSC)CC2)C(C2CC2)CCN1C(c1cc(F)n(C)n1)=O Cc1cc(C(N2CC3CC(NC(=O)CCC4CC(F)(F)C4)C2C3)=O)ncc1N N1(C(CC(CCC)C)=O)C2CCCC1CN(C(c1coc3ccc(C)cc13)=O)C2 C12(CNC(c3c(C)con3)=O)CCC1CCN2C(=O)CCc1cccnc1Cl C1(NC(=O)CCCN2CCCCC2)CCOCC1NC(C12CC(F)C1C2)=O C1(c2cn(C)nc2)CN(C(c2nonc2N)=O)CC1CNC(=O)CC1CC12CC2 CC1=NOC(C(=O)NCCN(CC(C)O)C(=O)CC2CCCC2)C1 C=CCCCC(=O)N1CC(CC(C)(C)CNC(c2ccc(F)cc2)=O)C1 C(CCC(C(=O)Nc1ccccc1C(=O)OC)N1CC(C)C(C)C1C)OCC CCCCCCCCCC(=O)NCC(CNC(=O)Cc1ccns1)CO Cc1cc(C(N2CC(NC(c3ncccn3)=O)CC23CCC3)=O)c(C)c(C)c1 c1(OCC(=O)NC2(C)CN(C(C3(C#C)CCC3)=O)C2)cc(C(F)(F)F)ccc1C CC1(C)CC1(c1ccccc1)CC(=O)NCCC1CN(C(=O)C(=O)NC2CC2)C1 n1(CC)ccc(C(=O)NC2(c3cn(C4CC4)nn3)CN(C(=O)C(N)=O)C2)cc1=O C12(NC(c3ccc(C)n3C)=O)CN(C(c3cn(C)c(O)n3)=O)CC1CS(=O)(=O)C2 n1(CC(N2CCC(OC)(CNC(=O)COC(F)F)C2)=O)ccc(=O)c(O)c1C CCCC(C(=O)N1CCC(C)C1C(N1CC(COC)C1(C)C)=O)N(C)C C(=O)(C(O)CC(C)(C)C)N1C(CNC(C2(C(F)F)CC(=C)C2)=O)CC2(CC2)C1 C1(CC(=O)N(C)CC2(CNC(=O)CCn3cccn3)CC2)COC(C)(C)C1 c1(CC)cc(C(=O)NC2CCN(C(=O)CCOC3CCCC3)C2)ncn1 c1(CNC(C2(C3N(C(C(CC(N)=O)O)=O)CCC3)CC2)=O)cn2cccnc2n1 N#CC1(c2ccccc2)CC2(CN(C(=O)Cc3ccc4c(c3)OCCO4)C2)C1 CCCCC(C(=O)N(C)CCNC(C1(C2CCCO2)CC1)=O)NC(N)=O S(=O)(=O)(CC(=O)NC1CC(NC(=O)CC(O)CSC)C1)NCC N1(C(CCc2n(C)cnn2)=O)CCCC(CCNC(c2cc(N)ccn2)=O)C1 C1(CNC(C2(c3ccncc3F)CC2)=O)CC2(CC2)CN1c1ncccn1 c1(C(N2CC(OC)C(NC(c3cnc(O)cc3C)=O)C2)=O)cc(Cl)ncc1N C1(C(N(CC(C(C)C)C)C)=O)COCCC1NC(c1cnsc1)=O c1(C(=O)NC(CCCC)CNC(=O)CC(=O)NCC2CC2)ncnc2c1CCC2 N1(C(CCCOC(C)C)=O)CC(NC(C2COCCN2C(C)C)=O)CC(O)C1 C1(C(N2CC(OCC)C(CO)C2)=O)(NC(=O)C(C)=CC(C)(C)C)CCC(C)(C)C1 c1(C(=O)NC2(CCNC(C=CCN(CC)CC)=O)CCC2)ccc(N)c(C)c1F c1(C(C)C)cn(CCC2CCN(C(=O)NC(C)(C)C)C2)nn1 Cc1ccc(O)cc1C(=O)NC1C2CCC1N(C(=O)CC1CN(C)C1)C2 C12(C(=O)NCCCC(C)(C)NC(C3(C(C)(C)C)CCC3)=O)CCCC1C2(F)F N1(C(c2ccnc(OC)n2)C(=O)NCC(F)F)CCC(F)(F)C(F)C1 N1(C(CCCC(C)(F)F)=O)CCC2CCN(C(c3cnc(S)nc3)=O)CC2C1 N1(Cc2cn(COC3(CC=C)CC=CCC3)nn2)CCc2sc(Cl)cc2C1 N1(C(CCC#C)=O)CCOC2(CCN(C(=O)CNC(c3ccccc3)=O)CC2)C1 C=CCC(C)C(=O)NC1CC12CC(NC(c1ccc(OC(C)C)cn1)=O)C2 N1(C(C)C(=O)NC(=O)NC2CC2)CCCC2(CNC(=O)C2)C1 c1(OCCC(=O)NC(C)C(C)NC(c2coc(Cl)n2)=O)ccc(F)c(Cl)c1 c1(NCC)cc(Cl)ccc1C(=O)NCC1CCC(NC(C23CC4CC2C3C4)=O)C1 C1(OC)CN(C(=O)CCC2CCOC2)CC1CNC(C1CCC(CC#N)CC1)=O c1(NC(CCCC)c2nnnn2CCCF)ccc(NC(=O)OC)cc1C N1(C(c2c(C)cc(C)nc2)=O)CCC(C2(NC(c3ccnc(C)c3C)=O)CC2)C1 C(C(CC)(CC)C(=O)N(CC(C)O)CCSN)NC(CC(C=C)(C)C)=O.CS.C C1(CC)CN(C(=O)COC(C)=O)CCN1Cc1cc(F)ncc1OCC(C)(C)C c1(CC(=O)NCC=CCNC(CCCOC)=O)csc2c(Cl)cccc12 N1(C(C(C)C2CC2)=O)CC2(COC(CNC(c3ccc(=O)oc3)=O)C2)C1 c1(C(N2CC(OC)C(NC(C3(C)CC4CCC(C3)S4)=O)C2)=O)ncnc(O)c1F c1(OC)nc(C(=O)NC(C)C(C)(C)NC(c2cc(C(F)(F)F)no2)=O)co1 C1(NC(c2c(C)n(C(C)C)nc2)=O)CN(C(C2CC(=O)N(C)C2)=O)CCC1O C(CC(=O)N1CCC(C)(C)C1CNC(=O)COC1(C)CCC1)(C(F)(F)F)OC c1(C(C)(C)C(N2CC3C(NC(C4CC4(F)F)=O)C3C2)=O)ccccc1Cl Cc1ccc(F)cc1C(=O)N(C(CNC(=O)C(C)(C)O)C1CC1)C C1(CNC(c2ccn(C(C)C)n2)=O)CC2CCC1N2C(=O)CC1C=CS(=O)(=O)C1 C12(NC(=O)Cn3cc(Cl)cn3)CCN(C(=O)CCc3cc[nH]n3)CC1C2 CC1CC(NC(c2nn(C)cc2Br)=O)CN1C(=O)COC1CCOCC1 c1(C(N2CC(CC)N(C(=O)CN3CCCC3C)CC2)=O)cc2c(cc1N)CCC2 CS(=O)(=O)c1ccc(C(N2CC3CCCC2(CNC(=O)CCF)C3)=O)cc1Cl N1(C(C2(OC)CCSC2)=O)CC(C)OC2(CCN(C(=O)Cc3cccnc3)C2)C1 N1(CCN(CCOC)Cc2cnc(C)o2)CCOCC1 N1(C(c2cccc(Br)n2)C(=O)NC)C(C)CN(C2CCOCC2)CC1C c1(CN2CCC3(C(C(N4CC(C)CC(C)C4)=O)C3)CC2)ccc2ncccc2c1 c12cccc(c1)N2.c12cn(nn1)C1CN(C1)C2=O.C(C(C)NC(=O)OC)SCC Cc1cc(N2CCSC(C(F)(F)F)C2)nc(C2C3CCCCCC23)n1 c1(C(N2CCCC(CCCCCC)C2)C(=O)NC2CC2)cc(OC)c(OC)cc1Cl CCCC(F)(F)C(=O)NC(C1CN(C(c2oc(C(F)F)cc2C)=O)CCO1)C N1(CC)CCC(C(=O)NC(C)CN(C(=O)Cc2n[nH]c(C)n2)CC)C1 C12(CNC(C(=O)O)=O)CC1CN(C1CCC1)C2=O.CC(C)(C)C(=O)NCCCN.N c1(CC)nc(C(=O)N(CC(C(=O)C(F)(F)CC)=O)CC(C)C)c(C)o1.N C1(NC(C(=O)NCCC(CCC)O)=O)CC(=O)NC1(C)C.C1(C)(C)C(=O)O1 C1(CNC(CC=CC)=O)(CO)CCN(C(=O)CNc2cccnc2C)CC1 C1(CN=C(N(C)CC(CC)(C)OC)NC2CCC2)CCC2COCCC2C1 N1(C(CC(CNC(C=CC=CC)=O)C2CCC2)=O)C2CCCC1COC2 n1(CC(N2CCC(O)(CNC(C(F)OC)=O)C2)=O)ccc(O)nc1=O Cn1nc(C(F)F)cc1C(=O)NC1CC12CC(NC(=O)C(C1CCOCC1)O)C2 CC1(C)CN2N3CC(C34CCCC4)C(=O)C12.c1(OC)cccc(Cl)c1 c1(C(N2CCN(C(COCC)=O)C(C)C2C)=O)cc([N+](=O)[O-])cnc1C N1(C(C)=O)CCCC1=CC(=O)NCCCN(C(=O)OC(c1ccc(Cl)s1)=O)C c1(C(N(CC)CC2CCC2NC(=O)C(C)(F)c2ccccc2)=O)ccc(F)cc1 C1(N(C(CN2CCN(C(c3cc(C)oc3)=O)CC2)=O)C)CCC(=O)N(C)C1 Cc1ccc(C2(O)CCN(C(=O)Nc3scnc3C(C)(C)C)C2)cn1 N1(C(C(C2CCC2)NC(c2c(C)c(=O)cc[nH]2)=O)=O)CCC2(CC(F)C2)C1 Cc1cc(C(=O)NC2CC(NC(=O)CCc3ccncn3)C23CCC3)ccc1F Cc1oc(C)c(C(N2CCN(C(c3ccc(F)o3)=O)CC2C)=O)c1C CC(C)CCC(=O)C(=O)NC(C(N1CCC(C)(O)C1)=O)C1CCCC1 CCC(C)CC(C(=O)NCC(F)Br)NC(c1sc(O)nc1C)=O c1(C(N2CCCC(CCC)(NC(=O)C=CC3CC3)C2)=O)cc(C)c(F)cc1F c1(CC(N2CC(CNC(C=C(C)C)=O)C(C)C2)=O)cc(C)ccc1N(C)C c1(C(N2CCN(C(CC)=O)CC2C2CC2)=O)cc([N+](=O)[O-])c(C)cc1C c1(C(=O)NC(C2CCN(C(C(C)=CC)=O)CC2)(C)C)cc2cccc(Cl)c2o1 C1(OC)CCC(C(=O)NCCC2(NC(c3ccoc3C(C)C)=O)CCC2)C1 C1(NC(c2cccc(OC(C)C)c2)=O)CC12CCN(C(c1cnns1)=O)CC2 N1(C(c2ncccc2Cl)=O)CCC2CN(C(=O)Cn3ccnn3)CCC2C1 N1(C(C(CC)CC(C)C)=O)CCC2(C=C(C(=O)N3CCOCC3C(C)(C)C)C2)C1 Cc1ccc(C(=O)NC2CC(NC(c3cn[nH]c3)=O)C(O)C2)cc1 CCC(CCC(=O)NC(C)(CNC(=O)C(C(C)C)c1ccncc1)CO)OC C(=O)(CC(C)CC(F)(F)F)N(C1CCN(C(C2CC2[N+](=O)[O-])=O)CC1)CC N1(C(CCOC(C)C)=O)C2CC1CN(C(=O)CC1CCC(C)(C)O1)C2 CC(CC(=O)NCC1(F)CC(NC(C2CCCN2C2CC2)=O)C1)c1cccnc1 CC1(C)CCC(Oc2ccc(Br)cc2-n2cc(CC(=O)OCC(=O)O)nn2)CC1 Cc1cc(N)cc(C(N2CC(NC(=O)Cn3cccn3)C(O)C2)=O)c1F c1(CC)ncoc1CNC(=O)C(CC1CCC1)NC(=O)CCCOC(C)(C)C c1(NC(CC(C)O)C)ccc(C(=O)Nc2nnn(C3CC3)c2C(F)(F)F)cc1 N#CC1CCCN(C(=O)NC(c2nccs2)c2ccncc2)C1 Cc1cccc2nc(C(N3CCCC3CCCNC(c3cnc(O)s3)=O)=O)cn12 c1(C(N2CCCC(NC(C3(C)C=CCCC3)=O)C2)=O)cc(C(F)(F)F)cc(N)c1 CCC(C)(CCNC(c1ccnnc1)=O)NC(=O)Cc1ccn(C)n1 C12(C(=O)NCC(C#C)CC)CCC(CN(C(=O)CCCC#CC)C1)C2 c1(C(c2nc(C3COCCO3)no2)N)ccc2cnccc2c1 Cc1cc(C(N2CCN(c3ccccc3OC(F)(F)F)CC2)=O)c(S(N)(=O)=O)s1 c1(C(=O)NCC2(O)CN(C(C=CCCCCC)=O)C2)ccc2scnc2c1 C1(NC(C=C(C)C(C)(C)C)=O)(CNC(=O)CCCN(C)C)CCCCC1C C(C(CC(F)(F)F)NC(C1(CC)CC1(F)F)=O)NC(CC(=O)NCC#C)=O C(=O)(CC(C)C(F)F)N1CC(OCC(=O)NC(CCSCC)C)C1 Cc1nc(N2CC3(CCCC3NC(c3csc4nccn34)=O)C2)ccc1C#N c1(NC(C)CF)ccc(S(=O)(=O)NCCNc2nn(C)nc2Br)cc1Cl n1(CC#C)cccc1C(N1CC(C(O)C(=O)NCC2CSCCO2)C1)=O CCCC(CNC(c1ccc(SCC)cc1)c1nnnn1C1CCC1)CCO CC1(C)CN(C(c2cscn2)=O)CCC1NCc1ccc(F)nc1C#N C1(CNC(C2CC(F)(F)CS2)=O)(CO)CCN(C(=O)COC2CC2)C1 C1(C(=O)NCC2(C(=O)OCC)CC2)CN(C(C23CCCC2C3)=O)CC2(CC2)C1 N1(C(c2cc(OC)n[nH]2)=O)CCOC(C)C1C(=O)NC(C)CCC=C(C)C O=C(C1CCc2nccn21)N1CCC(C(N2CC3OCCC3C2)=O)C1 n1(CC(=O)NCCC2(CCn3cc(Br)cn3)CCC2)ncc(O)nc1=O C1(C)(NC(c2cc(CNC(C(C)=C(C)C)=O)nn2C)=O)CCCCCC1 N1(C(C2(C#C)CCN(C(C3OC4CCC3C4)=O)C2)=O)CC(C)(C2CCC2)C1 N1(C(C2(CN3CCN(C(c4c(CC)nns4)=O)CC3)CC2)=O)CCCC(C)C1CC C1(NC(C(C)OCC=C)=O)CN(C(=O)CCc2nnc(C)n2C)CC(C)(C)C1 CS(=O)c1ccccc1C(=O)NCCN(C(C1CC12CCOCC2)=O)CC1CC1 CC1C(N(C(=O)CCn2cc(-c3cncn3C)nn2)CCO)CCCC1C c1(N2CCN(CCC)CC2)cnc2ccccc2n1.CCC(CC)C1CN1 c1(C(=O)NC(C)CN(C)C(C2(Br)CC2(F)F)=O)cc2c(ncn2C)[nH]1 c1(C(C)NCC2CCN(CC(C)C)CC2)ccc2ncoc2c1 N1(C(C2C(c3nc(=N)[nH][nH]3)CC2)=O)CCc2ccccc2C1 N1(C(C(c2ccc(Cl)s2)C)=O)CCN(C(c2cnn3ccsc23)=O)CCC1C C1(NC(C2(CCC)CCC2)=O)CC(O)CN(C(c2cc[nH]c2C2CCCC2)=O)C1 c1(CC(=O)NC(C2N(C(c3ccc(CC)[nH]3)=O)CCCC2)C)cc(F)ccc1F N1(C(COCCC#C)=O)CCC2CN(C(=O)C(F)(F)C3(O)CCC3)CCC12 c1(C(=O)NC(CN(C(=O)COCCCF)CC)C)[nH]cnc1CC c1(CNC(C(C2CCN(C(=O)C(O)c3ccsc3)CC2)C)=O)ccnc(Cl)c1 c1(SC)cc(C)c(C(N2CCOC(CN(C)C(C3(CO)CC3)=O)C2)=O)o1 N1(C(c2c(N=[N+]=[N-])cncc2)=O)CCC(C2CCN(c3ncc(F)cn3)C2)CC1 C1(NC(C(CCC=C)(F)F)=O)CS(=O)(=O)C2CN(C(=O)C(C)(C)CNC(C)=O)CC12 CC1(C)CCC(CC(=O)NC2C3CC2N(C(c2ccc(C4CC4)nc2)=O)C3)O1 c1(C(N2CCC(C)(CNC(c3nc(OC)c(C)s3)=O)C2)=O)cc2n(c1)CCC2 Cc1cc(=NC(C)c2nccs2)[nH]c(NC2CCCn3ncnc32)n1 CC1CCCCC1C(=O)NCC1CC(CNC(c2n[nH]c(C(C)(C)C)n2)=O)C1 N1(C(c2ccc(C(F)(F)F)cc2)=O)CCC(F)C(NCc2ccc(F)c(Br)c2)C1 c1(C(=O)NC(C)Cn2cc(CNC(c3nonc3N)=O)nn2)cc2c(s1)CCCC2 c1(C(=O)NC2(C)CCN(C(c3c(Cl)c(C)n(C)n3)=O)C2)ccc2c(c1)CCCS2 CC(C)C(C)CC(=O)N1CCCCC1CNC(=O)C(O)C1CCC1 C12(NC(Cc3ccc(OC)cc3Cl)=O)CCCC1N(C(c1nonc1N)=O)CC2 n1(CCCC=C)cc(NC(C23CC(F)C2C3)=O)nn1 C1(CNC(c2cnn3c2OCC3)=O)CCCCCN1C(c1ccc(C2CC2)s1)=O c1(C(C(=O)NCC(CC)NC(=O)C=Cc2cc[nH]c2)(C)C)cccc(OC)c1 C1(CC(=O)NCCN(C(=O)Cc2cc(C)[nH]n2)CC)CS(=O)(=O)C1 C1(C)(CNC(CN(C)CC)=O)CN(C(C2CCCCN(C)C2=O)=O)C(C)(C)C1 C1(NC(Cn2ncc(C)c2)=O)CN(C(c2occc2C2CC2)=O)C2(CCC2)C1 N1(C(C23C(C)OC(CC2)C3)=O)CCCCC2(CCN(C(C3CC=CC3)=O)C2)C1 Cc1n[nH]c(C)c1C(C)CC(=O)NC1CCC(NC(=O)C(=O)NCC(F)F)C1 c1(C(=O)NCC(CNC(C(N(C)C)C2CC2)=O)CO)sccc1S(N)(=O)=O Cc1nc(C(N2CCCC(NC(c3ccccc3C(C)(F)F)=O)C2)=O)[nH]c1C C(CN(C(C)C=CC(=O)OCc1ccccc1)C)(C(F)(F)F)OC C12(NC(c3onc(C)c3C)=O)CCCCC1N(C(c1sccc1F)=O)CC2 C1(NC(=O)CC2(CO)CC2)CC(F)(CNC(C2CC(C(F)(F)F)C2)=O)C1 C(=O)(C(C)CC(=O)OC)N(C1(CC(=O)N(C(CO)CO)CC)CC1)C C(CCCC(=O)NC1CCC(CCO)C1)N(C(Cc1cc(C)[nH]n1)=O)C N1(C(COC)=O)CCOC(CNC(=O)CC2(NS(C)(=O)=O)CCCC2)C1 c1(C(=O)NCCC(C)NC(CS(=O)(=O)NCC)=O)nnc2ccccc2n1 c1(C(N2CC(CNC(C3(CC)COC3)=O)N(C)CC2)=O)cc2n(n1)CC(F)C2 N1(C(C(C=C)O)=O)CCCCC(C2CN(C3CCN(C4CCCCC4)C3=O)C2)C1 c1(C2(Cc3n(CC(=C)C)c(N4CCC(CCCC)C4)nn3)CC2)c(Cl)cccc1Cl c1(C(C(=O)NC2CCCC2)N(CCC)C2CC2)cc(C2CC2)cc(C)c1 c1(CC)nc(C)c(C(=O)NC2CC3CN(C(=O)C=CC(C)(C)C)CC3C2)c(C)n1 c1(C2OCCN(C(c3csc(Cl)c3)C(=O)NCCSC)C2)ccc(C)cc1C C1(C(N2C(CN(C)C(c3cnc(O)nc3O)=O)CCC2)=O)C2CCCCCC12 Cn1ncc(Cl)c1CC(=O)NCC(C)(C)CCNC(=O)C=Cc1cnc[nH]1 C(=O)(CC(F)(F)C(F)F)NC(C1(O)CCCCC1)C(=O)N(CC(F)Cl)C N1(C(C(=O)NCCN(CCC)CC)=O)CCCC(C)C1.c1(C=O)cn(C)nc1CC N1(C(c2c(OC)ccc(I)c2)=O)CCOc2ncc(-c3cncn3C)c(C)c21 c1(C(=O)NC2C3(CN(C(C(CC=C)C)=O)C3)CCC2)ccc2c(c1)OCCN2C C1(C(N2C(C(=O)NCC3(O)CC(C)(C)C3)CCC2)=O)C2CCCCCC12 N1(C(CC2=NNC(=O)C2)=O)CCC(C2CN(C(=O)C(N3CC=CCC3)=O)C2)CC1 c1(C(=O)NCC(C)CN(C(=O)C(C)(O)C2CCC2)C)cc2n(n1)CCOC2 CCC(CCC(=O)N1CCC(C)(C(C)C)CC1)NC(C1CCCCC1(C)C)=O c1(C(=O)NCCC2N(C(C(C)OCC#C)=O)CCCC2)ccc(F)c2[nH]ccc12 N1(C(C=C(C)Cl)=O)CCC2(CC1)COC(CNC(c1cc[n+]([O-])cc1)=O)C2 c1(C(N2CC(CNC(c3c(C)nco3)=O)C(C)(C)C2)=O)cc(F)cc2ccoc12 C(=O)(CCC(C)(C)NC(=O)CC1CC(=O)NC1=O)NCC1N(CC)CC1 N1(C(C2C(C)(C)C2(C)C)=O)CCCC(C2CCN(c3ncc4c(n3)COC4)C2)C1 C(CCC[Si](C)(C)C)N(C(CCc1cc(C(=O)OC)c(C)o1)=O)C C1(CNC(C(C)NC(c2nc(C#N)cs2)=O)=O)NC(=O)CC1(C)C C(=O)(C(C)(C)CCC#N)N1CC2C(CNC(C(C)(C)COCC(F)F)=O)(CC2)C1 C12(C(N(C(CNC(COCCCCCC)=O)C)C)=O)CC3CC(C(=O)N1)C2C3 O=C1Cc2cc(C(N3CC(NC(=O)C4=CCC4)C4CCCCC34)=O)ccc2N1 N1(C(CCOC(CC(C)C)C)=O)C2CCC1CN(C(C13CC(CCO1)C3)=O)C2 N1(C(=O)NCC(c2n(C)ncc2)N2CCCC2)CC(O)CC1NS(C)(=O)=O c1(C(=O)NCC(C)(C)NC(CC2C(OCC)COCC2)=O)cccc(N)c1Br CCC(CC)CCC(=O)NC1(C(N2CCC(C(C)(C)O)CC2)=O)CC1(C)C c1(SC2C(CCN(CC(N3CCCC3)=O)C)C2)cnccn1 N1(C=O)CCC(C)(C)CC(C)(C)C1.Cc1ccc(N(C)C(=O)NC(C)(C)C)nc1 N1(C(c2ccc(CC)[nH]2)=O)CC2CCCC2(CNC(=O)Cc2nnc(C)o2)C1 C1(C)(C(=O)NCC(C)N(C(c2c(C)n(CCO)nc2)=O)C)CC(C)OC(C)C1 C1(C(=O)NCC2C(C(=O)NC(c3cc[nH]n3)C)CC2)CC(=O)CCO1 c1(SCC#C)cccc(C(=O)OCCCc2ncccn2)c1 C1(CN(C(=O)CC(C)(C)C)C)CCCN(C(=O)CSCc2ccc(F)cc2)C1 c1(C(N2CC(C(=O)NC)OCC2)=O)cc(C)[nH]c(=NC(=O)OC(C)(C)C)n1 C(C(F)(F)CCNC(=O)CCC1CCOCC1)n1cc(-c2cn(CC)nc2)nn1 C(=O)(CCCN(C)N=O)N1CC2C(CN(C(c3cc(CCC)oc3C)=O)C)C2C1 c1(C(=O)NC2C(CNC(C(F)=CC)=O)CCCC2)ccc(P(C)(C)=O)o1 C12(CC(=O)N(C)N(C(=O)C(=O)NCC)CCN(C)CC=O)CCCC1C2.C(C)(C)C c1(OC)ncc(C(=O)NCCOC2CCN(C(=O)CNC(C)=O)C2)nc1C Cc1cc(=O)c(C(=O)N(C)CCNC(=O)NCC2CCCC2)c[nH]1 C(=O)(CC1=CCN(C)CC1)NC(C1CN(C(C2CCC=CO2)=O)CCO1)C N1(C(C(N2CCC(OC(C)(C)C)CC2)=O)=O)CCCC2(C)CCCCC12 CC(=O)CCCC(C)C(=O)NCCN(C1CCCC1)C(C1CC1C1(C)COC1)=O CC1CCC=C1C(=O)Nc1cn(-c2ccc(OC(F)F)cc2)nn1 c1(NCC2COCCN(c3c4ccn(C)c4ncn3)C2)cc(F)ccc1[N+](=O)[O-] c1(NC(C(C2CCN(C(CSC(C)C)=O)C2)F)=O)ccncc1C1CC1 CC1CC(NC(=O)C=Cc2cccnc2)CCN1C(c1cnc[nH]1)=O N1(C(C(C)OCC#C)=O)CCC(CNC(C2(c3ccccc3)CCC2)=O)C(C)C1 C(=O)(N=c1ccn(C(F)F)[nH]1)C1(C(=O)OC(C)(C)C)CC(C(F)F)C1 c1(CC(=O)NC2C(NC(C3N(CC)CCOC3)=O)CC2)ccc2c(c1)CCO2 C1(C)(C(=O)NCc2n(CC)nnn2)CCCN(CC2(C)CSC2)C1 c1(NC(=O)CC2CCC(NS(=O)(=O)C3CC3)CC2)ccc(Cl)cc1CO c1(C(=O)NC(C)CNCCl)cc2c(Cl)cncc2s1.CC1CN2CCN1C(C=O)C2 CC(C)(C)CC(O)CC(=O)NC(CCC(=O)N1CC2NC(=O)OC2C1)C(C)(C)C N1(C(C=Cc2c(C)n(C)nc2)=O)CC(C)CN(C(c2cn(C)cn2)=O)CC1C CC(C)CC(O)C(=O)N1CCC(C)(NC(c2cnc(=N)[nH]c2)=O)C1 c1(NC(C2CCN(C(C3(C)N(C(C)=O)CCC3)=O)C2)=O)cc(C)c(F)cc1I N1(C(C2(NC(c3ccc(C#C)o3)=O)CC2(C)C)=O)CC2(CCOC(=O)N2)C1 C1(CNC(C2CC(=O)NC2)=O)CN(C(C2C3CC4C(C3)C24)=O)CCCO1 CN1CC(C(=O)NCC2CCCN(C(C3CCCCS3)=O)C2)NC1=O c1(C(=O)NC(CC)CNC(=O)C=C2CCOCC2)ccnc2cc(OC)ccc12 C=CCC(CNC(c1csc(CO)n1)=O)NC(C1(Cl)CC1(F)F)=O N1(C(c2cc(F)c[nH]2)=O)CC2(C1)CN(C(=O)C(F)(F)C=Cc1ccccc1)C2 c1(OC)cc(CN2CCC(NC(c3c(Cl)cccc3Cl)=O)C2)ccc1C(F)F N1(C(c2c(OC)scc2)=O)CCN(C(c2coc3c2COC3)=O)C(C)C1C Cc1sc(C(N2CC(CNC(C3CCC(=O)N3)=O)C(F)(F)C2)=O)cc1[N+](=O)[O-] C1(NC(C(C)OC2CC2)=O)COC2(C1)CN(C(=O)CCCCCn1cnnn1)C2 C1(CNC(=NCC=C)NCC(C)SC)CC(C)(C)CCC1O c1(C(N2CCCC(NC(C3(C)CCC(C)C3)=O)C2)=O)ccnc2ccsc12 c1(CC)ccnc(C(=O)N(C(C)CNC(=O)Cn2cc(C3CCOC3)cn2)C)c1 c1(C(=O)NCC2C(NC(=O)C(F)=CC3CC3)CC2)ccc2c(n1)CCC2 N1(C(C(N2CC(C(C)C)C(C)C2)=O)=O)CCC(CC(=O)NCCC(N)=O)CC1 C(C(CN=c1nnn(C)[nH]1)C(F)(F)F)NCC1(c2ccccc2Cl)CCC(C)C1 C(CCC)(C(=O)NCCCC(c1ccccc1)NC(C1(N(C)C)CC1)=O)=CCC N1(C(C(F)=C(C)C)=O)CCC(n2cc(-c3ccc(N(C)C)nc3)nn2)CC1 C1(NC(=O)Cc2cc[nH]n2)C2CCC1N(C(=O)CCc1cccc(F)c1Cl)C2 C(c1ccccc1F)=CC(=O)N(CC(CNC(C(C)N(C)C)=O)(C)C)C CN1CCC(C(N2CC3CCC3(CCNC(=O)Cn3cnc(=N)[nH]3)C2)=O)S1(=O)=O CCC(C)C(=O)C(=O)NC1CCCC1NC(=O)CC1C(=O)N(C)N=C1C CN1CCC(C)(NC(N2CCCC2Cc2cc(F)ccc2F)=O)CC1 C(=O)(C1=CCCCO1)NCC1CC(OC)CN1C(c1ccc(N)c(Br)n1)=O c1(OCOC)ccc(-n2nnnc2N(C)CCC2CCC(OC)CC2)c(OC)c1 n1(CC(=O)NC2CC(C(C(=O)NCC3(SC)CC3)F)C2)c(O)nnc1O C1(NC(c2ccccc2F)=O)CC2CC(C1)N(C(c1ccn3ccccc13)=O)C2 C=CCCCCC(=O)N1CCC(C=CC(=O)NC(COC)C(C)C)CC1 C1(C(N2CCCC(N3CCOCC3)CC2)=O)Cc2nccn2C1 Cc1cnc(C=CC(=O)NCC2CCCN2C(=O)C(C(C)C)c2cccnc2)[nH]1 C1(CC(=O)Nc2c(C(C)(C)C(F)(F)F)cccc2)CC2(CC2)CN1C(=O)CN c1(NC)cnc(C(N2CCC(C)(NC(=O)CN(c3ccccc3)C)C2)=O)cn1 CN1CC(F)(CNC(=O)CNC(c2cc(C3CC3)on2)=O)C1 c1(CCNC(C2CCN2S(=O)(=O)C(F)(F)F)=O)cc(Cl)cc(Cl)c1 CC1OCCN(C(=O)NC2CC3CC(O)C(C2)C3)C1(C)C N1(C(C=CCOC)=O)CC2(NC(c3ccc(S(N)(=O)=O)cn3)=O)CCCC2(F)C1 N1(CC(N2C(C(C(=O)NCCCCCSC)(C)C)CCC2)=O)CCNC(=O)C1 N1(CC)OCC(NC(c2occc2CNC(C2COCCC2C)=O)=O)C1=O N1(C(c2nc(C)oc2)=O)CC2CN(C(=O)C(C)(F)c3ccon3)CC(C1)O2 C1(C(N(CCCNC(CC(C)OC)=O)C)=O)CC(=O)N(c2cnn(C)c2)C1 C(CC(C(C)(C)C)NC(c1cn(C(F)F)c(C)n1)=O)N(C(COC(CC)C)=O)C C1(NC(CC2N(C(c3n(CC)ccn3)=O)CC2)=O)CC2CC(O)C1C2 C(=O)(C(C)C(C)(C)C)N1CC=CC(NC(C(C(C)C)c2ccc(F)cc2)=O)C1 C12CC3(CCN(CC3)C1=O)C2.c1(OC)cc(C(=O)Nc2csnn2)ccc1O CCC(CCCC(=O)NCC(C)(CC)C(N)=O)NC(c1nnsc1N)=O c1(NC)cc(C(=O)NC2CC(CNC(=O)C(F)C3CCOC3)C2)cc(Cl)n1 Cc1ncccc1C(N1CCC(C(C)(C)NC(=O)Cc2ccccc2C)CC1)=O C(CCC(O)C(=O)NCCN1CC=C(C)CC1)NC(C1(OC(C)C)CCC1)=O CCC(O)C(C)C(=O)NCC(CC)(CC)NC(c1nccn1C)=O c1(CC)nocc1CN(C(=O)CCOC1CN(C(=O)CN(C2CCC2)C)C1)C c1(C(C(=O)NC(C)CC(C)NC(=O)CCCC2CC2)O)cc(F)cc(F)c1 C(=O)(CC(CC(N)=O)CC(C)C)NCC(CC)(CC)NC(=O)COC1CC=CC1 C1(C2CCN(C(=O)C=CCO)C2)(NC(CN2CCCCC(OC)C2=O)=O)CC1 c1(N2CCC(C(C)C)C2)nc(NC2C3COCC23)nc2c1COC2 CCC(CCCC(=O)N(CC)OC1CC1)NC(=O)C(F)(F)C(O)C(C)C c1(C2CC(OC(C)C)C2)nc(C2CCCC2)nn1Cc1cccc(Br)c1 C1(CC(N2CCCC(CCNC(C3C(C)SCCC3)=O)C2)=O)CC2(CCC2)CO1 N1(C(Cc2c(C)cnn2C)=O)CC2CCCC2(NC(c2ccnc(S)c2)=O)C1 c1(C(=O)NCC2N(C(c3cc(C)on3)=O)CCC2C)c(C)sc2ccccc12 CCC(C)(CNC(=O)COCC(=O)OC)C(=O)N1CCCC(C)(CN(C)C)C1 N1(C(C23C(C)(C)C(CC2)C3)=O)CC(O)(C2(CNC(C3(O)CCCC3)=O)CC2)C1 C(CC(=O)NC12CC(C1)N(C(c1ccnn1C1CCC1)=O)C2)(C(F)(F)F)OC c1(C(C)C(=O)N(C)C)ccccc1S(=O)(=O)N(C(C)CC(=O)O)C C1(C2CC2)(C(=O)NCC2CCN(C(C(C)OCCC=C)=O)C2)CCOCC1 C1(O)(CC)CCN(C(=O)C=CC(C)(C)NC(=O)Cc2ccccc2C)C1 C(=O)(CC(N=c1cc(C)nc(N(C)Cc2ccc(Br)o2)[nH]1)C1CC1)NC C1(NC(C2CCC23CCC3)=O)CCCC12CN(C(c1cnc(S)nc1)=O)C2 c1(CC(=O)NC2C=CCN(C(C(n3cc(Cl)cn3)C)=O)C2)ccc2c(c1)CCO2 Cn1nccc1C1CC(NC(c2csc(Br)c2)C(=O)O)C1 N1(C(=O)COc2ccccc2O)CCC2OCCN(C(=O)CCC3CC3)C2C1 C12(CC(=O)NCCC(C)NC(C3CCCC3c3cnn(C)c3)=O)COCC(C1)C2 c1(C(=O)NC2CC(CC)(CC)N(C(c3snnc3C)=O)C2)cc2c(nn1)CCC2 c1(OC)c(C(=O)NCCNC(=O)C(C)Cc2cnco2)cc(F)cc1F N1(C(c2c(C)nc(CO)o2)=O)CC(NC(C2(F)CC3(CCC3)C2)=O)CC2(CC2)C1 C1(OC)CN(C(=O)CCn2nc(C)nc2C)CC1NC(=O)COc1cccc(F)n1 CN1CCN(C(=O)Cc2cncs2)C(CNC(C2CCCCN2S(N)(=O)=O)=O)C1 CN1C(=O)OCC1C(N1CCC(CCC(=O)NCCCCCF)C1)=O c1(CC(=O)NCC(C)N(C)C(c2cc[nH]c(=N)c2)=O)c(Cl)cccc1Cl C(C(CC(=O)NCC(c1cccs1)O)OC)NC(C=CCOC)=O c1(C(C)C(=O)NC2CC2CNC(=O)Cn2cc(Cl)cn2)c(F)cccc1F C(=O)(CC(C)C(C)(C)NC(c1cc(C)c(CC)o1)=O)N1CCC(C#C)C1 C#CC1(O)CCN(C(=O)C(c2ccnn2C)NC(C2CC3(CSC3)C2)=O)CC1 Cc1ccnc(C)c1C(N1CCCC(N(CC(N)=O)C2CC2)CC1)=O C(=O)(C(C)(C)CC1CCCCC1)N(CC(CNC(C1C(CCC)C1)=O)O)C C1(CNC(CC2C(CC)C2)=O)CCC(CNC(c2n[nH]cc2C2CC2)=O)O1 C1(C(=O)OC)CC2(CCC2NC(c2cnn(-c3ccccc3)n2)=O)C1 CCC(CC(=O)N(CCCNC(=O)C(COC)OC)CC)C1CC1.C1CCCC1 Cc1cc(CNC(=O)C(CCC2CC2)NC(=O)Cc2cccnc2)cnc1C c1(NC(=O)OC)cccc(C(=O)NCCCN(C(=O)C(F)(F)C2(O)CCC2)C)c1 c1(NC(C(c2cccc(Br)c2)(C)C)=O)cc(O)c(Cl)cc1Cl.C12CCN1C2=O N1(C(C(C(=O)OCC)F)=O)CCN(c2ncnc(CC)n2)CC1C c1(C(=O)N(CC(=O)O)Cc2cn(C3CCC3)nn2)cc(Br)c(C(C)(C)C)s1 CC1(NC(C2CC=CCN2C(=O)CN2CC=CC2)=O)CC(F)(F)C1 N1(C(C(C)N(C(=O)C=CC2CCOCC2)C2CC2)=O)CC=CC1(C)C S(=O)(=O)(c1cc(Br)ccc1Br)N1C(C(=O)Nc2ncc(Cl)nc2Br)CC(O)C1 c1(CC)ccc(F)c(C(=O)NC2CCC2NC(c2ccc(CN=[N+]=[N-])o2)=O)c1F c1(C(N(C)CC2(NC(c3sccc3C(C)(C)C)=O)CC2)=O)ccc(CO)cc1 C1(C(=O)NC2C(C)CN(C(C3NC(=O)CC3C)=O)C2)CNC(=O)CC1C n1(CC(=O)N(CC=C)Cc2ncccn2)ncc2cccc(Br)c2c1=O Cn1nc(C(=O)NCC2CCCN2C(=O)CCn2ccnc2)cc1O c1(OC)cc(NCCC2CCN(C(c3cc(C(C)C)n(C)n3)=O)CC2)ncn1 c1(C(N2CCCC(CN(C(=O)CC(O)C3CC3)C)C2)=O)cc2ccccc2n1C CC(=O)C(C)(C)CC(=O)N(c1cc(C)ccc1C)C(C)=O CC1CCn2ncc(C(N3CCC(C(C)NC(=O)C(C)(C)O)CC3)=O)c2C1 C1(C)(NC(CC(C=C)C)=O)CCN(C(=O)COc2ccc(Br)nc2)CC1 C1(O)(C(N(C)CC2CN(C(C3CCC(C)CC3)=O)CCO2)=O)CCCC(C)(C)C1 c1(C(N(CCOC)CCNC(=O)CC(C)n2cccc2)=O)cc(C#N)c[nH]1 N1(C(C(C=C)O)=O)CCC(O)(CCNC(c2cc(C)on2)=O)C1 C(CN=c1nc2scnc2c(Nc2cncc(C)c2)[nH]1)(c1ccsc1)N(C)CC CC1CC2(CCC2)CN1C(=O)C(=O)NC1CCC(C)(C)CN1 N1(C(C(F)=CC)=O)CCN(CCCCCNC(c2ccc(COC)s2)=O)CC1 C(=O)(C(O)CCc1ccccc1)NC(CC(C)NC(CCCC)=O)C CC1CN(c2ccc(C3CC3C(N3CCC4(CC4)C3)=O)cc2)S(=O)(=O)C1 N1(C(C2N(CC)CC2)=O)CC2CC2(CNC(=O)Cc2cc(Cl)sc2Cl)C1 C(=O)(C1=C(Cl)CCC1)NCC1C(NC(c2cn(C(C)(C)C)nn2)=O)C1 c1(CC(=O)NCCC(C)(C)NC(C#CC2(C)CC2)=O)c(F)c(F)cc(F)c1F c1(C(N2CC(CNC(CS(CC)=O)=O)C2)=O)oc2c(Cl)cccc2c1C C(=O)(C(C)C(C)NC(=O)CC1CC(N(C)C)C1)NCCC=C(CC)C n1(CCCCNC(c2ccn(C)n2)C)cc(C2(C(=O)NN(C)C)CC2)nn1 C(=O)(C1=NOC2(CCC2)C1)NC(C(=O)N1C(CCC)CCC1)(C)CO C12(C(=O)NCC(CC)NC(C3(CC(C)C)CCNC3=O)=O)CC(C)(CO1)C2 c1(C(C(=O)NCC(F)F)N(CC(C2CCC2)OC)C)cccc2cnccc12 C1(C(=O)Nc2ccc(C)c(Br)c2C)CCCC12CCN(C(=O)C(C)(C)F)C2 c1(CN2CC(CC(=O)OC)N(C(=O)C3=C(Cl)CC3)CC2)c(C)cc(C)nc1O Cc1ccc(CCC(=O)NCC2COC(CNC(c3ccsc3Cl)=O)C2)s1 C(CCNC(c1cocn1)=O)(C(=O)NCC1CC12CC2)OC N1(C(C(C)CF)=O)CCN(C(c2cccc(C(F)F)c2)=O)CC1C1CCC1 N(C(=NCCCCl)NCC1CCCCC1NS(C)(=O)=O)C1(C#C)CCC1 C(=O)(CC(C)(O)COC)NC(C1CCN(C(c2cc(C(=O)OC)sn2)=O)CC1)C Cc1cc(CC(=O)NC(C2CCN(C(c3conc3C)=O)C2)C)cc(C)c1 c1(C(C(=O)NC2(C(=O)NC(C3CCOC3)CC)CC2)SC)ccccc1 N1(C(CC2N(C(C3CC(=O)NC3)=O)CCC2)=O)CC2CCC(O)C(O)C12 N1(C(c2c(CC)[nH]cc2)=O)CCCC(CC(=O)NCC2(C(C)(C)OC)CC2)CC1 N1(C(C(OC)OC)=O)CC2(CCC2)CC1C(=O)NC1CCCC1CN(C)C N1(C(c2coc(CO)c2)=O)CCC2CCN(C(C3CCS(=O)(=O)CC3)=O)C2C1 C1(C(=O)NC(C)CCN2CCCC2)C2CCN(C(C3(C(N)=O)CC3)=O)CC12 Cc1nn(CC(N2CCC(C)(CNC(c3ccns3)=O)C2)=O)c(C)c1[N+](=O)[O-] Cc1cc(F)ncc1C(=O)NCC1(F)CC(NC(c2[nH]ccc2C)=O)C1 N1(C(C2(OCC)CCOCC2)=O)CCC2(CC1)CCN(C(=O)C#CC1CC1)C2 c1(NC2C(F)(F)CCN(C(CCN(C(C)=O)C)=O)C2)ncnc2c(F)cccc12 N1(C(C(=O)OC(C)C(=O)NC2(C)CCC2)C2CCCC2)CCOCC1.C(C)ON CC(C(=O)N1CCCC1C(=O)N(CCCN(C)C)C)S(N)(=O)=O c1(C(N2C(C)CC(NC(CC=C(C)C)=O)C2)=O)cc(C)c(Cl)cc1Cl C1(CC)CN(C)CCN1C(=O)C(=Cc1ccccn1)F C1(CCC)CN(C(C2(CC)CCCC2)=O)CCN1C(=O)CCc1ccc(O)cc1 c1(C(=O)NCC(CCNC(CC(C)C2CC2)=O)O)c[nH]c2cccnc2c1=O c1(C(=O)NC2C(CN(C)C(C3(F)CCC3)=O)CCC2)ccc(O)nc1Cl C1(NC(C2(c3ccccc3Cl)CCC2)=O)CCOCC1NCc1ccncc1 CC(C)(C)CC(O)C(=O)N1CCC(NC(c2ccc(C3CCCO3)[nH]2)=O)C(O)C1 C#CC1CN(C(=O)CC2CCCN(C(c3c(C)nsc3C)=O)CC2)CCO1 C=C(C)C(CC(=O)NCC(C(=O)NC1(CO)CC2CC2C1)C(C)O)OCC N1(C(c2ccc(OC)c(F)c2)=O)CCCC2(CCCN2Cc2cnc(Br)s2)C1 CC(C)C(N)CCNS(=O)(=O)C1CC1c1ccccc1 c1(OC)ccc(F)c(C(N2CC(F)CC2C(=O)Nc2ccc(F)cc2O)=O)c1 c1(C(=O)O)cccc2nccn12.N1CCC(O)(Cn2cc(CO)nn2)C1 C1(CC)(NC(C2(COCCNC(c3cnn(C4CC4)c3)=O)CCC2)=O)CCOC1.N N(C(=NCc1nc(C)cs1)NCC(=O)OC(C)(C)C)CCOC.C(C(F)F)SCC C(CCCCC(=O)N(CCCNC(C1CCC2C1C2(F)F)=O)CC)OCC C1(C(=O)NC2(C)CN(C(c3cccnc3S)=O)C2)CC(O)C(F)C1 C=CC(C)CC(=O)NC(C)CCNC(=O)CC1CCC1 C(=O)(C1CCc2cccnc21)N1CC(NC(c2c(CC)non2)=O)C(N=[N+]=[N-])C1 n1(CC)nc(C(=O)NCC(O)CNC(=O)CNC(c2ccc(C)cc2)=O)c(C)n1 c1(CC(=O)NCC(CCNC(COCCOCC)=O)F)c[nH]ccc1=O N1(C(C=CC(C)C)=O)CC2(CCC(CNC(C3(C)CNC(=O)C3)=O)O2)C1 c1(C(=O)NCC(C(N2CC=CC(OC)C2)=O)(C)C)cn(C)ccc1=O N1(C(COC)=O)CC2CC(NC(C3(C(C)C)CCC3)=O)CC2C1 C(N=c1nc2sccc2c(NCc2cncs2)[nH]1)c1scc(C(C)C)n1 N1(C(C(=O)Nc2c(C)cc(F)cc2)C)CC2CC(N)CC1C2 C(=O)(C1=CS(=O)(=O)CCC1)NC(C)C(=O)NC(c1ccccn1)C C(=O)(CCCCCCc1ccccc1)OCC(=O)NC(c1ccc(Cl)c(Cl)c1)=O c1(C(N(C(C)CNC(C2(O)CCC2)=O)C)=O)cc(Cl)nn1C CCCCC(O)CC(=O)NC1CC2C1CCN2C(=O)CC=C(C)C N1(C(=O)NCCCCOC)CC2CCCN(C(=O)C(C)OC3CC3)C2C1 C1(C)(C(N(CC(=C)C)CC)=O)CN(C(=O)C(C#N)CC)C(C)(C)C1 C1(C(=O)NC2CC(NC(c3ccnc(OC)n3)=O)C2)OCCOC12CCC2 c1(-c2c(C(N3CC(CO)CC3=O)C)cnn2C)n[nH]c2ccc(C(=O)O)cc12 C1(NC(=O)Cn2cccn2)CN(C(c2ccccc2F)=O)CC1CO c1(OC)cc(C(=O)NC2CCCC2NC(=O)CCN2CCC2)ccc1O N1(C(C2(c3cccc(OC)c3)CC2)=O)CC2CN(CCN(C)C)CC2C1 C1(NC(Cc2cc(CC)no2)=O)CCCC(NC(c2cnsn2)=O)C1 N(C(=NCCCF)NCC1CC1F)Cc1ccc(C2(C)CC2)o1 c1(C(=O)NCC2(F)CCC(CNC(COCC)=O)C2)ccc(C)c(Cl)c1N c1(C(=O)NCC2CN(C(c3cnc(C4CCCO4)s3)=O)C2)cccc2c[nH]nc12 CCCC(CC)CC(=O)N1CCN(C(C23CCC(F)(CC2)C3)=O)CC1C(C)C N1(C(C2(C=C)CC2)=O)CCC(NC(=O)CC2(C(F)F)CC2)C(C)C1 CCC(C(=O)N(CC)OCc1ccccc1)C(N1CCC(C)CC1C)=O c12ccn3ncc(c3n1)S(=O)(=O)N2C.C1(CNC2CN(C3CC3)C2)CCCC1 CC(C)(C)C(=O)C(=O)N1CCC(n2cc(COCCOCCO)nn2)C1 N1(C(=O)C(C2CCCCCC2)O)CCOC2CCNCC12 Cc1nc(NCCSC2CCCOC2)cc(N2CCC3(CCC3)C2)n1 C1(C2CCCC2)(C(N2CCC(c3cn(CCCCCCO)nn3)C2)=O)CCNC1=O N1(C(C2CN(C(Cc3c(C)ncs3)=O)CC(C)C2)=O)CC2(CCC(O)CC2)C1 c1(C(c2nnnn2CCOCCNC(C)=O)NC(C)=O)c(F)cccc1F c1(OCC)c(OC)cc(N2CC(C(=O)NCCN3CC4CC4C3)CC2=O)cc1Br C1(C)(C(=O)NCC2(CO)CC(C)C2)CN(C(C2CCCSC2)=O)C(C)(C)C1 Cc1ccc(N)c(C(=O)N(C2CC(NC(=O)Cc3sc(C4CC4)nc3C)C2)C)c1 c1(CNC(COCCCC#C)=O)cc(C)c(C(=O)N(CC(O)CF)C)o1 N1(C(C(C=C)O)=O)CCC(C)(C)C(CNC(=O)CCN2CCCC2)C1 N1(C(c2c(C)ocn2)=O)CCn2cc(C(=O)Nc3cnc[nH]3)nc2C1 C(=O)(C1=CC2(CCOC2)C1)NC1C2CN(C(C(c3c(C)ccc(C)c3)=O)=O)CC21 c1(C2C(C(=O)NCC3CN(C(C4(C(C)O)CC4)=O)C3)C2)ccc(N(C)C)cc1 C1(CNC(C(C)NC(CC)=O)=O)CCCCN(C(=O)CC2CC(=O)NC2=O)C1 C1(C(=O)NCC(CC)O)COCCN(C(=O)C(C2CCOCC2)O)C1 Cc1c(C(=O)NCCCN(C)C(C2(C)CC2)=O)nnn1C CN1C(=O)CCCC1C(=O)NC1CCC12CN(C(=O)COC1(C)CCC1)C2 CN=C(NCCF)NC1CCN(C(=O)C(C)C)C1.C1(C)CN1 C(=O)(C1CCS(=O)(=O)c2ccccc21)N(C)CCNC(=O)C(O)CC(F)F c1(C(N2CCC(CN(C)C(C3CCNC3=O)=O)C2)=O)cccc2ccncc12 CON=C(C(=O)NCC1CC(CNC(=O)C(C)CC2CCC2)C1)c1ccco1 C1(C(=O)NCCCC=CC)CN(C(=O)CCSC)CC1(C)C N1(C(c2nc(COC)sc2)=O)CCC2(CCCN2C(=O)Cc2cc(C)ns2)C1 c1(C(=O)NC2CN(C(c3ccsc3)=O)CC3(CC3)C2)cccc2cc(O)ncc12 N1(C(c2cccc(C)n2)=O)CC2CC1CN(C(C1COCCN1C)=O)C2 C(=O)(CC1=CCOCC1)NCC(CN(C(c1c(OCC)cccc1)=O)C)O N1(C(C(C)CC(C)(C)C)=O)CC2(CCCCN2C(C2CC2CN(C)C)=O)C1 c1(CN(C(C)C(C)C)C(c2cccc(OC)c2)=O)nccc2ccccc12 C1(NC(c2coc(CO)c2)=O)CC2CCC1CN(C(=O)C(C1(O)CCCC1)F)C2 CC1(C)CC(CNC(N2CCC(Cn3cccn3)C2)=O)OC(=O)N1 Cc1noc2nc(C(N3CC(NC(c4ccnnc4S)=O)C(C)(C)C3)=O)ccc12 CCC(C)(C)C(O)C(=O)N1CCN(C(=O)Cn2cnc([N+](=O)[O-])c2)C(C(C)C)C1 N1(C(c2occ(C)c2)=O)CC2CN(C(c3cccc(C(C)C)c3)=O)C2C1 N1(C(C2CCC(CCCC)O2)=O)CCC(N=c2[nH]nc(C3CC3)o2)CC1C c1(C(N2CCC(OCC(C)C)C2)=O)ccnc(CNC(C2CC2C(F)F)=O)c1 C1(CN(C(=O)CSc2nnnn2C)CC)CCCN(C(c2ncn(C)n2)=O)C1 CC1C(C(=O)O)CCN1Cc1cc(Br)c(Br)s1 C12(CNC(CCC=CC)=O)CC1CN(C(c1cnn(C)c1C)=O)C2 C1(NC(=O)CSC2CCCOC2)CN(C(=O)CCC2CC2)CCC1CO C(c1cc(Br)cs1)=CC(=O)N(C(CNC(CC1(CSC)CC1)=O)C)C c1(C(=O)NCC2CN(C(c3nc(C)sc3)=O)C2)cc2ccccc2cc1N C1(COC)CN(C(c2ccc(C(C)(F)F)cc2)C(=O)NC(C)(C)C)CCO1 c1(SC)nc(Cl)c(C)c(=NC2CC(CNC(=O)C3=CCCC3)C2)[nH]1 C1(C)(CNC(c2cc(CC)c(C)s2)=O)COCCN(C(=O)C(C)CC(F)(F)F)C1 C1(C(=O)NC(C)CCCCO)CCCN(C(=O)CCn2cccn2)C1C c1(CNC(c2nc(C(=O)NC(C)CCO)sc2)=O)c(F)cccc1F N1(C(C2(OC(C)=O)CC2)=O)CCC2CCN(C(c3nc4ncccn4n3)=O)CC12 N1(C(c2[nH]cc(C)c2)=O)CCC(C)C(CNC(C2(n3cncn3)CC2)=O)C1 N1(C(c2ccc(C)o2)=O)CC(CNC(=O)CCCOc2cccnc2)CC1(C)C c1(C(=O)NC(C(C)C)CO)cnn2cccc(-c3ccccc3)c12 CC1(C)CC(C(=O)NC2(CNC(=O)CN3CCCCC3=O)CC2)=NO1 N1(C(=O)CC2CCC(OC)CC2)CCCC(O)(CNC(C2CC(CC)(CC)C2)=O)C1 CC(C)(C)C(CNC(C1(CNC(=O)Cc2nc(=N)[nH][nH]2)CCC1)=O)CO C(=O)(C1=CC2(CCOC2)C1)N(C1CN(C(c2cnc(Cl)cc2Cl)=O)CC1(C)C)C N1(C(CCCCCC)=O)CCN(C(c2cn(C(C)C)nc2C2CC2)=O)CC(O)C1 C1(C(N(C(C)CNC(=O)COCCO)C)=O)CCC(NS(N)(=O)=O)C1 C1(C(=O)NC(C)CN(C(C2CC2c2ccn(C)n2)=O)C(C)C)CCC2CC2CC1 N1(C(c2c(COC)nn[nH]2)=O)CCN(C(C2CCCO2)=O)CC1C(F)F c1(C(C(=O)NCc2ccc(OCC#C)cc2)(C)O)ccc(Br)cc1F n1(CC(=O)NC2CCN(C(C3C(=C)C3)=O)C2(C)C)cnc2c(cnn2C)c1=O C(=O)(C1(C)CCCc2ccccc21)NCC1CN(C(C(C)=CC2CC2)=O)CC1O n1(CC)nc(Br)nc1C(N1CCCC(CC#N)C1)C(=O)NC1CCOC1 O=C(C1=NN(C2CCCC2)C(=O)CC1)OCCNC(=O)C1CC1 Cc1cc(CN2CC3C(C2)N3C(=O)Cc2c(C)cccc2C)c([N+](=O)[O-])c(C)c1 N1(C(c2c(C)sc(Cl)n2)=O)CCN(C(c2ccc(F)c(C(C)C)c2)=O)C(CF)C1 Cc1ccc2nc(C)c(C(=O)NCC3CCN3C(=O)CSCC(F)(F)F)cc2c1 c1(-n2ncc(C(=O)NC(C(C)NC(=O)CC3C=CCC3)CO)c2)ccc(O)cc1 N1(C(C(C=C)(C)O)=O)CCN(C(=O)CCNC(=O)NC)C(c2cccnc2)C1 C1(CC)C(C(=O)Nc2ccc(OC)cn2)CCCN1C(=O)C(C)c1ccco1 c1(C(=O)NC(C2(O)CN(C(c3cc(C4CC4)no3)=O)C2)C)cnc2sccn12 c1(N2CCC(C(N(c3ccc(C(C)=O)cn3)C)=O)C2)cccc2nccn12 Cc1oc2ccccc2c1CC(=O)NCC(=O)NC1CCCN(CC2CC2)C1 C1(CC(=O)NC(C)CCNC(=O)CSCc2ccccc2)SC2=NCCN2C1=O C1(CC)CN(C(c2cccc(Cl)c2OC)=O)CCC1NC(C1(CF)CC1)=O C1(NC(C2CN(C(C)C)C2)=O)CC2CC1N(C(c1cc(C(F)F)n(C)n1)=O)C2 C1(COC(=O)NCC(C(=O)OC(C)(C)C)F)COC2(CCCC2)C1 c1(NC(=O)OC)ccc2c(c1)CCN(C(=NCc1ccncc1F)NC1CC1)C2 C1(CC)CC2CCC(C1)N2C(=O)Cn1nc(C2CC2)n(C)c1=O c1(OC)ccc(F)c(F)c1C(N1CCOCC1C(N1CC(C)OCC1C)=O)=O CC1CN(C(=O)OC(C)(C)C)C(CNC(c2nccc(OC(F)F)n2)=O)CO1 C1(C(N(C2CCN(C(=O)CCCN(C)C)CC2)CCC)=O)COC2COCC12 C1(NC(c2ncc(N)nc2)=O)CC2CC(NC(=O)Cc3nc[nH]n3)CC12 c1(OCC(N2CC(CC)C(NC(c3ccoc3)=O)C2)=O)cccc(F)c1F Cc1cc(NC(C2C(NC(c3cc([N+](=O)[O-])n[nH]3)=O)C2(C)C)=O)cc(Cl)c1 N1(C(c2n(CC)cnn2)=O)CC(NC(=O)Cc2ccsc2C)CC(C)C1 N1(C(CC(=O)NC(C)C)=O)CCCN(C(=O)COCc2ccccn2)C(C)C1 c1(C(=O)NC2C(CNC(c3cc4sccc4s3)=O)CCC2)nnc2n1CCOC2 C(=O)(C#CC1CC1)NC(c1ccccc1)C(C)NC(c1c(CC)ncs1)=O C1(C(=O)NC2(C(=O)OC)CC(CO)C2)CCCC(C(=O)NCC(C)(C)O)C1 CC1CN2CCN12.C12(C=O)CC(CO)(CN1C(C1(C#N)CCCOC1)=O)C2 C1(C(N(CCC)CC)=O)CCC(C)(C)N(C(=O)CN2CCC(OC)C2)C1 S(=O)(=O)(CCCN1CCOCC1)N(C)C(c1ccc(Br)cc1)C1CC2CC1CN2 c1(OC)cc(C)c(C(N2CC(N(C)C(c3cncc(CC(C)C)c3)=O)C2)=O)cn1 c1(C(=O)NCC2N(C(=O)OC(C)(C)C)CC(O)C2O)cc(F)cc(Cl)c1N C=CC1COCCN1C(c1cc(C2CC2)[nH]n1)C(=O)NCCCC1CC1 c1(OC)c(Cl)cc(C(N2CCN(C(c3cnc[nH]3)=O)CC2CO)=O)c(OC)c1N N1(C(C(CC)F)=O)CCC(C2CC(c3ccccc3)(NC(=O)CN(C)C)C2)CC1 C1(NC(c2cc(Cl)on2)=O)COCCN(C(C2(O)CCSC2)=O)C1 N1(C(C(CCCC)N)=O)CCCC2CN(C(=O)C(=O)NC)CC12 C1(C(=O)NCC2C(C3CC3)CCN2C(c2cccnn2)=O)CCCCC1C1CC1 CC(C(=O)N1CCCCC1CCN(C(=O)C=C(Cl)Cl)C)S(C)(=O)=O C#CC1(C(=O)NC(C)CCC(C)C)CCN(C(=O)C=CC(F)F)C1 C1(C(=O)NCCC2CCCN2C(c2ccoc2)=O)C(C(F)(F)F)C1[N+](=O)[O-] CCC(CNC(=O)CCN(CCCO)C(C1CCC2CC1CO2)=O)C(C)(F)F c1(C(N2CC(F)(CNC(C(C)OCCOCC)=O)C2)=O)cn(C)c(=O)n1C N1(CC(C(C)(C)C)CO)CC2(CCOC(=O)N2)C1 Cc1ccc(Br)cc1C(=O)NCCC1C(C)CCCN1C(=O)C1=CCOC1 Cc1nn(C(C)C(=O)NC2(CO)CN(C(=O)C(F)(F)CO)C2)c(C)c1[N+](=O)[O-] N1(C(c2c(OCC)scc2)=O)CCC(CO)C(NC(c2cc(O)nn2C)=O)C1 C(CC(CC)C(=O)NCCn1ccc(C(=O)NCC2CC(O)CCO2)c1)=CC c1(C(C)NC2CCN(c3ccc(C)nc3)C2)cc(Br)ccc1Br C12(C(N3CC(O)(CCNC(C=CCOC)=O)C3)=O)CCCC1CC(F)(F)CC2 CC1CN(C(=O)Nc2ccon2)CC(C)N1C(c1cccc(F)c1F)=O C1(C(N2C(CNC(c3cncc(C#N)c3)=O)CC2)=O)CC2CCCC(C1)C2 CN1CCC(n2cc(C3(OC(=N)O)CN(C(=O)CO)C3)nn2)C1=O c1(CC(=O)N(C(CNC(CSCCC)=O)C)C)csc2ccc(C)cc12 Cc1cc(Cl)c(C(N2CCCN(C(c3cc4c(ccn4C)[nH]3)=O)CC2)=O)cc1F N1(C(C)C(F)(F)F)CCN(C(=O)C(CCOCCO)NC2CCCSC2C)CC1 Cc1ccc(C=CC(=O)N(C)CC2CCCN2C(=O)C=Cc2ccncn2)cc1 CC1ON=C(C(=O)NCC(O)CNC(c2ccc(C(C)(C)C)c(Cl)c2)=O)C1C C#Cc1cccc(NC(=O)C(F)CC2CN(C(C3(Cl)CC3(F)F)=O)C2)c1 c1(C(=O)NC(CNC(C(=COCC)C#N)=O)C)cc2ccccc2s1 C(C(F)(C(=O)NC)C(C)C)NC(C1(CC)CCCO1)=O.C12CC(C1)C(=O)N2 CC(N(C)N1CCCC(C)C1)C12CC1CCCN2CC#N CC1CCN(C(c2ccn(-c3cccnc3)n2)=O)CC1NC(=O)CC1CC1(C)C CN1Cc2ccc(C(N3CC4CCC3CN4C(=O)CNC(=N)N)=O)cc2C1 N1(C(C=C(C)Cl)=O)CC(C)N(C(c2ccc(-n3ccnc3)cc2)=O)CC1C Cc1cc(C(=O)NCCCC(C)(C)NC(=O)C(O)C(C)C)ncc1N Cc1ccncc1CC(N1CCCC1CN(C(C1CC1(C)Br)=O)C1CC1)=O C(CCC(=O)NCc1nocc1C(=O)NCC(C(C)C)OC)OC C(=O)(C1CC=Cc2ccccc21)N1C(CCNC(C2CC(C)C2)=O)CCC1 N1(C(C2(CNC(Cc3cn(CC)nc3)=O)CCCO2)=O)CCOC(C#N)C1 c1(C(N2CCC(NC(c3cnsc3)=O)C(CO)C2)=O)cc(F)cc2nn[nH]c12 c1(CN(C(c2ccc(OCC)cc2)=O)C)ccc(C(=O)OC)c(OC)c1 N1(CCC)CC(C(N2CCCC(N(C(=O)CCc3cnc[nH]3)CC)C2)=O)CC1=O CCC(C)CC(C(=O)NC1(CSC)CC(O)C1)NC(c1cncn1C)=O Cc1cc(N2CCC(CNC(c3cc4n(n3)CCC4)=O)C2(C)C)nc(C(C)C)n1 N1(C(c2n[nH]c(C)c2F)=O)CCCC2(C1)CN(C(C1CCC(=O)NC1)=O)C2 C12(C(N3C4CC(NC(COC)=O)CC3CC4)=O)CC3CC(C)(C1)CC(F)(C3)C2 C=CCCC(C(=O)NCC1(C)CNC(=O)O1)NC(C1CC1=C)=O C1(C(N(C2CCCCC2)CCNC(C2(C=C)CC2)=O)=O)CN2CCC1CC2 C(CCCCC(=O)N(CCNC(C1CCCSC1C)=O)C(C)C)NC(C)=O N1(C(Cc2nnc(C)o2)=O)CCOC(CN(C)C(c2c(C)noc2C)=O)C1 N1(C(c2cc(C(C)C)[nH]c2C(C)C)=O)CC(C)N(C(c2coc(CO)c2)=O)CC1C Cc1cc(N2CCC(C)(C)CC2)nc(=NCc2cnc[nH]2)[nH]1 c1(C(=O)NC(CC=C)CNC(=O)CCSC)cc(C(F)F)ncn1 N1(C(=O)NCCS(=O)(=O)NC(C)C)CCCC(C2CC2(F)F)C1 N1(C(CCCOC)=O)CCN(C(C23CC(C)(C2)OC3C)=O)CC1c1ccccn1 CC(C)C(F)C(=O)N1CC(N2CCN(C(C3(O)CCC3)=O)CC2)C1 CC1COCC(CNC(C2CC(O)(C)C2)=O)O1.C12(CC1)C(=O)N2C.C(=O)NC1CC1 C(=O)(CCC(F)(F)CN=[N+]=[N-])N1CCC(C)(CNC(CC(C)(C)OC)=O)C1 c1(CC(N2CC(NC(=O)COC3CCCC3)C(F)C2)=O)cc(F)cc(F)c1F CC1CC(NC(C2CCCN2C(C2CC(C)(C)CCO2)=O)=O)CC(C)(C)C1 c1(C(=O)NC2C(OC)CCC2)cc(CO)n(C)n1.C1(C(=O)N)(CO)CCCO1 C(=O)(C1=NN2CCC(C)N=C2N1)NCC(CNC(c1c(C)nc(O)[nH]1)=O)CO C1(C(=O)NCC23CCC2C3)CC(O)C(O)CC1CNC(C1CCC2(CCC2)C1)=O CC1(C)C(CNC(C2CC(=O)C2)=O)CCN1C(c1cccc(C(N)=O)n1)=O c1(CC)cccc(C(=O)N(c2cccc(OC3CCNC3)n2)CC)c1O c1(C(=O)NC(C(=O)OC)C2CC(C(=O)O)C2)cccc2c1S(=O)(=O)CCC2 N1(C(C(C)CN(C)C(c2cccc(C#N)c2)=O)=O)CCN2CCC1C2 CCCC(CNC(c1ccn(-c2cc(Cl)ccc2Cl)n1)=O)C(=O)O C1(C(=O)NCC(CNC(=O)Cn2nnc(=O)[nH]2)O)CCN(C2CC2)S1(=O)=O N1(C(C2CCC(C)O2)=O)CCN(C(c2ccccc2OCC#N)=O)C(CF)C1 c1(C(N2C(CCC(=O)NC(C)(CO)CO)CCC2)=O)cccc2ccoc12 C(=O)(C(C)(C)CN1CCCC1)N(C(c1ccncc1)C)C c1(CC)oc(C(N2CCC(CN(C(=O)CSS(C)(=O)=O)C)C2)=O)cc1C N1(C(CC(CNC(CC2OCC(C)(C)C2)=O)O)=O)CCOC(C#N)C1 c1(C(c2n(CCSC)nnn2)NCC(C)(C)CCC(C)O)ccc2c[nH]nc2c1 C(=O)(C(CC)C(=O)N(CC(=O)N(C)CC1(C)CCCC1)CC)OCC N1(C(C(=O)NCC(=C)C)=O)CCC2CCC1C2 O=C(CCCCc1cccc(O)c1)NC(CNC(c1cc(Cl)sc1Cl)=O)CO N1(C(C(C)OCC)=O)Cc2ccccc2C1CNC(=O)C1=NOC2CCCC12 N1(C(C(C(C)(C)C)O)=O)C2CCCC1CC(NC(=O)C=CC1CCCO1)C2 C(=O)(C(CNC(C1C2CC3C(C2)C13)=O)CC(C)C)Nc1cc(CC)cc(F)c1 Cc1ccc2c(=NC3CC4CCC34)[nH]c(N3CC(CO)C4(CCC4)C3)nc2c1 C(=O)(C1=NN(C)C(=O)CC1)N1CC2(CC(NC(C3(COC)CC=CCC3)=O)C2)C1 CCCCCC(O)C(C)C(=O)NCCc1ccc(O)nc1 Cn1ncc2c1CN(C(=O)CC1CCCN1C(c1ncccc1C(F)(F)F)=O)C2 c1(OC)c(CNC(=O)CN(CC(C)C)C2CC2)cccc1C(C)(C)C C(=O)(CCCC(=O)N1CCC(CCNC(c2ncc(F)cc2C)=O)C1)NCC N1(C(C(C=C)OC)=O)CCC(C)(C(=O)NC2CCOC(C)(CC)C2)CC1 c1(NC(C23CCCCC2C3(F)F)=O)ncc2c(n1)CCCCC2 N=c1[nH]c2ccccc2cc1C(=O)NCC1CC2CCCC2N1C(=O)CC(F)F c1(NC(C2N(C(c3ccc(OCC)nc3)=O)CC(O)C2)=O)cnc(C#N)c(Cl)c1 C1(C(=O)NC2(C(=O)NC(C3CCCCO3)C)CC2)C2CC(=O)CC12 C1(NC(c2c(N)non2)=O)(CNC(=O)COC2CCCCCC2)CCOCC1 C1(c2cn(CC3C=CCN3C(=O)CSc3ccncc3)nn2)(COC)CCCC1 C12(C(N(CCCNC(CCCc3c(C)ccs3)=O)C3CC3)=O)CC1COC21CCC1 N1(CCC(=O)NC2CC(NC(c3cnc(S)nc3)=O)C2)CCC(O)CC1 n1(CC(=O)NC2C(CNC(c3ccc(C(C)F)cc3)=O)CC2)nc(Cl)ccc1=O c1(CC(=O)NCCCSCC)cc(CNC(=O)CCn2cnnn2)oc1C C=C1CC(C(N2CCC(CNC(=O)COCCOCC)C2)=O)(CO)C1 C1(C(=O)OCC)C2CN(C(=O)CCN(C)C(C3CCCSC3C)=O)CC12 C(c1cccc(O)c1)=CC(=O)N(C1CN(C(C2CCCCS2)=O)CC1(C)C)C C=CCCCC(C(=O)N1CC2CCC(CC2)C1)NC(=O)C#CC(C)C N1(C(COCCCC#C)=O)CCC(NC(=O)C(c2c(C)noc2C)C)C(CO)C1 N1(C(COC)=O)C2CCC1C(CNC(c1ncsc1NS(C)(=O)=O)=O)C2 Cc1cnn(C)c1CC(=O)NC1CC(C(=O)NCCC(C2CC2)C2CC2)CC1O CN1CCC(C#N)(C(=O)NCC23CCCC2CCN3C(c2cn[nH]c2)=O)CC1 C1(c2n(C)nnn2)(NC(=O)NOCCC2CCOC2)CCCCC1 C(=O)(C(C)CC(N)=O)NCC1(F)CC(CNC(c2ccc(COC)cc2)=O)C1 C1(C(N2CC(COC)(NC(C3CC3c3nc[nH]n3)=O)C2)=O)CCc2nc[nH]c2C1 C1(C2CC2)(C(=O)NC(CC(C)NC(c2n[nH]cc2Cl)=O)C)CCC1 C1(C(=O)NCC2CCN(C(C3(CCC)CCNC3=O)=O)CC2)CC2(CCCC2)C1 N1(C(c2cc(Cl)cc(Cl)c2)C)CCC2(CCOC(C)C2)C1 Cn1[nH]c(C(N2CCCC(C3CCCN3C(=O)COc3ccsc3)C2)=O)nc1=O c1(CC)ccc(CC(N2CCC(CCCNC(=O)CN3CC=CC3)CC2)=O)cc1 C1(C)(OC)CCCC1(F)F.C(=O)(C1=CCSC1)N1C2CC(N)(C2)C1=O C1(C(=O)NC(CNC(Cc2c(C)con2)=O)C2CC2)CC2(CSC2)C1 O=C1CCN(CCn2ncc(Br)n2)C(=O)N1CC1CCCCCC1(F)F N1(CC(=O)NCCC(CNC(C2C(=C)C2)=O)O)C(=O)CN(C)C1=O CC(F)(F)C(F)(F)CC(=O)N(C1CCCCC1)CCNC(C1CC1(F)Cl)=O C(c1cccnc1)=C(C(=O)NC1CN(C(C(Br)=C(C)C)=O)C1)F N1(C(COCC=C)=O)CCCC(N2CCN(C(=O)C=C(C)CCC)CC2)C1 c1(C(N2CC(CNC(=O)C3=CCCS3)OCC2)=O)ccnc(Cl)c1Cl C1(NC(c2c(C)nc(C(C)C)s2)=O)CCN(C(c2ccn(C)c2C)=O)C12CCC2 c1(C(N2CCC3(C2)CN(S(=O)(=O)CCCCCl)C3)=O)ccc2nc(Br)nn2c1 CC1CCC(C(=O)NCC2CCCN(C(c3n[nH]cc3N)=O)CC2)CC1C C1(C(CC)(C)C)CCC(C(N2CCCC(N(C(=O)CCCOC)C)C2)=O)CC1 Cc1ccccc1COCC(N1CCCC(N(C)C(C23CC4CC2C3C4)=O)C1)=O c1(CC(=O)NCC(CN(C(=O)C=C2CCCC2)C)(C)C)cccc(F)c1O c1(NC(N)=O)ccc(S(=O)(=O)NOCC2CCOCC2)cc1 C1(NC(C(C)n2ccnc2)=O)CCC(N(C(=O)CNc2ccccn2)C)CC1 N1(C(c2n(CC)ccn2)=O)CC(F)(F)CC1C(N1CCN(C)CC1C(C)C)=O N1(C(C2(C(=O)OCC)CC2)=O)CCN(C)CC1CNC(C1OCCN(C)C1=O)=O c1(OC)ccccc1CN(C(c1nc(Cl)cs1)C(=O)NCCO)c1nccs1 N1(C(C=CCCCCC)=O)CCN(Cc2cnc(OC)s2)CC1C C1(C(N(CCC)C(C)C)=O)CC2(CC(NC(C3CCC(=O)O3)=O)C2)C1 Cc1ccncc1C(=O)NCCCOCCCNC(C1(O)CCCC1C)=O C1(NC(C2N(C(C)=O)CC(O)C2)=O)CCN(C(=O)CC2CCOCC2)C(C)C1 Cc1cc(C(N2CCN(C(C3CC3C3CC3)=O)C3CC23)=O)c(F)c(F)c1 Cn1ccc2c(C(=O)NCCC3=CCN(C(C4CCCS4)=O)CC3)ccnc12 C1(NC(c2ccccc2F)=O)CC(NCc2ccc(F)nc2)C12CCC2 C(N=c1cccc(S(=O)(=O)N(C)Cc2cnn(CC(C)C)c2)[nH]1)c1snc(C)n1 C1(NC(C2C(C(=O)OC)C2)=O)CC2CCC(C1)N2C(c1cnc(C)nc1SC)=O N1(C(CC2(C=C)CC2)=O)CC(C2CCCN(C(c3nn(C(C)C)cc3Br)=O)C2)C1 C1(C(=O)NC(C(=O)N(C)C)CO)CC12CCN(C(C13CC(CO1)C3)=O)CC2 CCCC(C(=O)N1C(C(=O)OC)CC1C)NC(=O)CCN(C)C C1(C(C)(C)NC(c2cnc(C(C)C)o2)=O)CCN(C(c2cc(Cl)n[nH]2)=O)CC1 c1(NCC)cncc(C(=O)NC(C)CC2CN(C(c3nc(=O)n(C)[nH]3)=O)C2)c1 c1(C(N2CC(O)(CN(C(C(CC)F)=O)C)C2)=O)cc(Cl)c(O)c(Cl)c1 Nc1cc(Cl)nc(Cl)c1C(N1CC2(C1)CN(C(=O)C(Cl)=CCl)C2)=O CCCCC(CC)CCC(=O)N1CCC(CCC(=O)NC23CCC(C2)OC3C)C1 c1(C(=O)NC2(COC)CCC2)oc(CNC(=O)Cc2ccc(C)o2)nc1C c1(C(=O)NCCN(CC(CC)OCC(F)F)C(=O)C=CC(=O)NC)ccc(Cl)o1 O(N=C1CCCCCC1)CC(=O)NCC1CN(C(CSCC#C)=O)C(C)CC1 c1(C(=O)NCCCCCNC(C2C3CCCC(=O)C32)=O)c[nH]c2cccc(F)c12 Nc1nccn2ncc(C(N3CCC(NC(=O)C=Cc4cccs4)C(F)C3)=O)c12 c1(OC(C)C)cc(F)c(NC(N2CCCC(C3COC(=O)N3)C2)=O)c(F)c1 CC1CC2(CCO1)CC2C(N1CCN(C(=O)CCC(C)(F)F)CC1)=O.CCC#N n1(C2CCN(C(CSC)=O)CC2)ncc2c1CN(C(=O)CCn1cccn1)C2 C=CCN=C(NCC1CCCCO1)NCC(F)(F)Oc1ccc(C#N)cc1 CCC(CNC(=O)NCc1c(C)cc(C)nc1O)(CC)C(F)(F)F C1(NC(c2cc(SC)c(N)cc2)=O)CN(C(=O)C(C)(O)C2CC2)CC2(CC2)C1 C1(C)(CNC(C(n2cnc(C(F)(F)F)n2)C)=O)CCN(C(=O)C2=CCSC2)C1 C1(C)(C(=O)NCCCN2C(C)CCC2)CCN(C(C2(C#N)CC(=O)C2)=O)C1 N1(C(C(CC)(CC)CO)=O)CCN2C(=O)C(NC(=O)C(C)C3(O)CCC3)CC2C1 c1(NC(CC)C(O)c2ccccc2)ncccc1S(=O)(=O)N(C)Cc1ccco1 C(=O)(CCCCC(OC)OC)N1CC(O)CC(NC(C(CCOC)C)=O)C1 c1(C(=O)NC23C(CN(C(CCCOCC)=O)C2)C3)cc(Cl)ccc1-n1ccnc1 n1(CCOC)cc(C(=O)Nc2cnn(-c3ccc(F)cc3)c2)c(=O)cc1C Cc1cc(=NCCN2CC3CC3C2)[nH]c(N2CCC(Cc3ncccn3)CC2)n1 N1(C(Cc2cc(C)no2)=O)CC(NC(C2CC23CC3)=O)C(n2ccnn2)C1 c1(NC(CNC(C=C(C)C(=O)O)=O)=O)ccc(Oc2cccc(O)c2)nc1 C1(CC(=O)NCC#CCNC(=O)Cc2ccsc2Cl)CCCCCO1 c12ccccc1C(=O)N1CCOC(C1)C(=O)N(C)CC(C)O2.CCCOCC CC(C)(C(=O)N1CC2CC(NC(C3(CC4CC4)CCC3)=O)C1C2)C(N)=O C(CCCCC(=O)NC1CC(C(C)(C)C)C1)NC(C1(CC=C)CC=CC1)=O c1(NC(CC)CC)cc(S(=O)(=O)NCCCN(C)CC2CCCO2)ccc1C#N C1(C(N(CC)Cc2ccc(F)cc2)=O)CCCCS1(=O)=O.C1(=O)CC2CC2CO1 O=C(C1Cc2ccccc21)NC1C=CCN(C(c2cnc3ccnn3c2)=O)C1 c1(NC(C23C(CN(C(C=Cc4cn(C)nn4)=O)C2)C3)=O)cccc([N+](=O)[O-])c1 c1(N(C)C)ccnc(C(=O)NCC2(CNC(C3COCCOC3)=O)CCCC2)c1 Cc1c(C(=O)N(C)CC2CCCCN2C(C2C=CC=CC=C2)=O)nnn1C(C)C C=CCCC(C(=O)NCC1(C#N)CCCC1)NC(=O)CCCC1CC1 C(C(F)(F)COC)(c1ccccc1)OC(C1CC1c1ccc(OC(F)(F)F)cc1)=O C(=O)(C(C)CCNC(=O)C(C)N(C(=O)COc1ccsc1)C)OC N1(C(c2csc(C)c2C)=O)CC(C(=O)NCCc2cncs2)CCC1C CC1CCSCCN1C(=O)NC12CCC(CC1N1CCOCC1)C2 CC1CCC(C)(C(=O)NCC2CN(c3nccnc3F)CCO2)C1 CCC(C)(C)CCCC(=O)NC(CC(C)(C)C)C(=O)NCc1ccoc1 c1(CC=CC(=O)N(C(C(F)(F)F)C2CC2)CC2CCCCO2)cc(C2CC2)[nH]n1 Cc1cc(C(=O)NC2CC3(C2)CN(C(c2cccc(CCO)c2)=O)C3)cc(N)c1 n1(CCCCn2c(C)ccn2)cc([N+](=O)[O-])cn1.N12CC(O)CC1C(=O)NC2=O N1(C(CC(C)CN(C)C)=O)CCC2(C1)CN(C(c1cc(O)cc(=O)o1)=O)CCO2 Cc1ccc(C(N2CCC(C)(CNC(=O)CCC(C)(F)F)C2)=O)cc1F C(CCC(C)(C)C(=O)NCC1CC(F)(F)CO1)NC(C(CC)N(CC)CC)=O N12CCC3(CC1)CC(CO3)NC(=O)COCC2=O.Cc1nnc(SCCN(C)C)s1 C1(C(=O)NCCNC(C2CCCN2c2ccccc2)=O)CC(CN)CCO1.CC(F)F C(=O)(CC(C)C(C)(C)C)NCCCCC1CCCN(C(c2c(C)ccnc2)=O)C1 CC1(C(=O)NCCC2CCC(NC(c3cn(CCF)nn3)=O)C2)CNC(=O)C1 C(=O)(CCCC1CCCO1)NC(C1CCN(C(=O)CC2CC2C2CC2)C1)C c1(C(=O)NCC2C3CN(C(C(CC(C)=O)(C)C)=O)CC32)noc2c1CCCCC2 C(CC(=O)N1Cc2ccccc2CO1)N(CCC(=O)NOC(C)(C)C)C c1(-n2c(CC(n3cc(C)cn3)C)nc(CC(CC)C)n2)cccc(Cl)c1C C#CCC(CC(=O)NCCCCCC=C)NC(=O)C(O)CCSC Cc1cc(C(F)F)n(CC(N2CC(NC(=O)CN(C)C(C)C)CC2CO)=O)n1 N(C1CCCc2ccoc21)C(C1COCCC1NC(C1CCNC1=O)=O)=O C#Cc1ccc(OCC(=O)N(CC(O)CN(C2CCC(CC)C2)C)C)c(OC)c1 c1(C(N2CC(NC(=O)CCCCC3CC3)(CO)C2)=O)cc2c(Cl)cccc2[nH]1 CC1(C)CC(CNC(=O)C(O)C2CCCC2)CN1C(c1c(Cl)cccc1Cl)=O n1(CCOC)nc(C(=O)NCCN(C(=O)C(CCSC)NC(N)=O)C)ccc1=O C(=O)(C1CCc2c[nH]nc21)N(CCCCN(C(C(C(=O)OCC)C(C)C)=O)C)C N1(C(C2COC(C)(C)O2)=O)CC2CCC1C1CN(C(c3c[nH]nc3F)=O)CC21 C1(COC(N(C)C(c2ccc(F)cc2)c2ccccc2)=O)CC2(COC2)C1 C1(NC(CCC2CCN(C(C=C)=O)C2)=O)CC(C)OC1=O c1(C(N2CCC(S(=O)(=O)NC(C)C)C2)=O)ccc2c(O)nnc(O)c2c1 CCCC(CCCNC(=O)C(C)(C)CO)NC(=O)CCNC(=O)C=CCl Cc1cn2c(=O)c(C(=O)NC3CC4CCC(C3)N4C(=O)COC(C)C)cnc2s1 N1(C(c2c(CCC)onc2C)=O)CC2COCCC2(NC(=O)CC2(C)CC2)C1 c1(C(N(CCNC(c2c(CC=C)cccc2)=O)CCOC)=O)cnc2n1CCS2 c1(C(=O)NC2C(F)CCN(C(CC(CC)C)=O)C2)cnc2c(c1)CCCC2 c1(C(=O)NCC2CN(C(COCCCC)=O)CC2C)cc(F)c(Cl)c(N)c1Cl C1(NC(COC)=O)CCC2(CC1)CN(c1cc(C)ncn1)C2 O=C(CCCCc1ccccc1)N1CC2CC1C2C(=O)N(CCO)CCO N1(C(C(C(CC)O)C)=O)CC2CCN(C(=O)CSc3cccc(OC)c3)C(C2)C1 c1(C(N2CC(NC(C(CCC)O)=O)C(O)C2)=O)cnc2cccnn12 C=C1CCN(C(=O)CC2CC(OC)C2)CC1.C(CCO)NC(C1CCC1)=O C(C1CN(C(C2(CC)CCOC2)=O)CC1C(N1CC(n2cnnc2)C1)=O)=CC c1(C(=O)Nc2cccc(NC(c3c(CC)non3)=O)c2)cc(C)c(F)cc1F S(=O)(=O)(c1cc(C(N)=O)c(Cl)s1)N1CCC(c2cc(C)c(C=CC(=O)NC)cc2)C1 C=C(C)CC(C(=O)N1CC(N(C)C(c2ccnc(C(F)(F)F)c2)=O)C1)NC(C)=O CC(C(=O)NC1CCC(CNC(c2ccccc2OCC#N)=O)CC1)C(C)(F)F C(=O)(CC(Cc1ccc(OC)cc1)NC(=O)C(C)(C)C)NCC(CC)O C1(C(=O)NCC(=C)CC)(OC)CCN(C(C2(N(C)C)CCCC2)=O)C1 c1(OC)ccccc1SC(F)(F)F.C1(C(=O)NC(C)C(c2ccccc2)O)CN1 C(=O)(C1=CCc2ccccc21)NCC1C(NC(C(C)(C)C(F)F)=O)CCC1 N1(C(c2cccnc2)=O)C2CCC1CC2.CC(CN(C1(C)CC1)C)C(=O)C(=O)CN N1(C(CSc2nc(C)sc2)=O)CCC(NC(=O)C(C)CN(C)C)CC1 C(=O)(CCCCN(C)C)NC1CCC(CC(N2CCC(=CCC)C2)=O)C1 N1(C(c2nc(C(C)C)sc2)=O)CC(CNC(=O)COC(C)=O)CC1C n12cc(nn1)CC(=O)NC(C)C2.c12csc(n1)C(C)NC2=O.C1(CNC(N)=O)CC1 C1(c2cn(-c3cnn(C)c3F)nn2)CC2C=CC1C2.c1(C2C(C)C2)cc(CC(=O)N)ccn1 C(=O)(C(C)C(O)C(C)CC)NCC(CC)N(C)C(c1cnc2nccn2c1)=O c1(C(N(CCCCN(C(C(C)OCCC=C)=O)C)C)=O)cn(C)nc1COC c1(C(N2CC3CC(CNC(CSCC(C)=O)=O)C3C2)=O)cccc2c(C)[nH]nc12 Cc1noc2cc(C(=O)NC3CC3NC(c3ccc(F)c(Cl)c3)=O)ccc12 C1(CNC(C(=O)NC2CCC(C(=O)OC)CC2)=O)CCCN2CCCCC12 C1(NC(C23OCC(C)(C2)C3)=O)CCSC12CN(C(C1CCCC1O)=O)C2 C(=O)(C(C)(C)CCC#N)NC1CCC(C)N(C(=O)C=C2CCN(C)C2)C1 C=CCC(CNC(c1ccc(Cl)s1)=O)C(=O)N1CC(N(C)C)C1 C1(C(=O)NCCN(C(=O)COCC(C)(C)C)CC)CCCC1O C1(CC(=O)NC(C(C)SC)C)CN(C(c2cn(C3CC3)cn2)=O)C(C)(C)C1 N1(C(c2ccoc2Br)=O)CCC2(CCCN(C(C3CCCOC3)=O)C2)C1 c1(C(N(CCCNC(C2C(F)(F)C23CC3)=O)CC)=O)cc2c(s1)CCCC2 Nc1ccc(C(F)(F)F)cc1.c12ccccc1Cn1ccnc1-c1ccncc1-2 C1(C(CN2CCN(C(C(=O)Nc3nc(SC)cs3)=O)CC2)=O)CCCCC1CC c1(C(N2CC(C=C)(CC(=O)NCC(C)CCO)C2)=O)c[nH]c(C)cc1=O C1(N(C)C(C2(CF)COC2)=O)CN(C(=O)CC2NC(=O)NC2=O)CC1O CC1CCC(CNC(c2ccc(O)nn2)=O)CN1C(=O)C1=CCCCO1 Brc1cnccc1-c1nc(CCC2CCOCC2)no1 CC1CCN(C(c2cccs2)=O)CC1CNC(C1CCCC2(CC2)C1)=O c1(C(=O)NC2CC2CNC(C2(C(F)(F)F)CC2)=O)cccc(=O)o1 C1(C)(CNC(c2cccc(C#C)c2)=O)CN(C(=O)CC(CC)CC)C(C)(C)C1 Cc1ccc(CC)c(F)c1.N12CCN(CC1)C(=O)C(=Cc1ccccc1)N2 C1(NC(c2nc(C)[nH]n2)=O)(CNC(C23CSCC2C3)=O)CCCCC1C C=CC1(C(c2nnnn2C2CC2)Nc2ccc(Br)c(C(F)F)c2)CCOCC1 C(C)(C)(CN=C(NC1CCc2ccccc2C1)N1CCN(C)C(=O)C1)NC(C)=O Cc1cccc2oc(C(N3CC(NC(=O)CCCS(C)(=O)=O)C3)=O)cc12 N1(C(c2c(C)c[nH]n2)=O)CC2CCCC(C1)N2C(=O)CNc1cccnc1 n1(CC)ccnc1C(N1CCC(C(C)NC(=O)C(CN(C)C)N(C)C)C1)=O N1(C(c2cc(C(CC)CC)no2)=O)CC(N(C)C(c2cc(Cl)no2)=O)C2(CC2)C1 C=CC(COC)N=c1ccnc(NCC2CCCN(c3ccccc3)C2)[nH]1 N1(C(CCOCCOC)=O)CC(C)(C)OCC1CNC(=O)CSC(F)(F)F c1(OC)ccc(CCC(=O)NC(C)CNC(=O)C(CO)c2ccccc2)cc1 Cc1cnc(C(=O)NCC(C(N2CCCCC23CC3)=O)N(C)C)cc1C c1(C(N2C(C)(C)C(CNC(=O)CC(=O)N(C)C)CC2)=O)ccc2[nH]c(=N)[nH]c2c1 c1(C(=O)NC(CCNC(c2c(CC)c[nH]n2)=O)C)nccc2ccccc12 c1(CN2C(C(=O)NC(C(=O)OC)CO)CC(F)C2)cnc2ccc(Br)cn12 C1(C(=O)NCC(=C2CN(C(C(CC)N3CCCC3=O)=O)C2)F)CCC2(CC2)C1 N1(C(c2cc3cn(C)nc3cc2)=O)CCc2occc2C1C(=O)O Cc1ccc(F)cc1-n1nc(C(O)C(C)C)nc1C(O)C(C)C.CO c1(C(=O)NCC2OCCN(C(C3(COC)CC3)=O)C2)c(I)ccnc1F N1(CC)CC(C(=O)NC2CC(NC(=O)OC(C)(C)C)C2)c2ccccc2C1=C N1(C(C(C)=C2CCCC2)=O)CC(OC)C(NC(=O)CCc2cncs2)C1 N1(C(C(C)C(F)(F)F)=O)CCOC2CN(C(=O)NCc3ccccn3)CC12 N1(C(c2n(CC)ccn2)=O)CCN(C(=O)CCSCC(C)C)CC(C)(C)C1 CCC(COC(F)(F)F)CC(F)F.C1C(=O)N1CCO N1(C(COCCC=C)=O)CC2CC2(NCCOCCOCCN(C)C)C1 C1(NC(C(CC)=CCCC)=O)CC(NC(=O)CC2(COC)CC2)C12CCC2 C(C1CCC(N)C1)NC(C1C(OCC(C)C)CC1)=O c1(N2CC(CNC(CC(C)N(C)C)=O)N(C)CC2)ncc2c(n1)COC2 c1(C(=O)NC(C)C(C)NC(=O)C=C(Cl)Cl)cccc2c(Br)cccc12 C1(NC(CN2CCC(OC)C2)=O)CCCCCC1NC(c1[nH]c(O)nc1C)=O C1(CNC(C2(OC)CCCOC2)=O)CC(C)CN(C(=O)CC2COCCOC2)C1 N1(C(C2CCN(c3cccnn3)C2)C(=O)NCC)CCC(c2cc(C)no2)CC1 CCCS(=O)(=O)CC(=O)NC1CN(C(=O)C(c2cnccn2)C)CCC1CO Cc1cccc(C(N2CC3C(N(C)C(c4cccc(CO)c4)=O)C3C2)=O)c1 NC1CN(C(=O)CCCC(=O)NCCC(F)(F)F)C2(CCCOC2)C1 N1(C(c2nc(CCC)oc2)=O)CCCC(C)C1CNC(c1coc(Cl)c1)=O N1(C(C(C(=C)C)(C)C)=O)CC2CC(NC(c3cc(C(F)(F)F)no3)=O)CC1C2 C1(NC(C(CC)C)=O)CC12CCN(C(=O)Cn1cnc(C#N)n1)C2 CC(C)C(O)C(C)C(=O)N1CC(C(=O)NC2CC(N3CCCC3)C2)C(C)(C)C1 C(=O)(C(C)(C)C(F)F)N1CCC(OCCNC(C(CCOC)SC)=O)C1 C(=O)(C(C)CS(C)(=O)=O)N1CCC(N(C(C(CSC)O)=O)CC2CC2)CC1 C1(C(=O)NC23C(CN(C(c4cnc(C(C)(C)C)[nH]4)=O)C2)C3)COCC2(CCC2)O1 C1(CC)CCC(O)(C(=O)NCCCN(C)C(c2cnn(CCO)c2N)=O)C1 N1(C(c2cnc(OCC)nc2)=O)CC(CNC(=O)CCC(C)OC)C(F)(F)C1 C1(NC(C(C)OCC=C)=O)CCN(C(=O)C=C2CCCC2)C1C1CC1 Cc1oc(C(=O)NCCN(C(C2CC2c2ccccc2F)=O)CC2CC2)cc1Br N1(C(C2C(=C)C2)=O)CCC2CC(NC(c3cc(N(C)C)ccn3)=O)CCC2C1 CC(C)CC(C(=O)N1CC(F)(F)CC1CO)ONC(=O)CCn1ccnc1 C1(NC(C2(C)CCCO2)=O)COC2(CCN(C(C3COC3)=O)CC2)C1 c1(CC(=O)NCC(C)NC(c2ncoc2C2CCCC2)=O)cnc(O)nc1O C#CCCCC(C)C(=O)NC1(CC(=O)N(C2CCC(C)C2)C)CC1 CCC(C(=O)N1CCC(N(C(c2cnncc2C(F)(F)F)=O)CC)C1)C(C)C c1(CCCC)cccc(C(=O)NCC(O)CN(C)C(c2nccc(C)n2)=O)c1N N1(C(C(=O)OC)C)CCN(C(=O)C=CC(=O)SC2CCCC2)C(C)C1=O C1(C)(c2nn(-c3cccc(C)c3)c(C3CCCC(C)CC3)n2)CCN(C(C)C)CC1 N#Cc1cc(Br)cc(Br)c1NC(C1COCCN1S(=O)(=O)CC1CCC1)=O N1(C(CC(C)C)=O)CC(CNC(=O)CCCSC)C2(CC2)C1 c1(C(=O)NC2CCN(C(C3CCCC3C(F)F)=O)CC2F)ccc([N+](=O)[O-])cn1 c1(NCCC(=O)NCC2C(C(=O)O)C2)ccccc1OC(F)(F)F C(=O)(C(C)(C)CCNC(=O)C(C)CO)NCc1cn(C(C)C)nc1 c1(C(N2CCC(C)(CNC(c3cc(F)cs3)=O)CC2)=O)c(F)ccc(F)c1O N1(C(C(=O)Nc2sc(CCC)c(C)n2)=O)CCC2(CCSC2)C1 C=CCC(C)(CC)C(=O)N1CCCC(CCNC(c2cnc(SC)n2C)=O)C1 N1(C(CC(=O)NCC)=O)CCC(C)C(NC(C2CN(C)C2)=O)C1 N1(C(C(C)N(C)C)=O)CCCC2(CCN(C(c3cnc4c(F)cccn34)=O)C2)C1 CCC(CC)C(C(=O)NC1(CCNC(=O)COc2ccccc2F)CCC1)OC C1(F)(CNC(C(C)SC)=O)CCC(NC(c2ccc(-c3ccc(Cl)cc3)s2)=O)C1 C1(NC(c2cccc(C(N)=O)n2)=O)C2CCC1N(C(=O)CC1C=CS(=O)(=O)C1)C2 C(C(C)CN=C(NCc1cnc(N2CCCC2)s1)NCC(C)(C)C)OCC N1(C(C2(C)CCCC2)=O)CCn2ncc(-c3cccc(C4(C)OCCO4)c3)c2C1 C1(C(=O)NC2C(NC(=O)CCc3ncc[nH]3)CC2)Cc2cccc(F)c2O1 N1(C(CCC)=O)CC(C(=O)NCCOCC(C)(C)O)C(CC)C1 CCCC(CCC)CC(=O)N1CC(C(O)C(=O)NCC2(CC(C)C)CC2)C1 C(=O)(N=c1c(F)c[nH]cc1Cl)N1CCN(C(c2cccc(S(N)(=O)=O)c2)=O)CC1 c1(NCC2C(C)CN(C(=O)C(CO)NC(N)=O)CC2)ncnc2ccc(Cl)cc12 C1(C(F)(F)C(=O)NC(C)C(C)NC(c2cc(C)[nH]n2)=O)(OC)CCCC1 C12(NC(=O)C=Cc3cn[nH]c3)CCCC1N(c1nc(Cl)nc3[nH]cnc13)CCC2 c1(C(N2CCCC(NC(CC3(C=C)CC3)=O)C2)=O)cc(C(F)(F)F)cc(C)n1 C1(CCC)CCC(c2csc(NC(=O)NCCC(F)(F)C3CC3)n2)CC1 c1(OCCC(N2CCCC(C(C)NC(C(C)=C3CC3)=O)C2)=O)c(C)cccc1C n1(CCCCN(C(=O)CCNC(=O)C(=O)O)CC)cc(-c2cnn(C)c2)nn1 C1(CC(=O)NC2CN(C(=O)CC3(O)CC3)CCC2CO)CC2(CCC2)CO1 C1(CCOC)CC(c2nnnn2C)(NCC(C)(C)C2CCCC2)CO1 C1(CC)CN(Cc2cnc(OC)nc2)CCN1C(=O)Cc1cnccc1OC C(CC(CC)C(=O)NCC1CC(NC(=O)CCCn2c(O)nnc2O)C1)=CC c12ncccc1C(=O)NC2.c1(NC2C(CC)C2)nccc(C(=O)OC)n1 C=CCC(C)C(=O)N1CCC(=CCNC(c2sccc2SC(F)F)=O)CC1 c1(CC(=O)NCC(CNC(C(C)NC(=O)NC)=O)C)c[nH]c2cc(F)ccc12 c1(COC(C2CC(=C3CC3)C2)=O)ccc(-c2noc(C3CCCO3)n2)cc1 CCCCCS(=O)(=O)CC(=O)N1CC2CN(C(C3OCC3(C)C)=O)CCC12 c1(NC(=O)NC)ccc(C(=O)NC2(C)CC(NC(c3cc(C)oc3C)=O)C2)cc1 c1(C(=O)NCC2(F)CN(C(C3C4CCC(=O)C43)=O)C2)ccc(F)c(Br)c1 C#Cc1cccc(C(N2CCCN(C(c3ncc(SCC)cc3Cl)=O)CC2)=O)c1 N1(C(C(COC)NC(C)=O)=O)CCC(C(C)C(=O)N2CC(COC)C2)CC1 C(=O)(C(C)CC(C)(F)F)NC1C(F)CCN(C(c2ncn(C(C)C)n2)=O)C1 C1(CNC(c2ccc(CC)[nH]2)=O)CC2CCC(C1)N2C(=O)CC1(C)COCCO1 CC1(C)NC(=O)CCC1NC(C1CCOCCN1C(=O)C(CO)C(F)(F)F)=O c1(CC2N(C(CCCC3(C)N=N3)=O)CCCC2)ccc(F)c(F)c1 C1(NC(C2CCC2)=O)CN(C(=O)CCCCc2ccccc2)CC2CC12 C1(C)(CNC(Cc2c(C)nc(S)s2)=O)CN(C(C2CCC(O)C2)=O)CCO1 C1(CC(=O)NCC(CNC(COCCOC)=O)CO)COCC1(C)C CCCCC(O)C(C)C(=O)N(CCCC(=O)NCc1ccc(O)c(C)c1)C N1(C(C(C)OCCCC)=O)CC(OC)CC1CNC(C1(CCCC)CC1)=O C1(NC(c2cnc(CC)s2)=O)(CC)CCCN(C(=O)CC2CCCC23CC3)C1 C(=O)(C(CC(C)C)C(C)C)N1CCC(NC(Cc2ccc(C)c(Cl)c2)=O)C(C)C1 C1(NC(c2n(CC)ncc2)=O)CCN(c2ncnc(O)c2Br)CC1F C1(C(N(CC(C2CC2)OC)CC)=O)CCC(C2CC2)N1C(c1cnns1)=O Cc1cc(C(N2CCN(C(=O)Cc3cncn3C)CC2CC2CC2)=O)ccc1Cl C(=O)(C1CC(=O)c2ccccc21)NC(CC=C)Cc1ccc(C)cc1F c1(N(CCn2c(=O)c2=O)C)nccn1C(C)(C)C.CC(C)C(C)C1CCC1 C1(NC(C(=O)NCC2CC2)=O)CC2CC(C1)N(C(c1ccc(Cl)c(F)c1O)=O)C2 C12(C(N3CC(NC(C4CN(C(C)C)C4)=O)C3)=O)CCCC1CC2 c1(OC)cc(C(=O)NC2CC2CNC(c2ncoc2C2CC2)=O)nn1C c1(C(=O)NCc2c(C(C)C)nn(C)c2)c2ccccc2nn1C C1(C2CC2)(CNC(C(C)CC2CCC2)=O)CCN(C(=O)CC2CC2)C1 N1(C(CCCC)=O)CCCCC1Sc1nnc(C2CNC(=O)C2)o1 CN1CCN(C(=O)CC2COCCO2)CC1CNC(c1cn(C2CC2)cn1)=O CC(CC(=O)NC1(CCNC(c2nccn2C)=O)CCCC1)P(C)(C)=O c1(C2C(OCC)C2)cccc(NC(C2CCOCC2)=O)c1.C1CCC2(CC2)C(=O)N1 C1(C)(C(=O)NC(c2noc(C)n2)CC)CN(C(=O)C(C)COC)CC1C C(C(C)(C)CCNC(=O)CCOCC(C)(C)C)OC c1(C(N(CCOCCCN(C(=O)CC2(C)CC2)C)C)=O)cc2ccccc2s1 C12(C(=O)NC(C)CN(C(=O)C=CCN3CCOCC3)C)CCC(CC1)C2 c1(SC)ccc(C)c(NC(=O)NC2CC(=O)N(Cc3ccc(C)cc3)C2)c1 c1(NC(C(=O)N(CC=C)CC2CC2)=O)ccc(F)c(C(F)(F)F)c1 O=C(NNC(=O)c1coc(C(F)F)n1)C(=O)C(O)C1CCC1 N1(C(C2CCCN(C(c3c(OC)cc(F)cc3)=O)C2)=O)CCC2(CCCC2)CC1 CC1CN(C(=O)CN2CC=CC2)CC(C)C1NC(=O)CC1(N(C)C)CCC1 C1(C(N(CCCCCNC(=O)CC2CCCO2)C)=O)COCC1(C)C c1(C(N2CC(NC(C=CCOC)=O)CC2(C)C)=O)ccc(S(C)(=O)=O)o1 C(=O)(C1=CCCCCC1)N1CCCCC(C(N(C2(C#C)CCCCC2)C)=O)C1 CC(C)(CCl)C(=O)NC1CCC(C(=O)NCC2(C#N)CCC2)CC1 C(CC(C)(C)CC(=O)N1CC(CC(C)NC(C2Cc3ccccc3O2)=O)C1)OC Cc1nc(N)cnc1C(=O)NCCC1(O)CN(C(=O)CCn2ccccc2=O)C1 c1(CN(CC(=O)NCC2C(c3cccc(C4CC4)c3)C2)C)cc(O)ccc1Cl c1(C(=O)OCc2ccc(C#C)nc2)occ2c1CCCC2 N1(C(C(c2cccnc2)C)=O)CCCCC1CC(=O)N(C)C CCCCC(C)(F)C(=O)NCC1(OC)CCCN(c2ncccc2C#N)C1 C(=O)(CCCCCN(C)C)N1CCC(C(C(=O)NCCCCN(C)C2CC2)(C)C)C1 c1(C(=O)NC(C(C)(C)O)C(=O)N2CCC(C)(F)C2)ccc2occc2c1 c1(N2CCCC(CN(C)C)C2)ncccc1S(=O)(=O)NCCCC(N)=O N1(C(C2CC(C)(C)C2)=O)CCCC1(C)CNC(C1CCCC(C(F)(F)F)O1)=O N#Cc1ccc(S(=O)(=O)N2C3CN(Cc4cc(Br)cs4)CC23)c(Cl)c1 N1(C(C(C)C)=O)CC(O)CC1CNCc1c[nH]ccc1=N N1(C(C(=O)Cc2ccccc2)=O)CC2(C1)CN(C(c1cnc(S)nc1)=O)C2 C1(COC)CN(C(C2CCCCCC2)=O)CCN1Cc1cccc(C(N)=O)c1 C1(C(=O)NCC(C)N(C(CC(=C)C)=O)C)CC(=O)NC(c2ccccc2)C1 C(=O)(CC1OCCc2ccsc21)N1CCCC(NC(c2cc(C)[nH]n2)=O)C(F)C1 c1(OC)ccc2nccc(C(=O)NC(C)CCNC(=O)C(C)(C)CF)c2c1 c1(-c2n(C)cnc2)cc2c(C(=O)N(C)C)cccc2[nH]1 c1(OC)ncc(C)cc1C(N1CC2CC(C1)N2C(=O)C1=COCC1)=O O=C1CCC(NC(c2ccnc(-c3ccc(I)cc3)n2)=O)CN1 c1(CC(=O)NCC2C3N(C(CCS(N)(=O)=O)=O)C(CC3)C2)cc(F)c(F)c(F)c1 C(C(=O)N=c1ccn(C2CC2)[nH]1)C1(C)CN(C(c2csc(O)n2)=O)C1 C12(CNC(CCC3(F)CC(C(=O)OC)C3)=O)CC3CC(CC(C3)C1)C2 c1(NC2CCCC(NC(COS(C)(=O)=O)=O)C2)ccc([N+](=O)[O-])cc1Cl Cc1ncsc1C=CC(=O)NC1(C(F)(F)F)CCC1.C12CC1CNC2=O N1(C(C(C2(C)CC2)NC(c2csnn2)=O)=O)CCC(C(N)=O)C1 C(CCCCCNC(C1C2CCC1CC2)=O)N(C(=O)C(C)(C)N1CCCCC1)C c1(C(=O)NCC2CN(C(c3cnc(Br)s3)=O)C2)cc2c(nn1)CCCC2 C(=O)(C(F)(F)C(O)C1CC1)N1C(c2cccc(OC(c3cccs3)=O)c2)CCCC1 C1(CC=C)(NC(c2ncccc2F)=O)CCN(C(=O)CCC(C)OC)CC1 Cc1nc(C(=O)NCC(CC(C)(C)C)O)c(C)o1.C1C(=O)NCCO1 Cc1cn2nc(N3CCC(F)(F)C(CNC(c4cc(Cl)ccc4Cl)=O)C3)sc2n1 C1(NC(C2CC(OCC)C2)=O)CCCC(NC(=O)Cn2cc(Br)cn2)C1 c1(NC(c2cn(-c3ccc(C)cc3)nn2)=O)coc2c1CS(=O)(=O)C2 Cc1ccc(C(=O)N(C2CCCN(C(c3cc(C)co3)=O)C2)CCF)nc1 c1(C(C)(C)C)ccc(CCNCc2ccnn2C2CCC2)c(F)c1 C(C(C(C)C(C)C)NC(=O)CCOC1COC1)NC(C(CC)c1ccccc1)=O N1(C(C(CC)(C)CO)=O)CCCC2(CCN(C(c3nc(C4CC4)oc3C)=O)C2)C1 c1(C(N2CCC(NC(c3ccnc(Br)c3F)=O)C2)=O)ccc2cc(F)ccc2n1 N1(C(CN2CC(NS(CC)(=O)=O)OCC2)=O)CCN(C(C)=O)CC1C C(C(O)CC(=O)C(CCNC(C)=O)=O)N.C1(N)CCC(OC(C)C)CC1 CC1OC2(C(=O)NCC(C)(C)NC(=O)C(c3ccc(C#N)cc3)C)CCC1CC2 c1(C(=O)NC(C2CCCCO2)C2CCCCC2)nc(Cl)sc1Br C1(C(N2C(CO)CC(NC(C=COCC)=O)C2)=O)CC(=O)NC(C)C1 N1(C(C(C(C)C)C)=O)CCC(C2(NC(=O)CCCNC(=O)C(C)(C)C)CC2)C1 N1(C(CCCOCC=C)=O)CCC(NC(=O)Cn2c(C)csc2=O)C(F)(F)CC1 Cc1cnc(N2Cc3ccc(Cl)c(Cl)c3C2)c(S(=O)(=O)N2CCCC(O)C2)c1 N1(C(=O)CN2CCOCC2)CCC2CCCN(C(c3cc(CCO)on3)=O)C2C1 c1(C(=O)NCC(C2CC2)NC(C(CC)F)=O)ccnc(O)c1 c1(C(N2CCC(C(F)(F)F)CC2CNC(=O)C(F)F)=O)nnc(O)nc1O c1(NC(CSCCNC(C(C)c2ccsc2)=O)=O)cc(CO)ccc1O c1(C(=O)NCC(C)NC(C(C)=C2CCC2)=O)cncc2n[nH]cc12 c1(OCCCC(=O)N2CCC(CCNC(=O)CC3CC34CC4)C2)ccc(Cl)cc1 N1(C(C(=O)NCc2ccc(C)cn2)=O)CCc2ccc(Cl)c(F)c2C1 C(CC1CC1)(C(=O)N1CC(CCCn2ccnn2)C1)NC(C(C)NC=O)=O Cc1ccc2c(c1)CC(C)N(c1nnc(C(C)OC)n1-c1ccc(Cl)cc1C)C2 C1(C(=O)NCC(C2CCCC2)NC(c2cc(CC)no2)=O)CCCC2C1C2(F)F C1(OCC)CN(C(c2cncnc2C)=O)CC1CNC(=O)C(C)c1cc[nH]n1.NC N1(C(c2c(OC)ccnc2)=O)C2CCCC1CN(C(c1cnn(C3CC3)c1)=O)C2 c1(C(N(CC(C)NC(C2CN(C(C)=O)C2)=O)C)=O)cccc(SCC#N)c1 C1(S(N)(=O)=O)(c2cn(C(C)C(=O)NCCC(=O)NC(C)(C)C)nn2)CC1 C1(CNC(C2C(C=C)C2)=O)CCCCN1C(c1cnncc1OC)=O CC(C)(C)CCC(F)C(=O)N1CCC(C(=O)NCc2cnn[nH]2)C1 C1(C(=O)NCC(CC#C)(C)C)CC12CCN(C(c1cccs1)=O)C2 CC(C)(CC1CC1)C(=O)N1CC(CNC(=O)CCc2ccccn2)C(O)C1 C1(NC(CC2(CS(C)(=O)=O)CC2)=O)CC2(C1)CC2NC(=O)CCN1CCCC1 c1(OCC)ccnc2sc(C(N3CCC(NC(=O)C(F)(F)CC)C(F)C3)=O)cc12 C1(OC)CN(C(c2cnc[nH]2)=O)CC1C(=O)NCC1(c2oncc2C)CC1 Cc1cc(Br)c(C(=O)NCCOC2CN(C(=O)CC3CCC4CC34)C2)cc1F CCCN=C(NCCc1ccc(C(C)C)cc1)N1CCCC(S(C)(=O)=O)C1 C(C)(CCC#N)(c1nnnn1CSc1ccccc1)NCC(=O)N(CC)CC C(=O)(C1CCC(NCCCCC2CCCCC2)c2ccccc21)OC C1(C2CCCN(C(C3CC3C3CC3)=O)C2)(NC(CSCCN(C)C)=O)CC1 C1(CN(C(COCc2nnc(C)s2)=O)C)CCCN(C(C2CCCCN2C)=O)C1 C1(C(N2CCC(O)(CNC(C(CC#C)CC=C)=O)C2)=O)Cc2c(F)cccc2O1 c1(N2CCN(C(C(=O)NCc3nc(C(CC)C)[nH]n3)=O)CC2)cc(C)cc(C)c1 N1(C(CN(C(CC2CC(=C)C2)=O)C2CCC2)=O)Cc2nncn2C(C)C1 C1(C(N(C2CC3CC3C2)C)=O)CC1C1CN(C(=O)CCc2nccs2)C1 C=CCCCCCC(=O)N1CCSCC1CCNC(=O)CC1C=CCC1 C=CC(C)(O)CC(=O)N1CCCC1CNC(=O)COC1CCC(F)(F)CC1 C1(CC(C)C)CCCN(C(=O)CC2(C)CCN(C(c3ccc(CO)nc3)=O)C2)C1 N1(C(C2CC(CC)C2)C(=O)NCCCOC)CCCOC(C2CCC2)C1 C(CCCCC(=O)NC(C(=O)NC(C)CC(C)(C)CN(C)C)C1CCCO1)=CC c1(C(=O)NCC2CN(C(C(COC)COC)=O)CC2C)n[nH]cc1[N+](=O)[O-] CC(CC(F)(F)F)C(=O)NC12CC(CNC(c3ccc(N)c(F)c3)=O)(C1)OC2C N1(C(C2OCC(C)C2)=O)CCCC(C)C1CNC(=O)CC1OCCC1C C(CC(=O)NC1(C2(OC)CCC2)CC1)(C(F)F)NC(C(CC#C)C1CC1)=O c1(C(=O)NC(CNC(COCCN(C)C)=O)C2CC2)cc2c(F)c(F)ccc2s1 CN1CCN(C(C2(C)CCCS2)=O)CC1CNC(C1CCCC(C)(C)C1)=O N1(S(=O)(=O)Cc2csc(Cl)c2)CC2CC1CN2CC(F)(F)F c1(N2CC(NC(CC(C(C)C)O)=O)C(C)C2)ncnn2c(Br)ccc12 c1(NC(C2CC(NC(C=C(C)C(C)C)=O)C2)C)nc(C)nc2sc3c(c12)CCC3 Cc1cccc(N)c1OCC1CCN(c2nccnc2F)CC1 c1(CC)c(C(N2CCCC(NC(=O)C(=O)C(C)(C)C)C2)=O)[nH]c(C)c1C(C)=O C(=O)(NNC(=O)CS(=O)(=O)C12CC(C1)C2)C1C(c2n(C)ccn2)CC1 C(CN=c1[nH]c(N2CCC3CCC(C3)C2)nc2ccsc12)NC(N(C)C)=O N1(C(CC(CCC)(C)C)=O)CCCC2(C1)CN(C(=O)C(CC)N(C)C)C2 C12(CNC(CN(CC)CC)=O)CCCC(CN1C(C1CC3CCC1C3)=O)C2 C1(C)(C(=O)NCCCCC(C)NC(C2OCCC2(C)C)=O)CCN(C)CC1 Cc1cccc(O)c1NC(c1ccc(NC(c2c(F)cccc2Br)=O)cn1)=O CCCCCCCC(=O)NCC(C)=CC(=O)N(CC(=O)OC)C1CC1 Cc1ccc2c(=NCC3CCC(C)C3)[nH]c(N(N3CCCS3(=O)=O)C)nc2c1 N1(C(Cc2cc(COC)on2)=O)CCOC(CNC(=O)C(C)n2cccn2)C1 CCCC(C)CC(=O)NCC1(NC(c2cnoc2)=O)CCOCC1 N1(C(CSC)=O)CCC(NC(=O)Cc2cnn(C(F)F)c2)C(F)C1 C(C(C)C(=O)N(C(c1cnccn1)C(=O)NC1CC1)C)OC.c1(C)cccnc1 S(=O)(=O)(c1ccc(NC(C)CS(C)(=O)=O)cc1Cl)NCC1(OC(C)C)CCOC1 N1(C(CS(=O)(=O)N(CC)CC)=O)CCC(C)(C)C1CNC(C1CCS1(=O)=O)=O C1(C(=O)NCC2N(C(C3(C)COC(=O)N3)=O)CC2)CC2(COC(=O)N2)C1 N1(CC)CC=C(CNC(C2CC2(C)CC)=O)CC1 CC1(CO)CCN(C(C2CC2NC(c2nc3ccccn3n2)=O)=O)CC1O c1(C(N(C(C)(CN)C2CC2)C)=O)cc(I)c(Cl)cc1F C(=O)(C(C)(C)CF)NC(C1CC(NC(c2cc(-c3ccc(Cl)s3)on2)=O)C1)C C1(CNC(c2c(CC)c[nH]n2)=O)(CNC(c2cncs2)=O)CCOCC1 N1(C(C2C(CCC)CCC2)=O)CCC(F)(CNC(c2csc(C)n2)=O)CC1 C1(CC(N2CCC(N(C(c3c(CC)c[nH]n3)=O)C)C2)=O)C=NN(C)C1=O n1(CC(=O)OCC)cc(C2(O)CN(C(c3occc3COCC)=O)C2)nn1 N1(C(c2cc(C)ncn2)=O)CCOC2CCN(C(c3ccc[n+]([O-])c3)=O)CC12 c1(C(=O)NCC(C)(CO)NC(C2C(OC)C2)=O)ccc(Cn2cnnc2)cc1 C1(C(=O)NC2C(CNC(CCc3c(C)ncs3)=O)CCCC2)CC12CCCCC2 N1(C(c2c(C)ccc(C)c2)=O)CCC2CCN(C(c3sccc3CSC)=O)C2C1 CC1(C)CCCC(O)(C(N2CC3OCC(NC(=O)CCC4(C)CC4)C3C2)=O)CC1 n1(CC(=O)NCCN(C(Cn2c(C)ncc2)=O)CC(C)O)ccc([N+](=O)[O-])n1 CC(C(=O)NCC1CCN(C(C2CSC2)=O)C1)S(N)(=O)=O c1(C(N2CC3(CCN(C(C4CC5(CCC5)CO4)=O)C3)C2)=O)ncnc2cc[nH]c12 N1(C(CCOCCC)=O)CCC2(CC2)CC1C(=O)NCCc1nnc(C)s1 Cc1cc2[nH]c(C(N3CCOC(C(=O)Nc4ccc(I)c(Br)c4)C3)=O)cc2s1 CCC(C)(C(=O)N=S(C)(=O)c1cc(Br)ccc1Br)c1cnc(Cl)c(Cl)c1 CC(C(=O)NC(C1CCCN(C(C23CC(CF)(CO2)C3)=O)C1)C)C(F)(F)F c1(C(C)NC2OC(C)CC2C)ccc(CNC(c2ccc(Br)o2)=O)cc1 N1(C(c2nc(Br)sc2C)C(=O)NCCOCC)CC2CCOC2C1 S(=O)(=O)(c1ccc(S(=O)(=O)N2CCCCC(N(C)C)C2)cc1)NC(COC)CO c1(CNC(C(=C)C)=O)ccc(-c2ccc(-n3ccnc3)cc2)cn1 C(C)(CC(=O)NCC(C)(C)CC1CN(C(c2cnns2)=O)C1)OC c1(C(=O)NC2C(NC(C(COC)(C)OC)=O)C2)ccc(Cl)c2ncccc12 N1(C(C2CCC3(CC3)C2)C(=O)NCC=C)CCC(S(=O)(=O)CC)CC1 c1(OC)ncc(S(=O)(=O)N2CC3(CC(=O)CO3)C2)cc1Cl C(=O)(C(C)(C)CS(C)(=O)=O)NC1CN(C(Cc2cc(C)c(O)cc2)=O)C1 N1(C(Cc2nc(C)[nH]n2)=O)CCC(NC(=O)CC(C)c2ccncc2)C(C)C1 N1(C(c2c(C)n(CCO)cc2)=O)CCCN(C(=O)C(C)c2cccs2)C(C)C1 N1(C(C2(O)CCCN(C(C)=O)C2)=O)CCC2CCC(NC(=O)CCF)C1C2 N1(C(C2C(C(=O)OC)C2)=O)CCC2(CCCCN(C(C3CSCN3C)=O)C2)C1 c1(C(=O)NC2C(NC(=O)C=CBr)C2)cccc(Cl)c1O CCC(CC(=O)NCC1(C(=O)NC2CCSC(C)C2)CC1)C1CCC1 C(=O)(CC(F)(F)C(F)F)NC1CCN(c2nc(=N)[nH][nH]2)C1 c1(C(=O)NCCCN(C(C(c2cnn(C)c2)OC)=O)CCO)ncn2c1CCC2 C1(NC(c2ccn(CCNC(=O)C(F)OC(F)(F)F)c2)=O)CCC2CC1CO2 Cc1nc(C(F)(F)F)ccc1C(=O)NCCC1CN(C(=O)CC2CCC2(C)C)C1 C(C(=O)NCC(C)(C(C)C)NC(C12CC(CC(F)F)(C1)C2)=O)(C(C)C)OC C1(C(=O)OC)(C(c2ccccc2)C)CN=C(N2CC3(CC=CCO3)C2)NC1 Cc1cc(C)c(C(=O)NCC2CN(C(C34CCCC3C4)=O)CC23CC3)c(N)c1 C1(C=C)(CC(N2CC(CC(=O)N(CC(C)N(CCC)CC(=O)OC)C)C2)=O)CCC1 C1(NC(CN(C)C(N)=O)=O)CN(C(c2cccc(OC(C)(C)C)n2)=O)CC1(C)C CCCCCS(=O)(=O)CC(=O)NCC(CNC(c1c(SC)cnn1C)=O)OC O=C(C#CC1CCCOC1)NCCC1CCN(C(=O)Cc2nncs2)CC1(F)F N1(C(C)C)CCC(C(=O)NCC2CCC(NC(=O)CCC3CC(F)(F)C3)C2)CC1 C1(NC(c2ccnc(N3CCCC3)n2)=O)C2CCC1N(C(=O)C=Cc1cccs1)C2 CC(CS(C)=O)C(=O)N1CC(O)(CNC(C2CC3(CCC3)C2)=O)C1 c1(C(=O)NC2CCCN(C(C=C(C)C(F)F)=O)C2)ccc(C)cc1F C1(NC(c2c(OC)cncn2)=O)CCCCC1(C)O.N12CCCC1CCC2=O c1(CC)cc(C(N2CCC2(C)CCO)C(=O)NCC(F)F)on1 CC(CN(C)C)CN=c1ccnc(N2CCC(c3ccc(F)cc3)C2)[nH]1 N1(C(COCc2c(C)ncs2)=O)CCC(C(C)(C)C)(NC(=O)C(C)C(F)F)C1 Cc1cc(=NCC2CCN(C(c3cncc(F)n3)=O)C2)[nH]c(S(C)(=O)=O)n1 C12(C(N(C)CCNC(=O)C(F)(F)CO)=O)CCCC1C2(F)F N1(CCC)C(=O)CCC1C(=O)NC(C1CN(C(c2cc(OC)nn2C)=O)C1)C C1(CC(N2C(C3(O)CN(C(=O)C=C4CCC4)C3)CCC2)=O)CC2CCC1O2 CC(C)CCCCCCNC(c1ccn(CCNC(c2nnc(S)n2C)=O)c1)=O CCCCC(CNC(c1c[nH]nc1-c1ccnn1C)=O)NC(=O)Cc1cncs1 C1(C(=O)NCCc2ccsc2)(CNC(C2CCC2)=O)CC12CCC2 N1(C(C2CCN(C(C)=O)C2)=O)CC(C2(NC(=O)CCCCC#N)CC2)C1 C1(N(CC(=O)NCC)CC)CCN(C(=O)CN(C)C(=O)OC(C)(C)C)CC1 C(=O)(CCCCN=c1nc2c(cnn2C)c(NC2CCCCC2O)[nH]1)N(C)C C(=O)(C(CC(C)C)C(C)C)N1CC(COC)N(C(=O)Cc2ccc(F)cc2)CC1 c1(CC)nn(C)c(CC)c1CN=C(NCC)NC1CCC(N(C)C)CC1 N1(C(C(C)C2CCCC2)=O)CC(CC(N2CC(S(C)(=O)=O)C2)=O)C2(CC2)C1 c1(C(=O)NC2CC(CCNC(CC3(C#N)CC3)=O)C2)ccc(-c2ccccc2)s1 C1(N(C)C(C2CCO2)=O)CCN(C(c2cc(-c3ccccn3)no2)=O)CC12CC2 c1(-c2cccc(C#N)n2)nc2c(s1)CN(C(=O)Cc1cc(F)c(F)cc1F)CC2 N1(C(C2CCCN(Cc3ccc(OCCN(C)C)cc3)C2)=O)CCCCC(F)(F)C1 C1(C(C(=O)N(CCCCCNC(=O)CC2(O)CCOC2)C)O)CCS(=O)(=O)CC1 c1(N(C)Cc2c(C)ccs2)[nH]c(=NC(C)c2ccccc2Cl)nc2scnc12 C1(CCCNC(C(n2ccc(Br)n2)C)=O)CCN(C(C2COC2)=O)CC1 C(=O)(C(C)(C)C(N)=O)N1CCC(C(C(=O)NCc2onc(COC)n2)C)C1 c1(CC(C)NC(C(c2cccs2)NC(C2CC(SC)C2)=O)=O)cnccn1 c1(NC(C(C)N(CCC)C(C2CS(=O)C2)=O)=O)ccc(O)cc1F C12CCN(CC1n1cc(-c3cnccn3)nn1)C2=O.CN1CC(F)CC1C(=O)O C1(C(=O)NCC23CC(NC(=O)Cn4cnc(C(F)(F)F)n4)(C2)C3)CCS(=O)(=O)C1 C1(C(=O)NCCCN(C)C)C2CCC(C2)C1Nc1nccc(C)n1 C(=O)(CCCCCS(N)(=O)=O)NC(C1CCN(C(CCCSC)=O)C1)C N1(C(C(C)CO)=O)CCCCC(C2CN(C(=O)Cn3cnc([N+](=O)[O-])n3)C2)C1 C1(CNC(c2ccc(CO)cc2)=O)CCN(C(c2cnn3ccsc23)=O)CC1O N1(CCCNC(=O)NC(CC)CCOC)CCCNC1=O CCCC(C)CCCC(=O)N1CCN(C(c2ncc(N)cc2C)=O)C(C(F)F)C1 N1(C(c2c(CC)nc(C)[nH]2)=O)CCCCC(NC(c2ccc(O)cc2)=O)C1 C12(NC(CCCOC)=O)CC(CNC(=O)CC3CC3C(F)(F)F)(C1)C2 C#Cc1cccc(C(=O)NCCC2(O)CCN(C(=O)CC=CC)CC2)c1 N1(C(C23CCCC2C3)=O)CCN(C(=O)C(F)=CC2CC2)C(CF)C1 N1(C(C(C)Cc2ccccc2)=O)CCCC12CN(Cc1ccc(F)c(Cl)c1F)C2 C1(C(=O)NCCC(C)N(C)C(C2CC(=O)C23CCC3)=O)Cc2ccccc2C1C c1(C(=O)NCc2occ(C(N(CC(C)(C)C)CC)=O)c2)cccc(C)c1O CN1CCc2cc(CC(N3CCc4nc(I)[nH]c4C3)=O)ccc21 C(=O)(CCCC(C)(C)C#N)N1C(CN(C(C(C)(C(C)C)OC)=O)C)CCC1 CC1CC(C(=O)O)(NC2(C3CCCO3)CCC2)CCO1 c1(C(=O)NC(C(C)NC(Cc2c(C)nc[nH]2)=O)C(C)C)ccc(F)cc1[N+](=O)[O-] CC1(C)CCN(C(C2CC3(CC(NCc4ccc[nH]4)C3)C2)=O)CC=C1 c1(C(N2CC(F)(F)C2)=O)ccccc1-c1ncccn1 Cc1cc(OCC(=O)NC2(C(=O)NCc3ccn(C)c3)CCCC2)cc(C)c1 C(CC1=CCN(C(=O)Cn2cc(Cl)cn2)CC1)NC(c1cccc(OCC)c1)=O C(=O)(C1=NNC(=O)CC1)NCCCN(C(C(CO)N(C)C)=O)C1CC1 N(C1c2ccccc2CC1NC(C1CNC(=O)O1)=O)C(C(CCC)(C)CC)=O Cc1nc(CN(C(=O)CCC2CCCN2C(=O)CC2(N(C)C)CC2)C)no1 c1(C(=O)NCCC2CN(C(=O)C=Cc3cc[nH]n3)C2)ccc2c(c1)CCOC2 c1(C(C)(F)F)ccnc(C(=O)NCCC2CN(C(C3CCC(=O)C3)=O)CCO2)c1 CC1(C(=O)N2CC(NC(C3CC3[N+](=O)[O-])=O)C2)COc2ccccc21 C1(NC(C2OCCN(C(CSCC)=O)C2)=O)CCN(OC)CC1 c1(OC)cccn2ncc(C(=O)NCC(C(C)C)NC(c3cccc(C)c3)=O)c12 N1(C(C(C2CC(C)(C)C2)OC)=O)CC(N=c2[nH]nco2)C(C)(C)C1 N#CCCCCCC(=O)NCC1(F)CCN(C(c2ccc([N+](=O)[O-])s2)=O)CC1 C1(C(=O)OCC2CC(=O)NCC2)CN2CCN1CC2 C1(C(=O)NC)CC(OC)CN1C(=O)Nc1cccc(C(=O)OC)c1 Cc1c(Cl)ccc(C(=O)NC(C2CN(C(=O)CCn3ccnc3)C2)C)c1Cl c1(CC)ccc(O)c(C(=O)NCC(C)(C(C)C)NC(=O)C(C)C2CCC2)c1 CCC(CC)CCC(=O)N1CC(NC(c2oncc2C)=O)CCC1C N1(C(c2cccc(Cl)c2Cl)=O)CCC2CN(C(C3(F)CCOCC3)=O)CC2C1 c1(C(=O)Nc2ccc(OC)c(C)n2)cc2ccccc2[nH]1 N1(C(C2OC3CCC2C3)=O)CCC2(CC1)Nc1ccccc1NC2=O C1(NC(C2(C#N)CCCO2)=O)CC2CC(NC(=O)C(C3CC3)C3CC3)CC12 C1(NC(CSc2nc(C)[nH]n2)=O)CCCCN1C(=O)C(c1cnn(C)c1)C C1(CC)CN(C(=O)COC2CCCCC2)CCN1C(=O)C(C)NC(C1CC1)=O C=CCC(CNC(c1nccnc1CC)=O)C(=O)NCc1cccc(O)c1 S(=O)(=O)(c1ccc(NCC(c2cnn(C)c2)(C)C)cc1Br)NCCC C(=O)(CC(C)CC(C)(C)C)N1CCN(C2CNC2)C(=O)C1.Cc1ccc(O)cc1C c1(C(N(CCC(C)NC(CCCCC#C)=O)C)=O)ccc2c(c1)C=CS2(=O)=O N1(C(CCCCSC)=O)CCC2C(C(=O)NC(CCO)C(C)(C)O)C2C1 C1(C(=O)N(CC(N(C(=O)CNC=O)C)C2CC2)C2CC2)OCCCO1 C=CCC(CC)C(=O)NC1CCCC1NC(=O)CCOCC1CC1 CC1C(=O)N(C)CCN1C(=O)C(=O)NCc1cccc2c1OCC2 S(=O)(=O)(c1ccc(Cl)nc1C)N1C(COC)CN(C(c2scc(C)c2Cl)=O)CC1 CC1=C(C(=O)N2CCCC2C2(NC(=O)C(O)C3CC3)CC2)C(C)(C)CCC1 C1(C)(CNC(C2C(CC)C2)=O)CCCN(C(=O)C(CC(C)C)N(C)C)C1 c1(C(=O)NCCC(C)NC(C2CCN(C)C2)=O)cnc2occc2c1 C(=O)(C=CS(F)(F)(F)(F)F)NCC(C1CC1)NC(c1cccc(C)c1F)=O N1(C(CN(C(C)C)C(c2cc(C(C)C)no2)=O)=O)C2CCC1CCSC2 c1(OC)ccc(CCCC(=O)NC2CCCCC2CNC(=O)CCCSC)cc1 c1(C(=O)NCCN(C(COCC=C)=O)C(C)C)nccc2cccnc12 Cc1ncc2n1CCC(NC(=O)NC1CCCN1CC1CCCCC1)C2 CCC(CC)(CCNC(=O)CCCCN(C)C)NC(=O)C(C)Cc1ccccn1 CCC(CC)C(=O)N1CCC1CO.N1(C2CC(C)(N)C2)CCN(C(=O)CC(C)CF)CC1 N1(C(c2nn(C)c(F)c2)=O)CC(NC(c2c(F)cc(F)cc2F)=O)C(C2CC2)C1 c1(C(N2CC(COC)N(C(=O)CC3OCCCO3)CC2)=O)ccc([N+](=O)[O-])cn1 n1(C(N2CC(C)(NC(c3cnn(CCF)c3)=O)C2)=O)nnc2c1CCCC2 C(=O)(C#CC1CCOCC1)NCCOCCNC(c1ocnc1CO)=O N1(C(C(N)=O)=O)C2CCC1CN(C(=O)NC1(C(F)(F)C(F)(F)F)CCC1)C2 N1(C(C2C(C)C2C)=O)CC(F)(F)CC1(C)CNC(c1cc(C(C)(F)F)on1)=O c1(N(C)C)ncc(NC(c2scnc2C(C)(F)F)=O)cn1 C1(CNC(C(C)(C)OC)=O)C(C2CC2)CCN1C(c1nccn2nccc12)=O c1(C(=O)NC2CCC(C(=O)NCc3ccc(C)o3)C2)ccc2ccoc2c1 C1(CC(=O)N(C)CC2(O)CN(C(C3(CSC)CCC3)=O)C2)CCCCC1O C1(NC(=O)CN2CC3CC3C2)(CNC(c2csc3cncn23)=O)CC2CCC1C2 c1(NC(C(C)O)(C)C)ccc(S(=O)(=O)NCCC23CCCC2C3)c2ccncc12 c1(OCCOC)ccc(NC(C2CC2(F)F)C)cc1 C(CCN(C(=O)Cc1nnc(C)o1)C1CC1)(C(C)C)NC(C(C=C)O)=O C=CCC(C)(C)CC(=O)N1CCCC1(C(=O)NC1CCOCC1C)C(C)C C(=O)(CC(C1CC1)NC1(CCO)CCC1)N(CC(=O)NCC1CC1)C C(CCCCC(=O)N1CCC(O)(C(C)NC(c2ccc(C)nc2)=O)C1)OC N1(C(c2n(C)cc(C#N)c2)=O)CCC2CCCC12C(=O)NCC(C)(C)C(F)F c1(C(=O)OC)c(NCC2(C(C)(C)C)CCN(C(=O)C(C)C(F)F)C2)ncnc1Cl CC1CC(CNC(C2(CNC(=O)CC3CCCC3O)CCC2)=O)CCO1 c1(C(N2C3CN(C(C(CN(CC)CC)F)=O)C(C3)C2)=O)cc2oc(C)cc2[nH]1 c1(C(N2C(C)CC(NC(Cc3ccc(C#C)cc3)=O)C2)=O)ccc(C#N)nc1C c1(CCC(C)NC(=O)C(N2CCSCC2C2CC2)=O)cc(F)c(F)c(F)c1 c1(C(=O)NCCC2(OC)CN(C(CCCC#C)=O)C2)ccc(C)c(CO)c1 CCC(C(c1nnnn1C1CCC1)NC1CC1c1cnn(C)c1)=Cc1ccsc1 C(C)(C(C)(C)C(=O)NC1(C2CC2)CC1)NC(C(C)OCCC=C)=O c1(C(=O)NC2CC2C(=O)NC(COC)CO)cc(N)ccn1 c1(CC(=O)NC(C(=O)NC(C(C)(C)OC)C)CC2CC2)cccc(F)c1 N1(C(C(C)SC(C)C)=O)CC(CNC(=O)CCCCC(N)=O)CC12CCC2 C(=O)(CCCC(=O)C(C)(C)C)NCCN(C(CN(CCCCCC)C)=O)C(C)C c1(NC(C2C(CNC(C)=O)CCCC2)=O)ccc(Cl)cc1C(F)(F)F C1(CCC#C)CCCN(C(C2(CC=C)CN(C(=O)C(C)C3(O)CCC3)C2)=O)C1 C(=O)(CC(N)C(F)(F)F)NCC(c1ccc(OCC(=O)OC)cc1)O Cc1csc(C=CC(=O)NC(CCNC(c2cnc(Cl)n2C)=O)C(C)C)n1 N1(C(CC=C)=O)CC2C3CCC(C2C1)N(C(C1(C)CC(O)CN1C)=O)C3 c1(C(=O)NC2CN(C(C3CC(=C)C3)=O)CC2C)ccc2c(c1)-c1ccccc1C2 c1(C(=O)NC(CN(C(=O)CNC(C)=O)CC)C)ccc(-n2nc(C)cc2C)cc1 C(=O)(CC(C(F)F)NC(C1CC1(F)F)=O)NCCC(=O)NCC N(C(=NCCC1(OCC)CCOC1)NCc1cscc1C)C(CC)C CCCC(CC)C(=O)NCC1(F)CCN(C(=O)CCCCC2CCCCC2)C1 c1(SCC)cccc(C(=O)NC2CCCC2NC(=O)CC2CCC2(F)F)c1O CC(C)CC(C(=O)N(C1CCN(C(C2C(C3CC3)C2(F)F)=O)C1)C)NC(N)=O c1(C(=O)NC2C(OC)CN(C(CNC(CC)=O)=O)C2)cc2sccc2s1 c1(OC)ncc(C(N2CC(O)C(O)C2CNC(=O)Cc2[nH]cnc2C)=O)c(C)n1 C=CCCCC(=O)NC(CC)C(C)NC(=O)COCCCN(C)C N1(C(C(C)NS(CC)(=O)=O)=O)CCC(NC(=O)C(C)(C)c2ccncc2)C(C)C1 Cn1cc(S(N)(=O)=O)cc1C(=O)NC1C2CCN(C(C3CCCCN3N=O)=O)C12 C1(NC(c2c(C)c[nH]n2)=O)CN(C(C2(F)CCOC2)=O)CC1C C1(NC(c2cccc(C)n2)=O)CCC12CN(C(C1COC3(CCC3)C1)=O)C2 NS(=O)(=O)N1CCC(C(=O)NCCNC(C2CCC(=C3CCC3)CC2)=O)CC1 C(=O)(CCCCC(C)(C)C)N1CCN(CC(=O)NCc2ncc(C)[nH]2)CC1 O=C(C#CC1CCCO1)NCC1CCC1NC(c1ncoc1CCC(F)(F)F)=O N1(CC(=O)NC(C)C2CC2)CCN(C(=O)N(c2ccccc2)C2CCC2)C(C)C1 N1(C(c2cc(Cl)ccc2F)=O)C2CCC1CN(Cc1ncccn1)CC2 N1(C(C(CCNC(C(C)N=[N+]=[N-])=O)O)=O)CCCC(F)(CO)C1 N1(C(C=CCN(C)CC)=O)C2CCC1CC(CNC(=O)COc1ccsc1)C2 C1(NC(CN(C(c2c(C)csc2)=O)C)=O)CCOC(C)(C)C1 c1(C(N2CCC(C)(CNC(c3nc(Cl)ccc3N)=O)C2)=O)ccc2nonc2c1 C(C1CCCCC1)=CC(=O)NCCn1ccc(C(=O)NCC(O)C2(Cl)CC2)c1 FC1CC(N=c2[nH]c(=NCc3ccc(C(F)(F)F)o3)[nH]c3c2COC3)CCC1 O=C1CCN(CCS(=O)(=O)N2CCCCC2)SC1=O FCC(CN=c1[nH]c(N2CC3CC2C3)nc2c1COC2)c1ccccc1 C(CNc1nc(C(F)(F)F)cc(C)n1)(C(C)C(C)C)NC(C(CCOC)OC)=O c1(C(=O)NCC2(O)CN(C(C3(C(N(C)C)=O)CC3)=O)C2)ccc(O)c(F)c1F CC1CN(C(c2c(Cl)nsc2Cl)=O)CC1N=c1ccc(C#N)c[nH]1 C(=O)(CCCC(F)(F)Br)NCC(C)(C1CC1)NC(C(C(CC)C)OC)=O Cc1nn(CCC(=O)NCC(C2CCC2)NC(C2CCC3(CC3)C2)=O)c(C)c1C c1(SC(C(C)NC(C2CC(C)C2)=O)CO)nocc1C(=O)NC C1(C(N(CCCF)CC)=O)C=CCN(C(=O)CC2CCC=CCC2)C1 N1(C(c2c(CC)c[nH]n2)=O)CCC(C(=O)NCc2csc(NC=O)n2)C12CCC2 N1(C(c2cc(C3CCCNC3)no2)=O)CCc2cc(Br)c(O)cc2C1 C12(CNC(CC(C)CF)=O)CC(NC(c3ccc4c(c3)CC4)=O)(C1)C1(CCC1)O2 C1(C(=O)NCC(C(C)(C)C)NC(C2CN(C3COC3)C2)=O)CCn2cnnc2C1 C1(C2CCN(C(=O)C(C(C)C)NC(=O)COC)C2)(NC(CCOC)=O)CC1 C1(NC(C(CC)(C)C(N)=O)=O)CCC2(CC1)CN(C(=O)CCCNC(N)=O)C2 C1(NC(C2(CC=C)CC2)=O)(CNC(=O)Cn2cnc(C)cc2=O)CCCCC1C C1(CC)COCCN(C(c2cc(CNC(c3cnoc3C(C)C)=O)no2)=O)C1 N1(C(C2C(CC)CCCN2C(=O)CCc2ccccc2)=O)CCC(O)CC(C)C1 c1(OC)cccc(C(=O)NCC(c2ccc(F)cc2)NC(=O)CC(C)(C)OC)c1 CN1CCN(C(N2CC3C(C4(NC(C5CC6C=CC5C6)=O)CC4)C3C2)=O)CC1 c1(C2C(C(=O)NCCCN(C(c3cncc(C)c3)=O)CC)CC2)ccc(F)cc1 c1(CC(=O)N(C2CCCN(C(=O)C(O)P(C)(C)=O)C2)C)c[nH]c2ccc(Cl)cc12 CCC(CC(=O)N1CC2CCC1CN2C(=O)C(C)CC(C)C)C(C)(C)C C1(C(=O)NCC(C)Cc2ccco2)CC(F)CN1C(=O)C(F)=CC1CC1 C(=O)(CCCC(=O)N1CCCC(NC(=O)CCCCN(C)C(C)=O)C1C)OC Nc1ccc(C(=O)NCCN(C(c2ccc(C(F)(F)F)cn2)=O)CC2CC2)nc1N C1(CCOC(C)C(=O)NC2CCN(C(=O)Cc3ccccn3)C2)CCCCC1 n1(CC)ccc(C(=O)Nc2cccc(NC(=O)COC3CC(F)(F)C3)c2)cc1=O C(C(=O)N(C)OC)NC(c1n(CCCSCC)nnn1)c1nccn1C(C)C.SCC C(=O)(C(O)CCNC(=O)COC1(C)CCOC1)NC C1(CN(C(=O)C(F)C2CCC2)C)COCCN1C(C12CCCCC1C2)=O C(=O)(C1=CCC(F)(F)CC1)NC(C(C)C)CCNC(=O)C(=O)NCC.C(CC(N)=O)SCC C12(C(=O)NC(CC)(CC)C(C)C)CCN(C(=O)C=Cc3cncs3)CCC1C2 c1(NC(C2(O)CCN(Cc3cc(F)c(F)cc3O)C2)=O)ccn2ccnc2c1 c1(C(N2CC3(CC(CNC(=O)CC4C=CCCC4)C3)C2)=O)cc2ccccn2n1 N1(C(CCc2cn(C)nc2)=O)CC=CC1(C)C(=O)Nc1csc(Cl)c1 CC#CCC(C(=O)NCc1cnc(C)[nH]1)NC(c1cnc(C)cn1)=O C1(CC(=O)NCCC2(NC(C3CCS3(=O)=O)=O)CCC2)CC2CC2C1 C1(C(=O)NC(C2CN(C(=O)C(O)C(C)(C)C)CCO2)C)C2CCC(C2)C1(C)C c1(C(N2C(CNC(CCC=CCC=C)=O)CC(OC)C2)=O)cc2c(nn1)CCC2 CC(C)S(=O)c1ccc(C(=O)NCCCN(C(=O)Cc2csc(=N)[nH]2)C2CC2)cc1 c1(CC)cc(C(=O)N(C)CC2C3CN(C(c4nocc4Cl)=O)CC23)oc1CC c1(N2CCC(CF)C2)nc2cc[nH]c2c(=NCC2CCCc3cncn32)[nH]1 CCCC(C(=O)NCC1CN(C(C2(C(=O)N(C)C)CC2)=O)C1)S(N)(=O)=O c1(NC(C2C(c3n(C(C)C)ncc3)C2)=O)cccc(CCCCOC(C)(C)C)c1 c1(C(N2CCC(CSC)C2)=O)n[nH]c2ccc(C(C)=O)cc12.C1C(O)C(=O)N1C C1(C(=O)NC(C(C)C)(C)CNC(C2(n3cnnn3)CC2)=O)OCCN(C)C1=O c1(C(N(C(C#C)C)C)=O)cccnc1CNC(C1(OCC)CCOC1)=O N1(CC(=O)NC2CCC(CCNC(c3c(C(C)C)cco3)=O)C2)CSCCSC1 c1(-c2n(C)cnc2)ccc(CN(CCC[Si](C)(C)C)C2CC2)cc1 c1(C(=O)NC2CC(NC(CCC(=O)c3ccccc3)=O)C2)coc2ccccc12 c1(C(N(C2CCCN(C(C(C)CF)=O)C2)C)=O)ccc(=O)n2c1CCC2 N1(C(COCc2ccc(C)cc2)=O)CCC2(NC(C3C=CC=CC=C3)=O)CC2C1 c1(OC)cc(CN(C)CC2CCN(C(c3csnn3)=O)C2)ccc1C(F)F C1(C(N(C(C)CCC)CC)=O)CCCCN1CC.c1(C(=O)NCC)cc(C(F)(F)F)ns1 C1(NC(c2ccc(CF)cc2)=O)CCCCN(C(=O)Cn2cc(C3CC3)nn2)C1 C(c1ccc([N+](=O)[O-])s1)=CC(=O)NCCC1(O)CN(C(=O)C=Cc2cccs2)C1 C1(C(N2CC(CCC#C)C2)=O)CC(F)(F)CN1C(=O)CCC(C)CC c1(CC(=O)NCC2CC(NC(=O)CN3CCCCC3)C(O)C2)cncc(F)c1 c1(CCC(=O)NC(C(C)(C)NC(Cc2cnc(C)s2)=O)C)cccc(F)c1F N1(C(c2cc(CC)nn2C)=O)CCN(C(c2cc(OC)ccn2)=O)CC12CC2 C1(C(N2C(C#C)CCC2)=O)CCN(C(=O)C=C(C)c2ccco2)CC1(C)C N1(C(C(CCC)=CCC)=O)CC2CCCC(C(=O)NC3(CO)CCSC3)C2C1 Cn1cc(C(=O)NC2CN(C(=O)Cc3cnsc3)CC2O)c(C2CC2)n1 Cc1nc(=NC(=O)C2CC23CCN(C(=O)Cc2ccc(Cl)cn2)CC3)o[nH]1 C1(NC(c2c(CC)n[nH]c2)=O)CC1C1CCCN(C(c2cc(C3(C)CC3)n[nH]2)=O)C1 CCC(C(=O)OC)NC(C1CC(CNC(c2cnn(C(C)C)c2)=O)C1)=O CCCCCCCCC(=O)N(C)CC1(CNC(C2COC(=O)C2)=O)CC1 C1(NC(c2cccc(C#C)c2)=O)CCN(C(=O)Cc2csc(=N)[nH]2)CC(O)C1 C(=O)(CC(CNC(=O)CC(C)(C)C)C1CCC1)NC(C#C)CC N1(C(c2ccccc2)C(N)=O)CCN(Cc2sccc2-c2nn[nH]n2)CC1 C1(C(=O)NCc2scc(C)n2)CCN(C(=O)C2(C)COCCO2)O1 N1(C(C(CC#C)C)=O)CC(NC(=O)C#CC2(C)COC2)C2(CCC2)C1 c1(C(N2CCC(C(C)NC(C3CC(=C)C3)=O)C2)=O)ccc2cncc(Br)c2c1 Cc1ccc2nc(NC(N3CC(C4(C(F)(F)F)CC4)C3)=O)cn2c1 C#CC1(C(=O)N(C2CCCC2)CC(C)C)CCN(C(C2CCCCC(=O)N2)=O)C1 C1(CC)CN(Cc2ccno2)CCN1c1ncc(F)cn1 C(=O)(C(CC)CC)N(CC(CC)CC)CCOCCOC C1(CNC(C2C(C(=O)OC)C2)=O)C(C)CCCN1C(=O)CCN(CCCCC)C N1(C(C(C)OCCC=C)=O)Cc2ccccc2C(NC(c2ccsc2C)=O)C1 C=CCC(C(=O)NC(C(=O)NCc1cocn1)C1CCCC1)C(C)C S(=O)(=O)(c1ccc(NCCC(O)C2CC2)c(F)c1)NC(c1cccnc1)C(C)C C(C(C)(C)CC(=O)NC(CCC(=O)NCCCCC(=O)NC(C)C)C(C)C)OC C(CCN=c1[nH]cnc2c1CCCCC2)NC(C1CC2CCC1C2)=O C(N1CCN(Cc2conc2C2(C)COC2)C(C)C1)SC Cc1cc(N)cnc1C(N1CCC(NC(=O)CN(CC(C)(C)C)C)C1)=O C1(C2CN(c3nnc(C)s3)C2)CN(C(C2(C(=O)OC(C)(C)C)CCC2)=O)CCO1 N1(C(C(N2C(=O)CCC2=O)C)=O)CCC(C)(NC(=O)CN(CC(F)F)C)C1 O=C(C1=C(Cl)CC1)NCCC1CC(CC(=O)NC(=O)C(c2ccccc2Cl)O)C1 C(C1CCN(C(C2(F)CC2)=O)CC1)=CC(N1CCC(C(=O)NC)C1)=O C=CCC(CNC(=O)C(CC(C)C)OC)C(=O)NC(C)C(C)(C)OC C(C)(C(C(C)C)NC(=O)CCCNC(N)=O)NC(CCCn1c(C)ncc1)=O N1(C(c2c(C)nn[nH]2)=O)CCCC(C)(NC(c2cnc(C(C)C)s2)=O)C1 c1(OC)cc(C(=O)NCCNC(=O)CC2CC(SC)C2)ccc1S(C)(=O)=O c1(C(N2CCC(CC=C)(NC(c3ccnc(C)c3)=O)C2)=O)ccc(C)nc1O c1(OC)ccc(C(N2CC3(C2)CN(C(C2(C)CC2C)=O)C3)=O)c(Br)n1 C(C1CCCCC1)=CC(=O)N(C(CNC(C1(C#N)CC12CC2)=O)C1CC1)C c1(CNC(C2SCCN(Cc3cccc(OC)n3)C2)=O)cccc(F)c1O CC(C)C#CC(=O)NCC(c1cccc(Cl)c1)NC(=O)C(C)N1CCCC1 N1(C(C=NOC)=O)CCC(F)(F)C(CNC(C2CC(SC)C2)=O)C1 c1(C(=O)NC2(C)CC(NC(C(CCC)OC)=O)C2)ccc2ncsc2c1 C1(C(=O)NCC2(N(C(C3CC(SC)C3)=O)C3CC3)CCC2)CC1C1CCOCC1 c1(CC(=O)N(CC(C)N(CC(N2CCC(C(=O)OC)C2)=O)C)C)cncn1C1CC1.C(C)=O c1(C(=O)NCCN(C(C(n2ncc(C)c2)C)=O)C)cc(C)c(F)c(S(C)(=O)=O)c1 C1(NC(C2CC(C)(O)C2)=O)CN(C(=O)Cc2ccc(Br)cc2)C2(CCC2)C1 C1(C(=O)Nc2cncnc2I)CCC2(CN(C(c3ccc(O)cc3)=O)C2)O1 c1(OC)ccc(C(N2CCN(C(c3cc[nH]c(=N)c3)=O)CC2)=O)cc1 CCS(=O)(=O)c1ccc(CNC(=O)Nc2nn(C)cc2C(F)F)cc1 C#Cc1cccc(C(=O)N(CC(N2CCCC(C)(N(C)C)C2)=O)C2CCC2)c1C c1(C(N2C(COC)CN(C(c3cnc(C)nc3)=O)CC2)=O)scc2c1OCCO2 CC(N=c1[nH]c2c(C(F)(F)CC3CC3)c(F)c(F)c(F)c(F)c(F)c1-2)c1cccs1 c1(C(N(C2CCCC2)CCCNC(CCCSC)=O)=O)ccncc1C(F)F C1(CCO)(CNC(=O)C(C)C2CCC2)CN(C(=O)C=CCC2(OC)CCC2)C1 C1(CNC(Cc2c(C)con2)=O)CCC(N(C(=O)Cc2ccc(F)cn2)C)CC1 C1(C(=O)NC2C(NC(c3ccncc3)=O)C2)CCc2nnnn2C1 CC(Cn1ccnc1)C(=O)NCC1CCCC1NC(=O)CC1CCCCO1 c1(OC)ccc2c(c1)C(C(=O)N1CCC(Nc3ncc(C)cn3)C(C)(C)C1)CC2 CC1=NOC2(C1)CC(C(=O)NC1CC(CNC(c3cn(C(C)C)cn3)=O)C1)C2 C1(C(CNC(c2c(CC)cco2)=O)(C)O)CCN(C(=O)Cc2nc(=N)[nH][nH]2)CC1 C1(CC(N2C(C=C)CC2)=O)CN(C(=O)Cc2nncn2CC)C2(CCC2)C1 c1(CCNC(C2C(C)OCC2)=O)ccc(CNC(=O)CC(F)(F)F)cc1 N1(C(C(CC)(C)C)=O)CCC=C(C(=O)C(CCc2ccc(O)cc2)=O)C1 c1(C(=O)NCC2N(C(c3ccc(SCC)cc3)=O)CC2)csc(S(C)(=O)=O)c1 C1(CNC(C2(CNC(C(C=CC)O)=O)CC=CC2)=O)CCOC1(C)C C1(N(C(=O)C=Cc2cnc[nH]2)C)CCC(NC(c2csnc2Br)=O)CC1 C1(N2CC(CNc3ncc(C(=O)OCC)nc3)C2)CCC(C)(C)CC1 c1(-n2cc(OCCN(C(CC=C)(C)C)C=O)nn2)ccccc1[N+](=O)[O-] C1(CNC(CCCSC(C)(C)C)=O)CC2CCC1N(C(c1ccccc1F)=O)C2 n1(CCOC)ncc(C(=O)NCCCN(CCSc2ncc(C)o2)C(C)C)c1C c1(C2C(C(=O)NCC(C)(C)NC(c3c(CCC)[nH]cc3)=O)C2)ccc(C)nc1Cl CCC(C)C(C(=O)NC1C2CC1CN(C(c1ccc(CO)nc1)=O)C2)NC(N)=O C(=O)(C1CCCc2ncccc21)N1C(CNC(c2nc(C3CC3)ns2)=O)CC1 CC(CCC(=O)NCc1csc(C(=O)NC2CCCC2(C)O)c1)N(C)C c1(NCC(CNC(C(C)OCC)=O)O)cc(C)nc(S(C)(=O)=O)n1 C#Cc1ccc(CC(N2CC3CC2C3CNC(=O)CC23CCCC2C3)=O)cc1 Cc1cnn(C)c1C(=O)NCCCCN(C(=O)C(c1ccc(Cl)s1)=O)C C(C)(CCC(=O)NCCC(C)NC(=O)C(=O)NCCC(F)F)OC(C)C N1(C(=O)COc2ccsn2)CCC(C2CCCN2C(=O)C(F)C2CCC2)CC1 Cc1cc(C)n(CNCCNC(c2cc(CC(C)C3CC3)on2)=O)n1 C(=O)(C(C(C)C)N(C)C)NC(c1ncc(C)[nH]1)C.N12CCC(C1)C2=O c1(OC)cc(Br)ccc1OCc1cc(Br)cc(I)c1 c1(C(=O)NCC(C(C(=O)N2CC(=CCC)C2)F)C)ncc2ccccn12 c1(C(=O)NCCCC(C)NC(C(C)OCC#C)=O)c[nH]c2ccc(F)cc12 CC1CC(NC(c2cccc(N)n2)=O)CCN1C(c1ccc(C(F)F)o1)=O N1(C(=O)NCC(CCCCC)=O)Cc2ccccc2C1CCO C1(S(N)(=O)=O)(C(N2CC(CCC)C(C(N3CC(c4ccon4)C3)=O)C2)=O)CCC1 C1(C(=O)NCC(N(C(C2(COC)COC2)=O)C)C2CC2)C2CC3C(C2)C13 c1(C(N2C(CN(C)C(C3CCC(=O)N3)=O)CCC2)=O)cc(Br)ccn1 c1(C(=O)NC(CNC(C(C(=C)C)(C)C)=O)C2CCC2)cccc2c1OCC2C c1(CC)ncc(C(N2CC(CCNC(=O)CSCC(C)C)C2)=O)c(C)n1 C1(C(=O)NC(C)C)(NC(C(=O)NCC)=O)CC1(C)C C1(NC(CC2(OC(C)(C)C)CC2)=O)C=CC(C(F)(F)F)C1.C12CC(C1)C(=O)N2 C1(NC(CC2CC(=C)C2)=O)CCN(C(c2cnccc2C(F)(F)F)=O)CC1F C(N=c1nc(N2C3CCC2CC(F)C3)c2c([nH]1)CCC2)c1cccc(C(N)=O)n1 C1(C(=O)Nc2cccc(C(=O)NC)c2)C2CC1CN(C)C2 C1(C(=O)NCCC(Cc2cccs2)NC(c2n(CC)ncc2)=O)CCCNC1=O c1(NC(N(C(CC)CC)CCO)=O)nccc2ccccc12 c1(C(N(CCCOCCNC(Cc2cc(CC)no2)=O)C)=O)ccc(F)cn1 c1(C(N2C(CNC(C(F)=CC)=O)CCCC2)=O)cccc2c1CC(=O)N2 C(=O)(CCCCCC(C)(C)C)NC1(CNC(C(C)CC(F)(F)F)=O)CC1 c1(C(N2C3CCC(NC(C4CCC=CCC4)=O)(C3)C2)=O)ccnn2ccnc12 c1(NC(Cc2nc(NC(CCC=C)=O)sc2)=O)ccc([N+](=O)[O-])c(F)c1 C(C(F)(C(=O)NCCN1CCCC1=O)C(C)C)NC(c1scc(C)c1)=O C1(NC(C=C(COC)C)=O)CC12CCN(C(C1(C#N)CCCOC1)=O)C2 c1(C(N2CCC3CN(C(C4=CCC(C)CC4)=O)CC32)=O)ccc2nn(C)cc2c1 N1(C(C(CN(CC)CC)F)=O)CCCC1(C)CNC(c1ccccc1SC)=O c1(NC(C=CCC2(NC(CC(C(C)C)O)=O)CCC2)=O)cc(C#N)ccc1O C1(NC(CCNC(=O)OCC)=O)CCCCN(C(c2cc(C(F)(F)F)no2)=O)C1 C1(NC(=O)C(C2CCN(C(=O)C(F)n3ccnc3)CC2)F)(CO)CCOCC1 c1(CC)ccc(C(=O)NC2CN(C(C3(C(F)F)CCCC3)=O)CC2F)c(C)c1 C1(NC(COCCCCCC)=O)CCCCN(C(c2cc(C)oc2CC)=O)C1 c1(C(=O)NCC(CC)N(C(CCC)=O)C)c(Br)ccc(F)c1F C1(C)(C(=O)NC2C3CN(C(c4cccc(OCC)c4)=O)CC32)CCN(C)C1=O c1(C(=O)NC2CCCC2NC(C2CCN(C(N)=O)CC2)=O)cc2ccnn2cn1 C1(CNC(CC(=C)C)=O)CN(C(C)C)CCO1.c12cc(ccn1)OC2 N1(C(c2c(COC)cc[nH]2)=O)CCN(C(c2cc(Cl)ccc2OC)=O)C(C)C1C C1(CCC)CN(C(=O)C(C)N(C)C(C)=O)CCN1C(=O)CCCc1cccs1 C(=O)(CCCS(C)(=O)=O)N1CCC(NC(c2cnc(C)s2)=O)C1C C#Cc1cccc(C(=O)N(CCNC(=O)CCC2CCCC2)CC2CC2)c1 c1(OC)cccc(F)c1C(=O)NC(C)C(C(C)C)NC(c1cc(F)cs1)=O C1(=CC(=O)NC(C2CCN(C(c3c[nH]nc3C3CCCO3)=O)C2)C)CCC(C)C1 c1(NC(C2CCCC(NC(c3ccc(C)cn3)=O)C2)=O)cnc(Br)c(Br)n1 c1(C(=O)NCC2CC3(CO2)CN(C(C2CCSC2)=O)C3)cccc2ccccc12 Cc1cccc(Br)c1C(=O)NCCN(C)C(C1C=CC=CC=C1)=O C1(CC)CN(C(=O)C=Cc2nccs2)CCC1NC(C1(C(F)(F)F)CC1)=O C=CC(CCC)CC(=O)N1CCCC(CC(N2CCC(C)=C(C)C2)=O)C1 Cc1cc(F)c(C(=O)NC(C2CCCN(C(c3cc(F)cn3C)=O)C2)C)cc1Br N(C(=NCC12CCC(CC1)OC2)N(C)Cc1cccs1)C(c1ccncc1)C c1(C(=O)OCC)ccc2c(c1)CC(NC(=O)NC1CC1c1cccs1)C2 C1(CNC(c2ccsc2)=O)CCCC2(CN(C(=O)CC(=O)Nc3nccs3)C2)O1 CCCCCC(C)(CC)C(=O)N1CC2CC(C1)N2C(c1cccc[n+]1[O-])=O C#CCCC(O)C(=O)N1CCCCC1C1CCN(C(c2c(Cl)cnn2C)=O)CC1 c1(OC)ccnc(NC(C2CCC(C)N2C(c2cncc(C)n2)=O)=O)c1I c1(OC(C(=O)NCC2CN(C(CC=CC=C)=O)CC2C)C)ccc(Cl)cc1C Cc1cc(Cl)cc(C(=O)NC2CCCC2CNC(=O)CSCC2CCCO2)c1C c1(N(CC(C)C(C)(C)C)C)ccc(Br)c(F)c1F c1(CC(=O)N(C(C)CNC(=O)C=Cc2cc[nH]n2)C)cncnc1O C(C(C)(C)C(=O)N(C1CCN(C(=O)Cn2nccn2)CC1)C)SC c1(Sc2[nH]nc(C(N3CCC(N(C(CCC)=O)C)C3)=O)c2Cl)cncc(C)c1 C(=O)(CC(C)P(C)(C)=O)NCC(CNC(C(=Cc1cccnc1)C)=O)O N1(C(CNC(C2CCC(C)O2)=O)=O)CC2CC1C2C(=O)N(CC(F)F)C c1(C(C(=O)NCC(C)CN(C)C(C2(C)CC(F)C2)=O)=O)cc(F)cc(Cl)c1 CC(C)CC(CC(=O)NCC(C)(C)CCO)NC(C1(n2cnnn2)CC1)=O c1(CC(N)=O)cccc(C(=O)NCc2c[nH]nc2C2CCC2)c1 c1(C(N(C2CC(NC(=O)CCC3CCOCC3)C2)C)=O)coc2ccc(O)cc12 N1(C(CC2CCC(=O)NC2=O)=O)CCC(C2CN(C(c3cc(Cl)c[nH]3)=O)C2)CC1 C1(CCNC(C2C(C)CCC2)=O)CCN(C(=O)COCCCN(C)C)CC1 c1(C(=O)NC2(C)CC(C(=O)NCC3(C)CCOCC3)C2)ccc([N+](=O)[O-])o1 c1(CNC(C2(OC)C(OC)CN(S(CCC)(=O)=O)C2)=O)cnc2ccsc2c1 c1(OC)cc(O)c(C(N2CCN(C(=O)C(C)C3CC3)CC(O)C2)=O)cc1Br C1(CCNC(c2ccc(CNC(=O)CC3CCCC3O)o2)=O)CC(=O)NC1=O C(N=c1cccc(S(=O)(=O)N2CCSC3CCCCC23)[nH]1)c1nc(C)c(Br)cc1 C12(C(N3CC4C(NC(CSc5n(C)ccn5)=O)(C4)C3)=O)CCC(F)(CC1)C2 N1(CC(=O)N(CCCNC(C2(CC#C)CCCO2)=O)C)Cc2ccccc2C1=O C1(CNC(Cc2nc(C)[nH]n2)=O)CC(C)(C)CN1C(=O)Cc1cnns1 N1(C(C(CC(C)C)C)=O)CC2(CCN(C(=O)C(O)CC3CCCCC3)C2)C1 C1(C(N(c2c(C)nsc2)C)=O)CCN(C(C2C3CCC(F)(F)C23)=O)C(C)(C)C1 C=CCCCC(C(=O)N1CCNC(=O)C1C)NC(=O)Cc1cc(C2CC2)no1 C1(NC(C(=O)NCC)=O)CN(C(=O)COCCc2ncc[nH]2)CC1C C(CCN(C)C)(C(=O)NC1CCNC(=O)C1)NC(C1(OC)CCCC1)=O C1(C(=O)NCC(C)C(N2CCC23CCC3)=O)CCC(=O)C(C)C1 c1(C(=O)NCC2C(NC(C(C)(CC3CCC3)OC)=O)C2)ccc(Br)cc1C#N CCC(CC(=O)N1CCN(C(=O)C(C(C)(F)F)c2ccccc2)CC1)C(C)(C)C Cc1ccc(C(C)C)c(C(=O)NCC(O)CCNC(c2c(C)[nH][nH]c2=N)=O)c1 N1(CC(=O)NC(CC2CN(C(C3(C)CCC(C)C3)=O)C2)C)CCCCCCC1=O N1(C(Cc2nc(C)[nH]n2)=O)CC2CN(C(c3nnn(C(C)(C)C)n3)=O)CC2C1 O(NC(=O)C(Cc1ccco1)NC(c1cnn(C)c(=O)c1)=O)CC=C c1(C(=O)NCC2N(C(CCC(=O)OCC)=O)CC(O)C2O)nnn2c1COCC2 N1(CC(N2CCC(NC(c3cn(CC)nc3)=O)CC2C)=O)C(=O)NC(C)(C)C1=O c1(C(=O)NC)[nH]c(=NCC2(CNC(c3cccc(C(=O)NC)c3)=O)CCC2)sc1C c1(CC)nc(C(=O)NC(C)(CNC(=O)CN(C(=O)C(C)C)C)CO)co1 c1(OCC)ccc(CNC(c2sccc2C)c2nnnn2C(C)(C)C)cc1OC CCC(C)C(CC(=O)NCC1CC(C(=O)OC)C1)NC(=O)Cc1cccnc1C c1(COC)cnc(N(C(C)CCc2cc(C)on2)C)nc1 c1(OC)ccc2cc(C(N3CCCC(NC(=O)CSC)C3)=O)[nH]c2c1 c1(C(=O)Nc2cc(C(=O)O)ccc2N2CCCCC2)cnc2ccncc2c1 c1(NC(c2cn3c(n2)SCC3)c2n(C)nnn2)cnc2[nH]cnc2c1 C1(CNC(C=C(C)Cl)=O)CC2CCC(C1)N2C(c1c(F)ccc(F)c1N)=O N1(C(=O)CCc2ncc[nH]2)CCC(C2(O)CCN(C(=O)C3=CCCS3)C2)CC1 C(=O)(C1=NOC(C)C1)NCC(C)CNC(=O)CN(C)S(N)(=O)=O CC.C1(=O)N(C)CCOCCNC(=O)O1.CC C1(C(N(C2(C(=O)NC3CCN(C(C)=O)C3)CCC2)C)=O)CCCN(C(C)C)C1 C1(C(N(C(C(=O)OCC)C)C)=O)CCCCC1CNC(=O)CNC(C)=O c1(C(C(=O)NCCC(=C)CNC(c2cc(SC)n(C)n2)=O)F)ccc(F)cc1 C1(C(=O)NCC2C(NC(c3n(C(C)C)ncc3)=O)C2)CCN(CCN(C)C)CC1 c1(C(=O)NCCNC(c2cccc(OC)c2OC)=O)cnc2snc(C)c2c1 N1(C(c2c(C)[nH]nc2C(F)(F)F)=O)CCOCC(NC(=O)C(C)CC2CC2)C1 CN1C2CCC1CN(C(=O)CCCCNC(=O)C(F)C1CCCC1)C2 C1(NC(=O)NC(C)Cc2ccc[nH]2)CCCC(C)(C)C1 C=CCCCC(COC(C)C)NC(=O)C(C)(C)C1CCOC1 c1(NCC(=O)NCCC(CCNC(C(C)C2CC2)=O)C)ccc(F)cc1F O=C(CSC(F)(F)F)C(=O)N=c1nc(-c2cccc(F)c2)[nH]s1 c1(C(=O)OCC)ccc(Br)cc1CSc1ccc(OCC#N)cc1 n1(CC)ncc([N+](=O)[O-])c1C(=O)NC(CN)CC(C)C C1(C)(C(N2C(C)CC2CO)=O)CCCN(C(=O)CN2CCNC(=O)C2)C1 N1(C(c2c(C)cc(C#N)cc2)=O)CCC2(CCCC2CNC(C2CC2C)=O)CC1 C1(CNC(C2(C)CCCC2)=O)CCCN(C(=O)C(O)CF)C1 c1(CO)ccc2c(c1)OCO2.C(C(O)C(=O)C(CNCc1ccccc1)=O)N(C)C N1(C(CCc2nnc(C)n2C)=O)CCC(O)(CNC(=O)C(C)C2(O)CCC2)CC1 N1(C(C2(C)CCCS2)=O)CC2CCCN(C(c3cn(CCC4CC4)nn3)=O)C2C1 CP(C)(=O)CN1CC(C(N2CC3CC(NC(=O)C=CC=C(Cl)Cl)C2C3)=O)C1 C1(N(C)C(c2nc(Br)c[nH]2)=O)CN(C(=O)CC2CCCC2)CC1(C)C CCC(C)(CC)C(=O)NC1CCCN(C(c2ccc(C(F)(F)F)cc2O)=O)C1 C#CC1CC2(CC(C(N3CCC(NC(C45CC(C)(CO4)C5)=O)C3)=O)C2)C1 C(=O)(C(C)C(=O)N1CC(O)(CNC(c2ccc(OC(F)(F)F)s2)=O)C1)OC C12(C(N3CC(OCC(=O)NC(C)CN4CCCC4=O)C3)=O)CC1CNC2=O c1(OCC(=O)N(c2nnc(C(=O)OC)s2)C(CC)C)ccc(C)cc1C C1(C(N2CCC2CNC(C2COC(=O)N2)=O)=O)(COCC)CCCCC1 C(c1cn(C(c2cccc(SC)c2)C)nn1)=CC(=O)OCC CC1(C)CC(CNC(c2cnco2)=O)CN1C(c1nc(=N)cc[nH]1)=O C1(CC)CN(C(=O)OC(C)(C)C)CCC1NC(=O)N(C)CCN1CC2CCC1C2 C1(CNC(C(C)OCC2CC2)=O)CCCCN1C(=O)CN(c1ccncc1)C C(CCC(N)=O)(C(=O)NC(CNC(c1cccnc1)=O)C1CCC1)N(C)C c1(OCC(=O)N(C2CC2NC(c2ccc(CO)o2)=O)C)cccc(F)c1F C#CC1CCN(C(C2OCCC2CNC(C2CC2c2ccco2)=O)=O)CC1 c1(C(N(CCOC)CCNC(=O)C(C)(O)C2CCOC2)=O)cncc2ccsc12 CCCC(CCC)C(=O)NC1CC(NC(c2cc(C3(C)COC3)no2)=O)CC1O c1(C(N2C(CNC(CCN(C)CC)=O)CC(F)C2)=O)cc(O)cc(O)n1 N1(Cc2ccc(CCN3CCOCC3)cc2)CCC(C2CCCC2)CC1 C(CCOC)(C(=O)NCCC(C)(C)COC)NC(C(CC)NC(C)=O)=O N1(C(C=Cc2n(C)ccc2)=O)CCN(C(=O)Cn2ccccc2=O)CC1C1CC1 c1(OCC)cccc(-c2nc(-c3ccncc3C)n(C3CCOCC3)n2)c1 C1(C(=O)NC(CC=C)CNC(=O)COCCF)CCC2(CCOCC2)O1 Cc1cnc(C)c(C(=O)NCc2ccc(C(N3C(C(C)C)CCC3C)=O)cc2)n1 c1(CNC(CSC(C)(C)C)=O)ccc(CNC(C2(F)CCOC2)=O)cc1 n1(CCC)cc(CNC2CCC(C(=O)N(C)CCOC)C2)cn1 C#Cc1cn(C)nc1C(=O)NC(C)C(C)NC(=O)CCc1cnn[nH]1 c1(C(N(C(CNC(C2C(C)(C)C2(C)C)=O)C2CC2)C)=O)cc(P(C)(C)=O)cs1 c1(C(=O)NCCCN(C(C(CC)O)=O)CCO)c(C)nc2ccnn2c1C c1(OCCC)ccnc(N2CCC(C)(CNC(=O)CC3CC4CC4C3)C2)n1 CC(C)CC(C(=O)N1CCC(c2cnn[nH]2)C1)C(N)=O.C12CCCCC1CC(=O)N2 C(CNC(=O)Cn1cc(C)cn1)(C(C)C(C)C)NC(C1(CC)CC1)=O C1(N(CCCN(C(=O)COc2ccsn2)CC)C(=O)CO)CC2CCCC(C1)C2 c1(C(N(C(C(=O)NCC(C)(C)CF)C2CC2)C)=O)cc2n(n1)CCC2 C1(C#N)(CCOC)CC(c2nnnn2CC2CC2)(NCCc2ncccc2Br)C1 N1(C(=O)CC2CCC2)CCC2CCCN(C(=O)CCn3cc([N+](=O)[O-])cn3)C2C1 C1(NC(c2cc(CC)on2)=O)CC2(CCN(C(C3C(C)CC3C)=O)CC2)C1 C(=O)(CCCC(C)O)N1CCC(N(C(=O)C(C2CCOCC2)F)CC#C)CC1 N1(C(c2cnn(CC(F)(F)F)c2C)C(=O)NCC=C)CCCc2c(C)cccc21 N1(C(Cc2c(C)non2)=O)CCCN(C(C2CCOC(C(C)C)C2)=O)CCC1 Cc1ccc(Br)c(-n2cc(C(N3CC(C4(NC(=O)C(C)O)CC4)C3)=O)nn2)c1 N(C(=NCCc1cn[nH]c1)NC(c1ccccc1F)C)CCSC c1(CN2CC3CCN(C(c4cc5c(s4)CSC5)=O)C3C2)c[nH]c2cc(F)ccc12 c1(OC)ccc(S(N)(=O)=O)cc1S(=O)(=O)NCC(O)C1CC1 N1(C(c2nc(OCC)sn2)=O)CCn2ncc(CNC(=O)C(C)CN(C)C)c2C1 C(C)(C)(CCC(=O)NCCCC(C)(C)NC(C1CC1CC(C)(C)C)=O)N(C)C CCC(C)C(O)C(=O)N1CCN(C)C(CNC(c2nccs2)=O)C1 CN1CCC(CCNC(C23CC(NC(=O)CCc4ncccn4)(C2)C3)=O)C1 c1(CCC)onc(C)c1C(N1CCN(C(c2cccnc2N)=O)CC1)=O N1(C(c2c(C)nn(C)c2)C(=O)NCC2CC2)CCN(C)C(c2nc(C3CC3)no2)C1 C1(C(=O)NCC2N(C(CCc3n(C)ccn3)=O)CC(O)C2)CC12CC(F)(F)C2 CCC(CNC(=O)CSC1CC1)(CC)C(=O)N1CCC(F)(CO)CC1 N1(C(C(c2ccccc2)CC)=O)CC2CCC(C1)N2C(c1cc(C)oc1C)=O c1(C(N2CC(C)(C)C(NC(=O)CCCCCF)C2)=O)csc(=NC2CC2)[nH]1 Cc1cc2[nH]c(C(N3CCN(C(C4CC4F)=O)C(c4ccccc4)C3)=O)cc2s1 CCC(CC)CCCC(=O)N1CCC=CC1C(=O)NCC1CCC(C)(C)O1 C12(C(=O)NC3CC(C#N)C3)CC1CN(C(c1cccc(=O)o1)=O)C2 c1(C(N2CC(COC)(NC(c3ccc(SC)cc3)=O)C2)=O)ccnc(C)c1O CC1OC2(C(=O)NCCNC(c3cc(C4CCCC4)n(C)n3)=O)CCC1C2 c1(CC)nnc2c(C(=O)NC3CCCN(C(c4cc(C)co4)=O)C3)cccn12 C1(C(C(=O)NC(C)CCNC(=O)C=CI)C)CCC(C)(C)CC1 C12(C(=O)NCC3C4CN(C(C5CN(S(CC)(=O)=O)C5)=O)CC43)CCC(O)(CC1)CC2 C1(NCc2cccc(C(=O)OC)c2)CC(NC2CCC(F)(F)CC2)C12CCC2 CCC(C(=O)OC)N(C(=O)CC1CCCC1NC(=O)CSCCC(C)C)C CC1=CCC(C)(C(=O)NCC2CN(C(=O)CC3(O)CCOCC3)CC2(F)F)CC1 C1(C(=O)NCC2CCC2)(CC)CCCN1C(=O)CC1CC1C1CC1 c1(C(N(C2CCN(C(C3CCC(C)S3)=O)CC2)C)=O)cccc2cc(Cl)ccc12 C(=O)(CC(C)C(F)F)NC1CC(NC(C2(NC(C)=O)CCCCC2)=O)C1 C1(CCC(=O)N(CC(C)O)CC(F)F)CCN(C(C2(N(C)C)CC2)=O)C1 N1(C(C2C(CCC)C2)=O)CCC(NC(c2cc(C3CC3)nc(O)c2)=O)CC(O)C1 N(C1CN(C(c2cc(C)c(F)c(C)c2)=O)CCc2ccccc21)C(CCOC)=O C1(C(=O)N(C2CC(Oc3ccccc3)C2)CC=CC(=O)NCCO)CCCCCC1 Cc1cccc(Br)c1C(C(N1CCSCCC1C)=O)NC(=O)CC1CCOCC1 N1(C(CSCCOC)=O)CC(C(=O)NCC2(C(F)(F)F)CC2)CC12CCC2 CC1=CC(C(F)(F)F)(C(=O)NCC2(C(C)(C)NC(N)=O)CC2(F)F)C=C1I C1(c2onc(CC)n2)CCCCN1CCC1CC1(Cl)Cl Cc1ccc2snc(C(=O)NCCC3CCCCN3C(=O)C(F)CC3CC3)c2c1 c1(C(N2C(C)C3CC2(CO)C3)C(=O)NCCCOC)cc(Cl)ccc1Cl N1(C(C(C(C)C)NC(C)=O)=O)CC(C)CN(C(c2csc3cncn23)=O)CC1C C1(CNC(Cn2cccc(C)c2=O)=O)CCCCN(C(=O)C(O)C2CC2)CC1 N1(C(CCc2c(C)nn(C)c2)=O)CC2(CCN(C(C3CCCC3O)=O)CC2)C1 Cc1cc(C(N2CC(NC(c3cc(N)cc(F)c3)=O)C(C)C2)=O)nc(C)c1 N1(C2CCN(CCOn3c(C(=O)O)cnc3O)C2)CCN(CCCCF)CC1 c1(C(N2CC(CC=C)(NC(C3CCCS3)=O)C2)=O)ccc2c(n1)CCCN2 CC1CC(NC(=O)CC(C)(C)O)CCN1C(=O)CN(C)C.c12nncn1CCS2 c1(OC)ccc(Cl)c(C(=O)NCC(C)(C)CNC(C2(C)CCCS2)=O)c1N C1(C(=O)NC2CC(C(C)NC(C3(N(C)C)CCC3)=O)C2)CCC2(CCC2)C1 N1(C(C(N2CCOCC2)C)=O)CCC(C(=O)NC2CCN(C3CC3)C2)C1C c1(CC(C(=O)N(C2CC3CNC2C3)Cc2ccco2)O)cccc(Cl)c1 C1(C(=O)NCCC2CCC(NC(=O)CC(C)CF)C2)(COC)CCOCC1 c1(C(=O)NCC2(CNC(C3=C(C)CC3)=O)CC2)cc(N(C)C)nc(Cl)c1 C#Cc1ccc(F)cc1C(=O)NC(C)CN(C)C(C1CCC1C(C)(C)C)=O CCC(C)(CNC(=O)C(O)CC1CCCC1)C(=O)NCCc1cccnc1C c1(OC)nccc(CO)c1-c1n[nH]c(CNc2ncc(Cl)nc2Cl)n1 C(=O)(CCCS(N)(=O)=O)NCCCCC(C)NC(C1CCCOC1C)=O c1(C(=O)NCC(CNC(C2C(C)C2)=O)C)c(F)cc(Br)cc1F Cc1ncc(C)c(NC(C)(C)CCNC(=O)CC2CC3(CC3)C2)n1 C1(NC(C2CC(C)(C)CN2C(=O)C=C(C2CC2)C2CC2)=O)CC2CC1C(O)C2O N1(C(C2(CC(C)C)CC2)=O)CC2=C(C1)CN(C(=O)C(C)n1ccnc1)C2 C1(CC(N2CC(CNC(c3cc(F)c[nH]3)=O)OCC2)=O)COC2(CCC2)CO1 c1(OC)ccc(C(C)NC(C2COCCN2C(c2ncccc2O)=O)=O)cc1 c1(C(=O)NCCNC(c2cc(-c3ccc(C)o3)[nH]n2)=O)c(OC(F)F)cccc1Cl N1(Cc2ccc(C)[nH]2)Cc2ccccc2C1C(=O)N1CCNC(C)C1 C1(O)(CNC(C(C)(C)CO)=O)CCCN(C(C2CCCN2C2CC2)=O)CC1 C1(C(=O)NC(C)CNC(=O)CC(C)N(C)C)(COC)C=CCC1.C1(=O)CN1 c1(SCCc2ccc(C)s2)cccc(C(N(CCC(=O)NCC=C)CC=C)=O)c1 C(=O)(C(C)=Cn1ccnn1)N1CC(CCNC(c2c(CCC)nco2)=O)C1 c1(C(N2CCS(=O)(=O)C(C)C2)C(=O)NCC)cnc2cc(C)nn2c1 N1(C(c2c(C)c(F)ccc2)=O)CC2CCC1CC2NC(C1(CC2CC2)CC1)=O c1(CC)ccc(C=CC(=O)NCC2C3CN(C(C4(C)CC4(Cl)Cl)=O)CC23)o1 N1(C(C=C(CC)CC)=O)CCC2(CC1)CN(C(C1CC(n3cnnc3)C1)=O)C2.C1CC1 c1(NC(C(N(C(C(CC)C)=O)C)C2CC2)=O)ccc(F)nc1 c1(C(N(C)CCN(C)C(C2(C#N)CCCO2)=O)=O)cnc2onc(C3CC3)c2c1 c1(C(N(C2CCN(C(c3sncc3C)=O)C2)CCC)=O)c[nH]c2cccc(F)c12 c1(C(=O)NC2CCCN(C(C3CCN(CCC)CC3)=O)C2)c(Cl)sc2nnsc12 n1(CCC)cc(C(=O)N(C)CC2(CNC(=O)Cc3cn(C)nn3)CC2)nn1 N1(C(c2cccc(OC)n2)=O)CC(C)(C)CC1C(=O)NC1CC(C)(O)C1 N1(C(CCc2[nH]c(=N)sc2)=O)CCCN(C(C2CCc3cncn3C2)=O)CCC1 c1(CC(=O)NCC(C)NC(C2(CF)COC2)=O)ccc(Cl)cc1F N1(CC2CCC(C(=O)O)CC2)CCCc2c(Br)cccc2C1 N1(C(CNC(CC)=O)=O)Cc2ccccc2C(NC(c2c(C)noc2C)=O)C1 N1(CCc2cccc(OCC#C)c2)CCC(CC)OC(C)C1 C(=O)(C(O)C(C)(C)C)NC(C(=O)N(CC(C)CN(C(=O)CC(C)(C)C)CC)C)C C(CO)(C(=O)N1CCC(OC2(C(=O)NCCC)CCC2)C1)NC(C)=O.C(CF)O c1(NC2CN(C(C=CS(CC)(=O)=O)=O)CC2C)ncnc2c1nnn2C c1(N2CCC(O)(C(C)NC(C(CC)N(C)C)=O)C2)nc2ccc(O)cc2s1 C1(C(=O)NCC(C)(C)NC(COCc2nnc(C)s2)=O)C(C)(C)C1(F)F C12(C(N3CCC(COC)(CNC(=O)CCC4CCC4)C3)=O)CCCCN1CCC2 C#Cc1ccc(C(=O)NC2(CC)CCCN(C(C3CC34CC(O)C4)=O)C2)cc1 C(=O)(C(CC(C)C)CC(C)C)c1ncc2c(N)n(ncn1)NCC(CC)NC2=O C(=O)(C(O)CCc1cnc[nH]1)NCc1cn(CCNC(CN(C(C(C)C)=O)C)=O)nn1 C(C(=O)NCC1CN(C(=O)CCC2CC2)C1)(C(C)C)OC(c1ccncc1)C c1(C(C)C)cc(C(=O)NCC2CCN2C(=O)COC2CC2)c(C(C)C)o1 C#Cc1c[nH]nc1C(=O)NC1CC(CNC(C2CC(c3cccc(F)c3)C2)=O)C1 Cc1ccc(C(=O)NCC2CC(C)CCN2C(=O)C=CCF)cc1S(C)(=O)=O C#CCC(C(N)=O)NC(C1CCCCN1C(=O)CCNC(=O)COC(C)C)=O CC1CC(CNC(=O)C(F)=CC2CC2)CN1C(c1ccnc(N2CCC2)c1)=O C(=O)(C1CCC(c2ccccc2)O1)NCCCNC(C1(C(=O)OC(C)(C)C)CC1)=O N1(C(C(COC)C)=O)CCC(F)(F)C(CNC(c2ccnnc2)=O)C1 C1(C(=O)NC2CC(C)(NC(=O)Cc3ccc(Cl)cc3F)C2)Cc2ccccc2N1 C(CC(=O)Nc1cc(CC)cc(C)c1)(C(F)F)NC(C1(C(=O)OCC)CC1)=O c1(NCc2nn(C)nc2Br)[nH]c(=NCCC(C)(C)S(C)(=O)=O)nc2sccc12 c1(C(=O)NC(CCCNC(C(C)OCCOCC)=O)C)ccc(C)cc1C C1(NC(c2ccc(CCC(N)=O)cc2)=O)CCN(C(C2CC=CCC2)=O)CC1F C1(C(N(CC(CNC(C(C(=C)C)(C)C)=O)O)C)=O)CC2(C1)CS(=O)(=O)C2 C1(CC)CCN(C(=O)C(CCF)NC(=O)CCCC2CC2)CCO1 Cc1cc(C23C(CCN(C=O)CC2)C3)nc2c1c(=O)n(C)c(=O)n2C C1(C#N)(C(=O)NC(CCOC)CNC(c2cc(C(N)=O)no2)=O)CCCC1 C1(CCC)(NC(=O)COCCF)CCCN(C(=O)C(C)N(C)C)C1 c1(C(=O)NC2CCN(C(C(C)N(C(C)=O)C)=O)C2)cc(S(C)(=O)=O)ccc1F N1CCC(C)N(CC2CSCCS2)CC1.C#Cc1cnc(-c2ccccc2)nc1 C(CC(=C)C)(C(=O)NCC1C(C)C1C)NC(CC=C)=O c1(CC(N2CC(CNC(c3c(CC)noc3)=O)C(C)C2)=O)ccc2c(c1)CCC2 CN1CCC(C(=O)NCCC2(C(=O)NCCN3CC=CCC3)CC2)C1=O Cc1cc(Cl)ccc1CC(=O)NC1CCCN(C(=O)CN2CC(=O)NC2=O)CC1 CC(C(=O)NCC1CN(C(=O)C(c2ccc(F)c(Cl)c2)(C)C)C1)C(F)(F)C(F)F c1(C(N(CCCNC(c2cnc(OC)nc2)=O)C2CC2)=O)c[nH]c2cc(C)ccc12 N1(C(C(CC2CC2)NC(C2CCCCC2)=O)=O)CC2CC1(CO)C2 C1(OC)CN(C(c2cccc(C(C)C)n2)=O)CC1NC(c1n[nH]cc1Cl)=O c1(NC(C2CCN(c3cccc(F)c3)C2=O)=O)cc(OCCCO)ccn1 c1(C(N2CC(CN(C(C=CCC)=O)C)OCC2)=O)ccnc(Cl)c1F Nc1cc([N+](=O)[O-])ccc1C(N1CCCN(C(c2c[nH]cc(F)c2=O)=O)CC1)=O N1(C(C2(C)CCC(=O)C2)=O)CC2(C1)CN(C(=O)Cn1cc(Br)cn1)C2 c1(C(=O)NC2CN(C(C3(OC)CC3)=O)CC2c2nccn2C)ccc(O)nc1Cl c1(C(C(c2cc(C)n(C3CCOC3)c2C)=O)C#N)ccc2c(c1)CCN2C C1(C(N(CC(=O)OC(C)C)C)=O)CCN(C(C2C3(CC3)C23CC3)=O)C1C(C)C c1(C(N2CC3C(CN(C(C(C)=C(C)C)=O)C)C3C2)=O)nn(C)c(C)c1Cl c1(CC)cncc(C(=O)NC2CCCCC2CNC(c2coc(C(N)=O)c2)=O)c1 C1(CC)C(=O)NCCN1C(c1cc(CNC(C2COC(=O)N2)=O)on1)=O c1(CC(=O)NCC2CCC(c3nn[nH]n3)C2)cccc([N+](=O)[O-])c1 N1(C(CCCOC)=O)CCCC(C2CCN(C(c3cccn4cnnc34)=O)C2)C1 C(CCCCC(=O)NC(C(N1Cc2ncsc2C1)=O)c1ccoc1)=CC N1(CCNC(C2(C#N)CC2)=O)CCC(NC(=O)CCCc2nccs2)CC1 c1(CC)c(C(=O)NCCCCN(C(=O)C(CO)NC(N)=O)C)nnn1C C1(CC)CN(C(=O)CSC)CCN1C(C1CCN1CC)=O N1(C(C2C(C)(C)CO2)=O)C(CNC(c2cncs2)=O)CC2CC12 Cc1nc2sccn2c1C(N1CCC(CNC(C2CC3(CC3)CO2)=O)C1)=O C1(n2cc(C(C)NC(C)C(c3ccc(C)cc3)O)nn2)CCCC1(C)O c1(NC(c2n(CCSC)nnn2)c2snnc2C)ccc2c(c1)OCC2 n1(CC(=O)NC(CNC(C(CCC)C)=O)C(C)C)ccc(C)cc1=O Cc1nc(=N)[nH]c(C)c1C(=O)NC1CC1.C12CN(CCO1)C(=O)CC(=O)NC2 c1(C(=O)NC2CCN(C(=O)Cc3ccc(F)cn3)C23CC3)cnc2[nH]ccc2n1 c1(CC)[nH]c(=N)sc1C(N1CC(NC(=O)CC2CCC2C)C(O)C1)=O N1(C(CCOCC)=O)CCC2C(NC(c3ccc(CN4CCCC4)[nH]3)=O)C2CC1 c1(CCC(=O)OC(c2ccc(F)cc2F)C)cccc(S(N)(=O)=O)c1 C1(C(=O)N(CCCn2cc(C3(F)CCCO3)nn2)C2CC2)CCCC2(CCC2)C1 C1(NCc2coc(SC)c2C)C=CC2CC1CO2 C1(OCC)CC2(C1)CC2C(=O)NCC(C)NC(c1cnc[nH]1)=O CC(CN(C(=O)Cn1ccc(CO)n1)C)C(=O)NCC1OCCC1C c1(NC(=O)C(N2C(C(=O)N(C)C(C)C)CCC(C)C2)=O)cc(Br)c(F)cc1N Cn1ncc(CNc2cc(N3CCC(NCCO)CC3)ncn2)c1Cl c1(N2CCCC(CNC(c3ccc(F)cc3Cl)=O)C2)cc2ncnn2cn1 CCC(C(=O)NC(CCCOC)C(=O)N1CCCC(C)(C)C1)C(C)(C)CC Cc1c(C(N2CC(NC(c3cnsn3)=O)CCC2C)=O)oc2c(F)cccc12 N1(CCC)CC(c2nc(-c3ccc(N)cn3)nn2CCN(C)C)CC1=O N1(C(c2c(C)nn[nH]2)=O)CCCCC(NC(C2(C(F)(F)F)CC=CCO2)=O)C1 N1(C(=O)NC)CCC(C(=O)NCC(F)CNC(C2(COC)CC=CC2)=O)C1 c1(CC)cnc(O)c(C(=O)NC(C)CCNC(c2[nH]nc(OC)c2Cl)=O)c1 C1(CC=C)(C(=O)NCCCc2ccc(C)s2)CN(C(=O)CC2CCCC2C)C1 c1(CN2CC(c3nc(COC)no3)CC2N(C)C)nc(C)c(CC)[nH]1 N(C(=NCC(C)N1CCCC1)NC1CCOCC1)CC1(S(CC)(=O)=O)CC1 C(=O)(C1=CCSC1)NC(C(C)NC(=O)CSC1(F)CC1c1ccccc1)CO c1(CC2(F)CN(C(c3n(C)ncc3CO)=O)C2)cc(F)ccc1F C1(C(=O)NC2CC3C2CCN3C(=O)C2CC2)Cc2cc(Br)ccc2O1 C(=O)(CC(C)(C)C(F)(F)F)NCC(C1N(C(CCNC(=O)OC)=O)CCCC1)(C)C C1(C(=O)Nc2c(OC)cccc2O)CCCN1NC(=O)CC1CCC(=O)N1 N(C1CC2(CCCC2)Oc2ccccc21)C(=O)C1=CCOCC1 c1(COC)cccnc1C(N1CCC(C)(NC(c2cocc2C(N)=O)=O)C1)=O c1(C(=O)NC2(OC(C)C(N3CC(CO)CC3(C)C)=O)COC2)cc(Cl)nnc1O Cc1ncc(Cl)c(C(=O)NC2(C)CC(NC(c3cn(C)c(=O)cn3)=O)C2)n1 C#CC1(C(=O)NCCCCC(=O)N2CCCC(CC)C2)CCCC1 N1(C(c2c(CCC)[nH]cc2)=O)C2CCC1CN(C(=O)CCCc1cccs1)C2 C12(C(N3CC4CC(NC(c5cc(COC)on5)=O)C3C4)=O)CC1COC21CCC1 N1(C(CCNC(COC)=O)=O)CC2CC(NC(C3CCC=CO3)=O)CC1C2 c1(C(=O)NCCN(CCOC)CC2CC=CC2)c(C)nn(-c2cccs2)c1O N1(C(=O)CCn2ccnc2)CC2CC1CN2C(C1(CO)CC1(F)F)=O c1(C(C(=O)NC(C)CN(C)C(C2CC2(F)F)=O)(C)C)c(F)cccc1F Cc1cc(C(=O)NCCC2(O)CN(C(c3cncn(C)c3=O)=O)C2)ccc1Cl C1(NC(c2ccc(CC)s2)=O)C2CCN(C(c3cc(O)ncn3)=O)CCC12 N1(C(C(C)Oc2ccccc2Cl)=O)Cc2n[nH]cc2CC1C(=O)O C=C(CNC(=O)C(=O)NCC(F)F)CCNC(=O)C(C)(C)c1sccc1Cl c1(N2CCC(C(N3CC(Cn4cnnn4)C3)=O)C2)cc(F)cc(F)c1 CCCCC(CC(=O)NC1CCOCC1OCC)NC(C1CCC1C(C)(C)C)=O c1(OC)nccc(N(C)C(=O)NC(c2ccc(C3CCCN3)cc2)C2CC2)n1 C12(C(=O)NCCCNC(c3cc(C)nnc3O)=O)CCC(CF)(CC1)CC2 C=C1CCC(C(N2CC3CC2(CNC(c2cc(Br)sc2C)=O)C3)=O)CC1 C=C(Cl)C(C)(C)C(=O)NC1CCCCC1NC(C1CC1Br)=O c1(OC)ccc(-c2csc(NC(=O)NC(C3CCOC3)CSC)n2)cc1 C1(c2cn(C(C(C)NC(=O)CC3CCC3)C)nn2)C(C)(C)C1(C)C CCCCC(C)CCC(=O)NCC1(C(N2CCC(CC)C2)=O)CC1 C=CC1(C(N2CCC(NC(=O)Cc3ccc(F)c(F)c3)C(C)C2)=O)CCCCC1 CC(=O)CCC(=O)N1CCC1CNC(c1ccc(COC)s1)=O c1(C(N(CC(CO)(CO)NC(C(C(C)C)F)=O)C)=O)cc(F)c(F)c(C#N)c1F c1(C(=O)NCCC2N(C(CCC=C)=O)CCOC2)cc(F)cc(F)c1F C(S(=O)(=O)CCNC(=O)CCC1(O)CCOC1)c1cn(C(C)C)nn1 n1(CCC)cc(C(=O)NCC=CCNC(C2CCS(=O)(=O)N2)=O)c(C)n1 C(C(C)(C)C(=O)NC1CC1c1cnn(C)c1)NC(C(CC1CCC1)OC)=O c1(C(=O)NCCC2(NC(c3cn(C(F)F)cn3)=O)CC2)ccc2c[nH]nc2n1 N1(C(c2c(COC)nc(C)nc2)=O)CCOC2(C1)CN(C(C1C3COCC13)=O)C2 Cc1ccc(C(=O)N(C2CCN(C(C3CCO3)=O)CC2)C(C2CC2F)=O)cc1 Cc1cc(C(=O)NC2CC(CNC(c3cc(O)cc(Br)c3)=O)C2)ccc1F CCCN=C(NCc1cccnc1C(F)(F)F)N1CC2C(C)C2C1 N1(C(CCC2C(C)C2)=O)CC(NC(=O)CC2CCC2)C(C2CC2)C1.c1ccncn1 CCC(C(=O)N1CCC(CCNC(c2sccc2Cl)=O)C1)c1cccnc1 c1(N2CC(CSC)CC(OC)C2)nc2c(c(=NCCC3CCCOC3)[nH]1)CSC2 c1(C(=O)NCCN(C(=O)NCCCOC)C2CC2)cnc(OC)c(Cl)c1 N1(C(C(COC)OC)=O)CCC(C)CC1.C1(C(N(CC(C)C)C)=O)CCCCN1C c1(C(=O)NCC=CCC(=O)NC(C(CC)C)CO)ccc2nccn2c1 c1(C(=O)NC(C2CN(C(=O)C(O)CN3CCCC3)C2)C)ccc(O)c(F)c1 N1(C(c2ccc(-c3nc(CC)on3)cc2)C)CCN(C(=O)CC)C(CC#N)C1 c1(CCC(c2nnnn2CCOCC)NCCCC)ccc(F)cc1 N1(C(CCC2CC(C)C2)=O)CCC(O)C1CNC(=O)CCC1CCOCC1 N12CC3(CCN(C3)CC1=O)C2.C(C1=CCCCCC1)(c1nnnn1C)N(C)C C1(C)(NC(C2(C)CCCN(C(c3ncc(C)nc3)=O)C2)=O)CC(C)(C)OC1=O C(=O)(C(F)C(C)CNC(=O)CN1CCCCC1)N(CCC(C)C)C1CC1 c1(OCC(=O)NC2CCC2NC(=O)Cc2cccc(C3CC3)c2)ccc(Cl)nc1 c1(C(N(C)CC2(O)CN(C(CC3N(CC)CCC3)=O)C2)=O)n[nH]c(C)c1C(C)=O CC1CN(C(c2cnc(-c3ccc(Cl)s3)s2)=O)CCC1NC(c1cnc(O)o1)=O N1(C(c2cc(C)sn2)=O)CCC2CCC(NC(=O)CCS(=O)(=O)N(C)C)C12 c1(C(N(CCCNC(CS(CC)(=O)=O)=O)C)=O)ccc2cccc(OC)c2n1 C1(NC(C2C(C)=CCS2)=O)CCC2(CCCN(C(=O)CCCCC#N)C2)C1 C1(CC)CN(C(C2(n3cncn3)CC2)=O)CCC1NC(c1cc(Cl)ccc1Br)=O C(CC(=O)NOCC(=O)NC)=CCC.C1C(O)CC(=O)N1 N1(CC(=O)NCC(C2CC2)NC(c2cnco2)=O)CCOC1=O C(=O)(C1=C(Cl)CCC1)NCc1ccc(C(=O)NCC(=O)OCC=C)s1 N1(C(c2cnc(C(=O)OCC)s2)=O)CCC2CSCC2C1 C(c1cc(Cl)ccc1Cl)=CC(N1CC2(CN(C(c3c(C)onc3CO)=O)C2)C1)=O N=c1cc[nH]c(C(N2CCC2CC(N2CCC(OCCF)C2)=O)=O)n1.C1(O)CC1 c1(C(N(CC(C)C(=O)NC2CN(C)CC2C)C)=O)ccc(C#N)cn1 C1(NC(C(c2ccc(C)o2)C)=O)CN(C(c2ccncc2Br)=O)CCC1F C=CC(C)CC(=O)NCC1CC(CNC(c2ccco2)=O)C1.c12ccncc1N2 Cc1nc(N2CCCC(C(C)NC(c3cc(Cl)sc3Cl)=O)C2)c(F)c(C)n1 C1(NCCC(C(C)C)OC)CCCN2CCSCC12 C1(CN(C)C(c2ncccc2F)=O)CN(C(C2(CO)CCOCC2)=O)CC12CC2 c1(C(N(CCNC(C(C)OCCOC)=O)C)=O)cnc(CO)nc1O.C1(C)CC1 C#CCC(O)C(=O)NC(CNC(=O)COCC1CCCC1)CC(C)C c1(CNC(C2(C(C)C)COC2)=O)cc(C(=O)N(CCCO)C)no1 N1(C(C2C(C)(C)CCCO2)=O)CCCC2CN(C(C3CCCS3(=O)=O)=O)CC12 C(=O)(C(C(=O)NC1(CNC(C23CC(F)C2C3)=O)CCCC1)C(C)C)OCC c1(OC)cc(C(C(=O)NC2CCC2)N(C)C(C2CCOC2)C)c(F)cc1Cl C1(C(NOCCCC#C)=O)(NC(=O)C(C2CC2)OCC)CCC(C)(C)C1 N1(C(C2C(C=C)CC2)=O)CC2CC(NC(c3cc(OC)cc(Br)c3)=O)C1C2 c1(NC(C2CCCC2NC(C2(Br)CC2)=O)=O)cc(Cl)c(F)cc1F c1(C(N(C(C)CNC(=O)C(F)OC(F)(F)F)C)=O)ccc(C#N)nc1O C=CCC(C)N=c1nc2c(cnn2C)c(N(CC)CC2CCCS2(=O)=O)[nH]1 c1(CC)cc(C(N2CC3C(NC(=O)CC4CCC4)C3C2)=O)oc1CC c1(CNC(C2CCN(c3ccc(C)cc3)C2=O)=O)n[nH]c2c1CCCCC2 C1(C)(NC(c2c(C)ncs2)=O)CCC(NC(=O)COCC(C)(C)C)CC1 C(=O)(CCCC(=O)N(C)C)N1CCC(N(C(c2ccc(F)s2)=O)CC)C1 C1(NC(Cn2ccc(C)n2)=O)CCC2(CC1)CN(C(=O)Cc1cc[nH]c(=N)c1)C2 C1(COC)(NC(C2CC2(F)Cl)=O)CCN(C(c2cc(CO)n(CCO)n2)=O)CC1 C12CCN(C1)C(=O)N(C(C)C)C2=O.CCC(C)(C)c1nn[nH]n1.C(C)(C)(C)OC=O c1(CC)nc(C(N2CCCC(CN(C(=O)C(C)OC3CCOC3)C)C2)=O)c(C)o1 C1(C(=O)NC(CCCCC)C2CC2)CC(C)(C)CCN1C(=O)Cn1c(C)ccc1C Cc1ccc(-c2ccc(C(=O)NC(C)C(CO)NC(=O)CC3COC(=O)N3)s2)o1 c1(C(=O)NCCCN(C(c2c(OCC)ccs2)=O)CCO)c[nH]c(=N)cc1C N1(C(C(CC)OCC)=O)CCCCCC1CNC(=O)Cc1ccc(O)nc1 CC(C)(C)CCCC(=O)NCCOCCNC(=O)CC1CCC(O)C1 c1(CC2CCN(CC(=O)N(c3ccc(F)cc3)CCCC)C2)ccc(O)c(C)c1 N1(C(C2C(NC(C3C(C(=O)OC)C=C3)=O)CC2)=O)CC(C)C(F)(F)C1 C1(CC)(NC(=O)C(N)=O)CCCN(C(=O)C(n2nc(C)cc2C)C)C1 c1(NC(C2OCCN(C(C3C(=O)CCC3)=O)C2)=O)nc2c(s1)COCC2 N1(C(c2cnc(CC)[nH]2)=O)CC2CCCC1(CNC(=O)COC1CC=CC1)C2 c1(C(=O)NC2C(C)CN(C(=O)C=CBr)C2)ccc2c(O)nc(S)nc2c1 N1(C(c2ccccc2CC)C(=O)NCCCC)C2CCC1C(C)C(CO)C2 c1(CC(=O)NC2CN(C(CCS(C)=O)=O)C2)coc2ccc3ccccc3c12 N1(C(Cc2cc(C)no2)=O)CCC(C)(CCNC(C2CCCC2F)=O)CC1 c1(OC)cc(OC)cc(NC(=O)CC2CCCN2C(c2ncccc2Cl)=O)c1 c1(C(N2CCCC(CCNC(C(C)P(C)(C)=O)=O)C2)=O)ccc2c(n1)COCC2 CC(C)C(C)C(C)CC(=O)N1CC=CC(NC(=O)C2=CCCCC2)C1 Cc1nc2c(s1)CCCC2C(=O)NCC12CC(NC(=O)C(C)C3CC3)(C1)C2 n1(C(=O)NCCC2CCN(C(=O)COC3CCCCC3)CC2)cnccc1=O C(=O)(C1=COCCO1)NC(C1CCCN(C(C(c2c(OC)cccc2)=O)=O)C1)C C1(C)(C(=O)NC(c2ccccc2)C(=O)OC)CCN(c2cc(O)nc(O)n2)CC1 C1(c2cn(CC(=O)N(CC(F)(F)F)CC)nn2)COC(C)(C)OC1 N1(C(C(C)=O)=O)CCC(NC(c2cc(C3CCOCC3)n[nH]2)=O)C(CO)CC1 c1(C(=O)NCCC2CCCC2)n[nH]c2c1CN(Cc1cc(F)c(F)c(Cl)c1)C2 N1(C(c2cnc(N(C)C)o2)=O)CCC(O)C(N(C)C(C2CCS2(=O)=O)=O)C1 c1(C(=O)NC(CC(C)NC(C=CC)=O)C)cc(OC)c(Cl)cc1Cl C1(NC(CC(C=C)CC)=O)CC1C1CCCN(c2cc(C(C)C)nc(SC)n2)C1 c1(OC)cccc(C(CNC(=O)Cc2sc(S)nc2C)NC(=O)CCC(F)F)c1 CC1(NC(C23CSCC2C3)=O)CC(NC(=O)CCc2nccs2)C1 c1(C(N2CC(C)(NC(c3n[nH]c(C)c3F)=O)C2)=O)nccn2ccnc12 N1(C(CC(CC)SC)=O)CC2(C)CN(c3cc(C(C)=O)ncn3)CC2(C)C1 C1(C(=O)NCC2(C)CC=CCC2)CCN(C(c2cc[n+]([O-])cc2)=O)CCO1 c1(NC2CCS(=O)C2)nccc(=NCCCc2cccc(O)n2)[nH]1 C1(C(C)CN(C(=O)C(=O)NC2CCC(F)(F)C2)C)CCC(F)(F)CC1 CC1=C(C(=O)N2CCC(C)(CNC(=O)C(C)C3CCC3)C2)CCO1 C(C(C(=O)NCC(=O)Nc1cncc(F)c1)C(C)(C)C)OC1(C)CCC1 C1(NC(c2nccnc2Cl)=O)CC2CC(C1)N(C(C1CC=CCO1)=O)C2 c1(CNC(c2occ(C)c2)=O)ccc2c(c1)CN(C(=O)CSc1ccncc1)C2 c1(C(=O)NCC(C)NC(c2cn(CC3CCCO3)nn2)=O)cn(C)c(=O)nc1O C(=O)(C1CCCc2ncnn21)NCC(C)NC(C(C(=O)OCC)C(C)C)=O C1(NC(c2c(C)nsc2N)=O)CCCCN(C(c2cc3sccc3[nH]2)=O)C1 C(CCc1cn(-c2cccnc2)nn1)(C(=O)O)NC(c1c(C(C)(C)C)c[nH]c1)=O c1(C(=O)NC23CCC(C2)N(C(=O)C=CC2CCCCC2)C3)ccc2n[nH]cc2n1 C(=O)(N=c1[nH]c(Br)cnc1Cl)C1N(Cc2n(C)nc(O)c2)CCSC1 C1(C(N2CCC(C)(CNC(c3cccc(OCC)c3)=O)C2)=O)CCC(=O)N(C)C1 CC1(C(=O)NCC(c2ccccc2)NC(=O)C=C2CC2)CCC(=O)NC1 Cc1nn(C)c(Cl)c1CNC1CC1C(=O)Nc1ccc(Br)cc1F C(=O)(C1=CS(=O)(=O)CCC1)N1CCC(C)(CNC(CC(CC)SC)=O)CC1 N1(CCC)CCOCC(C)(O)C1.c1(C2C(=O)NC3CC(C3)N2C)ccnn1C c1(C(=O)NC(CNC(C(C)N=[N+]=[N-])=O)(C)C)cnn2c1OCCC2 N1(C(CCSCCCC)=O)CC(NC(C2(O)CCSCC2)=O)C(C)(C)C1 C1(CCC(=O)NC(C)CCNC(C2CNC(=O)C2)=O)CCN(C)CC1 C(C(CCC(=O)O)C(=O)NCC(F)F)NC1=NCC(C)(CC)N1 C(=O)(C(F)C(C)CNC(c1ccc(C)c(F)c1)=O)N1C(C=C)CCC1 CC1(C)CCN(C(=O)C=CCF)CC1CNC(C1OCCO1)=O N1(C(c2nn(CC)nc2Br)=O)CCCCC2(CCN(C(C3(OC)CC3)=O)C2)C1 C1(C(N(C(C(=O)OC)C)C)=O)CC(O)C(O)CC1CNC(=O)C(C)(C)C(C)O C(=O)(CCCCC(C)(C)C)N(C(C)C(=O)NCCCC(C)(C)C)C C1(C)(N(C(C)C2CC2)CC2CCCO2)CCCN(c2cc(N3CCCC3)ncn2)C1 c1(CN(C(C)CC(=O)O)c2nnnn2C2CCCCC2)cccc2cccnc12 C1(CC(NOC(CC)CC)=O)C2CCCC2N1C(=O)CC1CCCN1C Cn1nc(CC(N2CC(O)(CNC(C3(C)CCCO3)=O)C2)=O)cc1C(F)(F)F C1(N(C)C(C2CCCCC2)=O)CC2CCC(C1)N2C(=O)Cc1ccno1 C=CCC(C)(C)C(=O)N1CCN(CC(N2CCC(C(=O)NC)C2)=O)CC1 c1(CCC)ccc(CC(=O)NCC(CNC(=O)Cc2ccc(F)cc2)CO)cc1 c1(C(=O)NC2(C)CCCN(C(c3c(CC)oc(C)c3)=O)C2)cnc2[nH]ccc2n1 c1(C(N2CC(C(=O)NC3CC(CC(=O)OC)C3)C(C)C2)=O)c(C)cc(C)nc1S C(=O)(C(C)CCC(C)(C)C)N1CCC(C)C(Nc2cc([N+](=O)[O-])ccc2N)C1 Cc1csc(C=CC(=O)NC2CC(NC(=O)CCCN3C(=O)CCC3=O)C2)n1 c1(C(N2CCC(C)(NC(=O)CC3C=CCC3)C2)=O)cc(F)c(O)c(Br)c1 N1(C(c2c(CC)sc(=N)[nH]2)=O)CCC(F)C(NC(c2ccn(C)c2)=O)C1 N#CC1C2CCC1CN(Cc1ccc(F)cc1C(=O)O)C2 C(=O)(C1=NNC(=O)CC1)N1CCC(CN(C(=O)CCOC2COC2)CC)CC1 C1(NC(CC2(CSC)CC2)=O)CCCC1CNC(=O)C(c1ccc(C)o1)C Cc1cc(C(N2C(C(N3CC=CCC3)=O)CC2C)=O)on1 N1(C(CC2CCCC(C)(C)C2)=O)CCCC2(C1)CN(C(C1CC13CC3)=O)C2 c1(C(=O)NC2C(NC(C(c3ccccc3)C)=O)COC2)nc(=N)cc[nH]1 N1(C(CCCCC)=O)CCOC2(CCN(C(C3CN(CP(C)(C)=O)C3)=O)C2)C1 c1(C(N2CCN(C(C(CCSC)O)=O)CC2C(F)F)=O)ncc(C#N)cc1Cl C(=O)(CC(C)COC(c1c[nH]nc1-c1ccccc1Cl)=O)NC C1(NC(CC=CCNC(C(CCC)NC(N)=O)=O)=O)CC2(CCCCC2)C1 C1(CN(C(c2cc(C(F)F)ns2)=O)CC)CCCN1C(c1cnc(N(C)C)o1)=O N1(C(C(C)N(C(C)=O)C)=O)CCC2CCCC12C(N1CCC(F)(CO)C1)=O n1(CC(N2CCCC(CN(C)C(C3CCC(=O)N3)=O)C2)=O)cc(F)ccc1=O CC(C)S(=O)(=O)N1CCN(C(c2ccc(Br)cc2)C(=O)NCCC#N)CC1 C1(O)(CN(C)C)CCN(C(C2C3CN(C(=O)CN4CCC(=O)CC4)CC23)=O)C1 C1(NC(=O)NCC(c2c(OC)cccc2)O)CCc2cccc(Br)c2C1 Nc1nc2c(cc1C(=O)N(C1CC1)Cc1cn(C3CCN(C(N)=O)C3)nn1)CCC2 C1(OCCC)CCN(C(c2cc(-c3c(SC)cns3)c[nH]2)=O)C1 C(C#Cc1cccc(Cl)c1)N1CCC(C)(NC(c2ncc3ccccn23)=O)CC1 C(=O)(CCC(F)F)NCC(CCOC)NC(=O)C(F)(F)c1cncs1 C(CCC(CO)SC)NC(C1CC(NC(c2c(CC)c[nH]n2)=O)C1)=O C1(C(N2CCCC(NC(C(=O)NC(C)C)=O)C2C)=O)CC2(C1)CC(C)(C)C2 c1(C(=O)NC(C)C(C)NC(C23CC(C)(C2)C3)=O)cccc2ccsc12 N1(C(Cc2cccc(OC)n2)=O)CCC2(CC1)CC2CNC(c1cc(C)ns1)=O C(=O)(C1=NOC2COCC12)N1CC(N(C)C(c2cnc(OC)cn2)=O)C2(C1)CC2 n1(C(Cc2ccccc2)C2C(C)C2)cnc2c(C(O)C(C)C)ncnc12 N1(CCN(C(=O)C(F)OC(F)(F)F)C)CCN(C(c2ccc(CO)cn2)=O)CC1 C1(CCC(N2CC(CNC(CCN(CCCCC)C(C)C)=O)C2)=O)CCCCO1 Cc1ccc(C(F)(F)F)cc1C(=O)NCCN(C(C1SCCC1C)=O)C1CC1 N1(C(c2cnc(C(F)F)s2)=O)CC2CC1CCN2C(C1CCCCS1(=O)=O)=O C1(CNC(C2CC(CC)C2)=O)(OC)CN(C(=O)CN2CCOC2=O)C1 CC(C)C(CNC(=O)Cc1nccn1C)C(=O)NC(c1ccc(F)cc1)CO C1(CC=C)(C(=O)NC(CC2CC2)CO)CN(C(=O)CC2CCCOC2)C1 N1(C(C2C(CC)C2)=O)CCC(CNC(=O)CNc2cccc(Cl)c2)C12CC2 CC(C)C(O)C(F)(F)C(=O)NC1CN(C(c2ccc3c(c2)CCN3)=O)CC1(C)C c1(C(N2C(CNC(c3ccc(OCOC)cc3)=O)CCC2)=O)cc2n(n1)CCC2 c1(C(N2C(C(=O)NCCCn3ccnc3)CCC2)=O)cc([N+](=O)[O-])c(Cl)cc1F Cc1ccc(C(CNC(=O)C(O)C2CCCC2)NC(c2cnc(C)[nH]2)=O)cc1 C(=O)(C(C(=O)OC1CCC(C(C)(C)C)CC1)OC)OCC C(=O)(C1=NOC(C)(C)C1)NC(C1CCCCC1)C(=O)N(C)CCC1CCCN1C N1(CCn2cc(C(CNCc3scc(COC)c3)C)nn2)CCCCS1(=O)=O c1(C(=O)NCC2N(C(C(c3ccccc3)C)=O)CC2)ccc(C(N)=O)cn1 C(=O)(C(CC)C(=O)NC(CO)C(C)NC(c1cc(F)ccc1C(C)C)=O)OCC c1(N2CC(C)OC(C(N)=O)C2)ccc(S(=O)(=O)N2CCS(=O)C(C)C2)cc1Cl C1(C(C)NC(c2csc(CO)n2)=O)CCCCN1C(=O)C=Cc1ccccn1 C(=O)(C1Cc2ccc(C)cc21)NCC(CC)(C)NC(=O)C=Cc1ccsc1 CN1CCC(C)(C(=O)NC2CCCCN(C(c3scnc3C(C)(C)C)=O)C2)C1=O c1(OC)cc(C(=O)NC2CC3CN(C(c4c(Cl)n[nH]c4C)=O)CC23)ccc1C#N CCCCC(CNC(=O)C(O)C(F)F)NC(=O)C(F)(F)c1csc(Cl)c1 c1(C(=O)NCCC2(O)CN(C(CC3C(CC)C3)=O)C2)cc(C)ccc1S(N)(=O)=O n1(CC=C)cc(C(=O)NC2CCN(C(=O)Cc3cscn3)C2)cn1 O=S1(=O)c2ccc(c(Cl)c2)NC2N1CC2.c1(C(CNSC(F)F)O)ccco1 c1(CCC)noc(CCCC(=O)NCCC(O)CNC(C2CCSC2)=O)n1 N1(C(CCC2CCN(C(c3cccc(C#C)c3)=O)CC2)=O)CC(C2=NOCC2)C1 c1(C(=O)NCC(C(C)C)(C)NC(C2CC(C3CC3)=NO2)=O)ccnc2[nH]cnc12 c1(C(=O)N(CC(=O)O)CC2CC2)cc2c(nn1)CCCC2 N1(C(=O)CCC2CCC2)CCN(C(=O)COc2ccc(Cl)c(Cl)c2)CC(CO)C1 N1(CC(=O)NC2C(O)CCN(C(C3=CCN(C)C3)=O)C2)Cc2ccccc2C1 C1(NC(C2CCN(C(c3c(CC)cno3)=O)C2)=O)CCCCC1(F)F N1(C(C2(CC)CC2)=O)CCC2CCN(C(=O)CC3CCC(=O)N3)C2C1 C1(NC(C(C)n2ccnc2)=O)CCN(C(=O)CCc2cccs2)C1C(C)(C)C C(=O)(C1=NNC(CC)C1)N(CCC(=O)N(C1CCOCC1)C)CC#C C1(C(=O)NCC=CCNC(CNC(C)=O)=O)CCc2nnc(O)n2C1 N1(CC)C(=O)NC(c2c(F)cnn2C)C2=C1CC(C(=O)O)NC2=O CC(CS(N)(=O)=O)NC(C1(NC(c2nc[nH]n2)=O)CCCC1)=O C1(CNC(c2cc3c[nH]cnc-3n2)=O)CC12CCN(C(c1coc(Cl)n1)=O)CC2 c1(CC(=O)NCC(=C2CN(C(c3ncn(CC)c3)=O)C2)F)n[nH]c2c1CCCC2 c1(C(=O)NCCCOCCNC(C2CC2[N+](=O)[O-])=O)cc2n(n1)CCCN2 C#CC1(C(=O)N(CCC(C)(C)O)C)CN(C(=O)CC2CC3C=CC2C3)C1 n1(CCOC2C(OC)COC2)c(C)cc(C(C2CC3(CC3)C2c2ccccc2)=O)c1C N1(C(c2ccc(SC)o2)=O)CC2(CCN(C(C3CCC(C)C3)=O)CC2)C1 N#Cc1cnc(N2CCCCC2CNC(=O)COCc2ccnc(O)c2)c(F)c1 C1(CCNC(C(CC#C)O)=O)CN(C(=O)COC2CCCC2)CC(C)O1 c1(CC)c[nH]c(C(=O)N(C)CC2CCCN2C(=O)C=C2CCN(C)C2)c1 S(=O)(=O)(CC(=O)NC(CCN(C(=O)CC1CCCC12CC2)C)C(C)C)NC CC1CC2CCC(C(=O)NCCC3CSCCN3C(=O)Cc3cc[nH]c3)CN2C1 c12nc(C)c(s1)CC(=O)NC2.C1(NC(C2CCCN2CC)=O)(COC)CCCC1 C12(NC(C(=O)NCC(F)F)=O)CCCC1N(c1nnc(O)s1)CC2 N1(C(COCC(=C)C)=O)CCC(CC(N)=O)(NC(c2nsc(OC)n2)=O)CC1 C1(O)(C(=O)NCC(=O)OCC)CCCN(C(c2cc(C3CC3)nc(O)c2)=O)C1 C1(C(CO)NC(COCCC)=O)CCN(C(c2cc(OC)cs2)=O)CC1 c1(NC(C(CN(C(c2c(C)cc[nH]2)=O)C)C)=O)cc(Cl)ccc1C#N C1(NC(c2ccnc(F)c2)=O)CC12CCN(C(c1cnc(OCF)cn1)=O)CC2 C1(C(N2CC(NC(C3(COC)C=CCC3)=O)C2)=O)Cc2cc(F)ccc2O1 C=CC(C)(O)CC(=O)N1CCN(C(=O)CNS(=O)(=O)CCCC)C(CC(F)F)C1 C1(C(N(C(CC)CNC(C2CC3CCC2CC3)=O)C)=O)CCn2ccnc2C1 C=C(Cl)CC(C(=O)N1CCCC(C(C)C)C1)NC(c1sccc1NC)=O C1(NC(c2c(C)cccn2)=O)COC2(CCN(Cc3ccc(I)cc3Cl)CC2)C1 C=CCCC(C(=O)NCc1cc(C)n(C)n1)NC(=O)Cn1cc(Cl)cn1 CC1CCC(O)CN1C(C1CC(NC(=O)CC2CCC(O)C2)C1)=O Cc1cc(N)c(C)nc1C(=O)NC1CCC(C)N(C(C2CC(C)(O)C2)=O)C1 N1(C(c2c(C)cc(C(=O)OC)o2)=O)CC2=C(C1)CN(C(=O)C=Cc1ccco1)C2 N1(C(c2cccc(C(C)C)c2)=O)CC2CCC(NC(=O)CC3(C4CC4)CC3)(C2)C1 c1(C(N(C2CCN(C(=O)Cc3cnnn3C)C2)C)=O)cnc(O)n(C)c1=O CC1CCn2cc(C(N3CCC(O)(C(C)NC(=O)Cc4ccno4)C3)=O)nc2C1 CC1CCc2nc(C(=O)NCCOC(C34CC5CC(C)(C3)CC(C)(C5)C4)=O)cn2C1 Cc1ccc2nc(C(N3C4CCC3CC(NC(C3CC3(Cl)Cl)=O)C4)=O)ccc2c1 C(CCC(C)NC(c1coc(-c2ccccn2)n1)=O)NC(C(C)n1cncn1)=O C1(COC)(CNC(c2[nH]nnc2C)=O)CCN(C(c2[nH]ncc2C#N)=O)CC1 c1(C(=O)NC2CN(C(c3cccc(C(C)C)c3)=O)C(C)C2)cc(N)ccc1O c1(OC)ccc(Cl)c(OC)c1C(=O)NCCC(C)(C)NC(=O)Cc1csc(C)n1 C(=O)(C1Cc2ccccc21)N1C(C)(CNC(c2c(C)cc(N)cn2)=O)CCC1 c1(C(=O)NCCN(C(c2c(C(=O)OC)ccnc2)=O)C)noc2c1CCCC2 CC(C)(C(=O)NC1CC(C(C)(C)O)C1)NC(=O)CC1COCCO1 c1(C(N(C2CCCN(C(=O)CCCCF)C2)C)=O)cccc(CF)c1 C(CC(C(C)(C)C)NC1CSCCN1C(=O)OC(C)(C)C)N(C)C C1(NC(CC=CC)=O)CCCC2CN(C(=O)CCCOc3ccccc3Cl)CC12 N1(C(CCN(CC)CC)=O)CC(NC(=O)Cn2cc(C(C)O)nn2)CC(F)C1 O=C(C1=CCCCC1)NCCCCNC(=O)C(c1c(F)cccc1F)(F)F O=C(CCC1CCCN(C(c2ccc(-c3ncc[nH]3)cc2)=O)C1)N=c1nc[nH]s1 c1(N(C2CC3CNC2C3)C(CNC(N)=O)=O)ccnc(CO)c1 C1(F)(C(N2CCC(OCC(=O)NCC(C)(O)C3CC3)C2)=O)CCCCCC1 C(=O)(CCC(C)(C)c1ccccc1)NCC(CNC(C(CC)CC)=O)(C)C C1(C(N2CCC(NC(c3c(O)nc(CC)c(C)c3)=O)C2)=O)Cc2cccc(F)c2O1 C(=O)(CCCCC(F)(F)F)N1CCOCC(CNC(CCC(CC)C)=O)C1 CC1C(NC(=O)Cc2c(Cl)cccc2Cl)CCCN1C(c1cc[nH]c1)=O Cc1sc(Br)nc1C(N1CCC(NC(=O)Cc2nnc(O)s2)CC1)=O C1(CNC(CCCCCC)=O)CC2(CO1)CN(C(=O)CNC(N)=O)C2 N1(C(c2cc(C(=O)OC)c(F)cc2)=O)CC(C)N(C(C)=O)CC1C N1(C(Cc2ccc(C)c(Cl)c2)=O)CC2C(C1)C(F)(F)C2(F)F C1(CNC(CCCc2nc(C)sc2)=O)CN(C)CCN1C(c1cn(C)cc1C)=O Cc1csc(C(=O)NCC(C)NC(C2CC23CCCC3)=O)c1Br C1(C(=O)NCC2(C)COCCO2)(CC)CCN(C(C2CCCO2)=O)C1 c1(C(N2CCC(C)(CNC(=O)C=Cc3ccccn3)C2)=O)cc2n(n1)CCCO2 C1(CC(=O)NC(C(=O)OC)CC2CCC3(CCC3)CO2)CC(C)(C)CC(C)(C)C1 c1(C(N(CC(C)CNC(C2CC3CCC2O3)=O)C)=O)csc2cc(Cl)cnc12 c1(C(N(C(CCNC(c2cnc(C(C)C)[nH]2)=O)C)C)=O)ccc2cccnc2c1 CC1CN(C(C2(F)CN(Cc3ncc(Cl)nc3Cl)C2)=O)CCC1O c1(N2CC(NCc3c(C)noc3C)C(F)CC2)ncc2[nH]ncc2n1 Nc1ccc(C(=O)NCC2(NC(c3ccc(-c4ccccn4)s3)=O)CC2)nc1F C1(C(N(C)CC2CCN(C(CNC(=O)OC)=O)C2)=O)C2CCC1CC2 C(=O)(C1CC=Cc2ccccc21)N1CCCC(OCCOC)C1 C1(CC)CCCC(C(N2CCC(c3cncn3C)C2)C(=O)NCCCSC)C1 CC(CCC(C)(C)C)C(=O)NC1(C)CCN(C(c2cnn(-c3cccnc3)c2)=O)C1 N1(C(C(C)C2CCC2)=O)CC2(CNC(=O)C=Cc3ccsc3)CC1CO2 N1(C(Cn2c(C)nnn2)=O)CCOC(C(C)NC(C2(C)CC(F)C2)=O)C1 c1(C(C)(C)C)ccc(O)c(CNCC2(C(F)F)CC2)c1 C1(NC(CCC#C)=O)CC(C)N(C(=O)CCc2cccc(OC(F)F)c2)C1 c1(CCC(=O)NCC(C)NC(=O)C(F)F)cc(Cl)no1 Cc1cnc(C(N2CC(C)CCC2C(=O)NCC2CCOCC2(C)C)=O)c[n+]1[O-] N1(C(C(c2cscn2)N(C)C)=O)CC(C(=O)OC(C)(C)C)C2(CC2)C1.C1(=O)CCN1 N1(C(Cc2c(C)ocn2)=O)CCCC(CN(C)C(C2COC(=O)N2)=O)C1 O=C(CC1OCCc2sccc21)NC1CCCN(C(=O)CN2CCCCC2)CC1 CC1=C(C(=O)NCC2CC(C(=O)NC(C)(C)C(O)CO)=NO2)SCCO1 CCC(C)(C)C(O)C(=O)N1CC(C(=O)N(C2CCOC2)C)CCC1(C)C CC(C(=O)N1CCC(CF)(NC(=O)CC2CN(C)C2)C1)S(N)(=O)=O N1(Cc2nc(-c3n(C)c([N+](=O)[O-])cc3)on2)CCCc2cccnc21 N1(C(C(c2cn(CC)nc2)=O)=O)CC2CCN(C(c3cn(C)nc3SC)=O)CC12 CCCCC(C(=O)NC(C)C)ON=C(C)C.c1(C(N2CCC2)=O)cc(CF)on1 c1(C(=O)NCC(CCNC(C(C)C(C)(F)F)=O)O)cccc2nonc12 CC(CN(C(=O)C(F)F)C)C(=O)NCC1(O)CC(O)C1 N1(C(=O)C2=CCN(C(=O)C(F)n3ccnc3)C2)Cc2cccc(F)c2C1 Cc1cc(C)n2cnc(C(=O)NCC(C)CNC(=O)C=C3CCC(C)C3)c2n1 CC1CN(C(=O)C=Cc2cc[nH]n2)CC(C)CN1C(=O)CN1CCCNS1(=O)=O C(c1ccsc1Br)=CC(=O)NC(C)CCNC(=O)CCc1cnco1 Cc1n[nH]c(C)c1CC(C)C(=O)NC1CC1CNC(c1cc(Br)cn1C)=O C1(NC(C(CC=C)CC)=O)COC2(C1)CN(C(c1cnc(N(C)C)cn1)=O)C2 C1(C)(C(=O)NCC2CN(C(c3c(SC)snn3)=O)CC2(C)C)CCCNS1(=O)=O c1(C(=O)NC(CNC(CCCNC(=O)NCC#C)=O)C)ccc2nc(O)[nH]c2c1 C(N=c1cc(C)[nH]c(=NCc2nc(=N)[nH][nH]2)[nH]1)c1ccc(COC)s1 N1(C(c2c(CC)cccn2)=O)CCC(C)C(NC(=O)C=C(C)C(F)F)C1 N1(C(CSCC)=O)CCC(NC(C2(O)CCOCC2)=O)C(F)C1 c1(CNC(C2C(C(=O)NC(c3ccccc3)CC)C2)=O)ccnc(Br)c1 C1(n2cc(-c3cnc(C)o3)nn2)CN(C(=O)C(=O)Nc2c(C)noc2C)CC1C c1(C(=O)OC)cnc(NCC2CCCCN2C(c2csc(C)c2C)=O)c(Cl)c1 CN1N=CC(CC(=O)NCc2cccc(NC(=O)C(F)=CC3CC3)c2)C1=O C=C(C)CCCC(=O)N1CCC(C(=O)NCCN=S(C)(C)=O)CC1CC c1(C(=O)NCC2C(NC(=O)C=CCO)C2)cccc2c1CCC(=O)N2 n1(CCOC)cc(C(=O)NCC(C)(C)NC(C23CC(F)(C2)C3)=O)nn1 CC1CN(C(=O)CCOc2ccc(Br)cc2)CC1NC(=O)C(O)C1CC1 Cc1nn(C)cc1C(N1CCC(NC(=O)C(C)NC(=O)C(C)(C)C)C1C)=O C1(C)(C(=O)NCC(C2CC2)NC(C(CCC(C)C)O)=O)C2CC3CC(C2)CC1C3 C1(C(N(CC(C)NC(c2c(C)nccn2)=O)C)=O)CC2CC1C1C2C1(F)F c1(C(N2CC(OCC)C(CNC(C3CCCC3(F)F)=O)C2)=O)ccc(F)c(Cl)c1 c1(CN(CC(=O)Nc2ccc(OC)cc2)C)ccc(F)c(Br)c1 c1(C(=O)NC2C(CNC(C3(CC)CCOC3)=O)CCC2)cc(O)nc(Cl)c1 Cc1cc2cc(-c3c[nH]nc3C(F)(F)F)ccc2nc1NC(c1ccsn1)=O Cc1noc(C)c1CC(N1CCOC(CNS(=O)(=O)CC2CC2)C1)=O c1(C(N2CC(CC)N(C(=O)C(C)n3ccnc3)CC2)=O)cccc2nn(C)cc12 N1(C(c2ccc(C(C)=O)[nH]2)=O)CC(C)(CNC(=O)C(O)CC(F)F)CC1(C)C N1(CC)C(=O)CCC1C(=O)NCC(CCOC)NC(=O)CCC1CC1 c1(C(N2C(C)CC(NC(C3C(C(=O)NCC#C)C3)=O)C2)=O)cnc2sccc2c1 C1(C(=O)NC(CCOC)C(=O)NC(c2nnnn2C)C)CC(C(C)C)=NO1 C1(CN(C(c2cccc(C)c2)C)Cc2ccc(C)o2)N(C)CCCC1(C)C C(=O)(CCCC(=O)N1CCN(Oc2ccc(CN(CC3CC3)CC)cc2)CC1)OC Cc1ccc(Cl)c(F)c1C(=O)NC1CCN(C(C2SCCCS2)=O)CC1C C(=O)(C1=CCCCC1C)N1CC(C(=O)NCc2cc(OC)ns2)C(C)(C)C1 C(=O)(C(C)(C)C(=O)NC1CCCN(C(C2CCN(C)S2(=O)=O)=O)C1)N(C)C N1(C(c2sc(=O)n(C)c2Cl)C(=O)NC)CCC(C2(O)CCC2)CC1 c1(NC(C2CC(C(=O)NC3C4CN(C(CC)=O)CC43)C2)=O)ncc([N+](=O)[O-])n1C N1(C(CNC(=O)OCC=C)=O)CCOCC1CN(C)C(c1cccnc1C)=O N1(C(C(CC)CCOC)=O)CC2(CCN(C(=O)CNC(c3ccoc3C)=O)C2)C1 S(=O)(=O)(c1cccc(F)c1)NC1C2(CCCC2)CNC1.C1(COCC)CCOC1 CC(CN=c1cc(C(F)(F)F)nc[nH]1)NC(C1(CCN(C)C)CC1)=O C1(NC(CSCc2nc(C)sc2)=O)CN(C(=O)C(c2ccccc2)F)CC1O C1(NC(=O)Cc2n[nH]cc2Br)CC2(C1)CC2NC(c1ccns1)=O C=CC(CC(=O)N1CCC(CN(C(C23CC(CO2)C3)=O)CC)C1)c1ccccc1 c1(C(C)C)ccc(NC(c2cn(CCNC(=O)C(N)=O)nn2)=O)cn1 Cc1nc(O)ccc1C(=O)NC(C)(CNC(C1CC(C#N)C1)=O)C(C)C c1(CCCC(N2CCC(NC(CCC(CC)C)=O)CC2)=O)nc2ccccc2o1 c1(N(CCNC(c2n(CC)ncn2)=O)CCOC)ccc([N+](=O)[O-])c(C)n1 C1(C(=O)O)CCCC(c2ccccc2)N1C(=O)Cn1cc(Cl)ccc1=O N1(C(C(F)OC)=O)CCCC(C2(NC(=O)CCn3cc(Cl)cn3)CC2)C1 C(=O)(C1=CCC2(COC2)OC1)NCC1CN(C(C=Cc2ccc(C)o2)=O)CC1O C(CC(=O)NC1CCN(C(C2CC(C)(O)C2)=O)C12CC2)(C(N)=O)NC(C)=O c1(C(=O)OC)cccnc1NC(C)CC(C)NC(C1CCC(C2CC2)O1)=O C1(C(N2CC3N(C(c4c(F)ccc(C)c4)=O)C3C2)=O)CCC2CCC(=O)N2C1 C(C(C)(C)C(=O)N1CCC(OCc2cn(-c3cncc(Br)c3)nn2)C1)SC CN1CC2CC1CN2C(C12CC(C)(CN1C(c1c[nH]c(C(N)=O)c1)=O)C2)=O N1(C(c2c(CC#N)ccs2)=O)CC(CNC(c2nsnc2O)=O)C2CC12 C1(C(=O)NCc2occ(C(N(CC(C)C)C3CC3)=O)c2)CCC(O)CC1 C1(NC(C(CO)NC(C(C)OCCC=C)=O)=O)CC2(CCCCO2)C1 CC(CF)C(=O)NCCN(CCC(N)=O)C(c1c[nH]cc1Cc1ccccc1)=O c1(N(C(N2CC(CO)CC(O)C2)=O)Cc2ccccn2)cccc2c1CCC2 n1(CC(=O)N(C2CCCCN(C(=O)C3=CCOC3)C2)C)ncn2cccc2c1=O c1(C(=O)N(NCCC(=O)NCCN2CCC2C)Cc2ccccc2)ccc(Cl)s1 C(=O)(CC(F)(F)C(C)C)N1CCN(C2CN(C(C3ON=C(C)C3)=O)C2)CC1 N#Cc1c[nH]ccc1=Nc1ccc2nc(NC3Cc4n[nH]cc4C(N)C3)ncc2c1 c1(NC(CCNC(c2nc(C(C)C)oc2)=O)=O)cccc(F)c1F CCC1=C(C(=O)NCCCN(C(=O)CCC2(C)CCC(=O)N2)C)CCCO1 c1(CC)cccc(C(=O)NC2CC(CCNC(c3ccc(O)c(N)n3)=O)C2)c1F CC1CCN(C(=O)CN2CC(C)(CCF)C2)CC1N1CCOCC1 c1(S)ccc(N)c(-n2cccc2)c1.C1(N(C)C)CCCC1C(F)F N1(C(C=CCC)=O)CCC2(CC1)CN(C(c1cc(Cl)cc(Cl)c1)=O)C2C(C)C n1(CC)nc(C(=O)NC2CCCCC2NC(=O)CCNC(=O)CO)c(Br)n1 CC(F)(F)C(C(=O)NC1CC(CCNC(c2cc(Cl)no2)=O)C1)c1ccccc1 C1(CC(=O)OCC)CCN(CCNC(N2CC(C(=O)N(C)C)C2)=O)CC1 N1(CC)CC(C(=O)NC2CCC(NC(=O)C(F)(F)C3(O)CCC3)C2)CCC1=O Cc1cnc(NCCCS(N)(=O)=O)c(S(=O)(=O)NCCCSC2CCCC2)c1 C(CCC1CCC1)(C(=O)Nc1ccc(Cl)nc1)NC(c1cncs1)=O C1(OCC)CCN(C(=NCCNc2ccc(CC#N)cc2)NCC)CC1C Cc1cc(O)ccc1CC(=O)NC1CCC(C)N(C(c2cc(C)n(C)n2)=O)C1 CC(CC(C)(F)F)C(=O)N(C)CC1(O)CN(C(=O)CCN2CCCCCC2)C1 C1(C(=O)NCCC(C)N(C(=O)CNC(C2CCOCC2)=O)C)CCCN1C=O C(CC1=CCN(C(c2ccc(O)c(O)c2)=O)CC1)NC(CC(CC)(F)F)=O C(C)(C)(CCNC(C1CC1(F)Br)=O)NC(C=CCOC)=O N1(C(CNC=O)=O)CCC(NC(=O)Cc2cnc[nH]2)C1 C1(C(=O)NCC(CNC(CCc2onc(C)n2)=O)O)OCC2COCCC12 c1(C(=O)NCCNC(C2CCN(C(c3cc(CC)on3)=O)C2)=O)ccncc1C N1(C(C2(CCOC)CCC2)=O)CCC2CCC(C1)N2C(C1CCC=CO1)=O C(=O)(CCCCCN=[N+]=[N-])N(CCN(C(C1N(C(=O)NC)CCC1)=O)C(C)C)C N1(C(C(=O)NC(CC)C)c2cc[nH]n2)CCS(=O)(=O)C(C)C1 c1(NC(C(N2CC3(CCOC3)C2)C(C2CCC2)OC)=O)ccc(F)cc1C c1(C(=O)NCC(CNC(Cc2c(C)noc2)=O)C)cnc(S)nc1 C(=O)(C(=O)C(C)(C)C)N1C(CN(C(=O)C2=NNC(C(F)(F)F)C2)C)CCC1 CCC(C)C(C(F)(F)F)NC(C1(CC)N(C(=O)OC(C)(C)C)CC1)=O Cc1cc(F)ccc1S(=O)(=O)N1CC(C)CC1c1cccc(F)c1 Cc1cc(C(=O)N(C2CC(NC(=O)CCC3CC(C)(C)CO3)C2)C)nn1C1CC1 N1(C(c2c(CCC)nco2)=O)CCC(O)(CNC(c2nnn(C(C)(C)C)n2)=O)C1 C(=O)(C(C)(F)C(F)(F)F)NCCOCCN(C)C(c1coc(C(F)(F)F)n1)=O c1(C(=O)NCC2CCN(C(C3C(C)CC4CC4C3)=O)C2)cn2cc[nH]c(=O)c2n1 C1(C(=O)NCC(CC)NC(=O)CC(C)(C)O)Cc2ccc(OC)nc2N1 C1(C2(O)CCN(CC(N)=O)CC2)(NC(COC(C)C)=O)CC1 C12(C(=O)NCCNC(c3cnc(CCC)s3)=O)CC(N=[N+]=[N-])C1C2 c1(C(=O)NCC2C(NC(Cc3cccc(C)c3)=O)CCCC2)cccc(F)c1Cl c1(C(N(c2nccc(C)c2)C)=O)cc(F)c(F)cc1Cl c1(OC)noc(C2CC2)c1C(=O)N(CCC(C)NC(C1(CF)CCOCC1)=O)C n1(CCCOC)nnnc1C(C1CC1C1CC1)NCc1ncnn1C1CC1 Cc1ccc(N)c(C(=O)NCC2CC(O)(CNC(=O)C=CC3CC3)C2)c1F Cc1nc(C(=O)CN2C(=O)CCCC2=O)ccc1-c1cccc(C(N)=O)c1 C(=O)(CC(C)C(=O)N1CC2C(CC(=O)NC(C)(C)CO)C2C1)OC C1(CNC(COCCCCC)=O)CN(C(=O)C(C)(C)COC)CCO1 N1(C(C2CC(=O)NCC2)=O)CCN(C(=O)Cn2cnccc2=O)C(CC(F)F)C1 c1(CN(C(c2ccc(Cl)cc2Br)C(=O)NC2COC2)CC)cc(Br)ccc1F C1(C)(CC(=O)NCC2ON=C(C)C2)CCN(C(C2CC(C#N)C2)=O)C1 C(CCC(C)(C)C)NC(=O)C(C)N(C=Cc1cccs1)CC CC(C(=O)N(C1CCN(C(=O)C(c2ccccc2F)(C)C)C1)C)C(C)(C)C C(=O)(C1=C(C)S(=O)(=O)CC1)NCCC(=C)CNC(c1cncc(C2CC2)n1)=O Cc1c(C(=O)NC2CC3(C2)CN(C(C2CCCOC2C)=O)C3)cncc1Cl c1(C(=O)O)noc(CN2CCCC(NC(C3CCCCO3)=O)C2)c1Br c1(C(N2CC(CCNC(=O)CC3(O)CCC3)OCC2)=O)cnc2c(c1)CNC2=O CC1(C)CCCN(C(=O)CC(C(F)F)NC(C2CC(O)C(F)C2)=O)CC1 C1(CNC(C(C)NC(N)=O)=O)CCN(C2CCN(C(=O)C=CBr)C2)CC1 CC(C(=O)NC1(CNC(=O)CCc2cc(Cl)cc(Cl)c2)CC1)C(C)C(C)(C)C c1(OC(C(=O)NN(C(C)C(=O)NC2(Cc3ccccc3)CC2)C)C)ccccc1 CCCS(=O)(=O)C(C)C(=O)N1CCC(CF)(NC(c2cn(C(C)C)nc2C)=O)C1 N1(C(C2CN(CC)C(=O)C2)=O)CCN(C(=O)Cc2cncn2C)CC1CO N1(C(=O)CC2CC(CF)C2)CCCC2(C1)CN(C(c1ncc(Cl)cc1Cl)=O)C2 C1(CCOC)(NC(=O)CSc2cccs2)CCN(C(=O)CS(=O)(=O)NC)C1 c1(C(=O)NCCCCCCN(C)C(C2CCCOCC2)=O)ccc(C#N)cn1 CCCCCC(F)C(=O)N1CCCC1CNC(=O)CCCCCOC C1(O)(CNC(CCOCCC)=O)CCCN(C(=O)Cc2ccc(C)s2)C1 c1(C(N(C2CCN(C(=O)C(F)F)C2)CC#C)=O)ccc(-n2ccnc2)cn1 c1(N2C(C(CCC)C)CCC2)nnc(Cc2ccccc2)n1CC(C)(C)OCC C(=O)(C(F)C(C)CNC(=O)CN(C(=O)C(C)C)C)NC(CCSC)C N1(C(C(COC(C)(C)C)N(C)C)=O)CCC(CNC(C2(CCF)CCC2)=O)CC1 CCC(CC(=O)NCC1(NC(C2CCC3(CCC3)CC2)=O)CC1)C(C)C CC1(C(=O)NCCC2(CNC(c3cnc(C4CC4)o3)=O)CC2)CC=CCC1 C1(NC(C2CCCC(F)C2)=O)COC2(CCN(C(=O)C(F)F)CC2)C1 N1(C(C(CCC)n2ccnc2)=O)CC(CNC(=O)Cn2nnc(C)n2)C2(CC2)C1 O(C1CCCc2ccccc21)C(C(C)NC(=O)Nc1cc(N)nc(Cl)c1)=O c1(C(N2CCN(C(C(C)SC)=O)C(CF)C2)=O)ccc2n[nH]cc2c1C CN(OC1CCCC1)C(=O)C(C)(C)CCNC(c1ccc2cccnn12)=O c1(C(=O)NC2CN(c3nc(C)c(Br)cn3)CC2F)c[nH]c2cccc(C)c12 Cc1cc(C)n(-c2ccc(CN(C(C)(C)C)CCc3cnc[nH]3)cc2)n1.C1=[SH]C1 N1(CC)CC(CC(C)(C)NC(c2ccsn2)=O)CC1=O.CC=CC c1(-c2nc(N3CCN(CCN4CCCC4)CC3)cc(O)n2)ccc2nc[nH]c2c1 C(CCCC(=O)N1CCN(C(=O)C(N)=O)CC1c1cn[nH]c1)(OC)OC c1(C(=O)NCC(CC(=O)NCCOc2ccncc2)OC)cnn(C)c(=O)c1 N1(C(C2(Cl)C(C(C)=O)C2)=O)CCC(CC2CCCC2)C(C)C1 c1(CSC(c2nc(C3CC(=O)N(C)C3=O)no2)CCC)c(Cl)cccc1Cl c1(OC)cc(Br)ccc1Cl.C1(OCCN2C(=O)C2)CN(C)C(=O)C12CC2 N1(C(CNC(CCN(C(=O)C=Cc2ccnn2C)C)=O)=O)CC(CO)C(C)(C)C1 Cc1cc(C#N)cnc1NC(=O)NCC1CC2(CC2)CO1 C1(CC(=O)NCCCCNC(C2C(CCOC)C2)=O)CCC(=O)C1C C1(C(N2CCC(N(C(C3=CCN(C)C3)=O)C)CC2)=O)CCc2nc[nH]c2C1 c1(C(N2C(CNC(CCC=C)=O)C=CC2)=O)cccc(CO)n1 CC(C)(C)C(O)C(=O)NCCC(=O)NCCOC(C1C(C(=O)NCCO)C1)=O c1(CC)ccccc1NC(C(c1ccc(OC)cc1)N(C)CCN(C)CC)=O c1(C(=O)NC2CCN(CCNC(C(CC)F)=O)CC2)ccc(C#N)cc1 C1(C(N2CCC(CC(=O)NC3CC(O)C(O)C3)C2)=O)Cc2ccccc2C1 c1(-c2cn(C(C(=O)NC3C(CC)C3)CCC(N)=O)nn2)nc2cc(F)ccc2s1 C=CC1(CC(=O)N(CC#CC)C)CN(C(=O)C=CC(=O)N(C)C)C1 c1(C(=O)NC2(CNC(C(C)c3ccon3)=O)CCCC2)ccc(F)c(Cl)c1 N1(C(c2ccn(COC)n2)=O)CCC2CCCC12C(=O)NC(CO)C1(C)CC1 c1(C(N(C2CCCC2)CCNC(C(C=CC)O)=O)=O)cnn(C)c1OC CCC(CC(=O)NCCN(CCCF)C)NC(C1(C2(C)CC2)CC1)=O C(c1ccc(Br)cc1)=CCC(N1CC(NC(C=CC=CCC)=O)C(C(F)F)C1)=O N1(C(Cc2scc(C)c2)=O)CCC(NC(C2CC2c2ccc(F)nc2)=O)CC1 C(=O)(CC(F)(F)F)N=CC(=O)NC(C)(C)CCNC(=O)COC1CCCCC1 Cc1cscc1C(N1CC(C(N)=O)(CNC(c2ocnc2C2CC2)=O)C1)=O C=C(C)CC(C(=O)N1CC(N2CC(O)C2)C1)NC(=O)CC(C)OC S(=O)(=O)(c1cccnc1NC1CN(CC2CC2)C1)NC1CC(C)SC1 c1(OCCC(=O)NCCN(C(=O)CCc2cscn2)C(C)C)ccc(F)c(F)c1 N1(C(C(CC)=CC)=O)CCC(Nc2ncnc(Cl)c2F)CC(C)(C)C1 N1(C(=O)CNc2ccsn2)CCCCC1CC(N1CC(F)(CC2CC2)C1)=O.CC C1(CC(=O)N(CCC(=O)NCCC#CCO)CCO)CCCC2CC12 C(=O)(C(C)(C)C(=O)N(C)CCN(C)C(C1CCCN(c2ccccn2)C1)=O)NC CCC(CC1CCN1C(C)=O)CCC1CCCC1 C1(CC)CN(C(=O)Cn2ccc(C)c2)CC1C(=O)NCC(C)C(=O)NC N1(C(CC(C)SC)=O)CC2(CCN(C(=O)CC3CCCS(=O)(=O)C3)C2)C1 Cc1cc(Cl)cc(C(=O)NC(C)C(C(C)C)OC(C)(C)C)c1C C(CN=c1nc(N2CCC(C#N)C2)c2c([nH]1)c(C)nn2C)c1c(C)cncc1 N#Cc1ccc(CN=c2cc(-c3ccccc3Cl)o[nH]2)c(Br)c1 C(C1=NOC2OCCCC12)C(COC(=O)Cn1cc(-c2ccccc2)sc1=O)=O C1(OC)CN(C(=O)CCCc2ncco2)CC1NC(c1cc(O)nn1C)=O Cc1ccc(C)cc1C(=O)NCC1CN(c2ncc(C(C)(C)O)cn2)CCO1 C(C(C(F)(F)F)N1CCNCC1)NC(C(=O)N(C1C(C)C1)C)=O c1(C(=O)NCCC2CCN(C(CCCNC(C)=O)=O)C2)cnc2n1CC(C)CC2 c1(C(N(CCOCCC(=O)NCC(COC)O)C)=O)ncncc1N C1(F)(CNC(C2CC3CCC2C3)=O)CCN(C(c2ccc(C3CC3)s2)=O)CC1 C1(NC(C2(OC)CCOC2)=O)CC2CCC1CN(C(c1cnc[nH]1)=O)C2 C1(C(=O)NCCn2nnc(C)n2)(COC)CN(C(=O)C2CC2)C1 C1(C(=O)NCC2(C)N(C(c3cc(C)c(C)nn3)=O)CCC2)CCOC2(CCC2)C1 CON1CC(C(=O)NCc2ccc(C(=O)N(C)C(C3CCCO3)C)s2)CC1=O C(=O)(CC1=CCN(C)CC1)N1C2C(NC(C(=Cc3ncc[nH]3)C)=O)CC(C2)C1 CN1CCC(=O)Nc2cc(C(N3CCC(O)(Cc4ccccc4)C3)=O)ccc21 c1(OC)c(C(N2CCC(CC3CC3)C2)C(=O)NCC(C)C)cccc1Br N1(C(COCCC(C)C)=O)CCC(CNC(=O)Cc2noc(C)c2C#N)C1(C)C c1(OC)ccc(CNS(=O)(=O)CC2CN(C)CC(C)O2)cc1Cl N1(C(CC2ON=C(C)C2)=O)CCC2CN(C(C3CC3C(F)F)=O)C2C1 C(=O)(CCCCCn1cc(CCCCC#N)nn1)N1C(C(N)=O)C(O)C(O)CC1 N1(C(CCN(C)CC)=O)CCCC(CO)(NC(=O)CCc2cncc(C)c2)C1 C1(NC(c2c(OC)cc(C)s2)=O)CN(C(=O)C2=C(Cl)CC2)C2(CCCCCC2)C1 c1(CC(=O)NC(C)C(C)NC(c2cc(CF)on2)=O)cccc2cccnc12 C1(CC#C)(C(=O)NC2CN(C(=O)C(C=C)=C(C)C=C)CC2F)CCCCO1 CCC(CCCC(=O)NCCN1CCC(CO)C1)NC(=O)CC1CC(C2CC2)C1 S(=O)(=O)(c1ccc2nc(N3CCCC(NC(=O)NC)C3)ccc2c1)N(CC)CC C1(NC(Cc2c(C)nc(S)s2)=O)CCN(C(C2(C3CCC3)CCC2)=O)CC(O)C1 c1(CCC(=O)NCC(C)N(C(=O)COCC(F)F)C)ccc(Br)cc1F c1(C(=O)NC2CC2C(=O)NC2CCN(CCCO)C2)cccc(OC(F)(F)F)c1 c1(CC(=O)NCCC(C)N(C(=O)CNC(N)=O)C)ncncc1Cl CC(C)C(O)C(O)C(=O)NCC=C(Cl)Cl C1(NC(C(C)=CC)=O)CC2(C1)CC1(CC(NC(c3ccn4c3CSCC4)=O)C1)C2 C1(CNC(C2CCCN(C)C2)=O)CC2CCC1N(C(=O)Cc1ccccc1O)C2 C1(CC(=O)NCC(=O)CCC2CCCC2)CC2(CC2)CO1 c1(CC)c[nH]c2ncnc(NC3CCCCC3NC(=O)CNC(=O)CC(C)C)c12 C1(C(N2C(C(C)O)COCC2)=O)CC2CN(C(C3CS(=O)C3)=O)CC2C1 c1(NC(=O)NS(CCCOC)(=O)=O)cnc2c(c1)c(O)nc(=O)n2C c1(CCC(=O)NC(C(=O)NCC2(C(N)=O)CC2)C2CCCO2)ccncn1 c1(C(=O)NC(CC)CNC(=O)Cc2ccc(C)nc2)ccc2nc(S)oc2c1 C1(NC(c2cc3c(s2)CCC3)=O)CC2CC1CN2C(=O)C(c1ccc(F)cc1)O N1(C(c2ccc(C)cn2)=O)CC2(C1)CN(C(C1CCc3n[nH]cc3C1)=O)C2 c1(-n2c(-c3ncn(C)c3C)nc(-c3nccc(OC)c3)n2)nc[nH]c2ncnc1-2 c1(C(=O)NC2C(NC(C(CC)(C)CC)=O)CCOC2)ccc2nnn(O)c2c1 C1(NC(C2(F)CN(C(=O)C3=COCC3)C2)=O)CC(CO)C(O)C1O c1(C(=O)NCC2CCCN2C(=O)C(F)(F)c2ccnn2C)noc2ccccc12 C#Cc1cnc(C(N2CCN(C(c3cn(C4CC4)cn3)=O)CC(O)C2)=O)c(C)c1 c1(C(N2CCCN(CCNC(C(C)OCC)=O)CC2)=O)cc2c(nn1)CCCC2 N1(C(C(C)(C)F)=O)CCCC2C1CCCN2C(=O)CN1C(=O)CC(C(=O)O)C1=O C1(C(N2CC(CC=C)(C(=O)NCCC3COCCOC3)C2)=O)CC(=O)C12CCC2 CN1CCCC(O)(CC(=O)NCCOC2CN(C(C3(C)CCC(=O)CC3)=O)C2)C1 N1(C(c2cc(CNC(C=CCC)=O)on2)=O)CCN(CC2CC2)CC1 C(=O)(C(C)P(C)(C)=O)NC(C(C)C)(C)CNC(c1cccc(Cl)c1N)=O C#CCC(CC(=O)NC(C)(C)C(C)(C)O)NC(=O)C(F)=CC1CC1 c1(C(c2nnnn2C2CCOCC2)NC(CC)C2CC2)nc(C)sc1C C1(NC(C(C)(C)C(F)(F)F)=O)CN(C(=O)CC2CCOCC2)CC2CCCC12 C(=O)(C(C)CC(C)(C)C)NCC(C)CC(=O)NCc1ccncn1 Fc1ccc2[nH]cc(-c3nc(C(F)F)nn3-c3cncc(Br)c3)c2c1 C1(C2(O)CCN(C(c3cccc4c3OCC4)=O)CC2)(NC(C2C(C)C2C)=O)CC1 N1(C(c2cc(C)oc2)=O)CCN(CC2CN(C(c3n[nH]cc3Br)=O)C2)CC1 c1(OC)cscc1C(=O)NCC1COC(CNC(=O)CCNS(C)(=O)=O)C1 Cc1nnc2n1CC(C(N1CCOCC1CCNC(c1cnccc1Cl)=O)=O)C2 CC1COc2ccccc2C1C(=O)NCC1CC(NC(c2cnc[nH]2)=O)C1 C1(NC(CCNS(CC)(=O)=O)=O)CN(C(=O)CC(=O)OCC)CC1F c1(C(=O)NC2CC(CCNC(C3C(C(C)C)(CC)C3)=O)C2)ccc(O)c(CO)c1 c1(C(N2C3C(CNC(C4C5COCC45)=O)C(C3)C2)=O)c(F)ccc2occc12 C12(C(=O)NCC3C(C)CN(C(c4cnn(C)n4)=O)C3)CCC(C1)OC2C Cc1cc(C(=O)NC2CC(NC(c3csc(C(C)C)n3)=O)C2)no1 C1(C(CNC(CN(C(C(Cn2cncn2)OC)=O)C2CC2)=O)O)CCC(C)(C)C1 N1(C(CNC(C)=O)=O)CCC(NC(c2c[nH]ccc2=N)=O)CC1 c1(C(=O)NC2C(NC(c3ccn(COC)n3)=O)C2)cc(C)c2ccccc2n1 CC(C)C(O)C(=O)N1CC(CC(=O)NCc2cccc(Cl)c2)C1 CC(C)C(CC(=O)NCCCCC1CC1C)NC(=O)CNC=O N1(C(C(C)NC=O)=O)CC=CC1CNC(=O)C(=O)NCC1CC1 CC1CCC(NC(=O)CC(C)(C)n2cnnn2)CN1C(=O)Cn1cnnc1 CC(CNC(=O)CC1CNC(=O)O1)C(=O)NCCOCCO c1(C(N(C2CCN(C(CSCCCC)=O)C2)C)=O)ccc(=O)n(CC(C)O)c1 c1(C(N2CCC(N(C(=O)CC3CC(C)(C)CO3)C)C2)=O)c(F)ccc2c1OCC2 C1(C(N2C(C)(CC(=O)NOCc3nc[nH]n3)CC2)=O)CCNC(=O)C1 c1(OC)cc(C(=O)NCCN(CC(C)O)C(=O)C=Cc2cscn2)cc(Cl)c1 C(=O)(C(C)S(N)(=O)=O)N1CCC(C(C)C(=O)NCC(O)(CO)CO)C1 C#CC1(O)CC(C(=O)NCC2(C(=O)NCc3cccc(F)n3)CCC2)C1 c1(C(=O)NC2C=CC(CNC(C3(O)CC(CF)C3)=O)C2)cc(F)cc(F)c1 C1(F)(C(=O)NCCN(C(c2cc(=O)c(OC)c[nH]2)=O)CC)C2CCCCC12 C1(C(N2CC(OC)(CNC(C3C4CCOCC34)=O)C2)=O)CCOCC1(C)C C1(NC(c2c(C(=O)OC)c[nH]n2)=O)CCN(C(C2(c3ccno3)CC2)=O)CC1 c1(SCCC(=O)NC2CCN(C(C3C(C#C)C3(C)C)=O)C2)ccc(C)c(C)c1 N#Cc1ccc(S(=O)(=O)NC(CO)CCF)cc1NC1CC(O)C1 C1(NC(Cc2c(C)ocn2)=O)CC2CN(C(C3CNC(=O)CC3C)=O)CC12 C1(CNC(C(C(C)C)CO)=O)CCN(C(C2CCCCN(C)C2=O)=O)CC1C C1(C(C)(C)O)CCC(C(=O)NCC2CC(NC(=O)Cc3cn[nH]c3)C2)CC1 N1(CCCCNC(=O)CCCc2ccccn2)CCCOC1=O C1(CNC(C(C)OC)=O)CC2(CCN(C(=O)CC(O)C(Cl)(Cl)Cl)CC2)C1 c1(OCC=C)ccc(Cl)nc1C(=O)NC1CC1NC(c1cnc(O)cc1C)=O C(C)(CCC(=O)NC(CNC(c1ncccc1-c1ccccc1)=O)C1CC1)OC C(=O)(C1=NOC(C)(C)C1)NC(CCN(C(c1ccc(CSC)c(F)c1)=O)CC)C c1(CC)oc(C=O)cc1C.C(=O)(CC(C)(O)C1CC1)N1CCC(C(C)N)C1 C(=O)(CCCC(F)(F)F)N1C(CNC(=O)Cn2cnnc2)CC2(CC2)C1 c1(C(N2CC(C)(NC(c3cc(C)cc(Cl)c3)=O)C2)=O)c(C)cc(F)cc1C C1(CCOC)CN(C(c2ccsc2)=O)CCN1C(=O)C(C)Oc1ccccn1 C1(C(C)C)CCOC1C(=O)NC1CC(CCNC(=O)C(O)Cc2ccccc2)C1 C1(C(N2CC3C(N(C)C(c4cnc(CO)s4)=O)C3C2)=O)CC2CCCN2C(=O)N1 Cc1cc(F)cc2[nH]c(C(=O)NC(C3(O)CN(C(C4COC(=O)O4)=O)C3)C)cc12 C(=O)(CCC(C)(C)C)NC1C(SC)CN(C(c2cc(-n3cccc3)ccn2)=O)C1 c1(N2CCN(CCCCS(C)(=O)=O)CC2)nccc(=NCCCCCF)[nH]1 CCCC(C(=O)NCC(C)(O)CNC(=O)CC(C)(C)O)OCC c1(OC)cc(O)ccc1NC(=O)C(C)(C)C1CCCN1C(=O)CSC(F)F C1(C(C)COC(C2(SCC)CCCCC2)=O)CC2(C1)OCCO2 C(=O)(C(C)(C)CC(=O)N1CC(NC(=O)C(C)(C)C(C)C)C(O)C1)OC C(=O)(CC1=CCCCC1)N(C)CC1(CNC(Cn2c(C)csc2=O)=O)CC1 C1(C(N2C(C(=O)NC)(COC)CCC2)=O)CCCCC(C)(C)C1 c1(OC)cnc(Cl)[nH]c1=NC(=O)C1C=CCN1Cc1cnc(-c2ccccc2)[nH]1 C(=O)(C(C)(C)COCCc1ccccc1)NC(CN(C(=O)C(F)=CCCF)C)C Cn1ccc(C(=O)NCC2(O)CC(CNC(c3ccccc3)=O)C2)n1 O=C(C#CC1CC1)NCc1ccc(CNC(C2CCCCC2O)=O)cc1 N1(C(CNC(=O)OCC=C)=O)CCOC2CN(C(=O)CC3CC=CCC3)CC12 N1(C(C)=O)CC2CCC(N=c3[nH]nc(C#N)s3)C2C1.CC1(OC(F)F)CC1 c1(CC(C)NC(=O)C(CN(C)C)NC(=O)CCCn2cncn2)nncn1C C1(NC(=O)Cn2cc(C3(CO)CC3)nn2)COC2COCC12 c1(C(=O)NCC2CCCCN(C(CC(C)C(F)F)=O)C2)cc2ccccc2n1C Cc1ccc2c(=NC3CCC(F)(F)CC3)[nH]c(=NCC3(n4nccn4)CC3)[nH]c2c1 CCC(C)CC(=O)NC1(CCNC(=O)C(C)C2CC2)CCC1 C(=O)(C(C)(CO)OC)NCCOCCCNC(=O)C(C)O.CCCCOCC C(=O)(C(CC(F)F)NC(c1ccc(C)cc1C)=O)N1CCCC(NC)C1 c1(NC(C(N2CCC(N)(COC)C2)=O)=O)cccc(N(C)C)c1F CC(C)C(C)(CNC(c1ccccc1-n1nccn1)=O)NC(=O)CCC1CC1C C1(NC(C2(OC)CC2C)=O)CC2(C1)CC(NC(=O)C(F)CC1CC1)C2 CS(=O)(=O)CCC(=O)NC1CCC(CCNC(c2cnn(C(F)F)c2)=O)C1 C1(C(=O)NC2CC(N(C)C(C3CN(C)C3)=O)C2)CCCN1c1cnccn1 C1(C2CCCC2)(C(=O)NCCN(C(C(C)CC(C)(C)C)=O)C2CC2)CCNC1=O c1(C(=O)NCC(C)NC(=O)COc2ccc(Cl)nc2)cnnc(O)c1 CC(CCNC(=O)C=Cc1ncc[nH]1)CCNC(c1ccsc1C(F)F)=O C(C(C)(C)C(=O)NCC1CC2C=CC1C2)NC(C(COC)C)=O CCCCC(C)CCC(=O)N1CC(NC(=O)COC2CCCC2)CC(C)C1 c1(C(=O)NC(C2(O)CCN(C(C=CSC)=O)C2)C)cnc2[nH]c(C)nc2c1 n1(CCC)[nH]c(=N)c(C(=O)CN(C2CCC(O)CC2)C)c1C c1(C(=O)NC(CSC)C)ccc(CNC(=O)C(O)c2ccsc2)o1 C1(C)(C(=O)NCC2C(NC(C3(OC)CC(CF)C3)=O)CC2)CCCCC1 C(=O)(C1=CC2CC=CCC12)NC(CNC(c1cccc(C(=O)OC)c1C)=O)(C)C C1(CNC(c2ncn(CC)c2)=O)CN(C)CCN1C(=O)CCc1cnc[nH]1 Cn1c(NC(=O)C(C)(C)Oc2ccc(-c3ccsc3)cn2)nc2cc(Br)ccc12 C1(OC)(CNC(=O)C(C)N2CCC2)CCN(C(=O)Cc2cncnc2O)C1 C1(C(=O)NCC2(O)CN(c3ncccn3)C2)CCC=CCCC1 C(CCCCCC(=O)NC1COCC1C)n1cc(-c2c(OC)cccc2)nn1 N1(C(CCn2cc(C(CC)NCC(C)C)nn2)=O)CC(C)OC(C)C1 c1(C(=O)OCC=CC(=O)OC)cc2c(Br)c(OC)ccc2[nH]1 C1(C(=O)NCCCC(CC)NC(c2cncc(C#C)c2)=O)CCc2nn[nH]c2C1 N1(C(c2cccc(C(C)=O)c2)=O)CCC(NC(c2oc(C)cc2C)=O)C(C)(C)C1 C(=O)(C(F)CCCC)NCc1cn(C2CCN(C(c3c(C#C)c[nH]n3)=O)C2)nn1 N1(C(C2CC(C)(F)C2)=O)CCC2CCN(C(c3cnc(C(F)(F)F)cn3)=O)CC12 Cn1c(C(=O)OC(=O)CCc2nnc(-c3ccc(Cl)cc3)o2)cnc1C1CC1 C1(C(N(C(CSCC)C)C)=O)CN(C(=O)CCc2conc2C)CCO1 N1(C(C(C=C)O)=O)CCC2CCN(c3ccc(C(=O)OC)c(C)n3)CC2C1 N1(C(c2csc3cccnc23)=O)CCC2(CC(NC(C3(O)CCC3)=O)CO2)C1 c1(CN2CCCCC(NC(c3cc(C)nc(Cl)c3)=O)C2)cnn2c1CCCC2 Cc1c(C(N2CCCC(N(C(=O)CC(C)CF)C)C2)=O)cc(C(C)C)n1C C1(C#N)(C(N2C(CCC(=O)NCC3(C(C)(F)F)CC3)CCCC2)=O)CCCCC1 Cc1c(C(N2CCCC3C2CC3O)=O)cnc2ncnn12 Cc1cnc2cccc(C(=O)NC3CCN(C(=O)Cc4cncs4)C(C)C3)n12 C(C)(C(O)C(=O)Nc1cccc(CNC(C2CC(N3CCOCC3)C2)=O)c1)OC C(=O)(C1CCCc2ccnn21)NCC1C(NC(=O)COc2cccc(Cl)c2)CC1 C(=O)(C1=CSCS1)NCC(C)(C1CC1)NC(C1CC(OC(F)F)C1)=O Cc1cc(C(=O)N(C(C)C(N2CCC(CNC(N)=O)C2)=O)C)c(C)[nH]1 C1(C(=O)N(CCCC(C)O)C)(NC(CC2CC(=C)C2)=O)CCC(C)(C)C1 c1(C(N2C(C3(O)CN(C(CC4CCN(C)C4)=O)C3)CCC2)=O)cnc(N)c(N)c1 c1(CCCC(=O)N(C2C3CN(C(CCC(=O)OC)=O)CC32)C)cc(C)ccc1C c1(C(=O)NC(C(C)C)CCNC(=O)Cc2cscn2)cc2c(cc1O)CCCC2 Cc1ccc(F)c(C(=O)NCCC2(NC(c3snc(O)c3Cl)=O)CC2)n1 N1(C(C(CCC)OC)=O)CC2CCC(C1)N2C(c1ccc(F)s1)=O CC1CCc2[nH]c(=NC(C)C(F)F)nc(N3CCC4(CC3)C(F)(F)C4(F)F)c2C1 CCCCC(O)CC(=O)NOCc1cc(Br)cs1 Cn1ncc2c1CN(C(C1CCN(C(=O)C(F)C(C)(C)O)C1(C)C)=O)C2 C1(NC(CCC(C)C)=O)CCN(C(=O)Cn2cnc(C#N)n2)C12CC2 C(=O)(CC(=O)NCC1(C(=O)NCC(O)C(C)O)CCCO1)N(C)C N1(C(CC)C(=O)N2CC(CNC(=O)C(F)CC)C2)CCc2ccccc21 c1(C(N2CC(NC(CC(C)(C)C3CC3)=O)C3C2C3)=O)cnc2nccn2c1 Cc1cc(N)cc(C(N2CCC(CNC(C3CC(C(C)C)=NO3)=O)CC2)=O)c1F O=C(CCS(=O)(=O)Cc1ccccn1)NC12CCCCC1NCCC2 N1(C(C2N(CCC)CCC2)=O)CC(C)CN(C(=O)C2=CCOC2)C(C)C1 C1(CNC(c2c(C)snn2)=O)CN(C(=O)Cn2nccc2C)CC12CCOCC2 CC1(C)CC(c2ccccc2)(C(N2CCC2CNC(C2(C#N)CC=CC2)=O)=O)C1 N1(C(c2c(CC)ocn2)=O)CC(C)C(C)(CNC(C2C(C)C2C)=O)C1 CC(C)(C)C(CN)CNCc1ccoc1C(=O)O C(=O)(C1CCc2c[nH]nc21)N(C(CC(C)C)C(=O)NCCc1cnn(C)c1)C N1(C(C2CCC(OC)C2)=O)CCC2(CCCC2NC(c2c[nH]cc2Br)=O)CC1 n1(CC=O)c(C)cc(O)cc1=O.C1(OC(C)(C)C)CCCN(C(=O)OC(C)(C)C)C1 C1(C(=O)NCC23CCCC2C3)CN(C(c2cccc(F)c2)=O)CC12CC2 c1(C(=O)NCCOC2CCN(C(c3c(C)nn[nH]3)=O)C2)cnc2c(c1)NCC2 c1(CC(N2CC(C)(NC(c3ncccc3O)=O)C2)=O)ccnc(Cl)c1F C1(C)(NC(C(CC2CC2)NC(CSC)=O)=O)CCCC1(C)C C1(C(N2CCC(N(C)C(C3(N(C)C)CCC3)=O)C2)=O)(OC)CCSC1 CN1CCCCCC1C(N1CCCC(C)(CNC(C2CCS(=O)(=O)N2)=O)C1)=O C1(CC(N2CC(c3c(C)nn[nH]3)(O)C2)=O)CCOC(COC)C1 CC(=O)CCCC(=O)NCC1CCC(NC(c2oc(C(C)C)nc2C)=O)C1 N1(C(c2nocc2Cl)=O)CCN(C(C2CCC(F)(F)C2O)=O)CC1c1ncc[nH]1 C1(C)(CNC(C(C2CCN(C(=O)CN3CCCCC3)C2)C)=O)CCCO1 C1(CC(=O)N(CCC(=O)NC(C)C)C2CC2)CCN(C(C2CCCCS2)=O)C1 C(=O)(C1=CCN(C(c2cc(C3CC3)[nH]n2)=O)C1)NC(C)Cc1cccs1 c1(C(=O)NCC2N(C)CCN(C(=O)CCS(C)(=O)=O)C2)cn2cccc(F)c2n1 c1(C(N2CC3C(NC(c4cscn4)=O)(CC3)C2)=O)c[nH]c2ccncc12 C1(C(=O)NCC=CCNC(C(CC)C(C)C)=O)Cc2ccccc2CO1 c1(CC(=O)NC2C(NC(C3(N=[N+]=[N-])CC3)=O)CCC2)ccccc1CC(N)=O N1(CCCOC(CNC(C(C)OC2CCCCC2)=O)=O)CCc2ccccc21 C1(CNC(c2c(C)ccc(C)c2)=O)C2CCCC1N(C(c1cn3c(n1)CCC3)=O)C2 N1(C(CCNC(C)=O)=O)CCC(C(F)(F)F)C(NC(=O)CCc2cc(C)on2)C1 C(CCCC#N)(c1nnnn1Cc1cccs1)NCC(C)CO N1(C(c2ccc(CO)o2)=O)CCN(C(=O)CC(c2cccs2)C2CC2)C2CCC12 c1(CN2CCC(CC(N3CCC(CNC(C)=O)C3)=O)C2)ccc(F)cc1Cl C(=O)(C(C(C)C)n1cncn1)NC1(F)CC(NC(CN(CC)CC2CC2)=O)C1 N#Cc1cnccc1NC(C1CCN1C(c1cccc(Cl)c1Br)=O)=O C1(N(C(C=C(C)C(F)F)=O)C)CCN(C(=O)Cn2c(C)ccc2C)CC1C c1(OCC(=O)NC(C)CCNC(=O)C(O)CF)ccc(F)cn1 N=c1[nH]c(C(=O)NCC(CNC(c2c[nH]nc2-n2cnnn2)=O)CO)cs1 c1(CC(C)C(=O)N2CCCC2C(C)NC(=O)CCC2CCCC2)cccc(Cl)c1 c1(C(=O)NCC(c2ccccc2)CNC(C2(N(C)C)CCCC2)=O)csc(Cl)c1 c1(N(CCS(N)(=O)=O)C)ncccc1S(=O)(=O)NCC1CCC(CC#N)CC1 C(=O)(C1CCCc2nccn21)N1CC2CN(C(CC(=O)OCCC(C)C)=O)C2CC1 c1(NCc2c(C)ccc(C(=O)O)c2)cc2c(cc1Br)OCO2 N1(C(c2c(C)cc(O)cc2)=O)CCC(NC(=O)COCCCN=[N+]=[N-])C(C)(C)C1 C1(C(=O)NCCCCNC(=O)C=CCN2CCCCC2)CC(=O)C12CCCC2 Cc1cc(F)c(C(=O)N(CCCNC(=O)C=CC2CCC2)C)cc1Br C1(NC(CC)=O)CS(=O)(=O)C12CCN(C(c1cn(C(F)F)c(C)n1)=O)CC2 C12(CNC(C3CCCC3)=O)CCCC1CN(C(c1cc3sccc3cn1)=O)C2 N(C1CCCc2ccoc21)C(C(C(C)NC(C(CCCC)CC)=O)(C)C)=O C12C=CC(C1)C(=O)N2.N1(C(C2CC2(F)F)=O)CC=CC1CF c1(CCC(=O)NCC(C)N(C)C(c2c(Cl)cncc2Cl)=O)ccc(F)c(Cl)c1 C(=O)(C(C)(C)CCCNC(C)=O)NCC12N(C(C(CC)OC)=O)CC(C1)C2.C(C)(C)C c1(NC(CC2(NC(c3ccc(CC)o3)=O)CCC2)=O)cccn(CCCO)c1=O N1(C(c2ccn(CCC)n2)=O)CC2CC1CC2NC(=O)C(Cl)=CCl Cc1[nH]nc(C(C)C)c1C(=O)NCCNC(=O)CC1CC1C(F)(F)F Cc1cnn(CC(N2CC(O)(C(C)NC(C3CC3c3cccs3)=O)C2)=O)c1 Clc1ccc2c(c1)CC(NCC1(c3ccccc3Br)CCCC1)C2 c1(C(N(C(CNC(C(CC)SC)=O)C2CC2)C)=O)cc2n(n1)CCCC2 C=CC1(CC(N2CCN(C(C3CNC(=O)N3C)=O)CC2CCO)=O)CCCCC1 c1(C(=O)N(C2(CNC(=O)COc3ccc(O)cc3)CC2)CC)ncc(Cl)cc1F CC(=O)CC(C)(C)C(=O)NC1C(C(=O)NCC2C3CCCCC23)C1(C)C C(=O)(CC(O)CC(C)(C)C)N1CCCCC(C(=O)NCc2c(C)ccnn2)C1 C1(CC(N2C(C)CC(CNC(c3onc(CC)n3)=O)C2)=O)CC2(CCCC2)CO1 O=C(C1=C2CCN=C2NC=C1)N1CCC2C(C1)CN2C(C1CC1[N+](=O)[O-])=O N1(C(CCCN(C)C)=O)CC2CCCC(CNC(=O)COc3ccccc3)C2C1 CN1CCN(C(C2(C)CCCN2C)=O)C(C(=O)N(CC(O)C2CCC2)C)C1 C1(CC)CC(C)CN(C(c2ccoc2CNC(=O)CCc2ccnn2C)=O)C1 c1(C2N(C(c3nc(Cl)cs3)C(=O)NCCOC)CCC2)cccc(C)c1 c1(CCN(C(=O)C(C)CN(C)C)CCC(=O)NCC(CC)O)ccccc1 c1(C(N2CC(C)C(CNC(=O)CC3CCCC3C)C2)=O)[nH]nc2cnccc12 C1(NC(=O)CCc2nncs2)CCOC12CCN(C(=O)C=CC1CCCO1)CC2 C1(C(=O)NCCCN(C(=O)C(C2CCOCC2)F)C(C)C)CCCSS1 C1(CNC(=O)C=Cc2cccs2)CN(C(=O)COc2ccsn2)C2CC12 C12(NC(CCN(CCC)C)=O)CCCN(C(=O)CCn3cncn3)CC1C2 c1(N(C)C)ccc(CCC(N2CCC(CNC(c3cnc(O)o3)=O)C2)=O)cc1 c1(CCNC(C23CCCN(CC2)C3)=O)cc(Br)ccc1Cl Cc1cccc(SCC(=O)N(C)CC2CN(C(c3cnc(C(F)F)nc3)=O)C2)c1 N1(C(C(C)(C)CC2CC2)=O)CC2CCCC(C1)N2C(c1ccc2c[nH]nc2n1)=O C=CCC(C(=O)NCC12CC1CN(C(=O)CC1CC(C)CC(C)(C)C1)C2)C(C)C c1(C(C(=O)N(CCCN(C(CCCC)=O)C)C)(C)O)ccc(F)c(Br)c1 C1(CNc2c(OC)cccc2)(OC)CCN(C(c2nncs2)=O)CC1 N1(C(c2c(CC)n[nH]c2)=O)CC=CCC1C(=O)NCC1(F)CCN(C)C1 C(c1cccc(Cl)c1Cl)=CC(=O)NC1CN(C(Cc2nnc(C)s2)=O)CC1C N1(C(C(C)n2cccc2)=O)CCCC(C(=O)NCC(C)(F)C(C)C)C1C CN1CC(C(=O)NCCCCN(C)C(C2CC3CCC2O3)=O)NC1=O C(=O)(C(C)(C)CO)N(C1CCN(C(C2(C(C)(F)F)CCC2)=O)C1)CC C1(CC(=O)NCCCC(C)NC(c2cnc(=N)[nH]c2)=O)CCCC(C2CC2)O1 Cc1cc(C=CC(=O)OCC2(C(=O)OCC(F)(F)F)CC2)ccc1F C(C)(C)(CC(=O)NC(C1CCCN1C(=O)Cn1nccc1C)(C)C)OC C1(C(=O)NCCN(C)CCO)C=CCCN1C(=O)Cc1ccncc1F c1(C(CC)C)cccc(NC(=O)CCN(CCCO)C)c1 C1(NC(C(C(C)(C)C)O)=O)CCC2CN(C(=O)CSCc3cccnc3)CC12 c1(C(=O)NC(c2cccc(I)c2)C)ccn2c(C3=CCNCC3)cnc2c1 Cn1nc(C2CC2)cc1C(=O)NCCOC1CCN(C(C23CCC2C3)=O)C1 CN=c1[nH]c(N2CC3CN(C(=O)CCc4ncc[nH]4)C3C2)ncc1F c1(C(N2CC(O)(CNC(CC(C)OC)=O)C2)=O)c(F)ccc2n[nH]cc12 N1(C(CN(C2CCC2)C)=O)CCN(C(C2CC3CCC2O3)=O)CC1CO C1(C)(CNC(CC=CC)=O)COCCN(C(=O)C(O)CCCC)C1 N1(C(c2cnc(OC)nc2)=O)CC(F)(F)CC1C(N1CCCC(C)C1CCO)=O c1(C(=O)NCCC(C)N(C(C(C)OC)=O)C)c(F)ccnc1Cl c1(C(C)C)cc(C(=O)N(C)CCN(C)Cc2csc(Cl)n2)on1 Cc1nc2cc(C(N3CCC(NC(C4CC4F)=O)C3C(C)(C)C)=O)ccc2s1 C1(C(=O)NCC2(N(C(=O)CCc3cn(C)nn3)C)CC2)CCn2nnnc2C1 c1(C(N(CC(C)NC(=O)CCOC2CCCC2)CC)=O)ccc(Cl)cc1C S(=O)(=O)(c1cn(C)nc1-c1cnn(C)c1)NCc1c(C)nn(C)c1Cl N1(C(C2C(=O)OCC2)=O)CCC2C(CCCN2C(=O)Cc2cnoc2)C1 N1(C2CN(C(=O)C=Cc3cnc[nH]3)C2)CCN(C(=O)C(CCSC)NC)CC1 C(=O)(C1=CC(O)CCC1)NC1CCCN(C(Cn2cnc(C#N)n2)=O)CC1 c1(C(N(CC(C)NC(=O)C(F)(F)c2csc(Cl)c2)CC)=O)cn2cc(C)sc2n1 C#Cc1cnn(CC(=O)NC(CCF)C(=O)NC2COC(C(C)C)C2)c1 Cn1nc(C(=O)NC2CCCC2NC(c2ccc(Cl)cc2)=O)ccc1=O CCC(CC)CC(=O)NC1CC(CC(=O)N(C2CC(C(N)=O)C2)C)C1(C)C C1(CNC(COCC#C)=O)CC(C)CCN1C(=O)C(C)Cc1cnco1 Cc1ccc(O)c(S(=O)(=O)Nc2ccc(O)c3ccccc23)c1 C1(C(=O)NCCC2(NC(C(c3cn(C)nc3)(F)F)=O)CCC2)CC2C=CC1O2 C1(F)(CNC(CCC#CC)=O)COCCN(C(=O)C(C)(C)OC(C)C)C1 N1(C(C(c2ccc(Cl)nc2)(C)C)=O)CC(NC(C2CC2C(N)=O)=O)C(N=[N+]=[N-])C1 N1(C(C(C)OCCC=C)=O)CCCC1CN(C)C(C1CCCC1CC)=O c1(SCC2(CNC(C3CCC3)=O)CC2)cnc(N2CCOCC2)c(F)c1 C(=O)(C(CCc1ccccc1)C1CC1)N(CCNC(CN(S(CC)(=O)=O)C)=O)C c1(C(N2CC(CC=C)(NC(=O)CCN3CCOC3=O)C2)=O)c(C2CC2)cnn1C C(CCC(=O)NCCCSCC)N(CCCOCC)C(C1(C2CCCO2)CC1)=O N1(C(Cc2nc(C)sc2C)=O)CCCC(NC(=O)CC(O)C(C)C)C1C c1(C(=O)NCC2C(CC(=O)NCC3(CCC)CCC3)CC2)cc(Cl)cs1 c1(C(N2C(C)CCC(CNC(c3c(C)ncs3)=O)C2)=O)nccc2c[nH]nc12 C1(NC(C=CCCC)=O)COC2C(NC(c3ocnc3C(F)(F)F)=O)COC12 C(=O)(C1CCC(=O)c2ccccc21)N1C(C(F)(F)F)C(C)S(=O)(=O)CC1 c1(OC)c(C)cc(C(=O)NCC2(NC(C3(F)CCS(=O)(=O)C3)=O)CC2)cc1Cl CCC(C)(C)C(O)C(=O)N1CC2(CCCC2C(=O)NOCC2(C)CCC2)C1 C#CCC(C)(C)C(=O)N1CCC(CCC(=O)N(CCCCC(=O)NC)C)C1 Fc1c(CNC2CN(c3ccc(C(F)F)c(Cl)c3)C2)cccc1C(F)(F)F c1(OC)ccc(C(=O)NCC2C3CCC(C3)N2C(c2ccon2)=O)c(OC)c1C CC(C)(C)S(=O)(=O)CC(=O)NC1CC(CNC(C2CC23CCC3)=O)C1 CC1(C)OCC2CC12C(=O)NCC(C(C)(C)C)NC(=O)Cc1ccc(O)cc1 c1(CNCC(CNC(C)=O)(C)C)nn(C)c2c1CCCC2 c1(C(N2CCC(C)(C(=O)NCC=CCSC)C2)=O)ccc2c(c1)CCC2 C(=O)(CCCCCN(C(=O)CC1(O)CCCCC1)C)NC(c1ncc(C)[nH]1)CC c1(C(=O)NC2C(C)CN(C(c3csnc3Cl)=O)C2)cc(Br)ccc1O c1(C(C2CC2)NC(=O)NCC2CC23CC3(F)F)ccc(-c2ccsc2)cc1 c1(CC(N2CCC(CNC(C(C)SC)=O)C2)=O)c[nH]c(=N)nc1O C1(CNC(COCC)=O)CN(C(c2cc(C(F)F)no2)=O)CCC1(F)F N1(C(C)=O)CSCC1C(=O)NCCCC(C)NC(c1csc(C)n1)=O CC1CN(C(c2cnc(C(C)(C)C)[nH]2)=O)CC1CNC(C1CC2CCC2C1)=O N1(C(CN(CCC)C)=O)CC2CC2(NC(=O)C(C)(C)n2ccc(C(=O)OC)n2)C1 c1(C(=O)NCC2C(NC(c3cccc(OC)n3)=O)CC2)cc2cccnc2o1 c1(C(=O)OC)ccc(C(=O)NCC2(F)CCCN(C(C3CCC3C)=O)C2)c(F)c1 S(=O)(=O)(c1ccc(C)c(C(=O)OCCC2CC3C=CC2C3)c1)NC c1(OC)cccc(C(N2CCCC2CC(=O)NCc2ccnn2C)=O)n1 C1(C(N(CC(CC)NC(C2(CC)CCC2)=O)CC)=O)CCc2nn[nH]c2C1 C1(C)(NC(C(C=C)NC(C)=O)=O)CCCN(C(=O)CCCn2ccnc2C)C1 c1(C(=O)NC(C)CCNC(c2cnn(C)c2Cl)=O)ccc2nc(N(C)C)sc2c1 N1(C(c2ccn(C)c2)C(=O)NC(C)C)CCOCC1CC(=O)OC(C)(C)C C1(C)(NC(CC2C(CNC(CSC(C)(C)C)=O)C2)=O)CCOC1 c1(C(N(CCN(C)Cc2ncnc(Cl)c2CC2CC2)C)=O)cnc(CO)nc1O N1(C(C(C)Oc2ccccc2F)=O)CCCC(NC(C2(C)CC2(F)F)=O)CC1 CC(=O)CCCC(C)C(=O)N1CCC(C)C1C(=O)NC1CC(C)CC(C)(C)C1 c1(OC)ccc(F)c(C(N2CCN(CC(=O)Nc3cc(Br)ccc3N)CC2)=O)c1 c1(N2C3CC(CNC(C4C(C)(C)C4(C)C)=O)(OC3)C2)nc(O)c2ccccc2n1 c1(C(=O)NCCCCN(C(=O)C(c2ccccc2)O)C)cccc(O)c1C CCCC(CC(C)C)C(=O)N(CCN1CCN(c2nccnc2F)CC1)CC c1(C(=O)NCC(c2ccccc2)CNC(C=CCC)=O)cnn(CC(C)C)c1 CCCC(C(=O)OC)C(=O)NCC(C)(C(C)C)NC(C1CC(OC)C1)=O N1(C(C(C)NC(C)=O)=O)CCN(Cc2cccs2)CC(C)(F)C1 c1(C(N2CCC(CC(=O)OC)(COC)C2)=O)c(Br)cc(O)cc1Br c1(C(N2CC(NC(C(C(C)C)NC(C)=O)=O)C(F)C2)=O)cccc(Cl)c1I c1(C(N(C2CC3CC(C(=O)OC)C2C3)C)=O)ccc2nc[nH]c2n1 c1(C(N2CCC(C)(CNC(c3nnn4c3CCC4)=O)C2)=O)cccn2ccnc12 c1(CC)cnc(O)c(C(N2CCN(C(=O)Cc3c[nH]nc3C)CC2CC)=O)c1 CC1CC(CNC(=O)CCC23CCC(CC2)C3)CN1C(C1CCCCCC1)=O N1(C(c2cccc(C(N)=O)c2)=O)CC(NC(C23CCC2C3)=O)C(C2CC2)C1 C1(CN(C(c2coc(C(N)=O)c2)=O)CC)CCCCN1C(=O)CC1(C)CCCC1 C1(O)(C(C)NC(c2conc2C2CC2)=O)CCN(C(=O)C(c2ccccc2Cl)C)C1 N1(C(C(C2CCCCC2)NC(C(CC#C)O)=O)=O)CCC(C)(C)CC1C Cc1nc2nnnn2c(C)c1CC(N1CC(NC(=O)C(N)=O)CC(O)C1)=O C1(N2CCC(c3c(OC)nccn3)CC2)CC(F)CN(C(C2CCCS2)=O)C1 c1(C(N2CC(CCCNC(C#CC(C)(C)C)=O)OCC2)=O)cnc2cc[nH]c2c1 C=CC(C)(CCOC)C(=O)NC(CCC)C(O)C(=O)NCCc1ccnc(C)n1 C=CCCCCC(=O)N(C1CCCC(N(C)C(c2ncoc2CC)=O)C1)C C1(C(=O)NC(C)Cc2cnccn2)CCC(NC(c2ncccn2)=O)CC1 N1(C(C2C(C)C2C)=O)CCC(C)(NC(c2cc(-c3ccccc3)on2)=O)C1 C(C)(C)(CS(=O)(=O)NC(C1(c2ccccc2)COC1)C)OC C1(NC(=O)C2=CCCO2)CCC2CN(C(=O)CN3CC(=O)NC3=O)CC2C1 C(=O)(C(C)(C)N(C1CC1)C1CC1)OC.C1(=O)C(Cc2ccccc2)N1.C(C)(C)C c1(C(=O)NC2C(CNC(CNC(=O)OCC=C)=O)CC2)ccc2ccccc2n1 c1(OCC(=O)N(c2c(C)non2)C)ccc2c(c1)C(=O)NCC(C)(C)O2 c1(C(=O)NC2CCC(C(=O)NCc3cccc(C)n3)OC2)ncc(C2CC2)cc1F C1(C(=O)NCC(C2CC2)NC(c2cc3c([nH]2)CCOC3)=O)Cc2cccnc2C1 C1(NC(Cc2c(C)nc(S)s2)=O)CCCCN(C(c2cc(F)cnc2Cl)=O)C1 N1(C(c2cc(OC)n[nH]2)=O)CCN(C(=O)CCCCCSC)CC1C1CC1 c1(C(=O)NC2C(OCC)C2)cccc2c1CCN(C(c1ncc(C(=O)O)[nH]1)=O)C2 C=C(C)CC(C(=O)N1CC(n2cccn2)C1)NC(C1CCOC1(C)C)=O C=C(C)CC(C(=O)NCc1cnc(O)cc1C)NC(=O)C(COC)CC Cc1[nH]c2ccc(F)cc2c1C(N1CCC1CNC(C1CC(F)(F)C1(C)C)=O)=O C1(C)(C(=O)NC2C(C)CCN(C(c3ccccc3Cl)=O)C2)Cc2ccccc2C1 c1(C(=O)NC2C(CNC(C=CCC)=O)CCC2)cn2cc(Cl)cnc2n1 N1(C(C(C2CCCOC2)OC)=O)CCCC(NC(c2ccc(C(C)C)nc2)=O)C1 C1(NC(c2c(C)cnn2C)=O)CCN(C)C12CCCN(C(=O)C(C)C1CC1)C2 N12CCOCCC1C2.c1(C(=O)OC)nnc(C2CC2)s1 c1(OC)cccc(Br)c1CCNC(=O)C(C)Sc1ccc(Cl)cc1 CC1(C)CC(CNC(c2cc[nH]c2C(F)F)=O)CN1C(=O)CC1COCCO1 C1(CNC(c2coc(Br)n2)=O)CC2(CCC2)CN1C(=O)CC1CC1 N1(C(CC(C)NC(N)=O)=O)CCC(C)(NC(C2CCC(F)(F)C2)=O)C1 Cc1cc(C(=O)NC2CCCCN(C(c3csc4nnsc34)=O)C2)ncc1F N1(C(CC2(CSC)CC2)=O)CCC(C(=O)NC(C)Cc2nc[nH]n2)C1C N1(C(C2(C)CN(C(CC3CCCC(OC)C3)=O)C2)=O)CC(O)(C2CC2)C1 C1(CC(=O)NCc2c(CCNC(C(CC)C)=O)ocn2)CCCC2(CCC2)O1 Cc1cccc(F)c1CC(=O)NC1CC(CNC(=O)C2=C(Cl)CCC2)C1(C)C Nc1cc(F)c([N+](=O)[O-])cc1C(N1CCCC(NC(=O)Cn2ccnn2)C1)=O C(=O)(C1=NOC2(CCCN(C(=O)C(O)C(C)C)C2)C1)Nc1c(C)ccc(OC)c1 N1(C(CC(C)C)=O)CC(NC(c2ccc(OC(F)F)cc2)=O)C(CC(C)(C)C)C1 CN1CCCC(C(=O)NCC(O)C(=O)NCCc2cn(C)cn2)C1 c1(C(C(=O)NC(C(C)NC(=O)C(Cl)=CCl)C)=O)ccc2c(c1)CCCC2 C(=O)(CC(F)(F)C(F)F)NCC1(C)CCCN1C(c1ccc(Cl)c(N)c1)=O c1(C(=O)NCC(CC)N(C(=O)C(C2CC2)N(C)C)C)cnc(COC)[nH]1 c1(C(=O)NC(CNC(c2cc(CCC)on2)=O)(C)CC)ccnnc1O C1(C(=O)NC(C(=O)NC(c2cccnc2)CC)c2ccco2)OCCC1C CC(CC1CC1)C(=O)N1CC(C)(OCC(=O)NCC(C)(O)Cc2ccccn2)C1 c1(C(=O)NC(CC=C)Cc2ccccc2)cnn2c(O)cc(C)nc12 N1(C(CCc2c(C)ncs2)=O)CCN(C(C2CCN(C(=O)NC(C)C)C2)C)CC1 C1(C(C)(C)NC(C2CC=CCC2)=O)CCN(C(=O)CCOC2CCOCC2)C1 C1(NC(C2(CC#C)CCOC2)=O)CN(C(c2ccc(C)nc2)=O)CC1C S(=O)(=O)(c1ccc2[nH]c(=NC(C)Cn3nc(C)cc3C)sc2c1)NCC=C C1(NC(C)=O)CN(c2nc(CC3CC3)ns2)CC1C C(=O)(CC(CC)NC(c1cnn(CCOC)c1)=O)N1CCC(CC=C)C1 N1(C(C(C)F)=O)CCC(CO)(CNC(C2CCCCCC2)=O)C1 C1(C(N2C(CCNC(c3c(C)scc3)=O)CSCC2)=O)CC(C2CCCC2)C1 C(=O)(C(C(C)(C)C)NC(c1ocnc1C)=O)NCc1snc(CC)n1 c1(CC(=O)NNC(=O)c2cc(Br)ccc2I)ccc2[nH]ccc2c1 C1(C(n2nnc(C(C)(C)C)n2)=O)COC2(CCCNC2)C1 C1(CC)C2CCC(O2)C1CC(=O)N(C(C)CSC)C C#CCCC(C(=O)N(CC(=O)OC)C)NC(C1CC2(CCC2)CO1)=O N1(C(CN(CC#C)C(c2n(CC#C)ccn2)=O)=O)CCC(C)=C(F)C1 N1(C(Cc2onc(C)n2)=O)CCC2(C1)CN(C(C13CC1COC31CCC1)=O)C2 N1(CCc2n(C)ncn2)CCC(=O)N(CCc2cccc3cc[nH]c23)C1=O C1(CNC(Cc2c(C)occ2)=O)N(C(C2CCS(=O)(=O)N2)=O)CCCC1(C)C N1(C(C2(c3ccccc3)CC(C)(C)C2)=O)CC(NC(C2CCCC2)=O)C2(CC2)C1 N1(C(CCC(=O)c2ccc(C)s2)=O)CCC(NC(=O)CCC(C)O)C(O)C1 C(=O)(CCCC(=O)N1CCC(NC(C2CCCNC(=O)C2)=O)C1(C)C)OCC C1(NC(C2(OC)CCN(C(=O)CCc3nc[nH]n3)C2)=O)CCC(=O)NC1C c1(NCCCC(C)NC(=O)OCC)cnc(C2CCC2)nc1O N1(C(c2c(CC)cco2)=O)Cc2[nH]nc(C(=O)N(C)CC3CC3)c2C1 C=CCC(C(=O)NC(C)CNC(c1csc(-c2cccc(Cl)c2)n1)=O)NC(C)=O c1(NCC2(C)CCCS2)nccc(=NCCCF)[nH]1 C1(C)(CNC(C2CCN(CC)C2)=O)CCCN1C(=O)Cc1cc(C2CC2)no1 C1(C)(C(=O)NC(C2CCN(C(CCc3cc(C)on3)=O)C2)C)CC2CC2C1 O=C(C(O)CC(F)(F)F)N1CC=CC1Cn1cc(C2CC3CC3C2)nn1 c1(CNC(c2nccs2)=O)ccccc1-n1cc(C(=O)O)nn1 c1(C(N2CCC(N(C(C3CCOC3)=O)CC)C2)=O)ccnc(C)c1N C12(CC(=O)NCC3CN(C(c4ncncc4Cl)=O)CC3O)CCC(CC1)OC2 c1(C(=O)NC23CC2CN(C(c2ncccc2O)=O)C3)ccc(F)cc1Cl C1(NC(c2ccc(OC)nc2)=O)CC2CCC1N2C(=O)CCC(=O)c1cccs1 Cc1nc(C(N2CCC(C(C)NC(=O)CCN3CCOCC3=O)C2)=O)c(C)n1C CCCCCCCC(=O)NCC1CC2(CC(NC(=O)C3=NOCC3)C2)C1 C1(CNC(c2nc(Cl)ccc2Cl)=O)CCCCCN1C(c1cccc(F)c1)=O c1cnn(CCO)c1C.c1(CNC(c2nnnn2C)C(=O)NCC=C)nc(C)cs1 c1(C(N2CCC(CNC(c3c(NCC)cccc3)=O)C2)=O)ccc(F)c(F)c1N c1(C(N(C)CC2(NC(c3cc(C)ncc3)=O)CC2)=O)n[nH]c2c1COCC2 N1(C(CCCCN(C(c2ncn(C(C)C)c2)=O)C)=O)CCCC(C)(N(C)C)C1 Cc1nn(C)cc1C1OCCC1CCN1CCCCC1.C(CCNC)OC C12(CNC(=O)Cc3ccco3)CC(C1)C(NC(C1(F)CC1)=O)CO2 c1(NC(C2OCCN(C(Cc3c(C)ccc(Br)c3)=O)C2)=O)ccc(C#N)c(F)c1 N1(C(c2c(Br)ccc(OC)c2)=O)CC2CCN(C(C3(F)CCC3)=O)C2C1 Cc1cc(C(=O)NCCN2CCOCC2C(C)C)nc(C)n1 n1(CC(=O)NCC(CNC(C(n2cnc(C#N)n2)CC)=O)OC)nc(C)cc1C C1(CN(C(c2nc(CC)oc2)=O)C)C2CN(C(C3CC34CCC4)=O)CC12 c1(CNC(C2C(C)(C)C2)=O)ncc(C(=O)NCCC(F)F)cn1 N1(C(CSCC)=O)CC2CC1C2CNC(=O)COCCc1ccccc1 c1(C(=O)NC2CCCC(NC(CCSCC)=O)C2)c[nH]c(=NCC(F)(F)F)cn1 N1(C(CSC(C)C)=O)CCC(NC(c2cccc(-c3cc[nH]n3)c2)=O)C1C1CC1 C(=O)(C1=C(C#N)CCC1)NC(CC#CC)C(=O)NCC1CCCC(C)(C)O1 N1(C(c2cnc(C)s2)=O)CCC(NC(=O)Cn2c(C)c(C)sc2=O)C(F)C1 CCC(C)(COC)C(=O)NC1CC2(C(C(N3CCOCC3)=O)C2)C1 C(=O)(C#CC(C)(C)CNC(c1c(C)ccnc1C)=O)NC(CCC=C)C N#Cc1ccc(CCC(N2CCCC2CNC(=O)CSC(F)(F)F)=O)cc1 c1(NC(C(CC2CC2)NC(c2sccc2F)=O)=O)ccc2ccncc2c1 C1(O)(CN(C(=O)C=CCC2CCCC2)C)CCCN(C(=O)CSCCC#N)C1 c1(CNC(C(C(C)C)NC(Cn2c(C)nnn2)=O)=O)ccc(F)cc1F C1(C(N2CC3C(NC(c4c(C)nn[nH]4)=O)(CC3)C2)=O)CCCC2(CCCCC2)C1 Cc1cccc2c1OCC2C(=O)N(C)CCNC(=O)CCN(C(=O)C=CCl)CCO C(CNC(=O)C(C)(C)CN(C(=O)C=Cc1ccco1)C)(CC(C)C)OC c1(C(=O)NCC2N(C(CC3(C)CC3)=O)CCC2)ccc(N2CCCCC2=O)cc1 C1(CC=C)(NC(=O)C(C)O)CN(C(=O)CCc2nccn2C)C1 Cn1cnc2ccc(C(=O)NCC3CCCC(NC(=O)C(O)C(F)F)C3)nc12 c1(C(=O)NCC2(O)CN(C(c3cc(COC)sc3)=O)C2)ccc2nnn(C)c2c1 c1(C(=O)NC2(CC)CN(C(c3cnc(O)o3)=O)C2)cc2ccccn2n1 C(=O)(C1=C(C)N(C)c2ncnn2C1)N(C)CC1C2CN(C(C(CSC)C)=O)CC21 C1(OC(=O)CCCOCc2ccccc2)CC(C)N(C(=O)OC)CC1C C1(C(N(C2CCN(CC)C2)C)=O)COCCC1NC(=O)CC(=O)OCC C1(CN(C)C(C2CCN(C(=O)C=Cc3cnn(C)c3)CC2)=O)CCC(C)(C)O1 N1(C(C(C)S)=O)CC2C(C1)N2C(c1cc(C(C)(C)C)on1)=O C(C(CNC(=O)CC1CCOCC1)C(F)(F)F)NC(CCc1cn(C)nc1)=O C(=O)(CC(C(C)OC)NC(c1cnncc1OC)=O)OC(CC)CC N1(C(c2c(CC)nc(C)[nH]2)=O)CCCC(NC(=O)C(c2cccc(C)c2)O)C1C N1(CC(=O)NCC2C(NC(C(CC=C)(C)C)=O)COC2)CCCCC(O)C1=O C1(C)(COC)CC(NC(c2ncc(N)nc2C)=O)CN1C(=O)CS(N)(=O)=O C1(C(NOC(C=C)C)=O)CN(C(=O)CC2CC3(CCC3)C2)CC(C)O1 N1(N2C(C(=O)Nc3cc(C=O)n(C)n3)(COC)C=CC2)CCCCCC1C c1(OC)ccc(CNC(=O)NC2CCOCC2F)c(Cl)n1 C#CCC(C)C(=O)N1CCCC1CN(C)C(C1OCCOC1C(F)(F)F)=O Cc1ccc(N(c2nnc(NC(COC(C)(C)C)=O)n2CC2CCOC2)C)cc1 c1(OCC)ccccc1C(=O)OCC(=O)NC(c1cccc(O)c1)C n1(CC)ccnc1C1OCCC1C(=O)NCCCC(=O)Oc1ccccc1 CCC(C(=O)NCC1CCN1C(=O)CCn1cncn1)NC(N)=O CCC(CC#N)C(=O)NCCCN(C)C(c1ccc(F)cc1CSC)=O c1(C(C2CCN(C(=O)COc3ccccc3)C2)C)cncc(Br)c1 C(N=c1nc(N2CCCC3(C2)CC3(F)F)c2c(ncn2C)[nH]1)c1snc(C)n1 C(=O)(C(CC(C)C)CC(C)C)N1CCC2(C(NC(C=C(CCC)C)=O)CCC2)C1 Cc1nc2cc(C(=O)NCC(O)CNC(=O)CC3CCOC3)ccc2n1C c1(N2CCC(C(=O)NC(CC)C)CC2)nccc(=NC2C=C(C)CCC2)[nH]1 C1(NC(C(C)OCCN(C)C)=O)CCN(C(C2CCCS2(=O)=O)=O)CC1F c1(CC)oc(C(N2CCC(C(=O)N(C)C(c3ccncc3)C)(CF)C2)=O)cc1C CC12CCC(C(=O)NC3CCC4CC4C3)(CC1)C2 c1(NC(C(CNC(C2CCN(CC)C2)=O)CC2CC2)=O)cc(C)c(O)cc1C c1(CN(C23CC2COC3(C)C)C)ccc(F)c2cccnc12.CC(C)(C)OC=O C1(CCC(=O)NCCOCCCN(C)C(C2CC2C2CC2)=O)CCC(O)CC1 C(=O)(C(C)CC(C)C(C)=O)NCc1ccc(C(N(CCC#C)CC)=O)o1 C(C(C)(C)CC(C)O)N(CC(N1CC(OCC(=O)NC2CC2)C1)=O)CC C1(NC(C2Cc3c(cn(C)n3)C2)=O)CN(C(=O)CC2=CCOCC2)CC1N=[N+]=[N-] c1(C(=O)NCC2(CNC(CC(CCC)C)=O)CC2)cnc2n(c1=O)CCS2 N1(C(c2cc(C#N)no2)=O)CC2CCC(C1)N2C(=O)C(O)CC1CC1 c1(C(=O)NC2C(CNC(C3CCCN(CC)C3)=O)C2)ccc(Cl)c(C(C)=O)c1 CC(CC(F)(F)F)C(=O)NC1(CNC(=O)Cn2cnc(Br)c2)CCCCC1 N1(CC(=O)NCC2CC(CNC(C3C(C)CC3)=O)C2)CCC(C)(C)C1 c1(C(=O)NCC2C3N(C(CCOCC(C)C)=O)C(CC3)C2)cc2scnc2[nH]1 N1(C(c2c(C)[nH]nc2C(F)F)=O)CCC(C)(CNC(C2CC(F)CN2C)=O)CC1 C1(O)(C(CNC(COC)=O)C)CCN(C(=O)CN(C(=O)COC)C)C1 c1(OC)cccc2cccc(C(=O)NCCCN(C(=O)CCF)C)c12 C(C)(C(=O)NNc1cccc(C(=O)O)c1C)Oc1ccc(C)cc1C c1(CNCC(C)S(C)(=O)=O)sc2ccccc2c1Br c1(CC(=O)NC2CC(CNC(C3C(C(=O)OC)CC3)=O)C2)cn(C)nn1 N1(C(CN(C(C)=O)C)=O)CCC(F)(CNC(=O)CC2CCC(F)(F)C2)C1 N1(C(CNC(C)=O)=O)CC2CCC2(CNC(=O)C(C)Cc2cnco2)C1 C=C1CCC(C(=O)NC(CNC(c2ccc(C(C)C)nc2)=O)C2CCC2)CC1 c1(C(=O)NC2CCC(NC(=O)CC3C=CCC3)CC2)ccc(F)c2ccncc12 C1(NC2(CSC)CC2)COCC(=O)N1C c1(C(=O)NCC(COC)NC(C2CC3(CCC3O)C2)=O)c(F)cc(F)cc1F C1(CNC(C2CC(CF)C2)=O)CN(C(c2cc[nH]c3nccc2-3)=O)CC12CCC2 Cc1nn2cc[nH]c(=O)c2c1C(=O)NC(C)CC(C)NC(=O)C(F)(F)C(C)O C1(C#CC(=O)Nc2cccc(NC(=O)C(C)NS(C)(=O)=O)c2)(CC)CC1 c1(NC(C)=O)ccc(C(=O)NC2CCCN(C(=O)C(C)Cc3cnc[nH]3)C2)nc1 N1(CCNC(C=C)C)CCN(c2nnnn2CCOC)CC1 N1(C(c2c(C(C)C)c[nH]n2)=O)CC(CNC(=O)C(C)C#N)CC(C)(C)C1 c1(C(=O)NCCCCC2C(C)C2)cc(CNC(c2ccsn2)=O)no1 C#Cc1ccc(OCC(=O)NCC(C(C)C)NC(C2CCN(C)C2)=O)cc1 c1(NC(C2C(C(=O)NCc3ncc(C)nc3)C2)=O)ncc(Br)c(C)c1[N+](=O)[O-] C1(N(C(CSC)=O)C)CCN(C(C2(F)CCOC2)=O)CC12CC2 c1(C(N(C2(CC(NOC(C=C)C)=O)CC2)C)=O)cc(O)n(C)n1 C1(N(CC(=O)NCC2(F)CCC2)CC)CCOCC1.C12=CC(=O)N(C1)C2 C(=O)(C1=CCC(C)CC1)N1CC(C(C)NC(c2csc(Br)c2)=O)C1 c1(C(CNC(c2cnns2)=O)NC(C2CC(C#N)C2)=O)cccc(Cl)c1 N1(C(c2c(CC)nc[nH]2)=O)CCC2OCCN(C(c3ccc(N)c(Cl)c3)=O)C2C1 C#CCCCCCC(=O)NC(c1ccccc1)C(=O)N1CCC1CC1CC1 C12CC(C3OC(C)(C)OC13)OC2=O.Cc1cc(C(N2CCCC2)C)c(C)n1C c1(C(C(=O)NCCSC)N(CC(C)(C)C)CC)nc(Cl)sc1Cl N1(C(C(C)OCCOCC)=O)CCC(C2CC2)(C(=O)N(CC(F)(F)F)CC)C1 C(=O)(C(C)(F)C(=O)NC1CCC1NC(c1cn(-c2ncccn2)cn1)=O)OC c1(NC(C2N=CN(C)C2)=O)ccc(N2CCNCC2)cc1F c1(C(=O)NC(CC)(C)CNC(C2CCCN2C)=O)ccc(Br)c(C)c1 c1(C(=O)NCC2CCC(NC(C3C(C=C)C3)=O)CC2)[nH]c2ccccc2c1CC C1(NC(C(C=CC)O)=O)CN(C(=O)CCc2ccncn2)CC1F C(=O)(C1=COCCC1)NC1(C(N2CCC(C(N)=O)C2)=O)CC(CO)C1 c1(C(=O)NCC2CCN2C(c2ccc3c(n2)NCC3)=O)c[nH]c2ccc(F)cc12 c1(-c2cn(CCN(C(c3cccnc3F)=O)CC)nn2)ccc(F)c(Cl)c1F C12CC(C13CCC3)NC(=O)C(CC)N2C.C(C)(C)N(C1CC1)CC(C)C N1(C(c2c(C)cccc2)=O)CCCC2CN(C(c3c(C)ccc(C)c3N)=O)CC12 C1(C(=O)NCC(C)N(C)C)CN(C(=O)CCOCCCOCCO)CC(C)(C)C1 c1(C(N2C(CNC(c3cc(O)cc(O)n3)=O)CC(O)C2)=O)c[nH]c2ncccc12 c1(CC(=O)NC)nsc2ccccc12.c1(N(CC)CC)ccc(C(=O)NC2CC2C)cc1 CC1CCC(C(N2CCOCC2CO)=O)N1C(c1ccc(C(F)(F)F)[nH]1)=O CC(C)CC(F)C(=O)NC1CCCC1NC(=O)CSCc1ccc(Br)cc1 n1(CC(=O)NCC2(NC(C(C)O)=O)CC2)ccc(=O)c([N+](=O)[O-])c1 CC(C)C(CC(=O)NCCCO)NC(C12CC(C(=O)OC(C)(C)C)(CO1)C2)=O Cc1nc(F)ccc1C(N1CCC(NC(C2CCC2)=O)C(F)C1)=O N1(Cc2cncc(OCC)c2)CCC2(CC1)CC2C(=O)Nc1cc(OC)ccn1 C(c1cncnc1O)=CC(=O)NC1(CNC(c2ccc(OC)nc2)=O)CC1 C1(C#N)(NC(=O)COC2(C)CN(C(C3N(CCC)CCC3)=O)C2)CCCC1 C12(C(N3CC(C)C(CNC(=O)C(O)C4CCC4)CC3)=O)CCCCC1C2(F)F C1(CCNC(C2(OCC)CCCSC2)c2nnnn2C)CCC(F)(F)CC1 C12(NC(C3C(CC)OCC3)=O)CCOC(CNC(c3cccc(N)c3)=O)(C1)C2 CN1CCC(CNC(=O)C(c2ccco2)NC(c2cc(C(F)F)[nH]n2)=O)CC1 C1(CNC(CN(C)CC)=O)(NC(=O)CCc2scnc2C)CCOCC1 CC1COc2c(C(N3CC4CC3CN(C(=O)CC3(O)CCCC3)C4)=O)cccc21 c1(N(C(C=C(CC)CC)=O)CC(C)NC(=O)C=CC2CCOC2)cccc(C)c1 C=C(C)C1CN(C(CC(=O)NCC(c2ccc(Cl)cc2)=O)=O)CCO1 c1(CN2CCC(C)(C(=O)NCCCN3C(=O)C=CC3=O)C2)c[nH]c2cccnc12 C(=O)(C1=CS(=O)CCC1)NC1C(NC(c2ccc(C#N)o2)=O)CCCC1 C1(NC(C(C)OCCN(C)C)=O)CCN(C(=O)CCc2cn[nH]c2)C12CC2 C1(C(=O)NCC2OCC(CNC(c3[nH]cc(CC)n3)=O)C2)COC(=O)N1C N1(C(c2cnn(C)c2Cl)=O)CC(C)(C)C(NC(c2cnn[nH]2)=O)C(C)(C)C1 c1(C(N2C3(CN(C(C4CC(OC)C4)=O)C3)CC2)=O)ccc2cccnn12 n1(CC)nnc(C)c1C(N1CCN(CC(C)NC(=O)C(C(=O)OC)OC)CC1)=O N1(C(C2C(OCC)CC2)=O)CCC(C(F)(F)F)C(NC(=O)C(F)CC2CC2)C1 c1(C(N(C2CN(C(C3CCN(C)S3(=O)=O)=O)CC2O)C)=O)c(F)cccc1Cl N1(C(C=CCC)=O)CCC(NC(C2CCCC(C)(C)O2)=O)C(F)(F)CC1 c1(C(=O)OC)ccc(OC)c(F)c1NCCCCCC1CCNCC1 C(=O)(N=c1[nH][nH]c2cccnc12)C1CCN(Cc2ccc(C)o2)C1 CN1C(=O)N(C)C(NC(=O)NOCC(F)F)C2=C1C(C)(C)N(C)C2=O C1(C(=O)NC2CCN(C)C2)COC2(C1)CN(Cc1ccccc1)C2.C1CO1 CC1(C)COCCC1OC(c1cnn(-c2ccccc2)c1N)=O C=CC(CC)CC(=O)NC1CN(C(c2sc(-c3ncc[nH]3)nc2C)=O)CC1F N1(C(C2CCN(CC)C2)=O)CCN(C(c2cccc(N)c2)=O)CC1CO c1(N(C)C)cncc(C(N2CCCC2(C)CNC(=O)CNS(N)(=O)=O)=O)n1 CC1(C)OCCC1CC(N1CCCC(CNC(=O)CCCn2cccc2)C1)=O C1(C(=O)NCCCOCCNC(c2c(=N)[nH]cnc2)=O)CCCS(=O)(=O)N1 N1(C(c2cc(C)ncc2)=O)CCN(C(=O)CCCCOC(F)(F)F)CC1C c1(CC)ccc(C(N2CCCCC2CNC(=O)CSC)=O)c(OC)c1 CCCC(C)CC(=O)N1CCC(N(CCC)C(c2cc(OC)nn2C)=O)CC1 c1(NC(C)=O)cccc(CC(=O)NC2CCCN(C(=O)C(F)(F)CO)C2)c1 C(=O)(C(C)CCC(C)(C)C)N1CCCC(CC)(NC(c2cc(F)ccc2C)=O)C1 C1(C(N(CC(CNC(c2cc(C)oc2C)=O)C)C)=O)CCC(=O)N(C(C)C)C1 c1(C(C(=O)NC2CC(NC(CN(C)CCO)=O)CC2O)O)cc(Cl)cc(Cl)c1 c1(C(F)F)cc2c(s1)CCCN(c1nccc(=NCCc3ocnc3CO)[nH]1)C2 CC(C)CC(C)(CNC(C1(c2ccsc2)CC1)=O)NC(C1CCCC(=O)N1)=O c1(C(N(CCCN(C(C(C2CC=CCC2)OC)=O)C)C)=O)cnccc1Cl c1(NC(=O)Nc2ccnn2CC2CCOC2)csc2ncccc12 c1(C(=O)NCC2C(CNC(=O)CCc3ccccn3)C2)cc2c([nH]1)CCCC2 C(=O)(C1=CCN(C(C2CC(=O)C2(C)C)=O)CC1)N1C(C)CSCC1 c1(N2CCC(NC(C3(SC)CCC3)=O)CC2C)nc(OCC)c2nc[nH]c2n1 N1(C(c2cc(SC)c(F)cc2)=O)CC(C)(C)OCC1CNC(=O)C(C)C(C)C C(C(C(=O)NC1CCN(C(=O)C(CC)C(C)C)C12CCC2)C(C)(C)C)OCC=C c1(C(N2CC(NC(C(COC)C)=O)C2)=O)cc(C)cc(Br)c1O c1(OC)ccc2c(n1)NC(C(=O)NC(C)CNC(c1ccc3n[nH]cc3n1)=O)C2 CN1CCOCC1C(=O)NC1CC(CC(=O)NCCC2CCC2)C1(C)C N1(C(Cc2cn(CC)nn2)=O)C2CCC1CN(C(=O)C(C)C(O)CC)C2 c1(SCC)ccc(CC(=O)NCC(C)(O)CNC(=O)C=Cc2ccc[nH]2)cc1 C1CN2CCN12.c1nc(C)ncc1Br.c1(C(COC)(C)O)ccccc1 c1(C(=O)NC2C(NC(c3c(OC)cncc3)=O)CCC2)cc(Cl)ncc1O C1(NC(CNC(CC)=O)=O)(NC(=O)CCOc2ccccc2)CC2CCC1CC2 CCC1=C(C(=O)NC(C)CN(C)C(c2cc(F)c(C3CC3)c(F)c2)=O)CCCO1 N1(C(c2c(C)n(C)cn2)=O)CCC(O)C(NC(=O)CN2CCCC2CO)C1 c1(C(=O)NCC(CC)NC(=O)COC2CC=CC2)cccc2cnsc12 C(=O)(C=CS(C)=O)NCC(CN(C(=O)CNC(=O)C(F)(F)F)CC)(C)C c1(C(N(CCNC(=O)CN2CCSCC2)C2CC2)=O)cc(F)cc2nccnc12 Cc1cc(CCCC(=O)NC(CNC(=O)CNC(C2CCC2)=O)C(C)C)c(C)s1 O=C(C1=C(Cl)CC1)NC1CCCC(C(=O)NCC(O)(C2CC2)C2CC2)C1 c1(C(C(=O)NCC(C)(C)CCc2nn[nH]n2)=O)ccc2c(c1)CCCC2N c1(CC)[nH]nc(C(N2CCC(C(C)NC(C3CCCO3)=O)C2)=O)c1Cl c1(C(=O)NCCC2CCCN(C(c3cc[nH]n3)=O)CC2)cc(F)c2cn[nH]c2c1 c1(-c2n(C(C3(C)CC3)C)nc(-c3cccnc3)n2)ccc2c(C#N)c[nH]c2c1 CCC(CC(=O)N(CCC(C)NC(c1cc(Cl)n(C)n1)=O)C)C(C)(C)C Cc1c(C(=O)NC2CC3CCC2N(C(C2(C)COC2)=O)C3)oc2ccccc12 C(=O)(CN=c1cc[nH]cc1)NC(c1cn(C)nc1)C(N1CCOC(C(=O)NC)C1)=O CCCC(O)C(=O)NCC1CCC1CNC(=O)Cc1cccnc1OC c1(C(=O)OC)cn(CC(=O)NCC2CC(NC(=O)C(C)n3cncn3)C2)nn1 c1(C(=O)NCC2(C(=O)OC)CCOC2)ccc2c(=O)c3ccccc3sc2c1 C1(CC=C)(NC(=O)C=CCO)CCN(C(=O)CC(C)Nc2ccc(F)cc2)C1 C(=O)(N=c1[nH][nH]c2ccccc12)C1CN(Cc2cccc(-c3c(N)cccn3)c2)C1 C#Cc1c[nH]nc1C(=O)NC(CO)C(=O)N1CCCC1CNC(N)=O CSC1=C(C(=O)NC23CCCC2CN(C(=O)CC2CCCCN2C)C3)CCCC1 c1(SCC(N2CCC(F)(CNC(=O)CCc3cnco3)C2)=O)cc(F)ccc1F C(=O)(CC(C)(C)C(C)=O)N1C(CN(C(C2CCCC(OC)C2)=O)C2CC2)CCC1 C1(C(N(CCN(C(c2ncncc2C)=O)CC)CC)=O)CCC2CCC(=O)N12 N1(C(C=C(C)Cl)=O)CC(NC(=O)C2=C(Cl)CC2)C(C2CC2)C1 C(CC(=O)NCCC(C)N(C)C(c1cnc(C(C)C)s1)=O)(C(C)C)OCC C1(OC)C(OC)CN(C(c2csc(-c3ccoc3)n2)=O)C1CNC(=O)C(C)O C1(C(=O)NC(c2ccc(O)cc2)C#C)CC(=O)N(C(C)(C)C)C1 c1(C(=O)NC2(CCNC(C(C)n3ccnc3)=O)CC2)csc2nccn12 O=S(=O)(c1ccc(NCc2ccccc2CO)c(F)c1)NCC1=CCCOC1 N(C(=NCCCF)NC1CC(C)Cc2ccccc21)C(C(CC)CC)CO c1(CCC)noc(CNC(=O)NCC2CCCN2C(=O)C(F)(F)F)n1 c1(CN2C(CNC(=O)CCc3nncs3)CC2)cccnc1 c1(NC(c2c(C)oc(S(C)(=O)=O)c2)=O)cccc(S(=O)(=O)C(F)F)c1 C1(CNC(C(C)O)=O)CC2(CCC2)CN1C(=O)C(O)C(F)(F)F C(CN=c1[nH]c2c(c(=NC3C=CC(C)(C)CC3)[nH]1)CCC2)c1c(C)ccc(C)c1 N1(C(c2cccc(C3(C)CC3)c2)=O)CCC(C(=O)NS(=O)(=O)C2CC2)C(CO)CC1 CC(C)(C)CCCC(=O)NC1CC(N2CCC2)C1.C12CCCC(CC1)C(=O)N2 C(=O)(CN=S(C)(C)=O)NCCC1CCN(C(c2ccn(C(CC)CC)n2)=O)C1 N1(C(C(C)=C(CC)C)=O)CCC(NC(=O)CC2CCN(CC(F)F)CC2)C(C)C1 C1(CC(=O)NC2(COC)CCCC2)C2CCCC2N1C(=O)C(C)CC(F)F N1(C(c2c(COC)c[nH]c2)=O)CCOC(CCNC(=O)CCc2ncnn2C)C1 c1(-n2c(C)cc(C(=O)NCC(C)OC(F)F)n2)ccc(C#N)cc1 CC(C)CC(O)C(C)C(=O)OCSC1(C)CCN(C(=O)OC(C)(C)C)C1 OC1CCCC1CCCn1nnnc1C(OC(F)F)C1CC1 Nc1ccc(C(N2CCC(CNC(=O)C(c3ccccn3)O)C2)=O)c(O)c1 C(C)(C)(C(C(=O)O)NC(C1CCC2(CC2)C1)=O)OC C1(NC(CN(C)C2CC2)=O)CC2CCC(C1)N2C(C1CCN1C1CCCC1)=O C1(CNC(C(C)(C)n2cnnn2)=O)CCN(C(=O)Cc2csc(=N)[nH]2)C12CCC2 C1(CC=C)(NC(C2CCS(=O)(=O)N2)=O)CCCN(C(=O)CCc2ncc[nH]2)C1 Cc1nc(C(=O)NC2(CNC(C3CCN(C)C3=O)=O)CC(F)(F)C2)c(C)o1 C1(C(N(C(C)CNC(C2CCNC(=O)C2)=O)C)=O)CC2(C1)CC1(CC1)C2 c1(C(N2CCCC(N(C(=O)CSc3nc[nH]n3)C)C2)=O)cnn2c1CC(F)(F)C2 N1(C(c2[nH]cc(C)c2)=O)CCCCC1C1(NC(c2n[nH]c(C)c2F)=O)CC1 c1(C(N2CC(C(C(=O)NC(CC)C3CCC3)O)C2)=O)ncccc1N c1(-c2c(C(=O)NCCN(C(c3cccs3)=O)C3CC3)[nH]cc2)ccc(F)cc1 C1(C(=O)NCC(C)N(C(=O)CCn2cc(C)cn2)CC)CCN(C)C1=O C(CN=c1nc(N2CCCC(COCCOCC)CC2)c2c([nH]1)CSC2)=CC C1(NC(Cc2cc(C)on2)=O)CC(N=c2[nH]c(Cl)ncc2C(N)=O)C1(C)C Cc1noc2ncc(C(=O)NC3CC4CC(NC(=O)C(Cl)=CCl)C4C3)cc12 C1(CC(=O)NC2CCN(C(c3c(CC)ncs3)=O)C2)CCC(C)(C)CC1 c1(CC)noc(C)c1C(N1CC(CO)(NC(c2cncn2CC)=O)C1)=O C#CCCCCCC(=O)N1CCC(C)(C)C1CNC(=O)CC1CC(C)(C)CO1 c1(C(CC(=O)O)CNCCCc2cccs2)ncc(Cl)cc1Br c1(NSc2ncc(CC)s2)cc(N2CCN(CCOC)CC2)nc(C)n1 Cn1nnc2cc(C(N3CCCN(C(c4ccoc4)=O)C(CO)C3)=O)ccc12 CCCC(C(=O)N1CCN(C(C2CC(=O)NC2(C)C)=O)C(CCO)C1)S(N)(=O)=O C(=O)(CCC(=O)NCCOCCCN(C)C(c1cc(Cl)cn1CC)=O)NCCC c1(C(N2CCC(O)(CCNC(C(C)C(F)F)=O)C2)=O)c(F)cc(F)cc1F N1(C(C(C)C2CCCO2)=O)CCC(C(=O)NCCC(C)(F)F)=C(F)C1 C(=O)(C#CC1CC1)NCC(C1CCC1)NC(CCCOCCC)=O c1(C(N2CCC(CNC(CSc3n(C)nnn3)=O)C2)=O)ccnc(N2CCC2)n1 Cn1ccc(COCC(=O)NC(c2ccccc2)c2cccs2)n1 N1(CCCC(=O)NCC(CO)NC(c2n(CC#C)ccc2)=O)C(=O)CN(C)C1=O C#CCCCCC(=O)NCC1CC(C)(C)CN1C(c1ncnc(C)c1C)=O C1(NC(Cc2nnc(C)o2)=O)CC2CC1N(C(c1n[nH]cc1Br)=O)C2 C1(CNC(CC2(O)CCCN(C)C2)=O)N(C(=O)Cc2cn[nH]c2)CCCC1(C)C C1(CC)CCCCC1NC(=O)CSCC.C12(CCCC1)c1cn(nn1)CCO2 C1(NC(CCCNC=O)=O)C=CCN(C(c2cnn(-c3ccccn3)c2N)=O)C1 C1(NC(C(Cc2ccc(OC)cc2)O)=O)CCN(C(c2cocn2)=O)CC1F c1(CNC(C(N2CCC(N3CCCC3=O)C2)C)=O)cc(C#N)cs1 CC1(C)CCCOC1C(=O)NC1CC(C(N2CC(n3ccnn3)C2)=O)C1 c1(C(=O)NCC(C2CC2)NC(C(COC)C)=O)c(Br)nc2n1CCCC2 c1(OC)cccc([N+](=O)[O-])c1CN1CC2CC1CN2C(c1cc(Cl)cc(Br)c1)=O c1(C(=O)NC2CC(C)CN(C(=O)C(C3CCCCC3)C)C2)cnn2cccc2c1 C#Cc1cn(C)nc1C(=O)NCC1CCCN1C(=O)C(=Cc1ccccc1)CC C#CC1(NC(=O)C(CC=C)NC(C2CC2CC(C)(C)C)=O)CC(F)(F)C1 C1(CN(C(=O)C=Cc2cn(C)nn2)C)COCCN1C(=O)CC1C=CCCC1 c1(C(=O)NCC2CC(NC(C(=O)NC)=O)C(O)C2)cc(C)n(C)c1C C1(O)(CCNC(C=CCOC)=O)CCN(C(=O)CNC(=O)C=Cc2nccs2)C1 c1(CN2CC(C)(C(=O)NCC3CCCO3)C2)cccc(O)c1O c1(OC)cccc(Cl)c1C(N1CC(Nc2cc(C(F)F)ncn2)CC1C)=O C1(CNC)CCCCN1C(=O)CC1C(=C2OCCCO2)CCC1 C1(C(N2CC3COCC3C2)=O)CCC(O)CN1C(=O)CC1CCCC2CC12 C#CCCC(=O)NN1CCCC1C(=O)NCc1ccc(C(N)=O)cc1 N1(C(C(CC)OC)=O)CC(NC(C2(CC(C)C)CCNC2=O)=O)C(C)C1 C#Cc1ccnc(C(=O)NC2CC(C(=O)NOCC(N)=O)C23CCC3)c1 C1(NC(c2scc(C)c2)=O)CCCCC12CCN(C(c1ccc[nH]1)=O)C2 c1(C(=O)NCC(C2CC2)NC(c2cc(C(C)(C)C)no2)=O)cnn2ccsc12 C1(NC(CS(CC)=O)=O)CC2CCC1N2C(c1c(C)ccn1C)=O N1(C(CSC2CCN(C)CC2)=O)CC2(CCC2NC(=O)CS(=O)(=O)N(C)C)C1 C12(CNC(C(C3CCCCC3)C)=O)CC(NC(=O)Cc3csc(=N)[nH]3)(C1)C2 CCC(N=c1[nH]c(=NC2COc3ccc(F)cc32)[nH]c2c1COCC2)c1cccs1 Cc1cc(=O)cc(C(=O)NCC2CCC3(CCC3)O2)n1C c1(CC(C)NC(c2cc(C(C)C)[nH]n2)=O)ccccc1Br CCC(CC)(CO)C(=O)N1CCCC(CC(=O)NCCCn2cncn2)CC1 N1(C(c2c(CC)nco2)=O)CC2CCCC(C1)N2C(C1CSC(C)=N1)=O C=CC1(C(=O)NCc2cnc(C)c(C)c2)CCN(C(C2CC(=C)C2)=O)C1 C1(NC(C(CC(C)C)C)=O)CN(C(c2cccc(CC#N)c2)=O)CC(F)(F)C1 N1(C(C(C2CC2)OCC)=O)C(C(=O)N(CC(c2nn[nH]n2)C)C)CC2CC12 c1(OC(C)C)cc(-c2nc(C(C)C)nn2-c2ccc(F)nc2)cc(Cl)n1 c1(CCC)cc(C(=O)N(CCOC)CCNC(=O)CCc2cccc(C)c2)n(C)n1 CCCC(CCCNC(c1cc(C(N)=O)[nH]n1)=O)NC(c1ccccc1COC)=O Cc1cc(CCCOC(C2(NC(=O)OC(C)(C)C)CCOC2)=O)cc(C)c1.C(C)(C)S C1(C(=O)NC2CC(C(N(C(C(C)SC)C)C)=O)C2)(N(C)C)CCCC1 c1(CC(CNC(=O)Nc2cnn(-c3cccnc3)c2)OC)ccc(F)cc1Br N1(C(c2c(Cl)csc2Cl)=O)CC2CC(Nc3ccc([N+](=O)[O-])cc3)CC1C2 c1(COC)nc(N2CC(O)(C(C)NC(=O)C)C2)cc(O)n1.c1(C2(C=O)CC2)cccs1 CN1CCC(F)(C(=O)NCc2ccc(N(C)C(N)=O)cc2)CC1 c1(OC)cc(C(=O)NC2CC2CNC(=O)CNC(=O)CC(C)(C)C)cc(F)c1F C12(C(=O)NCCC3CN(C(=O)CC(F)(F)F)C3)OCCCC1C2(F)F C(c1ccc(C2OCCO2)o1)=CC(=O)NCC(CO)NC(=O)C=CC1CCCC1 C12(NC(c3cc4n(c3)CCCNC4=O)=O)CCCC1N(C(=O)C1CC1)CCC2 c1(C(=O)NC2CC(C)(NC(C3CC3F)=O)C2)cccc(OCCF)c1 C(=O)(CCC(=O)NC(C)CC1(O)CCN(C(=O)C2=CCCS2)C1)OCC CCCCC(C(=O)NC1CC(NC(c2cn(C)ccc2=O)=O)C1)NC(N)=O c1(C(N(C2CCN(C(c3c(C)ccnc3)=O)C2)C)=O)cc2c(F)ccc(F)c2[nH]1 C(=O)(CCCC(F)(F)F)N1C(C(N(CCCC)C)=O)C(CC)CC1 Cc1nn(C)cc1CC(N1CCCC(C(N2CC=CC2C(=O)N(C)C)=O)C1)=O c1(C(CC)C(=O)NCCC(O)CNC(c2ccnn2C)=O)ccc2c(c1)OCO2 C(=O)(C(C#N)CCC)N1CCC(CC#C)(C(=O)NCc2ccccc2F)C1 C12(C(N(CCN(C(=O)CS(C)(=O)=O)C)C)=O)CCOC1CC(=O)NC2 c1(C(N2CCSCC(C(=O)OC)C2)=O)ccc2nonc2c1 C(=O)(C#CC1CCOCC1)N(CCC(=O)NCCN1CC(CF)C1)C C=CCCCC(C)NC(C1CSCCN1C(=O)C(C)SC)=O C(c1c[nH]cn1)=C(C(=O)N(CC(C)N(C)C(c1cnc(O)s1)=O)C)F N1(C(CC(C)OC)=O)CC2CCC1CN2C(=O)CC(COC)COC c1(CNC(=O)NC2C3(CC(OC)C3)C2)n[nH]c2c1CC(C)CC2 C=CCCC(C(=O)N(C)CC1OCCC1(C)C)NC(c1ccc(CO)o1)=O C1(C)(NC(C2CC(SCC)C2)=O)CC(NC(C2CN(C(=O)OC(C)(C)C)C2)=O)C1 c1(OC)cc(C(=O)NCCCCC(C)NC(=O)CN2CCCNC2=O)ncn1 Cc1nc(O)nc(S)c1C(=O)NCC(CC(C)C)NC(=O)Cn1ccnn1 N1(C(CN2C(C(N3CC(CC(C#C)C)C3)=O)CC(O)C2)=O)CCc2sccc2C1 C(=O)(C(C(C)C)C(C)C)NCCC(C)(C)NC(c1cc(C(=O)OC)c(O)cc1)=O C(=O)(CC1=CCCCC1)N1C(CNC(C2CSCCS2)=O)CCC1 c12nnc-1n2CC(C)C.N1(C(C(=O)NCCSC)C)CCOCC1 c1(OC)ccc2c(c1)C(C(=O)Nc1c(F)c(F)c(F)c(F)c1F)CC2 N1(C(C2CCC(CC)CC2)C(=O)NC)CC(C)c2ccccc21 N1(C(C)=O)CCCC1C(=O)NC1C=CC(CO)C1.c1(C=O)cscc1C1CC1 N1(C(Cc2ccn(CC)n2)=O)CC2CC2(C(=O)NCCC(=O)OC)C1 c1(C(=O)NCC2CN(C(CCNC(N)=O)=O)CC2O)nccc2c1NCCC2 N1(C(C2CCC(C(F)(F)F)CC2)C(=O)NCC=C)CCC(O)CC12CC2 C=CCC(C(=O)NOC(CC(C)C)C(=O)N1CC(n2ccnn2)C1)C(F)(F)F CC(=O)CCCCCCC(=O)NC(c1ccccc1)CNC(=O)Cc1nc[nH]n1 c1(C(=O)NCc2c(C(N(C)CC3CCCO3)=O)n[nH]c2)ccc(F)cc1F Cc1cc(Br)ccc1C(N1CCOC(CC(=O)NCC2CC(C)(C)C2)C1)=O C1(CNC(=O)Cn2cnnn2)CCN(C(c2cn(CCO)nn2)=O)C12CC2 C12CN(C(c3cc(C4CC4)[nH]n3)=O)CCC1NC2=O.c1(CC)ccccc1OC CCC(C)C(=O)N(C(C)CNC(=O)CC(C)C1CC1)CC c1(NC(C2CSC2)C)ccnc(C2CC2)c1 c1(OC)c(N)cc(C(=O)N(CCO)C2CC2)cc1Br CC(C)CC(C)C(=O)NCc1nc(C(=O)NCC2CCN(C)C2)co1 N1(C(C(C)n2cncn2)=O)CC2CCC1C(CNC(C1COC3COCC13)=O)C2 C1(C)(CC)C=C(C(=O)N2CC3C(CNC(c4cccc(O)c4Cl)=O)C3C2)C1 N1(C(CCC#C)=O)CC(NC(c2ccccc2C2(C)CC2)=O)Cc2ccccc21 Cn1ncc(Cl)c1CNC(=O)C(CNC(c1coc(CO)c1)=O)CC1CC1 c1(N2C3CC(CNC(C(C)(C)F)=O)C2CC3)ccc2nccnc2n1 CC1CC2CN(C(=O)NCCS(=O)(=O)C3CC3)CC2N1 c1(C(C)SCC(=O)NC23CC(CNC(CC(C)C)=O)(C2)C3)ccc(F)cc1 c1(CC(N2C(C)CC(NC(c3nnc(C)s3)=O)C2)=O)cnc2cccnn12 c1(CCCC2CCC2)ncc(C(=O)NCC(C(=O)C(C)NC)OC)[nH]1.C(C(C)C)O C1(NC(C(N2CCCC(O)C2)C)=O)CC2(C1)CN(C(c1ncccc1Cl)=O)C2 c1(SC)ccc(N)cc1C(N1CCN(C(C2CC2(C)Br)=O)CC1C)=O N1(C(C2CC(=O)OC2)=O)CCN(C(=O)COCc2ccc3c(c2)CC3)C(CO)C1 N1(C(CC2(CC)CCC2)=O)CCCC(C(=O)NCC(O)C(F)(F)F)C1 CC1(C(=O)NC(CO)C(C)NC(=O)C2=CCSC2)Cc2ccccc2NC1=O c1(N2CC(CNC(c3cc(F)c(F)c(F)c3)=O)OCC2)ncnc2c1COC2 N(C(=NCCCCl)NCc1ccccn1)C(C1CCCO1)C N1(C(C2CN(C(=O)OCC)C2)=O)CC2CCC1CN(C(c1[nH]nnc1C)=O)C2 N1(C(C(C=C)(C)CC)=O)CC(NC(c2coc(COC)n2)=O)CC2(CCC2)C1 c1(C(=O)NCCNC(COCCOCC#C)=O)c(F)cncc1Br c1(C(N2C3CN(Cc4cn(CC(C)C)nc4)CC2C3)=O)cccn2cncc12 c1(C(C)C)ccc(C(O)C(=O)NCC#CCNC(C2CC(O)C2)=O)cc1 N1(C(c2nscc2Br)C(=O)NCc2c(OC)cccc2)CCc2nn[nH]c2C1 C(Cc1ccco1)(C(=O)NCc1ccncn1)NC(C1C(C)(C)C1)=O N1(CC)CCN(C(C2CC(C)CN(C(=O)CN=[N+]=[N-])C2)=O)C(C)C1 C(C(CC(C)C)C(=O)N1CCC(CNC(c2sc(C)c(C)c2C)=O)C12CC2)OC C1(NC(C(C2CCN(C(c3cc(C)nc(C)n3)=O)C2)F)=O)Cc2ccccc2C1 N1(C(c2n(C(C)(C)C)ncc2)=O)CC2CN(C(=O)CC3CC4CCC4C3)CC(C1)O2 C(C(C)(C(C)C)NC(=O)C(C)c1cc[nH]n1)NC(C(c1cn(CC)nc1)=O)=O C#Cc1ccc(F)cc1C(=O)NC1CC1CNC(=O)C1=CCCCC1C Cc1cnc(C(=O)NCC2CCC2NC(C2(F)CCOC2)=O)cc1Br c1(NC(C2CSCCN2C(c2ccc(O)cn2)=O)=O)ccn2nccc2c1 C#CC1CCCN1C(c1ccc(C(=O)NC)cc1)C(=O)N(CC)Cc1nccs1 c1(C(=O)NC(CC)(CNC(=O)CN2CC3CCC2C3)CC)ccsc1S(N)(=O)=O c1(C(N2C(CN(C(=O)C(F)C3CCC3)CC)CCC2)=O)ccc(C#N)cn1 Cn1nc(Cc2nc(C3CC3)no2)c2ccccc12.N12CC3CN(CC3C1)C2=O N1(C(C(CC)(C)F)=O)CCC2(CC1)CCN(C(c1sc3nccn3c1C)=O)C2 N1(C(C(C)C2CCCO2)=O)CCC(C(CO)NC(=O)Cc2csc(=N)[nH]2)CC1 c1(CCC(=O)Nc2cccc(NC(C3CCS3(=O)=O)=O)c2)cccc(Cl)c1 C1(CCCC)CN(C(c2cnsc2C)=O)CCN1C(C1C(F)(F)C12CC2)=O CCC(C)CCCCC(=O)NC(CC(=O)N1CCSCC1)CC(C)C C(CCCN=c1[nH]c(=NC2CCNC(=O)CC2)[nH]c2cccc(F)c12)=CC c1(C(C(=O)NC2CC2)N(N2CC(OCC)C2)C)ccc(C(F)F)c(F)c1 c1(NC2CCCCN(C(C(CC)F)=O)C2)ncn(C)c(=O)c1Br N1(C(C(C)OCC)=O)CCN(C(=O)Cc2cnc[nH]2)CC1c1ccccn1 C1(CNC(=O)NC(C)(C(F)(F)F)c2ccccc2)CCC2COCCC2C1 CC(C)(C(=O)NCC(=O)NC1CC1c1c(C#N)c(=O)n(C)c(=O)o1)C1=CCSCC1 C(CCCCN=C(NCc1cnn2ccccc12)NCc1ccco1)SC CCC(C(=O)NC1C=CC(CNC(C2CC(n3ccnn3)C2)=O)C1)C(C)O C1(C)(NC2(CC(N3CC(C(O)C(=O)OC)C3)=O)CCCC2)CC2CCC1C2 N1(C(c2ccc(OC)nc2C)=O)CC(NC(=O)C(C)C)CC12CCCCC2 C1(C(=O)NC2CC(CNC(c3n(CC)ccc3)=O)C2)CC(c2cccnc2)=NO1 c1(C(=O)NC2(CO)CCCN(C(C(C)(C)OC)=O)C2)ncc(F)c2ccccc12 C1(C(N(CCCF)C)=O)CC(=O)N(c2ccccc2Cl)C1 c1(C(C)C(C)COc2ccc(F)c(Cl)c2)n[nH]c(=NCCCn2cnnn2)o1 C=CCC(C(=O)NCCCC(C)(C)NC(C1CC12CC2)=O)NC(C)=O C1(NC(CCOCCN=[N+]=[N-])=O)COCC1CC(=O)O c1(C(N2CCC3CN(Cc4c(F)cccc4Cl)CC23)=O)ccc2ncccc2c1 c1(CC)cc(C(=O)NCCC2(NC(c3ccc(F)s3)=O)CCCC2)ccc1Cl N1(C(C(C)CO)=O)CCCC(F)(CNC(C2CCCC(C)C2)=O)C1 C(C(C)NC(=O)CCCC1CCCC1)(C(C)C)NC(CCc1c(C)ncs1)=O C1(C(N(C)CCNC(C2CC(C)(C)CO2)=O)=O)CN=C2N=CNN2C1 CCC(CC(=O)NCC12CC(C1)C(NC(c1nc(O)sc1C)=O)CO2)C(C)(C)C C=CCCCC(c1nnnn1CCCSC)NCc1ccccc1CC Cc1ccc2oc(CN(C=O)Cc3cccc(Br)c3F)cc2c1 C1(NC(c2ccc(Cl)cc2)=O)CCC2(C1)CN(C(c1ccnc(F)c1Cl)=O)C2 C1(CC=C)(NC(=O)C(CCC)NC(C)=O)CCN(C(=O)C(=O)NCCOC)CC1 c1(C(C)C)ccc(C(c2nnnn2C2CCCCC2)NC2CCC2(F)F)c(F)c1 C(=O)(C1Cc2c(Cl)cccc21)NC1(CNC(CCSCC)=O)CCCCC1 C#CCCC(O)C(=O)N1CCC(CNC(=O)COc2ccc(F)cc2OC)C1 C1(CCNC(C2(C#C)CC2)=O)CCCN1C(=O)CCN1CCOC1=O N1(CC(=O)NCCCC(=O)NCCN2CCNC(=O)C2)C(=O)CCCC1=O c1(C(N(CC(C)N(C)C(C2(C)CCCN(C)C2)=O)C)=O)cn(C)c(=O)n1C Cc1ccccc1CCC(N1CCC(CNC(C2CC2c2ccccc2)=O)C1)=O NC(=O)CC(O)C(=O)N1CC(CNC(=O)CSCc2ccccn2)C1 N1(C(C=CC(=O)N(C)C)=O)CCC(O)CC1C(=O)NCCN1C(=O)CCC1=O N1(C2CC3N(C(C4CC(O)C4)=O)C(CC3)C2)CC(C2CCCCC2)C1 c1(C(=O)NC2CC(NC(C3C(CC)OCC3)=O)C2)cc2ncccc2o1 C1(NC(c2nc(CC)oc2)=O)CCCCN(C(=O)CC2CCCN(C)C2)C1 c1(C(=O)NC(CC2CCN(C(CCCOC)=O)CC2)C)csc2cccnc12 C(C(=O)NCC(C1CCC1)NC(=O)Cn1ccnn1)(C(C)C)OC Cc1cccc(F)c1C(=O)N(C1CC(NC(c2cc(O)cc(O)c2)=O)C1)C C=CCC(C(=O)NCC(=O)N(C)NCC(C)C)C(C)C.CC c1(CNC(c2cc(Cl)ccc2F)c2n(CCSC)nnn2)c(C)cnnc1O C12(C(N3C(CN=[N+]=[N-])CCC3)=O)CCC(NC(C3CC4(CCC4)CO3)=O)(CC1)C2 c1(OC)ccc(NC(=O)C=CCNC(=O)CSC(F)F)cc1N1CCCCC1=O c1(C(C(=O)NC2CCC(NC(C3(SC)CCC3)=O)C2)(C)C)cccc(C(F)(F)F)n1 C12(NC(CCCNC(=O)OC)=O)CCOCC1CN(C(=O)CC1(N(C)C)CC1)C2 Cn1cc([N+](=O)[O-])c(OCC(=O)NC23CCSC2CCOC3)n1 C1(C(N2C3C(NC(C(C)OCC)=O)CC(CC3)C2)=O)CC(C)c2nc(C)cn2C1 c1(C(=O)NCCC2(NC(C3C(C)OCC3)=O)CC2)cc(F)c(F)c(O)c1F c1(OC)ccc(Cl)c(-c2cn(CC(F)CCNC(=O)C(C)CC(F)F)nn2)c1 c1(NCc2ccc(C)cn2)ccc(OC(C)C(=O)O)c(F)c1 c1(C(N2CC(CCNC(C(CC)C(=O)OC)=O)C2)=O)cc2c(nn1)CCOC2 C(CC)(C(=O)NC1CC(C)(NC(c2cnc(O)o2)=O)C1)OCC Cc1nc(-c2nc(-c3ccc(C(F)(F)F)cc3)nn2CCS(N)(=O)=O)oc1C N1(C(c2[nH]cc(C(N)=O)c2)=O)CC2CC2C1CNC(=O)CCN1CCCS1(=O)=O C1(CNC(c2n(CC)ccc2)=O)(NC(=O)CCOC)CC2CCC1C2 c1(C(N2CCC(O)(CNC(c3onc(C)c3C)=O)C2)=O)ncnc2ccsc12 c1(C(=O)NC(CC2CC2)C(=O)NCCn2cnnn2)nccc2[nH]ccc12 N1(C(CC)=O)CCOC2(C1)CN(C(=O)C(C)(C)C)C2.Cc1nc(C(=O)OC)c(=O)[nH]c1C N1(C(C(C)(C)C)=O)C2CCC1C1CC1(NC(c1ccn3c1CCC3)=O)C2 c1(N(C)C)cccc(C(=O)NCC2(NC(=O)C(F)C3CCC3)CC2)n1 C1(C(=O)NC2C3CN(C(COC4CN(C(C)=O)C4)=O)CC32)CCCCC(=O)N1 c1(C(=O)NC)cccc(C(=O)NC2CC2CNC(c2cc(C)c(Br)o2)=O)n1 C#CC1CCCN(C(c2cccnc2CNC(=O)CC(C)C=C)=O)CC1 C1(CNC(C=C(CC)CC)=O)CN(C(c2cc(Cl)nnc2Cl)=O)CCC1(C)C C1(C(=O)OC)CCC2(CCN(Cc3cc(C4CCCC4)no3)CC2)C1 CCCCC(C(=O)N1CCCC1CNC(=O)Cc1csnn1)NC(N)=O c1(OC)cccc(CNC(=O)C(F)CC2CN(C(c3cc(C(C)C)no3)=O)C2)c1 N1(C(C(CC)C(=O)OC)=O)CC(C2CCCN(C(C3CCCC3)=O)C2)C1 C1(NC(CSC)=O)CCN(CCCN(C)C)CC(C)(C)C1.C12(C)CC(C1)C(=O)N2 N1(C(C(C)(C)C(F)F)=O)CC2(NC(=O)COc3cc(F)cc(F)c3)CCC1CC2 c1(CC)o[nH]c(=NC(=O)c2cc(C(C)C)on2)c1C CC(CCc1ccc(F)cc1)C(=O)NC(C1CN(C(c2ccsc2Cl)=O)C1)C Cc1cc(C(=O)NCC2(CNC(c3c[nH]ccc3=O)=O)CCC2)ccn1 C(=O)(CCC(C)(C)C#N)N(CC(C(=O)NC(C)Cn1cncn1)(C)C)C C1(C(=O)NCC(C2CCCO2)C(C2(n3cncn3)CC2)=O)CCC([N+](=O)[O-])CC1 N1(C(=O)CC2OCCO2)CCC2CC2(C(=O)Nc2ccc3c(c2)OCC3)CC1 c1(CCC(=O)NC2CCC2CNC(C2(c3ccc(F)cc3)CC2)=O)cccc(O)c1 C(=O)(CC(C)(C)CC)NC1(C(N2CCN(C(CC)C)CC2)=O)CSC1 C12CCN(CC1C)C2=O.C1(C(=O)NC(C(C)F)C)CCCC12CCC2 N1(C(=O)N(C(C(=O)OC)Cc2ccc(F)cc2)C2CC2)CCOCC1(C)C1CC1 C=CC(C)(C)CC(=O)N1CCC(N(CCO)C(c2sccc2OC(F)F)=O)CC1 c1(NC(C2N(C(c3ccccc3)CC)CCCC2)=O)ccn2c(C)cnc2c1 C1N=C2NN=C(S2)Cc2nc1cs2.C1(CO)CCCN(NC(C2CC23CC3)=O)C1 N1(C(CCC2CC(OC)C2)=O)CCOC(CN(C)C(c2csnn2)=O)C1 c1(C(=O)NCC2(F)CC(NC(c3cnc(OC)nc3)=O)C2)ncc2ccccn12 N1(C(C2C(C)(C)COCC2)=O)CCC2(C1)CN(C(c1cccc(F)c1C#N)=O)C2 c1(C(CNC(=NCC)NCCCC(=O)N2CCCCC2)O)cc(F)cc(F)c1 C1(CNC(C2CN(C)C(=O)N2)=O)CN(C(=O)CN2CCC2)CCC12CCOCC2 CS(=O)(=O)C1(NC(C2CC(n3cc(C4(CO)CC4)nn3)C2)=O)CC(=O)C1 C(=O)(C(C)(C)CCCC(=O)NC1(CCCNC(c2ccc(O)nc2)=O)CC1)OC CCC(C)C(O)C(=O)N1CC2C(NC(c3cc(CC)ccc3N)=O)C2C1.C(=O)OC Cn1c(O)nc(N2CCCC2CNC(=O)Cc2ccc(Br)cc2)cc1=O C1(CC)(NC(=O)CCc2nc(O)n[nH]2)CCN(C(=O)CN2CC3CCC2C3)CC1 C(C(CC(C)C)C(=O)NCC1CCC(NC(c2ccc3nsnc3c2)=O)C1)OC C1(CN(C(C)C#C)C(=O)OC(C)(C)C)CCC(NC(=O)CN(CCCC)C)CC1 C(C(C)(C)CC(=O)N1CCC(O)(CNC(=O)C(C)SC(C)C)C1)OC C(CC1=CCN(C(C2CC2CC)=O)CC1)NC(c1c(CC)nn(C)c1Cl)=O CC1CC(O)CN1C(=O)CCN(CCCO)C(c1cccc(Cl)c1)=O Cc1c(N(C(=O)Cn2cc(C3(O)CC3)nn2)C)cccc1F C(CCC(=O)NC(C1CCCN1C(=O)CSCC1CCCO1)(C)C)OCC Cc1ncsc1C(N1CCCC1C(C)(C)CNC(C1(O)CC1(C)C)=O)=O Cc1c(NCC(C)SCCCCc2nccs2)ncnc1Nc1cccs1 Cc1cc(C(=O)NCCC(O)CNC(=O)CCC2CC(F)(F)C2)ccc1[N+](=O)[O-] c1(NC(=O)CC2CCC(NC(=O)COCC3CC3)C2)cccc(O)c1 c1(C(=O)NC2CC(C)(COC)N(C(=O)C(C)C)C2)cc(F)cc2cnccc12 C1(C(=O)NCCc2cnc(C)o2)CCCCCCCC1 c1(C(C)C)cccc(C(N2CCCC(CN(C(=O)C(O)c3cnc[nH]3)C)C2)=O)c1 CC(C)S(=O)(=O)C(C)C(=O)NCC(=O)NCc1cn(CC2CCCC2)nn1 C1(CCC(=O)NCC2CC(CC)C2)CCCN(C(C2(CC(C)C)CC2)=O)C1 C1(n2cc(-c3scc(C)c3)nn2)CS(=O)(=O)C1c1ccccc1 C(=O)(C1CCCc2c1ncn2C)N1CCC(C)(CNC(CC(=O)OC)=O)CC1 N#Cc1cccc(CC(=O)NC2CCCN(C(=O)C=Cc3cncc(F)c3)C2)c1 c1(CC(=O)N(C(C)CNC(C2CC(N3CC(O)C3)C2)=O)C)ccccc1[N+](=O)[O-] N1(C(C2N(CC)CCOC2)=O)CC(NC(=O)C2=C(C)CCC2)CC12CCC2 c1(CC)ccccc1C(=O)N(CCC(=O)OC(C)(C)C)C(C)CC1CCNC1=O C(CCCCC(=O)NC1CCCCC1N(C)C)N(C(=O)C=CCN1CCCC1)C C=C1CC2(C1)CC(C(=O)NCC1(F)CCN(C(C3CCCN(C(C)C)C3)=O)C1)C2 CC(C)N(O)C(=O)C(=O)NC1(C)CC(NC(C2CCC(CCO)CC2)=O)C1 C1(C(N2C(C)(CCC)CC2)=O)CC(NC(c2cnsc2)=O)C12CCC2 N(C1=NCC(C2CCCOC2)N1C)C(CC)CNS(C)(=O)=O Cc1coc(C)c1Cc1csc(NC(=O)C(=O)NCc2ccccn2)n1 N1(C(c2c(C)cc(F)cn2)=O)CCCC2(CCN(C(C3CC(F)C3)=O)C2)C1 N#CC1(C(=O)N(CCC(=O)NCC2(n3ccnn3)CC2)C2CC2)CCOC1 C1(CC(=O)NCC2COCC2NC(c2snnc2C2CC2)=O)CC2C=CC1C2 C1(CNC(C2OCCN(C)C2)=O)CCN(C(=O)CN2CCOC2=O)C1(C)C N1(C(c2nc(C)[nH]n2)=O)CCC2OCCN(C(c3ccc(Cl)s3)=O)C2C1 c1(NCC(=O)N(CC(CC)NC(C2CCOCC2)=O)C)ccccn1 C1(C(=O)OC)(CC)CCCN(C(C2CN(C3CCC3)C2)=O)C1.N12CCCC1C2=O C1(F)(C(N2CC(N(C)C(c3cnn(C4CCCC4)c3)=O)C2)=O)CC12CCCCC2 N1(C(CC)=O)CCC(COC)(Oc2ccccc2)C1.C(=O)(C(CC)OC)NC N1(C(COC)=O)CCOCC(C)(CNC(c2noc(-c3cccc(F)c3)n2)=O)C1 C1(C(=O)NC(CNC(C(C)(C)N(C)C)=O)C2CCC2)CCC(=O)CC1(C)C c1(C(CNC(CSCC)=O)C)ccccn1.C12(CCC1)C(=O)N2 Cc1ccc2cccc(C(N3CC(NC(=O)Cn4cnnc4)C(C)C3)=O)c2n1 c1(OCC(=O)OC)cccc(CNC(=O)Cc2ccc(NC3CC3(F)F)cc2)c1 C1(c2ccc(OC)cc2)CN(C(c2ccsc2)=O)CCN1C(=O)C1=C(C)OCC1 C1(OC)CN(C(=O)CC2(CO)CCCC2)CC1NC(C12CSC(C1)C2)=O CCC(F)(F)C(=O)NC1CC(CCNC(c2ccc(-c3nc(=O)o[nH]3)cc2)=O)C1 c1(C(CC)OCCc2cc(C)on2)ccc(Oc2ccc(F)cc2)cc1 Cc1cc(C(N2CC(N(C(=O)CCS(C)=O)C)C3(CC3)C2)=O)c(C)c(C)c1 CC(C)CCC(F)C(=O)NCCOCCC(N1CCn2ccnc21)=O C(CCC1CC1C)(C(=O)NC1CC1c1ccco1)NC(C(=O)NCCOC)=O Cc1ccc2n1CCN(C(C(=O)N(c1ccccc1)CCC#N)C1CC1(Br)Br)C2C c1(C(=O)NCC2C(C(=O)Nc3ccccc3F)CCC2)cccc2ccnn12 n1(CC)cc(C(=O)NC23CC(C2)N(C(=O)C(C)SC(F)(F)F)C3)c2ccccc12 c1(CCCN(CC)CC2(F)CC2)ccccn1 c1(C(=O)NCCc2c(C)ocn2)c(CNC(c2cn(CCO)nn2)=O)nnn1C n1(C(C)C)ncc(C(=O)NCCN(C(=O)CC(C2CC2)C2CC2)CC2CC2)n1 Cc1cc(F)cc(NC(C2CCC(NC(c3ccc(Cl)nc3C)=O)CO2)=O)c1O C1(COC)(NC(=O)C2=CCOC2)CCN(C(c2cncc(O)c2)=O)CC1 Cc1nn(C)c(=O)c(C(N2CCCC(CO)(NC(=O)CC3CC(C)C3)C2)=O)c1C c1(CCC)ncc(C(=O)NC(C)(CNC(c2ccn(C3CC3)n2)=O)CO)s1 N1(C(C2(CNC(C(CC#C)O)=O)CC2)=O)CC(F)(F)CC1CO N1(C(C(C)Oc2ccccn2)=O)CC2CC(C1)N(S(=O)(=O)CCCCCl)C2 Cn1cc(C(O)C(=O)NC2CC(O)C2CC(=O)N(C2CC2)CC2CCC2)cn1 c1(N2CC(N(C)C)C(C)(C)C2)nc(N2CC3CC3C2)nc2cccnc12 c1(C(=O)NCC2C(NC(Cc3c(C)nn(C)c3Cl)=O)C2)ccc2ncn(C)c2n1 C1(C)(NC(CN2CC(CC)C2)=O)CCN(C(C2CCCC2CF)=O)CC1 N1(C(C2C(C(C)(C)C)C2)=O)CC2CN(C(C3CCCC3C3CC3)=O)CCC12 C(=O)(CCCCC1CC1)NCC(C1CCOC1)NC(COC(C)C)=O c1(C(=O)NCC(CN(C(C2CCCN(CCC)C2)=O)C)O)scc2c1CCCC2 C(=O)(C(C(C)C)N(C)C)NC1(CNC(C(CC)n2ccnc2)=O)CCC1 c1(C(N2CC3CC(NC(C4(O)CCCC4)=O)CC2C3)=O)cc2c(nc1O)CCC2 N1(C(=O)OC(C)(C)C)CC2(COC(NC(=O)NCCS)C2)C1.c1(CC#N)ccccc1 N1(C(CCSCC(N)=O)=O)CC(NC(=O)COCc2cccnc2)C2CC12 c1(C(c2n(CCCOC)nnn2)NCCN(C)C)c(Cl)n[nH]c1CC1CC1 CCC(CN(C)C)C(=O)NCCCN(C(c1sccc1SC)=O)CC N1(C(CCOCCC)=O)CCCC2CN(C(=O)CCNC(=O)NC)CCC12 N1(C(CNC(c2c(OCC)cccc2)=O)=O)CCN(C(C)=O)CCC1C C1(NCc2cn(CC)nc2)CCCCC1C(=O)Nc1nn(C)cc1Br c1(C(=O)NC2CC2)ccc(C(N)=O)cn1.C(=O)(C(=O)N(CCCC)C1CC1)NC(C)C N1(C(c2[nH]cc(C(N)=O)c2)=O)CCC2(CC1)CCN(C(=O)CC=C(Cl)Cl)CC2 C(C(=O)NN1CCCC1C(=O)NCC1(c2cccnc2)CCC1)NC(C)=O C1(O)(C(C(=O)N(CC(F)Cl)C)NC(C2CS(=O)C2)=O)CCCCC1 C(=O)(C(O)CC(C)(C)C)NC(C)C(CCc1ccccc1)NC(c1ccn(C)c1)=O N1(C(c2cc(C(C)=O)c(C)o2)=O)CC2(CC(NC(=O)Cc3[nH]cnc3C)CO2)C1 N1(C(C(C)Br)=O)C2CCC(C2)C1CNC(c1ccc(N)c(F)c1)=O Cn1c(C(=O)NC2(C3CN(C(=O)CC4CCC(C#N)C4)C3)CC2)ccc1[N+](=O)[O-] N1(C(C2CCC(=C)CC2)=O)CC(CN(C(=O)CCCN(C)C)C)C2(CC2)C1 C(=O)(C(O)CCCNC(=O)CCc1nccn1C)N(C1CCCCCC1)C C1(CNC(CC=CC)=O)CCCC12CCN(C(c1cnc3c(c1)CCC3)=O)CC2 c1(C(N2CCN(C(CC(=C)C)=O)CC2CCOC)=O)ccc2c(c1)nnn2CC C1(C)(C(=O)NCC2C(CNC(CSCC=C)=O)C2)CC(=O)N(C)C1 N1(C(Cc2c(C)n[nH]c2)=O)CCC(C)(CCNC(C2(C(C)C)CCC2)=O)C1 C1(NC(C(C(C)C)c2ccncc2)=O)CCCCN(C(c2ncccc2Cl)=O)C1 CC(C)CC(CC(C)C)C(=O)N1CC(n2cc(C(O)CC(C)C)nn2)C1 C(=O)(C(CC=C(Cl)Cl)NC(=O)Nc1ccccc1)Nc1cn(C)nc1CN N1(C(COc2cccc(NC(C)=O)c2)=O)CCN(C(=O)C(C)(C)C)CC1C1CC1 c1(C(C)NC(Cc2cccc(C)c2)C)cccc([N+](=O)[O-])c1 C12(CNC(C34CC(C3)C(c3ccccc3)N4)=O)CCCC1CCC2 c1(OC)cc(C(=O)NCCCCCCNC(=O)Cc2ccn(C)n2)cc(Cl)c1O c1(CCNC(=O)C(N2CCOCC2C2CCCOC2)=O)cc([N+](=O)[O-])ccc1F c1(NC2CC3CC(C(=O)OC)CC32)cc2c(cc1C(=O)OC)CCC2 c1(NC(N2CCC(C3CNCCO3)CC2)=O)ccc(OC(F)(F)F)cc1[N+](=O)[O-] c1(C(=O)O)sc2ccccc2c1CBr.n1(CCN2CC(n3cccn3)C2)cccc1 CC(C)CC(CNC(=O)C(C(C)C)C1CCC1)C(=O)N1C2CCC1CC(=O)NC2 C1(CC=C)(NC(=O)CCOCCCC)CCN(C(=O)C(O)CSC)C1 CC(C)CCC(C(=O)N1CCN(C)C(=O)C1C)NC(=O)C=Cc1ccc[nH]1 c1(C(N(C)CC2N(C(C(CC(C)C)OC)=O)CCCC2)=O)cc(F)c(Cl)cc1F c1(OC)noc(C(=O)NCc2ccc(CNC(C3CC(C)CO3)=O)cc2)c1Br C1(CN(C(COCC)=O)C)CCCN1c1nc(COC)ns1 CC1CCN(C(C2C=CC=CC=C2)=O)CC1CNC(=O)CN1CCN(C)CC1 c1(CNC2CC3N(CC(=O)NC(=O)NC)C(CC3)C2)ccc2c(c1)CC(C)(C)O2 CC1(C)CC(NC(C2(C)CC2(F)F)=O)CCN(C(=O)CC2(O)CCCCC2)C1 C1(N(C(C2CC(CC)(CC)C2)=O)C)CCN(C(c2cc(CC)cn2C)=O)CC1C c1(C(C)F)cccc(NC(C2CC(CCNC(C34CC(C3)C4)=O)C2)=O)c1 C1(CC)CN(C(C2CCC3(CCC3)C2)=O)CCN1C(c1cnnn1C)=O C(C(C)(C)CC(=O)NCC1CN(C(c2ccc(CN(C)C)nc2)=O)CC1O)OC C1(C(N2CCC(c3ccc(F)cc3)CC2)=O)CCN(c2nnc(C(F)F)s2)CC1 c1(C(=O)NC2CC3(NC(=O)C(O)C4CCC4)COC2C3)cc(O)c2ccsc2c1 c1(C(=O)NCCCC(=O)NCC)cc2cc(C(=O)OC)cc(Br)c2s1 C(=O)(C(CNC(c1cccnc1)=O)(CC)CC)NCC(=O)N(C)CC N1(C(c2c[nH]c(=NC)o2)=O)CCOC(C(=O)N(C(C)C(=O)OC)CC)CC1 N1(C(C(C)=CC)=O)CCC2(CC1)CN(C(=O)C(C)(CC)CC)C2 c1(C(N2CC3CN(C(c4c(C)ccc(Cl)c4)=O)CC32)=O)cc(Cl)cc2cc[nH]c12 C12(CNC(C3CCN3C3CCCC3)=O)CC(CO1)N(c1ncc(Cl)c(O)n1)C2 C1(CCNC(CC)=O)CC(OC)CN1C(=O)C(C)OC c1(C(N(C(C)CCNC(C2CNC(=O)O2)=O)C)=O)ccc(-c2cnc[nH]2)cc1 CC1(C(=O)Nc2ccc(O)cc2O)CCN(Cc2cccnc2O)CC1 N1(C(C2C(c3onc(CC)n3)CC2)=O)CCOC(CNC(=O)CCC2(O)CCC2)C1 N1(C(c2scnc2C(F)(F)F)=O)CCCOCC12CC2 C12(CNC(C3N(C(COCC(=C)C)=O)CCCC3)=O)CCCC1OCC2 N1(c2n(CCC#C)c(Cc3nccs3)nn2)CCC2CCCCC12 c1(C(CC)NC(=O)NC(C)C(=O)NCc2cccs2)cccc2ccoc12 c1(CCNC(c2n[nH]cc2-c2cnn(C3CCCCO3)c2)=O)ncccn1 c1(CN2C(C(=O)NCCCCCO)COCC2)ccc2nccn2c1 N1(C(Cc2ccc(C)s2)=O)CC2C(C(F)(F)F)CC2(NC(C2(C(N)=O)CC2)=O)C1 c1(CC(N2C(CC(=O)NCC3CCC(O)C3)COCC2)=O)cccc(Cl)c1F C1(O)(C(=O)NC(C2CN(C(C3CCCN3C3CC3)=O)C2)C)CCSC1 N1(C(CSc2ccc(C)cc2)=O)CCC2(CCCCC2NC(=O)NC2CC2)C1 C1(N=c2ccn(CCF)[nH]2)(C(=O)OC)CCN(n2nnnc2C(=O)OC)CC1 C(=O)(C1=NOC2(CCOC2)C1)NCCCN(C(CC(CC)C1CCC1)=O)CC c1(CN2CC3(C(C(=O)N(CCO)C4CC4)C3)C2)ccc(Br)cc1F N1(C(C2N(C(c3cccc(C)n3)=O)CC(F)(F)C2)=O)Cc2nc(C)nc(O)c2C1 Cc1c(Cl)c(C(=O)NC2CC2CNC(c2ccccc2C(C)(C)C)=O)nn1C c1(C(=O)NCC(CO)NC(=O)CC2CCC(=O)O2)c[nH]c2ccc(Cl)cc2c1=O CCCCC(C)CCC(=O)NC1CC(O)C1CC(=O)NC1CCCN(C)C1 C1(NC(c2cc(CC)oc2C)=O)CCC12CN(C(c1ccccc1CO)=O)C2 CC1CC(CNC(=O)CSC(=N)N)CN1C(c1ccc(Cc2ccccc2)[nH]1)=O C1(NC(=O)CN2CCCCCC2)CCC(O)CN(C(=O)C=Cc2ccncn2)C1 CCCC(CCC)=CC(=O)N(C)CC1C2CN(C(c3ncoc3CC)=O)CC12 C#CCC(CC(=O)OC)NC(c1ccc(CNC(C2CC2(Cl)Cl)=O)o1)=O C1(C)(C(N(CCCNC(Cc2[nH]n(CC(C)C)c(=O)c2)=O)C)=O)CCOC(C)C1 C(=O)(C(C(C)(C)C)N(C)C(C)=O)NCCN(CCC)C(c1cc(COC)on1)=O c1(C(=O)NCCCC(C)NC(C(CCSC)NC(N)=O)=O)c(F)ccc(F)c1Cl c1(C(=O)NC(C)CC(C)NC(=O)C=C2CCCCC2)cnc(O)c(Cl)c1 C1(NC(c2c(C)cc(C)[nH]2)=O)CC2CCC(C1)N2C(C1CCC(N=[N+]=[N-])CC1)=O c1(C(N2CC(OC)(CNC(c3snc(C)c3N)=O)C2)=O)cc(Cl)ccc1C(C)C C1(NC(CCn2ccc(C)n2)=O)CCC2CCN(C(=O)C=C(Cl)Cl)C1C2 N1(C(C(C)N(CC)CC)=O)CCC2CC12C(=O)NC12CCCC1C2 c1(NCCCCc2scc(C)n2)ccc(S(=O)(=O)N2CCP(C)(=O)CC2)c(Cl)c1 c1(C(N2CC(C=C)C(NC(=O)C(CC)=CC)C2)=O)cc([N+](=O)[O-])ccc1C N1(C(C2(C)CC(F)(F)C2)=O)CC(C(=O)NCc2cncnc2)C(F)(F)C1 CC(C(=O)N1CC(C)(NC(c2ccc(CO)s2)=O)C1)C1=CCCC1 Cc1[nH][nH]c(=N)c1C(=O)NCC1CCCC(NC(C2(CCF)CC2)=O)C1 c1(COCCNC(C(C)OCCCC)=O)cc(C(=O)NCCCSC)nn1C c1(C(C)C)ncc(C(=O)N(CCCCCNC(c2sccc2CN(C)C)=O)C)[nH]1 c1(OC)cc(F)c(NC(=O)NCCCCO)c(F)c1F.C(C)(=O)NC Cc1cc(C#N)nc(N2CCCN(Cc3cccc(Br)c3F)CC2)n1 N1(C(C2C(C)CC(=O)N2)=O)CCCC(CO)(CNC(=O)C=CC(F)(F)F)C1 C1(CC#C)(C(N2CC3CCC3C2)=O)CCN(C(c2c[nH]nc2C2CC2)=O)C1 Cc1ccc(CC(C)C(=O)NC2CC(NC(=O)CC3CCSC3)C2)cc1 CCC(C)CCC(O)CC(=O)N1CCC2(C1)CN(C(c1ccncc1)=O)CCO2 N#Cc1ccc(C(=O)NCC2(CNC(=O)CC3C=CS(=O)(=O)C3)CCC2)c(F)c1 c1(C(=O)NC2CC(COC)C2(C)C)cc2c3c(ccc2[nH]1)OCO3 Cn1c(Cl)nc2nc(Cl)nc(N3CCC(Nc4ccc(Cl)cc4)C3)c12 C1(CNC(CCC)=O)CC2(CCC2)CN1C(C1CN(C)C(=O)CCO1)=O CC1CCC(N(C(C)(COCCO)c2cccs2)C=O)C1 N1(Cc2cn(CC(C)(C)C)nn2)C(=O)NC(CCCC#N)C1=O CCCCCCCCC(=O)NCCC1(CNC(C2(C)CCCS2)=O)CC1 c1(C(N2CC(C(=O)NCC3CCOC3=O)C2)=O)cn2c(n1)CCC2 C(CCCCC(=O)NCCN1CC=CC1)c1cncc(OC)c1 c1(C(=O)NCCC(C)O)cn(CCNC(=O)C(c2cccn2C)=O)nn1 c1(C(N2CCN(Cc3ccc(Cl)c(Br)c3)C3CC23)=O)ccc(Br)cc1CO C(=O)(C1=CC2CCCCCC12)NCC1CCCN(C(c2c(C)sc(O)n2)=O)C1 c1(C(N(CCC)CCNC(c2csc(C3CCCCC3)n2)=O)=O)nc(Cl)sc1C c1(N2CCCC(NC(C3Cn4c(C)cnc4CC3)=O)C2)ccc2c(n1)CCC2=O N1(CCNC(=O)CCOCC(F)F)CCCN(C(C2CC3CCC2CC3)=O)CC1 C12(C(=O)NC3CN(C(C4CN(CC(F)(F)F)C4)=O)CC3O)CCCC1C2(F)F C(=O)(CCS(N)(=O)=O)NC(C)CN(C)C(c1cscc1Br)=O c1(OC)ccc(C)c(C(N2CCOCC(NC(c3cc(C)cn3CC)=O)C2)=O)n1 C1(C(N(C(C)C)C)=O)C2CCC1CN(C(c1c(F)cncc1F)=O)C2 CCC(F)(F)CC(=O)NCCC1CC(OC)CN1C(c1cscc1SC)=O C1(c2ccccc2)(CNC(CSC)=O)CC12CCN(C(C1CC13CC3)=O)CC2 Nc1c(NN2CCOC(C3CN(C(=O)CCC[N+](=O)[O-])C3)C2)cc(F)cc1[N+](=O)[O-] C(=O)(C1CCc2ccccc21)NCC(C)NC(C1CC(n2cnnc2)C1)=O C(=O)(C1=NN2CC(C)CN=C2N1)NCC1(NC(COCCCCC)=O)CC1 Cc1c(NCCC(=O)N(C2CCC(C)CC2)C2CC2)ncnc1N(CC(F)F)C C1(C(C)C)CCOC1C(=O)NCCN(C)C(c1ccn(CCNS(N)(=O)=O)n1)=O N1(C(C(C)=C(CC)C)=O)CC2CS(=O)(=O)CC2(CNC(=O)CCc2nc[nH]n2)C1 NS(=O)(=O)CC(=O)NC(C1(O)CCN(C(c2c[nH]cc2-c2ccc(Cl)s2)=O)C1)C1CC1 C1(CNC(=O)OC(C)(C)C)CCN(C(C2COCC(=O)N2C)=O)C12CC2 C(=O)(C1CNC(=O)c2ccccc21)NCCC(C)(C)CNC(=O)C1=CCCOC1 c1(C(N2CCC(C)(CNC(CC=C=C)=O)CC2)=O)cccc2ncsc12 c1(C(N(C)CCNC(=O)Cn2nnc(=N)[nH]2)=O)cc(C(F)(F)F)nn1C c1(C(N2CCN(C(CC3(C(=C)F)CCC3)=O)C(C)C2)=O)cc(S(N)(=O)=O)co1 O=C(CCC(F)(F)Cn1cc(C(C2CCC2)O)nn1)NCCn1ccnn1 C1(NC(C(C)C)=O)CN(c2nccnc2F)CC1C c1(CC)cc(C)ccc1C(N1CC(C(N)=O)(CNC(=O)C(C)c2cccs2)C1)=O CC(C)(C(=O)NCC(c1cccs1)O)C1CCCN1C(c1cc[nH]n1)=O N1(C(C(C(C)O)N(C)C)=O)CCOC(C(=O)NOC2(O)CCCCCC2)CC1 n1(CC)nc(C(N2CC(NC(=O)CN3CCC(C)CC3)CC2C)=O)c(C)n1 Cc1cc(Cl)nc(N)c1C(=O)NCC(C)(C)CNC(C1(C)C=CCC1)=O N1(CC(=O)OC)CCCC(CNCC2(C3CC3)CCCO2)C1=O c1(C(=O)NC(CNC(=O)CC2CC=CCC2)C2CCC2)ccc([N+](=O)[O-])cc1O N1CCCC(C)C1.C1(CC(=C)Cl)CCCN1C(=O)NCCCSC N1(C(C(C(CC)C)=O)=O)CC(C(N2CCCC2C(=O)N(C)C)=O)C2(CCC2)C1 C(CC(C(=O)NC1CC1)NC(=O)C(F)OC(F)(F)F)OCC.C1CO1 N1(C(c2c(C)nco2)=O)CC(C(N2CCC(CO)C(C)(C)C2)=O)CC(C)(C)C1 C1(CNC(C(CSC)C)=O)CCC2(CCC2)CN1C(=O)CC(F)(F)C(F)F Cc1cc2scc(CC(=O)NCCC3CN(C(=O)CC4CN(C)C4)CC3C)c2s1 CC1Oc2ccccc2OC1C(=O)N(C1CC1)CC1(n2cncn2)CC1 c1(OC)ccc(F)cc1C(C)NCC1CCCC(C(=O)OC(C)(C)C)C1 c1(NC(c2c(CNC(=O)OC(C)(C)C)nc(C)nc2)=O)cncc2nccn12 c1(CC(=O)NCC2(NC(c3ccc(C(=O)OC)s3)=O)CC2)cn2ccsc2n1 c1(-n2ncc(NC(C3C(C#N)CCCC3)=O)c2)nnc2ccc(Cl)cn12 CCS(=O)(=O)CCNC(C1(OC)CCN(C(=O)OC(C)(C)C)C1)C CN1C(=O)CCC1C(=O)NCC1(C(=O)NCC2CC(C)(C)CO2)CCCC1 C1(NC(c2csc(NC(c3cnc(O)nc3O)=O)n2)=O)Cc2ccccc2O1 C1(CC(N)=O)(NC(CCOCC)=O)CCN(C(C2CC(=O)N2)=O)CC1 N1(C(C(C(C)SC)O)=O)CCC2(CC(NC(c3coc4ccccc34)=O)C2)C1 c1(CNC(C2(CO)CCCO2)=O)ccc(C2CCCNC2)cc1.c1(C)ccccc1 n1(C(C(=O)OC)(C)C)cc[nH]c(=NC(=O)c2ccn3c(N)nnc3c2)c1=O C(=O)(C(C)Cc1cnco1)NCC1C(N(C(C)C(=O)N)C)CC1.N(C)C C1(C(N2CCC(C(=O)NC)C2)=O)CCCN(C(=O)Cn2c(O)nnc2O)C1CC c1(OCCC)ccc(NC(=O)CC2CCCN(C(=O)C(CO)NC(N)=O)C2)cc1 C1(CC)CC(C(N2CCC(C)(NC(=O)CCC(=O)NC)C2)=O)CC(=O)N1 N1(C(C(CCCC)NC(N)=O)=O)CC2(C1)SCCC2CNC(=O)C1=CCCC1 Cc1cc(=NC(C)C(C)F)[nH]c(=NCc2ccc(F)c(Br)c2)[nH]1 C1(N(C(C)=O)C)CCN(C(C2CC(F)(CO)C2)=O)CC1C Cc1ncccc1C=CC(=O)N(C)CC1COCCN1C(C1SCCCS1)=O C1(NC(CC)=O)C2CCC1N(Cc1ccc(C(=O)OC)c(Cl)c1)C2 c1(CC)cccc(F)c1C(=O)NCC(C1CCCC1)NC(=O)C(C)SC c1(-c2cncc(NC(N3CC(CNC)C3)=O)c2)ccc2oc(C(=O)OC)cc2c1 N1(C(COCCC)=O)CCN(C(=O)C(F)CC2CCC2)CC1CS(C)(=O)=O CCC(C)CC(C)C(=O)N1C2CCC1CN(C(C13CC4CC1(CO)CC4C3)=O)C2 C(=O)(C1=NN(C)C(=O)CC1)NCc1cc(C(=O)NCC2CCCCN(C)C2)no1 Cc1cnc(O)c(CNC(=O)C(CC(F)F)NC(=O)COCCF)c1 N1(C(C(CCCCC)O)=O)CC2(NC(=O)C(CC)CC)CCCC2(F)C1 S(=O)(=O)(c1ccc(Br)cc1Cl)Oc1ccc(NC(c2nccc(Cl)c2F)=O)cc1 Cc1nc(C(=O)NC2(CNC(=O)CN3CCCC3=O)CCCCC2)c(Br)s1 C(=O)(C#CC1(C)CCCO1)NC(CNC(C1C(CC)CCCC1)=O)C(C)(C)C C1(C)(CC)CC(NC(c2cc(CNC(C3CCCSC3)=O)on2)=O)C1 N1(C(c2ccccc2CO)=O)C2CCC1CN(S(=O)(=O)c1ccc(F)cc1)CC2 c1(C(=O)NCCCN(C(=O)CN2CCSCC2)C)nc(Cl)sc1Cl Cc1noc(C)c1C(=O)NC(C1(O)CCN(C(=O)C(=CC2CCCCC2)F)C1)C N1(C(C(CCC)(C)Cc2cccc(Br)c2)=O)CCc2ccccc2C1 Cc1[nH]c(C#N)cc1C(=O)NC(c1ccccc1Br)c1cc[nH]n1 N1(C(c2ccc(C)nc2)=O)CC(CNC(=O)CCCN2CCCC2)CC(C)(C)C1 c1(CC)cccc2c(CC(N3CCN(C(=O)C4=CCOC4)CC3C3CC3)=O)c[nH]c12 n1(-c2ccc(OCC)cc2)ncc2c(NCC3CC3(C)C)ncnc12 N1(c2cc(C)nc(CO)n2)CC23CCCC2(CN(C(=O)C=Cc2cnc[nH]2)C3)C1 N1(C(C(CN2CCN(C)CC2)NCN)=O)c2ccccc2OCC1c1ccccc1 C1(C(N2CCC(NC(c3csc4nnsc34)=O)C(O)C2)=O)CCc2nnnn2C1 C1(CNC(COCC(=C)C)=O)CN(C)CCN1C(C1CCOC1C(C)C)=O C12(CC(O)C1)C(=O)NCCC(=O)N2.C1(NC(=O)CO)CCCCO1.NC(=O)NC C1(N=[N+]=[N-])(C(=O)NC(C2(CO)CC2)C)CCN(C(c2scnc2Cl)=O)C1 C1(C(N2CCC(O)(CNC(C=COCC)=O)CC2)=O)CCc2c(n[nH]c2C)C1 Cc1ccc(C(=O)NCC2CN(C(C3Cc4nccn4C3)=O)CCCO2)c(C)n1 N(C1c2ccccc2C2CCC1CC2)C(c1cc(=N)[nH]cc1Br)=O C#CCC(CC#C)C(=O)NCCC1CCC(NC(c2ccccc2NC)=O)C1 c1(C(=O)NC2CC(NC(C(c3ccc(Cl)c(Cl)c3)(C)C)=O)C2)cnc2n1CCS2 c1(C(=O)NCC(CC=C)NC(=O)C(C)SC)cc(C)n(-c2ccn(C)n2)c1C C1(C)(CNC(CCN(C(=O)C#CC(C)(C)C)CC)=O)CCCCC1O CC(C)(C(=O)NCC1CC1C(=O)NCC1(C)CC(O)C1)C(F)F C1(NC(N(CC)CC)=O)CCCN1C(=O)C(c1ccccc1)NC(=O)CN(C)C c1(CCNC(N2CCN(C)C(CNC3=NCCC3)C2)=O)nnc2n1CCCCC2 n1(CC)nc(C2CC2)cc1C(N1CCCC1CN(C(=O)C=CCN(C)C)C)=O c1(C(C)Nc2c(C(N3CCC(C(=O)NC)C3)=O)cccc2)cc(OC)ccc1C c1(C(=O)NC2C(CNC(CC3(C#N)CC3)=O)CCCC2)ccnc2ccccc12 C1(CNC(C(F)=C(C)C)=O)CCC(C)N(C(c2cc(Br)sn2)=O)C1 N1(C(=O)Cc2ccc[nH]2)CCC(O)(CN2CCC2)C1.c1(C2C(=O)N2)ccccc1 C1(NC(C2(OC)CC2)=O)C2CN(C(=O)C(c3ccc(C)cc3)(F)F)CC12 N1(C(C(C)=C(C)C)=O)CCC2(CC1)CN(C(c1cc(Br)oc1C)=O)C2 Cc1nc(CNC(c2csc(CNC(C3CCCCS3)=O)c2)=O)sc1C C(CNC(c1ccc(NS(N)(=O)=O)cc1)=O)(CC(C)C)NC(C(CC)C)=O Cc1nocc1CCC(=O)N(CC(=O)NCC1CC(N(C)C)C1)C C1(C(=O)NCCCCCN(C(CCOC(C)=O)=O)C)COC2(CCC2)C1 N1(C(c2c(C)cccc2)=O)CCN(C(c2csc(C)c2C)=O)C(C)C1 C1(OC)CN(C(=O)C(C)Cc2cccc(Cl)c2)CC1NC(=O)C(F)=C1CCC1 N#CC1(C(=O)NCc2nc(CNC(=O)C(C3(O)CCCC3)F)cs2)CCOCC1 C(=O)(CS(=O)(=O)NC)NCC(CNC(C1(CC)COC1)=O)OCC c1(C(=O)NCC(CO)NC(C=CCC)=O)cccc(C2(O)COC2)c1 C1(CC(=O)NCC2(C(=O)NC(=O)C3CC3)CC2)CCCC1 C1(C(=O)NC2(CCNC(CNS(N(C)C)(=O)=O)=O)CCC2)CNC(=O)C(C)(C)C1 N1(C(C2N(C)CC2)=O)CCCCC1CC1CCN(C(=O)Cn2nnc(=O)[nH]2)CC1 CC1CCC(NC(=O)C(F)(F)C2CCCC2)CN1C(C1CN2CCC1CC2)=O c1(C(=O)OC)ccc2nc(C(=O)NC(c3cc(C)ccc3OC)C)c(F)n2c1 CC(C#N)C(=O)NCc1cc(C(=O)NC2(c3ncccn3)CC2)cs1 Cc1nc(C(=O)NCC(C(C)C)NC(c2cc(F)ccc2C)=O)c2ccsc2n1 Cc1onc(C(C)(C)C)c1C(=O)Nc1cccc(-c2nnnn2C)c1 c1(OC)ncnc(C)c1C(N1CC(NC(=O)CC(C)n2ccnc2)C(O)C1)=O C1(CNC(=O)C(F)Cc2ccccc2)CC2(CC2)CN1C(c1ccc(O)cn1)=O c1(C(N(C2CCCN(C(c3scc(C)c3Cl)=O)C2)C)=O)cn2c(n1)CCC(C)C2 N1(C(c2cc(CC)n(C)n2)=O)CCC2CN(C(=O)CCC(C)CN(C)C)CC12 c1(COC)cc(C(N2CCSCC2)C(=O)NC2(C)CC2)ccc1Br C1(O)(C(=O)NC2CCN(C(C(C)(C)C)=O)C2)CCCCC1 C1(NC(CCCOCC)c2nnnn2C2CCOCC2)CCc2n[nH]cc2C1C OCC1=CCN(c2nnc(-c3c[nH]nc3C(F)(F)Cl)n2CC2(C)CC2)CC1 n1(CC)c(C(=O)NC2CCN(C(=O)C(C)CC3CC3)C2C2CC2)cnc1O N=c1[nH]c(Cl)c([N+](=O)[O-])c(=NCC2CCCC2NC(=O)CC2CCCC(F)(F)C2)[nH]1 C1(CNC(C(N)=O)=O)CC12CCN(C(c1snnc1C1CC1)=O)CC2 N1(C(c2nc(CCC)oc2)=O)CCCC(N=c2[nH]n(C(C)C)cc2[N+](=O)[O-])CC1 c1(C(=O)NC(C=CC(=O)NCCCCCC)C)nc(C)ccc1F c1(C(=O)NCCCC2OCCN(C(C(C)(C)CO)=O)C2)ccc2nc[nH]c2c1F N1(C(c2c(C)oc(CO)c2)=O)CC(C)(C)CC1C(=O)NC1C2CCCCCC12 c1(C(C(=O)NCC(C2CCC2)NC(Cc2cc(CC)no2)=O)C)cccc(F)c1 Cc1cc(N2CC(N(C)C(=O)Nc3ccc(C(C)(C)C)s3)C2)nc(C)n1 c1(C(N2CC(C(N3CCC4(CCC4)C3)=O)C(O)CC2)=O)ccc2ocnc2c1 c1(NCC(c2ccccc2)CC)ccc(C(=O)NCC(N)=O)cc1 Cc1cc2c(N3CCN(CCC=Cc4ccccc4)CC3)nccc2n1C N1(C(C(C)S(C)(=O)=O)=O)CC(NC(=O)C(C)Oc2cccnc2)CC2(CC2)C1 C(=O)(C#CC1CCCCO1)NCCC(C)NC(=O)Cc1nnc2n1CCCC2 CC(C)C(CCNC(c1cc(F)c[nH]1)=O)NC(c1ccc[nH]1)=O c1(C(C2CC2)OCC)noc(-c2cc(-c3ccncc3)[nH]n2)n1 c1(C(=O)NC2CCc3n(C)nnc3C2)cnn2c1NC(C1CC1)CC2C(F)F c1(C(N2C(NC(CN3CC(SCC)C3)=O)CCC2)=O)ccc(C)c(Cl)c1F C1(F)(CNC(C23CC(O)C2C3)=O)CCN(C(c2ccccc2)=O)CC1 c1(OC)cccc2c1CCCC(N(CC(c1c(C)cccc1Br)=O)C)C2 C(c1ccc2c(c1)OCO2)=CCOC(C1C(C(C)C)CCC1)=O C(=O)(CCC(=O)NCc1nocc1C(N1CCCC1CF)=O)NCCC C1(C(=O)NC2CC3CN(C(C)=O)C(C2)C3)COc2ccc(F)cc2C1 C1(C(C(=O)OC)N(C)CCc2ccncc2)(CCl)CCCO1.CCCF N1(C(C(CCC)N(C)C)=O)CCCCCC(NC(c2conc2C)=O)C1 CC1(C)C(C(=O)NC2CCOCC2NC(=O)C=Cc2ncc[nH]2)C1(C)C c1(CCC)cc(C(=O)NC(C)CCNC(C2(CC3CC3)CCCO2)=O)ccc1Cl Cc1cc(C)c(CC(N2CC3CC2C3C(=O)NCC2CCN(C)C2=O)=O)c(C)c1 N1(C(C=C(CCC)C)=O)CCCC2(CCN(C(=O)CC(O)C(C)C)CC2)C1 CC1CC(=O)NC(C(=O)NC(CNC(=O)CCOc2ccc(F)cc2)C2CC2)C1 c1(C(N2CC3C(CNC(C4C=C(C)CCC4)=O)(C3)C2)=O)cc(C#N)oc1C C1(NC(C2C(=C)C2)=O)CCS(=O)(=O)C12CN(C(=O)CSc1ccc(F)c(F)c1)C2 N1(C(C(CCSC)O)=O)CC2CN(C(c3cc4ccc(F)cc4[nH]3)=O)CC2(C)C1 c1(C(=O)NCCC2(NC(Cn3ccc(C)n3)=O)CC2)cccc2cccnc12 c1(CCNC(c2ccncc2Cl)c2n(C(C)C)nnn2)ccc(F)nc1 c1(C(N(C2(CC(=O)NCC3C4CCCC34)CC2)C)=O)cnc(=N)[nH]c1 c1(OCC(=O)NCCCN(C(=O)C(CO)N(C)C)CC)ccc(Br)nc1 c1(OC)c(C(N2CC=CCC2C(=O)NC2CC(=O)NC2=O)=O)cnn1C c1(-c2cn(CN(CC(C)Cc3cccc(Br)c3)C)nn2)ccc(CC(=O)O)cn1 C1(C(N(C)C)=O)COCCN1C(C1CCCCN1C(c1ccc(O)cc1)=O)=O C(CC(C(N)=O)NC(=O)C(Cc1cc[nH]n1)NC(=O)CN1C(=O)CNC1=O)OC c1(C2CCN3CC(C3)N2)nnnn1C1CCCC1.O(C(F)F)OC(N)=O.CO C1(CNC(CC2CC(OCC)C2)=O)CC(C)N(C(=O)CCc2c(C)noc2Cl)C1 CC1CN(C(=O)Cc2cc[nH]n2)CC1(C)C(=O)NCc1cc(C#N)cs1 C(=O)(C(O)CF)N1CC(=C(CNC(C2CC(=O)N2)=O)F)C1 C1(C(=O)NCC(O)CF)CCCN1C(c1cn[nH]c1)=O N1(CCn2cc(C3N(C(C(CSC)OC)=O)CCOC3)nn2)OC(C)(C)CC1=O CC1(C)CCC(NC(=O)C(C)(C)CN2CCCC2=O)Cc2ccccc21 C1(CNC(C(COC)O)=O)CCN(C(c2cc(C)c(C)cn2)=O)CC1O c1(CCC(N2CC(CCNC(C(CCC)N(C)C)=O)C2)=O)cc(C)nc(C)c1 N1(C(C=CC)=O)CC(C)CC1C(=O)Nc1ccc(-n2nccc2C)cc1 C1(CNC(C(CN(C)C)N(C)C)=O)CCCN(C(c2occ3c2CCC3)=O)CC1 c1(-c2n(C(CC)C)ncn2)cccc(C)c1.C(CCC(C)C)(c1ccc(Cl)cc1)NC n1(CC)nc(C(N2CCCC(C(C)NC(=O)CSCC(F)F)C2)=O)cc1C N1(C(C2CC(C)=C(C)CC2)=O)CCC2(C1)CN(C(=O)Cc1n[nH]c(C)n1)C2 c1(N(C)C)ccccc1C(=O)NCCCOCCNC(=O)CC=C1CC1 C1(C)(CNC(C(C)(C)OC(C)C)=O)CCN(C(c2ccccc2CC#N)=O)C1 CCC(CCC(=O)NCC1CC2CC2N1C(c1cnc(C(C)(F)F)s1)=O)OC c1(CC)ccc(C(=O)NC2CCCC2CC(=O)NCc2cscn2)o1 CCCC(CCCNC(=O)Cc1ccsc1)NC(=O)C(C)(O)Cc1ccccc1 C1(CCOC)(NC(=O)C(C)NC(C)=O)CCN(C(c2ccc(Cl)cn2)=O)C1 C(CC(C(=O)N1CCCC(NC(c2cc(F)cs2)=O)C1)c1ccccc1)=C(C)C N1(C(CS(C(C)C)(=O)=O)=O)CCC2CCN(c3nccc(CO)n3)CC2C1 C(=O)(CN1C(=O)CSc2ccccc21)NC(C)CCNC(C1(C)CCC(=O)N1)=O C1(C(N(CCNC(=O)CC2OCCO2)CC)=O)CCC12CCC2.c1(S)ccccc1 C1(C(=O)NCC(C2CCCC2)C)CCCCC1(C)NC(C12CSCC1C2)=O C1(C(=O)NCc2cc(CC)[nH]n2)COCCN1C(c1ccc(C(C)(C)C)cc1)=O C1(N(C(=O)CC2CCCCO2)CCC)CCN(C(C2CCCC(=O)C2)=O)CC1 CCS(=O)(=O)CC(=O)NC1CCCCC1NC(c1[nH]ccc1-c1ccccc1)=O CC(C)(C)C(CNC(C1(O)CC1)=O)C(=O)NCCn1ncnn1 CCCCCC(O)C(=O)NCc1nc(C(N2CCC3CC3C2)=O)c(C)o1 c1(C(=O)NC(C(C)NC(CC2(OC)CC2)=O)C)cc(Br)cnc1O c1(CC(N2CCN(c3c(COC)cccn3)CC2)=O)cccc2c1OCO2 C1(CC)CN(C(=O)CCC2OCCO2)CCN1C(=O)CCc1nc(=N)[nH][nH]1 C1(C(=O)NCc2n(C)ncn2)CN(C(c2cc[nH]n2)=O)CCC1(F)F c1(OC)cccc(CC(=O)NCC2CN(C(c3cc(Cl)cn3C)=O)C3CC23)c1 N1(C(C(C(=O)OCC)F)=O)CC2COCC(C1)C2NC(c1cc(F)cc(Cl)c1)=O C(=O)(C1=CC2C=CC1C2)NCC(CC(=O)NCCOC(C)C)C1CCCC1 c1(NC(CC)=O)cccc(Nc2nc(C(c3nnnn3C)OC)sc2C)c1 N1(C(CCNC(=O)OC)=O)CCC(NC(c2cc(Cl)c(Cl)[nH]2)=O)C(CO)CC1 O=C(C1COCc2ccccc21)NC1CCC2(CC1)CCN(C(=O)CSC1CC1)C2 C1(NC(CN(C)C(=O)C2CC2)=O)C2CC(NC(c3cc(F)n(C)n3)=O)CC12 c1(C(N(CC(CNC(CNC(CCC)=O)=O)(C)C)C)=O)n[nH]cc1[N+](=O)[O-] CN1CCn2ncc(C(N3CC4(CNC(C5CCC(=O)NC5)=O)CCC3C4)=O)c21 c1(CC(=O)NCC(C)NC(c2cc(CN(C)C)c[nH]2)=O)csc2ccccc12 N1(C(C2C(CC)CCN2C(=O)Cn2ccccc2=O)=O)CCCNC(=O)CC1 C12(C(=O)NCC3(CNC(C4(C)CC=CCC4)=O)CCC3)CCC(CC1)C2(C)C N1(c2cc(CC)nc(C)n2)CCC2(CCCN(C(c3ccc(I)cc3Br)=O)C2)C1 C(c1ccccc1)=CCOCC(N1C(C(C)(C)NC(C=CCOC)=O)CCC1)=O C1(CCNC(COCCC)=O)CN(C(c2ccc(N)c(F)c2)=O)CC(C)O1 Cc1noc(C)c1C=CC(=O)N(C(C)CCNC(=O)C(F)(F)c1cccnc1)C c1(OCCC(=O)NCC2CN(C(c3cc(Br)co3)=O)CCO2)cccc(F)c1 c1(NC(=O)OC(N2CC(NC)(CO)C2)=O)cc(C(=O)OC(C)(C)C)cn1C Cn1nc(C(=O)NCC2C=CCN2C(C2CCCN(C(N)=O)C2)=O)ccc1=O C1(NC(c2ccc(O)nn2)=O)CCN(C(c2nccn3cnnc23)=O)CC(O)C1 c1(C(N(C2CCN(C(Cn3c(C)cnc3)=O)C2)C)=O)cc(Cl)ccc1F C1(C(=O)NC2CCC(NC(=O)CCc3cn[nH]c3)CC2)Cc2ccc(F)cc2C1 C1(C(=O)NCCOC2CCCC2)CCN(C(=O)c2ccccn2)O1 C=CC(C)(CC)C(=O)NCc1n[nH]cc1C(=O)NC1CCCC1 N1(C(CC2CC(C)(C)N(C(c3cc(C4CC4)on3)=O)C2)=O)CCOc2ccccc21 C(=O)(CC(C(F)F)NC(=O)C#CC(C)(C)O)N(C)CC1N(CC)CCC1 c1(C(=O)OC(C)C(=O)Nc2ccc(C#N)cc2F)ccccc1S(C)(=O)=O Cn1[nH]c(=NC(=O)c2ccnn2CC(F)F)cc1C(F)F Cc1c(F)cc(C(N2CCOC(C(=O)NCc3ccnc(Cl)c3)C2)=O)cc1Br C1(C(=O)NCC2CN(C(C(C)OCCOCC)=O)C2)OC(C)(C)OC1(C)C c1(OC)cccc(CNC(C)(C)C(=O)NC2CC2C(=O)Nc2onc(C)c2C)c1 C(=O)C1=Cc2ccccc2C1O.CC1CSCCN1 Cc1cc2c(cc1C)C(C(=O)N1CC(C)(NC(=O)CCS(C)(=O)=O)C1)CO2 C1(C2CCOCC2)(CNC(CCN(C)CC)=O)CCN(C(c2cc(C)[nH]n2)=O)C1 C(=O)(CC(C)(C(F)F)N(C)C)NCC(C)NC(c1c[nH]nc1C(C)(F)F)=O C(CC)(CCCC(=O)NC1(C)CCSCC1)NC(CCNC(=O)NC)=O CC1(C(=O)NC2CN3CCC2CC3)CCN(C(=O)CC2CCCC23CC3)CC1 C(CCCC(=O)NCC(CNC(C1(n2cnnn2)CC1)=O)CO)SC c1(OC)cccc(CO)c1.C(=O)(CC(C)(F)F)NCC(C)(C)CSC.C1CCC(=O)N1 C(=O)(CCC(C)NC(c1cc(CO)n(C)n1)=O)N(C)Cc1cnccn1 C(=O)(C1CCCc2ncnn21)NCC(C1CC1)NC(c1c(C)oc(C#N)c1)=O c1(C(=O)NC(C2CN(C(c3ccc([N+](=O)[O-])[nH]3)=O)C2)C)ccn2nnnc2c1 c1(NC2C(NC(C(C)OC)=O)CCCC2)ccccc1[N+](=O)[O-] Cc1c(C(=O)NCCCC(C)NC(C2(CCN(C)C)CC2)=O)cnc2ccnn12 C(C)(CCC(=O)NC(C)C=CC(=O)NCCc1ccn(CC)n1)SC C1(F)(CNC(c2cc(OC)no2)=O)CCN(C(c2nccnc2N)=O)C1 N1(C(C)=O)CC(O)(CC(=O)N(C(c2cnns2)C)C2CC2)C1 C1(CC)CN(C(c2cnn(C)c2N)=O)CCN1C(=O)CC1(N(C)C)CC1 N1(C(CS(N)(=O)=O)=O)CCC2(CC1)CC2(CO)CNC(c1c[nH]nc1F)=O C1(CC(N2CCC(C(C)NC(C3(CC)CCC3)=O)CC2)=O)CCC2(CCC2)O1 Cc1cc(=NC(C)C(C)CO)[nH]c(=NCc2cncc(Cl)c2)[nH]1 Cc1ccc(CCCC(=O)NCCC2(CNC(=O)OC(C)(C)C)CC2)cc1 N1(C(C2(CC=C)CC2)=O)CCOC(C)(CNC(=O)CC2OCCCC2(C)C)C1 c1(C(N2C(C)CC(CC(=O)NC(C(CC)CC)C)C2)=O)ccc2[nH]ccc2n1 N1(C(COCCC)=O)CCCC2(CCN(C(=O)Cc3ccc(F)cc3F)CC2)C1 c1(CC)cccc(OCCC(=O)NCC(C)CNC(=O)CC2CC(C)(C)CO2)c1 C1(NC(C2N(C(CC(=O)N(C)C)=O)CC(O)CC2)=O)CCCCC1N=[N+]=[N-] C1(CNC(C2(NC(C3CCCCCC3F)=O)CC(F)(F)C2)=O)C2CCCCCC12 C1(CC(=O)NCC(C)CNC(C2C3CCC(C3)C2(C)C)=O)Cc2ccccc2C1 c1(NC(N2CCCC(c3nncn3C3CC3)C2)=O)cc(OC(F)(F)F)ccn1 c1(C(N)=O)ccc(C(=O)N2CC(n3cc(CCn4cncn4)nn3)CO2)nn1 c1(CNc2cccc(C(C)(C)O)c2)ccc(C(F)(F)F)c(OC2CC2)c1 C1(CCC(=O)NCC2C(NC(CC=C=C)=O)CCC2)C(=O)NN=C1C C1(C(=O)NCC(C#C)CC)CCC(O)CN1C(=O)CC(=O)OC(C)=O c1(NC(c2ccnc(Br)c2)C)ccc(S(=O)(=O)NC(CO)CCF)c(Cl)c1 S(=O)(=O)(c1cccc(C(=O)NCc2ncn(C)n2)c1)NCC c1(CCC(N2CC(C)(NC(=O)Cc3cnns3)C2)=O)ccc(CO)cc1 C12CCC1C(=O)N2.C(C(=O)NC(C)C)(N(C(COCCOC)=O)C)C1CC1 C12(CC(=O)NC3(C)CN(C(=O)CN4CC=CC4)C3)CCCCC1C2(F)F CC1(CO)CCN(C(=O)CCOCCNC(c2ccc(C#N)o2)=O)CC1 C1(NC(C2(C)CCOC2)=O)CC(N=c2cc(Cl)nc(C3CCC3)[nH]2)C1 N1(C(c2cc(Cl)cc(Br)c2)=O)CCCC2(C1)CN(S(=O)(=O)C1CCCC1)CCO2 c1(C(=O)NC)ccc(S(=O)(=O)N(C)CCNCc2ccn(C)c(=O)c2)cc1 CC1CN(C(=O)CCCCF)CCC1NC(=O)C(c1ccc(F)cc1)C C=CCC(C)(CC=C)NC(=O)C(COCCOC)NC(C1(C)CCC(O)CC1)=O C1(CNC(C=CCN(CC)CC)=O)CCCC1NC(c1n[nH]cc1C1CCC1)=O c1(CCC(=O)NCC2(CNC(C3(C#N)C(C)C3)=O)CC2)cccc(Br)c1F C1(CNC(Cc2c(C)scc2)=O)CCN(C(=O)Cn2nnc(=N)[nH]2)CCC1(F)F c1(C(=O)NC(CSCC)C(=O)NC2CC(O)C2(C)C)ncccc1C C(C)(C)(C(=O)NCC(=O)NC1CCC1)OC(CC)C c1(C(N(C(CC)(C)C(=O)O)C)=O)cc2cc([N+](=O)[O-])ccc2s1 c1(CNC(c2cnc3n[nH]c(C)c3c2)=O)ccc2c(c1)OCCCO2 c1(NC(C(=O)NC(C(=O)OC)Cc2csc(Br)c2)C)ccc(C)cc1 Cc1ccc2c(C(N3CC(NC(C4CNC(=O)C4)=O)C4(CCC4)C3)=O)c[nH]c2c1 Cc1ccc(I)c(NC(C2CCCC2NC(c2cccc(O)c2F)=O)=O)n1 N1(C(CN2CCC(C)C2)=O)CC2CCC1CN2C(=O)COc1cn[nH]c1 c1(OC)ccc(OC)c(C(=O)NNC(=O)C2CC(I)C2)c1.c12ccc(cc1)o2 CCCC(C)CC(=O)NC(C)C(C)(C)NC(=O)Cc1cccs1 N1(C(CC2(CSC)CC2)=O)CC(C2(NC(=O)Cc3ccn(C(F)F)n3)CC2)C1 C1(C(N2CCC(CC(=O)OC(C)(C)C)CC2)=O)CCN(C(=O)N(C)C)CC12COC2 CCCCC(CC)C(=O)N1CC(CNC(c2nc(CC)oc2C)=O)CC(C)C1 c1(NC2C(C)N(C)C(=O)C2)cc([N+](=O)[O-])ccc1N(C)C c1(-n2c(C(c3cccs3)NC(C(=O)N(C)CC)C)nnn2)cccc(OC)c1 C1(CNC(=O)C(=O)N2CCC2CC2CCC2)CCCC2(CC2)C1 n1(CC(=O)N(C)C)ccc(C(=O)NCC2CCCC2NC(=O)C(C)(O)C2CC2)n1 C1(c2ccc(CC)o2)CN(C(C2CC(OC)C2(C)C)=O)CCO1 c1(OC)cc(NC(C2C3CC2(c2ccccc2)CO3)=O)ccc1C C1(CNC(C=CCCC)=O)CN(C(c2ccc(Cl)c(OC)c2)=O)CC(C)(C)C1 C(=O)(CS(=O)(=O)N1CCCCC1)NC(CC)CN(C(=O)C(C)NC(N)=O)C c1(CC(=O)NCCN(C(=O)C(F)=C(C)C)CC)cccc(Cl)c1 CCC1=C(C(=O)NCC2C(C)CCN2C(=O)CC(C)(C)C#N)CCCO1 C1(CCNC(=O)CN2CCCCC2)CC(F)(F)CN1C(=O)CN1CCC(CO)CC1 Cc1[nH]nc2ncc(C(=O)NCC3(C)CCN(C(c4ccc(Cl)nn4)=O)C3)cc12 S(=O)(=O)(c1c[nH]ccc1=NCCC1CCCOC1)NC(C)CCN1CCOCC1 C1(NC(C2(C(C)NC(c3ccc(O)nn3)=O)CCCO2)=O)CC(C)(C)C12CC2 N1(C(C)C)CCCCC1C(=O)NCCC(O)CNC(c1ccc(OCF)cc1)=O CC(C)C(F)(F)CCNC(=O)C#CCNC(=O)CC1(C)OCCO1 C(CC1CCC1)(C(=O)NC1CCN(C(C)C(=O)NCCC(C)C)C1)NC(C)=O C1(NC(C(CC=CC)CC)=O)CN(C(=O)COC)CCC1(C)C C1(C(=O)NC2CCOC23CCC3)(CO)CCCN(C(=O)COc2ccsc2)C1 C1(NC(C(CC2CC2)OC)=O)CC(F)CN(C(=O)CN2CSCCSC2)C1 CC1CCC(C)C1NC(=O)C(C1CC1)NC(=O)CCCC1CCCC1 C(=O)(C(O)CC(C)(C)C)NCC(=O)NCc1ccc(CN2CCCC(C)C2)o1 C(=O)(N=c1ccn(CC(=O)NC2CC3(CO)COC2C3)[nH]1)C1(OC)CCC1.C(C)=O C1(C(=O)NC2C=CCN(C(Cc3c(CC)noc3CC)=O)C2)CCC(N=[N+]=[N-])C1 c1(OC)cccc(C2(O)CN(C(c3ncc(N(C)C(C)C)cn3)=O)C2)c1 N1(C(C2(C)CCCCC2)=O)CCCC2(NC(c3cc(F)ccc3O)=O)CC12 c1(C(=O)NC2CC(C)N(C(c3cnn(CC4CC4)c3)=O)C2)cccc(Cl)c1F C1(n2ncc(C(=O)NCc3cnoc3)c2)CCN(C(=O)C=Cc2cccs2)CC1 c1(OC)ccc(CC(=O)NCC(C)N(C)C(c2ncc(Cl)cc2F)=O)c(OC)c1 O(NC(=O)C(CCOC)NC(=O)CCCCCF)CC1CC(=C)C1 C1(NC(C2(CCC)CC2)=O)COC2(CCCN(C(c3cccnc3CO)=O)C2)C1 C(C(CC1CC1)C(=O)NCC1C=CCOC1)NC(=O)CCc1csnn1 C#CC1(C(=O)NCCc2ccc(OC)cc2)CCN(C(=O)Cc2cccs2)CC1 C(C)(C)(CCC(=O)N1CC(CNC(=O)C(C(C)(C)C)c2cc[nH]n2)C1)OC C1(C)(COC)CCN1C(=O)CCCC1(NC(C2(C)CCCC2)=O)CCC1 CC(CC(C)(C)C)C(=O)NCC1CC(F)(CNC(=O)CC2CC3COCC23)C1 C12CCCCN(C1=O)C(=O)C(C)N2C.C1(OCC)CCCC1 C1(COC(CCCOc2c(OC)cccc2)=O)CN2CCC1CC2 N1(C(=O)Cc2nnc(O)s2)CCC2(CCN(C(c3ccn4nccc4n3)=O)C2)C1 c12ccc(cc1OC)C=CC(=O)O2.c1(NCC)c(Cl)cccc1[N+](=O)[O-] N1(C(C=CCC)=O)CC(C2CC2)(C(=O)NCC2CC2COC)C1 N1(CCNC(CCN(C(=O)C(C)(C)N(C)C)CC=C)=O)CCCC1=O N12CCC(C1)C(=O)N(C)CC2=O.C1(C#N)(CCC(=O)NC2CC2)CCC1 C12(C(=O)NC(C(C)C)CCN(C(=O)CSCC(F)F)C)CCC(N=[N+]=[N-])C1C2 CC(CN(C)C)CC(=O)N(CCCC(=O)NC(C)(C)CCCF)C C1(F)(C(=O)NC2CC(NC(C)=O)C2)CCCN(C(=O)CCC(C)(C)C)C1 c1(COC(C)C)ccc(NC(=O)C2CC2)c(-c2ccnn2C2CC2)c1 C1(Cc2cn(CC(C)(C)C)nn2)CCCN(C(c2c[nH]nc2C2CCOC2)=O)C1 CC1(C)COC(C)(C(=O)NCC2CN3CCN2CC3)CO1 N1(C(c2n(CC)ncc2Cl)=O)CC(CNC(=O)C2=COCC2)C2(CCC2)C1 c1(CNc2cc(N3C4(C(N(C)C)=O)CC(C3)C4)ncn2)sc2ncccc2c1N C1(C(C)C(=O)NCC(Cl)=CCl)CCN(C(C2(C)CCCCO2)=O)CC1 c1(C(=O)NC2(Cc3ccc(F)nc3)CCOC2)cccc2nn[nH]c12 C1(C(=O)OC)CCN(C(=O)C2C3CCN(C(c4cc(C#N)c[nH]4)=O)CC23)O1 C1(NC(=O)C(c2ccccc2)F)C=CCN(C(C2(CCF)CC2)=O)C1 N(C1CCCn2nccc21)C(C1=NOC(CNC(C2CC(N(C)C)C2)=O)C1)=O c1(NC(N2CCC(Cn3cc(Cc4ccc(F)cn4)nn3)CC2)=O)ccc(Br)cc1 c1(C2(NC(=O)NCCc3ccc(Cl)nc3)CCC2)cccc(Br)c1 c1(C(=O)NCc2c(CNC(C(C(C)C)C)=O)cccn2)ccn2nccc2c1 Cc1ccc2c(N3CCC(NC(c4c(O)cccc4Br)=O)C3)ncnc2c1 N1(C(C(C)(C)SC)=O)CCCC2(CC(NC(c3cnn(C(F)F)c3)=O)CO2)C1 C(C(CC(C)C)C(=O)NC1CCN(C(c2cn(C)nc2C2CC2)=O)C1)OC CCC(C)CC(C)N(C=O)Cc1ccc(-c2csc(C)n2)s1 c1(C(N2CCC(CCNC(c3ccc(C#N)s3)=O)C2)=O)cc2cc(Cl)cnc2o1 C1(C)(N)CN(C(=O)CCc2ccco2)C1.C12(CCC1)CC(=O)N2.C#CC C1(C(N2CCC(CF)(NC(=O)Cc3cnc(C)s3)C2)=O)(CC)CCNC1=O N1(CCOCCCOC)Cc2c(OC)ccc(OC)c2C(O)C1 C1(C)(NC(C=C(CC)CC)=O)CCCCC1C(=O)N(C)Cc1cncs1 c1(OC)ncc(CNC(C2(CC(N3CC(O)C(O)C3)=O)CC2)=O)cc1Cl C#Cc1ccc(CC(=O)NCC(C)(C)CNC(=O)C(F)(F)CC)cc1 C(=O)(C1=CC2(CCN(C(=O)CCC3CCCC3)C2)C1)N1CCC(C)(CO)C1 Cc1cc(C(=O)NCC2CCCN(C(C3CC34CC4)=O)C2)c(C)n1-c1nccs1 c1(-n2ccc(NC(=O)Nc3c(CC)cccc3F)n2)cc(F)cc(F)c1OCC N1(C(C(c2ccc(C)cc2)=O)=O)CCN(C(=O)Cc2cncs2)CC(O)C1 C(=O)(C(CO)C(C)(C)C)NC1CCN(C(c2c(C)ccc(C(F)F)c2)=O)CC1 C=CC(C)(CC)C(=O)NC1CN(C(c2cnc(C3CCCO3)s2)=O)C1 c1(C(=O)NCC(C2CCC2)NC(C2ON=C(CC)C2)=O)nc(OC)ccc1C O=C(N1NC2CCC1CC2)C1CCOC1SC(F)(F)F C1(NC(c2cc(C)on2)=O)CCN(C2CN(C(=O)OC(C)(C)C)C2)CC1 C1(C(N(c2nc(=N)[nH][nH]2)C)=O)CN(C(=O)C#CC2(C)COC2)CC12CCC2 Cc1ccn2cc(C(=O)NCC3(C)CCN(C(c4cncc(N)n4)=O)C3)nc2c1 Cn1ccc(C=CC(=O)NCC23CC(N(C(=O)CNC4CCOCC4)C)(C2)C3)c1 C1(CCNC(=O)CC)(OC)CCN(C(=O)CC2CC=CC2)C1 Cc1noc(C)c1CC(C)C(=O)NCC12CC1CN(C(=O)CC1CCCC1)C2 c1(NC(C(CCC)NC(=O)CC(C)SC)=O)c(C)[nH]c(C)cc1=O N1(C(C=C(COC)C)=O)CCCCC1CN(C(=O)COC)CC1CCCO1 N1(C(C23N(C(c4c[nH]nc4[N+](=O)[O-])=O)CC(C2)C3)=O)C(CO)CCC12CCC2 c1(CNC(c2cn(Cc3cccc(C#N)c3)nc2)=O)n[nH]c2ccc(O)cc12 CN1CCc2ccc(C(N3C4CCC3CC(NC(C3CC5CC5C3)=O)C4)=O)cc21 c1(C2C(C(=O)NCC(C3CCCC3)NC(c3ccc(CO)o3)=O)C2)cccnc1 N1(C(CN(C(=O)CC2CCOC2C)CC#C)=O)CCC=C(F)C1 C(C(F)(F)CN(C)C)NC(=O)N(CCSCC1CCCO1)CC.C=C1CC(CC)C1 C(N=c1cc(Cl)nc(-c2ccccn2)[nH]1)C1CCCC(CO)C1 N1(C(CC2(C)CCOCC2)=O)C(C(=O)NCC2CCCCC2)CCC12CC2 CC1(C)CC1(C(=O)NCC(C1CC1)N(C)C)NC(=O)Cn1[nH]cnc1=N C1(CC)CC(O)CCN1C(=O)Cn1cc(CCOC2CCOC2)nn1 Cc1cccc(N(CC(C)(C)C)C(C2CC2c2cccc(Br)c2)=O)c1 c1(CC(=O)NC2C(NC(c3c(CC)cccc3)=O)COCC2)ccc(C)c(O)c1 CCCC(O)C(=O)NCc1ccc(C(=O)NCC(C)(CC)CC)s1 C1(C(N(CC(N2C(C(C)O)CC2)=O)C2CC2)=O)CCCC1O c1(C(=O)NC2C(NC(C(C)Cc3ccco3)=O)CCOC2)ccc2c(c1)NCC2 N(C1CCCc2cc(CNC(N3CCC3)=O)ccc21)C(CCc1ccc(C)s1)=O c1(C(=O)NC(C)CN(C)C(C2(c3cc[nH]n3)CCC2)=O)cc2occc2n1C C1(C(=O)NC(CC(C)NC(C2CCCN2c2ccccc2)=O)C)CCCOCC1 C=CC(C)CC(=O)NC1CCN(C(=O)Cn2cccc2)C1c1ccccc1 C1(NC(C(CC)NC(C)=O)=O)CCCC1(C)NC(c1cc(Br)c[nH]1)=O C(C)(C(F)(F)C(F)(F)F)=CC(=O)NC1CC(NC(CCC=C)=O)C(O)C1 C1(C(N2C3CC(NC(C4N(C=O)CCC4)=O)(C3)C2)=O)CCc2ccc(F)cc2O1 C(=O)(C#CC1(C(F)(F)F)CC1)NCCC1N(C(CC2CCN(C)C2)=O)CCSC1 CC(CC(=O)NCCC(C)NC(C1COC1)=O)c1ccccc1 C1(NC(C(CC)=CC)=O)CC(C(=O)NCc2ccc(C#N)o2)C1(C)C C1(NC(CSCC(=O)OCC)=O)C2CC(NC(=O)COCCOC)CC12 N1(C(CCC=C)=O)CCC(CNC(=O)COCCSC)CC1C c1(C(=O)NCC(CCN(C)C(c2ccncc2)=O)OC)ccc(Cl)c(Cl)c1.CO N1(C(c2c(-c3ccc(C)o3)onc2)=O)CCC(NC(=O)C=CCO)C(C)C1 C1(C(C)C(=O)N(C)CCNC(=O)C2=CCSC2)CCC(F)(F)CC1 Cc1cc(C)c(CC(=O)Nc2cc(C(=O)O)cc3c[nH]nc23)c(C)c1 C1(CC(N2CC(OC)C(OC)C2)=O)CN(C(=O)C=C(C)C)CCC1C CCC(C)(COC)C(=O)NCC#CCNC(=O)C(C(C)(C)C)n1ccnn1 C(=O)(C(C(C)C(C)C)NC(=O)NC1(CC2CCC2)CC1)OC CC1CC(C)CCC1C(N1CCCC1c1nn[nH]n1)=O c1(SC)nc(Cl)cc(=NCC23CCC(NC(=O)C=C(C)c4ccco4)(CO2)C3)[nH]1 n1(C(C)C)ccc(C(=O)NC2CN(C(C3CCCO3)=O)CC2(C)C)cc1=O S(=O)(=O)(c1cc(C(F)(F)F)cc(N)c1)N1CCC(NCCC#N)CC1 c1(CC(=O)NCC2(C(=O)NC3(CF)CC3)CCCO2)ccccc1SC(F)(F)F Cc1noc(C(C)N(C(C(C)(C)C)c2ccccc2)C)n1 c1(C(=O)NC(CNC(C(C)OCC)=O)(C)CO)cc(OC(C)C)cc(Br)c1 Cc1cccc(OCCONC(=O)OC(C)(C)C)c1.C12(CCOCC1)CC(=O)N2 O=S(=O)(CCCCCN1CCCC1)c1ncco1 CC(C)CC(C)(CNC(=O)CC(C)(C)c1ccc(F)cc1)NC(=O)C1=CCC1 c1(OC)ccc2[nH]nc(C(=O)NC3CC3NC(C3CC4CCC3O4)=O)c2c1 c1(CC)ncnc(CC)c1C(=O)NCC1CCN(C(=O)CC23CCCC2C3)C1 N1(C(C(C)OCC2CC2)=O)CCC2(C1)CN(C(c1cccc3nsnc13)=O)C2 Cc1ccc(F)c(C(N2CCC(N(C(=O)Cc3nn(C)cc3Cl)CC)C2)=O)c1N N1(C(C(CC)O)=O)CCC2(CC1)CN(C(c1ccnc(C)c1N)=O)C2 N#CCS(=O)(=O)NC1CC(C(=O)Nc2ccc(C(N)=O)s2)C1 N1(C(C(C2CCCC2)NC(CN(CCOC)C)=O)=O)CCC(C)C(C)(C)C1 C(CCC(O)C(=O)Nn1ccccc1=O)NC(CSC)=O C(=O)(C(C)(C)C1CCN(C(C2CC23CCC3)=O)C1)NCC=C C1(C)(C(=O)NC2CCN(CCN3CCC(CC)CC3)C2)CC(C(C)C)=NO1 Cc1cc(C(=O)NC2CN(C(=O)Cc3ccc(O)cn3)CC2F)cc2ccoc12 C1(C(N(C)CC2(C)CCOCC2)=O)N(C(C23CC(CO)(C2)C3)=O)CC12CCCC2 n1(CC=C)cc(C(N2CC(CCNC(=O)C(C)(C)c3cc[nH]n3)C2)=O)cn1 Cc1cncc(C(N2CCOCC2CN(C)C(C2CC3CCC2O3)=O)=O)c1 c1(Cc2nc(CCC)on2)[nH]nc(CC)c1C.c12ccccc1S2 c1(C(=O)NCCC2CCN(C(C3(C#N)CCOC3)=O)C2)ccc(F)c(F)c1F c1(C(N2C3CC(CNC(C=C(C)C)=O)CC2CC3)=O)csc2ccc(F)cc12 N1(C(c2n(C(C)C)ncn2)=O)CCC(CNC(C2CCCS2(=O)=O)=O)CC1 C1(NC(C2C(C(C)(C)O)C2)=O)CCC(NC(=O)CCc2cnoc2)CC1 C1(F)(CNC(c2[nH]c(=NC)sc2)=O)CCN(C(=O)CCCCc2cnn[nH]2)CC1 CCCC(C(=O)NCC1CN(C(=O)CC2CC3CC3C2)CC1OCC)S(N)(=O)=O C1(NC(c2c(C(C)(C)C)cccc2)=O)C2CC(O)C1N(C(=O)C#CC1CCC1)C2 C1(OC)CCN(C(c2cc(CNC(c3cncc(C#N)c3)=O)ccn2)=O)C1(C)C C1(CNC(C2C(C)(C(=O)OCC)C2)=O)(OC(C)=O)CN(C(=O)Cn2cccn2)C1 c1(C(=O)NCC(C2CC2)NC(c2nc(C(=O)OC)sc2)=O)ccnc(C)c1 c1(CC(=O)NCCC(O)CNC(=O)C(=O)NCC(F)(F)F)ccc(F)cn1 C1(C(NOCC(=C)C)=O)CCC2(CC2)N1C(c1ncccc1Cl)=O c1(C(=O)NC2CN(C(CC(C)C(F)F)=O)CC2O)cnn2c1CN(C)CC2 N1(C(c2ncccc2CO)=O)CCCC1C1CCCN1C(=O)Cc1ccsc1 c1(C(=O)NCC2N(C(CC(C)OC)=O)CC(C)(C)C2)c(C)ccc2nsnc12 c1(CCCC(=O)N(CCNC(C2(C)CCCC2O)=O)CC)ccc2c(c1)OCO2 c1(CC)cc(F)c(C(=O)NC2CC(C)(NC(=O)Cc3cccc(O)c3)C2)cc1F c1(OC(C)C(=O)NCCCN(C(=O)CC2CC(=O)NC2=O)C)ccccc1Cl N1(C(C=Cc2ccc(C(N)=O)o2)=O)CCN(C(=O)C(F)=C(C)C)CC(O)C1 c1(C(=O)NCCNC(C2CCN(C(CC3(C)CC3(F)Cl)=O)C2)=O)cccc(=O)o1 N1(C(C(=O)NCCN2CCCC2)C2CCSC2)CC2COCC2C1 C12(C(=O)NCC(CC)NC(=O)CCCN(C)C(C)=O)CCC1CC2 c1(C(=O)NCCN(C(C2(C)ON=C(C)C2)=O)C)cc(C)c2c(O)nc(O)nc2n1 C1(C)(C(=O)NCC(CC)NC(=O)C=Cc2ccncc2)CC(OC)CN1C C1(NC(c2cc(CC)no2)=O)CC(O)(C2CCN(C(C3(C(C)C)CC3)=O)CC2)C1 C1(CNC(C2C(C)(C)C2(C)C)=O)CCC2(CCC2)C1NC(=O)CNC=O c1(CC)cc(C(=O)NC2CC(O)(CNC(c3cc(C(C)C)oc3C)=O)C2)sc1C CCCC(C)(CCC)C(=O)NCC1(NC(C2CC2c2ccoc2C)=O)CC1 N1(C(C2CCCC(C)C2)=O)CCCC2(CCCN(Cc3ncc[nH]3)C2)C1 CC1CN(C(c2cnc3n2CCC3)=O)CC(C)N(c2ccc([N+](=O)[O-])c(O)n2)C1 C1(CNC(C(CC)NC(C)=O)=O)CC2CCC1N2C(=O)CC(O)C1CCCC1 C1(C(=O)NCCC2ON=C(C)C2)CCN(C(=O)C2=CCCC2)CC1O c1(SCC)cc(C)c(C#N)cn1.C(=O)(C(O)CNC(=O)C(N1CCNC1=O)C)NCC C=C=C(C)CC(=O)N(CC(=O)NCC1CCC(=O)NC1)C1CC1 c1(C(=O)NCC2N(C(c3c(OC)cc(O)nc3)=O)CCC2)cc(Cl)c(N)c(Cl)c1 c1(OC)ccc(C(=O)NCCN(C(=O)C=Cc2ccc(C)s2)CC2CC2)nn1 C12(NC(c3c(C)ccs3)=O)CC1CN(C(c1cn(C3CCCC3O)nn1)=O)C2 c1(SCC)cnccc1C(=O)NC1CN(C(c2c(C)coc2C)=O)CC1F Cn1c(O)nc2ccc(C(N3CC(O)(CNC(c4cc(CF)on4)=O)C3)=O)cc12 C1(NC(C=COCC)=O)CCCCCN(C(c2ccc(C3CC3)nc2O)=O)C1 N1(C(c2csc(C)c2N)=O)CCCC1C1CCCN1C(c1cn(C)c(=O)nc1O)=O c1(C(=O)NCCc2ccc(C)c(F)c2)cccc2c1CCNC2 n1(CCC(=O)NC(CCCC)CN(C(C2CCCC2O)=O)CC)ccc(O)nc1=O Cc1ccc(C2CC2NC(=O)CO)cc1.N12CCN(CC1)C1CCC(CC1)C2=O n1(CC(=O)NCCCN(C(COCCCCC)=O)CC)cc(Cl)c(C(F)(F)F)n1 c1(C(=O)NC2CCN(C(C(CCC)C)=O)CCC2CO)nn(C)c2c1COCC2 C1(C)(NC(C2C(NC(c3cnc(CC)s3)=O)CCOC2)=O)CCCCC1C c1(C(N(C)Cc2cn(CC3CC3)nn2)=O)c2ccccc2nn1C N1(C(C=COCC)=O)CCCC12CCN(C(C1CCc3cnn(C)c3C1)=O)C2 c1(CC(N2CCC(NC(C(CCC)CC)=O)C2)=O)ccc([N+](=O)[O-])c(N)c1 C1(C(N2CCC(O)(C(C)NC(=O)CC3(O)CCCC3)C2)=O)(OC)CCCCCC1 C(=O)(C1=Cc2ccccc2C1)N1C(C)CC(CNC(C2CCCC(C)C2)=O)C1 CC(C)C(C(=O)NC1(CNC(C2CCN(C(=O)C(C)C)CC2)=O)CC1)C(C)C N1(C(c2c(C(C)C)nns2)=O)CCC(NC(=O)C(C)S(N)(=O)=O)CC(O)C1 C1(CNC(C2CC(C)(F)C2)=O)C2CCC(C2)N1C(c1csc(C(F)(F)F)n1)=O CS(=O)(=O)C1CN(C(c2cc3n(n2)CC2(CC2)C3)=O)CC1NC(C1CCOC1)=O C1(NC(C(C)N2CCC2)=O)CCCN(C(c2cn(C)nc2-c2cccnc2)=O)C1 C(=O)(CS(=O)(=O)Cc1cccs1)NCC(C)N(C(c1c(C)nn(C2CC2)c1)=O)C N1(C(C2CN(C(C)=O)C2)=O)CC(CC(=O)NC(CCO)CC(C)C)CC1(C)C c1(CC)cc(C(=O)NCC2(CN(C(=O)CN3CCS(=O)CC3)C)CC2)ncn1 C(=O)(N=c1ccn(C(F)F)[nH]1)C1(NC(c2onc(C)n2)=O)CCOCC1 N1(C(C(Cn2ccc(C)n2)C)=O)CCN(C(=O)C2=NNC(=O)CC2)C2(CC2)C1 C1(C(N(C(C)C)CCNC(=O)COc2ccsn2)=O)CCCC2(C1)CC2(F)F N1(C(Cc2c(C)con2)=O)CCC(C)(CCNC(=O)CC2CC=CCC2)C1 c1(CC(=O)NC2CCN(C(C(CC)=CC)=O)C2C)ccc2c(c1)COCC2 O=C(CC(O)CNC(C1CNC(=O)C1)=O)NCC(c1ccccn1)O c1(OC)cc(C(N2CCN(C3CCN(C(=O)C(C)O)C3)CC2)=O)c(F)cn1 C1(NC(c2cc(Cl)ccc2O)=O)(CO)CCCN(C(C2CC3CCC(C2)S3)=O)C1 N1(C(c2nc(CCC)oc2)=O)CC(=O)NCC1C(=O)NCC(CC(C)C)N(C)C c1(C(=O)NCC(C)(C)CC2CN(C(c3c[nH]c(=O)cn3)=O)C2)cc(CO)ccn1 C(CCCCCN)N(COC)CCC.c1(SC(CC)C(=O)NS(C)(=O)=O)ccc(OC)cc1 CC1(CNC(N2CCc3ncc(Cl)cc32)=O)CCCc2ccccc21 c1(C(=O)NCC2(NC(c3cnc(O)o3)=O)CCOCC2)cccc2c1OCO2 c1(C(N2C(C)CC(NC(CCc3n(CC)ccn3)=O)C2)=O)[nH]c(=N)ccc1C c1(C(N(CC(CN(C(C(CN(C)C)O)=O)C)O)C)=O)nccc2ncccc12 N1(C(COC(C)(C)C)=O)CCN(C(c2cc3cccnn3c2)=O)C2CCC12 C1(NC(CCc2cnc(C)s2)=O)CN(C(c2sc(C)cc2C)=O)CC1F c1(NC(C2CC(N(C)C)(C(F)F)C2)=O)cccnc1NC(C1CC2C=CC1C2)=O N(C(=NCC1CCSC1)N1CCC(F)(c2ccccc2)C1)(CC=C)CC C1(C(C)NC(CSCCC)=O)CCN(C(=O)CCCC2(OC)CCC2)CC1 c1(C(=O)NC(CC)CN(C(=O)CC(=O)NC2CC2)CC)ccc(C)cc1F C(=O)(C1=NN(C)C(=O)CC1)NCCC(C)N(C)C(c1cn2ncccc2n1)=O CC(C)(C)CCCCC(=O)N1CCOC(CNC(c2cc3ccncc3s2)=O)C1 C1(NC(CCC=C(C)C)=O)(CO)CCN(C(c2ccc(C)c(Br)c2)=O)CC1 C1(NC(=O)CCc2nncs2)CCC(CNC(c2csc(C(F)F)n2)=O)C1 C(=O)(C1=CCCN(C(=O)C(CC(C)C)N(C)C)C1)N1CCCC(CC)(CO)C1 c1(C(N(C)CC2CCCN(C(C3OCC(C)C3)=O)C2)=O)cnn2ccn(C)c12 c1(C(c2nnnn2CC)NC(c2cccnc2)CCOCC)ncc(SC)cn1 C(c1cccc(C(F)F)c1)=CC(=O)NCC(C)CN(C(=O)CCOC1CCC1)C C=CC(C)(C)CC(=O)NC1CC(CSC)N(C(c2cc(SC)ccc2C)=O)C1 N1(C(Cc2nc(=N)[nH][nH]2)=O)CCCOC(C(=O)NCC2CC(CO)CO2)C1 CCCC(CCC)CC(=O)N1CCC(N(C(=O)CC23CC(C2)C3)CCC)C1 Cn1ccc(C(=O)NCC2CC3(C2)CN(C(C2CC(C4CC4)C2)=O)C3)cc1=O c1(OCC2OCCN(C(=O)Cn3cc(CO)nn3)C2)ccc(Br)c(Cl)c1 C(=O)(C(C)(C)CC(=O)NC1CCCC1C(N1CC(=O)NC(C)C1C)=O)OC c1(C2(NC(C(C3CCCCC3)NC(C=C(COC)C)=O)=O)CC2)ccnn1C C(=O)(C(CCC(N)=O)n1cc(-c2c(C)nn(C)c2C)nn1)NC1C(CCC)C1 C1(OC)CCC(C)(C(N2CC(CNC(=O)C3=CCCCC3)C2)=O)CC1 Cc1[nH]nc2ncc(C(=O)NC3CC(F)(CNC(C4(C)CCC4)=O)C3)cc12 CCC(C)C(CC(=O)N1CC2(C1)CC(C)(O)C2)NC(=O)C(C1CC1)OC CS(=O)(=O)C1CC(C(=O)NC2CCC2NC(=O)Cn2nnc(=O)[nH]2)C1 N1(C(c2c(C)nc(CC)s2)=O)CCCC2(CC(NC(c3cncc(F)c3)=O)C2)C1 CC1(C)CCN(C(=O)C(O)CCN(C)C)CC1NC(=O)CCc1cccc(O)c1 c1(C(=O)NC2C(CNC(c3ccc(C)n3C)=O)CC2)ccc(F)c(F)c1F C1(n2cc(C3CN(C(CCC)=O)C3)nn2)CCOC(SC)C1 c1(C(=O)NC2CCC(NC(c3cnc(C)nc3)=O)C2)cc(F)ccc1[N+](=O)[O-] O=C1NC2(CO1)CC(C(=O)NC1COCCC1NC(=O)C(C1CC1)C1CC1)C2 C1(NC(CC2CC(C(=O)OC)C2)C(=O)OCCCN(C)C)CCN(C(=O)N)CC1 C1(C2CCN(C(=O)C(CC(C)C)SC)C2)(NC(CC2CC(CC)OCC2)=O)CC1 CCCC(C)(CC)C(=O)NC(C)CCN(C(=O)Cc1coc2ccccc12)C c1(NC(c2noc(C3CC3)n2)=O)ccc(NC(=O)C(O)C2(O)CCC2)cc1 O=C(CCS(C)=O)NCCC1(CNC(c2cc(C(F)(F)F)n[nH]2)=O)CC1 c1(C(N2CC(CCNC(c3ccc(OC)cc3)=O)(OC)C2)=O)ncc(N)nc1C C1(C(=O)NCCSCCC=C)(CC)CCN(C(=O)CCC=C(C)C)C1 CC(C)(C)C1C(=O)N(C2CCOC2)CCc2cn1nn2.C1(=CCC#N)CCCCC1 C(=O)(C(O)CCC(C)C)NCC1CCC(C(=O)Nc2cnc(OCC)nc2)C1 C1(C)(C(N(CCC(=O)OCC)C)=O)CCN(C(C2CCOCC2)=O)CC1 c1(OC)c(C(N2CCCC2C(F)(F)CO)=O)ccnc1F C(C(C)(C)CNC(=O)CN(C)Cc1ccccc1)N(C(CCOCCOC)=O)C CC1C(C(=O)OC(C)(C)C)CCN1C(N1CC(c2nncs2)C1)=O C1(C(=O)NC(C2CC(C3CC3)C2)=O)C(CC)CCN1C(=O)CN(C)CC c1(CC(=O)NC(CN(C(=O)COC2(C)CCCC2)CC)C)ccccc1[N+](=O)[O-] C1(N(C(c2cnc(=N)[nH]c2)=O)CC2CCCCC2)CC2CCCC(C1)N2 C#CCC(C)(C)C(=O)NC(c1nocc1C(=O)N(C)Cc1nc(C)no1)C c1(C(N(CCCNC(C(CC)C#N)=O)CCO)=O)cnc(O)c2cnccc12 Cn1c(C(=O)NCC2(F)CC(CNC(=O)CC3CCOC3(C)C)C2)cnc1O C12(CNC(c3c(OC)ccs3)=O)CCC(CC1)N(C(c1cc(C)ccc1O)=O)C2 N1(C(C(COC)O)=O)CCN(C(c2ccccc2C(C)=O)=O)CC1C1CCC1 c1(CS(CCn2c(C)cc(C)n2)=O)c[nH]c2ccc(F)cc12 C(N=c1nc(N2CCC3(CCCO3)C2)c2sccc2[nH]1)c1c(Cl)cccc1 C1(SCC#C)CN(C(=O)CC2(OCC)CC2)CC1C(=O)NCCC(=O)OC CC1=NOC(C)(C(=O)NCCCCN(C)C(C2(C3CCCO3)CC2)=O)C1 O(C=C(C(=O)NCC(c1ccc(F)cc1)C)C1CC1)CC N#Cc1nc(NCC2CCCC2)ccc1[N+](=O)[O-] N1(C(C=CCC)=O)CC(C(=O)NC(c2cccnc2)C)CCC1(C)C C1(OC)CN(C(c2csc(O)n2)=O)CC1C(N1CCC(CC2CC2)CC1)=O C1(CNC(=O)COC2CC2c2ccoc2)(NC(=O)C(F)C2CCCC2)CCCCC1 C1(NC(C(=O)NCc2ccc(OC)cc2)=O)CC12CCC(C(F)F)CC2 C1(CNC(C(CC)COC)=O)CN(C(c2ccnc(CO)c2)=O)CC(C)(C)O1 N1(C(CNC(=O)OCC)=O)CC2CCC(NC(=O)CCS(N)(=O)=O)CC2C1 Cc1c(C(=O)NCCOC2CN(C(=O)C3=CCCC3)C2)sc2[nH]cnc(=O)c12 Cc1ccc(OCCCC(=O)NCC2COCC2NC(=O)C(=O)NC2CC2)cc1 C(=O)(CC(O)(CC)c1ccccc1)Nc1cccc(NCC=C(C)C)c1 C1(CNC(C=CCC)=O)CN(C(=O)Cn2ccnc2C(C)C)CC2(CCC2)O1 N1(C(C(CC)C(C)(F)F)=O)CCC2(CCCN(C(=O)C3=CCCCC3C)C2)CC1 C1(N(C(=O)CC2C=CCC2)CC)CCN(C(=O)C(C)(C)CF)CC1 O=C(C1=C(Cl)CCC1)NC(CCC1CC1)C(=O)NCC1(O)CCOC1 N1(C(C(C)N(C(C)=O)C)=O)CCC2C(NC(=O)CCC(C)(C)F)C2C1 N1(C(c2c(C#C)c[nH]n2)=O)CCN(C(c2c[nH]nc2C(C)(C)C)=O)CC1C1CC1 N1(C(c2cc(C)c(Br)c(C)c2)=O)C(C(=O)NCCF)CC2CCCCC12 Cc1cccc(CNC2CCCCC2C(=O)NCc2cccc(O)n2)c1Br C1(NC(=O)Cn2cnccc2=O)CN(C(=O)C(F)C(F)(F)F)CCC1F N1(C(C(Cn2cccn2)NC(C2N(C)CCC2)=O)=O)CCn2nncc2C1 c1(NC(C(=O)NC(CC(C)NC(COCCC#C)=O)C)=O)cccc(C)c1F C(=O)(C1=Cc2ccccc2OC1)N1CC2C(NC(C3=C(C)OCC3)=O)CC(C2)C1 C1(CNC(COCC(C)C)=O)CC(C(=O)N2CCC2CF)=NO1.C1CCCC1 C12(NC(c3cn(C)nc3)=O)CCCC1CN(C(c1c[nH]cc(Br)c1=N)=O)C2 c1(-n2c(C(CC(=O)ONCC3(CO)CC3(F)F)O)cnc2)ccc(Br)cc1 c1(C(=O)OC)nccc(N2CCC(OCCNC(=O)COC3COC3)C2)n1 N1(C(c2cc(SCC)ncc2)=O)CCN(C(=O)C(O)C(F)(F)F)CC1CC(F)F C(C)(C)(C(=O)NCc1nc(CNC(=O)Cc2csc(S)n2)cs1)OC(C)=O C(C)(CCC(=O)N(C)CCN1CCN(C(=O)CSC2CCCCO2)CC1)OC C(=O)(CCC(C(C)C)NC(=O)C(C)CO)N(CCCO)CCC Cc1ccc(CC(=O)NCC2CCCCN(C(C3CCCO3)=O)C2)cc1C N1(CC(=O)N(C2CN(C(C3(c4cncs4)CC3)=O)CC2F)C)CCCS1(=O)=O c1(OC)ccc(C(=O)NC2CCC2NC(=O)Cn2nc(C)cc2C(F)F)c(Cl)n1 C1(CCC)(CO)CCN(C(=O)C(C2CCOC2)NC(=O)C(C)=NOCC#N)C1 C(=O)(CCC(CC)OC)NCCCCc1c(CC)onc1C.C1(=O)CCN1 C=CC1OCCC1C(=O)NC(C)CNC(=O)CP(C)(C)=O Cc1ccc(Cl)c2[nH]c(C(=O)NCCOCCCNC(C3CCC4CC34)=O)cc12 c1(C(C2(C(C)C)CC2)NCCC2CC(OC)C2)nnnn1CC1CCCO1 CN(C)NC(=O)CCC(=O)N1CC2CC1C2C(=O)NCC1CCC(F)(F)C1 N1(C(CCC)=O)CCC(c2ccc(C(=O)NCC3CC(O)CN3C)cc2)CC1 S(=O)(=O)(c1cc(Cl)ccc1F)N1C(C(N(CC(=O)N(C)C)C)=O)CC(F)C1 C1(CC(=O)NC(C)(C)CCNC(C2(Cl)CC23CCC3)=O)Cn2ccnc2NC1=O C1(C(C)C)(C(=O)NCC(C)CNC(=O)COc2ccccc2Cl)CCN(C)CC1 c1(CC)[nH]c(C(=O)NC2CN(C(C3(N4CCCCC4)CCCC3)=O)C2)nc1Cl C(C)(CCCC(=O)Nc1ccc(SC)cc1)NC(C1(C)CC(=C)C1)=O N1(C(CC2OCC(C)(C)C2)=O)CCC2(CCCN2C(C2CN(C3COC3)C2)=O)C1 Cc1nnc2n1CC(C(N1CCOCC(CNC(=O)CC(C)C)C1)=O)N(C)C2 N1(C(CC=C)=O)CC(NC(=O)Cc2cncn2C)CC1C C1(N(C)C(C2CCCN(C(c3ccc(C(F)(F)F)[nH]3)=O)C2)=O)CS(=O)(=O)C1(C)C c1(C(N(C)CC2(O)CCN(C(C(C(C)O)(F)F)=O)C2)=O)cnc2c(cnn2C)c1 c1(-c2ccc(COc3ccc(C(c4ncon4)F)cc3)o2)ccc(F)cc1 C(CCC(C)(C)C(=O)NC1CCC1)NC(CCC(C)OC)=O N1(C(C2CCC(C)O2)=O)CCN(C(=O)C(C)(C)c2cnc(C3CCC3)o2)CC1 CC(C)(O)C(F)C(=O)NCCC(O)CNC(C1CN2CCN1CC2)=O N1(C(N)=O)CCc2nc(O)cc(-c3ccccc3)c2C1.C1(=O)CN1C(N)=O NS(=O)(=O)c1sccc1C(=O)NCC1C2CCCC1N(C(c1cnco1)=O)C2 CC1(C(N2CC3(CCC3NC(c3cccc(Cl)c3F)=O)C2)=O)CCCS1(=O)=O N1(C(c2n(CC)ccn2)=O)CC(CC2CC2)C2(C1)CN(c1cc(O)nc(C)n1)C2 C1(=O)CC(CC)N1.C=C1CC(N(C)C(C2(COCC)CC2)=O)C1 c1(OC)ccc(C(C)(C)C)c(OC)c1.c12cc(ccn1)CNC2=O C1(CNC(C2C(CC)N(C)CC2)=O)CCC12CCN(C(c1oncc1C)=O)CC2 C=CCC(CC=C)C(=O)NCC1C(C)CCCN1c1cc2nncn2cn1 n1(CCCOC)c(N2CCCC2)nnc1C(C1CCC1)(C)C.c12nnc(o1)C2 Cc1ccc(C(N2CC(=C(F)CNC(=O)CC3CNC(=O)O3)C2)=O)c(O)c1 C1(NC(C(C)OC)=O)CN(C(c2ccnn2CC(C)C)=O)CC1CC(C)(C)C c1(C(=O)NC2CCCN(C(C3(CF)CC3)=O)CC2)ccc2c(O)n[nH]c2c1 c1(COC)ccc(C(=O)NC2CCCCC2NC(c2cnc(CN)o2)=O)cc1F c1(N2CC3CC(NC(C=Cc4c(C)ccnc4)=O)C3C2)ccnc(C#N)n1 C(=O)(C1=CCC(F)(F)CC1)N(CCC)CCNC(=O)CC1CC2CCC(C1)N2C N(C(=NCC1CCOC1)NCC(c1cccnc1)O)CC1(C=C)CCC1 c1(OCC)ccc(C(N2CCCC(C(=O)NC34CC(CO3)C4)C2)=O)cc1C CCC(C(=O)N1CC(O)(CCNC(C2CC(c3ccccc3)C2)=O)C1)OC n1(CC(=O)N(C(C(=O)N(C2CSC2)CC=C)C)C)cc(C)cn1 N1(C(CC(=C)C)=O)CC(NC(=O)C(C)OCCOCC)CC1CO Cc1nn(CC(C)C)c(Cl)c1C(=O)NCC(C)CN(C)C(C1(C)CC1(F)F)=O CC(F)(CNC(=O)C(N)c1ccoc1)Cc1ccccc1 c1(CNC(COCC#C)=O)cccc(NC(c2cncnc2CC)=O)c1 C(=O)(CC(C)(C)F)N(C1CCN(C(c2sc(CC)nc2C)=O)C1)CCC c1(CC)ncsc1C(=O)N(C1CCN(C(=O)CCc2cnc(C3CCC3)o2)C1)C Cc1nc(C)c(C(=O)NC2(C(=O)NC(C)CN(C)C)CC2(C)C)o1 N(C(=NCC1CCOC1)N(C)CC(C)C#N)(C(C)C)CCn1ncc(Br)n1 c1(C(=O)N(CC2CCN2C(=O)Cc2csc(C3CC3)n2)CC)cnc2ccnn2c1 C1(O)(c2c(CNC(CCCC)=O)nco2)CCN(C(c2n[nH]c(C3CC3)c2Cl)=O)C1 c1(C(N2CCC(NC(=O)NC3COCOC3)C2=O)C)ccc(Br)cc1 C1(CNC(C2CCCN(C(N)=O)C2)=O)CN(C(=O)CN2CC=CC2)CC1(F)F C1(NC(C)=O)C=CCN(C(=O)C=CC(=O)NCC2CC2)C1.C12CCN(C1)C2=O c1(NC(C2(CNCc3c(C)noc3C)CC2)=O)ccc2n[nH]cc2c1C Cc1c(C(=O)NCC(C)(O)CNC(=O)C=C(Cl)Cl)[nH]c2c(C)cccc12 C1(CC(=O)NCCCN(C(C2C(=C)C2)=O)CCO)COC(=O)C1 C1(C(=O)NC(C(=O)OCC)C2CC2)CCCCCCN1C(C1C2CCC(F)C12)=O C1(N(C(=O)C(C)C2CCC2)CC#C)CCN(C(C2CC2(Cl)Cl)=O)CC1 N1(C(c2cscc2Br)=O)CCN(C(c2n[nH]cc2F)=O)C2CC12 C1(C2CCCN(C(c3ccc4c(c3)COCC4)=O)C2)(NC(=O)C2=CCC2)CC1 c1(NC(c2cc3c(s2)CCCC3)=O)cnc2ccsc2c1 CC1c2c(Br)cccc2CCN1C(=O)NCCc1ccc(F)cc1F N1(C(c2cccc(SC)c2)=O)CC(NC(c2ccc(Br)c(Cl)n2)=O)C(F)(F)C1 c1(C(=O)NC)cccc(-c2cccc(N3CCCS3(=O)=O)c2)c1 CCCC(O)CN(C(=O)CCCNC(c1c[nH]nc1CC)=O)C C(CCCC(C)NC(=O)CC1(CO)CC1)NC(C(CC)Sc1ccccc1)=O N1(C(C2ON=C(C)C2)=O)CCN(C(c2cccc(F)c2O)=O)CC1CC(F)(F)F C1(C#N)(C(=O)NCC2N(C(C3ON=C(C)C3)=O)CCC2C)CC2C=CC1C2 C(=O)(C1=C(C#N)CCC1)NC(C1CCCN1C(c1cnn(CCF)c1)=O)C c1(OC)ccc(N(C(c2ccc(OC)nc2)C(=O)NC2CCCCC2)C)c(C)c1 Cn1cc(C(=O)NC2CCCCN(C(=O)C3=COCC3)C2)c2ccccc2c1=O c1(OC)cc(C)c(Cl)cc1S(=O)(=O)N1CCCC(NC(c2ccnnc2O)=O)C1 C1(CCC(=O)NC2CCC(CNC(C3CCC3)=O)C2)(N(C)C)CCCC1 N1(C(=O)CCc2ccc(C(F)F)cc2)CCCC(C2CCNCC2)CC1 CCC(CC(=O)N1CC(C(N2CC3CCC(C2)N3C)=O)CC1(C)C)C(C)C N1(C(C)=O)CCc2c(NC(c3csc(-c4cn[nH]c4)n3)=O)cccc21 N1(C(c2nccs2)C)C(=O)NCC(N2CCCSCC2)C1=O Cc1cc(C(N2CCC23CN(C(c2ccc(C4CCC4)cc2)=O)C3)=O)cc(Cl)c1 O=c1cc(CN2CC(CO)OCC23CC3)oc2ccncc12 c1(N(C(C)C)C(c2cccnc2)C)ncc(Br)c(N(C)C)n1 c1(SC)ncc(Br)c(N2CCC(CNC(=O)C(F)CC3CCCCC3)C(C)C2)n1 N1(C(Cn2c(=N)nc[nH]2)=O)CCC2(NC(=O)CCc3cccc(F)c3)CC2C1 C12(C(N3C(C(=O)OC)CCCC3)=O)COCC1CN(C(C1OC3CCC1C3)=O)C2 N1(C(c2cc(C)cc(Cl)c2)=O)C2CCC1CC(NC(C13CCCC1C3(F)F)=O)C2 C1(C(=O)NC2C(SC)COC2)CCCCN1C(c1cc(Cl)n(C)n1)=O C(=O)(C(C)(CSC)NC(=O)COCCSC)NCCCCC(=O)OC CC1CN(C(=O)Cn2cnnc2)CCC1N(C(=O)CCC(=O)N(C)C)C Cc1cc(C(=O)NC2CN(C(c3cnc(C#N)s3)=O)CC2CO)ccc1C(C)C N#Cc1cc(CN2CCC(C(=O)Nc3ccc(Br)c(Cl)c3Cl)C(O)C2)cc(F)c1 N1(C(CC(C(C)(C)NC(C(CC=C)OC)=O)C)=O)CCC(C2CCCC2)C1 C=Cn1nccc1C(N1CC(NC(=O)CC2CC(OCC)C2)C(COC)C1)=O C12CN(CCO1)C(=O)NC2C.C1(OC(C2CC(OC)C2)=O)=CC=CCCC1 N1(C(CCC(C)=O)=O)CC2(C)CC1(C(=O)NC1C=CCCCC1)C2 c1(C(N2CCCC3(NC(C4C(=C)CC4)=O)C(C2)C3)=O)cnc2c(Cl)cccn12 N1(C(c2cn(C(C)C)nn2)C(=O)NC(C)C)CCc2cc(F)cc(F)c2C1 N1(C(C(C)P(C)(C)=O)=O)CCCC2(CCN(C(C3CC(OC(F)(F)F)C3)=O)C2)C1 c1(C(N2C(CN(C(CN(C(C)C)C)=O)C)CCC2)=O)cnc2ncccn12 n1(CC(N2CCC(N(C(=O)CCC3CC(OC)C3)CC)C2)=O)nc(C)c(Cl)c1C c1(NC)c(C(N2CCC(C3N(C(=O)C(C)OC)CC3(C)C)CC2)=O)cccc1N c1(OCC)ccc(CC(=O)NCC(C)CN(C(=O)CCN2CCC(F)C2)C)cc1 N1(C(c2cnc(C(C)=O)s2)=O)CCC(NC(c2c(C)cnn2C(C)C)=O)C(C)C1 C1(CNC(CS(C(C)C)(=O)=O)=O)CC2(CCN(C(=O)CCCC#N)CC2)CO1 C1(NC(C(C)n2cccc2)=O)CCN(C(C2(C(C)(C)O)CC2)=O)CC1C c1(C(=O)NCCCNC(C2CC23CC(O)C3)=O)ccnc2[nH]ncc12 Cc1cc(C(=O)N(CC(C)N(C)C(C2CC2C(F)(F)F)=O)C)nn1C(C)(C)C Cc1nc2cc(C(N3CC(NC(=O)COC4CCCCC4C)C3)=O)ccc2o1 C1(C)(CNC(Cc2cn(CC)nc2)=O)CCCN(C(=O)COCC2CCOC2)C1 C1(C(N(C)CC2CCCC2)=O)CCN(C(=O)C(O)CC(F)(F)F)C(C)(C)C1 N1(C(C2CCN(C(C)=O)CC2)=O)CCC(CNC(=O)Cc2n[nH]cc2Br)CC1C N1(C(C(C)(C2CCC2)NC(c2c(C)csn2)=O)=O)CC(C)C12CCOCC2 C1(O)(C(N2CCC(CNC(c3cnc(COC)s3)=O)C2)=O)CCCCCC1 N1(C(CC(C)C2CC2)=O)CC2(C(N3CCCC3CCC(=O)O)=O)CCC1CC2 CC1OCCC1(C)C(=O)NCC(CO)NC(c1cccc(N2CCCC2)c1)=O N1(C(C2(C(=O)OC)CC=CCO2)=O)CCC(CNc2c(OCC)nsn2)C(C)C1 Cc1cnc(C(N2CCCC(C(N3CC(F)(F)CC3C)=O)C2C)=O)c(F)c1 CCCCS(=O)(=O)NCC(=O)NCC(C)(C(C)C)NC(=O)C(=O)Nc1ccc[nH]1 c1(C(N(C)CCN(C)C(C2(C)CCC(=O)NC2)=O)=O)cc([N+](=O)[O-])c(O)cc1N Cn1cc(SCC(=O)N(C2CC2)CC2CCCN2C(=O)C(O)CF)cn1 c1(N(CCOC(C(C)Oc2ccccc2)=O)C)nc(Cl)ncc1Cl C1(NC(c2cnc(C(C)=O)s2)=O)CN(C(=O)C(C)SC(C)C)CC2(CC2)C1 C(C(CC(F)(F)F)NC(C1CCCCC1O)=O)NC(c1ccnn1C(F)F)=O N1(C(c2n(C=C)ncc2)=O)CCCC2(NC(=O)C(CCC)CCC)CC2C1 n1(CCC(=O)NCCNC(C(C(C)SC)O)=O)cc([N+](=O)[O-])cn1 CCCCC(C(=O)NCC(C1CCC1)NC(=O)CNS(C)(=O)=O)N(C)C n12cc(nn1)CC(=O)N1CC2C1.c1(COCC)cn(NC(C2CCCCS2)=O)nn1 c1(C(C(C)N(C(=O)CC(c2ccc(F)cc2)C)CC)=O)ccc(F)cc1 N1(C(C2CC3(CC3)CN2Cc2c(C(C)(C)C)[nH]cn2)=O)CCn2cc(O)nc2C1 N1(C(C2C3(CC(NC(c4cc(C5CC5)no4)=O)C3)C2)=O)CC(F)(F)C(F)(F)C1 C1(C(=O)NCC2CCCN(C(c3cnc(C4CC4)o3)=O)C2)CC2(CCCC2)CO1 CC1CCCCCC1OC(C)(C)C.C12(C)CCCN1C(=O)C(CN)NC(=O)C2 N1(C(C(CC)=CC)=O)CCC2(CCCN2C(=O)C(C)Sc2ccccc2)C1 C(CO)(CO)(CN=c1[nH]c2c(c(=NCc3cc(Cl)n(C)n3)[nH]1)SCC2)OCC c1(CC)c(C(N2CC(NC(c3cc[n+]([O-])cc3)=O)C2)=O)[nH]c(C)c1C(C)=O C1(CC2CNC(=O)NC2)(CNC(C)C)CC=CCC1.C(C)(C)(C)O.C(=O)NC c1(CC(=O)N(C2CCCCN(C(C3C(=C)CC3)=O)C2)C)ccc(C)c([N+](=O)[O-])c1 CN1CC(C)(C(=O)NCc2n[nH]cc2C(=O)NC2CN(C)CC2O)CC1=O c1(C(N2CCC(c3ccc(C(F)(F)F)cc3)C2)=O)ccc(O)c(C(=O)OC)c1 C(=O)(C1CCCc2cccnc21)N(C)CC1CCCN1C(C1(C)CC(C#N)C1)=O C(=O)(C1=CC2(CCOC2)C1)NC1(CO)CCCN(C(C2(COC)CC=CC2)=O)C1 c1(C(C(=O)NCC(C)CC2(C(F)(F)F)CCCC2)(F)F)cc(F)cc(F)c1.C1CN1 C1(C(=O)NCC2(NC(=O)CC3CC4(CCO3)CC4)CCC2)CCC2(CCC2)CO1 c1(C(=O)NCC2(C(=O)NCc3nc(COC)on3)CC=CC2)cc(C)nn1CC C(CN=c1nc2c(cnn2C)c(NCc2cccnc2)[nH]1)C1C(C)C1 N1(Cc2cn(CCCCOCc3cc(NC(=O)OC)on3)nn2)CCCCC1=O C12C3CC4CC1CC(C4)(C3)NC(=NC)N2.c1(OC)c(Br)cnn1C.N12CC1C2 N=c1[nH]c(-c2cccs2)c(CC(N2CC(NC(C3CCC(CO)CC3)=O)C2)=O)s1 c1(CC)cc(C(=O)NCC2C=CCN2C(=O)CCC(=O)OC(C)(C)C)sc1C c1(CN(C(c2ccc(C3OC(=O)NC3(C)C)cc2)=O)CC)cnn2c1CCCN2 c1(OC)cc(Cl)cc(F)c1C(=O)NCC1CCCN1C(c1cccc(Cl)c1F)=O CCCC(CC)CCC(=O)N1CC(NC(=O)C(CCC)N(C)C)C2(CCCC2)C1 C1(N(CCOC)C(c2cnc(SC)[nH]2)=O)CCN(C(C2CCC3CC23)=O)CC1 Cc1cc(C(N2CCC(F)(CNC(C3CSCCS3)=O)C2)=O)c(C)n1C(C)C c1(C(=O)NC2CCCC(NC(C(C=C)(C)C)=O)CC2)cc2n(c1)CCCC2 c1(C(=O)NCC2(CNC(C3(C)CC3Br)=O)CCCC2)nccc(Cl)c1O c1(C(N2CC3C(NC(c4n[nH]c(C5CC5)n4)=O)(C3)C2)=O)ccc2nncn2c1 C(C(CNC(=O)C(c1cncc(F)c1)C)C(F)(F)F)NC(c1c(C)nn(C)n1)=O N1(CC(C)C)CC2(C)CN(C(=O)CC3CC3(C)C)CC2(C)C1 c1(C(N2CCSC(C(C)C)C2)C(=O)NCC)cccc(OCc2ccccc2)c1 n1(CC(CC)O)cnc2c(N3CCC(CO)=C(F)C3)ncnc12 c1(N2CCCC(C(N)=O)C2)nccc(=NCCC2(C(F)(F)F)CCC2)[nH]1 C#Cc1ccc(C(N2CC(OC)C(C(N3CCOC(CC(C)C)C3)=O)C2)=O)cn1 C(=O)(CC(O)CCSC)NCCCNC(C)=O c1(CNC(=O)C(O)C2CN(C(=O)CC(Cl)Cl)C2)ccccc1 C12(CNC(=O)COC3CCCOC3)CC(CO1)N(C(c1c(Cl)ccnc1F)=O)C2 c1(-c2n(CCC=C)nc(-c3cccc(C(C)OCC)n3)n2)cc(C)n(CC)c1C c1(C(=O)NC2CCN(C(CCCCNC(C)=O)=O)C(C)C2)cnc2[nH]cnc2c1 Cc1nnc(CCC(=O)NCC(C2CC2)NC(=O)Cn2nnnc2C)o1 C1(C(N2CCCC(O)(CNC(c3ccncc3F)=O)C2)=O)CCn2nccc2C1 CC1(C)C(CC(=O)NC)CC1O.n1(C2(N3CCCC3)CC2)cc(-c2ccccc2)nn1 CC(O)C(F)(F)C(=O)N1CC(CCCCNC(C2CN(C)CCCO2)=O)C1 c12csc(n1)CNC2=O.n1(CC(C2CCOC2)OC)cc(-c2cc[nH]n2)nn1 c1(OC)ccc(C(N2CC(CC(C(C)C)C(C)C)C2)=O)c(OCC(C)C)c1 N1(C(CNS(N)(=O)=O)=O)CCC(NC(=O)C(C2CC2)Sc2ccccn2)C(O)C1 c1(CC(=O)NC(CCNC(C2C(CCC)C2)=O)(C)C)cc(C(F)(F)F)n(C)n1 N1(C(C(=O)Nc2c(Cl)ccc(NS(C)(=O)=O)c2)=O)CCn2nncc2C1 C(=O)(CS(=O)(=O)C1CC1)N1C2C(NC(c3cnc(C(C)OC)s3)=O)C(CC2)C1 C1(NC(c2nnc(CC)s2)=O)CC2CCC1N(C(=O)CCCN1CCCC1)C2 C(=O)(CCCCC(C)(C)C)N(C1CCN(C(C2CC(CF)C2)=O)CC1)C C1(F)(CNC(CN(C(C)=O)C)=O)COCCN(C(=O)C(C)(C)CO)C1 N1(C(C)C)CC(CN(C)C(c2ccccc2CSC2(C)CCC(=O)N2)=O)CC1=O C1(CC=C)(NC(C2CCCC2(F)F)=O)CCCN(C(c2sccc2C#N)=O)C1 C(=O)(CS(=O)(=O)CCOC)NC1CCN(Cc2cnn(CCC)c2C)C1 C1(C(=O)NC(C)CN(C)C)(CC)CN(C(=O)C(C)c2ccsc2)C1 c1(OC)ccc(CN2CCC(O)C(C(=O)NC(c3ccc(I)cc3)C)C2)nc1Br C=CCCC(C(=O)NCCCCC(=O)NCC(C)(C)CC(C)C)C(C)C N#CC1CCC(C(=O)NC2CC(NC(=O)C(c3ccccc3)O)C2)CC1 Cc1ocnc1C(N1CC(C(C)(C)C)C1)=O c1(C(=O)NCC(CN(C(c2c(CC)cncc2)=O)C)O)cc(C)cnc1C(C)C c1(NC(C(=O)N(CCN(CC)CC)CC)=O)nccs1 N1(C(c2c(C)[nH]nc2Br)=O)CCC(NC(=O)CCc2ccsc2)C(CO)C1 C1(NC(c2c(CC)nc[nH]2)=O)CC(NC(=O)CCCn2cccc2)C12CCC2 C(C(C)N=c1nc(N2CCCCC(CO)C2)c2sccc2[nH]1)SC CC(C(=O)NCCC1CC(NC(=O)COCC2CCOCC2)C1)C(F)F C(=O)(C(O)CC(F)F)N(C1C2CN(C(COC(C)C)=O)CC21)C C(=O)(CC(C)C(=O)OC)N1CCC(N(C(=O)CC2CC(C)=NO2)CC)C1 c1(C(=O)NC(CCC)C(=O)NC2COCC2C(N)=O)cc(C)nc(O)n1 N1(C(c2ccc(CC)nc2)=O)CC(CNC(c2sccc2C)=O)CC12CCC2 N1(C(c2cc(C)[nH]n2)=O)CC2CC1CC2NC(=O)C(C)NC(c1ccco1)=O N1(C(Cc2c(C(=O)OC)csc2)=O)CCOCC(NC(c2cnc(S)n2C)=O)C1 c1(C(=O)NCC2N(C(c3c(CC)ocn3)=O)CCC2)ccc2c(c1)SCC(=O)N2 N1(C(c2c(C)ccc(Cl)c2)=O)CC(NC(=O)CC2CC(C)(C)C2)C(C2CC2)C1 S(=O)(=O)(c1ccc(Cl)c(Cl)c1)N1CCC(CN(C)Cc2cccc(F)c2)C1 c1(CNC(C2CC(C(F)F)(NC(C(C)SCCCC)=O)C2)=O)cccc(OC)c1 C(CCC(C)C(=O)NC1CN(C(c2ccc(-c3cccs3)[nH]2)=O)CC1C)OC C12(C(=O)NCC(C(C)(C)C)NC(=O)CCn3ccnc3)CCC(O)C1CC2 CC(CCNC(=O)OC(C)(C)C)N(C)C(C1(Br)CC1C(=O)O)=O c1(CC)cc(C(=O)NC2CCCCC2CNC(C2(C#N)CCCO2)=O)cc(O)n1 c1(NC(c2c(CC)[nH]cc2)=O)cccc(NC(C2CCCC(C(F)(F)F)O2)=O)c1 N1(C(c2cnc(OC)s2)=O)CCN(C(C23CC(C)C2C3)=O)CCC1C C1(OC)CCC2CN(C(C34CC3CCN4C(c3c(C)cccc3F)=O)=O)CC12 Cc1[nH]c2ccc(C(=O)O)cc2c1-c1cn(C2C=CCN2)nn1 c1(C(=O)NCC2CN(C(C(CC=C)C)=O)CC2C)ccc2c(c1)CCCS2 N1(C(C2C3CN(C)CC32)=O)CC2(CC(C(N3CC4CSCC(C4)C3)=O)CO2)C1 C1(C(C)O)CCN1C(C1(CNC(=O)CCn2ccnc2)CC1)=O c1(CC(=O)N(C2CCN(C(=O)C=Cc3cnc[nH]3)C2)CCC)cc(C)ns1 N1(C(C(C)OCCC=C)=O)CCC(C(=O)NCCCSCC(=O)NC)C1 C1(F)(CNC(C2CCC(O)C2)=O)CCC(CNC(C2CC(O)C2)=O)C1 C1(CC)CC2CCCC2N1C(=O)N=c1nc(C2CCOCC2)[nH]s1 C1(CCC(C)C)CCC(NC2CCCN(C(=O)OC(C)(C)C)C2)CC1 c1(C(N2CCC(C)C2c2cn(CCF)nn2)=O)cc(F)c(F)cc1Cl C1(CC(=O)NCc2c(NC)nccc2)CC(C)(C)CN1C(C1CC1C(C)(C)C)=O C(C(CC)C(C)C)(c1n(CCOC)nnn1)Nc1nccn1Cc1ccccc1 C1(NC(CCC#N)=O)CCN(C(=O)C=Cc2cccc(Cl)c2)C12CC2 CCC(O)C(C)C(=O)NCC1CCC1NC(=O)CSc1ccc(Cl)s1 N=S1(=O)CCN(C(C2CN(C(C3CCC(C4CC4)C3)=O)CC23CC3)=O)CC1 N1(C(C(C(=C)C)(C)O)=O)CC(NC(=O)C2=COCC2)CC2(CCOCC2)C1 C1(C(=O)NCCCC=CC(C)C)Cc2ccccc2S1 CP(C)(=O)CN1CC(C(N2CCC(NC(C34CCC(C3)C4)=O)C(F)C2)=O)C1 N1(C(Cc2c(OC)ccnc2)=O)CCCC2(C1)CN(C(=O)C(C)(O)C1CC1)C2 C1(NC(c2ccc(CN(C)C)[nH]2)=O)CN(C(=O)CNC(=O)C2CC2)CC1C1CC1 N1(C(CS)=O)CCN2C(C1)c1c(cccc1)CC2=O.C(CN(C)C)OC C1(CC(=O)N(C2CCN(C(CCc3scc(C)n3)=O)CC2)C)CCCC(C)(C)O1 O=[N+]([O-])c1cccc(C(O)CNC2CC(Cc3ccc(Cl)cc3)C2)c1 C(CC(C)NC(=O)COC)N(C)C.C1(CC(=O)NC2CC(CF)C2)CCOC1=O C(=O)(C1=CCCN(C(=O)CC2NC(=O)NC2=O)C1)N(CC(C)O)CC(C)O Cc1nc(C(C)NC(=O)C(CNC(=O)CCC=CC(C)C)N(C)C)no1 N1(C(C)=O)CCC(CNC(=O)CC2CC(NC(=O)C=CCn3cncn3)C2)C1 CC1(C)CC(CNC(=O)C=Cc2cnc[nH]2)CN1C(=O)C(O)CC(N)=O c1(CC(=O)N(C2CC(NC(c3c(CC)n[nH]c3)=O)C2)C)cc(OC)ccc1Cl c1(NC(=O)NC2CC(CS(C)(=O)=O)C2)ccc(O)cc1[N+](=O)[O-] C12=CC(=NC(C)C3CCN(CC3)C1=O)NC(C)=N2.c1(CC)cc(OC)cc(O)c1 C1(NC(C2CCCS2(=O)=O)=O)CC12CCN(C(=O)C=CC(F)(F)F)CC2 c1(C(=O)NCC2CC3(CC(NC(C4CC4(F)F)=O)C3)C2)ncc2cc(Cl)ccn12 N1(C(C(=O)NCC=C)CC2CCCO2)CCCC(O)(CO)C1 N1(C(C=CC=CC)=O)CCC(C2CCN(C(C3CCC(C(N)=O)CC3)=O)C2)C1 N1(C(CCNC(C)=O)=O)CCCCC1CC(C)NC(c1cnn(C2CCC2)n1)=O N1(C(CC(C)c2ccco2)=O)CC(C2CN(C(c3ccc4c(c3)CCO4)=O)C2)C1 N1(C(c2nc(C(=O)OC)sc2)=O)CCC(O)(C(C)NC(C2CCCC2O)=O)CC1 C(=O)(CC1=CCN(C)CC1)NCC(C)(CNC(=O)C(c1c(C)noc1C)C)OC N1(C(C(CC)CC(C)C)=O)CCC(C2(NC(=O)CSc3nncs3)CC2)CC1 C=C(C)CCCC(=O)N(CCC)CCNC(c1ccc(C)cn1)=O Cc1cnc(C(=O)NC2CC(C)CN(C(=O)C(C)(C)CC3CC3)C2)c(F)c1 Cc1ccsc1C(N1CC(O)(C(C)NC(C2CCCC2c2cnn(C)c2)=O)C1)=O C(=O)(CC(O)CC(C)(C)C)NCCn1c(C(=O)NC(C)Cc2nc[nH]n2)ccn1 c1(CN2CC3C(C(F)(F)F)C3C2)cc(Br)ccc1NC(=O)NCCS(CC)(=O)=O N1(C(c2n(C)nc([N+](=O)[O-])c2)=O)CC2CC(NC(C3CCC(=O)N3)=O)CC1C2 C1(C(C)C)CCC(C(=O)NCCCCCn2cc(C(C)C(=O)O)nn2)CC1 C1(C(=O)NC2(C)CC(NC(CS)=O)C2)CCC(C)(C)CO1.Cn1ccnc1CN Cc1nn(C)c2c(NCc3c[nH]c(=N)s3)nc(N3CCC4C(CCN4C)C3)nc12 N1(C(N)=O)CC(O)CC1C(N1CC(OCCNC(=O)C(C2CCCCC2)O)C1)=O C1(C(=O)NC(CNC(CCOCCOC)=O)CC)CCc2nc(C)ncc2C1 C1(C(N2CC(C)(NC(=O)COCC3CCCOC3)C2)=O)CC2CCC1NC2=O c1(C(=O)NC2CC(F)C2)cc2cc(F)ccc2s1 N1(C(C=Cc2n(CC)ccn2)=O)C2CCCC1CN(C(C1CCNC1=O)=O)C2 c1(NCCc2cc(C)ncc2)cc(=NCCOc2ccncc2C)[nH]c(C)n1 N1(C(c2c(Cl)cn(CC)n2)=O)C(C)CN(C(=O)C(n2ccnc2C)C)CC1C C1(C(N2C(C)CSCC2)=O)CCN(C(=O)CC2(C#N)CC2)CCO1 C1(NC(c2cc(C(=O)OCC)[nH]c2)=O)(CNC(C2CCC2(F)F)=O)CCOCC1 CC12CC(C(=O)NCC3(C)CCN(C(=O)COc4ccsc4)C3)(CCO1)C2 c1(OC)ccccc1CCCNC(C)CF C1(C(=O)NCC2N(C(CSC(C)C)=O)CC(O)C2)CCc2ccccc2O1 Cc1c[nH]cc(C(=O)NC(C)C(CO)NC(=O)Cc2ccc(F)cc2Cl)c1=O c1(CC(N2CC(C(C)NC(=O)CCN3CCOCC3)C2)=O)nc2c([nH]1)CCCC2 C1(NC(CCCC#C)=O)CCC2(CC1)CN(C(C13CCCC(CO1)C3)=O)C2 N1(CCN(C(=O)C(C)(Cl)Cl)C)CCN(C(=O)CCC2CCCC2)CC1 c1(OC)cc(C)c(CS(=O)(=O)Cc2c(C)cccc2Br)cn1 C12(CS(=O)(=O)N(CCC#N)CC3CCC3)CC3CC(CC(C3)O1)C2 c1(OCC)nc(N2CCC(NC(c3ccc([N+](=O)[O-])[nH]3)=O)C(O)C2)ncc1Cl Cc1nc(C(=O)NCCC2(O)CN(C(=O)CC3CCC(C)(C)CC3)C2)cc(O)n1 C1(CC(=O)N(CC(=O)NC(c2noc(C)n2)CC)CC2CC2)CCC(C)(C)O1 C1(NC(CCCCCN(C(=O)CCn2ccnn2)C)=O)CCN2CCCC2C1 C1(NC(C(COC)O)=O)CN(C(=O)CC2CC(C(F)F)C2)CCC12CCOCC2 c1(C(=O)NC2CN(Cc3ccc(OC)cn3)CC2F)ccc(OC)c(Cl)c1.N(C)(C)C CCC(CC)CC(F)C(=O)NCC(C)C(=O)N(C(COC)COC)C CN1CCN(C(=O)CC2CC3CC3C2)CC1CNC(C12CC1COC2(C)C)=O C1(C)(CC)CCN(C(=O)CC2COCCN2C(=O)Cc2cnsc2)C1 c1(CNC(=O)NCC2OCCc3ccccc32)csc2cccc(Cl)c12 N1(C(C2N(C)CCCC2)=O)CCC2(C1)CN(C(C1CCC(C(N)=O)O1)=O)C2 N1(C(C(=C(C)C2CC2)F)=O)CCC(NC(c2cnccn2)=O)CC1C Cc1cc(Cl)ccc1C(=O)NCCCCC1CCCN(C(=O)Cc2ccsn2)C1 c1(N2CC(NC(CCC(=O)OCC)=O)CC(F)(F)C2)ncnc2c1ncn2C C1(N(C(C=C(C)C)=O)CC2CC2)CCCN(C(=O)CC(C)n2cccn2)C1 C(=O)(C(C)S(C)(=O)=O)N1CC(C(C(=O)NC2C(C)C2C)OC)C1 C1(C(N2CC(OCCNC(c3ncc(N(C)C)nc3)=O)C2)=O)CCC12CCCO2 CCCCC(F)C(=O)N1CC(C(O)C(=O)NC2C=CCCCC2)C1 N1(C(c2c(COC(C)=O)nccc2)=O)CCN(C(c2c[nH]cc2C)=O)CC1CO C(C)(N=c1nc2c(ncn2C)c(N2CCOC(CF)C2)[nH]1)c1ccc(C)cc1Br Cc1n[nH]c(C)c1C(=O)NC1(CNC(=O)CCc2cnc(O)[nH]2)CCCC1 C=Cc1ccc(CC2=NOC3CCCN23)cc1.c1(Nc2ccccc2)ccc(O)cc1 N1(C(C2C(C)C2C)=O)CCN(C(=O)CN(C)C2CC2)C(C(F)F)C1 C1(CC)CN(C(=O)NC2(CNC(=O)CCn3cccn3)CC2)C(CC)CO1 N1(C(c2c(CNC(CCCC)=O)noc2)=O)CCC12CCN(C)C2 c1(C(=O)NCC2C(CNC(c3nc(C)c(C)s3)=O)C2)cccc2c1COCCN2 C1(NC(C2(SC)CC2)=O)CN(C(c2noc3cccc(C)c23)=O)C2CCCCC12 Cc1cnc(C=CC(=O)NC(C)(CNC(c2ncccc2O)=O)C2CC2)[nH]1 C1(n2c(-c3cc(C)n(-c4ccc(F)cc4)n3)nc(SC)n2)CCCCC1(C)C C(C)(C)(CCCCNC(c1cnc(C)nc1C)=O)NC(c1c(SC)ccs1)=O N1(C(C(C)CC2CCC2)=O)CCCC(CCNC(=O)CCc2ccc(F)nc2)C1 N1(C(c2cnc[nH]2)=O)CC2CCC1CN2C(c1ccc(-c2ccncc2)o1)=O C12(CNC(CN(S(CC)(=O)=O)C)=O)CC1CN(C(=O)Cc1cnoc1)C2 C(=O)(C(CNC(=O)C(C)CC)C(C)(C)C)NCc1cnc(COC)[nH]1 CCCC(CCN)=CC(N1CCCC(CN(C)C(C)=O)C1)=O C(=O)(Nn1nnc2c1CCCC2)C1(C=C)CCN(C(=O)CCC2CC2(F)F)C1 c1(OCCCC)ccc(S(=O)(=O)N2CC3CCC(C2)N3C(=O)C(C)C)cc1 N1(C(C(C)N=[N+]=[N-])=O)CCCC(N2CCOC2=O)CC1.C(=O)C(F)(F)F CC1Cc2cccc(C(=O)N(CCCNC(c3cnn(C)n3)=O)C)c2O1 C(=O)(C1=Cc2ccccc2C1)N1C(C)CCN(C(C=C(C)C)=O)CC1 C1(F)(CNC(C(C)CC2CCCCC2)=O)CC(N=c2ccc(C(F)(F)F)n[nH]2)C1 C1(CCC)CCCCCN1Cc1c[nH]nc1CCc1ccccc1 CCC(COC)C(=O)N1CCC1CNC(c1cnn(CC)c1CCOC)=O c1(C(=O)NC2C(CO)CCN(C(C(C)(C)OC)=O)C2)ccc(S(C)(=O)=NC)cc1 N1(C(c2c(C)cc[nH]2)=O)CCC(C(=O)NCc2ccnn2C)C12CCC2 N1(C(CCNC(C)=O)=O)CCC2CC2(C(=O)NC2CN(C3CC3)CC2C)CC1 C1(c2nnnn2C2CCOC2)(NC(c2ccns2)C)COCC(C)(C)C1 c1(C(=O)NCCN(CCC)C(C2CCC(NC)CC2)=O)cccc2c1CCOC2 C(=O)(C(N)C[Si](C)(C)C)N(C)CC1(CO)CCCC1 C(=O)(C1=C(Cl)CCCC1)N1C(CN(C(C(C)c2cc[nH]n2)=O)C)CCC1 N1(C(c2cc(C)no2)=O)CC(NC(C2(CC3CC3)CCCO2)=O)CC(C)(C)C1 N1(C(C(C)N(C(C)=O)C)=O)CC2(CCC2NC(=O)C(CCO)N(C)C)C1 N1(C(CCc2c(C(=O)NCCOC)c(C)[nH]c2)=O)CC(CO)C2(CC2)C1 C1(CNC(C(C)n2ccnc2)=O)CC2(C1)CN(C(=O)CC(C)(C)C#N)C2 c1(C(N(CCNC(C2CCO2)=O)CC)=O)[nH]nnc1C CCCC(C(=O)OC)C(=O)NC12CC(NC(=O)Cc3cnc(C)[nH]3)(C1)C2 C(CN=c1nc[nH]cc1C#N)(N(C(C1(CCOC)CC1)=O)C)C1CC1 CC1=CCC(C)(C(=O)NC(CCN(C(=O)C2=CCCC2)C)C(C)C)CC1 c1(C(=O)NC2CCN(C(=O)COC3COC3)C(C3CC3)C2)nc2cnccc2s1 c1(C(=O)NCC2N(C(c3ccc(C#C)cc3C)=O)CC2)cc2nc(=O)ccn2[nH]1 c1(C2C(=O)N2)cccc(P(C)(C)=O)c1.C(C(C)C(C)C)N(CCC(=O)OC)C C(=O)(C1=CC2(CN(C(N)=O)C2)OC1)NC1C(N(C(=O)COC2(C)CCCC2)C)C1 C12(C(N3CCC(C(=O)NC)C3)=O)CCCCC1C2(F)F.N12CCOC(C1)NC2=O C1(CNC(C2C(C=C)CC2)=O)(OC)CCN(C(c2cnsn2)=O)CC1 C1(C)(NC(C(CCCOC)NC(C2C(CC)C2)=O)=O)CC(C)(C)OC1=O c1(C(N2CCN(CC(C)(C)NC(=O)CO)CC2)=O)c(Cl)nc2cc(Cl)ccn12 c1(CC=O)ccccc1NC(=O)C=CCOC.C1(OCC)(CNC(CC)=O)CCC1 CC1CCC(C(=O)NCC#CCCO)N1C(=O)CC1CCOC1C c1(C(N(C(C)CNC(C2CC(SC)C2)=O)CC)=O)cnn(C)c1Cl N1(C(C(CN(C(c2cc(OC)no2)=O)C)(C)C)=O)CCCC2(CCC2)C1C N1(C(c2sc(C)c(O)n2)=O)CCN(C(C2(F)CC2)=O)CC(CO)C1 c1(C(=O)NC(C(C)NC(CC2(NC(C)=O)CC2)=O)C)ccc(CF)cc1 CS(=O)(=O)CC(=O)NCCCCCNC(C1(C(F)(F)F)CCCCC1)=O N1(C(COCCNC(CCC(C)(C)C)=O)=O)CCC2CC1C(=O)O2 C1(NC(c2c(C)nc(C)[nH]2)=O)CCN(C(=O)Cn2cc(C(C)O)nn2)CC1(C)C C1(CNC(COCCC)=O)CC2(CCC2)CN1C(=O)CCCc1cc(C)sc1C C1(C(=O)NCCOCCN(C)C(C2CCCOCC2)=O)CCC(=O)N(C2CC2)C1 C12(CCNC(C(CN(C)C)(F)F)=O)CCC1CN(C(C1(CC3CC3)CC1)=O)C2 C(C(O)(CO)CO)C(c1ccccc1)C1CCOC1.N1(C(=O)N)CCOCC1CF C1(C(=O)NC2C(CNC(c3ccncc3)=O)C2)CCn2c(O)nnc2C1 C(=O)(C1=NN(C)C(=O)CC1)NCCN(C(Cc1nnc(C)o1)=O)Cc1ccccc1 n1(C(C)C)cnnc1CNC(=O)CNC(=O)CCC1CC1(C)C N1(C(C(=O)N(C)C)=O)CCC(C)(NC(C2CC(C(F)F)C2)=O)C1 c1(C(NOC(CC)CC)=O)cccc(NC(C2C=C(C)CS2)=O)c1 C1(CNC(C(C)OCC2CC2)=O)CCCC(NC(c2cnc(O)n2C)=O)C1 c1(CN2CC3N(C(c4cc(Br)cc(I)c4)=O)C3C2)c(O)cc(O)cc1O N1(C(C(CCSC)O)=O)CCC(C(=O)Nc2ccc(F)nc2)C(C)C1 C1(NC(=O)CCNC(C2CCCO2)=O)CCCC1NC(c1c[nH]c(C2CC2)n1)=O c1(NC(N2CC3CCN(C(=O)OC(C)(C)C)CC32)=O)ccc(F)c(S(C)(=O)=O)c1 c1(C(=O)NC2CCN(C(C(C(C)C)C)=O)C23CC3)cccc(Cl)c1[N+](=O)[O-] CCCCCC(CC)C(=O)NCCOCC.C1(=O)C(CC)COCCCN1C C#CCC(C)C(=O)OCC1CCCN1C(C)C c1(OCCN(C(CNC(COC(CC)C)=O)C)C)cccc(F)c1 C#CCC(C)(CC)C(=O)NCC1CCC2(CN(C(c3cccc(=O)o3)=O)C2)O1 CC(F)(F)CC(=O)NCCN1CCN(C(c2cccnc2N2CCCC2)=O)CC1 c1(CC)c(C(N2CCC(NC(c3cccc(C(F)F)n3)=O)C2C)=O)ccn1C c1(C(N2C(CNC(c3c(N)non3)=O)CC2)=O)noc2cc(F)ccc12 c1(C(=O)NC2CN(C(c3cc(C(C)C)[nH]n3)=O)CC2(C)C)cc(O)cc(C#N)c1 C1(C2CN(C(=O)C(C)N(C)C)C2)(NC(C(C(C)C)NC(CN(C)CC)=O)=O)CC1 N1(C(CC(C)(C)NC(C2CCN(CC)CC2)=O)=O)CCOC2COCC12 C(=O)(C(C#N)C(C)(C)C)N1CCOCC(CNC(Cc2c(C)non2)=O)C1 c1(OC(C)(C)C)ccccc1Cl.C1(C)(C)C(c2nnnn2-c2ccccc2)N1 c1(OC)cc(C(=O)N(C)CC2(O)CCN(C(C3(NC(N)=O)CC3)=O)C2)ccc1F C12(C(=O)NCC3N(C(c4c(C)cc(C)o4)=O)CCC3)CCC(CC1)C2(C)C c1(NC(=O)Nc2c(CC)cccc2CC)c(F)cc(C#N)cc1Br CC1CCN(C(c2cc[nH]c2C2CCC2)=O)CC1C1C2CCN(C(CC)=O)C2C1.O N1(CC(=O)N(C2CCCN(C(c3cnnn3C3CC3)=O)C2)C)CCCCCC1 N(C1CCCc2cc(C#N)ccc21)C(=O)NCC1CCN(C)C1 c1(C(N(C(C)C2CC2)CC2CCCCCC2)=O)ccc(C#N)nc1 CC12CN(C(=O)Cc3ccc(F)cc3F)CC1(C)CN(C(C1CC1F)=O)C2 N1(C(CCC(N)=O)=O)CCC(F)(F)C(C(=O)Nc2cc(F)c(Br)c(F)c2)C1 c1(C(N2CCCC(N3CCOCC3)CC2)C(=O)NCCSC)ccc(F)c(Br)n1 N1(C(C(C=C=C)C)=O)CCOCC(C)(CNC(c2cn(C3CC3)cn2)=O)C1 C1(CC(=O)N(C2CCN(CC)C2)C)CN(C(=O)C(F)C2CCCC2)CCC1C C(=O)(C(C)S(N)(=O)=O)NC1CN(C(c2ccc(SC)o2)=O)CC1C.c1ccccc1 C1(CNC(C(F)OC)=O)CC2CCC(C1)N2C(=O)CC(C)n1ccc(C)n1 C(=O)(CS(=O)(=O)NC)N(C(CCNC(C1N(S(CCC)(=O)=O)CCC1)=O)C)CC C=C=CC(C)C(=O)NC(C)(C)COCCCNC(C1C=CCS1)=O C(=O)(C1COc2ccccc21)NCC(C(C)(C)C)NC(CNC(=O)NC)=O CC(CS(C)(=O)=O)C(=O)NCC(C1CC1)NC(c1cc2cccnn2c1)=O N1(C(CCC2CCCN(C(C3(C)C(C)C3)=O)C2)=O)CCC(C)(N(C)C)CC1 C1(NC(CN(CC)CC)=O)CCN(C(C2CCS(=O)(=O)C2(C)C)=O)CC1(C)C C(C1CCCN1C(=O)COC1CCOCC1)=CC(=O)NC1C(CN(C)C)C1 c1(C(N)=O)cnc(Cl)[nH]c1=NCCCNC(=O)C1=CS(=O)CCC1 C12(C(=O)NC(CC)CS(C)(=O)=O)C3C4C1C1C2C3C41C(=O)NC CC1CCC(NC(c2ncc(F)cn2)=O)CN1c1cc(Cl)nc(C(F)(F)F)n1 C(CC1CC1)(C(=O)N=c1ccn(CCOC)[nH]1)NC(C1CCC(CC)O1)=O N1(C(C2(CC)CC2)=O)CCOC2(CCCN(C(C3(C#N)CCN(C)CC3)=O)C2)C1 C1(Cc2cc(C)no2)CCN(C(=O)C(C)Oc2ccccc2)C1C=O.C(C)C c1(C(=O)NC(C(C(=O)NCCOC(C)C)C)C)cc(C#N)n(C)n1 c1(C(=O)NC2CCN(C(CCCOCCC)=O)C2)cnc2c(cnn2C)c1O Cc1ccccc1C1CC1C(=O)NCC1CC(NC(c2cnsc2)=O)C1(C)C CC1(CNC(C2CC3C=CC2CC3)=O)CCCN(C(=O)CCNC(=O)C=CCl)C1 CC(C)CC(C)CC(=O)NCCC(N1CCCC1Cc1nc2ccccc2o1)=O c1(C(=O)OCC(=O)OCCSCCCC)n[nH]cc1[N+](=O)[O-] C1(CC)CCN(C(=O)Cc2cnc(C)s2)C(C(=O)NC(c2ccccc2F)C)C1 c1(CCNC(C2N(CCCCCC)CCC2)=O)ccc(OC)c(C)n1 N1(C(COCCC(C)C)=O)CC2C(CC(=O)NCCSCCO)C2C1 N1(C(C2(NC(C3COCC(C)O3)=O)CCCC2C)=O)CCn2nccc21 n1(CC)nc(C)cc1C(=O)NC1CC(CNC(=O)Cc2c[nH]nc2C)CC1O C(c1cncc(C)c1)=C.c1(SCC)cc(C(N2CCCC2C(=O)N)=O)n[nH]1 c1(C(N(C2CCN(C(c3ccc(CCO)cc3)=O)C2)C)=O)ccc(O)c(Br)c1 C(C)(CCCCNC(=O)CCCC1(C)N=N1)NC(C1C(C)=C1)=O N1(C(CCC2CC(OC)C2)=O)CCCC(CC2CC2)CC1.C1C(=O)NCCO1 C1(NC(C2CCC=CO2)=O)CCN(C(c2cc3ccncc3[nH]2)=O)C12CCC2 N1(C(C=C(C)c2ccco2)=O)CC(NC(=O)C2=NOCC2)CC12CCOC2 N1(C(c2cc(OCC)ncc2)=O)CCC(C)CC1CNC(C1CC(C)=NO1)=O c1(C(=O)NCC2OCCN(C(C(CSC)C)=O)C2)cncn(C)c1=O N1(C(C(CC)c2ccccc2)=O)CCSCC1CNC(=O)C(=O)Nc1ncc[nH]1 C12(C(=O)NCC3OCCN(CC)C3)CC(CCO1)N(C(C1CC1(C)C(F)F)=O)C2 c1(C(=O)NC2CCCC(CN(C(=O)CCc3cn[nH]c3)C)C2)cc([N+](=O)[O-])c[nH]1 N1(C(CC(Cc2ccccc2Br)OC)=O)CCC(O)C(C2CCCC2)C1 c1(C(C(=O)NCC(F)CNC(=O)C(Cl)=CCl)=O)cc(Cl)cc(Cl)c1 CCCC(C(=O)OC)C(=O)N1CCC(CCC(=O)NCc2cc(C)sc2C)CC1 C(CCCC(CO)NC(=O)Cc1nccn1C)NC(C(C(C)C)n1cccc1)=O C1(NC(=O)CCCC2CCCCC2)(CO)CCCN(C(c2ccno2)=O)C1 c1(C(=O)NC2CCC(F)(CNC(CCCNC(C)=O)=O)C2)cnc2sccc2c1 N1(C(CC2CCC(C)C2)=O)CCC(O)(CNC(=O)COc2cncc(Cl)n2)CC1 CCC(CCOC)C(=O)N1CC(O)CC1(C)C(=O)NCCOCC(N)=O N1(C(C2CCN(C(Cn3ncc(C#C)c3)=O)CC2)=O)CCCNC(=O)C1 N1(C(c2cn(C)nc2)=O)C2CCC(C(N3CC(c4cc(O)no4)C3)=O)C1CC2 CN(C)S(C)(=O)=Nc1nc(C(N2CCC(NC(C3CC3F)=O)C23CCC3)=O)cs1 c1(OC)ccc(F)c(C(N2C3CN(C(c4cnc(O)[nH]4)=O)CC23)=O)c1F C1(CC(=O)NC(CCOC)CNC(c2noc(C3CC3)c2C)=O)CCC(C)CO1 Cc1cccc(O)c1C(=O)NCc1ccsc1C(=O)NC1CCCCCC1 C#Cc1cnc(C(N2CCC(C(=O)N(C)Cc3nncs3)CC2)=O)c(C)c1 N1(C(C2(CCOC)CCCC2)=O)CCC(NC(=O)CC2(C)CCCCC2)C(C)C1 c1(C(C)OC)ccc(C(=O)NCC23CC(C(F)F)(CO2)C3)cc1 N1(C(C(C(CC)C)N)=O)CCOC2CN(C(c3c(OC)cccc3C)=O)CC12 N#Cc1cccc(CCNC(=O)NCC2(O)CCC(CO)C2)c1 C1(CNC(c2ccc(OC)s2)=O)CCN(C(C2(OC)CCCOC2)=O)CC1C N1(C(C2(C#N)CCC2)=O)CCC2(CC1)CCN(C(C13CC(C1)S(=O)(=O)C3)=O)C2 c1(C(=O)NC(c2ccccc2)C#N)c(Cl)oc2ccccc12 CCCCCCn1nnnc1C(C1CC(F)C1)(C)NC(CCC)C1CCC1 c1(C(=O)NCC2C(NC(c3c(C(C)C)onc3)=O)COC2)nnn2c1CSCC2 C1(CC(N2CC(C3C(=O)N3)C2)=O)CC2(CCC2)CO1.N1(CC)CCC(C)C1 C#Cc1cccc(C(=O)NC2CCC(C(=O)Nc3nc(C)cs3)C2)c1 N1(C(C(c2ccco2)NC(C2CCC2)=O)=O)CCC(CC2CC2)CC1 N1(C(CCOc2ccc(OCC)cc2)=O)CC(NC(=O)C#CC(C)C)CC(O)C1 c1(NC(C2CCC(COC)O2)=O)cc2c(cc1O)=CC=CC=CC=2 n1(CC(=O)N(C2CC(NC(C3C(C)OC(=O)N3)=O)C2)C)cc(S(C)(=O)=O)cn1 C1(C(N(CCC(C)C)C)=O)CC12CCN(C(C1CCC(N)C(O)C1)=O)CC2 CC1=C(C)CC(C)(C(=O)NC(C)CC2CN(C(C34CC3COC4(C)C)=O)C2)CC1 c1(N(C)C(C2CCOC(C(C)(C)C)C2)=O)ccc(Cl)cc1C=CC(=O)O N1(C(C2(C)ON=C(C)C2)=O)CCCC(C2(NC(C34CC3C4)=O)CC2)C1 C(=O)(C#CC1CCCCC1)N1C(C(C)NC(c2cc(CN(C)C)on2)=O)CCC1 S(=O)(=O)(c1ccc(CBr)cc1)N1C(C)(NC(=O)Nc2c(Cl)cnc(C)n2)CCC1 C1(C)(C(=O)NCC2(NC(CCCN(C(C)=O)C)=O)CCCC2)CCC(=O)N1 c1(C(=O)NCC23C(CN(C(c4c(C)nsc4C)=O)C2)C3)ccc(C(C)C)cc1F N1(C(C(C)N(C(C)=O)C)=O)CCC(N2CCN(C(=O)C(C3CC3)SC)CC2)CC1 c1(NC(C(CC=C)CNC(=O)C(C)CCN(C)C)=O)cccc(N=[N+]=[N-])c1 NS(=O)(=O)c1ccc(SCC(=O)NC23CCC(CC2NC(=O)CO)C3)cc1 c1(C(N2CC3C(N(C(CCOC)=O)C)C3C2)=O)cc(F)c(OC)cc1N N1(C(=O)CCc2cnccn2)CCCN(C(=O)C=Cc2ccsc2)C(CO)C1 c1(SC)nc(C)cc(=NC2CC(F)(CNC(=O)Cc3ccc(OC)c(F)c3)C2)[nH]1 C#CCCCCC(=O)NCC=CC(=O)NC1CN(C2CC2)CC1C CC(C)C1=NOC(C)(C(=O)NC2CN(C(C3CCCC34CCC4)=O)C2)C1 CC1C(NC(=O)C(F)C(C)C)CC2CCC1N2C(c1ccc2cnccc2c1)=O c1(C(=O)NC2CC(CNC(C3CCCO3)=O)C2)cccc([N+](=O)[O-])c1Cl N(C(=NCCc1ccc(Cl)cc1Cl)NCc1cccs1)C1C(C)C1C N1(C(c2nc(C)[nH]n2)=O)CCCC(C)C1CCNC(C1(n2ccnn2)CC1)=O C1(NC(CN(C)Cc2cccs2)=O)CCN(C(=O)Cn2ncnn2)C(C2CC2)C1 N1(C(C(C)OCCC=C)=O)CCCCC(CNC(=O)C(C)(C)c2cc[nH]n2)C1 C=CC1COCCN1C(C1CCN(C(=O)C(C)OCCCC)C1)=O C1(CNC(C2N(C(CCC)=O)CCC2)=O)CCCN(Cc2cccc(C)n2)C1C C#Cc1cc(C(=O)NCCN(C(c2ccc(C(N)=O)s2)=O)C2CC2)cc(F)c1 N1(C(CCCCSC)=O)CCC2(CC1)CC2NC(C1CC(OC(C)(C)C)C1)=O N1(C(c2ncc(C)cc2F)=O)CCCC2C1CCN2C(=O)CCc1cnn(C)n1 N1(C(C(c2ccc(OC)cc2)O)=O)CC2CN(Cc3cccc(Cl)c3F)CC12 CCCC(CC)C(=O)NCCCCC(=O)NCC(C)(C)CC(C)C CC1(C)C=C(C(=O)N2CCC(O)(CCNC(c3csc(C(F)(F)F)c3)=O)C2)C1 C(CC(=O)O)(C(F)(F)F)NCCC.Nc1cc(OC)[nH]c1 N1(C(C(C)OC(C)(C)C)=O)CCCC(NC(c2csc(-c3ccco3)n2)=O)CC1 C=CCC(CC=C)C(=O)N1CCC(NC(C2(C3CC3)CCOCC2)=O)C(F)C1 Cn1c([N+](=O)[O-])cnc1C(=O)NC1CCCC1CNC(C1CCC(F)(F)CC1)=O C(=O)(CCS(C)(=O)=O)NC1C(C)(C)C(CNC(C2CCCC23CCC3)=O)C1 C1(NC(=O)CC2CCCCO2)CN(C(=O)CCc2ccccn2)CC1F C(=O)(C(F)CCC(C)C)NC(CC=CC)C(=O)NCC1(C2CC2)CCC1 C(=O)(C(C(=O)NCC(C)(C)CNC(=O)CCCn1cc(C)cn1)C(C)C)OCC C1(OCCNC(Cc2cc(OC)no2)=O)CC2CN(S(C)(=O)=O)CCN2C1=O c1(C(N2CC(NC(CNC(=O)OC)=O)C(C)CC2)=O)ccc2nc(Cl)nn2c1 c1(CN)cc(C(=O)OC(C)(C)C)ccn1.C12(C(=O)NC3CC3CNC(N)=O)CC(C1)C2 N1(C(C2C3CN(C(C(C(=O)OC)C)=O)C2C3)=O)CC2(CCOCC2)C1 Cc1ncc(NC(=O)CC2CCN(C(=O)CCc3ccncc3)C2)cc1Cl c1(C(C)(C)N(C)C)cn(CC(=O)NC(COC(C)(C)C)C(N)=O)nn1 C=CCCCCC(=O)NC1CCC(NC(c2c(C)nn(C)c2C(F)(F)Cl)=O)C1 C(=O)(CCCCCNC(c1nc[nH]n1)=O)NC1C(CCC=C)CCC1 c12c(sc3ccccc13)C(=O)N1CCCN(CC1)C2=O.C(C(C)C)OCC c1(C2(C(=O)NCC(CC)NC(=O)CC3CC(CC)C3)CC2)ccc(O)cc1 C1(NC(CCN(C(CCC)C)C)=O)CN(C(C2(CC)CNC(=O)C2)=O)CC1(C)C N1(C(c2ccccc2)=O)C2CC1CN(C(=O)COc1noc(CC)c1C)C2 c1(C(N2CC(CNC(C(C=C)(C)O)=O)OC(C)(C)C2)=O)cc(C#N)c(N)cc1O CN1C(=O)NCC1C(=O)NCC1CCC1NC(=O)C=CCN1CCCC1 C(=O)(C(C)(C)CF)N(C(C)CNC(=O)C(C)(C)N(C)C)CC N1(C(c2nc(COC)oc2)=O)CCC(CN(C(=O)CCC2CCCN2C)C)CC1 c1(C(N2C(CN(C(=O)CC(C)NC(C)=O)CC)CCC2)=O)cc(SC)ccc1O C12(C(N3C(CN(C(=O)CNC=O)CC)CCCC3)=O)CCCC1C2(F)F C(=O)(C(C)(C)CCC(F)(F)c1ccccc1)N1CC(C)C(O)C1 C1(CC(=O)NCC(CCNC(C(C)CC2CCC2)=O)O)CC(C2CC2)C1 CC(C)C(C)C(C)CC(=O)N1CCC(C)C(NC(=O)CC2CCC(C)CC2)C1C Cc1nn(C)cc1C(C)NC(=O)CCOCCCNC(=O)CN1CC(=O)NC1=O c1(C(C2CCCCC2)OC)cn(CC(C)NC(C2CC2C(C)(C)C)=O)nn1 CS(=O)C=CC(=O)NC1C2CN(C(c3c[nH]nc3C3CCC3)=O)CC12 c1(C(=O)NC(CC(=O)OCC)C)coc2c1CN(C(=O)C(C)c1cccs1)C2 C1(C(=O)NCCCN(C(C2CC(F)(F)C2(C)C)=O)CC)CC2C(C1)C2(C)C Cc1nncc(C(=O)N(C)CC2CCCN(C(=O)CN3CCNC(=O)C3)C2)c1C CCC(C)C(C)CNC(c1cc(=O)n(-c2ccc(Cl)cc2)[nH]1)c1ccccc1 c1(OC)cc(Cl)ccc1C(C)NC(c1ccc(C)c(Br)c1)C N1(CC)CCC(C(=O)N(CCCCNC(c2cnsc2)=O)CC)CC1 N1(C(c2ccn(CCC)n2)=O)C(C(=O)Nc2cccnn2)CC2CC12 c1(CC)scnc1C(=O)N(CC(C)(C)CNC(=O)C(O)C1CCC1)C Cc1cc(C(=O)NCC2CCN(C(=O)Cc3cncs3)C2)ncc1CO c1(C(=O)NC(C2CC(NC(=O)CCNC(C3CCC3)=O)C2)C)cnco1 N1(C(CCC=C(C)C)=O)C2CCC1CN(C(=O)CC1CC13CC3)CC2 C(CCC(C)(C)C(=O)NC1CC(OCC(=O)N(C)Cc2ccccc2C)C1)OC N1(C(c2onc(C)c2C(F)(F)F)=O)CCN(C(c2cc(N)c(Cl)cn2)=O)C(CO)C1 c1(N(C(=O)COC(C)(C)C)C)ccc(Br)c(S(=O)(=O)N2CCN(CCC#N)CC2)c1 C1(NC(C2OCC(C)(C)C2)c2ccccn2)CC2(CCCNC2)C1 C(=O)(C1=NOC2(CCC2)C1)NCC(CNC(C(c1ccc(CC)cc1)C)=O)OC CC1=NN(C)C(=O)C1CC(=O)NCC1(F)CC(NC(=O)CC2(C)CCCCC2)C1 C1(NC(C23N(C(C(C(=O)OC)OC)=O)CCC2C3)=O)CC2CC1CC2CO N1(C(c2nccc(OC)c2)=O)CC(C(=O)N(CC(C)C#N)C2CC2)C(F)(F)C1 C1(C(=O)NCCn2cc(COC)nn2)OCCCC1(C)C.C12(CC1)CC(=O)NC2 CC(C(=O)N1CC(NC(=O)CCc2ccccn2)C(N=[N+]=[N-])C1)C1=CCCC1 C1(CNC(=O)CCN2CCCS2(=O)=O)CCC2(CCCC2)O1 C(=O)(CCC(C)C#N)NC(C)CNC(=O)Cc1ccsc1Cl C1(NC(C=CC)=O)COC2(CCCN(C(c3ncn(-c4ccccc4)n3)=O)C2)C1 C1(CC=C(C)C)CCCC(N(C(=O)CCOc2cccc(Cl)c2)C2CC2)C1 c1(SC)cc(C(=O)NC(c2ccccc2)C(=O)N(CCC(O)CO)C)co1 N1(C(CCNC(=O)OCC)=O)CC2OC(=O)N(C3CCOCC3)C2C1 N1(C(CCC2C(C)C2)=O)CC(CNC(=O)CCOCCN(C)C)C(O)C1 CCCC(C)CCCC(=O)NCCCCN(C)C(c1cnc2cc(C)ccn12)=O c1(NC(C(CCC)CNC(C2CC(O)C(F)C2)=O)=O)ccn2nccc2c1 C1(NC(c2c(C)nc(COC)s2)=O)CC2CN(C(c3ccc(C(F)F)s3)=O)CC12 CCCS(=O)(=O)CC(=O)NC(C)(CNC(c1csc(O)n1)=O)CC(C)C Cc1nc2c([nH]1)CN(C(C1CCN(C(=O)C(O)C(F)(F)F)C13CC3)=O)CC2 C1(C(N2CCC(C(CNC(c3c(C)nsc3)=O)(C)C)CC2)=O)CC2(CCC2)CO1 C(=O)(CC(COC)CC)NCCOCCN(C(C1(C#C)CCCC1)=O)C C1(C(N2CC(OCC)(CNC(=O)C(C3CC3)C3CC3)C2)=O)CCC(=O)N(C)C1 CC(C)CC(CNC(c1cn(Cc2cccs2)nn1)=O)NC(C1CC1(C)C)=O C(C(=O)NC1CC1)(C1=NOC2COCC12)N(C)CCc1cccc(Cl)c1 C1(CNC(NCC(=O)N(CC)CC)=NCC2CCOC2)CN2CCCC1C2 N1(C(CC=CC=C)=O)CC(CC(=O)NC2(C(=O)N(C)C)CC2)(OC)C1 c1(NC(C2N(C(CCOCCN(C)C)=O)CC=C2)=O)ccc(F)c(CO)c1 C1(NC(C(CCN(C)C)NC(CC2(OCC)CCC2)=O)=O)CC12CCOCC2 N1(C(C2C(CNC(c3cc(C4CC4)no3)=O)C2)=O)CC2CC(O)CC1C2 N1(CC2C(C)SCC2)CCC(n2cc(C(C)(C)N(C)C)nn2)C(O)C1 N(C(=NCc1ccc(OC)c(F)c1)N1CCC(COCC)(CC)C1)C(CC)C C1(CN(C(C2(OCC)CCC2)=O)C)CCN(C(=O)C=C(C)C(F)F)C1 c1(-c2cn(CN(C(C(C)OC)C(=O)OC)C)nn2)ccc2c(c1)OCO2 C1(NC(=O)CC2CCOC2)CC2CC(C1)N(C(c1cc3ccsc3[nH]1)=O)C2 c1(N2CCCCC(NC(=O)CCn3cccn3)C2)ncnc2c1nnn2CC1CC1 c1(C(=O)NCC23CCCN(C(C=CC)=O)C2CCC3)cc(C)c2nc(C)cn2n1 C=CC(CC)CC(=O)NC(c1cn(-c2cccc(Br)c2)nn1)C c1(C(=O)OC)ccc(C(=O)NC(C)(C)C(C)NC(c2cccn2C)=O)o1 CC(CCCCNC(=O)C=Cc1ccncc1)NC(=O)CC12COC(C)(C1)C2 c1(C(=O)NC(C(C)NC(c2ccc(OCCF)cn2)=O)CO)csc2nccn12 C1(C)(C(=O)NCC23C(CN(C(C)=O)C2)C3)CCCNS1(=O)=O C(=O)(N1CC2(CC2)CO1)c1cc(NCC2CCN(C(C)=O)C2)ncn1 C1(NC(C2ON=C(C(C)C)C2)=O)CCC2(CCN(C(=O)COc3cn[nH]c3)C2)C1 c1(CN2CCC(NC(C(C)SCC)=O)C2C(C)(C)C)cn2ccncc2n1 c1(C(N2CCC(CNC(c3c(CC)[nH]nc3Cl)=O)C2)=O)ccc(F)c2occc12 C(=O)(CC(C(C)C)C(C)C)NC1CC2CC(NC(c3c(SCC)nccn3)=O)C2C1 C(=O)(CCCCCCCBr)N1C2CN(C(C3C(C)CCC3)=O)CC1CC2 CCC(CSCC)N=c1cc(C)[nH]c(=NCC(C)(C)NC(C)(C)C)[nH]1 CCCC(F)C(=O)OC(C)(C)C.C(=O)(CC(C)CN(C)C)N(C1CC(OO)C1)C c1(OC)cc(N)c(C(=O)NC2CN(C(c3ccncc3Cl)=O)CC2C)cc1OC Cc1cccc2c(C(N3CCC(NC(=O)C=C4CCC4)C(C)C3)=O)nccc12 CCC(C)(CC)C(=O)NCc1cn(CC2CCCN2C(=O)CCC2CCC2)nn1 C(=O)(C(O)P(C)(C)=O)NC(C)(C(=O)O)c1cn(C2CC2N2CC(=O)NC2=O)nn1 C1(CNC(c2ccc(C)cc2)=O)CCC(C)CN1C(c1ccc(Cl)c(C)c1)=O N1(C(c2ccc(CNC(C3C(CCC)C3)=O)s2)=O)Cc2c[nH]nc2C(C)C1 C1(O)(CN2CC(N(CCOC)C(=O)C3CC3)C2)CCCC(C(F)(F)F)C1 CCC(C)(CCC(C)C)C(=O)N1CCC2CN(C(=O)C(N)=O)CC12 C1(NC(=O)Nc2ccnc(N3CCOCC3)n2)CNCC2(CCC2)C1 N#CCCCCC(=O)N1CC(NC(=O)CCCc2cccc(Cl)c2Cl)C2CC12 N1(C(CC2N(C(c3c(C)ncc(C)n3)=O)CCC2)=O)CCc2ccsc2C1 C1(C2CCN(C(=O)C=CCO)CC2)(NC(C2CC3CCC(C2)N3C2CC2)=O)CC1 Cc1nnc2ccc(C(=O)NC(C)(CO)C3CCCC3)cc2c1C C(=O)(C#CC(C)(C)C)N(Cc1cccc(CNC(CC2CCN(C)C2=O)=O)c1)CC C(=O)(C#CC1CCOC1)N1CCC(N(C(=O)COCc2ccccc2)C)C1 c1(OC)cc(NC(=O)CC2COCCN2C(c2cc(O)no2)=O)cc(C)n1 C(=O)(CC(C=C)CCC)NCC(C1CCCC1)NC(COCC#C)=O c1(C(N2C(CCNC(CSCCC)=O)CSCC2)=O)ccc(Cl)c([N+](=O)[O-])c1 N1(C(c2c(C)c[nH]n2)=O)CCC(O)(CCNC(c2cn(CCC3CC3)nn2)=O)C1 C1(CNC(CC(C)c2ccccc2)=O)CCCCC1NC(C1CN(C)CCO1)=O c1(CC(=O)NCC2C(NC(C(c3ccccc3F)C)=O)C2)sc(O)nc1O c1(C(=O)NCC2CN(C(C3(F)C(C)OCC3)=O)C2)cc2c(=O)[nH]ccn2c1 CCCCCC(O)C(=O)NC1CCCC1CNC(c1nn(C)nc1Br)=O c1(CN2CCCC(CCCC)C2)cc(C)c(N2CCSCC2)cc1C N1(C(c2n(CC=C)ccc2)=O)CCN(C(=O)CCC(C)(F)F)C2CC12 c1(CNC(C2CC(OC)C2)=O)cccc(C(=O)NC(c2ccc(CO)cc2)C)n1 C=CCCC(F)(F)C(=O)NCc1cncc(C(=O)NCCNS(N)(=O)=O)c1 C1(C(=O)NCC(CCOC)NC(c2ccns2)=O)CCC(=O)N1C(C)C Cn1cc(Cl)cc1C(=O)NCC(C1CCN(C(c2cn(CCO)nn2)=O)CC1)F CCC(C)(C)CCCC(=O)NC(C)(C)CCCC(=O)Nc1ccc(C)c(C)c1 Cc1ccc2c(C(=O)N(C3(CO)CC3)CCCn3ccnc3)cnn2c1C Cc1cc(C(=O)N(C)CCOCCN(C)C(c2cocc2C)=O)ncc1Cl C1(NC(C2CCCN(C)C2)=O)CCN(C(c2[nH]nnc2C2CC2)=O)CC1CO N1(C(C(=Cc2cccs2)C)=O)CCCC(C)C1CNC(c1cn2c(n1)CCC2)=O C1(CC(=O)NCCN(C(=O)Cc2cncc(C(N)=O)c2)CC)COC(C)(C)CO1 S(=O)(=O)(c1cccc(Cl)c1Cl)N1CC(N(C)Cc2ccnc(F)c2Cl)C1 N1(C(CN(CC)CC)=O)CCN(C(=O)Cc2ccoc2C)CC1c1nccn1C c1(C(=O)NCC2CN(C(c3n(CC)cnn3)=O)CC2(C)C)ccc(Cl)c(F)c1F C=C(C)C1OCCC1C(=O)NCC1CC(NC(C2CC2C2CC2)=O)C1 C1(C(=O)NC(C(C)(OC)C2CC2)C)CN(C(=O)C2=NOCC2)CC2(CCC2)O1.C(C)(C)(C)O c1(NC(c2scc(-c3cccc(CCNS(C)(=O)=O)c3)n2)=O)cccc(Cl)c1Br c1(C2CC(OC)C2)ccc(NCc2cn(CCNC(=O)OC(C)(C)C)nn2)cc1 C12(NC(c3cc(C)[nH]c3)=O)CCN(C(=O)CCCc3cc(C)no3)CC1C2 c1(C(C(=O)N(CCNC(c2cn(CC)nn2)=O)C2CC2)OC)ccc(F)cc1C N1(C(C2CCN(C(c3c(C)nco3)=O)CC2)=O)CCC2(CC1)CC(F)(F)C2 C12(C(=O)Oc3nc(-c4ccc(OC)cc4)sc3)CCCCC1OCC2 O=S(=O)(c1cccnc1NCc1sncc1Br)NCC1CC2(CCC2)CO1 c1(C(=O)NCCC2(CNC(C3C(OC)CCC3)=O)CC2)ccc(=O)n(C)n1 C1(NC(CCCSC)=O)CC(C2CCN(C(C3CN4CCN3CC4C)=O)C2)C1 CCC(CNC(=O)C(Cc1ccco1)NC(C1CCC1C)=O)C(C)(F)F c1(C(=O)NC(C2CCCCC2)CNC(CCOC)=O)cccc2c1NCC2 C(c1cncc(O)c1)=CC(N1CC(C(C)NC(C2CCC(F)CC2)=O)OCC1)=O N1(C(c2cc(SC)ncc2)=O)CCOC2(C1)CN(C(c1cn(C)nc1C)=O)C2 C1(C(=O)NCCNC(C(N2CCC(C)CC2)=O)=O)CC2(CCC(F)(F)CC2)CO1 C(=O)(C(C)(C)NC(C1CCC1CNC(=O)Cn1cnnn1)=O)OC C(=O)(C1CCCc2nc[nH]c21)N1CCC(CNC(=O)CCCCCO)C1 c1(OC)cc(C(c2nnnn2C)NCc2cccc(C(F)F)c2C)c(Br)cn1 CC1=C(C)CC(C(=O)NCCCC2CCCCN2C(=O)CCCC2CC2)CC1 N1(C(c2ccc(N)c(F)n2)=O)C2CCC1CC(NC(C1(Cl)CCC1)=O)C2 C1(NC(C2N(C(N)=O)CCC2)=O)CN(C(=O)C=Cc2cc[nH]c2)C2CCCCC12 C#Cc1cn(C)nc1C(=O)NC(CC)(CC)CCNC(=O)C(F)CC1CC1 Cc1ccc(CCC(=O)NCCN(C(c2coc(C(F)F)n2)=O)C(C)C)s1 C1(NC(C2CC(O)C2)=O)CN(C(=O)Cn2nccn2)CC1n1ccnn1 c1(CC(=O)N(C2CCCN(C(CC(=C)C)=O)C2)C)cn(CC)c2ccccc12 C(=O)(CC(C)(C)CC)N(CC(CC)NC(c1cc(CC2CC2)on1)=O)C Cc1nc2ccccc2c(C(=O)NCCC2CCCCCC2)c1C CC1CC(NC(=O)COCc2ccc(C#N)cc2)CCN1C(=O)CCF C=C(C)C(CC(=O)NC(COCC)C(=O)NC1CCCC(=O)C1)OCC c1(OC)cc(C(=O)NC2C3CN(C(c4nccc(C)c4N)=O)CC23)ccc1C C1(C(N2CCc3nncn3CC2)=O)CCC(C2CCCCC2)CN1 C(N=c1[nH]c(C2CC2)nc(=N)[nH]1)c1c(CNC(CCSC)=O)cccc1C C1(NC(COC2CCCC(C)C2)=O)CCC12CN(C(c1cnc3n1CCS3)=O)C2 c1(C(=O)NC2CCCCN(C(c3c(C)snc3)=O)C2)nnn2c1CSCC2 CCC(C)C(C(=O)NC1(C)CC(C)(C)C1)N(C(=O)Cc1ccc2c(c1)CC2)C C1(C(=O)NCCS(CC)=O)N(C(c2cn(CCO)nn2)=O)CC12CCCC2 C(CCC(C(=O)NCCCSC(F)F)NC(=O)C(C1CC1)SC)OC.C(CO)O c1(C(=O)NC(CC(F)F)C(=O)N2CCC3CC23)ccc2cc[nH]c2n1 c1(OC)ccc(C(=O)NC23CC2CN(C(C2(O)CCCCC2)=O)C3)nc1Br O=C1CC(CC(=O)N2CC=CC2C(=O)NCCc2cn[nH]c2)=NN1 C1(CC)CN(C(c2ccc(F)c(C)c2)=O)CCN1C(c1cn(C)c(=O)nc1O)=O N1(C(c2c(CC)ncnc2)=O)CCCOC(CNC(=O)CCc2cncn2C)C1 N1(C(CCCN(c2ccc(Cl)cc2)C)=O)CCC2C(NC(c3cccs3)=O)CC12 N1(CCCOc2cc(C)on2)CCN(Cc2nc(C(=O)NC3CC3)nn2C)CC1 C1(N(c2n(C)ncc2)C(=O)CC2CCC(F)(F)CC2)CCCC12CCNCC2 c1(C(N2CCC(CNC(c3c(CC)occ3)=O)(CO)C2)=O)cc(F)ncc1OC N1(C(c2cnc(C)o2)=O)CCN(C(c2sc(=N)[nH]c2C)=O)C2CCCCC12 c1(C(=O)NCC2CCN(C(C3(COC)CCCO3)=O)C2)cccc(Cl)c1 C(CC(C)N=c1ccnc(CO)[nH]1)NC(c1c(NC(C)=O)c[nH]c1C)=O C1(C(=O)NCC(CNC(c2ncn(C)c2)=O)O)CCc2cc(Br)ccc2O1 N1(CC)CCC(c2nnnn2C(C)C)(NCC2CC(C)(C)CO2)CC1C C1(C(=O)NC2CN(C(c3c(CC)scc3)=O)C2)OCCOC12CCC2 c1(C(=O)NC2(C(=O)NC(CC)C(C)(F)F)CC(CO)C2)cc[nH]c(=NC)c1 c1(C(NNC(c2nc(C)sc2-c2ccccc2)=O)=O)ccc2c(c1)CCC(=O)N2 Cc1nc(C(C)(F)F)ccc1C(=O)NC12CCC(C1)N(C(C1(C)CCCO1)=O)C2 C1(C(N(C(C)CNC(=O)CCOC2CC2)C)=O)Cc2cc(F)ccc2O1 c1(C(N2C(C)(C(N3CCC3CO)=O)CCC2)=O)c(Cl)cccc1Cl Cc1cc(O)ccc1CC(=O)NC1CC2(C1)CN(C(=O)C(F)CC1CCOC1)C2 N1(C(C(C)=CC)=O)CCOC(CCCNC(=O)C(CC2CCCC2)NC(C)=O)C1 N1(C2(C(N(C)CCNC(=O)C(F)C3CCCC3)=O)CC2)CCCC1=O C1(COC(=O)CCCNCC2CCCCO2)CCCCCCN1 N#CC1C2CCC1CN(C(C1CCOCC1NC(=O)CCC1CC1)=O)C2 C(=O)(C1CCCc2sccc21)NCC(C)(C)NC(=O)CC(=O)NCCCC(F)(F)F c1(C(=O)NC2CN(C(c3ncc(C)nc3)=O)C2)cc2cc(C(F)(F)F)ccc2s1 c1(C(N2CCN(C(=O)C=CC3CCOC3)C(CCO)C2)=O)cc(Cl)ncc1Cl Clc1cc(-c2nnc(COc3ccccc3)n2CSCCc2ccco2)ccc1Br C1(C)CCC(=O)N1.C(C(C(=O)NCCN1CCC(C)C1)N(C)C)OC N#Cc1ccc2c(=NC(=O)C3CC4CC4N3Cc3cc4cccn4cn3)[nH][nH]c2c1 O=C1CCC2(CN(C(C34CC(CN3C(C3OCCC3C(F)(F)F)=O)C4)=O)C2)O1 C(=O)(C#CC1CCOCC1)NCC(C(C)C)(C)NC(=O)Cc1cc(C2CC2)on1 CC(C)S(=O)(=O)CC(=O)N1CCC(NC(C2CC2C(F)F)=O)C(C)(C)C1 CC(C)CCCCCCNC(c1cc(CCNC(=O)C(C)(O)C(F)(F)F)on1)=O c1(C(N2CC(NC(c3ccc(OC)nn3)=O)C(F)CC2)=O)cn2ncccc2n1 CC1CN(C(c2cc(O)ccc2F)=O)CCC1NC(C1(O)COC1)=O c1(OCC(=O)OCc2scc(C(=O)OC)c2)ccc(N(c2ccccc2)C)cc1 c1(CC(N2C(CNC(c3c(CC)nns3)=O)CC(O)C2)=O)ccc2occc2c1 N1(C(=O)CN2CCCC2CCO)CCC(O)(CNC(C2(CC(F)F)CC2)=O)CC1 c1(CC)ccc(C(C)(C)C(=O)NC2CCCCC2NC(=O)CNC(=O)CO)cc1 C(C(=O)NCCOCC)(c1ccco1)N(CCC#C)C C1(NC(C=C(CC)CC)=O)CCC2(CC1)CC(NC(=O)CC(=O)OC(C)(C)C)C2 Cc1nccnc1C(N1CCCC(c2cc[nH]n2)C1)C(=O)NCCCC1CC1 C1(C(=O)NCCN(C(=O)CCC2CCCOC2)CCOC)CN(C)C(=O)N1 C1(O)(Cc2cn(CCCC(=O)NC3(C)CC(C(=O)O)C3)nn2)CCOCC1 n1(CC(N2CC(CN(C(=O)CCC[N+](=O)[O-])C)OCC2)=O)ncc(O)nc1=O C1(C(N(CCCN(C)Cc2cc(CC)ncn2)C)=O)COc2ccc(F)cc2C1 C1(CNC(CCC(=O)NC)=O)CCN(C(=O)CC2CC(CC)=NO2)C12CCC2 N1(C(C(C(C)C)OC)=O)CC2(C(=O)NC3(CO)CCOC3)CCC1CC2 c1(C(=O)NCC(CC)NC(=O)CC2CCCCCO2)cn2c(n1)SCC2 C1(S(N)(=O)=O)(C(=O)NC2CC(CCNC(c3cc(C(C)=O)sc3)=O)C2)CC1 CS(=O)(=O)C1CCCN(C(=NCC2CCOCC2)NCC2CCCCO2)C1 C(=O)(CC1=CCOCC1)NC(C(=O)N(CC(F)Cl)C)Cn1cccn1 C(=O)(C1=CC(C)(C)C1)N1CC(CC(C)NC(C2CC3(CCC3)C2)=O)C1 c1(OCCN(C(c2ccco2)CC)C=O)ccc(F)cc1.C(C)(=O)O C1(C(=O)NC2CC(CNC(=O)CSc3ccncc3)C2)CC2C=CC1O2 Cc1cc(NC(C2CC(C)CN2C(c2cnc(Br)s2)=O)=O)cc(C)n1 C(=O)(C1CCCc2ccnn21)NCC1C(NC(CC(CN(C)C)(C)C)=O)C1 Cc1cc(C(N2CCC(C(C)NC(C3CCN(C)C3)=O)C2)=O)n[nH]1 C(=O)(C1CCN(C)c2ccccc21)N1CCC(=NC(NC(C)C(=O)O)=S)CC1 c1(C(N2CCCC(NC(C3C(C)CC(=O)N3)=O)(CO)C2)=O)ccc(C#N)c(O)c1 c1(CC(C)NC(=O)C(N2CCC(SC(F)(F)F)CC2)=O)ccc(Br)cc1 c1(C(=O)NCCCN(C(=O)C(C)Cc2cnc[nH]2)CC)cc[nH]c1C1CCC1 c1(C(=O)NCC2CCCN(C(C3C(OC(C)(C)C)C3)=O)C2)cnn2c1OCC2 Cc1oc(C(C)(C)C)cc1C(=O)NC1(C)CCN(C(=O)C(F)(F)C2CC2)C1 CC1CN(C(=O)CNC(C2CCCC2)=O)CC(C)N(C(=O)Cc2nccn2C)C1 N1(C(CN(C(C)C)C)=O)C(CNC(=O)C(C)n2cncn2)CC2CCCC12 C=C(C)CCCC(=O)NC1CN(C(=O)C(Cc2ccc(O)cc2)N(C)C)CC1F C1(NC(c2cc(CO)ccn2)=O)CCCC2CN(C(=O)Cn3cnnc3)CC12 N1(c2ccc(C(=O)OC)s2)CCC(NC(=O)CN2CCCCCC2)C(O)C1 C1(C(N(C)CC2(O)CN(C(=O)CN3CCCS3(=O)=O)C2)=O)CCCCN1N=O C=CCC(CCCCC)C(=O)NCC1(OC)CN(C(C2(C3CCC3)CC2)=O)C1 c1(CN(CC)CC2CC2)nnc2n1CCCCC2 c1(NC(N2CC(=CCC)C2)=O)cc(S(N)(=O)=O)ccc1O N1(C(CCNC(=O)OC)=O)CCCC2(NC(c3snc(Cl)c3Cl)=O)CC2C1 C(=O)(NNC(=O)CC1CCOC1C)c1c(-c2nc(C)c(C)[nH]2)c[nH]n1 c1(CN(CC(=O)N(C)Cc2csc(C)n2)C(C)=O)cc(Br)ccc1Cl c1(CNC(C2CC2NC(=O)COc2cc(Cl)ccc2Cl)=O)cccc2occc12 Cc1ccc2sc(C(=O)N(CCCN(C)C(c3cc(O)ncn3)=O)C)c(C)c2c1 C1(C(N(CCCNC(=O)CCc2ccsc2)C2CC2)=O)CC2CC(=O)C1O2 C=CC1OCCCC1NC(C1CN(C(=O)COc2c(C)cccc2Cl)CCO1)=O N1(C(c2c(C)ncnc2)=O)CC(NC(c2nn(C)cc2Br)=O)CC(C)C1 N1(C(c2c(OC)cncc2)=O)C2CCC1CN(C(=O)CN(C)C(C)C)CC2 Cc1ncc(C(N2CC(NC(C3NC(=O)OC3(C)C)=O)C(F)C2)=O)cc1Cl C(=O)(C1COc2ccc(Cl)cc21)NCC(C)(C)NC(=O)C(O)CN1CCCC1 c1(C(N(C(C)C)CCN(C(=O)C=CS(C)=O)C)=O)ccc2[nH]ccc2c1 C(=O)(C(C)C(=O)NC1(C(=O)N(C)Cc2cnn[nH]2)CC(CO)C1)OC N1(C(CCOCCOC)=O)CC(CO)C2(C1)CN(C(C1CC13CCOCC3)=O)C2 C1(CNC(C2CC(n3ccnc3)C2)=O)CN(C(c2n[nH]cc2Br)=O)CC1O C1(COC)COCCN1C(=O)C(c1cccs1)NC(=O)COCC(F)F C(=O)(C#CC1CCOC1)N1CCC(C)(CC(NOCCN(C)C)=O)C1 C1(NC(COCCSC)=O)CN(C(C2CCC([N+](=O)[O-])CC2)=O)C2(CCC2)C1 c1(CC(=O)NC(CC)CNC(c2cc(=O)n(C)cn2)=O)cc(Cl)cc2c1OCC2 C=CCC(CNC(=O)Cn1cc(Cl)cn1)NC(c1cn(C2CC2)cn1)=O Cc1nn(C)c(C)c1C(C)C(=O)NCCn1cc(CN2CCN(C)C(=O)C2)nn1 Cc1cccc(C(N2CCC(C(C)NC(c3cnc(O)c(Br)c3)=O)C2)=O)c1F C1(NC(Cc2nc(CC)sc2)=O)CC2CN(C(C3CCCC3(C)C)=O)CC12 N1(C(C(c2ccccc2)C)=O)CCC2CN(C(=O)CS(=O)C(F)(F)F)CC2CC1 c1(C(=O)NCC2CCN(C(C(C)OCC#C)=O)CC2)[nH]c2ccc(F)cc2c1Cl c1(C(=O)NC2CC(C(C)NC(c3cc(CC)no3)=O)C2)cnn(CC(F)F)c1C C1(NC(C(COCC)C)=O)CN(C(c2cc(CF)on2)=O)CC1(C)C CC(C)CC(C)CC(C)C(=O)N(C1CCCN(C(=O)CCF)C1)C C1(OC)CCCCC1n1cc(CNC(=O)CNC(=O)C(N2CCSCC2)C)nn1 Cc1c(C(N2C(C(=O)Nc3cnc(Br)c(Br)n3)CC3CC23)=O)cccc1F CC1=CCC(C(N2CCC(CO)(NC(C3CCC(C)(C)O3)=O)C2)=O)CC1 C1(CNC(C=C(C)Cl)=O)CCCCN(C(=O)Cc2cc[nH]c(=N)c2)C1 N1(C(=O)C(F)CC2CN(C(C3CCCNC3=O)=O)C2)CCn2c(O)nnc2C1 C1(NC(CONC(=O)NC(C)C)=O)CN(C(=O)CNC(C2CCC2)=O)CC1C.CN C1(CCCC)CCN(C(C2CCC(NC(=O)C(N3CCOCC3)C)C2)=O)C1 Cc1cc(C(=O)NCC(C2(O)CCN(C(=O)Cc3cc[nH]c3)C2)C)ccc1O C=Cn1ncc(C(=O)NCC2(C(=O)NCCCN(CC(C)C)C)CCCO2)c1N CS(=O)(=O)c1ccc(C(N2CC3CC(NC(C4(CO)CCC4)=O)CC2C3)=O)[nH]1 c12ccc(cc1)S(=O)(=O)CCN=C(NCC1CC3C=CC1C3)NC2.C(C)(=O)OC c1(C(=O)NCC(CN(C(=O)C(F)C2CC2)C)O)ccc(Cl)cc1 Cc1nn(C)c(C(=O)NC2CCN(C(=O)C(F)C3=CCCC3)C23CC3)c1Br C1(C#N)(OC)CC2(CCC(NCCCNS(=O)N(C)C)CC2)C1 CC1(C)C(C)(C(N2CC3CC(NC(=O)CCc4nccs4)C2C3)=O)C1(C)C C1(C(=O)NCCC(C)CCO)(CC)CCCN(C(=O)CC2CCCCCC2)C1 N1(C(C2(OC)CC(C)C2)=O)CCC(C(F)CNC(c2cc(C)no2)=O)CC1 C1(C(=O)NC(CNC(c2cc(C)c(Cl)cn2)=O)(C)C)CN2CCCC1CC2 C(=O)(CCCCCCNC(=O)C(O)C1CCCC1)NCC#CCN(C)C N1(c2nccc(OC)n2)CCC2(CN(C(=O)CC(C)(C)CCOC)CC(C)O2)C1 N1(C(C(C)(C(C)C)OC)=O)CCC2(C1)CN(C(c1cncs1)=O)C2 N1(C(=O)CC2CCC2)CCOC2(C1)CN(C(c1c(Br)nc3n1CCCC3)=O)C2 CC1(C)CN(C(C2CC2(Cl)Cl)=O)CC1C(=O)NCC1CCC2(CCC2)O1 CC(CC(=O)N1CCCC(NC(=O)COCC(=O)OC(C)(C)C)C1)C(C)(C)C C1(NC(C(C2CN(C(=O)CN(C)C(N)=O)C2)OC)=O)CC2CCC(C1)O2 c1(C(=O)NC(CCCC)CNC(=O)CSc2ccccn2)cc(OC)cc(C)n1 c1(C(N2CC(CNC(c3c(CC)nn(C)c3)=O)(OC)C2)=O)ncn2ccccc12 N1(C(=O)C2=NOC(c3ccc(F)cc3)C2)Cc2ccccc2OCC12CC2 C1(NC(C2CN(C(C)C)C2)=O)CCN(C(c2cc(C3CCC3)c[nH]2)=O)CC1CO c1(C(=O)NC(C(=O)NCCC)C)ccoc1CNC(c1ccoc1Cl)=O c1(-c2cc(NC(CC3C(C(=O)OC)C3)=O)on2)cccc(C#N)c1 CCCC(C(=O)N1CCC(O)(CNC(C2CCN(C3CC3)CC2)=O)C1)C(C)C c1(CC(C(=O)OCC)N(C(=O)CC(F)(F)F)c2ccccc2)cccc(F)c1[N+](=O)[O-] N1(C(C(C)=CC)=O)CCC2CN(C(c3cc(Br)ccc3C)=O)CCC2C1 C#CCC(C(=O)NCCCC(C)NC(c1c(C)noc1C(F)(F)F)=O)C1CC1 Cc1cccc(Cl)c1C(c1nnnn1C(C)(C)C)NC(c1ccn(C)c1)C c1(C(=O)NCCN(C(C2SC3C=CC2CC3)=O)C2CC2)n[nH]c2cc(Cl)ccc12 c1(C(N2C(CNC(CC=CC)=O)CC(C)(C)C2)=O)ccc2n[nH]cc2c1F c1(-c2cccc(C)n2)ccc2c(C(=O)NC(C#N)C(N)=O)nsc2c1 C(C(C(=O)NCC12CCCC1OCC2)C(C)C)NC(C1C(OC)(OC)CC1)=O N1(C(C(CSC)OC)=O)CC(NC(c2cccc(-c3ccccn3)n2)=O)C(O)C1 c1(NC(C(=O)NC2CC(C(F)(F)F)(OC)C2)C)ccc2ccccc2c1 c1(OC)ccc(F)cc1C(=O)NC(C(C)NC(c1cc(C)c(Cl)cn1)=O)C(C)C Nc1ccc(C(=O)NCC2CCN(C(C3(CO)CC(F)(F)C3)=O)C2)nc1 c1(OC)cc(OC)nc(C(=O)NCC(CNC(=O)CCC2CCCO2)CO)n1 C1(NC(C2C(=C)C2)=O)CCS(=O)(=O)C12CN(c1ccc3c(n1)CCC3=O)C2 CC1CCC(F)(F)CN1C(c1sccc1CNC(C1CC(=O)C12CCC2)=O)=O Cc1cc(Cl)c(C(=O)NC2CCCN(Cc3cc(C)sc3C)C2C)cn1 C1(CNC(C(COC(C)(C)C)N(C)C)=O)N(C(C2(C)CCC2)=O)CCCC1(C)C C1(C(=O)NCCCN(C(c2cnc(C(C)O)s2)=O)CC)(CO)CC(F)(F)C1 Cc1cnccc1CNC(=O)CNC(c1cc(Cl)cn1C)=O c1(C(C)(C)C)ccc(O)c(NC(C2CC(N)C2)=O)c1 C1(NC(C2CC(CF)C2)=O)C2CC3C1C3C2C(=O)NCCC1CC1C1CC1 c1(-c2ccc(NC(C(c3ccc(F)c(C)c3)CC)=O)cn2)cc(F)cc(F)c1F N1(C(CSCCCC)=O)CCC(C(=O)Nc2ccncc2OC)C(O)C1 c1(CC)cnc(O)c(C(=O)NCC2CCC2NC(C2CC2CC)=O)c1 C12(C(=O)NCC3CC(NC(C(CC(=C)C)C)=O)C3)CC(CO)(C1)OC2(C)C c1(OC)ccc(C(O)CCC(=O)NCc2cc(OC)ncn2)cc1OC C#CC(COC)CC(C)(C)C.C(=O)(C(C)C(C)CC)N1CC2C(C(NOCC)=O)(C2)C1 N1(C(C(C)=O)=O)CC2(CCOCC2C(=O)Nc2ccc3c(c2)OCO3)C1 CCC(c1ccc(OC)cc1)=CC(=O)NC1CC(NC(C2(CC)CCCC2)=O)C1 C1(NC(c2cn(CCC)nc2)=O)C(C)CN(C(c2cscc2Cl)=O)CC1C Cc1cnn2ccc(C(=O)N(CC(C)NC(c3cccn4nccc34)=O)C)nc12 c1(C(=O)NCC(CO)NC(C(C)C2CCC2)=O)csc(C(C)(C)C)n1 C1(NC(c2c(C(C)NC(c3nc(C4CC4)no3)=O)noc2)=O)CCCCC1(C)C C(CCC(=O)NC1C(C(=O)NC)C1(C)C)NC.N12CCC1(C)C2=O c1(C(N2C3C(NC(C(CC)OC)=O)C(C3)C2C)=O)cc2cccnc2s1 Cc1cc(C(=O)NC2CC(C)(NC(=O)CCN(CC(C)C(C)C)C)C2)cc(F)c1 N1(C(C2C(C)(C)CC2)=O)CCC2(CCN(C(=O)CN3CCC(=O)NC3=O)C2)C1 C1(C(N2CC(O)(CCNC(C3CC(C)(C)C3)=O)C2)=O)CCN2CCCC2C1 c1(CC(=O)Nc2cccc(C(=O)NCC)c2)ccc(N2CCCC2=O)c(F)c1 C1(C(N2C(c3cn(C(c4ccccc4F)C)nn3)CC2)=O)CC(=O)NC(=O)C1 CC(C)(C(=O)NC1CCN(C(C2CCCC3OCCC23)=O)O1)S(C)(=O)=O c1(C(N(C(C)CNC(C2CC3CCC2C32CC2)=O)C)=O)cc(F)cc2nc[nH]c12 Cc1ncnc2c1CC(C(N1CCN(C(=O)CCCN(C)C)CC1CF)=O)CC2 C1(CC)(NC(COC2CC(NC(c3coc(C)n3)=O)C2)=O)CCCC1O c1(C(=O)NCC(C)NC(=O)CC2C=CCCC2)nc(Br)sc1C1CC1 N1(CC(=O)NCC2CCCN2C(C2(CCO)CC2)=O)CC(=O)NC1=O CCCCCC(O)CC(=O)NCCCC(CCC)NC(C1CC1(Cl)Cl)=O N1(C(CCCC(=O)OC)=O)CC2COCCC2(NC(c2cncnc2C)=O)C1 C1(C)(CC)C=C(C(=O)N2CCCC2C2(C(=O)NCC3CC4(CC4)CO3)CC2)C1 CC1CCc2[nH]c(=NCc3n[nH]c(=N)s3)nc(N3Cc4c[nH]nc4C(C)C3)c2C1 CC1(C(N)=O)CCN(C(=O)CCOCCOCCO)C1.C12(CC1)C(=O)N2 N1(C(C(CSC)(C)NC(=O)C=C(C)C(F)F)=O)CCC(O)CC1C Cc1ccc(C(=O)NCC2CCC2NC(=O)CC2CSC2)cc1N N1(CCC(C(=O)OCC)C)CCCCC12CCNCC2 N1(C(C(C)Oc2cc(CN(C)C(c3ccns3)=O)on2)=O)CCCC(CO)C1 c1(CS(=O)(=O)N(C2CCOC2)CCCC)nn(C)cc1Cl C=CCCC(CC(C)C)C(=O)NCC1(NC(=O)CC2C=CCCC2)CCC1 N1(C(C2(CNC(C(C)OCCOC)=O)CC=CC2)=O)CC2(C=CCO2)C1 CC1CN(C(=O)C=C2CCSCC2)CCCN1C(c1sccc1I)=O C1(C(=O)NC(CCCCNC(CCC(=O)OC)=O)C)CN(CP(C)(C)=O)C1 c1(CN(C(C(COC)OC)=O)CCCNC(C2CC2(Cl)Cl)=O)cccnc1O N1(C(CCc2ccc(C)cc2)=O)CCC(F)C(NC(=O)C(F)C2CCC2)C1 c1(C(=O)NC2CC(NC(Cc3c(OC)nccc3)=O)C2)ccccc1P(C)(C)=O C1(C(N2C(C)CC2CO)=O)CC2CC2N1C(C1CC(=O)CCO1)=O Cc1cc(-n2cccn2)nc(N2CCC(N(C)C(C3(O)CCOCC3)=O)C2)n1 c1(C(=O)NCC(c2ccc(F)cc2)NC(C2CC2F)=O)ccc2c(n1)CCC2=O c1(N2C(C(C)(C)N(C(=O)C=CC3CCOC3)CCO)CCC2)cc(Cl)nc(S(C)(=O)=O)n1 Cc1nc(C(C)(C)C)oc1C(c1nnnn1C(C)(C)C)NC(c1ccccc1)C C1(C2(NC(CC3(COC)CC3)=O)CC2)CCCN1C(c1sccc1C)=O N1(C(c2cc(C)on2)=O)CCC(C(=O)OC2(Cc3ccc(F)cc3C)CC2)CC1C c1(CC(=O)N(CC(C)NC(C2CC23CC3)=O)C)ccc(Cl)c(Br)c1 N1(C(c2cc(C)n(-c3ccn(C)n3)c2C)=O)CCCN(C(=O)C2=CCC2)CC1C c1(OC)cc(C(=O)NC2CC3(C2)CC(NC(=O)CC2CCCCO2)C3)ccc1O c1(C(=O)NC(C(=O)N(CCOCC#C)C)Cc2cc[nH]n2)ccc(CC)cn1 c1(C(=O)NCC2N(C(C=C(C)CN3CCOCC3)=O)CCC2)ccc(O)nc1Cl N1(C(c2c(CC)ccs2)=O)CCCC12CCN(C(C1CCC3(CCC3)O1)=O)CC2 CC1(C)CCCN(C(=O)Cn2cccc2)C1CNC(C1CCC(C2CC2)C1)=O c1(C(N2CCCC(O)(CNC(CCCC)=O)C2)=O)ccc2c(c1)CCCC2 C12(C(=O)NC3(CNC(c4cc(C(C)(C)C)on4)=O)CCCC3)CC(C#N)(C1)C2 N1(C(C2(CCC=C)CC2)=O)CCN(C(C2CCC2C(C)(C)C)=O)CC1CC N1(C(=O)C=Cc2ccco2)CCC(O)C2(CCN(Cc3cncc(Br)c3)CC2)C1 C1(NC(C(C(C)(C)C)NC(C)=O)=O)C2CCC1CN(C(C1CC(C)(F)C1)=O)C2 C1(C(N2C(C)(CNC(c3ccc(F)o3)=O)CCC2)=O)Cc2ccccc2O1 C1(C(C(=O)N(CCCC)Cc2ccns2)NC(=O)COCCOC)CC(F)(F)C1 N1(CCCC)CCCCC1C(=O)NCC1C2CN(C(=O)CC3CCCCC3)CC12 C(=O)(C#CC1CCOCC1)NC(C(=O)NC(c1cnn[nH]1)C)(C)CO C(CC(C(=O)Nc1nc(C2CC2)no1)NC(C1C=CC1C(N)=O)=O)=CC.NCC c1(NCC2C(NC(CCc3ccc(C)nc3)=O)CCC2)c(Br)cccc1[N+](=O)[O-] C1(CNC(c2cccc(OC)n2)=O)CC2CCC1N(C(c1cc(CF)on1)=O)C2 C1(C(=O)NCCCCC#C)CC(OC)CN1C(C1CCC(C)(C)C1)=O N1(C(CN(S(C)(=O)=O)C)=O)CCC2(CCCN(C(c3cncc(C#N)c3)=O)C2)C1 c1(C(=O)NCC(C)CN(C)C(C2CCCCC2(F)F)=O)ccc2nn(C)cc2c1 N1(C(CSC)=O)CCC(C)C1CNC(c1n[nH]c(C)c1F)=O N1(C(C(C2CC2)OC)C(=O)NCc2ccc(OC)cc2)CCCC2CC1C2(C)C c1(C(=O)NC(C2(CNC(C3CC(CCC)C3)=O)CC2)C)cnn(C)c1C#N c1(C(=O)NCC2(CNC(C(C)O)=O)CCCC2)ccc(Cl)c(F)c1 n1(CC(=O)NCC23C(CN(C(C4CC(=C)C4)=O)C2)CC3)nc(C)c(C=NO)c1C N1(C(CCN(C(c2nc(CCC)oc2)=O)CC2CC2)=O)CCCCC1CO c1(C(=O)NCC(CC=C)NC(=O)C(C(C)C)OC)nccc(C)n1 c1(C(=O)NC2(CN(C(=O)Cc3cn[nH]c3)C)CC2)cc(-c2ccncc2)nn1C c1(C(=O)NC(CNC(C2CC(OC)C2)=O)(C)C2CCC2)ccn(C(C)C)c(=O)c1 c12cc(ccn1)C(=O)NCCCCn1cc-2nn1.C(CCOC)=CC=C C1(C#N)(C(=O)NC2C(NC(CNC(=O)OC)=O)CCC2)CCCO1 N1(C(C(C)Sc2ccc(O)cc2)=O)CCC(O)(CNC(=O)C#CC(C)(C)C)CC1 C1(C)(CC)CC(NC(c2cnccn2)=O)CN1C(=O)C=CCF c1(C(=O)NCC(N2CCCC2c2ccnc(Cl)c2)=O)ccc2[nH]c(=O)cnc2c1 Cc1cnc(Cl)c(C(=O)NC2CCCC2NC(=O)Cc2nnc(C)s2)c1 N1(C(C2(C(N)=O)CC2)=O)CC(CO)C2(CC2)C1 C1(C(=O)NCCN(C(C2C(C)C2c2ccccc2)=O)C2CC2)CS(=O)(=O)C1 N1(C(C2N(C(C(COC)C)=O)CCC=C2)=O)CC2C=CC1CC2 C12(COC(c3c(CC)cccc3)=O)CCC(CC1)C(C)(C)O2 N1(C(C(=O)NCc2c(C)cc(O)cc2C)=O)CCC(S(=O)(=O)C(C)C)C1 N1(C(C2N(C(C3C(C(C)C)OCC3)=O)CC(O)C2)=O)CCOC(C)CC1 N1(C(c2nc(CCC)oc2)=O)CCC2C(C(=O)NC(C3CCCC3)C)C2C1 C1(c2ccc(F)cc2)(C(=O)NC2C(NC(CC3(NC(C)=O)CC3)=O)C2)CCNC1=O c1(C(=O)NC2CC(NC(C(CC)=CC)=O)C2)ccnc(N(C)C)c1 Cc1cc2ncc1NC(=O)N2.C(Cc1ccccc1)(CC(N)=O)N(C)C C1(NC(C(CO)N(C)C)=O)COC2(CCN(Cc3ccc(O)cc3O)CC2)C1 C(=O)(C(CO)C(C)(C)C)N(CCNC(Cn1nc(C)c(Cl)c1C)=O)CC1CC1 c1(NCC2N(C(C3CN4CCC3CC4)=O)CCCC2)ncc(Cl)cc1[N+](=O)[O-] C(C(C)(C)CCCNC(=O)NC(c1cc(C#N)no1)=O)OC C1(NC(C=COCC)=O)CC(C)CN(C(=O)C(C)(C)CC)C1 C1(NC(C#CC(C)C)=O)CC12CCC(NC(c1nnc(C(C)(C)C)s1)=O)CC2 Cc1ccnc2c(C(=O)NC3CCCC3NC(=O)C(O)c3ccsc3)cnn12 N=c1[nH]cc(CCC(=O)NCCCCCNC(=O)Cn2cc(Cl)cn2)[nH]1 c1(N(CCC)C)ccc(S(=O)(=O)NC2CN(C(C)C)CCO2)cc1F N12CCC(CC1C)N2.C(=O)(C1=CCCSC1)N1CCC(C(C)OC)C1 C1(C(=O)NC(CNC(C2(OC)CCSC2)=O)C)CCC(OC(F)F)CC1 CCCC(C(=O)OC)C(=O)NC1CC(NC(=O)CSc2nnc(S)s2)C1 C1(c2cccc(OC)c2)CN(C(C2CCCC2)=O)CCN1C(C1(C)C=CCC1)=O C(=O)(C1Cc2ccc(F)cc21)N(C1CC(Nc2ncnc(O)c2Br)C1(C)C)C c1(CC(=O)NCCC(C)N(C(c2nc(C(=O)OC)sc2)=O)C)cc(C)ccc1F Cc1nc(CC(=O)NC2(CF)CCN(C(=O)CC3CCC(=O)C3C)C2)c(C)s1 c1(OC)ccc2c(c1)C(C(=O)NC(=O)NC1(O)CC(C)CCC1C(=O)O)CO2 C1(O)(C(=O)OC)CN2CCC1CC2.N12CC3CC1CN3C(=O)C1C(C(C)CC1)C2=O C1(N(C(C2CC(CCC)C2)=O)C)CCC(NC(=O)CC2(C)OCCO2)C1 n1(CC)nc(C(=O)NC(CNC(=O)C(F)C2CCC2)C2CCC2)ccc1=O N1(C(C(c2ccc(C)cc2)C)=O)CCC(NS(=O)(=O)Cc2ccccc2)C(O)C1 N1(C(C2CC(C)(CC)C2)=O)CCC(CNC(c2nn(C)nc2C)=O)CC1C c1(C(=O)NCC(CCCC)NC(=O)CSS(C)(=O)=O)ccc2nccn2c1 N1(CCn2cc(C3(CNC(COCC)=O)CC3)nn2)CCC(OC)C1C C1(C(N(CC(C)O)C(C)Cc2ccccc2)=O)C(C(=O)OC)C1(C)C C1(C(=O)NCC(C2CCC2)OC)CN(C(c2cn(C)cn2)=O)CC1C(C)C CC1=C(C(=O)N2CCC(CCNC(=O)Cn3ccnc3C(C)C)C2)CCC1 c1(NC(CC(CC)N(C(C(C=C)CC)=O)C)=O)cc(C)c(C)cc1C C1(C(N2C(C)CC(CC(=O)N(CC(C(C)C)C)C)C2)=O)CC(=O)CC(=O)C1 N1(C(c2c(C)sc(O)n2)=O)CCC(O)(CCNC(c2[nH]ccc2C2CC2)=O)CC1 N1(C(C23N(C(c4cn(CC)nc4)=O)CCC2C3)=O)CCC(C)(N(C)C)CC1 Cc1ccc(C)c(C(=O)NC(C(C)NC(=O)Cc2ccoc2C)C(C)C)n1 c1(CNC(CCOCCC)=O)ccccc1-n1cc(-c2sccc2C)nn1 c1(C(N(C)CCNC(C2(S(N)(=O)=O)CCC2)=O)=O)cc2c(=O)[nH]ccn2n1 C(=O)(C(C)C(O)C(C)C)OCCOc1cc(C)c(Br)cc1 S(=O)(=O)(c1ccccc1F)NCC(=O)NCC(C)N(C(Cc1c(C)noc1)=O)C CC1CN(C(C2CCCSS2)=O)CCN1C(c1coc(Br)c1)=O CN1CC(C(=O)N(C)CC2(O)CN(C(=O)C(c3ccccc3)O)C2)NC1=O N1(C(=O)NCCCCC#C)CCC(CC)(CC)C1 C1(NC(c2cnc(C(C)C)[nH]2)=O)COCCN(C(=O)C(C)Cc2ccnn2C)C1 C1(CC(=O)NC2(CO)CN(C(C3(CC#C)CCOC3)=O)C2)CCCS(=O)(=O)C1 c1(OC2CCCN(CC(=O)NC(c3ncc(C)[nH]3)C)C2)ccc(F)c(Cl)c1 c1(-n2c(C(c3n(CC)cnn3)NC3CC4(CCC4)C3)nnn2)c(C)cccc1Cl Cc1ccc2c(c1)CC(C(=O)NCC1CC(NC(=O)CC3(N(C)C)CCOC3)C1)O2 C12(O)CC(C1)C(=O)N2.c1(CC(C)NC(C)COC)ccco1 C12(NC(COCCC(C)C)=O)CCCC1N(c1ccc(C(F)(F)F)cn1)CC2 C(=O)(C(Cc1ccco1)CN)OC.N12CC=CC1NC2=O c1(NC(C2C(NC(C3(COC)CCC3)=O)C2)=O)cc(Cl)cc(Br)n1 C1(NC(C2(C(N)=O)CC2)=O)CC(C(=O)N2CC(COCC)C2CC)=CC1O C1(CC(=O)NCc2cccc(CNC(c3ccon3)=O)c2)CCC2(CCC2)O1 c1(C(=O)NC2(CC[SH](C3CC3)NC(C3CCN(CC(F)(F)F)C3)=O)CC2)ccncc1 Cc1cnc(CNC(c2ccc(CNC(=O)CC34CCCC3C4)o2)=O)o1 c1(C(N(CCOC)CCNC(=O)C(F)CC2CCC2)=O)sc(C)cc1Cl CC(=NOCC#N)C(=O)NCC(O)C(=O)NC1COC(C)(C)C1 c1(CSCC(=O)NCCN(C(CC(CC)O)=O)C)cc(C)ccc1C N1(C(C(C)NC=O)=O)CC(NC(c2cnn(C(C)(C)C)c2)=O)C(F)C1 C1(NC(Cc2c(C)cnn2C)=O)CCCN(C(=O)Cc2[nH]cnc2C)CC1F c1(C(=O)NCCNC(C2CCC(OC(F)(F)F)C2)=O)cnn2cc[nH]c(=O)c12 Cc1nocc1NC(C1CC1C(C)NC(=O)CCCc1cnn[nH]1)=O C1(C(C)(C)C)C(=O)N1.C(=O)(C(F)(F)CO)NCCOC1CN(C(C)=O)C1 c1(C(=O)NCC2N(C(c3cc(C)n(C4CC4)n3)=O)CCC2)cccc2nn[nH]c12 c1(C(=O)NCC(C)(CNC(c2cscc2C(C)C)=O)OC)cn(C)[nH]c1=N N1(C(C(=O)NCC)=O)CCCOC(CCNC(=O)CC(C)=C(C)C)C1 c1(C(N2CCC(F)(CNC(=O)C(C3CCCCC3)F)C2)=O)nccc(Cl)c1F c1(C(=O)NC2(CNC(c3cc(CC)ncn3)=O)CC2)ccc(S(=O)CC#N)cc1 C(=O)(CCC(F)(F)F)NC1CCCN(C(Cc2n[nH]c(=N)s2)=O)C1 N1(C(C(F)=CCC)=O)CCC(CNC(=O)CCS(C)=O)(COC)C1 C1(C(N2C(CNC(c3cnc[nH]3)=O)CC(OC)C2)=O)CN(C)C(=O)CCO1 C#Cc1ccc(C(N2CCCC2C2(NC(=O)Cc3c[nH]ccc3=O)CC2)=O)cn1 c1(OC)ccc(NC(C23CCC(C(=O)NCCF)(CC2)C3)=O)c(Cl)n1 Cc1cnc(Cl)nc1N(CC(C)CNC(c1cnccn1)=O)C N1(C(C(C)OCCC=C)=O)CC(N=[N+]=[N-])CC1C(=O)NCCn1ccnn1 C(=O)(CCCCCC#N)NCC1CN(C(COC(C)C)=O)CC(C)C1 C(c1ccccc1)=CC(=O)N(C1CC(C#N)C1)CC(O)CCC1CC1 N1(C(=O)OC)CCN(C(=O)CC(C)NC(C2CCCC2C)=O)CC1 c1(CCC(=O)NCCCN(C(C2CCN(C)C2)=O)C)cc(F)cc(F)c1 CCC(C)(C)CCCC(=O)N(C)CC1CCN(C(=O)CN2CC(C)C2)C1 C(C(C)(C)CS(=O)(=O)NC(C1CCOCC1)C(F)F)OC N1(C(CCC(=O)NC2CC(C)OC2)=O)CCN(Cc2ccccc2)CC1C1CC1 c1(C(=O)NC2(CO)CN(C(c3nccs3)=O)C2)ccn2nnnc2c1 CS(=O)(=O)c1ccccc1CN(C(c1[nH]ccc1-c1cncnc1)=O)C1CC1 C1(C(=O)NC(C=C)C)CC2(CCC2)CN1C(C1OCCCC1(C)C)=O Cc1ncc(CCNC(C2CC(C)N2C(=O)CCCC2CCC2)=O)s1 N1(C(c2c(C)nsc2N)=O)CC(CC(=O)NC(C)CCCCO)C2(CC2)C1 c1(N(C(C2(CC=C)CCCN2c2ncnc(=N)[nH]2)=O)CC)ccc(C)c(C)c1 c1(NC)cnccc1C(=O)NC1CCOC1C(=O)NC1COC(C(C)C)C1 c1(C(=O)N(CCCN(C(c2cccnc2N(C)C)=O)CC)CC)ccc(N)cn1 CC(C(CO)NC(=O)CC#N)NC(c1cnn(-n2ccnc2)c1)=O c1(C(N2C(CNC(CC=C=C)=O)CCC2)=O)ccc2cnc(C)cc2c1 c1(-c2ccc(NC(=O)CCOc3ccccc3)nn2)cc(F)ccc1CO N1(CCC(=O)NC(C)CCCCNC(=O)C=CC2CCC2)Cc2ccccc2C1 c1(C(=O)OC)cncc(C(=O)NCC(C)NC(c2ccn(C)c(=O)c2)=O)c1C c1(N(C(=O)C(C)O)C)cc(Br)ccc1Cl.C1(CC(=O)OC)CCN(C)C1=O N1(C(CCCCCC)=O)CCC2CCN(C(C3CN(CC)CCO3)=O)C2C1 c1(C(N2CCC(C(C)NC(c3ccc(CC)[nH]3)=O)CC2)=O)ncnc(O)c1F C(=O)(C(C(CC)CC)OC)N(C1CN(C(c2c(CC)nccc2)=O)CC1(C)C)C C(c1cccc(O)c1)=CC(=O)NCCN1CCN(C(C2CC23CCC3)=O)CC1 C12(CNC(CC(C)C(F)F)=O)CCCC1CN(C(c1ccc(CO)nc1)=O)C2 C12(C(=O)NC3CC(NC(C(N)=O)=O)C3)CCC(CC1NC1(n3cccn3)CC1)C2 c1(C(N2CCC(O)(C(C)NC(=O)C=CC3CC3)C2)=O)ccc(N)c(N)n1 C1(CC(=O)NC(C)(C)CCNC(C2(c3ccncc3)CC2)=O)CC2(CCC2)C1 C1(C)(C(=O)NC(CCNC(C(CSC)O)=O)Cc2ccccc2)CCC(F)(F)C1 C(=O)(C1=C(Cl)CCC1)NCC1CC(NC(C2CN(CCC)C(=O)C2)=O)C1 c1(OC)c(C(N2CCC(NC(=O)CC3CC34CC4)C(F)C2)=O)ccnc1Cl c1(NC(=O)Cn2cncc2N2CCOCC2)ccc2nnc(-c3ccsc3)n2n1 c1(C(N2CCOCC(CNC(C3N(C=O)CCC3)=O)C2)=O)occ2c1CCCC2 C#Cc1cccc(C(N2CC(NC(=O)C=Cc3ccccc3OC)C2)=O)c1F C=CCC(C)(C)CNC(c1oc(CNC(C2CCC(F)(F)C2)=O)nc1C)=O C(C(C)C(F)C(=O)NCc1ccccc1C#N)NC(COCC=C)=O c1(CCC(=O)NCCCN(C(=O)CC2CC2(Cl)Cl)C)ccnc2ccccc12 C1(NC(c2c(CC)cccn2)=O)CC(F)CN(C(C2CCCCN2C)=O)C1 N1(CC)CCN(C(C2CN(C(C3CC(SC)C3)=O)CC2OC)=O)CC1=O C(=O)(CC1=CCCCC1)N(C(C)C)CCN(C)C(c1ccc(C(C)(C)C)nc1)=O c1(C(=O)OC)oc2cccc(F)c2c1NC(=O)NCc1ccccc1C [nH]1ncn2nccc2c1=O.n1(CC(C)O)cc(CONC)nn1 c1(C(N(C2CCN(C(=O)CCC(F)F)C2)CC)=O)cnc2c(cnn2C)c1 c1(C(N2CCC(OCc3nc(C)on3)C2)=O)cccc2c(Br)cccc12 N1(C(c2cccc(C)n2)=O)CCC(CNC(c2ccc[nH]2)=O)C(C)C1 C(=O)(CC1Cc2ccccc21)N1CC(NC(CN(C)C)=O)CC(F)(F)C1 C1(C(N2CC3(CC(NC(C4CCN(CC)C4)=O)C3)C2)=O)CCC(=O)CC1(C)C CC(C(=O)N1CCC2CC12C(=O)NOCc1ccccc1)S(C)(=O)=O N1(C(C=Cc2c(C)ccs2)=O)CCCC(NC(=O)CN2CCCCC2)C1C C(=O)(CCC1=NNC(=O)CC1)NCCC1CCN(C(C2C(C)CC2C)=O)CC1 C1(NC(c2nc(Br)c[nH]2)=O)CCN(C(=O)Cn2cnnc2)C1c1ccccc1 C=CCCC(=O)NC1CCCC1CN(C)C(C1CC1c1ncc[nH]1)=O Cc1cc(CC(=O)NC23CCN(C(C4(C)CSC4)=O)CC2C3)ccc1O C(N=c1[nH]c(=NC2CN(C)C3(CCOCC3)C2)c2[nH]ccc2[nH]1)c1c(C)nccc1 C(CN=c1[nH]ccn2ncc([N+](=O)[O-])c12)c1cc(C)n(C)n1 Cc1cccnc1CN(C1CC1(C)C)Cc1nnnn1Cc1ccccc1 n1(CCN(CC)CC)cc(C#CCNC(c2nc(Br)ccc2N)=O)nn1 c1(C(=O)NC(c2ccccc2)CNC(=O)C(Cl)=CCl)nnn2c1CCC2 CC(C)(CCCF)C(=O)NCC12CC1CN(C(c1cc(C#N)c[nH]1)=O)C2 N1(C(C(CC=C)C)=O)CC2(CO)CC1(C(=O)Nc1ccccc1CCO)C2 N1(C(C2CCN(CC)C2)=O)CCC2CN(C(=O)C=Cc3cccc(Cl)c3)CC12 N1(C(C2CC(C(C)C)OCC2)=O)CCCN(C(c2csc(Cl)n2)=O)C(CO)C1 c1(C(N2CC(CC(N3CC(CC(C)C)C3)=O)(OC)C2)=O)ccc(O)nc1 CC(CC(=O)NCCN(C(=O)Nc1ccco1)CC1CC1)CCc1ccccc1 C1(CNC(c2cc(CNC(=O)C=CC(F)F)sc2)=O)(CO)CCOCC1 C(=O)(CC(C)(O)C(F)(F)F)NC(C)CCCNC(=O)CCC1CCCCCC1 N1(C(C2C(OC)(OC)CCC2)=O)CCC2(CCC2)C(CNC(=O)CS(N)(=O)=O)C1 C1(NC(C(CCC)OC)=O)CN(C(c2ccc(F)c(N)c2)=O)CCC1(C)C C12(C(=O)NC3CN(C(C(C)(O)C4CC4)=O)C4(C3)CCC4)CC3CC(C(=O)N1)C2C3 c1(-c2n(CCOC(C)C)nc(Cn3ccnc3)n2)nc2ncccn2n1 C=CC1(C(N2CC3(CNC(=O)CC4CC(=O)NC4=O)CCC2C3)=O)CCOCC1 C(=O)(C(C)(C)C(C)(F)F)NC1C(NC(C2C(c3cc(C)no3)C2)=O)COC1 c1(NC(C2CSCCN2C(c2cc(O)no2)=O)=O)ncc2c(n1)CCNC2 c1(C(=O)NCC(CNC(C(C)CN(C)C)=O)(C)O)ccc(F)c2cccnc12 C1(C(CNC(c2c(C)nn[nH]2)=O)(C)O)CCCN(C(=O)CCNC(N)=O)C1 S(=O)(=O)(c1ccc(C(=O)NC2CC(C)N(C(=O)C(C)=C(C)C)C2)cc1)NC NS(=O)(=O)C1CCN(C(C2CC(=O)N(C3CCS(=O)(=O)C3)C2)=O)C1 Cc1ccc(Cl)c(C(=O)NC2CC(NC(c3cnc(C#N)s3)=O)C2)c1 c1(CCC(=O)NCC2CN(C(C3CSCCS3)=O)C2)nc(-c2ccccc2)no1 N1(C(CCCC=C)=O)CC(=O)NCC1C(=O)NCc1c[nH]nc1C(C)C C(=O)(C1=NOC(C)C1C)NC1CC(NC(C(CC#C)C)=O)C1 C1(C(=O)NCC(CNC(C=C(C)C)=O)(C)O)CCCN1S(=N)(=O)N(C)C c1(OC)c(Cl)cc(C(N2CCC(NC(C3CC=C(C)CC3)=O)C2C)=O)nc1Cl c1(N2CCCC(CNC(C(n3ccc(C4CC4)n3)C)=O)C2)nc(Cl)ncc1Cl C12(NC(C(CC=CC)NC(=O)C3CC3)=O)CCC(C(=O)OCC)(CC1)C2 N1(C(C2CSCN2C(C2CC(CC3CC3)C2)=O)=O)CC(O)C(C2CC2)C1 C(=O)(CCCCC(F)(F)F)N1C(C2(C(=O)OC)CC2)CCC1 c1(OC)cc(C)ccc1COc1nc(N2CCC(O)C2)cc(C)n1 c1(OC)cncc(C(=O)NC2(CO)CCN(C(=O)CC3CC4(CC4)CO3)C2)c1C C1(CCN(C(Cc2nc(NC(C)=O)sc2)=O)CC)CN(C(=O)C=CCF)CC(C)O1 N1(Cc2ccc(CCCC)s2)CC(NC(=O)CC(O)C2CCCC2)CC(C)C1 N1(C(C2COC(C)(C)OC2)C)CCOCC1C1CCCO1 C1(CCNC(c2cn(CC(F)F)cn2)=O)COCCN1C(c1c[nH]nc1Cl)=O c1(C(=O)NCC(C)N(C(COC(C)C)=O)C)cccc2c1C(C#N)C2 c1(N(C)C)cccc(NC(C2CC(O)CN2C(=O)CN2CCSCC2)=O)c1 C(c1c(F)cccc1F)=CC(=O)N(C1CCC(CNC(c2cscn2)=O)CC1)C Cc1ccc2cc(C(=O)NC3CCN(C(C4C=CC(=O)N=N4)=O)C(C)C3)ccc2n1 C1(C(=O)NCC2(CO)CC(C)(C)C2)CC2C=CC1N(C(C1CC(C3CC3)C1)=O)C2 n1(C(C(N2CC(C)(NC(c3ncc(C)c(C)c3)=O)C2)=O)C)c(C)cc(O)cc1=O C(=O)(CC(C)CC(C)C)NCCCCC(N1C(C=C)CCC1)=O CCCC(C(=O)NC(C)Cc1cccs1)NC(C1(CC(C)C)CC1)=O c1(C(N(CCNC(=O)CCc2ccon2)C2CC2)=O)c(Cl)cccc1Br CCC(C(=O)N1CCCOC(CNC(=O)CC(C)(C)CCC)C1)C(C)(C)CC c1(NC(C2N(C(CSCC)=O)CC2)=O)cnc(OC)nc1 CC1(C)CC(C(=O)NC2(CO)CN(C(=O)CCc3cccnc3F)C2)CNC1=O N1(C(C)=O)C2CCC1CC(NCC13CCC(CC1)CN3)C2 C(=O)(C(CC(=O)NC1CC(CNC(C2CCNC2=O)=O)C1)C(C)=O)OCC C1(c2n(C)cnc2)CN(C(C2CN(S(C)(=O)=O)C2)=O)CC1NC(=O)CSC1CC1 C(=O)(C1=NOC2(CCOC2)C1)N1CC(CCNC(C(C)CS(C)(=O)=O)=O)C1 c1(C(=O)NCCC2CN(C(C=CS(C)=O)=O)C2)cc2c(=O)cc[nH]c2s1 c1(C(N2CC(OCCCC#C)C2)=O)ccc(CNC(=O)C(C2CCC2)OC)s1 Cc1cc(CNC(=O)C(C)C(C)NC(=O)C(C)NC=O)cc(O)n1 c1(C(=O)NCCC(CCNC(C2=CCC(C)CC2)=O)C)cc2cn[nH]c2cn1 C1(C(N2C(C)(C(=O)NC)CC2)=O)CC(O)CN1C(c1cc(O)ncc1F)=O C#Cc1cccc(C(N2CC=CC2(C)C(=O)NCC2(O)CC(CO)C2)=O)c1C N1(CC(C2(c3ccc(Br)cc3)CC(F)C2)=O)CCS(=O)CC1c1ccccc1 N1(C(C23CC(NC(C=CC)=O)C(OC2)C3)=O)CCC(CO)C12CCC2 C1(C(=O)N(CC(C)N(C(=O)CO)C)C)(CC)CCC(F)(F)CC1 c1(C(=O)NCC(F)CNC(C2CCCC23CC3)=O)cc(F)c(F)cc1F C(=O)(C1=C(C)OCCS1)NC(CNC(CCc1onc(CC)n1)=O)C C(=O)(C1Cc2c(Cl)cccc21)NCC1OCCCN(C(c2c(=O)ccn(C)c2)=O)C1 c1(C(=O)NCC2CN(C(Cc3nc(C)c(C)[nH]3)=O)CC2C)ncnc2sccc12 C1(C(=O)NC(c2ccc(CNC(=O)C=CCF)cc2)C)CC2C=CC1O2 N(C1c2ccccc2C2CC1C2)C(=O)CN1CSCC1=O c1(C(=O)NC(CN(C(Cc2c(C)ccnc2)=O)C)(C)C)coc2cc(F)ccc12 N1(C(C(COC)C)=O)CCC2(CCCC2NC(c2cc(O)nc(Cl)c2)=O)CC1 c1(OCC)cccc(C(=O)NCC(CNC(c2c(O)cccc2Cl)=O)OC)c1O c1(C(=O)NCCCCC(C)NC(=O)C(C)CCN(C)C)ccc(Cl)nc1N c1(C(N2CC(CNC(c3cn(C4CC4)cn3)=O)OCC2)=O)ncnc2sccc12 CCCS(=O)(=O)CC(=O)NCC1CCCN(C(C2CCC(C)(C)C2)=O)C1 N1(CC(c2ccc(Cc3ccccc3)o2)=O)CCCCC(n2ccnn2)C1 c1(CCC)cc(C(N2CC(C)(NC(C3CN(C)C(=O)N3)=O)C2)=O)ccn1 c1(C(N2C(C)CC(NC(C3CCC(CC)O3)=O)C2)=O)c[nH]cc(Cl)c1=O C1(NC(C(COC)O)=O)CCCC12CN(C(C1CCOC(C)C1)=O)C2 N1(C(C2(C)CC2(F)Cl)=O)C2CCC1CC(CNC(c1cc(C(F)(F)F)c[nH]1)=O)C2 C1(F)(CNC(CC(C=C)(C)C)=O)CCCN(C(C2CCN(C)C2=O)=O)CC1 C1(NC(=O)C=CCF)CCN(C(=O)CC(F)F)C1Cc1ccccc1 Cc1cc(O)c(C(C)NCC(Cc2ccccc2)C(=O)O)nn1 N1(C(C(C)(C)c2cscc2Cl)=O)CCC2(CCN(C(C3COC(=O)N3)=O)C2)C1 CCC(C)C(C(=O)N1CCCC1C1(C(=O)NCc2cnn[nH]2)CC1)NC(=O)OC C1(C(=O)NC2C(CNC(CNC(N)=O)=O)CCC2)CC1C1CCCCC1 O=C1CN(C(=O)C(O)Cn2cncn2)C(C(=O)NC2CCC(F)(F)C2)CN1 C1(NC(CNC(C(CC)C)=O)=O)CN(C(=O)CCn2ccnc2C)C(C)(C)C1 O=C(CCC(F)(F)F)NCC1C2CN(C(=O)Cc3cn4ccsc4n3)CC12 C(=O)(CCCC#N)NC1C(NC(c2n(C(C)C)ccc2)=O)CCC1 CC(C)C(C(=O)NCCCN(C(=O)C(F)(F)c1cscn1)C1CCC1)C(=O)OC c1(C(=O)NCC(c2ccccc2)N(C(C(C)CF)=O)C)ccc(=O)n(C)c1 c1(C(N2CC(CNC(=O)COC3CCCOC3)C2)=O)cccc2c1CCC(=O)N2 c1(C(=O)NC23C(CN(C(CC=CC)=O)C2)C3)ccc2c(c1C)OC(F)(F)O2 N(C1c2ccccc2CCC1(C)C)C(C1NCC(C)C1)=O c1(CC)ccc(CO)cc1O.N1(C2c3nnnn3CCCO2)CC(OC)CC1=O C1(C(=O)NC23CC(NC(C(C)OCCC(C)C)=O)(C2)C3)CCC(F)(F)C1 N1(C(C2CCCC(O)C2)=O)CCC2(CCCN2C(c2ccc(Cl)c(F)c2O)=O)C1 N1(C(C(C2CCCC2)NC(C(C(C)C)OC)=O)=O)CC2CCC1CC2 c1(C(C(=O)NC(c2nnnn2C)CC)N)ccccc1Cl C=C(C)CC(C(=O)NC1CC(N(C)C)C1)NC(=O)CCSCCCC N1(C(C(CC)NC(C)=O)=O)CCN(CC(C)NC(c2ccc(C)s2)=O)CC1 C#Cc1ccc(-c2cc(CN3CCN(C)CC3CO)n[nH]2)c(O)c1 C1(CC(N2CC(CNC(C3(C(N(C)C)=O)CC3)=O)C(O)C2)=O)CN2CCC1CC2 c1(NCc2c(C(N)=O)cc([N+](=O)[O-])cc2)ncc2c(n1)-c1ccccc1CC2 N1(C(CNC=O)=O)CCN(C(=O)CSCC(=O)OCc2ccccc2)C2CCC12 c1(C(N(CCCCCC)CCNC(CCC=C=C)=O)=O)cc(O)ccc1C(C)C c1(C(N2CC3CN(C(CC(CCOC)C)=O)CC3C2)=O)coc2c(C)cccc12 c1(N(CCSC)Cc2ccc(OCC(=O)OCC)cc2)nc(CC)ncc1Br C(=O)(CC1OCCc2sccc21)NC(C1N(C(c2sc(C)c(O)n2)=O)CCC1)C N1(CC)CC(C(N2CCCC2CNC(=O)Cc2cncc(C)c2)=O)CCC1=O C1(OC)CC(C(=O)NCC2CC=CCC2)N(C(=O)C=Cc2cn(C)nn2)C1 c1(-c2cn(C3C(C(c4ccccc4F)C)COC3)nn2)cc(N)ccc1F c1(NC(Cc2nc(N(CC(C)OC(C)=O)C)sc2)=O)ccc(CO)cc1.C(F)(F)F c1(C(N2CCCC(C(N)=O)C2)=O)cc2n(n1)CCN(C(c1cccnn1)=O)C2 N1(C(c2cc(C)nc(C)c2)=O)CCC2(CCN(C(=O)CC3CCCC3)C2)C1 CC1CC(C(N2CC=CC(NC(C3CCC(=O)N(C)C3)=O)C2)=O)CC(=O)N1 c1(C(=O)NCC(CNC(CNS(N)(=O)=O)=O)O)ccc(C(F)F)o1 C1(C(N2CCC(N(C)C(c3csc(C(N)=O)n3)=O)C2)=O)CCCCS1(=O)=O CC(C)(CCCNC(=O)Cc1ccc(Cl)s1)NC(C1CC1c1cccs1)=O O(NC(=O)CCC1CC1CNC(=O)COCC1CC1)CC(C)O C(=O)(C(C)(C)O)NCC(CNC(c1cnc(CC=C(C)C)s1)=O)OC c1(NC(CC=C)C2CC2)cccc(N2CCCCC2)c1 C(=O)(CCS(=O)(=O)N1CCCC1)NCC1N(C(c2cc(OC)no2)=O)CC1 c1(C(N(CCNC(CN(C2CC2)CC)=O)C)=O)nccc2c[nH]nc12 C12(CNC(C3C(C)CCC3)=O)CC1CN(C(c1cc(CO)on1)=O)C2 C1(C(=O)NCC(F)CNC(c2occc2CN(C)C)=O)(CC)CCOCC1 C1(C(=O)NC(c2nn[nH]n2)CC)CC(C)CCN1Cc1ccccc1 C(C(O)C(=O)NCc1cc(C(N2CCCC2C(=O)N(C)C)=O)co1)SC C(=O)(CC1=CCN(C(=O)C(C(C)O)NC(C)=O)CC1)NC(CCOC)C(C)C CC(CCC(C)(C)C)C(=O)NOCC(=O)NCC12CCCC1CCC2 CN1CCn2ncc(C(N3CC4CC(C3)N(C(C3C5COCC35)=O)C4)=O)c2C1 C12(C(=O)N(C3CC(CS(C)(=O)=O)C3)CCO)CC(Br)(CO1)C2.CC(C)(C)SC C1(C(=O)NC(C(C)NC(c2ccc(F)c(O)c2)=O)C)CCCC12OCCO2 c1(C(N2CCC(CCNC(CN(C3CC3)CC)=O)C2)=O)ccc(C(N)=O)cc1 c1(CCN2CCC(NC(c3ccccc3)=O)C2)ccc(F)cc1F C12(NC(c3cccc(OCCC)c3)=O)CCC(C1)N(C(c1ccc(Cl)s1)=O)C2 c1(CC(C2CCCC2)OC)ncccc1C(=O)NCc1ccc(-c2cc[nH]n2)o1 N1(C(c2scc(C(C)=O)n2)=O)CC2(CCN(C(C)=O)C2)C1 c1(C(N2CCC(=CCNC(C3C(=C)C3)=O)CC2)=O)cccc2ncnc(O)c12 CCC(CC)C(=O)NC1CC(CC(=O)OC)C1.C12CCN(C1)C(=O)NCC2 C1(O)(CNC(C(C)CCNC(=O)OC(C)(C)C)=O)CCN(C(=O)CC(C)F)CC1 C1(CNC(C(C)C2CC2)=O)(NC(c2cc(F)cc(F)c2)=O)CCC(F)(F)CC1 c1(N(CCC(C)(F)F)C)nc(=N)[nH]c(=NCC2CCOc3ccccc32)[nH]1 c1(CC(=O)NC(C2CC=CCC2)C(=O)NC2(COC)CC2)ccn(C)n1 c1(OC)cscc1C(C)(C)NC(=O)COC(C)C.N12CCCC1CC2=O C(CCC(O)C(=O)N(CC(C)(C)C)CC1CCCCC1)NC(C)=O n1(CC(=O)NC(C)CCCNC(=O)CC(O)C(C)(C)C)c(O)nc2ccccc12 N1(C(c2csc(C3OCCO3)c2)C(=O)NCCCOC)CC2CCCCC2C1 c1(C(=O)NC2C(C)CCN(C(C(=C(C)C3CC3)F)=O)C2)nn(C)c2c1CSCC2 N1(C(C(c2n(C)ccc2)=O)=O)CCCC(C2CN(C(C3(C)CCC3)=O)C2)C1 CCCCC(O)CC(=O)Nc1ccc(NC(c2occc2C)=O)cc1C Cc1cnc(NC2CCCN3CCCCC23)c(S(=O)(=O)NC23CCC(CC2)CC3)c1 c1(CN2CC(N3CCN(C(C4CN(C)C4)=O)CC3)C2)ccc(F)c(I)c1 c1(CC)cc(C(=O)NC(C)(C)CCCNC(c2ccc(F)s2)=O)cc(Cl)n1 N1(C(C2CCN(OC)CC2)=O)C2CCCC1CN(C(C1CN(C)C(=O)N1)=O)CC2 N1(C(CNC(C=CSC)=O)C)CCN(C(C2OCCC2C(C)C)=O)CC1 N1(C(C)(CC(C)C#N)c2n(CC=C)nnn2)CC2CCCN2C(=O)C1C C#Cc1ccc(C(N2CC3CC3(CNC(c3nnc(C)cc3O)=O)C2)=O)cc1Cl C1(C(N2CC(NC(c3c(C)con3)=O)C(F)C2)=O)CCc2ncnn2C1 Cc1[nH][nH]c(=N)c1C(N1CCC(CC(C)NC(c2[nH]ccc2C2CC2)=O)CC1)=O C(=O)(C(CC(C)(C)C)NC(=O)C(C)SC(C)C)N(CCCC#C)C c1(C(=O)NC(C2CCC2)C)c[nH]c2c(-c3ccc(NCCC#N)cc3)cccc12 C(=O)(C1=CCCC1)NCC(C)N(C)C(c1cn(C)nc1C(C)(C)C)=O c1(CC(=O)N(C2CCC(CNC(c3cc(C4CC4)on3)=O)C2)C)cncc(F)c1 C(CCC)(CCCNC(c1cccc(F)c1)=O)NC(C(CCC)C)=O C1(n2cnnn2)(CNC(C2C(NC(C3CC(CF)C3)=O)CC2)=O)CCCCC1 c1(-c2cc(C)nn2CC(N2CCOC3CC23)=O)ccc2[nH]c(C(N)=O)c(C)c2c1 C1(C(=O)NC(CO)C2CCC2)CCCCN1C(=O)C=CC1CCOC1 C(=O)(C(C)(C)COC)NC(C(C)NC(C1C(C=C)C1)=O)(C)C C1(NC(C(C)OCCCCCC)=O)C=CCN(C(c2sccc2CC#N)=O)C1 c1(C(=O)NCCCN(C(C)=O)CC)cc2cccnn2n1 c1(CNC(=O)NCC(C)(C)CN)cccc(C2CC2)c1 C(CN=c1cc(C2CC2)nc[nH]1)(N(C(=O)C(c1ccccc1F)(F)F)C)C1CC1 C1(NC(C2CCN(C)C2)=O)(CNC(c2snc(O)c2Cl)=O)CC2CCC1CC2 c1(C(N2CC(C)C(NC(C34CC3C4)=O)C2)=O)ccc2nc[nH]c2c1F C(C)(C)(CCCC(=O)NCCCCCCF)NC(CN(C)C)=O n1(OC)nccc1CNC(=O)NCCOc1ccccn1.C(CNCC)OC C123CCC(CC1)(C2)C(C)C1CCCN1C3=O.c1(COCC)ccc(OC)nc1 Cn1nnc(CNC(C23C=CC(CC2)C3)=O)c1C(=O)NCC1CSCCO1 C1(C(=O)NCC(F)C2CCC2)(COC)C=CCN1C(=O)C(C)c1ccco1 C1(NC(C2(C)CCNC2=O)=O)CC2CC1N(C(c1cc(C(N)=O)cs1)=O)C2 N1(C(COC)=O)CCC2(CC1)COC(C)C2NC(=O)CN C1(CNC(C=CCC(=O)N(C)C)=O)CCCN(C(c2cc(C#N)on2)=O)CC1 c1(C(=O)OC)cn(CC(=O)NC2CC2NC(=O)C(F)(F)C(F)(F)F)c(=O)nc1O c1(C(=O)NC2C(CNC(C(CC#C)(C)C)=O)CCC2)cc2nnn(C)c2s1 C1(C2(C)CC2)C(=O)O1.c1(CO)ccsc1.CC(C)(C)OC(=O)NC1CC1C(=O)NC N1(C(CCC(=O)NC2CC2)=O)CCC2CCC(NC(=O)CCCC3CC3)C1C2 c1(OC)ccc(C)c(C(=O)NC2CCN(C(=O)Cc3cnsc3)C2(C)C)n1 c1(NC(C2C(C(C)=O)C2(C)C)=O)ccc2c(c1)CCCS2 Cn1nc2c(c1C(N1CC(CCNC(=O)C(N3CCOCC3)O)C1)=O)CCCC2 c1(C(=O)NC2CN(C(C3C(C)OC(=O)N3)=O)CC2C)cccc2sncc12 C(C)(N=c1ccc(Oc2cccc(CO)c2)n[nH]1)c1ccc(CC)cc1 C(c1cccc(OC(F)(F)F)c1)=CC(=O)NCC1CCC(NC(C2CCC2)=O)C1 c1(OC)ccc(-c2nc(-c3ccccc3)nn2CCC(C)C)cc1C N1(C(C)C)CCC(C(=O)NCCc2csc(CN3CCCC(N(C)C)C3)n2)CC1 c1(-c2occc2)ccc(CNC(=NCC2CC2)NCC2CC2)cc1 Clc1ccc(-c2nc(-c3cnn(C4CCCC4)c3)n(C3CC4CCC3C4)n2)nc1 Cc1cc(C)c(C#N)c(NC2CN(C(c3ccc(F)c(Cl)c3F)=O)CC2C)n1 c1(C(=O)NCC2(NC(CC(C)CN(C)C)=O)CCC2)cc2cn[nH]c2cn1 C12(C(=O)NCCC3(CNC(c4n(CC)cnn4)=O)CC3)CCC(F)(CC1)CC2 c1(C(N2CC(NC(CCc3cnc(C)o3)=O)C2)=O)cc(F)ccc1NS(C)(=O)=O C1(C(=O)NCC2(CNC(c3c(C)nc(CC)o3)=O)CC2)CCC(C#N)CC1 C1(COC)(NC(C2CC(C(F)(F)F)CN2C(C2CC(F)(F)C2)=O)=O)CCOCC1 C1(=CC(=O)NCC2CCC(NC(c3ncc(Cl)cc3Cl)=O)C2)CN2CCC1CC2 N1(C(C(CC#C)C2CC2)=O)CC(C(=O)NC(C)CN(C)C)CCC1(C)C N1(C(C(CCC)OC)=O)CC2CC(C1)CN(C(c1cccc(C(F)F)c1)=O)C2 C(C)(C(O)C(=O)NCCN(C1CCCCC1)C(=O)Cc1sc(S)nc1C)OC CC(Cc1ccccc1)CC(=O)O.C(C(F)F)C1C(C)C1 c1(C(C)C)csc(C(C)NC(C)C(C)(C)OCCN(C)C)n1 C(=O)(CC1=CCOCC1)N(c1ccc(Cl)nc1)C1C(NC(CC2C(C)OCC2)=O)C1 N1(C(CCCC(C)C)=O)C2CCCC1CN(C(C1CS(=O)(=O)CCO1)=O)C2 Cc1cc(C(C)C(=O)N(CCNC(=O)CC2CCOC2)C2CC2)cc(F)c1 c1(OC)ccccc1CC(=O)C(N1CC(CNC(C2CC2C)=O)CC1C)=O CCC(CC)C(C1CCCC1)Nc1cn(Cc2ccc(F)cc2)nc1OC c1(CC(N2CC(N(C(CN(CCC#C)C)=O)C)C(O)C2)=O)ccc2occc2c1 C1(CC(C)C)C(=O)O1.c1(SCNC(C(c2ccccc2Cl)OC)=O)ccccc1C N1(C(C2(N(C)C)CC2)=O)CC(CNC(c2sccc2CO)=O)C2(CC2)C1 N1(C(c2nc(OCC)sn2)=O)C2CCC1C(NC(c1[nH]cnc1C)=O)C2 CC(C)C(C)(CNC(=O)CC(c1cccc(F)c1)O)NC(c1coc(O)n1)=O c1(C(=O)NC(COC)COC)cc(CCNC(=O)C(C)CC2CCCCC2)on1 N1(C(=O)CC2CCCC(C)C2)CCC(N(CCO)CC2CC(C(=O)OC)C2)CC1 c1(C(=O)NC2(CC=C)CN(C(c3ccc(SC)s3)=O)C2)ccc2c(c1)COCC2 c1(NC)ccc(C(N2CC=CC(NC(=O)Cc3cc(C)[nH]n3)C2)=O)cc1F C1CCC(=O)NOCC(=O)N1.C(C(N)C(=O)N(C)C)OCC C1(c2ccccc2)(NC(=O)NCCN(C)NC(=O)OC(C)(C)C)CCCO1 c1(SC)nc(C(N2CC(C(N)=O)(CNC(=O)C(c3cnccn3)C)C2)=O)cs1 c1(C(N2C3(CNC(CCSCC)=O)CCC3CC2)=O)cc2sc(Cl)cc2s1 c1(C(N(C2CC(C(=O)NCc3cnco3)C2)C)=O)ccccc1N1CCCC1 C1(CNC(CNC(c2ccc(Cl)cc2)(CC)C)=O)CCC2(CCC23OCCO3)O1 N1(C(C2C(NC(=O)CSc3ccc(F)cc3)CCC2)=O)C2COCC1CC(F)C2 c1(CC(=O)NC2C(C)N(C(=O)C=Cc3nccs3)CC2)ccc(C#N)nc1 c1(CNCC2N(C(c3cnco3)=O)CCOC2)c(Cl)ccnc1Cl CCCCCCOCC(=O)NCCOCCN(C(=O)CC1CSCCS1)C CC1CCC(NC(c2ccc(C(F)F)cc2)=O)CN1C(=O)C(F)=CCCl C1(NC(c2ccc(C=C)cc2)=O)CCN(C(=O)C(C)C#N)C12CCCC2 c1(OC)cnccc1C1CC1.c12ccc(o1)CNC(=O)C1CCN1C2=O C1(NC(C(C)(CO)NC(C)=O)=O)CC2(C1)CN(C(=O)Cc1ccsc1)C2 c1(C(=O)NCC(CC)(C)NC(=O)C(C)C2CC2)cc(C)cn2ccnc12 Cc1cc(-n2nc(CCN(C)C)nc2CC2CCCS(=O)(=O)C2)cc(Br)c1 N1(C(CCC=C(C)C)=O)CCC2CN(C(=O)CC3CCC(C)C3)C(C)C12 c1(CC)[nH]nc(C(=O)NCCNC(C2(SC3CC(SC)C3)CC2)=O)c1C N1(CCNC(CC2CC(CC)OCC2)=O)CCCN(C(c2n[nH]cc2C)=O)CC1 Nc1cc(-c2cn(C3CCN(C(C4CC5CSCC5C4)=O)CC3)nn2)ccc1Cl CC(CC(C)NC(c1ccnnc1Cl)=O)N=c1nc[nH]s1 C1(NC(C2(CC3CCCC3)CCCC2)=O)(CO)CN(C(=O)CCCC2CCC2)C1 C1(CC=C)(C(=O)NC(C=C)CO)CN(C(C2(SC)CCC2)=O)C1 CC(C)CC(CNC(c1ccc(C2CC2)cc1)=O)NC(=O)C(C)N1CC(C)C1 c1(CCNC(CC2OCCN(Cc3cn(C)nc3)C2)=O)coc2ccccc12 c1cc(NCC2CN(c3nncs3)CCO2)n2nccc2c1 CC1CC(c2ccccc2)CCN1C(=O)Cn1cc(-c2cscn2)nn1 C=CC(C)(CCOC)C(=O)N1CCC(NC(=O)CSc2cccs2)C(CO)CC1 N1(C(C2(C(=O)OC)CC2)=O)CCC(=CCNC(=O)C(C)(C)c2cc[nH]n2)CC1 n1(Cc2cccc(CC(=O)NCC(COC(C)C)O)c2)ccc2ccccc12 c1(C(=O)NC2CC2NC(=O)C(O)C2CC2)cc(O)nc(Cl)c1 c1(C(=O)NCC(C)N(C(=O)CCC2CCCOC2)C)ccc(CO)cn1 Cc1cncc(CN2CCC(CC(=O)NC3CC3C(N)=O)CC2)n1 C1(C2CCN(C(c3cc(CN(C)C)c[nH]3)=O)CC2)(NC(C(C)C2CC2)=O)CC1 c1(C(=O)NCC(C)NC(C2COCCN2C)=O)noc2ncccc12 Cc1cncnc1C(N1CCSCC1C(=O)NCCC1OCCC1C)=O c1(C(C)=O)cnc(N2CCC(NC(c3ccc(F)cc3F)=O)C2)c(C)c1 N=c1[nH]c2ncc(C(=O)NC3CCC3NC(c3cnn4c3CCCC4)=O)cc2s1 C1(CNC(C2CC23CCN(C(=O)C=Cc2ccccc2)C3)=O)C2CCCCCC12 CCC(CC(F)F)C(=O)N1CC(CCCCNC(c2nc(Cl)ccc2F)=O)C1 Cc1c(Cl)ccc(F)c1C(=O)N(CCCCC(C)C)C CC1(NC(c2ccc(O)nc2)=O)CCN(C(C2CCC(O)C2)=O)C1 C1(C(=O)NCC2N(C(C(C(C)(C)C)O)=O)CCCC2)CCCCN1S(N)(=O)=O c1(CC(N2CC(c3nnc(CC)s3)C2)=O)ccc(C)cc1F O=S(=O)(c1ccc(NC2CCCn3ncnc32)c(Br)c1)NCCCCCF c1(C(N(CCCCN(C(=O)CCC2CC2)C)C)=O)c(F)ccc(F)c1O C(=O)(CCN=c1[nH]ccs1)NCCCOCCN(C)C(C1CC2CCC(C1)O2)=O c1(CC)cccc(NC(=O)Nc2cc(CS(C)=O)ccc2Cl)c1C C1(NC(C2C(C)=C2)=O)CCCCC12CCN(C(=O)C1CCCc3ccnn31)CC2 c1(OC)cc(C)cc(C(=O)NCC2C(C)CCCN2C(=O)C(F)OC)c1C CN1CC(NC(=O)CCN(C(=O)CC2CNC(=O)O2)CCO)CO1 c1(CC(=O)NCC2CC3(CC3)CN2C(=O)COC(F)F)cccc2ccoc12 C1(C(F)F)(CNC(c2ccc(CF)cc2)=O)CCN(C(C23CCCC2C3)=O)C1 c1(C(=O)NC(CCC)CO)c[nH]c2cc(F)ccc12 N1(C(CC(CC)OC)=O)CCN(C(=O)CCc2nnc(O)n2C)CC(O)C1 c1(C(N2C(CNC(c3ncc(CC)cn3)=O)CCC2)=O)ccc(=O)n(CC)n1 C(C(C)(O)C(=O)NCCC(C)N(C(=O)COc1ccc(F)cc1)C)OC c1(OCCCC)ccc(C(=O)NC(C)CNC(c2ncsc2C(C)C)=O)cc1 N1(C(C2CCC(OC(F)(F)F)C2)=O)CCOC(C(F)(F)C(F)(F)F)C1 c1(COCC)noc(CN(C(c2ncnn2C)C(=O)NC(C)C)C)n1 N1(C(C2=CCC(NC(COC(C)(C)C)=O)C2)=O)CCn2nccc2C1 C(=O)(C1CCCc2cccnc21)NC1CN(C(c2c(N)c(C)n(C)n2)=O)C1 N1(C(C(=O)NCC(=C)C)CC2CC2(Cl)Cl)CCCCC1CN(C)C c1(-c2cn(CCCNC(c3c(C)oc(C(C)C)c3)=O)nn2)cccc(F)c1C C1(NC(C2(NC(C(C=C)OC)=O)CC(F)(F)C2)=O)CCn2nnnc2C1 C(=O)(C(F)(F)C(C)(C)O)NC1C2(CCN(C(COCCCOC)=O)C2)C1 c1(CN(C(c2nnc(C)s2)=O)C)ccc2c(c1)CCOC2 N1(C(=O)Nc2c(OCCC#C)cccc2)CCNC(=O)CC1 C1(CNC(c2n(C)nc(O)c2)=O)(CO)CC12CCN(C(=O)C(C)(C)CC#N)CC2 Cc1cn(C)nc1C(=O)NC(C)(CNC(C1(c2ccc(Cl)cc2)CC1)=O)CO C1(C(=O)NCCC(C(=O)NCC2(C)CC(O)C2)O)CC(=O)NC(=O)N1 N1(C(CCCCOC)=O)CCCC2(C1)CN(C(=O)CC(C)CF)CCO2 C1(C(N(C(CC)C(=O)N2CCC(Cn3ccnc3)C2)C)=O)CC2(CCC2=O)C1 Cc1ccc2oc(C(=O)NC3CC4C3CCN4C(=O)CCC3CC3C)c(C)c2c1 Cc1sc(S(N)(=O)=O)cc1C(N1CC(C)N(C(=O)CCS(=O)(=O)NC)CC1C)=O C1(C(=O)NC(Cn2cc(CCN(CC)CC)nn2)C)CC2(CO1)CC(F)(F)C2 C1(NC(C(CCOC)C)=O)CCC(O)CN(C(=O)Cc2ncc(C)o2)C1 C(=O)(N1OC2C=CC1CC2)C1C=CC(NC(c2ccc(C(N)=O)nc2)=O)C1 Cc1csc(C(C)C(N2CCCC2C(C)(C)NC(=O)COC(C)C)=O)n1 S(=O)(=O)(c1ccc(C(=O)NC2CC(CCNC(C3CCNC3=O)=O)C2)o1)NC C1(C(=O)NC2CC(N(C(C3CCC(CCC)CC3)=O)C)C2)CN2CCCN1CC2 C1(C)(C(=O)NCC(CNC(Cc2c(C)non2)=O)CO)CCCS1(=O)=O C1(NC(CNS(CC)(=O)=O)=O)CC2CCCC(C1)N2C(c1ccc(OC)nc1)=O C1(O)(CN(C)C)CCN(C(C2(c3nn[nH]n3)CCSCC2)=O)C1 CC1Cc2ccccc2N1C(=O)OCc1cccc(C(N2CCNC(=O)C2)=O)c1 N1(C(CC=CC=C)=O)CCCC(N(C(=O)CC2CCCOC2)CCO)C1 c1(C(=O)NC(C2CC2NC(=O)CSC)C)ccnc2cc[nH]c12.C1(C=O)(N)CCC1 c1(C(=O)NCCC(C)N(C)C(c2sccc2CC#N)=O)cncc(F)c1 N(C1CCc2c(Cl)ccc(Br)c21)C(c1ccc(C2CCC(=O)N2)cc1)=O C1(C(C)C)CCC(C(=O)NCC(C(C)(C)C)NC(=O)C2=COCCO2)C(=O)N1 c1(C(N(CC(C)NC(C2(CC)CCOC2)=O)C)=O)ccc(C(C)=O)cn1 c1(NC(C)=O)ccc(F)cc1C(N1CCC(CNS(=O)(=O)N(C)C)C1(C)C)=O N1(C(C2N(C(C(C)C)=O)CCCC2)=O)CC2COCCC2(NC(=O)C(F)F)C1 c1(CC2N(CC(F)(F)F)CCC2)nnc2n1CCOC2 C(C(=O)NC(COC)C1(C)CC1)(C1CN(C(=O)Cn2ncnn2)C1)OC C1(NC(c2c(CCC)[nH]cc2)=O)CN(C(C23CCC(CO2)C3)=O)CC1C(F)F C1(CC2CC2)CC2CC1C(O)C2O.O=C1CCSCCN1.C12CC(C1)C(=O)N2 N1(C(C2CCC(C(N)=O)C2)=O)CCN(C(=O)CC2CCOCC2)CC1CC(F)F c1(C(N2CC(C)C(NC(C3(F)CC3)=O)CC2)=O)cc(Cl)cc([N+](=O)[O-])c1O N1(C(c2ccc(OC(C)C)cc2)=O)CC(C2CN(C(C3CC(O)C(F)C3)=O)C2)C1 c1(C(N2CCC(O)(CNC(C(C)OC3CCCC3)=O)C2)=O)cc2ccccc2s1 C(=O)(C(C)(C)C(F)F)N(CCNC(C(n1ccc(C)n1)(C)C)=O)C(C)C C1(CC)(OC)CCCN(C(C2CCN(C(c3cc(C)[nH]c3C)=O)C(C)C2)=O)C1 N12CC3(CC1CO3)NC2=O.N1(C(C)(C)C)CCN(C(=O)C(Cl)(Cl)Cl)CC1 c1(C(N2C(CNC(c3ccncc3)=O)CCC2)=O)cc2ccccn2c1 c1(C(=O)NC(C(=O)NC(C2CCCC2)C#C)C)ccc(C(C)C)o1 CCN=c1[nH]c(C(=O)NC(C)(C)CNC(=O)CC2COCC(C)O2)cs1 C(=O)(C1=CC2CCC1C2)NCC(CN(C(CC(C)n1cccn1)=O)C)(C)C C1(CC(=O)NC(C(=O)NCCN(CC(F)F)C)Cn2cccn2)CC(=O)NC1=O C1(N(C(=O)C(C)=CCO)CC)CCN(C(C2(C)CCC(C)O2)=O)CC1 C1(NC(C2CCCO2)=O)CC2CC(C1)N(C(C1(O)CCCCC1)=O)C2 C(C(C)CN=c1cc(C(F)F)nc[nH]1)N(C)C(c1c(NC(C=C)=O)cccc1)=O N1(C(c2nc(CC)oc2)=O)CC2(CC(C(=O)NC3CCC(N(C)C)C3)CO2)C1 c1(C(N2C3C(CNC(CCSC)=O)CC(CC3)C2)=O)csc2cc(Cl)ccc12 C(=O)(CC(C)P(C)(C)=O)NCC(C(C)C)NC(=O)C=CBr CC(C)(C)CCCCC(=O)NC(C)(CO)C(=O)NCc1cc(C(N)=O)co1 c1(C(N2CCN(C(C(=O)NC(C)C)=O)CC2CC2CC2)=O)c[nH]c2cnccc12 N12CCN(C3CC13)Cc1cccnc1NC2=O.c1(CC)cccc(NC)c1F Cc1ccc(C(=O)NC2CC2NC(=O)C(c2ccc(Cl)nc2)(F)F)cc1N c1(C(=O)NCC2C=CCN2C(=O)COc2ccc(Cl)cn2)cccc(C2CC2)c1 C(c1ccc(F)c(OC)c1)=CC(=O)NCC(CCCC)NC(c1cc(Cl)no1)=O c1(C(=O)NC2C(CNC(c3c(C)occ3)=O)CC2)ccnc(C(F)F)c1 CC1CC(CNC(c2cc(-c3cccnc3)[nH]n2)=O)CCN1C(C1C=CCC1)=O c1(C(=O)NCCN(CCC)CC)cccnc1CNC(C1(C)COC(=O)N1)=O C(=O)(CCC(CF)CF)NCC1N(C(c2nc(COC)sc2)=O)CCCC1 c1(CN(C2CCCCCN(C(=O)CCCC(N(C)C)OC)C2)C)cn2ccsc2n1 C1(NC(CC(C)C#N)=O)CCCOC1C1CCN(C(C2(CCO)CC2)=O)CC1 N1(C(C)=O)CCCC(C(=O)NCC2CC=CCC2)C1.C12CC1CNC2=O c1(COC)cnc(OC)c(C(=O)NC2CCCN(C(=O)CC3(O)CCCC3)C2)c1 N1(C(c2c(C)nn[nH]2)=O)CC(NC(=O)C#CC(C)C)C(CC(C)(C)C)C1 c1(C(=O)NC2CCN(C(C3CC(n4cnnc4)C3)=O)C2)ccc([N+](=O)[O-])o1 N1(C(CC2CC(NC(c3nc(C)sc3C)=O)C2)=O)CCCC(O)C1C Cc1ccc(N2CCN(C(c3cc(C4(N)CCC4)on3)=O)CC2)cc1 C1(NC(c2cnc(C(C)C)s2)=O)CC2CC1N(C(C13CC(C)C1C3)=O)C2 C1(CNC(C2(O)CCC(C)CC2)=O)CC2(CO1)CN(C(=O)CC1CCSCC1)C2 C1(NC(c2cnns2)=O)CN(C(c2nccs2)=O)CC1C1CC1 CON=Cc1ccc(C(N2CCC(C)(C)C(NC(C3CCCOC3)=O)C2)=O)cc1 N1(C(c2c(C)cc(N)cn2)=O)CCC=C(C(=O)NCCCCC(F)(F)F)C1 N1(C(C(COC)C)=O)CCCCC1CNC(c1c(Cl)nsc1Cl)=O C1(C(=O)NCC(C#C)OC)CCN(C(=O)c2c(C)noc2CC)O1 c1(OCCNC(=O)NC(c2nc(C(C)O)n[nH]2)C)ccc(Br)cc1 C1(CNC(c2c(C)nc(C)[nH]2)=O)CCN(C(c2cc(Cl)ns2)=O)CCC1(F)F c1(C(N2CCC(NC(C(CC(=C)C)NC(C)=O)=O)C2C)=O)ccc(C)c(C)c1N C(CCO)(C(=O)NC1CCC(NC(=O)CCc2nc(O)n[nH]2)CC1)N(C)C C=CCC(C(=O)NC1(CNC(=O)CN2CCC2C)CCCCC1)NC(=O)OC C(CNC(=O)CC1CCC1)(CC(=O)NC1COCCCC1)OC C1(NC(C(C)=C2CCC2)=O)CCC2CN(C(C3CCc4nnnn4C3)=O)CC12 c1(OC)ccc2[nH]c(C(=O)NCC3CCN3C(=O)C(C(C)(C)C)OC)cc2c1 Cc1cnn2ccc(C(N3CC(NC(c4ncoc4C4CC4)=O)C(F)C3)=O)nc12 c1(C(=O)NCc2cccc(NC(CC(C=C)C)=O)c2)nc2cccnc2s1 C1(C)N(C(=O)OCCNC(C(CCC)O)=O)CCC1(C)C.C(C)(C)(C)O C1(OC)CC2CC(C(=O)NC(C)(C)CNC(c3cnn4c3OCC4)=O)CC12 C(=O)(C1CCOc2c(F)cccc21)N(C(C)CCNC(C1COC(=O)C1)=O)C N1(C(C=C(C)C(C)C)=O)CCOC(CCNC(=O)C2=CCSC2)C1 c1(-c2cnc(Sc3sc(C)c(C4CCC5(CC4)CC5)n3)o2)cccc(F)c1F C(C(CC(C)C)C(=O)N1CCC2(CCO2)C1)NC(CC(CC)O)=O N1(C(C(C)=C(CC)C)=O)CCN(C(C2(C)CCOCC2)=O)C(C2CCC2)C1 C1(CNC(C2CC(O)CN2C(=O)C(F)(F)Cl)=O)CCC(F)(F)CC1 C1(C(=O)NNC(=O)C(C)Sc2cccc(O)n2)(COC)CCC(=O)N1.C(C)(C)(C)O c1(CC(=O)NCCC(C(C)C)NC(c2ccc(=O)n(C)n2)=O)cc(F)cc(F)c1 C(=O)(C1=CCCOCC1)N1CC(NC(=O)CCC2CC2(F)F)C(F)CC1 C12(NC(c3ccc(F)s3)=O)CCCC1CN(C(C1C=CCC1)=O)C2 C1(C(=O)NCc2cncc(OCC)c2)CC2(CN1)CC2(F)F c1(C(C(C)C)NC2CCN(C(=O)NCC)CC2)cn2cc(Br)ccc2n1 C(C(=O)NC1COCC1NC(=O)CCc1ccc(Cl)nc1)(C(C)C)SC c1(OC)cc(NCC2OCCOC2(C)C)ccc1NC(N)=O N1(C(CC=CCC)=O)CC2(CC(NC(=O)C=CC=C(Cl)Cl)CO2)C1 c1(-c2n(-c3cn(CCOC)nc3)nc(CCOC)n2)ccc2c(c1)OCC2 C1(OC)CC(CF)N(C(=O)C(c2ccccc2)NC(=O)CN2CCOC2=O)C1 c1(C(=O)NC(CC(=O)NC(CC)CCCO)CC2CC2)ccn2cncc2c1 C1(NC(C#CCNC(C(CN(C)C)O)=O)=O)CCC12CCCC2 c1(C(N(C)CC2CCCCN2C(c2ncc(F)cn2)=O)=O)cc(O)nc(O)n1 c1(C(N2CC3(CCN3C(C3COCCOC3)=O)C2)=O)cccc2ccnn12 C(C(C)(O)C(=O)NCC#CCNC(c1cc(Cc2ccccc2)[nH]n1)=O)OC C1(C(=O)NCC#CCNC(c2ccc(O)cn2)=O)CCc2ncncc2C1 c1(C(=O)NCc2scc(-c3ccc(C#N)cc3)c2)ccc2c(c1)NCCC2 N1(C(CCC(C)(C)OC)=O)CC2CCCC2(CNC(c2ccnn(C)c2=O)=O)C1 C12(C(=O)NC(CC=C)CNC(=O)CCc3nc(=N)[nH][nH]3)CC1COC21CCC1 C1(C(=O)NCC(C)N(C(=O)Cc2cc(C3CC3)on2)C)CC12CC(C)(C)C2 CCCC(CC(C)C)C(=O)N1CC=C(CCNC(=O)CCc2ccn(C)n2)CC1 CC1CN(C(c2ccc(O)nc2)=O)CCN1C(c1cccc(N2CCCC2)c1)=O c1(C(=O)NCC2CN(C(c3cc(Cl)no3)=O)C2)ccc2c(c1)OCCO2 c1(C(N2CC(CN(C)C(c3ccsc3)=O)OCC2)=O)c(F)cccc1I c1(CC(=O)NCCC2CN(C(=O)C=CBr)CCO2)cn2ccccc2n1 CC1CCCC(C(=O)NC(C2CCOC2)CNC(=O)Cc2nc[nH]n2)C1 C1(CNC(C2CC(NC(C3CCC(C(=O)OC)C3)=O)C2)=O)CC12CCCCCC2 C1(C(=O)NC(C(=O)OCC=C)(C)C)(CC)CCN(C(=O)C(c2ccccc2)O)C1 c1(C(=O)NC(CCNC(C2C(C(C)O)C2)=O)C)ccc(Cl)c(F)c1F C(C)(CCC(=O)NC(CNC(C1CCN(C)C1=O)=O)CCO)OCC N1(C(c2cc(C)c(O)cc2)=O)CC2(C(N3CCS(=O)(=O)CC3)=O)CCC1CC2 C(=O)(C(O)C(F)(F)F)NC(C(=O)N(C(c1ccncc1)C)C)(C)C1CCC1 C(CCCC(=O)NCC1CC(NC(c2ccc(CS(C)(=O)=O)o2)=O)C1)NC(C)=O c1(CC(N2CC(C(C(=O)NC3(CCF)CC(O)C3)OC)C2)=O)nccn1C c1(C(N2CC(C(C)NC(c3ccc(COC)s3)=O)C2)=O)cnc(O)cc1OC CC12CC(C1NC(C1CC1F)=O)N(C(C1(c3ccc(F)cc3Br)CC1)=O)C2 CN1CCN(Cc2nc(C(N3CCC(O)CC3)=O)cs2)CC1 c1(C(=O)NCC=C2CCN(C(=O)C=Cc3cocn3)CC2)n[nH]c2c1COCC2 C(=O)(C(C1CCCO1)NC(C1CCC1C)=O)NCCN(C(C)C)C1CC1 c1(C(=O)NCC(C(C)C)NC(CC2(C(=C)F)CCC2)=O)ccc(C)n(C)c1=O N1(C(=O)CC2CCCC2)CCOC(Cn2cc(-c3cncnc3)nn2)C1 c1(OC)ccc(C(=O)NCCc2ccc(OC)c(C(N)=O)c2)cc1C(=O)O C1(NC(=O)Cc2cocn2)COCC1NC(c1ccn(CC(F)(F)F)n1)=O C(CC(C(=O)N(C)CCc1ccncc1)NC(=O)Cn1nccc1C)OC c1(C(N2CCC(NC(c3cc(C)sn3)=O)(CO)C2)=O)cnc(O)c(C)c1 Cc1cc2nc[nH]c(=NCC3C(C)CCCN3C(=O)C(O)C3CCC3)c2[nH]1 c1(C(CNC(c2sccc2C2CC2)=O)NC(C(COC)O)=O)ccc(F)cc1 c1ccc2c(c1)OCC2.c1(-c2ccccc2)cnccn1 C1(NC(c2ccc(C)o2)=O)CCCCC1C(=O)NC(c1ccccn1)CO c1(-c2nc(C(c3cc(C)[nH]n3)NCc3nnnn3C(C)C)on2)ccc(F)c(C)c1 N1(C(C(CC)Nc2cccnc2Cl)=O)CCCC(C2CN(C(C3(C)CC3)=O)C2)C1 C1(C(=O)NC(CNC(CCC#C)=O)C)CS(=O)(=O)CC12CC2 N1(C(C(C)(C)CO)=O)CCCC(C2CN(C(=O)CN3CCSCC3)C2)C1 C=CCN=C(NCC1(O)CCCOC1)N1CCCC(OC(C)C)C1 c1(C(=O)NC(C)C(C)NC(c2nc[nH]c2C(C)(C)C)=O)ccc2cnccc2n1 c1(C(=O)NCCC(C)N(C(=O)CC23COC(C)(C2)C3)C)cnc2nccnc2c1 C(CC(F)F)(C(=O)Nc1cccc(Cl)c1)NC(Cn1ccc(C)c1)=O C1(CN(C(=O)CCc2nc(=N)[nH][nH]2)C)CC(F)CN1C(=O)CN(C)C1CC1 C#Cc1cc(NC(ON=CC(C)C)=O)ccc1C C(=O)(C(CC)C(=O)OCC)NC(CCC)C(=O)NC1(CCF)CCC1 C1(CNC(CC=CCNC(C(C)C#N)=O)=O)Cc2nccn2C1 c1(CNC(C2C(CC)N(C(=O)C=C=C(C)C)CC2)=O)n[nH]c2c1CCC2 N1(C(C(C)(O)C2CCC2)=O)CCc2[nH]nc(CNC(C34CC5CC3C4C5)=O)c2C1 CC(C)CC(C(=O)N(CCCNC(C1CCCCC1)=O)C(C)C)NC(N)=O c1(CC)nc(C)cc(=NCCC(C)NC(C2CCC3CCCCN23)=O)[nH]1 N1(C(C(CC)NC)=O)CCN(C(N2CCC(SCC)(OC)CC2)=O)C(=O)C1 C1(NC(C=Cc2c(C)ccs2)=O)CC(F)CN(C(C2(N(C)C)CCC2)=O)C1 Cc1nn(C(C)(C)C)cc1C(=O)NCC1CC(NC(=O)C=CC2CC2)C1 C(=O)(C(C(C)O)N(C)C)NCC1C=CC(NC(c2cnn(CC)n2)=O)C1 C1(CNC(=O)NCc2cc(C)sc2)CCN2CCCC2C1 C(C(=O)N(CCN1CCCCCC1)C(C)C)(C(=O)NC)OCC c1(CN(C(=O)CCc2cnn(C)c2)C)ccc(CNC(=O)CC2CC3CC3C2)cc1 C1(O)(CN(C)C(C2CCC(OC)CC2)=O)CCN(C(=O)CN2CCC(C)(O)C2)C1 c1(C(=O)NCCC(=O)OCC2C(CC)C2(F)F)cc(Cl)cn1C C1(NC(c2c(C)cc(C)s2)=O)CCN(C(=O)C(C)(C)N2CCOCC2)CC1F C1(NC(c2ccc(SC)cc2)=O)CC2CCC(C1)C2NC(c1ccc(C)n1C)=O Cc1cc2ncn(CC(=O)NCC(F)CNC(=O)C(F)(F)C(F)(F)F)c2cc1C C(CC1=CCN(C(c2ncsc2C2CC2)=O)CC1)NC(Cc1cc(CC)no1)=O C1(NC(CC)=O)C2CCN(C(=O)Cc3csc4sc(C)cc34)CCC12 c1(C(N2CCC3(C(NC(CC4(CSC)CC4)=O)C3)C2)=O)ccc2cnnn2c1 C1(NC(CCc2cnc(C)o2)=O)CCN(C(=O)C=Cc2ccccc2)C1C Cc1noc(C)c1COCC(=O)NC(C)(C)CN(C(=O)CC1CCCS1(=O)=O)C c1(C(=O)NCC(C)NC(=O)C(c2ccc(F)cc2)(C)O)ccc(O)nc1Cl c1(C(=O)NC(C)C(C)NC(=O)CCCn2ccnn2)ccc([N+](=O)[O-])[nH]1 c1(C(N(C2CCN(C(c3cnc[nH]c3=N)=O)CC2)CC#C)=O)nc(C)oc1C C(=O)(C(C)(C)n1cc(Br)cn1)NCCCOCCNC(CC1CN(C)C1)=O C1(C(=O)NCC2N(C(CCOCC)=O)CCCC2)CCC(C#N)CC1 O=C(C1=C(Cl)CCC1)NC12CC(C(N3CCC(c4ncc[nH]4)C3)=O)(C1)C2 C1(NC(=O)C(c2ccccc2)F)CC2CC1CN2C(=O)Cc1ccc(F)cc1F c1(C(=O)NCCC(C(=O)NCC(n2ccnn2)C)OC)cc(O)ncc1F N1(CCCN(C(c2ccccc2)(C)C)C)CCC=C(Cl)C1 C(N=c1[nH]c(=NCCCc2ncc[nH]2)c2ncccc2[nH]1)c1ccc(COC)s1 C1(NC(CCC(C)OC)=O)CN(C(=O)C#CC2CC2)C2(CCOCC2)C1 c1(CC)nn(C)c(C(N2C3CCC2C(C(=O)Nc2ncc(COC)s2)C3)=O)c1Cl C1(C(=O)NCC2CC(NC(C3(C)CCC(C)C3)=O)C2)CCC2C(C1)C2(F)F CC(CN(C(=O)C=Cc1cccnc1)C)C(=O)NOCC(F)(F)F C(=O)(CCC(=O)NC1(C)COCCO1)NCC1N(C(CN(C2CC2)CC)=O)CC1 N1(C(=O)Cc2ccc(Cl)s2)CCOC(CNC(C23CCC(CO2)C3)=O)C1 C(=O)(C1=CC(O)C(NC(=O)Cn2ccnn2)C1)Nc1ccc(C(C)F)cc1 C1(C(=O)NCCC(=C)CNC(=O)C(C)(C)C(C)C)CC2CCCCN2C1 C1(CNC(C(CN(CC)CC)F)=O)CC2(CCC2)CN1C(c1cc(Br)c[nH]1)=O C1(C(N2CC(n3cc(CCCCC)nn3)C(C)C2)=O)Cc2ccncc2N1 c1(OC)ccc(Cl)cc1C(=O)NCC1CCCC1NC(c1nccs1)=O Cc1ccc2nc(C)cc(C(=O)NCC(C)N(C(=O)Cc3cn[nH]c3)C)c2c1 C1(C(N(CCCCCC)C(=O)C(N2CCNC(=O)C2)C)=O)COc2ccccc2O1 N1(C(C2CN(C)C2)=O)CCC(NC(C2CC(C3CC3)=NO2)=O)C1(C)C C1(NC(CC2C=CC(NC(c3c(CC)cc[nH]3)=O)C2)=O)C(C)CCC1C C=CCC(C)C(=O)N1CC2C(CNC(c3nnsc3C(F)F)=O)C2C1 c1(C(N2CCCC(N(C(=O)C3=C(Cl)CC3)CC)C2)=O)cnn2ccnc(N)c12 c1(C(N2C(CN(C(C3C(C)OCCO3)=O)C)CCC2)=O)ccc(F)c(Cl)c1 C1(NC(CSSC)=O)CC2CCCC(C1)N2C(c1ccnn1C)=O CCCCC(O)CC(=O)NC1(CO)CCN(C(c2cn(C(F)F)c(C)n2)=O)C1 C1(NC(C2C(C(C)(C)C)CC2)=O)CCCN(c2ccccc2)C1 c1(-c2nc(C(C)OC(c3[nH]cc(C(C)=O)c3)=O)sc2)ccc(F)cc1F c1(C(=O)NCC2C(CCC)CCCC2)nc2ccncc2[nH]1 CCCCCCCCCCCC(O)C(=O)N1CC(C2CN(C(=O)C(C)CC)C2)C1 c1(NC(C2CC2C(=O)NCc2nccnc2Cl)=O)ccc2[nH]ccc2c1 Cc1oc(C(=O)NC2C3CCN(C(=O)C=Cc4cnc[nH]4)C23)cc1Br c1(C(=O)NC(C(=O)NC2N(CCOC)CC2)COC(C)C)cnn2ccccc12 c1(C(=O)NCCN(C(c2c[nH]c(=NC)s2)=O)C)csc2nnsc12 N1(C(C2(C)CCCS2(=O)=O)=O)CCC2(CCC2NC(c2cncc(F)c2)=O)CC1 C1(C(N2CC(NC(CCNC(=O)OC)=O)C3(C2)CC3)=O)COC2CCCCC12 c1(C(=O)NC(C)CCC(=O)N2CCC(NC(=O)C3CC3)C2)cncc(C#N)c1 c1(C(N(C(CCNC(CCc2ccc(C)o2)=O)C)C)=O)cncc(P(C)(C)=O)c1 CC1CCOC(C(=O)NC(CN(C)C)CC(=O)N2CCCC(CCF)C2)C1 Cc1nn(C)c(C)c1C(=O)NC1CC(C(=O)Nc2ccc(Cl)c(F)c2)C1 N1(C(C(F)OC)=O)CCC(C2(CNC(c3nc(C)sc3C)=O)CCOCC2)CC1 c1(C(=O)NCC(CC(C)C)NC(C2CCCS2)=O)[nH]nc([N+](=O)[O-])c1Cl S(=O)(=O)(c1cc([N+](=O)[O-])ccc1C#N)Nc1onc(CCC(CC(=O)OC)C)n1 C12(C(=O)NC(C)CNC(c3ccccc3-c3cn[nH]c3)=O)COC(CCO1)C2 N1(C(C(COC(C)=O)C)=O)CC2CC(NC(=O)C(C)Cc3ccncc3)CC2C1 Cc1nocc1CC(=O)NC(C1CN(C(=O)CCN(C)CCO)C1)C N#Cc1cccc(C(O)C(=O)N2CCC2C(=O)NCC2CC3CC2CC3O)c1 c1(C(N2CCCC(CNC(=O)CC3CCCCO3)CC2)=O)ccc(Br)c(Cl)c1F c1(OC)ccc(Cl)c(C)c1C(=O)NC(CNC(c1cc(Cl)no1)=O)CO Cc1cccn2cc(C(=O)NC3CCC(NC(C4C(C)C4C)=O)CC3)cc12 C(C(=O)NCC1CCCCN1C(c1cnns1)=O)(C(C)C)SCC Cc1nc2ncccc2cc1C(=O)NC1(C)CC(NC(=O)C(C(C)O)N(C)C)C1 C1(C(=O)NCC(C)OCCO)CCC(O)CN1C(c1ccc(C#N)o1)=O CC1(C)CCCC1NC(N1CC(CC(F)(F)F)C1)=O N1(C(CCC(=C)Br)=O)CC(C)CN(C(=O)Cn2ccnn2)CC1C c1(NC2C(C)(CC)C2)ncc(C)cc1S(=O)(=O)N(C)CCOCCOC C(=O)(CC(O)CNC(=O)COC(C)C)NC(C1CCOC1)C#C C12(C(N3CC(C)N(C(C4CC(N(C)C)C4)=O)CC3)=O)CC3CC(C(=O)N1)C2C3 C1(C(=O)NCC(COC)O)CC12CN(C(=O)Cc1ccccc1SC)C2 C1(C(=O)NCc2ccnc(CO)c2)CC(F)(F)CN1C(C12CC(F)(C1)C2)=O Cc1cc(NC(c2ccnn2-c2ccccc2)=O)ccc1NC(C1CC(O)C1)=O C12(NC(c3cncc(C)c3)=O)CC(C)(C1)OC21CCN(C(=O)CCS(C)=O)CC1 CC1(C)C(N(C(=O)CN2CCCC2=O)Cc2cnc(O)nc2)C2CCOC12 N1(C(Cc2c(C)nc[nH]2)=O)CCC(CNC(=O)C(=Cc2cnn(C)c2)C#N)CC1 C(C1CCc2ncnn21)N1CCCC(CCNC(C(C)N2CCC2)=O)C1 Cc1ccc(Br)c(C(N2CCOC(C3CN(C(C4CCN(C)C4)=O)C3)C2)=O)c1 N1(C(C2CC(CNC(C(=Cc3ccccc3)C)=O)C2)=O)CCC12CCCOCC2 C=CCC(C)(C)CC(=O)NC(CC(F)F)C(=O)Nc1ccc2c[nH]nc2c1 Cc1nccc(Cl)c1NC(=O)COc1cc(Cl)ncc1Br C1(NC(Cc2nnc(C)s2)=O)CN(C(c2cccnc2C(F)(F)F)=O)CC1C N1(C(C2=C(C)OCC2)=O)CC(C)(C)OC2(C1)CN(C(=O)CCCC#N)C2 c1(C(N)=O)cc(C(=O)NCC2CC(NC(=O)CCN3CCC3)C2)c[nH]1 C1(F)(CNC(c2ccc(CN(C)C)o2)=O)CCN(C)C1 c1(C(=O)OCC)cnc(SC)nc1N1CCC(NC(c2occc2C)=O)C(F)C1 c1(CN2CC(CN)C(CC(=O)O)C2)c(-c2ccccc2)nc2ncccn12 C1(COC)CN(c2nnc3n2C3)CCO1.C1(O)(SC(C)C)CCCCC1 N1(C(=O)NCc2c(-n3cccc3)ccc(C)c2)CCC2(CCC(O)C2)C1 C1(C(=O)NC(C(O)CO)C2CC2)(CC)CCN(C(=O)CN=[N+]=[N-])CC1 Cc1cc(C(=O)NCC2CCN(C(=O)CC3(O)CCCOC3)CC2)nc(O)c1 c12nc(Cl)ccc1C(=O)NC1C(CC1)CN2.C1(C(=O)NC)(C(=O)OC)CCOCC1 C12(CCNC(C3CN(C(=O)CCc4ccon4)CCO3)=O)CCC(CC1)OC2 N1(C(C(CC)OC)=O)CCN(C(c2cc3nc(Cl)ccc3o2)=O)C2COCC12 C(=O)(CCCC(F)(F)Br)N1CC(CCOC)N(C(C2CC2C)=O)CC1 Cc1nn(C)c(Cl)c1C(=O)NC(CNC(=O)CN1CCCCCC1)C1CC1 c1(C(N2CCN(C(COCC)=O)CC2C)=O)ccnc2ccsc12 C(C(C(C)C(C)C)NC(=O)CCc1ccc(C)cc1)NC(CN(CCC)C)=O N1(C(C(CC)C)=O)CCC(CC)(NC(c2cc(Br)n[nH]2)=O)CC1 N1(C(CSCC)=O)CCN(C(=O)C(C)CN(C)Cc2ccccc2)CC1C(C)C C(=O)(C1=COCCC1)NC1C(CNC(C(C)n2ccnc2)=O)CCC1 c1(C(N2C(C)C(NC(C3(Cl)CC3)=O)CCC2)=O)cnn2cc[nH]c(=O)c12 C1(=CC(=O)NCCOC(C(=O)N(C)CC)C2C(C)C2)CCN(C)C1.C(C)(C)(C)OC=O C1(NC(c2c(C)noc2C(F)(F)F)=O)CC2CC1N(C(c1cncn1C)=O)C2 c1(C(=O)NCCC(C)NC(C(CC)=CC)=O)c[nH]n(CC=O)c1=N.C(C)(C)OCC CC1(C(=O)NCC(CC(F)(F)F)NC(c2cnc(O)s2)=O)CCCC1(F)F N1(C(CCC(C)C)=O)CCC(F)(C(N2CCCC2CCO)=O)CC1 N1(C(=O)COC(F)F)CCC(NC(C23CC4CC2C3C4O)=O)C(CO)CC1 C1(C(N2C(CNC(C(C(C)O)N(C)C)=O)CCC2)=O)CC(c2ccccn2)=NO1 c1(C(N2CCCC(F)(CNC(C(C)OCCCC)=O)C2)=O)ccc2nc[nH]c2c1 C12(C(=O)NC(c3nc[nH]n3)CC)CCC(O)(CC1)CC2 CC1CCCC(C)N(C(=O)C(C2(O)CN(C(=O)C3=COCC3)C2)F)C1 c1(CC)cc(OC)cc(C(=O)NC2CC2NC(c2ccc(C)o2)=O)c1 N1(C(C(CC(C)C)F)=O)CC2CCN(C(c3ccc([N+](=O)[O-])[nH]3)=O)CC12 c1(OC)ccc(CN2CCC(C(N3CCOCC3CC(C)C)=O)C2)cn1 CC1CN(C(=O)COCC(F)F)CCN1C(c1cnc(O)s1)=O c1(C(=O)NC2CN(C(C3(C(=O)NC)CCC3)=O)C(C)C2)cccn2c(C)nnc12 CN1C(=O)NCC1C(=O)NCC1CCC(NC(=O)COCC2CCOCC2)C1 N1(C(C(C)C#N)=O)CCN(C2CCCN(C(c3cccnc3C3CC3)=O)C2)CC1 N1(C(C2COC2)=O)CC(C(N2CCCC2CC2CC2)=O)C2(CCC2)C1 C(=O)(C(F)C(F)(F)F)N1CC(C(C)NC(=O)CC#N)OCC1 c1(C(N(C2CCN(C(=O)C=Cc3cncs3)CC2)C)=O)cc(O)cc(F)c1 CC1CC(C(=O)NC(C2(O)CN(C(=O)CC3CCCOC3)C2)C)CC(C)C1 C=C(C)CCC(=O)N1CCC(NC(=O)CCOc2ccccc2)C1c1cccs1 N1(C(Cc2cccc(C)c2Cl)=O)CC2CCCC2(NC(c2cnn(C)c2C)=O)C1 C#CC(C)(C)C(=O)N(CC(C)N(C(=O)CC=C(Cl)Cl)C)C C(=O)(CC1=CCOCC1)N1C(C(=O)NCc2n(CC)nnc2C)CC(O)C1 C(=O)(C1=CNC2=NCCC2=C1)N1C(C)C(NC(=O)C(O)Cc2ccccc2)CC1 CC1CN(C(C23CCC(C)(C2)OC3)=O)CC(C)C1NC(=O)COCCN(C)C CCC(C)C(C)C(=O)NCCCC1(NC(c2cnn(CCC#N)c2)=O)CC1 N1(C(C)=O)CCc2sccc2C1C(=O)NCC(CNC(=O)OC(C)(C)C)N(C)C c1(N(C)C(=O)CCF)cccc(N)n1.C12(C(=O)NC(c3ccccc3)C)C3C4C5C3C1C5C24.N C1(C(=O)NCC2CCN(C(CCC3CCC(C)O3)=O)CC2)COCCC1(F)F c1(C(=O)NC23CCCN(C(CCCCOC)=O)CC2C3)ccc(F)c2occc12 C12(C(N(CC(C)NC(=O)C=Cc3cncn3C)C)=O)CC(CO)(C1)OC21COC1 N1(C(COCC=C)=O)CCN(C(=O)C(C)C)CC1CCOC c1(C(=O)NCC(=C)C(=O)OC)c(C)cnn1C C1(C(=O)NC(CNc2nccc(C(C)(C)C)n2)C2CC2)CCc2ccccc2O1 c1(CNC2CCC(C(=O)NCc3nnc(C)o3)C2)cc([N+](=O)[O-])cc(O)c1O c1(C(C)C)ccc(C#N)c(N2CCC(C[N+](C(c3ccno3)=O)([O-])N(C)C)CC2)n1 C(C(C)(O)C(=O)NCC(C)NC(=O)CCCOCc1ccccc1)OC N1(C(C(CCC)O)=O)CC2(C=C(C(=O)NC3(CO)CCC4(CC3)CC4)CO2)C1 C1(C)(NC(=NCc2c(OC)cccc2)NC2CSC2(C)C)CCC2(CC1)CC2 C(=O)(C(O)CC(=O)OC(C)(C)C)NCCCCN(C(c1c(CC)nc[nH]1)=O)C C(=O)(C(C)CC(C)C)N(c1nccc(C)n1)C(C)CC(C)(C)C c1(C(N(CC(C)NC(=O)CCSC)CC)=O)oc(CO)cc1C C1(C)(NC(=O)NCc2cnc(-c3c(OC)cccc3)s2)CC2CCC1C2 C1(C)(OCCC(=O)NC(C2CCN(C(C3(CO)CC3)=O)C2)C)CCCC1 c1(-c2nc(C(C3CC3)OC)nn2C2CCCC2(C)C)cc2nccnc2cc1F CC1CN(C(=O)CN2CCC2)CC1NC(=O)C(C)(O)Cc1ccccc1 c1(C(=O)Nc2ccc(C(N3CCCC(CO)C3)=O)c(Cl)c2)cc(O)nc(Cl)c1 C#CC1CCCN(C(=O)CCCN(C(=O)COc2cccnc2)C(=O)C2CC2)C1 Cc1cccc2oc(C(=O)NC3CNCC(O)C3)cc12.C1(C(=O)N)C2CC3C(C2)C13 c1(C(N2CC(C)(NC(=O)COCC(F)(F)F)C2)=O)c(Br)ccc(F)c1F c1(C(=O)NC2(C)CN(C(CC3(C(=C)F)CCC3)=O)C2)cc(C)nc(C(F)(F)F)n1 N1(C(=O)NC2N(C(c3c(C)c[nH]c3)=O)CCC2O)CC(O)C(O)C1CO C1(NC(C(CC)SC)=O)CN(C(=O)CCCC(=O)OC(C)(C)C)CC1(C)C C1(CNC(CNc2ccc(OC)cc2)=O)CCCN(C(=O)CCC=C(C)C)CC1 C1(CCNC(c2ccoc2C2CC2)=O)CCCN(C(C2CCSC2)=O)C1 N1(C(c2c(NCC)scn2)=O)CCN(CCNC(C2(C(C)C)CCC2)=O)CC1 c1(C(=O)NCCC(C)NC(=O)CNC(=O)CNC(N)=O)n[nH]c(CC(C)C)n1 c1(NC(C)=O)cccc(NC(=O)CC2(C)CN(Cc3cncc(C)n3)C2)n1 C1(CC(=O)CC2(C(=O)NCc3cccc(C)c3)CC2)COc2ccccc2O1 C1(C2CC2)(NC(COC(CC)(C)C)=O)CCN(C(=O)C(C(C)(C)C)NC=O)C1 c1(NC(C2CCC(N(c3nccs3)C(CC)=O)CC2)=O)cc(=O)n(C)c(O)n1 c1(OC)ccc(CCC(=O)NC2COCC2CNC(=O)C(F)=CC2CC2)cc1C n1(CC)nc(C)c(C(N2CC(O)(C3CCCN3C(=O)CC3CC(=O)C3)C2)=O)c1C c1(C(C)C(=O)NC(C)COCc2cccc(F)c2)cc2ccccc2o1 C1(C)(COC)C=CCCN1C(=O)N(CC(=O)Nc1ccc(I)cc1)CC c1(CC)[nH]nc(C(N2CCC(C(=O)NC3CN(C)CC3C)C2)=O)c1C CCCCCCCCC(F)C(=O)N1CC(O)(CCNC(c2coc(CO)c2)=O)C1 Cc1nc(NCC2(CNC(=O)CN(C3CCCC3)C)CCCC2)c(C)c(O)n1 N1(C(CC)=O)CC(F)CC1CNC(C1CC(C(=O)OC)C1)=O CN1CCC(C)(C(=O)NCC2CC(C(=O)NC3(C4CCC4)CC3)=NO2)CC1 c1(OC)ccc(Cl)c(C(=O)NC2CC(C)(NC(C3CCCC(C)CC3)=O)C2)c1N Cc1cc(C)n(C(C)C(=O)N(C2CC(NC(c3n[nH]cc3Cl)=O)C2)C)n1 CC(C)C(CO)CCNC(=O)NC1CCOCC1C(F)(F)F c1(OC)cnc(N2CCCC(NC(c3c[nH]cc3C)=O)C2)nc1 N1(C(C2CCCCCO2)=O)CCC2(CCN(Cc3cc(Cl)cnc3Br)C2)C1 CC(C)CC(C(=O)NCC(C)N1CCC1)C(N)=O.C12(CSC1)C(=O)N2 C1(CCCC)CCCN1C(=O)C(C)N(C(c1ccnn1CC)=O)C1CC1 C(c1cncnc1O)=CC(=O)NCC(O)CCNC(c1cnoc1C1CC1)=O c1(OC)ccc(CNC(=O)C(=O)NC2C3CC2N(C(=O)CS(C)(=O)=O)C3)cc1 C1(C(N(CC(C)NC(=O)CCCc2ccncc2)CC)=O)CC(=O)N(CC)C1 CC(C)CC(C)CC(C)C(=O)Nc1nc2cc(Br)ccc2n1CC(=O)O C=CCCCCC(=O)N1CCN(C(c2cccn(CC)c2=O)=O)CC1C CCC1=C(C(=O)NCC2CCCC2NC(C2CCN(C3CC3)CC2)=O)SCCO1 C(=O)(C(C)(O)C(C)C)N(C1CCCSC1)CC(N1CCN(C(CC)=O)CC1)=O C(=O)(CCCS(C)(=O)=O)N1C(CNC(C(C2CCC2)OCC)=O)C(C)(C)CC1 C=CCCCCC(=O)N1CCC(C(N2CC(CS(C)=O)C2)=O)C1CC C1(C)(CNC(C2(CCC)CC2)=O)COCCN(C(=O)C=CC2COC(C)(C)O2)C1 C=CC(C)(O)C(=O)NC1CCC1NC(=O)Cc1nnn(-c2nccs2)c1C CC(C)CC(C)CC(=O)NC(CNC(=O)COCc1ccccc1)CC(C)C N1(C(C(C(=C)Cl)(C)C)=O)CCCC2(NC(=O)CCc3csc(C)n3)CC2C1 c1(C(N2CC(CNC(CC(=C)Br)=O)C3(C2)CC3)=O)c(C)ccc(F)c1O O(N1CCC(CC(=O)NC(C)CCNC(C2(C3CCCO3)CC2)=O)CC1)CC N1(C(C(CC)C)=O)CCC2C(NC(c3cnn(Cc4cccc(F)c4)c3)=O)C12 C1(NC(C2(CNC(C3C(OC(C)=O)C3)=O)CC3(CC3)C2)=O)CCN(OC)CC1 N1(C(C2CCCCC23CCC3)C(=O)NCCC#N)CCOc2cccc(Br)c2C1 c1(C(=O)NCC(C(C)C)NC(C2CSCCS2)=O)cc(C(F)(F)F)ncc1Cl C(=O)(N=c1ccn(C2CC2)[nH]1)O.c1(C2CN(C(=O)OC(C)(C)C)C2)ncncc1F CCC(CC(=O)N(C(C)C(=O)N(C1CN(C)C1)C)C)C1CC1 N1(C(CC2CC(OC)C2(C)C)=O)CC(C)OC2(CCN(C(=O)CS(N)(=O)=O)C2)C1 Cc1ccc(C)c(C(=O)NCCCNC(c2nsnc2O)=O)c1 C=C(Cl)C(C)(C)C(=O)NCC(C1CCOC1)NC(c1cc[nH]c1C1CC1)=O CCCC(C(O)C(=O)NCc1ncn(C(C)C)n1)NC(C1CCC(O)CC1)=O n1(CC(C)C)cc(CCCNC(=O)CN(C(=O)OC(C)(C)C)C2CC2)nn1 N1(C(c2c(OCC=C)c(C)ccc2)=O)CCCC2C1CCN2C(c1cnn[nH]1)=O C1(NC(CNS(NC)(=O)=O)=O)CCC2(CCN(C(C3CCO3)=O)CC2)C1 CCC(CC(=O)NOCCCC1CC1)NC(=O)CC(CC)SC C=CC1(C(N2CCCC(NC(C3CCC3CF)=O)CC2)=O)CCCCC1 CN1CCN(C(c2ncoc2C2CC2)=O)CC1CNC(=O)C#CC1(CO)CC1 N1(C(CCCNC(=O)OC)=O)CCC(O)C1C(=O)NCCn1cnccc1=O Cc1cc(=N)[nH]cc1C(N1CC2(CNC(C3(CCF)CCC3)=O)CCC1C2)=O Cc1c(CC(=O)NC2CC(NC(=O)C(C)(C)F)CC2O)sc2ccccc12 C(C(CC(C)C)C(=O)N1CCC(CO)C(NC(c2cnc[nH]2)=O)C1)OC CC1CN(C(C2CC2c2ccccc2)=O)CC1CNC(C1CCCSS1)=O CC(C)(CC(F)F)C(=O)NC1CC=C(C(=O)N2CCNC(=O)CC2)C1 C(=O)(C1CCCc2nccn21)N1CC(N(C(c2ccc(C)s2)=O)C)C2(C1)CC2 c1(C(N(C(CNC(=O)CN(S(C)(=O)=O)C)C2CC2)C)=O)cc(F)cc(F)c1 N1(C(C2C(CC)(COC)C2)=O)CCC(CO)(CNC(C2(SC)CC2)=O)CC1 CC1(C)CC(NC(c2cnc(C(F)F)[nH]2)=O)CN(C(c2ncccc2CO)=O)C1 C#CCCCC(C)C(=O)NCC1CC1NC(=O)Cc1cncc(OC)c1 C1(NC(=O)Cc2cnc[nH]2)CCC(F)(CNC(C2CC(=O)N(CC3CC3)C2)=O)C1 N1(C(Cc2c(C)nn(C)c2)=O)CCC2(CC1)CC(NC(c1ccsc1)=O)CO2 C(=O)(CC(O)CC(C)(C)C)NCC12OCC(NC(CC(C(N)=O)NC(C)=O)=O)(C1)C2 c1(C(c2cccs2)NC(C2CCC(C(C)(C)C)CC2)=O)ccc(F)cc1F C1(CC(C)(C)CC(C)(C)C)C(=O)N2CCCNC(=O)CC(C)C(CC)CCC12 C#Cc1ccc(F)nc1NC(=O)NCCc1ccc(OC)c(CC)c1 N1(C(c2nncn2C)C)CCn2ccnc2C1C(=O)O CCC(CC)C(c1nnnn1CC1CC1)NCC1(C)CSC1 C1(C(C)NC(=O)CNc2ccccc2)CCCCN1C(c1cccc(Cl)n1)=O C(=O)(C(C)(C)C(F)F)NCC1CN(C(C=CC)=O)C(C)C1 C1(NC(CSC)=O)CCC2(CCN(C(=O)CCOc3ccccc3F)C2)C1 C1(N(C(c2nc(CC)oc2)=O)C)CCN(C(c2ncncc2Cl)=O)CC1 c1(CC2CN(C(CNC(=O)CCC3CCCC3)=O)C2)ccc2n[nH]cc2c1 N1(C(CN2C(C)CC2)=O)CCCC12CCN(C(c1cnc(S)[nH]1)=O)C2 N1(C(C(C)n2ccnc2)=O)CC(C)(C)CC1CNC(=O)CSC(F)(F)F N1(CC)CCOCC1C(=O)NCC(C)(C)NC(c1ncccc1OC(F)F)=O C(=O)(C(CC(C)C)n1ccnc1)N1CC(OC)C(NC(=O)CCCSC)C1 c1(C(N2C3CCC(CCNC(c4c(C)c[nH]c4)=O)(C3)C2)=O)nn(C)c2c1CCC2 C=CCC(C)(C)CCNC(=O)C(CO)NC(C1CCC(NC(C)=O)CC1)=O C1(C(N2CC(CN(C)C(c3ccnc(CO)c3)=O)OCC2)=O)Cc2nccn2C1 N1(NC(C2C3(CN(C(C4CN(C)C4)=O)C3)C2)=O)CCN(S(=O)(=O)N(C)C)CC1 Cc1cc(CCC(=O)NC(C)CCCNC(=O)C(C(C)C)NC=O)ccc1Cl c1(CC)ncc(C(=O)NCC(O)CNC(=O)CCCSC(C)(C)C)c(C)n1 C1(C(C(=O)NCC2(O)CN(C(C(C3CCOC3)OC)=O)C2)C)CCC(C)(O)CC1 c1(C(N(C2CN(C(C3(F)CC3)=O)CC2(C)C)C)=O)cc2n(c1)CCOC2 N1(C(c2nc(C)n(C)c2)=O)CC(N=[N+]=[N-])CC1C(N1CCC1C)=O c1(C(=O)OCc2ncc(-c3ccccc3Br)o2)cc2cccnn2c1 c1(CC)cc(NC(=O)NC(c2ccncn2)C)c(C)cc1F C(=O)(C(C1CC1)N(C)C)NCCN(C(=O)C(=O)NCC(F)(F)F)CC c1(CNCc2ccc(-c3ccc(C(C)(F)F)cc3)nc2)cccc(F)c1[N+](=O)[O-] C(CC(CC)C(=O)N1CCCCC(CNc2c(Cl)c(C(=O)O)nn2C)C1)=CC Clc1csc(C(F)(F)F)n1.n12nnnc1C2 C(=O)(C1=CC2(CCN(C(c3cccc(C)c3F)=O)C2)C1)N1CC2C(OC)CC(C2)C1 C1(Cc2cn(CCC=C)nn2)CCCCN1C(c1cnc(Cl)[nH]1)=O C(C(C)N=c1[nH]c(N2CC(n3cnnc3)C2)nc2ccsc12)c1c(C)ncs1 C1(CCOC)(NC(=O)CCC2OCCO2)CCN(C(c2c[nH]cc2Br)=O)C1 c1(C(=O)NC2CCC(Cn3cc(COC)nn3)C2)ncccc1C(F)F c1(NC(C(=O)NCCC(C)(C)C[N+]([O-])=O)=O)ccc2c(c1)ncn2C1CCCC1 c1(CC)c[nH]nc1CNC(=O)NC(C(C)(C)C)c1ccc(C)o1 c1(C(N2CC(N(C(c3c(C)cc(O)cc3)=O)C)C2)=O)c(C)oc2cc(O)ccc12 c1(S)ccccc1.C1(C#N)(C(=O)NCCCN(C(C(C)SCC)=O)CCO)CC1 Cc1ccc(C)c(SCC(=O)NCC2CN(C)CCN2C(=O)COC(C)C)c1 C=C(C)CCCC(=O)NCC12CC1CN(C(=O)C(C(C)C)n1cccn1)C2 n1(CC(=O)NCC2N(C(C(F)=C(C)C)=O)CCC2C)cc(C(N)=O)c(O)nc1=O O=C(CCCCC(F)(F)F)NC1(C2CCCN(C(c3ncc[nH]3)=O)C2)CC1 n1(CC)cc(Cl)cc1C(=O)NCC1(NC(=O)Cc2cc(C)ns2)CCCC1 C(C(C(=O)N1CC(OC)C1)C(C)C)NC(c1c(CC)nccc1)=O c1(OC)cc(CNC(C)CN2CCOC2=O)c(OC)c(C)c1[N+](=O)[O-] c1(C(=O)NC2CN(C(C3CCCS3)=O)C3(CCC3)C2)cccc2c1CNC2=O C1(C(N2CCCC2)=O)CCN(C(N)=O)CC1.C1(=O)C=CC(=O)N(C)CCCN1C C1(CCOC)CN(C(C2CCCCC2C)=O)CCN1C(=O)CCC1CCOCC1 C(=O)(CC(CC)CC(C)C)N(C(C(N1CCC(C#C)(O)C1)=O)C)CCC C1(NC(C(CC)F)=O)CC2CC(NC(c3cc4ccccc4o3)=O)CC2C1 Cc1cncc(CNC(=O)CN2CCN(C(=O)OCC(C)(C)C)CC2)c1 C1(NC(C2CCCN(C(CCN(C)C)=O)C2)=O)CCOCC1(C)C O=C1COc2cc(C(N3CCC(F)(F)C(F)(F)CC3)=O)c(Br)cc2N1 c1(Cc2n(CC)ccn2)nnc(N2CCOC(CC)C2)n1CC(C)C C1(NC(C(C)C2CCC2)=O)CCCCC12CCN(C(C1CCC(=O)C(C)C1)=O)C2 C1(CNC(C)=O)CCCCN1C=O.C1CCCN1C(c1cnc(C)[nH]1)=O N1(C(C(COC)C)=O)CC(CNC(=O)C=Cc2ccnn2C)C2(CCOCC2)C1 C1(N(C(C2C(NC(CC3CC(CSC)C3)=O)CC2)=O)C2CC2)CCCC(C)(C)C1 CCC(CC)C(C)C(=O)N1CCNCC1.C(=O)(C(C)(C)CC(C)C)N1CC2C(N)C2C1 C(CCCCCCCO)NC(C1N(C(C2N(C)CCC2)=O)C2C(C1)C2)=O C1(N(C(=O)Cn2cc(C3CCOC3)cn2)C(=O)C2CC2)CCOC12CCCC2 N1(C(C(F)=CCC)=O)CCC(C)C(CNC(C2CC2c2ccoc2C)=O)C1 O=C1NCC2CN(C(=O)COC3CCC(F)(F)CC3)CCC2N1 C1(CC(=O)NC2(CNC(c3c(O)cccc3F)=O)CCC2)CCCCC1(F)F CC1CCOCC1C(=O)NCc1ccnc(C(=O)N(C)Cc2ccccc2F)c1 CC#CC1CCN(C(=O)C(F)C2CC(NC(=O)C(COC(C)=O)OC)C2)C1 c1(C(=O)NCC(CC)NC(CCCC=C)=O)ccc2cnccc2n1 c1(COC2CCN(C(C3CN(C(CC)C)C(=O)C3)=O)C2)ccc(O)c(OC)c1 N1(C(Cc2ccc(SC)cc2)=O)CCC(NC(=O)COCCF)CC1C N1(C(=O)C2=COCCO2)CC2(CCCN(C(c3cc(F)c(F)cc3O)=O)C2)C1 N1(C(C2(OC)CCCC2)=O)CCCCC(N(C)C(C2OCCOC2C)=O)C1 c1(OC)cc(Cl)c(S(=O)(=O)N2CCCCC2P(C)(C)=O)cc1Cl CC1(C)CC(CC(N2CCC(OCCO)C2)=O)N(C(C2CCCOC2)=O)C1 CC1CC(NC(=O)CCC(C)(C)F)CCN1C(c1nn(C)c(Cl)c1Cl)=O c1(C(N2CCN(C(C3(F)CCCC=C3F)=O)CC2)=O)[nH]nc2ccncc12 N1(C(C(=O)NC)=O)CCc2ccc(NCC3CCCN(CC)C3)cc2C1 c1(CC)cc(Cl)ccc1C(=O)NCC(C)N(C)C(C1(C)CCOC1)=O C(=O)(C(F)(F)C(C)O)NCCC1CCC(NC(c2cccc(OC)c2)=O)C1 C1(CC(=O)NCC)CN(C(=O)CCOCCN(C(=O)CC2CSC2)C)C1 C(=O)(CCCC(F)(F)C(F)(F)F)NCC1(OC)CCN(C(=O)C=CSC)CC1 c1(C(N2CCC(C(=O)Nc3cccc(C#N)c3)C2(C)C)=O)cc2scc(Cl)c2[nH]1 C1(NC(c2cc(C(C)=O)oc2)=O)CCC12CCN(C(=O)C(C)=CC(C)(C)C)CC2 C1(C)(CNC(c2ccc(CC)cn2)=O)CN(C(c2coc(Cl)n2)=O)CC1C C1(NC(=O)C=CC(F)F)CCCCN(C(C2CCCCS2)=O)C1 c1(C(=O)NC2(CF)CCN(c3nnc(C(C)C)o3)C2)cc2cnn(C)c2s1 c1(N2CC3C(C)(C)C3C2)nc(=NCC2(Br)CC2)nc(N2CCC(c3ccco3)C2)[nH]1 C1(F)(C(=O)NCC(CC=C)NC(=O)C(c2cn(C)nc2C)O)CCC(F)(F)CC1 C(=O)(CC1C(=O)Nc2ccc(F)cc21)NC1CC(NC(C2(CSC)CCC2)=O)C1 Cn1ncc2c(C(N3CC4CC3CN(C(C3CCNC3=O)=O)C4)=O)ncnc12 CN=c1[nH]nc(CC(N2CCC(NC(=O)Cc3ccn(C(C)C)n3)CC2)=O)s1 C1(SC)CCCN(C(C2CCN(Cc3cc(OCC)no3)C2)=O)CC1 CS(=O)C1(C(=O)O)CCN(C(c2coc(C3CCOCC3)n2)=O)C1 C(=O)(C1CCOc2ccccc21)N(CC(C)O)CCNC(Cc1c(C)ccs1)=O N1(c2ccnc(NCc3cc(C)c(Br)s3)n2)Cc2cnc(CO)nc2C1 Cc1nc(CC(=O)NC(C)Cc2cnccn2)cs1.C12(CCCO1)C(=O)NC2 C=CCCC(C)NC(C1CC(OCC(C(c2cn(CCC3CC3)nn2)=O)C)C1)=O c1(CC(=O)Nc2cc(Cl)ccc2Nc2ccccc2Cl)c(Cl)cc(Br)cc1Cl N1(C(C2C(C)OCCO2)=O)CCC(C(=O)NCCN2CCCC(O)C2)C12CCC2 CCCCC(=O)C(=O)N1CCCC1C(C)NC(=O)CC1CCSC1 C1(C(=O)NC(CC#C)CC)CN(C(c2nn(C)cc2Cl)=O)CC12CCC2 C(=O)(CS(=O)(=O)CCOC)NCC=CCNC(CN(C1CC1)CC)=O C1(NC(c2c(CCC)n[nH]c2)=O)CCN(C(=O)Cn2cnnc2)C(C)C1 c1(C(=O)NCCC2CCN(C(CCCCC#C)=O)C2)cc(C)c(Cl)cc1F Nc1cnc(Cl)c(C(N2CCC(CF)(NC(c3cncc(OCF)c3)=O)C2)=O)c1 C(=O)(CCCCC(F)F)N(C1C(C)CCN(C(c2cc(C)nn2C(F)F)=O)C1)C Cc1ccc(Cl)c(C(=O)NCC(C)N(C(=O)C=Cc2cccnc2)C)c1 C1(C(=O)NC(C2CCN(C(=O)CCc3cn[nH]c3)C2)(C)C)CCC2CC1C2(C)C c1(OCC)cc(F)cc2ccoc12.C1(=O)CC(C(=O)OC)O1 C#CCC(CC#C)C(=O)NCC(C)CN(C(=O)CSc1ccc2c(c1)CCC2)C N1(C(c2nc(OCC)oc2)=O)CC(CNC(=O)C(F)C(F)(F)F)CC(C)C1 C1(NC(c2cc(OC)ncc2)=O)CN(C(c2ccc(C)nc2O)=O)CCC1C N1(C(C=Cc2ccc(CC)o2)=O)CCCC(CO)(NC(=O)CC2C=CCCC2)C1 C1(C2(O)CCN(C(c3c[nH]c(=N)o3)=O)CC2)(NC(CC(C)(C)O)=O)CC1 C1(C(N2C(C(=O)NCCCC)C=CCC2)=O)CCCCC(=O)N1 c1(NC2CCN(C(C(N3CC(C)(C)C3)C)=O)CC2)cccc(Cl)c1Cl CN(C)S(=O)(=O)N(C)CC(=O)NCC1CCCCN(C(C2(F)CC=CCC2)=O)C1 N1(C(C2CC(=C)C2)=O)CC2CC(C1)CN(C(=O)C(CCC)CC(C)C)C2 c1(C(=O)NC2CN(C(C=C(C)c3ccc(F)cc3)=O)C2)ccc(O)c(N=[N+]=[N-])c1 CC(C)C(C)C(=O)N(CCCNC(=O)C(c1cccnc1)NC(N)=O)C1CC1 C1(CC(=O)OCC)CCCC1.N1(C=O)CCC(NC(=O)C(C)N(CC(C)C)C2CC2)C1 CN1C(=O)NCC1C(=O)NCC1(CNC(c2cc(Cl)no2)=O)CCC1 c1(NCc2ccc(Cl)s2)ccc(C#N)c(C(F)(F)F)c1.C123CC(C1)(C2)C(=O)N3C C1(Nc2c(C)cncn2)C(C)CN(CCC2CCCN2C(=O)C(C)C)CC1C CC(O)C(C(=O)NCCC1CN(C(C2(n3cnnn3)CC2)=O)CCO1)N(C)C C123CCN(CC1C2)C(=O)CO3.c1(C(=O)OC(C)(C)C)cccc(OCC(F)F)n1 Cc1ccccc1C=CC(N1CCOCC1CCNC(C1CC(Cl)(Cl)C1)=O)=O c1(N2C(C(N3CCCC3c3ccc(C(=O)O)cc3)=O)CCC2)cc(Cl)cnc1F O=C(CCOCCCF)NNC(=O)N1CCC(N2CCCCC2CCO)CC1 CC(C)CC(C(=O)NCc1cnn[nH]1)N(C(=O)Cc1cccs1)C c1(CSC)cc(C(=O)NCC2C(CNC(C3CCS3(=O)=O)=O)C2(F)F)ccc1F CCC(F)(F)C(=O)N1CCC(C(C)NC(c2cn[nH]c2)=O)CC1 CCC(CC)C(=O)NCC(C(C)C)NC(c1cc(-c2ccn(C)n2)on1)=O c12cc(C)c(c(C)c1)C(=O)NCC(SC1CC1)C(=O)N2.CCSCOOC.O.C(C)C C1(C(C)C)CN(C(=O)C(=O)NCC(F)(F)CC2CC2)CCO1 Cc1ccc2[nH]cc(C(N3CCCC(N(C(=O)CC(C)C)C)C3)=O)c(=O)c2c1 c1(CC(=O)NC2CC3CCCN3C2)c[nH]c2ccc(Br)cc12 C1(CNC(CCOCC)=O)CCCC1C(=O)NCCCCN(C)C(=O)C1CC1 C1(CNC(C2(COC)CCC2)=O)CCc2cn(C)nc2C1.C1(C(=O)N)CC1C(=O)C1CC1 N1(C(CC(C)P(C)(C)=O)=O)C2CCC1C1CC1(NC(=O)CCc1ncc[nH]1)C2 C(=O)(CCCCCCNC(c1c[nH]cc1C)=O)N1CCC(COCC)C1 c1(NC(C2C(CNC(C(C)OC3CCCC3)=O)C2)=O)cccn2ncnc12 CCCCC(C)CCC(=O)NCC1(O)CCN(C(c2coc3c2COC3)=O)C1 C1(C(=O)NCC2CCN(C(c3cc(CCC)nn3C)=O)C2)CCN2CCOCC12 c1(C(N2CC(NC(=O)C(C)S)CC(C)C2)=O)cccc2[nH]ncc12 C1(NC(CCC)=O)CCC(C(=O)OC2(C)CC(NC(=O)CSCCOC)C2)C1 C(=O)(C(C)(CSC)NC(C1CC(CCC)C1)=O)NC(CCC)C1CCC1 Cc1c(C(=O)NC(C)CN2CCN(C(C3CN(C)C3)=O)CC2)sc2nccn12 C(=O)(C(C)CC(=O)N(CC(CO)(CO)NC(=O)C(C1CC(F)(F)C1)O)C)OC c1(CC(N2CC(C=C)C(NC(=O)CSC(F)F)C2)=O)cnc2cccnn12 C1(C(N2CC(C(C)C)N(C(=O)CCc3cccs3)CC2)=O)CCc2nn[nH]c2C1 CC1CC=CCC1C(N1CCC(C(C)(C)NC(=O)C(=O)NCC(F)(F)F)CC1)=O C(=O)(CCCCCCCCCO)N(CCNC(C(C)OCC(C)C)=O)C C1(NC(c2nn(CC)c(O)c2)=O)CN(C(=O)C(C)Cn2ccnc2)CC1N=[N+]=[N-] c1(OC)cccc(C#N)c1NC(C1CC1C(=O)Nc1c(C(N)=O)cnn1C)=O Cc1ccc(CNC2CC(NC(c3cnn(C)n3)=O)C2)o1 c1(CC)cc(C(=O)NC(C)CCN(C(=O)C(c2c(C)n[nH]c2C)C)C)ccc1C C1(NC)CCN(CC(c2cc(Br)sc2Cl)=O)CC1 c1(C(C)C)ccc(C(=O)NC2CCC(CNC(C34CCCC3C4)=O)CC2)cc1F N1(C(C(CC)C)=O)CC(NC(c2cc(F)ncc2Br)=O)C(F)(F)C1 c1(CCNC)cccc(NC(=O)NC(C)CCc2ccc(Br)s2)c1 C1(S(C)(=O)=O)(C(=O)NCC(C2CCCC2)NC(c2c(C)con2)=O)CC1 C1(NC(C2CC(=O)NC2)=O)CCC2(CC1)CC2NC(C1CCCCCCC1)=O Cn1nc([N+](=O)[O-])cc1C(N1CC2CC(NC(=O)CCC3CC3(F)F)C2C1)=O C(C1(CO)CCc2ccccc21)NC(=NCC=C)NCCc1ccccc1OC CCC(CC)CCCC(=O)NC(CO)C(C)NC(c1nccc2[nH]ccc12)=O c1(C(N(CCNC(C2(OC)CCOC2)=O)C2CC2)=O)ccc2[nH]c(=N)oc2c1 C1(O)(CNC(CC(=C)C)=O)CC2CCC(C1)N2C(c1ccc(SC(F)(F)F)nc1)=O CC(C(=O)N(CC(C)O)CCNC(=O)C(c1ccc(Br)s1)=O)C(C)O C1(NC(=O)C=C(C2CC2)C2CC2)CC(F)CN(C(=O)CCC2CC2(F)F)C1 c1(NC(C(CCOCC)NC(c2n[nH]c(C)c2C)=O)=O)cc(C)ccc1O Nc1c(Cl)cnc(C(=O)NC2CCC(CNC(C3CC=CC3)=O)C2)c1Cl c1(C(N(CCNC(C2CC(C)(C)C2)=O)CC2CC2)=O)cc2c(cn1)CCCC2 C1(NC(c2nc3ccccc3o2)=O)CC2CCC(C1)N2C(=O)C(F)(F)Cl Cn1cnc2sc(C(=O)NCC34CCC3CN(C(c3cccc(O)n3)=O)C4)cc12 C1(NC(C(COC)O)=O)CC2CCCC(C1)N2C(c1cccc(C)n1)=O c1(C(=O)N(CC)CC2CCCC2NC(=O)C(F)C(F)(F)F)ccn2nccc2c1 c1(Cn2cc(C(CC(=O)O)NC3CCCCC3F)nn2)cc(Cl)ccc1[N+](=O)[O-] c1(C(N2C(COC)CCC2)C(=O)NCCSC)nn(C)cc1C CC1(C)C(NC(=O)CC2(c3ccon3)CC2)CC1CNC(c1nc(=N)[nH][nH]1)=O C1(C(=O)NC(CNC(c2cccc(F)c2F)=O)C2CCC2)CC2C=CCC(C1)C2 Cc1cccc(C(O)C(=O)N(CCNC(C2(C3CCCO3)CCC2)=O)C2CC2)c1 C(=O)(CCCC(C)(C)C)NC(CC)CN(C(=O)CCC(=O)c1ccc[nH]1)C C1(C(=O)NC(C2CSC2)=O)CN(C(C)C)CC12CCC2.C1(=O)CC(C)N1 C(=O)(CCC(F)F)NC(C)(C)CNC(C1(n2cccn2)CCC1)=O CC(CC(C)(C)C)C(=O)NCCN1CCC(NC(=O)CCC#N)CC1 Cc1cc(C(F)(F)F)nc(N2CCC(C(C)NC(C3(CO)CCCO3)=O)C2)n1 CCC(C)CCCC(=O)NC1COCC1CNC(c1cccc(F)c1)=O C=CCCCCCCCCC(=O)N1CC(NC(=O)C(C)CC(N)=O)C2(CCC2)C1 N1(C(CCCN=[N+]=[N-])=O)CCOC(c2cn(C3CCOC3)nn2)C1 CC1(C)C(NC(=O)CN2CC3CC3C2)CCN1C(C1SCCCS1)=O C1(NC(CCN(S(C)(=O)=O)C)=O)CCN(C(C2(F)CCC2)=O)CC1F N1(C(C=C(C)C)=O)CCN(C(c2ccc(-c3ccccc3)cc2Cl)=O)CC(O)C1 C(CC1=CCN(C(=O)CN2CCCC2CO)CC1)NC(=O)Cc1ccns1 C=CCC(CC=C)C(=O)NC1CCN(C(=O)CC(c2ccc(OC)cc2)C)C1C C#CCCCCC(=O)N1CC2(CNC(=O)CC(C)SC)CC2(C(F)(F)F)C1 N1(CC)CCCCC1C(=O)N(CC(C)C(=O)NCC1CS(=O)(=O)C1)C C1(C(N2CC3C(CNC(COCCC)=O)(CC3)C2)=O)CNC(=O)CC1(C)C Cc1nn(C)c2sc(C(=O)N(CC(C)NC(c3ccc4cc[nH]c4n3)=O)C)cc12 C(=O)(CC(C(C)OC)NC(=O)CP(C)(C)=O)NCC(CC(=O)OC)C c1(C(CO)NC(c2cc(CS(C)(=O)=O)no2)=O)ccc(F)cc1F c1(NC(=O)NCCCn2cncn2)ccccc1Cc1ccccc1F C(=O)(C1CCCc2ccccc21)NCC12CCC(Nc3ncc(C#C)cn3)(C1)CO2 C(=O)(CN=c1[nH]c(N2CCC3(CC2)N=N3)ncc1Br)NCCC C=CCC(CC(F)F)C(=O)N1CC2(NC(=O)C(C)C(F)(F)C(F)F)CCC1C2 N1(C(Cc2cncc(C)c2)=O)CCC(NC(C2CC2CN(C)C)=O)C(F)C1 c1(C(N2C(C(C)NC(C3(C(F)F)CC3)=O)CCCC2)=O)cc2ccc(Cl)cc2o1 C1(C(N2C(CC(=O)NCc3c(C)n(C)nc3)CCCC2)=O)CCCCC(=O)N1 C1(O)(CNC(c2cnc(=N)[nH]c2)=O)CCCN(C(c2ccc([N+](=O)[O-])s2)=O)C1 c1(NC(=O)CC2CC(C)C2)ccc([N+](=O)[O-])c(C(F)(F)F)c1.C1(C(=O)NC)CC1(F)F C(=O)(CCCCCC#N)N1CCC(CC(N2CC(C)OCCC2)=O)C1(C)C C1(C(=O)NCC2OCCN(C(Cn3c(C)ncc3)=O)C2)CC(=O)NC(C(C)C)C1 C(=O)(C1=CCCCO1)N(CCN(C(=O)CC1CCS(=O)(=O)CC1)C(C)C)C Cc1nc(C(N2CCCC(O)(CNC(C3C(Cl)(Cl)C34CC4)=O)C2)=O)c(=O)[nH]c1C c1(C(=O)OCC)c[nH]c(=NC(CNC(=O)CSc2nc[nH]n2)C(C)C(C)C)cn1 c1(-c2ccccc2)c(N)sc2ccccc12.CC1CC2N(C1)C(c1ccccc1)C2.N(C)(C[Si](C)(C)C)CC.C c1(C(C(=O)NC2CCN(CCCNC(=O)CC3CC3)C2)(F)F)cccc(F)c1F c1(CC)c(C(=O)NCC2(O)CCN(C(c3c[nH]nc3Br)=O)C2)cnn1C C(=O)(C#CC1CCCO1)N1CCCC(C(=O)NCCNC(C=NOC)=O)C1 N1(C(c2ccc(CCCC)cc2)=O)CCN(C(c2nc(C)oc2C)=O)CC1CC c1(C(=O)NCC2CN(C(C=COCC)=O)C(C)CC2)cc(Cl)c(N)cc1OC c1(C(=O)NCC2CCN(C(CSC)=O)CC2)cccc(OC(CC)CC)c1F CC1COCCN(C(c2c(I)ncn2C)C(=O)NCC(F)F)C1 N1(C(C=C(COC)C)=O)CCC2CCCC12CNC(=O)CSc1ccc(C)c(C)c1 C(=O)(C1=CC(O)CC1)C(=O)CC1CC(C2CC2)C1.C(=O)(CNC)N(C)C c1(C(=O)NCCCCNC(C2CC3CC(OC)C3C2)=O)ccc(S(C)(=O)=O)cc1 n1(C(=O)N(O)Cc2ccccc2)nc(COC2CC=CC2)cc1-c1ccncc1 Cc1ncc(NC(=O)NCc2cncc(I)c2)c(F)c1Br Cc1ccccc1C=CC(=O)N(C1CCN(C(C2CC(C)(O)C2)=O)C1)C O=C(C(F)C1=CCCCC1)N1CC(F)(F)CC1CNC(C12CCCCC1C2)=O c1(N(CCCCCC=C)C)ccc(S(=O)(=O)N2CCC(CC(C)C)C2)cc1Br CC1c2sccc2CCN1C(CC1CCCCC1)C(=O)NCCSCC#N C1(NC(c2cc(C(C)C)on2)=O)C=CCN(C(C2(P(C)(C)=O)CC2)=O)C1 c1(C(C)NC(=O)C(C)O)ccc(F)cc1F.c1(CSCC(=O)O)scnc1C C1(N(C)C(C2CCC(n3cc(CC4COC4)nn3)CC2)=O)CC(O)C1(C)C c1(C(F)(F)F)ccc2c(c1)C1(CC1)CN(c1nnnn1CC1CCCCO1)C2 c1(C(=O)OC)csc(C(=O)NC2CC(NC(=O)C(C3CCCCO3)OC)C2)c1 C1(C)(C(=O)NC(c2nc(C)sc2)C)CN(C(c2cccc(O)c2C)=O)C(C)(C)C1 c1(C(N2CCN(C3CCC(NC(CN(C)C)=O)C3)CC2)=O)nc2ncccn2n1 c1(C(=O)NC2C(NC(COCc3ncc(C)o3)=O)CCC2)cnn(CCO)c1N c1(NCC2(C)CCSCC2)ccc(S(=O)(=O)N2CCC(F)(C(N)=O)C2)cc1Br C(C(=O)NCC(C)CNC(c1cnc(CCC(F)(F)F)s1)=O)(C(C)C)OC C#Cc1cccc(C(=O)NC(C)CNC(=O)Cn2cnc3c2CCCC3)c1C CON1CCC(NC(N2CCOC(Cc3cccnc3)C2)=O)CC1 c1(CNC(C(C2CCCCCCC2)N(C(CC)CC)CC)=O)cccc(C)c1F CC1CN(C(c2c(Br)cccc2[N+](=O)[O-])=O)CC(C)N(C(c2cc[nH]c2)=O)C1 c1(C(N(CC(C)N(C(C(C)OCC2CC2)=O)C)C)=O)ccc2c(c1)N(C)CCO2 C1(NC(C2C(OC)C2)=O)CN(C(C2CCc3nnc(C)n3C2)=O)CCC12CCC2 N1(C(CCC#C)=O)CCC2(CNC(=O)CN=S(C)(C)=O)CCCCC12 CCCCCCC(=O)NCC1(F)CCCN(C(=O)C(=O)NCCC(N)=O)C1 C(=O)(C1CCc2c[nH]nc21)N1CC(CCCCNC(C(CC)C)=O)C1 C1(NC(CC(CC)O)=O)CC2(CCCCN2C(C2(C3CCCO3)CC2)=O)C1 C(C(=O)N(CCCNC(=O)CCc1ccc(Cl)nc1)CCO)(C(C)(C)C)SC c1(CCC(N2CCCC(N(C)C(=O)OC(C)(C)C)C2)=O)cc(F)cc(Br)c1 c1(OCC)cc(C(=O)NCCN)ccc1OC.C(=O)(C(C)N1CC(C)C1)C1CC1 c1(OC)ccc(C(=O)N(C2CCCC2)CCNC(C2COC(=O)N2C)=O)nc1Cl C1(CN(C(=O)CCc2csnn2)CC)CCCN(C(c2cc[nH]n2)=O)C1 c1(C(N2CC(O)(C(C)NC(CN(C)CC)=O)C2)=O)ccnc(Cl)c1Cl n1(CC(C)NCC)cc(CNC(C2(N(C)C)CN(C(=O)C=CC3CC3)C2)=O)nn1 c1(CCC(=O)NCCCNC(C(C(CC)C)OC)=O)ccc([N+](=O)[O-])cc1.C(C)(=O)N CC1C(C(=O)NCCSCCCO)CCN1C(c1cc[nH]n1)=O N1(C(CC2CN(C(C(CC)SC)=O)CC2C)=O)CC2COCC2C1 C12CC(=NO1)C(=O)N1CCC(C1)C(=O)NC2.C1(CC(=O)OC)(COC)CC1 c1(CC(=O)NCCC2N(C(c3cnc(CC)s3)=O)CCC2)ccc(C)c(C)c1 C(=O)(C(O)P(C)(C)=O)N(C(C)CCNC(=O)Cn1cnc(Br)c1)C NC(=O)CC(C(=O)NCCF)NC(=O)Cc1cccnc1 C=C(C)CC(C(=O)NCCC(=C)CNC(=O)Cc1cnn(CC)c1)NC(C)=O.OCC O(NC(=O)C(CCOC)NC(=O)C(C)O)CC(=O)NCC c1(C(=O)NC(C)CCNC(=O)CCC2(C#N)CCC2)cc(Cl)cc2ccccc12 c1(N2C(CNC(C=Cc3cc(C)cc(C)c3)=O)CCC2)ccc([N+](=O)[O-])cc1Br c1(CCC)ccc(N)c(C(=O)NCCN(C)C(C2CC2C2CC2C)=O)c1 C#CCCCC(C)C(=O)NC(C)(CNC(=O)CSCC(F)F)CC(C)C c1(C(C)C(=O)NCC2CC(NC(C3COCCO3)=O)C2)ccc(F)cc1 C1(C(N2C(C)CC(NC(c3ccc(N)cc3Cl)=O)CC2)=O)CC2(C1)CC(C#N)C2 C12(NC(Cc3c(C)noc3Cl)=O)CC(CNC(=O)CC3C=CCC3)(C1)OC2(C)C NS(=O)(=O)CCC(=O)NC1CN(C(=O)CSCCN2CCCC2)CC1C(F)(F)F C1(CNC(C2CCO2)=O)CC(O)C(O)CC1c1cn(C2COCC2C(F)F)nn1 c1(CCC)ccc(C(=O)NC(C)CN(C)C(c2cc(CS(C)(=O)=O)on2)=O)s1 C(=O)(C1=CCN(C(=O)CCC=CC)C1)N(C(C)CCNC(C)=O)CCC C(N=c1nc2c(cnn2C(C)C)c(NCCC#N)[nH]1)c1c(C)[nH]c(=N)s1 C(=O)(CCC(C)S(C)(=O)=O)N(C)CC1CCN(C(C(CC(=C)C)NC(C)=O)=O)C1 C(=O)(C#Cc1ccccc1Cl)N(c1ccccc1)C(C)Cc1cnn(C)c1 C12(C(=O)NC3C(NC(c4c(C)[nH]nc4Br)=O)CCC3)CCCC1CCC2 C#CCCC(C(=O)N1C(CO)CCC1CO)NC(C1SCC=C1C)=O C1(C(=O)NCCCCNC(c2ccc(NC=O)cc2)=O)CCCC2(CC2)C1 N1(C(C(CSC)C)=O)CC2(CCC(CNC(c3cc(F)ccc3Cl)=O)O2)C1 c1(CN(CCNC(c2nccc(C)n2)=O)CC)cc(O)nc(-c2ccccn2)n1 N1(C(c2ccn(C(C)C)n2)=O)CCCC(NC(=O)C(F)=CCCF)C1 n1(CC(=C)C)nnnc1C(c1cc(C(=O)OC)co1)NC(CC)CC c1(C(N2CCC(C)(CNC(c3ccc(C)cc3O)=O)C2)=O)nc2c(s1)COCC2 n1(CC)ccc(CC(N2CC(O)(CC(=O)N(C)Cc3ncc[nH]3)C2)=O)n1 c1(OCC)cc(C(=O)NCCCN(C)C(c2ccc(F)c(SC)c2)=O)cc(F)c1 C(=O)(CC(F)(F)CC(=O)N1CCC2(CC2C(=O)Nc2c(C)cc(C)cc2C)C1)OC c1(C(=O)NC(CCSC)C(=O)NCC2CSCCO2)cccc(C)c1C c1(OC)ccc(F)c(S(=O)(=O)N2CC3CCCC2C3NC(=O)OC(C)(C)C)c1 C=CCC(C(=O)Nc1ccccc1)N(C)C.N12CCCC(C1)CNC(=O)CC2 N(C1CCCc2ccccc21)CC(=O)NCC1CC2(CCCO2)C1 Cc1nn2cc(C(N3CC(NC(c4c[nH]c(Br)c4)=O)CC3(C)C)=O)nc2s1 c1(CCCC(=O)NC2C(NC(C(CC#C)O)=O)COC2)ccc2c(c1)OCO2 C1(C(=O)NC2CC(OC)CN(C(C3(C)CCCO3)=O)C2)CC2CCCC(C1)C2 N1(C(c2ncn(C(C)C)n2)=O)CCC(CNC(=O)CCCn2cccc2)C(O)C1 C(C(O)C(=O)NCc1cccnc1)NC(c1nc(-c2ccccc2)no1)=O c1(C(=O)NC2C(CNC(=O)C(=O)NC3CC3)CC2)cc2cccc(F)c2o1 N1(C(CSCCC)=O)CCN(C(C2CC(SC)C2)=O)C(c2ccc(F)cc2)C1 Cc1ccc(NC2CCCCC2CNC(C2(C)CC(O)CN2C)=O)c([N+](=O)[O-])c1 N1(C(C(C2(C)CC2)NC(C(CC)N(C)C)=O)=O)CCC(COC)CC1 C=CCCC(F)(F)C(=O)NCc1cc(C(=O)NC2CCCC2SC)co1 C1(NC(CCC(=O)NCC)=O)CN(C(c2snc(O)c2Cl)=O)CCC1C(F)(F)F S(=O)(=O)(c1ccc(C(=O)Nc2cnc3ccnn3c2)o1)N(C)C Cc1c(Cl)c(C(N2CC3C(NC(C4CCCCC4(C)C)=O)C3C2)=O)nn1C c1(NC2CN(C(CS(CC)(=O)=O)=O)CC2C)ncnc2c(Cl)cc(Cl)cc12 C(=O)(CCCCCN(C)C(C1CC(C)N(C)C1)=O)NC(N1CCNC1=O)C c1(C(N(CCC(N2CCCC(CC=C)C2)=O)C2CC2)=O)cc(O)nc(O)n1 N1(C(=O)Nc2c(NC(C)=O)cccc2)CC2C3CCC(C3)C2(C)C1 c1(C(=O)NCCC(CNC(C2CCc3nc[nH]c3C2)=O)O)nnn2c1CSCC2 C=CC1(C(N2CC(CN(C)C)C2)=O)CCN(C(=O)C(CN(C)C)CC)C1 Cc1cnc(NCc2ccc3cnccc3c2)n2ccnc12 c1(C(N2CC(C)C(NC(c3ccc(N)c(Cl)c3)=O)CC2)=O)cccn2ccnc12 c1(C(=O)N=c2cc[nH][nH]2)noc2c1CN(C(C1CCCCO1)=O)CC2 C(C(=O)N1CCC(CSC)C1)(C(C)(C)C)NC(=O)COc1cccnc1 C12(CNC(C#CC(=O)N(C)C)=O)CCCC(CN1C(C1CNC(=O)N1)=O)C2 c1(C(N2CC(C(=O)NCCC#CCC)(CC)C2)=O)cccc(=O)n1C C1(CNC(c2c(NC)scn2)=O)CC2(CCC2)CN1C(=O)CCCCCO C1(C(C)C)CN(C(=O)CC2CCN(C(=O)CCc3cccs3)C2)CCO1 C(CC(C)C)(C(=O)NCC1COC(=O)C1)NC(C(c1ccc(CC)o1)C)=O Cc1[nH]c(=NCC2(O)CN(C(=O)C=CC=C(Cl)Cl)C2)ccc1[N+](=O)[O-] N1(C(C2(C(C)N(C(=O)C(F)CC3CCOC3)C3CC3)CC2)=O)CCC(F)(F)C1 C(CCCC(CO)NC(c1cnc(S)[nH]1)=O)NC(C(C)CF)=O C1(C)(CC)CCCN(C(C2CC(C)CCN2C(=O)C(c2ccn(C)c2)C)=O)C1 CC1CCCN(C(=O)CN2CCSCC2)C1CCNC(c1cn2ccsc2n1)=O C1(N(C(c2c(CCC)nco2)=O)C)CN(C(C2CCS2(=O)=O)=O)CC12CC2 C=CC(CC)C(=O)NC(CC(=O)NCC(c1ccsc1)O)C1CC1 C1(C(N(CCNC(COC)=O)C)=O)(CC)CCCO1.c1(C(=O)N)cccs1 c1(CNC(C2C(=C)C2)=O)ccc(C(=O)NC(C2(O)CCCC2)(C)C)s1 c1(OCC)ccc(NC(=O)CCCNC(=O)C(C)C)cc1S(=O)(=O)NC CCC(CC)CCC(=O)NCC1CC(NC(=O)C(C(C)C)NS(N)(=O)=O)C1 C1(CNC(CCCSC)=O)CC(NC(=O)Cc2cc[nH]c(=N)c2)C12CCC2 CCC(C)(COC)CNC(N1CCC(c2cccc(C)c2)C1)=O C1(C(=O)NCCc2ccccc2)(CNC(=O)COCC2(O)CCC2)CC12CCC2 c1(C(=O)NC2CCN(C(C3COCC(C)(C)O3)=O)C2)cnc2c(c1)CNC(=O)N2 c1(OC)cccc(C=CC(=O)NC(c2nnnn2C(C)C)CCC2CCCC2)c1 CC#CCC(C(=O)NCCC1CCCC1(C)C)NC(=O)CCCCC#N C1(C(N2C3CC(CNC(=O)Cc4ccoc4)C2CC3)=O)CCn2nnnc2C1 C1(CNC(C(CC2CCCC2)OC)=O)CN(C(C2(C)CCCCC2)=O)CCCO1 N1(C(C(C)C(C)(F)F)=O)CC2(CCCCN2C(c2ccnn2C2CC2)=O)C1 Cc1nn(C)c(=O)c(C(N2CC3CCC2C(NC(c2csc(Cl)c2)=O)C3)=O)c1C c1(NC(C2SCCN(Cc3cc(C)c(F)nc3)C2)=O)c(Cl)ccc2nsnc12 c1(OC)cnccc1C(=O)NCC1(NC(C2CC2c2nc[nH]n2)=O)CCCCC1 N1(C(c2nc(C)sc2)=O)CC2CC1CC2CNC(c1cnn(CC(F)F)c1)=O c1(Cc2c(SC(N3CCc4ccsc4C3)=O)ccc(F)c2)cc(F)c(F)c(F)c1 C1(C)(N(C(C)=O)Cc2ccc(Br)cc2)CCN(C(=O)C(N2CCSCC2)=O)C1 Cc1nc(N2CCN(C)C(CNC(c3cncc(Cl)n3)=O)C2)cc2nncn12 C(c1ccco1)=C(C)C(=O)NCC(C(=O)NCC1(n2ccnn2)CC1)N(C)C N1(C(C2N(C(c3cc(OC)no3)=O)CCC2)=O)CCC(O)(C(N)=O)CC1 N1(C(CNC(c2[nH]cc(C(C(C)C)=O)c2)=O)=O)C2CCC1CN(C(=O)CO)C2 c1(C(CN(C2CCCC2n2ccnn2)C)=O)cc(F)cc(Br)c1 C1(C)(C(N2CCC(C(C(C)C)NC(C3C(=C)C3)=O)CC2)=O)CCN(C(C)=O)CC1 CC1(C)CC(O)CCN(C(=NCc2nccs2)NC2CCS(=O)(=O)C2)S1 C1(NC(=O)C(CCF)NC(c2sccc2Cl)=O)CCc2n[nH]cc2C1 C1(C(=O)NCc2cc(C(=O)NC(C34CC(CO3)C4)C)n[nH]2)CN2CCN1CC2 C1(N(C(C(CC)O)=O)C)CCC(NC(=O)CC2C=CCCC2)CC1 c1(C(=O)NC2(C)CCN(C(=O)Cc3cc(C4CC4)on3)C2)cc(O)ncc1Br CC(N=c1nc2scnc2c(NCC2CCN2C(C)(C)C)[nH]1)c1cc(Br)ccc1F N1(C(C(C(C(C)C)O)(F)F)=O)CCC2(CC1)CN(C(=O)CCCCF)CCO2 C(C)(CN=c1[nH]c(Cl)ncc1Br)(C1CC1)NC(CCC1CC(OCC)C1)=O N1(C(c2c(CC)c[nH]c2)=O)CC2CC(NC(=O)CCn3ccnc3)CC1C2 CCCCCCCCCC(=O)NC1C2CC1N(C(=O)C(F)C(F)(F)F)C2 Cn1nc(C(=O)NC2COCC2NC(=O)C(C)(C)c2cscn2)cc1OC(F)F C=CCCCC(C(=O)NCCC(C)CCO)NC(=O)C(COC)CC(C)C CC(CCCCNC(=O)Cc1ccc(C(N)=O)nc1)NC(c1ccsn1)=O c1(C(N(CCCN(C(C(CC)NC(C)=O)=O)C)C)=O)nccc2ccsc12 Cc1ccc(C)c(C(N2CCC(CNC(c3cnn[nH]3)=O)CC2)=O)c1C c1(C(=O)NCCC(CNC(=O)CCOC2CCOC2)O)ccnc(OC(F)F)c1 C1(CC)CC(C(=O)N(CCNC(=O)C(C)NC(N)=O)CCOC)C1 C(=O)(CCCCC(=O)N1CCN(C(c2c[nH]cc(C)c2=O)=O)C2CC12)OC c1(C(N(CC(C)NC(c2c(Cl)cnn2CC)=O)CC)=O)onc2c1CCCC2 c1(C(N2C(CN(C(=O)Cc3csnn3)C)COCC2)=O)ccnn2ccnc12 C1(C(=O)O)CN(CC(=O)NC(CCCCSC)OC(C)(C)C)C2(CCC2)CO1 Cc1cc(=O)n(CC(N2CCC(O)(CCNC(=O)C(O)C3CCCC3)C2)=O)cn1 N1(CCCC)CCCCC1C(=O)NC1CC(CNC(=O)C(C)Cc2cnc[nH]2)C1 N1(CC2(CSC)CC2)CCCC(O)CC1 C1(NC(C(CSC)C)=O)CCN(C(c2cn(CCCN(C)C)nn2)=O)C(C)C1 C1(C(NOCCCOC)=O)CC2(CCN1C(=O)C1=NOC(C)C1)CC2 C1(C)(C(N(C2CN(C(c3n[nH]c(C)c3C)=O)C2)C)=O)CCC(C)C1(C)C c1(OCCC)cccc(CN2CC3(CC3C(=O)Nc3nsnc3NC)C2)c1 N1(CC(C)NC(c2cc(CCC)[nH]n2)=O)CCN(C(=O)CC2CC2)CC1 CC1(C)CCN(CC(N2CC3CC3(CNC(C3CC(C#N)C3)=O)C2)=O)CC1 c1(OC(C)C)cnc(C(=O)NC(C2CCN(C(c3ccn(C)n3)=O)C2)C)cn1 C(CC(F)C(=O)NC)NC(c1n(CC)ncc1)C(=O)OC N1(C(CCc2onc(C)n2)=O)CCC2CCC(NC(c3ncsc3C)=O)C1C2 S(=O)(=O)(c1cccc(NCc2c(C)nn(C)c2Cl)n1)NC1C(CCCC)CCC1 c1(C(N2C(C(=O)Nc3c(OC)c(C)sc3)C=CC2)=O)cn(C)c2ccccc12 N1(C(C2(OC)CCCC2)=O)CC2CC(NC(=O)CN3CCOCC3=O)CC(C2)C1 C1(CNC(c2cc(C)c(C)s2)=O)CC(F)(F)CN1C(=O)CCCc1cccnc1 C1(C(=O)NC(c2nccc(=N)[nH]2)C)COCCN1CC=Cc1cnccn1 Cc1c(C(=O)NC2(C)CCN(C(C3CC3c3nccn3C)=O)C2)n[nH]c1C1CC1 c1(C(N2CCN(C(C(C=C)O)=O)CC2CC(F)F)=O)ccc2[nH]ccc2c1 Cc1c(C=CC(N2CC3CCC3(NC(c3cccc(=O)n3C)=O)C2)=O)cnn1C N1(C(c2c(C)n(CCO)cc2)=O)CCC(NC(C2(C)CCCCO2)=O)C(CO)C1 C1(CNC(=O)CCC(=O)N(C)C)CC(C(=O)N(C2(C(=O)OC)CC2C)C)CCO1 Cc1nc(N2CCCC(CO)(NC(=O)Cc3csc(C4CC4)n3)C2)cc(O)n1 Cc1cscc1C(=O)N(CCCCN(C(=O)CCCc1ccccn1)C)C CC(C)C(O)C(F)(F)C(=O)NC1CC(C)N(C(c2csc3cncn23)=O)C1 C1(CC)CCCN(C(=O)CC2(C)CCN(C(=O)CCCNC(=O)OC)C2)C1 N1(C(Cc2cc(CN3CCOCC3)[nH]n2)=O)CCOC(CNC(=O)C=CC)C1.O=CN CC(C)C(C#N)C(=O)N1CC(CNC(c2ccn(C(C)(C)C)c2)=O)CC1(C)C C(c1cncc(F)c1)=CC(=O)NC(CC)CNC(=O)CCNC(=O)CO C1(CNC(C2C(CC)(COC)C2)=O)C(C(F)F)C1(C)C.c1(C(=O)N)ccc(F)o1.C1CN1 c1(C(=O)NCCCN(C(c2ccc(CC)nc2C)=O)C)ccn2c1CCCC2 c1(C(N(CCOC)CCNC(=O)C=C(C2CC2)C2CC2)=O)c2c(nn1C)CCC2 C1(N(C(CCCC#C)=O)C)CN(C(=O)CCCC2CCCC(=O)N2)CC1(C)C c1(C(N(CC(CC)NC(C2CC2Cc2ccccc2)=O)C)=O)ncn(C)c1C C1(CCNC(C2C(F)(F)C23CC3)=O)CCCN(C(c2ccsc2Cl)=O)C1 c1(C(N2C(CN(C(CCC)=O)C)COCC2)=O)cccc(C)c1N c1(SC)snnc1C(=O)N(CCCNC(=O)CCCn1ccnc1C)C(C)C c1(CCNOC)cccc(F)c1.C1(=O)C(C)O1.C1(=O)CN1.C(C)=O C1(C(=O)NCCNC(C2C3CN(C)CC32)=O)CC12CC(F)(F)C2 c1(-c2ccc(C)cc2)cc(=NC(=O)C(F)(F)C(F)(F)Cl)[nH]o1 c1(C(=O)NCCC(C)N(c2nccc(C(C)(C)C)n2)C)ncnc2c1cnn2C C1(CNC(=O)CN2CCS(=O)CC2)C(O)C(O)CN1C(C1CC1c1ccoc1)=O Nc1ccc(-c2cn(C3CC(NC(=O)Cn4ccnn4)C3)nn2)cc1 c1(C(=O)NC(CNC(c2cn(C)nn2)=O)CO)ccc(S(=O)(=O)NC2CC2)cc1 C(=O)(C(C)(C)S(=O)(=O)C1CC1)NCCOCCNC(C1CC(C)(C)C1)=O c1(-n2c(C(CCC(C)CCO)CC)nnn2)ccc2c(c1)CCC2.C1(C)(N)CC1 c1(CNC(C(N(C(C(CN(C)C)O)=O)C)C2CC2)=O)cc2ccccc2[nH]1 C12(C)CCN(C1)c1ccc(s1)-c1c(ccs1)CCN(C)CC2C.CCO CCC(CO)(C(=O)NCCOC1CCN(C(c2coc(C(F)F)n2)=O)C1)OC N1(C(c2ncc(C)c(Cl)c2)=O)CCC2(CCCN2C(c2nc(=O)n(C)[nH]2)=O)CC1 N1(C(C(C)(C)OC)=O)CCCOC(CNC(c2cc(OC)n[nH]2)=O)C1 c1(C(=O)OC)cc(C(=O)NCc2ccccc2-n2cnc(C)c2)c2cccnn12 N12CCN(CC1CCO)C(=O)c1nc(cs1)CC2=O.C1(OC)(CF)CCC1 c1(NC(C)=O)cc(C(=O)NC2CC(CCC(c3ccsc3CO)=O)C2)ccc1C Cc1ccn2c(C(=O)NC3CCCCC3NC(C3(C(F)F)CCC3)=O)cnc2c1 N1(C(C(COC(C)=O)C)=O)CCC(C)C(NC(=O)Cn2cncn2)C1C N1(C(C2CCCC(C)(C)O2)=O)CC2CN(C(=O)Cc3cnn(C(F)F)c3)CC2C1 N1(C(c2c(CC)scc2)=O)CC2CC(NC(c3ccoc3C3CC3)=O)C1C2 CCS(=O)(=O)CC(=O)N1CCN(C(c2c[nH]nc2Cl)=O)CC1CC#N C(C(O)CCNC(=O)Nc1c[nH]cc1-c1ccc(Cl)s1)NC(=O)OC(C)(C)C C(=O)(C(CC(C)(C)C)OC)NCC(=CC(=O)NC(CC(=O)OC)(C)C)C C(=O)(CCCC(F)(F)CO)NC(CCCC)CNC(=O)CN1CCC(C)C1 N1(C(C2CC(=C)C2)=O)CCCC2(CCN(C(c3cccc4nn(C)cc34)=O)C2)C1 N1(C(c2n(C)nnc2)=O)C2CCC1CC(CNC(c1ccn3nncc3c1)=O)C2 CCS(=O)(=O)C1CN(C(=O)C(n2cc(-c3nc(C)ncc3Cl)nn2)C)C1 c1(CN2C(C(=O)NC(c3ccncc3)(C)C)CNCC2)cc(Cl)c(Cl)cc1O c1(-c2cn(CCCCCNC(c3cnns3)=O)nn2)cccnc1F Cc1cncc(-c2cn(CC(=O)NC3CCN(C(c4csc(C)c4)=O)C3C)nn2)n1 c1(-c2scc(CC)c2)nc(-c2ccc(C)cc2)nn1C1CCCOC1 C1(C(N2CC(C)(NC(CCNC(C(C)(C)C)=O)=O)C2)=O)CC2CCC1NC2=O Cc1cc(N)cc(C(=O)NC(C)(C)CN(C(=O)C2=CCOC2)C)c1F CCC(CNC(c1csc(C(=O)NC(C)C)n1)=O)N=c1[nH]c2ccc(O)cc2s1 c1(C(=O)NCC(N2CCC(F)C2)C)ccc(-c2cnoc2)cc1 C(CC(C)(C)CC(=O)N1CC2CC1CCC2NC(c1coc(SC)c1)=O)OC C(=O)(CCN(OC)C(=O)C(F)CC1CCOC1)NCC(=O)OC CCCCCCC(C)CC(=O)NCC(O)CNC(C1CN2CCN1CC2)=O CCC(O)CC(=O)NCC1C(CNC(C23CCC(OC)C2C3)=O)C1(F)F C(=O)(C1Cc2c(Cl)cccc21)N1CC(=C(CNC(C(c2cnn(C)c2)C)=O)F)C1 c1(C(N(CCOCCN(C(=O)C2=CCCCC2)C)C)=O)ccc2c(c1)CCCC2 CC(C)CCCCCCNC(=O)C(CC(F)F)NC(=O)OCc1ccccc1 C1(CNC(Cc2ccn(C)c2)=O)CC2CCC(C1)N2C(=O)C(O)CC(F)(F)F c1(OCC)cccc(CN=C(NC(C)C)NC2CCN(C(=O)OC)C2)c1 CC(C)C1(C(=O)NCc2ccc3c(c2)nnn3C)Cc2ccccc21 C1(C)(CNC(Cc2cc(C)no2)=O)CCN(C(C2CCCCC2O)=O)C1 N1(C(C2CCN(C(c3cnn(C)c3N)=O)C2(C)C)=O)CC(CO)C2(CCC2)C1 C1(C(=O)NCC(CO)NC(c2cccc(C(C)(F)F)n2)=O)CCCS(=O)(=O)C1 C(C(C)C)(C(O)C(=O)N1CC(CNC(C2CN(C)C2)=O)CC1(C)C)OC N1(C(C(C)=C(CC)C)=O)CCC(CC)C1CNC(=O)C(C)CC C(=O)(C(C)(C)CC(=O)NCC(CNC(C12CCCCC(F)(C1)C2)=O)CO)OC CCCC(C)(C)CC(=O)N(C1CN(C(=O)C(C2(O)CCCC2)F)CC1(C)C)C C(=O)(C1=NOC2COCC12)N(C(C)CN)C.O(CP(C)(C)=O)C(=O)C N1(C(C)=O)CCC2(CC1)CC2C(=O)NC(C)(CCCl)c1nn[nH]n1 c1(NC(=O)NC(CSC)(C)C)ccc(N2CCSCC2)cc1 N1(C(c2c(C)nc(C3CCCO3)s2)=O)CC2CC(NC(=O)CC(C)(F)F)CC1C2 Nc1cccc(Cl)c1C(N1CCC1CNC(=O)CCCCc1ccccc1)=O C#Cc1cncc(C(=O)NC2CN(C(C3(SCC)CC3)=O)C2)c1 C1(CC(=O)NCc2n(CC)nnn2)CC2(C1)CN(C(C1CCSC1)=O)C2 C1(C(=O)OC)(NCCN2CCC(NC(C3CCCNC3=O)=O)CC2)CS(=O)(=O)C1 C1(NC(CNS(N)(=O)=O)=O)C2CN(C(c3csc(Cl)c3Cl)=O)CC12 N1(C(CCN(CCOC)C)=O)CC(F)(F)CC1CNC(=O)Cc1csc(C)c1 Cc1ccc(Cl)c(-c2cn(C(C)C(=O)NC3(C(N)=O)CCCOC3)nn2)c1 N1(C(=O)OCCC#C)CCCN(N2CCC(C)(c3cc(C)[nH]n3)C2)CC1 c1(C(=O)NCC(C)NC(COCc2onc(C)n2)=O)cc(F)cc2nn(C)cc12 C=CCCCC(=O)NC1CCC(NC(=O)C(c2ccc(O)cc2)(C)C)CC1 C1(NC(=O)NCCCCSc2cccc(Cl)c2)CCSC2(CCC2)C1 CC(CC(=O)NCC(O)CN(C)C(c1ccn(Cc2ccccc2)n1)=O)N(C)C c1(CC(=O)NC(C2C(C(NOC(C)CO)=O)C2)C)ccn(C)c1 CCC(C)(C)C(=O)NCC1CCCCC1C(=O)NCc1cn(C)cn1 c1(C(=O)NC(CC)C(=O)N2CCC2(C)C(=O)OC)cc(O)cc(F)c1 C(=O)(C(O)C(F)F)N(CCOCCCN(C(=O)CC1C=NNC1=O)C)C C(=O)(C(F)(F)Cc1ccc(F)cc1)NC1C(NC(C2CC(C(F)F)C2)=O)COC1 C(=O)(C(C)(C)CC1CC1)N1C(C2(O)CN(C(CCCOCC)=O)C2)CCC1 C(=O)(C(O)CC(F)(F)F)NC(CN(C(c1cccc(NC(C)C)c1)=O)C)C c1(-n2c(CCO)nc(CSCCC)n2)ccc(OC)c(-c2ccnn2C)c1 C12(CCNC(C(CC=C)C)=O)CCC1CN(C(c1csc(C(F)F)c1)=O)C2 N1(C(c2[nH]cc(C(C)=O)c2C)=O)CC(C)CN(C(=O)CC23CCC(CC2)C3)CC1C C1(C(=O)NCCC(C(=O)NCC(CC)(F)CC)O)Cc2nccn2C1 c1(CC)nn(C)cc1C(=O)NC(CO)C(C)NC(=O)CN1CCC1C C1(C(N2CCCC2CCOC)=O)CC2CC1CC2(F)F.n12cc(nn1)C1(CC1)C2 N1(C(C2CSCCS2)=O)CCC(O)(c2cn(Cc3ccno3)nn2)CC1 C1(NC(C2CNC(=O)N2)=O)CC2CCC1N(C(=O)C(c1ccc(F)cc1)O)C2 C(=O)(C1CCCc2cccnc21)NC(c1ccc(F)cc1)CN(C)C c1(C(C)C)ccc(O)c(C(N2CCC2CNC(C2CC2CN(C)C)=O)=O)c1 C(CCN=C(NCC12CCCC(C)(CO1)C2)NC1CC1)OC(C)=O CC1=C(C(=O)N2CCC(NC(=O)CCCCN(C)C)CC2C)CCS1(=O)=O c1(C(N2CCC(NC(CC3(OC)CCC3)=O)C(CO)C2)=O)c(C)ccc(C)c1C c1(C(COC(C)(C)C)NC(C=CC(=O)NC(C2CC2(F)F)COC)=O)cccs1 N1(C(C2CC(C)OC2)=O)CCN(Cc2cn(CC3(C)CCC3)nn2)CC1 c1(C(N(C2CC(NC(C3N(C(C)=O)CCC3)=O)C2)C)=O)cc2ccnc(Cl)c2[nH]1 c1(CC)ccc(C(=O)OC)cn1.c12ncc(s1)CCNC(=O)N2 CCCC(C(=O)N1CCC(C(=O)Nc2cnccc2OC)C1C)N(C)C c1(C(=O)NC(COC)CNC(=O)Cc2cnsc2)cc(C#N)[nH]c1C C(CO)(CC(O)c1ccccc1)NC(C1(O)CC(OCCO)C1)=O C1(CC=C)(NC(=O)CCn2ccc(=N)[nH]2)CCCN(C(C2(C)CC2Br)=O)C1 O=S(=O)(c1ccc(N2CCCC(C3CCC3)C2)c(F)c1)NCc1cc(Br)ccn1 C1(CC(N2CC(OC)(CO)C2)=O)CN(C(C2COC(C)C2)=O)C(C)(C)C1 N1(C(C2C(=C)C2)=O)CC(C)(CNC(=O)Cn2ncccc2=O)CC1(C)C C1(O)(CNC(C2(COC(C)C)CC2)=O)CCN(C(=O)C#CC(C)C)CC1 C1(NC(CC)CC2CCCCO2)CCCN(C(=O)C(C)(C)CC)C1 Cc1cccc(C)c1CC(=O)NCCC(C(C)C)NC(c1cncn(C)c1=O)=O c1(NC2CCC(C(=O)NCc3nccc(OC)c3)CC2)ncc2cc(Br)cn2n1 C(=O)(C1=NOC2(CCCN(C(=O)C(C)n3cccn3)C2)C1)NCc1occ(C)n1 N1(C(C(C2CN(C(=O)CSc3nncs3)C2)O)=O)CC2(CCC2O)C1 C1(CCNC(=O)NCCC2CCCO2)CCCOC1 c1(CNC(C2(C(N)=O)CC2)=O)ccccc1CNC(=O)CSC1CCCOC1 C1(COC)CN(C(c2ncsc2C2CC2)=O)CCN1C(c1cnn2ccsc12)=O Cc1cc(F)c(N)cc1C(=O)NC1CN(C(=O)CCc2ccc3[nH]ccc3c2)C1 C1(CNC(CCCC(C)=O)=O)CN(C(C2CC2CF)=O)CC(C)(C)C1 Cc1ncc2n1CCC(C(=O)Nc1ccc(CNC(=O)C(C)(C)CO)cc1)C2 C1(C(=O)NCC(C)Cn2ccnc2)CCN(C(c2sccc2F)=O)C12CCC2 N1(C(CC)=O)CCOC2CN(C(c3ccc(Cl)c(OC)c3N)=O)CC12 Cc1ccsc1C=CC(=O)NC(C1(CNC(=O)CC(F)(F)Cl)CC1)C CN1CCN(C(c2cccc(C3CCOCC3)c2)=O)CC1CNC(=O)CC1CC1 N1(C(C(CC)CC)=O)CCN(C(=O)CCc2ccc(Cl)nc2)C(CC)C1 c1(-c2nc(NC(c3cccc(F)c3I)=O)sc2)cnc2[nH]ncc2c1 Cc1ccc(OCC(N2CC(NC(=O)C(C)C3CCOC3)CC2C)=O)cc1 N1(C(=O)OC(C)(C)C)CC=C(C(C)(C)C(=O)NCCCSCC2CCCOC2)C1 N1(Cc2c(C)nns2)C(=O)CCN(Cc2noc3c2CCCC3)C1=O CC1CN(C(c2ccnc(Cl)c2)C(=O)NC2CCC2)CCO1 C1(N(C(c2c(CC)nn[nH]2)=O)C)CCN(C(=O)C=C(C2CC2)C2CC2)CC1C Cc1nc(C(N2CC(O)CC2CNC(=O)C(C)CF)=O)c2ccccn12 c1(C(=O)NC2CCN(C(C3C(C)CCS3)=O)CC2)cc2nccc(Cl)c2s1 c1(C(=O)NC(C(C)NC(=O)CC2CCC2)C)cc2n(n1)CCCC2 c1(CC)ncc(C(=O)N(C2CCN(C(C3C(C)(C)C3(C)C)=O)C2)C)c(O)n1 C1(N(C(Cn2cc(C(C)O)nn2)=O)C)CN(C(c2ccc(OC)s2)=O)CC1O C1(NC(CN(C(C)C)C)=O)CCCN(C(C2CCCCC2c2ccnn2C)=O)C1 c1(C(=O)NCCN(C(=O)CC(c2ccc(F)cc2)C)CC)ccc(C)nc1OC S(=O)(=O)(c1c[nH]ccc1=NCC1CCOC1)N1CCCC(C(C)C)C1 c1(C(=O)NCCCCN(C(C(C)N(C)C)=O)C)cncc2cccnc12 c1(CCC(=O)NC23CC(NC(=O)C(O)CC4CC4)(C2)C3)cnccn1 c1(OC)c(Br)ccc(F)c1C(=O)N(Cc1ccccc1)Cc1cncnc1 N(C1CCCc2ccoc21)C(C(CC(=C)Cl)NC(c1ncccc1N)=O)=O c1(NC(CNC(C2(SC)CC2)=O)C2CCC2)ncnc2scc(Br)c12 CC1CC1C1CC1C(=O)N(C)CC1CCN(C(=O)CS(C)(=O)=O)C1 c1(CC(C(=O)N(C)CC2N(C(C(C3CC3)OC)=O)CCC2)C)ccc(Cl)cc1 C(=O)(C1=CC(C)CC1)NCC(C1CC1)NC(Cc1cc(C)sc1C)=O Cc1cc(CCC(=O)NCC2CCN(C(c3cc[nH]c(=N)c3)=O)C2)ccc1Cl CCC(CCC(=O)NCc1ncnn1C)NC(=O)C=C(C)C(C)(C)C C1(CNC(CC(C)(C)F)=O)COCCN(C(=O)CCc2cncc(F)c2)C1 CN1CCOCC1CNC(=O)CC1CCCN(C(=O)COC2CCCCC2)C1 C(=O)(CC(C)(O)COC)N(C(CC)C)Cc1cc(C)cc(C)c1 Cc1cc(C)c(C(=O)N(C2CCN(C(=O)CC(C)F)C2)C)o1 C(c1ccccc1[N+](=O)[O-])=CC(N1C2CN(C(CC(CC)SC)=O)C(C2)C1)=O CN=c1[nH]c(=NC(C)c2nnnn2C)[nH]c(=NCC2(C)CC2(C)C)[nH]1 C(c1ncccc1C)=CC(=O)NC1C(NC(c2cccc(C)n2)=O)CCC1 C(=O)(C(C)(CC)CC)N(CCC(=O)NCCOC(C)(C)C)CC#C C1(CN(C(CCc2n(C)c(=O)on2)=O)C2CC2)CC2CCCC(C1)C2 C#Cc1ccc(C(N2CC3C(CNC(C4CC(OC)C4)=O)C3C2)=O)c(F)c1Cl Cc1cc(C=CC(=O)NC(C(C(C)C)NC)c2ccccc2)cc([N+](=O)[O-])c1O c1(C2(N3CCC(O)CC3)CC2)nc(N2CCCC(F)(F)C2)c2c(F)cccc2n1 c1(COC)cncc(NC2(c3nnnn3CC3CC3)CSCCSC2)c1 N1(C(c2cc(OC)ncc2)=O)CCN(C(c2c[nH]c(=N)o2)=O)C(C)C1C N1(C(C(CC2CCC2)NC(c2ccc(OC)o2)=O)=O)CCCN(C)CC1 c1(-c2cn(CC3CN(C(CC)=O)C3)nn2)ccccc1SC.C12CCCN1C2 C#CC1(CNC(c2nc3c(s2)CCC3)=O)CCN(C(=O)NC(C)(C)C)C1 N1(C(C(C(CC)CC)C)=O)C2CCCC1CC(Nc1ncnc(Cl)c1F)C2 C(=O)(C(C(C)C)C(C)C)NC1CCC(N(C(c2ccc(OC)cn2)=O)C)CC1 N1(C(c2ccc(OC)cc2)=O)CCC2(CC1)CC(NC(c1ccon1)=O)CCO2 N(C1CCc2cccnc21)C(=O)CC1COCCN1C(=O)C1CC1 Cc1cc(C(=O)NC2(CNC(=O)Cc3cn[nH]c3)CCCC2)c(F)cc1Br C1(NC(C(C(C)C)NC(C=CCCC(C)C)=O)=O)CCCCC1(F)F C1(NCCC(CC=C)(C)C)CCCC2(CC1)CC2 CC(C)(C)C(=O)NCC(=O)NC1C=CC(C(=O)NCCc2c[nH]nc2O)C1 c1(OCC(=O)N(C2CCN(CCC#N)C2)CC)cccc(C)c1 c1(CS(=O)(=O)NC2CCC(CC)C2)ccc(Cn2ccccc2=O)cc1 N1(c2nc(CC)nc(=N)[nH]2)CCC(NC(=O)C=CI)C2(CCC2)C1 c1(CC(N2CC(F)(CNC(CNC(C=C)=O)=O)C2)=O)ccc(C(F)F)cc1 CCC(C(=O)NCC12CC1CN(C(C1CCOCC1(C)C)=O)C2)C(C)(C)CC C(=O)(C(F)(F)C(F)(F)Cl)N1CC(COC(c2c(Cl)ccc(OCC)c2)=O)OCC1 N1(C(COC2(C)CCC2)=O)CCC(C)(C)C1CNC(c1cncnc1)=O C1(C(=O)NC(c2cn(C)nn2)CC)CCCC1CNC(c1cc(C(F)F)[nH]n1)=O C1(C(N2CC(CNC(c3nc(C(=O)OC)sc3)=O)C2)=O)CCCC2(CCOC2)O1 C1(C)(NC(C(CC)NC(=O)C(n2ccnc2C)C)=O)CCCCC1 N1(C(C2=CC(C)C2)=O)CCN(C(C2CCCCC2)=O)C(C2CCC2)C1 c1(C(=O)NC(CN(C(=O)C=CS(C)=O)C)(CO)CO)cc2ccccn2n1 C1(CN(C(C=CCCC)=O)C)COCCN1C(=O)Cc1cc(Br)cs1 N1(C(C(CC)NC(C)=O)=O)CC2(CCC(NCc3cccc4[nH]ncc34)C2)C1 c1(C(C(N2CCC(N(C(=O)C=Cc3ccsc3)CC)C2)=O)O)cccc(C)c1 O(NC(=O)C(CCN(C)C)NC(=O)C(n1ccnc1C)C)CC#C c1(C(=O)NCC2C(C)CN(C(=O)CNS(C)(=O)=O)C2)cnc2nc(O)ccc2c1 Cc1ccc(C(N2CC(=O)CC2C(N2CC(C(N)=O)C2)=O)=O)cc1O CC(CC(F)F)C(=O)NC(C)(C)C.C12(CC13CCC3)CN(C)Cc1cn(nn1)C2 c1(C(=O)NCC2CC(F)CN2C(c2cc3ccccc3[nH]2)=O)ccn2ccnc2n1 Cc1nc2cc(C(N3CC4CC4(CNC(=O)CCOC4CC4)C3)=O)ccc2n1C N1(CC(=O)NCC(CNC(c2cc(Br)co2)=O)OC)OC(C)(C)CC1=O n1(CC(N2C(C)CC(CNC(C3(n4ccnn4)CC3)=O)C2)=O)cc(F)ccc1=O C1(OC(=O)CCOC2CCOC2)CC=CCC1C(F)(F)F C1(CNC(c2nnn(C)c2N)=O)CC(NC(c2c(F)cccc2Cl)=O)C12CCC2 N1(c2n(CC)c(CC3CCCCC3)nn2)CCC2CCCC2C1 n12c(nnc1N)SCC2.C1(SCC)CCO1 c1(C(C)C)ncc(C(N2CCCC2CCNC(=O)CN2CCCC2C)=O)o1 N1(C(C2(C(C)(C)OC)CC2)=O)CCC2C(NC(c3ncc(C)cn3)=O)C2C1 N1(C(C(F)OC)=O)CC(NC(=O)CN(CC(=O)NC(C)C)C)C(O)C1 c1(CC(=O)N(C)CC2OCCN(C(C3C(C#C)C3(C)C)=O)C2)csc2nccn12 C(=O)(CCCC(=O)NCc1cn(CCOC)nn1)OC.C12(CCC1)C(=O)N2 C(=O)(CC(C)C(=O)NC(C)CCNC(=O)C(c1ncccc1OC)(F)F)NCC N1(C(CCC=C=C)=O)CCCCC(CNC(=O)COc2ccc(C(C)C)cc2)C1 c1(C(=O)NCC(CO)NC(C(CCC)C)=O)c[nH]c2ccc(F)cc12 c1(C(N2CCC(N3CC(CC)CC3=O)CC2)C(=O)NC(CC)(C)C)cccc(Br)n1 n1(CC(=O)NC(C(=O)NCC(COC)C)Cc2cn[nH]c2)c(O)nnc1O C1(C(C)(C)NC(CCSC)=O)CCCN(C(C2(C#N)CCCO2)=O)C1 CC(CCCCNC(=O)C(C1CCC1)C1CCC1)NC(=O)CSc1nncs1 Cc1ncccc1C=CC(=O)NCC1CC(NC(C23CC(C)(CO2)C3)=O)C1 C1(C(=O)NC2(C3N(C(CC4C(OC)COCC4)=O)CCC3)CC2)CC2(CCCC2)C1 N1(C(C2(F)CCN(C(CNC=O)=O)C2)=O)CCCC2OCCC12 c1(C(=O)NC2C(CNC(C#CC(C)(C)C)=O)CCC2)cncc2cccnc12 c1(OCC)ccc(CC(=O)NCC2(C)CCCN2C(c2nc(=O)n(C)[nH]2)=O)nc1 C1(CC(=O)NC(C(C)NC(C(C=C)(C)C)=O)CO)CC2(CCC2)CCO1 n1(CCC=C)nc(C2Cc3ccccc32)nc1-c1ccc(-c2nncn2C)nc1 C1(C(N(S(C)(=O)=O)C)=O)CCN(Cc2ccc(CF)cc2)CC1.C1CN1 C1(C(=O)NC(CNC(C(COCC)(C)C)=O)(C)C)CC12CC(C)(C)C2 C1(CC(=O)NC2(CNC(C3(CC)CCCCC3)=O)CCOC2)CCC(C)(C)CO1 C1(NC(CCCCCC)=O)CN(C(C2C(C)C2C)=O)C2(CCC2)C1 CS(=O)(=O)c1cscc1C(N1CC(NC(=O)CCCNC(N)=O)C2(CC2)C1)=O C(=O)(CCCCCN(C)CCC1CCCC(C)C1)OCCCC CC(CC(=O)N1CCCC1(C)CCC(=O)N(C)CC1(O)CCCC1)C(F)(F)F N1(C(c2cnn(C)c2Br)=O)CCC(CO)C(NC(c2cc[nH]c2)=O)C1 c1(C(N2CC(C(N(c3ccccn3)CC)=O)OC(C)C2)=O)ccc(C#N)c(C)c1 CN1CCN(C(C2CC(C)(C)CCO2)=O)C(C(=O)NCCC(C)(F)F)C1 CCCS(=O)(=O)CC(=O)N(C1CCN(C(CNc2cc(Cl)ccn2)=O)C1)C CC(O)C(C)(C)CNC(C1(CNC(c2ccn(C3CC3)n2)=O)CC1)=O c12ccc3c(c1)CN(CC3)C2=O.Cc1ccc(S(=O)(=O)N2CCN(C)CC2C)cc1 C1(NC(c2c(CC)nccn2)=O)CCN(C(=O)CCn2c(C)csc2=O)C12CC2 N1(C(c2cnn(CCCC)c2C)=O)CCC2CCCN(C(=O)C3CC3)C2C1 c1(C(=O)NCC(C2CCC2)NC(CC2CCN(C)C2)=O)ncccc1Cl C(c1ccc(C)cn1)=CC(=O)N(CCCOCCNC(CN(C1CC1)CC)=O)C c1(C2C(C(=O)NCCN(C(C3(CC#C)CC3)=O)CCOC)C2)ccc(OC)cc1 C1(CNC(CCN(CC)CC)=O)CN(C(c2snc(O)c2Cl)=O)CC1(F)F C1(NC(c2c(CC)onc2C)=O)CC2(C1)CN(C(=O)C(C)=C(C)C)C2 c1(C(=O)NCC2(OC)CCN(C(C34CC(C)C3C4)=O)C2)c[nH]c2nccc-2c1C CCS(=O)(=O)CCCNC(=O)CC1CN(C(=O)C(c2ccccc2)O)CCO1 c1(C(=O)NCC2C=CC(NC(C3CC(C)(C)OCC3)=O)C2)nnn2c1CCCC2 C1(NC(=O)CCC2CC2CC2CC2)CN(C(c2ccnc(S)c2)=O)CC2CCCC12 C1(N(C(=O)Cn2cnnc2)C)CCC(NC(=O)CC2CC2c2nc[nH]n2)CC1 CCC(C)CCC(O)CC(=O)N1CCCC2(C1)CN(C(=O)CSc1nncs1)C2 c1(NC(C2CC(OC)CN2Cc2cnc(Cl)cc2Br)=O)c(Cl)cc(Br)c(Cl)c1Br c1(OC)cc(OC)cc(N2CCC(C(=O)Nc3cccc(OC)c3)CC2)c1 N1(C(CCCCCC)=O)CCN(C(c2nccnc2C)=O)CC12CCC2 C(=O)(C1COc2ccc(Cl)cc21)NCCN(CCC)C(c1cnc[nH]1)=O CCCCC(C)CCC(=O)NCC(Cc1ccccc1)NC(C1C2COCC12)=O Cn1cc2ccc(C(=O)NC3C4CN(C(C56COC(C5)C(O)C6)=O)CC34)cc2n1 CC1Cc2ccc(Br)cc2CN1C(=O)C(C)(C)CS(N)(=O)=O N1(C(CC(C(=C)C)OCC)=O)CCCC2(CCN(C(c3sc(O)nc3O)=O)C2)C1 c1(CC(=O)NC2C(NC(C3C(C)OCCC3)=O)COC2)cc(Cl)ccc1Cl C(=O)(C(C)(C)C(F)F)NCCN(C(=O)CCCCCSC)CCC N1(C(C(c2c(C)cccc2)C)=O)CCN(C(=O)CC2(O)CCC2)CC1C(C)C C1(NC(=O)Cc2cccc(Cl)c2)CCC12CN(C(=O)CSC1CCOC1=O)C2 CCCS(=O)(=O)C(C)C(=O)N1CCC(CCN=c2ccc(C)n[nH]2)C1 C(=O)(NN1CCCC1C(N1CCCC1CO)=O)c1cccc(C)c1O C1(C(N2CCC(N(C(=O)C(O)COC)CCC)CC2)=O)CCOCC12CCC2 N(C(=NCCCCl)NCc1nc(Cl)cs1)C1CC(OCC)C1SC CC1(C)CCOC1CC(=O)NC(C(=O)NCCSCC1CCC1)c1ccoc1 C1(CNC(=O)C(O)C(F)(F)F)CCCC2CN(C(=O)C=Cc3ncc[nH]3)CC12 c1(C(=O)NC2C(NC(c3nccc(C)n3)=O)CS(=O)(=O)C2)c(F)ccc(O)c1F CC1=C(C(=O)NC(Cn2cccn2)C(=O)NCC2CC2c2ccoc2)CC1 c1(C(=O)NCC(CNC(c2ccc(COC)s2)=O)CO)sc(CO)nc1C N#CC1CNCC12CC(NC(=O)NNC(=O)C1CCOCC1)C2 C(=O)(C1=C(F)CN(C(c2cc(Cl)cs2)=O)CC1)N1CC2C(=O)C2C1 c1(CC(=O)OC)ccnc(N2CCC(CN(C(=O)CN3CCCCCC3)C)C2)n1 Cc1cc(C(=O)NCCOCCCN(C(=O)CC2(C)CC2F)C)cc(C)n1 c1(C(=O)NC2CN(C(C(CC(C)C)O)=O)CC2F)ccc2c(O)nnc(O)c2c1 c1(C(=O)OC(c2cccc(C(F)(F)F)c2)C2CC2)cc2ccccc2[nH]1 N1(C(c2cncc(Cl)c2)=O)CCC2(CNC(C34CCCC3CCC4)=O)CCCC12 N1(C(C(C)SCC)=O)CCC2(CCC2)C(NC(=O)C(C)CCc2ccccc2)C1 C1(C)(CNC(CSCC)=O)CN(C(c2c(-c3nccs3)noc2C)=O)CCO1 c1(CCC(=O)NC(C)C(C)(C)NC(C2CC2C2CCCO2)=O)cc(F)ccc1F N1(C(c2c(CC)csc2)=O)CC(NC(c2cnc(Cl)s2)=O)CC(O)C1 N1(C(N(CCN(C(=O)CN2CC3CC3C2)C(C)C)C)=O)CC2C=CC1C2 CC1=NOC(C(N2CCCC(CNC(C3CC(C(F)F)C3)=O)C2)=O)C1C c1(OCC2N(c3c(OC)cncn3)CCC2)cc(Br)c(C)nc1Cl c1(NC(c2ncc(OC)nc2)=O)cnc(Cl)cc1C(=O)Nc1cccc(O)c1Br N1(C(COC(C)C)=O)CC2(CCC(CNC(c3cc4cccnc4s3)=O)O2)C1 c1(C(N2CC3C(NC(=O)Cc4nc(C5CC5)n[nH]4)C3C2)=O)cncc(Cl)c1Cl C1(CCC)CN(C(c2nc(O)sc2C)=O)CC1NC(=O)CCOC1CCCCC1 c1(C(C)C)cn2c(nc1=O)CCN(N1CCSC(C(C)C)C1)CC2 CCC(C)CCC(=O)N1CCN(C(c2ccc(C)nc2O)=O)C(C(F)F)C1 N1(C(C2N(CC)CC2)=O)CCC(C)C1C(N1CC(C(C)(C)O)C1)=O CC(C)C(CC(=O)N(CC(C)N(C)C(c1cccc(C(N)=O)c1F)=O)C)C(C)C c1(CC(N2CC3CC(Nc4c(C#N)ccnn4)C3C2)=O)ccc2cccnc2c1 Cc1nn(CC(N2CCC(NC(c3coc(O)n3)=O)C(F)C2)=O)cc1[N+](=O)[O-] C(=O)(C1CCc2cc(Br)ccc21)N1CC(N(C(C2CCN(OC)CC2)=O)C)C1 c1(C(=O)NCC2C(C)CN(C(c3snc(O)c3Cl)=O)CC2)cnn2ccn(C)c12 Cc1c(Br)c(C(N2CCOCC2CNCc2cc(Br)nn2C)=O)nn1C c1(C(=O)NC2(CCNC(C=CCC)=O)CCC2)ccc(Br)cc1F C1(CNC(C(COCC)C)=O)CC2CCC(C1)N2C(c1cc(C)c(C)nn1)=O C1(O)(CN(C)C(c2cn[nH]c2)=O)CCCN(C(=O)C(F)(Cl)c2ccccc2)C1 C(CC(=O)N1CC(N(C)C)C1)N(CC=C)C(C)=O.C1=CC=C1CC CC1(C)CC(NCC2CN(c3ncc(F)cn3)C2)CCN(C(=O)CN=S(C)(C)=O)C1 C1(C(=O)NCC2(C)CCC2)C=CCN1C(c1nccs1)=O Cc1cnc(Cl)c(C(=O)NCC(C)NC(c2cccc(CCN(C)C)c2)=O)c1 N12CC(C)(C)CC1c1c(C)c(n[nH]1)C2.C1CCC(=O)N1.C(=O)O C(=O)(C(O)CC(C)C)NCC(CC)(CC)NC(C1CCN1S(C)(=O)=O)=O C1(NC(=O)CCc2ccccn2)C2CCN(C(c3ccc(=O)oc3)=O)C12 C(=O)(CC(C)CNC(c1nnnn1CCN1CCOCC1)CCC1CCC1)NC c1(C(=O)OC(C(=O)OCC)Cc2ccccc2)cncc(F)c1 C12(C(=O)NC3C(NC(=O)CCc4cc[nH]n4)CC3)CCCN1CCC2 N1CC(C)(C)CCC1CNC(C=C(COC)C)=O.C1(C(=O)NC)CN(C2CCC2)C1 N1(C(CCCc2nnc(C)n2C)=O)C2CCC1C(NC(c1c[nH]nc1C1CC1)=O)C2 C1(C(=O)NC2CCN(C(COCCC)=O)C2CC)CC2CCC(C1)C2O C(CCCCF)NC(C1(NC(COCC(=C)C)=O)CSC1)=O CCC(C)C(C(=O)NCC(N1CCSC(C)CC1)=O)N(C)C c1(C(CNC(CC(C)F)=O)NC(=O)C=CC2CCCC2)ccc(F)cc1F C=CCC(CNC(=O)C(c1cncn1C)OC)NC(c1cc(C(F)(F)F)[nH]n1)=O Cc1cc(S(=O)(=O)NC2CCc3ccc(Br)nc32)cc(C(=O)O)c1F Cc1nc(Br)ccc1C(N1CCOC(CNC(=O)Cc2cccc(C#N)c2)C1)=O c1(C(N2CC(CN(C(C3CC(C)OCC3)=O)C)C2)=O)cc(O)cc(C#N)c1 C1(CCNC(C2C(CC)OCC2)=O)CC(F)(F)CN1C(=O)CNC(=O)NC c1(C(C(N2C(C(C(=O)NCC(=O)N(C)C)(C)C)CCC2)=O)N)ccc(O)cc1 C1(NC(CCOCCOC)=O)CCN(Cc2nc(C)no2)C1 N1(C(c2nc(C)c(C)[nH]c2=O)=O)CC2CCC(Nc3cc(C(C)C)ncn3)C2C1 C=CC1CCCN(C(C2CN(C(=O)Cn3cnnc3O)CC2C)=O)C1 CC1CCc2nc(C(N3CC4CC4(CNC(C4(N(C)C)CC4)=O)C3)=O)cn2C1 C1(NC(=O)C(CC2CCCC2)C(C)C)C(C)(C)C(NC(=O)NC2(C)CC2)C1(C)C C(CC1=CCN(c2cc(C(F)F)ncn2)CC1)NC(Cc1ccc(C)cc1Br)=O Cc1cc(C(N2CC(NC(c3cccc(=S)n3O)=O)C(CO)C2)=O)cc(N)c1 n1(CC)nc(C)c(C(=O)NCC(CNC(=O)CCC(=O)OC)OC)c1Cl C(=O)(C(C)CCCC(C)=O)N1CCN(C(c2cc(CC)no2)=O)C(C(C)C)C1 Cc1coc(C(C)(C)C)c1C(=O)NCC1CCC(NC(c2cnnc(O)c2)=O)C1 C=CC(C)C(C)C(=O)NC1CCN(C(=O)C(C)=C2CC2)CC1 C1(C)(NC(COC(CC)CC)=O)CCN(CC2CC(NC(C)=O)C2)C1 C#CCCCCCC(=O)N1C2CCC1CN(C(C1CC1(c1ccccc1)C)=O)C2 c1(NCc2n(C)cnc2)ccc(NC(c2ccc(CO)cc2)=O)cc1F C1(CN=[N+]=[N-])COCCN1C(c1ccc(CNC(c2cc(Br)co2)=O)nc1)=O C1(CNC(C(c2ccc(C)cc2)(C)O)=O)CCCCCN1C(=O)C(O)CC(N)=O c1(C(C)C)cc(=NCC(C2CCCC2)NC(C2COC2)=O)[nH]cn1 C(C)(CO)(C(=O)NC1CCN(CCO)CC1)NC(c1c(C)[nH]cc1)=O C1(C)(COC)CCCC1NC(C12CC1CN(C(=O)C(C1CC1)C1CC1)C2)=O C(C(C(C)C)NC(C1CCN1C1CCCC1)=O)NC(CC1CC(OCC)C1)=O C12(C(=O)OC)CN(C(=O)CCSc3ccccn3)CC(CO)(C1)C2 N1(C(c2c(Cn3cc(C4C(C)(C)C4)nn3)cccc2)=O)CCC(O)C1(C)C c1(NC(c2cnn3c2OCC3)=O)c(Br)cc(Cl)cc1Br CC1(C)CC(NC(=O)CCn2cc[nH]c(=O)c2=O)CN1C(C1CCC1)=O N1(CCCC(=O)NCCCOCCNC(c2ccc(Cl)o2)=O)C(=O)CCC1=O CC(C)C(C)(C)C(=O)NCCSCC(=O)NC1CC1c1ccncc1 C(=O)(C(C)(C)C(N)=O)N1CCC(CN(C)C(c2cnn(CC(F)F)n2)=O)CC1 C1(C(=O)NC2CCCN(C(C3(c4ccccc4)CC3)=O)CC2)CC2C=CC1CC2 C1(F)(C(=O)NCCC2(C(N(CC)CC3CCCO3)=O)CC2)CCOC1 C1(CC(=O)NC(C)CCNC(=O)CC(C)n2cccn2)(OC)CCCC1 C12(CCNC(c3ncn(C)c3)=O)CCC(CC1)N(C(=O)C(F)C(F)(F)F)C2 N1(C(c2c(SC)csc2)=O)CC2CN(C(c3c(C(F)(F)F)ncn3O)=O)CCC12 N1(CC#N)CCN(C(=NCCC(CO)CO)NCC(c2ccc(Cl)cc2)O)CC1 c1(C(=O)NC2C(CNC(C3C(CC)OCCC3)=O)CCCC2)cc(O)nc(O)n1 c1(C(=O)NC(C2CCCC2)CNC(C(CC)C2CCC2)=O)cccc2nncn12 C1(C(=O)NCC=CC2CC2)CC2CCC1N2C(c1ncccc1F)=O c1(C(N(C)CC2CCN(C(CC)=O)C2)=O)ccc(Br)c(F)c1OC C1(CC)C(C(=O)OCC2(C(C)CCO)CCC2)CCN1C(=O)OC(C)(C)C CCC(O)CC(=O)N1CCCCC1CCNC(=O)C(c1ccc(C)o1)C Cc1cc(Cl)ccc1OCC(=O)NCC1(NC(c2occc2Cl)=O)CC1 c1(C(C(=O)NCC(C)(CO)NC(c2cc[nH]c(=N)c2)=O)O)ccc(Cl)cc1F N1(C(c2csc(C)c2)C(=O)NCCC)CCN(S(=O)(=O)N(C)CC(F)(F)F)CC1 C=CCN=C(NCc1csc(Cl)c1)NC1CCC(C#N)C1 N1(C(CN(CCC)C)=O)CC(NC(=O)C2=NOCC2)C2(CCS(=O)(=O)CC2)C1 c1(NC)ccc(O)c(F)c1.c1(OC)ccnc(N2CCC(CNC(C)C)CC2)n1 C(=O)(C(O)P(C)(C)=O)NCC1CC(NC(C(C(=O)OC)C)=O)C1 c1(NC(C2CCCCC2)(C#C)C)ccnc2[nH]c(C)nc12 C12(CNC(=O)OC(C)(C)C)CC(CN(C3CCN(CC(F)F)CC3)C1)C2 N1(C(CC2C(C)(C)CCO2)=O)CCC12CS(=O)(=O)C2 c1(OC)ccc(C(N2CSCC2C(=O)N(C2CC2)CC2COC2)=O)cc1C N1(CC)CCCC(C(=O)N(CC(C)CNC(C2CC2F)=O)C)C1 Cc1noc(C)c1CC(=O)NCC(=O)N(CCCNC(=O)CC1CC(F)(F)C1)C N1(Cc2ccc(CS(=O)(=O)NC)cc2)CCCC(C(=O)NC(C)C(=O)O)C1 N1(C(c2c(Cl)cccc2Cl)C(=O)NC(CC)(C)C)CCCCC(C)(F)C1 CCCCCCC(C)CC(=O)NCC1CN(C(=O)CSCC(F)F)CC1(C)C C1(NC(c2c(C)nc(CO)nc2)=O)CC2CN(C(=O)Cc3ccsc3)CC2C1 C1(C(=O)NCCN(C(C2CCC(OC)C2)=O)C(C)C)CCN(C)CC1 N1(C(c2cc(OCCOC)n[nH]2)=O)CC2CC(C)N(C(=O)C(CO)C3CC3)C2C1 Cc1ccnc(N(C2CCCN(C(c3ccncn3)=O)C2)C)n1 N1(C(c2c(C)[nH][nH]c2=N)=O)CCC(NC(=O)CN(C2CCCC2)C)C(CO)CC1 C1(C(=O)OC)COC(CCNC(=O)CC2CCN(C(c3cnc(C)o3)=O)C2)C1 N1(C(CC(c2ccc(C)cc2)C)=O)CCOCC(NC(C2CCS2(=O)=O)=O)C1 Cc1ccc2c(c1)S(=O)(=O)N2N.C(=O)(C(C)(C)C(=O)N(C)C)OCCSC.C(C)(C)N CC1C(C(=O)N(CC(O)CNC(c2ncn3c2CCC3)=O)C)OC2CCCCC12 N1(C(C2(CNC(=O)CCc3ccncc3)C(C)(C)C2)=O)CC2(CC=CC2)C1 N1(C(CC2C(CC)C2)=O)CC(CNC(=O)Cc2noc(C)c2C#N)C2(CCC2)C1 N1(C(COC(CC)C)=O)CC(NC(c2cc(SC)n(C)n2)=O)C(C)C1 Cc1ccc(C(F)(F)F)cc1C(=O)Nc1ccsc1C(=O)Nc1cn(C)nc1C N1(C(C(COC)COC)=O)CC(NC(=O)CCN(C)C)CC(C)C1 C1(C2CC2)(NC(c2cccc(CC)n2)=O)CCN(C(=O)Cc2ccc(F)cc2)C1 c1(NC2CCC(NC(C(C)(C)c3ccc(C(=O)O)s3)=O)C2)ncc([N+](=O)[O-])cc1F CC1CCCC(C)N1CCC(=O)NC(CNC(c1conc1C1CC1)=O)C1CC1 c1(C(N2C(CNC(C(CSC)O)=O)CC(O)C2)=O)cc(C)c(C)cc1Cl Cc1cc2nc(C)c(CCC(N3CCC4(CCC(O)C4)C3)=O)c(C)n2n1 C1(SC)CCC(C(=O)NCc2nc(CNC(=O)C=CC3CCC3)cs2)C1 C1(CCNC(=O)CSc2ccccc2)CCCCN1C(=O)CCCCSC1CC1 C(C(C)(C)CC(=O)NNC(=O)c1ccccc1Oc1ccccc1Cl)SC N1(C(CCCSC(C)(C)C)=O)CC(CNC(c2csnc2C2CC2)=O)C(O)C1 C1(C(=O)NC(CC(C)C)CNC(C2CC(C)OC(C)C2)=O)CCCC2(CCC2)C1 c1(C(N2CC(NC(c3cc(OC)no3)=O)C(O)C2)=O)cc(C)c(O)nn1 C1(F)(C(N2CC(O)(CNC(c3c(CC)nco3)=O)C2)=O)C2CCCCC12 CCC(C)(C(=O)N1CC(CN2CCN(C(C3CCCN3CC)=O)CC2)C1)C(N)=O C(=O)(C(C(F)(F)F)C(F)(F)F)N1CC(NC(c2c(CC)nc[nH]2)=O)C(C)C1 C(=O)(C1=C(C#N)CCC1)N(C(C(=O)NC1CC(O)(CO)C1)C1CC1)C c1(CNC(C2C(CC(C)C)C2)=O)cc(C(=O)NCC2CCC(=O)N2)cs1 C(CC(C)(C)C#N)(C(=O)c1ccc2cc1OCON2)N1C(CC)COC(C)(C)C1 N1(C(c2c(C)nc(C)o2)=O)CCCC2CN(C(C3CC(=C(F)F)C3)=O)CCC12 C1(NC(C(CC)(C)C)=O)CC2(C1)CC(NC(=O)C1=COCCC1)C2 C12(C(=O)NCC3CC(=O)N(C)C3=O)CCCC1N(C(=O)CCCC(C)(C)C)CC2 c1(OC(C(=O)NCC(CC)N(C)C(c2ocnc2C)=O)C)cccnc1 C(=O)(CC(CNC(C1(C#C)CCC1)=O)CC(C)C)N1C(C)(NC(C)=O)CC1 Cc1ccnc(NC(C)CCNC(c2ncn(C(C)C)n2)=O)n1 C1(CNC(C2=C(C)CC2)=O)CCN(C(c2c(C)nsc2C)=O)CC1C Cc1cc(C#N)cc(C(=O)N(C)CCC2CCN(C(=O)COCCCF)CC2)n1 N1(C(c2c(OC)ccnc2)=O)CC(NC(c2[nH]nnc2C2CC2)=O)CCC(O)C1 c1(C(N2C(C)C(NC(c3cnc(C(F)(F)F)nc3)=O)CC2)=O)cccc(Cl)c1Cl c1(C(N2CCC(NC(CC)=O)CC2)=O)csc(N=S(C)(C)=O)n1 c1(C(N2CCN(C(c3ccc(C)c(Cl)c3)=O)CC2C)=O)cn2cnnc2cn1 c1(NC)ccc(C(=O)NCC2COCCN(C(c3nncs3)=O)C2)c(Cl)c1 C1(C)(CC)C=C(C(=O)NC2CN(C(=O)C=CC=C(Cl)Cl)CC2C(F)F)C1 C(=O)(CCCCCCCCCO)NC1C=CCN(C(c2c[nH]c(=N)o2)=O)C1 NC1CCC=CCCC1C(N1CCCCC1C1CCOCC1)=O c1(C(=O)NCC(=O)NCC(=O)NCC(C)CN(C)C)ccc(Cl)cn1 C12(C(=O)NCC3C(C(N4CC(N(C)C)C(O)C4)=O)C3)CCC(C1)C2(C)C C(=O)(C(C(C)(C)NC(=O)C(C(C)F)OC)NC(c1ccc(CO)s1)=O)OC CC1=CCC(C(=O)NC2C=CCN(C(c3sc(C(C)(C)C)nc3C)=O)C2)CC1 Cn1c(COC(c2n[nH]c(C3CC3)c2Cl)=O)cc2ccsc12 N1(C(CCN(C(C)=O)C)=O)CCC2(CC(C(=O)NCc3c[nH]nc3C)CO2)C1 N1(C(C)=O)CC(OC(COC(c2nccc(C(F)F)n2)=O)=O)CCC1=O C1(NC(C2(N(C)C)CC2)=O)CN(C(=O)Cc2cccc(Cl)c2F)C2(CCCC2)C1 c1(NCC)ncccc1C(N1CCC1CNC(=O)C(C)CCc1ccc(F)cc1)=O CCC(CC(=O)NC(C(=O)N1CCC(O)(CN(C)C)C1)C(C)C)CC(C)C C12(C(N(C)CC3CCCC3(C)C)=O)COCC1CN(C(=O)CC1CC(F)(F)C1)C2 C1(COC)(NC(=O)C(C)c2ccsc2)CCN(C(=O)C(F)=C(C)C)C1 Cc1nc2ccc(C(=O)NC3C4CC5CN(C(c6cccs6)=O)C3C5C4)cc2s1 c1(OC)ccccc1CC(=O)N(C(C)CNC(=O)C(=CC1CCCN1C)C)C c1(N(CC(CC2CCCC2)C(=O)NCCCCN=[N+]=[N-])C(C)=O)ccc2c(c1)CC2 C1(CNC(C(CC)=CC)=O)CN(C(=O)CSc2ccccc2)CC12CCOCC2 c1(NCC(N2C(CNC(C3CN(CC(F)(F)F)C3)=O)C=CC2)=O)cncc(Cl)n1 C1(C)(C(N(CCC2CCN(C(C(C)(C)OC)=O)CC2)C)=O)CCN(C)C1=O Cc1cc2c[nH]nc2cc1C(N1CC(O)(CCNC(C2(C)CCOCC2)=O)C1)=O c1(C(=O)OC)cncnc1C(=O)N(Cc1ccc(C(F)(F)F)nc1)Cc1cscn1 C(=O)(C(O)CCCNC(=O)Cc1ccccc1C)NCCC(C(=O)OC)O c12ccc(nc1)CCNC2C.C1(C(=O)N(C)CO)CCC(O)C1.C(CO)OC Cc1sc(N)c(C(=O)N(CC(C)CNC(C2CC2C(C)(C)C)=O)C)c1C N1(C(C=CC(C)C)=O)CC2(C1)CN(C(=O)CN(C)C)C2.C1(O)CCN(CC#N)CC1 C1(NC(C=CSC)=O)CCC(NC(c2cncc(-c3ccncc3)c2)=O)CC1 C1(CNC(CC(C)SC)=O)CCN(C(=O)CN(C)Cc2ccc(C)cc2)C1(C)C C(C)(C(=O)NCC1CC1C(C)(F)F)(C1CCC1)NC(C(C)C1CCC1)=O C1(CNC(C=C(C)C)=O)CCN(C(=O)Cn2cc(C#N)cn2)C12CCC2 C1(C#N)(C(=O)NCC2(OC)CN(C(=O)CC3CC(C)(C)C3)C2)CC2(CCC2)C1 c1(C(=O)NCC(CNC(C(C)(CO)OC)=O)CO)nccc2ccsc12 C(CC(C(=O)NCCCNC(C)=O)NC(=O)C=CCOC)=CC CCC(CC)C(=O)NC1CCC(NC(=O)Cc2cnco2)CC1 C1(CNC(c2n(CC)ncc2)=O)CC(NC(=O)C(C)(C)C#N)CCO1 c1(C(=O)NC2CC(CCNC(C(CCC)NC(N)=O)=O)C2)ccn(CC)c(=O)c1 N#Cc1ccc(C(=O)NCC=CCNC(=O)CCc2cnc(C3CC3)o2)s1 C1(CNC(C(C)OC)=O)CCC(NC(C2(O)CC(c3ccccc3)C2)=O)C1 c12ocnc1C2.C(=O)(C(C)OC(C)=O)N(CCNC(C1CC1F)=O)CC c1(CC(=O)N(C2CCC(NC(=O)CCN(CCO)CCO)C2)C)ccccc1 c1(N(C(C(=O)NC(C2(CC)CC2)=O)CC)C)ccnnc1C.C1(C2CC2)CCCN1C N1(C(c2ccn(C)c2)=O)CCN(C(=O)CC2CCOC(C(C)C)C2)C2COCC12 N1(C(C=CC(=O)NCCC2CCCO2)=O)CCC(N2CCC2)C1 C1(C(c2nnnn2C2CC(F)(F)C2)(C)NC2(CC(C)C)CC2)CCN(C)C1 Cc1cccc2[nH]cc(CC(=O)N(C3CN(C(C4COC(=O)C4)=O)CC3O)C)c12 N1(C(Cc2cc(C)cc(C)c2)=O)CC(C(=O)N(CCF)C2CC2)CCC1(C)C c1(CN2CCCC(O)(CC)C2)ccccc1S(N)(=O)=O CCC(CC(=O)NC1CC(C(F)C(=O)N(CCC#N)C)C1)C1CCC1 C1(C(F)(F)F)(C(=O)NC(CNC(COCCC)=O)C)CCN(C)C1 CCC(C)CCCC(=O)N(C)CC1CCCN(C(C2(NC(C)C)CC2)=O)C1 C1(NC(C(C)Cc2ccco2)=O)CCCC2CN(C(=O)C(=O)C3CCCC3)CC12 CC1(C)C2CCC(C(=O)NC34CCCC3CN(C(=O)C3=CCOC3)C4)C1C2 c1(C(=O)NC(C(C)NC(C=C(C)c2ccco2)=O)(C)C)ccn2nccc2c1 N1(C(c2nc(C)oc2)=O)CCCC(C(C)C(N2CCC(F)(CO)C2)=O)C1 O=C(C(O)CC(F)(F)F)NC1(C(=O)NC2C=CC(CO)C2)CC(O)C1 C1(NC(C(CCC#C)O)=O)CN(C(C2(CC#C)CC2)=O)CCC1(C)C c1(C(=O)NC2CN(C(CC(C)F)=O)C(C)CC2)cc2ccccc2s1 c1(C(=O)NCC(CC)NC(CCCC(=C)C)=O)ccc2nc(O)n(C)c2c1 CN1C(=O)CCC1C(=O)NCCCNC(c1sccc1Br)=O c1(C(N2CC3(C2)CN(C(=O)CCC(F)F)CCO3)=O)ccc2ccccc2c1F C1(NC(c2c(C(=O)OCC)c[nH]c2)=O)CCCCC1NC(c1nnc(S)n1C)=O C(=O)(CC(C(F)F)NC(C1(CO)CC(F)C1)=O)N1C(C(C)O)CC1 C(=O)(CC1OCCc2ccsc21)NCCC(C)N(C(c1[nH]cc(C)c1)=O)C c1(CNC(c2cc[nH]n2)C)nc(-c2ccccc2)cc(O)n1 C1(CNC(C2CCC3(CC3)C2)=O)CN(C(=O)C2=COCC2)CCC12CCC2 c1(C(=O)NCCC2(NC(c3cc(F)c[nH]3)=O)CC2)ccc(-n2ccnc2)cc1 c1(CNC(CCC#CC)=O)cc2cc(Br)ccc2[nH]1.C(C)(C(=O)OC)SCC C(CNC(C1CC1F)=O)(CC(F)(F)F)NC(CC1(C)OCCO1)=O CN1CC(C(=O)NCC(C2CCCC2)NC(c2ccc(=O)oc2)=O)C(C(F)(F)F)C1 Cc1ccc(-c2nc(CCN(C)C)nn2CCc2ccccn2)c2cccnc12 C(C(C(=O)N1CCCC(C(C)C)CC1)C(C)C)NC(c1c(CC)ccs1)=O C1(C)(CNC(C(CC)N2CCCC2=O)=O)CCCN1C(c1n[nH]c(C)c1Cl)=O n1(CC)cc(C(=O)N(C2CCCN(C(=O)C=CC3CCC3)C2)CCO)c(CC)n1 Cc1cc(Cl)c(C)c(C(=O)NC2CN(C(=O)C(C)(C)CC(C)C)CC2C)c1N C1(CCNC(=O)C=CC2CCC2)CN(C(C2COC(=O)N2)=O)CCS1(=O)=O N1(CCCC(=O)N(c2c(C)cccc2)CC(=C)Cl)CCN(C(C)=O)C(C)C1.C(C)(=O)OCl C1(C(C2CCOC2)OC)CCC(C(=O)NCC(C(=O)OC)C)CC1 N1(Cc2c(OC)ccc(Br)c2F)CCC(F)(F)C(NC(c2nc(C)cs2)=O)C1 CC1CN(C(=O)CS(N)(=O)=O)CCCN1C(=O)Cc1ccc(C#N)cc1F C(C(F)(C(=O)NC1(CC(C)C)CC1)C(C)C)NC(c1cn(CC)nc1)=O Cc1cscc1C(=O)NCC(O)C(=O)NCCNS(C)(=O)=O Cc1c(F)cc(C(=O)NC2CCCN(C(=O)C(C3CCCCC3)O)C2)c(F)c1N C1(CNC(CNS(CC)(=O)=O)=O)(OC)CCN(C(C2COC(=O)O2)=O)C1 N1(c2cn(C)nc2)CC(C(N2CC(NC(=O)Cc3cccc(Cl)c3)C2)=O)CC1=O c1(C(N2C(CN(C(C3CC(C(C)=O)C3(C)C)=O)C)CCC2)=O)cccc(Cl)c1N N1(Cc2c(C)nn(CC)c2C)CCCC2(C1)OCCO2.C12CCCN(C1)C2=O S(=O)(=O)(CCC(=O)N1CC2CCC2(CCNC(C2CC=CC2)=O)C1)N(C)C CC1(NC(=O)CC=CCN)CCN(C(c2cccc(C3CNC(=O)C3)c2)=O)C1 C(CC(C)(C)C)(C(=O)N(CCCN(C)C)CCO)NC(C(C)S(C)(=O)=O)=O N1(C(c2cccc(C)c2)=O)CC(C(=O)NCc2ccncc2)CC(F)C1 C(=O)(CC1CCC(C)(C)c2ccccc21)N1CC(CC=C)(NC(=O)CC(C)O)C1 Cc1c(C(=O)NCCCNC(c2ccccn2)=O)sc2ccc([N+](=O)[O-])cc12 c1(C(N(C2CCN(C(=O)C=CCN3CCOCC3)C2)C)=O)ccc2nnnn2c1 C(=O)(C(C#N)C(C)(C)C)N1CCC(CC)C1C(=O)NC1(CO)CC(C)C1 C(=O)(C#CC1CCCCC1)NC(C(CC)C)C(=O)NCCOC1(C)CCCC1 C1(C(NOCCC(C)C)=O)(CNC(=O)CC2(C)CC2)CC12CCC2 Cc1ccc(CNC(C2(CNC(=O)CC(O)C3CC3)CCC2)=O)o1 C(C)(C(=O)NC1CC(N(C)C(C2CC2c2ccsc2)=O)C1)OCC C1(CC)CCC(C)N(C(=O)NC(c2n[nH]cc2CSC)C)C1 C1(NC(C(C(C)C)NC(C2C(C)C2C)=O)=O)CCC(C)(C)CC1 C1(OCC)CC2CN(C(c3ccc(CNC(c4ncccc4F)=O)o3)=O)CC12 c1(CCC(=O)Nc2ncc(C(=O)NC)nc2)cccc(Br)c1O C1(C(N2CC(NC(c3cscc3C(F)F)=O)C2)=O)CC2CCC1CC2 c1(C(N2CCC(CNC(C3CCC4(CCC4)C3)=O)C2)=O)c(Cl)ccc2c1OCO2 CN1CCC(CC(=O)NCC2C(CNC(c3nn[nH]c3Cl)=O)C2(F)F)CC1 CC(C(F)(F)C(F)(F)F)=CC(=O)NCC(C1CCCC1)NC(C1CC2CC1C2)=O c1(C(c2n(CCSC)nnn2)NCC2(C(N)=O)CC2)sc(Br)nc1Cl C1(C(=O)NCCc2cnn[nH]2)CC=CC(NC(c2sccc2F)=O)C1 C1(CCCNC(=O)CCOCCOC)CCCCN1C(=O)CCc1cncs1 c1(C(=O)NC2CC(C)(C)N(C(=O)CNS(=O)(=O)C3CC3)C2)cc(F)c(Cl)cc1F C(=O)(C(C)(C)C)N(C(CN(C(CCOCCOC)=O)C)C)C1CC1 c1(C(=O)NC(C2CCOC2)CNC(C(CC)=CC)=O)cnc(S)n1C1CC1 N1(C(c2c(C)nn(C)c2)=O)CCCC12CN(C(=O)Cc1ccc(Cl)cc1)C2 C1(CN(C(=O)CC2C=CCC2)C)CCCN(C(=O)C(F)(F)CN2CCCC2)C1 C(CC(C)(C)CC(=O)N1CC(C(=O)NCc2cccc(C)c2O)CC1(C)C)OC N1(C(CCC)=O)CCN(C(c2cc3cccnc3s2)=O)CC(O)C1 N1(C(C(C2CCCCC2)OCC)C(=O)NC2CC(F)(F)C2)CCN(C)CC1CC CCC(C)(CNC(C1C2CC3C(C2)C13)=O)C(=O)NCC(C(=O)OC)OCC c1(OC)ccc(C(N2CCOC(C(=O)OC(C)(C)C(F)(F)F)C2)=O)nn1 C1(C(=O)NC2C(CNC(CCNC(COC)=O)=O)C2)CCOCC12CCCCC2 N1(C(C23CCC(OC)C2C3)=O)CC2(CCCN(C(=O)C(C)C3CC3)C2)C1 C=CCCC(F)(F)C(=O)NC1CN(C(C2(N(C)C)CCC2)=O)CC1C N1(C(c2n(CC#C)ccc2)=O)CCCC(CC(=O)NC2(C(=O)OC)CC2)C1 Cc1cc(C(=O)NC2CCCC(CNC(=O)C(C)(C)C(N)=O)C2)cc(F)c1C C1(C(=O)NCCOCCCO)(NC(C2CCSC2)=O)CC(F)(F)C1 c1(N2CCC(C3CCN(C(=O)C(C)(C)N4CCC4)C3)CC2)ccc(C#N)nn1.CS(=O)C C(c1ccc(OC)c(O)c1)=CC(=O)NC1CC(C)(NC(C(C=C)O)=O)C1 CC(C)C(C)C(CNC(=O)Cc1c(Cl)cccc1Cl)NC(=O)CC1CC(=O)C1 c1(SCC)cc(C(N2CCCC2CNC(=O)C(=Cc2ccccc2)C)=O)ccn1 C1(OC)(CNC(c2cc(C)nc(C)n2)=O)CCN(C(=O)Cc2cn(C)nn2)CC1 c1(CN(C(c2nc(C)sc2)=O)C)ccc(CNC(c2ccnnc2)=O)cc1 C(c1ccc(F)cc1)=CC(=O)NCCC(C)NC(c1onc(CC)c1C)=O n1(CC(=O)OC)nnc(CNC(c2nncn2C(C)C)c2nnnn2C)n1 N1(CC)CC2(CN(C(=O)CC(CNC(=O)CC(C)n3ccnc3)C3CCC3)C2)C1 C1(NC(C(c2ccccc2)OCC)=O)CCN(C(=O)CC23CCC(CC2)C3)CC1 C1(C(=O)NCC2N(C(CCc3onc(CC)n3)=O)CCCC2)CCCS(=O)(=O)N1 N1(C(c2c(C)c(F)ccc2)=O)CC2(CCCC2NC(c2cc(=O)n(C)cn2)=O)C1 N1(C(=O)NC2CC3CCC2O3)CC2CCC(C(F)F)(C2)C1 CC1(C)OCC(C)(CNC(=O)C(=O)NC2CCOC(=O)N2)O1 C1(CC)CN(C(c2cc(C)oc2COC)=O)CC1C(N1CC(N(C)C)C(C)C1)=O c1(NC(CC)CNC(=O)C=Cc2cccnc2C)cc(S(C)(=O)=O)ncn1 c1(C(=O)NC2CC(C)N(CC3Cc4ccccc4O3)CC2)ccccc1[N+](=O)[O-] c1(C(=O)NCCc2ccc(I)cc2)cc(S(=O)(=O)N2CCCC2)ccc1F CCCCN(CC)N1CCC(C(=O)NCC(=O)OC)CC1 N1(C(C2CN(C)C(=O)N2)=O)CC2OCCN(C(C3CCCCN3N=O)=O)C2C1 S(=O)(=O)(c1cc(Br)ccc1Cl)NC1CCN(C(CC(C)(C)C)=O)C1 CCC(CC)CC(=O)NC1CC(C)N(C(c2ccc(C)cc2)=O)C1 C1(C(N2CCC(O)C(F)(F)C2)=O)CCn2c(O)nnc2C1 N1(C(c2c(C)nc(C)s2)=O)CCOC(C(=O)Nc2cccc(CO)c2C)CC1 C1(C(=O)OC)CC(OC(C)C(N2CC(F)(OC)C2)=O)CN1C(=O)OC(C)(C)C C=C(CC)CN=c1[nH]c(=NCCCc2nccs2)[nH]c2c1CCC2 C1(C(=O)NCC2CC(C)N2C(=O)CCC2CCCCC2)C2CN(C)CC12 c1(C(N2C3C(NC(CCC(=C)C)=O)CC(C3)C2)=O)cc(=O)c2cc(O)ccc2o1 C1(O)(C(=O)NCC(C(=O)N(CC(O)C2CC2)C)N(C)C)CCOCC1 Cc1cnn(C)c1C(N1CC(NC(C2(C)CC2(C)C)=O)C(F)C1)=O C(=O)(C(C)(F)C(=O)N1CCC(CN(C(=O)Cc2ccnc(F)c2F)C)C1)OC c1(C(=O)NC2C(NC(c3cn(CCOC)nn3)=O)CCC2)cccc(OCCF)c1 CCC(F)(F)CC(=O)N1CCCC(C)(NC(c2cc(C)nc(O)n2)=O)C1 CC1C=C(C(=O)N(C)CC2(O)CCN(C(=O)C(c3ccc(F)cc3)F)C2)C1 C1(C(=O)NC(C)Cc2ncco2)C(C)OCCN1C(c1sccc1C#N)=O C1(CC(=O)NCC2CCCCS2)CN(C(=O)CC2CSC2)CC12CC2 c1(C(=O)OC)ccc(C)nc1NC(C1CC(NC(c2csnn2)=O)C1)=O C(=O)(CC1=CCOCC1)N(C1CCN(C(C(CC(=C)C)C)=O)CC1)CC1CC1 Cc1[nH]nc(Cl)c1C(=O)NCC(C)CNC(=O)CCC=CBr C1(NC(CN(S(C)(=O)=O)C)=O)CCOCC1C(=O)NCc1ccnnc1 N1(C(C(CC=C)NC(=O)CCC2CCCC2)=O)CC(F)(F)C(F)(F)C1 c1(C(=O)NCC(CCOC)NC(c2csnc2Cl)=O)c(C)cc(C)oc1=O C1(C(=O)NC2(CF)CCN(C(C=Cc3scc(C)n3)=O)C2)CCCS(=O)(=O)C1 N1(C(CSCCCC)=O)CCC(CCOC)(NC(=O)C(O)CSC)CC1 C1(C(=O)NCC2(F)COCCN(C(C(CC)(C)C)=O)C2)Cc2cc(Cl)ccc2O1 C12(CNC(c3ccc(C)cn3)=O)CCCC(CN1C(c1sc(C)c(C)c1C)=O)C2 C1(C(N2CCCN(C(CN3CCN(C)CC3)=O)CC2)=O)C(O)C(=O)N(C)C1C N1(C(=O)C#CC2CC2)CCC2(CCN(C(c3cc4cnccc4o3)=O)C2)C1 C1CC2CCCCC(C1)C1(CCOCC)OCC(C1)N2 c1(C(=O)NCc2cc(C(N3C(C)CCC3)=O)no2)cc(N)cc(F)c1 c1(C(=O)NC2CC(NC(c3c(N)ccc(C)c3)=O)C2)noc2cc(F)ccc12 c1(CNCc2ccc(F)cc2I)cn2cccc(F)c2n1 Cc1ccc([N+](=O)[O-])c(S(=O)(=O)NC(C2C(O)C(=O)N(C)C2C)=O)c1C N1(C(c2c(C)cno2)=O)CCN(C(C2CCc3nccn3C2)=O)C2CCC12 C=CCC(CC(C)C)C(=O)NC(C)(CNC(C1CCN(C(=O)CO)CC1)=O)CC c1(C(=O)NCc2ccc(C)o2)c(Cl)ccc(Cl)c1Cl.N12CC3CC3(C1)C2 C1(NC(C(C=C)O)=O)CCN(C(c2ccc(C(C)=O)c(C)c2)=O)C(C)C1 N1(C(CC2(NC(C3C(C)CCO3)=O)CCC2)=O)CCCCC(CO)C1 C#CC(C)(C)C(=O)N1CCCC(N(C)C(c2cccc(CS(C)=O)c2)=O)C1 N1(C(C2=C(C)CCCC2)=O)CC2(CCCCN(C(=O)C=Cc3ccccc3)C2)C1 N1(C(c2cccc(OC)c2F)=O)CC2CCCC2(NC(c2cnco2)=O)C1 C(CNC(=O)CCCCN(C)C)(C(C)C(C)C)NC(c1nc(C)c(C)s1)=O C1(CNC(C=CC)=O)CC2CCC1N2C(c1cccc(CO)c1)=O CC1(C)CCCC(CO)(NCCNC(c2cc(Cl)cc(Cl)c2)=O)C1.O(N)C c1(C(N2CC(CNC(C(F)=CC)=O)N(C)CC2)=O)cc2ccccc2s1 C1(C(N(CC(CNC(CCCC=C)=O)C)C)=O)CC(C)(C)CCO1 CC1CCC(Cl)=C(C(=O)NC(C)(CNC(=O)CCS(=O)(=O)N2CCCC2)CO)C1 c1(-c2nc(CC)nn2CC2CCCOC2)ccc2n1CCNC2 c1(CN2CCC(CC(=O)OC)C2C)cnc(F)c(F)c1 C1(NC(C(CC2CN(C(c3c(C#N)scc3)=O)C2)F)=O)CCN2CCC1C2 C1(NC(Cn2c(C)cnc2)=O)CN(C(=O)C(c2ccccc2)C)C2CCCCC12 C1(C(=O)NCC2CCN(C(COCC=C)=O)C2)C2CCC1(c1cscn1)C2 C1(CN(CCc2cccs2)CC)CCC2C(CC1)C2(F)F Cc1cn2cccc(C(N3CC4CC4(CNC(C4COC(=O)O4)=O)C3)=O)c2n1 c1(C(N2CCC(CNC(C(C)N(CC)CC)=O)C2)=O)sc(N(C)C)nc1Cl N1(Cc2ccc(OC)nc2Br)CC2(CN(C(=O)CSC(C)=O)CC2CO)C1 N1(C(Cc2ccn(C)n2)=O)CCCC(C(=O)NCCn2cccn2)CC1 N1(C(C(CCCC)N(C)C)=O)CC2CC(C(N3CC(=O)NC4(CC4)C3)=O)C(C2)C1 C1(C(=O)NCC2(C(=O)Nc3c(C)cc(Br)cn3)CC2)CCc2nc[nH]c2C1 C1(C2(O)CCN(C)CC2)(C(=O)NC23C(CN(C(C(CC(C)C)O)=O)C2)CC3)CC1 C1(C(N2CC(CNC(=O)CC3CCCC34CC4)C2)=O)CCC2(CCCCC2)C1 N1(C(C(C=C)(C)O)=O)CCC(F)(F)C(CNC(=O)CCCc2ncco2)C1 c1(C(=O)N(CC2C(C(=O)NCc3c(C)nsc3)CCO2)Br)ccc(F)cc1F.C1CC1 Cc1noc(C)c1CC(=O)NC1CCC(NC(=O)C(O)Cc2cnn(C)c2)C1 c1(C(N2CCC2c2cc(F)cc(Cl)c2)=O)nccc(Cl)c1F C=C=CCCC(=O)N(c1ccnc(C2(NCC(=O)OC)CC2)c1)Cc1cscn1 Cc1nn(C)c(C)c1C(N1CCOC(CNC(c2ccc(I)cc2Br)=O)C1)=O C(=O)(C1=CCCOC1)N1C(C)(C(N2CCN(C(C)=O)CC2)=O)CC1 c1(C(=O)NC(CNC(CCC#N)=O)CO)cnc2ccsc2c1 S(=O)(=O)(c1cc2ccccc2s1)NCC1N(Cc2cc(C)cc(Br)c2)CCC1 C1(C(=O)NCCCn2cnnn2)CN(C(C2CCCOC2)=O)CC12CC2 c1(C(=O)NCC2N(C(C3(OC)CCC3)=O)CCC2)ccc(C)cc1[N+](=O)[O-] N1(C(CCC)=O)CCC2(C1)CN(C(c1cc(Cl)cc(Cl)n1)=O)CCO2 C1(CCC(=O)N(CC#CC)C)CCCCN(C(=O)C(C)(C)CO)C1 N12CCC(C13CCC3)C2=O.c1(OC(C)Cn2cnc(=N)[nH]2)ccc(F)cc1 c1(NC2CCC(NS(C)(=O)=O)CC2)nc2cc(OC(F)(F)F)ccc2o1 C=C(C)CN=C(NCC1COC1)NCC1CC=CCC1 C1(C(=O)NC(Cc2cnc[nH]2)CO)(SC)CCOCC1 c1(C(=O)Nc2ccc(NC(CCNC(N)=O)=O)nc2)cc(Cl)c(Cl)cc1O C1(NCc2nc(C)cc(OC)n2)CC2CCCCN2C1=O C1(NC(c2cc(OCC)ns2)=O)CCN(CC(=O)O)CC1 C1(CNC(C(C)NC(CC)=O)=O)CN(C(=O)CCOC(C)C)CC1O c1(CNC(COC2(C#C)COC2)=O)cc(C(=O)N(CC(F)F)CC(C)O)n(C)n1 N1(C(C2CCC2(F)F)=O)CC2CC(C1)N2C(=O)CC1CCCC12CC2 c1(CC)cc(C(=O)NCC(C(C)C)NC(=O)CSCCOC)ncn1 C1(OC)CC(CNC(C23CC(C(F)(F)F)(CO2)C3)=O)N(C(c2ccoc2)=O)C1 c1(CNC(C(C)(C)SC)=O)ccc2c(c1)CCN(C(=O)CCC(C)N(C)C)C2 c1(C(C(=O)NC)N(CC(N2CCC(F)(F)CC2)(C)C)C)cc(C#N)ccc1F N1(C(=O)CCn2ccnc2)CCC2CN(C(C3CCCCS3)=O)CC2C1 N1(C(C2CC(OC)C2)=O)CCN(C(=O)CC(C)c2ccncc2)CC1CC(F)F C1(C(N2CCCCC(NC(c3ccc(Cl)cn3)=O)C2)=O)CCCC12CCOCC2 c1(OC)nc(C)nc(Cl)c1NC(C1CCCN(C(c2oc(C)cc2C)=O)C1)=O C1(C(=O)NC2C(NC(C=CC(CC)C)=O)CCC2)CC2C=CC1C21CC1 C1(N(CC(=O)Nc2scc(C(=O)OCC)n2)C)CCCS(=O)(=O)C1 c1(C(N(CC(CNC(CC(C)(C)OC)=O)C)C)=O)ccc(C)c(F)c1Br C1(CC)(CC)CN(C(=O)CCCCCNC(C2CC23CCCC3)=O)CCO1 N1(C(C=CC(=O)OC)=O)CCC2(NC(c3cc(F)c(OC)c(Cl)c3)=O)CCCC12 c1(C(=O)NCC2CC(NC(C(CCC)CC)=O)C2)cc(C)c(C)nc1C N1(C(C2CCC(C(C)C)NC2=O)=O)CCCC2(CCN(C(C3(CO)COC3)=O)C2)C1 Cc1nc(CO)oc1C(=O)NCC(N1CCN(C(C2CCC(=O)N2)=O)CC1)C N1(C(CCOC2CN(C(C(CCCCC)O)=O)C2)=O)CCC2(CNC(=O)C2)C1 CC(CC(=O)N1CC(C2CN(C(=O)Cc3c(F)cccc3F)C2)C1)P(C)(C)=O c1(C(N(CC(C)NC(c2cc(SC)oc2)=O)C)=O)onc(C)c1C Cc1nn2cc(C(N3CCC(CNC(=O)C4=CC(C)CC4)CC3)=O)nc2s1 c1(C(=O)OC)cnccc1C(=O)NCC(O)CNC(C1NC(=O)OC1C)=O c1(OC)ccc(CNC(N2CCC(c3nc(=O)o[nH]3)C2)=O)c(C(F)F)c1OC CC(C)CC(O)CC(=O)NC1C(C(=O)NC(C)C(=O)N2CCCC2)C1(C)C N1(C(C2CCC(O)CC2)=O)CCC2CN(C(C3CC(C(F)(F)F)C3)=O)CC12 N1(C(c2ncc(CC)cn2)=O)CCC12CN(C(=O)C(C1CCOCC1)C)C2 N1(c2ccc(C(=O)NC(CN(C(C(F)=C(C)C)=O)C)C)cc2)CC(C)OC(C)C1 N1(C(c2cc(C(F)F)[nH]n2)=O)CCC(n2cc(-c3ccccc3)nn2)C(O)C1 c1(N(CCCS(C)(=O)=O)C)nnc(-c2ccc[nH]2)n1CC1CCCOC1 c1(C(=O)NC2C(CNC(C(C)SCCCC)=O)CC2)cc(N)c(Cl)c(O)c1 CCC(C(=O)NC(C)CNC(=O)NC(C)C)NC(c1csnn1)=O N1(C(C(CC)SC)=O)CC(F)(F)CC1CNC(C12CC(C1)S(=O)(=O)C2)=O N1(Cc2n(C)ccn2)CCC2(CC1)CC(NC(c1csc(C3CC3)n1)=O)CO2 c1(C(N2CC(O)(CNC(CCCN(C(C)=O)C)=O)C2)=O)cc(C#N)ccc1Cl C1(CC(=O)O)CCCN(C(C2(CN(CC(F)F)C3CC3)CCCCC2)=O)CC1 C12CC13CCN(CC3)CC(=O)N2.c1(SCC)ccc(OC)c(OC)c1.N(CC)(CC)C c1(C(=O)NCC(CNC(C(=O)NCC)=O)O)ccc(Cl)nc1.C1CO1 c1(C(=O)NC2CCN(C(c3c(C)n[nH]c3)=O)C2)cccc2c1COCCN2 N1(C(C(C=C)(F)F)=O)CC2(NC(=O)CCNC(=O)OCC)CCC1C2 c1(C(=O)NC2CCC(CNC(C(CCSC)O)=O)CC2)ccnn2ccnc12 c1(C(N2C(CN(C(c3c(CC)noc3C)=O)C)CCC2)=O)cc(C)nnc1O O(NC(=O)C(c1cccnc1)NC(c1ccc(O)cn1)=O)CCOCC#C C1(CC)CN(C(c2nnsc2C)=O)CCC1NC(c1ccc(C)cc1C)=O C1(C(=O)NCCN(C(=O)C=CC2(C)COC2)C)(COC(C)C)CCOC1 C1(F)(C(=O)NC(CC)COC)CCCN(C(=O)C(C)OCC(C)C)C1 c1(C(=O)NC2(CNC(C3C(C)(C(=O)OC)C3)=O)CCOC2)ccnnc1O N1(C(C(C=CCCC)O)=O)CCOCC1CN(C(=O)CN1CCOCC1=O)C c1(C(=O)NCC(CCCC)NC(C2(CCC=C)CC2)=O)ccc2c(c1)CN(C)C2 CS(C)(=O)=NS(=O)(=O)CCNC(c1nnnn1CC1CCOC1)c1csnn1 C1(CNC(=O)NC2C(OCOCC)CCCC2)CC(C)OC(C)C1 Cc1c[nH]c(=NCc2ccn(C3CC3(F)F)n2)cn1 C1(CCNC(C2CCC=CCC2)=O)CCCN(C(c2coc(O)n2)=O)CC1 N1(C(CC(C)C)=O)CCC2(CC(NC(c3cnc(-c4cnn(C)c4)s3)=O)CO2)C1 c1(CC(=O)N(CC(CNC(C2(C#C)CCCC2)=O)O)C)cnc2c(=O)[nH]ccn12 C(=O)(C1=CCC2(COC2)OC1)NCC1(C)CCN(C(=O)CC2CCCOC2)C1 C(CC(C)C(=O)NCc1cc(C(=O)OC)co1)OC.C12CCCC1C(=O)N2 N1(C(c2c(COC)scc2)=O)CC(C)CN(C(c2cncc(OC)c2)=O)C(C)C1 CC1CCN(S(=O)(=O)CC(=O)NCC=CCNC(C2CC=CCC2)=O)CC1 N1(C(c2c(C)scn2)=O)C2CCC1CN(C(C1(C)CC1Br)=O)C2 c1(C(=O)NC2COCCN(C(C(CN(C)C)(C)C)=O)C2)ccc2nccnc2n1 c1(C(=O)NC2C(F)(F)CCN(C(C3=C(C)CC3)=O)C2)ccc2nccc(Cl)c2c1 c1(C(=O)NCC2N(C(c3cccc(OC)n3)=O)CC3CC32)cnc2nc(C)oc2c1 CN1CC=C(CC(=O)NCC2CC(F)(CNC(c3nc(C4CC4)cs3)=O)C2)CC1 C(=O)(C(C)(C)CS(N)(=O)=O)NCC(CC)NC(c1ccc(CO)c(Cl)c1)=O C(c1cccnc1)=CC(=O)N(C1CCCCC1)CCNC(c1cc(SC)oc1)=O c1(C(=O)NCCCCCNC(c2[nH]c(=NC)sc2)=O)ccc2c(c1)S(=O)(=O)NC2 CC(CC(=O)NCCOCCN(C)C(C1CC(C)(C)CCO1)=O)C(F)(F)F c1(CC(=O)NCCCCCNC(c2c(CC)noc2C)=O)nc2ncccn2n1 c1(-c2nnc(NC3CC(c4cn(C)nc4)SCC3)o2)cc(Cl)ccc1Br C(CNC(c1ccc(C(F)F)s1)=O)(CC(F)(F)F)NC(c1c(C)ncs1)=O c1(CC)ccc(O)c(C(=O)NC2(CNC(C3CCCCC3F)=O)CCCCC2)c1 C(=O)(C1=CC2(CCN(C(=O)CC3CCCC3O)C2)C1)NCC(CCC)CCO c1(OCC)ccccc1C(=O)NCC1(C)CCCN1C(=O)CC(C)n1cccc1 c1(C(=O)NCC(C2CC2)NC(CCSCCCC)=O)ccc(-c2csc(C)n2)s1 c1(C(N2CC(C)(C(=O)OC)C2)=O)ccc(CNC(C2CNC(=O)O2)=O)nc1 c1(C(=O)NC(C2C(NC(COc3cn(CC)nc3)=O)C2)=O)cc(SC)ccc1C C1(C(=O)NC2C(c3ccc(OC)cc3)C2)CCNC2(CCC2)C1 O=C(C(O)C1=CCCCC1)N1CCCC(C(=O)NC2CCCN(O)C2=O)C1 Cn1cccc(C(=O)NC2CCC(CCNC(=O)C(C)(C)N=[N+]=[N-])C2)c1=O C(=O)(C(C#N)CC)N(C(C)C(N1CCOCC1COC)=O)CC N1(C(c2c(C)ccnc2)=O)CCC2(CC1)CC2NC(c1c(F)cccc1Cl)=O C1CC(C)(C)CC(=O)Nc2cn1nn2.c1(CN2CCC(NC)C2)cccc(Cl)c1 C1(C2CCN(C(c3cc(F)c(C)cc3O)=O)C2)(NC(C(=CC2CCCC2)C)=O)CC1 c1(C(=O)NC23C(CN(C(CSCC#C)=O)C2)CCC3)c[nH]c2cccc(Cl)c12 Cc1cccc(C)c1CNC(=O)C(N1CCCCC1c1cnc(=N)[nH]c1)=O c1(C(=O)NC(c2nccc(O)n2)C)coc2c1COC2 N1(C(C2(C(=O)NC)CCC2)=O)CCCOC(CNC(=O)Cn2cnnc2)C1 N1(C(C2CCC=CO2)=O)CCOCC12COC2 C(=O)(C(C)C(O)C(C)C)N1C(C)CCC(C(=O)NC(c2ncc[nH]2)CC)C1 N1(C(c2c(CC)n(C)nn2)=O)CC2CCC2(CNC(=O)C(F)=C2CCC2)C1 c1(CCC(N2CCC(CC(=O)N(C(C(=O)OCC)C)C)C2)=O)cccc(O)c1 c1(C(=O)NCC(CNC(CC)=O)(C)O)[nH]c2ccc(C(C)C)cc2c1C CC(C(=O)NCC1CCN(C(=O)CN2CC3C=CC2C3)CC1)C(F)F Cc1cccc(C)c1N=c1[nH]nc(CN2CCC(CN)CC2)s1 C1(C)(NC(C2(F)CCN(C(COCC(C)C)=O)C2)=O)CCC(=O)NC1=O CC(C)CCCCN(C(NOC(=O)C(C)COc1ccccc1)=O)C N1(C(c2ccc(Cl)nc2O)=O)CCn2c(Cc3ccccc3)nnc2C1 c1(C(=O)NC2(CCNC(C(CC)OCC)=O)CC2)ccc(O)c2ccccc12 c1(OC)nc(C)ncc1C(=O)NC1CCN(C(C2CC(C)(F)C2)=O)C1C C1(NC(COCC(C)C)=O)CCOC(C2CCN(C(=O)CP(C)(C)=O)CC2)C1 N1(C(C(C=C)(C)CC)=O)CC2CCCC(NC(=O)C(C)(C)N3CCCCC3)C2C1 C(C)(CNC(=O)Cc1ccn(C)n1)(CO)NC(CN1C(C)CC1)=O N1(C(C2C3CC2N(C(c2c(Cl)cccc2Cl)=O)C3)=O)CCC2(CCCO2)C1 Cc1ccc(Cl)cc1C(=O)NCCCCC(CO)NC(c1coc(C(F)F)c1)=O Cc1cc(C(=O)NCC2(NC(c3cnc(O)n(C)c3=O)=O)CCC2)ncc1N C#CCC(C(=O)OC)NCCC1CC(C(=O)O)C1 C(C)(CCC(=O)NCC=C1CCN(C(=O)COc2ccsc2Cl)CC1)OC C1(CNC(c2cc(CCC)n(C)n2)=O)(NC(=O)C(CC)OCC)CCCCCC1 c1(NC(c2nc(C(=O)NC3CC3(F)F)sc2)=O)ccnc(SCCO)c1 C(c1ccc(O)c(OC)c1)=CC(=O)N(C(CNC(C(CC)(C)CO)=O)C)CC N1(C(C(CCC)N(C)C)=O)CCN(C(C23CC(CC(C)C)(C2)C3)=O)C2(CC2)C1 N1(C(CC(CC)SC)=O)CCC(C(N2CCCC(OC)C2)=O)C(C)C1 Cc1c(C)c(CC(=O)NCCN2CC=CCC2)c(C)c(C)c1Br c1(C(N(C2CCN(C(C34CCC3C4)=O)C2)C)=O)cnc2ccc(Br)cc2c1 CCCC(C)CC(=O)NCCN(C)C(c1cnccc1N(C)C)=O c1(C(N2CCC(C(C)(C)C)(CNC(C(C)SCC)=O)C2)=O)cc2c([nH]1)CCOC2 C=CC(C)(C)CC(=O)NC(CCSC)C(=O)NCc1csnc1OC c1(C(N(CCCNC(C2CC(OC)C2)=O)C2CC2)=O)cccc(OC(F)F)n1 C1(CNC(C2CC(OC)CN2C(c2ccnn2C2CC2)=O)=O)CCCN(C)C1=O C1(NC(C2CCCCO2)C(=O)OCC)CNC(=O)CN1C(=O)OC(C)(C)C C(=O)(C1=CCS(=O)(=O)C1)NC1CCCN(C(C2NC(=O)OCC2)=O)CC1 C(=O)(C(C)C(C)C)N(CCCC=CC(NOCC(=C)C)=O)C1CC1 N1(C(c2ccc(C(C)O)cc2)=O)CC(N(C(=O)CCc2nc[nH]n2)C)C2(CC2)C1 C(=O)(C(C)(C)C(=O)OC(C)(C)C)N1CC(N(C)C2CC2)C(O)C1 C1(CN(C(C2(OC)CC2)=O)C)CCCCN1C(=O)CCOc1cccc(C)c1 N1(C(C2(NC(C)=O)CCCC2)=O)CCC(NC(c2ccoc2)=O)C(O)C1 N1(C(CCC2(C)N=N2)=O)CC2CC(C(=O)NCCCC(F)F)C(C2)C1 N1(C(c2c(CNC(C3CC=C(C)CC3)=O)nccc2)=O)CCC2(CCO2)C1 c1(C(=O)OC(c2ccc(OC)cc2)COC)cc(O)nc(Cl)c1C#N C1(C(N(C(CSC)C)C)=O)CC(O)CN1C(c1cnncc1O)=O C1(NC(COC)=O)CCN(c2ccnc(C(C)(C)C)n2)CC1O N1(C(CC(N2CCC3(CN(C(C=NOC)=O)C3)C2)=O)C)CCc2ccccc2C1 N1(C(CC(CC)C2CC2)=O)CC(CO)C2(C1)CN(C(c1ccc(O)c(F)c1)=O)C2 C(=O)(C(CO)C(C)(C)C)N1CC(CN(C(=O)C=Cc2cnccn2)C)OCC1 N1(C(C(C)N(C(C(=O)NCCC)=O)C)=O)CCCC(C)C1CO c1(C(N2CC(C)(C(=O)OC(C)(C)C)C2)=O)cc2cc(Br)sc2[nH]1 c1(NC(C(=O)NC2CCC(CC)C2)=O)ccc(CCC#N)cc1 Cc1cc(C(=O)NCCC2CCCCN2C(C2CCCN2N=O)=O)sc1C N1(C(c2cc(C)oc2)=O)CCCC(N2CCN(C(c3ccc(C)o3)=O)CC2)C1 C1(NC(c2c(CC)n(C)cc2)=O)CCCCCC1NC(=O)C(CC1CC1)OC c1(C(N2CCC(NC(CCC=C)=O)C(C)C2)=O)cc2ccc(F)cc2nc1O C(=O)(C1=NOC(C)C1)N1CC(CNC(c2c(C)coc2C)=O)OCC1 C=CC(CC)C(=O)NC1CCCCC1C(=O)N(CCCC(=O)OC)C c1(C(=O)NCC(C)(C(C)C)NC(CN(CC)CC)=O)cc(F)c(O)c(Br)c1 C1(C)(C(N(CCC(C)NC(c2cc(OC)ncc2)=O)C)=O)CCCNS1(=O)=O CCCCC(CC)C(=O)N1CCC2(C1)CN(C(C1(F)CCC1)=O)C2 C1(C(=O)NC2(C)CN(C(c3ccc4nccn4c3)=O)C2)CCn2ncnc2CC1 C(=O)(N=c1cc[nH]cc1Cl)c1ccc(C)c(-c2nc(C(=O)O)cs2)c1 C(=O)(C1=C(C)OCCS1(=O)=O)NCC1(O)CC(CNC(CCCC(=O)NC)=O)C1 c1(CC(C)NC(C2(n3cc(C(CC)(C)O)nn3)CC2)=O)ccc2cccnc2c1 N#Cc1cnc2ccc(=NCc3cn[nH]c3)[nH]n12 N1(C(C(COCC)NCCOC(C)=O)=O)C(N(C)C)CCC1C1CC1 c1(CC)c(C(=O)NC2CC(OC)C2)c(O)nc2[nH]nc(O)c12 C(=O)(CS(=O)(=O)CCO)N1CC(c2ccc(OC)cc2)N(C(C)=O)CC1 C1(CN(C(=O)CC2C(C)(C)C2(C)C)C)CCCCN1C(c1cnn(C2CC2)c1)=O c1(OCCC(N2CCC(CN(C3CCCN(CC)C3)C)C2)=O)ccc(F)cc1Cl c1(-c2nccc(NC(=O)Cc3ccc(F)c(Cl)c3)c2)ccc2c(c1)OCCN2 C1(O)(C(N2CC(NC(CC(C)N(C)C)=O)C(O)CC2)=O)CN2CCC1CC2 N1(C(c2[nH]cc(CC)c2)=O)CCN(C(N2CCN(CC3CC(O)C3)CC2)=O)CC1 CC1CCC(NC(C2CCNC2=O)=O)CN1C(=O)C(C1CCCCCC1)O CC(C)C(CCNC(c1cnsn1)=O)NC(c1cncnc1C1CC1)=O c1(OC)ccc(C(=O)NCCN(C(=O)C2=NOC(C)C2)CC(C)O)cc1O c1(C(N2CC(C(=O)NCC3CCN(C)C3)C(O)CC2)=O)[nH]nc2ncccc12 C1(NC(C2(CC)CCC2)=O)COCCN(C(c2cc(=N)[nH]c(Cl)n2)=O)C1 Cc1cc([N+](=O)[O-])ncc1C(N1CCC(NC(=O)CC(=O)C(F)(F)F)C(C)C1)=O C1(NC(Cc2nc(C)sc2Cl)=O)CC2(C1)CN(C(C1CCCSC1)=O)C2 c1(CCC(=O)N(C)CC2(O)CN(C(C3(SC)CC3)=O)C2)nc2cccc(Cl)c2[nH]1 C(C1CCN(C(C2(Cl)CCCCC2)=O)CC1)=CC(=O)NC(CC)C(C)C C(F)(F)(C(F)(F)C(F)(F)F)N1CCN(C(=O)Nc2cccc(COCC)c2)CC1 c1(OC)ccc(C(C)C(=O)NCCNC(C2(C)CC2C)=O)cc1 C1(C(N(CC(=O)NC2CCC(C(N)=O)C2)C)=O)(CNC(=O)C2CC2)CC12CCC2 c1(N(C)C)ccc(CCC(=O)NCC2CN(C(C3(C)CS(=O)(=O)C3)=O)C2)cn1 N1(C(C2(C#C)CCC2)=O)C2CCC1CN(C(=O)CSCc1ccc(Cl)cc1)C2 CC(C)C(F)(F)CC(=O)NCC1CCCC(CNC(C2(C)CC2)=O)C1 c1(N2CC(N(C)C)C2)ccc(N2CCC(SC(C)=O)C2=O)cc1Cl c1(C(N2CCN(C(CCOC)=O)CC23CC3)=O)oc(=O)c2ccccc2c1C C1(NC(c2c(CC)ncs2)=O)CN(C(c2ccc3c[nH]nc3c2)=O)CC1N=[N+]=[N-] C(=O)(C(CC(C)C)OC)NC(CNC(C(OCC)NCc1nccs1)=O)C(C)C N1(C(c2c(Cl)cnc(OC)n2)=O)CCC2(CCC(NC(C3CC3C(N)=O)=O)C2)C1 CC1CCC(=CC(=O)NCC(C)CNC(C2CC3(CC3)CO2)=O)CC1 c1(C(=O)Nc2cn(C)c(NCc3c(Br)ccnc3Cl)n2)cc(Cl)ccc1I C1(C(=O)NCC2CC3C=CC2O3)(NC(C(CC)O)=O)CCOCC1 C1(NC(C(C)(C)OC)=O)CCC2(CCCN(C(c3ccc(C(C)C)nc3)=O)C2)C1 CC(C)C(CC1CCCCC1)C(=O)NCCCN(CCO)C(C1CCSC1)=O N1(c2cc(C)ncn2)CCN(C(=O)CC(C)n2ccnc2)C(C)C1 C1(C(=O)NCC2CC3(CN(C(C(CSC)O)=O)C3)C2)CS(=O)(=O)CC(=O)N1 C=CCC(CC=C)NC(N1CCOC(C)C1)=O CCC(C#N)C(=O)NCC1CCCC1NC(C1(O)CCOCC1)=O N1(C(=O)Cc2csnn2)CCN(C(=O)CCOc2ccc(Cl)cc2)C(CCO)C1 Cc1[nH]c2c(F)cccc2c1CCNCc1ccccc1OC(F)F N1(C(C(C)O)=O)CC23CCCC2(C1)CN(C(C1CS(=O)(=O)C1)=O)C3 C1(NC(c2c(CC)occ2C)=O)CCN(C(=O)COCCOC)CC1C N1(C(CN2CCC(C)CC2)=O)CCCC(N(C)C(C2(C)CCCS2(=O)=O)=O)CC1 c1(OC)cc(C(=O)NC(C2CCN(C(=O)CSCCC(F)(F)F)C2)C)ccc1F c1(CNC(CC2(C)CCN2C(=O)C=CC=Cc2ccccc2)=O)c(F)cccc1F C(=O)(C(Cn1cccn1)NC(C1C=CCS1)=O)N(C)CC1CC(=C)C1 Cc1ccc(C(=O)NCC2CCCC(NC(=O)CNS(=O)(=O)N(C)C)C2)cc1O C=CC(C)(O)CC(=O)NCC1CCCC(CNC(=O)Cn2ncc(Br)n2)C1 c1(N(C)C)cc(CC(=O)NCC2CCC(NC(=O)CSC3CCCCO3)C2)on1 C(=O)(C1=C(C#N)CCC1)NCC(C(=O)NC1CC(C(F)(F)F)C1)N(C)C Cc1cc2cccc(CNC(C3(Cc4ccccc4)CCNC3)=O)c2[nH]1 C(=O)(C(C)(CC)C(N)=O)NC1CN(C(c2c(SCC)cccc2)=O)CC1COC C1(CNC(CCN(C(C2C(C)(CC)C2)=O)C2CC2)=O)CC2CCC(C1)C2 Cc1ccc(N)cc1C(=O)NCC1CN(C(c2nc(C(C)(F)F)cs2)=O)C1 C(c1c(C)cc(C)cc1C)=CC(=O)NC1C2CN(C(C=C(CC)CC)=O)C(C2)C1 Cc1cc(CC(=O)NC2CC2CNC(=O)CNC(C2CCCCCC2)=O)ccc1Cl c1(C(=O)NCC2CCN(C(C3(O)CCC3)=O)CC2)ccc2nc(O)oc2c1 C1(C(=O)NC(CC(=O)OC)C)CN(C(c2c(F)cccc2Cl)=O)CCC1O CC(C)(C)C(C(=O)NCC1(C)CCN(C(=O)C2=CCCO2)C1)C1CCC1 C(C1=CCN(C(=O)COc2cccc(C(F)(F)F)c2)CC1)NC(CCC(N)=O)=O CCCC(C)(O)CNC(c1cn(CCNC(c2scc(C)c2C)=O)cn1)=O C1(NC(C(Cc2c(C)noc2C)C)=O)C2CC1N(C(=O)C1=CCC1)C2C CCCC(O)CC(=O)NC1CCCN(C(c2cc(C)ccc2Cl)=O)C1C N1(C(CCc2ccc(C(=O)NC(c3cccc(Br)n3)C)[nH]2)=O)CCC(C#N)C1 n1(CCOCC=C)c(N(C)CC2(C)CC(O)C2)nnc1-c1ccc[nH]1 C=Cc1cnn(C)c1C(=O)NC(C)CNC(=O)CCCN1CCCC1=O Cc1cccnc1CCC(N1CCC(CO)(NC(C2CCC(C)CC2)=O)C1)=O N1(C(=O)NCCCN(c2ccccc2)C(C)(C)C)CCC(C2CCC(=O)N2)CC1 NC(=O)CCC(N)C(=O)N1CC2CCC(C1)C2C(=O)NC1(c2ccccc2)CC1 C1(CNC(CC2(COC)CC2)=O)CN(C(=O)CC2NC(=O)NC2=O)CC(C)(C)O1 c1(C(=O)NCC(C)NC(C2CC(OC)C2)=O)cc(CO)n(C)n1 C(S(=O)(=O)CC(=O)NCC1(C(=O)O)CCCO1)c1ccc(C)o1 c1(OC)cc(C(=O)NC2(CCNC(C3CCC(C)O3)=O)CCC2)ccc1Cl C#Cc1cccc(CC(=O)NC(C)CN(C(=O)Cn2cc([N+](=O)[O-])cn2)CC)c1 CC1(C)CN(C(C23COC(C2)C(O)C3)=O)CC1CNC(=O)CC(=O)N(C)C N1(C(c2cc(C)sc2C)=O)CCC(NC(c2cccc(C3CC3)n2)=O)C(O)C1 C1(C(=O)NCC(C(C)C)OC)(OC)CCCC1 N1(Cc2ccc(C(N)=O)o2)CCc2ncccc2C1.N12CCC3(CC1)CC3C2=O C(=O)(C1CCc2ccccc21)N(CC(=O)NCCCF)C1COC1 c1(CC)ccc(C(=O)NCC2(F)CC(CNC(=O)CC3CCCN3C(C)C)C2)s1 C1(OC)CC2(C1)CC(C(N1CCOCC(CNC(=O)Cc3nonc3C)C1)=O)C2 CCC(O)CC(=O)NC1CCC(CCC(=O)NCc2cnn(CC)c2)C1 C1(NC(CCOC)=O)CCC(N(C)C(c2cnn[nH]2)=O)CC1 C(=O)(C1=CCCC1(C)C)N(CCOC)CCNC(C1(CC2CCCCC2)CCC1)=O Cc1nc(CNC(=O)CC2CC(F)(F)C2)oc1C(=O)N(C)CC1OCCC1(C)C c1(CC(=O)NC2C(OC)CN(C(=O)C(C)CF)C2)c[nH]c2cccc(F)c12 c1(NC(=O)NC2CN(C(CCOc3cccc(C)c3)=O)C2)cc(S(C)(=O)=O)co1 c1(NC(C2C3(CN(C(CCOC)=O)C3)C2)=O)cccc2[nH]nc(I)c12 C1(NC(COCCC)=O)CN(C(c2ccccc2N)=O)CCC12CCC2 C1(CNC(c2c(OC)c(C)sc2)=O)CN(C(C2CC2C(C)C)=O)CC1(C)C N1(C(C(C)Oc2ccccc2Cl)=O)CCC2CCN(C(=O)CCCF)C2C1 C(=O)(CC1OCc2ccccc21)NC(CNC(c1cn(CCC)nn1)=O)(C)C c1(C(N(C2CC3CNC2C3)Cc2cccc(C)c2O)=O)cc(F)c(Br)cc1F CCC(C)CCC(O)CC(=O)NCCN(C(=O)CS(=O)(=O)C(C)(C)C)CC C(C)(C)(CC(=O)NCc1cnnn1C)n1cc(CCCN(C)C)nn1 N1(C(c2c(-c3cn(C)nc3)ocn2)=O)CC2CC(C1)C2NC(=O)Cc1csnn1 CC(=O)CCCC(C)C(=O)NC(c1ccccc1F)CNC(=O)CC1(C)CC1 C1(CNC(C2C(C)CC=CC2)=O)CN(C(c2ncccc2F)=O)CCC1(F)F C(C#Cc1cccnc1)NC(C(C(C)NC(=O)CCC(F)(F)F)(C)C)=O C1(CNC(CSCC=C)=O)CCC2(CCC2)CN1C(c1cccc(N(C)C)c1)=O C1(C(C)C)C(=O)N2CCN(CC2)CCO1.Cn1cnnc1C(N1CCCC1CO)=O N1(C2CCN(CC=C)C2=O)CCC(C)(NC(=O)CC2(OCC)CCC2)CC1 C1(C(=O)Nc2c(SC)cccc2)CC12CCN(C(=O)OCC(C)C)CC2.C(C)(C)C N1(CC)C(=O)NC(c2ccc(Br)c3[nH]ncc23)C(C(=O)OCC)=C1C1=CNCC1 c1(OCC(=O)C2CC2c2cccc(Cl)c2)nccn2nc(Br)cc12 N1(C(C(c2ccc(C)cc2)C2CC2)=O)CC2CCCC(C1)N2C(C1(C(N)=O)CC1)=O c1(C(=O)NCCC(CNC(C=CC(CC)C)=O)O)cc(Cl)c(C)cc1OC C1(C(=O)NCC2C(C)CCN2C(=O)CC2CCCC(=O)N2)CC(C2CC2)=NO1 N1(C(c2nc(C)nn2C)=O)CCC2CN(C(=O)CCC3(C)CC3)CC2C1 C1(C2CC2)(CNC(c2scc(C)c2C)=O)CCN(C(C2(C(F)F)CC2(F)F)=O)C1 c1(C(C2(NC(C(C)CC3CCOC3)=O)CCSCC2)OC)c[nH]c2ncccc12 c1(CC(=O)NC(C)C(CO)NC(C2CC2(F)F)=O)cccc(OC(F)(F)F)c1 c1(CS(=O)(=O)NCc2ccc(C(O)C(F)(F)F)cc2)ccc(Br)cc1 N1(C(C(C(=O)OC)OC)=O)CCN(C(c2cnc(C)[nH]c2=N)=O)C2(CC2)C1 c1(COC)cc(N2CCCC2CC(=O)NCC2(C(F)(F)F)CC(C)(C)C2)ncn1 N1(C(c2ccc(C)c(I)c2)=O)CCC2CN(C(=O)COC(C)C)CCC12 CC1(C)CN(C(=O)CC2CCC=CCC2)CCN(C(=O)C(C2CCOCC2)=O)C1 Cc1cccc2oc(NC3CC(CNC(=O)C4=C(Cl)CC4)C3(C)C)nc12 C#Cc1cc(F)c(C(=O)NCCC2CCCCN2C(=O)C(O)C(F)F)c(F)c1 C(CCC(C)C)=CC(=O)NCCOCCNC(C=C(C)C(F)F)=O C(=O)(C1=NN(C)C(=O)CC1)N(CC(=O)NCc1c(CC)onc1C)C c1(C(=O)Nc2c(OCC)cc(C)cc2)cnn2c1NCC(C)C2 c1(C(N2CCC(N(CC(CC)C)C)C2)=O)cccc(-c2ccc(O)nn2)c1 N1(C(c2cc(CC)oc2C)=O)CCC(NC(=O)C2=CCCO2)C(C)C1 c1(C(N2CC3(CN(C(CCS(C)=O)=O)C3)C2)=O)cc2cc(Cl)c(Cl)cc2[nH]1 C1(C(N(CCCN(C)C(c2ccc(C(C)(C)C)cc2)=O)C)=O)CCC(C)(F)CC1 C(=O)(C(C)CC(C)CC)N1C(CC)CCC1C(=O)NC1CC(C)N(C2CC2)C1 C12(C(=O)NCCCN(C(Cn3ccc(C)n3)=O)C(C)C)CC1COC21CCC1 c1(C(N2CC(NC(C(C)C3CC3)=O)C(C)C2)=O)ccn2c(O)nnc2c1 C1CC(C)(C)C(=O)N2CCC(C2)Cn2cc1nn2.C1(CSC)CC(N(C)C)C1 C(=O)(CCCCC#N)NC(C(C(C)C)NC(c1cc(Br)cn1C)=O)C N1(C(c2c(CC)n[nH]c2)=O)CCC12CN(C(C1CC3(C1)CC(F)C3)=O)C2 c1(C(=O)NCCCC(C)NC(=O)CC2CC2)c(Cl)n[nH]c1C1CC1 Cc1cc(C(N2CCC(NC(c3cccc(C)c3Cl)=O)C2)=O)[nH]c1C#N CCC(C)C(C(=O)NCc1ocnc1C(=O)NCc1nn(C)c(=O)n1C)OC CCCCC(CC)C(=O)NC1(CF)CN(C(C2C(C)CCN2C)=O)C1 c1(-c2ccc(COC)cc2)ccc(OC)cc1-c1nccn1CCl.C1CCOC1 c1(C(N(CC(C)N(C(C(C)=CC)=O)C)C)=O)cc(S(=O)(=O)N(C)C)oc1C C1(N(CC(=O)O)C)CCCN(c2ccc(C(F)(F)F)cc2)C1 C1(C(N2CCCC2c2cn(C(C3CC3C(=O)O)C)nn2)=O)COCC2(CCC2)O1 N1(C(C=CC=CC)=O)CCN(C(=O)Cc2cncc(O)c2)C(C)C1C C1(C(N2CCN(C(=O)CN(C(=O)CC(C)O)C)CC2)=O)(CC)CCCCC1 N1(C(C2C(OC)CC2)=O)CCS(=O)(=O)C(CCNC(=O)CN2CCN(C)CC2)C1 Cc1cccnc1CC(=O)NCCc1n[nH]cc1C(=O)NCCN1CCCCC1 C1(NC(C2C(CCOC)C2)=O)(CO)CCN(C(c2cc(C(N)=O)n(C)n2)=O)C1.C1(C)CC1 N1(C(C(CC=CC)NC(=O)Cc2cc(C)no2)=O)CCN(C)CC(O)C1 c1(C(N2C(C(C)C)CN(C(c3cc[n+]([O-])cc3)=O)CC2)=O)cn2c(n1)COCC2 N1(C(c2c(CCC)n[nH]c2)=O)CC(NC(C2(CC)CC2)=O)C2(CCC2)C1 C1(C(N2CC(C=C)C2)=O)(COC)CCN(C(c2oc(C)nc2C)=O)C1 CN1CC(C(=O)NCC2COCCN2C(=O)C(N)=O)CC1=O C1(C(=O)NCC=CCNC(CC2CC(CC)C2)=O)CCCC2CCCN12 C(=O)(C(O)CCCCC)NC(CCC=C)C(=O)Nc1cccnc1OC c1(C(=O)N(CCNC(C2(Cl)CC23CCC3)=O)C2CC2)cnc2c(c1)COC2 c1(C(=O)NCC2CN(C(CS(CC)(=O)=O)=O)C2)cccc2[nH]nc(O)c12 C1(C)(CC)CCC(N(C)C(=O)OC(CO)C(C)C)CC1 CCC(C)C(C)CNC(=O)C(C1CN(C(=O)Cc2nccn2C)C1)OC CC(CCC(=O)N1CCC(O)(CN(C(=O)Cn2ncccc2=O)C)C1)SC1CC1 C(=O)(C1CCCc2nc(C)[nH]c21)OC(c1cccc(Br)c1)COC C1(C(C)C)CCN(C(C2(O)CCCC2)=O)CC1.C12(CCCC1)CNC(=O)NC2 C(=O)(C(F)CCC(C)C)N(C1CCCN(C(CN2CC(CC)C2)=O)CC1)CC CC1CN(C(=O)Cn2ncnn2)CC(C)N(C(c2cc(CO)[nH]n2)=O)C1 C12(C(N(C(C)CNC(c3ccncc3)=O)CC)=O)CCCCC1NCC2 Cc1ncc(NC(=O)C(CC2CCCC2)NC(=O)CC2CC2(C)C)cn1 Cc1nc(N2CC3(CC3)CC2C(N2CCn3cncc3C2)=O)c2sccc2n1 C(=O)(CCS(C)=O)N1CC(N(C(C2CCN(CCSC)C2)=O)C)C1.CO c1(CC(=O)NCC(O)CNC(=O)NCCCC(=O)N(C)C)cccc(F)c1 Cc1nn(C)c(C)c1C(=O)N(CC(C)N(C)C(C1CCCCS1(=O)=O)=O)C c1(NC(=O)Nc2c(C(=O)OC)cnn2C)cc(CC2CCCC2C)ccc1Br C1(C(N)=O)CN(C(C2CCCN2Cc2scnc2Cl)=O)CCO1 C(CC(F)F)(C(=O)NCC1(O)CC(O)C1)NC(c1cc(=N)[nH][nH]1)=O Cc1cc(N)cnc1C(=O)NC(C1CN(C(=O)CC2CCC(C)C2)C1)C C1(C(=O)NCC2(C(=O)NC(C=C)CO)CC2)CCCCNC1=O C=CCC(CNC(=O)C(C)(O)COC)C(=O)NC(C12CCC(CO1)C2)C Cc1ccc(CC(=O)NCCCC(C)NC(=O)CCCc2ccccn2)o1 C(C(CNC(=O)CCC1NC(=O)NC1=O)S(C)(=O)=O)NC(c1c(C)nsc1)=O CC#CC1CCN(C(=O)CC2(NC(C3(N(C)C)CC3)=O)CCC2)C1 c1(OC)cccc(C(=O)NC2C=CCN(C(C3CC3C)=O)C2)n1 C(=O)(CCC(c1ccccc1)NC(N)=O)N(CCN(C(=O)C(Cl)=CCl)C)C C1(C(N(C23CC(C2)C3)C)=O)CC(O)C(O)CC1CNC(=O)C(C)(C)n1cccn1 C(=O)(C1CCc2nnc(C)n21)N1CC(NC(C=C(C)Cl)=O)C(O)CC1 C1(CNC(=O)CNC(=O)C2CC2)CC2CC(C1)N(C(c1ccc(O)nn1)=O)C2 C(=O)(CC(O)CC(C)C)N1CC(NC(C(C(C)(C)C)NC(C)=O)=O)C(C)C1 c1(OC)cc(C(N2CCCC(O)(CNC(C3CCS(=O)(=O)C3)=O)C2)=O)cc(F)c1 CCC(C)(CC)C(=O)N1CC(O)(CN(C(=O)CC2CC23CC3)C)C1 c1(OC)cc(NC(=O)CC2CCC(NC(C3CCSCC3)=O)CC2)cc(OC)n1 C1(NC(C=C(C)C)=O)(CNC(=O)CC(=O)NCC=CCl)CCCCC1 c1(C(=O)NCCC(=C)CNC(=O)C(C(C)O)NC(C)=O)nc(Cl)sc1Cl N1(C(Cc2n(C)nnc2)=O)CCC(NC(C2CC3CC3C2)=O)C(O)C1 N1(C(CC(CNC(c2c(C)cn(C)c2)=O)C)=O)CCC2(CCOC2)CC1 Cc1cc(=O)n(CCc2nc(C3CC3)no2)c(=O)n1C1CC1 c1(C(=O)NC(CCNC)C)cccc(-c2ccc(C)cc2)c1 C1=CC(=O)Nc2ccc1cc2.c1(OCC)cccc(CN(C)C)c1F C(CC(F)F)(C(=O)NCc1coc(C(C)C)n1)NC(C1CC(OC)C1)=O C(=O)(C1CCC(NC(C2C3C=CC(O3)C2C(F)F)=O)c2ccccc21)OC C=CC1(NC(=O)C(CC2CC2)NC(=O)C2=CC(C)(CC)C2)CCCCC1 C(=O)(CC(O)CCC)N1CC=CC(NC(COCCCCOCC#C)=O)C1 N1(C(C2CCCC(C)C2)=O)CC(NC(=O)Cc2ccc(Cl)cn2)C(F)(F)C1 N1(C(c2cc(OC)cc(Br)c2)=O)CC2ON=C(CNC(=O)C3=CCC3)C2C1 N1(C(C(C)N2CCC2)=O)CCC2CN(C(=O)CCSCc3ccccn3)C2C1 N1(CC2CCC(=O)C2)CCc2c(CNC(C3(C4CCCO4)CC3)=O)cccc2C1 Cc1cccc(C(=O)N(CCCCN(C)C(c2conc2C2CCCO2)=O)C)c1 c1(C(N2C(C(N3CC(c4n(C)ncc4)C3)=O)CCC2)=O)cc(I)c(F)cc1F N1(C(C)=O)CCCC(C(=O)Nc2cccc(-n3ccc(C)n3)c2)(CO)C1 c1(C(=O)NC(C(CC)C)c2nnnn2C)cc(OC)c(C)o1 CC1COCC(CC(N2CCC(C)(C(N3CC(O)CC3CO)=O)C2)=O)O1 c1(CN2CCC(NC(c3cncc(C)c3)=O)(CF)C2)cnc(F)cc1C Cc1c(C(N2CC(NC(c3cc(C#N)cs3)=O)CC(O)C2)=O)cccc1[N+](=O)[O-] N1(C(C(C)(C)C(N)=O)=O)CC(NC(C2CCOC2(C)C)=O)C2(CCOCC2)C1 c1(C(N2C(CNC(CCc3cc(C)[nH]n3)=O)CC2)=O)n[nH]c2c1NCCC2 C1(CNC(C(C(C)C)F)=O)CC2CCC1N2C(c1cccc(O)c1Cl)=O C1(NC(CN(CC)CC)=O)CCC(O)CN(C(C2(C)CC3(CCCC3)C2)=O)C1 N#Cc1cccc(Cn2nc(CC3CC3)nc2-c2cc3sccc3[nH]2)c1 c1(CC(=O)NC(C)C)noc(C)c1C#N.C1(=O)C#CC(=O)N(C)CCOC2CN1C2 C(=O)(C(C)C(C)NC(C1CCN(C)C1)=O)OCC.N12CCC(C1=O)NC(=O)C2 C12(C(N(CCC(C)C)CCC(C)C)=O)CCC(C(N3CCC(O)C3)=O)(CC1)CC2 N1(C(c2ccn(C(C)C)n2)=O)CCCC(CNC(c2cncc(F)c2Cl)=O)CC1 CC12CC3CC(C(=O)NC4CN(C(=O)C=CBr)C4)(C1)CC(C)(C3)C2 N1(CC(=O)NCC(CC)N(C)C(c2ccc(OC)o2)=O)CCOCC1 c1(C(N(CCNC(CC(=C)C)=O)CCOCCO)=O)nccc2ccn(C)c12 C1(NC(c2cc(Br)no2)=O)COC2(CCN(C(=O)C=C3CCSCC3)C2)C1 C(c1ccc(-c2ccc(F)cc2)s1)=CC(N1CCC(NC(c2ccsc2)=O)C1)=O C(=O)(N=c1ccn(C2CC2)[nH]1)C1(F)CCN(C(C(c2cncnc2)C)=O)C1 c1(C(=O)NCC2(C)C(NC(C=CC(C)C)=O)CCC2)ccc(O)nc1Cl c1(N2CCCC(NC(C3C(C)C3)=O)CC2)ncc2c(ccn2C)n1 CCC(F)(F)CC(=O)NCC1CCN(C(C2CC2(C)C(F)(F)F)=O)CC1 c1(OC)cc(C)c(NC(C2CC2NC(c2cccc(OC)c2)=O)=O)cc1Br Cn1cc(C(=O)NC2(CNC(=O)C(N3CCOCC3)C3CC3)CCCC2)cn1 C12(C(=O)NCCC3CCN(C(CCCn4ncc(C)c4)=O)C3)CCC(CC1)C2 c1(CC(=O)NCCC(C)NC(C2CC(OC)C2)=O)ccccc1S(C)=O C=CCCC(C(=O)NCCC1CCCN(C)C1)NC(C1CC(=O)N(CC)C1)=O c1(C(N2CC(O)(C(C)NC(C3CC(=C)C3)=O)C2)=O)cn2cc(Cl)cnc2n1 CC(C)(C)C(CN1C(=O)NC(C(C)(C)C)C1=O)C(=O)NC1CCNC1=O C1(C(=O)NCC(C2CCCC2)NC(c2sccc2F)=O)CCC(C(F)(F)F)CC1 N1(C(C(c2c(C)c3c(s2)cccc3)=O)=O)CC2CCC(C1)N(C(=O)C(Cl)=CCl)C2 C1(CNC(C=CC(C)C)=O)CCC(F)(CNC(=O)CC2C=CS(=O)(=O)C2)C1 C(CC(C)C)(C(=O)NCc1ccc(F)cc1C)NC(C(C)OCC#C)=O C1(C(N(CCC(C(C)C)OC)C)=O)COCCN(C(C2CC(F)CN2C)=O)C1 C(=O)(C(CCC(C)C)NC(c1ccnc(C)c1C)=O)NC(C=C)C(F)(F)F N1(C(C(=Cc2ccc(Br)o2)C)=O)CC(NC(C2(C(C)C)CC2)=O)CCC(O)C1 N1(C(C#CC(C)C)=O)CCC(C)CC1CNC(=O)C(C)(C)c1cnn(C)c1 c1(C(=O)NCC2(C)N(C(CN(C(C)=O)C)=O)CCC2)ccccc1N=[N+]=[N-] CC(C)C(C)(CNC(c1ccc(F)cn1)=O)NC(=O)CN1CCC(C)C1 c1(C(C)NC(COC)=O)ccc(CNC(c2cc(Br)ccn2)=O)cc1 c1(C(=O)NC2CCCC(N(C(=O)Cc3csnn3)C)C2)ccc2[nH]c(=N)[nH]c2c1 c1(C(=O)NC2CCN(CC=C)CC2C)noc2cc(Cl)ccc12 C(=O)(C(CNC(C1CC(O)CN1C)=O)C(C)(C)C)N(CC(C)O)CC(C)O N1(C(C2(COC(C)C)CC2)=O)CCOC(CN(C(=O)C(C)N2CCC2)C)C1 N1(C(C=CC=CCCCCC)=O)CCN(C(C2(O)CC(C)(C)C2)=O)CC(C)(C)C1 c1(C(=O)NC(CC)CNC(=O)CCC2CC2(Cl)Cl)ccncc1F C1(NC(CCC=C=C)=O)COC2CN(C(C3CN(C(=O)C(F)(F)F)C3)=O)CC12 N1(C(COC(C)C)=O)CCCC(C)(C)C1C(=O)NC(C)C(C)O c1(CC)ccc(C2C(=O)C(=O)NN2C)c(C)c1.C(CCC(C)O)N.c1(N)ccco1 CCC(C)C(C(=O)NC1CCN(C(C2SCCCS2)=O)CC1F)NC(N)=O CC(C)CCCC(C)C(=O)N1CCC2CN(C(c3cc(O)nc(Cl)c3)=O)C2C1 N1(C(CSC(C)C)=O)CCOC(CNC(c2cncn2-c2ccc(F)cc2)=O)C1 C1(OC)CCCC(CC(N2CC(C(F)(F)F)C(CNC(=O)C#CC3CC3)C2)=O)C1 N1(C(C=C(COC)C)=O)CCC(C2(NC(=O)CCNC(C3CCCO3)=O)CC2)C1 C1(CNC(CC)=O)CCN(C(=O)COCC2CCCO2)CC1C1CC1 N1(C(c2ncc(CC)nc2)=O)CC2(C1)C(NC(=O)C1=C(C)CCC1)CCS2(=O)=O N1(S(CC)(=O)=O)CCCC(C(N2CCC(CNC(C3(CO)CCCC3)=O)C2)=O)C1 C1(CCCC)CN(C(c2ccc(C(=O)OCC)cc2C(F)(F)F)=O)CCN1C(C)=O N1(C(CC=CC=C)=O)CCCC1(CNC(=O)COC(C)CC)COC C(C)(CS(C)(=O)=O)NC(C(=O)N(C1CCN(S(C)(=O)=O)CC1)CCCC)=O c1(OC)ccc(CC(=O)OC(C2CN(c3nccnc3F)CCO2)C)cc1F C(=O)(C(O)CC(F)F)N(C1CCN(C(C2CC(F)(CO)C2)=O)CC1)C CN1C(=O)CCCC1C(=O)NC1C2CC1N(C(=O)CCCF)C2 Cc1nc(C)c(CC(N2CCN(C(=O)NC3CC3)C(CC(F)(F)F)C2)=O)c(O)n1 C(=O)(C(CC(C)C)C(N)=O)N1CCC(NC(CCN(CCC)C)=O)C(F)C1 N1(C(c2ccc(Cl)s2)C)CCn2cnc(-c3ccc(-c4ccccc4)s3)c2C1 C(=O)(C(CC(C)C)NC(=O)CC(O)CC1CC1)N(C(C(=O)OCC)C)C C1(C(=O)NC(CN(C(CSCC(C)C)=O)C)(C)C)CCCOC1c1cn[nH]c1 C=C1CCN(c2cc(OC(C)=O)ncn2)C1C(=O)NCCOCCN(C)C.CO C1(NC(C(CCC)O)=O)CCN(C(=O)C=C(C)I)CC(C)(C)C1 C1(NC(C(C=C)(C)C)=O)CCCCCC1C(=O)NCC(O)CC(C)(C)C C1(CC)Oc2cc(C(C)NC(C3(CO)CCCC3)=O)ccc2NC1=O c1(C(=O)NCC(CC=C)NC(c2n[nH]cc2Cl)=O)ccc2nc(CC)cn2c1 CC1CN(C(=O)CCN(C(=O)CN2CCCC2C)C)CC1(F)F Cc1ccc2c(c1)CC(C)N(Cc1cn(Cc3ccccn3)nn1)C2 C(CCC(O)C(=O)N1CCC(N(C)C)C(C)C1)NC(C1(C(C)C)CC1)=O C1(C(=O)NCC(=O)NCCN(C(=O)C(C)(C)C)C(C)C)CCc2c[nH]nc2C1 C1(NC(=O)COC2CCCCC2)CCCN(C(C2(C(F)(F)F)CC(O)C2)=O)CC1 CCCC(C(C)CC)NCC(N1CCCC1c1ncno1)=O C(=O)(C(C)CC(F)(F)F)NC1N(C(CCCCCOC)=O)CC(OC)C1 Cc1ccc2[nH]c(C(=O)NCC3CN(C(=O)C(C)C(C)C)C(C)(C)C3)cc2c1 C(=O)(CS(=O)(=O)CC(C)C)NCC1(OC)CN(C(=O)C(N2CCN(C)CC2)C)C1 c1(C(=O)NC2CCN(C(=O)CN3C(=O)CSC3=S)C2)ncc(C2CC2)cc1F C(CC)(C(=O)N1CCC(CCNC(=O)C(=O)NCC(F)(F)F)C1)OCC c1(C(=O)OC)cc(S(=O)(=O)NCC(O)COc2ccccc2OC)c(Br)cc1C C(C(=O)NC1C=CCN(C(=O)CSc2n[nH]c(O)n2)C1)(C(C)(C)C)N(C)C N1(C(CC2(C(=C)F)CCC2)=O)CC2(C)CN(C(=O)CCOCC3CC3)CC2(C)C1 c1(NCC2(NC(=O)C(=O)NCC(F)F)C(C)CCCC2)ncc2c(n1)CCCC2 c1(OC)cncc(C=CC(=O)NCCCNC(=O)CC2CC3C=CC2CC3)c1 C(=O)(C(C)(C1CCC1)NC(=O)CN(C)C1CC1)N(CC(C)OC)C N1(C(CCC(C)(C)O)=O)CCC2CCCC12CNC(=O)C(F)(F)c1cscn1 c1(CNC(C(N2CCOC(C)(C3CC3)C2)C)=O)ccc(F)c(F)c1 C=CCCCCC(=O)NCC1(CC(N2CCC(CO)C2(C)C)=O)CCOCC1 Cc1ccn(C)c1C(=O)NCC(C(C)(C)C)NC(=O)C=CCO CCC(C)(C)CCCC(=O)N1CCCC1CCNC(C1CC(C)=NO1)=O Cc1csc(CCCC(=O)NC2CN(C(=O)C=CBr)C2)n1 c1(OC)ccc(C(=O)N(C)CCOCCN(C(=O)C(F)C2CCC2)C)nc1Cl N1(C(C2COCCN2C(c2ccc(CF)cc2)=O)=O)CC2(CCC1CO)CC2 C(=O)(C(O)CCCNC(C1COCC1(C)C)=O)NCCc1cn(CC)nc1 c1(C(N(CC(CC)NC(C2C=CCCC2)=O)CC)=O)cccnc1-n1ccnc1 CCC(CC)CCCN(C)C(c1cc(SCc2ccccc2)[nH]n1)=O C1(C(N2CC(OCCNC(=O)Cn3cnnn3)C2)=O)OCCC1C(C)(C)C N1(C(C2(C(=O)NC(C)=O)CC2)=O)CCN(C(C2CC2(F)F)=O)C(CO)C1 C1(OC)CCN(C(=O)C(CNC(=O)CCCC(C)=O)C(C)C)CC1(C)C c1(C(C(=O)NC(C(=O)OC(CC)(C)C)C)N(C)CCF)ccc(C2CCC2)cc1 C1(C(=O)NC2CC(NC(C3CC3(Cl)Cl)=O)C2)CCCN2CCCC12 C=CC1(CC(=O)NC(c2cn(C)cn2)C)CN(C(=O)COC(C)CCC)C1 C1(NC(CNC=O)=O)CN(C(C2CCCN2C2CCC2)=O)CC1C(F)F C12(NC(CCOCCOCC)=O)CCC1CN(C(c1snnc1C(C)C)=O)C2 N1(C(Cc2ccc(C)o2)=O)C2CCC1CN(C(c1ocnc1C)=O)C2 C1(NC(CCC=C(C)C)=O)CC2(CCC(NC(C34CCC(F)C3CC4)=O)CC2)C1 N1(C(C(C(C)(C)C)O)=O)CCC(C(N2CCCC(S(N)(=O)=O)C2)=O)C2OCCC12 CC(C)CC(CNC(=O)Cc1sccc1Cl)NC(c1ccc[n+]([O-])c1)=O C1(CNC(Cc2nnc(C)s2)=O)CCCC(CNC(c2c[nH]nc2C2CC2)=O)C1 C(=O)(C(C)CC(=O)OC)OC(C(=O)NC1CC2(C(=O)OCC)C(C1)C2)C(C)C c1(C(=O)NC2C(NC(c3c(C)cc(F)cn3)=O)C2)c(F)ccc(C)c1Cl Cc1ccc(C#N)cc1-c1cn2cnc(C(=O)Nc3ccnnc3)c2s1 Cc1cc(C(=O)NCC2CN(C(c3ccc(C#N)o3)=O)CCO2)cnc1F N1(CCC(=O)NC2COCCN(c3n[nH]c(=N)s3)C2)Cc2ccccc2C1 CC1=NOC(C)(CC2CC(n3cc(CCOC(=O)CC4CCOC4)nn3)C2)C1 N1(C(C(CCC)O)=O)CCCC(NC(C2(C(F)(F)F)CCCCC2)=O)CC1 N1(C(CCN(C(c2n(CC)ccc2)=O)CCO)=O)CCCOC(C)C1 c1(C(N2CCC3(NC(CSCCC#N)=O)C(C2)C3)=O)cc2c(F)cccc2[nH]1 N1(C(CC(CC)(C)C)=O)CCC2CN(C(c3csc(C(F)(F)F)c3)=O)CC12 C1(NC(CCC)=O)CN(C(=O)CC2CCC(F)(F)C2)Cc2ccnn2C1 c1(C(=O)N(c2ccc3n[nH]cc3c2)C)ccc2cc(Cl)ccc2c1.CC(C)(CO)SC CN1CC(O)CCC1C(=O)NCCCNC(=O)C(c1ccnn1C)O n1(C(C)C)cc(C(N2CC(C(C)NC(=O)CCc3nncs3)C2)=O)nn1 O=C(C1CCCc2nc[nH]c21)NC1CCN(C(c2cccs2)=O)C12CCCC2 c1(-c2nc(C(CC)C)nn2C(C2CCOCC2)C)cc(F)ccc1C(F)(F)F C1(C(N(C)CC2(CNC(=O)CCS(C)(=O)=O)CC2)=O)CC2CCC1CC2 C=CC(CC)C(=O)N(CC(N1CCC(C(F)(F)F)C1)=O)C1CCC1 c1(NCC(C(CC)C)O)ccc(S(=O)(=O)NC(C)(COC)CC)cc1Br c1(C(C)Nc2cccc(C(OCC)OCC)c2)cc2ccccc2o1 CC1CN(C(=O)CC2(C)CN(C(=O)C(=O)C3CC3)C2)Cc2nncn21 C(=O)(CCCC(F)(F)CO)NCC(CNC(C(C(=O)OCC)(C)C)=O)OC Cc1cc(C(N2CCC(NCc3cccc4nn(C)cc34)C2)=O)n2nccc2n1 C1(C(N)=O)(OC)CCN(C(c2ncoc2CNC(C2CCN(C)C(=O)C2)=O)=O)C1 c1(C2C(NC(=O)C(N3CCC(N4CC=CC4)C3)=O)CCCC2)ccc(Cl)c(Cl)c1 C(=O)(C1=CCC(F)(F)CC1)NC1(CC)CN(C(=O)C(c2ccccc2)C)C1 N1(C(c2c(C)nc(C3CCC3)o2)=O)CCCCCC1CNC(C12CC(F)C1C2)=O N(C(=NCCF)N1CCN(c2ccccc2)C(=O)C1)Cc1n(C)ncc1 c1(C(N2CC(NC(C(C(C)C)C)=O)C(C)(C)C2)=O)cc(Br)cc2nc[nH]c12 Nc1c(C(N2CCC(NC(C3CSCCS3)=O)C2)=O)cnn1CCO c1(C(N2C(C(=O)NCCC=C=O)COCC2)=O)ccc(F)cc1Cl N1(C(c2c(C)nco2)=O)CC2CC1C2NC(c1cc(Cn2cccn2)on1)=O C(=O)(C#CC1(C)CCCO1)NC(c1cn(C)nn1)C(=O)Nc1cn(C)nc1 N1(C(C=CCC)=O)CCC2(CCCN2C(=O)CCN2CCCCC2)C1 C(=O)(C1=CC2CCCC12)NCC(C1CC1)NC(=O)Cn1cc(C(F)(F)F)cn1 N1(C(C(C2CC2)OCC)=O)CCCC(N(C)C(c2[nH]nc(C(F)(F)F)c2C)=O)C1 c1(C(=O)NCC2N(C(c3c(C#C)c[nH]n3)=O)CCCC2C)cc(C)cc(Cl)c1N c1(NC2CN(C(C)C)C2)ccc(S(=O)(=O)NCCC2CC2)cc1C#N c1(SC)nc(N(CC(O)CN(C(=O)CCS(C)(=O)=O)C)C)cc(C)n1 n1(C(C)C(=O)NCCc2cc[nH]c2)cc(CCCN(C)C)nn1 C12(CNC(C(CCC)F)=O)CCC(NC(=O)Cc3cncs3)(CO1)C2 Cc1cccc(-c2cn(-c3ccc(C(=O)NC4COCC4CO)nc3)nn2)n1 C1(NC(CSCCN(C)C)=O)C=CCN(C(=O)COc2ccccc2F)C1 c1(C(=O)NC2CCCC2C(=O)Nc2ccc(Br)nc2Cl)cc(Br)cnc1[N+](=O)[O-] N1(C(C2N(C(C)=O)CCC2)=O)CC(F)CC1CC(=O)NCCCC(O)CO c1(C(=O)NC(CC)CNC(c2cnn(C3CCOCC3)n2)=O)cc2n(n1)CCO2 C(=O)(CC(C)CC(C)C)NC1CC(OCC(=O)NCC(C=C)O)C1 Cc1nc(C(N2CCC(CC(=O)NC(CO)C(C)O)C2)=O)cn1C O=S(=O)(c1ccc2c(c1)CCO2)NC1C2CN(Cc3ccc(Br)c(O)c3)CC12 C(=O)(CCC(C)S(C)(=O)=O)NC(CNC(c1c(N)ccc(C)c1F)=O)C1CC1 c1(C(C(=O)NCC)N2CCC2C(C)C)cc(F)cc(Br)c1OC C#Cc1cncc(C(N2CCCCC2CCNC(=O)C(C)N(CC)CC)=O)c1 Cc1ccnnc1C(=O)N(CCCCN(C(=O)CCn1cccn1)C)C c1(CCCC)ccc(C(N2CC(CNC(c3coc(C)n3)=O)CC2C)=O)cc1N N1(C(c2c(C)nn(C)n2)=O)CCCN(C(=O)CCCc2ccccc2Cl)CCC1 n1(C(C)C)ncc2c(NCc3ccn(C)n3)nc(N3CCC(C(C)O)C3)nc12 CN1CCNC(=O)C12CC(c1ccc(N3CCN(C4CCCC4)CC3)cc1)C2 Cc1cccc(Br)c1C(C(=O)N1CCC1C(C)C)NC(C1CSC1)=O n1(CC(=O)NC2CCC(NC(CCOCC)=O)C2)cc(C(=O)OC)c(O)nc1=O N1(C(CCSCC)=O)CCN(C(C)=O)C2CC12 N#Cc1cc(S(=O)(=O)NCC2SCCS2)ccc1NC(Cc1ccco1)CO C(CC(CC)CO)NC(CC1CCN(C(CC=C)=O)C1)=O C1(CNC(C(C)CN(C)C)=O)CC2CCC1N(C(c1ncc(Cl)cc1F)=O)C2 C1(C(C)C)CN(C(=O)Nc2ccccc2C2CC2(F)F)CCN1C c1(C(N2C(C)CC(c3ccoc3)C2)=O)cc(Cl)c2c(c1)CCCN2 c1(OCC(N2CCOCC(NC(C3(CF)CC3(F)F)=O)C2)=O)cccc([N+](=O)[O-])c1 C1(NC(CCSCCC)=O)COC2(CNC(c3cnc(C(C)O)s3)=O)CC1C2 N1(C(C2C(C)C2C)=O)C2CCC1C(CNC(c1cnco1)=O)C2 CC1(C)CC=C(C(=O)N(CCCC2CCCC2)CCO)CC1 Cc1cnc2c(C(=O)N(C3CC(NC(c4c(C)ncnc4C)=O)C3)C)cnn2c1 Cc1nc(C)c(C(=O)NCCNC(=O)C(c2cccc(C)c2)O)[nH]1 Cc1cc(C(N2CCC(O)(CCNC(C3CCC(O)C3)=O)C2)=O)nn1C(F)F c1(CC(=O)NCCC2CN(C(c3c(C(C)C)scn3)=O)C2)cncc(C#N)c1 CCCC(CCC)C(=O)NC1COCCC1NC(c1cccc(O)n1)=O CS(=O)CCC(=O)NCCCC1CCCN1C(=O)CC1CCCSC1 CC1(C(=O)NOCC2(C)CCSCC2)CC(O)CN1C(c1nc[nH]n1)=O CC(C)C1=NOC(C(=O)NCC(C2CCCC2)NC(c2ccc(F)c(F)c2)=O)C1 C1(NC(c2c(CC)noc2C)=O)CCN(c2ccc(OCCOC)nn2)CC1F N1(C(c2c(C)cccc2)=O)CCN(C(=O)C(N2CCSCC2)C)C(CCO)C1 C12COCCC1CC(=O)N2.C(=O)(C1=CSCS1)NCC1(OCC)CCCC1 N1(C(C)=O)CCOCC1CNC(=O)C(O)C1CCCC1.C1CCC2(CC2)C(=O)N1 C1(C(=O)CNC(=O)Nc2cccc(OCC3CC3)c2)CCC(F)(F)CC1 n1(CC(=O)NCC(CC)NC(C2COCCC2C)=O)cc(Br)ccc1=O N=c1[nH]ccc(F)c1C(=O)NC1CCOC1c1ccccc1 CC1(C)COc2c(C(=O)NCC(O)CNC(=O)C#CC3CC3)cnn2C1 CCC(C)C(O)C(=O)NCC(C(C)C)NC(=O)C=Cc1ccc[nH]1 C1(NC(c2ncn(CCNC(c3c(C#N)scc3)=O)c2)=O)CC2CCC(C1)C2O c1(C(=O)NCC2C(CC)CCN2C(=O)C(C)n2ccnn2)cnc2ccccn12 C(=O)(CCCS(C)(=O)=O)NC(C(C(C)C)C)CNC(c1cocn1)=O S(=O)(=O)(c1cccs1)N(CC(=O)NC1CCCN(C(=O)OCC)C1)C C(C(C)C(=O)NC(CNC(=O)CN1CC(C)(C)C1)C1CC1)OC(C)=O N1(C(CN(C2CC2)CC)=O)CC(C)N(C(c2cnc(C(F)F)s2)=O)CC1C C1(N(C(=O)Cc2cc(C3CC3)no2)CC)CCCN(C(c2cnco2)=O)C1 c1(C(CSC)NC(CC2(O)CCCN(C(C#C)=O)C2)=O)ccc2ncccc2c1 Cc1ccc(Cl)cc1C(N1CC(NC(=O)CC2CCC2(C)C)C1)=O Cn1cnc2cc(C(=O)NC3CN(C(c4cncs4)=O)CC3C(F)F)ncc12 c1(C(=O)NCC(CCNC(=O)C(=O)NC2CC2)OC)cc2c(nn1)CCC2 O(NC(=O)CCC1CCCCN(C(=O)CCOC2CCC2)C1)CCC C1(C(=O)NCC2N(C(CC)=O)CCCC2C)CCc2nnn(C)c2C1 C1(c2nnnn2C(C)C)(NCCOCC)CC(C)(SCc2cccc(C)c2)C1 C1(CC(=O)N(C)CC2CCCN2C(C2CCC(N(C)C)C2)=O)CCCCCC1 C1(COC)(CNC(=O)CCC(C)OC)CCN(C(C2CCCO2)=O)CC1 N1(C(c2nc(C)oc2C)=O)CC2CCN(C(C3CCS3(=O)=O)=O)C2C1C N1(C(=O)Nc2ccc(C(=O)OC)cc2F)CCC2OC(=O)OC2C1 c1(OC)ccc(S(=O)(=O)N2CCCN(C(=O)Cn3ccc(C)n3)CC2C)cc1F CN1CCN(C(c2ccc(C#N)o2)=O)CC1C(=O)NCC1CNC(=O)C1 N1(C(=O)C(C2CC2)C2CC2)CCC(C)C1.C(CC(=O)O)N(CCC1(OC)CCC1)C c1(C(=O)NCCCn2cc(C3(O)CCOCC3)nn2)nc2c(cc1Cl)OCCO2 C1(CC)(CCl)CCN(c2ccc(-n3c(C)cnc3O)cn2)C1.C(C)CS(=O)(=O)CC c1(NC(c2[nH]cc(C)c(=O)c2)=O)ccc(S(C)=O)cc1 N1(C(CCC=C(C)C)=O)CCC2(CCCN(c3nc(C)ncc3F)C2)CC1 c1(COC)ccnc(C(=O)NC(CCO)C(F)F)c1 C(C(C)(C(C)C)NC(c1csc(Cc2ccc(F)cc2)n1)=O)NC(COCC)=O C1(NC(C(CC)F)=O)CN(c2c(Cl)cc([N+](=O)[O-])cc2Cl)CCC12CCOCC2 c1(C(=O)NC2C(CC)CCC2)nc(NC(c2nccnc2OC)=O)sc1Br C(=O)(C(C(C)(C)O)NC(=O)CC(Cl)Cl)N(CCN(C)C)CC c1(CC)cc(C(=O)NCC2(NC(C3CC(=O)N(CC(C)C)C3)=O)CCC2)n(C)n1 N1(C(C(C)SCCCC)=O)C2CCC1CC(NC(c1ccccc1C(C)C)=O)C2 N1(C(c2ccc(C)[nH]2)=O)CC(NC(=O)CC2CCC(C)(C)O2)CCC1C c1(C(=O)NC2COCCN(C(c3c(C)nsc3)=O)C2)c(O)ncc2c1CCC2 C1(CNC(c2nn(CC)c(C)c2)=O)CN(C(c2ccc(F)c(N)c2)=O)CCCO1 C1(CNC(COCC)=O)CN(C(C2(c3nc(OC(C)C)no3)CC2)=O)CC1(C)C N1(c2cc(C)nc(Cl)n2)CC2(COC(CNC(C3(F)C(C)(C)C3(C)C)=O)C2)C1 c1(C(=O)NC(C)CCNC(=O)Cc2sccc2C2CC2)ccc(C(F)(F)F)cn1 N1(C(CN(c2ccc(Cl)cc2)C)=O)CC(F)(F)CC1(C)CNC(C1CCCC1)=O Cc1cccc(C)c1NC(C1(C)CCN(C(c2ccc(F)c(Cl)c2)=O)CC1)=O N1(C(c2c(OC)scc2)=O)CC(C)(C(=O)NCC2CCSC2)CC1(C)C C1(OCCCN(C)C(C2CC2NC(=O)CSC(F)F)=O)CCOC1=O CC1=C(C)CC(C(N2CC3(CC(NC(C4CCCN4C=O)=O)C3)C2)=O)CC1 CC#CCCC(=O)N1CC(C(C)NC(=O)CCc2ccccc2OC(F)(F)F)C1 O=C(CC(C(F)(F)F)NC(c1cscn1)=O)NCc1cccc(F)c1 c1(C(C(=O)NCC2CC2)N(C2(CC)CC2)C)cccc(Br)c1F c1(-c2cn(-c3ccc(OC)c(F)c3)nn2)ccc2nc(C(=O)OC)cn2c1 C1(N(CC)Cc2ccccc2C(F)(F)F)CCc2nc(C(=O)O)ncc2C1 N1(S(Cc2ccc(C)cc2)(=O)=O)CCC(F)(F)C(C(=O)Nc2cc(Br)nn2C)C1 C1(CCN(C)C)CN(C(c2ccc(Cl)o2)C(=O)NCc2ccc(F)cc2)CCO1 c1(CC)cc(C(=O)NCCC(C(C)C)NC(=O)C(C)NC(C)(C)CC)ccc1C N1(CC(=O)N(C)CC2CN(C(C(C)OCC3CC3)=O)C2)CCc2sccc2C1 C(CC(C)CCNC(c1ccnn1CC1CCCC1)=O)NC(C=CC)=O.C1CO1 N1(C(C2N(CCC)CCC2)=O)CCN(C)C(NC(C2CNC(=O)C23CC3)=O)C1 C1(OC)CC(C(N2CCC(c3cnn[nH]3)C2)=O)N(C(=O)Cc2ccc(O)cc2)C1 Cc1cccc(CC(=O)NCC(C)CNC(C2(Br)CC23CCC3)=O)c1 N1(C(C(=O)NCCCNC(C(C)C)=O)=O)CCC(C)C(C)(C)C1.C(=O)(C(C)N=[N+]=[N-])N N1(C(c2ccncn2)=O)CC(CNC(C2(F)CCOCC2)=O)C2CC12 c1(CC)ncc(C(=O)NC2(C(F)F)CC(NC(c3cccn3CC)=O)C2)c(O)n1 c1(C(=O)NC(CN(C(=O)CC2CCCN(CC)C2)CC)C)ccc(OC)cc1F C12(CNC(CN3CCN(CC)CC3)=O)CCCCC1N(C(=O)C=CC(C)C)CC2 N1(C(c2c(C)ccnn2)=O)CCN(C(C2CCN(C(N)=O)CC2)=O)CC(C)(F)C1 c1(N2CC=CC(OC)C2)nc(N2CCN(C)C(C(C)(C)C)C2)nc2c1COC2 Cc1[nH]c2cnc(Cl)cc2c1C(N1CCOC(C(C)NC(=O)C(C)C2CC2)C1)=O CN1CCC2CN(C(C3CC4CC4N3C(c3cccc(CO)c3)=O)=O)CC12 C=C=CC(C)C(=O)NCC1CCN(C(=O)Nc2cc(-c3ccc(F)cc3)no2)C1 CCC(CNC(=O)NC(c1ccc(C)c(C)c1)C)C(C)(F)F C1(F)(CNC(CC2(C=C)CCC2)=O)CCCN(C(c2ccnnc2O)=O)C1 CN1CCN(C(C2CCOCCN2C(=O)C=CC2CCOC2)=O)CC12CC2 N1(CC(N2CCN(C(CSc3ccc(OC)cc3)=O)CC2)=O)C(=O)CN(C)C1=O C1(F)(CNC(C(CC)Cc2ccc(N)cc2)=O)CCN(C(C2CC2F)=O)CC1 C1(NC(C2CN(C)CC(C)O2)=O)COC2(C1)CN(C(c1cccc(N)c1N)=O)C2 C1(NC(CCC(C)SC)=O)CCCCC12CCN(C(C1C(CC)C1(F)F)=O)C2 C1(C2CCC(=O)NC2)(C(N(C)CC2CCN2C(=O)CC(C)(C)C2CC2)=O)CCC1 C1(CNC(C2(NC(C)=O)CCC2)=O)CC2(CC2)CN1C(C1C2CC3C(C2)C13)=O Cc1c(N2CC(N3CCCC3)C(C)C2)ncnc1N1CCCC(c2cn[nH]c2)C1 C1(C(=O)NCC(CC(C)C)(C)O)CN(C(=O)C(=O)NCC2CC2)CCC1(C)C C1(CNC(C=CCC)=O)CC2CCC1N(C(=O)C(C1CC1)C1CC1)C2 N(C1CCCc2n[nH]cc21)C(C1C(NC(C(CC)NC(N)=O)=O)C1(C)C)=O C1(NC(C(CC)O)=O)CCN(C(=O)CCc2ccc(C)cc2)C12CC2 C12(NC(c3ccc(C)c(C)n3)=O)CCCC1N(C(C1CCN(C)CC1)=O)CC2 CC(C)C(CC(=O)NC1CN(C(c2ccnc(Cl)c2O)=O)CC1C)C(C)C Cc1ccc(C(N2CCC(c3nnc(C(F)F)o3)C2)C(=O)N(C)C)cc1 c1(C(N(CCN(C(=O)C=C2CCN(C)C2)CC)CC)=O)ccnc(C2CC2)c1 c1(C(=O)NCC(CNC(C(c2ccccc2F)OC)=O)F)cccc(SC)n1 N1(C(C(=Cc2ccco2)C)=O)CCCC(NC(c2ccsn2)=O)CC1 c1(C(=O)Nc2c(C(N3CCCC(OC)C3)=O)scc2)ccc2n[nH]cc2c1 N1(C(=O)C=CC2CCCCC2)CCN(Cc2cccc(Br)c2)C(CO)C1 c1(CC(=O)NCC(CN(C(C2CCC(=C)CC2)=O)C)C)ccc(Cl)cc1F C(=O)(C(C)S(N)(=O)=O)N1CCC(C(=O)NCC(C(C)C)(C)F)(CF)C1 c1(C(N2CCC(CO)(CNC(C3CC(O)C3)=O)CC2)=O)cccc(Cl)c1O c1(Sc2cc(NCCCOC)nc(-n3c(CC)nnc3CC)n2)ccccc1[N+](=O)[O-] c1(C(=O)NCC2N(C(CCSC)=O)CCCC2C)ccc(S(=O)(=O)NC)o1 CC(C)CC(C(=O)N1CC(NC(C2(CN(C)C)CC2)=O)CC(O)C1)N(C)C C(=O)(C(F)C(C)CNC(=O)C=CC(F)F)N1CC(NC(=O)OC)C1 N1(C(c2cc(OC)no2)=O)CCCCC(NC(C2CCC(F)(F)C2)=O)C1 C1(C(N2CCC(COCC)C2)=O)CC2CC1CN(C(C1CC13CCC3)=O)C2 C1(CC(=O)NCC2CCN(CCC3CC3(Cl)Cl)CC2)NC(=O)NC1=O c1(C(=O)NC2CN(C(CC=C=C)=O)CC(O)C2)ccc(C)c(F)c1N C12(C(N3CC(CC(C)NC(c4cncnc4)=O)C3)=O)CC3CC(C(=O)N1)C2C3 CC(C)(C)C(CO)C(=O)NCC1C(O)C(O)CN1C(c1ncncc1Cl)=O C1(C(=O)NCC2(CC(F)F)CCC2)CCN(C(c2cccc(O)n2)=O)CC1 N1(C(C(C)CC(F)F)=O)CCC2(NC(c3ncoc3-c3cccs3)=O)CCCC12 c1(C(N2CC(CNC(CC(=C)C)=O)C(C(F)(F)F)CC2)=O)ccc(Cl)c(F)c1F C1(C(=O)N(CCCC(=O)NCc2cccnc2Cl)C)(CC)CCCC1O C1(C(N2CC(N(C(=O)COc3ccon3)C)C(O)C2)=O)CCC(C2CC2)CC1 c1cc(C)cc(C)n1.C12CCC(CC1)CNC2=O.CCC(C)NC(=O)N C(=O)(CCC1=CCCCC1)NC1CN(C(c2cc(C)n(C)c2C)=O)CC1(C)C c1(CC(C(=O)OC)NCc2coc(=N)[nH]2)ccc(C)c(C)c1 N1(C(c2cc(CC)nn2C)=O)CC(NC(c2cccnc2S)=O)CCC1C C1(CNC(C(C)S(C)(=O)=O)=O)CC12CCN(C(c1cc(CO)on1)=O)CC2 C=CCC(CC)C(=O)NCc1ccnc(C(=O)NCC2CCCC(C)O2)c1 N1(C(C(C(C)(C)O)F)=O)CCN(C(c2coc3c2COC3)=O)C2CCCC12 N1(C(C(CC)N(C)C)=O)CCC(CC(C)NC(c2cnns2)=O)CC1 Cc1ccc(SCC(=O)NC2CC(N(C)C(c3ccncc3N)=O)C2)cc1 N1(C(C(CSC)C)=O)CCCC(N(C)C(C2CCCC(=O)N2)=O)CC1 N1(C(CC2CCC(NC(c3c(OC)nccc3)=O)CC2)=O)C2CCCC1COC2 c1(CC(=O)NCCC(C)NC(c2cc(OCC)n[nH]2)=O)nc(C)sc1Cl N1(C(=O)NCC2(C(C)C)CCC2)C(N2CCCC2)CC1C N1(C(CC2(NC(=O)OC)CCC2)=O)CC2(CO)CC1(C(=O)NC1CC1F)C2 c1(C(=O)NC(CC)(C)CNC(=O)C(C)Cc2cnn(C)c2)cc(O)n(C)n1 C1(NC(C2CC(CC)(CC)C2)=O)CN(C(C2(C(C)(F)F)CC2)=O)CC1F CC1CC=C(C(=O)N2CC3CC2(CNC(=O)CCOC2CCOC2)C3)CC1 Cc1cc(=O)n(C)nc1C(=O)NC1CCCC1NC(=O)COC1CCOC1 C1(NC(C2CC(C)C2)=O)CCC(N=c2cc(C(F)(F)F)nc(Cl)[nH]2)CC1 N1(C(C(N)=O)=O)CCC2(CCCC2CNC(C2CCn3cncc3C2)=O)CC1 c1(N(CC(=C)C)C)nnc(-c2ccc[nH]2)n1CC(=O)NCCC1CC1 N1(C(c2cc(COC)no2)=O)CCCC2(CCCN2C(C2CC2F)=O)C1 N1(C(C(COCC)NC(=O)CSC(F)F)=O)C(=O)CNC1=O.C1CN1 C(=O)(CCCCC(N)=O)NCC(C1CCN(C(c2c(C)cc(CC)o2)=O)CC1)C C1(CC=C)(C(N2CCC(C(C)(C)C)CC2)=O)CCCN1C(=O)COCCCC=C c1(C(=O)OC(C)C)ccc(S(=O)(=O)N2CC3(CCCN3C(=O)C(C)CN)C2)cc1 Cc1c(Cl)ccnc1CNC(C1CCCN1C(=O)C(C(C)C)N1CCCCC1)=O CC1CCc2nc(Cl)nc(N(C)CC3CCN(C(C45CCC(CC4)C5)=O)C3)c2C1 N(C(=NCCCCl)N1CCN(S(=O)(=O)c2cccs2)CC1)CC1CC(C)C1 CC#CCCCC(=O)N1CCC(C(=O)Nc2ccc(F)c(C)c2F)O1 c1(NCc2cccc(O)c2)nc(C(F)(F)F)n2ccncc12 C(N=c1[nH]c(=NCC2(Cl)CC2(F)F)c2[nH]ccc2[nH]1)c1cc(C)oc1C C(=O)(C1=CCCN(C(=O)C#CC2(C)COC2)C1)NCC1(C)N=C(C)SC1 C1(NC(CC2(COC)CC2)=O)CCC(n2cc(-c3ncccc3N)nn2)CC1 Cc1cc(F)ncc1C(N1C2CN(C(c3ncsc3Br)=O)CC12)=O c1(C(CC)NC(N(C(C#C)C)C2CC2)=O)ccc(Cl)cc1Cl c1(CNC(=O)CCOCCOCc2ccccc2)ccc2c(c1)CC(=O)N2 C(CC(C)C)(C(=O)N(c1cc(OC)cc(C)c1)CCC)OC C1(F)(CNC(CN(C)C2CC2)=O)CC(NC(=O)Cc2ccsc2)C1 C(CC(C)(C)C)(C(=O)N1CCC(C)(C)C1C(=O)NCC(c1nccs1)C)OC n1(CC(C)C)cc(CNC(c2nnnn2C2CC2)CCc2nccs2)nn1 CCC(C(=O)N(CCN(C(=O)CSCc1cccnc1)C)C1CC1)C(C)C C12CCCCC1OCC(=O)N2.c1(CC(C(=O)O)SCC)cccc(C)c1 c1(OC)ccc(OC)c(C(N2CCC(F)(CNC(=O)CNS(=O)(=O)C3CC3)C2)=O)n1 C1(C(=O)NCC(CC)NC(c2c(Cl)ccc(C)c2N)=O)CCC([N+](=O)[O-])CC1 C1(C(=O)NCC(C)(O)CO)(COC)C=CCN1C(c1csnc1C)=O c1(C(N2CCCC(CC)CC2)C(=O)NCC=C)ccc(C)cc1Cl c1(OC)cc(C(=O)NC2CN(C(c3cc(N)ccc3C)=O)C3CC23)ccc1Br N#CC1CCC(C(=O)NC2CC(OCC(=O)NCCCC3CC=CC3)C2)C1 CC1(C)CCN(C(c2cc[nH]n2)=O)CC1CNC(=O)C(C#N)C1CC1 C1(CNC(C=CC=CC)=O)CN(C(=O)Cc2conc2C)CC1O C1(C(N2CC(C(C)NC(Cn3c(C)cnc3)=O)C2)=O)C(C(F)(F)F)C1[N+](=O)[O-] C1(c2ccccc2)(NC(C(CO)OC)=O)CCN(C(=O)CCc2nc(O)n[nH]2)C1 N1(C(c2c(OC)nccn2)=O)CC2CCCC2(C(=O)NCc2ncoc2CO)C1 N1(C(c2cnc(CC)s2)=O)CCOCC1CC(=O)NCCC[Si](C)(C)C c1(CNC(=NCCCCC)NC2CC3CCC(C2)N3CC)cc(O)c2ccoc2c1 c1(OC)nc(C)cc(=NC2C3CC2CN(C(c2cc(C)nn2C)=O)C3)[nH]1 C(=O)(C(C(C)NC(=O)CC1CCC(C)(C)O1)C(C)C)N(CCCC=C)C N1(C(Cc2ncc(CC)[nH]2)=O)CCC(C)(CNC(=O)C(C)(C)c2cncs2)CC1 CCCCCCC(CC)C(=O)NCC1(C)CCCN(C(=O)Cc2ccc(C)s2)C1 c1(CC(N2C(CCCNC(C(CC)(C)F)=O)CCC2)=O)nn(C)cc1[N+](=O)[O-] C1(CC)CCC(c2cccs2)CC1.C12(C)CC(C1)NC2c1nnnn1CCOC c1(CN2CCN(C(C3CNCCO3)=O)CC2)cc(F)cc(I)c1 c1(OC)ccc(C(=O)C(=O)NC2CCCN(C(C3CC3(C)C)=O)CC2)cc1OC CCC(CNC(=O)C(F)CC(C)(C)C)(CC)C(=O)Nc1cn(CCF)nc1C C1(NC(c2cc(COC)no2)=O)CCN(C(c2cc(Cl)cn2C)=O)C1C CCCCC(CC)C(=O)NCCC(C)N(C)C(c1cnc2n1CCS2)=O C=CCC(CNC(C1C=C(C)CS1)=O)C(=O)NC(c1ccc(O)cc1)C NS(=O)(=O)CC(=O)N1CC(O)(CCNC(=O)CS(=O)(=O)NC2CC2)C1 C(=O)(N=c1cc(-c2ccc(Br)cc2)[nH][nH]1)c1cc(OCC)c(O)cc1 CCC(C)C(O)C(C)C(=O)NCC(C)=CC(=O)NC(C)CC1CC1 c1(C(=O)NCC2CCC(NC(c3c(CCC)n(C)nc3)=O)C2)cccc(C)c1O CC1CN2CCN1CC2C(N1CCCC(n2cc(CCC(=O)CCO)nn2)C1)=O C1(CC)CCCC(CNC(c2ccc(O)cc2)C(F)(F)F)C1 C(=O)(CCC(C)(F)F)N(C)CC1N(C(CC=CCC)=O)CCOC1 N1(C(Cc2cncc(OC)c2)=O)CC2CCC(C1)C2C(=O)Nc1cc(O)ncn1 C1(NC(c2cnn3ccsc23)=O)COC2(C1)CN(C(=O)CCC1CC1(F)F)C2 CCC(C)CCCCC(=O)N(C1CN(C(c2cnsn2)=O)CC12CC2)C N1(C(Cc2ncc(C)[nH]2)=O)C2CCCC1CC(NC(C1CCCCO1)=O)C2 c1(NC(C(CC(=C)Cl)NC(c2cc(C3CC3)[nH]n2)=O)=O)cccc2c1CCC2 C(CC(=O)NC1CC(NC(=O)COc2nn(C)cc2[N+](=O)[O-])C1)(C(F)(F)F)OC C(=O)(CC1C(=O)Nc2ccccc21)NCC1CN(C(C2CC2F)=O)CC(C)(C)O1 OCC(CN=c1[nH]c(=NCc2cncs2)[nH]c2c1CCC2)C1CCOC1 c1(CCC(=O)OC(C)C(=O)N(c2ccccc2Cl)C2CC2)cccc(S(N)(=O)=O)c1 c1(C(=O)NC2CN(C(=O)C3CC3)CCC2(F)F)cc(F)c([N+](=O)[O-])cc1F C1(NC(N2CCN(C)CC2)=O)CCCN1N1CCc2ncsc2C1 CC1CN(C(C2COC(=O)C2)=O)CCCN1C(=O)C=CSc1ccccc1 C=C=CCCC(=O)NCCC(C(=O)NCC(c1cnc[nH]1)C)OC c1(SCCC)ccccc1C(=O)NCC1CN(C(=O)CC2CC(C)(C)C2)CC1C c1(CNC(c2ccn(CCC)n2)=O)cccc2c1CCN(C(C1CC1CC)=O)C2 N1(C(C2CCC(CNC(CCC=CC)=O)O2)=O)CC(OC)C2(CC2)C1 Cc1ccc(C(N2CCSCC2CCNC(=O)CC(F)(F)Br)=O)cc1N Cc1cc(C(=O)Nc2cccc(NC(=O)NC(c3cccs3)C)c2)ccc1Cl N1(C(C(C2CC2)OC)=O)CC2CC1C2NC(c1cn(C)nc1-c1nccs1)=O c1(NC(CCC2CCN(C(CC(C=C)CC)=O)C2)=O)cccc2ccoc12 n1(CC(=O)NC2CCN(C(C(C(C)C)n3ccnc3)=O)C2)cc(Br)ccc1=O CC1CCN(C(=O)C=CI)CCN1C(C12CC(C)C1C2)=O C1(NC(COCCC)=O)CCN(C(=O)C=C(C)C)CC1F.c12cccnc1OC2 CCC(CC)C(C)C(=O)NCC1CCCCN(C(=O)C(C)(C)CCCF)C1 CC(CC(=O)NCC1CC2CCC1O2)C(C)(C)NC(C1(C)CC(F)(F)C1)=O C1(C)(NC(C=C(C)CNC(=O)C(C)CC(C)C)=O)CCCC1(F)F c1(C(=O)NCC(C2CCN(C(=O)C3=CCC3)CC2)C)cc(Cl)cc(F)c1F C=CCC(CNC(c1sccc1OC)=O)C(=O)N1CCCC(C(C)C)CC1 N1(C(CC2(CC)CCC2)=O)CCN(C(=O)C(C)CC(OC)OC)C(CO)C1 c1(OCC)nc(Cl)ccc1C(=O)NCCC1(CNC(C2CCO2)=O)CC1 C1(C(=O)OC)(C(=O)NCCCOCCNC(=O)Cc2cscn2)CC1C.C(CO)S c1(CN(C(=O)CCC2(C)CN(C(=O)CC3C=CCCC3)C2)C)cc(CO)cs1 CC(C(=O)NCc1cn(C2CCN(C(=O)CC3(C)OCCO3)C2)nn1)S(N)(=O)=O C12(C(=O)NCC3C(C)(C)CN(C(=O)Cc4ccsc4)C3)CCC(CC1)C2(C)C N1(Cc2ccc(OC)cc2Br)CC(C)(C)C(O)C(C)(C)C1 c1(C(N2CCN(C3CC3)C(c3cn[nH]c3)C2)=O)ccc(-c2ccncc2)c(F)c1 Cc1c(C(F)(F)F)nn(C)c1NC(C1CCN1CC1(C2CC2)CC1)=O CCCC(C)C(=O)N1CCC(CO)(NC(=O)C(O)C2CC2)C1 C(=O)(C(CNC(=O)CCCC1CC1C)(CC)CC)N1CCC(OC)CC1 C1(C(=O)NCC(CNC(c2cc(C)[nH]c2)=O)C)CCc2nnc(C)n2C1 N1(C(C2(CC)CCCCC2)=O)CCC(NC(=O)CCCCOC(C)=O)C2(CCC2)C1 N1(C(C2(C)CCOCC2)=O)CC(C2CCN(C(=O)NC(=O)C(Cl)(Cl)Cl)CC2)C1 CC(C)CC(CNC(c1nc[nH]c1C(C)(C)C)=O)NC(C1(S(N)(=O)=O)CC1)=O c1(OCC)cnc(C(N2CC(NC(C3CC4(CCC4)C3)=O)CC(O)C2)=O)c(Cl)c1 c12nc(ncc1Cl)NCCCOCCNC2=O.c1(C(=O)OC)ccc(OC)nc1 c1(C(=O)NCC(C)CNC(C2CC2C)=O)csc(C2CCCCC2)c1 c1(C(=O)NC(C(=O)Nc2c(CC)ncnc2)Cn2cccn2)cc(F)ccc1O C#CCC(C)(C)C(=O)NCC(C1(O)CCN(C(c2c(F)cncc2Cl)=O)C1)C C1(C(N2C(CCC(=O)NC3CCCC(CF)C3)CCC2)=O)CCC2(CC1)N=N2 N1(C(CCOCCC)=O)CC2CC(NC(=O)CC34CCC(C)(C3)OC4)C1C2 CCCC(C)(CC)C(=O)NC1CCC(N(C)C(c2ccc(Cl)c(N)c2Cl)=O)CC1 C1(NC(C(C(C)C)NC(c2ccc(=N)[nH]n2)=O)=O)CC12CCCCCC2 N1(C(C2(OCC)CCOCC2)=O)CCN(C)C(CNC(c2cnoc2C)=O)C1 CC1CN(C(=O)CCc2cncc(F)c2)CCN1c1ncc(C#N)cn1 c1(NC(CCC=C)Cc2ccccn2)ccc(C2CCC2)cn1 C1(C)(CC(=O)NC2C(C(N(C3CCN(CC)C3)CC)=O)C2(C)C)CCCCO1 C=CC1(CC(=O)N(CCCC)C)CN(C(=O)COCC2CC2)C1 C1(C(=O)NCC2(CCNC(c3cnn(CC4CCCO4)c3)=O)CC2)C=CCCC1 c1(C(=O)NC(CCCNC(C(C)N(C(C)=O)C)=O)C)nc(O)sc1C C=CC1(CC(=O)NCCC2CCC(NC(=O)C=Cc3cccs3)C2)CCC1 CCC(CCCC(=O)NC(CO)CCCO)NC(=O)CCC(Cl)Cl c1(NC(C2CCCCN2C(c2cnc(O)cc2O)=O)=O)nccn2ccnc12 c1(C2(C(N(CC(C)NC(=O)CNS(C)(=O)=O)C)=O)CC2)cc(Br)ccn1 N1(C(C2N(CC(C)(C)C)CC2)=O)CCC(n2cc(CNC=O)nn2)C1 c1(C(=O)NC(CC)(CNC(=O)CSCc2cccs2)CC)cc2[nH]ccc2s1 C1(=CC(=O)NCCN(C(C2(O)COC2)=O)CC2CC2)C2CC3CC(C2)CC1C3 c1(C(=O)NC2CCC(CNC(=O)CC3CCS(=O)(=O)C3)C2)nc2c(s1)COCC2 N1(C(c2cccc(SC)c2)=O)CCC(NC(C23CCCC2C3)=O)C(C)(C)C1 C1(CNC(C(CC=C)(C)C)=O)COC(C)(C)CN1C(c1cnn(C)c1SC)=O C1(C(C)NC(C2(OC)CCC2)=O)CCCN1C(c1cc(C)[nH]n1)=O Cc1ccc(C(N2CCC(CCC(=O)NCc3ccncc3C)C2)=O)n1C c1(CNC(CCC2CCC(NC(Cn3ncc(C)c3)=O)C2)=O)cccnc1F C1(C(=O)N(C(C)CNC(=O)CCc2ncccn2)C)(CC)CCCC1 C1(CC(=O)N(CCCCC)C)CC(NC(C2SCC=C2C)=O)C1(C)C N1(C(C(Cn2cncn2)NC(C2CCN(C)CC2)=O)=O)CC2CC1C1CC21 C1(NC(c2c(C)ncc(C)c2)=O)CN(C(c2cncs2)=O)C2(CCC2)C1 C1(CC(=O)NCC(CCC)NC(c2conc2C(C)(C)C)=O)CCC=CCC1 N1(C(c2cc(C)c(O)nc2)=O)CC2CN(C(c3ccn(C(F)F)n3)=O)CC(C1)O2 N1(C(C(C)N(CCC)C(C2CC2C2(C)COC2)=O)=O)CCOC2COCC2C1 CCC(C(=O)N1CCCC(C(=O)NC(c2cc(C)on2)C)(CC)C1)C(C)(C)CC c1(OCC)cccc(C(=O)NCC2CN(C3CCCCCC3)C2)c1Cl C1(CC(=O)NC(C(=O)NC(C)CC2CCCO2)(C)C2CCC2)CCCN(C)C1 c1(C(=O)NCC(CNC(C2C(COC)C2)=O)O)sccc1Br C(CC(=O)NNC(=O)NC(c1ccccc1)C)N1CC(C)C(C)C1 C1(NC(Cc2n(C)nnc2)=O)CC(C(=O)NCCN2CCCC(O)C2)=CC1O C(=O)(CCCCC(F)F)NC1CCCCN(C(c2c(N)nccc2)=O)C1 Cc1ccccc1C(N1CCCC(N(C(=O)Cc2nc[nH]n2)CCN(C)C)C1)=O c1(C(N2CCC(CC)C2CNC(=O)CC(C)(C)N(C)C)=O)nsc2ccccc12 S(=O)(=O)(c1ccc(Br)c(F)c1F)NCC1N(C(C(C(C)C)O)=O)CCOC1 N1(C(c2ccc(N(C)C)nc2)C(=O)NCC(F)F)CC2C3CCC(C3)C12 C1(C(N2CC(C(N3CCCOC(CC)C3)=O)(CC)C2)=O)OCC2CCCC12 C1(NC(C2CCC(CNC(CCSC)=O)O2)=O)CN(C(C)C)CC1C N1(C(C2C(CC)OCCC2)=O)CCC(CNC(c2ccc(C)nc2C)=O)C12CC2 C(c1nc(NC(=O)C(C)N)cs1)=CC(=O)OC Cc1cc(C(N2CC(NC(=O)CC3CCOC3=O)C(C)(C)C2)=O)cc(Br)c1 c1(C(=O)NC(C(C)(C)NC(c2c(CCC)occ2)=O)C)nc(Cl)sc1Cl C1(C(N2Cc3c[nH]nc3C2)=O)CCC2CCC1N2C(=O)C(F)C(F)(F)F c1(C(N2CCCC(NC(C=C(C)C)=O)C2)=O)cccc(S(=O)(=O)NCC2CC2)c1 c1(COC)ccccc1OC.C1C(O)CC(=O)N1C C(C(C(=O)NC(c1ccc(Cl)cc1)C)N(CCC(C)C)C)(C1CCCC1)OC C1(CNC(=O)C=Cc2ccccn2)CC2(CCN(C(=O)CO)C2)CO1 C1(NCc2c(F)cc(OCc3ccccc3)cc2)CCC2(CCNCC2)O1 c1(C(N2CCCC(C(C)Nc3cccc(C(F)(F)F)c3)C2)=O)cc(C)c(Br)cn1 C1(C(=O)NCCOC(c2c(OC)scc2)=O)CCN(C(=O)CCc2cnc[nH]2)CC1 C12(C(N3CCC(N(C(CNC(CNC(C)=O)=O)=O)C)C3)=O)CCCC(C)(C1)OC2 CN1CC=C(CC(=O)NC2CCOCC2NC(c2cnnn2C2CC2)=O)CC1 C(=O)(C1=CNC2=NCCC2=C1)N1CC(OCCNC(c2c(C)cccn2)=O)C1 O=C(N=c1c(F)c[nH]cc1Cl)CCCSC(F)F.C1CN1 N1(C(C=CCC)=O)CC(CNC(c2c[nH]cc2C)=O)C(C)C1 C(=O)(C(CO)C(C)(C)C)N1C2C(CNC(c3cc(CC)c(O)cc3)=O)C(CC2)C1 C(N=c1[nH]cnc2cc(F)c(F)cc12)C1(NC(CC(COC)OC)=O)CC1 C1(CNC(CCC(=C)C)=O)CN(C(=O)C(C)OCCc2ccccc2)CC1(C)C C(=O)(CCCN=[N+]=[N-])N(C1CCCN(C(c2c(C)cc[nH]c2=N)=O)CC1)CC N1(C(C2(C)COC2)=O)CCC2CN(C(c3ccc(I)cc3)=O)CCC12 Cc1cccc2cc(CC(=O)NCC3CCCN3Cc3c(F)cccc3F)[nH]c12 c1(C(N2CC(NC(=O)Cn3nccn3)C(F)C2)=O)c(F)ccc(Br)c1F N1(C(=O)OC)CCCC(C(=O)N(CCCNC(=O)C(C2(O)CCCC2)F)C)C1 C1(CNC(C(C)C)=O)CCN(c2cc(NC3CCC(O)C3)ncn2)CC1 C(=O)(C1CC(=O)Nc2ncccc21)NCCNC(c1[nH]c2ccn(C)c2c1)=O c1(C(N2C(C(N(C(C#C)C)C)=O)C(O)CC2)=O)ccc2c[nH]nc2c1 N1(C(C(C)NC(CC)=O)=O)CCCC(C2CCCN(Cc3noc(C4CC4)n3)C2)C1 c1(C(c2nnnn2C(C)C)NCCc2nc(CC)sc2)n[nH]c2c1COCC2 c1(C(N(CCCN(C(=O)Cc2cc(Cl)cs2)C)C)=O)cncn(C)c1=O N1(C(C2(C(=O)OC)CC2)=O)CCC(C)N(C(=O)Cn2cnc(C#N)n2)CC1 C1(F)(CNC(C(C)OC)=O)CC(NC(=O)Cc2[nH]cnc2C)C1 C12(C(N3CC(C)N(C(c4cc(F)cc(Cl)c4N)=O)CC3)=O)CCCCC1C2(F)F C1(CNC(Cn2c(C)c(Cl)cn2)=O)C2CCC(C2)N1C(c1cnc(O)cc1O)=O c1(OC)ccc(O)c(C(=O)NC(c2ccc(-c3cnn(C4CC4)c3)cc2)C)c1 N1(C(C2ON=C(C(C)C)C2)=O)CCC2C(CCCN2C(=O)C=CCN2CCCC2)C1 c1(C(=O)NC2CC(C(CC(N3CCC(CC(C)C)C3)=O)C)C2)cc2n(n1)CCO2 C(C1c2ccsc2CCN1C(c1ccc(C(C)(F)F)cn1)=O)NC(C1C(C)C1)=O N1(C(c2c(C(C)(C)C)ocn2)=O)CCCC2C1CCN2C(C1CC1(C)C)=O c1(OC)cc(NC(=O)C(C)N(C)C)nc(NC2CCC(NC)CO2)n1 c12c[nH]cc1C2c1nnnn1-c1ccccc1.NS(=O)(=O)NCCCN CC(C)(CC(=O)N1CC(CC(F)C(=O)NCC(c2nn[nH]n2)Cl)C1)C(F)F c1(CN2CCCC(C(=O)NCCCCCN(C)C)C2)ccnc(F)c1Cl c1(C(=O)NCc2cc(C(=O)NC(C)C(C)(C)O)on2)cc2ccccn2n1 C1(CNC(C(CC)O)=O)CCCN(C(=O)CCCOC(C)C)C1 N1(CCN)CCCNC1=O.O=C(C=CSc1nc[nH]n1)N1CC(C2C(=O)N2)C1 N1(C(COCC)=O)CC2CCC(C1)N2C(=O)C(C1CCOCC1)C N1C(=NCCCF)NCC2CCCC12.C1(S(=O)(=O)N2CCOCC2)(CC#N)CC1 C1(OC)CC(NC(=O)C(CC(C)C)NC(N)=O)CN(C(=O)C(C)(O)C2CC2)C1 N1(C(C(c2ccc(C)o2)C)=O)CC2CCN(C(C34CC5CC3C4C5O)=O)CC12 C12(C(N3C(C(C)(C)NC(C4CC4(F)F)=O)CCC3)=O)CCC(C1)OC2 C12(C(N3C4(CNC(C(C(=O)NC)(C)C)=O)CCC3CC4)=O)CC=CCN1CCC2 c1(CC)ccc2c(C(N3CCC(CNC(=O)C(C)C(C)C)C(O)C3)=O)coc2c1 C(N=c1[nH]c(=NCCc2cn[nH]c2)[nH]c2c1CCCCC2)C1CCCCO1 N1(C(C)=O)CCC2(CC1)COC(CNC(c1ccc3nnc(S)n3c1)=O)C2 Cc1cc(O)cc(=O)n1CC(=O)NCC1(C)COCCN(C(C2(C)CCC2)=O)C1 Cc1ncnc(C(N2CCC(NC(c3[nH]nnc3C)=O)C2)=O)c1C CCCC(C)CCCC(=O)N1CC(NC(c2cncc(OCC3CCC3)c2)=O)C1 N1(C(c2c(C)nsc2)=O)CCCC2(NC(=O)CCN3CCOCC3)CCCC12 N12CCOCC1C(=O)OCCCCC2.C(=O)(CC(=O)Nc1ccccc1)NC C(=O)(C=CS(C)(=O)=O)N(C1CCC(NC(c2cnncc2O)=O)CC1)C CC(C)C1=CCC(c2nc(C(C)(C)C)nn2C)CC1 c1(C(N2CC(C)(NC(C3N(C(C)=O)CC(O)C3)=O)C2)=O)cnc(O)cc1C N1(CC)CCc2cc(NCc3c[nH]nc3C(C)(C)C)ccc21 C1(CC(N2C(COC)CCC2)=O)N(C(c2c[nH]c(=O)cn2)=O)CCC1(C)C c1(C(=O)NC(C)CCNC(C2CS(=O)(=O)C2)=O)ncn2c1CCC2 C1(CNC(CC(C=C)CC)=O)CCCC2(CN(C(=O)CSC(F)F)C2)O1 N1(C(c2scc(CNC(C=CC)=O)c2)=O)CCOCC1COC c1(C(N2CCC(CNC(C(C)(C)C)=O)CC2)=O)cc(F)c(Br)cc1[N+](=O)[O-] Cc1c(C(=O)NCC2(C)CCCN2C(=O)C=Cc2ccccc2)cncc1Cl c1(CC(=O)N(C(C)C)CCN(C(=O)CN(c2ccccc2)C)C)ccc(Cl)cn1 C1(CCCC)(C(=O)NCCN(C(=O)C=C(C)Cl)C)CCC1 N1(C(C(CC(=O)OC)C)=O)C2CC=C(C(=O)N3CCC(F)(F)C3)C1CC2 C1(c2cn(CC(C)NC(C3CC3C3CCOC3)=O)nn2)(COC)CCCO1 N1(C(CCCCCOC)=O)C2CCC1CC(NC(C13CCC(CC1)O3)=O)C2 CC1CN(C(C2(C#N)CC2)=O)CC1CCNC(c1ccc(CO)cc1)=O C1(CC)CCCN(C(=O)C(C)NC(C2CCC(=O)N2)=O)CC1 c1(OC)cc(C(=O)NC(C)(CNC(=O)C(C)C2CC2)CC(C)C)c(Cl)cc1Cl c1(C(N2CCC(C)(CNC(CCCOC(C)=O)=O)C2)=O)c(C)nn(CCO)c1C C1(CN(C(C(C)OC)=O)C)CN(C(c2ccc(CC(N)=O)cc2)=O)CC12CC2 CC1CCC=C1C(=O)N1CC(CC(C)NC(=O)C=Cc2ccccc2)C1 c1(OC)cnc(C(=O)N(CC(O)CNC(c2ncccc2C(F)(F)F)=O)C)cn1 N1(C(Cn2nc(C)oc2=O)=O)CCCC(NC(C2CC23CCCC3)=O)CC1 N1(C(c2nc(C)sc2)=O)CCC(C)CC1CNC(=O)CC1(O)CCCCC1 C1(CC(=O)NCC2CCCN2C(=O)Cn2nnc(-c3cccs3)n2)CC2CC1C2 c1(C(N2C(C3(NC(C=CCOC)=O)CC3)CCC2)=O)cc(C)c(F)cc1C N1(C2(C(=O)NC(=O)OC(C)(C)C)CC2)CC2C3CCC(C3)C2(C)C1 C12=CN=C(Cl)NC1=NCC1CCCC(C1)O2.n1(CC(=O)NCC)ccsc1=N C1(C(=O)NC2CCC2CNC2CC2)CSCN1C(=O)Cn1nnc(C(F)F)n1 C1(OC)C(NC(=O)NCCc2cc[nH]n2)COC12CCC2 c1(C(=O)NCC(C)(C(C)C)NC(C(C(C)C)C)=O)c[nH]c(=O)c2ccnn12 Cc1cc(NC(c2cn(C)nc2-c2ccco2)=O)ccc1NC(=O)C(F)C(C)C c1(C(=O)NCCOC2CCOCC2)cc(NC2CC2)cc(Br)c1 N1(C(CCN(CCC)C)=O)CC2CCC1CN2C(C12COC(CC)(C1)C2)=O C1(CNC(CNC(N)=O)=O)CC(F)CN1C(C1CCSCC1)=O CCC(O)C(C)C(=O)NCc1cccc(CNC(c2cc(C)no2)=O)c1 c1(C(=O)NCC2(O)CN(C(c3nn(CC)c(O)c3)=O)C2)c(Cl)cccc1Cl c1(CC2(CNC(C3(N(C)CC)CC3)=O)CC2)ccccc1.C1(C)C(=O)N1 N1(C(CCc2ccc(C)o2)=O)CCC2(CCN(C(=O)C(C)(Cl)Cl)C2)C1 CCCC(CC)C(=O)NCC1CCCN(C(c2ccc(N)c(SC)c2)=O)CC1 c1(CN2C(CC(N3CC(C(=O)OC)NC(=O)C3)=O)CCC2)onc2ccccc12 C(=O)(C1=C(Cl)CCCC1)N1C(C2CCN(C(CCOCCOCC)=O)C2)CCC1 c1(OC)cc(C(=O)NC(C)CCNC(=O)C(C(C)C)OC)cc(F)n1 CN1CCN(C(C2COCCC2NC(=O)Cc2cnsc2)=O)CC1=O CC1CN2CCN1CC2C(N1CCN(C(c2nnc3ccccn23)=O)CC1)=O C1(C(=O)N(C(C=C)(C)CC)CC)CCCN1NC(=O)C(O)CN1CCCC1 C1(C(=O)NCC(C(C)C)NC(=O)Cc2cscn2)CCc2n[nH]cc2C1 C12(CNC(=O)CN3CC4C=CC3C4)CCCC1N(c1ncc(C(F)F)cn1)CC2 Cc1cnc(C(=O)NCC2CC2NC(=O)CCCn2c(C)csc2=O)cn1 C1(CC(=O)NCC(CC(C)C)NC(C(CC)CC)=O)COCC2(CCC2)O1 C1(C(N(C)CC2CCC(NC(=O)Cn3cncn3)CC2)=O)CCC2CC1C2(C)C c1(NCCOC(CC)(C)C)ncc(C)cc1S(=O)(=O)N1C2CCC1CC2 C1(C(=O)NC(C2CCC(n3cccc3)CC2)C)CCCC(CN)C1 C(=O)(C(CNC(C1(C)CCCS1)=O)N(C)C)NCCC1CC(C)C1 CC1CCCC(CO)(NC(=O)N(C2CCCC(c3ccccc3)CC2)C2CC2)C1 CC1=C(C)CC(C)(C(=O)NC(C)CCNC(=O)C#CC2CCCC2)CC1 C1(NC(C2(COC)CCC2)=O)COC2(CCN(C(c3ccc(F)cc3)=O)C2)C1 c1(-c2cnc(CC(=O)NC(C(=O)N(CC=C)CC)CCC)nc2)ccc(C)c(Cl)c1 C1(C(N2CC3CC(C)C3C2)=O)CC2CN(C(=O)C3=CCCOC3)CC2C1 N1(C(c2c(C)ncc(N)c2)=O)CCN(C(=O)C2=CCCC2C)CC(C)(F)C1 N1(C(c2cnn(C(C)C)c2Br)=O)CC2CC1CC2NC(=O)Cc1ccco1 N1(C(c2c(CC)scn2)=O)CC(Cn2nc(C)cc2C)CCC1C.C12CC1NC2 C12(OCC)CCC(Nc3c(C(=O)O)cc(CN4C(=O)CSC4=O)cc3Br)(CC1)C2 N1(C(c2ccncc2)=O)CCC2CCN(C(c3ccc(C(F)F)cc3)=O)C2C1 Cc1cc(F)ccc1C(N1CC(N(C(=O)C(C2CCC(=O)N2)C)C)C1)=O C(CC(C)(C)C(c1nnnn1CCCF)NC1CCC1Sc1ccccc1)OC Cc1ccc(C(N2CC3CC(NC(=O)C(=Cc4c[nH]cn4)F)C2C3)=O)c(=O)n1C C1(NC(C(C(C)C)NC(C)=O)=O)CCCCCC1NC(=O)C#CC1CC1 C#CC1(C(=O)Nc2ccc(CCF)cc2)CCN(C(=O)CCn2cc(C)cn2)C1 C=CC1(C(N2CCNC(=O)C2C)=O)CCN(C(=O)CCc2ccn(C)n2)CC1 N1(C(C(Cc2c(C)cccc2)C)=O)CC2(CCCN(C(C3CCCCO3)=O)C2)C1 c1(CN(C2CCN(C(CCCN(C)C)=O)C2)C)ccc(C#N)cc1[N+](=O)[O-] C1(C2N(C(C(C)=C3CC3)=O)CCC2)CCN(C(c2ccc(C3CC3)o2)=O)CC1 N1(C(C(CC)CC)=O)CC(CC(=O)NC(c2ncc(C)cn2)C)CC1(C)C CC1CC(N=c2ccc(Br)c(S(=O)(=O)N3CCC(CF)CC3)[nH]2)CC(C)(C)C1 c1(N2CCC(CNC(C3CC34CCOCC4)=O)CC2)cc2nncn2cn1 N1(C(C2C(C=C)C2)=O)CCC2(CC1)CN(C(=O)C1=COCCO1)CC(C)O2 C1(C(=O)NCCC2CCN(C(CCc3nc(=N)[nH][nH]3)=O)C2)CCn2nncc2C1 CC(C)(CC1CC1)C(=O)N1CCN(C(=O)CNC(=O)COc2cncc(Cl)n2)CC1 C(=O)(C1=NOC(C)C1C)NCC(C1CCCC1)NC(c1c(OC)nc(Cl)cc1)=O C1(NC(C2Cc3nccnc3C2)=O)CCC2CN(c3ccncn3)CCC2C1 C(C(=O)NC(C)(C)C#CC)(C(C)CC)N(C(C1CC(O)(CC#C)C1)=O)C N1(C(C(CC)NC(c2ccco2)=O)=O)CCC(CNC(=O)CCSC)CC1 c1(OC)cc(C(=O)NCC2CCN(C(c3ccc(Cl)cn3)=O)C2)c(O)c(Cl)c1 C1(C(C)NC(C2(CCCC)CC2)=O)CCCN1C(=O)CCn1cccc1 C1(CCNC(COCCOC)=O)CCCN1C(=O)CC1(C)CCOC1 N1(CCCSC2CC2)CC(C(F)(F)F)CC1C(N(CC(F)(F)F)C1CC1)=O c1(C(=O)NC(c2cn(-c3ncccc3F)nn2)CCC)ccc(Br)c(Cl)c1C c1(CC(=O)NC2(CNC(C(CSC)C)=O)CCC2)ccc(Cl)cc1C C1(C)(C(N(CC(N2CCN(C(CCC=C=C)=O)CC2)=O)C)=O)CCC(C)(C)CC1 N1(C(c2cnc(CC)o2)=O)CCCC(C(=O)NC2CCN(C)CC2)C1 C(c1ccc2c(c1)OCO2)=CC(=O)NC1(CF)CCN(C(C2(CO)CC2)=O)C1 C(=O)(C1OCCn2ccnc21)NCC1(CNC(c2nccc(C)n2)=O)CC1 C(c1ccc(OC2CN(c3nnnn3C)C2)cc1)=CCNC(C(C)OC)=O CC(C)CC(C(=O)NCC1(O)CCCOC1)N(C)C(c1cnnn1C)=O C1(NC(CCC=C)=O)CC2CCC(C1C)N2C(=O)C(C)CNCC(F)(F)F C1(NC(c2cnc(CC(C)C)s2)=O)CC2CCC1N2C(C1(F)CCOC1)=O C1(n2cc(-c3c(CC)c(C)no3)nn2)CCCN(C(=O)CN(C)C(C)=O)CC1 N1(C(C(CC)(F)F)=O)CC(NC(c2cnc(C(C)(C)C)[nH]2)=O)C(C)(C)C1 CC(CCCCNC(C1(C2CCCO2)CCC1)=O)NC(C1CCCNC1=O)=O c1(C(N2CCCC(C)(NC(c3cc(C)sc3)=O)C2)=O)oc2c(Cl)cccc2c1C c1(OCC(=O)NC2(C(=O)NCC3(CO)CCOC3)CCC2)ccccn1 C1(NC(c2ccc(C(=O)OC)[nH]2)=O)CN(C(C2CCC=CO2)=O)CC1(C)C N1(C(C(C)NC(N)=O)=O)CCC2CCC(NC(c3cc4cccnc4s3)=O)C12 C1(C(N(C)C)=O)CCC2CC2C1.c12cn(nn1)CC(=O)NC2.C12CC(C1)C2 C1(C)(C(=O)NCC2(CCNC(c3c(C)n(C(C)C)cc3)=O)CC2)CCNC(=O)N1 N1(C(C(C)Nc2scc(C)n2)=O)CCCCC(N(C)C(c2[nH]c(O)nc2C)=O)C1 N12NN=NC1=NCC=C2.c1(C(NNC(=O)OC)=O)cc(OC)cc(OC)c1 N1(C(C2(N(C(c3c(C)cco3)=O)C3CC3)CCC2)=O)CCC2(CCO2)C1 C1(CC(N2CCC(C)CC2)=O)CN(C(c2ccccc2)=O)C2(CCC2)C1 C1(C)(C(=O)NCCC2(O)CCN(C(C=C(C)c3ccsc3)=O)C2)CCC(C)CC1 c1(C(=O)NC2CCCNCC2O)ccc([N+](=O)[O-])cc1Cl C1(CC(N2CC(N(C(=O)CC3CCCCC3F)C)C2)=O)CCC(F)(F)CC1 c1(C(=O)NC(CNC(C2N(CC)CCC2)=O)C(C)C)cc2cccc(OC)c2[nH]1 Cc1cc(C(=O)N(CCn2cc(Cn3ccnc3C)nn2)C2CC2)c(C)c(C)c1 C(=O)(C1=CCC2CCC1N2C(=O)C(C)(C)CC)N(CC=C)CCO CCC(C)C(O)C(C)C(=O)NC(c1nocc1C(N1CC(C)(CCO)C1)=O)C C1(C(N2CCCC2CNS(=O)(=O)C(F)F)=O)CCCN1CCC(F)(F)F c1(CNC2CCC(CC(=O)OC)C2)cccc2c(C)csc12 C(=O)(C(O)CCNC(C1(SC)CN(C(C2CN(C3CC3)C(=O)O2)=O)C1)=O)OC C=CCCC(C(=O)NOCC1(C)CCC1)NC(c1cc2n(n1)CCC2)=O C(=O)(C1=CCCCC1C)NCC1C(CNC(C2(CC=C)CCC2)=O)C1 C(=O)(CCC(=O)N1CCC(CCC(N2CCC(CC(=O)NC)C2)=O)CC1)NC C1(NC(C2(C)CCC(C)C2)=O)CCN(C(=O)N)CC1C.C1(C(N)=O)C2CC3C(C2)C13 C1(C(F)F)CCCC(N=c2[nH]c3c(c(=NCCC45CCC(CC4)C5)[nH]2)CCC3)C1 c1(C(N2CCC(CC(=O)NC(CC=C)CO)C2)=O)c(F)ccc(C)c1Cl C(c1cccc([N+](=O)[O-])c1)=CC(=O)NCCNC(C1(c2ccncc2)CC1)=O C1(NC(C(=O)OC)CN(C)C)CCC(C)CC1OC.C1(C)CCCCO1 C1(C(=O)NCCOC2CCN(C(=O)C=CCO)C2)CC12CC(O)C2 C12CCN(CC1)c1cccc(n1)N(C(C)C)C2=O.N1(CC(C)C)CCCC1 C(=O)(C1=CCCCC1)N1CCC(N2CCC(NC(=O)C(F)n3ccnc3)CC2)C1 C1(NC(C(=O)NCc2ccc(Br)cc2Br)=O)COc2ccccc2NC1=O C1(NC(C2N(CC(C)C)CCC2)=O)CCCN(C(=O)CSC(F)(F)F)CC1 c1(C(N(C(C)(C)C)Cc2nc(C)sc2)=O)cccc(C2=CCOCC2)c1 N1(C(C=NOC)=O)CCC2(CCN(C(=O)C(C)n3cccc3)CC2)C(C)C1 c1(CC(N2CC(CNC(C(C)(C)SC)=O)C(C)CC2)=O)sc2ccccc2c1C c1(CC)nc(C)[nH]c(=NCC2CN(C(c3cccc(NC(C)=O)n3)=O)CC2C)n1 c1(C(C)=O)ccc(C(=O)NCC)[nH]1.C(C)(C)(C(=O)N1CCC(O)C1)OCCO Cc1cc(NC(=O)NC2(C(N)=O)CCOC2)cc(F)n1 C(CCC(C)(C)c1cn(C2CCC(NC(=O)CCC=C(C)C)C2)nn1)OC c1(C(N2C(CCNC(=O)C3CC3)COCC2)=O)cc(O)nc(Cl)c1 C1(F)(CNC(c2ccc(SCCCO)cc2)=O)CCN(C(C2CS(=O)(=O)C2)=O)C1 c1(OC)cccc(C(C)=CC(N2CCOC3(C2)CN(C(C24CC(C2)C4)=O)C3)=O)c1 Cc1nc(C(=O)NCCN(C(=O)C(C2(O)CCCC2)F)Cc2ccccc2)co1 C(=O)(N=c1cc(C2CCCC2)[nH][nH]1)c1c(-c2ccc(C#C)cc2)cncn1 c1(NC(C2C(C(=O)NCC(=O)NCC3CC3)C2)=O)cnn(C2CCC2)c1 Cc1cc(CC(=O)NC2CN(C(=O)CCCC(N)=O)CC23CC3)ccc1Cl N1(C(c2c(CC)nn[nH]2)=O)CC2(CC)CC1(CNC(C1CN(C(N)=O)C1)=O)C2 N1(C(C(C2CC2)OC)=O)CCC(CNC(C2CC3C=CC2CC3)=O)C(F)(F)CC1 S(=O)(=O)(c1nc(N2CCC(SC(F)F)C2)ccc1Br)NC(CC)(C)COC n1(CC)ncc(C(N2CCC(CNC(C3(CF)CC3(F)F)=O)C2)=O)c1C C(=O)(CCCS(C)(=O)=O)NCC(c1cccc(Cl)c1)NC(CCCOC(C)C)=O c1(C(=O)NC2CCCN(C(C3C(CCOC)C3)=O)CC2)c(N)cc(Cl)cc1F c1(C(C(=O)NCCOC)N(CC(n2ccnc2)C)C)c(C)cc(C)cc1C Cc1cnc2c(C(=O)NC3CCC4CC3CN4C(C3(C(N)=O)CC3)=O)cccn12 c1(OC)cccc2cc(C(=O)NC3(CNC(=O)CC4CC4)CCCCC3C)oc12 C1(NC(c2c(OC)nsc2)=O)CN(C(=O)CN(C)C2CC2)CC1C CCC(CC)(CC)C(=O)N1CCC(N(C)C(c2cc3ccccc3[nH]2)=O)C(C)C1 CC(CNC(C1CC=CCC1)=O)C(=O)NCC1CN(C(C)C)C1 CC1(C(=O)NC2CC(=O)N(C3CN(C(C4(C)CCC(=O)N4)=O)C3)C2)CCCOC1 N1(C(CC(=C)C)=O)CCN(C(c2cccc(OC)c2)=O)C(c2ccccc2Cl)C1 c1(C(N(CCN(C(=O)C=CSc2ccccc2)C)C)=O)ccc2cnn(C)c2c1 C(=O)(C(CC(C)CC)N(C(=O)CCCOCC)C)NCC(F)F c1(CCC)ccc(NC(C)CN(C)C(c2ccc(=O)oc2)=O)c([N+](=O)[O-])c1 O=C1NCC(C(=O)NCCC2CCN(C(=O)CCCc3cc[nH]n3)C2)N1 Cc1ccc(Cl)c(O)c1C(N1CCC(N(C(=O)C(C)C2CCCC2)C)CC1)=O c1(C(=O)NCC2N(C(CC3CN(C(C)=O)C3)=O)CCC2(C)C)cc2cccn2cn1 N1(C(c2nccc(C)n2)=O)CC2CCCC1(CNC(C1CCC(C)(C)C1)=O)C2 C1(NC(C23CC(C)C2C3)=O)CC2(C1)CC(CNC(c1c[nH]c(=O)cn1)=O)C2 c1(-n2c(C)ccn2)cccc(NC(c2nnnn2C(C)C)CCC2OCCO2)c1 N1(C(c2cc(COC)no2)=O)CC(CNC(c2cccc(OC)n2)=O)C(C)(C)C1 C12(CNC(CN(CCC)C)=O)CC(NC(C3CCC(C)(F)CC3)=O)(C1)C(C)O2 C1(CNC(c2cnc(C)o2)=O)CN(C(=O)CC(C)(C2CCC2)N(C)C)CC1O C1(NC(c2ccnc(OC)c2)=O)(CNC(c2ccc(Cl)[nH]2)=O)CC2CCC1C2 c1(C(C(=O)NCC(F)F)N(CC)CC2CC2)c2c(nn1C)CCCC2 c1(C(N2CCC(N(C(c3cc(OCC)n[nH]3)=O)CC)C2)=O)cc(CO)n(C)n1 c1(OC)ccc(C(=O)NCCCCCNC(C2CC(C)(C)CO2)=O)cn1 c1(C(=O)NCC2(CN(C(=O)C(F)CC3CCOC3)C)CC2)sccc1C#N C(CC(=O)N(C1CCC1)CCCn1nccn1)N(C(C1CCC1)=O)CC c1(C(=O)NC(CN(C(CC(=C)C)=O)C)CC)nc(Cl)c(Cl)s1 C1(N(C)C(C2(C)CC2(F)F)=O)CCCC2CN(C(c3ccc(=N)[nH]n3)=O)CC12 c1(CC)nn(C)cc1C(c1nnnn1CCC1CC1)NC1(c2ccccc2)CC1 Cn1cncc1C(c1ccccc1)OC(C1C2CNCC12)=O N1(C(C(C)OCCCC)=O)CCCC(C(=O)N(C)CCc2cc[nH]n2)CC1 c1(NC(C)C(c2nnnn2CCCF)C2CC2)cc(F)cc(S(N)(=O)=O)c1 CC(N=c1cc[nH]cc1S(=O)(=O)NC1CCN(C(=O)CO)C1)c1ccsc1 c1(C(N2CCCC3(NC(CS(=O)(=O)NC)=O)C(C2)C3)=O)cccc2oc(C)cc12 c1(OC)cncnc1N1CC(NC(c2ccc(OC)nc2)=O)C1 C12(NC(c3cnc(C)[nH]3)=O)CCCC1N(C(c1ncncc1Cl)=O)CCC2 n1(CCC)ccnc1CNC(c1scnc1Br)c1nnnn1C1CC1 O=C(C=Cc1ccc(F)cc1F)Nn1cccn1.C(c1cccc(F)c1)=C N1(C(C(C)(C)Cl)=O)CC(C(=O)NCCCn2cnnc2)CC(F)C1 C12(C(N3CC(N(C)C(C4OC5CCC4CC5)=O)C3)=O)CCC(=O)N1CCS2 C#CCCC(O)C(=O)N(C)CCN(C)C(c1cc(F)ccc1N(C(C)C)CC)=O C(=O)C1SCCc2sccc21.C1(C(=O)O)CCC2C1C2(F)F c1(C(=O)NC(CN(C(c2ccncc2NC(C)C)=O)CC)C)cc(C)c(O)nn1 c1(C(=O)NCC2C(NC(C(C)(C)N(C)C)=O)CCC2)cnc(=N)[nH]c1 c1(CSC)cc(C(=O)N(C)CC2CCN(C(c3coc(C)n3)=O)C2)no1 O=C(C1Cc2cccc(Br)c21)NCC1CC(=C2CC2)C1 c1(C(=O)NCC2(C)CCC(NC(=O)C(F)F)C2)cc2cc(F)ccc2o1 C1(CC=C)(NC(C2CC2CF)=O)CCN(C(c2sccc2C)=O)CC1 S(=O)(=O)(c1ccc(CC(=O)NCC2CC2NC(=O)CC2(O)CCC2)cc1)NC N1(CC(=O)N(CC(C)NC(C2CC2F)=O)C)CCNC(=O)C1 N1(C(C2(CC)CC(C)(C)C2)=O)CCC2(C1)CN(C(C1CC1OC)=O)C2 CCC(C(=O)NC1CC(CCNC(=O)C(C)(C)C2(C)CC2(F)F)C1)n1cncn1 c1(CC)nc(O)c(C(N2CC3CCC(N(C(=O)C(=O)NC)C)C3C2)=O)cc1C c1(C(N2CC(C)C(NC(=O)COC3CC3)C2)=O)cc2ccc(Cl)cc2o1 c1(OC)c(CNC2CCn3c(Br)cnc3C2)ccc2ccccc12 C=CC(CCC)CC(=O)NCC(CNC(=O)Cn1ncn(C)c1=O)S(C)(=O)=O C1(n2cccn2)(C(=O)NCC(C)CO)CCN(C(c2ncn(C)n2)=O)CC1 C1(CC)CN(C(=O)CCC2(C)CN(C(=O)Cc3cccnc3)C2)CCS1 Cc1cc(O)c(Cl)cc1C(=O)NC1(CNC(C2CC2(C)Br)=O)CCC1 C1(SC2C(C(C)(C)C)CC2)CCN(C(N2CCCCC2C2CC2(F)F)=O)CC1 C1(OC)CN(C(=O)C(C)NC(=O)CO)CC1N.N1(CC(=O)NC2CC2)CCOC1=O N(C1CCC(NC(=O)COCC2CCCC2)c2ccccc21)C(CC(C)(C)C)=O CCCC(C(=O)NC(C)(CNC(=O)CCOc1ccccc1)CO)NC(=O)OC CCC(CCCC(=O)NC(C)(C)C(F)(F)CC)NC(=O)CN(C)C(C)C Cc1cnc(NC(=O)NC(Cc2ccccc2)C(N)=O)c(C(N)=O)c1 C1(C(=O)NC23CCCN(C(c4c[nH]cc4Br)=O)CC2C3)CCCC2CCCCC12 N1(CC)CC(C(N2CC(NC(c3c(Cl)sc(C)c3C)=O)C(C)C2)=O)CCC1=O C1(CNC(c2nnn(CC)c2C)=O)CCN(C(C2(OC)CCC2)=O)CCC1(F)F C(=O)(C(C)S(N)(=O)=O)N1CCC(O)(CNC(C(C=C)c2ccccc2)=O)C1 N1(C(c2ccc(C)cc2O)=O)CCCC2(C1)CN(C(C1CCC(C)O1)=O)CCO2 c1(CNC(C2(C)CCCC2)C)ccc2cc(F)ccc2n1 N1(C(c2c(CC)cco2)=O)CC(=O)NC2CN(C(=O)C(C)S(N)(=O)=O)CCC12 c1(N2CCC(O)(C(C)NC(CC(COC)COC)=O)CC2)nc(OC)ncc1C N1(C(C2CC(CC)C2)=O)CCCC(CSC)C1.C12(CCCC1)C(=O)NCC2 C(CC(C(=O)NCC1CC1C(C)C)NC(=O)CC1CCOC1=O)OC c1(SC)ncc(C(=O)NCC(C)NC(c2ccc(C3CCC3)cc2)=O)c(O)n1 C1(C(=O)NCCCN(C(c2ccc(=O)n(C)n2)=O)CC)CCCN2CCCC12 C=C(C)CC(C(=O)NOCCCC1CC1)NC(=O)CC(C)n1ccnc1 CC1CCOCC1C(N1CCN(C2CCCC2NC(=O)Cc2cc[nH]n2)CC1)=O N1(C(C2(C)C(C)(C)C2)=O)CCCOC(CNC(c2csnc2Cl)=O)C1 N1(N2CC(C)(NC(CNC(=O)OC)=O)C2)CCN(C(c2ccc(Cl)cc2)=O)CC1 N1(C(C2C(C)=C2)=O)CCC2(NC(=O)CC3CC4CCC3O4)CCCCCC12 C1(CNC(CCc2onc(CCC)n2)=O)CCCCN1C(=O)C(C)CNC(C)=O N1(C(C)C)CC(C(=O)N(C)CCOCCC(=O)N(CC(C)O)C(C)C)CC1=O c1(CC(=O)NC2C(NC(c3c(C)[nH]nc3Br)=O)C2)cn(C)c2ccccc12 CCCC(F)C(=O)NC1(CNC(C2CCN2C2CCCC2)=O)CCOCC1 c1(OC)ccc(CN2CC3C(CNC(=O)CCC(C)C)C3C2)c(OCC(C)C)c1 C1(CNC(COC(C)=O)=O)C=CCN(C(=O)CS(C)(=O)=O)C1 C(CC(C(=O)NO)Nc1cn(-c2ccccc2C(F)(F)F)nn1)SC C(=O)(C(C)N(C(=O)CC1(NC(=O)Cc2csnn2)CCC1)C1CC1)OC N1(C(c2[nH]cc(C(N)=O)c2)=O)CCN(C(C2CC(=O)NC(=O)N2)=O)C2CCC12 C1(OC)CC2(C1)CC(C(=O)NC1CCN(C(=O)Cc3cnc[nH]3)CC1O)C2 N1(C(CNC(=O)OC)=O)CCC(N(CCOC)C(C2CC(C)=NO2)=O)CC1 C1(C(=O)NCC(CNC(c2nc(CC)sc2)=O)F)CCCC2(CCCCC2)C1 N1(C(C(=O)NCCCC)C2=CCSC2)CCc2cccc(F)c2C1C Cc1ccnc2c1CN(C(c1ccc3c(n1)N1CCC(O)C31)=O)CC2 C1(C(=O)NC(C2(OCC)CCC2)C)CC=CCC1NC(c1ncncc1Cl)=O N1(CC=C)CCCC(NC(C2CCN(C(C)=O)C2)=O)C1 N1(C(C2C(c3ccn(C)n3)C2)=O)CC2CC(NC(c3ccc(O)nc3Cl)=O)CC2C1 C1(C(=O)NC)CCN(C(C)C(=O)Nc2ccccc2C(C)C)CC1 C(=O)(CC1=CCOCC1)NC1(CC(=O)NCC(C)OCCO)CCC1 c1(OC)cccc(NC(C2CC23CN(Cc2cccc(I)c2F)C3)=O)c1OC C(C)(C(C)(C)C(=O)N1CCOC(CCF)C1)NC(C(C)C(F)F)=O C1(NC(c2csnn2)=O)CC(F)CN(C(=O)COc2ccc(F)cc2C(F)F)C1 c1(OC)ccnc(CN(C)C(=O)NCC2CCOC(=O)N2)c1OC C1(C(C)C)CCC(=O)N1.Cc1[nH]ccc1C(=O)NOCC1CCCO1 C(C)(CC(F)(F)C(F)F)(c1n(CCCC)nnn1)NCCNC(C)=O c1(NC(CCNC(c2c(C)ccnc2)=O)(C)C)ncnc(O)c1Br c1(C(N(CC)CC2CCN(C(=O)CC(C)F)CC2)=O)cnc2c(c1)OCC(=O)N2 Cn1ncc([N+](=O)[O-])c1C(=O)NCC1CC1NC(=O)C(C)(C)COCC(F)F C=Cc1ccc(C(=O)NCC(C)(C)CC(=O)NCCCC2CCCCC2)cc1 C#Cc1ccc(C(N2CCOC(CC(=O)N(C3CC3CCOC)C)C2)=O)cc1 c1(C(C(=O)NCC=CCNC(C(C)SC(C)C)=O)O)ccc(F)c(Cl)c1F C1(c2cc(CNC(CC=CCC)=O)on2)CCN(C(C2CC2(Cl)Cl)=O)CC1 c1(C(=O)NCCC2CSCCN2C(C2CC=CCC2)=O)cc(F)c(Cl)cc1F C1(NC(C2CC2C2CCCCC2)=O)CN(C(c2csc(Cl)c2)=O)CC2(CCC2)C1 C1(NC(c2ccc(CC(=O)OC)cc2)=O)CN(C(=O)C(C)C2CC2)CC(C)(C)C1 C(=O)(CC(O)CNC(C1(N(C(=O)CC2CC2(C)C)C)CC1)=O)OCC CCC(CC(=O)N1CCC(C(C)NC(C2CC(C)=NO2)=O)C1)C(C)(C)C C(C(C)(C)CNC(=O)CC1CCC1)N(C(=O)CN(C)C(C)=O)CC c1(C(=O)NC(C2(O)CN(C(CCC(C)C)=O)C2)C)cc2ncccn2n1 C1(CC)CN(C(=O)CC(C)F)CC1C(N1CC(OC(=O)NC)C1)=O C12CC3(C1)CC(C3)CN2C(C(C)C1CCOC1)=O.C(=O)(CCS(C)(=O)=O)NC1CC1 C1(NC(COCC(=O)OC)=O)(CO)CCN(C(=O)COC2CCCC2C)CC1 C1(C(N2CC3C(CNC(c4ncccc4F)=O)C3C2)=O)CC2(C1)CC1(CC1)C2 c1(N2CCN(c3n(C)ccn3)CC2)cnc(Cl)c2cccnc12 C(=O)(CC(F)(F)C(C)(F)F)NC(CNC(C(CCC)C)=O)(C)CO C(C)(C(=O)N1CCC(NC(c2ncccn2)=O)CC1)(C(C)C)OC C12(CNC(=O)COC(F)(F)F)CCC1CCN2C(c1cn(C2CC2)cn1)=O c1(C(=O)NCC(C)(C)NC(C23COCC2C3)=O)c(Cl)ccc(O)c1N C1(C(=O)NCCc2n(CC)cnn2)CC2(CCC2)CN1C(C1CCC(O)C1)=O CC1(CNC(C2CC3CCC2CC3)=O)CCCN(CCn2cncn2)C1 CN=c1[nH]cc(C(=O)NCC2CC(O)(CNC(c3cc(Cl)n(C)n3)=O)C2)s1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(C)CNC(c1ncoc1-c1ccc(F)cc1)=O CC1(CC(=O)NCCNC(c2cc(CO)co2)=O)CCOC1 C1(C(=O)NC2CC(OCC(=O)NC3C(C)(COC)C3)C2)CCOC(C)(C)C1 Cc1ncc(Br)c(C(=O)NC2CCN(C(=O)CC3CCC(C)(O)CC3)C2)n1 N1(C(CCCC=C)=O)CCC2CC2(NC(=O)Cc2cccc(C)c2)CC1 N1(C(C2ON=C(CC)C2)=O)CC2CC(C(=O)N(C(C)C(=O)N(C)C)C)(C2)C1 N1(C(C2(CC)COC2)=O)C(CN(C)C(CCC(C)C)=O)C2CCCC12 C1(CNC(CCSC)=O)CN(C(c2csc3nnsc23)=O)CCCO1 C1(C(N2CCC(C)(CC)C2)=O)C2CCC(C2)N1C(c1coc(OC)n1)=O N1(C(C2C(=C)C2)=O)CCC(C2CCN(C(C3(OC)CCSCC3)=O)CC2)C1 C1(CNC(C(CC#C)CC#C)=O)CC2(CCN(C(=O)C(=O)Nc3ccco3)C2)CO1 c1(C(N2CCC(N(C(C3CCC3(C)C)=O)CC)C2)=O)c(C(F)F)nn(C)c1C C1(C(N2CC(OCc3cc(C(=O)NCc4ccccc4)no3)C2)=O)C2CCCC12 CC1CCN(C(=O)N(C)C)CC1.C1CCCN(c2cncc(N3CCCCC3)n2)C1 C(CCCC(CO)NC(C1CCOC1)=O)NC(c1c(OC)c[nH]n1)=O N1(C(C(C=C)(C)C)=O)CC2CN(C(c3nccc(C)n3)=O)CC2C1 N1(C(c2ncccc2CC)=O)CCC(NCc2cnc(OC)nc2OC)C(O)C1 C1(C(=O)NC(C)C(c2ccccc2)O)(CC)CCSCC1 CCCCC(O)CC(=O)N1CC(NC(=O)C=Cc2ccnn2C)C2CCCC12 C#Cc1cccc(C(=O)NCCC2CCCN(C(c3ccc(O)cc3)=O)C2)c1 Cc1nc(NC(C)CN(C)C(C2CCC(C)O2)=O)c2c3c(sc2n1)CCCC3 c1(NC2C(NC(c3cn(CCOC)nc3)=O)C2)cc(C)ncn1 C1(C(N)=O)CCCN(C(=O)CC2CC(F)CN2C(=O)CC(O)C2CCCC2)C1 CN1CC=C(C(=O)N(CCC(=O)NC2CCOCC2(C)C2CC2)C(C)C)C1 c1(N2C(C(N3CC(C)C3)=O)CCC2C)ncnc2c1cc(I)n2C c1(C(=O)NC(Cc2ccccc2)C(=O)NC(CO)CCC2CC2)ccccc1Cl C1(C)(NC(C2CC(C)N2C(=O)C2=CCCCC2)=O)CCCCC1(C)C c1(OC)nc(N2CC3CC2CN3C(c2cnc(O)[nH]2)=O)ncc1Br c1(C(C(=O)NCc2cnc(C)n2C)N(C)CC)cc2cc(C)c(C)cc2o1 C1(C)(NC(CNC(C(C)(C)C)=O)=O)CCNC1=O.C12COC(C1)C(=O)N2 C1(CNC(C=C(C)C)=O)COCCN(C(c2cc(F)ccc2OC(F)(F)F)=O)C1 N1(C(=O)Cc2cnccc2Cl)CCCC(c2cn(CC3CCCOC3)nn2)CC1 c1(C(=O)NC(C(=O)OC)CN2CCOCC2)cc2cc(Cl)ccc2s1 C1(CN(C(=O)Cc2nccn2C)C)CCCCN1C(c1cccc(CF)c1)=O Cc1nc(NCCC2CC(=O)N(C)C2)cc(N(C)Cc2csc(C)n2)n1 C#Cc1ccc(OCC(N2CCCC2CCCNC(=O)C(CC)=CC)=O)cc1 c1(C(=O)NC2C(NC(=O)CC3(O)CCCOC3)CCC2)coc2c(F)cccc12 N1(C(CC=CC=C)=O)CC2(CCC(CNC(=O)C(C)(C)N3CCCC3)O2)C1 c1(CC)cccc(C(=O)NC(CNC(c2cnn(CC)c2)=O)C(C)C)c1C C#CCCCC(C)C(=O)N(C)CCOCCNC(c1cc2occc2s1)=O Cc1nc(C2CC2)sc1CC(=O)NCC(C)CN(C)C(C1CC(=O)N(C)C1)=O N1(C(C(c2ccc(C)cc2)C)=O)CC2CC(C1)C2NC(C1C2COCC12)=O C(C(C)(O)CC(=O)N1CC(NC(c2cc(C)n(C3CC3)c2C)=O)C(O)C1)OC Cc1nc(=N)[nH]cc1C(=O)NCCC1CCCN(C(C2CCS2(=O)=O)=O)C1 C1(CNC(c2c(C)nc[nH]2)=O)CCCCN1C(C1(CO)CCCO1)=O N1(C(C(C)=CC2CC2)=O)CC(CO)C2(C1)CN(C(=O)CC1CC1)C2 N1(C(CCCOC(C)C)=O)CC(NC(c2cnn(C)c2F)=O)C2CC2C1 c1(NCC(=O)NC(CNC(C(C)Cc2ccccc2)=O)C)ccc([N+](=O)[O-])cc1 C(CNC(=O)C(C)Cc1ccncc1)(CC(F)(F)F)NC(c1c(C)nn(C)n1)=O N1(C(CNC(=O)C2CC2)=O)CCOCC(NC(c2cccc(CCO)c2)=O)C1 N1(C(Cc2c(C)nsc2)=O)CC(C(=O)NC2CCN2C(C)(C)C)C2(CC2)C1 N1(C(CC2(C)CC2)=O)CCOCC1CNC(C1CCCN1C(c1ccccc1)=O)=O c1(OCC(=O)NC2CN(C(CC=CC)=O)CC2O)cccc(C)c1F C(C)(C)(CCN(C)C(C1CC2CC2C1)=O)NC(C1CC(SC)C1)=O C1(NC(C(CC)=CC)=O)CCCC(CC(=O)NOCc2cn(CC(=O)OC)nn2)C1 c1(SCC(=O)NC2CC(NC(c3c(C)cco3)=O)C2)cccc(F)c1 C1(C(=O)N(CCF)Cc2cscn2)CN(CCF)CCC1O c1(C(N(CC(C)N(C)C(c2ccnnc2)=O)C)=O)c(F)c(F)c(F)c(F)c1F N1(C(c2c(OC)c([N+](=O)[O-])ccc2)=O)CC(NC(C2CC2F)=O)CC12CCCC2 c1(CCC=C)ccc(-c2noc(-c3cccc(C)c3)n2)cc1 N1(C(C2C(C)CC2)=O)CC(O)(CCNC(c2cn(Cc3ccccn3)nn2)=O)C1 C(=O)(CC1=Cc2ccccc2C1)NCC(CNC(C1CCC2(CC2)C1)=O)OC C1(NC(c2cnn[nH]2)=O)CN(C(c2cccnn2)=O)C2CCCC12 C1(C(=O)OC)CN(C(=O)NCCc2csc3cc(C)ccc23)CC2(CCC2)O1 C1(C(=O)OC)CC2(C1)CC(C(N1CCC(CNC(=O)C(C)SC(C)C)C1)=O)C2 c1(CN(C(=O)C(C)OCCN2CCCC2)CC)ncc(C)[nH]1.C1(C)CCCO1 c1(NC(c2c(C(C)C)onc2)=O)cnn2ccsc12 c1(CC)ncccc1C(N1CCC1C(=O)NCCCS(C)(=O)=O)=O n1(CC)c(C(=O)NC2COCCN(C(=O)C(C)(C)CC)C2)cc2ccccc12 c1(OC)ccc2c(CC(N3CC4(CC(NC(C5CC5C)=O)CO4)C3)=O)c[nH]c2c1 C(=O)(CN=c1cc[nH]cc1)N1CCCC(F)(C(=O)NC2CCN(C)CC2C#N)C1 c1(C(CC(=O)OCc2c(C(=O)OCC)scn2)C)ccc(Br)cc1 CC(c1ccco1)=CC(=O)NCC(C)(C)CNC(c1cnc(C2CC2)s1)=O C1(NC(C2(C)CSC2)=O)CCC(NC(c2cncc(-n3ccnc3)n2)=O)CC1 Cc1noc(CC(N2CC(NC(=O)CCc3nnc(C(C)C)o3)C2)=O)n1 CCCCCCC(=O)N1CCCC(F)(CNC(=O)CCC2CCC(C)O2)C1 C1(C(C)=O)CC(C)CN1C(c1cccc(OCc2ccc(F)cc2)c1)=O C1(C(=O)NC2CC2C(F)(F)F)CCCN(C(c2c[nH]nc2-c2ccoc2)=O)C1 C12CN(CCN1C(=O)CCC(N)=O)C2=O.c1(C(=O)NC)cnc(C(F)(F)F)cc1Cl CC1C(C)N(C(=O)C=CCO)CCN1C(=O)CS(N)(=O)=O C1(CNC(c2cnn(CC)c2C)=O)CCN(C(=O)C(C)C(=O)OC)C1(C)C C(=O)(C(C)CC(C)C(C)=O)NC1CCC(CC(NOCCCC(=O)OC)=O)C1 C1(C)(CC(=O)NC(c2nccn2C)C)CCN(C(=O)Cc2ccccc2)C1 c1(C(=O)NCC=CCNC(CN(C)C(=O)C2CC2)=O)cccc(-c2ccsc2)c1 CC1(C(=O)NC2CC(F)(CNC(C3CCC(=O)N3)=O)C2)CCCNS1(=O)=O N1(C(=O)C=CC=C(Cl)Cl)CCC2(CCN(C(c3cccn4ccnc34)=O)C2)C1 N=c1[nH]c2ncc(C(=O)NCC3CC4CCC3N4C(=O)C#CC3CCC3)cc2s1 C(=O)(CCCCCCCCSC)N(CCN(C(=O)C1=C(C)OCCS1)CC)CC c1(CSC)cc(C(=O)NCC2(NC(=O)Cn3cnnc3)CC2)ccc1F N1(C(=O)C=CCOc2cccc(F)c2)CCN(C(C2C3COCC23)=O)CC1 CC1CN(C(=O)C(C)(O)F)CC(C)N1C(=O)CC1(C)CCOC1 C(=O)(C(CC(C)C)C(C)C)N1CCC(NC(CCc2cnc(C)s2)=O)C(O)C1 C1(C(N(C)Cc2n(CC)ccn2)=O)C2CCN(C(=O)CC3CCCC(C)O3)CC12 c1(C(C)=O)cc(=NCC2CCN(C(C3CCCN3S(C)(=O)=O)=O)C2)[nH]cn1 C1(CNC(CC2(OC)CN(C(C3CCCSC3C)=O)C2)=O)CN2CCC1CC2 c1(NC2C(C=C)CN(C(c3c(C)cc(Br)cc3C)=O)C2)nccc2[nH]ccc12 C12(NC(C3C(CCC)CCC3)=O)CCC(NC(=O)CCC3CC(OC)C3)(CC1)C2 C(=O)(C1=Cc2ccccc2OC1)N1CC(NC(c2c[nH]c(Br)c2)=O)C2C1C2 c1(CC)oc2ccccc2c1C(=O)NC1CCC1CNC(c1csc(Cl)c1)=O CC1CN(C(c2nsnc2O)=O)CCC1CNC(=O)C(C)(C)Cc1cnn[nH]1 C#CC1(C(=O)NCC(CC(C)C)OC)CCN(C(c2c[nH]cc2C)=O)C1 N1(C(C2CC(NC(=O)NC(=O)OC(C)(C)C)C2)C)CC(C)OC2(CCOC2C)C1 c1(C(N(C)CC2(CNC(c3ccc(CO)o3)=O)CC2)=O)ccc(F)c(Cl)c1 c1(C(=O)NC2C(NC(C=C(C)C(C)C)=O)CC2)cn(C2CC2)nn1.C1CCCO1 N1(C(C(C)(C)F)=O)CCN(C(c2ccc3nccn3n2)=O)CC(CO)C1 C1(CC=C)(NC(c2n[nH]c(C3CC3)c2C)=O)CCN(C(=O)C(C)C(C)O)C1 CC1N(C(C2OCCC2CNC(=O)C2=CCN(C)C2)=O)CCCC1(C)C N1(C(C(CC)C)=O)CCC(C2CC2)(CNC(=O)CCc2c(C)noc2C)C1 c1(C(N2C(C3(C(=O)NCCC(=O)OC)CC3)CCC2)=O)cccc(OC)n1 CCN=C(NCC12CCC(C1)C(=O)N2)N1CCc2cccc(C)c2C1 c1(CC(=O)NC(CC)CN(C(=O)C2=CCCCO2)C)cccc([N+](=O)[O-])c1C C1(C(N(C(C(C)C)CO)Cc2cccc(Cl)n2)=O)CCCN(Cc2cn[nH]c2)CC1 N1(C(CCNC(=O)CO)=O)CCCC2(C1)CN(C(=O)C=CC1CCCCC1)C2 Cc1ccc(F)c(C(=O)NCC(CO)NC(c2csc(-c3ccsc3)n2)=O)c1 N1(C(C(=O)N(C)C)=O)CC2CC(=O)CC1C2.c12cnc(s1)CNC2=O c1(C(=O)NCC2(O)CCN(C(C(n3ncc(C)c3)C)=O)C2)cc2n(c1)CCOC2 C1(C(=O)NCCCCC2C(C)C2)C2CC(O)C(C2)N1C(=O)CC12CCCC1C2 c1(C(=O)OC)cc(N2CCOC(CNC(C3CCSC3)=O)C2)nc(C)n1 c1(C(N(CC(CNC(CCC#C)=O)C)C)=O)c(Cl)ccc(C)c1N C1(CC=C)(NC(C2CCN(C)C2=O)=O)CCN(C(c2nc(F)ccc2Cl)=O)CC1 C(C)(CCC(=O)N(CCC(=O)NCCCc1n[nH]c(C)n1)C)OCC CC(c1ccccc1C)=CC(N1CC(CNC(=O)Cc2cccnc2)C(C)C1)=O N1(C(C2N(C(c3c(C)c(F)cnc3)=O)CCSC2)=O)CC(O)CC(C)(C)C1 c1(OCC)ccc(C(N2CC(NC(=O)Cc3cncs3)C(O)C2)=O)cc1OCC N1(C(C=CC=CC)=O)CCC(NC(c2coc(Cl)n2)=O)CC(O)C1 c1(C(N(CCCNC(=O)C(C)CN(C)C)CC)=O)cccn2nccc12 N1(C(C2(C(=O)OC)CC2)=O)CCC(O)(CN(C)C(C2CCC(C)(C)C2)=O)CC1 c1(OC)ccc(C(=O)N(C)CC2CN(C(=O)CCC3(O)CCC3)CCO2)cc1F C1(NC(c2cc(C(=O)OC)no2)=O)CCC(N(C)C(c2cn[nH]c2)=O)CC1 Cc1ccc(C(=O)NC(C)(CNC(=O)C(C)C(F)(F)F)CO)c(O)c1C CC(C)C(C)(C)C(=O)NCC1CC2CC1CN2C(C1CCCN1S(C)(=O)=O)=O c1(C(=O)OC)cncn1C(c1nc(COC(C)=O)cs1)C c1(C(=O)OCc2n(CC)nc(Br)n2)ccc(Cl)c(C#N)c1 S(=O)(=O)(c1[nH]c(=NCC2C(C)(C)C2(F)F)ccc1Br)N(C)CC1CSC1 N1(C(C(C)(C)OCC)=O)CC(CNC(c2ccc(-c3ccccc3)[nH]2)=O)C(C)C1 c1(CNC2CC(C(=O)Nc3cnc(C(=O)OC)nc3)C2)ccc(F)c([N+](=O)[O-])c1 C1(COCCCF)CC(C)CCC1(c1nnnn1C)NC1CC1 c1(OCCC(N2CC(CNC(C(C)(C)OC)=O)OCC2)=O)ccc(Cl)c(Cl)c1 c1(OCC)ccc(CNC(C2CCCC2COC)=O)cc1.c1(COC)ncno1 CC(C)(C(=O)NCC12CC1CN(C(=O)CCNc1ccccc1)C2)C(N)=O C(c1cc2ccccc2o1)=CC(N1CCC(NC(C2CC=C(C)CC2)=O)C1)=O C(=O)(CC1=CCN(C)CC1)NCC(CC)NC(C1CCC(OC(F)F)CC1)=O c1(CC(N2CC(C(Cn3cc(C4(C)CSC4)nn3)F)C2)=O)cc2ccccc2s1 c1(C(C)C)nc(C(=O)NCc2ccoc2C(=O)NCC=C(Cl)Cl)co1 Cc1cccc(F)c1CC(N1CC2CC(NC(=O)CCC3CC3(Cl)Cl)C1C2)=O C(=O)(N=c1[nH][nH]c2cc(Cl)ccc12)c1ccc(NC(=O)CCc2ccsc2)cn1 CCCCC(CC)CCCNCC1CCN(C(=O)Cc2ccc(Br)cc2)C1 N1(C(CCC2(C)CCCN2C(C2CCOC2)=O)=O)CC(C2CCCCC2)C1 N1(C(c2ccc(CNC3CC3)cc2)C(=O)NCCCF)CCCC2(CCOC2)C1 CC1CCC(CNC(c2cc[nH]c2)=O)N(C(c2cnc(-c3ccccc3)o2)=O)C1 C12(NC(C(C)Sc3ccccc3)=O)CCC(CNC(=O)C(C)(C)C#N)(CC1)OC2 C=CCN=c1[nH]c(N2CCC(OCCO)CC2)nc2cc[nH]c12 c1(OCC)cc(C(=O)NCC2CCC(N(C)C(c3ccsn3)=O)CC2)cc(F)c1 C(C1=NOC2CN(C(C34CCCC3CCC4)=O)CC12)NC(c1cnc(C)[nH]1)=O C(=O)(C1=COCCC1)NC(C(=O)N(C(CO)C1CC1)C)(C)Cc1cn[nH]c1 C1(NC(=O)CN(C(=O)C(Cl)(Cl)Cl)CCO)CC2CCC(C1)N2 c1(C(N(CC(C)NC(=O)CN2CC3CC3C2)C)=O)ccnn1CC(F)F c1(C(=O)NCC2CN(C(CCC(=C)C)=O)CC2C)cnc2ccccn2c1=O C1(C(=O)OC)COC(NC(=O)NCC=CC)C1.O(C(=N)O)CCS c1(C(=O)NC2C(C(=O)NCC3C(OCC)CC3)C2(C)C)cc(F)ccc1F C1(CNC(C=CC(CC)=CC)=O)CCC2(CCC2)C1NC(=O)C1=COCCC1 C1(C(C(C)C)NC(=O)CC2CC(C)N(C(C)=O)C2)CC2C=CC1C2 c1(OCC)c(Cl)cc(C)nc1C(=O)NC1CN(C(C2CCCOC2)=O)CC1C C(C(CC(C)C)OC)NC(c1n(CCCSC)nnn1)(C)CCc1ccc(Cl)cc1 N1(C(C(C2N(C(c3n(CCC)ncc3)=O)CCC2)(C)C)=O)CC(O)C(C)(C)C1 N1(C(Cc2cccc(C)c2)=O)CC(C(N2CCC(OCCO)C2)=O)CC(F)(F)C1 c1(C2(F)CCC(NC(=O)CCc3cc(I)c[nH]3)C2)cc(F)cc(F)c1 CC1(CNC(=O)Cn2nc(Cl)ccc2=O)CC(F)(F)CN1C(C1CCCSC1)=O N1(C(c2cccc(NC)n2)=O)CC2(CCN(C(=O)C=CC3CCC(=O)CC3)C2)C1 C1(C(N(CCNC(=O)CCSC(F)(F)F)CC)=O)CCC(C)(C)O1 c1(C(=O)NCc2ccc(CSC)cc2)nnn2c1CSCC2 c1(CC(=O)NC(C(CO)NC(CC2(C=C)CC2)=O)C)cnc2ccccc2c1 C=CCC(C)(C)CC(=O)NCC12CCC(C1)N(C(=O)CCc1cc(OC)no1)C2 c1(C(N(C2CCCN(C(CCC=CC)=O)C2)CCO)=O)ccc(C(F)F)cc1F C(=O)(CCS(N)(=O)=O)N1CCC(CCC(N2C(C)CSCC2)=O)CC1 C1(NC(=O)CCc2ccccc2)CC2CCC1N(C(c1cn(CCF)nn1)=O)C2 c1(C(=O)NCC(C)NC(=O)CC2(c3ccccc3)CC2)cc(F)ccc1OCF CC(C)(CCCN(c1ccccc1)CC(O)CSC#N)c1ccccc1 C1(C(=O)NC2CCN(C(=O)CCCCC(F)F)CC2O)(OC)CCCC(C)(C)C1 c1(C(=O)NCC(CC(C)C)NC(C2C(=C)C2)=O)cc(C)nc2c(C#N)cnn12 N1(C(CSCCCC)=O)CCN(C(=O)CCCc2ncc(C)o2)CC(C)(C)C1 C1(COCC)CCN(CC(O)CNC(=O)CCC2CCCN2C)CC1 C1(O)(CN(C(=O)C(O)Cc2ccccn2)C)CCCN(C(=O)COCC2CC2)C1 C1(C(=O)NC23CCN(C(CN=S(C)(C)=O)=O)CC2C3)CCCC12CCOCC2 c1(C(=O)NCC(C)CN2CCCC2)ccc(N2CCCC2)nc1 C1(F)(C(=O)NC2C(NC(c3cc(Br)no3)=O)CCC2)CC=CCC1 C1(NC(C(C)CCN(C)C)=O)CN(C(C2Cc3ccccc3N2)=O)CC1(C)C C1(NC(C2CCC(=O)NC2)=O)CN(C(=O)COCCF)CCC1F c1(C(=O)OC)cc(NCC23CC2CN(C(c2ccno2)=O)C3)ncn1 C1(C(=O)NCC(N2CC(C(=O)NCC)C2)=O)CSCCN1C(C)=O.C1(=O)CN1 Cn1[nH]nnc1=NC1CCCCCN(C(c2cc3ccccn3n2)=O)C1 N1(C(c2cnc(C)nc2)=O)C2CCC1CC(C(N1CC(n3cnnc3)C1)=O)C2 N1(C(c2cn(C)nn2)=O)CCC2(CC(NC(=O)C3=COCCO3)CO2)C1 N1(C(C)=O)CCC(C2CCCN2C(=O)N(C)C)CC1.c12ccc(cc1)s2 N1(C(CC(=O)NC2CC2)=O)CCOCC1C(=O)NCc1cccc(F)c1 C1(C(=O)N(CCO)CCO)CC(O)CCN1C(c1ncccc1Cl)=O CN=c1[nH]nc(CC(N2CC3C(CN(C)C(C4CCOCC4)=O)C3C2)=O)s1 c1(C(=O)NCCC2C(C)CN(C(=O)C=CC(F)(F)F)C2)cc2ccsc2c(O)n1 C(=O)(CCC(C)(C)NC(C1CCC(C)C1)=O)NCc1cnn(C2CC2)c1 N1(CCC)C(=S)NC(c2cnc(O)c(C)c2)C(C(=O)OCC)=C1c1[nH]cnc1C c1(CC(=O)N(CC(C)NC(=O)COCc2ccnc(O)c2)C)ccc(C#N)nc1 CC1C(NC(c2nc(Cl)ccc2F)=O)CC2CCC1N2C(=O)CCCC(F)(F)F CC(C)CC(C)(CNC(=O)CCCC1CC1)NC(=O)CC1CCOC1 C1(NC(c2cn(C)nc2)=O)C2CC1N(C(=O)CC1(CO)CCOCC1)C2 N1(C(Cn2c(C)ncc2)=O)CCN(C(C)CNC(c2conc2C(C)C)=O)CC1 C1(C(=O)NCCN(CCC)C(C2(CO)COC2)=O)CCCC1c1ccccc1 c1(C(=O)NCC(CC)NC(=O)CC(C)N(C)C2CC2)cn(C(C)C)cn1 C1(N(C(c2conc2CN)=O)CC)CCN(C(=O)C(C(C)C)n2cnnn2)CC1 N1(C(C(F)=C(C)C)=O)CC2CCN(C(c3cc(N(C)C)ccc3F)=O)CC2C1 c1(NCC(c2cccnc2)(C)OC)nccc(=NCC2(N(C)C)CCC2)[nH]1 N(C1CC2(CCN(C(=O)CO)CC2)Oc2ccccc21)C(c1cncc(C)c1)=O c1(CCC(=O)NCC(CC=C)NC(C2CCCC23CC3)=O)ccccc1Br C(=O)(CC(F)(F)C(C)(F)F)NCC1C(C)CCN(C(c2cncc(Cl)c2)=O)C1 c1(N2CCC3(CCN(C)C3)C2)nc(N2CCC(Cl)=C(Cl)C2)c2c(n1)CCOC2 n1(CC)ncc(C(=O)NC2CN(C(=O)C(c3ccn(C)n3)C)CC2C)c1Br C(=O)(CC1=Cc2ccccc2C1)NCC1C(NC(c2cnn(CCC)c2C)=O)C1 CC(C)CC(C)CS(=O)(=O)Cc1cc(Cl)ccc1Cl N1(CCNC(=O)CC2CCC(NC(c3cocn3)=O)C2)CCCC(O)C1 N1(C(CSC)=O)CC(n2cc(C3CCCCN3C(C)=O)nn2)C(O)C1.C1(=O)CN1 C(=O)(CCC(C)C)NCCC(=O)NC(C#C)C(C)C C1(C2(CN(CC(F)(F)F)C(=O)NC(C)C3CC3)CC2)CCCCO1 CC1=C(C(=O)NCC2(O)CCCN(C(=O)C(F)n3cccn3)C2)CCC1 C(=O)(C(O)C(C(C)C)OC)NC1(CC=C)CN(C(=O)C=CC(C)(C)SC)C1 N(C(=NCC1CC1)NCC1CCOC1)NC(C(C)(C)C)=O.C1(C)CNC1 c1(C(N2CC(NC(Cc3cn(CC)nc3)=O)C(O)C2)=O)c(F)cc(F)cc1F Cc1cc(C(=O)NC23CCC(CC2NC(=O)CCNC(=O)CO)C3)cnc1O N1(C(C(C)OCc2ccncc2)=O)CCCC(C)(C(=O)N(C2CCC2)CCF)C1 c1(C(=O)NC(C2CCN(C(C=CC(C)=O)=O)C2)C)cc(C(N)=O)ccn1 C(=O)(CCCN(C)N=O)NC(C1OCCN(C(c2c(C)cns2)=O)C1)C c1(NC(C)=O)ccc(CC(=O)NC(C)(CO)CCF)cc1 CC1CC(C(=O)NC2CC(NC(=O)CCCCC#N)C2)CC(C)C1 N1(C(CC2(C)CC2)=O)CCC(NC(c2cc(=O)c(O)c[nH]2)=O)C(C)(C)C1 C#CCCCCCC(=O)N1CCC(N(C(=O)CCc2ccsc2)CC)CC1 CC1CC(NC(c2ccc(CO)s2)=O)CN(C(c2ncccc2Br)=O)C1 c1(CC)ncc(C(=O)NCC=CCNC(=O)C(O)C2CCCC2)c(O)n1 N1(C(CCOCC)=O)CCN(C(c2cc[n+]([O-])cc2)=O)CC1c1ccc(F)cc1 CCC(C)C(O)C(C)C(=O)NCC1CCC(C(N2CCOC(C(C)C)C2)=O)C1 CC1CN(C(c2cc(Cl)ccc2-n2cncn2)=O)CCCN1C(=O)C1=CCSC1 N1(C(CCOCCOC)=O)CCC2(CC1)CCN(C(=O)Cc1cn(C)nn1)CC2 C(=O)(C#CC1CCCCC1)N1CC(C(=O)NC(C)CC2CCCCCC2)OCC1 C1(C(N2CCOCC2)=O)CCC2(CCCC2)CC1.C(=O)(C(=O)N)NC1C(C)C1 O=C(CCCC(F)(F)F)NC(C1CCN(C(c2cccnc2)=O)CC1)(C)C C(=O)(CS(=O)(=O)C(C)C)NCC1(C)CCC(NC(C=C(COC)C)=O)CC1 Cc1cccc(C(=O)N(c2cc(CNC(C3(C)CC3(F)Cl)=O)ccn2)C)c1 c1(C(=O)NC2CCC(c3nn[nH]n3)C2)cc2n(n1)CCOC2 C1(CN(C(COC(CC)CC)=O)C)CCCN(C(C2CC2CF)=O)C1 C1(C(=O)NC(CC=C)CNC(=O)CSCc2ncc[nH]2)CCC(N=[N+]=[N-])CC1 C1(NC(C(C=CC)O)=O)(CNC(c2ccc(C)c(O)n2)=O)Cc2ccccc2C1 C1(C(=O)NCCC(=O)N(CCC(=O)OC)C2CC2)OCCC1(C)C CCC(F)(F)C(=O)NCC1(NC(=O)C(C)c2cccs2)CCC1 c1(CN2CC3CCN(C(C(C)NC(C)=O)=O)C3C2)ccc2cccnc2c1 Cc1cn2cc(C(N3CCC(NC(c4ccnn4C)=O)C3(C)C)=O)nc2s1 C(=O)(C(O)C(C(F)(F)F)NC)NC1Cc2c(C(=O)OCC)n[nH]c2C1 C1(CN)CCCN(C(=O)C(=O)NCCOCC2CCCC2(O)c2ccccc2)C1 c1(C(=O)OCC(C2C(CS(C)(=O)=O)C2)=O)cccnc1 Cc1ccc(CC(=O)NC(C(=O)NCC2(C)CCCC2)C2CCCC2)o1 c1(CC(=O)NCC(CC)NC(=O)CCc2ccncn2)ccccc1Br Cc1ccc(CSCCC(=O)NC2CC(NC(c3cc(C(C)(F)F)n[nH]3)=O)C2)s1 C1(NC(Cc2scc(C)c2)=O)C2CCC1N(C(C1CC(C3CC3)=NO1)=O)C2 N1(C(COCCC#C)=O)CCC2(CC1)CC2NC(=O)C(c1cccnc1)OC c1(COC)nc2c(s1)CCCC2.C1(C)(C)C(C)NC(=O)N1 c1(CC(=O)NCCCCNC(c2ccc(SC)o2)=O)c[nH]c2ccncc12 N1(C(C(C=C)c2ccccc2)=O)CC2(CC(NC(c3ccnnc3)=O)CO2)C1 C1(C#N)(C(N2C(C)CN(C(=O)Cc3ccccc3)CC2)=O)CC12CCCC2 N1(C(C2CCC(OC)C2)=O)CC2(CC(NC(=O)CCc3cncc(C)c3)CO2)C1 N1(C(C23CN(C(CCCC(C)(C)C)=O)C(CC2)CC3)=O)CCC2CCNC(=O)C12 C1(NC(C2C(CC)CCN2C(c2scnc2C)=O)=O)CCCN(O)C1=O C(=O)(C1CCCc2n[nH]cc21)N1CC(F)CC(NC(=O)CC(Cl)Cl)C1 Cc1c(Cl)ccc(CC2CC2)c1F.N12CCC(C(F)C1)C(c1ccccn1)NC2=O CCC(C)CC(=O)N1CCC(N(C(=O)C(C)Oc2ccccn2)C)CC1 c1(NC(CC2N(Cc3cccc(OC)c3)CCOC2)=O)ccc2nn(C)cc2c1 C1(NC(C(c2ccc(F)cc2)OC)=O)C=CCN(C(=O)CNc2nccs2)C1 N1(C(C(C2CCOCC2)C)=O)CC(n2cc(C(C3CCCOC3)C)nn2)C(C)C1 C(=O)(C(O)C(C)C)N(CC(N1CC(c2nc(C)on2)C1)=O)C1CC1 CC1CN(C(=O)CC2CCOC2(C)C)CCCN1C(C1CC2C=CC1O2)=O c1(C(=O)NCC2CCN(C(CCC(=C)Cl)=O)CC2CC)c(Cl)ccc(F)c1N C1(C(N(C)Cc2cccc(C)c2)=O)CN(c2ccc(C(=O)O)cc2)CC(F)(F)C1 c12ccc(cc1)[nH]c2=O.C(C)(C=O)C1CCCO1.C(COCCOCCO)OC CC1CC(CNC(=O)C2=NOCC2)CN1C(=O)CNC(N1CCCC1)=O c1(C(N2C(C(N3C(C(=O)OC)CC(C)C3)=O)CC2)=O)c(C)cccc1C C1(C(N2CC(CNC(c3cc(Cl)c(F)cc3F)=O)C2)=O)CCc2ccccc2C1 C#CCCCCCCCC(=O)N1CC(CNC(c2cc(CO)n(C)n2)=O)C(C)C1 C1(CC)CCN(C(c2cc(CO)on2)=O)C(C(=O)Nc2cnc(SC)nc2)C1 N1(C(CCC=CCC=C)=O)CC(F)(F)CC1(C)CNC(=O)CCc1cocn1 C(=O)(CCCC#Cc1ccccc1)NCC(C)(C)NC(=O)CC1CC(=O)NC1=O C1(C(C)(C)C)CN(C(C2CCC(CO)CC2)=O)CCN1C(C1COC1)=O Cc1cccc2c1OCC2C(=O)NC(=NCCC(=O)NCC)Nc1nc(O)c2ccccc2n1 N#CC1CC(N=c2cccc(S(=O)(=O)NCCN3CCSCC3)[nH]2)C1 C1(C(=O)NCc2ccc(C(=O)O)o2)CCCC12CCOCC2 C1(NC(c2cc(CC(C)C)[nH]n2)=O)C(C)(C)CN(C(=O)CSCC#N)CC1(C)C c1(C(C)C)cnn(C)c1CNC(=O)NCC(C12COC(C)(C1)C2)C C(=O)(CC(C)(C)O)NC1(CCC(=O)NCCN(C2CC2)CC)CCCC1 C1(c2cn(C3C(SC)CN(C(=O)C(C)(C)CCSC)C3)nn2)CCCC(C)(C)O1 N1(C(C(F)=C(C)C)=O)CC2C(CNC(c3nc(O)sc3C)=O)C2C1 c1(NC(C(CCC)N(C)C)=O)ccc(NC(=O)C(CC)C(C)C)c(F)c1 c1(OC)ccc(CCC(N2CCC(C)(CNCc3ccn(C)c3)C2)=O)cc1O C1(C2(O)CCC2)(CNC(C2(OC)CCN(C(c3ccn(C(F)F)n3)=O)C2)=O)CC1 CC(C)CCC(C)NC(C1CCCN(C(=O)CCc2cncs2)C1)=O Cc1ccc2sc(C(=O)NCC3(NC(c4cnsc4)=O)CCC3)c(C)c2c1 C#Cc1ccnc(C(=O)N(C2CCN(C(C3C4C5CCC(C5)C34)=O)CC2)C)c1 CC(C)CCCCC(=O)N1CCCC(CNC(c2ccc(C(C)F)cc2)=O)CC1 n1(CC)ncnc1C(N1CCC(C(C)NC(=O)CCc2cnc(C)o2)C1)=O C1(C(=O)NCc2cc(C(C)C)no2)CCCN(C(=O)Cc2cc[nH]n2)C1 c1(C(=O)NC(CCCC)CNC(=O)CS(=O)CC)cc2cccc(OC)c2o1 c1(NC(=O)NCc2cccc(-n3nccn3)c2)ccc(CO)nc1 N1(C(c2scc(C)c2Cl)=O)CCN(C)C(CNC(=O)COc2cccc(Cl)c2)C1 CCC(C)(CO)C(=O)NCCOCCN(C(=O)CCOc1cc(C)ccc1C)C N1(C(CN(C2CC2)CC)=O)CCC(CNC(c2ccccc2Br)=O)CC1C c1(C(=O)NCC2(C)CN(C(C3CCCC(=O)N3)=O)CCO2)n[nH]c2c1COCC2 c1(C(=O)NC(CC)CNC(C2(c3cccs3)CCCCC2)=O)ccc(C)c(Cl)c1 Cc1ccc(-c2nc(-c3ccc(N(C)C)cn3)nn2Cc2cccs2)nc1C c1(C(=O)NC2CCN(c3ncccc3[N+](=O)[O-])C2)c(F)ccc(Cl)c1F Cn1cnc(N2CCC(O)(Cc3c(F)cccc3F)CC2)cc1=O C1(C(=O)NCCn2cc(C(=O)NC34CCC(CC3)CC4)nn2)CC2(C1)OCCO2 C(=O)(C(O)P(C)(C)=O)N(C)CCN1CCN(C(C23CC(C#N)(C2)C3)=O)CC1 C(=O)(C(C)S(=O)CC)N(C1CCN(C(=O)C(C)NC(=O)COC)CC1)CC C(C(N=[N+]=[N-])C(=O)N1CCN(C(c2cc(OC)cnn2)=O)CC1C1CC1)OCC N1(C(C(c2c(OC)cccc2)O)=O)CCC2CN(C(C34CCCC3C4)=O)CC2C1 C1(NC(C(C)=CC2CC2)=O)CCC(C)N(C(C2C(Cl)(Cl)C23CC3)=O)C1 CC1CCC(CNC(C2(n3cnnn3)CC2)=O)CN1C(=O)C(C1CCCCC1)C c1(OC)ccc(C)cc1C(=O)NC1CN(C(c2cc(Cl)ccc2F)=O)CC12CC2 C1(NC(c2ccc(CC)cn2)=O)CC=C(C(=O)N2CC(=O)N(C)C2)C1 c1(C(N2CCC3CC3C2)C(=O)NCCSC)cc(C(F)(F)F)ccc1Br C(c1ccc2c(c1)OCCO2)=CC(=O)NOCC(c1ccc(F)cc1F)=O c1(OC)cccc(C(CNC(C2CC23CCC3)=O)NC(c2cnc(O)s2)=O)c1 C1(CNC(C2CCCO2)=O)CN(C(c2cnc(S)[nH]2)=O)CC1C(F)(F)F C1(C(=O)NC(C(=O)OC)Cc2cccc(F)c2)CC2OC(C)(C)OC2C1 C(=O)(C#CC1(CC)COC1)NCC(CC=C)NC(=O)C=C(C)c1ccco1 c1(C(N2C(CNC(CN(CCCCCC)C)=O)CC2)=O)cc(C)cc(Cl)c1 CCCC(C)(CC)C(=O)NC(C)CCN(C)C(c1ccccc1NC(=O)NC)=O Cc1cc(C(N2CC3CC2(CNC(=O)CCCC2CC2)C3)=O)cc(N)c1 CCC(CC(=O)N1CCC(F)(C(=O)NC2CCOC2=O)C1)CC(C)C C1(C(N2CCN(C(CCCCCC)=O)C(C)CC2)=O)C2Cc3ccccc3C12 C(C(C)(O)C(=O)OCC)NC(c1scc(CC)n1)c1nnnn1C1CC1.C(C)(C)(C)O c1(CNC(c2ccsc2Br)=O)ccc(Cl)c(Cl)c1Cl C(=O)(C1SCCc2sccc21)NCCN(C(=O)C1CCc2cccnc21)C C1(C(N(C2CCN(C(CCc3n(C)ccn3)=O)C2)CC2CC2)=O)CC(F)C(=O)N1 CCCCC(O)C(=O)N(CCCNC(C1CCCN1C=O)=O)CC1CCCC1 N1(CC)CC(O)CC1c1ccccc1.C1(=O)C(=O)NCCSCCN1 c1(C(=O)NC2CCN(Cc3ccc(Br)cn3)CC2F)cnn2c1CCCC2 CCC(CC)C(=O)N1CC(NC(=O)CSc2ccc(-c3ccc(F)cc3)n2C)C1 N1(C(C(C)N2CCC2)=O)CCCC1(C)CNC(c1cn(CC(F)F)cn1)=O C(=O)(C(C)CC(F)F)NC1CCC(N(C(C(C)Cc2ccco2)=O)C)CC1 N1(C(COCCOCCOC)=O)CC(NC(C2C=CCC2)=O)CC12CCOCC2 C(C(=O)NC(C)C=CC(=O)NC(c1cnn[nH]1)(C)C)(C(C)C)SCC N1(C(CCC(C)OC)=O)CC(C(=O)NCC2(F)COC2)CC2OCCC12 C(C(=O)NCCCC(C)NC(C1CC(C(F)F)C1)=O)(C(C)C)NC(=O)OCC c1(C(=O)NCC(CC)NC(=O)C2CC2)csc(C2CC2)n1 C1(NC(c2cn(CC(CC)O)nn2)=O)CCN(C(C2(O)CCC2)=O)CC1CO c1(C(C)(C)C)ncc(C(=O)NC2(C)CC(NC(c3ccn(C4CC4)n3)=O)C2)s1 N1(C(CCC(=C)Br)=O)CC2COCCC2(NC(=O)CCC2CCCO2)C1 c1(OC)ccc2nc(N3CC4CC4C3)nc(N3CCC4(CCCC4)C3)c2c1 CC(CCC(C)(C)C)C(=O)N1CCC(C)C(NC(=O)CC2COC(=O)C2)C1 c1(C(=O)NCC2OCCN(C(C(CC)C(=O)OC)=O)C2)n[nH]c2cc(C)ccc12 N1(CC)CCCCC1C(C)(C)CNC(=O)C(=O)NCC1CCCN1CC(F)F c1(Cc2nc(C(CC)C)nn2-c2ncnn2C)ccc(F)c(F)c1 N1(C(CCN(C(C=CCN(C)CC)=O)C(=O)C2CC2)=O)CCCC(n2ccnn2)C1 C(=O)(CCC(C)(C)C#N)N1C(C)CC(NC(C(C)OC2CCCOC2)=O)C1 Cc1cc(F)cnc1C(=O)NC(C)CNC(c1ccc(OCC(C)C)cc1)=O C=CC(CC)C(=O)NC(c1cccnc1)C(=O)NCC(=C1CCCCC1)F C1(C(=O)NCc2cc(C(N(C3CC(C(=O)OC)C3)C)=O)no2)CC2(CC2)CN1C c1(C(=O)NC2(CO)CCN(C(C3C(C)(C(F)(F)F)C3)=O)C2)coc2c1CCCC2 Cc1cc(C(C)C(=O)N2CCC2CNC(C2CC(C)OC2C)=O)cc(F)c1 c1(-c2onc(C3OCCN(C(=O)CCCSC(F)(F)F)C3)n2)ccc(F)c(F)c1 N1(C(C(C)Nc2ccccc2)=O)CCC(NC(=O)CC2CCOC2)C(F)C1 C(=O)(C1=CCC(C)CC1)N1CCC(CNC(CC2(C(=O)OC)CC2)=O)C12CC2 c1(C(=O)NC(C(N2C(C#C)CC2)=O)CN(C)C)ccc(CO)cn1 c1(C(C2CC2)NC(CNC(c2cccc(Br)n2)C)=O)ccc(Cl)cn1 N1(c2cc(C(N)=O)ncn2)CC2CCCC(NC(=O)CCCc3cnn[nH]3)C2C1 C1(CNC(C2ON=C(C)C2)=O)CCC2(CN(C(c3ccc(C)cc3N)=O)C2)O1 c1(SC(C)(C)NCC(=O)N(CC(C)(C)C)C)ccccc1Cl Cc1ncnc(C(=O)N(C)CCN(C(=O)C(O)CN2CCCC2)C)c1C c1(C(CCOCCN)=O)cnc(Cl)c(C2CC2)c1.C12(C(=O)C3CC3)CC(CN1C1CC1)C2 C#Cc1cc(C(=O)NCC2CCCCN2C(=O)C(O)CC)cc(Br)c1 c1(CC2(C(=O)NC3C(NC(=O)C(F)C4CCCC4)CC3)CC2)c(Cl)cccc1Cl n12c3c(cc(cc3)c1=O)NC(=O)C2.C1(C(=O)OC)(CC)CCCN(C(N)=O)C1 c1(CC2CCN(Cc3c(OC)cccn3)C2)ccc(F)c(Cl)c1 CC1(C(=O)NCCN2CCN(c3cncc(C#N)n3)CC2)CCc2ccccc21 CC(C)(C)C(C(=O)N(CCCn1cc(C2COC=CO2)nn1)CC)N1CCCC1=O C(=O)(CCCC(=O)N1CC2CC(NC(=O)CSc3nc[nH]n3)C1C2)OCC N1(C(C(c2ccc(C(F)(F)F)cc2)(C)C)=O)CCCC(C)(O)CC1 Cc1cc(C)c(C(=O)N(C2CCCCN(C(C3CN4CCN3CC4)=O)C2)C)cn1 N1(C(c2ccc(Cl)c(F)c2)=O)CCC2(CC1)CC(NC(C1(C3CC3)CC1)=O)CO2 c1(C(N(CCCCC)CCO)=O)cc(CNC(c2c[nH]nc2C)=O)on1 N1(C(c2c(N)ccc(C)c2)=O)CCOC2(CCCN(C(c3ccc(F)o3)=O)C2)C1 N1(C(c2ccc(C)c(C)c2)=O)CCC2C1CCN2C(c1ccn(C)c1)=O C(CC1=CCN(C(=O)Cn2nnnc2C(C)C)CC1)NC(CSC(C)C)=O C1(n2cnnn2)(CN2C(C(=O)NC34CNC(C3)C4)CCC2)CCSCC1 C1(NC(C2(NC(C(CCC)C)=O)CCCC2C)=O)CCOC(C)(CC)C1 c1(C(c2nnnn2C)Nc2scc(C3(OC)CCC3)n2)ccc(I)cc1 C1(NC(c2ccc[nH]2)=O)CN(C(c2ccc(OCC3CC3)cc2)=O)CCC1CO N1(C(CCNS(CC)(=O)=O)=O)CCOCC(CNC(=O)C(C)C2CC2)C1 c1(C(N2CCC(NC(C3CC(C4CC4)=NO3)=O)(CO)C2)=O)ccnc([N+](=O)[O-])c1 Cc1cc(C)n(CC(=O)N(CCCCCCNC(=O)CC2CCSCC2)C)n1 c1(CN(C)C)cc(CNC(=O)Nc2cccc(N(C)C)c2)ccc1F N1(C(c2cc(C#N)on2)=O)CC2CN(C(c3cc(C4(C)CC4)n[nH]3)=O)CC2C1 c1(C(=O)OC)cn2c(n1)CN(C1CCN(C(c3ccc(C)nn3)=O)C1)CC2 C1(NC(CC2CC(C)(C)C2)=O)CC2CCC1(NC(=O)CCc1ccc[nH]1)C2 C1(NC(C(CC=C)C)=O)CN(C(c2[nH]nnc2CC)=O)CC2(CCC2)C1 c1(C(=O)NC(CC(C)NC(=O)CNC(=O)C(C)(C)C)C)cccc(Br)c1Cl C(=O)(C(COC)N(C)C)NCC(COC)OC(=O)CC(Cl)Cl c1(OCCCC)ccc(C(=O)NC2CN(C(C3(C)CCCC3O)=O)C2)cc1 c1(C(=O)NCC(C)N(C(CC(C=C)C)=O)C)cc(Br)c2nc(C)oc2c1 CCCC(C(=O)N1CCCN(C(=O)C=C(C)c2cnn(C)c2)CC1CO)C(C)C c1(C(N(C2CCN(C(C3CCCC3OC)=O)C2)CC)=O)nc(=O)n(C)[nH]1 N1(C(Cc2cc(C)sc2C)=O)CCCCC(CNC(=O)CNC(=O)C2CC2)C1 C1(OC)(CNC(=O)C(N2CCCCC2=O)C)CCN(C(=O)CCCN(C)C)C1 C(=O)(C(C)CC(C)(C)C)N(CCCCCCNC(C(c1c(C)cncc1)C)=O)C c1(C(=O)NCc2ccc(C(N3CCNCC3C(F)(F)F)=O)s2)ccc(O)c(F)c1 c1(CC)cccc(CNC(C2CN(C(=O)CCc3cnc[nH]3)CCO2)=O)n1 C1(C)(NC(C(CC=C)N(C)C)=O)CCC(NC(C2CCC(C)(C)C2)=O)CC1 N1(C(C2CC3CN(C(C4N(CC)CCC4)=O)CC2C3)=O)CC2(COC(C)(C)C2)C1 C1(C(=O)Nc2ccc(-c3cnccn3)cc2)Cc2cccc(F)c2O1 c1(NC(=O)C(=O)N(C)C)cnc(C(=O)NCCC(C)N(C)C)cn1 C(=O)(CC(O)CC(C)(C)C)N(C)CC1(NC(Cc2c(C)cc(Cl)cc2)=O)CC1 CCC(CC)C(F)C(=O)N(C(C)C(N1CCCC(C)C1CO)=O)C N1(C(c2c(C)cc(C#N)cn2)=O)CCC2(CCC2)C(NC(c2ccncn2)=O)C1 C(C(=O)NOCCO)(c1cn(C)nn1)NC(C1CCSC1)=O N1(C(c2c(OC)cccn2)=O)CCC2CC1CN(C(=O)C1=CCCCC1)C2 CC(C)CC(C)(C)C(=O)NCC1C=CC(NC(=O)CC2SC(=N)NC2=O)C1 N1(C(CC=CC)=O)CCN(C(=O)C(O)Cn2cncn2)C(COC)C1 c1(CNC2(C(=O)OC)CC(O)(C(F)(F)F)C2)nc2c(C(F)(F)F)cccc2s1 S(=O)(=O)(c1c[nH]ccc1=NCC1CCC(C(F)(F)F)O1)NCC1N(C)CC1 c1(OC)cccc(O)c1CN1CCC(NC(=O)Cc2nc[nH]n2)CC1C C(c1nc2ccccc2[nH]1)=CC(=O)N(CCCNC(C1C2CC2C2CC12)=O)C c1(C(=O)NCCC2(O)CCN(C(C(C)(CO)OC)=O)C2)c(F)cccc1Cl c1(OC)c(F)cc(NC(C2C3CC2N(Cc2ccc(F)c(C)c2)C3)=O)cc1Br c1(C(N2CC3(CC(NC(C(C)NC(N)=O)=O)C3)C2)=O)cc2c(cc1Cl)NC(=O)C2 c1(C(=O)NC(CC(C)C)Cn2cc(CC3(O)CCSC3)nn2)ccccc1C#N N1(C(c2cnnc(O)c2)=O)CCCC(C(N2CCCCCC2CO)=O)CC1 CCCCCCCCNC(C1(CC)CCN(C(=O)CS(=O)(=O)NC)C1)=O C1(C(=O)NC(C2CN(CCOCC)C2)C)CCCC12CCOCC2 C1(C(N2CC(OC)(CNC(=O)C(C)OC(C)(C)C)C2)=O)C2CCC(=O)C12 N1(C(c2n(C=C)nnc2)=O)CCC2(CC1)COC(CNC(c1cscc1C)=O)C2 c1(CNC(C(C)(CO)NC(Cc2cn(CC)nc2)=O)=O)nn(C)c(=O)n1C NC1(C(=O)NC2CC3CCCCN3C2)CCCCCC1 C(=O)(C1CCCc2nncn21)NC1CC2(CN(C(c3c(C)csc3)=O)C2)OC1 N1(C(C2CCC(CC)O2)=O)CCC(O)CC1C(N1CC(CC(C)C)C1)=O C1(C2CCC2)(C(=O)OC)CCN(S(=O)(=O)Cc2ccc(Cl)c(Cl)c2)C1 CON1CCC(C(=O)NC2COCC2NC(=O)C2=C(C)CCC2)CC1 c1(CC)cc(Br)ccc1C(=O)Nc1cccnc1C(N1CC(O)C(F)C1)=O N1(C(CCCOC)=O)CC2CC(NC(c3c(C)ccc(Cl)c3F)=O)CC1C2 Cc1nsc(Br)c1C(=O)OC1CN(C(=O)C(C)(C)CCl)C1 c1(CNC(C2CCN(C(COC)C)CC2)=O)cc2c(o1)C(C)(C)CCNC2=O C1(C(=O)NCC(=C2CCCCC2)F)(CNC(C2CCCSC2)=O)CC(C)(C)C1 C1(O)(CNC(C(C2CCOCC2)OC)=O)CCCN(C(c2cc(OC)ns2)=O)C1 CC1=C(C(=O)N2CCOCCC2C(N2CCC(F)CC2)=O)COCC1 N1(C(c2ccn(C(C)(C)C)n2)=O)CCCC2(CCN2C(=O)COC(F)F)C1 c1(C(=O)NC(C2CCN(C(=O)CN(C)CCO)C2)C)cc2c(O)ccc(F)c2[nH]1 C(CCC(=O)N1CCC(CN(C(=O)CC2CC(C)(C)C2)C)C1)SC C(=O)(C(O)C(F)(F)F)NC(CNC(C1C(C)(C)CCO1)=O)CO C1(C(=O)OC)CN(C(=NCC(C)c2ccnc(Br)c2)NC2CC2)CC1C(=O)OC C1(CNC(c2c(OC)n[nH]c2)=O)C2CN(C(c3ncccc3N(C)C)=O)CC12 Cc1cc2n(n1)CCN2C(c1cccn1-c1ncn2c1CCC2)=O c1(C(=O)NCC2CN(C(c3cccc[n+]3[O-])=O)CCCO2)ccc2cccnn12 c1(C(C(=O)NC(C2CC(NCc3c(C)ncs3)C2)=O)O)ccc(F)cc1 Cc1cc(C)n2nc(-c3nc(-c4cccs4)nn3-c3cc(F)cc(F)c3)cc2n1 NCCC(=O)N=c1ccn(C(=O)Cn2nnc(-c3ccsc3)n2)[nH]1 c1(NC(C)=O)nc(C)c(Br)cc1S(=O)(=O)NC(C)C(c1ccc(Cl)cc1)C CC1(C)CC=C(C(=O)N2CCC(CCNC(C3NC(=O)OC3(C)C)=O)CC2)CC1 N1(CC2(c3cn(CC)nn3)CC2)CCCN(C(=O)C=Cc2ccc(C)cc2)CC1 N1(C(=O)CN2CCC(O)CC2)CCC2C(NC(c3cnc(C4CC4)o3)=O)C2CC1 N1(C(C2C(NC(CC3(NC(C)=O)CC3)=O)C2)=O)CCC(O)(c2cnn[nH]2)C1 CCC(CC(=O)NC1CC(C)N(C(c2ccc(C3CCC3)nc2)=O)C1)C1CC1 C1(C(=O)NC2CCC(NC(C(C)=C(C)C)=O)C2)C2CCC1(c1ccc(O)cc1)C2 C1(S(N)(=O)=O)(C(=O)NCCN(C)C(c2cnn(CC(F)F)c2)=O)CCCC1 CC1(C)C(CNC(=O)NCc2ccccc2OC(F)(F)F)CCS(=O)(=O)N1 c1(CN(C)C)cnccc1C(=O)NC1CCC1NC(C1(CC2CC2)CCC1)=O C(=O)(CCC(C)(C)N(C)C)NCC1N(C(c2ncn(CC)c2)=O)CCOC1 Cc1ccc(Cl)c(C(N2CCC(C(=O)NCc3ccc(F)cn3)C(O)C2)=O)c1 c1(C(N2CCC(CN(C)C(c3cc(Cl)ns3)=O)C2)=O)ccc2c(c1)C(=O)C(=O)N2 N1(C(C(COC)NC(C)=O)=O)CC2CC(NC(=O)CN3CCSCC3)CC1C2 N1(CC(C)C)CCC(C(=O)N(C2CCN(C(=O)C3=CCSC3)C2)C)CC1 C(=O)(C1CCCc2cncn21)N1C(CCNC(=O)C=CC2CCCCC2)CCC1 CCCCCCCCCCCCNC(C1(C)CCNC1=O)=O N1(C(C=CCC)=O)CCCC1C=CC(N1CCOCC1CC1CC1)=O CC1CCC(CC(N2CC3(C2)CN(C(=O)CC2CC4(CCC4)CO2)C3)=O)CC1C c1(C(=O)NC2(CCCNC(C3C(OC)CCC3)=O)CC2)cccc2ncnn12 C(C(C)CC(=O)NC(c1ccccc1)CO)NC(c1c(CC)con1)=O C(CCCC(F)(F)F)NC(C1CCC=CCCC1)c1n(CCCCCC)nnn1 C=CCCCC(C)(C)C(=O)N1CC2(C1)CN(C(c1ncc(N)cc1C)=O)C2 C1(C(=O)NC2CC(CCC(=O)NCC(C(C)C)(C)F)C2)CCC=CCCC1 C1(C(N2CC(C(N)=O)(CNC(C(C)OCC=C)=O)C2)=O)CCCN(C(C)C)NC1=O c1(C(=O)NC(C2CCN(C(=O)Cc3cnoc3)C2)C)cc(O)cc(C#N)c1 N1(C(c2ccc(CN(C)C)nc2)=O)CCC2C(C1)CN2C(c1cncnc1)=O CC1CC2(CCN(C(=O)C(N3CCOC3=O)C)CC2)CN1C(c1cnsn1)=O CCC(O)C(C)C(=O)NC(C)(C)CC(=O)N1CC(SC)C1 C1(c2n(CCC)nnn2)(NCCc2cncnc2)CC(C)(C)CCC1C C1(NC(=O)CNC(=O)NCC2CCCC2)CC(O)CN(C(c2ccsn2)=O)C1 N1(C(C=CCOC(C)(C)C)=O)CC(CN(C(=O)Cn2ncnn2)C2CC2)C1 C12(NC(CCCOCCC)=O)CCCN(C(c3c[nH]c(=N)o3)=O)CC1C2 c1(C(N2CCC(OCCO)C2)C(=O)NCC=C)cnc(CC(C)C)[nH]1 N1(C(C2(C)CC=CCC2)=O)CCCN(C(c2cc(Cl)nnc2O)=O)C(CO)C1 CC1(C)CCCC(CNC(C2CC(NC(=O)CC3NC(=O)NC3=O)C2)=O)O1 CC1CC(NC(=O)C#CC(C)(C)C)CCN1C(=O)C(=O)N(c1ccccc1)CC1CC1 C1(C(NCCC(=O)OC)=O)CCC(C)O1 c1(CSCCC(=O)N(CCOC)CCNC(C2(C(F)F)CC2C)=O)ccccn1 C(C(C(=O)N(C(CF)CF)C)n1cc(C2CCCOC2)nn1)OCC Cn1nnc2ccc(C(=O)NC(C3CCCC3)CNC(=O)CC3(C)OCCO3)cc12 N1(C(C(C)OCCCC)=O)CCC(C(C)C(=O)NCCCCCCO)CC1 CC1(C)C2CCC(C(N3CCCC3CNC(C3CCC4CC4C3)=O)=O)C1C2 C(=O)(C1CCCc2ccnn21)N1CC(C(N)=O)(CNC(C23CC(C)C2C3)=O)C1 C1(C)(CNC(c2c(C)ccn2C)=O)CCCN(C(C2CC2CC2CC2)=O)C1 C1(c2cn(CCCOC)nn2)CC2CCC1N2C(=O)CCCc1cccc(Cl)n1 c1(C(=O)NC(C)CCCCNC(C2CCOC2)=O)c[nH]c2ccc(F)cc2c1=O C1(CC(=O)N(CCC)CC2CC2)CCCN(C(c2cnn(C)c2)=O)CC1 C1(N(C(c2cc(C(C)=O)[nH]c2)=O)C)CN(C(=O)CCc2ccn(C)n2)CC12CC2 C1(C(N(C2CCN(c3snc(Cl)c3C#N)C2)CCC)=O)COc2ccccc2O1 N1(C(c2ccc(C)c(F)c2)=O)C2CCC1CN(c1ncnc3c1ccn3C)CC2 N1(C(CC2CC(OC)C2)=O)CCC(NC(=O)C=CCn2cncn2)C12CCC2 C(=O)(C1COc2ccccc21)NCC1(C)C(C)CN(C(c2c(C)noc2)=O)C1 CC1OCCC1(F)C(N1CCC1(C)CC(=O)NCC1(CC2CC2)CC1)=O n1(Cc2n(CC(C)C)c(N(CCC=CBr)C)nn2)cnc2ccccc12 c1(C(=O)NCC2CC(NC(c3ccc(C)cc3C)=O)C2)c(N)cc(F)cc1F C1(CNC(c2cnc(C3CCOCC3)s2)=O)CCC2(CN(C(=O)CO)C2)O1 c1(NC(C)=O)cnc(O)c(C(=O)N(CCNC(C2CC3(CC3)CO2)=O)C2CC2)c1 c1(C(=O)NCC(CO)NC(C2N(CC)CC2)=O)c[nH]nc1-n1cnnn1 c1(C(N2CC(NC(c3cnc(-c4cccs4)s3)=O)C2)=O)[nH]cc2c1CCCC2 C1(C(N2C(CCCC)CCC2)=O)CN(C(c2nc(C)sc2C)=O)CC12CC2 C1(C(=O)NCCCCCC#C)CC12CCN(C(C1(C#C)CC1)=O)C2 N1(CC(=O)NC(C(=O)NCCOCC2CC(=C)C2)C2CCC2)CC2CC2C1 Cc1ccc(NC(=O)C(CC2CC2)NC(C2CC(C)(O)C2)=O)cc1 C#Cc1cnn(CC(=O)NCC2CCCC2NC(C2CC(C)=NO2)=O)c1 Cc1cc(NC(=O)C(F)OC(F)(F)F)ccc1NC(C1CC1C)=O CCC(CC)C(C)C(=O)N1CCCC(N(C)C(c2cc[nH]c2C)=O)CC1 CC1CCCC(C)N1CCC(N1CCC(C)(NC(=O)CCc2cnn[nH]2)C1)=O C1(C(=O)NC2(C3N(C(C(CC)CC)=O)CCCC3)CC2)CC12CC(F)(F)C2 C(=O)(C1CCCn2cncc21)NCCC(C)(C)CNC(c1cccc(F)c1)=O c1(CCC)cc(C(=O)NCC2CCCN(C(c3cn(C4CC4)cn3)=O)C2)n(C)n1 C(CCC(=O)N1CC(COC)(NC(=O)C(C)N2CC(C)C2)C1)OCC CC(C)CCC(C(=O)NCc1cnn[nH]1)NC(C1CCOC1=O)=O N1(C(CN(C)C)=O)CCC(C(N2CCC2CC2CC2)=O)(CO)C1 C=CC(C)(CC)C(=O)NCC(C)(Cn1cccn1)NC(c1cc(F)n(C)n1)=O c1(C(=O)NC(CNC(Cc2ccc(C)o2)=O)(C)CO)n[nH]c2c1CCOC2 c1(C(C(=O)NCC2C(OC)COC2)C)ccc(Cl)c(Cl)c1.n12cc(nn1)SCC2 Cc1cc(F)ccc1C(=O)NCC1CC2CCC1N2C(=O)C(c1cnn(C)c1)C Cc1cc(=NCc2cnn(C)c2)[nH]c(=NCC2NC(=O)c3ccccc32)[nH]1 CCCCS(=O)(=O)NC(C(=O)NC1CC1NC(=O)CC1(C)OCCCO1)C(C)C N1(C(=O)CCn2cc(CN3CCCC3=O)nn2)CCc2[nH]nc(O)c2C1 N1(C(c2c(CNC(C(C=CC)O)=O)cco2)=O)CCN(CC(=O)NC)CC1 Cc1cccc(C(CNC(=O)C(O)CF)NC(C2CCCC2O)=O)c1 C1(CC)C(NC(=O)CCc2cscn2)CCCN1C(=O)Cn1nccn1 C=C1CCC(C(N2CC3CC2C3C(=O)NC2CC(C(F)F)C2)=O)CC1 N1(C(c2cncc(-c3ccoc3)c2)=O)CCC2(CCNC2)CC1 N1(C(C2(NC(c3c(C)ncnc3)=O)CC(F)(F)C2)=O)CCc2c(cnn2C)C1 C1(NC(c2n(C(C)C)ccc2)=O)CC2CCC1N2C(=O)CCC1(C)CC1 C(C(C(C)(C)C)NC(c1ccnn1C(F)F)=O)NC(C(c1cn(C)nc1)(F)F)=O N1(C(N2CCCCC2)C(=O)Nc2ccc(C)nc2)CCc2nc(CN)ncc2C1 C1(C(=O)NCC23C(CN(C(CN(C(COC)=O)C)=O)C2)C3)CCn2ccnc2C1 C1(NC(C(CC)N(C)C)=O)C2CCC(C(=O)O)CC2C1 C1(CC)CN(C(=O)CCc2cnc(C)s2)CCN1C(c1cnc(CO)nc1C)=O c1(CN2C(C(=O)NC3CCS(=O)(=O)C3)CC(OC)C2)ccc(F)cc1O C1(NC(COCC)=O)CCC(NC(C2CCC3(CC3)C2)=O)CC1 c1(OCC(=O)N(CCCCCNC(=O)C(C)(C)C(N)=O)C)nn(C)cc1[N+](=O)[O-] N1(C(C2(C(=O)OC)COC2)=O)CCCC2(CCCN2C(=O)C2=CCCSC2)C1 CC(C(=O)NC1CC1C(=O)N(CC1CCCCC1)Cc1ccnn1C)S(C)(=O)=O c1(C(N2CC(C)(NC(CN(C)CCO)=O)C2)=O)cc(C(N)=O)ccn1 C1(CNC(c2onc(C(C)(C)C)n2)=O)COCCN1C(=O)CC1CCCCO1 C1(CC)CN(C(=O)CC2CCOCC2)CCC1NC(=O)CN(c1ccccc1)C CCCC(C)CCCC(=O)N(CCNC(=O)CN1CCC(C)CC1)CC1CC1 n1(CC(=O)NC(CNC(C2C(SC)CCC2)=O)C)ncc2cc(C)cnc12 c1(C2CCN(C(C(=O)NCC3(SC)CCC3)=O)C2)cccc([N+](=O)[O-])c1 c1(NC(C2CN(C(=O)CN3C(=O)C=CC3=O)CCC2O)=O)cnccc1[N+](=O)[O-] Cc1nc(C#N)cc(=NCC2CCCCN(C(=O)C(=O)NCC3CC3)C2)[nH]1 C1(C(=O)NCC(N)=O)COc2ccc(-c3cnn(CCO)c3)cc2C1 Cc1coc(C)c1C=CC(=O)NCCOC1CN(C(C2CCCC(=O)C2)=O)C1 N1(C(c2cc(C)nn2C2CC2)=O)CC2CCC1C(CNC(C1CC1C)=O)C2 C12(C(=O)NCCN(C(C(C)OCCC=C)=O)C)CC3CCC(CC(C3)C1)C2 c1(C(C(=O)Nc2ccc(F)cc2)N(C(CC(=O)OCC)C)C)ccccc1Br C(CCN=c1ccc(S(C)(=O)=O)c[nH]1)N(C(=O)C(C)NC(=O)CC(C)(C)C)OCC C1(NC(=O)Cn2ncnn2)CC2CC1CN(C(c1cn3ccccc3n1)=O)C2 C1(C(=O)OCC(=O)NCCC2CC3C=CC2C3)CC2(CCC(F)(F)CC2)CO1 C1(C(=O)NC2(C(=O)NC3(C(C)(F)F)CC3)CC(CO)C2)CC12CCOC2 C1(NC(C(CNC(C2CCCN2C2CC2)=O)N(C)C)=O)CC(O)C(O)C1 n1(CC)nc(C)c(C(=O)NCC(F)CNC(=O)CCC2(C)CC2)c1C c1(C(=O)OC)cc(OCC23CCC(CN(C(=O)OC)C2)C3)cc(S(C)(=O)=O)c1 C(=O)(C(F)(F)C(C)(C)O)N1CCC(NC(C(CN(C)C)O)=O)(NC(C)NCCCBr)C1.C(C)SC Cc1cnc(C(=O)NC23CC(NC(C4CC(=O)N(C(C)C)C4)=O)(C2)C3)c(F)c1 C(=O)(CCO)NC(C)CCN.c1(C(N2CC(C(N)=O)C2)=O)coc(NC(N)=O)n1 c1(OC)cnc(F)c(C(=O)N(CC(C)CNC(c2cccn2C)=O)C)c1 CN1N=CC(CC(N2CCC(CC(=O)NCC#CC(F)(F)F)CC2)=O)C1=O C1(NC(c2cc(C)oc2)=O)CCOC12CCN(C(=O)C(C)(C)O)CC2 C(CC(C)C)(C(=O)N1CCCC1CNC(C1CC2(C1)CC(O)C2)=O)NC(C)=O N1(C(c2n(CC)cnn2)=O)CCCC(N(C(=O)C(c2ccc(Cl)cc2)O)C)CC1 C(c1cnccc1C)=CC(=O)NC(C(C(C)C)NC(C=NOC)=O)C c1(C(N2CC(N(C(c3cc(C)c(F)cc3)=O)C)C2)=O)ccc2c(c1)C(=O)OCC2 c1(C(N2CC(NC(C3(C)COC3)=O)C(F)C2)=O)cc2cc(Cl)cnc2o1 Cc1ccc(SCC(N2CC(CC(C)NC(c3ccoc3Cl)=O)C2)=O)c(C)c1 c1(C(=O)NC2CCN(C(=O)CNC=O)CCC2CO)cc(=O)c2ccccc2[nH]1 c1(C(=O)Nc2cc(CC(=O)NC(CCSCC)C)on2)cccc(O)c1 C(CN=c1ccnc(NC(=O)C(F)(F)CN2CCCC2)[nH]1)CCN(CC)CC C1(CNC(c2occc2C2CC2)=O)CCCN(C(c2cscc2Cl)=O)CC1 CCCC(C(O)C(=O)NC1CCCCC1(C)C)NC(c1cnn(CC2CC2)c1)=O c1(C(=O)NCC2CCCCN(C(C3OCCO3)=O)C2)cc(O)nc2c1CCCC2 CC1CC2(CC(C(=O)NCC3(CNC(C45CSCC4C5(F)F)=O)CC3)C2)C1 C1(CNC(c2cc(OC)ns2)=O)CC12CCN(C(C1(c3ccno3)CC1)=O)CC2 c1(C(=O)NC2(CO)CC3CCC2C3)cnn2ccncc12 C(CC(=O)NCC(F)Cl)(C(C)OC)NC(c1c(CC)n(CC)nc1)=O C1(CNC(C(C)OCCOC)=O)CC2(CC2)CN1C(=O)CCC1OCCO1 CCS(=O)CC(=O)NC(CNC(c1ccc(C(N)=O)o1)=O)C(C)C C1(NC(C(C)NC(C)=O)=O)C2CCCN(C(c3cncc(CO)c3)=O)C2C1(C)C C(C(CC(=O)NCC1CC12CC2(F)F)C1CCC1)NC(CCC)=O c1(OC(C)C)cccc(CC(=O)N(CC(C)(C)NC(C2CCCOC2C)=O)C)c1 C(CC(F)F)(C(=O)N1CC(C)(C)C1CO)N(C)C(c1ccn(CCF)n1)=O C=CC(C)(CCOC)C(=O)NC1CN(C(c2c(C)ccc3nonc23)=O)C1 C(CN=c1[nH]c(N2CCCC(Cc3cnn(C)c3)C2)nc2c1SCC2)N(C)CC C(CC(O)CN)NC(=O)CN.c1(C(C(=O)NC2CC2)=O)ccc(C2CCCO2)[nH]1 C12(NC(C(=O)NCC(CC)O)=O)CCC(OC(C)(C)C)(CC1)C2 CCCC(CNC(C1CC2(CCO1)CC2)=O)C(=O)N(CCCF)CC CCCC(C)(CC)C(=O)N1CCCC(NC(C2CCCC(F)C2)=O)C1 O(NC(=O)C(CNC(c1cnc(C)s1)=O)C(C)(C)C)Cc1cccc(C)n1 N1(C(C2C(C(=O)OC)CCCC2)=O)CCN(C(C2CCCC2F)=O)C(CCO)C1 CCCC(C(=O)N(CC)CC1CCCN1C(=O)CNC(C)=O)OC C1(NC(C2C(CC)CCN2C(c2ccoc2Cl)=O)=O)CC(C)(C)OC1=O Cc1ccccc1CC(=O)Nc1ccc(C(=O)NCCCCO)nc1 C12(C(N(CC#C)CC=C)=O)COCC1CN(C(=O)COCC(C)(C)C)C2 C1(C(C)C)CN(C(c2cc(Cl)no2)=O)CCN1C(=O)CCc1cnn(C)n1 c1(C(N2C(CN(C(=O)CC3CC(F)C3)CC)CCC2)=O)cn2cc[nH]c(=O)c2n1 c1(C(N2CCC3(C(C(N(C)CCC4CC4)=O)C3)C2)=O)cnc2ccoc2c1 C(=O)(CCC(C)S(C)(=O)=O)NCCOCCNC(C1(C(=O)OC)CCCCO1)=O Cc1cc(C(=O)NCC2COCCN2c2ncncc2C#N)cc(C)c1O C(=O)(C(C)(C)C(=O)N1CCC=CC1C(=O)Nc1cc(C)ccc1F)OCC c1(CNC(C2N(C=O)CCC2)=O)nc2c(s1)CN(C(=O)CC1CCCC1)CC2 c1(C(=O)NC2CN(C(c3cccc(C)c3)=O)CC23CC3)ccc2n[nH]cc2c1 O(NC(=O)C(C)(C1CCC1)NC(c1cc(C(N)=O)c[nH]1)=O)C(C)(C)CO C1(CC(=O)NCC2CCC(NC(=O)CN3C(=O)CNC3=O)C2)CC2(CCC2)C1 C1(C(N(CCCC(N2CC(O)(CC=C)C2)=O)C)=O)CCN(C)C(=O)C1 c1(SC)cccc(F)c1C(N1CC2CC1C2NC(=O)C(n1nc(C)cc1C)C)=O c1(CC(=O)NC2CCC(NC(CC(C)F)=O)CC2)cccc2c1SCCC2 C(CN=c1[nH]c(=NCCOCC2(C)CCC2)c2cc(F)cc(F)c2[nH]1)OC(C)C CC1OC2(CO)CC1(C(=O)NCCC1(NC(=O)CC3CC=CCC3)CCC1)C2 C12CCCCC1C(=O)N2.N1(C(c2c(SCC)cno2)=O)CCCC1(C)CN=[N+]=[N-] c1(NC(CCNC(C2(C)COC2)=O)(C)C)cc2c(cn1)C(=O)CCC2 C1(CNC(C2CCC(NC(C3(c4cc[nH]n4)CC3)=O)C2)=O)CCC(F)(F)C1 C1(C)(CNC(C(CSCC)NC(=O)CCc2cc(C)no2)=O)C=CCCC1 c1(C(N(c2cccc(OCC)c2)C)=O)cnc(O)c(C)c1.C12CC(C1)NC(=O)C2 C1(NC(c2cc(CF)on2)=O)CCCC(NC(c2cc(Br)cs2)=O)C1 N1(C(COCc2c(C)cccc2)=O)CCC2(CCCN2c2nc(Cl)ncc2F)C1 C(=O)(C(C)C(O)C(C)C)NCC1ON=C(C(=O)NCCC(COC)(C)C)C1 c1(NC(=O)NC(CC#C)Cc2ccccc2)ccc2cnn(CCCCOC)c2c1 C1(OC)COCC1N(C(=O)C#CCNC(=O)C(N)=O)C CN1CCCN(C(C2CC3CCC2N3C(=O)CN2CCSCC2)=O)CCC1 n1(CC)ncc([N+](=O)[O-])c1NC1CN(C(=O)NC2CCC(SC(C)(C)C)C2)C1 C(=O)(CC(CN(C)C)C(F)F)NC1C(N(C(C=C(C)C(F)F)=O)C)CCCC1 C1(NC(C=CC)=O)CCN(Cc2ccc(CCCCCC)s2)CC1O C1(NC(c2n(CC)ncc2Cl)=O)C(=O)NCCC1C C1(CNC(C2CN(CC(F)F)C2)=O)CN(C(=O)CCNc2ccccn2)CCO1 c1(CC)ccc(-c2ncccc2C(=O)NCC2CC3C=CC2C3)cc1 c1(C(=O)NC2C(NC(CN(C)CC)=O)CC2)cc(S(N)(=O)=O)c(F)c(F)c1F Cc1c(F)ccc2[nH]c(C(N3CCC(NC(=O)CC(C)C)C(F)C3)=O)cc12 N1(C(=O)N(Cc2ncccc2F)Cc2ccc(F)cc2)CCOCC1CO N1(C(c2csc(Cl)n2)C(=O)NCCCOC)CCOC(C(C)(C)O)C1 N1(C(C2CCN(C)C2)=O)CC2CN(C(=O)COc3ccccc3)CCC12 N1(C(C(C(C)NC(CC=CC=C)=O)C)=O)CC2(CCC1CO)CC2 N1(C(C2(C)ON=C(C)C2)=O)C(C)C2CC1C2NC(c1ccc(Cl)o1)=O C(CC(=O)NC1(C)CC1C)OCCCNC(COCC=C)=O c1(C(N(C(CN(C(C2(CCOC)CCC2)=O)C)C)C)=O)cc2ccncc2s1 N1(C(C(=O)NC(C)C)=O)CCC2(CCCN(C(=O)CN(C)S(=O)(=O)N(C)C)C2)C1 c1(C(N2CC(O)(CNC(COCc3c(C)cccc3)=O)C2)=O)cc2occc2[nH]1 c1(C(F)(F)F)ccccc1CCCc1noc(-c2cnc(-c3ccccn3)s2)n1 c1(NC(Cn2cc(-c3ccc(C)c(C(F)(F)F)c3)nn2)=O)cc(Cl)c(O)c(Cl)c1 C(=O)(CC(C)(O)COC)N1C(C(=O)NC(C(=O)N(C)CC)C)CC1 Cc1ccn2ncc(C(N3CCC4(CC3)CC(NC(C3CCCO3)=O)C4)=O)c2c1 c1(C(=O)NCC2COCCN2C(C2CC23CCSCC3)=O)ccnc2ccsc12 CC(C(=O)N1CCCCC(NC(=O)COCC2CCCC2)C1)C(C)(C)C C1(NC(=O)C=Cc2ccoc2)CCOC12CCOC2.c1(C2CO2)ccccc1 CC1(C(=O)NCC2(F)CC(NC(=O)CC3(C)CCCO3)C2)CCCCO1 C1(CNCC(Br)=C(C)C)(CO)CC2(C1)CC(F)(F)C2 c1(CCOC(c2cnnc(C3CC3)c2)=O)ccc(F)cn1 CC1(C)CCC(C(=O)NCCc2ccccc2F)CN1C(=O)C(C)(C)C(C)(C)O C1(NC(c2ccc(COC)o2)=O)CC12CCN(C(=O)C1=CCCC1)CC2 C1(C)(C(=O)NCC2(F)CCC(NC(C(CCOC)C)=O)C2)C(C)(C)C1(C)C c1(C(C)C)nc(C(=O)NC(C)(CNC(c2nocc2Cl)=O)CO)co1 C12(C(=O)NC3(CC=C)CCN(c4snc(C)c4C#N)C3)CC=CC(C1)OC2 CCC(F)(F)C(=O)NC(CC(=O)NCCN1CC=CC1)C1CC1 c1(NCc2c(C)non2)cc(NCc2nncn2CC(C)C)ncn1 CN1CCOC(C(=O)NCC2CCCN2C(C2(C(C)(C)O)CCC2)=O)C1 N1(c2nc(OC)nc(C)c2)CC2CCC1C1CN(C(=O)C3=CS(=O)CCC3)CC21 C(c1cccnc1)=CC(=O)NCC(=O)NCC(C)NC(c1c(OC)csc1)=O c1(C(N(CC(CC)NC(c2c(CC)occ2)=O)CC)=O)ccnc(C)n1 N1(C(=O)C2=C(Cl)CC2)CCC2CCN(C(=O)Cc3csc(Br)c3)C2C1 Cc1cccc(SC(C)C(N2CCC(CF)(NC(c3cccnc3)=O)C2)=O)c1 Cc1cc(NC=O)ncn1.c1(C(=O)NC(C)CN(C)C(=O)OC)csc(NC(C)(C)C)n1 c1(C(=O)NC2CC3CC2N(C(=O)C(C2(O)CCCC2)F)C3)nc2ccccc2[nH]1 N1(C(CC2CC(OC)C2)=O)CC2CC(C)N(C(=O)CCc3cc(C)no3)C2C1 CCC(C)(C(=O)NCCOC1CN(C(c2cc(C(=O)OC)ccc2O)=O)C1)C(N)=O Cc1ccc(C(=O)NCC(c2cccc(O)c2)CO)c(O)c1 c1(C(N(C(C(=O)Nc2ccc(OC)cc2)C)C)=O)cc(=O)cc(Cl)[nH]1 Cn1nnc(Br)c1CNC(=O)NCC1CCOC1 c1(C(=O)NC2CC(NC(C(CC)NC(=O)OCC)=O)C2)ccccc1OC(C)C S(=O)(=O)(c1c(C)nn2cc(Br)cnc12)NCC=CS(CC)(=O)=O C(=O)(C1=CS(=O)CCC1)NCc1ccc(CNC(=O)CCC2OCCCO2)cc1 N1(C(c2cnn(C)c2F)=O)C2CCC1CN(C(=O)CC1CCOC(C)(C)C1)C2 N1(N(C(c2ccccc2)CO)C)CCOCC(C=O)C1.C1(C=O)CC(C)(O)C1 c1(C(C)C(N2CCN(C(c3ccco3)=O)CCC2C)=O)ccccc1S(N)(=O)=O C(CC(CC)C(=O)N1CCCC1(C)CCC(=O)NCC1CC(OC2CC2)C1)=CC N1(C(C2(C#C)CCCCC2)=O)CC2CCC(C(=O)OCCC(C)SC)(C2)C1 C1(NC(CC=C)=O)(CNC(c2sc(-c3cccc(F)c3)nc2C)=O)CCOCC1 c1(SC)cc(F)ccc1C(=O)NCCC1COCCN1C(C1CC1C(F)(F)F)=O C1(C(=O)NCC(c2ccccc2)CNC(=O)CC2C=CCCC2)CC2C=CC1O2 N1(C(Cc2ncc(C)[nH]2)=O)CCC2(C1)CN(C(=O)COC1CCCCCC1)C2 C(=O)(CC(C(F)(F)F)NC(=O)CCC1CCN(Cc2cccc(F)c2C)C1)OC c1(C(=O)NC2C(NC(CC(=C=C)C)=O)C2)ccc2cccc(O)c2c1 c1(CC(=O)NC2CN(C(C(CC(C)C)(F)F)=O)CC2C)coc2cc(O)ccc12 C12(NC(CC3C(OCC)COCC3)=O)CCCN(C(c3ccno3)=O)CC1C2 N1(C(C2CS(=O)(=O)CC(=O)N2)=O)CC2CC3CC2C1C3NC(=O)C#CC1CC1 C1(NC(C(C)=C(C)C)=O)CC1C1CCCN(C(=O)CC2CC3CCC(C2)N3C)C1 N1(C(CSc2ccc(C)cc2)=O)CC(CO)C2(C1)CN(C(=O)C(=O)NCC1CC1)C2 C1(N(C(C(C)N(C(C)=O)C)=O)C)CN(C(c2occc2C)=O)CC1(C)C C1(F)(CNC(=O)CCc2nnc(S)nc2O)CCN(C(c2cnc[nH]2)=O)CC1 c1(C(=O)NCCC2CC(NC(C3C(CC)OCC3)=O)C2)c(C)[nH]c2ncccc12 C1(CNC(CC2CC(CC)OCC2)=O)CC2CCC1N2C(=O)Cc1cnsc1 C1(C(=O)NC2CCN(CC#N)CC2O)CCC2COCCC2O1 N1(C(C(C)(F)F)=O)CCCCC1C1(NC(c2cnc(C(F)F)s2)=O)CC1 c1(C(N2CC(CNC(CCSC)=O)OCC2)=O)cnn2c1NCC(C)C2 CCCS(=O)(=O)C(C)C(=O)N1CCCC(CNC(c2nocc2Br)=O)C1 C1(C(N(CCN(C(c2c(C(C)C)c[nH]n2)=O)C)C(C)C)=O)CCCOC1C c1(CC)cc(C(N2CC(NC(C3CC3C)=O)C(O)C2)=O)sc1-c1ccc(F)cc1 c1(C(=O)NCC2CC(OC)CN2C(c2cc(O)nn2C)=O)nccc(N)c1Cl c1(C(N2C(CNC(C3(CC)COC3)=O)COCC2)=O)cc(Cl)c(Cl)n1C c1(OC)cncc(C(=O)NC(C(=O)N(C)CCc2cccs2)C2CC2)n1 N1(C(c2c(C)oc(Cl)n2)=O)CC(=O)N2CCOCC2(CNC(=O)C(C)N(C)C)C1 CC1CCN(C(=O)CN2CCC(OC(=O)CCC(C)(F)F)C2)CC(C)O1 C(=O)(CN1C(=O)Cc2ccccc21)N1C2CC(NC(C(C)CN(C)C)=O)(C2)C1 CC1CN(C(C2(C)CN(C(c3ccnc(Br)c3)=O)C2)=O)CCc2ccc(Cl)cc21 C1(C(N(CCCO)C)=O)COC2(CCN(C(=O)C=CC(=O)O)CC2)C1 c1(CNC(C(COC)NC(C2CCCC2O)=O)=O)cccc(F)n1 c1(C(C)C)cccc(C(=O)NC(C)C(C)(C)NC(=O)CC2(O)CCOC2)c1F C1(CC(=O)NC(C#C)CC2CCC2)CN(C(c2cc(C)c(C)o2)=O)C(C)(C)C1 CC1NC(=O)N(CCC(=O)NON2CCN(C)CC2)C1=O.CCC(F)(F)F C1(C)(CC)CC(NC(=O)COC(=O)CO)CN1C(c1cc(N)ccn1)=O N1(Cc2cnc(C)o2)CCC2(CCCN(C(c3ccc([N+](=O)[O-])o3)=O)C2)C1 CCCCC(CNC(=O)C(C)(C)c1ccno1)NC(=O)CCC1CCCOC1 c1(OC)cc(C(=O)NC2CCN(C)CC2)ncc1-c1ccc(CNC(C)=O)cc1 N1(C(Cc2n(C)ncc2)=O)CCCCCC1C1CCCC1=O c1(C(=O)OCC)cc(NC(C2CC(C)N2C(c2ncccc2C)=O)=O)n(C)n1 c1(C(=O)NC(C(=O)NC(C)Cc2ccco2)C(C)O)ccnc(O)c1F C#CC(CNC(=O)CC1CCCN1C(=O)C(N1CCCCC1)C)CC(C)(C)C C1(CNC(=O)OCC)CC(C)CN(C(=O)C(=O)NCCC2CCC(C)(C)C2)C1 c1(C(=O)NC(C)(CNC(c2ccc(Cl)o2)=O)C2CCC2)ccc(F)cc1C1CC1 C1(C(N2CC(C)C(NC(c3ccc(=O)oc3)=O)C2)=O)CCC(C)(C)CO1 N1(C(C2(CCOC)CCC2)=O)CCC(CCC(=O)N(C)C(C2CCOCC2)C)C1 Cc1cccc(NC(CN2C(C3CC3)CCC2)=O)c1.C12(C(=O)N(C)CC3CC3)CC1C2 C1(CC)CCCN(C(c2cc(C)[nH]c2C)=O)C1C(=O)NCCN(C)C(N)=O CC(c1cnn(C)c1)=CC(=O)NCC(C)(C)CN(C)C(c1cnc2n1CCC2)=O C(CCCC(C)(C)C)OC(=O)NCC(C)NC=O.C(C)(C)(C)O.C=CCOCC c1(C(N2CCCC(N(C(C(C)N(CC)CC)=O)C)C2)=O)c(C)ccnc1C C(C(C(=O)NC1CN(C(=O)C(F)n2ccnc2)CC12CCC2)C(F)(F)F)OC CCC(C)(C)CC(c1nnnn1-c1ccccc1Cl)Nc1ccc(F)c(I)c1 CC(C)(C(=O)N1CC(n2ccnn2)C1)C1=CCN(C(C2CCCCS2)=O)C1 N1(C(C2(C#C)CCC2)=O)CC2(CCN(C(C3CCN(C)C(=O)C3)=O)C2)C1 Cc1ccc(CC(C)C(N2CCC(O)(CN(C)C(C3CC3C(N)=O)=O)C2)=O)cc1 N1(C(c2ccc(OCC)cc2)=O)CCC(NCc2cccnc2OC)C(C)C1 N1(C(CNC(CCC)=O)=O)CCCC2C1CCN2C(c1cc(CO)c(C)o1)=O C1(NC(c2cccc(OC)c2O)=O)CN(C(=O)CCC(N)=O)CC12CCOCC2 Cn1cc(C(N)=O)cc1C(=O)NCC1CCCN(C(=O)Cn2nccn2)C1 C1(NC(=O)C#CC2CC2)CC2CC1CN2C(c1cc2[nH]ccc2s1)=O c1(NC(C)C(=O)N(C)Cc2nnc(CC)s2)cc(Cl)ccc1C#N c1(C(C)CNC(=O)CNC(=O)CCc2ccccc2F)ccc(F)cc1 C1(C)(C(=O)NC2CC(NC(c3c(OC)c(Cl)ccc3)=O)C2)CC(C2CC2)=NO1 CC(CNC(C1CCC(C2CC2)N1C(=O)CC(C)(F)F)=O)CCCO C12(CNC(c3c(C)nc[nH]3)=O)CCC1CCN2C(=O)CNC(N1CCCC1)=O c1(C(N2C(CNC(C3CCCOC3)=O)CC(O)C2)=O)ccc2ncccc2c1 c1(NC(C2CC23CCCC3)=O)cccc(NCc2cn(CC3CCCC3)nn2)c1 C#CC1CN2CC(NC(=O)CC(c3ccccc3Cl)C)(CO1)CO2 C1(NC(c2scc(C)c2)=O)CCCN(C(c2cc(Cl)c(Br)cn2)=O)CC1 c1(C(N(C2CCCC(NC(c3ccnc(C)n3)=O)C2)C)=O)c(C)nn(C)c1C N1(C(C#CC(C)(C)C)=O)CCc2[nH]nc(CNC(C3CC3F)=O)c2C1 Cc1cc(Cl)c(C(=O)NCC(C)NC(c2cc(S(=O)(=O)N(C)C)c[nH]2)=O)cc1F N1(CCOCC)CCCC1(C)NC(CC1(C)N(C(C=CCOC)=O)CC1)=O c1(NC(CCC)=O)ccc(NC(=O)C(C)Cc2cccc(F)c2)c(C)c1 c1(CNC(CN(C(=O)CCn2ccnc2)CCC)=O)cnc(CC)[nH]1 CC1(C)CC(NC(=O)C2=CSCCO2)CN1C(=O)CCCN1CCOCC1 N12CCC(O)(C1)C2=O.CCCC(C)N(CC(N)=O)C(=O)CC1CC=CC1 C=C1CCC(C(=O)NC(C)(CNC(C2CC=CCC2C(F)(F)F)=O)C(C)C)CC1 c1(C(N2C(CCNC(C(=O)NCC)=O)CCC2)=O)cccc(CC#N)c1 C1(CC(C)C)CNCCN1C(C1CC(C)(C(C)(C)C)C1)=O C1(NC(C2(NC(C3N(CC)CC3)=O)CCN(C)C2)=O)CCC2(CC1)N=N2 c1(CC(N2CC3(CCN(C(C(C4CC4)OC)=O)C3)C2)=O)ccc([N+](=O)[O-])cc1F CC1CCC(NC(=O)CCC2NC(=O)NC2=O)CN1C(=O)C(Cl)=CCl N1(C(=O)Cn2nc(-c3cccs3)oc2=O)CCN(C(C2CCOC2)=O)CC(O)C1 Cc1cc(F)ncc1C(=O)NCC1CCN(CC(C)O)CC1 N1(C(C2CN(C(C3CC(C)=C(C)CC3)=O)CC2C)=O)CCCC(O)(C2CC2)C1 CC(CCC(=O)N(CC(C)C(=O)NCc1ccccn1)C)N1CCCCC1 C(CN=c1[nH]c(C(F)F)nc2c(C)csc12)(C1CCOC1)OC Cc1nnc(C(=O)NCC2(NC(=O)Cc3cncs3)CC(F)(F)C2)n1C C1(C(=O)NCC(C(C)(C)C)NC(C(C)(F)F)=O)CCn2c(Br)cnc2C1 N1(C(c2c[nH]nc2-c2cccnc2)=O)CCOCC12COC2 FC(F)(F)CCNC(=S)NC1(c2ccccc2)CCOC1 N1(C(c2ccc(C)cn2)=O)CCCN(C(C2(F)CCCOC2)=O)CC1C(C)C c1(C(C(=O)NCC(CCCC)NC(=O)CCCC(F)F)=O)ccc(F)c(C)c1 C1(C(=O)NC2CCC2NC(=O)Cc2cnc(-c3ccco3)s2)CC=CCC1 CC(C)C(CNC(=O)CSc1ccccc1)NC(c1cc[nH]n1)=O Cc1nc2n(n1)CC(C(N1CCC3(CC1)CC(NC(=O)C(C)(F)F)C3)=O)CC2 c1(C(N(C(C(CC)C)C(=O)N2CCC(F)(C#N)C2)C)=O)ccc2nccn2c1 c1(CC)ccc(F)cc1CC(=O)N(C(C)CN(C(=O)COC(C)C)C)C C1(CC(=O)NC2(CC=C)CCN(C(=O)Cc3cncs3)C2)CCCCC12CC2 c1(C(C(=O)NC(CC)C)N(C)CC2CCCNC2=O)ccc(OC)cc1Cl N1(C(c2occ(C)c2)=O)CCC(C2CCN(C(=O)C(C)(C)NS(C)(=O)=O)C2)C1 c1(C(N(C(C)C(=O)NC2CCC3(CC2)CNC3)C2CC2)=O)ccc2occc2c1 CC1CC(c2cccc(F)c2)N(C(=O)C(c2ccccc2Cl)N)C1 c1(C(=O)NC(CC(C)NC(c2cocn2)=O)C)nc(O)nc(O)c1F N1(C(CCN(C(C)=O)C)=O)CC2CC1CCC2NC(C1CNC(=O)N1)=O Cc1ccc(F)c(Br)c1C(=O)NCC1CC1CNC(=O)CNC(c1ccoc1)=O Nc1cccc(C(N2CCOCC(NC(C3CC3C3CCCC3)=O)C2)=O)c1O Nc1cncc(C(N2CCCCC2CCNC(c2cc(Cl)c(Cl)s2)=O)=O)n1 N1(C(c2c(OC)nc(C)cc2)=O)CC=C(C(=O)NCCOCCCF)CC1 N1(C(Cc2ccc(CC(C)C)cc2)=O)CCC2(CC1)CC2NC(c1ccco1)=O c1(C(N(CCC(C)NC(CCCC(C)C)=O)C)=O)ccc2nnn(C)c2c1 CC#CCCCC(=O)N(C(CC)CC(N1CCN(CC)C(=O)C1)=O)C N1(C(C2(F)C(C)OCC2)=O)CC(C)CN(C(c2cc(C(C)(C)C)on2)=O)CC1C C1(CCSCC(=O)NCCOCCOCC(=O)OC)COCCC1C c1(OC)cnc(C(N2CCC(NC(=O)CSCc3ccnn3C)CC2)=O)cn1 c1(C(=O)NC2C(NC(C(N3CCC(O)CC3)C)=O)COC2)ccn2cncc2c1 C1(C(F)(F)F)(C2CC2)C(=O)Nc2cccc(c2)N1.C(=O)(C(F)(F)F)N(C)C CC1CN(C(c2ccc(C(F)(F)F)cn2)=O)CCC1NC(=O)C(O)CN(C)C C1(NC(C(COC)N(C)C)=O)(CNC(=O)CCN2CCOC2=O)CCCCC1C Cc1c(C(=O)NC2CN(C(C3(c4ccn(C)n4)CC3)=O)CC2C)ccn1C1CC1 C(=O)(CCCCCC(C)C)N1CC(CNC(COCCC=C)=O)OCC1 C(=O)(C(O)C1=CCCCC1)NC1CN(C(c2cnc(OC)c(C)n2)=O)C(CO)C1 CCCC(C(=O)N(CCCN(C)C(c1cccc2ccnn12)=O)C)S(N)(=O)=O c1(C(=O)NCCN(C(=O)CCCC2CCCC2)CCC)ccn(CC(F)(F)F)c1 C(=O)(C(O)CC(F)(F)F)N1CCC(N(C(=O)CC2CCC(C)(C)CO2)CC)CC1 c1(C(N(C)CC2CN(C(C(C)=C(C)C)=O)C2)=O)ccc(NC(=O)C(C)(C)C)cc1 n12nc(cc1C(=O)O)NC(=O)CN(C)CC2.C1(CC)CCCN1C(=O)CC(C)C c1(C(=O)OCC(C(=O)NC)C)cc(C)sc1S(N)(=O)=O CCC(CNC(=O)CCS(C)(=O)=O)(CC)C(=O)NCC1(C)CC1(C)C N1(C(C(C=C)O)=O)CCN(C2CN(C(=O)CC3COC(=O)C3)C2)CC1 C1(C(N2C(CCC)CCC2)=O)CCCCCN1C(=O)CC1CC(F)(F)C1 N1(C(C2(CC)CCCC2O)=O)CC2=C(C1)CN(C(c1cc(F)ccc1C)=O)C2 c1(C(N(C)Cc2cc(F)ccc2Cl)=O)c[nH]c2cc(Cl)c(Br)cc12 O=C(C1=COCC1)N1CCCC(NC(C2(CC3CC3)CC2)=O)C1 C(=O)(C(C)(F)C(=O)NC(CNC(c1ccc(OC)nn1)=O)C1CCC1)OC N1(CC(c2cccc(Cl)c2)OC)CCCC(C)C1.C1(=O)NCCN1 C1(CNC(c2c(CC)occ2)=O)CN(C(C2(NC(N)=O)CC2)=O)CC1C N1(c2c(C)cnc(C)n2)CC2(CC(NC(c3cnc4ncnn4c3O)=O)CO2)C1 Cc1ccc(OC(C)(C)C)c(-c2csc(=NCc3cnn(C)c3)[nH]2)c1 c1(OC)cncnc1C(N1CCN(Cc2ccc(C)o2)CC1)=O CCC(CC(=O)NCCN(C(c1[nH]c(C)cc1C)=O)C1CC1)C1CCC1 CC(=O)CC(C)C(=O)N1CC2CC1CN2C(c1nc(-c2ccccc2)oc1C)=O c1(CC(=O)NC(C)CNC(=O)C=CC(F)(F)F)ccc(Cl)c(Cl)c1C C12(CNC(C(C)OCC(N3CC(N(C)C)C3)=O)=O)CCCN(CC1)C2 C1(C(N(C2CC(O)(c3ccncc3)C2)C)=O)C2Cc3c(Br)cccc3C12 c1(C(N2C3(CNC(C(C)(C)C#N)=O)CCC3CC2)=O)cnc2[nH]c(O)nc2c1 c1(C(=O)OC)cc(CN2C(C(=O)Nc3cnnc(Cl)c3)CC3CC23)ccn1 C1(C(=O)NC(CC(=O)OC)(C)C)CN(C(=O)CC2(C)CCOCC2)C2(CCC2)C1 N1(C(C(C)NC(COC)=O)=O)CCOCC1C(=O)NC(CO)C(C)(C)C CN1CC2CN(C(=O)C(=O)NCCC3CCCC3O)CC2C1 c1(CCC=C)ccc(C(=O)NCCOC2CCCN(c3ncccn3)C2)cc1 c1(CC)ccc(F)c(-c2cccc(NC(c3cc(O)ccc3Br)=O)n2)c1 C(=O)(C1=NOC(CNC(C2C3CC(=O)CC23)=O)C1)NC1(CO)C(C)(C)C1 C1(C(=O)NCC2(O)CN(C(CCCCOC)=O)C2)CCn2nncc2C1 Cc1noc(C)c1C(C)CC(=O)NCC1CCCN1C(C12CCC1CC2)=O c1(C(=O)NCC(C)(C)NC(C(CC)SC)=O)cnc2[nH]nnc2c1 c1(CC(=O)NCC(CCCC)NC(=O)CCCNS(C)(=O)=O)cccc(F)c1F C(=O)(C1=CC2(CCOC2)C1)N(CCC(N1CCN(C2=NCC2)CC1)=O)C1CC1 c1(C(=O)NCCC(C)NC(c2c(CC)ocn2)=O)cnc(OC)c(C(F)(F)F)c1 c1(C(=O)OCC)ccc(N)c(Br)c1.C1(C(=O)OCC)CC(F)(F)CN1C(C1(Br)CC1)=O c1(C(=O)NC(CNC(C(C(CC)C)O)=O)(C)C)ccc(OC)c(N)c1F C(=O)(CC1=CCCCC1)N1CC(NC(c2c(CC)nns2)=O)C(C)CC1 N1(C(CC2(COC)CC2)=O)CC(C2CC2)(C(=O)NCC2CCC(=O)N2)C1 N1(C(CC2CCC(C)C2)=O)CCCC(CCCC(=O)N(c2ccc(Cl)cc2)CC#N)C1 c1(C(N(CCCCNC(CS(CC)=O)=O)C)=O)c(C)[nH]c2ccc(F)cc12 C1(NC(C2C(C(N)=O)COC2)=O)CCCCN(C(c2cnc(C)nc2C)=O)CC1 c1(C(=O)NC(C2CN(C(c3ccccn3)=O)CCO2)C)cc(F)c(O)c(Cl)c1 O=C1NCCN2CCN(C(c3cccc(N4CC5CCC4C5)c3)=O)CC12 CCCC(C)C(=O)NCC12CC(NC(=O)C(C3CCOCC3)OCC)(CO1)C2 N1(C(C(C)CC(C)(C)C)=O)CCC2(CC1)CN(c1cccc(F)c1C#N)CCO2 C1(C(=O)NC(CO)CCO)COCCN(C(C2(n3cnnn3)CCOCC2)=O)C1 Cc1coc(C(=O)NCCCCc2cn(-c3ccccc3C(C)C)nn2)c1C C#CCCCC(=O)N(CC(C)(C)NC(=O)Cc1cc(=O)n(-c2ccccn2)[nH]1)C N1(C(c2c(CCC)nco2)=O)CC(NC(=O)CCc2cccc(O)n2)C(O)C1 c1(CC2(C)CCCC2)nc(CCCO)nn1-c1ccnnc1 c1(C(=O)OC)cccc(C(=O)NCC2CCCCC2NC(c2n[nH]cc2C)=O)n1 c1(C(=O)NC2C3CN(C(c4ccc(C(N)=O)o4)=O)CC23)cc(F)ccc1F Cc1ncc(CNC(C2CCCC2NC(C2(O)CCSC2)=O)=O)o1 CC1CC(C)(C(=O)N(C2CN(C(c3occ4c3CCOC4)=O)C2)C)CC(C)O1 C1(NC(CCSCC)=O)COCCC1C(=O)NC(CC)(CC)CO c1(-c2cc(CC(=O)Nc3cccc(C=C)c3)ncc2)cc(S(C)(=O)=O)ccc1F CCC(CC)C(C(=O)NCCn1cc(C(=O)N(C2COC(C)(C)C2)C)cn1)OC C(C(C)(C(C)C)NC(=O)CSc1nncn1C)NC(c1cc(C)oc1)=O c1(SC)cc(C(=O)NCCCCNC(=O)CCN2CCCC2)ccc1Br N1(C(c2c(C(C)(C)C)ncs2)=O)CCCC(C)(CNC(=O)Cn2cc(Cl)cn2)C1 c1(CC(=O)N(C)CCN(C)C(C2CCCCN2S(C)(=O)=O)=O)cncc(C#N)c1 C1(CNC(Cc2n(C)ccn2)=O)CC(N=c2nc(-c3ccccc3)[nH]s2)C1 Cc1cc(C(N2CCC(NC(=O)CN(C3CCCC3)C)C(O)C2)=O)c(C)n1C N1(S(CCC)(=O)=O)CCCCC1C(=O)N(CC(C)N(C)C(c1nocc1C)=O)C N1(Cc2ccc(C(C)C(F)(F)F)cc2)CCC(O)(C2CCC2)CC1 C1(NC(c2ccc(OC)c(Cl)n2)=O)C2COCC1CN(C(=O)CC1CC(C)C1)C2 c1(C(=O)NC2CC(NC(c3csc(C(F)(F)F)n3)=O)C2)c(F)cc(F)cc1Cl c1(OC)cc(CCCC(=O)OC2CCC2c2ccccc2)cc(F)c1 C1(C(N2C3CCC2COC3)=O)CN(C(=O)Cc2ccc(O)cn2)CCC1(F)F C1(CCCC)CCC(NC(=O)CN(C(c2c[nH]cc2C)=O)CC)C1 N1(C(CNC(CC)=O)=O)CCC2(CCC2NC(=O)CC(C)C2CCCCC2)CC1 N1(C(CC2ON=C(CC)C2)=O)CC2CN(C(=O)C(C)(C)C(C)(C)C)CC2(C)C1 C(=O)(CC(C)CC(C)C)N1C(CC(=O)NC(CCOC)(C)C)C2CCC1C2 CC(O)C(O)C(=O)N(C)CCNC(=O)C(=O)Nc1cccc(Cl)c1 S(=O)(=O)(c1cccc(S(=O)(=O)Nc2nccs2)c1)Nc1cc(C)c2c(c1)CCC2 Cc1nc(C)n(CC(=O)NCC2C3CN(C(=O)CC4CC=CCC4)CC23)n1 C(=O)(C(F)CC(F)(F)F)N1CC2C(C(C3CCCCN3)=O)C2C1 c1(NC(=O)NCCCNC(C)=O)nc(Cl)c2ncnc-2[nH]1 c1(-c2c(OCC)cc(F)cc2)n[nH]c2c1CN(C(c1cc(O)nc(Cl)c1)=O)CC2 C(F)(F)(C(F)(F)F)OCC(=O)NCC1(O)CN(C(C(C2CCCCCC2)C)=O)C1 C1(CN(C(=O)CC2CCCN(C(c3ccn(C(F)F)n3)=O)C2)C)CCCC1(C)C C(N=c1cc[nH]c(=NCCCCC(N)=O)[nH]1)C1(CN)CCCC1 c1(C(C)CC(=O)N(C2CN(C(C3CCOC3=O)=O)C2)C)cc(F)cc(F)c1 c1(C(N2CCC(C(=O)NC(CC)(C)COC)C2)=O)cc(C)cc(F)c1 CCCC(C(=O)N(CC(CC)NC(=O)C(O)CN(S(C)(=O)=O)C)C)OC N1(Cc2cc(C)no2)CCC(C(C)NC(=O)C2=C(Cl)CC2)CC1 C1(C2CN(C(C3CC4(CC4)CO3)=O)C2)(NC(C(CC#C)O)=O)CC1 N1(C(c2cc(C)n(C(C)C)c2)=O)CCCN(C(c2ncsc2C)=O)CC1C(C)C CC(C)CC(C)C(=O)N1CC(NC(=O)CC(O)CN(C)C)C(C)C1 C(CCCC(C(=O)NC(C)C)N1CCCC(N(C)C)CC1)OC C1(F)(CNC(c2ccnnc2)=O)CCCN(C(C23COCC2C3(F)F)=O)C1 c1(C(N2CCC3CN(C(CC4(C)CCCO4)=O)C3C2)=O)cncc2cnccc12 c1(C(=O)NC2CC(C)(CC)N(C(=O)Cc3ccc(Cl)s3)C2)ccc(O)c(C)c1C C(=O)(C1CCCn2nccc21)NC(C1CCN(C(c2c(Cl)cc(C)s2)=O)CC1)C C1(C)(CNC(c2c(CCC)n(C)nc2)=O)CN(C(C2COC(=O)N2)=O)CCO1 C1(CN(C)C(c2ccn(C(C)(C)C)n2)=O)CCCN1C(C1COC(=O)C1)=O Cc1cn(C=CC(=O)NC2CCC(N(C)C(c3conc3C)=O)C2)s1 c1(C(N(CCCC)C)=O)cc(Cn2cc(CCCCCO)nn2)oc1C c1(C(N2CC3C(CNC(CC=C)=O)C3C2)=O)c(F)cc(Br)cc1F c1(C(C)=O)ccc(N2CC(CC(C)N)C2)nc1.C(=O)(C=CC(N)=O)NC(N)=O Cc1nn(C)cc1C(=O)NCCCCC1CN(C(C2(C#N)CCCC2)=O)C1 Cn1cnc2c1CC(NC1CCCN(CCN)C1)CC2 N1(C(CC(C)OC)=O)CCC(NCc2ccccc2F)C(C)C1 N1(C(CCC#C)=O)CCN(C(=O)C(C)OCCOC)CC1CC(C)(C)C C=Cn1nncc1C(=O)NCCC(=O)N.C(C)(CC)(CC)CCCOC CC1CN(C(=O)CCn2ccccc2=O)CCC1NC(c1cnco1)=O n1(CCCN2CCN(CCC(=O)N(C)C)CC2)ccc2cccnc12 C1(C(N(OC)CCO)=O)CCC2C3CCC(C3)C12 c1(CC)[nH]nc(C(=O)NC(C)CCCCNC(=O)C=Cc2cnc[nH]2)c1Cl N1(C(COC(CC)C)=O)CCC(C(C)NC(=O)Cc2csc(Cl)n2)CC1 N#Cc1cc(C(=O)NC2CCCC2NC(c2ccc(=O)oc2)=O)ccn1 C(CC(=O)N1CCN(C)CC1CO)(C(F)F)NC(C(C)=NOCC#N)=O N1(C(c2onc(CC(C)C)c2C)=O)CC(C(=O)OC(C)(C)C)C(C2CC2)C1 C1(C(C)C)CN(C(=O)CCCNC(=O)Cc2ccc(F)cc2)CCCO1 C1(CNC(CC(C)=C(C)C)=O)CC(C)CCN1C(=O)C(C)c1ncco1 c1(NC2CN(C(CC(C)(C)OC)=O)CC2C)cc(C)nc2ncnn12 Cc1ccccc1OC(C)C(N1CC(NC(=O)COCCCF)C(O)C1)=O C(C)(C)(CC)CCOCC(=O)N(CC(=O)NC(C)(C)C1CC1)CC#C N1(C(c2n(C)ncc2Cl)=O)CCC2(CCC2)C(CNC(=O)C=CCO)C1 CCCCC(CC)CN=c1nc2ncn(C)c2c(NCc2c(Br)cnn2C)[nH]1 CC1CCCN(C(=O)COc2ccc(Cl)c(C(N)=O)n2)C1CNC C1(C(=O)NCC(C)CNC(=O)CN2CCC(=O)NC2=O)(CC)CCC(F)(F)CC1 C(=O)(CCN=c1[nH]ccs1)NCCN(C(Cc1c(C)cccn1)=O)CC(C)O C12(CNC(CC3CCN(C)CC3)=O)COCCN1CCN(C(=O)C(O)C1CC1)C2 C1(C(=O)NC2(C)CC(NC(CC(C(C)C)O)=O)C2)CNC(=O)CC1(C)C c1(CNC(C(CC#C)O)=O)nnc2n1CCN(C(=O)CSCCC(F)(F)F)C2 c1(COC)nocc1C(=O)NCC(O)CNC(C1CCC(=O)O1)=O c1(C(=O)NCC2CN(C(C(C=CCCC)O)=O)CC2O)cnc2sccc2c1 c1(C(=O)NC2CC3N(C(C(CC)C#N)=O)C(CC3)C2)nc2ccccc2cc1Cl c1(OCC)ccc(C(C)C(N2CCCC2C(C)NC(c2coc(O)n2)=O)=O)cc1 c1(CCC(N2C(C(=O)Nc3cc(C)ncc3)CCCC2)=O)cccc([N+](=O)[O-])c1 c1(C(N(C)CC2CCCN(C(C(F)OC)=O)C2)=O)c(C)nn(C)c1F C(c1cccc(F)c1F)=CC(N1CC(NC(c2cnc(C)s2)=O)C2C1C2)=O C1(NC(c2n(C=C)nnc2)=O)CCN(C(c2ccc(CCC)cc2)=O)CC1C CCS(=O)(=O)C=CC(=O)N1CCOCC1CN(C)C(c1cccc(C(F)F)c1)=O C1(C(C)C)CCC(CC(=O)N(CCN(C(=O)CC2CCN(C)C2)C)C(C)C)CC1 C1(NCCCOCCCl)CCCCC1.O=C1CN1C1CC1 CC12CCC1CN(C(C1CCCCN1C(C1CC1[N+](=O)[O-])=O)=O)C2 C1(C2(C)N=N2)CCN(C(=O)CCn2cc(C(C3CCOC3)N(C)C)nn2)C1 c1(C(N2CC(NC(C(C)(C)c3ccccn3)=O)C2)=O)ccccc1[N+](=O)[O-] CC1CN(C(=O)C(C)(C)n2cc(Br)cn2)CCN1C(C1CC2OC1C1CC21)=O C(C)(C)(C(C)CC(=O)c1nc(C(F)(F)F)c(Br)s1)NCC1CC(=C)C1 C1(C(N2CCC(C(C)O)C2)=O)(CC)CN(C(=O)CN2CCCC2=O)C1 N1(C(CN(CCC)C)=O)C2CCC(C2)C1C(N1CC=CC1CN(C)C)=O C=CCN(OC)C(=O)C(Cn1ccnn1)NC(=O)C(C)n1cncn1 C1(C(N2CC(NC(C3(F)CCN(C(C)(C)C)C3)=O)C2)=O)CC2(CCC2O)C1 C=CC1CCCN(C(=O)C=CC(C)NC(c2ccncc2Cl)=O)C1 N1(C(N)=O)CC(O)CC1C(=O)NC1C2CC1N(C(=O)CSC1CCCCO1)C2 Cc1n[nH]c2nc(O)c(C(=O)N(CCCNC(C3(C)C=CCC3)=O)C(C)C)cc12 C(CCN(C)C(c1cnn(C)c1F)=O)(C(C)C)NC(C1CCC(CC)O1)=O C#CC1(C(=O)NOCCCC(F)(F)F)CCN(C(=O)C(F)C(C)(C)O)CC1 C(C1CCCCC1)=C(C(=O)NC(C1(O)CN(C(=O)CN2CCC(F)CC2)C1)C)F C1(C(N(CCOCCCN(C(=O)Cn2ccnn2)C)C)=O)CCC=CCCC1 C1(C2CCN(C(=O)CC3CCCCO3)CC2)(NC(CSCC(N)=O)=O)CCC1 CC(CC1=CCCCC1)NC(c1c[nH]nc1CNC(C1(C)CCOC1)=O)=O CCCCCC(C)CC(=O)NCC1(C(=O)NC2CCCC2CN(C)C)CC(=C)C1 N1(C(CCCCNC(CC2C(C)(C)C2(C)C)=O)=O)CCSC2CCCC12 C(CCC(C)C)(C(=O)NCC(C)(C1CC1)C1CC1)NC(COCCC)=O c1(C(=O)NCc2oc(C)c(C(N3CC(c4nn[nH]n4)C3)=O)n2)cc(O)ccc1F CN(CCCC(=O)NC1CC2(CCN(C(c3cccn3C)=O)C2)C1)N=O c1(CC(=O)NCC(C2CCC2)NC(C2CC(=C)C2)=O)cc(OC)ccc1[N+](=O)[O-] C1(C)(CNC(c2[nH]cc(C)c2)=O)CCCN(C(c2cnc(C(F)(F)F)nc2)=O)C1 c1(CN(C)CC2CN(C(c3c(CC)occ3)=O)C2)cc(-c2nn[nH]n2)cc(O)c1 CC(C)C(C(=O)NC(C)CCCNC(c1ccnn1C(F)F)=O)C(C)C C1(F)(C(=O)NCC(CO)NC(CCCCCC)=O)CS(=O)(=O)CC12COC2 C(=O)(C(C)(C)COC)NCCN1CCC(NC(C2(C(F)F)CC(=C)C2)=O)CC1 C(=O)(C1COc2ccccc21)N1CC(C(=O)OC)C(O)C1 N1(C(n2c(C)nc(C)n2)=O)CCCCC(N(C(=O)C(=O)N)C)C1.C(C(F)F)NC(C)=O C(=O)(CC(C)(O)CCCC)N1CCC(CC=C)(NC(c2ccsn2)=O)C1 C(=O)(C(O)P(C)(C)=O)N1C(C(CNC(C2(OC)CCCC2)=O)(C)C)CCC1 C(C(C)(O)C(F)(F)F)N(CCOC)C(=O)Nc1ccc(OC)nc1 Cc1ccc(NC(C23CCC2CN(C(c2ccc(Cl)o2)=O)C3)=O)cc1O c1(C(N2C3CC(NC(C4CC(F)C4)=O)(C3)C2)=O)ccc(-c2ccncc2)c(F)c1 c1(C(N2C(C(N)=O)CC2C(N2CCC(O)(CO)CC2)=O)=O)cc(O)ncc1F Cc1cc(C)c(C(N2CC(C(C)NC(=O)C(c3cn(C)nc3C)C)C2)=O)c(S)n1 Cc1ccnc(O)c1C(=O)NCCCCC1CN(C(C2CCOC(C)C2)=O)C1 CC1(NC(c2cc(C(N)=O)c[nH]2)=O)CCN(C(=O)CCn2cc(Br)cn2)C1 N1(C(Cn2nnc(=N)[nH]2)=O)CCC2CCN(C(c3cccc(F)c3)=O)CC12 C1(CC)CCc2sc(C(=O)NC3(CN(C)C(C4CCC(C)CC4)=O)CC3)cc2C1 c1(CC(=O)NCc2c[nH]nc2CNC(C2C=CCS2)=O)ccc(F)cc1 c1(CN2CCC(NC(c3c(C=C)cccc3)=O)C2)ccc(I)c(F)c1F C(=O)(CCCC(C)(C)C)NCCC(C(=O)NCC1(COC)CCCC1)O c1(C(N2CCC(C(C)NC(=O)OC(C)(C)C)CC2)=O)ccc(C(C)(C)C)nc1 CCCCC(O)C(=O)N1CC(=O)CCC1.C(C)(C)(C)C(=O)OC(=O)C1CC1 C1(NC(C2(c3ccc(C)cc3)CCC2)=O)CCCCN(C(=O)C#CC2(C)CC2)C1 N1(C(c2c(OC)cccc2O)=O)CCC(C2CCN(C(=O)C3=C(Cl)CCC3)C2)C1 C(CCCCC(=O)N1CCSCC(C)C1)N(C(=O)C(c1cnn(C)c1)O)C CC1CSCCN(C(C2CCC2CNC(=O)C(c2ccn(C)n2)C)=O)C1 CC1(C)C(C(N2CCCC2CNC(c2ccc3ccnn3c2)=O)=O)CCS1(=O)=O C(CCCC(CO)NC(C1(C2CCCO2)CC1)=O)NC(=O)C1=CCSC1 c1(OCCC(N2CC(CNC(c3n(CC)ncc3)=O)C2)=O)c(C)cccc1C S(=O)(=O)(c1ccc(N2CCC(COC)C2)c(Br)c1)NCC(C)OCC=C C(=O)(C(F)(F)CO)NCC1(CNC(C2(c3ccc(F)cc3)CC(C)C2)=O)CCC1 C1(C(C)C)CN(C(c2nccc(C(F)F)n2)=O)CCN1C(C1(C)COC1)=O Cc1c(F)ccc(C(=O)NC2(CCO)CN(C(C3(Cl)CC3(F)F)=O)C2)c1Cl c1(C(=O)NC2CCN(C(CCCC(C)=O)=O)CC2CO)cnc2sc(C)cn12 c1(OC)ccc(CNC(C2(C)CCN2Cc2cccc(C(C)C)c2)=O)cc1 C1(C(N2CC(CCNC(CNS(N(C)C)(=O)=O)=O)C2)=O)CC2(C1)CC1(CCC1)C2 c1(CNC(COCC#C)=O)ccc2c(c1)CN(C(=O)C(C)(C(C)C)OC)C2 C1(C(=O)N(CCCCCNC(=O)C(=O)NC2CC2)C)(CC)CC(C)(C)C1 c1(CN(C(C(CN(C)C)NC(C(C)OCOC)=O)=O)C)cccc2ccccc12 C1(C(=O)NCC2C(C(=O)NCC[Si](C)(C)C)OCC2)CC(F)C(=O)N1 N1(C(C(C)NC(CC)=O)=O)CCC(C(=O)Nc2ccc(C)c(CC)c2)=C(F)C1 c1(C(=O)NCCOC2CCN(C(C3C(C)=C3)=O)CC2)cc(F)cc(C)c1N c1(N2CCCCC(NC(CCC(=O)NC)=O)C2)ccc2c(n1)CCC2=O C1(CN(C(=O)C=CSc2ccccc2)CC)CCCN1C(=O)CC(C)c1ccco1 n1(CC(=O)NC2CCCN(C(C3CCC(CC)O3)=O)C2C)cnc2ccccc12 N(C(=NCC1CN(C2CC2)C1)NC1CCOc2ccccc21)C1CCS(=O)(=O)C1 C1(C(=O)NCc2c(CC)nccn2)CC(C)(C)CN1C(=O)C(C)NC=O c1(CNC(C(C2CCCC2)OCC)=O)ccc(CN(C(=O)CC2(C)CC2)C)cc1 CCC(CCC(=O)NOCC1CCCO1)NC(C1CC(C)(O)C1)=O c1(C(C2CC(SC)C2)NC2CC2)nnnn1CCO.c1(C2(C=O)CC2)ccsc1 N1(C(c2cc(C(C)C)on2)C(=O)NCCC2CC2)CCC(F)(F)CC1 c1(CNC(C2C=CC(NC(C3C(CC)CCO3)=O)C2)=O)scc(C)c1C N1(C(CC(C)C(F)F)=O)CCCC12CCN(C(c1ccc(N=[N+]=[N-])cc1)=O)C2 CN1CCN(C(=O)CCCC2CCCC2)C(C(=O)NC2(C3CCCO3)CC2)C1 Cc1ccc(C(N2CCC(C)(CNC(c3ccoc3CC(N)=O)=O)C2)=O)c(O)c1 c1(N2CC(C(N)=O)(CNC(c3cc(C)cc(C(F)F)c3)=O)C2)ncn(C)c(=O)c1Br N1(C(Cn2c(C)csc2=O)=O)CCCC2C1CCCCN2C(=O)C(C)S(C)(=O)=O N1(CCC(=O)NC(c2ccccc2)C)CCCC1P(C)(C)=O c1(NC(COC(C2CC(CSC)C2)=O)=O)nc2cccnc2s1 C(=O)(CCCCCC(C)O)NC1(CNC(c2ccc(C)c(Cl)c2)=O)CCC1 Cc1ccncc1C=CC(=O)NC1CN(C(c2nnc(O)nc2O)=O)CC1C C1(NC(C2(CC)CC2(F)F)=O)CCCCN(C(c2cccc(C#N)c2)=O)C1 CC1(C)OCC2CC12C(=O)NCC#CCNC(c1ccc(C(N)=O)c(Cl)c1)=O C1(c2ccc(OC)cc2)C(C(N2CCOC(c3cc[nH]n3)C2)=O)CCC(=O)N1C c1(C(N2CCc3c[nH]nc3C2)C(=O)NCC2CC2)ccc(Cl)c(Br)c1 C(CN=C(NCc1cnc(C)cn1)N1CCN2C(=O)OCC2C1)OCC C(CCOC)(C(=O)N1CC2C(C(N)=O)C2C1)NC(CCOCC#C)=O C(=O)(CC(F)(F)C(F)F)N(C1CCN(C(C2(C)CCOC2)=O)CC1)CCOC C1(NC(c2c(C(C)C)nns2)=O)CCCN(C(C2C(C)C2C)=O)CC1 C12(OC)CCCC(C(=O)NCCCn3cc(C4C5CCCCCC45)nn3)(CC1)C2 C1(CC(=O)O)CC(F)(F)CN1C(=O)CC12CCC1CCN2 C(=O)(C(C)(C)CCC#N)NCC1C(NC(c2n(C)c(S)nc2)=O)CCC1 Cc1c(C(N2CCC(NC(C3CCC34CCC4)=O)C2C)=O)ccc2cncn12 CCC(F)(F)CC(=O)NC(C(=O)N1CCCCC1)C(C)C c1(C(N2CCC(NC(c3cnc(C)nc3C)=O)C2)=O)ccc(Br)cc1C#N C12(C(N3CC4C(NC(c5n[nH]cc5Br)=O)(C4)C3)=O)CCC(C1)S(=O)(=O)CC2 C1(NC(c2cn(CC(CC)O)nn2)=O)CN(C(c2ccc(Br)o2)=O)CC(C)(C)C1 CC1CN(Cc2cccc(S(N)(=O)=O)c2)Cc2c(Br)ccc(F)c21 c1(C(=O)NCC(CNC(C=C(C)Cl)=O)C)cccc(C2(C)CC2)c1 CC1(C)CC(C(=O)NC(C2CCCC2)CNC(c2c[nH]nc2Br)=O)C1 C1(OCC)COCCC1NC(=O)C(=O)NCC(c1ccccc1)N1CCCC1 N1(C(c2ccn3ncc(CC)c3n2)=O)CCC2(CCC2CNC(=O)C(N)=O)CC1 c1(CC(=O)NC2C(C)CN(Cc3ccccc3)C2)ccc2c(c1)CCC2 c1(SC)cccc(C(=O)NC(CNC(c2cn(C)nc2C2CCC2)=O)CO)c1 c1(C(N2CCC(NC(CCC3C(C)(C)C3)=O)C2)=O)cc(Cl)ccc1O c1(NC(C(CSC)(C)NC(C2CC23CCCCC3)=O)=O)cc(C)c(C)cc1C c1(N(C2CCCN(C(CC)=O)C2)C(C2CCC2)=O)nc(=N)[nH]c(C)c1C c1(CNC(N(CC(COCC)C)C)=O)cc(OC(C)(C)C)cc(Cl)c1F Cc1cnc(F)c(-c2cn(CC3CN(C(C4CCCC(C5CC5)O4)=O)C3)nn2)c1 C#CC1CN(C(=O)C(C)OC)CCN1C(c1ccc(C(C)=O)cn1)=O C1(NC(=O)C2=CCOC2)CC(F)CN(C(=O)C(=Cc2cccc(F)c2)F)C1 C(CCC(C)CC(=O)NC12CC(C(=O)Nc3ncc(CCO)s3)(C1)C2)=C(C)C N1(C(C(C)(C)SC)=O)CC(CNC(c2ccc(C3CC3)cn2)=O)C(n2ccnc2)C1 Cc1ncncc1NC(c1ccc(-c2cnn(C(C)C)c2)cn1)=O S(=O)(=O)(c1cc2ccccc2s1)NC1C(C#N)CCCC1 CCC(C)(C)CC(=O)N1CCN(C(=O)Cc2cc(OC)no2)CC1c1cn[nH]c1 Fc1cccc(-n2nccc2CNCCc2ccc(Br)s2)c1 C#CC1(NC(C2CC(=O)N(C3CCN(C)CC3)C2)=O)CCC(C)(C)C1 c1(CN(C)C(C2(CCN)CC2)=O)cccc2[nH]ccc12.C1(CC(=O)CN)COCCO1 C1(Cc2n(C)ccn2)CCCN(CC2C=CCOC2)C1 Cc1[nH]c2cc(Br)ccc2c1C(N1CC(CNC(=O)C2=CCOC2)C1)=O C1(CC(=O)NC2CC(C(C)NC(c3ccnnc3)=O)C2)CCCC1O C1(CC(=O)NC)CN(C(=O)Cc2occc2C)CCN1C(C12CC(C1)C2)=O c1(C(=O)NC2CCC(CNC(C3N(C)C(=O)CC3)=O)C2)[nH]cc2c1CCCC2 CC(C(C)(C)C(=O)NCC1CCCC(=O)N1)NC(c1cccc(O)n1)=O c1(NCCC(C=C)C)[nH]c(=NC(C)CF)nc2c1ncn2CC C1(COC)CCCN(CC(N2CCCC2)=O)C1.C12(CC1)CC(=O)N2 N1(C(c2c(C)nn(C)c2)=O)CCN(C(=O)C(C)CN2CCOCC2)CC1CCO CC1CC(O)CN1C(=O)CCC1CCN(C(C2CC23CCCC3)=O)CC1 C1(NC(c2c(OC)ccc(Cl)c2)=O)C(C)CCN(C(=O)CC2COCCO2)C1C CCCS(=O)(=O)C(C)C(=O)N1CCCC1C1(NC(c2nc(O)sc2C)=O)CC1 CC1CCC(C(N2CC(C)(C)CC2CNC(c2cc(O)n(C)n2)=O)=O)CC1C C1(CCNC(c2cc(CC(C)C)sc2)=O)CCCCN1C(=O)C(C)C1CCCC1 C1(C)(NC(C(C)SCc2ccc(N)cc2)=O)CCCN(C(C2(C(N)=O)CC2)=O)C1 Cc1cc(COC(C)(C)C)oc1C(=O)NC(CNC(c1[nH]nnc1C)=O)C n1(C2CCCN(C(=O)Nc3cc(C)nn3C3CCOCC3)C2)nc(O)ccc1=O N1(OCC)CCCC(C(=O)NC2CCC(NCCSCCO)CC2)C1 C1(CN(C(C2CC(C(=O)OC)C2)=O)C)CN(C(c2cccc(Cl)c2)=O)CCO1 N1(C(c2c(C)nn(C)c2)=O)CC2CCN(C(C3(S(N)(=O)=O)CC3)=O)CCC2C1 C1(C(=O)NC(CCOC(C)=O)C(=O)O)CC2(C1)CC21CC1 CC(C)CCCC(C)C(=O)NCC1CC(C(N2CCn3nccc32)=O)CO1 c1(NC(C(=O)NCCSCCC=C)=O)cc(Br)cnc1Cl C(=O)(C(C(C)CC)N(C)C(c1cncn(C)c1=O)=O)NCC(C)OCC#C CC1(CNC(C2C3CC2N(C(=O)CC24CCCC2C4)C3)=O)CCC(=O)N1 CCC(CN=c1[nH]c2c(c(=NCc3ccnc(O)c3)[nH]1)CCC2)N(C)C C1(C(=O)NCc2cc(OC)ns2)(CNC(CC(=O)NCC)=O)CC12CCC2 CC1=NOC(CC(=O)NCC2CN(C(=O)CCc3ccncc3)C2)C1 CC(C(=O)N1CCN(CCN(C)C(C2(N3CCCC3)CC2)=O)CC1)C(F)(F)F CCCC(C(=O)NC1CCN(CC2CN(C3CCC3)C(=O)O2)CC1)OCC N1(C(C=C(C)C)=O)CC(CNC(=O)Cc2cc(O)nnc2O)CC12CCC2 c1(CC(N2CCN(C(C(CC#C)O)=O)C(CCCC)C2)=O)ccc2nn[nH]c2c1 C(=O)(CCCc1nc(C2CC2)no1)N(CC(C)N(C(=O)Cc1cscn1)C)C N1(CC)CC(C2=NOC(C)C2)C1.C1(CC2CCC2)C(=O)N1.N12CCCC1C2=O C1(C(=O)NCC(C)C)CC(NC(c2ccc(O)cn2)=O)C1(C)C CN1CCOC(C(=O)NCCCC2CCN(C(=O)C(C)(C)c3cncs3)CC2)C1 c1(CCC)nc(C)c(C(=O)N(C(C)CN(C(=O)CN2CC=CC2)C)C)o1 c1(C(N(CC(C)NC(=O)CCN(C)Cc2ccccn2)C)=O)csc(CSC)n1 C1(NCCC(=O)NC(N)=O)CC2CC1N(C(=O)CCNC(C1CCCCC1)=O)C2 C=CC1(C(=O)N(CCCNC(=O)CC(C)N(C)C)C(C)C)CCC1 CCC(C)CC(=O)NC1C2CC1N(C(c1coc(Br)c1)=O)C2 N1(C(C(C)=NOCC#N)=O)CC=C(CC(=O)NC2(CO)CC(F)C2)CC1 c1(C(N2CCC(O)(CCNC(C3(F)CCCOC3)=O)C2)=O)cc(F)cnc1O C1(C(N2CCCC(NC(C(C)CN3CCOCC3)=O)C2)=O)CN2CCC1CC2 c1(C(C(=O)NCC(F)F)N(C2C3COCC23)C)cc2ccc(Cl)cc2o1 C1(C(=O)NCCC#C)CCN1C(C1CC1(C)C)=O C1(CN(Cc2cccc(C(C)(C)C(N)=O)c2)Cc2ccccc2)CC(=O)NC1(C)C Cc1cc(C(N2CC(CO)C3(CC3)C2)C(=O)NCC2CCOCC2)cc(C)n1 CC1(C)CN(C(=O)Cn2ccc3ccccc23)CCC1NC(=O)C(=O)C(F)(F)F C1(C(=O)NC)CCCN(C(C2(F)CCN(C(C3CCCSC3)=O)C2)=O)C1 N1(C(C(C)n2cccc2)=O)CCC(NC(=O)C=CI)C(O)C1 N1(c2ncnc(C)c2F)CC2CCCC(NC(=O)C(C)CC(F)(F)F)C2C1 CCC(CC)(CC(=O)OC)C(=O)NCC=CCNC(=O)CCC1CCOC1 c1(Cc2c(C3CCN(C(=O)NCC(c4ccccc4)C)C3)n[nH]c2)ncccc1F N1(C(C(C)OC)=O)CCC(C(C)C(=O)N(CC(C)O)C(C)C)C1 C=C1CON(C(=O)CC2CC(C)N(C(c3cc(C4CC4)on3)=O)C2)C1 N1(C(c2c(OCC)ccs2)=O)CCC2(CCCN(C(=O)C3=COCC3)C2)C1 CC1CN(C(=O)C(c2cc(Cl)ccc2Cl)=O)CC(=O)N1 c1(C(N2CC(C)(NC(C3CC(N4CCCC4)C3)=O)C2)=O)cccc(C2COC2)c1 O=C1CC2(CO1)CN(C(C1CN(C(=O)C(c3ccccc3)F)CCO1)=O)C2 c1(C(=O)OCC2CC(CC)C2)cc2cccc(Br)c2s1 CC(C)(CCNC(C1CCCS1)=O)NC(=O)COCCc1cccs1 Cc1cc(-c2cc(-c3nccn3CC3COC3OCC)ccn2)cc2cnn(C)c12 C1(CNC(c2nc(C)oc2)=O)CCC(C)(C)CN1C(=O)Cc1cccnc1O c1(N2C(CNC(c3c(OC)ccc(F)c3)=O)CCC2)ccc2c(n1)CCCC2=O C(C)(CC1=CCCCC1)NC(CC1(OC)CN(C(C2CCCC2)=O)C1)=O N1(C(C=C(C)c2cccs2)=O)CCC(NC(=O)Cc2ccccc2C)C(CO)C1 CCCC(C)CC(=O)N1C(CC(N2CCC2COC)=O)C2CCCC12 C(=O)(CCCCCC(C)(C)C)NCC(C)N(C(c1cc(C)ncc1C)=O)CC C(=O)(C(F)C1=CCCCC1)N1C2CC(NC(C34CCCC3CCC4)=O)CC1CC2 C(=O)(C(C)(C)CS(N)(=O)=O)NCC1C(C)CCN1C(c1ncc(C(F)(F)F)s1)=O CC1=CC(C)CN(CCNCc2ccc(N3CCOCC3)cc2)C1 C1(NC(CC2CC(NC(c3cc(COC)no3)=O)C2)=O)C(=O)OC2CCCC12 c1(OC)cc(C(N2CCCC2CN(C(=O)C(C)(C)C(N)=O)C)=O)c(Cl)cc1Cl C1(C(=O)NC(C2CCN(C(CCSC)=O)C2)C)C(=O)NN=C1C CCC(C(=O)N(C(CNC(c1ccc2snnc2c1)=O)C1CC1)C)C(C)(F)F N(C1CCCc2occc21)C(CC1CCN(C(C(=O)N(C)C)=O)CC1)=O C(CCCCNC(=O)CCOCCCOC1CCCC1)NC(CN(C)C(N)=O)=O N1(C(c2ccc(OC)nc2)=O)C2CCC1CN(C(=O)C(C)CC(C)C)C2 Cc1cccnc1C=CC(=O)NCC(C1CCCN1C(=O)CC(C)C(C)C)(C)C C(C)(C)(CC(c1nnnn1C1CC1)NCCc1ccccc1C1CC1)OC n1(CC(=O)NC(C)(C)CCNC(C2(C(F)F)CCCO2)=O)cc(S(C)(=O)=O)cn1 c1(C(=O)NCC(c2ccc(F)cc2)NC(C(C)(C)C2CC2)=O)cc2scnc2[nH]1 Cc1cccc2c1CCN(N1CCCC(c3nc(C(F)(F)F)cs3)C1)C2 C(=O)(CC(C(C)OC)NC(=O)CC1CCCCO1)N1CCCC(CC=C)C1 C1(C(C)C)CCCCC1CNC(=O)N(CCN(C)C)Cc1ccccc1 C(C(CCC(F)(F)F)N=c1cc(C)[nH]c(=NCc2nc(C(C)(C)C)co2)[nH]1)OC C1(CNC(=O)Nc2ccnc(C)n2)CCC2(C1)OCCO2 c1(C)ccc(C(F)(F)F)cc1F.N(C1=NCCNN1)C(CC)CC#N.SC CC1CCC=C1C(=O)N1CCN(C(c2cc3occc3[nH]2)=O)C2CC12 CC1CN(C(=O)CN2CCC(C(N)=O)CC2)CC1NC(c1cn(C2CC2)nn1)=O N1(C(C(C)(C)OC(C)C)=O)CCC(NC(=O)C#CC2(C)CCCO2)CC(C)(C)C1 Cn1ncc(C(N2CC(O)(CNC(c3cnoc3-c3ccoc3)=O)C2)=O)c1C#N Nc1ncc(C(F)(F)F)cc1C(=O)NCCCNC(c1cc(Br)n[nH]1)=O Cc1c(C(=O)NC(CNC(c2c[nH]c(Br)c2)=O)C2CCC2)cccc1CO C1(CNC(C(C)O)=O)CN(C(=O)C(C)(C)Oc2ccccc2)CCC12CCC2 C1(N(C)C(C2CC(=O)N(C3CCCC3)C2)=O)C2CN(C(=O)C(C)=O)CC12 C12(C(=O)NCCN(C(C(=O)NC(C)C)=O)C3CC3)COC(CO)(C1)C2 C1(CNC(C(COC)C)=O)(COC)CCCN1C(c1cncc(C(N)=O)n1)=O C(=O)(C(CCCC(=O)OC)N1CCCC1C(C)(C)O)N(CCCC(=O)NCC)C C1(C(=O)N(C(C)CC2CC2)C)(CC)CCCN(C(C2CCCOCC2)=O)C1 C12(NC(c3ccc(OC)cc3C)=O)CCCC1N(C(=O)C(F)=CCCF)CCC2 C#CC1(O)CC(C(N2CC(CNC(c3nccs3)=O)C(O)C2)=O)C1 c1(OCC)cccc2[nH]cc(CN=c3[nH]c(C(=O)Nc4ccc(Cl)cc4)cs3)c12 N1(C(=O)C2=COCCOC2)CC2CC(N=c3[nH]nc(CO)s3)CC1C2 Cc1cnc(N2CCC(CCO)C2)c(S(=O)(=O)NC(C)CC(C)(C)C)c1 c1(C(=O)NC2C(NC(C(CCN(C)C)O)=O)COC2)cc(O)c(O)c(O)c1 Cc1ccc(Cl)c(C(N2CC(NC(=O)CC3CCCSC3)C3(CC3)C2)=O)c1 N1(C(c2c(Cl)cc(C)s2)=O)CCC(C)C(CNC(c2ncccc2N(C)C)=O)C1 N1(C(c2occc2C2CC2)=O)CCC2(CC1)CN(C(C1(C3CC3)CCC1)=O)C2 C#CCCN=C(NCCC1COC1)NC1CCC1(C)C N1(c2nc(C)c(Br)cn2)CCc2nn(C)c(C(=O)Nc3cnc(Cl)cc3I)c2C1 c1(CC(=O)NCCCCNC(C(c2ccc(F)nc2)C)=O)ccc(Cl)nc1 c1(C(=O)NCCC(C(C)C)NC(c2ccnc(OC)n2)=O)ncc(C)cc1F C#CCCCC(=O)NOC(CC(C)C)C(=O)NC(C)CCC(F)(F)F C#Cc1ccc(CNC(=O)CN2CCN(C(=O)Cc3ccc(F)c(C)c3)CC2)cc1 C1(O)(CC(=O)NCC(CNC(C2CC2CC(C)C)=O)OC)CCCCCC1 Cc1cc(C(N2CC(O)C(O)C2CNC(C2CCS(=O)(=O)N2)=O)=O)ccc1O C1(NC(C(C)(C)CCl)=O)CC2CCC(C1)N2C(c1ccc(I)cc1F)=O C(=O)(C(C)C(O)C(C)C)NC1(CNC(C=Cc2cccc(C)c2)=O)CC1 CC1CCCN1CC(=O)NCCc1ocnc1CNC(c1cnsn1)=O c1(C(N2CCC3C(NC(C(CCSC)OC)=O)C3C2)=O)cc2ccccc2o1 N1(C(C2C(c3ccn(C)c3)C2)=O)CCN(C2CCN(C(C3CC3(C)Br)=O)C2)CC1 C12(C(N3C4C(CNC(C)=O)CC(CC4)C3)=O)CCCCCC1OCC2 CCC(CC)CCC(=O)NCCCNC(=O)C=C1CN2CCC1CC2 c1(CCC)cc(C(=O)NCc2cc(-c3ccco3)nn2C(C)(C)C)ccc1F CC1CCN(C(=O)CCc2ccc(Cl)cc2)C(C(C)NC(=O)C(=O)NC2CC2)C1 Cc1ccncc1CCC(=O)N(CCC(C(C)C)NC(=O)C(F)CC1CC1)C C1(C(N2C(C(=O)NC(CC)C3CCC3)CC2)=O)C2CC(=O)CC12 C12(C(=O)OC)COCC1CN(CC1CCCN1C1CCCCC1)C2 CC1CN(C(c2ccc(Cl)nc2N)=O)CC(C)N(C(=O)CCN2CCCC2)C1 Cc1cc(-c2cn(C3CCC(C(=O)NCCN4CC(C)(O)C4)C3)nn2)ccn1 C1(C(N2C(CNC(CNS(N)(=O)=O)=O)CCCCC2)=O)CCc2cncn2C1 S(=O)(=O)(c1cnc(C(C)(C)C)s1)N1C(C)CN(CC(=O)N(CC(C)(C)C)C)CC1 C1(C(=O)NC2(C(N(CC)Cc3cnccn3)=O)CC(O)C2)CCC2(CCC2)O1 CN1CCN(C(=O)COC2CCOCC2)C(CNC(=O)CC2CC(N(C)C)C2)C1 CC(C)(CNC(=O)Cc1ncccc1F)CC(=O)NC1CCCC(O)C1 C(CCCCCOC)(C(=O)NC1COC1)N(CCCCCCCC)C C1(C)(Cn2cc(CN(C)C(=O)C3CC3)nn2)CCN(C(c2cnc(N)cn2)=O)C1 Cc1cc(C(=O)NCC2COCC2NC(c2cccc(N(C)C)n2)=O)nc(C)c1 N1(c2c(S(=O)(=O)N3C(C)COCC3)cncc2)CCCC2(CCNC2=O)C1 C(=O)(C(C)(C)CO)NC1CCC(NC(c2c(CC)non2)=O)C1 c1(C(=O)NC2CCC(CCC(=O)NC3(CCCC)CCC3)C2)ncc(C)cc1F C1(NC(=O)COc2ccccc2)CC2CCC1N(C(C1(CO)CCCCC1)=O)C2 N1(C(=O)Cc2nncs2)CCN(N2CCCC(c3ccon3)C2)CC1 CCCCC(CNC(C1(C)CCC1)=O)NC(=O)CCCc1ncc(C)o1 N1(C(C(C)NCc2nc(C)sc2)=O)CCCC(C)(C(=O)NC(C)(C)C)C1 N1(C(C2N(CCC)C(=O)CC2)=O)CC2(CCC2)CCC1CNC(=O)C(C)SC N1(C(c2nc(CCC)oc2)=O)CCC2(CC1)CCN(C(C1CCC1COC)=O)C2 C=CC(C)(C)CC(=O)N(CCNC(=O)CNC(c1cccc(Br)c1)=O)CC CC(C)CS(=O)(=O)CCC(=O)NCC(C)(F)CNC(=O)CC1CC(=O)NC(=O)C1 c1(C(=O)NCC2(C)CCN(c3cnc(F)cn3)CC2)ccc2n[nH]cc2c1Cl C1(CNC(C2CN(C(C)=O)C2)=O)CCC(C)CN1C(=O)Cc1c(C)cnn1C C12(CC(=O)NC3CCN(C(CC=C(C)C)=O)C3C3CC3)CCC(CC1)OC2 C1(NC(NC(COC)C)=NCCCc2cc(C)no2)CCOC2(CCCC2)C1 c1(CSC)cc(C(=O)NC2CN(C(c3csc(O)n3)=O)CC2C)ccc1F N1(C(CNC(=O)OC)=O)CC2(CCN2C(=O)C(C)C2CCCO2)C1.c1ccccc1 c1(C(=O)NC2CCCN(C(CCCCCC)=O)CC2)nc(O)nc(O)c1N C1(=O)CC(C2CC2)CN1C12CC(F)(C1)C2.c1(OCC)ccccc1 C1(NC(CC(CC)(F)F)=O)CC2CN(C(=O)CC(=O)OCCC(C)C)CC2C1 CC(C)N=c1[nH]c(N2CCNC(=O)C23CCC3)nc2c1COC2 CC1CC(C(=O)N2CCC(NC(C3CN4CCN3CC4)=O)C2)c2ccccc2N1 C1(c2nnnn2C2CC2)(NC(CCNCc2ncc(CC)o2)=O)COC(C)C1 CC1CN(C(=O)CC2CCOC2=O)CC1(C)CNC(=O)Cc1cccc(F)c1Cl C1(NC(C2C(OC)CC2)=O)CC2CCC1CC2NC(=O)Cc1ccc(F)cc1C c1(C(N2CC(OC)(CNC(=O)CCP(C)(C)=O)C2)=O)nc(=N)[nH]c2ccccc12 c1(CC)c(C)[nH]c(C(=O)N(C)Cc2ccnn2C)c1C C1(CC)CN(C(c2ccc(Cl)cc2O)=O)CCN1Cc1sc(Cl)nc1Cl c1(C(N(CCCNC(CCNC(=O)OCC)=O)C)=O)c(F)ccc(F)c1C C1(N(C(COCC#C)=O)CC)CCN(C(=O)C(F)C(=O)OCC)CC1 C1(=O)CCN=C(N2CCC(n3cc(C)cn3)C2)NCCC2CCN1C2.CN C1(C(=O)NC2(CO)CCN(C(C(C)(C)C3CC3)=O)C2)CN2CCCC2CO1 CCCCCC(CC)C(=O)N(CC(C)NC(c1cccc(C(N)=O)c1N)=O)CC C1(CC)CN(C(c2cc(C(F)(F)F)cnc2O)=O)CCN1C(c1c[nH]nc1F)=O C#CC1CC2(CC2)CN1C(=O)C(C1CCOC1)NC(=O)COCC(C)C C1(CCN(C(=O)Cc2ccco2)C)CCN(C(C2CCN(C3CC3)CC2)=O)CC1 N1(C(Cc2ncc(C)s2)=O)CCC(O)C(NC(c2nn(C)cc2C(F)(F)F)=O)C1 C(=O)(CC(C)CN(C)C)N1CC(CNC(C(c2ccc(Cl)cc2)OC)=O)C1 N1(C(Cc2ccc(C)cc2)=O)Cc2n[nH]cc2C1C(=O)N1CC(C)C(F)(F)C1 N1(C(c2c(C)coc2C)=O)CC2CCC2(CCNC(c2csc(Cl)c2)=O)C1 C1(CC(=O)OCCCc2cnc[nH]2)CCC(C(=O)NCCCN2CCCC2)CC1 CC(O)(Cn1ccccc1=O)C(=O)NCC1CC(NC(=O)CC2(F)CC2)C(O)C1 C1(COC)(CNC(C2CC(OC)C2)=O)CCN(C(C2CC2C)=O)C1 c1(C(N2CC(=C(C(N3C(CC)CCC3)=O)F)C2)=O)cccc(CO)n1 C(=O)(CC(C)(C)COC(C(CC)CC)=O)OCC1CCCC(C)(C)O1 C1(NC(c2cc(C)c(O)nc2)=O)C(CNC(=O)CCC2CC2)CCC12CCC2 c1(C(N2CC(CN(C(c3c(C)cccc3)=O)C)C2)=O)c[nH]c2c(O)cccc12 C1(C(=O)NCC2(OC)CCC2)CCN(C(c2cnc(C3CC3)o2)=O)C1 c1(CC)c(C(=O)NCC2CCCN(C(=O)CNS(=O)(=O)CC)C2)csc1C c1(C(=O)N=c2cc[nH]c(F)c2)c[nH]c2cc(Cl)c(Cl)cc12 C1(CC)CN(C(c2cnn3cc[nH]c23)=O)CCN1C(c1ncccc1F)=O N1(C(CC=C=C)=O)CCN(C(c2ccc(C3CCCO3)[nH]2)=O)C(CS(C)(=O)=O)C1 CCC(CC(=O)N(C1(CC(=O)NC(C2CSC2)C)CC1)C)C1CCC1 c1(C(N2CCC(N(C(=O)CC3CCOC3(C)C)C)C2)=O)ccc2cnnn2c1 N1(C(CC(CC2CC2)NC(C(C)C(F)F)=O)=O)CCCC2(C1)N=N2 N1(C(CCCNC(C)=O)=O)CC(C)C(C)(C(N2CCC(O)C(C)C2)=O)C1 C12OCCN(C(c3ccccc3OC)=O)CC1N(C)N2.C(=O)(C(C)C#N)OCC c1(NC)cc(C(=O)N(C2CCN(C(c3cnccc3OC)=O)C2)CC)cc(Cl)n1 n1(CC(N2CC3C(CNC(C(c4cccnc4)C)=O)C3C2)=O)cc([N+](=O)[O-])cn1 c1(C(N2C(C)C3CC2C3NC(=O)CN=S(C)(C)=O)=O)ccc([N+](=O)[O-])c(O)c1 C(CCC(=O)NO)NC(C1N(C(C(=O)NC)=O)C(C)C1)=O c1(OC)ccc(C(N2CCCN(C(C3CCCCS3)=O)CC2C)=O)c(F)c1N C1(NC(C2(OCC)CC2)=O)CCC2C(C1)C2(F)F.c12cccc(c1)Cn1cc-2nn1 CCC(CC(=O)NC(C)C(=O)NC1CN(CC)CC1C)c1ccccc1 C#CCCCCC(=O)NCC(CC(F)(F)F)NC(c1ccccc1OC(F)F)=O CC(F)(F)CCC(=O)OCC1CCC(=O)N1C(=O)C(C1CCCCC1)O N1(C(c2c(C)ccc(N)c2)=O)CC2(C1)CN(C(=O)CCC1CCCCC1)CCO2 C12(CNC(Cc3n(C)ncc3Cl)=O)CCCCC1CN(C(c1ccon1)=O)C2 C=C(CN)CCOCCCC(=O)Cn1cnnn1.C(=O)CC(C)C C(=O)(CCCCCc1cccs1)NCC(CNC(c1c(OC)cccn1)=O)(C)O CONC(=O)C(=O)N1CCOC(C(=O)N(C)Cc2nnc(C)o2)C1 C1(C(=O)NC(CC)Cn2cncn2)CCCCCN1C(=O)C(n1nccc1C)C CC1(C#CC(=O)NC2COCC2C(N2CCC3(CC2)CC3CO)=O)CCCO1 N1(C(c2cc(C)n(C)c2C)=O)CCC2C1CCN2C(c1n[nH]cc1[N+](=O)[O-])=O c1(C(=O)NC2CC(NC(C3N(C(C)=O)CC(O)C3)=O)C2)ccc2cnccc2c1 c1(CC)ccc(OC)c(C(=O)NC2CN(C(C3(N(C)C)CCCSC3)=O)C2)c1 Cc1cc(C=CC(N2CC3(CNC(C4(F)CCOC4)=O)CC2CO3)=O)c[nH]c1=N c1(C(=O)NCC2N(C)CCN(C(CSSC)=O)C2)cc(C)nc2ncnn12 C(=O)(C1CC(=O)N(C)c2ccccc21)N(CC(C)NC(CSCCCC)=O)C c1(C(N(C2CCN(C(C(n3ccc(C)n3)C)=O)C2)C)=O)ccc2c(c1)OCCC2 C1(OC)CN(C(=O)OC(C)(C)C)CC1F.C12(CO)CN(C1)C(=O)C(C)CNC2=O c1(C(=O)NCC(CC)(C)NC(c2cncc(O)c2)=O)cn2c(n1)CCC(C)C2 C#Cc1cnc(C(=O)NC2CN(C(c3cn4ccsc4n3)=O)CC2SC)cc1C C(=O)(C1=NNC(=O)C1)N1CC(O)(C(CNC(C2CN(C)C2)=O)(C)C)C1 c1(C2(C(=O)NCC(CO)NC(c3cncc(OC)c3)=O)CC2)cc(C)ccc1F N(C1CCc2ccc(F)cc21)C(c1nnnn1C(C)C(=O)NCCF)(COC)C N1(C(C2(CC=C)CCCN2C(=O)CC2CCC(C)(C)C2)=O)CCOC(C)CC1 Cc1cc(C(N2CCNC(C(N3CCCC(C)(O)C3)=O)C2)=O)ccc1F Cc1ncnc(O)c1C(=O)NCCC1CSCCN1C(C12CCC(C)(C1)OC2)=O c1(C(N2C(C(N3CC(C)(C(N)=O)C3)=O)CC2C)=O)ccc(F)cn1 c1(CCC(=O)NC(CNC(c2cn(CC3CC3)nn2)=O)C2CC2)ccccc1F N1(C(CCc2cc(C)no2)=O)CC2(CC2)CC1CC(=O)NC1CCC2CC1CO2 C1(NC(c2n(CC)nc(C)c2)=O)CCN(C(=O)Cn2ccnc2)CC1F C(=O)(CC1OCc2ncccc21)N(C)CC1N(C(CCC(=O)OC)=O)CCC1 CCCCCC(C)CC(=O)NCCCOCCN(C)C(C1CCC2(CC2)C1)=O N1(CC(=O)N(CCNC(=O)CCCNC(=O)C2CC2)CC)C(=O)C(C)C(C)C1=O C(=O)(C(C)(C)C)NCC(C)(C)NC(CN(c1nccn1C)C)=O C(=O)(CCCCCCN=[N+]=[N-])NC1C(NC(CC(COC)(C)O)=O)C1 C(CC(O)CC(=O)Nc1cc[nH]c1C(N)=O)NCC1C(NC(=O)OC(C)(C)C)C1 C(S(=O)CC(=O)OC)C1CCC(OCC(=O)OC)CC1 N1(C(C2CC(CNC(C34C(C)OC(CC3)C4)=O)C2)=O)CCC2CC1C(=O)N2C N1(CC(=O)N(C(C)C)C)CCN(c2cc(C3CCCNC3)ncn2)CC1 Cc1nc2ncnn2c(C)c1C(=O)NC(CNC(=O)C(C)(C)CO)CC(F)(F)F N1(C(C(CC=CC)NC(c2n[nH]c(C)c2Cl)=O)=O)CC2(CCC2)CC1C CCC(C)CC(C(=O)NCCC(=O)NC)NC(c1ccoc1)=O C1(COCC(=O)Nc2ccc(F)cc2)(CNC(C2(C)CCCO2)=O)CCOCC1 c1(C(=O)NC2(CNC(C(C(C)SC)O)=O)CCC2)nc2ccccn2c1F C#Cc1ccc(C(N2CC(NC(=O)C(c3cc(F)ccc3C)=O)C(C)C2)=O)nc1 N1(C(C2(CCC=C)CC2)=O)C2CC=C(C(=O)NCC(C)C(C)(C)C)C1CC2 C1(C)(C(N2CC(O)(C(C(=O)NC(C(C)C)C3CC3)F)C2)=O)CNC(=O)C1 C1(C(=O)NCC2C3CN(C(C=CCCC)=O)C2C3)CC2(CCCC2)CO1 C(C(=O)N1CC2(C=CCO2)C1)(C(C)CC)N(C(c1c(CC)con1)=O)C C1(C(=O)N(c2ccccc2)CC2(NC(CC3(C#N)CC3)=O)CC2)CC2(C1)CC1(CC1)C2 C1(CNC(c2ccon2)=O)CC(C(F)(F)F)CCN1C(=O)CN1C(=O)CNC1=O N1(C(C(C)=CC2CC2)=O)CCOC2(CCN(C(c3coc(C#N)c3)=O)C2)C1 C(CCF)(C(=O)NOC1CCOC1)NC(C(n1c(C)ccn1)C)=O N1(C(c2n(C)nc(CC)c2Br)=O)CCC2(CC1)CC(=O)N2.N12CCC(O)C1C2=O CCCC(CC)C(=O)NCCC1(O)CN(C(C2COCCN2C=O)=O)C1 N1(C(C(C)(C)NC(=O)NCC)=O)CC(OC)CC(NC(=O)C(C)N2CCC2)C1 N1(C(C(C)N(CC(CC)O)C(=O)CC2CC2)=O)CC(C)OC(C)C1 c1(CCC(=O)NC(CN(C(C2CC(=C)C2)=O)C)Cc2ccccc2)c[nH]c(=N)[nH]1 C1(C)(CNC(CN(C(C(CO)OC)=O)C2CC2)=O)CC2CCC1C2 c1(C(N2CCCC(F)(CNC(C3CCCC3)=O)C2)=O)cc(F)c2ccccc2c1 N1(C(C(CCSC)NC(C2CCCC(C)(C)C2)=O)=O)CC2(C1)OC(=O)NC2=O C(CCCC(=O)NCCOCCNC(c1ccccc1O)=O)OCC Cc1nc2ccc(C(=O)NCC(F)CNC(c3ncnc(C)c3C)=O)cc2[nH]1 C1(CC#C)(C(=O)NC2CCC(CC(=O)NCC3CC4(CC4)C3)C2)CCOC1 c1(C(=O)OCCC2(O)CN(C(=O)OC(C)(C)C)C2)cnnc(C2CC2)c1 c1(CNC(=O)C2=COCCC2)nnc2ccc(-c3ccc(F)c(F)c3)cn12 C1(CC(=O)NC(C(C)SC)C)COCC1NC(=O)C(O)Cn1cncn1 N1(C(c2coc(C(F)F)n2)=O)CC2OCCN(C(c3ccn(C(F)F)n3)=O)C2C1 CC(O)C(C)(C)C(=O)NCC1(CNC(C2(C(=O)N(C)C)CCC2)=O)CC(F)(F)C1 c1(C(N(CC(CN(C(CCN(CC)CC)=O)C)O)C)=O)ccc([N+](=O)[O-])o1 C(C)(C)(C(C)CC=O)NC(CC1(SC)CC1)=O.c1(CNC(C)=O)nc(CO)n[nH]1 CC(CCC(C)(C)C)C(=O)N1CC2(CC(C(=O)NCCCOC(F)(F)F)CO2)C1 c1(CCN(C)C(c2n[nH]c(O)n2)=O)nnc(C2CCC2)n1C CC(C)C(CCN(C)C(C1(C(C)(F)F)CC1)=O)NC(=O)CCCF C1(CC(=O)NCCN(C(C2CC(OC)C2)=O)C)CCCN1CC(F)(F)F C1(O)(CCNC(c2cc(OCC)no2)=O)CCCN(C(C2CCCC23CC3)=O)C1 C1(NC(CCN(C(C)=O)C)=O)C=CCN(C(c2ncsc2Br)=O)C1 C1(C(=O)NCCCN(C(C(C)OCC#C)=O)C2CC2)CCCN(C)C1 c1(C(N(CCNC(C2CC(OCC)C2)=O)CC)=O)ccc(CO)nc1.C1(N)CC1 c1(C(=O)OCC)ccc(CC(=O)NCCNC(C2CC2C(F)F)=O)cc1 c1(OC)c(F)ccc(F)c1C(=O)NC1COCC1CNC(C12CC1C2)=O C(C(O)C(=O)N1CC(NC(=O)OCC)C1)=CC c1(CC)ccc(C2CN(CC(C)N(C)C)C2)cc1 C1(CC(=O)NC(c2ncnn2C)C)CC2(C1)CN(C(C1CCCC1)=O)C2 C1(CC(=O)NC(CN(C(=O)CC2CCC(F)(F)C2)C)(C)C)CC2(CCC2)CCO1 Cc1cc(C(=O)NC2(C)CC(NC(c3cc(=O)n(C)cn3)=O)C2)c(Cl)cc1F Cc1cnn(C)c1CC(N1CC2C(CC(=O)NC3COCC3C)C2C1)=O CCC(C)(C)C(O)C(=O)N1CC2(CC2)CC1C(=O)NCCc1ccncc1F C1(CNC(C(C)N(C(C23CSCC2C3)=O)C2CC2)=O)CC2(CC2)CO1 c1(C(=O)NC(C2N(C(C=CCCC)=O)CCC2)(C)C)cnc(O)n1CC C1(C(C)C)CN(C(=O)C2=CC(C)(C)C2)CCC1NC(=O)CN(C)CCO c1(NC(=O)NCc2cccnc2Br)csc2ccncc12 c1(C(N(CC(C)C)C2CC2)=O)occc1CNC(C1C=CCC1)=O CC1CCc2[nH]c(=NCc3ccc[nH]3)[nH]c(=NCCCCCCCC3CC3)c2C1 N1(C(C2CCC(OC)CC2)=O)C2CCC1C(C)C(NC(C1CCCO1)=O)C2 N1(C(c2cnn(C)c2Cl)=O)CC(C(=O)NCCC2(CO)CCC2)C2(CCC2)C1 CCCCCCNC(=O)C(c1cc(C)co1)N1CCC(C(N)=O)C1 C1(C(=O)Nc2cnc(N)cn2)CCN(CC2N(C(C(C)(C)C)=O)CCC2)C1(C)C C1(C(N(C)CC2(O)CCN(C(=O)CC3CCCC3)C2)=O)CC(=O)NC(C)C1 C(CCSC)(C(=O)NCC(n1cc(CC2CC2)nn1)C)NS(CC)(=O)=O.C(CCO)O C1(NC(C2OCC(C)C2)=O)CCN(C(=O)CC2CCCCC2(C)C)C1(C)C C1(C(=O)NCC(CC)NC(c2ccc(C#N)cc2)=O)CCCc2ccccc2C1 CC1CN(C(C2CC2C(F)F)=O)CCCN1C(c1cccc2[nH]ncc12)=O c1(C(N2CC(O)(CN(C)C(C3CC4C=CC3C4)=O)C2)=O)c(F)ccc2[nH]ccc12 Cc1ccc(C(=O)Nc2ccc(N3CCN(S(=O)(=O)CCCCl)CC3)cn2)cn1 n1(CC=C)c(N2CCC(CS(=O)(=O)CC)CC2)nnc1-c1cccc(C)c1 CCC(CCC(=O)NCc1ncccc1C)NC(=O)C(OC)OC C1(CNC(CCOCCC)=O)CC(O)CN1C(=O)C(O)C1CC1 C(=O)(CCCCOCC)N(CCC(=O)N1CC(CCCC)C1)CC#C N1(CC(C)C)CCC(C(N2CC(O)(CNC(C3OCCC3C(C)C)=O)C2)=O)CC1 CCC(C)CC(C)C(=O)NC1CCC2CC1CN2c1ccc(C(C)=O)cn1 C1(C(N(CCN(C(=O)CC2CCC(C)(C)C2)C)C)=O)CCn2cncc2C1 Cc1c(CNC(C2C3CC4C(C3NC35COCC3C5)C24)=O)oc2ccccc12 C1(C(=O)OC(C)(C)C)CCCC2(CCCC2)C1.C(C(=O)C(C(C)C)NC(=O)O)OC c1(NC(C2(F)CC(N(C(C3(C(C)(C)C)CC3)=O)C3CC3)C2)=O)nc2c(s1)COCC2 c1(OCC)cc(C(=O)Nc2cccc(O)n2)c(-c2ccc(CCO)cc2)cn1 CCC(CC)C(CCC)N1CCC(c2ccc(-c3nnc(Br)s3)cc2)CC1 CC1(C)CCC(C(=O)NC2CCCCC23CC3)CN1C(C1CC2(CCO1)CC2)=O c1(N(C(CN(CCC#C)C)=O)C)cc(OC)nc(Cl)c1 C1(NC(C2C(NC(c3ccc(COC)s3)=O)CCO2)=O)CC2CC1CC2O N1(C(c2c(C)nc(O)[nH]2)=O)CCC2(CCCC2NC(=O)C(=O)NCC2CC2)CC1 C(=O)(CC(CC(C)C)NC(c1[nH]cc(C)c1C)=O)NCc1ncc(C)nc1 C1(NC(COCc2cc(C)on2)=O)CC2(NC(=O)CCc3cccs3)COC1C2 C1(NC(COCC#C)=O)CN(C(c2c[nH]cc(F)c2=O)=O)CC2(CC2)C1 Cc1nn(C(C)C)c(C)c1C(N1CC(NC(C2CCC(C)(C)O2)=O)C(C)(C)C1)=O c1(OC)ccc(C2(NC(C3CSCN3C(C3(C(F)(F)F)CC3)=O)=O)CCC2)cn1 C1(NC(C2C(C)C2(F)F)=O)CN(C(c2nccnc2C(F)(F)F)=O)CC2(CC2)C1 C1(C(N2CCC3CN(C(c4cc[nH]n4)=O)C3C2)=O)Cc2ccccc2C1 c1(Cn2c(-c3cnn(C4CCC4)c3)nc(C(C)OC)n2)cc(F)cc(F)c1 c1(CCC(N2C(CNC(C(C)CO)=O)C(C)(C)CC2)=O)cccc2c1OCO2 n1(CC)nc(C)c(C(=O)N(CC(C)NC(=O)CCc2c(Cl)cncc2Cl)C)c1C C(=O)(C(O)C(C)(C)C)NC1(CCC(=O)NCC(C)(C)CC2CCCC2)CCC1 c1(C(N(CCC(C)(C)NC(C=CC=CCC)=O)C)=O)cc(Cl)ccc1OC(C)C c1(OC)ccc(Br)c(N)c1C(=O)NC1CN(C(=O)C(C)CF)CC1C c1(CC(N2CC(CNC(c3ccno3)=O)C(O)C2)=O)c[nH]c2cc(Cl)ccc12 N1(C(C(CO)OC)=O)CCCC2(C1)CN(C(c1cc(F)cc(C)c1N)=O)CCO2 c1(CC(C)C)ccc([N+](=O)[O-])cc1.C1(=O)C(C)N1C1CC1 C(=O)(C1=CCCC1)NC(c1ccc(F)cc1)C(=O)OC1(C)CSC1 C1(CC(=O)NCC(=CC(N2C(COC)C=CC2)=O)C)CCOC1(C)C C(CS(=O)(=O)CC(=O)NC1COC2(C1)CN(C(C1CCSCC1)=O)C2)OC c1(CC(N2C(C(N3CCOC(CO)C3)=O)CSCC2)=O)c(F)cccc1F N1(C(C2(CC)COC2)=O)CCC2(COC(CNC(c3nc(C)sc3C)=O)C2)C1 c1(C(C(=O)N(CCC)CC)(C)C)cccc(N)c1 C1(CNC(C(CC(=C)C)NC(=O)CN(CCCCCC)C)=O)CCCCN(C)C1 N1(C(c2n[nH]c(CC)c2C)=O)CCCC(F)(CNC(C2C3COCC23)=O)C1 c1(C(N2CCC(C(C)NC(c3c(C)coc3C)=O)C2)=O)ccc2c(c1)CCC2 CC(C)C(C)CC(=O)N1CC(O)(CN(C(=O)C(N2CCC(C(N)=O)CC2)=O)C)C1 c1(C(=O)NC2(C(=O)NC3CCCCC3C#N)C(C)(C)C2)ncn2ccccc12 C1(C(=O)NC(C2CCN(c3snc(C(C)C)n3)CC2)C)CCc2ccccc2C1 c1(CNC(=O)CNC(c2ccc(Br)s2)=O)cc(Cl)cnc1F Cc1cc(NC(=O)CC2CC(O)CN2C(=O)C(C)CO)cc(C)c1 CCC(CC(=O)OCCCNC(=O)NC1CCN(c2ccn(C)n2)C1=O)C1CC1 CC(C(=O)NCC(O)CNC(c1cnc(C(F)(F)F)nc1)=O)P(C)(C)=O CC(C)C(C#N)C(=O)NCCN(C)C(c1cccc(N2CCCC2)n1)=O c1(C(=O)Nc2c(C(=O)OCC)ccc(OCC)c2)cnc2[nH]cnc2c1 N1(C(CC2(N(C)C)CC2)=O)CC(C(=O)NC2CC(O)C23CCC3)C2(CCC2)C1 c1(C(N(CCCC(=O)OC)c2ccccc2)=O)ccc2nc(Br)nn2c1 C1(CNC(C(C)OC)=O)CC2(CCN(C(=O)C=Cc3ccc(C)nc3)CC2)C1 C1(C(N2CCC(CC(=O)NC(c3cscn3)C)CC2)=O)CC(=O)OC1(C)C C(=O)(C(O)CC(N)=O)NCCOC(C)(C)CNC(C12CCCC(CO1)C2)=O c1(CC)cn2c(C(=O)NC3CC(NC(=O)CC4CC4(Cl)Cl)C(O)C3)cccc2n1 N1(C(C(C2CCCCC2)C)=O)CCC(C)N(C(c2ncnn2C)=O)CC1 C12(C(=O)NC(CC#C)C(=O)NCc3csc(C)n3)CC(C)(CCO1)C2 C1(C(=O)NC2CN(C(c3ccn(CCC)n3)=O)CC2C)CCn2nnnc2C1 S(=O)(=O)(c1ccc(C(C)(F)F)cc1)NCC(C)NC(=O)C(=O)N(C)CC1CCC1 n1(CC(=O)NC(C2N(C(CCCC)=O)CCC2)C)c(C)c(C)sc1=O C1(NC(C2CC(F)(F)C2)=O)COCCN(C(=O)CC23CCCC2C3)C1 CCCC(CC(=O)NC1CC(C2CCC2)C1)NC(=O)CC1(O)CCC1 Cc1cc(CCC(=O)NC2CCCC2NC(=O)C=C2CCCC2)cc(C)c1 C1(NC(C2(C)CCCOC2)=O)CCN(C(c2ccc(N)c(F)c2)=O)CC1F C1(C(=O)NC2C(C)CN(C(c3cccc(=O)n3C)=O)C2)CC2(CCOCC2)CO1 C(C(C)(C)CC(=O)N1CCC(CO)C(NC(c2n[nH]c3c2COC3)=O)C1)OC N1(C(CCC2(C)CN(C(=O)C(F)(F)C(F)(F)F)C2)=O)C2C=CCC1CCC2 N1(C(C2C(CC)(CC)C2)=O)CC(NC(c2cn(C3CC3)nc2C)=O)CC(C)(C)C1 CCCCCC(O)CC(=O)NC1(C)CC(C(=O)NC2CCOC2C2CC2)C1 N1(C(CCC(C)=O)=O)CCCC2(NC(c3ccoc3C)=O)CC2C1 Cn1cnc2[nH]c(=NCCSCCO)nc(N3CCN(CC(N)=O)CC3)c12 c1(C(=O)NC(CC=C)CNC(c2cc(C)c(Cl)c(C)c2)=O)ccc2nncn2c1 c1(OC)cc(C(=O)NCC(C)(C)CNC(c2c[nH]nc2C)=O)c(N)cc1F C1(C(=O)NC2C(CC(=O)NCCOC)CCCC2)CCCC(C#N)C1 Cn1nnc(CNC(C2(N(C)C)CCC2)=O)c1C(=O)NC1CC(C)(C(N)=O)C1 N1(C(COCCCC(C)C)=O)CCOC(CN(C(=O)CCC2CCC(=O)N2)C)C1 C(CC(O)C(=O)NC1CCCC1CN(C)C(C1CSC1)=O)SC c1(C(=O)NC(C(C)NC(CC=CCC)=O)C)ccccc1COC C1(F)(CNC(c2cc[nH]n2)=O)CCN(C(C2CCCC2C(F)(F)F)=O)C1 c1(CNCC23C(O)(CCC2)CC3)nccc2c(Br)cccc12 C1(NC(CCNC(C)=O)=O)CCCC1CNC(=O)CC1C=CCC1 N1(C(C(C)OCCOCC)=O)CC(F)CC1CNC(c1c[nH]nc1C)=O C(=O)(CC(O)CNC(c1cccc(O)n1)=O)NCC(NOCC)=O c1(CC(CC(=O)NC(C)C(C)(C)F)CO)c(F)cccc1F C(=O)(C(=O)C(C)(C)C)N1CC(=C(CNC(c2c(OC)cccc2)=O)F)C1 N1(C(CSC)=O)CCC(NC(c2cc(C)ccc2Br)=O)CC1C N1(C(=O)Cc2ccccc2)CCC2CCCN(C(=O)CSn3cnnc3)C2C1 Cc1cc(C)c(C(=O)NCC2(CNC(=O)COc3cccc(Cl)c3)CC2)[nH]1 Cc1cc(=NC(=O)C(=O)N2CC3CCC2C(NC(=O)CN2CCCC2=O)C3)[nH]o1 Cn1ncc([N+](=O)[O-])c1N1CCC(O)(CCNC(=O)Cc2cccnc2)CC1 c1(OC)ccc(OC)c(CC(=O)N(C2CC(NC(C3CC=CCO3)=O)C2)C)c1 Cc1cc(Br)ccc1C(=O)NCC12CC1CN(C(c1cnc(O)nc1O)=O)C2 C1(NC(c2scc(OC)c2)=O)CCC(C)(CNC(C23C=CC(CC2)C3)=O)C1 c1(C(=O)NS(=O)(=O)CCc2ccccc2)cccc(CN2CCCC2)c1 Cc1cc(C(N2CCN(C(C3CC4(C3)CC4F)=O)CC2C(F)F)=O)cc(=O)n1C C(CC(C(=O)N1CC(NC(c2csnc2Cl)=O)C(F)C1)NC=O)SC c1(-c2nc(-c3c4ccc(CC)cc4oc3)on2)ccc2c(c1)CCN(C(C)=O)C2 S(=O)(=O)(c1ccc2oc(O)nc2c1)N1C(C)CCC1C(=O)Nc1cc(Cl)ccc1Br C1(N2C(=O)CN3CC(C3C(C)(C)C)C2)CC2(CCCC2)C1.C(C)(C)(C)OCC C1(CNC(C(C)N(C(C)=O)C)=O)CC2(CC2)CN1C(C1C2CC3C(C2=O)C13)=O C1(C(=O)NC2CCCN(C(CCn3c(C)cc(C)n3)=O)C2)CCOCC12CCC2 CC1CN(C(=O)CCC2CCCCN2C(c2ccc(=N)[nH]c2)=O)CC(=O)N1 N1(C(C(C2CCOC2)OCC)=O)CCC(NC(=O)CCc2ccc(C)s2)C(F)C1 C1(NC(C2CCC(C(=O)OC)C2)=O)CC2(C1)CC(NC(=O)C=CC(C)C)C2 C1(CC(=O)NCC2CCC(NC(c3[nH]cc(CC)c3)=O)C2)CCCC(=O)N1 Cc1nc2cc(C(N3CC(NC(C4(CCO)CC4)=O)C(C)C3)=O)ccc2n1C C1(NC(C(F)=C(C)C)=O)CCN(C(=O)C(CO)c2ccccc2)C1(C)C C1(NC(C2CCN(C(C)C)CC2)=O)CC2CC(NC(=O)C(F)F)CC2C1 O=[N+]([O-])c1cc(CNCC2CC3(CCOCC3)O2)cc(Br)c1 C1(N(C(C2CC(NC(CN3C(C)CC3)=O)C2)=O)CC2CC2)CCN(C)C1 C(=O)(C(C)(C)C1=CCSCC1)N1C(CN(C(CC=CC)=O)C)CCC1 c1(C(=O)NC(CC2CN(C(C=CC)=O)C2)C)c[nH]c2cc(F)c(F)cc12 c1(CC)c(C)nc2ncnn2c1N1CC(NCc2ccccc2)OC(C)C1 N1(C(C2C(C)C2C)=O)CC2(NC(=O)CS(=O)(=O)C(C)(C)C)CCCC2(F)C1 C1(CCN(C)C)C2CC1CN(C(=O)CCC(N)=O)C2.c12ccc(cc1)[nH]2 Cn1c(NC(C2CC2c2ccc(Br)s2)=O)cc2ccsc12 CC1(C)CN(C(=O)CC2(C#N)CC2)CCC1C(=O)Nc1ccc2nccn2c1 C1(CNC(CC(COC)C)=O)CCCCN(C(=O)C(F)C(C)C)C1 c1(CN2CCC(C(C(F)(F)F)NC(C=C(C)C)=O)CC2)c[nH]c2ncc(C)cc12 c1(C(=O)NC2(CCNC(C3CC(C)OCC3)=O)CCCC2)cc2c(nn1)CCC2 C(C(CC(=O)O)NC(c1ccc(-c2nn[nH]n2)[nH]1)=O)OC Cc1oc(C(C)C)cc1C(=O)NC1CCN(C(=O)CC2CN(C)C2)CC1 n1(CC(=O)NCC2CN(C(C(CC)OCC)=O)CC2C)cccc(N)c1=O c1(C(N2CCCC(NC(CCCC#C)=O)(CO)C2)=O)noc2ccc(Cl)cc12 Cc1c(C(=O)NC2CC2NC(C2CC(=O)N(CC3CC3)C2)=O)cncc1Cl CC1(C)CC(=O)OC1CNC(C1CC(CNC(=O)COCC(F)F)C1)=O CC(CN=c1nc(N(C)CCc2nccs2)c2[nH]ccc2[nH]1)S(N)(=O)=O c1(CC)cnc(CNC(C2CCN(C(=O)Cn3nnnc3C)C2)=O)s1 C1(CNC(CNS(NC)(=O)=O)=O)COC(C)(C)CN1C(C1CCC(=O)N1)=O n1(CCC(=O)NCCN(C2CSC2)CC)cc(Br)ccc1=O c1(C(=O)NC2CC23CCN(Cc2cncs2)CC3)ccc(Br)c([N+](=O)[O-])c1 Cc1cncc(NC(C2C(CNC(=O)Cc3ccc(O)cc3)C2)=O)n1 C(=O)(C(COC)CC(C)C)N1CC(O)(C(C(=O)Nc2c(CC)ccc(C)c2)F)C1 C1(CNC(CC(C)n2cccn2)=O)CN(C(c2cncs2)=O)CC(C)(C)C1 c1(-c2c(C)occ2)nc(C2=NOC(C)C2)n(-c2cc3ccccc3[nH]2)n1 C1(NC(CC2OCCN(C(C3(C)CCCCC3)=O)C2)=O)CCCCC12CC2 C1(N(C(CCc2c(C)nn(C)c2)=O)C)CN(C(=O)Cc2csnn2)CCC1O C1(CNC(c2c(CC)nco2)=O)CC2(CC(NC(=O)CC(C)CN(C)C)C2)C1 c12ccc(cc1)n2CC.N1(C(C)=O)CCC(C)(CNC(=O)CC2CCOC2)C1 C1(NC(COCc2onc(CC)n2)=O)CC2CN(C(=O)CC(C)(C)C#N)CC12 CC(C)CC(C(=O)NCC(CC(=O)N(CCN=[N+]=[N-])C)C1CCC1)C(C)C c1(C(N2CCC(NC(c3cc(CC)no3)=O)CC2)=O)cc(=O)c(OC)cn1C Cc1c(Cl)nc(C(N2CCCC2CNC(=O)C(O)C(C)C)=O)n1C N1(C(CCOc2cncc(C)n2)=O)CCCCCC1C(=O)NC(C)C C1(C)(NC(c2ccc(C)o2)c2nnnn2C)CCS(=O)(=O)C1 CC(C(=O)OC=CC(=O)N1CC(n2cc(COCCO)nn2)C1)S(N)(=O)=O Cc1cc(NC(=O)COC(=O)C(c2cccc(Br)c2)C)ccc1[N+](=O)[O-] c1(CC)cc(C(=O)N(C2C3CN(C(=O)C(=O)NC(C)C)CC23)C)oc1CC C1(C(=O)NCC2(C)CCC(C)C2)CN(C2CCOc3cc(Cl)ccc32)C1 CCCCC(CC)C(=O)NCC1CCCC(CNC(=O)C#CC2(C)CC2)C1 N1(C(c2ccc(CC3CCC3)cc2)C(=O)NCC)CCOC2CCN(C)CC12 CC(C)(C)C(C#N)C(=O)N1CCCC1C1(C(N2CC3(CCNC3=O)C2)=O)CC1 c1(N2CCC(Cc3ccc(C(=O)NCC)cn3)CC2)nc(C(C)C)ccc1C#N Cc1cc2scc(CC(=O)NC34CCN(C(C5(CC(F)F)CC5)=O)CC3C4)c2s1 c1(C(=O)NC2CCN(C(CS(CC)=O)=O)C2)ccc(OC)c2cccnc12 Cc1cc(Cl)ccc1OCCCNC(=O)C(N1CCS(=O)(=O)C1)=O c1(NC(CC2N(C(CC(C)C)=O)CCC2)=O)c(F)ccc(F)c1[N+](=O)[O-] S(=O)(=O)(c1cccs1)NC(C(N1CCN(C(C(COCC)C)=O)CC1)=O)C c1(NC(c2ccc(C(=O)C(F)(F)F)cc2F)C)cccc(CS(=O)(=O)C(C)C)c1 N1(C(=O)CCOCCCO)CCC(N(CCO)C(C2(O)CC2)=O)C1 CC(C(=O)NCC1CC(O)(CNC(C2CCCCCC2)=O)C1)C1=CCCC1 C(CNC(C1(C)CC1C)=O)(CCNC(C1CCCOC1)=O)OC C(=O)(CCCN(C)C(c1ccccc1)C)NCC1(CNC(CSC)=O)CC1 C1(NC(C2OCC(C)(C)C2)=O)C2CCC1N(C(=O)C(C)(C)OCC(F)(F)F)C2 c1(C(=O)NCC2CN(C(C(CC)CC)=O)C(C)(C)C2)c[nH]c2cccc(C)c12 c1(SCC(=O)NCC(CNC(CC2N(CC)CCC2)=O)OC)ccc(F)cn1 c1(C(c2n(CCOCC)nnn2)NC)cc(C(=O)OC)c2n1CCOC2 c1(C(=O)NCCCN(C(COc2cc(C)c(Cl)cc2)=O)C)ccnc2[nH]nnc12 N1(C(C2(C(=O)NC)CC2)=O)CCC(NC(C2CCC(N(C)C)C2)=O)CC1C c1(C(=O)NCC2CCN(C(C3CN3C3CC3)=O)C2)c(F)ccc2ccncc12 c1(OC)ccc(NC(c2cccc(NCc3ccncc3)c2)=O)cc1Br C1(C(CO)NC(CCC=CCC=C)=O)CCN(C(c2ccc(SC)cc2)=O)CC1 C#CC1(C(=O)NCc2csc(CC)n2)CN(C(C2(C(C)=O)CC2)=O)C1 Cn1cncc1C=CC(N1CCCC1C1CCCCN1C(c1cc[nH]n1)=O)=O C1(C(N(CCC#C)CCO)=O)CCN(C(=O)C(=O)C(C)C)C(CC)C1 Cc1nc(CCCC(=O)NCCC(C)N(C)C(c2coc(Cl)n2)=O)cs1 C=CC1(C(N2CCC(NC(=O)C(C)CCOC)C(C)C2)=O)CCOCC1 C(=O)(C(C)(C)CCNC(=O)CC1CSCCS1)NCCC1N(C)CCC1 C1(CCC)(NC(C2CCN(C)C2)=O)CCCN(C(c2snnc2COC)=O)C1 N1(C(C2CC(C)(C)C2)=O)CCC(C2CCN(C(C3COC(=O)N3)=O)CC2)CC1 N1(C(=O)CN2CCCC2)CC2CC(C1)CN(C(c1ccc(F)cc1F)=O)C2 N1(C(CCS(=O)(=O)NC)=O)CCC2(CC(NC(=O)CCS(=O)(=O)NC)CO2)C1 CCC(C)C(CC(=O)N1CCC(CO)C(C)C1)NC(C1(COC(C)C)CC1)=O C1(CN(C(c2cc(SC)oc2)=O)C)CCCCN1C(c1cc(C2CC2)ccn1)=O C(=O)(C(C)(C)c1cccs1)NCCN(C(=O)CCc1cc(Cl)cs1)C(C)C C(=O)(C1=NOC(C)C1C)N1CCCC(CNC(CC(=O)OC)=O)C1 C1(C)(CNC(C(C)NC(=O)Cc2ccccc2)=O)CCN(C(=O)C(N)=O)CC1 N1(C(c2cccc(C)c2F)=O)CC(CNC(=O)CC(F)F)CC12CCC2 C(CC(C)C(=O)N1CCCC1C(C)(C)NC(=O)C(C)C1CCCO1)OC C(=O)(C(S(C)(=O)=O)C1CC1)NC1CN(C(c2cc(CC)oc2C)=O)CC1O N1(C(C2C(O)CCN(C(c3nc(C(C)C)oc3)=O)C2)=O)Cc2cccc(F)c2C1 C=CCCCCCC(=O)NCC1CCC(n2cc(C3C4CCOCC34)nn2)CC1 C1(NC(CCOCC)=O)CN(C(C2CCN(C3CC3)CC2)=O)C2(CCCC2)C1 Cc1ncnc(O)c1C(N1CC(NC(=O)Cc2cncnc2O)C(F)C1)=O C1(NC(c2ccc(CNC(C(C)S(C)(=O)=O)=O)cc2)=O)CCn2cncc2C1 Cc1cc(C(=O)NC2(CO)CN(C(C3CCC4CC34)=O)C2)nn1C(C)C1CC1 C1(CC)CCC2(CC1)CCN(S(=O)(=O)NC(c1ccoc1)C)CC2 C12(CC)CC(C1)C(C(=O)OCCCNc1ccc(N(C)C)cn1)CO2 N1(C(C2(CNC(c3c(C)n(C)nc3)=O)CCCCC2)=O)CCC(O)C(F)C1 C1(OC)CC(CCNC(c2ccnc(S)c2)=O)N(C(c2ccnc(C)c2)=O)C1 C1(C(=O)NCC(CNC(c2n(C)nc(C3CCC3)c2)=O)F)CCC2CC2CC1 C#CC1CC2CCC1N(C(=O)CC1CCC(NC(=O)C=CCOC)CC1)C2 C(=O)(CC(O)CC(C)(C)C)NC(CC(C)NC(COc1c(CC)cccc1)=O)C N(C1CCCc2c1cnn2C(C)(C)C)C(N(CCC)CCN(CCC)CC)=O C(=O)(C1=NNC(=O)CC1)NC1(CO)CCN(C(CC(C)CN(C)C)=O)C1 CC1C(NC(c2cnc(C(C)(C)C)s2)=O)CCCN1C(=O)Cc1cn[nH]c1 N1(C(c2cn(C(C)C)nc2)=O)CCN(C(=O)COCCSCC(F)F)CC1 C1(C(=O)NC(C2CCN(C(C3(C(N)=O)CC3)=O)C2)C)CC(F)(F)CS1 CC1CCCC1(C)C(=O)N(CC(C)NC(=O)Cc1ccsc1Cl)C C12(CNC(CCCC(C)O)=O)CCCCC1N(C(=O)CCOCCN(C)C)CC2 CCCC(C(=O)NC1COCCC1NC(=O)C=CC(=O)OC(C)(C)C)N(C)C c1(C(N2CC(C)C(NC(=O)CCOC3CC3)C2)=O)ccc(C(F)F)cc1F Cc1cc(C(=O)NCc2csc(CNC(=O)CN(C3CCCC3)C)n2)ncc1N Cc1cc([N+](=O)[O-])cc([N+](=O)[O-])c1N1CCCC(NC(c2cocc2C)=O)C1 C=CC12CC(CCN1C(=O)Cc1c(C)n[nH]c1C)C2 Cc1nc(C(N2CCC(C(C)CNC(=O)CCCCN(C)C3CC3)CC2)=O)cn1C CCCCCCCCC(C)C(=O)N1CCC(N(C(=O)C=C2CCCCC2)CC)CC1 C1(CC(=O)NCC(=C)CCNC(c2n[nH]c(CC)n2)=O)CCC(=O)N1CCOC c1(C(C)C)cc(C(N2CCCCC2C2C(C(=O)NC(C)C)C2)=O)nc2ncnn12 CCCCC(C(=O)NCC(C)CC(=O)NC(C)(CC)CCO)N(C)C c1(OC)ccc(C(=O)NCCCN(C(=O)C2=COCCC2)C2CC2)c(F)n1 C(=O)(N1OC2CC1C(O)C2O)C1C(NC(c2c(NC)nccc2)=O)CCOC1 c1(NC(C2C(NC(c3c(C)noc3C)=O)CCCC2)=O)ncnc(O)c1Br N1(C(C2N(C(C)=O)CS(=O)(=O)C2)=O)CC2CC1CN2C(=O)CSC(F)(F)F Cc1c(C(N2CC3(CC(NC(c4ccco4)=O)C3)C2)=O)cnc2ncnn12 N1(C(c2c(CC)onc2C)=O)CCC(F)(C(=O)Nc2ccc(C)nc2)CC1 n1(CC(=O)NCCNC(C(CCC)(C)OC)=O)cnc2ccccc2c1=O CC(CC(F)F)C(=O)NC1CCCCC1CNC(C1(N(C)C)CC1)=O C(C)(C(CC(=O)NC(C)C1CC1)NC(=O)Cn1ncccc1=O)OC C1(CNC(C(COC)O)=O)CCN(C(=O)Cc2cn3c(C)csc3n2)CC1(F)F CCC(C(N)=O)NC(=O)CNC(=O)C(C)(C1CCCCC1)OC C(=O)(C(=O)N=c1cc(C)n(-c2ccc(C)cc2)[nH]1)Nc1cnc(C(=O)NC)nc1 N1(CC(=O)NC2(C)CC(NC(CCc3n(C)cnn3)=O)C2)CCC(=O)NC1=O c1(C(=O)NC(CC)(C)CNC(=O)C(C)=C(C)C)cc(N)cc([N+](=O)[O-])c1 C(=O)(C1=C(C#N)CCC1)N1C2CN(C(c3onc(CC)c3C)=O)CC1C2 N1(C(c2nc(C)nn2C)=O)CC2(CCCN(C(C3CC(C)(C)CO3)=O)C2)C1 C(C#Cc1ccccc1Cl)N(C(=O)CC1CCCCC1)C N1(C(C(C=C)(C)C)=O)CC(NC(=O)COCc2ccccc2Cl)CC2(CC2)C1 c1(C(=O)O)cccc(-c2cccc(COC)c2)c1N.N12CCCC1C2(C)C Cc1cc(=NCC2CC(=O)NC(C)C2)[nH]c(=NCCC2CN(C)C2)[nH]1 C=CC(CC)CC(=O)NCC1CCN1C(=O)C(C)(C)C(F)F C1(NC(C(C)CO)=O)CCCC12CCN(C(c1cc(C(F)F)ccn1)=O)C2 N1(C(c2c(C)cn(C)c2)=O)CC2CC(NC(c3cnn(CC(C)C)c3C)=O)C1C2 c1(CCC(=O)NC23CC(NC(C4C(C(=O)OC)CC4)=O)(C2)C3)ccc(C)cc1 C1(C(=O)OC)CCc2nc(=NC(=O)Cc3cnn(C(C)(C)C)c3)[nH]n2C1 C(C)(C(=O)NCC1CCCN1C(=O)Cn1nc(C)n(C)c1=O)(C(C)C)NC(C)=O c1(C(=O)NCC2CN(C(C=NOC)=O)CC2(C)C)cccc2nc(S)oc12 C1(C(N(CC(N2CC(N(C)CCO)C2)=O)CC2CC2)=O)CCN(C)C1 C1(CNC(=O)NCc2ccccc2F)C(Cl)(Cl)C12CC2 C1(C(=O)NCC(CC(C)C)OC)(CNC(C(C)NC(CC)(C)C)=O)CCCCC1 c1(N(CCOC)CCNC(c2cccn2C)=O)cc(OC(F)F)ccc1[N+](=O)[O-] C1(CNC(c2ccc(C3(CC)CC3)s2)=O)C2CCC(C2)N1C(C1CCCC(=O)N1)=O C1(CNC(CNC(CCC)=O)=O)(CNC(C2CCS2(=O)=O)=O)CCOCC1 C1(C(=O)NCCC(C)O)CCC2(CCN(C(=O)COCC3CC3)CC2)C1 Cn1ccc2c(CNC(C3CC4(C3)CC4(F)F)=O)ncnc12 C1(CNC(C(COC)(F)F)=O)Cc2ccccc2CN1C(c1ccc(Cl)cn1)=O c1(C(=O)NC(C2CCCCN2C(c2ccc[n+]([O-])c2)=O)C)c(F)cc(Cl)cc1F CC(C)CC(O)C(=O)N1CC(O)(C(F)C(=O)N(C2CCCC2C)C)C1 C1(C2CCCN(C(c3cnc(Cl)cc3Cl)=O)C2)(NC(c2cc[n+]([O-])cc2)=O)CC1 c1(CC)nnc2n1CC(NC(c1cn3cc(Br)cc(C)c3n1)=O)CC2 c1(CN(CCCNC(c2cn(C)nc2)=O)C(=O)COCCCO)ccccc1Cl c1(C(N(C(CCNC(c2cc(C(C)=O)c(C)o2)=O)C)C)=O)onc2c1CCCC2 C(=O)(C1CCCc2n[nH]cc21)N1C(C(C)(C)NC(c2cnc(C)s2)=O)CCC1 C1(C(=O)NC2CC(=O)N(C)C2c2nccn2C)CCC2(CCC2)CN1 C1(NC(C2CCC(C)O2)=O)CC2(C1)CC(NC(=O)CC(C)c1cccs1)C2 C1(NC(c2n[nH]c(C)c2Br)=O)CN(C(=O)CC2CC2(C)C)C(C)(C)C1 N1(CC=CCNC(=O)NCC(=O)OC(C)(C)C)CCCS1(=O)=O C1(CCCC)CN(C(C2(C)CC(C)=NO2)=O)CCN1C(c1csnc1C)=O CC(C)CC(O)C(=O)N1CCCN(C(c2cccc(Cl)c2)=O)CC1 C1(NC(c2ccc(C(C)C)o2)=O)CCN(C(C2(C)CCC2)=O)CCC1CO C(=O)(C#CC1CCCC1)NCC1C2N(C(c3n(C(C)(C)C)ncc3)=O)C(CC2)C1 C1(NC(C23CC(COC)(OC2)C3)=O)C2CCC1N(C(=O)CC1(CSC)CC1)C2 C(CC)(CC(F)(F)F)NC(C1N(C(C(CC=C)OC)=O)CC(=O)C1)=O N1(C(c2cc(CNC(CCSCC)=O)on2)=O)CC2(CCC(C)OC2)C1 C1(C(N2C3C(CNC(C(CC=C)C)=O)C(C3)C2)=O)CCC2(CCC2)CO1 Cc1[nH]nc(C(=O)NC2CCC(CCNC(c3cccn3C3CC3)=O)C2)c1Cl C1(C)(NC(C(C)(F)F)=O)CCCN(C(c2ccc(C(F)(F)C(F)F)cc2)=O)C1 N1(CC(=O)NCC(CCNC(c2ccc(C(N)=O)o2)=O)O)CCCCCC1 N1(CCOCC=C)CCCC(C)(CNC(=O)CSCC=C(C)C)C1 C=C(Cl)CCC(=O)NCC=CCNC(c1sc(C(C)OC)nc1C)=O N1(C(C2CC(N(C)C)C2)=O)CCN(C(=O)C(F)CC2CC2)C(CC(F)F)C1 N1(C(C(C(C)O)C)=O)CCC(C2CCN(C(c3ccc(F)c(O)c3)=O)C2)CC1 C(c1cccc(Cl)c1Cl)=CC(N1CC2C(CNC(c3cnc[nH]3)=O)C2C1)=O CC1(CNC(=O)Cn2ccc(Br)n2)CCCN(C(=O)Cn2ncnn2)C1 c1(C(N2CC(CNC(c3c(C)cn(C)n3)=O)C2)=O)cc(Br)c(Cl)cn1 c1(C(=O)NC2(CC)CN(C(c3cccc(F)c3N)=O)C2)ccc(OC)nc1Cl C(=O)(CCCC(=O)C1C(C(=O)NCC2CC2CNCC)C1)NCC C1(CC(=O)NC2CC3(CC3)C2)CCC(NC(C2(CC)CC(CO)C2)=O)CC1 c1(CC)nnc(N)n1CC.c1(C(N(C2CCSC2)C)C)ccccn1 c1(CCC(=O)NC2CCC(CNC(CSCCCC)=O)C2)n[nH]c2c1CCCC2 c1(OCC(=O)OC2CCCN(C(CC)=O)C2)ccc(C)cc1C N(C(=NCc1ccc(Cl)nn1)N1CCC(Cc2c(C)noc2C)C1)C(CC)C C1(N(C(C)CN)C)C2C3CC4C1C1C2CC3C41.c1(CC(=O)C=O)nc(CN)cs1 C12(CNC(CC(=O)OC)=O)CC1CN(C(c1ccccc1NC1CC1(F)F)=O)C2 N1(C(c2cc(OC)n[nH]2)=O)CCCCC1C(=O)NCC(O)C1CCC1 c1(CC)c(C(=O)NCCN(C)C(C2CCCN2C=O)=O)[nH]c(C)c1C(N)=O C1(CCNC(COC)=O)CC(F)(F)CN1C(C1CC1CC(C)C)=O CC1CC(CNC(=O)CC23COCC(C2)C3)CN1C(c1ccnc(C(N)=O)c1)=O n1(NC2(c3cccs3)C(C)C2)nc(-c2cnn(C)c2)nc1C.c1(SCC)cnnn1CCO CC1CCN(C(C2CCC=CCC2)=O)CCN1C(c1cnc2c(c1)COC2)=O C1(C(N2CC(OC)C(NC(c3cnns3)=O)C2)=O)CC(c2ccccn2)=NO1 c1(OC)cccc(C(=O)N(C)CCN(C(=O)CC2(c3ccon3)CC2)C)n1 N1(C(C(C)=CC)=O)CCN(C(C2C(OCC)C2C)=O)CC1c1ccccc1 C1(C(=O)NCc2cn(-c3cnc(NC)nc3)nn2)CCc2ccc(F)cc2O1 C1(CCOC)CN(C(c2cc(Cl)n(C)n2)=O)CCN1C(C1CC2(CCC2)CO1)=O C=CCC(C(=O)NC1(C)CC(NC(=O)CC2CCCC2)C1)C(C)(C)C C1(NC(C2(C#N)C(C)(C)C2)=O)CC2(C1)CC(CNC(c1cscc1C(F)F)=O)C2 N1(C(c2ccsn2)=O)CCCN(C(c2ccc3ccsc3c2)=O)C(CO)C1 C1(C(=O)OCc2ccccc2)CCN(C(C2CCCN2c2ccncn2)=O)C1 CC(CC(=O)NCCCC(N1CCC(O)C(F)(F)C1)=O)C(C)(C)C N1(C(C2=CC(O)C(NC(Cc3cn(CC)nn3)=O)C2)=O)CCN2C(=O)CCC2C1 C1(NC(c2n(C)nc(C)c2Cl)=O)CC2CC(C1)N(C(=O)CSc1cnn(C)c1)C2 C1(CNC(CC2(C)CC2)=O)CCCC2(CN(C(c3ccc4cncn4c3)=O)C2)O1 CCN=c1[nH]c(C)c(C(N2CCCN(C(=O)CC3CCC34CCC4)C(C)C2)=O)s1 c1(C(=O)NCC(CNC(=O)CCc2nc[nH]n2)OC)sc(O)nc1C c1(N2CCC(CNC(C(C)C3CCC3)=O)C2)nc(Cl)nc2c1cnn2C CC1(C(=O)NC2CCN(CCCNC(c3cncs3)=O)C2)CC=CCO1 C12(C(=O)NC3CC(NC(C4CCC(CC(C)C)C4)=O)C3)CCCC1C2(F)F c1(OC)cnc(C(=O)NC2CCOCC2)cn1.C12(CCC1)CC(=O)NC2 n1(CC)cc(CC(N2CCC(NC(c3cn(C4CCC4O)nn3)=O)C2)=O)nn1 N1(C(C(C)C2(O)CCC2)=O)CC2(CCC(C(N3CCC(F)(F)C(F)(F)C3)=O)O2)C1 c1(CC)ccc2c(c1)C(N1C(=O)NC(CCCF)C1=O)CC2 N1(C(CC(C)n2cccc2)=O)CC2(C1)CN(C(=O)COCc1nccs1)C2 c1(C(N2CCC(O)(CNC(=O)C(F)C3CC3)C2)=O)cc2ccnc(Cl)c2[nH]1 c1(C(c2nnnn2C2CC2)NC(CC)(C)COC)ccc(C#N)c(OC)c1 c1(CN(C(=O)CC2(CC)CCCCC2)CCOCC)ccc(C(F)F)c(F)c1 C(CCCCCNC(=O)COC1CCCC(C)O1)n1cc(CCCC(C)O)nn1 Cc1c(N)ccc(C(=O)NCCCN(C)C(C2(C)CC2Br)=O)c1F C(CC(=O)N1CCC(C)(CN(C)C)C1)(C(F)(F)F)NC(c1c(C)nc(C)s1)=O c1(C(=O)NC(CCCCNC(C(C=C)(C)CC)=O)C)ccc(Cl)c(S(C)(=O)=O)c1 C(N=c1[nH]c(=NCCC(=O)NC2CC2)c2[nH]ccc2[nH]1)C1C(CCC=C)C1 C1(C(N2CC(F)(F)C2C2CC2)=O)CC2C=CC1N(C(=O)Cc1cnsc1)C2 c1(OC)c(Br)csc1CNC(=O)NC1(OC)CCCC1 C1(NC(C(C)(C)n2ccnn2)=O)CC12CCN(C(C1CCC(F)(F)C1O)=O)CC2 C1(C(=O)NC(CC#C)(C)C(=O)OC)CC2(CCN1C(C1CCC(F)CC1)=O)CC2 N1(CC(CC)OC)CCC2CC(C(=O)NC3CCC(O)CC3)C2C1 C1(C(C)C)(CNC(C2CC2(C)C)=O)CCN(C(C2CCN2C)=O)C1 c1(C(=O)NCC2CN(C(C3=C(C)OCC3)=O)C2)cc(C(C)C)nc2onc(C)c12 C#Cc1ccc(C(N2CC(C(=O)Nc3ccc(Cl)nc3)CC(C)C2)=O)cc1 c1(CC)nc(C)ccc1Cc1onc(C2(Oc3ccccc3)CC2)n1 c1(OC)ccccc1C(=O)NCC1CN(C(c2cnns2)=O)C2CC12 Cc1ncn(C)c(=O)c1C(=O)NC(CO)CCCCNC(=O)C=C(Cl)Cl c1(C(N2C(CNC(C(CC)(C)OC)=O)CCCC2)=O)cn2cc(C)c(C)cc2n1 O=C(C1=CCSC1)NC1CCCC1CNC(c1nccc(C(F)F)n1)=O C12(C(=O)NCc3cn(CCNC(C4CCCO4)=O)nn3)COCC(C1)OC2 N1(C(c2cc(OC)n[nH]2)=O)CCCCC(NC(c2cn(C(C)(C)C)nc2C)=O)C1 C1(O)(CNC(CCN(CCCCC)C)=O)CN(C(c2cc(C3CC3C)on2)=O)C1 CCC(C)C(O)C(C)C(=O)NCC1CC(NC(c2ccc([N+](=O)[O-])s2)=O)CCO1 CC1CCC(NCC2CC3C=CCC(C2)C3)Cc2ccccc21 N1(C(c2c(C)con2)=O)C2CCC(C2)C1CC(N1CCC(C(C)C)CC1)=O C1(C(N2CCCCC(Nc3cc(C)ncn3)C2)=O)CCC2C(CC1)C2(F)F Cn1cc2cc(CNC(C3(c4cc(Br)ccn4)CC3)=O)ccc2n1 c1(OCC(=O)NC(C(C)NC(C2CC2(F)F)=O)(C)C)c(F)c(F)c(F)c(F)c1F CC1CCN(C2(c3cn(C4COCC4NC(=O)C(C)(C)F)nn3)CC2)CC1 N1(c2n(Cc3[nH]ccc3)c(CC3CCOCC3)nn2)CCCC2(COC2)C1 C1(NC(CC2(NC(C)=O)CC2)=O)CC(CNC(c2ccc(F)cn2)=O)CC1O Cc1cc(=NC(=O)C(C(C)C)Sc2nc(-c3ccc4ccccc4n3)no2)[nH]o1 Cc1cc(N2CCC(CNC(=O)Cn3nnnc3C(C)C)C(C)C2)nc(Cl)n1 C(=O)(CC(O)C(C)(C)C)N1CCC(N(C(CCCc2ccc(C)cc2)=O)CCO)C1 N1(C(c2nc(C)n(C)n2)=O)CC2=C(C1)CN(C(C1CN3CCCC1C3)=O)C2 N1(C(C2CNC(=O)N2)=O)CCOC2(CCN(C(c3ncsc3C(F)(F)F)=O)C2)C1 N1(C(c2nc(-c3scc(C)c3)n(-c3ccccc3Cl)n2)=O)CCn2cccc21 c1(C(N(C(CNC(C2(F)CCCC2)=O)C2CC2)C)=O)ccc2nnnn2c1 C1(OC(N2CC(C(C)NC(c3cnnn3C)=O)C2)=O)NC(=O)OC1C C(=O)(CC(CC(C)C)NC(=O)C(F)C(CC)CC)NCC(CC)n1cccn1 c1(NC(C2N(S(CCC)(=O)=O)CCOC2)=O)cc(OC)cc(C#N)c1 c1(C(C)C(=O)NCCn2cc(-c3cnc(C(=O)N(C)C)o3)nn2)cncc(F)c1 N1(C(=O)Cn2ccccc2=O)CCC2C1CCN2C(C1CCCOC1)=O C(=O)(CC(C)C(C)(C)NC(=O)CCC1CC1C)NCc1c(C)nc(C)[nH]1 N1(C(C2CN(C(=O)NC3CCN(CC)CC3C)C2)=O)CCC(C=CC(=O)CC)CC1 C(=O)(C1CCCc2cncn21)N1CC(NC(c2cc(=N)[nH]cc2)=O)C2(C1)CC2 C1(CC(=O)Nc2cc(O)ncn2)CCN(C(c2cccs2)=O)CC1 C1(OC)CN(C(=O)CCOc2ccccc2Br)CC1NC(=O)Cc1cc[nH]c1 C1(C(=O)NCCC2CCCN(CC3CC4(CCC4)C3)C2)CCCS(=O)(=O)C1 C1(F)(CNC(C2(C)CC(F)C2)=O)CCN(C(=O)C(c2cc(Cl)cc(Cl)c2)O)CC1 CC1(C)CCCC(C(=O)NCC2CCN2C(=O)COC2(C)CCOCC2)CC1 N1(C(CSCCOC)=O)CCCC(N2CCN(C(C3(C)CCCOC3)=O)CC2)C1 C(=O)(N=c1[nH]nc(-c2ccccn2)s1)C1CCN(C(=O)CSc2cnon2)C1 C(C(CCC(F)(F)F)C(=O)O)NC(C(=O)N(CC)CC1CCCC1O)=O CC1=C(C(=O)N2C(C(N3CCC3CO)=O)CCC2C(C)(C)C)CCO1 C(=O)(C(C(C)NC(C1CC2(CC2)C1)=O)C(C)C)NCCC(=O)NCC(C)C S(=O)(=O)(c1ccc(Br)cc1NC(c1nncs1)=O)NC(C)=O.C1C(CO)N1 c1ccc(C)c(O)n1.N1(C(C=C(C)C)=O)CCN(C(C23CCC(C2)C3(C)C)=O)C2CC12 C1(C(c2nnnn2C2COC2)NC2(COC)CCCC2)CCCCCC1 c1(OCC)cc(C(=O)NC)ccc1OCc1ccc(Cl)s1.C12CCN(C1)C2 c1(CNC(C(=O)NC(C)(C)CF)Cc2cncs2)cccc(C(=O)OC(C)(C)C)c1 C1(NC(c2ccc(C#N)cn2)=O)CN(C(c2cocn2)=O)CC12CCC2 C12(NC(C(C)C3CCCO3)=O)CC3CC(C1)CC(CNC(=O)C(F)C1CC1)(C3)C2 C(=O)(C(CNC(c1ccc(C)c(C)n1)=O)C(C)C)N(CCC#C)CC N1(C(CC2CN(C)C2)=O)CCN(C)CC1CNC(=O)CC1(C#N)CCC1 c1(OC)ccc(Br)c(C(=O)NC(C)(CNC(=O)CCC2CC2C)C2CCC2)c1 c1(C(N2CCN(Cc3ccc(O)cc3)C3CC23)=O)ccc(Cl)c(F)c1F CC12CN(C(C3CC3(F)Cl)=O)C(C(=O)NC3(C4CCC4)CC3)(C1)C2 CC1CCN(C(=O)CCn2ccccc2=O)C(CNC(C2CC2C#N)=O)C1 C1(C(=O)NCC(CO)NC(c2cc(C)n(C)n2)=O)(CC)CCC(O)CC1 N1(CC(=O)NCC2CCC(O)C2)CCN(C(c2cnc(S)nc2)=O)CC1 C1(O)(CC2(C(=O)NCC)CCCC2)CCN(C(=O)COCC2CCCO2)C1 CS(=O)(=O)CCCC(=O)N1CCN(C(c2cccc(O)c2)=O)C(CF)C1 C(=O)(C(C(C)C)C(C)C)N1CCC(c2ccccc2)(NC(c2c(C)noc2)=O)C1 Cc1ncccc1C=CC(N1CCCN(C(C2CCN(C)C(=O)C2)=O)CC1)=O c1(OCC(=O)NCC(CNC(=O)C(C)S(N)(=O)=O)OC)ccc2c(c1)CCC2 C1(C(N(CCOC)C)=O)CCCC(NC(c2nnccc2C)=O)C1 c1(C(N(CCCNC(COCC#C)=O)C)=O)n[nH]c(-c2ccccc2)c1C C(N=c1nc(N2CC(CO)C3(CC3)C2)c2c([nH]1)c(C)nn2C)c1c(C)nn(C)c1 C(C(O)C(=O)NC(C)CCNC(=O)C(C)Nc1ccccc1)SC c1(C(N2CCOC(CN=c3ccnc(CO)[nH]3)C2)=O)ccc(Br)c2ncccc12 c1(C(N(C2CCCN(C(C3C=CCC3)=O)C2)CC)=O)cc(Cl)cc(Cl)c1F CC1CC(=O)NCC1C(N1CCC(CO)(CNC(c2nc(=N)cc[nH]2)=O)CC1)=O C1(COC)(CO)CCN(C(C2CCC(NC(c3ccc(OC)o3)=O)CC2)=O)CC1 C(C1CCOCC1)=CC(=O)NC(C1CC1F)=O.c12cccc(c1)NC2=O.C1CS1.NCO c1(OC)ccc(F)cc1C(N1CCOC(CNC(=O)CCc2cncn2C)C1)=O CC(=O)CCCC(=O)N1CCC(C(N2CC3CC2C3)=O)O1 N1(C(c2c(C)cn(C)n2)=O)CCCCCCC1C(=O)NC(C)Cc1cccnc1 c1(CC(=O)NC2CC3(C(NC(C(C)C(F)(F)F)=O)C3)C2)ccc2ccccc2c1 CC1CCc2[nH]c(=NC3C=C(c4ccccc4)C3)nc(N(C)CC3(CO)CC3)c2C1 N1(C(c2c(C)nsc2C)=O)CCC(NC(c2nccn2C)=O)C(CO)CC1 C1(NC(C2(CNC(C(CC)N(CC)CC)=O)CC2)=O)CCc2ccc(F)cc2C1 N1(C(C(C)OC)=O)CCC2CN(C(C3(C(F)(F)F)CCCCC3)=O)CC2C1 N1(C(C2CC3(CC(=O)C3)C2)=O)CCN(C(C2CC=CC2)=O)CC(O)C1 C1(C(=O)NCCN(C(=O)CC2COC(=O)C2)CCC)(C(F)F)CCOCC1 N1(C(CCCOC(C)C)=O)CCC2CN(C(=O)Cc3c[nH]ccc3=O)CCC2C1 N1(C(C=CC)=O)CCC2(CC1)CC(C)N(C(c1ccccc1C(N)=O)=O)C2 C1(C(=O)NC2CCC(NC(CCC#CC)=O)CC2)CCOCC12CCCC2 c1(NC(C2(CCNC(CSCC)=O)CC2)=O)cc(Br)ccc1C#N c1(SCC2(O)CCCN(C(=O)Nc3c(C)cccc3)C2)cc(C#N)ccc1Cl C12(C(=O)NCC3(CCOCC)CC3)CC1CCN2C(c1cnnn1C)=O c1(C(N2CCC(C(N3CCC4(CC3)COC4)=O)C(F)C2)=O)cccc2c1CCC2 N1(C(C2CCSC2)=O)CCC(C2(O)CCN(C(=O)CCC(F)F)C2)CC1 C1(C(=O)NCCn2nc(C)nc2C)(OC)CCN(Cc2ncc[nH]2)CC1 C1(C(N(C)CCOCCC(=O)NCC=CC2CCOC2)=O)CCOC1(C)C C#CCCCCCCC(=O)N1CCCCC1CNC(c1cc(N)c(O)c(F)c1)=O C1(CNC(NNC(=O)NCCOC)=O)CC2(CCCCC2)C1 n1(CC)ccc(C(N2CCN(C(C3CN(C(=O)NC)C3)=O)C(C)C2)=O)cc1=O c1(CCC(=O)N(CCc2ncc(CC)[nH]2)CC)ccc(C)nc1 C1(CC(=O)NCC2C3CN(C(C(C=CC)O)=O)CC32)CCCS(=O)(=O)C1 CCC(CCOC)C(=O)NCC(CCNC(=O)C(C)S(N)(=O)=O)OC N1(C(c2ccn(C)n2)=O)CC2CCC(CNC(=O)CC(F)(F)C(F)F)C2C1 C(CCCCC(=O)Nc1ccc[n+]([O-])c1)N(C)C(C1(Cl)CC1(F)F)=O C(C1CCCN1C(=O)CC(C)F)=CC(N1CCC(C(C)C)C1)=O N1(C(CSCCCC)=O)CC(O)(C2CCCN2C(=O)CCOCC(F)F)C1 c1(OC)ccc2c(c1)CCC2C(=O)NCC1C(=O)N1.C(C)(CC(C)C)NC(C)=O C12(NC(c3ccc(OC)c(Cl)n3)=O)CCCC1N(C(=O)C(C)(C)OC)CCC2 N1(C(C(N2CCCCCC2)C)=O)C2CCC1C1CC1(NC(=O)CCC(C)(C)F)C2 Cn1cnc2ccc(C(N3CC(NC(C45CCC4C5)=O)C4(CC4)C3)=O)cc12 Cn1cc(-c2cn(C3CCCC(F)C3)nn2)c(-c2ccc(Br)s2)n1 C1(NC(C2CC3CC2CC3NC(C2(F)CC=CCC2)=O)=O)CC2(CCOC2)C1 CC(C)CC(C(=O)NC1CCN(CCCNC(=O)CC2CN(C)C2)C1)N(C)C N1(C(C2CC(O)(CC#C)C2)=O)CCC2C(CCCN2C(=O)C=Cc2cocn2)C1 C1(NC(C(c2cncnc2)C)=O)CN(C(c2cnc[nH]2)=O)CC2(CC2)C1 Cc1cc(C)c(C(=O)N(CC(C)CNC(=O)Cn2nnnc2C(C)C)C)[nH]1 CC1(C)CC(C(=O)NC2CCN(C(C3CCOCC3)=O)CC2(C)C)C(C)(C)O1 N1(C(c2c(C)cco2)=O)C2COCC1CN(C(=O)C(n1cc(Br)cn1)C)C2 CC1OCC2(CCNCC2)C1N(S(=O)(=O)C(Cl)(Cl)Cl)Cc1ccc2c(cnn2C)c1 C1(O)(CNC(C2CN(C)C(=O)C2)=O)CC(N=c2cc(Cl)nc(CS(C)(=O)=O)[nH]2)C1 c1(CCC(=O)NCC(C)CNC(=O)CNC(N)=O)cccnc1 c1(OC)cc(C(C)NCC2(C)CCN(C(=O)OC(C)(C)C)C2)cc(Cl)c1 C1(C(N2C(C)CC(CNC(=O)CCSC(F)(F)F)C2)=O)CC2CCC(C1)S2 C(=O)(CCCCCN=[N+]=[N-])NC(CCCC(=O)N(C1CCCC1)CC#CC)C O=C1CC(CC(=O)N2CCC(C(F)CNC(c3c[nH]c(C(F)F)c3)=O)CC2)=NN1 C(=O)(N=c1ccn(-c2ccc(Cl)cc2Cl)[nH]1)N(CC#N)C1CC1 c1(C(=O)NCC23CC2CN(C(c2ccsc2)=O)C3)cnn2c1OCC(F)C2 c1(OC)cc(NC(=O)C=C(C)C(C)(C)C)ccc1-c1ccc(O)cc1 C1(C(=O)NC2CN(C(C=NCCCC=CC)=O)CC2C)CCCCN1S(N)(=O)=O C1(CNC(c2n(C)ncc2)=O)CN(C(c2ccc[nH]2)=O)CCC12CCOC2 C1(C(=O)NC(CSC)(C)C(=O)N2CC(C3CCCO3)C2)CCC(C)(C)CC1 c1(C(N2CC3C(NC(c4ccc(NC)cn4)=O)(CC3)C2)=O)ncc2[nH]ncc2n1 c1(C(=O)OCC)cnc(CNCCN2CCCC2c2cccnc2)s1 CC1=C(C)CC(C)(C(N2C3CCC2C(CNC(C2CCCC(O)C2)=O)C3)=O)CC1 C(=O)(CCCCNC(=O)OC(C)(C)C)NCCc1onc(CSC)n1 c1(C(=O)NCCc2cccs2)csc(=NCC(O)c2ccccc2)[nH]1 C(=O)(C(=O)C(C)(C)C)NC1CC(O)(CNC(COCc2cc(C)on2)=O)C1 c1(C(=O)NCC2CN(C(C(CC=CC)CC)=O)C2)cc(F)cc(F)c1N c1(C(=O)NC2(COC)CCN(C(=O)C(F)(F)CO)CC2)ccc2c(c1)OCCC2 CC(O)C(C(=O)N1CCC(COC(C)(C)C)C1)NCCn1cnc(C(=O)NC)n1 C1(C(F)F)(OC)CCCN(c2ncnc(NC(C)CCCCCO)c2C)C1 c1(CN2CC3(C(NC(c4ccc(O)nc4)=O)C3)C2)cc2ncccc2[nH]1 C1(CO)(CC2C(N(C)C(=O)NC(=O)C=CC(=O)N(C)C)CCC2)CC(C)(C)C1 C1(COC)(CNc2cc(NC3CCS(=O)(=O)C3)ncn2)CCOCC1 CCCCCC(F)C(=O)NC(CC(=O)N1CC(OC)CC(C)C1)C(F)F c1(C(=O)NCC2N(C(c3ccc(SCC)cc3)=O)CCC2)cnc(O)c(F)c1 N1(C(C2=CC(C)(C)C2)=O)CC2(CCCN(C(C3Cc4ccncc4C3)=O)C2)C1 C1(CN(C(c2cnc(C)[nH]2)=O)CC)CCCN(C(c2cnn(CC(F)F)n2)=O)C1 c1(CC)ccc(C=CC(N2CCC(CNC(C3CC(C)N(C)C3)=O)C2)=O)cc1 C1(C)(C(=O)NC(c2cnc[nH]2)C)CCN(c2nccc(Br)n2)C1 C(C)(N=c1cc[nH]c(-c2nccs2)n1)c1c(Br)ccc(C)c1 C1(CC(=O)NC(CN(C(C=C(C)C(C)(C)C)=O)C)C)CCCCC12CC2 N1(Cc2n(C(C)C)ncc2)CCOC(C(=O)NCc2nc(Br)cn2C)C1 Cc1cc(C)c(OCCN(C)C(=O)NC(C)CCCC(C)C)c(C)c1 CC(=O)CCC(=O)N1CCN(C2CCCN(C(c3ncccc3C)=O)C2)CC1 C1(C(CC)(C)C)CCC(CC(=O)N(C(C)CCNC(=O)C(CSC)OC)C)CC1 CCCC(C)(CCC)C(=O)NC1CC(C(=O)NCc2cn(C)nc2C)C12CCC2 N1(C(CCCNC(N)=O)=O)CCC(F)(CNC(=O)Cc2cccc(O)c2)CC1 c1(C(N2CC3C(CNC(CC(C=C)CC)=O)(C3)C2)=O)ccc(C)c(OC)c1F CC1CC(C2CN(S(=O)(=O)CCOc3ccccc3C(F)(F)F)C2)=NO1 N1(C(=O)OC)CC(O)CC1C(=O)NCCC(O)CNC(c1cccc(C)c1)=O CCCCCCCC(=O)NCC1(OC)CN(C(c2c[nH]cc(Br)c2=N)=O)C1 C(=O)(C1CCCc2ccnn21)N1CCC(N2CCCS2(=O)=O)C1.C12CC1C(O)C2 c1(C(=O)NC2CCN(C(C3CCSCC3)=O)CC2)coc2cc(O)ccc12 C1(NC(=O)CC2CCCC2O)COCCN(C(c2cnc(C3CC3)[nH]2)=O)C1 C1(CCCNC(C2C(=C)CC2)=O)CCCN1C(c1cnc(O)o1)=O c1(C(=O)NC(C(C)NC(CCC(=C)Cl)=O)(C)C)cccc(Cl)c1OC C1(NC(c2cc(OCC)no2)=O)CN(C(c2ncncc2Cl)=O)CC12CC2 c1(C(=O)NCC2N(C(C(CC)N(C)C)=O)CC(F)C2)cncc2cnccc12 C(=O)(C(C)CNC(C1CCC(=O)N1)=O)N(C(COC)COC)C c1(OC)cc(C(=O)NCC(C)NC(c2cnn3ccsc23)=O)c(F)cc1N C(=O)(CCC1=CCc2ccccc21)NC1CC2(N(C(C=CCCC)=O)C2)C1 C1(N(C(c2ccc(C(C)C)o2)=O)C)CCCCN(C(=O)CCn2cnnn2)C1 c1(CC)ccc(C(=O)NCC2(NC(C3CC(F)(CO)C3)=O)CC2)[nH]1 C(C)(C(=O)NCC1CCC(NC(=O)CCCn2cncn2)C1)(C1CC1)OC CCC(CO)C(=O)N(CC(O)CN(C)C(c1ccc(C(N)=O)o1)=O)C C1(CC=C)(NC(C2OCC2(C)C)=O)CCN(C(=O)COC2CCCOC2)CC1 C=CC(CCC)CC(=O)N(CCC(N1CCCC(CC)(CC)C1)=O)CCO N1(C(C)=O)CCCC(Cc2ccc(NC(=O)CCCSC)cc2)C1.c1(=O)c(=O)[nH]1 c1(C(N2CCC3C(NC(C(C)OCC)=O)C32)=O)n[nH]c2c1CCCC2 C1(NC(C2CCCCS2)=O)CN(C(=O)CCCCC(F)F)CC1C1CC1 c1(C(N(CCNC(CCCOc2cccc(C)c2)=O)C)=O)cnc2scnc2c1 c1(NC(C(C)NC(C=CC(CC)C)=O)=O)cccc(CCF)c1 C1(CN(C(C(CO)OC)=O)C)CCCN(C(c2ncccc2N)=O)C1 c1(C(=O)NCc2ocnc2-c2cn(CC3CCCC3)nn2)ccc2cccnn12 Cc1[nH]c(=N)nc(O)c1C(c1ccc(OCCSc2nn[nH]n2)cc1)(C)C c1(C(N2C(C)(C(N3CC(OCC(=O)NC)C3)=O)CCC2)=O)c(F)cncc1F CCC(N)(C)C(=O)NCc1ccc(SC)o1 C1(NC(Cn2cc(-c3c(Cl)ccc(OC)c3)nn2)=O)CCC2(CC1)COC2 C(=O)(C1OCCc2ccccc21)N1CC(CNC(C2C(C=C)CC2)=O)(COC)C1 C1(C(=O)NC2CCC(C(=O)NC(C)C(C)n3cccn3)C2)(OC)CCOC1 c1(NC(C2N(C(c3cc(C)[nH]c3)=O)CC2)=O)c(Br)cc(Cl)cc1C#N C(=O)(CCC(F)(F)C(F)(F)F)N1CCC2(C(NC(C3CC(=C4CC4)C3)=O)C2)CC1 CC(C)(O)CC(=O)NCC1CC1CNC(c1cnoc1-c1ccccc1)=O C12(C(=O)Nc3cc(C(=O)OC)no3)C3CC1C1C(C(=O)NC4(C)CCCCC4)C3C21 C(=O)(C(O)(C(F)(F)F)c1ccccc1)NC1C(NC(=O)C=C(Cl)Cl)C2CCC1C2 N#Cc1c[nH]c2c(F)c(F)c(F)cc2c1=NC(=O)c1ccc2[nH]ccc2n1 CC(CCCC(=O)NCc1cnns1)NC(c1cn(C)nn1)=O N1(C(c2cc(CO)[nH]n2)=O)CCCC1C=CC(=O)NCC(O)CF C(=O)(C(CO)C(C)(C)C)N(CC(C)C(N1CCC2(CCO2)C1)=O)C C1(CC)NCCC1S(=O)(=O)C(c1ccccc1C)C(C)(C)C N1(CC)CC(NC(=O)C(C)N(C(=O)COC(C)=O)C)C1 c12cc(no1)C(=O)NC2.C(CC(=O)NCCCNC(N)=O)(C1CC1)OC Cc1ccc(NC(c2cccc(C)c2)=O)cc1.C1(CNC(=O)CN(C)C)CCC1CF c1(C(N(CCC(C)NC(=O)CC2CC(C)(C)CO2)C)=O)snc2ccccc12 C1(NC(COCC(C)C)=O)(CO)CCN(C(=O)C(c2cccc(Br)c2)O)C1 Cc1c(CC(=O)NCCC(O)CNC(=O)C(C)NC(C2CCC2)=O)ncn1C CC1CN(C(=O)CC(F)(F)F)CCCN1C(=O)CCn1ccc2ccccc12 CC1(C)CC1(CO)CNC(C1CCN1C(=O)C(O)CN1CCCC1)=O C1(C(=O)NC(CC#C)CC#C)CN(C(=O)CC2CCCCC2O)C(C)(C)C1 N1(c2nc(NC(c3nnc(SC)s3)=O)c(C)s2)CCS(=O)(=O)CC1 C(=O)(CCC(CF)CF)N1CCCCC(CCC(=O)N(C2CC(C)CC(C)C2)C)C1 C1(NC(c2c(OC)nsc2)=O)CCC(C)(NC(=O)CN2CCCOC2=O)CC1 O=C1CCCC(C(=O)OCC2CCCSC2)C1 Cc1cc(CNC2CC(C(=O)Nc3cnc(O)c(C)c3)C2)c(O)c(C)c1 c1(OCC)ccccc1C(=O)NC1C2CN(C(c3ccc(C(F)(F)F)o3)=O)CC12 c1(C2N(OCCOCCOC)CCOC2)ccc(F)c(F)c1 c1(-n2c(Cn3ccc(C)n3)nc(-c3ccc(Cl)s3)n2)cc(Cl)cc(Cl)c1 C1(CC(=O)NC2CC(C(C)NC(C3(CC4CC4)CC3)=O)C2)CCC(=O)CC1 n1(CC)cnc2c(N(C)Cc3cccn3C)nc(=NC(C)c3cn(C)cn3)[nH]c12 CS(=O)(=O)C1CC(C(N2CCN(C(=O)C3=CCC3)C(C3CCC3)C2)=O)C1 C(=O)(C1=CS(=O)(=O)CCC1)N1C(C)CCC(NC(C2(COC)CCCO2)=O)C1 N1(C(CC2(OCC)CCC2)=O)CCC(C)(NC(=O)C(=O)N(C)C)C1 c1(OC(c2cnn(C)c2Br)C(=O)OC)ccc(N(C)CC2(CO)CC2)cc1 N1(C(C(c2ccc(N(C)C)nc2)C)=O)CCN(C(=O)C2=COCCC2)C(C)C1 CC1CNC(=O)CN1C(=O)C(Cn1cncn1)NC(c1cnnc(O)c1)=O C1(CNC(c2ccc(O)cc2O)=O)CN(c2ccnc(CO)n2)CCC1(F)F C(CC(O)C(=O)N1CCC(F)(C(=O)N(C(C)C)CC2CCCO2)C1)SC C1(C(N2C(CCNC(C(N(C)C)C3CC3)=O)CCC2)=O)CCCCC(=O)N1 c1(C(=O)NCC2CC(NC(c3cc(C(C)(C)C)n[nH]3)=O)C2)ccn2cccc2c1 N1(C(C2C(C(C)C)C2)=O)CCC(F)(C(=O)NC2C(O)CC2O)CC1 C(CCN=c1nc(N2CCC3(CC2)CS(=O)(=O)C3)cc(C)[nH]1)NS(NC)(=O)=O N1(CC(=O)NCC(CC)NC(=O)C(C(C)C)c2cccnc2)CCC(=O)NC1=O c1(C(=O)NC2CN(C(c3cc(C(C)=O)sc3)=O)CC2C)ccn2nncc2c1 C1(CC(=O)NC(CO)C(=O)NCCN2CCCOC2)CCCOCC1 C1(CNC(c2c(CC)oc(C)c2)=O)COCCN(C(=O)CC2CCOC2=O)C1 CN1CC(F)CC1C(=O)NCC1COCCN1C(c1cnc(CC(C)(C)C)s1)=O n1(CC(N2CC(C)(NC(c3ccc(C(C)=O)o3)=O)C2)=O)ncc2ncccc12 N1(C(=O)OC(C)(C)C)CCC(NC2CCC2Sc2ccccc2)C1 C(C(=O)N1CCC(C(=O)NCc2cnn(C)c2)O1)N(CCC)C c1(CCn2c(C(c3cnc[nH]3)OC(N(C)C)=O)nnn2)ccc(N(C)C)cc1 c1(NC(CC(=O)OC)C2CCC2)cc(C)nn1CCCOC C1(NC(=O)Cc2ccc(O)nc2)CC2CC1CN(C(c1ccc(Br)o1)=O)C2 C1(N(C(C)CO)C(c2cccc(OC)c2F)=O)CCC2(CCNCC2)CC1 C=CCCC(C(=O)Nc1cccc(OCC)c1)NC(C1CCCCCC1)=O CCCCC(O)C(=O)N(C(C)CCNC(c1ncncc1C)=O)C CC(C(F)(F)F)NC(=O)C(c1ccco1)NC(=O)CCC1CCCC1 C(=O)(CCN=C(NCC(C)SC)N1CCC(F)(CSc2ccccc2)CC1)NC c1(C(N(CCCNC(COCCOC)=O)C2CC2)=O)cc(Br)nn1C N1(C(C(C)(C)NC(=O)OC)=O)CCCC(C)(C(=O)NC2(C)CC=CC2)C1 c12nc(Br)cnc1NC2=O.n1(C(C(=O)OC)C)cc(C(C)N(C)C)nn1 N1(C(C(C)CC(N)=O)=O)CC(Nc2ncc(C(C)(C)O)cn2)C2(CCOCC2)C1 Cn1ccc(C(=O)NC2(C)CCCN(C(C3CC4CC4C3)=O)C2)cc1=O c1(CN2CCCC(NC(C3ON=C(C)C3)=O)C2)nc(O)[nH]c(=N)n1 CCCC(CCCNC(c1cccc(C(F)F)c1)=O)NC(c1nc(O)sc1C)=O Cc1nn(CC(N2CC(NC(c3cccs3)=O)CCC2C)=O)c(C)c1C#N N1(C(CC(C=C)CCC)=O)C2CCCC1CN(C(=O)C=Cc1cnc(C)s1)C2 C#CC1CN(C(=O)C=CCN(C)C(C2(C)COC(=O)N2)=O)CC1O CCC(O)CCN=c1[nH]c(=NCCNC(=O)N(C)C)[nH]c2ccccc12 c1(OC)ccc(Cl)c(CC(N2CC(O)(CCNC(=O)C(F)=CC3CC3)C2)=O)c1 NC(Cc1nc(C2CCCC2)no1)C(=O)N1CCC(O)C1 CCCC(CNC(=O)CN1C(=O)CCCC1=O)C(=O)Nc1cnc(C(C)C)nc1 C1(CN(C(COC(C)C)=O)C)CCCCN1C(c1cccc(-n2cccn2)c1)=O c1(C(=O)NC2CCN(C(C(C)CCN(C)C)=O)CC2)cc(N)c(F)cn1 c1(C2(F)C(C(N3CC(NC(=O)C(F)(F)C4CCCC4)C3)=O)C2)ccccc1 c1(NC(=O)NC2CN(C(C(C)(C(C)C)NC(C)=O)=O)C2)cc(Cl)cc2c1OCC2 N1(C(c2c(C)cn(C)c2)=O)CC2CN(C(c3c(Cl)n[nH]c3C)=O)CC2(C)C1 CC1(C)CCC(C(=O)NCCC(O)CCO)CN1C(c1cnc(S)nc1)=O c1(C(N2CC(CNC(C(NOC)=O)=O)OCC2)=O)ccc(C(N)=O)cc1C CC1C(NC(=O)C(=O)N(CC(O)C2CC2)C)CCN1Cc1ccccc1 C1(CC=C)(NC(C2CCOCC2)=O)CCCN(C(C23COC(CF)(C2)C3)=O)C1 c1(CC(=O)NCC(CC)N(C)C(c2cnsn2)=O)cc(F)cc2c1OCOC2 N1(C(CCC2CC(NC(CCC3N(C)CCC3)=O)C2)=O)Cc2ccncc2C1 c1(C(=O)NCC(C2CCC2)NC(c2nn(C)c(O)c2)=O)cc(F)cc(F)c1 N1(C(C(CSC)OC)=O)CCCC(C(=O)NCc2nc(C)ns2)C1 N1(C(C2CCC(CC)C2)=O)CCC(C(C)(C)NC(C23CC(C)C2C3)=O)CC1 Cc1cc(C(=O)NC(c2nocc2C(=O)NCC2(O)CCOC2)C)cc(C#N)c1 C1(C(N(C(C)C)CCc2ccccc2)=O)CCn2ccnc2C1 c1(C(N2CCC(CC)(NC(C3CNC(=O)N3)=O)CC2)=O)cc(F)c(F)cc1N N1(CC=C)CCC(N(C(c2nn(C)cc2Cl)C(=O)NC(C)(C)C)C)C1=O C(c1cccc(Cl)c1)=CC(=O)NCC(C1CCCC1)NC(CSC)=O C1(SC)CN(C(=O)NCc2ccc(F)cc2)CC1n1cc(CC(O)C(C)(C)C)nn1 N1(C(CC(CC)NC(=O)CCc2nccn2C)=O)CCOCC(O)C1 c1(C(=O)NCCC2=CCN(C(c3cc(C)[nH]n3)=O)CC2)cnn2c1CC(C)CC2 C1(CC(=O)NCCCOCC)CCCN1Cc1cnc(C)o1 c12ccc(nc1)NC1(C)CCN(C1)C2=O.c1(C2(C=O)CC2)ccccc1Cl.CO CC1(C)CC(C(N2CC3C(C(N)=O)C3C2)=O)(CO)C1.N12CCOCC1C2=O N1(Cc2ccc(CC)s2)CC2CCN(C(c3cc4cccnc4s3)=O)C2C1 c1(C(c2nn[nH]n2)NC2(CC)CCC2)cccc(NC)c1C N1(NC(C(C2(O)CN(C(c3ccc(CC)o3)=O)C2)F)=O)CCC(O)(C(C)C)CC1 N1(C(C2C(C(C)O)C2)=O)CCCC(C)(C)C1CNC(c1ncnc2ccsc12)=O C(C(F)(F)C(=O)NC1CC(NC(c2cncnc2-c2cccs2)=O)C1)OC C1(C(=O)NC2CCC(NC(CCOCC(C)C)=O)C2)CCc2nc(=N)[nH]cc2C1 CC1CCN(CC(=O)NCCn2cc(C(=O)NCC=C3CCOCC3)nn2)C1 N1(C(C2(CC=C)CC=CC2)=O)CCC2CN(C(=O)C(C)(Cl)Cl)CCC2C1 N1(C(C2CC2)=O)CCN(C2CN(C(N)=O)C2)CC1.C12CN(C1)C2=O.CCSCC S(=O)(=O)(c1cccnc1)NCC(=O)N(C)CC1CN(C(C(CCC)O)=O)C1 N1(C(=O)C(O)CC(F)(F)F)CC2CCC(C1CO)N2C(c1ncc[nH]c1=O)=O Cc1ccccc1CNc1cc(N2CCCC(C3CCCCO3)C2)ncn1 CC1CCC(C(N2CCSCC2CCNC(=O)CC2CCC(C)(C)C2)=O)CC1 c1(Nc2cnc(O)nc2O)nccc(=NC2CC(N3CCCCC3)C2)[nH]1 [N-]=[N+]=NCCCC(=O)N1CCCOC(CNC(=O)CCc2ccsc2)C1 C(=O)(C1=C(C)CCCC1(C)C)N1CC(C)CC(NC(C(CCC)OCC)=O)C1 c1(C(N(C)CC2N(C(CNC(=O)NC)=O)CCC2)=O)ccc(Cl)nc1N N1(C(C(c2cncnc2)C)=O)CC(N(C(=O)C2=CC(C)C2)C)C2(CC2)C1 N1(C(c2ccc(Cl)c(Cl)c2Cl)=O)CCOC2(CCN(C(C3CC3(F)F)=O)C2)C1 C1(CC(=O)N(CC(C)(C)NC(CCOCCC(C)C)=O)C)(CC(C)C)CCCC1 c1(OC)ccc(Cl)c(CN2CCC(NC(C3Cc4nccn4C3)=O)C2)c1F N1(C(CCSC)=O)CCC2(CCCC2C(=O)Nc2ccc(F)c(Br)c2)C1 c1(NC(C2C=CC(NCc3ccc(C=O)s3)C2)=O)cc(Br)c([N+](=O)[O-])cn1 N1(C(CC(C(F)(F)F)NC(CNC(C(CC)C)=O)=O)=O)C2CCCC1CN(C)C2 C1(CNC(C(CC=CCC)C)=O)(CO)CCN(C(=O)COCc2nc[nH]n2)CC1 c1(CC)cc(C(=O)NCC2CN(C)CCN2C(c2cocc2C)=O)c(C)nn1 C(CC(C)C(=O)N1CC(C(N)=O)(CNC(=O)CCN(C)CC)C1)=CC N1(C(c2c(OC)scc2)=O)CCCCCC1C(=O)NCc1cnc[nH]1 c1(CC)ccc(N)c(C(N2CC(NC(=O)CCC(C)SC)C(SC)C2)=O)c1 c1(-n2cc(C(C3N(C(C(=O)N(C)C)=O)CCC3)C3CC3)nn2)c(F)cncc1F S(=O)(=O)(c1cc(Br)c(C)cc1F)NC(c1ccc(OC)cc1)CCO N1(c2cc(CC(C)C)ncn2)CCC2(CC1)C(NC(=O)C1=COCC1)CS2(=O)=O Cn1ncc(Cl)c1C(=O)Nc1cnn(Cc2ccccc2Cl)c1 c1(OC)ccc(N=c2scc(-c3ccc(Br)o3)n2C(C)(C2CC2)OC)cc1C C(CC)(CCCC(=O)NC(c1ccccc1)C)NC(c1c(CC)n(C)nc1)=O c1(NCCCOCC)[nH]c(=NCC2(CO)CC(C)(C)C2)nc2scnc12 CC1(NC(c2csc(C3CC3)n2)=O)CC(NC(=O)CCn2cc(Cl)cn2)C1 Cc1nn(C)c(C)c1C(=O)NCC1CN(C(=O)CCc2cncnc2)CCN1C N1(C(C(CCC)O)=O)CCN(C(c2cc3cscc3s2)=O)C(CCCC)C1 C(CS(=O)(=O)CC(=O)N1CCCC(C(=O)NCc2ccc(Cl)cn2)CC1)OC N1(C(CC(=O)OC)=O)CCN(C(=O)CC(C)N(C)C)CC(O)C1 N1(C(C)=O)CCC2(CCCN(C(=O)Nc3cc(-c4ccncc4C)ccn3)C2)C1 C(=O)(C(C(=O)NC(C)(CNC(=O)C(c1ccccc1C)(F)F)CO)OC)OC C1(NC(C(NOC)=O)=O)CC2(CCN(C(=O)CC3CCC(C)(C)CO3)CC2)C1 C1(N(C(CCOCCOCC)=O)CC)CCCN(C(=O)Cc2ccc(C)s2)C1 C1(C)(NC(c2cc(OC)ncn2)=O)CCCCC1C(=O)NC(c1cccs1)(C)C c1(C(N2CCC3CC23C(=O)Nc2cccnc2)=O)ccc2cc[nH]c2n1 C1(CNC(C2C(=C)C2)=O)CC2CCC1N(C(=O)CCCCC(F)F)C2 Nc1ccc(C(N2CCC(NC(C3(C=C)CC3)=O)C(O)C2)=O)nc1N N1(C(COC(CC)CC)=O)CC(NC(C2(C)CCN(C)CC2)=O)CC(C)(C)C1 N1(C(CCSC)=O)CCN(C2CCCN(C(c3coc(Br)n3)=O)C2)C(=O)C1 C1(NC(C(CC)CCOC)=O)CCC2CN(C(c3cc(C)ccn3)=O)CCC2C1 C(=O)(C(C)(C)C(F)F)NCCC1CCN(C(c2c(CC)c[nH]n2)=O)C1 N1(C(C(CC)C)=O)CC(NC(c2cc(F)c[nH]2)=O)C(O)C1 c1(OC)ccncc1C(=O)NCC(O)CNC(C1(CC2CC2)CCC1)=O c1(C(=O)NC2C(C)CN(C(C3CCCSC3)=O)C2)cc(O)nc2[nH]c(=N)ccc12 n1(CC#C)cccc1C(=O)N(CCCNC(=O)C(F)(F)C1CC1)C(C)C C1(NC(CC(COC)COC)=O)CC2(CO1)CN(C(=O)OC(C)(C)C)C2 C(=O)(C(C(=O)N1CC(NC(=O)CCCc2ccccn2)C(O)C1)C(C)C)OCC C(C(C(=O)N1CCC(CNC(=O)C(C)(C)c2ccno2)C1)C(C)(C)C)OCC=C S(=O)(=O)(c1c[nH]c(=N)c(C)c1)Nc1n[nH]c(C)c1C(F)(F)F C(=O)(C(O)C(C)(C)C)N1CCC(NC(CC2CCN(C(C)=O)CC2)=O)(CO)C1 C(N=c1nc2c(cnn2C)c(NC2CCC2C(N)=O)[nH]1)C1(C)N(C)S(=O)(=O)CC1 c1(-n2c(N3CCC(C(=O)OCC)C3C)nnn2)ccc(C)c(C)c1 c1(CC)cc(F)c(C(N2CCC(CN(C(=O)CC(C)COC)CC)C2)=O)c(F)c1 Nc1cc(C(=O)NCC2CCCN(C(c3cc4sccc4[nH]3)=O)C2)nc(O)c1 C1(CC)(CC)CCCN(C(=NCc2ccccc2CO)NCC2CCCO2)C1 c1(C(=O)OC)ccc2c(c1)CCC2NC(=O)C(=O)N(C)Cc1noc(C)n1 c1(C(CCN(c2ccc(F)cc2)CC)=O)cc(OC)c(OC(C)=O)cc1F c1(CNC(C=CC(C)(C)C)=O)ccc2c(c1)CN(C(c1cc(C#N)cs1)=O)C2 c1(OC(C)=O)cccc(SCC(N2CCC(N(C(=O)CC(C)(C)C)C)CC2)=O)c1 N1(C(C2N(C(c3c(OC)nsc3)=O)CCC2O)=O)CCCC2(C=CCO2)C1 c1(CNC(CN(CCCCCC)C)=O)cccc(CNC(C2CC(C)CO2)=O)c1 N1(C(COc2ccc(OC)cc2)=O)CC2(CCCN(C(=O)C#CC(C)(C)C)C2)C1 c1(OC)cc(F)c(CN2C3CN(Cc4ccc(F)c(Cl)c4F)CC23)c(F)c1 c1(OC)ccc(C(N2CC(NC(c3sc(F)cc3C)=O)CC2C)=O)c(Cl)c1 CCCCC(CC)C(=O)NCCCCN(C(=O)C(c1cccs1)=CC(C)(C)C)C CC1CCCC(CCNC(C2CN(C(=O)Cc3ccc[nH]3)C2)=O)C1 N1(C(C)=O)CCC(OCCC2COCCO2)C1.C1(=O)C=CC[NH+]([O-])CC1=O.C1CC1 C(=O)(C(F)C(C)C(F)(F)F)NC(CN(C(=O)Cc1c(O)ncnc1O)CC)C CC1(C)CN(C(=O)CC(C)(C)NC(=O)COC2CCC2)CC(C)(C)O1 c1(CNC(c2cnc(CCC)s2)=O)ncccc1CNC(C1CC(SC)C1)=O N1(C(C=C(C)C(C)(C)C)=O)CC2CCCC(Nc3ncccc3[N+](=O)[O-])C2C1 CC1(C)CCCC(CC(N2CCC(O)(CNC(=O)CN3CCC(O)CC3)C2)=O)O1 c1(OC)cc(N2CCC(N(C)C(c3cc(C)ccc3C)=O)CC2)ccc1Br c1(C(=O)NC(C2CCCN2C(c2ccc(C(N)=O)o2)=O)C)ccc([N+](=O)[O-])nc1 CC1CCN(S(=O)(=O)NCC(=O)NC(C)CNC(c2ccccc2)=O)CC1 C1(C(N2C(C)(C)C(NC(=O)C(F)(F)C(F)(F)F)CC2)=O)CCCC2CCCCC12 Cc1cc(CN2CC(NC(=O)Cc3cccc(Br)c3)CC(C)C2)cc(F)c1 c1(OC(C)C(N2CCC(C)(C(=O)NCc3ccccn3)C2)=O)ccc(Cl)nc1 c1(C(C)C)ccc(N)c(C(=O)NCCC(C)(C)NC(=O)Cc2cnccn2)c1 c1(C(N2C(C)(CO)COCC2)C(=O)NCCC2CCCO2)ccc2c(c1)COCC2 c1(CC(=O)NC2(C(N(C(C)COC)CC=C)=O)CC2C)c(C)n[nH]c1C C1(CC(=O)OC)C2CCC(C2)N1C(C1CCCCC1)C(=O)NCCC(=O)N(C)C N1(CC#C)CCCC1COC(=O)CCC1CC1CC1CC1 C(=O)(C1=CS(=O)CCC1)N(C1CCN(C(=O)Cc2csc(Cl)c2)CC1)CC(C)C C(=O)(C1=CC2CCCC12)Nc1cccc(NC(COCC2CCC(C)(C)O2)=O)c1 C1(C(N2CC(O)(CNC(C(CCC)N(C)C)=O)C2)=O)CCOCC1(C)C C1(C(=O)NCCOCC(N)=O)(NC(C(C)OCCOC)=O)CCOCC1 S(=O)(=O)(c1ccc(Br)cc1F)N1CCC2CN(S(CC(=O)OC)(=O)=O)CC2C1 C(C(C)(COC)C(=O)NCC(O)C(=O)N(C)CC1CCC1)OC N1(C(C(Cc2cnc[nH]2)NC(c2n(CC)ccn2)=O)=O)CCC(C)C(F)(F)C1 c1(NC(C2(C)CCN(C(c3ccc(Cl)nc3)=O)CC2)=O)cc(Cl)c(Cl)cc1Br C(=O)(C(CCF)NC(c1c[nH]c(C#N)c1)=O)N(C(C)C)C CCCCCCC(C)C(=O)NCC(C)(CC)C(=O)N1CC(C(N)=O)C(CCC)C1 C(CCC(=O)NC(c1ncn(C)n1)C)(C(C)C)NC(Cc1cc(C)on1)=O C1(C(=O)NCCC=C)COCCN(C(=O)NC)C1.C(=O)(CCO)C1CC1.C1CO1 CN1CCCN(C(C23CCC2CN(C(=O)C(C)(F)c2ccon2)C3)=O)CCC1 Cc1ccc(SCC(N2CC(CNC(=O)CC3CC3)C(C)C2)=O)cc1 C1(OC)CCC2CN(C(=O)CC3CCN(C4CC(F)(F)C(=O)N4)C3)CC12 C#CCC(O)C(=O)NCC1(C)CCCN1C(c1nnn(CC(N)=O)c1C)=O CCC(CC)CCCC(=O)N1CCC(C(C)(C)NC(c2nn(C)c(Cl)c2Cl)=O)C1 N=C1NC(=O)C(CC(=O)NCC2(F)CC(NC(=O)CCC(F)F)C2)S1 c1(CN2C(C)CC(c3c(C)cccc3)C2)cc(F)cc(I)c1C N1(C(CC(C)N(C(CC=CC)=O)C)=O)CC(C)C(C2CC2)C1 Cc1ccnc(-n2cc(C(N3CCCC3CNC(=O)CC3CC=CC3)=O)cn2)c1 c1(C(=O)OCC)cc(COC(C)(C)C)ccc1[N+](=O)[O-].C1C(=O)N1C C1(NC(C(C2CCC2)OC)=O)CC2CC(NC(C3(CC(C)C)CCC3)=O)C2C1 c1(C(C(=O)NC(C(=O)OC)Cn2cccn2)O)ccc(Cl)cc1F c1(C(=O)NCC2(F)CC(NC(c3cncc(CO)c3)=O)C2)ccc2occc2n1 c1(C(=O)NC2(CF)CCN(C(C3C(C(C)O)C3)=O)C2)c2c(nn1C)CCCC2 Cc1ccc(N)c(C(=O)N(C2CCN(C(C3(C4CCC4)CC3)=O)C2)C)c1F C(=O)(C1CCCc2n[nH]cc21)NC(CCCC)CNC(=O)Cn1ncnn1 C(=O)(C(CCCC=C)NC(C1CCCCCN1C)=O)NCCCCC#C C1(NC(c2cn(CCOC)nc2)=O)CCN(C(=O)COc2ccc(O)cc2)C12CC2 CCCC(CC)C(=O)N1CCN(C(=O)CN(c2cnccn2)C)C2CC12 C1(CC)C(=O)N1.C1(C)C=CC(=O)N1.C(C(=O)N(C)C)OCCSC N1(C(c2nccc(C)c2N)=O)CCC(C2CCN(C(=O)CNS(N)(=O)=O)C2)C1 Cc1nc(C(=O)NCCC2(CNC(c3cc(F)c[nH]3)=O)CC2)ccc1[N+](=O)[O-] Cc1c(C(=O)NC2CC(NC(=O)Cc3ccc(C4CCC4)cc3)C2)cccc1F C(=O)(C1=C(C)CCC1)NC(CC)CNC(C1CCCN(C)C1)=O c1(CC(=O)N(CC(CC)NC(=O)CC2CN3CCN2CC3)C)cccc(C)c1F CCCCS(=O)(=O)CC(=O)NC1CCCN(C(=O)CC2CCCCC2O)C1 C1(CNC(C2CC2F)=O)CN(C(c2ncncc2Cl)=O)C2(CCC2)C1 N1(C(C2(COC)CC2)=O)CCC2(CC(C(=O)Nc3cnn4cccnc34)=NO2)C1 c1(OC)ccn2ncc(C(=O)NCCCN(C)Cc3ccc(C#N)s3)c2c1 N(C1CCc2c(Cl)cccc21)C(=O)Nc1cccc(C)c1[N+](=O)[O-] S(=O)(=O)(c1cccc(N2CC(C)OC3(CCCC3)C2)n1)NC1(CC)CCC1 c1(NC(c2ccc(C#C)s2)=O)ccc(Cl)cc1C(=O)OC.C12(CCCC1)NC2 N1(C(c2c(C)cc(N)cn2)=O)CCCN(C(=O)C(C)Sc2ccccc2)CC1C c1(C(=O)NCCC2CN(C(C3CC(SC)C3)=O)CC(C)O2)cc2sccc2[nH]1 c1(SCC)ncc(C(=O)NCCCCCO)cn1.N12CCNC(C1)C2=O n1(CC(=O)NC2CCN(C(COCCC)=O)C2)c(C)cc(O)cc1=O N1(C(c2n(C)c(Br)nc2)=O)CC(NC(=O)C=CCN2CCCC2)C(C2CC2)C1 CC1(C)CC(OCC(N2CC(n3cc(C4(O)CCOC4)nn3)C2)=O)C1C(F)(F)F c1(NC(CC2(C)CN(c3ncc(OC)cn3)C2)=O)ccc2nncn2c1 C=CC1(C2(C(=O)NC(CNC(=O)CCCCC(C)C)C3CC3)CCC2)CCC1 c1(SCC)cnc(N2CCOC(CNC(c3cnnn3C)=O)C2)nc1 Cc1nnc(NC(=O)NC(CC(C)C)c2nn[nH]n2)o1 c1(C(N2C(CNC(CSCC#C)=O)C(C)CC2)=O)ccc(C(F)F)nc1O C(=O)(CC1=CCN(C(=O)C(c2cnn(C)c2)C)CC1)N1C(CC(C)C)COCC1 c1(NC(c2noc(NS(C)(=O)=O)n2)=O)cc(S(=O)(=O)C(F)(F)F)ccc1F CN1CCC(C(=O)N(c2ccccc2)C2CCNC2)CC1.c12cncnc1OC2 Cc1cnc(C(=O)NC(C2CCN(C(c3nn(C)c(C)c3N)=O)C2)C)cc1Cl c1(CCSC(F)F)nc2c(c(=NCCc3nc(O)n[nH]3)[nH]1)CCC2 c1(NC(=O)OC)cccc(NC(c2cnc(NC)cn2)=O)c1C.N12CC(C1)C2=O C1(C(C)O)COc2ccccc2O1.C=C(C)CC(C)C(=O)Oc1ccc(CO)cc1 c1(C(N2C(CNC(c3ccc(C(C)C)cc3)=O)CC3CC32)=O)cc(F)cc(F)c1 Cc1cc(NC(c2c(C)noc2C)=O)ccc1NC(c1cc(C)c(Br)o1)=O C(CCC(=O)NCc1nocc1C(=O)NCC(O)C1CC1)N(C(C)=O)C N1(C(c2c[nH]c(=N)s2)=O)CCN(c2ccccc2CNC(c2ccns2)=O)CC1 Cc1cc(C(=O)NC2C3CN(C(=O)Cc4cccs4)CC23)cc(C)n1 S(=O)(=O)(c1csc2ccccc12)Nc1nn[nH]n1.CC1(C)C2CN3C(C12)C3=O CC1(C)CN(C(c2ccccc2Cl)=O)CC(CNC(=O)CSCC#N)O1 c1(OCC)ccc(C(=O)NC2CNCC(OC(C)(C)C)C2)n2nc(C)nc12 c1(C(=O)NCCC(CCNC(C(C)SC)=O)C)ccn2ncccc12 C1(C(=O)NC2CC(C)N(C(=O)CCCn3cccn3)C2)CCCC2CCCCC12 C(C(C)(C)C(N)=O)NC(C(C)OCC)=O.C1CC(=O)N(C)CCO1 C1(NC(c2c(CCC)nns2)=O)CN(C(=O)C(CC)n2cncn2)CCC1CO C1(CNC(CN(C(=O)C2=CCSC2)CC(C)C)=O)CN(C(C)C)C(=O)O1 N1(C(c2cn(CCO)nn2)C(=O)NCCC)CCCC(O)(CCOC)C1 c1(C(=O)NCC2CC(C)(C)N(C(=O)Cc3cccs3)C2)cccc2cnccc12 c1(C(=O)NC(C)C(C)NC(c2ccc(C(N)=O)o2)=O)noc2c1CCCC2 N1(C(c2n(C)[nH]c(=N)c2)=O)CCCCC(C2CN(C(=O)CSc3nncs3)C2)C1 N1(C(C(C)Oc2ccc(CO)cc2)=O)CCC(NC(c2cc(F)cs2)=O)C(O)C1 C1(CN(C(c2c(C)nc[nH]2)=O)C)C2CN(C(=O)CC(C)c3ccccc3)CC12 N#Cc1cnc(NC2CCN(C(=O)CCC3CCOCC3)C2)c2sccc12 C1(CCNC(C2CC(C(=O)OC)C2(C)C)=O)CN(C(c2cnsn2)=O)CCCO1 N1(C(C(N(C(COC(CC)C)=O)C)C2CC2)=O)CCC12CCN(C)C2 c1(C(=O)NCC(CNC(CCN(C(CC)CC)C)=O)C)ccc(=O)n2c1CCC2 CC1CCC(C(=O)NOCCn2cc(Cl)cn2)CN1C(c1ccn(C(F)F)n1)=O c1(OC)c(C(=O)NC2CC(n3cc(C4CCCC4)nn3)C2)cccc1Cl C1(CC(C)C)CCCCN1C(=O)C(CN(C)C)NC(C1OCCC1C(C)C)=O c1(CNC(c2ncc[nH]2)=O)noc(C(F)(F)F)n1 C1(NC(Cc2ccc(OC)cn2)=O)CCCCN(C(=O)C(=O)NC2CC2)C1 CC(C)C(C#N)C(=O)N1CCC(NC(c2ccc(C3CC3)c(F)c2)=O)C1 Cc1c(C(=O)NC(CNC(=O)C2=CCCS2)C(C)(C)C)ccn1C(C)C c1(C(=O)NC(CC)(C)CNC(=O)C=CC(F)(F)F)ccc(Cl)cc1O C1(C2CCN(C(c3ccn(C(C)(C)C)n3)=O)C2)(NC(CCC(C)(F)F)=O)CC1 C12(C(N3CC(C)C(CNC(=O)C#CC4(C)COC4)CC3)=O)CC3CC(CC(C3)O1)C2 CCC(F)(F)C(=O)N(CCNC(C1CC(C)C1(C)C)=O)C1CC1 Cc1cc(C(=O)N(CCCCC(=O)N2CCCC(F)C2)C)c(C)cn1 Cc1cc(C(=O)N(C2CCN(C(C3CC(Cl)(Cl)C3)=O)C2)CCO)c2c(c1)CCO2 C1(NC(C(CC(=O)OC)C)=O)CC(O)(C2CCN(C(=O)Cc3cc[nH]n3)CC2)C1 CC(CCNC1CCCCN(C(=O)OC(C)(C)C)C1)N=c1ccnc(N(C)C)[nH]1 Cn1cc2c(C(=O)NCC3(NC(c4ccc([N+](=O)[O-])cn4)=O)CCC3)cccc2n1 N1(C(=O)C(C2CCN(C(c3csc(O)n3)=O)C2)F)CC2CC(O)CC1C2 c1(C(=O)NCC2N(C(Cc3ccc(C)s3)=O)CC(F)C2)cnn2c1NCCC2 c1(NCCSCCOC)cc[n+]([O-])c(F)c1 Cc1ccc(C(C(=O)NC2COC2)N(C2CC3CCC2C3)C)c(C)c1C N1(C(=O)CC2COCCO2)CCC2(CCCN(C(C3CCC4CC34)=O)C2)CC1 c1(C(N(C2CCCCC2NC(c2cnc(C(F)F)cn2)=O)C)=O)ccnnc1O C1(NC(C=C(C)CNC(C2CC3(C2)CC(C)C3)=O)=O)CCc2nn[nH]c2C1 c1(C(=O)NC(CN(C(C#C)=O)C)C)scc(-c2ccccc2)c1-c1ccccc1 CCCCC(=O)NCCCC(=O)NC(c1cscn1)CO N1(C(Cc2ccc(C)cc2)=O)CCC2(CC1)CN(C(=O)C(C)(C)C)CC2C(=O)O C1(CNC(C(c2ccccc2)C)=O)COCCN1C(c1cc(CCO)on1)=O C1(OC2CC(NC=O)C2)CC(F)(CNC(C2C(Br)(C(=O)OC)C2)=O)C1.OC C1(O)(C(CNC(c2cn(CCC)nc2)=O)C)CCN(C(=O)CCC(F)F)C1 N1(C(Cn2ncc(C#N)c2)=O)CC2CCCC1CN(C(=O)CCNC(=O)CO)C2 Cc1cccc2cc(C(=O)NC3CCCCN(C(=O)C=CCF)CC3)nn12 c1(NC(CC2CC(NCn3cc(C(=O)OCC)nn3)C2)=O)cc(COC)cnn1 C(=O)(C(O)CCCc1ccccc1)NC1CC(NC(C(CC)OC)=O)C1 N1(C(CC2CCCC(C)C2)=O)CC2(CCCN(C(=O)COC3(C)CCCC3)C2)C1 CC1CCC(C(=O)Nc2ccc(-n3cccn3)c(F)c2)C(=O)N1 C1(CC(=O)N(CCCCN(C(=O)CCNC(=O)CO)C)C)CCC(=O)NC1 Cn1cnc(Cl)c1C(N1CCCC(OC(F)F)C1)C(=O)NC1CC1 C#CCCC(C(=O)NCCOC)NC(=O)NC(C)Cc1c(F)cccc1F N1(C(C2CC(N(C)C)C2)=O)CCC2C(C1)C2(F)F.C12(CCC1)CC(=O)N2 Cc1cc(C(N2CCC(C)(CC(=O)N(C)CC3CCCS3)C2)=O)c(C)cn1 c1(C(=O)OC)cc(OC)cc(NC(=O)C(c2ccc(Cl)cc2)CO)c1Cl CC1(C)CCCC1N.c1(C(NOC(=O)Cn2cc(C3CC3)nn2)=O)cccnc1 N1(C(C2=C(C)OCC2)=O)CCC2CC2(C(=O)NCCCCCCF)CC1 N1(C(c2ccc(=O)oc2)=O)CCC2CN(C(c3cocn3)=O)C2C1 c1(CNC2CC(NC(c3cnc(C(C)C)s3)=O)C2)ccc(C(F)(F)F)nc1 N1(C(C)=O)CCN(C(c2cnc(N(C)C)nc2)=O)CC1n1ccnn1 C12(CNC(=O)CN3CCCC3)CCC(CC1)N(C(C1CCC3CCC13)=O)C2 CC1(C)OCC2CC12NC(C1CNC(=O)CN1C(C1CC(=O)CC(=O)N1)=O)=O C1(CNC(C2CCN(C(=O)CSCc3cccnc3)C2)=O)CC2(C1)CC2(F)F C=CCC(C(=O)NC(CC=CC)C(=O)N(CCCCCO)C)C(C)C C(=O)(C1=CCN(C(=O)Cc2cnccc2C)CC1)NC(C1CCCCO1)CC N1(C(C(CC)SC)=O)CCC2(CCCN(C(C3CCC(F)(F)C3)=O)C2)CC1 O=C1CSCC(C(N2CCCCC2CNC(=O)C(O)Cn2cncn2)=O)N1 C12(C(N(CCNC(C(C)OC)=O)CCOC)=O)CCC1CC2 N1(C(c2ccc(CNC(C(C)(C)CO)=O)nc2)=O)CCC(CO)(CO)CC1 C(C(=O)N(C1CN(C)C1)C)(C1CC1)NC(CC1(N(C)C)CC1)=O C(=O)(C(C)(C)CC(C)(C)C)N1CCC(CNC(C(C(CC)CC)F)=O)C(C)(C)C1 CCCCCCCC(=O)N1CCCC(NC(=O)COC2CC=CC2)C1C N1(S(=O)(=O)Cc2cc(Cl)c(Cl)[nH]2)CCCC(n2nccn2)C1 C1(C(=O)NCCC(C(N2CCCC(O)(CO)C2)=O)OC)CCCCC(=O)C1 c1(CNC(CCN(C(=O)Cn2cc(C3CCC3)nn2)CC)=O)ccc(OC)cn1 c1(CC)nc(C)ncc1C(=O)NC(C1CCN(C(=O)C(C2CCOCC2)=O)C1)C C1(CN(C)C(C2CCC(F)(F)C2)=O)CCN(C(=O)CCC2CC2(Cl)Cl)CC1 C1(NC(CNC(N)=O)=O)CCC(NC(=O)CSc2ccccc2)C1 C(c1cncc2ccccc12)=CC(=O)NC(CNC(c1ccc(C)nc1)=O)CO CC1=C(C(=O)N(C)CC2(CNC(C3(C)CC4CC4C3)=O)CC2)CCO1 N1(CC(=C)Br)CCC(C)C(NC(c2coc(C(C)(C)C)n2)=O)C1 N1(C(C(CC=C)N(C)C)=O)CC(NC(c2cc(CO)oc2C)=O)CC1(C)CC C1(OC)(CNC(c2ncccn2)=O)CCN(C(=O)CCSC2CCCC2)C1 c1(C(N(CCN(C(c2cnc(SC)s2)=O)C)C)=O)cnc2onc(C)c2c1 c1(C(N2CCCC2N2CCCC2=O)=O)cccc(-c2cnc[nH]2)c1 C1(C(=O)OCC)CC2(CCN(CC(c3ccc(OC)cc3)C)CC2)CO1 c1(C(N(CC(CC)NC(c2[nH]c(O)nc2C)=O)C)=O)sc(F)cc1Cl n1(CC(=O)NCC(C)N(C(=O)CCN2CCCCC2)C)cc(C2CC2)cn1 N1(C(C2(C)CCCO2)=O)CC2CCC1CN2C(=O)CCOc1cccc(F)c1 C1(NC(C2CSCCS2)=O)CN(C(C2(F)CCCC2)=O)C2CCCCC12 c1(C(=O)NC2(C3N(C(CC(=C=C)C)=O)CC3)CC2)cc2ccccc2n1C CC1C(=O)NC(=O)CN1C(=O)C(C(C)(C)C)NC(=O)Cc1ccon1 N1(C(c2cnn(C(C)C)c2Cl)=O)CCCC2C(CCCN2C(C2CCC2)=O)C1 c1(CC)nc(Cl)nc(N2CCC(CNC(=O)CNC(C3CCCC3)=O)C2)c1C#N C(=O)(C(O)CC(C)(C)C)N(C1CCCN(C(C(C)c2ccco2)=O)CC1)C c1(COC(COCCCC)=O)ccc(Cl)c2cn[nH]c12 CCCCC(O)C(=O)NC1CC=CCC1C(=O)NCC(CC)CC Cc1oc(Cl)nc1C(=O)NCC1CCCC(CNC(=O)CCCn2cccn2)C1 C1(C#N)(c2cn(CCCC(=O)NC(CC=C=C)=O)nn2)CCCCC1.C1CCC1 C(=O)(C(CC1CC1)NC(c1ccsc1OC)=O)N(C)CC C(=O)(C1Cc2ccccc21)NC1(CC=C)CN(C(c2ccc([N+](=O)[O-])cc2)=O)C1 C1(C(=O)NC(C(C)C)C)CCCN(C(c2cn(C3CC3)nn2)=O)CC1 N1(C(c2c(C)coc2)=O)CCN(C(CNC(=O)CCF)C(F)(F)F)CC1 CCC(CC(=O)NCC(C(F)(F)F)OC)NC(c1sncc1C)=O C(=O)(C(C)(C)CF)N(CCCNC(c1ccc(SC2CCOC2=O)cc1)=O)CC C(N=c1[nH]c(=NCC(C)C(C)(F)F)[nH]c2c1CCCC2)c1cccc(OCC)n1 N1(C(C2N(C(C3C4C5CCC(C5)C34)=O)CC3C(C)(C)C32)=O)CCC12CCCSC2 C1(NC(C(CN(CC)CC)F)=O)COC2(C1)CN(C(c1c[nH]c(=N)cc1C)=O)C2 C(c1nnn(C)n1)=CC(N1CC(C(C)NC(c2c(CCCC)ocn2)=O)C1)=O C1(O)(Cn2cc(CCCC=C)nn2)CCCN(C(c2csc(C3CC3)n2)=O)CC1 N1(C(C2C(C)C2)=O)CCCC(C2CCCN(C(c3n[nH]cc3Br)=O)C2)C1 C1(C(N(C2CCC2)CCC)=O)CCN(C(=O)C(C)CC2CCC2)CC1 C1(C=O)CC(C)OC(C)C1.c1(NC)ncccc1C(=O)NCC(C)NC1CC1CF c1(C(N2C(CNC(C(CC)NC(N)=O)=O)C=CC2)=O)sc(COC)nc1C C1(NC(C(CCNC(C(=Cc2ccco2)C)=O)O)=O)CCCN(C)CC1 C1(NC(C2ON=C(C)C2)=O)(CO)CCCN(c2nnc(C)o2)C1 Cc1ccc(OCCCN(C)C(C)=O)cc1.c1(CCO)cnn(-c2ccccc2)c1 N(C(=NCCc1ccc(F)cc1)NC(c1cc(C)on1)C)CCC1(OC)CCC1 C(CCCCNC(C1CCCN1c1ncccn1)=O)N(C(=O)C=Cc1cncs1)C C(=O)(C(CCc1ccccc1)C(C)C)NCC1C(NC(C(C)(C)OCC)=O)CCC1 c1(CC(=O)NCC(C)(CO)NC(C2CC2(Cl)Cl)=O)ccnc(O)c1 C1(CC(=O)NCCCCC2(NC(C3(CO)CCCO3)=O)CC2)CCC(=O)N1 C1(NC(Cn2c(C)csc2=O)=O)CC(C)CN(C(=O)CSc2nncn2C)C1 N1(C(C(C)SCc2ccccn2)=O)CC2(NC(=O)C(c3ccccc3)C)CC1C2 Cc1ccc(C(=O)NC2CCOC(C(=O)N(C)CC3C(C)(C)C3(C)C)C2)c(O)n1 c1(C(=O)NCC(CNC(c2nocc2C2CC2)=O)OC)cc(OC)ccc1F c1(OCCN(C)C(=O)NC2COC(=O)O2)ccc(O)cc1 c1(C(N(C)CC2OCCN(C(CC3CCCN(C)C3)=O)C2)=O)csc([N+](=O)[O-])c1 N1(C(C)=O)CCN(C(C2CSCCN2C(=O)CC=C(Cl)Cl)=O)C(C)C1 C(=O)(C(C)C1=CCCC1)N1C(C(C)NC(c2nccc(OC)c2OC)=O)CCC1 C1(C(=O)NCC(C(=O)NC(CCOC)C)OC)CCCC(=O)N1C C12(NC(c3cc(OC)n[nH]3)=O)CCCC1N(CC(=O)NC1CCC1)CC2 C1(CNC(CN(C(=O)CS(N)(=O)=O)C)=O)CCC(NC(=O)C2CC2)CC1 C1(NC(C2(C=C)CC2)=O)CCCC(NC(c2ccnc(OC(F)F)c2)=O)CC1 N1(CCNC(=O)Nc2cnn(C(C)C)c2Cl)CCc2nc[nH]c2C1c1cccnc1 C12(NC(CC3(C=C)CCC3)=O)CC3CCC(C1C2)N3C(=O)CC1CC=CC1 C1(CCC)(NC(=O)CN2CC3CC3C2)CCN(C(C2CC(F)C(=O)N2)=O)CC1 C1(C(=O)NC2(C)C(C)(C)C2)CCCCC1NC(=O)CC(O)CN(C)C CCCCCCCC(=O)NCC1(F)CC(NC(=O)C=Cc2ccc(OC)cc2)C1 c1(C(=O)NCC2C(OCC)CN(C(CC(=C)C)=O)C2)cnn2c1OCC(C)C2 N1(C(c2c(C)cc(CNC(c3n(CC)ncc3)=O)o2)=O)CCC(F)(F)CC1 c1(C(=O)NCCCCNC(C(C=CCCC)O)=O)cc(C)ncc1Cl Cc1cc(NCCOCC2(S(N)(=O)=O)CC2)cc(C)c1 c1(CC#N)ccccc1NC(=O)C(=O)Nc1ccc(C(F)F)cc1 Cc1ncsc1C=CC(N1CC(NC(c2csc(C(N)=O)n2)=O)C(O)C1)=O CC1(CNC(c2cc[nH]n2)=O)CCC(NC(C2(CS(C)(=O)=O)CCC2)=O)C1 N1(CC2CCC(C)(C)CO2)CC2(CO)CCC1CC2 c1(CC(N2CCC(N(C(C=NOC)=O)CC)CC2)=O)c(C)nn(CC(C)C)c1C c1(OCC)cnc(C(=O)N(CC(O)CNC(C2CN(C3COC3)C2)=O)C)c(Cl)c1 C1(CC(=O)NCC2(NC(c3cncc(C)c3)=O)CCCCC2)CCC(=O)NC1=O O(NC(=O)C(F)N(C(C)=O)CC)CCCC.C1(=O)CC2(CC2)CN1 c1(C(N(CC(CC)NC(=O)COc2cccc(C)c2C)C)=O)cc(N)c(F)cn1 N1(NC(C2N(Cc3scc(NC(C)=O)n3)CCOC2)=O)CC2CC2C1C#N c1(C(N2CC(OC)C(NC(C3(CF)CC3)=O)C2)=O)ccc(O)cc1[N+](=O)[O-] c1(NC(C2N(Cc3ccc(C(C)(C)C)cc3)CC2)=O)nc(O)nc(O)c1[N+](=O)[O-] C(=O)(CCC(F)(F)C(F)F)NCC(C)NC(c1cc(C=C)cc(F)c1)=O c1(CC)ncccc1C(N1CCOC(C(=O)NC(c2ccc(C)cn2)C)C1)=O N1(C(c2cncc(NC=O)c2)=O)CC2CCC1CN(C(=O)CSc1cccs1)C2 Cc1nc(CNC(C2(N(C)C(c3n[nH]c(C4CC4)n3)=O)CCC2)=O)oc1C C1(C(=O)NC(c2cn(CC)nc2)C)CCc2c(ncn2C)C1 c1(C(=O)NC(CC2CN(C(CCC=C)=O)C2)C)c(C)nn2cccnc12 C1(NC(=O)Cc2cnsc2)CN(C(c2ccc(O)nn2)=O)C2CCCCC12 N1(C(c2occ(C)c2)=O)CC(N(C(=O)Cc2cocn2)C)C2(CC2)C1 Nc1ccc(F)c(C(N2CC(NC(=O)CC3CCSC3)C(O)C2)=O)c1F C1(NC(C(=O)NCC)=O)CN(C(c2cnnn2C)=O)C2(CCOCC2)C1 CS(=O)(=NCC(=O)OC1CCCOC1)c1ccc(Cl)cc1 N1(Cc2ccc(C)cc2)CCC(O)(C(=O)NCCc2ncc(C)[nH]2)CC1 C1(NC(c2ccccc2C(F)F)=O)CC12CC(NC(C1CCCOCC1)=O)C2 C(=O)(C(F)C(C)C)NC(CCNC(c1nc(C)sc1)=O)C CCC(CC(=O)NC12CC(CNC(=O)C(F)C3CCOC3)(C1)OC2(C)C)C(C)C C#Cc1ccnc(C(N2CCC(C)C2CNC(c2cn(C)nc2CC)=O)=O)c1 N1(CC)CC(C(=O)NCCC2CCCN2C(c2cncc(OC)c2)=O)CC1=O N1(C(C=CCOC)=O)CCCCC1CN(C)C(C1CCC(N(C)C)C1)=O C12(CNC(=O)CN3CCCCCC3)CCC(CN1C(=O)CNc1ccccn1)C2 CC1(NC(c2cc(C(F)(F)F)cs2)=O)CCN(C(c2ncccc2F)=O)C1 N1(C(C(C=C)(C)C)=O)CCCC(NC(=O)C(CC2CCCC2)CC)CC1 c1(OC)ccc(F)cc1C(=O)N(C)CC1CCCCN1C(C1CC2(CCC2)C1)=O CCCCC(O)C(=O)NCC(C1(O)CN(C(=O)Cn2nc(C)c(C)c2C)C1)(C)C c1(CC)nc(C)c(C(=O)NC(C)CNC(=O)CCNC(C2CCCO2)=O)o1 CC1(C)OCC2CC12C(=O)NC1COCC1NC(C1SC2C=CC1CC2)=O c1(C(=O)NCC(C)NC(CC(CCCC)O)=O)cc(C)nc2c1nc(C)n2C CC(C(=O)NCCC1(C(N2CCN(CC3CC3)CC2)=O)CC1)S(N)(=O)=O C(=O)(N=c1cnn(-c2ccc(Br)cc2)[nH]1)NC1(C)C(C)OCC1 C(=O)(C(CC(F)F)N(C(=O)C(C)=CC(C)(C)C)C)NC(COC)C(C)C CN1N=C(C(=O)N2C3CCC2C(C(N2Cc4ccccc4C2)=O)C3)CCC1=O c1(OCC)cc(Cl)ccc1C(=O)N(C1CCN(C(C2CC2F)=O)CC1)CCO c1(C(N(CCC(C)NC(C2CCO2)=O)C)=O)ccc(F)cc1Cl c1(OC)cccc(C(=O)NCC2(C)CN(C(C3CCCN3N=O)=O)CC2C)c1F N1(C(CCCOCC)=O)CCC(C(=O)NC2CCCC(N(C)C)C2)CC1CC C(=O)(C1CC(=O)c2c(F)cccc21)N1CC(N(C)C(c2nc(=N)cc[nH]2)=O)C1 c1(CC(N2CCN(C(c3c(C)cno3)=O)C(CC#N)C2)=O)ccc2c(c1)CCC2 C(C(C)(CC(C)C)NC(=O)CC1COCC1O)NC(c1c(C)nccc1)=O c1(C(N2CCCC(NC(C(C)OCC)=O)(CC)C2)=O)ccc2c(c1C)CCC2 C1(NC(C2C(=C)C2)=O)CC(F)(F)CN(C(=O)CN(CC)CC)C1 N12CC(O)CC1CNC(=O)C1CCC(O1)C(OC)C2.c12ccc(o1)C2.C(SC)SC C1(=O)CCCCN(C(C)C)C(C2(O)CCC2)C(=O)N1.C(=O)(C(C)(C)SC)OC c1(C(=O)NC2CC3(CN(C(c4c(C)ccn4C)=O)C3)C2)nc2ccccc2[nH]1 N1(C(CC(CC)(C)C)=O)CCC2(CC1)CC(C)N(C(=O)CCCC(N)=O)C2 c1(OC)nc(Cl)ccc1CN1CC2CC2(C(N2CCSCC2)=O)C1 CC1(C(N2CCCC(CNC(c3cc(C(F)F)cs3)=O)CC2)=O)CCC(=O)NC1 c1(C(N2CCC(NC(c3c(=N)cc[nH]c3)=O)CC2)=O)cc2cnccc2cc1F c1(C(=O)NCC2C(NC(CC(=O)OCC)=O)CCC2)ccc(CC)c([N+](=O)[O-])c1 C1(CNC(C(C)(c2ccccc2)OC)=O)CN(C(C2(Br)CC2)=O)CC1C(F)(F)F C(CCC(=O)NNc1ccc(C(F)(F)F)cc1)Sc1ccc(C)cn1 CCC(C)(C)CCCC(=O)N(C(C)CC(=O)NC(C)CCC(C)C)C N1(C(COCCOC)=O)CCC(NC(=O)CC(=O)O)C1 c1(CCC(=O)NCCCN(CCO)C(c2cc(C3CC3)no2)=O)cnc(O)[nH]1 O(NC(=O)C(C(C)CC)N(C)C(c1sccc1CC)=O)CC(=C)Cl C1(CC)(NC(c2ocnc2C)=O)CCN(C(=O)CCCC2CCCC(=O)N2)CC1 C=CCC(C(=O)NCCc1cccs1)NC(c1nnsc1N)=O CC(C)C(F)C(=O)N1CCC(C(C)NC(=O)C(C)CC2CC2)C1 CC1(C(N2CCC(NC(c3ncoc3-c3cccs3)=O)C2)=O)CCCS1(=O)=O CCC(CNC(C1COCCN1C(=O)C(C)C)=O)(CC)NC(=O)CCCC#N CSC1=C(C(=O)N2CC(=O)CC2COC2CCCCC2(F)F)CCCC1.C1COC1 C1(NC(c2cn(C)[nH]c2=N)=O)CCN(C(=O)Cn2nccn2)CC(C)(C)C1 C1(NCCC(=O)NC(=O)CC2C3COCC23)CCC(C(=O)NC2CC2)CC1 N1(C(C(C)N(C)C)=O)C2CCC1C(F)C(NC(C13CCC(CC1F)C3)=O)C2 C1(CNC(CCC#C)=O)CN(C(=O)C(C)(O)C=C)CC1(C)C C12(N(c3ccc(C)cc3C)C(C=C(C)C)=O)CCC1CN(C(=O)C(=O)NC1CC1)C2 c1(CCC(C)NC(C23CC(CN2)C3)=O)cccc(-c2ccccc2)c1 N1(C(Cc2cncc(C)c2)=O)CC2(CCCC2NC(=O)CCN=[N+]=[N-])C1 C(C(C(=O)NCCc1nnc(O)o1)NC(=O)C(C)=C(C)C)OCC C[Si](C)(C)C1(C(=O)NCCOCCCNC(c2csc(O)n2)=O)CC1 c1(C(=O)NC(C(C)NC(c2cc(C)c(C)nn2)=O)CO)cc2cccc(C)n2n1 c1(C(=O)NCC(C)(C2CCC2)NC(C(C2CC2)OC)=O)csc(CS(C)(=O)=O)n1 c1(C(N2CCC(CC(C)C)C2)C#N)ccc(Cl)cc1 c1(C(=O)NCC2CCC(NC(c3c(SC)cccc3)=O)C2)cnc2c[nH]nc2c1 N1(C(C(C=C)(C)O)=O)CC2CC(NC(=O)C#CC3CCC3)C1C2 c1(C(=O)NCCN(C(CCCCC=C)=O)C2CC2)ccc2nc(C)ccc2c1 CC1CC(N)CCCN1C(=O)Sc1ccccc1.C1(=O)COC1=O.C(C)(C)(C)O c1(C(N2C(CCC(C)(C)OC)CCCC2)C(=O)NC(C)C)cc2sc(C)cc2[nH]1 c1(-c2nc(-c3cc(OC)c(O)nc3)n(C3CCC3)n2)cc(Cl)cc(S(C)(=O)=O)c1 N1(C(CCCOCCC)=O)CCC(O)(CNC(c2ccn(C)n2)=O)C1 C(C)(C(C(=O)NCCS(N)(=O)=O)C(C)C)NC(c1c(C)cccn1)=O N1(CCC(=O)NCc2cc(C(=O)NCCc3ccsc3)co2)CCCCC1 C1(O)(C(C)C)CCCN(C(=O)C2=CCC(NC(=O)CCNC(N)=O)C2)C1 c1(CC)ccnc(C(N2CCCC(NC(=O)C(S(C)(=O)=O)C3CC3)C2)=O)c1 C(=O)(C(C)CC(F)(F)F)N(CCC(c1cccs1)N(C(CSCC=C)=O)C)CC C#CCC(C(=O)N1CCC(F)(F)C1)NC(=O)C(C)CCOC N1(C(C2C(C)C2)=O)CCCC(N(C(=O)C=CC2CC2)C)CC1 c1(C(N2CCCCC(CNC(=O)C3=CCCSC3)C2)=O)ccc2nccn2c1 C1(NC(C(C)OCCOC)=O)(CO)CN(C(=O)C(F)C2CCC2)C1.C(COC)S n1(CCCNC(C(n2cc(-c3cc(C(=O)OC)sc3)nn2)C)=O)c(C)csc1=O C(=O)(C1=C(C)CCCC1)OC.c12ccc(cc1)NC(=S)NC1(CCC1)COC2=O c1(C(C)C)cn(CC2C=CCN2C(=O)CNC(c2ccco2)=O)nn1 c1(C(=O)NC2CCN(C(C(C)OCCC#C)=O)CC2O)cccc2ccn(C)c12 C1(CC(=O)OC)CCCN1C(=O)CCc1ncnn1C.C1(C)(C)CNC(=O)CO1 n1(CC)cc(C(=O)N(C)CCOCCCN(C(=O)CC(O)C2CC2)C)cn1 N1(C(c2cc(C(C)(C)C)no2)=O)CC2CC(CNC(C3CNC(=O)C3)=O)C2C1 C(CN=c1ccc(C(N2CCCC2CCCNC(c2ccsc2)=O)=O)c[nH]1)OC N1(C(CC(CCCCC)O)=O)CCC2(NC(c3nocc3C)=O)CCCCCC12 CC(C)(C(=O)N1CCC2(CC2C(=O)NC2C=CC2C(=O)OC)C1)C(F)F C(CC(C)C)(C(=O)N1CC(OC)CC1CSC)N(C(C=CC=CCC)=O)C N1(C(C(=O)NC2CCCC(C(C)C)CC2)=O)CCC(F)(F)C(C)C1 Cc1ccnnc1-c1ccc(CN(CC(C)O)CC2CC(F)(F)C2)s1 C1(C(=O)NCCn2c(CC)ncc2)CC(O)CN1C(=O)CC1CC1(C)C Cc1c(C(=O)NC2(C)CCCN(C(C3OCCCO3)=O)C2)[nH]c2c(Cl)cccc12 N1(C(C(CC)CC)=O)CC=C(C(=O)NC(c2cn(C)nc2C)C)CC1 C(CCC(C)C(=O)NCC(CNC(c1cnoc1C)=O)CO)OC N1(C(Cc2c(OC)nccc2)=O)CC2CC(NC(C3CCCC(O)C3)=O)CC1C2 Cc1[nH]nc2ncc(C(N3CCC(F)(CNC(C4CC4(C)Br)=O)CC3)=O)cc12 Cc1c(F)ccc(Cl)c1C(N1CCC(NC(C2CCC(C)CC2)=O)C(C)(C)C1)=O c1(C(=O)NC(C2CCN(C(C(C)OCC3CC3)=O)C2)(C)C)ccc(C2CC2)cc1 c1(C(N(C)CCOCCNC(=O)CC2CCOC2)=O)cccc(-n2cncn2)n1 c1(C(=O)NC(C(C)C)CCN(C(=O)C(C)(C)CN(C)C)C)cc2c(ccn2C)[nH]1 c1(C(=O)NC(C2(CNC(CN3CC(C)C3)=O)CC2)C)c2c(nn1C)CCOC2 c1(C(N2CC(NC(c3c(CC)c[nH]n3)=O)C(C)C2)=O)cccc(F)c1OC(F)F c1(OC)cc(C(N2CC3CC(NC(c4ccc(C)nn4)=O)C2C3)=O)ccc1C c1(C(=O)NC(CCCCNC(C(CC)(C)O)=O)C)ncc(Cl)cc1O N12CCCC(C1)N(Cc1cccs1)C(=O)C2C.c1(CNC(=O)OC)nnn(C)n1 N#Cc1cccc(N(C2CCNCCC2C)C(c2cccc(I)c2O)=O)c1 c1(CC)c(C(N2CCN(CCN)CC2)=O)cnn1-c1ccc(C)cc1 N1(C(CC(COC)C)=O)CCC2C1CCCN2C(=O)CN(c1ccccc1)C C1(C(=O)NCC2(O)CCCN(C(c3nccc(C)n3)=O)C2)CC2C=CC1C21CC1 c1(OC)cc(C(=O)NCCSc2cn(Cc3nc(C(=O)O)cs3)nn2)cc(C)n1 N1(C(C(CC#C)CC#C)=O)CC(NC(=O)CCC(=O)NCC)CC12CCOC2 C1(OC)CN(C(n2ccnc2C)=O)CCC1NC(=O)CC1CCCCO1 C(=O)(C(F)CC(C)C)N1CC(F)(CNC(C(C)OCCCC)=O)C1 c1(OC)cccc(C(=O)N(CCN2CCCCCC2)C(C)C)c1 c1(C(N2C(CNC(C3CC4C=CC3C4)=O)COCC2)=O)cnc(O)nc1O Cc1cccc2c(CN3C(C(=O)Nc4cnn(C)c4C#N)CC4CC34)c[nH]c12 N1(C(C2CCN(C(c3c(CC)ocn3)=O)C2C(C)C)=O)CCCC(F)(F)C1 Cc1cccc(CN(C(=O)C(CC2CCCC2)NC(c2ccc(CO)o2)=O)C)n1 c1(OC)c(C(=O)NC23CC(C2)N(C(=O)CCOCC(C)=O)C3)c(C)nn1C N1(C(c2ncn(C)c(=O)c2)=O)CCC(C2(O)CCN(C(=O)COCCF)C2)CC1 c1(C(N2C(CCNC(=O)CC3CCC4CC4C3)CCC2)=O)ccc2nccn2c1 C1(C(=O)OC(C)(C)C)CC2(CCN(C(=O)NCCCc3ncn(C)n3)C2)CO1 C1(C2CN(C(C3CCC(N(C)C)CC3)=O)C2)(NC(C=C(CCN(C)C)Cl)=O)CC1 C1(CC(=O)NC2CCCC(NC(C3(SC)CCC3)=O)C2)CCCNC(=O)C1 c1(NCc2cc(OC)c(F)cc2)cc([N+](=O)[O-])c(C(N)=O)cc1OC C1(C(=O)NC(C)CN(C)C(c2ccccc2CO)=O)CC2(C1)OCCO2 N1(C(c2n(C)ncc2C#N)=O)CCC(F)(F)C(CNC(=O)CC2CS(=O)(=O)C2)C1 c1(C(N2CCC3CC23)C2CN(C(CC=CC=C)=O)C2)ncc(C#N)cc1C Cc1cn2cccc(C(=O)NC(C)C(C)NC(C3(CCN(C)C)CC3)=O)c2n1 n1(CC)cc(C=CC(=O)NC2(C(=O)OC(C)(C)C)CC=CCC2)c(C#N)n1.C(N)=O C1(C(N2CC(C)C(CNC(=O)C(O)C3CCC3)C2)=O)C2CCC1(C)C2(C)C C1(C(=O)NCC2CCCC2NC(C2(C(F)F)CC2)=O)COc2ccccc2O1 N1(C(C(C)SCC)=O)CCCCC2(CCN(C(=O)Cn3ccnc3C)C2)C1 c1(C(N2CC(NC(C3(OC)CCCOC3)=O)C2)=O)cccc2[nH]c(=N)oc12 C1(NC(CS(CC#C)(=O)=O)=O)CCc2ncccc2C1=O C#Cc1cc(NC2CCC(S(C)(=O)=O)C2)ccc1Cl C(=O)(C(O)CC[S+](C)C)N(C1CC(NC(c2ccc(C#N)s2)=O)C1)C C1(C(N(C(CC)(C)C)CC)=O)CCCCN(C(=O)C(OC)OC)C1 C1(C(=O)NCC2(OC)CCN(C(=O)C=CC3CC3)CC2)CCc2ccccc2C1 N1(C(c2c(C)nns2)=O)CCC(O)(C(C)NC(c2cncc(N(C)C)c2)=O)C1 c1(C(=O)NC(CC)CNC(=O)CN2CC3CC3C2)ncc(C#N)cc1C c1(C(=O)NC2(CCCNC(C(C3CCCC3)OC)=O)CC2)cc(C)c(=O)n(C)c1 C(=O)(C1SCc2cccnc21)NC(C)Cn1cc(C2CCCC2O)nn1 c1(C(N2CCCCC(NC(c3c(C)nc(C)s3)=O)C2)=O)ccc2sccc2c1 CCCCS(=O)(=O)N1CCCC1C(=O)NC(C)(C)CN(C)C(C1(F)CC1C)=O c1(C(CNC(C2C(C)C2)=O)NC(=O)CCc2cncn2C)ccccc1F N1(C(C(CCOC)C)=O)CC2(CC(NC(c3cc(Cl)n(C)n3)=O)CO2)C1 C1(C(N2C(CNC(c3cc(Cl)ccc3Br)=O)CC(O)C2)=O)CC2OC1C1CC21 c1(C(N2CCC(C(C)NC(c3cn(CC=C)nn3)=O)C2)=O)cc([N+](=O)[O-])n[nH]1 c1(N(CCNC(=O)CC2COC(=O)C2)CC)ncc(C(C)(C)O)cn1 CC1CC(NC(C2C3CCCOC23)=O)CN(C(=O)CCC2CCCC2)C1 CC1=C(C)CC(C(=O)N(C2CN(C(C3CCCCNC3=O)=O)C2)C)CC1 C1(CNC(=O)C(F)n2cccn2)CC2COCC2N1C(c1cccc(Cl)c1)=O C12(NC(C3CC=C(C)CC3)=O)CCCC1CN(C(c1cnoc1C1CCC1)=O)C2 c1(CC)ncc(C(=O)NCCC2(OC)CN(C(c3cc(C)[nH]n3)=O)C2)c(C)n1 c1(C(=O)NCCC(CNC(c2nc(CCC)oc2)=O)O)cn(C)[nH]c1=N c1(C(=O)OC)cccn(CC(=O)NC2CCC(NC(C3(C(N)=O)CC3)=O)C2)c1=O c1(C(N(CCNC(COCc2onc(C)n2)=O)C)=O)cc(C#N)c(N)cc1O N1(C(CONC(c2cc(F)cnc2O)=O)=O)CCC(C2CCOC2)C1 N1(C(=O)Nc2ccc(C#C)cc2)CCCC2(CCN2C(c2cccnc2)=O)C1 c1(NC)ccc(C(=O)NCC2CN(C(=O)CCC3CCOC3)C(C)(C)C2)cc1F N1(C(c2ncn(C)n2)=O)CCC(F)C(NC(=O)COCCc2cccc(F)c2)C1 c1(C(=O)NC(CC)(C)CNC(C2CN(C)C2)=O)occ(C)c1C N(C1C(=O)Nc2cc(Cl)ccc21)C(c1ccc(C)cc1C(F)F)=O c1(C(=O)NC(C)CCCNC(c2cnc(C(F)(F)F)nc2)=O)cccn(C)c1=O C(c1sccc1C)=CC(=O)NCC(C)NC(CC1CC(OC)C1)=O CC(C)(C)C(CNC(C1CCC12CCC2)=O)NC(=O)CCc1ccccc1 C#CCC(C)(C)C(c1nnnn1Cc1c(F)cccc1F)NCc1ccccc1 Cc1cc(Br)c2c(c1)CCCN2C(C1C(Cl)(Cl)C12CC2)=O C1(NC(Cc2nc(C)oc2)=O)C2CN(C(=O)CCC3CNC(=O)N3)CC12 N1(C(c2oc(C)c(CO)c2)=O)CC2CCC(C1)C(NC(=O)CC1C=CCC1)C2 C(=O)(C(C)C(C)(C)C)NCC(c1ccc(C)cc1)NC(=O)Cc1nn(C)cc1Cl CC(CC(=O)NCC1(NC(=O)Cc2nc[nH]n2)CCCC1)n1cc(Br)cn1 Cc1cc(NNC(=O)NC2CCN(CC(F)F)C2)nc(S(C)(=O)=O)n1 N1(C(C(C)=O)=O)CC(C)C(C)(CNC(c2ccc(F)c(CO)c2)=O)C1 N1(C(C2C(C)CCC2)=O)CCC2(CCC2NC(=O)Cc2ccc(F)cc2Cl)CC1 O=[N+]([O-])c1cc(NCc2cc3cc(Br)ccc3s2)nc(F)c1 C(C(C)(C)CC(=O)NCC(CC(F)(F)F)NC(C)=O)OC c1(C(=O)NC2C(C)(C)C2c2ccccc2)ccc(F)cc1Nc1ncccn1 C1(N(C)Cc2scc(C(=O)OC)n2)CCC(O)CC1 CCC(CC(=O)NCC1CCC(C(=O)NC(c2nccn2C)C)CC1)C(C)C c1(C(=O)NCC(CC)NC(c2sc(F)cc2C)=O)c2c(nn1C)CCCC2 C1(CC(c2cccnc2)(C)O)(NC(CCO)N(C)C)CCOCC1 C(C(C(C)(C)C)NC(=O)CC1CCSCC1)NC(C1(COC)CCCC1)=O c1(C(=O)OC)nc(N2CC(C)(NC(=O)CN3CC4CC4C3)C2)c2ccccc2n1 c1(C(N2C3CN(C(c4ccc(OC)c(F)c4)=O)CC32)=O)cnc2ccc(Cl)cn12 C1(NC(=O)CC2(O)CC2)CCC(NC(C2(CF)CCOCC2)=O)CC1 N1(Cc2c(C)ccc(Cl)c2)C2COCC1CN(C(c1cc(C3CC3)no1)=O)C2 CC1=C(C(=O)N2CCCOC(CNC(c3ccc(Cl)cc3)=O)C2)CCC1 C1(CNC(=O)CC2CC=CC2)CN(c2ncccc2[N+](=O)[O-])CCC12CCOC2 CCC(CC)CCC(=O)NC(C)(C)CCNC(C1CC(C)CO1)=O O=C(C1CCCc2ccnn21)NCCC1CCCN1C(c1cc(C2CC2)[nH]n1)=O c1(CNC(=O)Nc2cn(C(C(=O)OCC)(C)C)nc2)cc(CC)ccn1 N1(C(C(CCOC)NC(=O)CCc2ccn(C)n2)=O)CCCC(CCO)CC1 N1(C(C23CC(C)(C2)C3)=O)C2CCC1CC(O)(CN)C2.C(=O)C(CCN(C)C1CC1)N(C)C N1(C(c2cc(C)n(C(F)F)n2)=O)CCN(C(=O)Cc2c[nH]nc2O)C(CCO)C1 C1(C(=O)NC(C(N2CC(C)OCC2)=O)(C)C2CCC2)CCC=CCCC1 c1(C(=O)NC2CCC(NC(c3cc(C)cc(O)c3)=O)C2)ccc2c(c1)OCCO2 N1(C(C=C(C)c2ccc(F)cc2)=O)C2CCCC1CN(C(=O)C(=O)C(C)(C)C)C2 CC1CC(C)OC1CNC(=O)CCCNC(N)=O N1(C(C(C)OCC2CCCC2)=O)C2CC1CN(C(=O)C(CO)N(C)C)C2 N1(C(CCCOC)=O)CC(C(=O)NC2C=CCCC2CO)CC(C)(C)C1 c1(CC(C)NCC#CCN(C)C)c(F)cccc1F CC1OCCN(C(=O)CC2CCSC2)C1C(=O)NC1C=CCC1 C(=O)(C(F)C(F)(F)C(F)(F)F)N(CC(N1CCC(C)(F)C1)=O)C C1(C(=O)NCCc2onc(CC)n2)CC(F)CN1C(=O)CCc1nncs1 c1(CNC(C(C)=C2CC2)=O)nc(C(N2CCC(F)(C(C)C)C2)=O)c(C)o1 C(=O)(C(C(C)(C)C)SC)NCC1CN(C(c2n[nH]c(CC)c2Cl)=O)C(C)C1 c1(OC)c(C(N2CCC(C)C2C(=O)N(C)Cc2cc(C)n(C)n2)=O)cnn1C c1(CN2CCC(CC(=O)Nc3n(C)ncc3Br)C2)ccc(F)nc1F CN1CCC(C2(C(N3CCC4(C3)CN(C(C3(O)CCOCC3)=O)C4)=O)CC2)CC1 c1(CNC2CC(c3cn(CCO)nc3)OCC2)cnc(F)c(Cl)c1 CC(F)(C(=O)N1CCC(NC(=O)Cn2cc(Br)ccc2=O)C1)C(F)(F)F CNS(=O)(=O)NCC(=O)NCC1COCC1NC(=O)C(c1cnn(C)c1)O N1(C(C(C2CCC2)OC)=O)CC2CCC2(CNC(=O)Cc2nncn2C(C)C)C1 C1(CC)OCCC1C(=O)NCc1csc(C(N2CC(OCC(C)C)C2)=O)c1 C(C(C)(F)C(C)(C)F)NC(CC(C1CC1)NC(C(C)C1CCCC1)=O)=O N1(C(=O)C(F)C2CCC2)CCC(CC2COCCN2C(C2CCSCC2)=O)CC1 Cc1ccnc(C2CCN(Cc3cnn(-c4ccccc4C)c3O)C2)n1 C1(C)(C(N2CC3C(CN(C(COC)=O)C)C3C2)=O)CC2C=CC1C2 N#Cc1ccsc1C(N1CCC1C(=O)N(C1CCOC1)CCO)=O C1(CC(=O)NCC(CCOC)NC(c2oc(SC)cc2C)=O)C(C)(C)C1(C)C S(=O)(=O)(c1ccc(Br)cc1NCC(C)CO)NCC(CC)O C1(O)(CNC(=O)C(O)c2ccsc2)CN(C(=O)CCc2ccncc2)C1 C(=O)(C(C(F)(F)F)C(F)(F)F)N1CCCC(N(C(CCCOC)=O)C)C1 Cc1cc(C(F)(F)F)ncc1C(=O)NCC(C(C)C)NC(c1cc(=O)cc[nH]1)=O C1(C)(CNC(CCN(C(CC)CC)C)=O)CCCN1C(C1CC2(CCC2)C1)=O N1(C(CN2CC(C)C2)=O)CCC2(CC1)CC(C)N(C(=O)C(C1CCCCCC1)C)C2 C1(NC(C2(C3CC3)CN(C(=O)C=CC3CCCC3)C2)=O)C2CCC3C(C2)CC13 C1(NC(CCCC=C)=O)CN(C(=O)CC2CCCC(C)(C)O2)Cc2nccn2C1 c1(C(=O)NCCN(C(=O)CCc2ccsc2Cl)C(C)C)occc1F c12cncc(c1)N2.N1(C(=O)NCC2CC23CC3)CC(CF)C1 c1(C(N2CCC(NC(C(CC)F)=O)C2C)=O)cnc(O)cc1OC c1(NC(CNC(c2c(CC)noc2)=O)=O)ccccc1SC(C)(C)C Cc1nn(C)cc1C(O)C(=O)NCCCC(C)(C)NC(c1ccncc1)=O C(=O)(C(CC(F)F)C1CCC1)NCC(CNC(c1c(C)nc(N(C)C)s1)=O)(C)C c1(C(N2CC(NC(c3cnc(C)nc3C)=O)C(F)C2)=O)ccc2c(c1)C=CCC2 C1(CNC(CNS(CCCC)(=O)=O)=O)CCC12CCN(C(=O)C(C)(C)CF)CC2 C(=O)(C1CCCc2c[nH]nc21)N1CCCCC(NC(C2CC3C=CC2C3)=O)C1 C(=O)(NNC(=O)NC(Cc1ccco1)CO)c1ccnc(C)n1 c1(NC(c2c(NC(c3cccnc3F)=O)c[nH]n2)=O)cc(Cl)ncc1Cl C1(SCC)C(C(=O)NCCCC2(C)CC2)CCCN1C(C1CC1c1ccco1)=O c1(OC)nn(C)cc1C(N1CCC(CNC(=O)C(c2cccnc2)O)C1)=O N1(C(c2cc(CC)ncc2)=O)CC2(C(=O)O)CC1CO2 C(=O)(C1NCCc2ccccc21)NC(C)Cn1cncn1 c1(OC)nccc(C)c1NC(=O)NC(CC(N)=O)c1ccccc1 C(C(F)(F)C(=O)NC(C1CCN(C(=O)CC2CC(F)(F)C2)CC1)CO)N(C)C Cc1cc(N2CC(CCCNC(=O)OC(C)(C)C)OC(C)C2)nc(C)n1 C(=O)(CCCCSC)N1C(CN(C(C2CCC(C)CC2)=O)CC)CCC1 C1(CCCC)CN(C(=O)C(C)C(C)(C)C)CCN1C(=O)CCCNC(C)=O N1(C(C(C)CN(C)C(c2ccc3c(c2)CC3)=O)=O)CCC2(COC(C)C2)C1 N1(C(C2(C)CCCS2)=O)CCCC2CN(C(C3CCCC4(CC4)C3)=O)CCC12 C(C(C)CN=c1[nH]c(Cl)nc(C)c1[N+](=O)[O-])NC(C1(OC)CCC1)=O C(=O)(C(=O)N=S(C)(C)=O)NC1CC(NC(c2cccc(C(=O)NC)c2)=O)C1 C1(NC(c2cnn(C(F)F)c2)=O)CC2CC1N(C(=O)Cc1csc(C3CC3)n1)C2 Cc1cn(CC(N2CC3CC(NC(C4CCNC(=O)C4)=O)C2C3)=O)c(=O)nc1O N1(C(C2=C(C)OCC2)=O)CCN(C(C2C3CC4C(C3=O)C24)=O)C(=O)CC1C C(CC(F)(F)Cn1cc(-c2ccnn2C)nn1)NC(C(C)O)=O N1(CC#C)CCN(C(C2CN(C)CCN2C(=O)CCCn2cccc2)=O)CC1=O CCC(C)C(=O)C(=O)OCc1cc(F)ccc1F c1(N2C(COCC)CN(c3cc(C)ncn3)CC2)ncc2ccc(F)cc2n1 C1(NC(=O)Nc2ccccc2)CC(F)CN(C(C2CC3C=CC2C3)=O)C1 C1(C(=O)NCCOCCC(=O)NCCC2CCCOC2)CCCOCC1 c1(CCC(N2C(C(=O)NC(c3ccccc3Cl)CO)CC2)=O)ccc(F)nc1 Cc1[nH]cc(C(N2CC3(COC(CNC(=O)CCC4(C)CC4)C3)C2)=O)c(=O)c1Cl Cc1sc(Cl)c(C(=O)NCCCN(C)C(C2CC(=O)N(c3cn[nH]c3)C2)=O)c1C C(=O)(C(O)C(C)(C)CC)N1CCC(O)(C(C)NC(CC(=O)NCC)=O)CC1 c1(SCC)cc(CC(=O)N(C)CCN(C)C(=O)C2CC2)on1 C1(OCC)CCN(C(=O)CC2(CNC(C3CC4(CC(=O)C4)C3)=O)CC2)C1(C)C N1(C(CNC(c2ccc(F)cc2)c2c(C)ncs2)=O)c2ccccc2CCC1C C1(NC(C(C)CC2CCC2)=O)CC(F)CN(C(c2coc(C3CC3)n2)=O)C1 c1(C(=O)NCC(C2CCOC2)OCC)ccc(OCC(C)C)nn1 C1(C)(CNC(C(C)NC(COC)=O)=O)CN(C(c2nocc2C2CC2)=O)C(C)(C)C1 N1(C(c2cn(C)nc2)=O)CCCCC1CNC(C1CC1(c1ccccc1)C)=O C(=O)(C(F)C(F)(F)F)NCCNC1CCC(CC(=O)N(CCN(C)C)C)CC1 CC1CCC(CNC(c2cccc(C(F)F)n2)=O)CN1C(c1ncn(C)n1)=O N1(C(CCN(CCC)C)=O)CCC(C(=O)NCc2ocnc2C2CC2)(CO)C1 c1(OC)cc(C(N2CC(NC(C3(OC(C)C)CC3)=O)CC2C)=O)c(Cl)cc1Cl C1(C)(CNC(CNC(C(CC)C)=O)=O)CN(C(=O)CC2(C#N)CCC2)CC1C c1(C(=O)NC2CC3CN(C(c4nn(C)c(O)c4)=O)C2C3)cccc(P(C)(C)=O)c1 c1(NC(C(=O)NCc2cccc(F)c2)=O)nc(Br)cn1C(F)(F)F Cc1csc2ncc(C(=O)NCC(C(C)C)NC(C3CCCS3(=O)=O)=O)n12 c1(NCCN(C(=O)CCCN2CCOCC2)CCOC)nc2ccc(O)cc2s1 c1(C(N(CCN(C(C2CCCN2CC)=O)CC)CC)=O)cn2cc(Cl)cnc2n1 c1(-c2cccc(OC)c2)ccc(S(=O)(=O)NNC(=O)C2CCC(=O)N2C)cc1 c1(COCCOC)cc(C(=O)NCC2CC2NC(c2ccoc2Cl)=O)ccc1F C(=O)(C(C#N)CC)NCCCC(c1ccccc1)NC(c1c(CC)cco1)=O Cc1nc(C(=O)NCC(F)CNC(=O)C=CS(C)=O)sc1C CC1CCCN(C(=O)Cc2csc(-n3cc(Br)cn3)n2)C1CO c1(C(N2CCCC(C=O)C2)=O)cc2nc[nH]c2cn1.CC(C)C(C)N(N1CCCC1)CC N1(Cc2c(C)nc(-c3ccc(Br)cc3)o2)c2ccccc2CC1C C(=O)(C(C)(CNC(=O)C(F)OC(F)(F)F)CC)NC(CCCCC)C c1(OC)ccccc1C1(C(N2CC(NC(=O)CC3CN(C)C3)C(C)C2)=O)CCC1 c1(OC)cccc(C(C)NC(N2CCC(CCOc3csnn3)C2)=O)c1 C1(NC(CC)=O)CCC(NC(C)C(=O)NC)CC1 C(=O)(CCCCCNC1(C(=O)OCC)CCCO1)N(CCC)CCC1CC1.COC N1(C(CCOCC#C)=O)CCC(CNC(=O)COCC(C)(C)C)C1 c1(N(C)C)ccc(C(=O)NCC(=O)Nc2cnn(C(C3(O)CCC3)C)c2)cc1 CCC(CC)CC(=O)NC(CC)C(=O)NCc1cn[nH]c1 C1(C(F)(F)F)(NC(C(=O)NC(C)CNC(c2ccco2)=O)C)CCN(C)C1 n1(CC)nc(C)cc1C(=O)NCc1nc(C(=O)NC(C)(CO)CCF)c(C)o1 C1(C(=O)NCc2c(CN(C(C(F)OC)=O)C)cccc2)CC2(CCC2)CO1 N1(CC(=C)C)CCN(C(=O)COC2CCN(C(c3ccsc3)=O)C2)CC1 N1(C(C2CCC(C(=O)OC)CC2)=O)CCC2(CCCCC2NC(=O)CCF)C1 C1(NC(C2(CC=C)CCN(C(=O)C(C3CCOCC3)C)C2)=O)CC2(C1)CN(C)C2 C=CC1(CC(=O)NCC2C=CCN2C(C2CC23CC3)=O)CCOCC1 C(=O)(CC(F)(F)c1ccccc1)NCC1N(C(C=C2CCC(C)C2)=O)CC1 N1(C(c2nccc(OC)c2)=O)CC(NC(c2csc(C#N)c2)=O)CC(F)C1 N1(C(C(C)SCCCC)=O)CCCCC(NC(c2nc(C(C)C)ncc2Cl)=O)C1 C12(C(=O)NC3C(CNC(C4(C)CCC4)=O)CCC3)CC3CC1C2C3O CC1CNc2ccccc2C1CNC(N1CCC(N(C)C(=O)OC(C)(C)C)C1)=O c1(CCOC)cn(C2CC(C(=O)NCCSC3CCC3)C2)nn1 C1(NC(CC)S(C)(=O)=O)CCC2(CC1)CC(CNC(=O)NC(C)(C)C)C2 C1(NC(COc2ccc(OC)cc2)=O)CC2C1CCN2C(c1cc(F)ccc1O)=O C1(O)CCC(N(C)C(C2CC2C(=O)NCCOC2CCCN(C)C2)=O)CC1.CO.O c1(OC)ccc(C(=O)NC2CCC(CC(=O)NC3CCOC3)C2)cc1 c1(CC)ccc(C(=O)N(C)CC2(O)CN(C(C3(C)CC(F)C3)=O)C2)nc1 N1(C(C(C(C)C)NC(=O)OC)=O)CCC(C2CC2)(NC(=O)C2=C(Cl)CC2)C1 c1(-c2cccc(N(C(CCC(C)SC)=O)CC3CC3)c2)cccc2nc(C)nn12 N1(CC2OCC(C)(C)C2)CC2CCCC(NC(=O)Cc3ccc(CO)cc3)C2C1 N1(C(C2N(C)CCC2)=O)CCC2(C(=O)NCCCc3cnccn3)CCCC12 N1(C(CC(CCC)O)=O)CCC(NC(C2(C)CCC(=O)NC2)=O)C(CO)CC1 N1(C(=O)NCCC(C)(C)C(N)=O)CCC(F)C(c2on(C)c(=O)c2)C1 C1(C(N2CC(CCCCC)C2)=O)CCCCN1C(=O)Cc1cn(C)nn1 C1(COCCOC(CCC)=O)CC2(C1)CC1(CC(NC(=O)OC(C)(C)C)C1)C2 c1(C(=O)NCC(CNC(C2C(C)(C)CC2)=O)O)ccccc1SCC(N)=O c1(C(=O)NC2C(CNC(C3(CC)CC3(F)F)=O)C2)ccc(O)c([N+](=O)[O-])c1 CCCC(C)C(=O)NC(C)(CC)CCNC(c1c[nH]nc1C1CC1)=O c1(CC)onc(C(=O)NCC(C)(CNC(c2scnc2Cl)=O)OC)c1C C(=O)(C(CC)CC(C)C)NC1(c2ccccc2)CN(C(CCCC)=O)C1 N1(C(Cc2ccn(CC)n2)=O)CC2CCCC(C1)N2C(=O)C(c1ccnn1C)C c1(C(C(=O)NC2CC(F)(CNC(C3(CC=C)CC3)=O)C2)O)ccc(Cl)cc1F N1(C(C(C)Cc2cnn(C)c2)=O)CC(NC(C2(O)CCCC2)=O)CC(C)(C)C1 c1(C(=O)NCC2(CN(C)C(C3CCSCC3)=O)CC2)cscc1C(F)F CCCCS(=O)(=O)NC(C)C(=O)N(C(CNC(=O)C(C)=C(C)C)C1CC1)C CC1(C)CCC(N=c2[nH]c(NC3COCC3Cn3ccnc3)nc3c(F)cccc23)C1 C=CC(C)CC(=O)N1C(NC2CCCN(C(=O)OC(C)(C)C)C2)(CC)CC1 CCCC(F)C(=O)N(C(C)CNC(C1CN(S(=O)(=O)C(F)(F)F)C1)=O)C C(=O)(C(C)(C)CCCO)NCC1CC(C)N(C(=O)CC2CCOC2)CC1 c1(CC(N2CC(O)(CCNC(C(CC)C)=O)C2)=O)cncc(Br)c1 c1(NCCN2CC(CS(=O)(=O)NC)OCC2)cccc2c1OCCO2 c1(-c2cc(C(=O)NCCCC=C)sc2)ccc(OC)cc1F Cc1cccc(OCC(=O)NCC(C)N(CC(=O)NC2CCCC2)C)c1C C(=O)(CCC(C)(F)F)NCC(C1CCN(C(c2c(C)cc[nH]2)=O)CC1)(C)O C1(O)(CNC(C(N2CCCCC2=O)C)=O)CCCN(C(=O)C(=O)NC2CC2)CC1 c1(CN2CC(C(=O)NCc3ccccn3)C(O)CC2)cc2ccccc2[nH]1 Cc1ccc(-c2nc(C(C)N(C)C)n[nH]2)cc1OCCC1CC1 N1(C(C(=O)NC(COC)C)=O)CC(O)CC12CCCC2 CCC(C)(CO)C(=O)NCC(C)(F)CNC(c1cc2n(n1)CCO2)=O C(C)(CO)(C(=O)N1CC(N2CCC2)C1)NC(C=CC(C)C)=O N1(C(=O)C=CCF)CCC(N(C(c2ccnc(OC3CCC3)c2)=O)C2CC2)C12CC2 C#Cc1cncc(C(N2CCC(F)CC2C(=O)NC(C)C(C)(C)O)=O)c1 C1(NC(C(COC)C(F)(F)F)=O)CC2COCC(C1)N2C(=O)C(O)CCSC C1(C(=O)NCCNC(COC)=O)COCCN1C(=O)C=CCOC CS(=O)(=O)CCCC(=O)N1CCCC(CNC(C2CCc3[nH]nc(O)c3C2)=O)C1 C1(O)(C(C)C)CCN(C(C2(CO)CCN(C(=O)CCSC3CC3)C2)=O)C1 c1(OC)cc(C)sc1C(=O)NCC1CCN1C(=O)C(O)CC1CCCCC1 c1(CCC)cc(C(=O)NC(C2CCN(C(C3CCCN3CC)=O)CC2)C)nc(Cl)n1 c1(OC)cc(NCc2cccnc2O)c(OC)cc1Br c1(CCNC(C2(CS)CC2)=O)csc(Cl)n1.c1(CO)cn(CCN2CCCC2)nn1 Cc1oc(C(C)(C)C)cc1C(=O)N(CC(C)NC(C1(O)CC1)=O)C c1(CCC(=O)N(CCNC(c2n(CC)ncc2)=O)C)ccc(Cl)cc1Br c1(NC(N(C)CCc2noc(CSC)n2)=O)c(C)cccc1C CN1CC(O)CCC1C(=O)NCCC1(NC(=O)CNC(c2cccs2)=O)CC1 CN1CCC(CC(=O)NCC(C)(C)CN(C)C(c2cnc(C3CC3)s2)=O)C1 C1(CC(=O)NCC(N(C)C(C2CCCOC2)=O)C2CC2)CCS(=O)(=O)C1 c1(CCC)ccccc1C(=O)NC1CCN(C(c2ccc(C)cn2)=O)C1 c1(C(C)=O)cc(C(N2CC=CC2CNC(=O)C=Cc2scnc2C)=O)ccc1C N1(C(CCCCSC)=O)CCCCC(NC(C2SC3C=CC2CC3)=O)C1 C1(C(=O)NCCCOC=C)CC12CC(NC(c1nccs1)=O)C2 N1(C(CCCN(C(C)=O)C)=O)CCC2(C(=O)NC(C)CCC(C)(C)C)CCCC12 c1(C(=O)NCCN(C(=O)COCCCC(C)C)CCC)cccc2c1CCC2=O c1(C(C(=O)NC(c2cccc(OC)c2)C(F)(F)F)(C)C)c[nH]c2ccccc12 N1(C(CC2(COC)CC2)=O)CCC2(CC2NC(C2(C(C)C)CNC(=O)C2)=O)C1 N1(C(C(CC2CC2)NC(C(C=C)(F)F)=O)=O)CCC2(CCCOC2)C1 N1(C(CC=C)=O)CCC(C2(O)CCN(C(=O)Cc3cnn4ccccc34)C2)CC1 C#Cc1cncc(C(N2CCCC(C(O)C(F)F)C2)=O)c1 C(=O)(C(F)C(C)CNC(=O)C(N1CCOCC1)C)Nc1ccc(CC)cn1 C1(NC(=O)C(C2CCOCC2)O)CSCCO1.C1CCC(=O)NC12CCC2 c1(N2CCC(C=O)C2)ncnc(Cl)c1C(C)C.c1(NC(CC)=O)ccc(S)cc1 N1(C(CCN(C(c2nc(CC)oc2C)=O)C2CC2)=O)CCCC12CCOC2=O c1(C(=O)NCCN2CCCCC2)n[nH]c2c1CN(C(C1CCOC1=O)=O)C2 C1(CNC(CC2(N(C)C)CCC2)=O)CCN(C(=O)CSCCC#N)CC1(F)F C(=O)(C1COc2c(C)cccc21)NC(CC)(CC)CCNC(=O)Cc1ccon1 CCCCCCN1CCC(CC(=O)N(CC(N2CCOCC2)C)CCC)C1 C(C(CC(F)(F)F)NC(c1ccc(Br)cn1)=O)NC(C1CCC(=O)N1)=O C1(C)(NC(CC2CCC(C)(C)O2)=O)CCN(CCC2CC2)CC1 CCCCC(=O)N1CCC1C(=O)NC(COC)C(=O)OC c1(CCCC(=O)NC2CCN(C(C3(OC)CCCC3)=O)C2)cc(C)sc1C N1(C(CNC(=O)OC)=O)CCC2(CC1)CC2NC(c1ccn(CCO)c1C)=O Cc1ccc(C)c(CC(N2CC3CC2CC3NC(=O)CC2CCCCCC2)=O)c1 C#Cc1cc(C(=O)NC(C)CCNC(c2cnc3[nH]cncc2-3)=O)ccc1C N1(C(CC(CC)(C)O)=O)CCC2(C1)CN(C(c1ncoc1-c1ccc(F)cc1)=O)C2 C1(C(N2CC(NC(c3ccc(COC)o3)=O)C(C)C2)=O)CS(=O)(=O)CCO1 c1(CC(N2CC(NC(C(CC)C)=O)C(CC)C2)=O)ccc(C(C)=O)cc1Cl C1(C(N(C)CC2(CNC(=O)C=CBr)CC2)=O)CC(C2CC2)=NO1 N1(C(C2CCC(CC)O2)=O)CCC(F)(C(=O)NCC(C)(C)CSC)CC1 c1(C(N2CCC(C(=O)NCC(C)C(C)(F)F)(CO)C2)=O)c[nH]c2nccc-2c1 c1(CNC(CC2N(C(c3cn(CC)nc3)=O)CCC2)=O)ccccc1C(F)(F)F CCCCCCCCOCC(N1CCN(C(c2cnsc2)=O)CC1CCO)=O CN1CC(CC(=O)NC(C)(C)CCNC(C2COCCO2)=O)c2ccccc21 C(N=c1[nH]c2cc(F)ccc2o1)C1(O)CCCN(C(c2cnn(CC)n2)=O)C1 C(=O)(CC(C(F)F)NC(C1CCCSC1)=O)NCC1(C)CC=CCC1 C(CCCC(=O)NC1(CNC(C2C3CC(=O)CC23)=O)CCCC1)SC c1(C(=O)NCC=CCNC(C(C)(c2ccccc2)OC)=O)cnc(SC)n1C c1(C(=O)NCc2ccc(C(F)F)cc2)cc(Br)cc2[nH]ncc12 c1(CC)cc(C(=O)NC2CC(C(=O)NCCn3cc(CC)cn3)C2)on1 C12(C(=O)NCCCNC(=O)Cc3ccc(F)c(F)c3)CCCCC1CCC2 C=CCCCCCCCCC(=O)N1CCN(Cc2cc(O)ccc2Cl)C(C#N)C1 c1(C(=O)OCC2=CCS(=O)(=O)C2)cc(F)c(OC2CC2)c(F)c1 C=C=CCC(=O)NCC(C)(F)CNC(=O)CCCC1CCCC1 C12(C(CNC(=O)N(C)Cc3csnc3C)OC)CCC(CC1)C2 N1(C(COC)=O)CC=CC(NC(C23CC(c4ccccc4)(CO2)C3)=O)C1 c1(C(C(=O)NCc2ccnn2C)N(CC)CC)cccc(C(C)C)c1 c1(CC(=O)NCC(CN(C(C(C(C)C)CO)=O)C)C)nc2c([nH]1)CCCC2 C1(NC(CCCC=C)=O)COCCN(C(=O)C(C)Cc2cccnc2)C1 Cn1cc(C#N)cc1C(N1CC=CC(C(=O)NCCN2CC=CC2)C1)=O CC1(CNC(=O)C(F)(F)CO)CCN(C(=O)CN2CCN(CCO)CC2)CC1O N1(C(CCCC)=O)CCC(N2CCOCC2)C1C c1(CC)ncc(C(=O)NC(C2(CNC(C3CC34CC4)=O)CC2)C)c(C)n1 C1(CNC(c2c(CC(=O)OC)scc2)=O)COCCN1C(C12CSCC1C2)=O C(C(=O)N1CC(O)CC1CNC(=O)C(F)(F)c1csc(=N)[nH]1)(C(C)C)OC C1(NC(c2cc3ccsc3[nH]2)=O)CCC2CC1CN2C(=O)Cc1nncs1 C(=O)(CC1=NN(C)C(=O)C1)N1C2CCC(NC(CC3CCC(C)CC3)=O)C(C2)C1 c1(SC)ccc(C(N2CC(C(N)=O)(CNC(C3CNC(=O)N3)=O)C2)=O)o1 C1(C(N2CC(CC(C)NC(c3ccc(SC)s3)=O)C2)=O)CCOC(C)(C)C1 Cc1cccc(C(=O)NCC2CCCN(C(C3(O)CCOC3)=O)CC2)c1F C=C1C(NC(=O)N(C)NC(=O)c2cccc(I)c2)CC2CC1C2(C)C C1(NC(c2c(C(C)C)onc2)=O)CC(C2CCN(C(=O)C3CC3)C2)C1 c1(Cn2nc(CC)c(-c3noc(C4CCCO4)n3)c2)nnc2n1CCCC2 c1(C(=O)NCC2N(C(C(Cn3ccc(C)n3)C)=O)CCC2)cc(F)c(O)c(Cl)c1 C(=O)(CC1OCc2cc(Cl)ccc21)N1CCN(C(c2c(SC)nn(C)c2)=O)CC1 Cn1ccc2cc(NC(C3CCCN(S(=O)(=O)c4cccs4)C3)=O)cnc12 C(c1ccc(C)nc1)=CC(=O)NC1C=CCN(C(C2(CSC)CCOCC2)=O)C1 c1(CN(C(c2n(CC)c(N3CC4CC(C)C4C3)nn2)=O)C)ccc(Cl)c(Cl)c1 c12nn(C)nc1NC2=O.n1(C(C(=O)OCC)C)cc(-c2ccncc2)nn1 CCCCCC(=O)N1CCCCC1CCNC(=O)C(N1CCOC(CC)C1)C N1(C(=O)NC(C(CC)(C)C)c2ccccc2)CCCN2C(=O)CCC12C C(=O)(C1=CC2CCC=CCCC12)N(C)CC1CN(C(c2c(C)nn(C)c2Cl)=O)C1 C1(NC(C(C)(C)c2cscc2Cl)=O)COCCN(C(=O)COCCCF)C1 C1(C)(NC(=O)OC)CCN(N2CCSCC2)CC1 C1(C)(COC)CCCC1NC(c1cc(CNC(c2cnc(Cl)n2C)=O)[nH]n1)=O C1(NC(=O)Nc2c(OC)cccc2)CN(C(c2csnn2)=O)CC1C#N C1(C(=O)NCCc2n(C)cnc2)(CNC(C2CC(C)(C)CO2)=O)CC(F)(F)C1 Cc1coc(C)c1C(N1CCC(C)(NC(=O)CSc2nnnn2C2CCCC2)C1)=O CC1CCCN(C(C2CCOCC2NC(c2cc(Cl)cn2C)=O)=O)C1 C1(CNC(C(OCC)OCC)=O)CC2(CO1)CN(C(C13COCC1C3)=O)C2 C1(NC(c2c(C)ccn2C)=O)CN(C(C2CCCN(C(=O)OC)C2)=O)CC12CCC2.C c1(C(N2CCC(CCNC(c3ncn(C)c3)=O)C2)=O)ccc2cccc(O)c2c1 C1(OC)(CNC(=O)CC2CC(C)C2)CCN(C(C2CC(O)C2)=O)CC1 CCC(C)(CNC(c1cc(C)n(C)n1)=O)C(=O)NCc1cncc(F)c1 N1(C(C(C)C2CCCC2)=O)CCN(C(C2CN3CCC2CC3)=O)CC2(CC2)C1 N1(C(c2ccc(C3CC3)s2)=O)CCOC(C2CC2)CC1.C12CCC1C(=O)N2 N1(C(CC(C(C)C)OCC)=O)CC2CCN(C(=O)C(C)(CC)CC)CC2C1 CCC1=C(C(=O)N2CC3CCC(C2)C3NC(=O)CCC(C)OC)CCCO1 CC1(C)C=CC(NC(=O)C(C)(C)C2CCCN2C(C2CCC2)=O)CC1 c1(C2CC(CC(=O)N(CC(C)NC(c3nncn3C3CC3)=O)C)C2)ccccc1 CC1CC(C(=O)NCCN(C2CCCCC2)C(c2cccc(C3CC3)n2)=O)=NO1 C=CC1(C(=O)NCC2OCCC2C(=O)NCC(=O)OC2CC2)CCOCC1 C1(CNC(=O)Cc2csnn2)CN(C(=O)Cc2cccc(C3CC3)c2)C2CC12 N1(C(c2cc(OCC)n[nH]2)=O)CC(NC(=O)CCOC(C)=O)CC2(CCC2)C1 C=CCCCCCCCCC(=O)NCCC(O)CNC(C1CN(C)CCO1)=O N1(C(C=NOC)=O)CC2ON=C(CNC(c3cc(Cl)c4n[nH]cc4c3)=O)C2C1 C=C=CC(C)C(=O)NCc1cccc(NC(=O)C(C)NC(N)=O)c1 c1(C(=O)NC2CC(NC(=O)C=Cc3cn[nH]c3)C2)ccc2nc[nH]c2c1 c1(C2(C(N3CC(N(C)C(C4CC5(CC5)C4)=O)C3)=O)CC2)ccnc(Cl)c1 c1(C(C(=O)NC2CC(NC(C3CC(=C)C3)=O)C2)C)ccc(OC)cc1 N(C)(C(=NCc1ccccc1)NCC1CC2CC1C2)CC(C=C)(F)F Cc1cc(C(=O)N(CC(C)NC(=O)C#CC2CCC2)C)c(C)n1CC(F)(F)F N1(C(C2CCCCS2)=O)CCN(C(c2nc3ccccc3[nH]2)=O)C2CCCC12 c1(C(=O)NC(C(=O)NCCCOC)C)cn(CCNC(C)=O)nn1 c1(C(=O)NC2CC(NC(C3C(C(N)=O)C3)=O)C(O)C2)csc2nccn12 c1(OC)cc(C)cnc1C(N1CC(CCNC(C2CCCCN2C)=O)(OC)C1)=O C(CCCCCC(=O)NCCC1(O)CN(C(C2C(C)(C)C2(C)C)=O)C1)SC N1(C(=O)NCc2ncc(CC)s2)CCC2(CCNC(=O)O2)CC1 c1nc(NC2CCCSC2)cc(N2CCCC(c3n[nH]c(CO)n3)C2)n1 C(=O)(CCC1=NNC(=O)CC1)N(C1CCC(NC(c2csc(C(F)F)c2)=O)CC1)C C(c1ccc(O)cc1)=CC(=O)NC(C)(C)CCNC(=O)CCCC(F)F C(=O)(C(CC)CC)N.C1(CC(=O)NCC2(CC)CC2)(NC=O)CCC1 n1(CC)c(C(=O)N(CC(C)C(=O)NCCn2nncc2C)C)cnc1O CC(Cc1ccccn1)N=c1nc2sccc2c(NCc2ccncc2)[nH]1 Cc1cc(=NCCc2nc(C(C)C)n[nH]2)[nH]c(N2CCC(C)(CO)C2)n1 c1(C(N(CCN(C(c2ccoc2C(C)C)=O)CC)CC)=O)ccc(SC)cn1 c1(C(N(CCC)CCNC(=O)CCNS(=O)(=O)CC)=O)cccc(C(C)(C)C)c1 c1(NC(C(CNC(C(C)N(CC)CC)=O)N(C)C)=O)cc(C)ncn1 C1(C(=O)NCCN(CC=CC(=O)NC(C=C)C)C2CC2)CCCC1C(C)C C(=O)(C(C)S(N)(=O)=O)N1CC2C(CNC(C3(CCC)CCOC3)=O)C2C1 Cc1cc(C(N2CCC(NC(C3CCCCN3N=O)=O)CC2C)=O)c(O)nn1 N1(C(CCCOCC(C)C)=O)CC2(CCC2NC(=O)C(=O)NC2CC2CO)C1 CC1CCC(C)N1Cn1c(N2CCN(C3CCCC3)CC2)nnc1-c1ccc[nH]1 CCS(=O)CC(=O)N(C1CC(NC(=O)CCCOc2ccccc2F)C1)C c1(OCC(=O)NCCSCCCCNC(C)=O)ccc(F)cc1 N1(C(CCN(CC=C)C(C2CCCCNC2=O)=O)=O)CC2CC1C(F)(F)C2 c1(C(C(N2CC(c3cn(C(C)CO)nn3)(C)C2)=O)(C)F)ccc(Br)cc1 c1(C2(C(C(=O)C(CO)CC(F)(F)F)=O)CC2)cccc(Br)c1Cl.N c1(C(N)=O)cn(C)nc1NC(C1N(C(C2(CC#C)CCOC2)=O)CC1)=O CCS(=O)(=O)CC(=O)NCCC1(C)CCN(C(=O)CC(C(C)C)OCC)C1 c1(OC)c(C(=O)NC2CCN(C(c3csc(C)n3)=O)CC2C)cc(F)cc1F C1(C(N2CCC(CNC(C(CC)NC(C)=O)=O)C2)=O)CC2(C1)CS(=O)(=O)C2 c1(OCC)cccc(CCC(N2CC(CNC(=O)Cn3cccc3)C(C)C2)=O)c1 c1(C(=O)OC)ccc(C(N2CC(NC(C3C(C)(C)C3(F)F)=O)C(F)C2)=O)n1C C(=O)(C1CCCc2ncccc21)N1C(C)CC(CNC(C2CNC(=O)N2)=O)C1 C1(CN=c2ccnc(N(C)C)[nH]2)CN(C(=O)OC(C)(C)C)C2(CCCC2)C1 C1(C(N(C(CC)C#N)CC)=O)CCCC(NC(=O)CCC)C1 N1(C(CC2CC(C)(C)C2)=O)CCCCCC(NC(=O)C(O)CC(C)(C)C)C1 CCC(O)C(F)(F)C(=O)NC1CC=C(C(=O)NC(C)CCn2cncn2)C1 c1(C(CNC(CCOCCC)=O)NC(=O)C(C)c2cccs2)cccc(Cl)c1 Cc1ccncc1C(=O)NCC1CC(NC(=O)CC2(C(F)(F)F)CC2)C(O)C1 c1(C(N2CC(C)C(NC(C3CC(=O)N3)=O)CC2)=O)cccc2c1OCCCO2 C12(NC(C(CC)C(C)C)=O)CCC(CN(C(=O)C(F)(F)C(F)F)C1)C2 C1(C(=O)NCC2(O)CN(C(c3ccc(CC(C)C)s3)=O)C2)CN(C)C(=O)CCO1 N1(C(CNC(C)=O)=O)CCC2C(C1)CN2C(c1cccc(N2CC=CC2)c1)=O C1(CC(=O)NC2CC(n3cc(CNC(CCC=C)=O)nn3)C2)C(=O)NN=C1C C1(CCN(C)C(c2c[nH]c(=N)s2)=O)CCN(C(C2CCC3CCC23)=O)CC1 N1(C(c2c(CC)cco2)=O)CC(CNC(=O)CN2CC(C)(OC)C2)CCC1C N1(C(Cn2c(C)nc(C)n2)=O)CCCC2(CCCN2C(=O)C(=O)NCC2CC2)C1 c1(N2CCCCC(C)C2)ccc(Br)c(S(=O)(=O)N(C)Cc2ncn(C)n2)n1 c1(N2CC(NC(CSCCCC)=O)C(C)CC2)nc(Cl)nc(COC)c1COC Cc1c(N)ccc(C(=O)N(CCCCNC(C2CCN(C(N)=O)CC2)=O)C)c1F CC(C)C(C)C(=O)NCc1cccc(CN(C)C(C2CC(C)(C)C2)=O)c1 Cc1coc2ccc(C(=O)NNC(=O)Cc3ccccc3)cc12 N1(C(=O)CSC2CC2)CCC2(CCN(C(C3C=CCCC3)=O)C2)C1 N1(C(C(N)=O)=O)CCN(C(c2csc(C(F)(F)F)n2)=O)C2CCCCC12 C1(C(=O)NC2CC(C)C2)CCCC1CNC(C1(COC(C)C)CC1)=O N1(C(c2c(Br)c(C)n(C)n2)=O)CCC(F)(F)C(NCc2cc(Br)c(O)c(Br)c2)C1 C1(NC(N)=O)CCC(C(=O)NCC2(CNC(=O)CC34CCCC3C4)CC2)CC1 Cc1cc(C)n(CCC(=O)NCC2CC2CNC(=O)C(O)C2CC2)n1 c1(C2(C(=O)NCCCN(C(CCC=C)=O)C)CC2)ccc(OC)c(OC)c1 c1(OC)cc(NC(=O)NC2CCN(CC#N)CC2)c(Cl)c(C(=O)NC)c1 Cc1nc(C2CC2)ccc1C(N1CC(NC(C2OCC2(C)C)=O)CCC1C)=O c1(OCCCOCCCO)nc(-c2ccc(CO)nc2)nn1CC1CCOC1 C(=O)(C(C)(C)CC#N)NC1CC2C(NC(C=Cc3occ(C)n3)=O)C2C1 N1(C(C2CCCN(Cc3cc(F)cc(F)c3)C2)=O)CCN2CC(O)CC2C1 c1(C(=O)NCCCN(C(C2CCCSC2)=O)C2CC2)nccc2[nH]ccc12 C(N=c1nc2c(cnn2C)c(N(C)CCn2cccn2)[nH]1)c1[nH]nc(C(C)C)n1 C(C(=O)OC)(C(C)CC1CCOCC1)N(CC(=O)NCCSC)CCC c1(C(N(CC(C)N(C(CCC#C)=O)C)C)=O)cc(C(F)(F)F)cnc1OCC N1(C(Cn2c(C)nc(C)n2)=O)CCC2(CC2C(=O)NCC2CC23CC3)C1 c1(C(=O)NCC2(C(N3CCN(CCO)CC3)=O)CC2)cc(Cl)ccc1Cl C(=O)(CC(F)(F)F)NC(c1cccnc1)C(=O)NC(c1ncc(C)[nH]1)(C)C C1(NC(CC2(C)CC2(F)F)=O)CCN(C(C23CC(CO)(C2)C3)=O)CC1(C)C C1(NC(CNC(C)=O)=O)CCCC(NC(=O)CNC(=O)CCC2CCCC2)CC1 c1(COC)cc(C(=O)NCCC2(NC(c3csc(CO)n3)=O)CC2)on1 N1(C(C(CC)C)=O)CCC2(CC1)CN(C(=O)C(C(C)OC)N(C)C)CCO2 C(C(F)(F)C(=O)N1CCC1CNC(c1cnn(CC(C)C)c1)=O)OC C1(NC(c2cc(CCC)ncc2)=O)COCCN(C(=O)Cc2nc(C)sc2C)C1 CC(CC(=O)NC1(CO)CN(C(c2ccnc(C3CC3)c2)=O)C1)C(F)F c1(C(=O)OC)ccn(CC(F)(F)F)n1.C(=O)(CC1CCC1)NCC=CCN c1(OC)ccc2cc(NC(C3CCCC(c4cccnc4)C3)=O)ccc2n1 c1(C(=O)NCc2cc(CNC(=O)CC3CC3C(F)(F)F)co2)c(F)cccc1F C1(CNC(C2CCC(=O)N2)=O)C2CN(C(c3cnnc(O)c3)=O)CC12 c1(COCCNC(C(c2cccc(F)n2)N(C(C)C)C2CC2)=O)ccc(F)cc1 C1(C(N2C(C)CCN(C(C(C(C)C)SCC)=O)CC2)=O)CCCC2(C1)CC2(F)F C(=O)(C(C)(F)C(F)(F)F)N(CC(CC)NC(=O)CCc1ccc(Cl)cc1)C C(=O)(C1=CCCN(C(=O)CCCn2cncn2)C1)NCC(N1CCCC1)C N1(C(C(N2CCCCC2)C)=O)CC2CN(C(=O)C(C)(C)c3ccnn3C)CCC12 C(=O)(C1CCCn2ccnc21)NC1CCC(NC(C(C(C)C)(C)O)=O)CC1 N1(C(c2c(C)n[nH]c2C)=O)CCC2(COC(CNC(c3nnn(C)n3)=O)C2)C1 C#CCC(C)(C(=O)NCc1ccsc1C)NC(=O)Cn1ncn(C)c1=O N1(C(=O)OC)CCN(CCCNC(=O)CC2CCN(C)C2=O)CC1C(C)C c1(OC)ccc(C(N2CCCC2C2(NC(C3CC3(F)F)=O)CC2)=O)cc1Cl N1(C(c2ccc(CC)s2)C(=O)NCC(C)C)CCOC(CC(C)C)C1 O=[N+]([O-])c1cc(-c2noc(-c3cnc(-n4cccn4)s3)n2)co1 C1(NC(C2C(C)(C)C2C#N)=O)CCN(C(=O)CCCNC(N)=O)CC1C(N)=O c1(C(N(CC(C)(C)C)CCN(C)C)=O)csc(-c2ncc[nH]2)n1 C1(O)(C(CNC(C(=O)NCC)=O)C)CCN(C(=O)CCC2CCCC2)C1 C(CCCCC(=O)NCCC1COCCN1C(=O)C(O)C=CC)=CCC=C N1(C(Cc2c(C)nc(C3CC3)s2)=O)CCC2CN(C(=O)CCC(C)(C)C)CC2C1 CC1c2ccccc2OC1C(N1CC(NC(=O)CC2(O)CCCCC2)C(O)C1)=O N1(C(C(CC)OC)=O)CCCCC(CNC(c2ccc(C(N)=O)nc2)=O)CC1 Cc1[nH]nc(C(=O)NCCC2CC(NC(C3(C4CCCO4)CC3)=O)C2)c1F CC(CS(C)(=O)=O)C(=O)N1CCC(C(F)CNC(=O)C=CC=C(Cl)Cl)CC1 CCCCCC(O)C(=O)N1CC2(CC(CNC(=O)CC3C=CCC3)C2)C1 C12(C(=O)OC)CCCC1N(C(=O)C(F)Cl)CC2 N1(C(c2ccc(OC(CC)C)cc2)=O)CCC(NC(=O)CSC)C(F)C1 C#Cc1ccc(C(=O)NC2CCC2NC(c2cn(C)nc2C(C)C)=O)cc1C c1(OCC)ccc(F)c(CNC(N2CCC2CC(C)C)=O)c1 N1(C(C=CC)=O)CCC(CO)(CNC(C2CC3CC3C2)=O)C1 Cc1ccc2c(=NCc3cc(C(C)C)no3)[nH]c(=NCC(C)C#N)[nH]c2c1 Cc1cc(Cl)c(C(=O)N(C(C)CNC(c2cnsn2)=O)C)cc1C C(C(C)NC(c1cccn1C1CC1)=O)(C(C)C)NC(C=CC(CC)=CC)=O C=CCC(CC)C(=O)NCC1CC(NC(c2cncc(NCC)c2)=O)CCO1 C1(NC(CNC(C=C)=O)=O)CC2(C1)CC(C(=O)NC(c1cccnc1)C)C2 C1(C(=O)NC(COC)C2CC2)CC12CCN(C(=O)Cc1cncnc1O)C2 CCCC(CC)C(=O)NCc1cn(CC(C)NC(=O)CC2CC=CC2)nn1 C1(CNC(C=NOC)=O)CCN(C(C2CCN(CCS(N)(=O)=O)CC2)=O)C(C)C1 S(=O)(=O)(c1ccc(C(C(=O)OCC)NC2CC2(Br)Br)cc1)NC c1(C(N2CC3C(NC(C(C=CCC)O)=O)C3C2)=O)ccc(O)c(Cl)c1 CC(C(=O)N1CC(C)(C(=O)NCC2CNC(=O)O2)C1)C(F)F N1(C(C(C)(C)C2CCCO2)=O)CC(CCNC(=O)Cc2cccnc2)C(C)C1 c1(C(N2CCCC(NC(C3(CN(C)C)CC3)=O)C2)=O)cc(Cl)ccc1C(F)F c1(C(=O)NCC=CCNC(c2cc(OCC)ns2)=O)c(C)cnn1C(C)C C1(NC(CCC=CC(C)C)=O)CCC(C)N(C(C2CN3CCN2CC3)=O)C1 CC1CCC(CC(=O)NC2(C)CN(C(=O)Cn3cc(C#N)cn3)C2)OC1 N1(C(=O)OC(C)(C)C)Cc2cccc(Cl)c2C1.CC1C2CCCN1C2=O C(=O)(C1=C(Cl)CCCC1)N1CCN(C(C(COCC)C)=O)CC1CC c1(C(N2CC(CCC)N(C(=O)C(C)CN(C)C)CC2)=O)cc2ccc(C)cc2[nH]1 c1(C(N2CCC3CN(C(CCS(C)(=O)=O)=O)C3C2)=O)cccc2ccncc12 C1(C)(CNC(C2(CC=C)CCCC2)=O)CN(C(=O)CC(C)n2ccnc2)CC1C c1(C(N(C(C)CN)C)=O)c(Cl)ccc(I)c1F Cc1ccc2c(c1)C(NC(=O)C(=O)NC(C)CC(C)(C)c1ccccc1)C(C)C2 C(C(=O)NCCC1CCCN1C(c1ccnc(C(=O)OC)c1)=O)(C(C)C)OC C1(C(F)(F)F)(C(=O)NCC2C(NC(C(C)=C(C)C)=O)CCC2)CC2C=CC1CC2 CC1=C(C)CC(C(=O)NCc2nocc2C(=O)NCC2CC2(F)F)CC1 N1(c2n(Cc3cccc([N+](=O)[O-])c3F)nnn2)CCC12CCCS(=O)(=O)C2 C(=O)(C(F)(F)C(O)C(C)C)NC1C(NC(c2cc(CC)on2)=O)COCC1 N1(C(C=CC)=O)CCC2(NC(=O)CS(=O)(=O)CCC)CCCC12 C(C(C)(C)CCC#N)N(C(C=CCCC)=O)C.C1C(C(C)CC)N1 C1(C(N(C2CCC(C(=O)N(CC(O)C3CC3)C)CC2)C)=O)CC(O)C(F)C1 c1(NC(CC2N(C(c3c(SCC)cccc3)=O)CCOC2)=O)c(C)ccnc1Br C(=O)(C(C)S(N)(=O)=O)NC1CCCN(S(Cc2cccc(C)c2)(=O)=O)C1 C1(NC(C#CCNC(C2C(OC)(OC)CC2)=O)=O)CCCCN(C)C1=O C1(C(=O)NC2C(OC)CCC2)CN(C(c2[nH]ccc2C2CC2)=O)CCC1(C)C c1(C(=O)NC2CCN(C(C3(C)CCC3)=O)CC2F)ccc(P(C)(C)=O)nc1 N1(C(CCC(C)N(C)C)=O)CCC2(CCCC2NC(=O)C(C)(F)C(C)(C)F)CC1 c1(CNC(=O)CSCCNC(=O)CC23CCCC2C3)ccnc(O)c1 C1(NC(C2(CC)CC2)=O)CN(C(C2CCC2(C)C)=O)C2CCCCC12 c1(OC)ncc(C(=O)NCC(C)CNC(C2CCOC2C)=O)nc1C N1(C(C2(OC)CCC2)=O)CC2CC(C1)C(CO)C2NC(C1CCCCC(=O)N1)=O O=S(=O)(c1cnn2ccccc12)N1CCC2(CCCC(CO)O2)C1 C1(NC(CN(C)CCO)=O)CCC(N(C(=O)CCc2cnc(C3CC3)o2)C)C1 N1(C(C(c2ccc(C)cc2)C)=O)CCN(C)CC1CNC(c1cccn1C)=O N1(C(CC2(NC(CSCCC(C)C)=O)CC2)=O)CCCC12CCOC2=O c1(CNC(=O)NCC(=O)NC2CC2C(F)F)cccc(-n2cccn2)n1 C1(NC(c2ccco2)=O)C2COCC1CN(C(C1CC13CCCC3)=O)C2 C(c1cn(C)c2ccccc12)=CC(=O)N(C1CC1)Cc1cc2cc(C)[nH]c2cc1 CC1(C)CCCC(C(=O)NC2CC(NC(=O)COCc3ccnc(O)c3)C2)O1 C1(CNC(c2sccc2F)=O)C2CN(C(c3cc(-c4ccccc4)co3)=O)CC12 CCCC(CC)C(=O)N1CCN(C(=O)CC23CC(C2)C3)CC1CO Cc1oc2cc(C(C)N(C(=O)C3CC3)CC3CCOC(C(F)(F)F)C3)[nH]c2c1C N1(C(c2[nH]cc(CC)c2)=O)CCC(CNC(=O)Cc2cc(F)ccc2C)C(C)C1 CC(C(=O)NCCCOCC(C)(C)NC(c1cnccn1)=O)C(C)S(C)(=O)=O Cc1cc(CNC(C23CC(C(=O)Nc4ccnn4CCO)(C2)C3)=O)c(F)cc1Br Cc1cc(C(N2CCCC3CC23CNC(c2sccc2Cl)=O)=O)cc(=O)n1C CCCC(C(=O)N1CC2C(CNC(=O)CN3C(=O)CNC3=O)C2C1)C(C)C Cc1cc(CC(=O)N(C(C)CNC(=O)CCN2CCCCC2)C)cs1 C(=O)(C(C)C(C)C)NC1(COC)CN(C(=O)C(O)CCN(C)C)C1 C=CCCC(C)(C)CNC(=O)C(O)C1CN(C(c2nc(C)c(C)s2)=O)C1 c1(C(=O)NC(CC(C)NC(c2cc(C)nnc2)=O)C)cc(Cl)ccc1C(C)C CCC(C)(CO)C(=O)NC1CC(C)(NC(c2cn(CC3CCOC3)nn2)=O)C1 C1(CCOC)(NC(=O)CC2(CNC=O)CCCC2)CCCC1.C1CC(OCC)C1 C1(NC(C(F)=C(C)C)=O)CN(C(c2ccnc(O)c2)=O)CC1C N1(C(CC(CC)C2CCC2)=O)CCC2(CC1)CC2NC(c1nsnc1O)=O Cn1nc(Br)c2ncnc(N3CCC(C)(C)C(CNC(=O)CN4CCCC4)C3)c12 Cc1ccc2nc(C(=O)NCC(O)CN(C)C(C3CC(CC4CC4)C3)=O)cn2c1 C=CCC(C(=O)N(C)CCNC(c1cccc(-n2c(C)cnc2O)c1)=O)C(C)C c1(NC(C2(C)CCCN(C(=O)Cc3cccs3)C2)=O)cc(Br)cnc1[N+](=O)[O-] C1(NC(C2C(C)(CC)C2)=O)C2CC3CN(C(c4cc(C)cc(C)c4N)=O)C1C3C2 c1(C(CN(C(C=CSC)=O)C)O)cc(Cl)cc(Cl)c1 C1(CN2CC(O)(CNC(c3n(C)cnc3)=O)C2)CCS(=O)(=O)CC1 N1(CC)CCC(NC(=O)CCCNC(=O)CC2CCCSC2)CC1 CC(C)CCCCOc1cccc(CNC2COC(=O)N2)n1 N1(c2nc(C)nc(NCC3CCCC4(CCC4)O3)c2)CCCc2[nH]c(=N)[nH]c2C1 C1(C(N(C2CCN(C(c3cc(C4CC4)on3)=O)C2)CC)=O)CCOC2(CCC2)C1 N1(C(COCCC)=O)CC(N(C)C(c2cc(F)ccc2O)=O)C(C)(C)C1 C(=O)(N=c1cccn[nH]1)c1csc(NCc2nn(C)c(C(F)(F)F)n2)n1 C(CC(=O)OC)(N=c1ccn(Cc2ccccc2)[nH]1)c1n(CC)nnn1 N1(C(C2(CC)CCC2)=O)CCC2(CCCN2C(c2ncn3ccccc23)=O)C1 C1(CCC(=O)NCC(C(C)C)NC(COCC(=O)NC)=O)CCC(C)NC1=O C12(C(=O)NCc3c(C)ccnc3C)CCCC1N(C(=O)C=CC(=O)N(C)C)CC2 C12(CNC(c3cc(C)n(C)c3)=O)COCCN1CCN(C(=O)C=CC(F)(F)F)C2 N#Cc1c[nH]c(=NCC2CCCC(O)C2)c2sccc12 c1(CNC(N2CC(CS(C)(=O)=O)C2)=O)ccc(Cl)cc1.c12cnc(s1)s2 Cc1ncc(-c2ccccc2C(CC(=O)O)NCc2ccc(Br)cc2F)c(=N)[nH]1 N1(C(C(=O)N(C2CCN(C(CCCN(C(C)=O)C)=O)C2)CCO)C)CCOCC1=O N1(C(C2(NC(C3CCC4(CCC4)C3)=O)CCSC2)=O)CCC(F)C(F)C1 C1(CC=C)(NC(=O)CC2C=CCC2)CCCN(C(=O)CC=CC)C1 c1(C(=O)NCCCN(C(=O)CC2CC(CF)C2)CC)cc(O)ccc1[N+](=O)[O-] C1(C(=O)NCCN(C(CC(C)CF)=O)C)CCC(C)(O)CC1 C(=O)(C1=C(Cl)CCOC1)N(C1CC(NC(=O)C(c2cccc(Br)c2)O)C1)C N1(C(CN(C(C(C)C)=O)C)=O)CCC(NC(C23CCC(C2)C3)=O)CC1C1CC1 CC1CCC(C)(C(=O)NCC2(NC(=O)C3=NOCC3)CCCCC2C)C1(C)C C1(C(=O)NCC(c2cnc[nH]2)C)CC=CCN1C(=O)Cn1[nH]cnc1=N CC1(C)CCCC(C(N2CCN(C(=O)CCc3cncc(O)c3)C3CC23)=O)O1 c1(C(CN(C(=O)CC23CC(C2)C3)CC)(C)O)ccccc1.C12CCN1C2=O N1(C(C=CCN(C)CC)=O)CCN(C(=O)CN(C2CCC2)C)C(CC(F)F)C1 N1(C(C(CC2CCCCC2)OC)=O)CCC(C)(NC(=O)CCc2cnoc2)C1 C(=O)(CC(C)(F)F)N(CC(C)O)CCNC(C(CC)NC(N)=O)=O C=CC1CN(C(=O)C(C)(C2CCC2)NC(c2ccc(C)c(C)c2)=O)CCO1 c1(CC)ccc(Br)cc1.c1(C(=O)NCC2(CN3C4CC(C4)C3)CC2)cnn(CC)c1 N1(CCNC(CN(C(=O)CCc2ccon2)C(C)C)=O)CCCCCC1 C12(C(=O)NC3CC(NC(c4cccc(C(F)(F)F)c4)=O)C3)CCCN(CC1)C2 [N-]=[N+]=NC1CCC(C(=O)NCC2(CNC(C3CCCC(=O)N3)=O)CC2)CC1 C(c1cscn1)=CC(=O)NCCOC(CNC(C1C(C(C)C)(CC)C1)=O)(C)C C(=O)(C(C)(C)CCNC(C)=O)N(CCCCN(C(C1C(OCC)C1)=O)C)C c1(OC(C(=O)NCC(N(C(C2CC(=C)C2)=O)C)C2CC2)C)ccc(Cl)cc1Cl C1(CC(N2CC(C(C(=O)NCC3CC(OC)C3)O)C2)=O)CC1C1CC1 c1(CNc2c(Br)ccc(C(=O)O)c2)cc2c(s1)CCNC2 C1(NC(c2cc(COC)on2)=O)CCCCC1C(=O)NC1CC1CCF c1(C(=O)NC(C2CN(C(=O)CCC3CCCCO3)C2)C)ccnc(Cl)c1N c1(C(=O)NC2(C)CC(NC(C3N(C)CCOC3)=O)C2)nc(O)nc(O)c1N N1(c2n(CC(OC)OC)c(C(C)OC(C)C)nn2)CCCC2(CCC2)C1 C1(CNC(CC(CC)C)=O)CN(C(c2cnc(C(C)(C)C)[nH]2)=O)C(C)(C)C1 C1(CNC(CN(C(C(C)C)=O)C)=O)CN(C(C2CCOC2)=O)CC12CCC2 C(=O)(CS(C)(=O)=O)NCC(C1CCCN1C(=O)CCn1ccnn1)(C)C c1(C(=O)NCC(C)NC(COC(CC)C)=O)cccn2nnnc12 N1(C(c2c(COC)cccc2)=O)CC(C)N(C(=O)C(C)(F)F)CC1C CN(C(=NCC(CCO)C1CCCC1)NC1CC1)CCC1CCCCC1OC(F)F N1(C(C(C)(C)OC)=O)CCC2(CCN(C(=O)CNC(=O)CCCCO)C2)C1 C#CCC(C(=O)N(C)CCN(C(c1ccc(C(F)(F)F)[nH]1)=O)C(C)C)C1CC1 N1(C(c2cn(C(C)C)nn2)=O)CCC(N(C(=O)CC2(O)CCOC2)C)C2(CC2)C1 CON1CCC(C(=O)NC2CCCC(NC(=O)C(=C3CCCCC3)F)CC2)CC1 C(=O)(C(C)(C)C1CCCN1C(=O)CCC1(C#N)CCC1)NC(C1CSC1)C N1(C(C2(C)CC(=C)C2)=O)CCC(F)(Cc2cn(CCC3CC3(Cl)Cl)nn2)C1 c1(C(C)Nc2cc(N(CCCSC)C)nc(C)n2)nnc2n1CCCC2 C1(NC2CN(C(=O)OC(C)(C)C)OCC2)C(=O)NCC12CCCO2 c1(CC(=O)NCC(C)N(C(=O)C(F)F)C)ccoc1 C(N=c1[nH]c(=NC2CCSC2)c2[nH]ccc2[nH]1)c1cc(C(C)(C)C)ncc1 c1(C(=O)NCCC(C)NC(C2C(=C)C2)=O)cnc(N2CCOCC2)s1 N1(C(=O)NCc2cc(F)ccc2Br)CCC2(CCCC2Cc2ccc(O)cc2)C1 Cc1cc(O)c(C(N2CCN(C(=O)CCc3nnc(C)n3C)C(C)C2)=O)cc1Br C#Cc1cnn(C)c1C(=O)NCCCN(CCO)C(c1cocc1C)=O c1(OCC)ccc(S(=O)(=O)N2CCOCC2C(=O)NCC(C)CC)cc1OC C(C(C)(C)CC(=O)N1CCC1CNC(=O)Cc1ncc(C)s1)OC C(CS(=O)(=O)CC(=O)N1CC(NC(=O)Cc2ccsn2)CC2(CC2)C1)OC c1(NCC2CC(C(N3CCC(O)C(O)C3)=O)C2)cc(F)c(F)cc1Cl N1(C(=O)NCC(C(C)(C)O)(C)C)Cc2cccc(C#N)c2C1 N1(C(C2C(CC)CN(C(c3ccc(C(N)=O)[nH]3)=O)C2)=O)CC2CCCC(O)C2C1 c1(OC)ccnc(C(c2nnnn2C2CCCC2)NCc2ccc(Br)cc2)c1C c1(C(=O)NCc2nccnc2Cl)c[nH]c2ncc(-c3ccco3)cc12 CC(C)CC(C)(O)C(=O)NCC(CC(N1CCC2(CCSC2)C1)=O)C1CCC1 C1(CNC(c2ccc(C(N)=O)[nH]2)=O)CCCN(c2nnc(C(N)=O)s2)C1 C1(C(=O)Nc2ccc(OC)nc2Br)CC(N=c2nc[nH]c3[nH]c(Br)cc23)C1 O=C(OCC(F)F)C(F)(F)CCNC(=O)Cc1ccc(O)nc1 CCC(F)(F)CC(=O)NCC(C)CNC(C1CN(C(=O)N(C)C)C1)=O.OCC Cc1cc(=NC(C)CC#N)[nH]cc1S(=O)(=O)NCCN1C(=O)c2ccccc2C1=O Cc1c[nH]cc(Br)c1=NC(=O)c1csc(-c2ncc3ccccn23)n1 Cc1noc(C)c1C(=O)Nc1nc(CC(N2CCOC(C)C2)=O)cs1 C(=O)(C1=NNC(=O)CC1)N(CC(CC)NC(=O)COc1ccc(C)cc1F)C C1(C)(OC)CCCN(c2nnc(Cc3cccc(C)c3Cl)n2C)C1 C1(NC(C(C=C)O)=O)CN(C(c2ccc(Br)cc2CC#N)=O)CCC1CO Cc1c(F)ccc(C(=O)NCCCCNC(=O)C=Cc2cn[nH]c2)c1C#N C1(C(=O)NC(CNC(C=C(C)C(C)(C)C)=O)C)CCS(=O)(=O)C(C)C1 C(=O)(N=S(C)(=O)CC1CC(=O)N(C)C1)c1c(C(C)C)onc1 C(=O)(C(CNC(c1ccc(O)c(F)c1)=O)CC(C)C)NC(C=C)C(F)(F)F C1(F)(CNC(C2COC2)=O)CCC(NC(c2cn(-c3ccc(F)cc3)nn2)=O)C1 c1(C(N2CCC(N(C(CC(C)(C)C)=O)C)C3(C2)CC3)=O)nc2cc(F)ccc2s1 Cc1onc(C(N2CCCCC2CNC(=O)Cc2cnn(C)c2)=O)c1Br Cc1cc(C#N)nc(N2CCN(CC(N3CCCC(C)C3)=O)CC2)n1.C(C(C)C)N N1(C(c2ccc(OC)nc2)=O)CCC2(CCN(C(=O)C(Br)=C(C)C)CC2)C1 c1(NC(C)=O)cc(F)c(F)cc1-c1ccnc(C(=O)Nc2cncc(CO)c2)c1 CCCCC(C)(CO)NC(C1CC2CCC1N2C(=O)CC(=O)N(C)C)=O C(=O)(C1=CCCOC1)NCC=C1CCN(C(CCN(C2CCCCC2)C)=O)CC1 Cc1[nH]c2ccc(C(=O)NC(C)CC3CN(C(C4CCC(F)C4)=O)C3)cc2c1C Cn1ccc2cccc(C(N3CCC(F)(CNC(C4CC4(F)F)=O)C3)=O)c12 C1(C(=O)NCc2ccco2)CC12CCN(C(=O)CCc1cccnc1F)CC2 c1(C(=O)NCCC2CN(C(C(C)N(C(C)=O)C)=O)C2)ccnc(CO)c1 N1(C(c2c(C)nc(CC)o2)=O)CC2CCC(NC(=O)Cc3csc(C)n3)CC2C1 C=C=CCC(=O)NC(C)CN(C)C(c1cc(-c2cnccn2)[nH]n1)=O C12(C(=O)NCC3N(C(C4C(CC)OCC4)=O)CCOC3)CC1COC2(C)C C1(CNC(CN(C(C)=O)C)=O)CN(C)CCN1C(c1n[nH]c(C2CC2)c1Cl)=O CCCCC(CC(=O)N1CCNC(=O)C1CCO)NC(c1cc(O)n(C)n1)=O c1(C(=O)NC2C(C(=O)NCCOC)C2)ccc(F)c(S(=O)(=O)N2CCOCC2)c1 N1(C(C2CC(SC)C2)=O)CCC(NC(c2ccn(C)c(=O)c2)=O)CC1C1CC1 c1(CC(=O)NC(CN(C(C2(CC)CCCCC2)=O)C)C)cc(C)cc(Br)c1 Cc1nn(C)c(C)c1-c1cnc(CNC(C2CC3CCC2O3)=O)nc1 C1(C(=O)NCC(C)F)C2CCCC2CN1C(C1CC1(C)C(F)F)=O C1(CC)C(NC(C2CN(c3ncco3)C2)=O)CCCN1C(c1cc[nH]c1)=O C1(CC(=O)NCCC2CC(C(=O)NCC(NOCC)=O)C2)COCCOC1 N1(C(C23CC(C2)C3)=O)CCC(C(=O)NCc2ccc(Br)nc2)C(O)C1 C1(OC)CN(C(=O)CCn2cc(C)cn2)CC1NC(c1cc(C(F)F)nn1C)=O CCC(C)C(=O)C(=O)N(C)CCOCCNC(=O)C(COC)NC(=O)OC c1(C(C)C)ncc(C(=O)N(C)CC2(CNC(C3(C#N)CC3C)=O)CC2)[nH]1 Cc1cc(C)c(C(N2CC(NC(c3n[nH]c4c3CSCC4)=O)C(F)C2)=O)cc1C Cc1cc(C)n(CC(=O)N(CC(=O)NC(c2ncc[nH]2)C)C)n1 c1(C(=O)NCC(CO)NC(COc2cn(C)nc2)=O)ccn2nccc2c1 CC(C)CC(CNC(=O)CN1CC2CC2C1)C(=O)NCCc1csnn1 Cc1nc2cc(C(N3CC4(C)CCC4(NC(C4CC=CCC4)=O)C3)=O)ccc2s1 C1(NC(c2n(CCC)ccc2)=O)CCCC(NC(C2COC(=O)N2)=O)C1 C1(NC(C2C(C)=C2)=O)CCCC12CN(C(C13CCC(N(C)C)(CC1)CC3)=O)C2 c1(C(=O)NC2CC(C)N(C(=O)CC3CC(F)C3)C2)cnc2c(c1)CCCO2 Cc1nc(C(=O)N(C(c2cccnc2)C)Cc2ccccc2)[nH]c1C C(=O)(C1Cc2ccc(Cl)cc21)N(C)CC1CCN(C(c2csc(C(N)=O)n2)=O)C1 N1(CCC(CCC)C)CCC2(CC1)CC2C(=O)O.C(=O)C(C)SCC c1(CC2(NC(c3ccc(C4CC4)o3)=O)CCC2)ccncn1 Cc1cc(Sc2ccc(CN)cn2)cc(O)c1 c1(C(=O)NC2(C)CCCC2O)cc(C2(NC(=O)OC(C)(C)C)CC2)cc(O)c1 c1(C(N2CCN(C(c3c(OC)nccc3)=O)C(C)C2)=O)[nH]nc2ncnc(O)c12 C1(CC(=O)NC2(C)CN(C(=O)CNC(=O)CCCC#N)C2)CN2CCC1CC2 c1(C(=O)NCCCCCN(C(c2cc(C(C)C)on2)=O)C)ccncc1F N1(C(CN(C)C)=O)CCC(NC(C2(C(F)(F)F)CCCC2)=O)C(C(N)=O)C1 c1(C(C)=O)cc(S(=O)(=O)NC2COC3(CCC3)C2)oc1C C(=O)(C1=C(Cl)CCC1)NCC1OCCN(C(C2C(c3c(C)cccc3)C2)=O)C1 C1(COC(Cc2c(C)cc(Br)cc2)=O)C2CCCC(F)(F)C12 N1(C(C(C)(C)OCCC)=O)CCCC(NC(c2cnoc2C)=O)CC1 CCCC(CC)CC(=O)NCC1(C)CN(C(c2ccccc2C#N)=O)CCO1 C12(NC(c3cc(F)ccc3Cl)=O)CCCN(C(=O)CSc3cccc[n+]3[O-])C1C2 C1(CCNC(=O)CCC2CC2)CCCN(C(C2SCCS2)=O)CC1 CCC(CNC(c1cc(OCC)no1)=O)N=c1[nH]n2cc(C)nc2s1 c1(NC(c2n(CCCSC)nnn2)c2cnc(C)s2)cccc(-c2cnco2)c1 C1(C(=O)NC(c2ncnn2C)C)CC2(CCC2)CN1C(C12CCCC1C2(F)F)=O C1(NC(c2n(CC)nnc2C)=O)CN(C(c2cnc3n2CCC3)=O)CC1C1CC1 c1(CC)csc(CNC(=O)N(C)Cc2cccs2)c1 C1(F)(C(N2CCC(c3cccc(C)c3)C2)=O)CN(C(C(C)(C)C)=O)CC12CCC2 O=C(O)C1CN(S(=O)(=O)Cc2cccc(Cl)n2)Cc2n[nH]cc21 CC(CC(C)C(F)F)NC(=O)C(C)(C)CNC(c1ccc(Cl)cc1)=O N1(C(c2nc(CCOCC)oc2)=O)CCCC(NC(=O)C(O)C(C)C)CC1 C(=O)(CN=S(C)(C)=O)N(CC(C)O)CCNC(c1ncsc1-c1ccccc1)=O c1(C(NOCC(=O)N(C(C)C(C)(C)C)C)=O)cncc(Cl)c1 c1(C(=O)NCCCCCNC(CC2C(C)CCC2)=O)ccc(O)cc1F c1(C(=O)NC23CCCN(c4nnc(C#N)s4)CC2C3)c(Br)ccc2ccccc12 C#CC1CN(C(c2cnc(C(C)=O)s2)=O)CCN1C(C1CC2(CSC2)C1)=O C12(NC(CS(C)(=O)=O)=O)CCCCC1N(C(C1CC(=C(F)F)C1)=O)CC2 Cc1nc(C)c(C(=O)NCC23CC(CO2)N(C(C2CCCS2)=O)C3)nc1C CC1=C(C(=O)N(C(C)CN(C(=O)CC(C)C2CCCCC2)C)C)COCC1 CC(CC(F)F)C(=O)NCC1CN(C(c2cnc(-c3cnccn3)s2)=O)CCO1 C1(NC(C2(C(C)O)CC2)=O)CC2(C1)CC(NC(C1CC1C)=O)C2 C1(C(=O)NC(C)C(=O)NCC2(C)CCCOC2)CC2(C1)CC21CC1 O=C(C1=CCCN(C(C2(O)CCCCCC2)=O)C1)N1CCC2C(C1)C2(F)F C=Cn1nncc1C(N1CCC1CNC(c1cnn(-c2cccc(Cl)c2)n1)=O)=O Cc1cc(Cl)c(C(N2CCC(CNC(=O)CNS(=O)(=O)N(C)C)CC2)=O)cc1F N1(C(c2c(C)noc2C)=O)CCOC2(CCCN(C(c3cc[nH]c3C)=O)C2)C1 C(=O)(C1=CCC(C)(C)CC1)N1CC(N(C(c2occ(C)c2)=O)C)C(O)C1 C1(CNC(C2(n3cc(-c4cncs4)nn3)CCCOC2)=O)CC(O)C12CCC2 N1(CC(C(=O)OC)N)CCSC(CC(F)(F)F)C1 Cc1ccc(SCC(N2CC(CCNC(C3CCC3n3ccnc3)=O)C2)=O)cc1 C(=O)(CC1=NNC(=O)C1)N1CCN(C(CC(CC)C2CC2)=O)C(C(C)C)C1 N1(C(c2nc(C(C)C)oc2)=O)C2CCC(C(=O)NCCC(C)(C)C)C1CC2 C1(C(=O)NCCCC)CC=CCN1C(=O)C(C)c1cc[nH]n1 C1CC(=O)O1.C1(C(=O)OCC)CN(C(=O)C(C)NC=O)C1.C12(CC1)C(=O)NC2.NC c1(C(=O)NCC=C2CCN(c3cc4nncn4cn3)CC2)cnn2ccccc12 N1(C(c2c(C)nn(C3CCOC3)c2)=O)CC(NC(c2scnc2Cl)=O)C(C)(C)C1 C(=O)(CC(C(F)F)NC(c1cnn(C)c(=O)c1)=O)NC(c1cnn(C)c1)CC c1(CN(C2CCSC2)C)[nH]nc([N+](=O)[O-])c1Br c1(C(=O)NC2CCN(C(CCOCC)=O)CC2C)[nH]c2ccc(OC)cc2c1C c1(-n2cc(C3N(C(c4snnc4C4CC4)=O)CC=C3)nn2)c(Cl)cccc1Cl c1(C(N2CCC(C)(NC(c3c(CC)scc3)=O)C2)=O)ccnc2ncccc12 C1(NC(C2C(C)C2)=O)CC(c2ccccc2)CN(C(c2c(C)cccc2F)=O)C1 c1(C(=O)NC2CCN(C(C(c3ccccc3)C)=O)CC2C)ccc2nonc2c1 Cc1cc2c(CC(=O)NCCC3CC(NC(c4cc(O)ncn4)=O)C3)csc2s1 Cc1ccc(CCNC(=O)NCC2(c3c(C)cccc3C)CC2)c(Br)c1 C1(CC(=O)N(CCC(C)NC(COCCC#C)=O)C)CCC(=O)N1 c1(C(N(C2CC3CN(C(C(C)OC)=O)C2C3)C)=O)c[nH]c2cccc(F)c12 CC1CCC(C(N2CC(OCCNC(c3cc(Br)no3)=O)C2)=O)C1 C1(C)CC(C)(C)OCC(=O)N1.N1(C(C)=O)CC(C(=O)NCC(=O)N(C)C)C1 N1(CC(c2c(F)cccc2F)C)CCC(=O)N(CC23CCCCC2C3)C1=O CC1(C)CCC=C1C(=O)N1CC(NC(c2ncccc2Br)=O)C(O)C1 C1(CC(=O)NCC2C(CNC(c3nc(C)sc3)=O)C2)(OC(C)C)CCCSC1 C#CC1CCCN(C(=O)C(Cc2ccccc2CNCC2CCCO2)CC)C1 c12cc(ccc1C)C(=O)N2.C(=O)(C(C)CC(C)C)NCC1OCC(C(C)=O)C1 c1(NCCS(CCOC)=O)cc(OC)c2c(c1)CCCO2 N1(C(C2C(CNC(C(C)=CC(C)(C)C)=O)CC2)=O)CC(CO)C2(CC2)C1 CC(CC1CC1)C(=O)N(C1CN(C(=O)CC2CC2)C1)C N1(C(c2c(C)cco2)=O)CCC(C)(C(=O)NCC2=NOC(C)C2)C1 C=C=C(C)CC(=O)N1CC2C(CNC(=O)C(C)(C)CC3CC3)C2C1 C1(CNC(c2onc(C)n2)=O)CCCCC1NC(c1cc(C)ncn1)=O N1(C(C2(COC)CCOC2)=O)CCN(C(=O)Cn2ccnc2C)CC12CCC2 CCCCCCCCOCC(=O)NC1CCN(C(C2COC(=O)N2)=O)C1(C)C c1(C(=O)NCC(CN(C(=O)C=C2CCSCC2)C)(C)C)cc(Cl)ccc1C(F)F C(C)(C(C(=O)NC1(C)CCC(C)C1)C(C)C)NC(c1c(O)ccc(C)c1)=O C1(CNC(C(CCC)N(C)C)=O)CN(C(=O)CC2(C)CCC2)CCC1(F)F c1(CSCC)nc(-c2cn(C3COCC3CC)nn2)n(C(C)COCC)n1 N1(CCC(=O)NCC(CC)NC(c2ncc(F)cn2)=O)CCCC(N(C)C)C1 Cc1nc(O)[nH]c1C(=O)NC1(CF)CCN(C(=O)C(C)(C)C2CCCO2)C1 c1(C(=O)NC(COC)C)c[nH]c2cc(-c3cc(OC(C)C)ccc3F)cnc12 c1(NC(C2N(C(c3cc(CC)on3)=O)C3C(C2)C3)=O)ccc(C(C)C)nc1C N1(C(COC(C)C)=O)CCN(C2CCN(C(=O)CCc3nc(O)n[nH]3)CC2)CC1 C1(CNC(N2CC(c3cccc(C)c3)(F)C2)=O)COc2cscc2O1 C1(C(=O)NCC(CN(C(C(CCC)NC(C)=O)=O)C)C)CCc2n[nH]cc2C1C c1(CC2(C(=O)NCC(C)NC(Cc3nnc(C)o3)=O)CC2)ccc(Cl)cc1 N1(C(C(=O)NC2CCN(c3ccc(Br)cc3)C2)=O)CCC12CCC(O)C2 C12(NC(=O)CCn3cccnc3=O)COC(CNC(C3CC34CCC4)=O)(C1)C2 c1(C(=O)NCC(C)N(C(CC(C)CF)=O)C)cc(N(C)C)ccc1F C(=O)(C(F)C(F)(F)F)NC(C1(C(N2CC3(C(C(=O)OC)C3)C2)=O)CC1)C c1(NC(C(C)OC)=O)ccc(NC(=O)CC2CC=CCC2)cc1C Cc1nn(CCO)c(C)c1I.C12(CCCN(C(=O)OC(C)(C)C)C1)C(=O)N2 Cc1cnc(Br)c(NC(C2CC23CN(Cc2cncc(Cl)c2)C3)=O)c1 n1(C(CC)C)cc(CC2CCN(C(=O)C(c3ccccc3)F)C2)nn1 CCCCCC(F)C(=O)N1CCC(C=CC(N2CC(C)CCC2CC)=O)CC1 C(=O)(C(C)(C)CO)NCCC1CC(C(N(C(CC)C(=O)OC(C)(C)C)C)=O)C1 c1(C(N(CC(C)NC(C23CC(C)C2C3)=O)C)=O)ccc2c(n1)CCC2 N1(CCNC(CCN(C(C)C)C(C2CCSC(C)C2)=O)=O)C(=O)CCC1=O N1(C(CC(C)C(F)F)=O)CC2CCC(CNC(c3ccoc3Cl)=O)C2C1 O(NC(=O)C(C(C)C)C(C)C)CC(=O)NC1(c2nc(C)on2)CC1 C1(C(N2CC(N(C(=O)COC3CCC(F)(F)CC3)C)C2)=O)COCC2(CCC2)O1 N1(CC(C)C(=O)NCC(c2cccs2)C2CCC2)C(=O)CCC1=O N1(C(C2(CC=C)CC=CC2)=O)CCC(N(C)C(C2CCCS2(=O)=O)=O)CC1 C(C)(C)(CCCCC(=O)N1CCC2CN(C(C3(C)CC(C#N)C3)=O)CC2C1)OC N1(Cc2c(OC)ccs2)CCC2C(CCCN2C(C2CCCOC2)=O)C1 C1(NC(=O)CCCCO)CC2CC(C1)N(Cc1nc(C(F)F)n[nH]1)C2 C=CC(C)(C)CC(=O)N1CCC(C(=O)N(CC(C)(F)F)C)C1C(C)C N1(C(C(CC)N(C)C)=O)CC2CC(C1)N(C(C1CCCOCC1)=O)C2 N1(C(C(CC)O)=O)CCC2(CC(NC(=O)CCN3CCNC(=O)C3)C2)C1 N1(C(C(=O)NC2C(N)C2)=O)CCC(F)(c2ccc(Cl)cc2)CC1 C(C(C)(CNC(C(CC)n1ccnc1)=O)COC)NC(C1C(C)C1)=O.OC c1(CC(=O)NCC(C)N(C)C(c2cc(Cl)cn2C)=O)nnc(S)n1C C(=O)(C1=NNC(C(F)(F)F)C1)N1CCC(N(C)C(C2CC(Cl)(Cl)C2)=O)C1 c1(C(=O)NCC2CN(C(CC3(CCC=C)CC3)=O)C2)cc(C)n(NC(N)=O)c1C c1(C(=O)OC)nc(NC2CCN(C(=O)CC(C)C(F)F)CC2(C)C)c(F)c(Cl)n1 c1(C(=O)NCC(C)(C)NC(c2ncc(Cl)cc2Cl)=O)cc(F)cc2nc[nH]c12 n1(CC=C)c(N(CCCNC(=O)Cc2c(C)noc2C)C)nnc1C(C)(C)C C1(CC)C(=O)N(C)CCN1C(=O)CN1CCC(N(C(=O)CCc2ccc[nH]2)CC)C1 c1(CC(=O)NCC(CCCC)NC(c2csnn2)=O)c(F)cncc1Cl C(=O)(C1=C(C)N(C)c2ncnn2C1)NC(CN(C(c1cnc(OC)s1)=O)CC)C C(=O)(C1=CS(=O)CCC1)NCCCN(C1CCCC1)C(c1c(NC)cncc1)=O Cc1cc(F)ccc1CC(=O)Nc1nc(Cl)ccc1C(=O)Nc1csc(Br)c1 C#CC1CCCN1C(c1cncc(N(C)C)c1)C(=O)Nc1ccc(OCC)cc1 N1(C(CC(C)C(F)(F)F)=O)CCC2(CCN(C(C3COC(=O)C3)=O)C2)C1 C1(CCC(=O)NCCCCNC(=O)CCOCC2CCCO2)CCCCO1 c1(C(=O)NCCNC(C2N(CCC)C(=O)CCC2)=O)cccc2c1CC(=O)N2 c1(C2(F)C(C(N(CC(CN(C(=O)C=CC(=O)N(C)C)C)O)C)=O)C2)ccccc1 N1(S(C)(=O)=O)CCN(C(=O)CCCC2CC2)CC1.C123CC(C1)(C2)C(=O)NC3 C1(C(=O)NCC2(C)CCC2)CCN(C(c2ccc(F)c(O)c2)=O)CCO1 N1(C(CC(=O)NCC)=O)CC(CNC(=O)C(F)C2CCOC2)CCC1C c1(C(=O)OC)cc(C(N2CC3CC2(CNC(c2cnc(C)[nH]2)=O)C3)=O)ccc1C C1(NC(c2cc(C(C)=O)c(C)o2)=O)CCCCCN(C(=O)CC2CCC(=O)N2)C1 N1(C(C2C(OCC)C2C)=O)CCC(F)C(NC(c2cnn(C3CC3)c2C)=O)C1 C(=O)(C(CO)C(C)(C)C)N1CC(CC(C)NC(=O)C(O)C(F)(F)F)C1 C(=O)(CCCCN=[N+]=[N-])NCCOCCNC(c1c(OC)cncc1)=O Nc1c(C(=O)NC2(CNC(c3ccc(O)nc3)=O)CC2)ccc(F)c1F c1(C(=O)NCCCC(C)NC(C(C2CCOCC2)OCC)=O)cncc(N)n1 CC(Cc1cnc[nH]1)C(=O)NC1CC1CNC(c1cc(Cn2cccn2)on1)=O c1(N2CC(NC(C(C3CCC3)OC)=O)C(C)C2)nc(Cl)ncc1Cl [SH](=O)(=O)c1cc(N2CC(CC)C(c3ccc(F)cc3)CC2)ccc1OC.OC C#CCCN=C(NCC1CCS(=O)(=O)C1(C)C)N1CCN(CCOC)C(=O)C1 N1(C(C(C)(C2CCOCC2)OCC)=O)CCC(CO)(CNC(=O)C(C)SC)CC1 N1(C(C=CC=CCC)=O)CC2CC1CN2C(=O)CN(C)C(c1cccs1)=O N1(C(C(CCCC)(C)F)=O)CCCC2(CCN(C(c3nc(C)ccc3F)=O)C2)C1 N#CC1(C(=O)NCC(O)Cc2ccccc2)CC2CC2C1 C1(NC(C2(C(c3cn(C4CN(C(=O)C5CC5)C4)nn3)=O)COC2)=O)CCC2(CC2)C1 N1(C(CCC=CC)=O)CCC(NC(=O)C(F)(F)C2(OC)CCCC2)C(O)C1 c1(C(C)NC(=O)C(CO)OC)ccccc1NC(C1(SCC)CCCC1)=O CC1C(C)N(C(=O)NC2(c3ccccc3)CC2)CCN1C(=O)CCCC#N c1(C(C(=O)NC(C)(C)C(C)NC(=O)C(F)F)OC)cccc(F)c1 C1(C(=O)NCC=CCSC)C(C2CC2)CCN1C(c1ncccc1Cl)=O CC(C)(CCNC(=O)C(C)(C)F)NC(c1cn(CC(N2CCCC2)=O)nn1)=O N1(C(c2c(CCC)n[nH]c2)=O)CCCC12CCN(C(c1cnc(C)cc1C)=O)C2 C(=O)(C(CC(C)C)ONC(C1(C)CC(=O)N(C)C1)=O)N(CCSC)CC C12(CNC(C(OC)OC)=O)CCCCC1CN(C(=O)CCSCC(N)=O)C2 C1(NCC(=O)NCCCN2CCN(C(CS(CC)=O)=O)CC2)CCOC(C)(C)C1 Cc1ccc(OCCOC2(CNC(C3CC3C(=O)NCCO)=O)CCC2)cc1F CCC(C)C(N)C(=O)N1CC2C(C(=O)Nc3ccnn3-c3ccccc3)C2C1 Cc1nn(C)c(C(=O)NCCCN(CC(C)C)C)c1Cl Cc1[nH]c2ccnn2c(=O)c1CC(=O)N1CCC12CN(C(=O)CN(C)C(C)C)C2 Cn1ccc2sc(C(N3CCC(n4cc(-c5cccnc5F)nn4)C3)=O)cc12 C12(CCCC1)C(=O)N2.C(=O)(C(F)n1cccn1)NCCC1(C(=O)OCC)CC1 CC(CS(C)(=O)=O)C(=O)N1CC(O)(CN(C)C(c2ncncc2F)=O)C1 C=CCC(CC)C(=O)N1CC(c2ocnc2C(=O)NCc2cccc(OC)c2)C1 N1(C(c2cnccc2Cl)=O)CCN(C(C23COCC2C3(F)F)=O)C2(CCC2)C1 c1(C(N2CCC(OC)(CNC(c3ccoc3Cl)=O)C2)=O)cc2c(nn1)OCCS2 c1(OC(C(=O)NCC2(CNC(CCCOC)=O)CC2(F)F)C)ccc(F)c(F)c1 C(C(=O)C1CCOc2ccccc21)OC(Cn1cc(-c2c(C)cccc2)nn1)=O N1(C(C(c2cccc(C(F)(F)F)c2)C)=O)CC(NC(=O)CNC(N)=O)C(C)(C)C1 C1(c2n(CC)nnn2)(NCCOc2ccc(Cl)cc2C)CCCC(C(C)C)CC1 N1(C(=O)OC(C)(C)C)C2COC3C2OCC13.C1(C(C)N(C)C)CCCN(C=O)C1 N1(C(C(C(C)C)OC(C)C)=O)Cc2occ(C(=O)NCC(O)CN(C)C)c2C1 c1(CC)cscc1CC(=O)NC(CN(C)C)CC Cc1cc(=NCCc2c[nH]c(=N)s2)[nH]c(N2CCCC(SC(F)(F)F)C2)n1 c1(OCC)ccc(CN2CC3CN(C(=O)CCSC)CC23)cc1C C1(NC(C2CC(C(F)(F)F)(OC)C2)=O)CN(C(=O)CCC#N)CC2CC12 N1(C(C(COC)(C)C)=O)CCC(C2CC2)(NC(=O)C(O)C(C)C)C1 CN1CC2(CCN(C(=O)NCc3sccc3C(F)(F)F)CC2CO)C1 CC(Cc1ccnn1C)C(=O)NCC#CCNC(=O)CCNC(=O)CO Cc1ccnc(C(=O)NC2CC(CC(=O)NCC(C)OC(F)F)C2)c1F CCS(=O)(=O)CC(=O)NCC1(OC)CN(C(=O)CCCCO)C1 c1(-n2cc(C3(O)CN(C(c4csc(Cl)c4Cl)=O)C3)nn2)ccc2cccnc2n1 CCCCC(C)CCC(=O)N1CC2CC(C1)CN(C(=O)CCn1cccn1)C2 C1(C)(CNC(c2ncc(C)cn2)=O)CCCN(C(=O)CC(C)c2ccncc2)C1 CN1C(=O)C(F)CC1C(=O)NCCC1CC(NC(=O)C=CI)C1 c1(C(N(C2C3CN(C(=O)C(O)C(F)F)CC23)C)=O)cccc(F)n1 N1(C(c2c(COC)ncs2)=O)CCN(C(=O)Cc2nonc2C)C(C2CC2)C1 c1(C(=O)NC2CC(NC(c3cc(CC)c(C)s3)=O)C(O)C2)cc(F)c(O)c(F)c1 c1(CC2(NC(C3(Cc4cccc(Cl)c4)CC3)=O)CC2)cccc(Br)c1F C1(OC)CCC(C(N2CCCC(CNC(=O)CC(C)SC)C2)=O)CC1 N1(c2c(C)c(NCC3CC(=O)N(C)C3)ncn2)CCOC2CCCC12 N1(C(c2ccc(C(=O)OC)[nH]2)=O)CCC2(NC(C3(F)CC3)=O)CCCC12 C(=O)(CCCCCC(C)O)N(C(C)C)CCNC(=O)CCc1nnc(C(F)F)o1 C=CC(C)(CCOC)C(=O)N1CC2CC2(CNC(=O)CNC(C2CCOCC2)=O)C1 C=CC(CCC)CC(=O)NC(c1ccc(O)cc1)CO C1(COCC(=O)NCCC2CCCCC2O)(NC(C2CCC2)=O)CC(F)(F)C1 c1(OC)conc1C(=O)NC1(CC(=O)N(CCCO)C(C)C)CCC1 c1(CC)nc(CC(Cc2cn(C(C(=O)NC(C)=O)C)nn2)C(C)C)cs1 c1(-c2n(C3C(C)OCC3)nc(-c3ccoc3)n2)cnc(-c2ncccn2)nc1O O=C(C#CCCCF)N(Cc1cnn(C(F)F)c1)CC1CCC1 CC1CCC(C(C)NC(C2CC(N(C(C3OCCC3C)=O)CC3CC3)C2)=O)C1 N1(C(C(CCC)N(C)C)=O)CC2CCC(C1CO)N2C(C1CSC1)=O n1(-c2c(SC)n(C)nc2)cnc2c1CCCC2.c12ccc(nc1)[nH]c2=O c1(C(N(CC=C)CC=C)=O)cn2cccc(-c3ccnn3C(C)C)c2n1 CC(CN(C)C(C1CCN1C)=O)C(=O)N1CCC2CC12 N1(CC(=O)NCCC(=C)CNC(C2CC3CCC(C2)C3)=O)C(=O)NC(C)(C)C1=O CCCCC(C(=O)N(C)CCOCCC(N1CC(F)(COC)C1)=O)C(C)C C1(CNC(c2c(OC)nsc2)=O)C2CCCC1N(C(=O)C=Cc1csc(C)n1)C2 CC(C)C(C(=O)NCCc1ccsc1)n1cc(CN2CCN(C)CC2)nn1 n1(C(N2CC(CCNC(CC=C)=O)OCC2)=O)ccc(=O)n(C)c1=O C(CCCCC(=O)N1CCCCC1CNC(=O)C1=CCSC1)N(C)C N1(C(c2ccc(C)c(C3CC3)c2)C(=O)NCC)CC(C)C12CCOCC2 C(=O)(C(F)C(C)CNC(c1cccnc1S)=O)NC1CCN(CC)C1 c1(C(=O)NC2C(NC(=O)C(c3ccc(F)cc3F)=O)C2)cc(Cl)ccc1O N1(C(c2cccc(C)n2)=O)CCN(C)CC1C(=O)NCCN(C)CCF C1(CC)CCN(C(C2CCN(C)CC2)=O)C1CNC(C1CC(CN(C)C)C1)=O N1(C(CNC(C)=O)=O)CC(NC(=O)C=Cc2ccccc2C#N)C2(CCOCC2)C1 c1(C(N2CCC(NC(CC=CCC)=O)C2C)=O)cc2c(nn1)CCCC2 c1(C(C(=O)NCC(CN(C(C=CCN(C)CC)=O)C)C)SC)ccccc1 c1(CCC)cnc(SC)nc1C(=O)NCC12CC1CN(C(=O)CC1CCCOC1)C2 Cc1cc(C(=O)NCC2CC2NC(c2cccn2CC(N)=O)=O)n(C(C)(C)C)n1 C1(NC(CC2N(CC)CCOC2)=O)C2CC1N(C(=O)Cc1ncn(C)c1C)C2C c1(C(C)(C)C)ccc(S(=O)(=O)Nc2ccc(Cl)c(N3CCCC3=O)c2)cc1 CC(C)C(C(=O)N1CC(NC(=O)CSCC(=O)N(C)C)C1)N(C)C C1(C(=O)NC(CCC)C2CC2)C=CCCN1C(=O)CCCCNC(N)=O c1(C(C(=O)N(CCCC(C)(C)C)C)N)cc(F)ccc1F CCC(CNC(=O)C(F)C1CCOC1)(CC)C(=O)N1CCC(C(N)=O)(N(C)C)C1 c1(C(=O)NC(C2CCCOC2)C(=O)NCC2CCCO2)ccc2c(c1)OCO2 Nc1cnc(Cl)c(C(N2CCC(F)(CNC(C3CC3CF)=O)CC2)=O)c1 Cn1cc(C(=O)NCC2CCCN(C(=O)CC3(O)CC3)C2)c(O)n1 N1(C(CCOCC)=O)CCCC(NC(C2CC(C(C)C)C2)=O)C(F)C1 c1(NC2CC(C(C)NC(CC)=O)C2)ncnc2scnc12 c1(C(=O)NC(C)CCNC(C2CC2F)=O)ccc2c(n1)CCC2 N1(C(C(CCN(C)C)O)=O)C(C(=O)NCCN2CCCC2=O)CCC12CC2 c1(C(=O)N(C2CC(C)N(C(=O)CCOCCN(C)C)C2)CC)ccn2ncccc12 c1(NC(=O)NCc2nnc(-c3c(OC)cccc3)o2)cc(C)cc(C)c1OC c1(C(=O)NC(C)CCCNC(C2(CCO)CC2)=O)ccc(CN(C)C)cc1 Cc1cc(O)ccc1C(N1CC2C(NC(C3CC4(CCCO4)C3)=O)C2C1)=O N1(C(C)C)CC2CC1CN2C(C1C=CCN1C(C1CC2CC1CC2O)=O)=O c1(C(=O)NC(C(C)NC(C2CCN(C3CC3)C2=O)=O)(C)C)cn2c(n1)CCCC2 C(=O)(C1CCCn2nccc21)NCC12C(CN(C(c3c(C)n[nH]c3C)=O)C1)CC2 c1(C(=O)NCC2N(C)CCN(C(=O)CNS(N)(=O)=O)C2)ccc2ncccc2c1 Cc1cn(C(C)(C)CC(=O)NCC2(O)CN(C(=O)CCCC(C)O)C2)c(=O)nc1O c1(C(N2CC(CNC(C3CN(C(C)=O)C3)=O)C(O)C2)=O)c(C)nn(C)c1Cl Cn1cncc(C(=O)NCCNC(c2ccc(=O)oc2)=O)c1=O c1(C(=O)OC)ccccc1C(=O)NCC(C)N(C(=O)Cc1ccoc1)C c1(C(CNC(C2COCCO2)=O)NC(c2ccc(CC)[nH]2)=O)ccccc1CC c1(N(c2nnc(O)nc2O)C)nc(C#N)c(Cl)s1.C12CCCN1C2=O C1(C2CCN(C(c3ccn4ccnc4n3)=O)CC2)(NC(C(CSC)C)=O)CC1 O=C(NNc1ccc2ccccc2c1)NC(c1ccccc1)Cc1cccnc1 C=C(Cl)C.C(C(C)CSCC)NC(C)=O c1(NC(c2n(CC)nnn2)c2csc(C3(SC)CCC3)c2)ccc(Cl)cc1 Cc1ncc(Cl)cc1C(=O)NC1CC12CCN(C(=O)C=Cc1cnn(C)c1)C2 N1(C(CC=C(C)C)=O)CC(CNC(C2(C)CCNC2=O)=O)OC(C)(C)C1 Cc1cc(C(=O)NCC(C)NC(c2cccc(-n3cccn3)n2)=O)c(C)cn1 Cc1csc(C(=O)NCC(C)(F)CNC(=O)CCC2CCCN2C)c1C c1(OC)c(C(=O)N(CC(CC)NC(C2CC(C)(C)CO2)=O)C)cccc1Br n1(CCC(N2C(CNC(C3C(=C)C3)=O)C=CC2)=O)nc(C)c(C)c1C CC1CC(C(=O)NCCC2(O)CN(C(=O)CNC(=O)C3CC3)C2)CC(C)C1 c1(-c2c(C(=O)NC(c3ccccc3)C(=O)OC)ncnc2)cccc(C(C)=O)c1 CCCC(CCCNC(c1cnc(S)[nH]1)=O)NC(=O)Cc1c(C)cnn1C N1(C(C2(C)CCC(=O)C2)=O)CC(CO)C2(C1)CN(C(c1ccc(C3CC3)s1)=O)C2 CC1(C)CCOC1CNC(=O)C(Cc1cc[nH]n1)NC(=O)C(F)=CC1CC1 CC1C(NC(c2cnc(C(F)(F)F)s2)=O)CCN1C(=O)Cc1csc(S)n1 C1(CNC(C(C)(C)OC)=O)CN(C(c2ccc[n+]([O-])c2)=O)CCC1(C)C C(CC1CCC1)(C(=O)N1CC(O)(CNC(c2cc(C(N)=O)co2)=O)C1)NC(C)=O CCCCCC=CC(=O)NC(COCCOC1CC1)C(=O)NC1CC1CC C1(NC(c2[nH]nc(OC)c2Cl)=O)CCN(C(=O)C2=NNC(=O)C2)CC(O)C1 C(=O)(C(F)C(C)CNC(c1cc(OC)no1)=O)N1CC(O)(CC)C1 N1C(=NCc2sccc2Cl)NCCC1C1CCCO1.C1(C(C)(C)C)CCCCO1 Cc1c(C(=O)N(CCCN(C)C(c2cc(Cl)c(Cl)[nH]2)=O)C)nn2c1OCCC2 C1(NC(c2cnc(CC)s2)=O)CCCC(Nc2nccc(-n3ccnc3)n2)C1 C(=O)(CC(C)C(=O)NCC1(C)CCCN1C(c1ccc(Br)cn1)=O)OCC C1(NC(CN2CC(C)(C)C2)=O)CCN(C2CCN(C(=O)CC3CC(F)C3)C2)CC1 C1(NC(c2ccn3ccnc3c2)=O)CN(C(C2CC2Cl)=O)CC(F)(F)C1 N1(C(c2ccc(CNC(c3c(C(C)(C)C)[nH]cn3)=O)cn2)=O)CCC(F)C(O)C1 N1(C(c2c(C#N)ccs2)=O)CCN(C(c2csc(Cl)c2Cl)=O)CC(O)C1 C1(C(=O)NCC(CO)NC(=O)CCc2ccsc2Cl)CC(C2CC2)C1 Cn1cc(C(=O)NCCOCCC(N2CC3(CSC3)C2)=O)ccc1=O c1(OC)ccc(CN2CCN(C(=O)CCc3ccccc3)CC2)cc1Cl c1(C(=O)NCC=CCNC(c2ccsn2)=O)cccc(SC(F)(F)F)c1 C1(C(=O)NCC2(CCCO)CC2)CN(C(c2conc2CC)=O)CC1CSC c1(C(CNC(C2OCCO2)=O)NC(C(C)OCCOC)=O)ccccc1 C(=O)(N=c1ccn(C2CN(Cc3ccc(O)c(C)c3)C2)[nH]1)c1ccc(OC)cc1 c1(NCC(C)NC(C(CC)OC2CCCCC2)=O)cc2nnc(C)n2cn1 CCCC(C(=O)N(C(C)(C)CC(=O)N1CCC1CF)C)C(C)C C(CCCCCNC(=O)CNC(=O)C(c1cccnc1)O)n1cc(CC(C)C)nn1 N1(C(C(C)(C)C2CCN(C(=O)CC3CCCCO3)C2)=O)CC(F)C(F)C1 c1(SC(C(N2CCC(C)(C(=O)NCC=C)C2)=O)C)nc2ccc(C)cc2[nH]1 c1(C(C)C)cc(CC(=O)NC(C)(CNC(=O)C(C)NC(N)=O)C(F)(F)F)on1 N1(C(CC=CC)=O)CCC2(CC1)COCC(CNC(C1(C)CS(=O)(=O)C1)=O)O2 C1(CC)CCN(C(=O)CC2CC=CC2)C(C(=O)NCCN2CC(C)(O)C2)C1 N1(C(C(CN(C)C)NC(C=C)=O)=O)CC2CC(CO)C(C2)C1 C1(CCC#C)CCN(C(c2ccc(COCC)cc2)C(=O)NC2COC2)CC1 c1(C(N2CC(N(CC(C)C)C)C2)=O)ccnc(CNC(=O)CCn2cccn2)c1 C1(C(N2C(CNC(C3(S(N)(=O)=O)CC3)=O)CC(O)C2)=O)CC2(C1)CC1(CC1)C2 Cc1c(C2CCCN2C(=O)C(=O)NCc2ccc(Cl)s2)cnn1C CC1CCCC1(C)C(=O)NCC#CCNC(=O)Cc1cccc(O)c1 C1(NC(C2(CC=C)CCCN2C(=O)CSC2CC2)=O)C2C=CC(C2)C1COC c1(C(=O)NCC2(NC(=O)COc3ccon3)CCCC2)cc2ncccc2[nH]1 N1(C(CN(C)CC)=O)CCCOC(CNC(c2cc(OC)cc(Cl)c2)=O)C1 C(=O)(CCCn1cc(-c2csc(C)n2)nn1)NCCNC1C(C(=O)OC)C1 c1(CC2(O)CCN(C(c3ncc(C(C)C)s3)=O)CC2)csc2ccccc12 N1(C(c2c(CCC)occ2)=O)CCC(NC(=O)Cc2cnn(C)c2)C(C)C1 c1(C(N2C(C)CCN(C(CCN(C)CC)=O)CC2)=O)n[nH]c2c1CC(C)CC2 c12ccc(cc1F)CNc1cc(nc(C)n1)N2C1CC1.C(C)(C=C)S.CCO c1(C(N2CC(CC=C)(NC(=O)CCCOC)C2)=O)cccc(Cl)c1OC(F)(F)F c1(C(=O)NC2C=CCN(C(CC(CCC)C)=O)C2)sc2nnc(S)n2c1C c1(C(=O)NC2(C3CCCN3C(C3CCSC3)=O)CC2)ccc(O)c(F)c1F Cc1csc2c(N3CCC(NC(=O)C=Cc4ccc(Cl)cc4)C(F)C3)ncnc12 c1(C(N2CC(CNC(C=CC(=O)N(C)C)=O)C2)=O)ccc(-n2cccc2)nc1 N1(C(C2C(C)OC(=O)N2)=O)CCCC2(CCN(C(c3sccc3CO)=O)C2)C1 N1(C(C2(C)C(C)C2)=O)CC(O)(CNC(C2(c3cccs3)CC2)=O)C1 C1(C(=O)NC(C(=O)N(CC(C(C)C)C)C)C)CCC2(CC2)C1 S1(=O)(=O)c2cccc(c2)C(=O)N1.CCCCN(CCCN(C)C)CCCN1CC1 C12(C(=O)NC(CNC(C(C(CC)C)O)=O)C3CC3)CCC(CO)(CC1)CC2 C1(O)(CN(C)C)CCN(C(C2CSCN2C(c2cnn(C)c2Cl)=O)=O)C1 c1(CCC=CC(N2CC(NC(C3CC(CCC)C3)=O)C2)=O)ccccc1 S(=O)(=O)(CC)N(CC(=O)NCCOCCNC(C1C(OC)C1)=O)C c1(OC)cc(CN2CCC(NC(=O)OC(C)(C)C)C2)cc([N+](=O)[O-])c1O c1(NC(C2CC(O)CCN2Cc2scnc2Cl)=O)cc(Br)c(F)cc1I C1(NC(CCS(=O)(=O)NC)=O)CCSC12CN(C(=O)CSCc1ccccn1)C2 c1(C(=O)NC2CCOC2C(N2CC3CCC=CC23)=O)cc2ccccn2n1 n1(CC)ccc(C(N2CCC(CNC(=O)C#CC3CC3)(OC)C2)=O)cc1=O c1(N2CCC(CC(C)NC(C3CCC(=O)N3)=O)CC2)ccnc2ncnn12 C1(CC(=O)NCCC2(C)CC2)CCCCC1NC(=O)CCc1nccs1 C1(C(N2CC(N(C(CCc3cn(C4C(C)C4)nc3)=O)C)C2)=O)CCCN1N=O C1(CC=C)(C(=O)NCC2C(C)(C)C2(C)C)CCCN1C(c1cnn[nH]1)=O c1(CN(C(C(C2(O)CN(C(c3nc(Cl)cs3)=O)C2)C)=O)C2CC2)cccc(F)c1 N1(C(C(COC)C)=O)CC(C)OC2(CCN(C(c3cc[nH]c3C)=O)CC2)C1 C(C(COC)CC(=O)NC1CCC(C)N(C(=O)C(C)C)C1)OC C12(C(=O)NCC3C(C)CCN3C(=O)CN3CCCNC3=O)CCOC(C)(C1)C2 Cc1nc(NC2CCOCC2F)c2ccsc2n1 Cc1cc(N)c(C)nc1C(=O)NCC1(NC(C2CC3CC3C2)=O)CCOC1 C12(C(=O)NCC(C)N(C(CC3C(C)CCO3)=O)C)CCC(F)(CC1)CC2 N1(C(C2CN(C)CC(C)N2)=O)CCC(C2(N)COC2)CC1 C1(C(=O)NC(C)CC(O)CO)N(C(=O)CCOCC2CCC2)CC12CCCC2 c1(C(N2CC3C(CNC(C(CNC(C)=O)(C)C)=O)C3C2)=O)cnn2c1N(C)CC2 C1(CNC(C2C(C)(CC)C2)=O)CCN(C(=O)C2=CC(C)(CC)C2)C1(C)C Cc1ccc(C(N2CCC(C(=O)NCC(C)(O)C3CC3)CC2C)=O)c(C)c1 C1(=O)C(CC(C)C)O1.Cc1nc(C)n(CCNC2(C)COCCO2)n1 C1(C(N(CC(CO)(CO)NC(C2CCC2C#N)=O)C)=O)CCCCC(C)(C)C1 N1(C(c2c(C)nc[nH]2)=O)CCN(C(c2ccc(O)c(F)c2)=O)C(CCO)C1 C1(C(=O)O)CC(NC(c2cnn(Cc3ccc(Br)cc3)c2)=O)CCN1 CCC(C)(C)C(=O)C(=O)NCC1OCCC1C(N1CC(O)(COC)C1)=O N1(C(C2C(OC)CC2)=O)CC2C(NC(=O)CCCC3OCCO3)C2C1 CC(C)C(O)C(C)(C)C(=O)NC(C)C(N1CC2(CCC1CO)CC2)=O C(=O)(N=c1cc(C(N)=O)n(C)[nH]1)C1N(C(C2C(C(=C)C)OCC2)=O)C2CCC1C2 C1(SCC(=O)N(C2CC(C#N)C2)CC(=O)NC2C(C)C2)CCNC(=O)C1 c1(NC(C(c2ccc(OC)cc2C)N(CCCC)C)=O)c(C)cc(C)cc1C c1(C(N2C(CNC(CC(=O)NCC)=O)CCC2)=O)cc2c(cc1Cl)OCCO2 c1(C(=O)NC(C2CCCCC2)CNC(C2CCC(F)(F)C2)=O)cnccc1Cl C=CCC(C)(C)CC(=O)NCC1CC(NC(=O)COCCOC)C1 c1(C(N2C(C(=O)NC(COC)C)CC3CC32)=O)ccn2cncc2c1 CC1(C(N2CCC2Cc2ccccc2)=O)CCN(C(c2cscn2)=O)CC1 C(=O)(C(F)C(C)(C)O)NCC1CC(OC)CN1C(=O)CNC(c1ccoc1)=O C1(C(C)C)CN(C(=O)C(C2CCCO2)NC(=O)CCC2CC2(C)C)CCCO1 C1(NC(CCOCCOC)=O)CC(CNC(c2cccc(N)n2)=O)C1(C)C Cc1cc(I)ccc1C(C(=O)Nc1ccc(Cl)cc1F)N(c1ccccc1)C C(=O)(CC(C)C(F)F)N1CCC(CN(C(CCC2CC(C)C2)=O)C)C1 C1(NC(c2[nH]cc(C(C)(C)C)c2)=O)CCCC(C(=O)NCc2ccc(Br)nc2)C1 O(NC(=O)C(C)NC(=O)COC(c1cc(CSC2CCC2)[nH]n1)=O)CC c1(C(=O)NC(C2(O)CCN(C(C(C)NC(C)=O)=O)CC2)C)cc(C)cc(C)c1N C#Cc1ccnc(C(N2CCC(C(=O)N(C3CC(CCO)C3)C)(CC)CC2)=O)c1 C1(CCC(=O)NCC=CC)CCCCN(C(C23CC(SC)C2C3)=O)C1 c1(OC)cccc(C(=O)NC(c2cccnc2)C(=O)NCc2ncn(C)n2)n1 S(=O)(=O)(c1cccs1)NC(C(C)C(=O)NCC1C=CCN1C(=O)CNC1CC1)=O c1(C(=O)NC(CNC(C2(CC)CC2(F)F)=O)(C)C(C)C)cc(Cl)cc2c1CCC2 c1(OC)ccc2c(c1)CCC2C(=O)N(C(c1csc(-c2cccs2)n1)C)C1CC1 C1(NC(C)=O)CCN(C(=O)OC(C)(C)C)C12CC2.C12C3CN(CC13)C2=O C1(C(N(CCC(C)C)C)=O)CCN(C(=O)C(C)N(C)C)CC(O)C1 c1(NC(C(=O)N(CC(C(C)c2ccccc2)O)CC)=O)ccc(Cl)c(C(F)(F)F)c1 C1(NC(C(C=CCCC)O)=O)CC2CCC1CC2NC(=O)CN(C)C(C)=O C(CCCCC(=O)NCc1c(O)cccc1F)N(C(CC1(N(C)C)CC1)=O)C c1(C(=O)NCC2(C)CC(NC(Cc3c(C)ccs3)=O)C2)nc2ccccn2n1 C1(C(NOC(C)(C)C)=O)COCC1NC(=O)CC1CC(N(C)C)C1 c1(OCCC)nc(C)ccc1C(=O)NCc1cn(CC(C)NC(=O)C(N)=O)nn1 C1(CCC(=O)OC)C(=O)OCC2(O)CCN1CC2.c1(CC)noc(C(=O)NC)n1 N1(C(C(N2CCCCC2=O)C)=O)CCC2(CC(NC(=O)CSC3CC3)C2)C1 Cc1cc(=NCC(C)NC(=O)CC(C)C)[nH]c(C)n1.SCC CC1C(NC(c2scnc2C(F)(F)F)=O)CCCN1C(C1OCCC1C)=O CC1CC(c2scc(C(=O)NCC3(O)CCCCC3)n2)CN1Cc1ccccc1 C1(CC)CN2CCCC2CN1CC1CC2CC1CC2O c1(C(=O)NCCN(C(=O)C(C)=C2CCC2)CCC)ncn2c1COCC2 CC(C)C(C)C(=O)NCC1CN(C(c2conc2C2CCCC2)=O)CCO1 N1(C(c2cc(C)ncn2)=O)CCC(NC(C2CC(C)CCO2)=O)C(F)(F)CC1 C1(C(C)(C)N(C(C)C)C(CCC2CC(C)(C)O2)=O)CCNC1=O CC1(C)C(=O)CC1C(=O)NCC1CCN(C(C2(CC3CC3)CCCC2)=O)CC1 c1(C(=O)NC2C(NC(C3C(C)(C)CCC3)=O)CC2)ccc(Br)cc1O c1(N(C(=O)C=C2CCN(C(=O)Cc3cncnc3)C2)C(C2CC2)=O)ccccc1 CCCC1C(=O)NC2CC(C2)C(=O)N1C.C1(C(=O)OCC)(N(C)C)CC1 N1(C(c2c(SC)cccc2)=O)CC2CC(NC(c3cnc(O)s3)=O)C1C2 C(C(C(=O)NCCn1cccn1)C(C)C)NC(CCOCCOCC)=O C1(Cc2nn(-c3ccc(OC)cc3)c(-c3cc(OC)ccn3)n2)CC2CCC1O2 C1(C(F)(F)F)(C(=O)NC(C2CCOC2)CNC(C2CCCC2)=O)CCCCC1 C1(C(=O)NC(C(C)O)(C)C)CCN(C(=O)C(=O)NCC2CC2)CC1O C1(CNC(c2cc(C)nn2C)=O)CC2CCCCC2N1C(C12CC(C#N)(C1)C2)=O Cc1ccc(C=CC(=O)NC2CC(NC(=O)C(C(C)O)NC(=O)NF)C2)cc1 c1(C(=O)NC)cccc(C(N2CC(NC(C3(C)CSC3)=O)C3CC23)=O)n1 CC(Cn1ccnc1)C(=O)NC(C)CC(C)NC(=O)C(F)(F)c1cscn1 N1(C(c2c(C)noc2)=O)Cc2ccc(CNC(c3cnc(O)c(Cl)c3)=O)cc2C1 N1(C(c2cc(OC)c(Cl)s2)=O)CCCC(NC(c2cc[nH]c2C2CC2)=O)CC1 C1(CCC(=O)NC(C2C(C(=O)NCC3(CC)CCC3)C2)C)CCC(=O)C1 N1(c2nc(CC)c(C)cn2)CC2CCCC(NC(C3CCS(=O)(=O)CC3)=O)C2C1 c1(OC)ccc(Cl)cc1CN1CCC(C(C)NC(=O)CCc2ccn(C)n2)CC1 C1(COCC(=O)NC2(C(=O)NCC3CCC3(F)F)CC2)CCCOC1 Cc1cc(F)cc(C(=O)NCC(O)CNC(C2CCC(C)(C)C2)=O)c1N c1(C2C(C(=O)NC(CN(C(c3n(CC)ccn3)=O)C)C)C2)ccc([N+](=O)[O-])cc1 N1(C(C2(NC(=O)C(C)c3ccco3)C(C)C2)=O)CCCN(C)C(=O)C1 C1(C(=O)NCCCCCN=[N+]=[N-])CCC2(CC1)CNCCO2 C1(F)(CC)CCN(NC2COCC2n2ccnc2)C1 N1(C(C(c2ccccc2)N(C)CC)=O)CCN(C(C2CC(C(=O)OC)C2)=O)CC1 C(=O)(CCC(=O)c1cccnc1)NC(c1cccc(Br)c1)C#N c1(C(=O)NC(C)C(CO)NC(c2ccc(N)cn2)=O)cc2nc(F)ccc2o1 C(=O)(C1CCc2c[nH]nc21)NC(C1CCCCC1)CNC(C12CC(CCO1)C2)=O C#CC1CCCC(Nc2ccc(Br)c(C(F)(F)F)c2)C1 N1(C(CC2C(C)=NOC2=O)=O)CC(NC(=O)CN2CCCNC2=O)CC(C)(C)C1 N1(C(C(CCC)CC)=O)CCCC2C(NC(c3oc(CC)nc3C)=O)C(C)(C)C12 N1(C(C(C(C)(C)C)O)=O)CC(CO)C2(C1)CN(C(C13CCCC1CCC3)=O)C2 c1(OC)cc(Cl)c(C(N2CC(NC(C3(C4CC4)CC3)=O)C3(CC3)C2)=O)cc1Cl C1(NC(=O)C2=COCC2)CCCCN(C(=O)CCc2ccc(Cl)cc2)C1 c1(C(=O)NC(CNC(C(C(C)C)NC(N)=O)=O)(C)C)ccc2c(O)nncc2c1 C1(N(C(C=C(C)Cl)=O)C)CCCC2CN(C(c3c[nH]cc3Br)=O)CC12 c1(CNC(CC2(COC)CC2)=O)nc2c(s1)CN(C(=O)C#CC(C)C)CC2 c1(C(N2CCC(C(C)NC(C3(C#N)CC=CC3)=O)C2)=O)cc(F)cc(F)c1 C1(CC(C)C)C(C)CCCN1CC(=O)NCc1sc(-c2cnn(C)c2)nc1C N1(C(C2N(CCC)CCCC2)=O)CCN(C(c2snc(O)c2Cl)=O)CC1CCC Cc1cncc(C(N2CCN(CCCNC(c3cc(O)nn3C)=O)CC2)=O)c1Cl N1(C(C2CC(CNC(C(C)OCCC=C)=O)C2)=O)CC2CCCC(O)C2C1 Cc1cc(C(=O)NC2(CO)CCN(C(=O)C=Cc3cc[nH]n3)C2)cc(C)c1O c1(CNC(C2(CC)CC2)=O)ccc(CN(C)C(C2CCCC2CC)=O)cc1 C(CCOCCO)(C(=O)NCC(C1CC1)N(C)C)NC(C=NOC)=O CC1(C)OCCC1CCNC(C1CN(C(C2(C(=O)O)CCNC2=O)=O)C1)=O C1(C(=O)NC2(CO)CN(C(C3(C(C)C)COC3)=O)C2)CC2C=CC1O2 C12(CNC(C(CC)OC)=O)CCC(CNC(=O)C3=C(Cl)CCC3)(CC1)CO2 c1(C(=O)NC2(CNC(C3(Br)CC3)=O)CCOCC2)cc(=O)c2ccccc2o1 c1(C)nc(-c2cncc(F)c2)nn1C(C)C(F)(F)F.C12(C(C)(C)O)CC(C=O)(C1)C2 CC(C)(C)C(O)CCC(=O)N1CCCC1CNC(=O)CCCc1cnccn1 CC(C)(CNC(c1c[nH]nc1CNC(=O)C=Cc1ccoc1)=O)CCO CN1CC2(CC2)CC1C(=O)NC1(C(=O)NCC2NC(=O)NC2=O)CCC(C)(C)C1 Cc1nn(C)c(C)c1C(=O)NC(CNC(C1(O)CCC1)=O)CO CCCC(C)(O)CC(=O)N1CC(CN(C)C(c2ccnc(C(N)=O)c2)=O)C1 Cc1cc(NC(C2(C(C)NC(C3CC(C)CCO3)=O)CC2)=O)c(F)cc1F C1(CC(=O)N(C)CC2(O)CN(C(C=CCN(C)CC)=O)C2)CC2(CCCC2)CO1 c1(CCNC(C(=O)NC2CCc3n(cc(C)n3)C2)=O)ccc2c(c1)NC(=O)CO2 C1(C2CCCN(c3ccnc(C(C)C)n3)C2)(NC(C=CCCC)=O)CC1 Cc1cc(C)c(C(N2CCOC(C3CN(C(=O)CCCCCF)C3)C2)=O)c(C)c1 c1(CC(=O)NCC(CCCC)NC(c2c(C)coc2SC)=O)cccc(C)c1Cl C#Cc1c[nH]nc1C(=O)N(C1CCN(C(c2ccc(F)s2)=O)CC1)CCC CCC(CC(=O)NC(c1ccccc1F)CNC(=O)C=CC(F)(F)F)C(F)F CCC(F)(F)C(C)(C)C(=O)NCC=CCNC(=O)CSc1ccccc1O C1(C2CN(C(=O)COCC3CC3)C2)(NC(c2n(C)nc(C3CC3)c2)=O)CC1 c1(C(=O)NCC2CN(C(c3ccc(OC)cc3F)=O)C2)ccc2c(c1)COC2 C(CNC(=O)C(c1cccc(OC)c1)C)(CC(C)C)NC(c1ccn(CC)n1)=O C(=O)(C(CC(F)F)N(C(=O)CC1(N(C)C)CC1)C)N(CCCCO)CC C1(CNC(C=C(CCC)CCC)=O)CCN(C(c2cnc(S)nc2)=O)C(C)C1 c1(C(N2CC(NC(C3CC(=C)C3)=O)C(C3CC3)C2)=O)ccc(C2=CCCC2)cc1 c1(CN(C(CCCOC)=O)C)cccc(CNC(c2coc(Cl)c2)=O)c1 C(=O)(C(C)CC(=O)N1CC=CC(NC(=O)CCSc2nnnn2C)C1)OC C(C(C)(C)CC(C)O)NC(C(CN(C(C1C(C(C)C)OCC1)=O)C)(C)C)=O n1(CC(=O)NC2CC(O)CN(N3CCCC3CO)C2)ccc2c(F)cccc12 C(=O)(CC(C(F)(F)F)P(C)(C)=O)NCC(CN(C(=O)CN1CC2CC2C1)C)O c1(C(=O)NC(CNC(C2(CC)CCNC2=O)=O)C(C)C)cccc(C)c1N Cc1nn(C)c(C)c1C(=O)NC1CC(NC(=O)C(c2ccc(Br)cc2)(C)C)C1 Cc1ccc(C)c(OCC2(F)CCN(C(=O)NCCOC(C)(C)C)CC2)c1 C(=O)(CCC(C)(F)F)N1CC(SC)C(NC(=O)CCCOc2ccccc2)C1 c1(CC)nn(C)cc1C(=O)NCCOC1CC(CNC(=O)Cc2cn(C)cn2)C1 c1(C(N2CCC(NC(C3C(F)(F)C34CC4)=O)C2)=O)nnn2ccccc12 c1(CN(C(=O)C(CCC2CCC2)NC(=O)CCOC2CCC2)C)ccnc(F)c1 C(=O)(C1=CCS(=O)(=O)C1)NC(C)(CNC(C1CCCN1C)=O)CO Cc1c(C(=O)NC2(CNC(c3cnc(O)n3C)=O)CCOC2)nn(C)c1Br N1(C(C=C(CC)CC)=O)CCC2(NC(c3occ(C)c3C)=O)CC2C1 N1(C(C(C)CC2CCCC2)=O)CCC(NC(=O)CC2CC(C)(C)C2)CC1 N1(C(=O)OC(C)(C)C)CCN(CCCCC#N)CC1.C12CCCC(O1)N2 c1(OC)ccc(C(=O)NCCNC(=O)CC(C)n2ccnc2CO)c(F)c1Cl C1(C(=O)OC(c2ccc(NC(C)=O)cc2)CC(=O)OCC)CCN2CCOCC12 Cc1cc(C(=O)N(C2CCCCC2N(C)C(C2CC(O)CN2C)=O)C)cc(F)c1 N1(C(=O)C(C)O)CC2CCC(NC(C(C)(C)OC(C)C)=O)(C2)C1 c1(C(=O)NC(CNC(c2cn(CC=C)nc2)=O)C)cc(C#N)cn1C C1(c2ccccc2)(NC(n2cccc2)=O)CCCN(C(=O)CC2COCCO2)C1 C1(C(=O)NC2CC(OC)C2)COC2(C1)CN(C(=O)COc1ccc(C)cc1C)C2 N1(C(c2c(C)sc(O)n2)=O)CCN(C(=O)COC2(C)CCCCC2)C(C)C1 N1(C(C2(C#C)CC2)=O)CCC=CC1C(=O)NCc1ccc(Cl)nc1 c1(CCNC(N(C(c2ccccn2)C)C)=O)cc(O)cc(Br)c1 N1(C(C(CCC)S(N)(=O)=O)=O)CCC2(CC1)CCN(C(=O)C(CC)C(C)O)C2 N1(Cc2cc(C)c(Br)cc2)CCC2(CCCN(C(c3ccc(CO)nc3)=O)C2)C1 N1(C(c2cc(CC(C)C)on2)=O)CCOC(CC(C)C)C1.C12(CC1)C(=O)N2C CC1CN(C)CC1(c1nnnn1Cc1cccs1)NC(c1ccc(CO)c(Cl)c1)=O c1(C(=O)NCC(C2CC2)NC(Cc2cc(C)sc2)=O)cc(C)c(C)c(F)c1 c1(C(=O)NCC2CCCN(C(CC3CC(C)C3)=O)C2)cc(O)nc(Cl)c1 C(CN=c1nn[nH]n1-c1ccccc1)N1CCN(C(=O)CCC2CCCCC2)CC1 c1(SC(C)C(=O)NC2CN(C(c3nnnn3C)=O)C2)ccc(C#N)cc1 N1(C(C2CC(C)(C)C2)=O)CCCC(O)(CNC(C2(Br)CC23CCC3)=O)C1 c1(N(CC(N)=O)C)nc(=N)[nH]c(=NCCc2ccc3ccccc3c2)[nH]1 c1(CNC(c2ccccc2-c2cccc(Cl)c2F)=O)cc(F)cc(Br)c1F c1(C(=O)NC(CC(C)NC(C(C(C)C)OCC)=O)C)c(OC)ccc(F)c1OC c1(CN2CC3CN(c4ncc(CCC)cn4)CC32)c(Br)cccc1[N+](=O)[O-] CC1c2nccn2CCN1C(C1CCC(NC(=O)Cc2cncnc2)C1)=O CC1CC(CNC(=O)COC2(C)CCC2)CN(C(=O)COC2CC=CC2)C1 C=CC(O)(C(=O)N1CC2CCCC(NC(C3SCCCS3)=O)C2C1)C(F)(F)F C(=O)(CC1=CCN(C)CC1)N1C(C)CC(NC(C2CC(=O)NC(=O)C2)=O)CC1 Cc1nn(C)cc1CNC(C(C1C(C)CCC1)=O)=O.N(C)C C1(C(=O)NC(C(C)C)CNC(=O)Cc2nccn2C)CC1C1CCOCC1 C(=O)(C(CNC(=O)Cc1nonc1C)C(C)C)NC(C(=O)OCCC)C c1(CCN(C(c2c(C)oc(-c3ccc(Cl)cc3)c2)=O)C(C)C)cc(Cl)cc(Cl)c1 c1(C(=O)NCC=C=C)oc(CNC(=O)COC)nc1C CC(C)(C)C(CO)C(=O)NCc1cc(C(=O)NCCc2cccc(O)c2)n[nH]1 c1(CNC(C2CSCN2Cc2cc(C(C)C)on2)=O)csc(C#N)c1 N1(C(C(C(C)C)(C)O)=O)CCC(C2(NC(c3ccncc3Br)=O)CC2)C1 C1(N(C(CC(C)C2CC2)=O)C)CCC(NC(c2cccc(C(C)(C)C)n2)=O)CC1 c1(C(=O)OC)ccc(C(N2CCCC2CC(=O)Nc2ncc(O)cc2Cl)=O)c(F)c1 c1(OC)ccccc1CNC(C1(CN(C)C(C2CC=CC2)=O)CC1)=O c1(C(N2C3CCN(C(CSc4n(C)nnn4)=O)C(C3)C2)=O)nnn2c1CCCCC2 C1(C(=O)NC2(C(=O)NCC(C)CC3CCC3)CC(F)(F)C2)Cc2ccccc2C1 C1(CC)CNC(=O)CN1C(c1conc1C(C)NC(=O)CCOCCOC)=O CC1(C)CC(C(=O)NC2(CO)CC2)CN1C(=O)C(O)CC1CCCC1 c1(CCC(N2CCC(NC(C3(NC(=O)OC)CC3)=O)C2)=O)nnc(O)nc1O N1(C(CCC#C)=O)CCCCC1C1CCCN1C(c1ccc2nc(O)oc2c1)=O N1(C(C2(CNC(c3nn(C)c(CO)c3)=O)CC(C)(C)C2)=O)CC2CC1CS2=O Cc1cc(N)c(C(N2CCCN(C(C34CC(Cl)(CO3)C4)=O)C(C)C2)=O)c(F)c1 c1(CCC)cc(C(=O)N(CC(C)(C)C(=O)OCC)C)c(C)o1 CC1CCCCC1(C)NC(=O)NCC12COC(Cc3cccc(Cl)c3O)(C1)C2 C1(CC)CN(C(=O)CC2CSCCS2)CCC1NC(c1c(CO)noc1C)=O c1(NS(CC)(=O)=O)ncnc(N2CCC(c3c(C(C)C)cccc3F)CC2)c1C c1(N(C(C)CNC(C2(c3ccccc3)CC2(F)F)=O)C)ccn2c(Br)cnc2n1 C1(CCNC(=O)Nc2cc(O)nn2-c2ccccc2)CC2CCC1CC2 C1(NC(CC=CC)=O)CC2CC1CN(C(=O)C(C)=C(C)CC)C2 C(CC1CC1)(C(=O)N1CC(c2cc(O)n[nH]2)C1)NC(=O)CO N1(C(C(CC)COC)=O)CC2(CCC(NC(c3cccc4c3COC4)=O)CC2)C1 N1(C(c2c(CC)ncnc2)=O)CCCCC(NC(C2CC2Br)=O)C1 c1(CNC(C2CN(C(C3CN(C(=O)NC)C3)=O)C2)=O)ccncc1F C(=O)(CC(C)(C)C(=O)OCC)NC(CC=C)C(=O)Nc1cnccc1CC N1(C(c2cc(C(F)F)[nH]n2)=O)CCCC2(CCN(C(C3CCC=CO3)=O)C2)C1 C#Cc1ccc(F)c(C(C(=O)NCC2CC2)N(C)Cc2nc3ccccc3s2)c1 C1(O)(CCNC(c2cncs2)=O)CCN(C(c2c[nH]cc2Br)=O)C1 N1(C(C2CC(C)OCC2)=O)CCCC2C1CCN2C(=O)COc1ccc(F)c(F)c1 Cc1cc(C(N2CC(CC(=O)NCCCc3ccsc3)CC2(C)C)=O)ccc1F c1(CNC(CC2C(C)=NNC2=O)=O)nc2c(s1)CCN(C(=O)C(C1CC1)N(C)C)C2 c1(C(=O)Nc2cccc(CC)n2)cc2nc(-c3ccc4c[nH]nc4c3)ccc2[nH]1 O=C(C1NCC2(CC2)c2ccccc21)NCC12COC(CO)(C1)C2 C1(NC(CCCSC)=O)C=CCN(C(=O)C(C)(C)Cc2ccccc2C(F)(F)F)C1 N1(Cc2ccc(OC)c(-c3ccc(C(C)=O)cc3)c2)CC(C2(C)CCCCC2)C1 C#CC1CCCCN1C(=O)CCN(C(c1cc(C(N)=O)[nH]n1)=O)CC N1(C(Cc2cc(C)nn2C)=O)CCOC2CCN(C(C3CNC(=O)CC3C)=O)CC12 c1(C(C)C)ccc(C=CC(=O)NCC2CN(C(=O)CC3CSCCS3)C2)cc1 C(=O)(CCCCCCSCO)N1C(CC)(CO)CCC1.c1(C(=O)O)nc(Cl)oc1C C1(CC)CN(C(C2CC2c2ccn(C)c2)=O)CCN1C(c1nn[nH]c1Cl)=O CCCC(C(=O)NCC(O)CNC(c1sccc1NS(C)(=O)=O)=O)N(C)C N#CC1(CNC(=O)C(CO)NC(=O)CC(O)C2CCCC2)CCCC1 N1(C(c2ccc(N(C)C)nc2)C(=O)NC(CC)C)CCC(OC)(CO)CC1.CC c1(C(N2CCCC(F)(CNC(CC(C)SC)=O)C2)=O)cc2ccccc2o1 CC(C)C(C)CC(=O)N1CCN(N2CCCC2)CC1C.CC(F)(F)F C(=O)(C#CC1CCCC1)NC1CCC(CNC(C2COC(C)(C)O2)=O)C1 c1(SC)ccncc1S(=O)(=O)N(C)Cc1cscn1.CC(CSC=O)C(F)F C(=O)(C1CCCn2cnnc21)NCCCC(C)NC(c1cnns1)=O c1(Nc2nn(CC)nc2C)ncc(C)cc1S(=O)(=O)NCC1CCN(C)C(C)C1 c1(C(N(CC(CCCC)CC)C)=O)ccccc1S(=O)C(F)(F)F c1(CC(N2CCC(C)C(CNC(c3cnsc3)=O)C2)=O)ccccc1S(C)(=O)=O CCC(C)(C)CC(=O)NCC(=O)N(CC)Cc1cn(C(c2cnn(C)c2)C)nn1 N12CCCC(C1)N(CC)CCC2=O.c1(C(C(=O)NC)O)ccc(F)cc1 c1(C(N2CCC(CS(C)(=O)=O)C2)C(=O)NCCOC)ccc(C2CC2)cc1 Cc1cncc([N+](=O)[O-])c1NCP(C)(C)=O.N12CCN(CC1)CC2=O c1(CC(=O)NC(C)CN(C(=O)CCS(N)(=O)=O)C)cccc2occc12 c1(C(=O)NCC(CCOC)NC(=O)C(C)O)cc(NC(C)=O)ccc1C c1(NC(N2CCC(CC3(COCC)CC3)CC2)=O)ccc(OC)c(OC)c1 c1(C(N2C(C(=O)Nc3ccc(C)nc3)CSCC2)=O)ccn2cncc2c1 C1(CC(N2CC(NC(COC)=O)C2)=O)CCN(C(=O)CC2CCC(C)(C)O2)CC1 C(CN=c1[nH]cnc(CC)c1F)N(C(C(C)OCCCC)=O)CC Cc1n[nH]c(C)c1CC(C)C(=O)Nc1nc(CN2CCOCC2)cs1 c1(OCC)cc(N2CCOC(CNC(c3cnnn3CC)=O)C2)ncn1 Cc1nnc(C(=O)NCC2CCCC2NC(=O)C(F)CC2CC2)s1 C1(C(=O)Nc2c(C)cc(C#N)nc2)CCCCCCN1C(C1CC2(CSC2)C1)=O C(C(=O)N1CC(O)CCO1)N(C(=O)C(C)CSCC)CC#C c1(N2CC3CN(C(Cn4ccc(C)n4)=O)C3C2)ncnc2c1ncn2C1CC1 c1(C(=O)NC2CCN(C(c3c(C)n[nH]c3)=O)CC2F)ccc2oc(O)nc2c1 C(C)(CCC(=O)NCCC(O)C(=O)NCCC(O)C(F)F)OC C(C(C(=O)NCCc1cc(C)no1)NC(=O)CCOC1CC1)OC.O=CC1CC1 c1(NC(C(C2CCC(C)CC2)OC)=O)ccccc1CSC CC(C)(O)C(F)C(=O)NCC(C1CCCCC1)NC(c1c[nH]cc1Br)=O C1(OCC)C=CCN(C(=O)NCc2sc(Cc3ccccc3)nc2C)C1 C1(NC(c2ccc(O)cc2F)=O)CC12CCC(NC(C1CC3CC3C1)=O)CC2 c1(C(=O)NC(CCCNC(c2cccc(C)n2)=O)(C)C)ccnc2[nH]c(C)nc12 C(=O)(C(CC(C)C)OCO)N(CC(CC)NC1CN(C)C(=O)N1)C c1(C(c2n(CC)nnn2)NC2COCC2C(C)(C)C)cc(OC(C)C)cc(=O)o1 N1(C(c2ccoc2Sc2ccccc2)=O)CCCCC(NC(=O)COC2CC2)C1 C1(NC(C2N(C(C(C3CCOCC3)C)=O)CC3CC32)=O)CCCCNC1=O Cc1cccc2cc(C(=O)NC3CCCCC3NC(c3ccnc(O)c3)=O)[nH]c12 Cc1ncc([N+](=O)[O-])cc1C(=O)NC(c1ccccc1)C(C)NC(=O)C=CCO C12(NC(CC(C)OC)=O)CCC(C1)N(C(c1nccn1C(C)C)=O)C2 CS(=O)(=O)c1coc(C(N2CC3(NC(c4cc(CCCO)on4)=O)CC2C3)=O)c1 C1(C(=O)NCCC2CN(C(c3ccc(OC)c(N)n3)=O)C2)CCCCC(=O)N1 C(C(CCOC)NC(C1(C)CC(C(=O)OC)C1)=O)NC(CC=C)=O C(c1cncc(C)c1)=CC(=O)NC(CC=C)CNC(c1c[nH]nc1CCC)=O c1(NC(c2ncc(-c3cn(COC)nc3)c(C)c2)=O)cnc(Br)c(Cl)n1 C(=O)(C(C)CC(=O)N1CCC(NC(=O)C(C)OCc2ccccc2)CC1C)OC c1(C(COC(C)C)C)cn(CCCC(=O)NCC2CCC(F)C2)nn1 C1(C)(CNC(c2ccc(OC)cn2)=O)CCCN(C(C2CCCOC2)=O)C1 C(N=C(NCC(F)F)N1CCN(C)C(C(C)(C)C)C1)C1CC(=O)N(C)C1=O N1(C(C2CC(C)OCC2)=O)CC2CC(NC(c3ccc(F)o3)=O)CC2C1 Cc1nc(C(N2CCC(NC(c3cc[nH]c3C3CC3)=O)C2)=O)cc(O)n1 c1(NC(c2ncccn2)CC)cc(NC2CCOC2C2CC2)ncn1 C1(NCC(C)NC(c2ccnn2CC(F)(F)F)=O)CC(F)(CC2C(C)C2(F)F)C1 C1(CNC(=O)CC2(C(F)(F)F)CC2)CCC2CCC1N2C(=O)C(F)=CC1CC1 C1(CC(=O)NC(C(C)NC(c2nc(COC)sc2)=O)(C)C)CC2(CCC2)C1 C12(C(=O)NCCC=C)CCC(C(=O)Nc3c(C)nn(CC)c3C)(CC1)CC2 N1(C(C2CC(CC)C2)=O)CCC(CNC(C2(COC)CCC2)=O)C(O)C1 C(CCCCCC(=O)NC1CCC(Cn2cc(-c3ccccn3)nn2)C1)SC C(=O)(CCCCCF)NCC(CC=C)NC(C1(Br)CC1(C)C)=O Cc1cc(C2=NNC(=O)CC2C)c[nH]c1=NCc1c(C)cc(C(F)(F)F)cc1C CC1(C#N)CCCN(C(C23C(NC(C4CCCO4)=O)C4CC2C3C4)=O)C1 N1(C(CC2CCN(C)C2=O)=O)CCN(C(=O)CSc2cnn(C)c2)CC1CO c1(CN2CCC(C(=O)Nc3c(Cl)ccnc3Cl)C(O)C2)cc(CO)ccc1O C(=O)(C(C)(C)C(C)O)NCC(CC)NC(c1snc(C)c1N)=O C1(CC=C)(NC(C2COCCN2C)=O)CCN(C(=O)CCc2nc(O)n[nH]2)C1 CCCCCC(O)C(=O)N1CC(O)(CCNC(C2CC2C(F)(F)F)=O)C1 C1(C(=O)NCCN2CCOC(c3ccccn3)C2)CCC2(CCC2)CC1 O(NC(=O)C=CC(=O)NCC(c1ncc(CC)s1)=O)CC(CC)C C1(CNC(C=CCOC)=O)CN(C(=O)C(CC)CCOC)CC12CCC2 CC1CC(C(N2CC(CO)C(C)C2)=O)CN(C(c2ccn(C3CC3)n2)=O)C1 c1(C(C(=O)NC(CC)C)N(CCCCNC(C)=O)C)ccc(-c2ccccc2)s1 C(C(=O)N=c1ccn(CCc2cccs2)[nH]1)c1cn(C)nn1 C1(NC(=O)NCc2c(OC)cccc2OC)CC(O)CC(C)(C)C1 N1(C(C=CC=CC)=O)CCCN(C(=O)CC2COCCO2)CC1CO c1(CN2CCN(C(c3c[nH]c(Br)c3)=O)CC2)cc2ccncc2[nH]1 N1(C(c2cccc(C#N)c2)=O)CC2CN(C(c3ccc4ncnn4c3)=O)CCC12 Cc1nn(C)c(C)c1CCC(=O)N1CC(CNC(=O)C=C2CN3CCC2CC3)C1 c1(C(=O)NCCCN(C(CCc2n(C)ncc2)=O)CCO)nc2c(s1)COCC2 N1(C(=O)CC2CCCC2)CCC(C(=O)NCc2ccccc2F)(CO)C1 N1(C(c2c[nH]c(=NC)s2)=O)CCN(C(=O)CC2CCCCC23CC3)CC1C1CC1 C(=O)(CCCn1cc(C(C)(C)C(N)=O)nn1)NC(c1cccnc1)COC c1(CC(=O)NCC(C(=O)N2CCC(OCC(N)=O)C2)N(C)C)cccnc1F n1(CC(N2CCC(C)(CCNC(C3(C#C)CC3)=O)C2)=O)cc([N+](=O)[O-])ccc1=O c1(C(=O)NC2C(c3ccc(C)cc3)C2)ccc(Br)cc1Cl c1(C(C)C)cccc(C(=O)N(CC(C)NC(C2CC2c2cncnc2)=O)C)n1 CN1CCn2nc(C(N3CC4CCC3C(CNC(c3cnsn3)=O)C4)=O)cc2C1 C#CCCN=C(NCCc1ncc(C)s1)N1CCC(F)(F)CC1 CCCC(C)(CCC)C(=O)NCC=CC1(C)CCC(NC(c2ncn(C)n2)=O)C1 c1(C(=O)NC2CC(CCNC(CSC)=O)C2)ccc(F)c(C(F)(F)F)n1 N(C)(S(=O)(=O)N1CCN(C(C(=O)NC2CC2)C2CC2Cl)CC1)CC c1(C(=O)NCC2(C)N(C(C3C(C=C)OCC3)=O)CCC2)c(C)nn(C)c1Br C1(CNC(c2c(CC)n(CC)nc2)=O)CN(C(=O)CNC(N)=O)CC12CCC2 c1(OCCC(=O)NC2C(NC(C3(C)CCCO3)=O)C2)ccc(S(N)(=O)=O)cc1 c1(CN(C(c2nc(C3CC3)n(C)n2)C(=O)NCC)C)cc(C)nc(Cl)c1 Cn1cc(N2CCC(CC(=O)NC(C)(C)CCNC(=O)C(=O)N(C)C)C2)cn1 C12(C(=O)NCC3CN(C(CCCC#N)=O)C3)CC3CC(C1)C(=O)C(C3)C2 C(=O)(N1CC(O)C(O)CO1)c1c(C2(C#N)CC2)cccc1 N1(C(C2(OC)CC2)=O)CC(C(N2CC3CC2CO3)=O)OC(C)C1 C(c1cc(Br)cs1)=CC(=O)NCC1CCC1NC(=O)CCc1cccnc1 N1(C(C2CN(C(C)C)C2)=O)CCCCCC1C(=O)NCC1CN2CCC1C2 N1(CC)CCN(C(C2CCC(N3CC(O)C3)C2)=O)CC1.c12cc(cs1)NC2=O N1(C(CCC)=O)CCCC(C2CC2N(C2CCCC2)C(=O)CC2(N3CCCC3)CC2)C1 O=C1OC2CC(C(N3CCC(NC(=O)CCn4cc(Cl)cn4)C34CC4)=O)CC2O1 C1(C(=O)NC2C(COC)CCC2)CC2CCCC2N1C(c1ccc(O)c(F)c1)=O c1(OCC)ccc(NC(=O)CC(CC)NC(=O)C=CCO)cn1 Cc1nccc(C(=O)NCC(O)C(=O)N2CCC(c3cnn[nH]3)C2)n1 C1(CCNC(=O)C(C)CSC)(OC)CCN(C(c2cn(C(C)C)nn2)=O)C1 c1(C(=O)NCC2CN(C(CCCCCC)=O)CC2(C)C)cc(C#N)c(F)cc1F C1(CCNC(C(n2cc(Cl)cn2)C)=O)CCCN1C(C1CC(C)(O)C1)=O O=C(C(CO)C(F)(F)F)N1CCCC(CCNC(C2(c3nccs3)CC2)=O)C1 C#CCC(C)(C(=O)NCCCC1CCOC1)NC(=O)C=Cc1ccc[nH]1 N1(CCCC)CCCCC1C(=O)NC(c1nnc(C)s1)C(=O)OCC C(=O)(CCCCC(C)CC)N1C(CCNC(CCC(C)OCC)=O)C(C)CCC1 C1(C(C)NC(C2(CC)CC2)=O)CCCCN1C(c1sc(-c2cccs2)nc1C)=O CN1C(C)(C)C(CNC(N2CCCCC(C)(F)C2)=O)CS1(=O)=O CC(C)C(O)C(C)N=c1nc(N2CC3NC(=O)OC3C2)c2c([nH]1)CCC2 C(=O)(C(C(C)C)C(C)C)N1C(C(N(CC(CC)O)CC)=O)CC(O)CC1 c1(C(=O)OC)ccc(CCNC(=O)NC(c2cnc(Cl)s2)C2CC2)cc1 C1(NC(c2cncc(Cl)c2)=O)CC2CC(NC(C34C=CC(CC3)C4)=O)CC12 c1(C2CC(=O)NC2)ccc(C(=O)NCCn2cc(CCO)nn2)cc1 C1(NC(CC=CC(C)(C)C)=O)C2CC3C1C3C2C(=O)NCc1nc(CN(C)C)n[nH]1 N1(CC)C(=O)CCC1C(=O)NC1CC1CNC(=O)CCc1nc(C)c(C)[nH]1 N1(C(C2(C)CCC3CC3C2)=O)C2CCC1CC(NC(c1cccnc1S)=O)C2 C1(NC(CN(CCOC)C)=O)(CNC(C2(n3ccnn3)CC2)=O)CCOC1 N1(C(CS(CC)(=O)=O)=O)CC2CCC(C1)C2N(C1COCCC1O)CC C1(C(=O)NC(c2nnc(O)o2)C)CN(C)CCN1C(c1ccncc1Cl)=O CCCC(CC(C)C)C(=O)NCC1(C)CN(C(c2ncc[nH]c2=O)=O)CC1C c1(C(=O)NCC2CC(NC(=O)C(F)CC3CCC3)C2)ccc2ncncc2c1 c1(OC)cc([N+](=O)[O-])ccc1C(=O)NC(C)CNC(c1oc(C(F)F)cc1C)=O c1(CC)ccc(C(=O)NC2CN(C(C3CCC3OC)=O)C2)c(Cl)c1 C1(C(=O)NC(c2cnc[nH]2)C)COCCN(C(c2cnn(C)c2)=O)C1 C(c1ccccc1)=C(CC)C(=O)NC1(C2CCCCN2C(c2c[nH][nH]c2=N)=O)CC1 N1(C(CCCCC(=O)OC)=O)CCC2CCN(C(=O)C(C)=C(C)C)C2C1 Cn1ccc(C=CC(N2CCC(NC(C3CC3c3cccnc3)=O)C2)=O)c1 c1(C(=O)NCC(CCOC)NC(C2CCC(=O)NC2)=O)cccc2c(C)[nH]nc12 CN1CCCCCC1C(N1CCCC(CCC(=O)NC2(CO)CCSC2)C1)=O c1(CC(=O)NCC2CCC(F)(CNC(C3CN(C)C3)=O)C2)ccc2c(n1)CCC2 C1(C(N2CCCC(CNC(C=C(C)C)=O)C2)=O)CC12CCOCC2 c1(C(N(C(CNC(CC2(OC)CC2)=O)C)C)=O)oc(C(C)C)nc1C c1(C(N(C2CC(NC(c3ccnn3C3CC3)=O)C2)C)=O)cc2sccc2cn1 c1(N(C)CC2CCSCC2)nc2c(c(=NC3COCC3F)[nH]1)COCC2 CCCC(C)(O)C(=O)NCC1CC(F)(CNC(=O)CN2CCCC2)C1 C(CCC(C)C(=O)N1CCCC(CC(=O)Nc2cc(C)cc(F)c2)C1)OC CC(C)C(C(=O)NCC1CN(C(C2CCN(C(N)=O)CC2)=O)CC1C)N(C)C C12(CNC(C3(CC#C)CC3)=O)CN(C(=O)C(c3ccccc3F)C)CC(F)(C1)C2 c1(OC)ccc(CNC2CC(C(=O)NCCF)C2)cc1OCCC(C)C C(=O)(CCCC(N)=O)N(C1CC(NC(CC(CC)OC)=O)C1)C C1(C(=O)NCc2cc(C)ncc2)CC12CCN(C(c1cc(Cl)ncc1F)=O)C2 c1(C(=O)NCC(CC)NC(=O)C(C)Cn2ccc(C)n2)ccc(O)cc1Cl C(=O)(CCCSC)N(C1CCN(C(C2(F)CC2)=O)C1)CC c1(C(N2CC(C)(c3cn(CCO)nn3)C2)=O)ccc2c(c1)CCC2 Cc1cc(N)c(C(N2CCCC(NC(C3C=CC=CC=C3)=O)CC2)=O)cc1F c1(C(C)C)ccc(Br)c(C(c2nnnn2C)NCCC2(C)CCOCC2)c1 N1(C(C(C)O)=O)CC2(C1)OC1(CO)CC2(NC(=O)Cc2ccnc(F)c2F)C1 C#Cc1ccc(C(=O)NC2CCCC2NC(=O)C(C)C(O)CC)cc1 N1(C(CSC)=O)CC2COCCC2(NC(c2cc(OC(C)C)ccc2Cl)=O)C1 C(N=c1[nH]c(N2CCCC(N3CCCC3)C2)nc2c1SCC2)c1c(F)cc(Cl)cc1 C1(NC(C=Cc2nnc(C(C)C)o2)=O)CCCC12CN(C(=O)Cc1cscn1)C2 c1(NC(CC2CCN(C(c3c(C)c(Cl)ccc3)=O)C2)=O)cc(F)c(F)cc1F c1(C(=O)NCCNC(=O)NC2(CS(C)(=O)=O)COC2)ccc(S(C)(=O)=O)s1 c1(CCC(=O)NC2C(CNC(c3c(CC)cno3)=O)C2)ccc2cnn(C)c2c1 N1(C(C(C)Cc2cnn(C)c2)=O)CC(NC(=O)COCCO)CCC1C C1(NC(C(C=CC)O)=O)CC2CCC1N(C(=O)CC1(CS(C)(=O)=O)CC1)C2 CN1CCOC(C(=O)NCC2CC(NC(C3CCSCC3)=O)C2)C1 c1(OCCC)ccc(CNC(N2CCC(c3ccc(C)cc3C)C2)=O)c(C)c1 C1(NC(CC=CCC)=O)CCCN(C(C2CCCCCN2C)=O)CC1 C1(C)(NC(C2(C)CC(C)(C)C2)=O)CCCN(C(=O)CC2CC3(CC3)CO2)C1 CC1OCCC1C(=O)NCC1CCN1Cc1ncsc1Br CC1(C(=O)NC2CC(CNC(C3CCCCC3(C)C)=O)C2)CCCC(F)(F)C1 C(=O)(CCCS(N)(=O)=O)NC(C1CN(C(CSc2nnc(C)s2)=O)C1)C CCC(CC)CC(=O)NCCCN(C(=O)C(C)n1cncn1)CCO C1(C(=O)Nc2cncnc2)(CNC(C(C2CCOC2)OC)=O)CCC(F)(F)CC1 C1(C)(C(=O)NCC(C)NC(=O)C(c2ccccc2F)(C)F)CCCCNC1=O C1(C(=O)NC(CCCCNC(c2c(C)cnn2C)=O)C)CCn2c(O)nnc2C1 N1(C(C23COC(c4ccccc4)(C2)C3)=O)CCCN(C(C2CC(CF)C2)=O)CC1 C1(NC(c2cccc(C)c2)=O)(CNC(=O)CNC(=O)CN(C)C)CCCCCC1 CC(C)(CCCC(=O)NC1CCC2CCC1C2)NC(c1ccn(C2CC2)n1)=O c1(C(=O)NCC(CNC(C2N(C(C)=O)CCC2)=O)O)cc(Br)cn1C(C)C c1(C(=O)NC(CC)CNC(=O)C(C)CSC)c(C)nn(-c2ccccc2)c1C C(C)(C(C)C(=O)NCC(C)N(C)C)NC(C(COC(C)=O)C)=O n1(CCCSC)nnnc1C(C1CC1(C)C)NCc1ncsc1C c1(C(=O)NCCCCCCN(C)C(C2(F)CCCC2)=O)ncn2ccccc12 c1(C(=O)NC2C(NC(=O)Cn3nccn3)CCC2)c(Br)csc1Cl Nc1cccc(F)c1SCC1CCCNCC1 N1(C(CC2(CC=C)CCCC2)=O)CCC2(CC1)CC2CNC(C1CC(C)C1)=O C(C1CCCN1C(=O)C(O)Cn1cncn1)=CC(N1CCC1CO)=O N1(C(=O)COC2CCOCC2)CC(NC(C23CCCC2C3(F)F)=O)C2CCCC12 C(=O)(C1=C(Cl)CCOC1)NC1CCC(C(C(=O)NC(CC#C)CO)(C)C)CC1 n1(CC)nc(C2CC2)cc1C(N1CC(OC)CC1CNC(=O)CC1CCOC1)=O C1(C(=O)NC2C(NC(c3cc(CC)nnc3C)=O)CCC2)CCCC2(CCC2)O1 C1(N2CCOCC2)(CC)CCN(CCCCn2ccnc2)CC1 c1(CNC(CSCCNC(C(COC(C)=O)C)=O)=O)oc(C)nc1C C1(C2CCCC2)(C(=O)NC2CCN(C(C3N(C(C)C)CCC3)=O)CC2O)CCC1 C1(C(N2CC(C)(NC(C(C)NCCCCCC)=O)C2)=O)COC2COCC12 C(=O)(CC1C(=O)Nc2ccc(Cl)cc21)N1CCN(c2c(N)cc(Cl)c(Cl)c2)CC1 N1(C(C(COC)NC(=O)NC2(CO)CC2)=O)CC(NC(c2ccccc2)=O)C(C)C1 C(C(N=c1[nH]nc(C)s1)C(C)C)NC(c1cncc(NC)c1)=O N1(C(C(CSC)(C)NC(=O)CC2CC3(CC3)CO2)=O)CCC(F)(F)CC1C c1(CNC2CCC(C(=O)NCc3nccc(C#N)c3)OC2)cnc2[nH]ccc2c1 C1(C(=O)NCC2C(CNC(C(C)Cc3cnn(C)c3)=O)C2)OCC2CCCCC12 C12(C(=O)NCCOC3CN(C(c4n(C)nc(O)c4)=O)C3)CCC(CF)(C1)OC2 C1(CNC(=O)Cc2cnsc2)CN(C(c2cnc(C(F)(F)F)s2)=O)CC12CC2 Cc1ccc(C(=O)C(=O)NCC2CC2CNC(=O)CC2CCCOC2)cc1 c1(C(=O)Nc2cccc(NC(C3ON=C(C)C3)=O)c2)ccnc2[nH]c(C)nc12 c1(OCC)ccccc1C(=O)NCC1CCCC1NC(=O)CCn1cncn1 CCC(Cc1cccc(C)c1)C(=O)N(CCCCCCNC(=O)C=CCOC)C C1(C(=O)NC(C(=O)OCC)CCc2n[nH]c(C3CC3)c2F)OCC2CCCCC12 N1(C(C(C)NC=O)=O)CCN(C(C2COCCO2)=O)CC1CC#N CC1CN(C(c2cnc(Cl)s2)=O)CCC1N(CC(=O)Nc1ccccc1)C C(=O)(CC1CCC(=O)c2ccccc21)N1CCC(CNC(=O)COC2COC2)C1 C#CCC(C)(CC)C(=O)N1CCCC(CCC)(NC(=O)COC(F)(F)F)C1 N1(C(C2CC(N(C)CC)C2)=O)CC(NC(=O)Cc2conc2C)C2(CCOCC2)C1 Cc1ccc(C)c(S(=O)(=O)NC2CCCCN(S(=O)(=O)c3cccnc3)C2)c1 Cc1nc(C)c(CC(=O)NC(CNC(=O)C(c2ccc(F)cn2)(F)F)C(C)C)s1 N1(C(C2C(NC(c3ccc(F)s3)=O)CCO2)=O)CC2CCC(C1)C(=O)N2 N1(C(Cc2cc(C)nn2C)=O)CCC(C(=O)NCCN(C)C2CC2)C12CCC2 C(=O)(C1=CCC(C)(C)CC1)N1CCC(C(C)C(=O)NC2CS(=O)(=O)C2)CC1 N1(C(c2cc3nc[nH]c3cn2)=O)CCC2CCC(C1)N2C(c1cnncc1O)=O C(=O)(CC(CC)CCCC)N1CC(NC(C(C(=C)C)(C)C)=O)C(O)C1 c1(C(=O)NC2CN(C(CCC=C=C)=O)CC(C)C2)cccc2ncsc12 C1(NC(c2ccsc2)=O)CN(C(c2nccnc2Br)=O)CC1F CS(=O)c1cccc(C(=O)NCC(O)CNC(c2sccc2-n2cccc2)=O)c1 c1(C(N2C(CC)CN(C(C3CCSC3)=O)CC2)=O)cnc2c(F)ccc(F)c2c1 c1(C(=O)NC(C(=O)Nc2c(C)nc(Cl)nc2)CC2CC2)ccn2ccnc2c1 N1(C(c2cnc(C(C)(F)F)s2)=O)CCC2(C1)CN(C(C1CCC3C1C3(F)F)=O)C2 C1(NC(CCCC=C)=O)CC(C(=O)N(C)CCC2CCCO2)=CC1O c1(CCCCn2cc(-c3ccc(CNC(=O)CCCF)s3)nn2)ccc(F)cn1 c1(C(N2C(C(=O)Nc3cncc(CO)c3)CC2)=O)cc(F)c(F)cc1Cl c1(-c2cc(C)cc(C#N)c2)cnn2c1CN(Cc1ccc(C)nc1)CC2 c1(CNC(C(CC)NC(=O)COc2cn[nH]c2)=O)cnc(OC)cn1 C1(SC)CN(C(=O)Cc2cc(F)ccc2Cn2ccnn2)C2(CCC2)C1 N1(C(C(CCC)OC)=O)CC2CCC(NC(c3cc(O)cc(Br)c3)=O)(C2)C1 c1(OC)ccc2[nH]cc(CC(=O)NCCCNC(c3ncnc(C)c3C)=O)c2c1 O=C1NC(=O)C2(CCN(C(C3CNCC3c3ccc([N+](=O)[O-])cc3)=O)C2)N1 N1(C(C2=C(C)CC2)=O)CCN(C(C2(C(F)(F)F)CC2)=O)CC1c1ncc[nH]1 CCCC(=O)NCC(C1CC1)NC(=O)C(C)NC(=O)OC(C)(C)C N1(CCC)C(=O)CCC1C(=O)NCCN(C(=O)C(C)SC(F)(F)F)CC1CC1 C#CC1(C(N2CCCC(CC(=O)NCC3CC3)C2)=O)CCCCC1 c1(C(=O)NCC(CO)NC(=O)CN2CCS(=O)CC2)cc2n(n1)CCCCC2=O c1(SCC)cccc(C(=O)NC2CC2CNC(=O)CO)c1 C(=O)(C(C1CC1)N(C(=O)Cc1cnoc1)C)NCCN(CCC)CCC c1(C(=O)NC(COC)(C)C(N)=O)ccc2c(n1)CN(C(c1coc(C)n1)=O)CC2 C(=O)(CC(C)(C)C(F)(F)F)NCCC1CCN(C(CCNC(=O)OC)=O)C1 c1(CC)cc([N+](=O)[O-])ccc1C(=O)N(CC(C)NC(=O)C(c1ccccc1)C)C Cn1nccc1C1=CC2CCC(C1)N2c1cc(C#N)c2c(Br)cnn2c1 C1(CC(=O)N(C)Cc2c(C)cncc2)CN(C(=O)COCCF)CC(C)(C)C1 N1(C(C(CCSC)NC(C2(C(=O)N(C)C)CC2)=O)=O)CCN2CCC1CC2 c1(C(C)C)ncc(C(N2CC(O)(CNC(C3CC4CC4C3)=O)C2)=O)n1C c1(SC)cccc(NC(=O)C(C)=CCNC(=O)C(n2ccc(C)c2)C2CCOC2)c1 C(C(CC(F)(F)F)NC(=O)CSCc1nnnn1C)NC(C=CC(=O)N(C)C)=O C=Cc1cncc(C(=O)NC(CNC(=O)CCc2ncccn2)C(C)(C)C)c1 N1(C(Cc2cc(C)sc2)=O)CCN(C(=O)C(C)Cn2ccnc2)C(CO)C1 C1(C(N2C(CC)C(NC(=O)CCc3ccc(C)s3)CC2)=O)COC2(CCC2)C1 c1(OCC=C)cc(C(N2CC3CC3C2)C(=O)NC2(C)CC2)ccc1OC C1(C(N(CCNC(c2cncc(C(C)(C)C)c2)=O)CC)=O)CC12CCCOC2 C1(C(C)(C)C)COCCN1C(C1CCCN(C(c2cccnc2)=O)C1)=O C1(CNC(c2ccc(F)s2)=O)CCCN1C(=O)C(Cc1ccccc1)C1CC1 Cc1oc(C(=O)NC(C)CCNC(=O)CC2CN3CCC2CC3)cc1S(N)(=O)=O c1(C(C2CCCOCC2)=O)nccnc1CCC(F)(F)F CCC(C)C(C(=O)OC)OC(=O)Cc1csc(NC(c2cncn2C)=O)n1 C1(CC(N2C(C(=O)NCC(C(C)C)O)C(C)CC2)=O)CCC(=O)C1C n1(CC#C)cc(COC(c2cncnc2C(C)C)=O)c2ccccc12 CC1CCC(C)(C(N2CCN(CCCCCNC(c3sccc3F)=O)CC2)=O)C1 CCS(=O)(=O)CC(=O)NC(CNC(=O)C(C)OCCN(C)C)(CC)CC C(C(C)(C)C(=O)N(C1CN(C)C1)C)N(C(C=CCC)=O)C CCCC(C)(O)C(=O)NC1COCC1NC(c1c(Cl)cccc1Cl)=O C(c1ccco1)=C(C)C(=O)NC(CC(=O)NCC(C)C(C)C)C1CC1 C=CCC(CC(C)C)C(=O)N1CCC(O)(CN(C)C(c2cccc(F)c2Cl)=O)C1 C(=O)(C(CNC(=O)C(C1(O)CCCC1)F)C(C)C)N1CC(NC(=O)OC)C1 n1(CC(=O)NCC2N(C(CCNC(=O)C=CCl)=O)CC2)nnnc1CC1CC1 C(=O)(C(CO)C(C)(C)C)N1CC(O)(C(C(=O)N(CCn2c(C)ncc2)C)F)C1 C#Cc1cncc(C(=O)NC2CN(C(C3CC=CCO3)=O)CC2(C)C)c1 C(=O)(CC(C)C(C)C)NCC(=CC(N1CCN(C(CC)CC)CC1)=O)C c1(C(N2CCN(S(=O)(=O)CC3CC3)C3(CCC3)C2)=O)ccc(O)c2ccccc12 Cn1ccnc1S(=O)(=O)NC1CN(CC2OCCO2)C1 C(=O)(CC(C)(C)C(=O)NCC(O)CN(C)C(c1nc(C)n(C)n1)=O)OCC c1(OC)c(C)csc1C(N1CCSCC1CCNC(C1(SC)CC1)=O)=O CCC(CC(=O)NCCCOCCOCCNCc1cc(C)nn1C)CC(C)C C1(OC)CC2CC1CN(C(=O)CC(C)(C)CNC(=O)C(F)(F)C1CC1)C2 C1(NC(C(CCOCCO)NC(=O)C=C2CCC2)=O)Cc2ccccc2C1 C1(C(=O)NC(C2(CNC(c3c(C(C)C)noc3)=O)CC2)C)CN2CCCN1CC2 C1(C(=O)Nc2ccc(C)cc2O)(CC)CCCN(C(=O)C(=O)NCC(C)C)C1 C1(NC(COC(CC)(C)C)=O)(CO)CCN(C(=O)CCC(C)SC)C1 Cc1cccc(CC(=O)NCC(C)(C2CC2)NC(=O)CCc2cn(C)nn2)c1F c1(C(=O)OCCNC(N2CCCC(CC#N)C2)=O)ccc2c(c1)C(=O)NCC2 CCCCCCCC(C=O)N1CCCc2ccc(CC)cc21 Cc1nn(C)c(C)c1OCC(=O)NCC(C)NC(=O)C=C1CCC(C)C1 N1(C(COCC)=O)CCC2C1CCCN2C(C)=O C1(CC(N2CCC(NC(CN(C(C)=O)C)=O)(CO)C2)=O)CCCC(C)(C)O1 CC(C)(C(=O)NC1CC(CCC(=O)NC(C(N)=O)C2CC2)C1)n1cccn1 CC(C)CC(C(=O)NCC(F)CNC(c1ccoc1)=O)N(C)C(=O)OC(C)(C)C c1(NCC=CCOCC)[nH]c(=NCc2cccc(OC)n2)nc2ncn(C)c12 c1(C(=O)NCCCCc2nc(C)sc2)cccc(S(=O)(=O)CC(F)(F)F)c1 c1(C(N2CCC(C(C(=O)NCc3n(CC)cnn3)C)C2)=O)ccncc1N C(=O)(C(C(C)C1CCCC1)N1CCOC(C(C)(C)O)C1)NC(C)C c1(CC(C)NC(=O)NC(c2nc[nH]n2)C)ccc(Cl)s1 C1(C(=O)NCC2CCC(C)N(C(=O)Cc3ccoc3)C2)CN2CCCN1CC2 C1(COC)CC(CNC(C2(C)CCCCO2)=O)N(C(=O)C=CC(=O)N(C)C)C1 c1(CCC(c2n(CC)nnn2)(C)NC(C)CCSC)ccccc1F c1(C(=O)NC(CCCNC(CCC(C)OCC)=O)C)ccn2c1CCCC2 c1(CSCC(=O)NC2CCN(C(C3CC(O)(C(F)F)C3)=O)C2)ccc(F)cc1 C(C)(C(C)(C)C(=O)NCC)NC(c1n(CCCC)nnn1)c1cc(C2(C)CC2)n[nH]1 C1(NC(C(CC)NC(N)=O)=O)CCC12CN(C(=O)CCCOc1ccccc1)C2 C(CC(=O)N1CC(OC)C1)N(CC)CC.C(C)(C(=O)NC)NCC C(C(=O)N(CCC(C(C)C)NC(=O)C1=CCOC1)C)(C(C)C)(C(C)C)NC(C)=O N(C1CN(C(=O)C(CO)NC(N)=O)Cc2ccccc21)C(CC1(C=C)CCC1)=O C(=O)(CC(O)c1cc(C)cs1)NCC(CNC(=O)Cc1ccsc1)OC Cc1nc(C(C)(C)C)nc(C)c1C(N1CCC(CNC(C2C=CCC2)=O)CC1)=O N1(C(C2CC2C(C)(C)O)=O)CCN(C(=O)CCNC(=O)OC(C)(C)C)C2CCC12 Nc1ccc2nccc(C(=O)NC(c3ccccc3Cl)c3nccn3C)c2c1 c1(CC(=O)OC)ccc(CN=C(NCC2CCCO2)NC2CCCC2(F)F)cc1 c1(COC(C(N2CCCC(O)C2)C)=O)ccc(C#N)cc1 C(C(C)C(F)F)NC(CC=CCNC(CC1(C)CC1)=O)=O Cc1ccc(CC(=O)NCCN(C(=O)CCn2cnnn2)CC2CC2)c(C)c1 c1(C(N2CC(C(N)=O)(CNC(C(CC)n3ccnc3)=O)C2)=O)sc(CO)nc1C N1(C(CCOCCOC)=O)CCOCC(C(=O)N(C(C)C)CC2CCCS2)C1 C(CCCCC(=O)N1CCCC2(CCC2)C1)=CCCC.C1(=O)CSCCN1 c1(N2CC(CC)OCC2)nc(N2CCC(C)C(C)(C)C2)nc2ccsc12 Cc1cc(C(=O)N(C2(C(=O)NC3CC(n4cccn4)C3)CCC2)C2CC2)c(C)cn1 c1(OC)ccc2c(n1)NC(C(=O)NCC1(C)CCCN1C(=O)C1=CCCOC1)C2 C1(NC(C(COCC)OCC)=O)CCC(NC(c2cn(CCO)nn2)=O)C1 c1(CC(=O)NC(CNC(CC=CC)=O)CCOC)ccc2c(ccn2C)c1 c1(OC)ccc(CCC(=O)NCC2CCN(C(C3C(Cl)(Cl)C34CC4)=O)C2)c(F)c1 c1(C(N2CC(COC)(CNC(c3ccccc3C)=O)C2)=O)cccc2c1COC2 CC1CN(c2ncc(C(=O)NC3CC3c3ccc(F)cc3F)cn2)CC(C)O1 C(CC1(C#N)CCC1)(C(=O)NC(C)CC)N(C(C=C)C1CC1)C1CC1 C(CC(=O)NCC1C2CCC(C2)N1C(=O)CSC(C)C)(C(N)=O)NC(=O)OC c1(C(=O)NCC2(NC(C(C)OC3CCCCC3)=O)CCOC2)cc(N)cc(O)c1 C(C#Cc1cccnc1)NC(C1(CNC(C2CCC(O)C2)=O)CC=CC1)=O Cc1ccc(C(N2CCC(NC(C3CC3(C)C)=O)C23CC3)=O)cc1Cl c1(C(C(=O)NCC(O)C2CC2)NC(c2ccc(Cl)o2)=O)cccnc1 C(=O)(C(CC(C)C)NC(=O)CCP(C)(C)=O)NC(c1c(C)noc1C)C C1(N(C(CSCCN(CC)CC)=O)C)CCCN(C(=O)CC2CCC(C)(C)C2)C1 c1(C(=O)NCCCC(C)NC(C(C(C)C)SC)=O)cnn2c(=O)cc[nH]c12 CCCCC(C(=O)NC)NC(C1CCCN(C(C2(C(C)C)CCC2)=O)C1)=O N1(C(c2csc(Cl)c2)=O)CC2COCC2(C(N2CCOCC(CO)C2)=O)C1 N1(C(CSCCC)=O)CCN(C(=O)C=Cc2ccc(C(N)=O)o2)CC(O)C1 C#Cc1cc(C(N2CCC(CC)C2C(=O)N(C2(CC)CC2)C)=O)ccc1C C(=O)(CC(C)(C)C)NC(C)C(=O)NC1CCN(C(c2c[nH]c(C(N)=O)c2)=O)CC1 N1(C(C2(Cl)C(C(C)=O)C2)=O)CCC(C(=O)NC2CCCNC2=O)(CF)C1 C(=O)(CCCC(C)(C)NC(=O)CC1CSCCO1)N1CC(C)(C#N)C1 C1(NC(=O)C(C)c2ccsc2)(CC(N(CC)Cc2ccco2)=O)CCCC1 c1(C(=O)Oc2cccc(OCC)c2)nnn2ccccc12.C12CCCN1C2 CC1C(C(=O)NCCC2(CO)CC2)CCCN1C(C1CC2(CC2)CO1)=O CC(C)CC(CNC(=O)C(C(C)C)N(C)C)NC(=O)CC(C)(F)F C(=O)(C(F)(F)CCn1ccnn1)N1C(C(N(CC)CC23CC(C2)C(C)O3)=O)CC1 c1(C(=O)NCC(C)(CO)NC(c2nc(C)sc2)=O)ccc(N(C)C)cc1C c1(C(=O)NCC(CC)N(C(=O)CCOC2CCC2)C)cnn(CCF)c1 Cc1cnc(C)c(C(N2CC(NC(c3cscn3)=O)CC(O)C2)=O)c1 CC1CCC(CCNC(=O)NCC2CC2c2cncs2)O1 N1(C(C(C)NC=O)=O)CCC(n2cc(NC(c3ccnc(Br)c3)=O)cn2)CC1 C=CCCCCCC(=O)NC(=O)CCc1ccn(C)n1.C12(CC)CN(C1)C2=O CC1CN(C(c2cn(C(F)F)cn2)=O)CC1NC(=O)C=Cc1ccco1 c1(CC)ccc(C(=O)NC(C)(C)CNC(=O)C(O)CC2CC2)cc1Cl c1(OC)ccc(C(=O)CCC(=O)OCC2CCCC(O)C2)cc1 c1(N2C(CNC(c3c(CC)nc[nH]3)=O)CCC2)ncnc2c1CCS2 c1(CCC(N2CCCC(N(C(C3C(C(C)C)C3)=O)CCO)C2)=O)ccc(Cl)c(F)c1 N1(Cc2cnc(CC)s2)CCCCC1NC(=O)Nc1ccc(F)cn1 CC1(C(=O)NC2CCC(CCNC(C3CC3C3CC3)=O)C2)CC2(C1)CC(F)(F)C2 C(CCCCC=O)NC.N1(C(=O)CC2CCCSC2)CC2(C1)CC2(F)F N1(C(C(CCC)N(C)C)=O)CCC(C)(C)C1C(=O)NC1CC1(C)C(F)F c12ccncc1N2.C(CC(=O)NC1(C(=O)NC)CC1)N(CCC)C.C1(O)CC1.CC N1(C(C2=C(C)CC2)=O)CC2(CCN(C(C3CCN(C)C3=O)=O)C2)C1 C(C(C)(CC(C)C)NC(=O)CC1CCCC1)NC(C1(C(=O)OCC)CC1C)=O C(=O)(Nn1cnc2ccccc12)C1N(C(C(C(C)C)C#N)=O)CC2CC21 N1(C(C2N(C(CCC)=O)CCCC2)=O)CCC(CNC(=O)CC(C)(F)F)C12CC2 c1(C(N2CC(C(C)NC(C3CC(C)(O)C3)=O)OCC2)=O)cnc2c(c1)CCOC2 C(N=c1ccn(C(C)(C)C)[nH]1)(c1c(C)ncc(SCC)c1)c1n(CC)nnn1 N1(C(c2c(C)n(C)nc2)=O)CCC(NC(c2cnc(O)n2C)=O)C(C(C)C)C1 c1(C(=O)NC(C)CN(C)C(C2C=CCC2)=O)ccn2cc(C3CC3)nc2c1 CCCCN(OC)C(=O)C1CCCCCC1Nc1ccc(Cl)s1 c1(C(=O)NCC(C2CC2)NC(C2(SC)CC2)=O)ccc2c(c1)C1CCC2O1 C1(CCC)CCC(C(N2CC3C(NC(c4nnc(C(C)(C)C)s4)=O)C3C2)=O)CC1 N1(C(C2C(OC)CN(CC)C2)=O)CCN(C(=O)Cn2ccnn2)CC1CF C(=O)(CC(C)CC(=O)O)Nc1c(C)c(-n2cc(C3(C(=O)O)CC3)nn2)ccc1 C(=O)(C1=CC2CCC(C1)C2)N1CCC(CC)CC1C(=O)N(CCCC(O)CO)C c1(C(=O)NC2CN(C(CCNC(=O)NC)=O)CC2C)cnc(N(C)C)c(Cl)c1 c1(SCC(=O)NCC(CCOC)NC(=O)CCC2CCC2)ccccc1F C1(N(C(Cc2cn(CC)nc2)=O)C)CCN(C(c2nnn(C(C)C)c2C)=O)CC1 c1(C(N2CC3C(CNC(C(C)Cc4cnc[nH]4)=O)(C3)C2)=O)cnn2cccnc12 C1(COC)CC12CCN(CC1CCCN(C(=O)OC(C)(C)C)C1)CC2 C1(OC)(CNC(=O)CCCCN(C)C)CCN(C(c2ccccc2CC#N)=O)C1 c1(NC(C2C=CCN2Cc2cccc(-n3ccnc3)c2)=O)cc(F)cnc1Cl C(CCC(O)C(=O)N1CC2CC1CC2O)NC(CCn1ccc(C)n1)=O C(C(C)(CC(C)C)NC(=O)C(C)Oc1ccccc1F)NC(c1c(C)onc1)=O CC(C)C1=NOC(C(=O)NCC2(O)CCN(C(=O)CSc3nncs3)CC2)C1 N1(C(CC(=C)C)=O)CCC(COC)(NC(=O)CC2CN(C)CC2O)CC1 C1(C(N2CC3(CC(NC(C(CN(C)C)O)=O)C3)C2)=O)CCc2nncn2CC1 c1(C(N(CCOCCNc2snc(C(=O)OC)n2)C)=O)cc2cnc(Cl)cc2s1 c1(C(N(CCC)CCNC(=O)CC2CCC(O)C2)=O)ccc(OC(C)C)cn1 C1(C(=O)NC(CNC(Cn2ncc(C)c2)=O)C)CN(C)CC(C)O1 CCCC(O)(CCC)CC(=O)NCCCCC(C)NC(=O)C(C)=CC CC1(C)CCC(O)(C(=O)NCCC2CCN(C(=O)CN3CC4CCC3C4)C2)CC1 c1(NC(N2C(C)(C)CC(C)(CO)C2)=O)cncc2ccc(F)cc12 C1(C(=O)NCc2c(C(=O)NC(c3c(C)noc3C)C)[nH]cc2)CC(=O)NC1(C)C Cc1cccc(CNC(C(F)(F)C2CCC2)=O)c1.C1CCN1C(C)(C)C N1(C(C2(CC)CCC2)=O)CC2CC(C(=O)N(C)CC3CCOC3C)CC2C1 c1(C(=O)NCC(c2ccccc2F)(F)F)cc2cc(Br)cnc2o1 c1(C(N2CC(O)CC2CNC(C23CCCC2C3(F)F)=O)=O)cc(O)cc(O)c1 n1(CC)c(C(=O)NC2CCCCC2CC(N2CCCC(COC)C2)=O)cnc1O CC1(F)CCCCN(C(C2CC(NC(C3CC4(CSC4)C3)=O)CCO2)=O)C1 c1(C2(N)CC2)c(F)cccc1F.C12(C=CCC1)C(=O)N1CC(C1)C(C)NC2=O.CO c1(NC(C(c2cccc(Cl)c2)C)=O)cccc(C(=O)NCC2CCCO2)c1 C(=O)(C1=C(F)CN(C(c2csc(CO)n2)=O)CC1)Nc1c(C)ccc(C)c1 C#CC(CC(C)(C)C)NC(c1cc(CNC(C2CC(C)(F)C2)=O)ccn1)=O c1(OC)c(C(=O)NC2CC(NC(=O)CCNC(C)C)C2)cccc1Br N1(C(c2cc(-c3cn(C)nc3)[nH]n2)=O)CC2CC2(NC(=O)CSC(F)F)C1 c1(OC)cccc(CC(=O)NC2CCN(C(=O)C(O)C(C)(C)C)CC2F)c1Cl C(=O)(C1CCc2cc(Cl)ccc21)N(C1CCN(C(=O)CSSC)CC1)CC#C C1(C(C)C)CCCCC1NC(=O)CN(C(=O)CC1CC=CC1)C(C)C CCC(C)CC(=O)N1CCC(n2cc(CNC(=O)CC3CC3)nn2)C1 CC1(CC(=O)NCC=C2CCN(C(c3cc(C(F)F)cs3)=O)CC2)CNC(=O)C1 CCC(CO)CCNC(C1CC1CNC(c1ccc(Sc2ccccc2)nc1)=O)=O C12CN(C(=O)CCCN(C)C)CCN1C(=O)C(C)COC(=O)C2.COCSC C1(OCCNC(C(C)OCC2CC2)=O)CCN(C(c2cnc(O)o2)=O)C1 O=C(CC(F)(F)c1ncccc1Br)NC(c1cccc(F)c1)c1ccc(F)cc1 c1(N(C(=O)CCOC2CC2)C)cnc(CNC(C2(CCO)CCC2)=O)s1 O=C(CC(O)c1ccccc1)NC(C1(NC(=O)C(O)C2CCCC2)CC1)CF c1(C(=O)NCCN(C(=O)C(C)(O)C(C)C)CC)cc(Br)cc(Cl)c1C C=Cn1nncc1C(N1CCCC(CNC(=O)C(C2CCCCC2)O)C1)=O C1(C)(CNC(C(C)O)=O)CN(C(C2C=CCCC2)=O)C1 CCCC(C)CC(=O)N1CCN(C(=O)CCCSc2ccc(F)cc2)C(CO)C1 c1(CC(=O)NC(C2CN(C(c3cc(C)no3)=O)C2)C2CC2)cc(Br)ccc1F N1(C(=O)Cc2ccccc2)CCC2OCCN(C(c3cc(F)cnc3O)=O)C2C1 C(CC(=O)NCC1C2CN(C(=O)C=CCN(C)C3CC3)CC12)(C(C)C)OCC C=C1CCN(C(=O)C(CCC)N(C)C)C(C(=O)NCC2CN(C)CCO2)C1 C1(C(N(C(CC)CO)C)=O)CCCN(C(C2CC(=C3CCC3)C2)=O)CC1 c1(C(=O)OC)cnc(C(c2nnnn2C2CC2)NCc2[nH]nnc2C)cn1 N1(CC)C(=O)CCC1CC(=O)NCC1(O)CN(C(=O)CSCc2ccccc2)C1 C1(NC(=O)NCC(CC(=O)NC2(CCCCO)CC2)OC)CC2CCCC(C1)C2 S(=O)(=O)(c1cccs1)NC(=O)CC(CCOC)CNC(=O)C(F)=CCCF c1(C(N2CC(c3cn(-c4ccc(C)nc4)nn3)(C)C2)=O)sc2ncnn2c1C c1(OC)ccc(NC(=O)C(N2CCN(c3cc(Cl)nc(C)n3)C(C)C2)C)cc1F c1(SCC(=O)NC(CC)CN(C(=O)C(F)OC(F)(F)F)C)ccccc1C Cc1cc(=NCC2OCCc3ccccc32)[nH]cc1S(=O)(=O)N1CCCNC(=O)C1 N1(C(c2nocc2C)C(=O)NC(CC)C)CCN(C)C(C(=O)OC)C1 c1(NC(Cc2onc(C)n2)=O)cnc2c(c1)CN(Cc1cncc(O)c1)CC2 c1(C(=O)NCC(=O)NCC)cc(Oc2c(C)nn(C)c2C)nc(Cl)c1 N1(C(C)=O)CCc2ccccc2C1CC(=O)Nc1cc2ccsc2c(O)n1 c1(CC(=O)NCC2N(C(CC(=C)Br)=O)CCC2)cc(F)c(N)cc1F N1(C(c2c(OC(C)C)nccc2)=O)CCN(C(C2CC3CC2CO3)=O)CC(O)C1 N1(C(CC(CC)C)=O)CC2(CC2)CC1CC(=O)NC1CCN(C(C)C)C1 C(=O)(C(C)C1=CCCC1)N1CC2CN(C(c3[nH]cc(C(C)=O)c3)=O)C2C1 C(N=c1[nH]c(=NCCCc2nc[nH]n2)c2sccc2[nH]1)C1N(C)CCN(C)C1 N1(CC(=O)OC)CCC(NC(=O)CC(C)O)C(F)C1 c1(OC)ccc(Cl)c(C(N2CCCC(NC(C3(OC)CC(O)C3)=O)C2C)=O)c1N CCC(CC(=O)N1CC(F)CC1C(=O)N(C(C)CC(N)=O)C)C(C)(C)C N1(C(COCCOC)=O)CCC(NC(=O)CN(C)CCO)C(C(N)=O)C1 c1(C(N2C(CCC(N3CC(CCC)OCC3)=O)CC2)=O)ccc(C)c(C(=O)OC)c1 C1(C(N)=O)CCC(C(=O)NCC=CCNC(C2(C(F)(F)F)CC2(F)F)=O)O1 N1(C(c2c(CC)noc2)=O)CC2CC1CN(C(=O)COc1ccc(F)cc1F)C2 CC(=Cn1ccnn1)C(=O)Nc1cccc(NCc2nnccc2C#N)c1 C(=O)(C1CNC(=O)c2ccnn21)NCc1nc(O)cc(C(=O)OC)n1 C1(C)(C(=O)NCC(C(C)C)NC(C2(CC)COC2)=O)CC=CCC1 N1(C(=O)NC2C(CN(C3CC3)CC)CCC2)CCOC(c2ncno2)C1 c1(C(N2C(CNC(CC(=C)C)=O)C(CC)CC2)=O)ccc(=O)n(C)n1 C1(C(=O)NC(C#C)C)CC=CCN1C(=O)CCNC(N)=O c1(CC)c(C(=O)NCCOC2CN(C(=O)C(F)=CC3CC3)C2)cnn1C C1(O)(CNC(C(C)c2ccco2)=O)CCN(C(=O)Cn2ccnn2)C1 N1(C(C2(C=C)CCC2)=O)CC(NC(=O)C(C)OC)C(c2nccn2C)C1 C1(N)(C(=O)NC(c2cn(C)nn2)CC)CCCCC1 C1(C(=O)NC2CC(C)N(C)CC2)CN(C(C2CC(N(C)CC)C2)=O)CC12CCC2 Cc1c(C(=O)NCC2CC2CNC(c2cnncc2C)=O)cccc1Br N1(C(c2n(CC)nnc2)=O)CCCC2CN(C(=O)CC3CCOC3)CCC12 c1(CC)ccc(F)cc1NC(C1CCN(C(=O)CC=C(C)C)CC1F)=O C1(NC(COC2(C)CCCC2)=O)CCCCCC1C(=O)N(CC(F)F)CC(N)=O Cc1cc(C(=O)NCC2CN(C)CCN2C(=O)C(C)CC2CC2)cc(C(F)F)c1 CC1(C)CN(C(c2csnn2)=O)CC1NC(=O)C(c1ccccc1)n1cccn1 c1(C(=O)NCC2CC(NC(C3(C)C=CCC3)=O)C2)cnn2ncccc12 c1(C(=O)NC(C(C)C)(C)CNC(=O)C(C)N2CCC2)ccc(Cl)c(Cl)c1 C(=O)(CC(C)CCCC)NCC(CC=C)C(=O)NC(CO)C(N)=O O=C(CCC(CF)CF)NCC1CCN1C(=O)CCc1nc(O)n[nH]1 N1(C(C(CCC)C)=O)CCN(C(C2CCCCN2C(C)=O)=O)C(C)C1 c1(C(N2CCC(C(C)(C)C)(CNC(C(C#C)(C)C)=O)C2)=O)cc(C)nc(Cl)c1N C(CCC(O)C(=O)NC1CCC1(C)C)NC(c1n(CC)ncc1)=O c1(CNC2CCN(C(=O)OC(C)(C)C)CC2F)c(Cl)cc(Br)cc1Cl C(=O)(C1c2ccccc2OCC1(C)C)NC(CC)CNC(C1CC1CC(C)C)=O c1(C(=O)NC2CCN(C(C3C(C(=O)OC)C3)=O)CC2)cc2ccccc2cc1Cl CC1C(NC(=O)Cc2ccccn2)CCCN1C(c1cc(CF)on1)=O C12(C(=O)NCCCCNC(=O)CCC(F)(F)F)CCCCC1NC(=O)CC2 N1(C(CN(C(=O)OC)C)=O)CC=CCC1C(=O)NCC1CC(O)C1(C)C c1(C(=O)NC2CC(C)N(C(=O)CC3CS(=O)(=O)C3)C2)cnc(F)c(Cl)c1 C1(C(=O)OC)CN2CCCN1CC2.c1(SCC(=O)N2CCC2)nc(C)cc(C)n1 C(=O)(CCCCCCNC(C1CC(CC)(CC)C1)=O)N(C(CC)C)C C(c1cccc(Br)c1)=CC(=O)NCC#CCNC(CNC(C)=O)=O CCCCCCCCOCC(=O)N(CC(C)NC(c1nc(=N)cc[nH]1)=O)CC C(CCCCCNC(C1CC2CCC2C1)=O)N(C(=O)CNC(c1ccncc1)=O)C N1(C(C2(CSC)CCC2)=O)CCC(NC(=O)CSS(C)(=O)=O)C(C)C1 c1(OC)cc(OC)c2[nH]c(C(=O)NC3(C)CCN(C(=O)C(C)C(C)O)C3)cc2c1 C1(NC(CN(C(=O)Cn2ccnc2)C(C)C)=O)CCN(C)C(=O)C1 c1(C(C)OC)cc(C2CC2)no1.C1(=O)CCOCCCN(C)C(=O)CN1 N1(C(c2ncc(OC)nc2)=O)CC(NC(C2CCCC(=O)N2)=O)CCC1C Cc1c(Br)cccc1NNC(=O)c1cc(-c2cccnc2)nn1C c1(-c2c(OC)cccc2)cc(=NC(=O)Nc2ccc(C)c(F)n2)[nH]o1 S(=O)(=O)(c1ccc(=NCCC(=O)N(C)CCO)[nH]c1)NC1CC(C)(C)OC1(C)C N1(CC)CC(C(=O)NC(C)CCCNC(=O)Cc2cc(C)no2)NC1=O C1(C(N2CC(C3CCCO3)C2)=O)C2CC(O)C(C2)N1CCn1ccc(C(=O)O)n1 C(=O)(C(C)(C)CCCNC(=O)C=CC(F)F)NC1CCC(CCCC)C1 CC1CC(NC(=O)CC2(O)CCN(C)CC2)CCN1C(=O)C1=COCCO1 Cc1ccc(F)c2c1N(C(C1CC1c1ccc(F)nc1)=O)CCC2 CC1CN(C(=O)CC(C)C(F)(F)F)CC(C)N(C(=O)CCCN(C)C)C1 c1(C(=O)NCC(C)CNC(=O)CC2CCCCC2)noc2c1CC(F)(F)CC2 CC1(NC(C2(C(F)F)CCCO2)=O)CCN(C(=O)CSCc2ncc[nH]2)C1 c1(NC(C)=O)cccc(C(N2CCCC(CN(C)C(C3CCCSC3)=O)C2)=O)n1 c1(NC(C2C(C(=O)OC)C2)=O)cc(Br)c(CSC2CC2)cc1Sc1[nH]cnc1C C(CC(=O)N1CCCCC1CCCO)(C(F)F)NC(=O)COC1CC=CC1 C(CCCCC(=O)NC1CC(N2CCCC2)C1)N(C(Cc1ccn(CC)n1)=O)C Cc1ncnc(O)c1C(=O)NC1CCC1NC(=O)CCc1ccc(O)c(F)c1 c1(C(N2C3(CNC(C(C)(F)F)=O)CCC2CC3)=O)ccc2c(c1)NC(=O)C2(C)C n1(CC)nnc2cc(C(N3CCCC(NC(C4CC5(CC5)C4)=O)CC3)=O)ccc12 c1(OC)cnc(C(=O)NC2CC2NC(c2cccc(C)n2)=O)c(F)c1 c1(C(N2C(CNC(C3Cc4cccnc4C3)=O)CC2)=O)noc2ccc(F)cc12 c1(C(=O)NCCCCC2CN(C(c3cc(C)nnc3)=O)C2)cc(Cl)c(Cl)n1C Cc1c(Br)c(C(=O)N(CCCNC(=O)CC2(C)CC2F)C)nn1C c1(C(N(C2CCN(C(C3CCOCC3)=O)CC2)C(C)C)=O)cnn2ccsc12 C(=O)(C(CC)C(=O)NCC=CC(N1CCC(CCO)CC1)=O)OCC c1(C(N2C3(C(=O)OC)CC3CC2)C(=O)NCCCC2CC2)c(Cl)cccc1Cl N1(C(CC=CC)=O)CCN(C(=O)C(C)O)CC1C1CCC1 c1(OCC(=O)N(C(CCNC(COC(C)C)=O)C)C)cccc(Cl)c1Cl O(NC(=O)C1=C(F)CN(C(c2cn(C)ccc2=O)=O)CC1)C(C(C)C)CO c1(NCC(=O)NC(C)C(C)(C)NC(c2cccs2)=O)cc2ncn(C)c2cn1 N1(C(COCC)=O)CCN(C(=O)CN(C(=O)C(C)NC=O)C)CC1 CC1(CCO)CC(O)CN1C(=O)CCCNC(=O)COC1CC1 c1(C(=O)NCC23C(CN(C(c4ccc(CCC)[nH]4)=O)C2)C3)cn2c(n1)COCC2 CCCC(C(O)C(=O)N1CC(=O)NC(CC)C1)NC(c1nccc(C)c1F)=O CC(C)CC(C(=O)N1CC(C)OC(C)C1)N(C)C(c1c[nH]ccc1=O)=O n1(C(C)C)nncc1C(=O)NC(C)(C)C(C)NC(=O)CNC(c1ccccc1)=O N1(C(c2cnn(CC)c2Cl)=O)CC2(CC(NC(c3c[nH]cc3Br)=O)C2)C1 C1(C(=O)NCCCCC(C)C)(NC(c2c(CC)occ2)=O)CCCC1C c1(C(=O)NCC2N(C(c3c(O)ccc(C)n3)=O)CCC2)cnn2ccc(O)nc12 CCC(C)(C)CC(=O)NC1CN(C(C2(C)COC(C)CO2)=O)CC1F CC(CCCO)NC(=O)COC(=O)C(CC1CCCOC1)c1ccccc1 CCCC(O)CC(=O)N1CC(c2cn(CCCn3cccn3)nn2)C1 c1(C(CC)NC(=O)CC2(NC(=O)COC3CC=CC3)CC2)ccc(C)cc1 c1(C(=O)NCCCN(C(=O)CCC(C)(C)F)CCC)cccc2cncn12 CN1CCCCC1CCNC(=O)C(C)(C)CN(C(=O)CC1(C)CC1)C C(=O)(C(C)(C)C(=O)N1CCC(CNC(c2nocc2Br)=O)CC1)OCC c1(N(C(=O)CN2CCCC(O)C2)C2COC2)ccc(Cl)cc1Cl c1(C(N2CC(NC(c3nc(CCC)sc3)=O)(CO)C2)=O)cn(C)c(C(F)F)n1 CCC(C)C(C(=O)N1CC(O)CC1Cn1cc(COC)nn1)N(C)C N1(C(CCC2C(C)C2)=O)CCCCC(N(C)C(c2ccnn2CC(F)F)=O)C1 c1(C(=O)NC23CCN(C(C(F)=CC)=O)CC2C3)oc2ccc(Cl)cc2c1C N1(C(c2cc(C(N)=O)[nH]n2)=O)CCOCC(C(=O)NCC2CCCC2)C1 C(=O)(C1CCCn2nccc21)NCCOCCCN(C(=O)Cn1nnc(=N)[nH]1)C CC(C)C(C(=O)NC1CCN(C(=O)COCC(=O)OC(C)C)C1C)c1cnn(C)c1 c1(OC)cc(C)c(C(N2CCC(O)C(N(C)C(c3cc(C)n(C)c3)=O)C2)=O)cn1 c1(CN=C(NC(c2ccn(C)c2)C)NCC2CC2)cc(Cl)cc(Cl)c1F C(=O)(CS(=O)CC)NCC1CCC(NC(CCC=CCC=C)=O)C1 c1(OC(C)C)cccc(CC(N2CCCC2(C)C(=O)NCCc2cnc[nH]2)=O)c1 C1(CCC(=O)NC(CN(C(=O)CCOCCCCO)C)(C)C)CCC(=O)C1 n1(CC(=O)N(C(C)CCNC(c2nccc(Cl)c2F)=O)C)nnc2ccccc12 C#Cc1ccc(C(=O)NCC2CCC(CNC(C3(C)CCCC3C)=O)CC2)nc1 CC1(C)CCC(CC(N2CCCC(C)(CNC(C34CCC(C3)OC4)=O)C2)=O)OC1 N1(C(c2c(SCC)cccn2)=O)CC=C(CNC(c2sccc2Cl)=O)CC1 c1(CC(=O)NCC(CNC(C23OC(C)C(C2)C3)=O)(C)O)cnc2ccccc2c1 c1(C(=O)NCc2ncc(OC)nc2)ccc2c(n1)CN(C(=O)C=CC(C)C)CC2 Cc1nn(C)c(C)c1C(=O)C(=O)NC1CC1NC(C1(C)CCN(C)CC1)=O C1(OCC)CC2(C1)CC2C(=O)NC1CCCC1CNC(c1ccnc(OC)c1)=O c1(SCC)ccc(OC)c(C(N2CC=CC(NC(=O)C(C)C(O)CC)C2)=O)c1 c1(C(C)=O)cccc(C(=O)NC(C)CCNC(=O)CCN(c2cnccn2)C)c1 CONCC(O)C(=O)NCC(c1ccc(-c2nn[nH]n2)cc1)C Cc1cnn(C)c1CC(=O)NCCC1CN(C(C2OCC2(C)C)=O)CCO1 C(C(C)(C)C#CC(=O)NC1CCCC1(C)N(C)C)NC(C1COCC(C)O1)=O N1(C(c2ccc(CC)nc2)=O)CC2CCC1C(CNC(=O)CC(F)(F)F)C2 c1(C(C2CCC2)NC(c2ccsc2)C)nnnn1C1CC1 C1(C(=O)NC2(C)CN(C(C=C(CCN(C)C)Cl)=O)C2)COc2c(Br)cccc2C1 c1(NC(C(CC)c2ccccc2)=O)ccc(CC(N2CCC(CO)C2)=O)cn1 Cc1nn(C)cc1C(C)NC(=O)CCC1CCC(NC(=O)C(C)C(C)C)C1 c1(CC)ccc(C(=O)NCC2CC3CC3N2C(=O)C(C)NC(N)=O)c(OC)c1 c1(OC)ccc(C(N2CCCC(NC(C3CC(F)(CO)C3)=O)C2)=O)cc1 c1(C(N(C2CCN(C(c3ncc(F)cc3N)=O)C2)CC)=O)cc2c(s1)CCC2 c1(C(N(CCCNC(=O)C(C)OC(=O)C2CC2)CC)=O)cc(O)cc(C#N)c1 CCS(=O)(=O)c1ccc(CCC(=O)OCc2ncc(Cc3ccccc3)o2)cc1 N1(C(c2ccc(C)[nH]2)=O)CCC(NC(=O)C(c2cnn(C)c2)O)C(C)C1 c1(C(=O)NCC23C(CN(C(CC4CC(=C)C4)=O)C2)CC3)ccc(S(C)(=O)=O)cc1 c1(C(=O)NC(CNC(C2N(C(C)=O)CCC2)=O)C2CC2)sc(CO)nc1C O=C(C1CCCCc2ccccc21)NCC1CC(O)CN1C(c1ccc(Cl)o1)=O N1(C(c2cnc(CC)nc2O)=O)CCN(C(=O)C(O)C(C)(C)C)C(CC2CC2)C1 C(=O)(C1=CCc2ccccc21)N1CC(O)(CNC(C2CCC3CCC(=O)N23)=O)C1 C(=O)(C1CCc2c[nH]nc21)CCN1C(CC(=O)N(CCCCO)C)C(C)(C)CC1 c1(C(=O)NCC2(NC(=O)COCC3CCCO3)CCCC2)ccc2nc[nH]c2n1 C1(NC(C(C)O)=O)CCC2(CCN(C(=O)CNC(=O)C(C)(C)C)CC2)C1 N1(CCSCC(=O)OCCC)CCC(C2(C3CCCCC3)CC2)C1.C(C)=O c1(COC(C(C)OCC2CC2)=O)cc(Cc2ccco2)c2n[nH]cc2c1 Cc1cnc2n1CC(C(=O)NCCNC(=O)C1=C(Cl)CCCC1)CC2 C1(CC(=O)N(C)CC2CCCO2)CCCN(C(=O)CC#N)CC1 C1(Cc2nccc(C(=O)OCC)c2)CC2CN(C(c3nc(CC)no3)C)CC12 N1(C(C(C)CC(N)=O)=O)Cc2ccccc2C(NC(c2c(Cl)nsc2Cl)=O)C1 C(=O)(CCC(=O)NC1CC(NC(=O)CC2COCC(C)O2)C1)N(CC)CC c1(C(C(=O)NCCCC)N(C)Cc2cc(C)n(C)n2)ccc(F)cc1C C(CCSC)(C(=O)NCC(c1ccccc1)NC(C1(O)CCOC1)=O)OC C(=O)(C1CCCn2cnnc21)NCC1N(C(c2cc(C(N)=O)oc2)=O)CC=C1 CCCC(O)(CCC)CC(=O)NC1(CNC(=O)C(C)CC)CCC(C)(C)CC1 C(=O)(CN=c1[nH]c(=NCCNc2ccc(C(F)F)cc2)[nH]c2ccsc12)NCC Cc1nn(C)c2[nH]c(=NC(C)c3nnc4n3CC(C(=O)O)C4)ccc12 O=C(NNc1nccn2nccc12)c1ccccc1Cn1cccn1 CC(CC(=O)NCC1(O)CCCN(C(c2cncc(F)c2Cl)=O)CC1)C(C)(C)C C1(C2CC2)(CNC(CC(C=C)CC)=O)CCN(C(c2cccc3c2OCO3)=O)C1 c1(C(=O)NCC(CC)NC(=O)COCC(C)C)cncc2c(O)nccc12 c1(C(=O)NC2CCN(C(=O)CCC3CC3)C2)cc(Cl)cc(Cl)c1[N+](=O)[O-] C12(C(=O)NCC3N(C(C4CCN(C)C4)=O)CCC3)C3CC(CC13)C2(F)F C(C)(C)(CC(=O)N1CC(O)C(O)CO1)NC(c1n(CC)ncc1)=O n1(CC)c(N2CCCC(CS(N)(=O)=O)C2)nnc1-c1cc(C)no1 CCCCC(C(=O)N(C1CN(C)CC1O)C)NC(c1cc(F)c[nH]1)=O N1(C(c2c(C)nn[nH]2)=O)CC2(C=C(C(=O)N3CCC(F)C3)CO2)C1 N1(C(CCC(C)OC)=O)CC2CCN(C(=O)COc3nn(C)cc3[N+](=O)[O-])CC2C1 CC1=NOC(C)(CNC2CC(NC(C3CC(=C4CC4)C3)=O)CC2O)C1 n1(C(C)C)nccc1-c1cn(CC2CN(C(C3CCC(C)O3)=O)C2)nn1 C1(NC(C2CCN(C(=O)NC)CC2)=O)CC(O)CN(C(=O)Cn2cc(Cl)cn2)C1 CC1(C(=O)NCCNC(c2ncccc2N)=O)CCNC(=O)C1 C1(NC(C(C)Oc2cccnc2)=O)CC(O)CN(C(=O)CCCC#N)C1 C#CC1(C(N2CC(c3[nH]nnc3C)C2)=O)CCN(C(=O)C2=C(Cl)CCC2)C1 c1(OC)noc(C(=O)N(C2CC(NC(=O)C(c3cccnc3)C)C2)C)c1Br C1(C(N(CCCN(CC)CC)C)=O)CN(C(c2nc(O)sc2C)=O)CC1F C12(CNC(c3ccc(C)c(Br)c3)=O)CN(C(=O)Cc3ccon3)CC1CCO2 N1(C(c2c(C)cc(C)s2)=O)CCC2(CC1)CN(C(C13CCOC1CCOC3)=O)C2 C1(CNC(C2N(C(c3cc(C)[nH]n3)=O)CC(O)C2)=O)CCCCC1(C)C N1(CC)CCC(C(=O)NC(C)CNC(=O)CC2COC(C(F)(F)F)C2)C1 c1(C(N(CC(C)NC(C2(C)CC(F)(F)C2)=O)C)=O)cc(Cl)ccc1Br c1(NC(C(c2ccnn2C)NC(CCCSC)=O)=O)cnn2c1OCCC2 C12(C(C(=O)NC)N(CCC#N)CCN(C)C)CCC(CC1)C2.C(COC)S N1(C(C2C(C)(C)C2NC(=O)CCC2CCCC2)=O)CCCCC2(CCC2)C1 C(C)(C)(CC(F)C(=O)NC(C)CCN1CCCC1)NC(CNC(C(CC)C)=O)=O C(=O)(CC(O)CNC(=O)CCNC(C)=O)N(CC(F)F)CC O=C(C1CCCc2cncn21)NC1CN(C(c2cnc(-c3cccs3)s2)=O)C1 CC(C)(C)C(C#N)C(=O)N1CCC(OCC(=O)NCc2cc(Cl)ccn2)C1 C1(C(=O)NC(C2CN(C(C(C)OCCN(C)C)=O)C2)C)CCCOCC1 C1(C(=O)OCC2CC2)CCCN(C(c2ccccc2)=O)C1 C#CC1(NCC(=O)Nc2cc(C(F)(F)F)ccc2C)CCCOC1 CC1CC(C)C(C(N2CCC(=CCNC(c3ncc(Cl)n3C)=O)CC2)=O)O1 N1(C(C=CC(C)C)=O)Cc2nccn2CC(NC(=O)C(C)(C)F)C1 CC1OC2(CO)CC1(C(=O)N(CC(C)NC(c1ccc([N+](=O)[O-])o1)=O)C)C2 C12(CC(N3CCC3CNC(C34CCC(CC3)CC4)=O)=O)CCCCC1C2(F)F c1(C(N2CCCC(C(C)(O)CNC(C3(F)CC3)=O)C2)=O)ccc2ccncc2c1 C1(C(N2CCCC(NC(c3cncc(SC)c3)=O)C2)=O)CC12CCC(F)(F)CC2 C1(CCC=C)CCCN(CC2(CC=C)CN(C(=O)CN(C3CC3)CC)C2)C1 C#CCCCCCCC(=O)NCC(CC(C)C)C(=O)N1CC(C)OCCC1C Cc1ccc(C(N2CCC(NC(c3cnc(C)cc3Cl)=O)C2(C)C)=O)c(C)n1 C1(C(=O)NCCCOC=C)CCC(O)C1.C(=O)(C=CCCC)NCCS c1(C(=O)OC)ccc(OC)nc1NCCCOCCN(C(=O)CC(C)(F)F)C S(=O)(=O)(c1c(C)cccc1C)Oc1c(CC)cccc1 C#CCCCCCCC(=O)NCC=CCNC(C1CN(C)C(=O)N1)=O C(N=c1[nH]cnc2c1SCCC2)C1CC(NC(=O)C=CBr)C1 N1(C(C(C2CN(C(=O)CC3CCC(F)(F)C3)C2)OC)=O)CC2CCC1CC2 N1(C(Cc2c(C)cccn2)=O)CC2CCCCC2(CNC(C2CCSCC2)=O)C1 CC1C(NC(=O)C(C)OCc2ccccc2)CCCN1C(=O)C=CCO Cc1cc(C(=O)NC2CC2CNC(=O)C=Cc2cnn(C)c2C)cc(C)c1 Cc1cc(C)n2nc(C)c(C(=O)NCCCC(C)(C)NC(=O)C3CC3)c2n1 CCC(F)(F)C(=O)NC(C)CNC(=O)CCC1COC(C)(C)O1 C1(C(=O)NCCCCN(C(=O)CN(C2CCC2)C)CC)CCOCC1(C)C c1(C(C(=O)NC)N(C)CC)nc(C(c2ccccc2F)OC)c2n1CCCC2 C1(C(N(C(C)CCNC(c2cc(C#N)cn2C)=O)C)=O)CCCC(F)(F)CC1 c1(C(C(=O)Nc2cccc(OC)c2)N(C)C)cc(C)cc(C)n1 N1(C(CN(C)C2CC2)=O)CCCCC1C1(NC(c2cnc(S)n2C)=O)CC1 C1(C(C)C)C(C(=O)NCCC2CCCC23CC3)CCN1C(c1cc(C#N)c[nH]1)=O C(=O)(C(C(C)(C)C)n1ccnn1)NC1CC(CNC(CC(C)F)=O)C1 C(=O)(C1CCCn2nccc21)NC1(c2ccc(C)cc2C)CCCOC1 S(=O)(=O)(c1ccc(C#N)c(NCC(OC)OC)c1)NC(c1c(CCC)nns1)C N1(C(c2ccc(C#C)cc2F)=O)CC(C)CN(C(=O)COc2ccsn2)CC1C C(C(C(C)(C)C)NC(=O)C=Cc1sccc1C)NC(CCCN(C(C)=O)C)=O CCCCC(C)(F)C(=O)NCCC1CCN(C(=O)CCC(C)(F)F)C(C)C1 c1(OC)cc(CNCC(c2nnnn2C2CC2)C2CC2(C)C)ccn1 C1(NC(Cn2cc(CNC(C3(N(C)CC)CC3)=O)nn2)=O)CCCN(C(C)=O)C1 CCC(C)CCC(O)CC(=O)N(C(C)CCNC(c1sc(C)nc1C)=O)C Cc1oc(CO)cc1C(N1CC(CCNC(C2CCC(C(F)(F)F)CC2)=O)C1)=O c1(C(N(CCNC(C(C)CS(C)=O)=O)C2CC2)=O)cc(Cl)c(N)c(Cl)c1 c1(CC)cccc(C(=O)NCCN2CCN(C(=O)COc3cnn(C)c3)CC2)n1 C(C(C)C)(C(O)C(=O)N1CC(O)CC1(C)C(=O)NOCCN(C)C)OC C(c1ccc(OC)cc1C)=CC(=O)NCC1CC(NC(CNC(CC)=O)=O)CC1O CCCCCCC(=O)NCCCSC1CCC(OCC(=O)NC)C1 n1(CC(=O)NC2C(C)(COC)C2)cc(CN2CCCCC2)nn1.C1CC(=O)N1 c1(COCC(=O)NCCCNC(C2CCCOCC2)=O)ccc(Cl)cc1 c1(COCC)ccc(NC(=O)C(C)(C)NC(C)=O)cc1 C1(N(C(c2c(C)occ2)=O)CCF)CCCN(C(=O)CC2(N(C)C)CCCC2)C1 C12(C(=O)NC(C)CC3CN(C(c4ccc(C(N)=O)[nH]4)=O)C3)CC(C1)C(CO)O2 Cc1noc(C)c1C(C)CC(=O)OC1CCN(c2ncccn2)C1 N1(C(COCC(=C)C)=O)CC(CNC(=O)C(C(C)(C)C)OC)CC(C)C1 c1(NC(c2cc(OC)c(C)cc2)=O)n[nH]c2c1CN(Cc1ccnc(Br)c1F)C2 C(=O)(C1CCCc2nccn21)N1CCC2(CN(C(C3C(C)C3)=O)C2)C1 Cc1cc(C2(NC3(c4nnnn4CCC4CC4)CCC(C)SC3)CC2)ccc1F Cc1ccc(C#N)cc1S(=O)(=O)N1CC(F)CC1C(=O)NCc1ncn(C)n1 N1(C(C(c2cccnc2)OC)=O)CC2CCC1C(NC(C1CCCC(O)C1)=O)C2 Cc1c(C(=O)Nc2cc(F)ccc2Br)oc2c(Br)cccc12 c1(C(=O)OC)c[nH]c(C(N2CC(NC(c3cc(C(N)=O)c[nH]3)=O)C2)=O)c1 c1(C(N2CCCC(N(C)C(c3cscc3Cl)=O)C2)=O)cnc(O)c(F)c1 c1(CN2CC(NC(C(CC)(C)C)=O)C(F)C2)ccc(Br)c(OC)n1 c1(OC)ccc(CN2CCC(C(C)C(=O)Nc3ncc(O)cc3C)CC2)cc1F c1(C(=O)NC2C(O)CCN(C(C(C)(C)c3ncco3)=O)C2)ccc2sncc2c1 C#CC1(O)CC(C(=O)NCC2CCCCN2S(C)(=O)=O)C1 CC(CC(=O)NCCCCC1(NC(=O)C=Cc2ccc[nH]2)CC1)C1CC1 C(c1ccc(F)cc1)=CC(N1CC(C(=O)Nc2cccc(CC)c2)OCC1)=O Cc1nn(-c2ccc(F)cc2)c2sc(C(=O)NC(c3ccc(O)c(F)c3)C)cc12 Cc1[nH][nH]c(=NC(=O)C2CCC2C(C)(C)C)c1C CC(C)CC(C)(O)C(=O)N1CC2(C(=O)N(C3CC3)Cc3nc[nH]n3)CC1CO2 Cc1cncc(C(N2CC(=C(F)CNC(=O)CC3COC(=O)N3)C2)=O)n1 N1(C(c2nocc2Br)=O)CCN(C(=O)C=Cc2cc[nH]c2)C(CC2CC2)C1 Cc1nc(C(N2CCC(CN3CCCC3)C2C)C(=O)NCCCF)c(Br)[nH]1 c1(C(NNC(=O)CC2(NS(=O)(=O)O)CCC2)=O)cccc2c3c([nH]c12)CCCC3 Cc1cc(C(=O)CNC(=O)C(F)(F)F)cc(C)c1.N12CCC(C)(CC1)NC(=O)C2 CC1CCN(C(=O)CCCC(N)=O)CC1NC(=O)CSc1ccc(F)cc1 C#Cc1cccc(C(N2CC3CC(NC(=O)C(C)(CC)CO)CC2C3)=O)c1Cl N1(C(c2c(OC)scc2)=O)CC23CCCC2(C1)CN(C(=O)CC(C)(C)C#N)C3 N1(C(C(C)OCC)=O)CCN(C(=O)Cc2c(C)cccc2F)C(CO)C1 O=C(CC(C(F)F)c1ccccc1)NCC1CN(C(=O)CC2COCCO2)C1 c1(CC(=O)N(C)CC2CN(C(c3ccn(C)n3)=O)CCO2)c(F)cccc1Cl C1C(C)(C)C(=O)N1C(C)C.C1(O)(CNC(CCOC(C)C)=O)CCN(C)C1 Cc1cccc(-c2nccn2C(c2csc(N3CCCC3=O)n2)C)c1F C1(CNC(c2cc(Br)co2)=O)C2CCC(C2)N1C(C1CCS(=O)(=O)N1)=O C1(CNC(=O)CCc2ccncn2)CN(C(C2CC(F)C2)=O)CC1C(F)(F)F N1(C(C2C(C)(C)CC2)=O)CCCN(CCNC(c2cc(Cl)c(Cl)s2)=O)CC1 c1(C(=O)NCC2(C)CN(C(c3cccc(O)c3)=O)C2)c(F)cc(Cl)cc1I c1(C(=O)NCC(C)N(C(c2ccc(SC)o2)=O)CC)c(C(F)F)nn(C)c1C Cc1cc(C(=O)NC(C)(CNC(=O)C(c2c(C)noc2C)(C)C)CO)nc(C)n1 c1(C(c2n(CCOCC)nnn2)NCCc2ccccn2)c(Br)cnc(Cl)c1F CCC(C)(C)C(C)CC(=O)N1CCC(N(CCO)C(c2cncc(Cl)c2Cl)=O)C1 C1(CC(=O)NC(CC)CNC(c2cc(C)c[nH]2)=O)(C(F)(F)F)CCC(=O)NC1 C1(NC(=O)CSCC(F)F)CC2CC1CC2C(=O)NCCSc1ccccc1 Cc1cccc(N(C)C(C2(CNC(=O)OC(C)(C)C)CC(F)(F)C2)=O)c1 C(C(CNC(c1ncoc1Br)=O)C(F)(F)F)NC(C(CC)=CC)=O C12(C(=O)NC3CN(C(c4ccc(-c5c[nH]nn5)cc4)=O)C3)CC=CCN1CCC2 CN1CCC(CCC(=O)NCC2(N(C)C)CCOCC2)CC1.C12(CCC1)C(=O)N2 N1(C(CC(C)OC)=O)CCCCC2(C1)CN(C(=O)C(C)Sc1ccccc1)C2 N1(C(c2cc(C)[nH]c2)=O)CC(CC(=O)NC(CO)CC(F)(F)F)CC1(C)C c1(NC2CC(O)C2)ccccc1C(=O)OC(c1n(CCCCOC)nnn1)C1CC1 N#Cc1ccc(C(=O)NCC2CC(NC(C3CCS(=O)(=O)N3)=O)C(O)C2)cc1F c1(O)cn(CCO)c(=O)nc1O.CC1CC(CSC)CCN1C(=O)OC(C)(C)C N1(C(C(C(COC)C)C)=O)CCCC2(C1)CN(C(c1ccc(F)c(O)c1)=O)C2 C1(NC(C=CC(=O)N(C)C)=O)CC2CN(C(c3ccc(C#N)o3)=O)CC12 C=C(C)CC(C(=O)NC1CN(C(=O)C(c2ccccc2C)O)CC1C)NC(C)=O c1(N)ccc2sccc2c1.N1(C(CN(CCC#N)CCO)=O)CCOC(COC)C1 C(=O)(C1Cc2ccccc21)N1CC(OC)(CNC(c2nnccc2C)=O)C1 Cc1nn(C)c(C(N2CCC(C(=O)Nc3cc(CO)ccc3Cl)C(O)C2)=O)c1F C=CCC(CC(C)C)C(=O)OC(C)C.c12cnn3cc(cnc13)C(=O)OC2 C1(CC=C)(C(=O)NCCC(C)F)CCN(C(C23CCC2C3)=O)C1 c1(C(N(C(CNC(C2C3(CC(OCC)C3)C2)=O)C)C)=O)ccc([N+](=O)[O-])cc1N CCCCCCCC(=O)NCCn1cc(CNC(=O)C(C)CN(C)C)nn1 CCC(F)(F)CC(=O)NCC1(CC(=O)Nc2cn(C)nc2C#N)CC1 C(=O)(CC(C)(C)CC(F)F)NC(CC(C)NC(=O)CSc1n[nH]c(O)n1)C CCCCC(C(=O)NC(c1cn(CCOC)nn1)C)N1CCCCC1 Cc1cnn(C)c1CC(N1CCC(NC(c2nn(CC(C)C)cc2Cl)=O)C1C)=O C1(CCCC)CCCN(C(=O)NCC2(Cc3ncc(C(F)F)s3)CCC2)C1 c1(CC)ccc(C(=O)NC(Cc2cc[nH]n2)C(=O)NCc2nnc(O)n2C)nc1 N1(C(C2(C)CC=CCC2)=O)CC2(CCCN(C(C34CC5CC3C4C5O)=O)C2)C1 C1(NC(c2nnn(C(C)(C)C)n2)=O)CC12CCN(C(=O)Cn1ccnc1)CC2 c1(C(=O)NC2CCN(C(CCCOC)=O)C2)ccc(C(F)F)nc1 C(=O)(C1=CCCCC1)NC1CC(CNC(c2c(CC)cccn2)=O)C1(C)C C(=O)(CCC(C)(C)F)N1C(C)CC(CNC(CCc2ccc(SC)cc2)=O)C1 N1(C(C(C)(C)F)=O)CCC2C(C1)CN2C(C12CC(c3ccccc3)C1C2)=O Cc1nc2cc(C(=O)N(c3cc(Br)ncc3Cl)C3CC4CNC3C4)ccc2s1 N1(C(C2(OC)CCCOC2)=O)CCCC(O)(CC(=O)NCC=CCC2CCC2)C1 C1(C(N2C(CNC(C(C)C)=O)CC(C(F)(F)F)C2)=O)CCn2c(O)nnc2C1 N#Cc1ccc(NC(C2CN(C(=O)CCCCBr)CCC2(F)F)=O)c([N+](=O)[O-])c1 c1(CC(C)(C)OCC)cn(CC(F)CCNC(=O)C(C2CCCC2)OC)nn1 C1(CN(C(c2c(C)csc2)=O)C)CN(C(=O)CCc2ccnn2C)CCO1 O=[N+]([O-])c1ccc(C(c2nnnn2-c2ccccc2)NCCc2cn[nH]c2)cc1 c1cc2c(cc1NC(=O)NC)OCCO2.N1(CC)Cc2cccc(O)c2C1 c1(C(=O)NCC2N(C(C3C(OCC)C3)=O)CCC2C)ccnc2ccc(O)cc12 C1(C(N(CCNC(c2csc(C)c2N)=O)C2CC2)=O)CC2CCC(C1)S2(=O)=O c1(NC(c2c(CNC(=O)CCn3cncn3)nccc2)=O)c(O)cccc1F C(=O)(C(C)S(N)(=O)=O)NCC1CN(C(c2oc(CC)c(C)c2)=O)CC1O CC1(C)CN(C(=O)C2=CCSC2)CC1NC(=O)CCCc1ncco1 N1(C(c2cc(C)c(C)o2)=O)CC(C)(C)CC1CNC(c1cccnc1Cl)=O C1(CC)CCC(C)N(C(C2CC(c3cccc(Cl)c3)C2)=O)C1 CCCC(C#N)C(=O)NC(CC1CC1)CC(=O)NCc1ccc(C)s1 C1(CNC(c2c(C)noc2C)=O)CCN(C(c2coc(O)n2)=O)CC1C c1(C(C)(C)O)cc(C(=O)NCC(O)CNC(C2CC2(F)F)=O)ccn1 Cc1nccc(N2CCCC(NC(=O)C(O)(C3CCC3)C3CC3)C2)n1 C1(NC(c2nc(C)sc2)=O)COCCN(C(=O)CSC(C)(C)C)C1 CCCN(OC)C(=O)CC(C(C)OC)NC(=O)CC1CCCSC1 C1(NC(C2N(CC)CC2)=O)CN(C(c2cc(N3CCCCC3)ccn2)=O)CC1F C1(O)(C(C)NC(c2c(C)nc(C)[nH]2)=O)CCN(C(C23CCCC2C3)=O)CC1 N1(CC)CCC(C(=O)NCC2CC(C)N(C(=O)C(N3CCC(C)CC3)=O)C2)CC1 N1(C(CC2CC(NC(CCSCC)=O)C2)=O)CCCC(CC(C)C)C1 c1(OC)ncc(C(=O)N(CC(C)N(C)C(c2csc(C)c2C)=O)C)cn1 CC(C)C(F)(F)CC(=O)N(C)CCNC(c1cc(C#N)ccc1Br)=O c1(SC)cc(C(=O)NC2CN(C(=O)CC(C)CF)CC2CC2CC2)nn1C c1(OC)ccc(C)cc1C(=O)NCC=CCC(=O)N(CCC(C)C)C c1(C(N2CCC(O)(CCNC(c3cc(F)cnc3Cl)=O)C2)=O)ccc(Cl)c(F)c1 C1(F)(C(=O)NCC(C)NC(c2cc3n(n2)CCC3)=O)CCS(=O)(=O)C1 C1(CNC(c2cc(OC)no2)=O)CCCC2(CN(C3CCCc4ccccc43)C2)O1 c1(C(=O)NC(CNC(c2c(C)n(C)cn2)=O)C)cc2c(s1)CCC(C)C2 c1(CCCNC(CCCCC)c2nnnn2CC)c(F)cccc1F S(=O)(=O)(c1ccc(N(C)CC2(C)CCCO2)c(F)c1)NCc1c(C)cn(C)n1 Cn1ccc(CC(N2CCC(n3cc(-c4cncn4C)nn3)C2)=O)n1 N1(C(C(COC(C)=O)(F)F)=O)CC(C(=O)NC23CC(C)(C2)C3)CC(C)C1 C(=O)(C(C)CC(C)C(C)=O)N(CCC(=O)NC(CC)CC(=O)OC)CCO c1(C(=O)NCC2N(C(c3c(OC)nccc3)=O)CCCC2)ccc2ccncc2c1 N1(C(C2NC(=O)C(F)C2)=O)CCC(C(F)(F)F)CC1CNC(=O)CC1CSCCO1 O=C1OCc2nc(C(=O)NCC3(CO)CCS(=O)(=O)CC3)c(Cl)cc21 c1(C(=O)NCCCCOC)ncc(C(C)(C)C)cc1N N1(c2[nH]c(N3CCC(O)C3)nc(=NC)n2)CCCC2(CC(=O)N(C)C2)C1 c1(OC)cnc(C(=O)NCC(CC(C)C)NC(c2c[nH]c(Br)c2)=O)nc1 n1(CC(=O)NCC2(CNC(CSC(C)C)=O)CC2(F)F)cc2ncccc2n1 C(=O)(C(CC)CCOC)N1CC(O)(C(C(N2CC(C#C)C2)=O)F)C1 Nc1cccc(Cl)c1C(=O)NCC1(CNC(=O)CC2CCC3CC3C2)CC1 c1(OC)ccc2cc(C(C3CCCCC3)N3CCC3c3noc(C)n3)oc2c1 c1(OC)ncnc(NC(C23CC2CN(C(c2sc(C)nc2C)=O)C3)=O)c1OC c1(N2CCN(CCOC(C(C)(C)NC)=O)CC2)nc(C)ncc1C(=O)OC n1(N(C(=O)C(C)C2CCCN2)C(CS)Cc2ccco2)ccc(C)n1.CO CC1(C(=O)NCC=C(Cl)Cl)CC(O)CN1C(C1C=CC=CC=C1)=O CC(O)C(C(=O)N1CC(NC(=O)C(F)=CCN(C)C)C1)NC(=O)OC(C)(C)C c1(N2CCCC(NC(c3c(C)csc3)=O)CC2)ncnc2cc(Br)ccc12 C12C3CC1N(C3)C(=O)C(=O)c1ccc(cc1)OC2=O.C1(C(=O)OC)CCC1 C1(C(C)C)CCC(C(=O)NC2CCCC2NC(=O)CC2CCCN2C(C)C)CC1 C1(CC=C)C2CC1NC(=O)Cn1cc(nn1)CCCN2.C(C)(C)(C)SC(C)C O=[N+]([O-])C1CCCCCC(NCC2CCN(Cc3ccccc3)CC2(C)C)C1 c1(C(c2nnnn2-c2ccccc2Cl)NCC2CC(C)(C)OC2)ccc(F)c(F)c1 C(=O)(C1=CCCOC1)NC(C1CCN(C(Cc2c(CC)n[nH]c2CC)=O)C1)C N1(C(C)=O)CCC(C)C(CN(c2c[nH]nc2C2CC2)C(=O)C=Cc2ccncc2)C1 c1(CC)ccc(C(N2CCC(C(F)C(=O)NCCC(F)(F)Cl)C2)=O)o1 c1(C(=O)NC2CN(C(C(F)=CC)=O)C2)ncccc1OC(F)F N1(C(CC2CCCC(C)(C)O2)=O)CCN(C(C2CCCS2)=O)CC12CCC2 CC(C)C(O)CC(=O)NCC1CCCCC1C(=O)NC(C)CCc1cn[nH]c1 C(C(C(=O)N1C(C)COCC1C)C(C)(C)C)n1cc(-c2nc(C)c(C)s2)nn1 N1(C(CNC2CC2)=O)CCC(C)C1c1ccccc1.C1CS(=O)(=O)N1CC Cc1ccnc(C(=O)NCC2CN(C(c3csc(C(C)(C)C)c3)=O)C2)n1 c1(NCC(COC)C(F)(F)F)cnc(Cl)c(N(C)C)c1 C1(NC(=O)CSC(F)F)CCN(C(=O)CCc2ccc(F)cc2)CC1F c1(-c2nc(SCc3ccc(C)s3)n(CC(F)F)n2)ccc2ccccc2n1 CC(C)CC(C)C(=O)NCC(C)(CO)NC(=O)COCC(C)(C)C c1(C(N(CC(C)(C)NC)C)=O)c(Br)cnn1C.c1(C(=O)OC)ccc(C2CC2)cc1 C1(NC(c2[nH]n(C)c(=O)n2)=O)CN(C(c2csc(CC(F)(F)F)n2)=O)C(C)(C)C1 C1(CCOC)(C(=O)N(CC(C)NC(=O)C(C)C#N)C)CCCC1 CC1(C(N2CCCC(CNC(C3CCCC3)=O)C2)=O)CC=CCO1 C(CCC(=O)NCCCCCF)N(C)C(c1ccsc1Cl)=O C1(C(=O)NC2(CC)CCC2)CC2CN(C(c3cccc(=O)o3)=O)CC2C1 Cc1ccc(Cl)cc1C(=O)NCC1CCN1C(C1CC=CCC1)=O C=C(C)CC(C(=O)NC(CCC)CCCC)NC(=O)C1=NOCC1 N1(SC)CCN(C(=O)C(C)OCCN(C)C)C(C)C1.C1C(=O)NCCO1 c1(NC(CC)CNC(=O)CCCSC)cc(C)nc2c(C)cnn12 c1(C(=O)NC2CCC3(C(NC(C(COC)C)=O)C3)CC2)ccc2nc(S)[nH]c2c1 c1(C(N2CC(Cn3cc(-c4cn(CC)nc4)nn3)C2)=O)ccc(OC)cc1 N1(C(c2nc(-c3cccc(C)c3)oc2)C(=O)NC2CC2)CCC(C)(C)C1C N1(CCN(C(=O)Cn2cc(-c3ccc(N)cc3F)nn2)C)CC(=O)CCC1=O CC1C(C(=O)NCC(C2CCC2)NC(c2coc(C3CCCCC3)c2)=O)C1(F)F c1(CC(=O)NC2C3CN(C(CNC(=O)OC)=O)C2C3)c(C)nc2ncnn2c1C C1(C(=O)NCC(F)C2CCC2)(SC)CN(C(=O)CNC(C2CCCC2)=O)C1 C(=O)(C1=CS(=O)CCC1)NCC12C(CN(C(CCc3ccn(C)c3)=O)C1)CC2 C1(NC(C2CC23CC3)=O)CC2CCC1CN(C(=O)C=CCO)C2 c1(C(C(=O)N(CCN(C(c2c(CC)c[nH]n2)=O)C)C(C)C)C)cncc(F)c1 C(=O)(N=c1cc[nH]c2cc[nH]c12)C12CC(NC(c3c(OC)ccc(C)c3)=O)(C1)C2 CCC(CO)C(=O)NCC#N.c12ccc(cc1)OCC(=O)N1CC(C)(C1)O2 c1(NC(C2N(C(COCC=C)=O)CCC2)=O)cc(CO)ccc1OC c1(NC(C2CC(NC(=O)Cc3ccc(F)cc3F)C2)=O)cc2ccc(Br)cc2s1 c1(C(CNC(=O)CN2CCC(C)C2)NC(CC=C)=O)ccc(C2CC2)cc1 c1(C(N2CCCC(C(C)NC(C(CC)N(C)C)=O)C2)=O)noc2ccccc12 c1(OC)cccc(N2CC(C)(NC(=O)C(C3CCOCC3)C)C2)c1[N+](=O)[O-] N1(C(CCC(C)OC)=O)C(C(=O)NC2C(O)C3CCOC23)CC2CCCC12 C1(NC(C2OCCN(C(c3[nH]cc(C)c3)=O)C2)=O)CC2(CCOC2)C1 c1(C(=O)NCC2(O)CCCN(C(CCNC(N)=O)=O)C2)cc2n(c1)CCOC2 c1(C(C)(C)NC(=O)CNC(C2CCOC2=O)=O)ccc(-c2ccncc2)cc1 c1(C(N2CCN(C(COCc3ccc(C)cc3)=O)C(C)C2)=O)cc(O)c(F)cc1N CC1C(NC(=O)CCc2cnoc2)C(C)CCN1C(c1cc(C#N)on1)=O C1(C(=O)NCCN(C(=O)CC2(C)OCCO2)CCC)CCc2cc(C)ccc2O1 C(=O)(C1=CCC(C)(C)CC1)NCC1(OC)CCN(C(=O)CC2CC(F)(F)C2)C1 n1(CC#N)nc(-c2cccc(CC3(n4cccn4)CC3)c2)nc1Cc1ccco1 N1(C(c2cncc(NC)c2)=O)CC(NC(c2cc(Cl)cn2C)=O)CC(C)C1 c1(N(C(=O)C(c2cccs2)NC(=O)C=Cc2ccco2)CC)ccccc1F c1(C(N2C(CC(=O)NCCC(=C)C)COCC2)=O)cc(C)c(C)cn1 c1(C(=O)NC2CCN(c3ccc(C)cc3)CC2)ccc(OC)c2c1CCNC2 C(=O)(CC(F)(F)C(F)(F)F)N(C1C(NC(c2nc(C(C)C)oc2)=O)CCCC1)C Cc1cc(C(=O)NC2CN(C(=O)Cc3ccc(F)c(F)c3)CC23CC3)ncc1N c1(C(=O)OCc2c(CC)noc2)ncnc(C)c1C c1(OC)cccc(CNC(=O)C(c2ncsc2C)N2CCC(SC)C2)c1 N1(C(c2cncc(F)c2)=O)CC2(C1)CN(C(=O)C(c1cccc(Br)c1)O)C2 N1(C(CCC#C)=O)CCC(O)(CCNC(=O)C(C)(C)Nc2ccccn2)C1 C1(F)(CCC)CCN(CC(OCc2ccccc2)OC)C1 CCCC(CC)C(=O)N1CCCC1(CNC(=O)CSC(F)F)COC c1(C(=O)NCCC2CCCN2C(=O)CC2CCCOCC2)cncc2c1CCC2 CCCC(CCC)CC(=O)NCC1CN(C(=O)C(O)C(F)F)CC1SC Cc1ccc(C=CC(N2CCC(C(C)(C)NC(=O)CC3(O)CCC3)CC2)=O)o1 C(c1ccc([N+](=O)[O-])cc1)=CCNC(=O)NC12CC(C(F)(F)F)(C1)C2 CC1=C(C(=O)NCC2(F)CCCN(C(=O)C(N3CCOC3=O)C)C2)COCC1 N1(C(C(C)c2cncs2)=O)C2CCC1CC(CNC(=O)CCc1cc(Cl)no1)C2 C(CCCCC(=O)NC(Cc1cn(-c2ccc(F)cc2F)nn1)C(=O)O)SC O=C(C#CC1CCCC1)N1CCCC(CCC(N2CCC(CO)CC2)=O)C1 CN1CC(NC(C2CCN(C(c3ccc(=N)[nH]c3)=O)C2)=O)CC1CO c1(CN(C(CN(C(C2CC(OCC)C2)=O)C)=O)C)c(C)cnn1C C(CCC(=O)NCC(O)C1CCC1)(C(C)C)NC(c1cc(C)sc1N)=O Cc1ccc(N(C(=O)CC2CC2CNC(c2cc(O)cs2)=O)C)cc1C N1(CCC)CCN(C(=O)C(=O)NC(c2ccccc2)c2nc(C)cs2)CC1C N1(C(c2noc(CC)c2C)=O)CC2CCC(C1)N2C(C1CCCCN1N=O)=O C1(NC(c2c(C)nc(CC)o2)=O)CCN(C(=O)CN2CCCC2C(N)=O)CC1C C#Cc1cncc(C(N2C3CCCC2CC3)=O)c1 c1(C(=O)NCCC2C(C)CCCN2C(=O)CCCF)ccc2c(c1)COCC2 C(C)(CC(C)C#N)(c1n(CC=C)nnn1)NCCn1ccnc1 C(=O)(C(=O)NNc1nc2ccc(Cl)cc2s1)NCCC N1(C(C(C=C)O)=O)CCCC1(C)CNC(=O)Cc1cncc(C)c1 c1(OC)cc(C(=O)N(CCC(C)NC(c2ccccc2Br)=O)C)cc(F)c1 C1(C(=O)NCC2(F)CC(CNC(C=C(C)Cl)=O)C2)CC12CCCOC2 CC1CN(C(c2cn(CCO)nn2)=O)CC(C)CN1C(c1cc(F)cnc1O)=O CC(C)C(S)C(=O)N1C(C(=O)NCC2CCCCO2)CC2CC12 N1(C(c2cncc(C)c2)C(=O)NC2CCOCC2)CCC2(C)C(F)(F)C2(C)C1 C1(NC(c2cocn2)=O)CC(O)CN(C(=O)CCCOc2cc(F)ccc2F)C1 C1(CNC2C(C(C)(C)C)C2)CCCN(C(c2cc(Br)ccn2)=O)C1 C1(NC(=O)CSCC2CCCO2)CC(CNC(c2c[nH]c(Br)c2)=O)CC1O N1(C(C=C(C)C(F)F)=O)CCCC(CN(C(=O)C(C)CN2CCCC2)C)C1 N1(C(C2(C=C)CCN(C(=O)CCC3CCC3)CC2)=O)CCC2CN(C)CC2C1 N1(C(C(N)=O)=O)CC=CC(C(=O)NC(c2ccccc2)C(N)=O)C1 N1(C(c2nocc2Br)=O)CCCC12CCN(C(=O)C(F)(F)C1CC1)CC2 C1(C(=O)NC2CC(NC(CCCN(C(C)C)C)=O)C2)CCOC(C2CC2)C1 CC1=C(C(=O)NC2COCCN(C(C3COC4COCC34)=O)C2)CCO1 CC(C)(C)C(C(=O)N1CCN(C(C2(CCF)CC2)=O)CC1)NS(C)(=O)=O c1(CNC(CC(=O)NCC(CN(C(COCCOC)=O)C)O)=O)ccccc1 C(=O)(C1=NN2CCC(C)N=C2N1)NC1C(CNC(C2ON=C(C)C2)=O)CCCC1 C1(C#N)(C(=O)NC(C=CC(=O)NCC(c2ccncc2)C)C)CCCOC1 c1(C(=O)NCC#CCNC(CCCN(C)C)=O)ccc(N)c(C(F)(F)F)c1 c1(NC(=O)NCC2(C(=O)OCC)CCCO2)c(OC)ncn1C1CC1 C(c1cccc(F)c1)=CC(=O)NCC(C)CNC(c1ccc(SC(F)(F)F)o1)=O c1(N)cc(C)ccc1C.C1(c2n(CCSC)nnn2)(NCCC2CC2)CCCOC1 C(CC(CNC(c1sccc1F)=O)NC(c1ccsc1C)=O)OC N#Cc1cc(NC(C2CN3CCC2(F)CC3)=O)c(F)cc1F c1(C(N2CC(NC(C(C)CC3CC3)=O)C(C)C2)=O)cnn2cc(Br)cnc12 N1(C(C=CC=CCC)=O)CC(OCC(N2CC(C(C)C)C2)=O)C1 c1(CC)ccc(CNC(c2ccc(CNC(C3(C)CC3)=O)nc2)=O)nc1 N1(C(C2(CC#C)CCN(C(=O)CCCN=[N+]=[N-])C2)=O)CCc2ccccc2C1 C(CCNC(=O)CC1CC2CCC1O2)(C(=O)N1CC(O)(C(C)OC)C1)OC c1(OC)cnc(C(N2CCCC2CN(C)Cc2ccc[nH]2)=O)c(F)c1 N1(C(C=Cc2n(C)cnc2)=O)CCCCC(CNC(c2ccc(C(N)=O)s2)=O)C1 CC1CCOC(C(=O)N(C2CCCN(C(c3ccccc3C(F)(F)F)=O)C2)C)C1 C1(C(N2C(CNC(c3c(CC)cno3)=O)CCCC2)=O)CC(C)(C)OC1(C)C n1(CC)ncc(Cl)c1C(=O)NCC1CCN1C(=O)Cc1ccc(C)nc1 C(=O)(C1SCCc2sccc21)NC1CC(NC(c2cccn3c(O)nnc23)=O)C1 C1(NC(=O)C=Cc2ccoc2)CC(CNC(=O)C(C2CC2)C2CC2)C12CCC2 c1(N2C(CNC(C(C)SC)=O)CC3(CCC3)C2)nc2ccc(Cl)cc2s1 c1(CC)cc(=NC(=O)CNC(C23CCC(CO2)C3)=O)[nH][nH]1 c1(CC)[nH]nc(C(N2CCCC(CNC(c3csc(C(C)C)n3)=O)C2)=O)c1Cl CC#CCCC(=O)N(CCN(C)C(c1ccnn1-c1ccncc1)=O)C(C)C c1(NC(C2N(c3nccc(OCC)n3)CCC2)=O)cc(F)c(Br)cc1OCC C12(NC(C=CC(=O)NC3CCCO3)=O)CCCC1N(C(=O)C(O)C1CCC1)CC2 C1(CNC(CCSCC)=O)C2CN(C(c3cnn(C)c3Cl)=O)CC12 c1(C(C)C)nc(NC2CCN(C(C)C)C2)cc(=NCC2OCc3cc(Cl)ccc32)[nH]1 C1(CCN(C)C)(C(=O)NCC(O)CNC(=O)CCc2ccncn2)CCCC1 CC(C)CCCCC(=O)N(C1CCN(C(=O)C(C)C(C)n2cccn2)CC1)C C1(CCC(=O)NCC2CC2NC(=O)CCCc2ccc(Cl)cc2)CCC(O)CC1 C1(NC(C2CCN(C(=O)OC)C2)=O)CCN(C(=O)CSCC(C)C)CCO1 CCC(C)(C(=O)NC(C)CC1CN(C(c2ccncc2O)=O)C1)C(N)=O C12(C(N3CC(N(C(c4c(C(C)C)occ4)=O)C)C3)=O)CC3CC1C2C3O C1(C(=O)NC(C)Cc2cnccn2)CN(C(=O)CN=[N+]=[N-])CC1C1CC1 C1(C(=O)Nc2cccc(Cl)c2)COC2(CCN(C(=O)C(F)Cl)CC2)C1 c1(OC)cc(C(N2CCC(C)(C(=O)NC3CCC(C#N)CC3)C2)=O)cc(Br)c1O c1(NC(C)=O)nc(C(=O)NCC2CC23CCC3)cs1 C(=O)(C(C)(C)C(C)(C)O)NCCCCN(C)C(C1CNC(=O)C1)=O CC1(C(N2CC(F)(C(=O)NCCC3CC3)C2)=O)CC(=O)C1 C(=O)(N=c1cnn(CC(=O)OC)[nH]1)c1[nH]cc(CC)c1C C1(CCC)CN(C(=O)C(=O)N(C)CCC)CCO1.C(C(C)O)N c1(NC(=O)Nc2n(C)c3c(n2)cccc3Cl)cc2c(cc1[N+](=O)[O-])NCC2 c1(OC)ncc(Cl)cc1C(N1CCC(N(C)C(C2COC(C)C2)=O)CC1)=O C1(CNC(C(C)(N(C)C(C2CC=CC2)=O)C2CC2)=O)CC2CCC1C2 c1(NC(=O)NC(Cc2nn[nH]n2)CO)ccnc2c(Br)cccc12 C(=O)(CC(C(F)(F)F)NC(=O)C(C)(C)OCC)NC(C#C)C(C)OC C1(C(=O)NCC(CC)N(C)NC(=O)Cn2cnnn2)CCCC1CC c1(C(N2CC(N(C(=O)CC3CCNC3=O)C)C2)=O)ccc(C(C)(C)C)nc1 N1(c2nc(OC)c(C)cn2)CCCC2(CN(Cc3ccc(Br)cc3O)CCO2)C1 n1(CC)ncn(NC(=O)C2(F)CCN(C(=O)CCc3ccco3)CC2)c1=O c1(C(c2nnnn2C2CCCC2)NC(C2CCCO2)C(C)C)csc(Br)c1 c1(NC2CC(C(C)C)C2)cc2ccccc2cc1I N1(C(c2ccc(C)cc2)=O)CCN(C(c2cc(C(F)(F)F)ns2)=O)CC(O)C1 C=CC1CN(C(c2nccnc2CC)=O)CC1NC(c1cc(C(F)(F)F)c[nH]1)=O O=C(C1=COCCO1)NC1CCC(CC(N2CCCC3CC3C2)=O)C1 C1(C)(NC(C2CCCC(C(=O)OC)C2)=O)CCN(C(c2ccncc2O)=O)CC1 Cc1ccc(C(=O)NC2CC2NC(=O)COCC(c2ccccc2)C)o1 C(=O)(C1=CC(C)(C)C1)NC(C(=O)NCCOCCC#C)COC c1(CCC(=O)N(C(C)CC(N)=O)C)ccc2[nH]ccc2c1 C1(NC(CCNC(=O)C=CCl)=O)CC2CC(C1)N(C(C1CCCS1)=O)C2 CCC(C)(C)CC(=O)NC1CCOCC1NC(c1csc(CS(C)(=O)=O)n1)=O S(=O)(=O)(c1c(C)noc1C)N1CCC(C(C)C(N2CCC(Br)CC2)=O)CC1 c1(C(=O)NC2(C)CCN(C(c3ccnc(O)c3F)=O)C2)cc2scnc2[nH]1 c1(N2CC(C(=O)Nc3cc(C(N)=O)n[nH]3)OCC2)ncc2c(Cl)cccc2n1 C1(CC(=O)Nc2ncccn2)CCCN(C(=O)CC2CCCOC2)CC1 c1(N(C)C)ccc(C(=O)NC2COCC2CN2CCC(NC(=O)C3CC3)C2)cc1 CCCCC(CCCC)C(=O)NCC1(CNC(=O)CC2CC2(C)C)CCCCC1 c1(C(N(C2CCCN(C(c3csc(O)n3)=O)C2)C)=O)cc2cccn2c(O)n1 Cc1ncc(C=CC(=O)N(C2C3CN(C(=O)CC4(O)CCCOC4)CC23)C)s1 c1(C(C)=O)cc(Br)c(C(N2CC(CNC(c3ccncn3)=O)C2)=O)s1 N1(C(C2CC2Cl)=O)CCC(NC)CC1.Cc1ccsc1CC N1(C(C2(CC)CNC(=O)C2)=O)CC2CCCC(NC(C3CN(C(C)=O)C3)=O)C2C1 C1(OC(CC(=O)OCCN(C)C)=O)CCCC12CCCN(C(=O)OC(C)(C)C)C2 C1(NC(C2Cc3nccn3C2)=O)CCC2CN(C(=O)COc3ccon3)CC12 c1(C(C)=O)cccc(C(N2CC(NC(=O)C=C(C)C(F)F)CC23CC3)=O)c1C c1(CC)cc(NC(C2C=CC(NC(=O)Cc3ccsn3)C2)=O)ccc1C N1(C(C2CCC(CC)C2)=O)CC2(C)CN(C(=O)C(C)(C)CF)CC2(C)C1 CS(=O)c1ccccc1C(=O)Nc1ccc(N2CCCCC2=O)c(Cl)c1 C1(NC(C2CCC(O)CN2C(c2coc(C(F)F)c2)=O)=O)C2CCCC1COC2 c1(C(=O)NC2(COC)CC2(C)C)nc2ccccc2[nH]1 C(=O)(CCC1CCc2ccccc21)N1CC2CN(C(C3CC(=C)C3)=O)CC2(C)C1 c1(C(N(CCCNC(C(CC=CC)CC)=O)C2CC2)=O)ccc2c(C)noc2n1 N1(C(C2(C)CC2(F)Cl)=O)CCC(N(CCO)C(c2cc(C3CC3)ccn2)=O)CC1 c1(C(N2C(C(=O)NCCC3(C)CCCO3)CC(C)C2)=O)cccn2nccc12 c1(C(N(C2CCCN(C(C3N(CC)CC3)=O)C2)C)=O)cc2c([nH]1)CCCC2=O c1(OCCNC(C2C(c3c(C)cccc3)C2)=O)cccc2nccn12 C(=O)(CC(C)C(C)(C)NC(c1cccn1C)=O)N1CC(C(CC)C)C1 C1(C(=O)NCC2OCCN(C(C=Cc3ccn(C)c3)=O)C2)C2(CCC2)C12CCC2 C1(NCC2CN(C(=O)OC)C2)C2CC1CN(C(=O)C=CSc1ccccc1)C2 c1(OC)cc[n+]([O-])c(C(=O)NCC2CCCN2C(=O)CCNC(N)=O)c1 c1(C(N(CCC)CCNC(=O)CC2CC(CC)C2)=O)ccc(O)cc1 CCCC(C)(C)C(=O)N(C1CCCN(C(=O)C(C2CCC2)C2CCC2)C1)CC c1(SC)cc(C)c(-c2cn(C3CN(C(C4CC4c4ccnn4C)=O)C3)nn2)o1 N1(C(C2C(C)C2)=O)CC2COCC(C1)C2NC(c1ccc2cc(CN)oc2c1)=O C1(C(=O)NCCOCCN(C)C(C2C=CC=CC=C2)=O)CCCCN1S(N)(=O)=O C(=O)(C(O)CF)N(C1CCCCC1)CCNC(=O)Cn1cccn1 c1(C(=O)NCCCN(C(C2(OCC)CCC2)=O)CCO)ccc2cnccc2n1 c1(CC(=O)NC2CCCN(Cc3nccnc3Cl)C2)c(F)cccc1Cl C(=O)(C(F)(CNC(c1cnco1)=O)C(C)C)NC(c1c(C)noc1C)C CC1C(C(=O)NC(C)(CNC(=O)CC2CC(C)(C)C2)C(C)C)CCN1C N1(C(C2CCOC2)=O)CCC2CN(Cc3c(O)cc(F)cc3F)CC2CC1 N1(Cc2ncc(C)c(Br)c2)CC2(CCC(C(=O)Nc3cc(CCO)nn3C)O2)C1 Cn1cc(C(N)=O)c(=NC(=O)C2CCCC2C(=O)NCc2cccc(Cl)n2)[nH]1 Cc1ncc(Cl)c(C(N2CC3CC(NC(=O)Cc4ccnn4C)C2C3)=O)n1 c1(N(C(C)C)C(c2ccc(-c3cccc(C#N)c3)o2)=O)cc(Br)cc2[nH]ncc12 N1(OC(C=CC)=O)CCOC(C(N2CCCC2(C)C(C)(C)C)=O)C1 C1(CCOC)CN(C(C2(OC)CCOC2)=O)CCN1C(c1n[nH]cc1Cl)=O c1(C(N(C2CCN(C(C=CCOC)=O)C2)C)=O)cnc(O)n(C2CC2)c1=O c1(C(N2C(CNC(CCCC=C)=O)CCC2)=O)ccc(Br)c(N)c1 c1(C(=O)NCC(CC)NC(c2ccc(CC(N)=O)cc2)=O)cc(S(N)(=O)=O)co1 C(CNC(c1cn(C(C)C)cn1)=O)(C(=O)NC1(C(C)(F)F)CC1)N(C)C C#CC1(O)CC(C(=O)N(CCCn2cc(-c3c(C)noc3C)nn2)C2CC2)C1.CO C1(C(=O)NC2COCCN(C(c3c(CC)occ3)=O)C2)CCCCC(C)(C)C1 O(NC(=O)C(C)CCCC(C)=O)C(C(=O)NC1CCCN(CC)C1)CC(C)C c1(CC)ccc(C(=O)NC(C)CN(C(=O)CN2CCC(C)(C)C2)C)cc1[N+](=O)[O-] C1(C(=O)NC2CCC(C(=O)OCC)CC2)CC2(CCC2)C1OC C=CC(C)C(=O)NC1(C)CC(C(=O)NCC)C1.C12(CC1)C(=O)N2 N1(C(C2CCC(C(C)C)CC2)=O)CC2CCC1C2NC(=O)C(C)c1ccsc1 C1(F)(CNC(CCCCCO)=O)CC(CN(C(COC(CC)(C)C)=O)C)C1 c1(C(N2C(C(CNC(C(C)(CO)OC)=O)(C)C)CCC2)=O)cccc2c1NCC2 C(=O)(CCCCc1ccc(C)cc1)NC1CC(CCNC(CN(C(C)=O)C)=O)C1 CC1CCCC(C(=O)N(C)CC2COCCN2C(=O)C(C)C2CCC2)C1 c1(C(=O)NC(CNC(C(CC)(C)OC)=O)C)cc2sccc2cn1 N1(C(C=Cc2ccc(C#N)o2)=O)CC(NC(C2CC=CCO2)=O)CC2(CC2)C1 c1(C2N(C(CCn3cc(C(C)OC)nn3)=O)CCCC2)ccc2ncccc2c1 O=C(CCC(F)F)NC1CCN(C(c2cccn2Cc2cccnc2)=O)C1 N1(C(C=CCC)=O)CCOC(CNC(C2CC(F)C(=O)N2)=O)C1 C1(C2CCN(C(c3coc(SC)c3)=O)C2)(NC(C2(OC)CCCC2)=O)CC1 C(=O)(CCC(F)(F)F)NC1C(CNC(C2(C(=O)OCC)CCO2)=O)CCCC1 C(=O)(CC(P(C)(C)=O)P(C)(C)=O)N1CCC(O)(CS(=O)(=O)N(C)C)CC1 N1(C(CCN(C(c2c(NC)nccc2)=O)CCO)=O)CCC(C)C1(C)C N1(C(C(C)CO)=O)CCC2(CCN(C(c3cn(C)nc3O)=O)CC2)C(C)C1 CC(C)C(F)(CN(C(=O)C1CC1)C1CC1)C(=O)N1CCOC2CC12 c1(C(=O)NC2C(SC)CN(C(=O)Cc3ncc(F)cc3F)C2)cc(C)nc(C)c1 CCCCS(=O)(=O)NC1CCC(Nc2cc(OCC)ncn2)C1 Cc1cccc(F)c1C(=O)N(CCC(=O)NC1CCCC(C)C1)CCO C1(COOc2ccc(C(C)(C)CN3CCOCC3)cc2)CN2CCCCC2CO1 c1(C(=O)NC2CN(C(CC3(C)CC3(F)Cl)=O)C2)cc(Cl)ccc1F c1(C(C(=O)NCCSC)N(CCC(C)C)C)oc2ccc(F)cc2c1C c1(C(=O)NCC(C)N(C(=O)C#Cc2ccccc2)C)ccc([N+](=O)[O-])cc1F N1(C(c2c(C)nc(CC)s2)=O)CCC(CNC(C2(CCN(C)C)CC2)=O)C(C)C1 N1(C(C(C)NC(=O)Cc2ccon2)=O)CCCC(C)(C#N)C1 C=C(C)C1OCCCC1C(=O)NCC(C)(C)CNC(=O)C(C)=CC c1(C(=O)NC2CCN(C(c3c(C)ccnc3C)=O)C2)cc(F)cc2c1CCC2 C12CCCC13CN(C3)C(=O)C1(CC1)C(=O)N2.c1(OCC)cc(CCC)cnc1C C(=O)(C(CNC(=O)CC1CCCCO1)C(C)C)N(C(CCCC)C)C C1(NC(C(C)SC)=O)CCC(N2CCN(C(c3oc(C)nc3C)=O)CC2)CC1 C(=O)(C(C)(C)S(=O)(=O)C1CC1)NCCCN(c1c(Br)cnc(C(C)C)n1)C(C)C N1(C(C(C)C(C)(F)F)=O)CCC(NC(=O)C(=O)NCC2CC2)C2(CCC2)C1 Cc1nnc2ccc(C(N3CCOC(C(C)NC(=O)C(C)C(C)(F)F)C3)=O)cn12 Cc1cc(CN2CCCC(CCC(=O)NCc3cnoc3)C2)cnc1Cl c1(OC)ccc2c(c1)CC(C(=O)NC1CCN(C(c3cnco3)=O)C(C)C1)O2 c1(C(CC)O)nc(-c2ccc(C3CCCC3)nc2)n(Cc2cccc(Cl)c2)n1 CCC(CC)C(F)C(=O)N1CCC(C(=O)NC2(C)CCCC2(F)F)CC1(C)C N1(C(C(CC)c2ccccc2)=O)CCN(C)C(CNC(c2ccc(CO)cc2)=O)C1 C1(C)(C(=O)NC2CC(N(C(=O)CC3CCCO3)C)C2)CC2(C1)CC(F)(F)C2 c1(OC)ccnc(C(N2CC3CCC3(CCNC(=O)C(C)(C)C(F)F)C2)=O)c1C C(C(CC)(CC)C(=O)NCCc1scnc1C)NC(C(COCC)N=[N+]=[N-])=O C(=O)(CCCC(=O)N1CC(C)C1C(=O)NCCOCCN=[N+]=[N-])OC C(=O)(CCCCCCNC(C1CN(C)CC(C)O1)=O)NCc1scc(C)n1 c1(N2CCC(O)(C(C)NC(=O)COCP(C)(C)=O)C2)c([N+](=O)[O-])cnn1C c1(C(c2nnnn2-c2ccc(F)cc2)NCC(CO)OC)nc(Br)sc1C C1(C(=O)NCCOC2CN(C(c3cn(CCOC)nc3)=O)C2)CCCCC1C Cc1cnc(C(N2CCN(CC(C)NC(=O)CC3(O)CCOCC3)CC2)=O)cn1 N1(C(c2cc(C)c(Cl)s2)=O)CCC2(CCC2CNC(=O)CCc2cn[nH]c2)CC1 C=CCCC(CCC)(c1nnnn1CCOC)NCC1(CSC)CC(F)(F)C1 c1(C(=O)NCC(CNC(CC(CC)CC)=O)O)ccc(F)c(C)c1N c1(NC(C2N(C(=O)OC)C(C)C2)=O)ccc(C(=O)Nc2cncs2)cc1 N1(C(CCOC(C)C)=O)CC2CCC(CNC(=O)Cn3ccccc3=O)C2C1 c1(C(N2CC(CNC(C(C(C)C)O)=O)C3(C2)CC3)=O)cc2occ(Br)c2[nH]1 c1(NC(C2(C)CN(S(=O)(=O)C3CCCCC3)C2)=O)ccc2c(c1)OC(F)(F)O2 S(=O)(=O)(c1ccc(NCc2nnnn2-c2ccccc2)cc1Cl)NC(CC=C)C C(C)(C(C(=O)N1CC(C2CCCC3CC23)C1)C(C)C)NC(C1C(OCC)CC1)=O C1(O)(CN(C(=O)Cc2cn(C)cn2)C)CCN(C(C2CC2F)=O)C1 C12(C(N(CCNC(c3ccc(COC(C)=O)s3)=O)CC)=O)CCCC(=O)N1CCC2 C1(C)(OC)COC(COC(c2ccc3scnc3c2)=O)C1(C)C CC(C)C(CC(=O)N1CC2(CSC2)C1)NC(C1CCC(C)CC1)=O c1(OCCCC(=O)NC(CCNC(C(F)=CCC)=O)C(C)C)ccc(Cl)c(Cl)c1 C1(CC=C)(NC(=O)C(C)C(C)O)CCCN(C(=O)C(C)(C)F)C1 C1(CC(=O)N(C(c2ccccc2)CNC(c2csc(C3CC3)n2)=O)C)C=CCCC1 C(=O)(C1=CCc2ccccc21)N1CCN(C(C(C)C(N2CCCC2)=O)=O)CC(O)C1 CCC(O)C(C)C(=O)N(CCC(N1CCC(C)(CN(C)C)CC1)=O)C1CC1 N1(C(CCCCC)C(=O)Nc2ccc(F)cc2)CCC2(C(=O)OC)C(C1)C2(F)F c1(OC)cc(C)c(C(N2CCC(O)(C(=O)Nc3nccc(I)n3)C2)=O)c(C)c1 C(=O)(C1=CC2CCCCC12)N(CCOCCNC(Cc1c(C)ccnc1)=O)C C1(NC(c2cnc(C(C)O)s2)=O)CN(C(=O)Cc2ccn(C(C)C)n2)CCC1CO C1(CNC(c2scc(C)c2)=O)CC2(CC2)CN1C(=O)C(c1ccccc1C)C c1(C2C(C(=O)NC3CCC(NC(C4C5CCOCC45)=O)C3)C2)ccc(Cl)cc1 C1(O)(C(C2CCC2)NC(C2(C)CC(F)C2)=O)CCCCC1 CCCC(CC(=O)C(C(CCF)N)=O)N.C(=O)(CC(O)C(C)C)OCC Cc1cnncc1C(=O)N(C)CC1CCCN1C(=O)CNC(N)=O c1(C(=O)NC23CC(NC(CC4N(C)CCOC4)=O)(C2)C3)cc2ccccc2cc1Cl c1(OC)cc(CC(=O)OC)cc(N)c1C(C)C.c1(C(=O)CCC2CC2)cc(C(C)=O)c[nH]1 N1(C(C(c2ccc(C)cc2)F)=O)CC2CCN(C(c3cc(N)cc(O)c3)=O)C2C1 C(=O)(C(CCSC)OC)N(C1CCN(C(c2cccc(F)c2)=O)CC1)CC c1(NC(CC(CC=C)NC(=O)C(C)SCCCC)=O)cnc2ccnn2c1 c1(OC)ccn2cc(C(=O)N=c3cnn(C(C)C)[nH]3)nc2c1 C#CCCC(O)C(=O)N(CC(C)NC(=O)CCC(C)(C)c1ccccc1)CC C1(NC(C2C(C)C2)=O)CN(C(c2cc3[nH]ccc3s2)=O)CC2(CC2)C1 c1(C(N(CCNC(C(C)OCC2CC2)=O)C)=O)ccc2c(c1)CCN2C c1(CC(=O)NCC(C)CN(C)C(c2cn(C3CCOC3)cn2)=O)sc(O)nc1O N1(C(CC(C)N(CC=C)CCC)=O)CCCCC(NC(C)=O)C1 N1(C(C(C)=CC=C)=O)CCC2(CC2)CC1C(=O)NC(c1nc(C)no1)C C(=O)(C(O)(CO)C(F)(F)F)NC(c1csc(-n2cc(C3CCC=CO3)nn2)n1)C c1(NC(C2CC=CCC2C(N2C(C(=O)OC)CCC2)=O)=O)cc([N+](=O)[O-])ccc1F CCC(C)(C)CC(=O)N1CC2CC2(CNC(c2cncs2)=O)C1 C1(OC)CC(NC(c2cnn(-c3ccccc3)c2Cl)=O)C12CCOCC2 N1(C(C(c2ccn(C)c2)C)=O)CC(CC(=O)NC2CN(C)NC2=O)CC1(C)C C1(COC)(NC(=O)C(F)n2cccn2)CCN(C(=O)CCN2CCCC2)C1 c1(CN2CC(C(=O)Nc3ccc(F)c(Cl)c3F)SCC2)ccc2ncnn2c1 c1(C(=O)NCC(CC)NC(CC(CC)O)=O)cc(F)cc(Br)c1 c1(C(N(C2CCOC2)CC(=O)OC)=O)ccccc1N1CC(C(F)(F)F)OC1=O Nc1c(C(=O)NC(CC2CCCC2)CC2CCCC2)cc(Cl)nc1F Cc1cc(C)c(SCCNC(=O)C(N2CCCC23CCNC3)=O)c(C)c1 C1(C)(CNC(C(C)(C)OCCC)=O)CN(CC(Cl)=CCl)CCO1 c1(C(=O)NC2CN(C(C(C(=O)OC)C)=O)CC3C2C3)cc(C)nc2c1cnn2C CCC(C)C(O)CC(=O)N1CC(C(N2CC(C)S(=O)C(C)C2)=O)(SC)C1 N1(C(CCC(=O)NCCN(CCCC=C)C)=O)CCc2sccc2C1 C(=O)(C(C)(C)CC1CN(C(=O)NCCC2(N(C)C)CCC2)C1)OCC C(=O)(C(C)(F)C(C)(C)F)NC(CN(C(c1ccc(OCC)nc1)=O)C)CC C1(C)(C(=O)NC(CC)CCCO)CCCN(C(c2ccc(Cl)cc2)=O)C1 N1(C(C=CC)=O)CC(CNC(c2n[nH]cc2C)=O)CC(C)C1 C1(CNC(C2(SC)CC2)=O)C2CCC1CN(C(c1c(Cl)ccc(O)c1Cl)=O)C2 n1(CC)ncnc1C(=O)NCC1C=CCN1C(=O)CCc1cc(C)on1 N1(C(c2c(C)nc(CCCC)s2)=O)CCC(NC(=O)C(C)C(C)CC)C(C(N)=O)C1 c1(C(=O)NCC(CC)NC(=O)Cn2ncc(Br)n2)cnc2nccn2c1 Cc1c(C(N2CC(O)(CNC(=O)Cn3ccsc3=N)C2)=O)oc2c(C)cccc12 C(=O)(CCCC(C)(F)F)N1CCC(NC(c2c(CC)nc(C)[nH]2)=O)C1CC c1(CN(C)C)ccsc1C(=O)NC1CCCC1NC(=O)CNC(C1CCC1)=O C(F)(F)(C(F)(F)F)CC(=O)NC(C)CCNC(=O)C(C1CCCCC1)N(C)C C1(CN(C(c2n(COC)ncc2)=O)C)CCCN(C(c2cc(=O)cc[nH]2)=O)C1 C1(CN(C(=O)C(C)OCc2ccccc2)CC)COCCN1C(=O)C#CC1CC1 c1(NC(Cc2cc(C#N)cc(Br)c2)=O)ccc2c(n1)OCCO2 c1(C(N2C(C)CC(NC(=O)C=Cc3cn(C)nn3)C2)=O)ccc(F)c2c1OCC2 C(CCC(C)C(=O)NCC(C)CNC(c1cccc(C)c1N)=O)OC CCCS(=O)(=O)C(C)C(=O)N1CC(CO)(NC(c2nc(O)sc2C)=O)C1 N1(C(CCN(CCC)C)=O)CCN(C(C23CCN(CC2)C3)=O)CC1C C12(CN(C)C(c3ccccc3O)=O)CC(CO1)N(C(=O)C(C)(C)N1CCCC1)C2 Cc1cnc(S(C)(=O)=O)nc1NC1CC(C)CN(C(C23CCCN2CCC3)=O)C1 c1(C(N2CC3CN(C(C(CCC)O)=O)CC32)=O)ccn2cnnc2c1 C1(NC(C(C)=C2CCC2)=O)CCN(c2nccc(-n3nc(C)cc3C)n2)C12CC2 N1(c2cc(COC)nc(C)n2)CCCC(C2CC2NC(c2nc(O)sc2C)=O)C1 Cc1cc(N)cnc1C(=O)NC1CCC1NC(=O)C(c1ccc(Cl)cc1F)O C1(C(C(=O)NCC(=C)Br)(C)C)CCCN(C(C2CCC(C)O2)=O)C1 C(=O)(N=c1cccn[nH]1)c1c(N(C(c2ccc(Br)c(O)c2Br)=O)CCl)cncc1 C1(NC(C#CC(C)C)=O)COCCN(C(=O)C(F)C2CCC2)C1 c1(C(=O)OC(C)C(=O)NC2CCNC(=O)C2)ccc(C2CC2)nn1 C(C1CCCc2cccnc21)NC(=O)C(N1CCC12CC(O)C2)=O CC1(CNC(=O)CN(C(=O)CCC2CCC2)CC2CC2)CNC(=O)O1 C1(NC(c2coc(C(F)F)n2)=O)CCCCCC1Nc1ncnc(O)c1Br C#Cc1nc(C(N2CC(O)(C(C)NC(C3CC3(C)C)=O)C2)=O)cs1 C=CCCC(C)(C)C(=O)N1CCC(NC(C2CN(C3COC3)C2)=O)C(F)C1 c1(NCCc2n(C)cnc2)nc(NC2CSc3ccccc32)nc2c1ncn2C C(=O)(C(O)C(C)(C)C)NC1CC(NC(c2oc(C)c(CO)c2)=O)C1 c1(C(C)=O)cn(CC(=O)NC2(CC(=O)NCCN3CC=CCC3)CCC2)nn1 Cc1noc(C(=O)NCC2CCCN2C(C2CC2(C)Br)=O)c1C C(C)(C(=O)NCC(CNC(C1CCN(C)C1)=O)S(C)(=O)=O)(C(C)C)NC(C)=O C(=O)(CC1=CCCCC1)N1CCC(C(CO)NC(CC2(OC)CCC2)=O)CC1 N1(C(c2ccc(CC)cn2)=O)CCC(CNCC(O)CO)C(F)(F)C1 C1(CNC(COc2c(C)ccc(Cl)c2)=O)CC(C)(C)CN1C(=O)C(CO)N(C)C C12(CC(=O)NCc3c(C(N(C4=CC=CCCC4)CC)=O)c[nH]n3)CCC(CC1)C2 c1(CC)cccc2ccc(C(=O)NC3CC(C)(NC(=O)CC4CC=CC4)C3)nc12 c1(CC)sc(C(=O)NC2CN(C(C3C(C)(C)C3(F)F)=O)CC2OC)cc1C CC1CCCC1N(CCO)C(c1cn(C(C)C)cn1)=O.c1(C2CC2)ccco1 C1(NC(c2cccc(C#C)c2)=O)CN(C(C2CC(O)C2)=O)CCC12CCOCC2 N1(C(C2C(C)(C)COCC2)=O)CCN(C(=O)CC2NC(=O)NC2=O)CC2(CC2)C1 C(=O)(CCCCCNC(=O)CCn1cccc1)NCCC(CC)CO Cc1cccc2[nH]c(NC(C3CC3C(C)NC(=O)C3CC3)=O)cc12 c1(C(=O)NCC(NC(c2cc(CC3CC3)on2)=O)CF)cc2ncccc2s1 Cc1cc2ccc(C(N3CC4CCN(C(c5ccc(C)n5C)=O)CC34)=O)cn2c1 N1(CCC(N2CCC(C(C)NC(c3c(CC)cco3)=O)C2)=O)CCCS1(=O)=O C#CC1CCN(C(=O)C(C)NC(=O)C=C2CCC(C)CC2)CC1 Cc1nccc(C(N2CC(C)C2C(N2CC(N3CCCCC3)C2)=O)=O)c1N CN1CC=C(C(=O)NCC2CCOC2C(=O)Nc2cc(Cl)cnc2O)C1 C1(CCC(=O)N(C(CC)CNC(=O)Cc2ncc(C)[nH]2)C)CCC(=O)NC1 c1(OCC#C)ccc(C(=O)NC2(CO)CCN(C(C3(Cl)CC3(F)F)=O)C2)cc1 CC1(C)OCCC1C(=O)Nc1cccc(CNC(=O)C(F)Cc2ccccc2)c1 CCC(C)CC(C)C(=O)N1CCC(CCNC(CO)C(=O)OC)(C(=O)OC)CC1 c1(C(N2CC(C)C(O)C2)=O)ccc2c(-c3cccc(O)c3)c[nH]c2c1 CC1CCCn2ncc(C(=O)NC(CNC(=O)C=Cc3cscn3)C(C)(C)C)c21 CC1CCC(F)(C(N2CC(NC(=O)COc3cc(F)cc(Cl)c3)C(C)C2)=O)CC1 C1(CC(=O)N(CCOC)CCNC(=O)CCOC(C)(C)C)CCCCC1C C(=O)(CC1OCc2ncccc21)N1C(CNC(c2c(OC)c(Cl)ccc2)=O)CC1 CC1(C)CC(C(=O)NCCCC2CCC2)CN(C(=O)CC2CC3CCC3C2)C1 c1(CC)ccc(F)cc1F.c1(S)ccc(C(=O)N(C)CCN(C)C(C2CNC2)=O)cc1 C1(F)(C(N2CC3CN(C(Cc4ccc(C)c(C)c4)=O)C3C2)=O)CCCCC1(F)F c1(C(C(=O)NC2(C)CC2)N(CC)Cc2cccc(F)c2)cccn2ccnc12 CC1CN(c2cc(Cl)nc(C3(C)CC3)n2)CCC1NC(=O)C=Cc1cnn(C)c1 c1(C(=O)NCC2C(C(=O)NC3C(CN(C)C)COC3)CCC2)n[nH]cc1[N+](=O)[O-] CC(C)(C(=O)NCC1(F)CC(NC(C2OCC2(C)C)=O)C1)C(F)F N1(C(c2c(CC)scn2)=O)CCC(CNC(C2CC23CC(O)C3)=O)C1(C)C Cc1c(C(N2CC(C)(NC(C3CC4CCCN(C3)C4)=O)C2)=O)ccc2cncn12 c1(OC)cc(C(=O)NCC(C)(F)CNC(=O)OC(C)(C)C)cnc1Cl C(C(C(=O)NCCCN(C)C)N(C)CCOC1CCCCC1)(C1CCCC1)OC c1(C(C)(C)C(=O)NCCCCCCNC(=O)CC2(C)CC2F)cc(F)cc(Cl)c1 C1(=O)CCNC(=O)C(C)N1CC.C1(COC(C)=O)CC1C c1(C(N2CCC(CC=C)(NC(=O)CN=S(C)(C)=O)C2)=O)cc(O)c2ccsc2c1 C1(C(C)C)Cn2nccc2CN1C(C1CC2CCC1N(C(C1C=CCN1)=O)C2)=O N1(CC)CCCN(C(=O)Nc2cncc(C(F)F)c2)CC1 C(=O)(C(CC(C)C)N(C)C)N(CCOCCN(C(Cc1cc(C)sc1)=O)C)C CC1(CNC(C2CCCCO2)=O)CCCN(C(c2ccnn2C2CCC2)=O)C1 C(=O)(C1=CCc2ccccc21)NCc1nnc(C(=O)OCC)s1 c1(C(=O)NCCC2CC(NC(Cc3ccc(C)s3)=O)C2)ccc(O)cc1F C(=O)(CC(P(C)(C)=O)P(C)(C)=O)N(C)CC1(O)CN(C(C2C(C)OCCC2)=O)C1 C12(C(N3CCC4C(NC(C(C)=C(C)C)=O)C4C3)=O)CCC(N(C)C)(CC1)CC2 C1(CC(=O)N(C(CSC)C)C)COCCN1C(c1ccsc1C)=O n1(CC)nc(C(=O)NCC2(F)CCC(NC(=O)CC(C)O)C2)c(Br)n1 O=C1CCCC(CC(N2CCC=CC2C(=O)NCC(F)CO)=O)C1 C(=O)(CC(C)(C)CC(=O)NCC(CO)NC(C12CC1CN(C(C)=O)C2)=O)OC c1(NC(COc2c(C)cccc2)C)ccc(S(=O)(=O)NC(CO)C(C)C)c(Cl)c1 C1N=C2C=CN=C(N2)CN2CCCC12.c1(N2C(=O)NC(=O)C2)ccc(F)c(Cl)c1 N1(C(c2c(C)sc(Cl)n2)=O)CC(NC(=O)Cc2csc(Cl)n2)C(C)(C)C1 C1(C(N2CC(O)(CCNC(c3ccc(O)nn3)=O)C2)=O)C2CCCOC12 Cc1cccc2c(CC(=O)NC(C)CC(C)NC(=O)Cn3ccnc3C)c[nH]c12 c1(C(N2CCC(C)(NC(C3CCC(C)(O)CC3)=O)CC2)=O)ccc2nn[nH]c2c1 Cc1[nH]nc2cc(CNc3nnn(CC4CCCOC4)c3C)ccc12 C12CCCCC1OCC(=O)NCCCNC(=O)C2.C1(C(=O)N)CC(C(C)C)C1.CC C=CC1CN(C(=O)CCN(C(=O)CCn2cnc(=N)[nH]2)C2CC2)C1 C1(C)(C(N(C)Cc2c(C)occ2)=O)CCN(C(=O)CCOCC2CC2)CC1 c1(OC)ccnc(-c2cn(CCCC(=O)NC(c3cccc(C)c3)C)nn2)c1 C(C(C)(CNC(=O)CCNC=O)OC)NC(C(C)OCCCC)=O N#Cc1ccc(C(N2CC(NC(c3ccc(F)cc3O)=O)C2)=O)c(F)c1F N1(C(C2(C(F)F)CC(=C)C2)=O)CCC(CC)(NC(C2CCOC(=O)CC2)=O)CC1 C12CCCN1C(=O)C1CCC(C1)C2.C(C)(C)(C)OC(N(C1CC1)CC)=O c1(N2C(CNC(c3cccc(C(N)=O)c3)=O)CCCC2)nc2ncc(Cl)cc2s1 CC(CN(C)C)C(=O)N1CCCC1C1(O)CN(C(C2(C3CCCC3)CC2)=O)C1 C1(CSCC)(NC(CC2N(C(=O)OC)CCC2)=O)CCN(C(=O)CC=C(C)C)C1 C#Cc1ccc(Cl)c(C(=O)NCC2(F)CCC(NC(=O)CC(C)C(F)(F)F)C2)c1 N1(C(C(C)=CC)=O)CC(O)CC1CNC(=O)C(c1ccc(CC(C)C)cc1)C CC(CC(=O)NC1CCN(C(c2cc3cc[nH]c(=O)c3s2)=O)C1)CC(C)(C)C C1(N(C(C(CC)N(C(=O)CSC)C)=O)C(C)C)CCCCCC1 C1(NC(=O)Cc2ncc(Cl)s2)CCC2CN(C(c3cc[nH]n3)=O)CC2C1 C(=O)(C1=C(Cl)CCC1)N(C)CCC1CCN(C(=O)COC(C)(C)C)CC1 C12(COC)CN(C(=O)Cc3cc(C)no3)C(CNC(=O)C=CS(C)=O)(C1)C2 c1(C(=O)NC2CCC(C)N(C(c3ccncc3Cl)=O)C2)cc2n(n1)CCNC2=O C=C=C(C)CC(=O)N1CCCC(CNC(=O)CCCCc2ccccc2)C1 N1(C(Cc2ncc(C)[nH]2)=O)CC2CCC1C1CN(C(=O)COC3CCOC3)CC21 N1(C(C(=O)NCC(=C)C)C(C2CCCC2)OC)CCC2COCCC12 C1(CNC(c2c(OC)cc(F)cc2)=O)(CNC(=O)C(C)C)CC2CCCC2C1 C1(CCC)(C(N2CCC2COCCNC(=O)C(C)C2CCCO2)=O)CCNC1=O C(C)(C)(C#Cc1cn(-c2ccc(F)cc2F)nn1)NC(C(CC)C1CCOC1)=O N1(C(CNC(CCCCC)=O)=O)CCCC(NC(c2cnc(O)n2C)=O)CC1 c1(OCCNC(Cc2c(CC)cccc2)=O)cccc(OC)c1[N+](=O)[O-] N1(C(C=CCN(C(=O)C(C)(C)n2cnnn2)C)=O)CCn2nncc2C1 CC1=C(C(=O)N(CCNC(C2C=CCCC2)=O)C(C)C)CCCC1 C1(CC(=O)N(C(c2ccccc2)CNC(C(C=C)OC)=O)C)CCC2(CC2)CO1 N1(C(c2ccc(COC(CC)C)cc2)=O)CCN(C(=O)CS(N)(=O)=O)C(C)C1 C1(C2CN(C(=O)Cn3cnc(=N)[nH]3)C2)(OC)CC1.c12nc(co1)C(=O)NC2 C1(NC(C(C)NS(C)(=O)=O)=O)C2CC1N(C(=O)C(c1cccc(Cl)c1)(C)C)C2 C12CC(O)(C1)COC2=O.c1(C(=O)N)cncnc1.CN(CCO)C(C1CC1)C1CC1 c1(C(N2CCC(NC(C3CN(C(C)=O)C3)=O)C(O)C2)=O)cc(Br)cc(N)c1C c1(C(N2CC(NC(=O)CSC3CC3)C(CO)CC2)=O)cc2nc[nH]c2cn1 c1(CC)cc(C(=O)NCC2(NC(c3cnn(C)n3)=O)CCOC2)c(C)nn1 c1(NC(C2C3CN(c4ncc(F)cn4)CC23)=O)cc(F)cc2[nH]ccc12 C(=O)(C(CC(C)C)NC(C12CCC(C1)C2)=O)N(CC(CC)C(C)C)C CC1=C(F)CN(C(C2COCC2NC(c2ccccc2C)=O)=O)CC1 c1(C(=O)NC2(C(=O)NCC3(COC)CCC3)CCCC2C)cnc(C)c(C)c1 C(=O)(CCCC(C)CC)N1CCCC(C(C(=O)NC(C#C)(C)C)C)C1 C1(NC(c2cc(Cl)cs2)=O)CCN(C(c2cc(C(F)F)ncn2)=O)C12CC2 N1(C(C2(CC)COC2)=O)C2CCC1CN(C(c1ccc(SC)c(Br)c1)=O)C2 CCCCC(CC(=O)NCCCN1CCCCC1)NC(=O)CC1C=NN(C)C1=O N1(C(NOCC=C)=O)CC(O)CCC1NCCS(C)(=O)=O C1(CNC(=O)C(Cl)=CCl)CC2(C1)CN(C(c1cc(C3(O)COC3)on1)=O)C2 c1(NC(C2CC(F)(F)CN2Cc2cnc(Cl)s2)=O)nc(Br)ccc1O c1(C(N2CCCC(CNCC3(C)N(C(C)=O)CCC3)C2)=O)cnn2ccsc12 CC1CC=C(C(=O)N2CCN(C(=O)CSc3ccccn3)C(C)C2)CC1 c1(C(N2CC(O)(CN(C(CCC#CC)=O)C)C2)=O)nccc2occc12 CC1(C(=O)N(C2CC(NC(=O)COCCCN=[N+]=[N-])C2)CC2CC2)CCCC1 C(=O)(CC(C)C(=O)OC)N1CCC(C(=O)NCCOCC#C)(CO)C1 Cc1noc(N)c1CC(=O)NC1CCC(Cn2cc(-c3nccnc3C)nn2)C1 C(=O)(CCCC(C)(C)C)NC1CCCN(C(C(C(C)C)NS(C)(=O)=O)=O)CC1 c1(CC(=O)N(CC(C)NC(=O)C(C)NS(C)(=O)=O)C)ccsc1 C1(C(NOCCOCC)=O)CCCN(C(c2ncncc2OCC)=O)C1 C1(CNC(C2(C)CC2)=O)CCCN(C(C2CCOC2(C)C)=O)C1 C1(CNC(C23CC(C)(C2)C3)=O)CCC2CN(C(c3cccc(Cl)c3Cl)=O)CCC12 C1(C(N2CCN(Cc3ccc(CC)cc3)CC2)=O)CCNC(C2CCCO2)C1 CC1CC(N=c2[nH]nc(CO)s2)CCN1C(=O)CCn1cnccc1=O S(=O)(=O)(c1cccc(Cl)c1Cl)N1CC2CN(C(CCC(=O)OC)=O)C2C1 CC(=O)CC(C)(C)CC(=O)NC1CCCC2CN(C(=O)C(O)C3CCC3)CC12 CC1(C)CCCC(C(N2CCOC(CCNC(C3CCCC34CC4)=O)C2)=O)O1 N1(C(CC2(C=C)CC2)=O)CCC2(C1)CN(C(c1c(Cl)ccc(OC)c1N)=O)C2 CCC(c1ccc(C)cc1)=CC(N1CC(NC(=O)CS(=O)(=O)NC)CC(F)C1)=O c1(C(=O)NCC(CNC(CC)=O)NC(=O)CCOCC)ccnc(C2CCC2)c1 C1(CC(=O)Nc2cc(N(C)C)n[nH]2)CCCCN1C(=O)NC(c1ccccc1)=O CC1CCC=C1C(=O)NC1C2CC3C(C2)C13C(=O)NCc1nccc(O)n1 c1(CN2CCCC(CC(=O)N)(CO)C2)ccc([N+](=O)[O-])cc1Cl.C1(C(C2CC2)C)CC1 c1(C(N(C)C)=O)cc(-c2cnc(NCc3cncs3)c(O)c2)ccc1O C(=O)(C(CC(C)C)NC(C1CC(C)(C(N)=O)C1)=O)N1C(CSC)CCC1 c1(C(=O)NC2C(C(N3C(C)CC3(C)C)=O)COCC2)cccc2ccoc12 C1(NC(CCC2(C)N=N2)=O)CCCC1CNC(c1ccnn1C1CCC1)=O C(=O)(C1=NN2CCCN=C2N1)N1CC(CC)OCC1CC(=O)NOCCOC N#Cc1ccc(C(=O)NCCOCCCNC(C23CCCC2C3(F)F)=O)nc1 CC1ON=C(C(=O)N2CCC(N3CCN(C(c4ccsn4)=O)C3)CC2)C1C CN1CCC(C)(C(=O)NCCC2CCN(C(C3(C)CC3(F)F)=O)C2)CC1 C1(C(=O)NCc2ccc(C)cn2)C(C)OCCN1C(c1ncoc1C)=O C(CC(C)N(C)CC)(C(=O)NCSc1ccccc1)N1C(CC)C(C(=O)OC)CC1 c1(CCC(=O)N(C2CCN(C(=O)CCCCC3CC3)C2)C)n[nH]c2ccccc12 C(CCO)(C(F)(F)F)NC(=O)NCC(CC)Oc1ccccc1C n1(C(C)C)ncc(Cl)c1C(=O)NC1COCCC1NC(=O)C=CC1CCCN1C c1(NC(C2CCCN2Cc2sc(Cl)nc2Cl)=O)cccc2nc[nH]c12 Cc1[nH]c(C#N)cc1C(=O)NCC(C)CN(C)C(C1CC2CCCCC12)=O C=CCCCC(C(=O)NC(C)C(=O)OC)N1CC(C)C(C)C1C C1(C(=O)NCc2cccc(C#N)n2)CC2(CCC2)CN1C(c1cc(O)ncn1)=O Cc1nc(C)c(CC(=O)NCc2cnccn2)s1 C1(NC(CCC#N)=O)CCCC(NC(c2cccc(-n3cncn3)c2)=O)C1 C(=O)(CC(O)CNC(=O)C(C(C)C)N(C)C)N(CC#C)Cc1ccco1 Cc1nn(C)c(C)c1CCNC(=O)CNC(C)CCc1ccccn1 C(C)(C)(CCNC(=O)CC1(O)CC1)NC(CSCC)=O N1(C(c2c(C)nncc2)=O)CCc2nc(O)cc(C(=O)N(C3CC(C)C3)C)c2C1 C1(O)(CNC(CC(C(C)C)O)=O)CCCN(C(c2ncncc2Cl)=O)CC1 Cc1ccc(-n2ncc(C(N3CC(NC(C4(C)CSC4)=O)C3)=O)c2N)cc1 C1(NC(CC(=O)OCC)=O)CCCCCC1NC(c1[nH]nnc1CC)=O C1(C2CCCCC2)(NC(COC2CCN(C(CSC)=O)C2)=O)CC1 C(=O)(C(F)CC(C)(C)NC(c1cccnc1CC)=O)NCc1c(CC)nco1 N1(C(CCC=C(C)C)=O)CC(CNC(c2cc3c[nH]cnc-3n2)=O)OC(C)(C)C1 CC(F)(F)C(F)(F)CC(=O)NC1CCCCC1NC(C1CCCO1)=O C1(CC(=O)N(CC(C(=O)NC)C)C)CN(C(C2COCCO2)=O)CC1C c1(CC(C)(C)NC(N2CCC3(C=C3)CC2)=O)c(O)ccc(F)c1F N1(C(c2ccc(CC)c(N)c2)=O)C2CCC1CN(C(=O)CCc1cccnc1)C2 Cc1cc(Br)c(F)cc1C(=O)NC1CC(C(=O)Nc2cnc(Cl)cc2C#N)C1 C(=O)(C(C)CC(=O)N(C(C)CNC(=O)Cc1ccsn1)C)OC N1(C(C)=O)CCC(N(C(=O)C=CC(C)C)CC2CCCO2)C1 C(=O)(C(C(C)(C)O)NC(C1CCN(CC)C1)=O)NC1(C#C)CC1 CC1(C)CCN(C(=O)CN2CCCNC2=O)C1C(=O)NCCC1CC2CCC1O2 c1(NC(=O)NC2(CC)CCC2)cn(C2CCOCC2)nc1C C(=O)(CCCCC(=O)NCC1CC(NC(c2cc(C3CC3)nn2C)=O)C1)NC CC(C(=O)NCC(O)CN(C)C(c1cc(Cl)nn1C)=O)P(C)(C)=O C1(C(=O)NCCC2N(c3nnn(C)n3)CCSC2)CCOC2(CCCC2)C1 N1(C(C(C)=C2CC2)=O)CCC(NC(c2csc(-c3cccnc3)n2)=O)C(O)C1 N1(C(c2c(C)noc2C2CC2)=O)CCC(C2CC2)(CNC(=O)C(C)N(C)C)C1 N1(C(C2N(C(N)=O)CCCC2)=O)CC2CCC1C2NC(c1ccnc(Cl)c1N)=O C1(C(N2C(C(=O)O)CSC2)=O)CCn2c(cnc2C(F)(F)F)C1 c1(NC(=O)NC2C(CC=C)CCC2)cc(F)c(F)cc1C(F)(F)F C1(CC(=O)NC(C(C)C)CC2CC2)CC(NC(c2nccnc2N)=O)C1(C)C CC(N=c1[nH]c(N(C)CCO)nc2c1CCCCC2)N=c1ccc2ncccc2[nH]1 C=CCC(C)(C)CNC(=O)C=CC(C)NC(=O)C(C)SCC c1(CC(=O)NCC(CO)NC(=O)COC2CCCC2)cnc2nccn2c1 Cc1nn(C)c(Br)c1C(=O)NC1CC1NC(C1CC2C(C1)C2(F)F)=O C1(CC(=O)OC)CCCN1C(=O)CSCC(=O)NC1CN(C(C)=O)C1 CC1CCN(CC(=O)N(CC(C)(C)NC(c2coc(CN(C)C)c2)=O)C)C1 N1(C(CCc2onc(C)n2)=O)CCCC(CC(N2CCCC(C(C)C)C2)=O)CC1 CCCC(C)(CCC)C(=O)NC1CC(C)(NC(c2c(C)sc(C)c2Cl)=O)C1 C1(C(=O)NC(CCCC)(C)CO)CCN(C(=O)C(CC)C(C)O)O1 Cc1ccccc1C(N1CC(NC(C2(C)CNC(=O)N2)=O)CC1C)=O N1(C(COC(C)C)=O)CC(NC(c2ccccc2C(F)(F)F)=O)C(O)C1 c1(NC(N2CCC(CC3(CF)CC3)C2)=O)cc(OC(F)(F)F)ccc1Cl C1(OC)CC(NC(=O)C=C(C)C)C12CCN(C(c1cc(O)cc(C#N)c1)=O)CC2 c1(C(C)CC(=O)NC2(CC(F)(F)CCOC(=O)N(C)C)CC2)c[nH]c2ccccc12 C1(C)(CNC(CCCOC(C)C)=O)CCN(C(=O)CC2(C#N)CCC2)CC1 CCC(C)CC(=O)N(CC(C)N(C)C(c1ccc(Oc2ccccc2)nc1)=O)C N1(C(C(CN(CC)CC)F)=O)CCC(C)C(NC(=O)CC23CC(C2)C3)C1 C1(NC(C2(OCC)CC2)=O)CC(C(=O)NCCC2CCCC3CC23)=CC1O Cc1cccc(Br)c1C(C(=O)N1CC(C(C)C)C1)NC(=O)C(F)C1CCCC1 N1(CC2C(=O)NN=C2C)CCN(C)CC(C)C1.C=CC12CCN(C1)n1cc2nn1 c1(N2CC(C)(CC(=O)Nc3ncc(C4CC4)s3)C2)ncc2cc(Br)cnc2n1 c1(C(=O)NCCOCCNC(c2cnn(CC)n2)=O)cccc2c1OC(C)C2 Cc1ccc(C23CC(C(=O)NC(C)CCBr)(CO2)C3)cc1 N1(C(c2c(C)nccn2)=O)CCOC2(CCN(C(C3CCCC(C)CC3)=O)C2)C1 C#CC1CCN(C(c2ccc(CNC(=O)C=CCN3CCC3)nc2)=O)C1 Cc1cc(Br)ccc1NC(=O)NC(c1ccc(F)cn1)c1cscc1N(C)C C1(C(=O)NC2CC3CN(C(Cc4[nH]c(=N)sc4)=O)CC32)CCC2(CCC2)CC1 c1(C(N(CC(c2cccs2)O)C)=O)cc(S(N)(=O)=O)c(Cl)o1 CCCCC(C)CCC(=O)Nc1ccnc(C(=O)OC)c1.C12CC(C1)C(=O)N2 N12CCCC(C1)C2=O.C1(C(=O)NCCNC(=O)C(C)=O)(COC)COC1 C1(OC)CCN(Cc2cccc(F)c2Cl)C2(CC2)C1 N1(C(c2ncn(CC)n2)=O)CCC(CCNC(c2ccc(=N)[nH]c2)=O)CC1 CC1CN(C(=O)CC2COCC(C)O2)CC(C(=O)NC2C3CCC2CC3)O1 CN1CCN(C(c2ccc(Cl)nc2)=O)CC1CNC(=O)C(F)(F)C1CC1 C1(N(C(C=C(COC)C)=O)CC2CC2)CC2CC1N(C(=O)CN1CCCC1=O)C2 N(C(=NCc1cc(C)on1)N1CCC(C)(C2CCCO2)C1)Cc1nnn(CC)n1 C1(CNC(c2cc(C(=O)OC)no2)=O)CC2(C1)CN(C(C1(C)CC(C)=NO1)=O)C2 C1(C(N2CC(N(C(C3ON=C(C(C)C)C3)=O)C)C2)=O)CCc2c(cnn2C)C1 c1(C(N2CC(O)CC(NC(c3c(CC)ocn3)=O)C2)=O)ncn2ccccc12 Cc1ccc(F)c(C(N2CCC(NC(=O)CCC3CCCOC3)C(CO)C2)=O)n1 N1(C(CCC(=C)C)=O)CCC2C(NC(=O)CC(=O)NCc3nccs3)CC12 N1(C(CN(CCC)C)=O)CCC2C(CCCN2C(c2cc(N)cc(O)c2C)=O)C1 Cc1cc(C)n(-c2cc(NC(c3ccccn3)C)ncn2)n1 C(CC(C)(C)CC(=O)N1CCC(C2CCCN2C(c2cnn(C)n2)=O)C1)OC c1(C(C(=O)NC2CN(C(CC=CC)=O)CC(O)C2)=O)cc(F)c(F)cc1F c1(CC)ncc([N+](=O)[O-])cc1Cl.C12(F)CCN(C1)C(=O)C1CC(n3cc2nn3)C1 C(c1cnc[nH]1)=C(C)C(=O)N(CC(C)N(C(=O)CCc1nc(C2CC2)no1)C)C C1(OC)CC2(C1)CC(C(=O)NCC1CCCC1NC(c1cccc(F)c1C)=O)C2 CCCC(CNC(=O)CC1(NC(c2ccn(C)c2)=O)CCC1)CCO Cc1cc(C(=O)NC(CNC(=O)CC(O)C(C)C)CO)c(C)n1-c1ccccc1 N1(C(=O)C#CC2CCC2)CCC2(CCCCN(C(=O)C(O)Cn3cncn3)C2)C1 CCC(CCOC)C(=O)NCC1(C)CCCN(C(=O)CCF)C1 N1(C(CCCC2C(C)C2)=O)CC2CCCC(NC(C3(CO)COC3)=O)C2C1 Cc1sc2ncc(C(=O)NC3CN(C(=O)C(C)c4ccco4)CCC3C)n2c1C c1(C(N(CCOCCNC(CCSCC(C)C)=O)C)=O)cccc2c1SCCC2 Cn1cncc1C=CC(=O)NCc1ncccc1C(=O)NC(CO)C(=O)N(C)C c1(CNC(C(C)N(C(C=CC)=O)C2CC2)=O)cc(C(N)=O)co1 CCCC(O)CC(=O)NCC(C)(C)CC1CN(C(=O)C(C)(C)C(C)O)C1 C12(CCNC(CCC3CNC(=O)N3)=O)CCC(CC1)N(C(C1COC(=O)N1)=O)C2 N1(C(CN(CC)CC)=O)CCC2(CCCCN(C(=O)C(C3CC3)C3CC3)C2)C1 CC(C)C(CCNC(C1CC(=O)N(C(C)C)C1)=O)NC(c1c(Cl)cnn1C)=O C12(C(=O)NCC3CC(C(=O)OCC)C3)C3C(=O)C4C5CC(C14)C2C35.C(N)CC C1(C(=O)NCCOC2CCN(C(Cc3c(C)n[nH]c3)=O)C2)CN2CCN1CC2C N1(C(C(c2cccc(Cl)c2)OC)=O)CC2CC(NC(=O)CSC3CC3)C1C2 C12(CNC(CC(C)(C)O)=O)CCC1CCN2C(=O)C1=COCCO1 c1(C(N2CCCC(NC(C(C(C)O)(C)C)=O)C2)=O)cnc2c(ccn2C)c1 c1(C(N2CC(N(C)C(c3cnc(S)[nH]3)=O)C2)=O)cccnc1O C(c1ccc(C(F)F)o1)=CC(=O)NC(C)CNC(C1CC(C(F)(F)F)CO1)=O Cc1cc(C)c(C(=O)N(C2CCCN(C(=O)COCCF)CC2)C)cc1C N1(C(CCCC(=O)NCCC)=O)CCCN(C(=O)Cc2cnsc2)C(C)C1 N1(C(C(C)(C)OC)=O)CC2CC1CC2NC(C1CC(C)(C)CCO1)=O C1(C(N(CCCC)CCCO)=O)CC2CCCC2N1C(=O)CC1CC=CCN1C c1(C(N(CC)CC2CCCCN2C(=O)C=C(C)C)=O)ccc2cnccc2n1 C(=O)(C(=O)C(C)(C)C)NCC(C(=O)N(CC(C1CC1)OC)C)C N1(C(c2ccc(C(F)(F)F)o2)=O)CCN(C(=O)CCF)C(c2cccc(F)c2)C1 c1(NC(=O)Nc2ccc(C(C(C)C)=O)cc2)ccc2c(O)cccc2c1 c1(NC(c2n(C(C)C)c3c(n2)scc3)C)ccc(F)cc1C#N Cc1ccc(C(=O)N(CCC(=O)N(C2CCC2)C)C2CC2)cn1.C1C(=O)N1 CC1CCCC(C(C)NC(C2(C)CC=CC2)=O)C1 CC1(C)CC(NC(c2n[nH]c(O)n2)=O)CN(C(C2CC3CC3C2)=O)C1 N(C(=NCCc1ccc(Cl)nc1)N(C)Cc1ccc(Br)s1)CC(=C)C c1(C(C)=O)ccc(C(=O)NC2CCN(C(=O)CC3CC4(CCC4)C3)C2C)nc1 CC(C)CC(O)C(=O)NCC1(NC(c2coc(C3CCCC3)n2)=O)CCC1 C1(C(=O)OCc2c(CC)nco2)CCC(=O)N1C(=O)CC1CC1C n1(CC=C)nc(-c2cccnc2)nc1-c1ccc(C)s1 C1(C(=O)NC23CC(C(=O)NCc4cc(COC)[nH]n4)(C2)C3)C2CCC(C2)C1C C(C(C(C)C(C)C)NC(=O)C(F)(F)c1nccs1)NC(c1c(CC)noc1)=O N1(C(=O)OC(c2c(COC)ccs2)=O)CC(c2cn(C3CC(O)C3)nn2)C(O)C1 c1(CCC)c(C(=O)NC2CCCC(NC(=O)C(C3CCC3)OC)C2)nnn1CC c1(CN2CCCC(C(=O)Nc3ccc(C(F)(F)F)s3)C2)ccc(C(F)(F)F)cc1 Cc1ccc(C(=O)NCCC2(NC(C3C(C)C3C)=O)CCCC2)c(O)c1 c1(CC)cccc(C(=O)NC2CC(NC(=O)CN3CCC(C)CC3)C2)n1 c1(C(N(CCN(C(=O)CCCC2CC2)C(C)C)C)=O)cccc(Cl)c1N c1(C(=O)OCC)nonc1COC(=O)C(C)(C)c1cscn1 c1(-c2cn(C)nc2)ccccc1C(=O)NCC1CN(C(=O)C=C2CCC2)CC1O N1(C(c2c(NCC)cccn2)=O)CCC2CCN(C(=O)CCCCSC)C2C1 C1(CC2COC(=O)N2)COCCN1C(C(n1cc(CCC2CC2)nn1)C)=O C1(C2(C)CC2)CN(C(C2(CF)CC(=O)C2)=O)CC1NC(=O)Cn1nnnc1.CO C1(CCNC(C2ON=C(C)C2)=O)CSCCN1C(=O)C(n1cc(C)cn1)C N1(C(CCC#C)=O)CCN(C(=O)COc2ccc(F)cc2Cl)CC1COC C(=O)(NNc1cc(F)ccc1Br)c1c(Br)ccc(C#N)c1 N1(C(CCc2cc(C)[nH]n2)=O)CCC(CNC(C2CC(C)(C)C2)=O)C(F)(F)CC1 c1(C(=O)NCCN(CCC)C(C2CC(C)CO2)=O)ccsc1S(N)(=O)=O C1(NC(c2cc(C(C)=O)oc2)=O)CN(C(c2ccc(C)o2)=O)CC2(CC2)C1 CCCCN=C(NCC(N1CCOC(C)(C)C1)C(C)SC)NC1CCCCC1C Nc1cncc(C(=O)NCCNC(c2cn(-c3ccc(Cl)cc3)nn2)=O)c1 CC(CN=c1[nH]c(=NCC2CC3(CCC3)CO2)[nH]c2c1SCC2)N1CCOCC1 C1(N(C)C(c2cc(Cl)c[nH]2)=O)CCN(C(c2cc[nH]n2)=O)CC1 C(CCC(C)NC(=O)CC1CCCC1O)NC(COCC(C)C)=O C1(CC)CCN(C(=O)C2=CCCC2)C1CNC(C1CCN1CC)=O N1(C(CCc2cc(C)no2)=O)CC2CCC2(CCNC(=O)CCC(N)=O)C1 C1(C(=O)NC2(C)CN(C(=O)CCC3CCCO3)C2)CCC(C2CCCO2)O1 CC1CC(NC(C2CC3CC3C2)=O)CCN1C(c1cc(N)ccc1N)=O CC(CC(=O)N1CC2CN(C(=O)Cc3cnc4cccnn34)CC2C1)C(F)(F)F C12(C(=O)NCCC3CC(NC(c4cn(C5CCOC5)cn4)=O)C3)CCCCC1C2 CC1CC(NC(C2CCC(CCO)CC2)=O)CCN1C(=O)CCS(C)=O C(=O)(C(CC1CC1)NC(c1cncs1)=O)N(CCC)CCC c1(COCC(=O)NCC2CCC(NC(CCCCC)=O)C2)ccnc(OC)c1 C#Cc1cccc(C(N2CCCC(O)(CC)C2)C(=O)NC(C)C)c1 C12(NC(C(C(C)C)OC)=O)CCCC1N(C(=O)C=C(C)c1ccccc1)CCC2 CC1CC(NC(c2cn(C)nc2C(F)(F)F)=O)CN1C(c1nncn1C1CC1)=O CC1CCN(C(=O)CC2CS(=O)(=O)C2)C1CNC(C1OCCCO1)=O CCCC(CNC(C1CCCCN1C(=O)C(C)(C)C)=O)CCC C1(NC(CCC=C)=O)CN(C(c2sc([N+](=O)[O-])cc2Cl)=O)CC1C1CC1 C1(C(N2C(CNC(C3CCC(F)(F)CC3)=O)CCC2)=O)Cc2cc(F)ccc2O1 c1(C(=O)NCC(C(=O)N(CC(O)CO)CC)CC2CCCC2)ncccc1Cl C1(NC(=O)C=CC2CCC2)CN(C(=O)C(c2ccc(F)cc2)(F)F)CC12CC2 C(CC(=O)NCC(O)C1CCC1)(CC(C)C)NC(Cn1nnc(C)n1)=O c1(CCC(=O)N(c2ccc(O)cn2)CC(=O)OC)ccc(F)c(F)c1.C1(CCC)CN(C)C1 C1(C(=O)NCc2ccc(C(=O)NC(c3noc(C)n3)CC)cn2)CC2CCCC2C1 C=C(C)CCCC(=O)N1CC2CC1(C(=O)Nc1ccc(O)cc1)C2 C(c1ccccc1)=CCN(CC(=O)NCC(CC)NC(=O)C=CC1CC1)C c1(OCC)cc(C(=O)NC(C)CNC(=O)C(c2cccc(F)c2)(C)O)oc(=O)c1 C1(NC(C(COC)C)=O)COCCN(C(=O)Cn2cccc(C)c2=O)C1 N1(CC(=O)NCC(CC)N(C(=O)C=NOC)C)CCCCC1C C1(C(C)NC(CNC(CCOC)=O)=O)CCN(C(=O)C(C2CC2)OC)CC1 Cc1cc(C#N)ccc1S(=O)(=O)NC(C1CCN(C(=O)C(C)C)C1)C C1(N(C(CN(CCC)C)=O)C)CN(C(=O)C(c2ccc(F)cc2F)C)CC1(C)C Cc1ccnc(NCC2CCCCN2C(C2CC23CCOCC3)=O)c1[N+](=O)[O-] N1(C(CNC(CCC)=O)=O)CCOC2(C1)CN(C(=O)C#CC1CCCC1)C2 c1(N2C(CC)CNC(=O)C3CCN(C(=O)N2)C3)cc(F)c(F)c(Cl)c1F CC1C(C(=O)NC2COC(C(F)F)C2)CCCN1C(c1cccc(O)n1)=O N1(C(C(C)Cc2cnc[nH]2)=O)CC(NC(=O)C2=CCC2)CC(C)(C)C1 C12(CNC(c3n(C)ncc3)=O)CN(C(C3(S(N)(=O)=O)CCCC3)=O)CC1CCO2 C(N=C(NC1CC1)N1CCc2c(ccc3ccccc23)C1)C1CCS(=O)(=O)C1 S(=O)(=O)(c1ccc(C)c(Cl)c1)N1CCC(NC(c2c(F)cc(C)cc2Br)=O)C1 C=C1CCC(C(=O)NC(C)CCC(=O)N2CCCC(OC)C2)CC1 CCC(CC(C)C)C(=O)NC(CNC(C1(C(C)C)CC1)=O)CC(F)(F)F C1(C(=O)NCC(C)N(C(=O)C(C)(C)Cc2cnn[nH]2)CC)C2CC(F)(F)CC12 C(=O)(C1CCCc2ccccc21)NCC1CC(NC(C(C(C)O)N(C)C)=O)C1 c1(C(N2CC(CCC=C)(C(=O)NCC(F)Br)C2)=O)cncc(C)n1 N1(C(C(CCCC)F)=O)CCC(C(=O)Nc2cccc(C(C)=O)c2)C12CCC2 C(N=c1[nH]c(=NC(C)Cc2ccc(F)cc2)c2ncccc2[nH]1)c1c(C)c[nH]n1 C1(C(=O)NCC(C)CC2CC2)CN(C(=O)CN2C(=O)CCC2=O)C2(CCC2)C1 CC(C)CC(O)C(=O)NCC1C(C)CCCN1C(=O)CN1C(=O)CN(C)C1=O c1(C(=O)NC2CCC(N(C(=O)C=CC3CCC3)C)C2)cccc2c1NCC2 C(C)(N=c1[nH]nc(C#N)s1)c1nc(-c2occ(OC)c(=O)c2)on1 C(=O)(CC1CC(=O)c2ccccc21)NCCCN(C)C(C1(C)CCCC1)=O c1(CC)cc2cc(S(=O)(=O)NNC(=O)c3cnn(CSc4ccccc4)c3)sc2s1 c1(CN(CC(=O)N(C)C)Cc2cc(OC)[nH]n2)ccc(O)c(Cl)c1 O([Si](C)(C)C(C)(C)C)CC(C)NC1CC1CC1CC(OC)C1 c1(NC2CCC(N(C(=O)C3=CCSC3)C)CC2)cc(=O)n2ccccc2n1 C1(C(C(C)NC(=O)C(C)OC)NC(CNC(CCC)=O)=O)CCCCC1 C(=O)(C1=C(F)CN(C(=O)CC2CCCCC2O)CC1)NC1(C#C)CCCOC1 Cc1nc(C)c(CCC(=O)NCCC2CCCN(C(c3csc(O)n3)=O)C2)s1 N1(Cc2nc(CCOCC)on2)CC2(CC(NC(=O)Cc3cnoc3)CO2)C1 C#CCC(C(=O)NCCC(O)C(C)C)NC(C1CCOC1(C)C)=O C1(C(=O)NC2C(NC(c3cc(C)[nH]n3)=O)CCCC2)CC(C2CCCC2)C1 N1(C(C)=O)C2CCC1CC(CCNC(=O)CCCN1CCc3ccccc31)C2 c1(C(N(CC(O)CN(C)C(c2cn(C3CCC3)nn2)=O)C)=O)cnnc(O)c1 C1(NC(c2c(C)nco2)=O)CCCCC1NC(c1ccccn1)=O N1(C(N2CCS(=O)CC2)=O)CCCC2(CCCC2)C1 C1(CC(=O)NC(CCC)C2CC2)CCCC(NC(=O)C=Cc2ccncn2)C1 C1(CNC(CCSCCC)=O)CN(C(c2c(OC)cccc2C)=O)CCC1C c1(OC)cc(C)c(C(N2CCN(C(c3ccc(C(F)(F)F)cc3)=O)CC2)=O)cn1 c1(OC)c(C(N2CC(CNC(=O)C(F)(F)C3CCCC3)C(O)C2)=O)cnn1C c1(C(=O)NC2(C(=O)NOC3CCC3)CC(F)C2)c[nH]c2nccc-2c1 C1(C(=O)NC(CN(C)Cc2c(COC)noc2)C)COc2ccc(F)cc2C1 C(=O)(CCCC(CC)NC(c1cccn1CC)=O)NC1CN(CC)CC1C C(=O)(C(CCSC)N(C)C)NCCC(CNC(=O)C(O)CC1CCCC1)OC c1(COCC(c2ccccc2)C)cn(CCC(=O)NC2CC2C(F)F)nn1 C(=O)(C(C#N)CCC)N1CC(CCC=C)(C(=O)N(C)CC2CCCC3CC23)C1 C12CC1N=C1N=C(SN1)SC2.Cc1cnc(N(C)C)c(O)c1 CCC(CCC(=O)NCCC(O)CNC(=O)Cc1cccc(F)c1OC)OC C(=O)(CC1OCc2ccccc21)NCC1(C)N(C(=O)OC(C)(C)C)CCCCC1 N1(C(C2CCC(CNC(C3(C=C)CCC3)=O)O2)=O)CC=C(C)CC1 N1(S(CC#N)(=O)=O)CC2(CCN(C(C3CCN(c4cccc(F)c4)CC3)=O)C2)C1 c1(C(=O)NC2C(C(C)C)C2)occc1CNC(=O)COCCN(C)C.C1(C)CC1 c1(CCC(=O)NC2(CC=C)CN(C(c3cncc(NC)c3)=O)C2)cncc(C)c1 c1(CNCC2N(C(CCOC)=O)C3C(C2)C3)ccc2cc(O)ccc2c1 N1(C(C(C(=O)NC)(C)C)=O)CC2CCN(C(C3(CC4CC4)CCCO3)=O)CC2C1 Cc1cc(C#N)c[nH]c1=NC1CN(C(C2CC23CC(O)C3)=O)CC1C C#CCCN=C(NCCCSC)NCC1CSCC(OC)C1 CCCCCCCCOCC(=O)NCC1N(C(=O)C#CC(C)(C)C)CC1(C)C c1(CC(=O)NC(C(=O)N(CC#C)CC#C)C2CCC2)ncn(C)c1C C1(C(=O)NCC2CN(C(CCN(C(C)=O)C)=O)C2)COC2CCCCC12 S(=O)(=O)(CC(=O)NC(C)CCCCNC(=O)CC1NC(=O)NC1=O)NC N1(C(c2cccc(OCC)c2)=O)CC2(CNC(=O)C(O)C(C)OC)CC(F)(C1)C2 Cc1cccc2[nH]c(=NCC3C4CN(C(C5CC5(Cl)Cl)=O)CC34)sc12 N1(C(C2C(OC)CCC2)=O)CCC(O)C(C(N2CCC(CO)(OC)CC2)=O)C1 C1(CN(C(c2cc(-c3cccs3)on2)=O)CC)CCCN1C(C1CC1CF)=O C#CC1CCC(C(=O)N(C2CN(C(=O)CN3C(=O)CN(C)C3=O)C2)C)CC1 N1(C(CCCN(C(C)C)C)=O)CC2COCCC2(NC(C2CCC2)=O)C1 CCCC(C)(C)C(=O)NCC1CN(C(c2ccn(C3CCCCC3)n2)=O)C2CC12 C(=O)(C(C)N(OC)C(=O)c1sccc1CNC(=O)CC(C)(C)N(C)C)OC c1(CNC(=O)OC)cn(CC2C=CCN2C(c2ccn(COC)n2)=O)nn1 c1(OC)c(C(=O)N(C)CCNC(=O)C=Cc2nccs2)csc1C C#Cc1cc(NC(=O)C(c2ccccc2)NC(c2cscc2Cl)=O)cc(F)c1 N1(C(c2cc(C)c(Br)cc2)=O)CCC2(CC1)CC2C(=O)NCc1cccs1 N1(C(C23CCC(CC2F)C3)=O)CCC12CC(C(N1CCN(C3CC3)CC1)=O)C2 Cc1ccc2ccccc2c1C(N1CC(CNC(=O)CC2=NNC(=O)C2)C1)=O N1(C(C(OC)OC)=O)CCC2(CCCN2C(C2(C(=O)N(C)C)CC2)=O)CC1 c1(NC(C2C(CC)CCN2C(C2CC(=O)NC2(C)C)=O)=O)ccc(O)cc1C C(=O)(CCC(C)(F)F)NCC=CCNC(C(C)(COCc1ccccc1)OC)=O Cc1cc(C(=O)NCCCCCCNC(=O)C(O)Cc2cnc[nH]2)c(C)o1 N1(C(C(C(C)NC(=O)Cc2cn[nH]c2)(C)C)=O)CC(C2=NOCC2)C1 N1(C(C2CCC(CCC)CC2)=O)CCC(CC)(NC(=O)Cc2ccnn2C)CC1 c1(C(N(C)Cc2cn(C)nn2)=O)n[nH]c2c1CN(C(c1cc(Cl)ns1)=O)C2 c1(CC(N2C(C)CCC(NC(=O)CCF)C2)=O)ccc2c[nH]nc2c1 c1(N2C(CNC(=O)CCCC(F)(F)F)CCC(C)(C)C2)nc2c(F)cccc2o1 c1(OC)cc(CNC2CCC(C(=O)Nc3cc(F)ccc3Cl)C2)cc(Br)c1OC C(CCCC(C)(F)F)NC(C1(CC=C)CCCN1C(c1occc1COC)=O)=O C1(CC(=O)N(C2CN(C(c3cnc(CC4CC4)s3)=O)C2)C)CCCCC1O C1(N2CCCCC(C)C2)CCOC12CCN(C(=O)OCc1ccccc1)CC2 c1(C(N(C(C)CNC(c2cc(Br)n(C)c2)=O)C)=O)cnn2c1CN(C)CC2 C1(NCCC(C=C)C)CCC2(CC1)CNCCO2 Cc1cc(C(N2CC(NC(=O)COC3CCCC3)C(F)C2)=O)c(Br)cn1 O=C1C2CC3C1C3C2C(N1C(C(N2CC(O)(C(F)F)C2)=O)CCC1C1CC1)=O Cc1ccc(NC(C23CC(C(=O)N(c4ccccc4)C)(C2)C3)=O)nc1C N1(C(C(CC)C)=O)CCC(C2CCN(C(c3sc(S(N)(=O)=O)cc3C)=O)CC2)C1 c1(C(N(C(C)CNC(=O)CC2CCCC(=O)N2)CC)=O)ccc(C)nc1N c1(NC(C(C)NC(C2(C=C)CCOCC2)=O)C(C)C)nc(Cl)nc2[nH]c(O)nc12 c1(NC(C(C2CC2)NC(Cc2scc(C)c2)=O)=O)cnc2c(c1)CCC2 CCC(CC)C(C(=O)N1CC(OC)C(CC(=O)NC(c2cccnc2)C)C1)OC N1(C(c2c(SC)c[nH]n2)=O)CCN(C(=O)CO)CC1.C12(CC1)CC(=O)NC2 Cc1ccc([N+](=O)[O-])c(C(N2CC(CNC(=O)C(F)(F)C(C)O)CC2(C)C)=O)c1 C1(c2ccccc2)(NC(C=COCC)=O)CCN(C(C2CCCC2)=O)C1 C1(NC(C2(COCC)CC2)=O)CCCC(C(=O)N(C)CC2(F)CCC2)CC1 n1(CC(C)C)ccnc1CNC(=O)NC(c1nc(O)n[nH]1)C Cc1cc(NC(C2CC(F)CN2c2nccc(C(F)F)n2)=O)ccc1Cl Cc1cc(C2CC2C(=O)NCC2CC(NC(=O)C(O)CC3CCCO3)C2)cc(C)c1 Cc1cc(CCNC(=O)C(C)C(C)NC(=O)C(C)(C)F)cc(C)c1 c1(C(=O)NC(CNC(CCC(C)C)=O)C2CCC2)c[nH]c2cccnc12 N1(C(=O)CCCC2CCCC2)CCCN(C(c2ccc(C(F)F)o2)=O)CC1 C(=O)(C1=CCSC1)NCC(CN(C(=O)CC1CCCCC1)CC)(C)C Cc1cn2cc(C(=O)NC(C)(C)CNC(C3(CCF)CCOCC3)=O)nc2s1 N1(C(CCCCCC)=O)CC2(C1)CN(C(c1nc3c(s1)COCC3)=O)CC2CO N1(C(C(c2ccc(C)cc2)C)=O)CCCCC(NC(=O)Cn2ncc(Cl)c2C)C1 O=S1(=O)CC=CCC1CN1CCCCC1C1CCCNC1 c1(SCC(=O)NCC(CN(C)C(c2cccc(Cl)c2)=O)O)ccc(F)cc1F C1(C(N2CCC(CN(C)C(C3(NC(N)=O)CC3)=O)C2)=O)CCCS1(=O)=O C1(NCC2(C(=O)OC)CC3(CC3)C2)CCCN(C(C)=O)C1 N1(C(C(C)CSC(F)(F)F)=O)CC(NC(c2csc(O)n2)=O)CC12CCOCC2 C(=O)(C(C(C)(C)C)N1CCCCC1=O)NC(CC)(CNC(=O)Cc1ccco1)CC c1(C(C(=O)NCC(CNC(C=CCCC)=O)OC)(C)F)ccc(F)cc1 CN1CCCC(CNC(c2ccc(CNC(C3CC3(F)Cl)=O)nc2)=O)C1 Cc1ccc2scc(CC(N3CCN(C(=O)C#CC4CCC4)CCC3C)=O)c2c1 N#Cc1ccc(C(=O)NCCC2(CNC(=O)CC(F)F)CCC2)c(C(F)(F)F)c1 C1(NC(CCCOC)=O)CC(C)CN(C(=O)C(=O)NC2CC2)C1 C(=O)(C(C)(O)C(F)(F)F)N(C)CCC1CCN(C(c2scnc2Cl)=O)CC1 c1(OCC)cncc(C(=O)NCC2CC(O)CN2C(=O)C(C)OCC(F)(F)F)c1 C1(C(=O)NC2CCCN(C(C(N3CCNC3=O)C)=O)C2)Cc2cc(Cl)ccc2O1 n1(CC(=O)NC2CCCC2NC(c2ccc(F)o2)=O)cnnc1O c1(C(=O)NCCN2CC(O)CC2C2CC2)ccnc(-n2ccnc2)c1 N1(C(CN(C2CCC2)C)=O)CC(F)CC1CN(C(=O)COCC1CCCCO1)C CC(C)CC(C(=O)NC(C)CCCCNC(c1ccc(N)c(O)c1)=O)C(N)=O c1(C(=O)NC(CCNC(C2C(CC)C2)=O)(C)C)cnc(O)c(Cl)c1 c1(C(=O)NCc2cc(C(=O)NC3C(C)CCC3)n[nH]2)ccnc(O)c1 C(CCCCC(=O)NCc1ncccc1C(=O)NCCC1CC1)SC C(=O)(C=C1SCC(=O)N1C)NCc1c(N(C2(C(=O)NCC)CC2)C)cccc1 N1(C(c2c(SCC)cc(Cl)cc2)=O)CC2CCC(C1)N2C(=O)C(C)CC(C)C CC(C)CC(C(=O)OC(=N)O)NC(=O)C(n1cc(CN2CCCC2)nn1)C N1(C(C(N(C(C2C(C=C)OCC2)=O)C)C2CC2)=O)CC2CCC(O)C(O)C12 C1(OCCn2cc(-c3c(C)ccs3)nn2)CCCN(C(C2CS(=O)C2)=O)C1 C12(NC(c3c(C)cc(F)cc3)=O)CCC(CN(C(c3c[nH]nc3C(F)F)=O)C1)C2 c1(C(=O)NC2CC3CC(NC(CCCOC)=O)CC32)cc(F)c(C#N)c(F)c1 C(=O)(C#CC1CCCCC1)N1C2CC(NC(=O)C#CC3CCOC3)CC1CC2 c1(NC(C2C=CCCCN2)=O)cccc(-n2cc(CCCCO)nn2)c1 N1(C(C(C)NC(N)=O)=O)CCC(CNC(c2cc(C(C)(C)C)n[nH]2)=O)C(CO)C1 c1(NCC(CCC=C)O)ccc(S(=O)(=O)NCC2CC3(CCCCC3)C2)c(Br)c1 N1(C(c2cccn3nccc23)C(=O)NC(C)C)CCC2(COC(=O)N2)C1 N1(C(C2C(CC)CN(C(=O)CC(C)N(C)C)C2)=O)CCCC(C)C1C N1(C(=O)C=C2CCC2)CCC2CCCC12CNC(C1(Br)CC1(F)F)=O C1(N(C(=O)Cc2cncnc2O)C)CC2CC1N(C(=O)CNS(N)(=O)=O)C2 c1(SC)cc(C(N2CCOCC2CCNC(=O)CC(C)CN(C)C)=O)ccc1N CCC(F)C(=O)NCC1(NC(C2CC(O)(C(F)(F)F)C2)=O)CC1 c1(CC(=O)NCCCN(C(CC(CC)C)=O)C2CCCC2)cc(Cl)ccc1OC c1(C(=O)NC2CCCCN(C(c3n(C)nc(O)c3)=O)C2)cccc2nc(S)oc12 C1(CC)CCC(N=c2[nH]c(=NCc3cc(N)ccc3F)[nH]c3ncn(C)c23)C1 c1(CC(Cn2cc(CCSCC)nn2)CO)ccc(F)cc1 C1(CC(=O)NC(CC)C(F)(F)F)CN(C(=O)CC2(O)CCCOC2)C(C)(C)C1 Cc1cccn2nc(C(N3CC(NC(=O)CC4CCOC4)C(C)(C)C3)=O)cc12 c1(CN(C(=O)C(O)C2CN(C(=O)CCN(CCO)CCO)C2)C)ncn(C)n1 C1(CC(=O)OC)CCC2(CO1)CN(C(=O)C(c1ccc(F)cc1F)OC)C2 C1(Nc2onc(-c3ccc(C)cc3)n2)C2CC3CC(C2)CC1(CO)C3 N1(C(CCNC(=O)NC)=O)CC(NC(c2cnc(S)[nH]2)=O)CC12CCCOC2 c1(OCC)ncc(C(=O)NC2CC(NC(C3CC(N4CCOCC4)C3)=O)C2)cn1 c1(CNC(C2CC(NC(c3c(C)cno3)=O)C2)=O)ccnc(C)n1 C(=O)(C1=CCOCC1)NCCN(CC(C)O)C(=O)CN1CCCNS1(=O)=O O(NC(=O)C(CC)NC(c1cc[nH]c1)=O)CC(COCC)O C1(NC(CC=C)=O)CCN(c2ncc(C)cn2)C1(C)C N1(C(c2cc(C)nnc2)=O)CC2C(C1)N2C(c1cccn(C)c1=O)=O C1(NC(C(C2CC2)SC)=O)(Cc2cccs2)CCCN(C(c2coc(CO)c2)=O)C1 O=C(CCC1CCN(C(C2CC23CC3)=O)C1)NOCC1CC2CCC1O2 C1(CC(=O)NC(CCOC)CNC(=O)C(C)C)CCN(C)CC1 c1(N2CCC3(CCN(C)C3)C2)nc(=NCc2cncs2)[nH]c2c1CCCCC2 C1(NC(N(C2CCNC2=O)Cc2cnc(CC)s2)=O)CC2CCC1CC2 c1(CNC(=O)COCCN(C)C)cc(C(=O)Nc2c(C)ncs2)on1 c1(CC(=O)NC2C(NC(C(CCC(C)C)O)=O)CCC2)ccc2ccccc2c1 C(=O)(C1SCCc2sccc21)N(CCC(C(C)C)NC(c1cccc[n+]1[O-])=O)C C1(C(=O)NC(CNC(=O)COCCOCCOCCO)(C)C)CCC(=O)NC1 C1(C(N(CCOC)CCNC(c2cocc2Br)=O)=O)CCC2CC2CC1 CC1CCc2nc(CNC(=O)NCC(C)(C)C(F)(F)F)sc2C1 C(=O)(C(O)CCCC)NC1CC2C(NC(C(C)NC(CC)=O)=O)C2C1 CC(C)(C)CC(O)CC(=O)NCC1(C(N2CC3(CCCC3)C2)=O)CCC1 c1(N(C)CC2(OCC)CCOC2)cc(C)[nH]c(=NC(CC(C)C)C(N)=O)n1 C=CC1(CC(N2CC(NC(C3CCC3COC)=O)CC2CO)=O)CCCCC1 N1(C(c2c(Br)c(C)n(C)n2)=O)CC2CN(C(=O)CN=S(C)(C)=O)CCC12 c1(N2CC(CN(C(C(C)CN(C)C)=O)C)OCC2)[nH]cnc2nc(Cl)cc1-2 CN1CCN(C(=O)Cc2ccon2)CC1CNC(c1cccc(C2CCC2)c1)=O CC1CC=C(C(=O)NCCn2ccc(C(N3CCN4CCCC4C3)=O)c2)CC1 Cc1ccc(C=CC(N2CCCC2C(C)NC(=O)C(C)C)=O)nc1 N1(C(c2nc(OC)oc2)=O)CCC2(CC1)CN(C(c1ncc(C)nc1OC)=O)C2 c1(CC)nc(C)c(C(N2CCC(OCCNC(c3nc(Cl)oc3C)=O)CC2)=O)s1 C1(C(=O)NC(CCC=C)C2CC2)CCCN(C(=O)C(O)C2CCCC2)CC1 C1(C)(NC(c2nc(=O)n(C)[nH]2)=O)CCN(C(CNC(CCNC(C)=O)=O)=O)CC1 C(=O)(C(Cc1ccccc1)CF)NCC(C)(C)F C1(C(=O)NC(C(=O)N(CC(CCC)C)C)COC(C)C)CCC(=O)N1C C1(C)(C(=O)NC2CC(CNC(C(C)OCc3ccccc3)=O)C2)CCOCC1 Cc1c(C(=O)N(CCCOCCNC(=O)C2=NOCC2)C)[nH]c2ccc(F)cc12 CC1(C)CN(C(c2cccnc2Cl)=O)CCC1NC(=O)CC1CC2CC2C1 c1(CSC(C)C(=O)NC(c2ccccc2)C2CCC2)nc(C(C)(C)C)n[nH]1 C1(NC(c2c(C)nn(C(C)C)c2)=O)CCN(C(C2CC(O)(C(F)F)C2)=O)C1(C)C C1(CC(=O)NC(C#CC#C)(C)C)CN(C(c2ccnnc2C)=O)CC12CC2 C1(C(=O)NCC(CCC)OC)CC2CCC(C1)N2C(=O)CCc1cccn1C CC(c1ccco1)=CC(=O)NCC1CN(C(C2(C)CC(F)(F)C2)=O)CC1C CC1CN(C(=O)CC2CC2(Cl)Cl)CC(C)N(C(c2ccn(C)c(=O)c2)=O)C1 C(=O)(C(=O)C(C)(C)C)N(C1CCC(NC(c2cn(CC)nc2C(C)C)=O)CC1)C N1(C(C(C)N2CCC2)=O)CCN(C(c2csc(C(F)F)n2)=O)CC1C(F)F c1(SC)ccc(OC(C)(C)C(=O)N(C)CCNC(=O)CC2CCCCCO2)cc1 N1(C(C(C)(C)OCC)=O)CCC(CNC(=O)CC2(O)CCCCC2)C1(C)C c1(CC(=O)NCC(=O)NCc2ncccc2O)ccc(Cl)cc1Cl Nc1c(Cl)cnc(C(=O)N(CCCNC(C2CC=CCC2)=O)C2CC2)c1Cl c1(C(N2CC(NC(=O)CC3CSCCS3)C2)=O)ccc2nc(Cl)ccc2c1 C1(CNC(c2ccc(F)c(F)c2F)=O)CC2COCC2N1C(C1(F)CCCC1)=O C(=O)(C1=CCCC1)N(C(C(N1C(COC)CCC1)=O)C)C1CC1 c1(C(=O)NC2CCC(C)(CNC(C(=O)NC(C)C)=O)C2)cc2cccc(F)c2s1 c1(C(N2CCC(N(C(c3cc(Br)c[nH]3)=O)CC)CC2)=O)ccc2nc(C)oc2c1 Cc1cccc(C(=O)N(C(C)CN(C(c2[nH]c(O)nc2C)=O)C(C)C)CCO)c1 C12CC(S(=O)(=O)N(C(C)=O)N3CCC(CC3)N1)C2.c1(NCC(=O)OC)nccs1 C#Cc1ccc(Cl)c(-c2nc(Cc3ccncc3)nn2CC(C)C2CC2)c1 C1(C(=O)NC2CC(CNC(C34CC(C)C3C4)=O)C2)CCC12CCC2 Nc1ccc(C(=O)NC2(CCNC(C3CC3C(F)F)=O)CCC2)c2c1CCCC2 C(=O)(CC(CNC)C(F)(F)F)NC(CCN(C(C(CC)NC(C)=O)=O)C)C.C(C)=O c1(C(N(CC(CC)NC(C2CCCC23CCC3)=O)C)=O)ccc(P(C)(C)=O)nc1 Cc1cc(F)cc(C(=O)N(CC(O)CN(C)C(c2ccc(C(F)F)o2)=O)C)c1N N1(C(=O)CCNc2ncccn2)CCC2CN(C(c3csc(CO)n3)=O)C2C1 c1(SCC)ccccc1C(=O)NC1(C)CC(NC(C2(CCO)CC2)=O)C1 c1(C(N2CC(OCCNC(C3CC4(C3)CC4F)=O)C2)=O)cc(F)cc([N+](=O)[O-])c1 N1(C(C2C(C(=O)OC)C2)=O)CC2(COC(CNC(C34CCC(C3)OC4C)=O)C2)C1 CC#CCCCC(=O)N1CCC(CCNC(c2cc(C)cc(C)n2)=O)C1 c1(CNC(N(CC(C)CN)C)=O)csc(-c2ccccc2)n1 C#Cc1ccc(F)c(C(=O)NC(C)CN(C(=O)C(C)(C)c2ccccc2)C)c1 C1(N(C(CNC(c2cccc(C)c2)=O)=O)C)CC2CC1N(C(=O)CN(C)C1CC1)C2 c1(C(N(Cc2c(CN)cccc2)Cc2ccccc2)=O)ccc(I)c(Cl)c1 CC(C)C(N=[N+]=[N-])C(=O)NCC1CCN(C(C2(CO)CCCO2)=O)C1 N1(C(C2(CSC)CCC2)=O)CCOC(CNC(=O)C(C)c2cc[nH]n2)C1 C1(C(N(CCN(C(CC2CN(C)C2)=O)C)C2CC2)=O)CCC(C)CC1C(=O)OC.NC C1(O)(C(C)NC(=O)Cn2ncccc2=O)CCN(C(c2cccnc2)=O)CC1 N1(C(c2cc(C)ncc2C)=O)CCOC2(CCN(C(c3cc(C)n(C)n3)=O)C2)C1 N1(C(c2ccc(-n3cc(Br)cn3)cc2)C(=O)NC2CCC2)Cc2c[nH]nc2C1 CC(C)(C)CCC(=O)C(=O)NC1CC(CNC(c2ccc3c(c2)CCO3)=O)C1 c1(C(N(C)CC2CCN(C(c3c(CCC)occ3)=O)C2)=O)cc(OC)nc(Cl)c1 C1(C(N2CC(O)(CNC(C3(C4CC4)CCCO3)=O)C2)=O)(COC)CCCO1 C1(C(N2CCCC(C(=O)NCC3(CO)CCCO3)C2)=O)CC2CCCC2C1 c1(CC(=O)NC(CSCC)C(=O)N2CC(C(C)OC)C2)ccc(O)nc1 c1(C(N2C(CNC(c3cc(CC)ncc3)=O)CCC2)=O)c(C)c(C)cc(C)c1C c1(OC)cc(CNC(=O)CC(C)(C)N(C(=O)Cc2ccn(C)n2)C)n(C)n1 C1(NC(C2(CC=C)CC2)=O)CC2(CCCN(C(c3cc(C)c(F)cc3F)=O)C2)C1 C(=O)(CCC(C)c1ccccc1)NC(CCNC(C(C)(C)OC(C)C)=O)C C1(CNC(c2cn(C3CC3)nn2)=O)CCCN(c2ncccn2)C1 c1(C(=O)NC(c2ccc(OC)cc2)CNC(CC)=O)cc2ncccc2s1 c1(C(N2CC(C(=O)NC)C2)=O)ccc(OCc2cccc(OC(F)(F)F)c2)cc1 C1(C(=O)NC2(COC)CN(C(c3cc(F)ccc3O)=O)C2)CCCCNC1=O C(=O)(NNS(=O)(=O)c1ccc(Br)c(Cl)c1)C1(CC)CCCO1 CC1(C)C(NC(c2cc(Cl)sc2Cl)=O)CCN1C(c1cc(N)c(F)cn1)=O CC1CCN(C(c2ccc(Oc3cccnc3)cc2)C(=O)NC2COC2)CC1C c1(C(C)NC(=O)NCC2CC2C(=O)NC2CC2CO)cccc(Br)c1 C(CCCC(=O)NC(C1CCN(C(C2(C(C)(F)F)CC2)=O)C1)C)OC C12(C(=O)NC(CN3CCCC3)CO)CCN(C(C3CN4CCC3CC4)=O)CC1C2 C(CCC(O)C(=O)NCC(C)C(F)(F)F)NC(CC1CC(OC)C1)=O N1(C(c2c(CC)nc(C)cc2)=O)CCC(NC(=O)OC(C)(C)C)C(C)(C)C1 C1(CNC(C(CC2CCCC2)NC(CC=CC=C)=O)=O)CC(C2CC2)=NO1 c1(C(=O)NC2CC(CNC(=O)C(O)c3ccsc3)C2)scc2c1OCCO2 c1(C(=O)NCCC2CN(C(C(C)CC3CCC3)=O)C2)cc(N)cnc1Cl N1(C(c2ccc(Cl)c(Br)c2)C(=O)NC(C)C)CCOc2ccncc2C1 C(C)(N=c1nc2scnc2c(NCC(C)(C)N2CCCC2)[nH]1)c1cccc(OC)c1 CCC(F)(F)CC(=O)NCC1CC1NC(=O)COCCCF C(CC(=O)N1CCCc2ccnn21)N(C(c1ccc2cncn2c1)=O)CC1CC1 C1(C(N(CCC(=O)OCC)C)=O)CN(C(=O)Cc2cccc(O)c2)CCC1O C#CC1(C(=O)Nc2ccc(F)cc2)CN(C(c2cc(CO)oc2C)=O)C1 C#Cc1cncc(NC(=O)CCCNC(C)=O)c1.N12CCCCC1C2=O C1(CNC(C(CCC)CC)=O)CN(C(=O)Cc2c(Cl)cnn2C)CCC1(F)F C(=O)(C(CNC(=O)C(c1ccccc1)C)CC(C)C)NCc1cccc(CC)c1 c1(SC)cc(C(N2CC(CNC(c3c(C)[nH][nH]c3=N)=O)CC2C)=O)nn1C C1(NC(C2C(COC)C2)=O)CCCC1NC(c1cn(CCC(C)(C)C)nn1)=O c1(CNC(C2OCC(COC)C2)=O)ccc2c(c1)CCCS2(=O)=O C#CCC(C(=O)NC(C)CC)NC(=O)CN(C1CC(=O)C1)C C(=O)(C(C)CCCC(C)C)NC1(C(N2CCC(C(=O)NC)CC2)=O)CCCCC1 c1(OC)cnc(Br)cc1NC(=O)CC1CC(NCc2ccccc2Cl)C1 c1(C(=O)Nc2scc(C(N3CC4OC(C)CC4C3)=O)n2)cncc(S(C)(=O)=O)c1 CC1(NC(=O)C=Cc2cccnc2)CCCN(C(C2CCCOCC2)=O)C1 c1(C(N2CCCC2c2oc(C)nc2C)C(=O)NCC(=C)C)nn(C)cc1C c1(OC)cccnc1C(=O)NCC#CCNC(=O)CN1CCCNC1=O N1(C(C(CC)(CNC(=O)CCCC2CCCO2)CC)=O)CCC2(CNC(=O)O2)C1 CC1(C)CC1(C)C(=O)NC1CCC(NC(c2csnn2)=O)C1 C=C1CC2(C1)CN(C(C1(CNC(C3CCC(=O)N3)=O)CCCCC1)=O)C2 N1(C(C=CC(C)C)=O)CCC(C)(C)C1CC(=O)NCCCC1(C)CC1 CS(=O)(=O)C=CC(=O)N1CCCCC(NC(=O)CC2CCC3CC23)C1 c1(C(=O)NC2CC(NC(c3cncc(SC)c3)=O)C2)cc2c(Cl)cccc2[nH]1 N1(CC)CCCCC1CNC(=O)C(CCC1CC1)NC(c1cc(Cl)n(C)n1)=O C1(C(=O)NCC(CC(=O)NC(CCCC)CC)O)CN2CCN1CC2 Cc1cccc(C(C)NC(=O)C(=O)NC(C2CSCCS2)(C)C)c1 c1(C(C)(C)C)ccc(CNC2CC(n3cc(CCCO)nn3)C2)o1 Cc1cc(C(=O)NC(C)CC(=O)N(CCCO)CCO)c(C)cn1 C1(F)(C(=O)NC(CCOCC)C)CCN(C(C2CC(N(C)C)C2)=O)C1 Cc1ncc2n1CCN(C(C1COC3(C1)CN(C(c1cnccn1)=O)C3)=O)C2 C1(CNC(CC(C)NC(N)=O)=O)CN(C(=O)C(C)(F)F)C2(CCOCC2)C1 c1(C(=O)NCC2C(NC(c3ccc(OC)nc3)=O)COC2)ccc(N)cc1Cl C(=O)(C1CCc2nccn21)NC1C2CN(C(C=Cc3occ(C)n3)=O)CC21 C1(C2N(C(=O)NC)CC(=O)NC2)CCN(C(=O)C2CC2)CC1C(F)(F)F CCC(CC)C(C(=O)N1CCC1(C)CC(N1CCOC(C2CC2)CC1)=O)OC c1(N(C)CC2CC3CC3C2)nc2c(c(=NCC3CCC(C(F)(F)F)O3)[nH]1)SCC2 c1(C(N2C3(CNC(COCCOC)=O)CCC3CC2)=O)cc2c([nH]1)CCCC2=O C1(OC)CCC2CN(C(=O)C(C)(CSC)NC(c3ccccc3CO)=O)CC12 C1(C(N(CCCCCNC(c2n(CCOC)ncc2)=O)C)=O)CCC(C)CC1 c1(CC)ncoc1CNC(=O)CC1CCN(C(=O)CCc2cnoc2)C1 CCC(C)(C(=O)OC)NC(=O)NCc1cc(N2CCCC2)ncn1 c1(OC)ccc(CSCc2cn(-c3ccc(C)c(OCC4CC4)c3)nn2)c(OC)c1 c1(OCC)ccc(F)c(CN2CCC(=O)N(CCC3=CCCCC3)C2=O)c1Br C1(CC)CCN(C(=O)CC2(OC)CCC2)C1C(N1CC(CO)C(O)C1)=O C(=O)(C1CCCc2c1ncn2C)NCC(CNC(CCC)=O)C(F)(F)F C1(CC(=O)NCC2(C(N)=O)CN(C(=O)CSCC3CCCO3)C2)NC(=O)NC1=O Cc1nc(C(C)C)cc(=NC2CCCC23CNC3)[nH]1.C(C)(C)(C)OC=O N1(C(c2cc(OC)nn2C)=O)CCOCC(F)(CNC(=O)C=CSC)C1 c1(CC(=O)NC2CCC(NC(Cc3[nH]c(=N)sc3)=O)C2)ccc(F)cn1 C1(CCN(C(=O)Cn2cnccc2=O)C)CCN(C(=O)CSC(F)(F)F)CC1 C1(CNC(C2C(NC(COCCC)=O)CCC2)=O)COCC(=O)N1C N1(C(Cc2c(C)con2)=O)CCC2(CC1)CN(C(c1ccc(F)c(N)c1F)=O)C2 N1(C(=O)CSC2CCC2)CC2(CCCN(C(c3cn(CCC4CC4)nn3)=O)C2)C1 C12(NC(=O)CC3CCN(CCF)CC3)CCCC(CN(Cc3cccnn3)C1)C2 C1(CN2CCC(O)(c3ccc(F)cc3)C2)CC[Si]2(CCCC2)CC1 N1(C(C2(C)CCCN(C(=O)CC3CCCNC3=O)C2)=O)CC(O)C2(CCCC2)C1 c1(CC)cccnc1C(=O)NCC1(NCC#CCNC(C2CC2C)=O)CCCC1 N1(C(C)=O)CC2CN(C(=O)CC(C)(F)F)CC2(C(F)(F)F)C1 N1(C(C(CCSC)O)=O)CCC(C2(NC(=O)Cc3cccc(C)c3Cl)CC2)CC1 N1(C(C=Cc2n(CC)ncc2)=O)CCCC2(NC(C3CC3(C)Br)=O)CC2C1 C1(C(N(CC(CNC(CCCN(C(C)=O)C)=O)C)C)=O)CC2(CCO1)CC2 C1(C(=O)NCCCNC(c2cccc(C3(F)COC3)c2)=O)CCCC2(CC2)C1 C1(C(C)NC(=O)CCC2CCCOC2)CCN(C(=O)C(C)(C)CF)CC1 c1(OCC)ccccc1NC(=O)CCC1CCC(NC(=O)CCN(C)CCO)C1 Cc1cc(C(=O)OC2CN(C(=O)OC(C)(C)C)CC2OC(C)C)ncc1C(F)F N1(C(C2CCC(C(F)(F)F)CC2)C(=O)NC2CCC2)CCCC2(CCCCO2)C1 c1(C(=O)NC2C(NC(CNC(N)=O)=O)C2)ccc(-c2ccc(F)cc2)cc1F c1(OCC(N2CC(C(C)NC(c3cnc(C(C)C)[nH]3)=O)C2)=O)cccc(F)c1 CC(C)CCCC(=O)NC(CC(=O)NCC1(O)CCC1)C1CC1 C1(CC(=O)NC(CC2CC(C)(C)OC2)=O)CC2CCC1(NC(=O)C(F)(F)F)C2 CC1=C(C(=O)NC2CCCCC2NC(c2cc(Cl)nnc2O)=O)CCC(C)(C)C1 N1(CCn2c(N3CCC(COCC)C3)nnc2C(C)(C)CC)CCOCC1(C)C CCC(C(F)(F)F)NC(=O)CCCNC(=O)C(C)(C)CC1CC1 c1(C(C2CCCN2C(=O)OC2COC2)=O)cccc(Cl)c1 CCCCC(C(=O)NC(C(=O)N(C)CCOCCCO)C1CCCO1)NC(N)=O Cc1c(CC(=O)NCC2CCCCN2C(=O)Cc2coc(C(F)F)n2)cnn1C C1(NC(Cc2c(OC)cccc2)=O)CN(C(c2cc(C3CC3)no2)=O)CC12CC2 C1(C(=O)NC2CCN(c3ncc(OCC)cn3)CC2)CC2CCCN(C1)C2 C1(C(CNC(c2c(CC)cno2)=O)F)CCN(C(=O)C(C)(C)NC(=O)OC)CC1 C1(O)(CNC(c2ccccc2OC2CCC2)=O)CCN(C(c2ccnnc2)=O)C1 c1(C(N(C2CCC(NC(=O)CC3CSCCO3)C2)C)=O)cnc2ccnn2c1 c1(C(N(C2CCN(C(=O)CCCc3cccc[n+]3[O-])C2)C)=O)ccc(N)cc1F CCCC(CC)C(=O)N1CC2CC2(NC(c2c[nH]c(C(F)(F)F)c2)=O)C1 O=C1NC(CCCNC(c2ccc(OCC(F)(F)F)cc2)=O)c2ccccc21 N1(C(C(C)NS(CC)(=O)=O)=O)CCCC2(CCN(C(=O)C=CC(=O)N(C)C)C2)C1 C(c1ccc(F)cc1)=CC(N1CCCC(CN(C)C(C2CC2(C)Br)=O)C1)=O N1(C(C(CC)CC)=O)CCC(C2CCN(C(c3nccc4ccncc34)=O)C2)C1 C1(C(=O)NCC=CCNC(c2onc(OC)c2Br)=O)CN2CCN1CC2 N1(C(C)C)CCC(CNC(=O)CNC(c2n[nH]c(=N)[nH]2)=O)C1 c1(C(N(C(CC)CO)CC2(CO)CC2)=O)ccc(-c2sccc2C)s1 C(CCC(=O)N1CC(F)(CNC(=O)C(C)C2CCOC2)C1)N(C(=O)OC)C N1(C(c2c(CC)con2)=O)Cc2ccccc2C(CNC(=O)C(O)CC(N)=O)C1 CCC(C)C(CC(=O)NCc1cnc(C)cc1C)NC(c1ccncc1NC)=O N1(C(C(C2CC2)OC)=O)CCCCC2(CCN(C(=O)CCCC(C)C)C2)C1 c1(CC)c(C(=O)NCc2ccoc2C(=O)NC(C)C(F)(F)F)ccn1C CN1CCN(C(=O)Cc2ccc[nH]2)CC1C(=O)NC(C)(CO)C1CCC1 N1(C(c2cc(CC)oc2C)=O)CCC(C2CCCN(C(C3(C)CC(F)C3)=O)C2)C1 c1(C(N2CC3N(C(COCC)=O)C(CC3)C2)=O)nc(C)n2c1CCCC2 CCCC(O)C(CO)NC(=O)C(C1(O)CN(C(=O)Cn2c(C)ccc2C)C1)F CC(CC(F)(F)F)N(C(=O)C(c1ccco1)NC(C1CCCC1)=O)C C1(C(=O)NC2(CC(=O)NC(C3(CO)CC3)C)CCC2)CCN(C)C1 C1(CNC(c2c(C)nns2)=O)CCN(C(c2c(Cl)nsc2Cl)=O)CC1C c1(C(N2CC(C(C(=O)NC(CCCC)COC)OC)C2)=O)cc(O)cc(F)c1 C1(C(=O)NCC2(CNC(C(CC)(C)O)=O)CCC2)CN2CCN1C(C)C2 C1(NC(CSC(C)C)=O)CCCCC1CNC(C1CCCC1)=O n1(CCC)nnnc1C(c1nocc1COC)NCCCOC C1(C(N2CCC(NC(C3(C=C)CCCC3)=O)C2)=O)CC(=O)CC(=O)N1 C1(C(N2CC3C(N(C(c4nc(C)n(C)n4)=O)C)C3C2)=O)CCN(C)S1(=O)=O N1(C(c2scc(OC)c2)=O)CCN(C)CC1CNC(c1ccc(O)nc1)=O C1(CN(C(=O)C(c2cncn2C)N(C)C)C)CCN(C(=O)CSCC(F)F)C1 C1(C(=O)OC)Cc2ccc(O)cc2CN1C(c1ccc(CC(C)C)cc1)=O C=CC(C)(CCOC)C(=O)N1CCCC(C)(CNC(c2onc(Br)c2C)=O)C1 C1(CC)(NC(C2CCC3(CCC3)O2)=O)CCCN(C(c2c[nH]cc(C)c2=O)=O)C1 Cc1c(C(=O)NCCC(O)CNC(=O)C=CCF)cnn1C(C)C(C)(C)O CC(CO)C(=O)NC(CNC(c1ccoc1C1CC1)=O)C1CC1 C(=O)(CCC(=O)NN(C)C)NC1CC(C)CN(C(c2cncs2)=O)C1 c1(C(N(CC(CC)NC(C2CC2C(F)(F)F)=O)C)=O)ccc2cc[nH]c2c1F C1(C(=O)NC(C(C)NC(=O)Cn2cc(CN(C)C)nn2)(C)C)CC(F)C(=O)N1 N1(C(c2cccc3cc(C)[nH]c32)=O)CC(C(=O)O)C2(C1)CN(C(=O)C(C)CN)C2 c1(C(N2CCC(C)(CNC(C(CC=C)C)=O)C2)=O)c(C)ccc2ccccc12 C1(C(C(=O)NCCN(C(=O)CCNC(C2CCC2)=O)CCC)O)CC(F)(F)C1 c1(C(c2nnnn2C2(C)CC2)Nc2ccc(C)cc2)ccc2c(c1)CC(C)(C)O2 c1(-c2n(C)c(COC3CCc4ccsc43)nn2)cc([N+](=O)[O-])ccc1N c1(C(=O)NC(c2ccccc2)C(C)NC(C2CSC2)=O)ccc([N+](=O)[O-])cc1F c1(SCC(=O)NCC2N(C(CC(=O)OC)=O)CC2)ccc(Br)cc1C Cn1c(C(=O)NC(CNC(c2cncc(-c3cc[nH]n3)c2)=O)C2CC2)cnc1S CC1CN2CCN1C(C(=O)NCC1CCN(C(c3ccc(F)c(Cl)c3N)=O)C1)C2 c1(C(N(C2CCN(C(=O)CC=C)C2)CC#C)=O)c(F)cccc1Cl C1(NC(c2cc(SCC)ncc2)=O)CC(O)CN(C(c2sccc2C(C)=O)=O)C1 Cc1nn(CC(=O)NC2CC(CNC(=O)CCF)C2)c(C)c1C=NO C(c1cccc(F)c1)=C(C(N1CC(CNC(=O)C=C(Cl)Cl)C(O)C1)=O)F C1(CNC(CCCN(C(C)C)C)=O)CCC(NC(C2CCC23CCC3)=O)CC1 C1(NC(C2C(SC(C)(C)C)CN(C(=O)CSCC)C2)=O)CC2C(C1)C2(C)C c1(NC(=O)NC(CCC)C)ccncc1-c1cncc(C(=O)NC)c1 Cc1ccccc1-c1cc(C(=O)NCC2COC(CNC(c3cnsc3)=O)C2)no1 C1(C)(C(=O)NC2(C)CN(C(c3ccc(CC)cn3)=O)C2)CCC(=O)N(C)C1 C1(NC(COCCC)=O)CCCC(NC(=O)CC2CCOCC2OCC)C1 S(=O)(=O)(c1ccc2ccccc2c1Br)NCC(CCN)O.C12CCC(C1)N2 N1(C(c2c(=N)cc[nH]c2)=O)CCCC2CCN(C(=O)C=C3CCC3)CC12 C12CCCC1C(=O)N(C)C(=O)NC2.C1(CC)CC(CC(=O)OC2CCSC2)C1 C1(NC(CC(CC)(C)C)=O)CCN(C(=O)COC2CC2(F)F)C12CCC2 N1(C(C=CC2N(C(CSC(C)C)=O)CCC2)=O)CCCC12CCCC2 C1(C(=O)NC)CCN(C(=O)C(C2CC2)N(C)C(C2C3CCCCC23)=O)CC1 c1(C(N(CC(C)N(C)C(C2C3CCCCC23)=O)C)=O)ccc(C#N)c(O)c1 Cc1cc(F)c(C(C(=O)NCC2CCCO2)N(c2cccc(CO)c2)C)cc1F C1(C(=O)NC23C(CN(C(C4(CC#C)CC4)=O)C2)C3)C2CCN(CC2)S1(=O)=O CCCC(C(O)C(=O)Nc1cnsc1)NC(c1c[nH]nc1Cl)=O C#Cc1cccc(C2CCN(C(c3csc(Cl)c3)C(=O)Nc3ccccc3)CC2)c1 O=C(CC(F)(F)C(F)(F)F)NCC(C1CCOC1)NC(=O)CSc1n[nH]c(O)n1 C1(C(c2nnnn2C(C)CC)NC(COCC)C(C)C)CC2C(C1)C2(F)F N1(C(c2c(C)[nH]cc2)=O)CCCCCCC1C(N1CCC1C(C)O)=O c1(C(=O)NC2C(C)CN(C(c3cc(O)cc(F)c3)=O)C2)ccc2ccoc2c1 CC1CCCC1(C)C(=O)N(CCCN=[N+]=[N-])C.N12CC(C1)OCC2=O c1(C(N2CC3CCN(C(C4C(C)C4)=O)C3C2)=O)ccc2c(c1)OCCC2 c1(OC)cc(C(N2CC3CC3(CNC(C3CCCC3F)=O)C2)=O)ccc1O C1(C(=O)NC2(C)CC2(C)C)(NC(CC=CCC)=O)CCC(C)(C)C1 CC1CC=CCC1C(=O)NCCC1(O)CN(C(C2(C(=O)N(C)C)CC2)=O)C1 CCC(O)C(C)C(=O)NCc1ccccc1N1CCN(C(=O)C=CCSC)CC1 C1(O)(CNC(c2ccccn2)=O)CCOCC1.C12COCC1NC2=O Cc1cnc(C(=O)NC2CCC(C(=O)NCC(C)(O)C(F)F)CC2)cn1 c1(NC(C(C)CC2CC2)=O)ccc(Cl)c(NCCNS(C)(=O)=O)n1 CC(C)C(F)C(=O)NCC1CCC(NC(=O)C(C)(C)C2CCCCO2)CC1 c1(NC(C)CN2CCCCC2)ccc(S(=O)(=O)NC2C=CCC2)cc1Br c1(C(N2CCCC(NC(=O)Cc3ccsc3)C2)=O)cccc2c1NCC2 c1(C(C(=O)NC(C(=O)N(C)CC)C2CC2)C)cccnc1 N1(C(c2cnc(C)nc2)=O)CC2CC(C1)N2C(=O)CC1CC2C=CC1C2 Cc1cc(C(F)C(=O)N(c2cccc(CC(F)(F)F)c2)C)ccc1F N1(C(C(C)NC(C=C)=O)=O)CC2CCCC(C1)C2C(=O)Nc1cc(O)ncc1Br c1(CC(=O)NC2C(CNC(C3(CC)CC3)=O)C2)sc(C2CCC2)nc1C c1(OC)ccc(OC)c(NC(=O)COC(C2CCCCC2(F)F)=O)c1 CC(C)CC(C)(CNC(c1ccc(Cn2cncn2)cc1)=O)NC(=O)C(F)OC c1(C(N2CC3(CC(CC(=O)NC(c4ncc[nH]4)C)C3)C2)=O)ccc2nncn2c1 CC(C(=O)N1CC(OC2CCN(C(=O)Nc3ncc(CO)[nH]3)CC2)C1)S(C)(=O)=O CC(C(=O)NCCCN(C)C)N(C(=O)C(C)n1cccc1)C1CC1 C1(NC(c2n(CC#C)cnn2)=O)CN(C(C2SCC=C2C)=O)CCC1C(F)(F)F C1(NC(C2(CC=C)CC2)=O)CN(C(c2ccc(=O)n(C(C)C)c2)=O)CCC1O C(CNC(=O)NCc1cccnc1F)(CC(=O)N1CC(NC(N)=O)C1)OC C#CCC(C(=O)NC)NC(C1(C(=O)NCC2CCCC(=O)C2)CCC1)=O c1(OC(N2C(C(CC)C)CCCC2)=O)ccc(OC)c(C#N)c1 C(C(C)CN=c1cc(C(F)F)nc(SC)[nH]1)NC(C(C)OCC)=O c1(C(C)C)cnc(Cl)[nH]c1=NC(C)CCNC(=O)Cc1c[nH]c2cccnc12 c1(C(=O)NC2CCC2CNC(C23CCCC2C3)=O)cccn(C2CCC2)c1=O C1(NC(c2cn[nH]c2)=O)CCN(C(C2CCC=CCCC2)=O)CC(O)C1 C1(C(N(CCC(F)(F)F)CC)=O)(NC(c2ccc(N)cn2)=O)CCC(C)(C)C1 CC(CNC(c1cnc(O)o1)=O)C(=O)NOCc1ccccc1F C(=O)(C(C)(C)n1ccnn1)N(C(C1CCCCC1)CNC(c1ncn(C)n1)=O)C C(C)(CCC(=O)NC1CCC1NC(=O)CCCCN1CCCCC1)OCC C1(C(=O)NCCC2CCCN(C(C3CCCCC3)=O)C2)CCCNC1=O C1(OCC)COCCC1N=c1[nH]c(=NC(CF)CF)c2ncccc2[nH]1 C1(C(=O)NC(CCCOC)(C)C)CNC(=O)CN1C(=O)C=CC1CCC1 c1(C(N2CC(CCOC)N(C(=O)C=CC(C)C)CC2)=O)cc(C)cc(C)c1C C(=O)(C(C)(O)C(F)(F)F)NC1C(CSC)CN(C(=O)CCC=C(C)C)C1 CN1CCCC(C(=O)NC(=O)CCN(C)C)C1.c1(C2C(=O)N2)cn(C)nn1 C1(CNC(c2ccc(C(C)C)cc2O)=O)COC(C)(C)CN1C(=O)CC C(CC(=O)NOCCc1ccccc1)N(C(C1CCN1C)=O)C(C)C1CC1 c1(NCc2ccc(CC)s2)ccc(S(=O)(=O)N2CC=CC(O)C2)cc1C#N c1(CC)nc(C)c(CC(N2CCCN(C(C3CCOC3C)=O)C(C)C2)=O)c(C)n1 c1(C(N2CC(NC(C3C(C)(C)C3C#N)=O)C(C)(C)C2)=O)ccc2sncc2c1 CCC(CC)C(C(=O)NC(C1CCCN1C(C1(C)CCC(F)(F)CC1)=O)C)OC C12(C(=O)NC(CC#C)(C)C)COC(C1)C(NC(C1(C)CC(C)=NO1)=O)C2 O=C(C1=NOC2CN(C(=O)C(O)O)CC12)NCCC(F)(F)F.C12C3C=CN(C13)C2=O CS(=O)(=O)c1ccccc1SC(C1CC=CCC1NC(=O)C(=O)Cc1cccs1)=O CS(=O)C=CC(=O)N1CC(CNC(c2coc(C3CCC3)n2)=O)C1 C1(CNC(c2c(CCC)n(C)nn2)=O)CN(C)CCN1C(=O)CS(=O)(=O)CC C(C(=O)Nc1ccc(N(C)C)nc1)(C(C)C)NC(COC(CC)(C)C)=O C1(O)(CNC(c2c(C)ccnc2C)=O)CCCN(C(=O)C2=CCCCO2)CC1 C(c1ccccc1C#N)=CC(N1CCC(NC(C(C)(CO)OC)=O)C1C)=O N1(C(Cc2c(C)scc2)=O)C2CCC(C2)C1CNC(=O)C(C)(C)CF c1(OC)cc(C(=O)N(C)CCN(C(=O)C#CC2CCCO2)C)cc2c1OCCO2 C1(CC(C)C)(C(=O)NC(CN(C(C(C)OCCCC)=O)C)(C)C)CCNC1=O n1(CC=C)nnnc1C(c1ccc(CCCOC)o1)NC(C)CCF C1(CNC(Cn2ccc(C)n2)=O)CN(C(c2ccnnc2S)=O)CC12CC2 C12(C(=O)NC(C)CCNC(c3cc(F)c[nH]3)=O)CCCC(C1)OC2 N1(Cc2ccc(C#N)s2)CCC2(CCCC2C(N2CCc3ccccc3C2)=O)C1 C1(NC(COCC(=O)NC)=O)CN(C(=O)CN(C)C2CC2)C2CCCCC12 C1(c2cn(CCC3CCN(C(Cc4cn(CC)nc4)=O)C3)nn2)CC2CCC1O2 c1(C(C)NC(C(CSCC)NC(=O)Cc2csnc2C)=O)cccnc1F c1(CC(=O)C2(C(=O)NCc3cc(NCCC45CC(C4)C5)n[nH]3)CC2)c[nH]nc1O c1(NC(=O)NC2CCN(C(Cc3nc(C)[nH]n3)=O)C2)ccccc1C C(=O)(C#CC1(CC)COC1)N1C(CC(=O)NCC(C(CC)CC)O)COCC1 c1(OC)cncc(C=CC(=O)NCC2(CNC(c3cccnc3O)=O)CCC2)c1 c1(C(=O)NC2C(NC(c3ccc(C)c(N)c3)=O)C2)csc2c1CCCC2 c1(OC)ccnc(C(=O)NCC(C2CCC2)NC(c2cncc(C)c2)=O)c1OC N1(C(CCC#CC)=O)CC(NC(c2nnn3ccccc23)=O)CC12CCOC2 N1(C(C2C(NC(c3ncc(F)cc3F)=O)CC2)=O)CC2C(C1)C2(F)F C(CC(CC)C(=O)N(C)CC1(NC(c2sc(C)nc2Br)=O)CC1)=CC c1(C(=O)NCC2(CNC(c3ncccn3)=O)CC2)ccc2c(c1)C(=O)NC2 C1(CC(N2C(C)(CNC(c3cnn(C)n3)=O)CCC2)=O)CCCCC12CC2 C1(=O)CCC(=O)NC(C)CC(C)N1.C(=O)(CCCNC(C)=O)NC(C)(C)C c1(C(N2CC(C(C)C)N(C(=O)CN(S(C)(=O)=O)C)CC2)=O)cc(S(N)(=O)=O)co1 C1(C(C)C(=O)NCC(C)(O)C2CC2)CCN(C(C2(C)CCCOC2)=O)CC1 N1(C(CCCC=C)=O)CCC(C)C(CC(=O)NC2(c3nn[nH]n3)CC2)C1 Cc1ccc(C(=O)N(C)C)c(NC2CCOC(c3ccnn3C)C2)c1 C1(OCC)CC2(C1)CC2C(=O)NCCC(C)NC(=O)CN(C1CCSC1)C c1(C(N2CC(F)(CNC(C=C3CCN(C)CC3)=O)C2)=O)[nH]nc2c1COC2(C)C C(C)(C(C)NC(C1CC1CNC(=O)CNC=O)=O)(C1CC1)OC CC1Cc2cc(NC(=O)NCc3cncc(Br)c3)ccc2N1S(C)(=O)=O c1(C=O)c[nH]c2cnccc12.C12(C(=O)NCC(C)N)C3C4C1C1C2C3C41CO N1(C(c2ccc(F)c(F)c2O)=O)CCCC2C1CCN2Cc1cc(Br)cc(Br)c1 C(CCC(C)CC(=O)N1CC2(C1)CN(C(=O)CC1(C)CCS(=O)(=O)N1)C2)=C(C)C C(C(=O)OC)(C(C)C)NC(C1(C=O)CCOCC1)=O.c1(CC(CSC)O)ccccc1 C1(CNC(=O)C(F)n2ccnc2)CC2CN(C(C3(n4cnnn4)CC3)=O)CC2C1 S(=O)(=O)(c1ccc(NCc2cccc([N+](=O)[O-])c2)nc1)NCC(CC)(CC)CO C1(CCNC(COCC(=C)C)=O)CC(OC)CN1C(C1CCC(F)CC1)=O c1(C(=O)NC(CC)CNC(c2c[nH]c(=NC)o2)=O)nn(C(C)C)nc1Br c1(C(N2CC(C3CN(C(C4CCCCCCC4)=O)C3)C2)=O)ccc2c(c1)CCC2 c1(CNC(C(C)C(C)(C)C)=O)ccc2c(c1)CCC2NC(c1c[nH]ccc1=O)=O N1(C(c2[n+]([O-])ccc(OC)c2)=O)CCC(C2CCCN(C(c3cnc[nH]3)=O)C2)C1 c1(C(=O)NC(c2ccc(N3CCCCCC3)cc2)C)ccc(S(N)(=O)=O)o1 c1(C(=O)NCCC23CN(C(CCCCC)=O)C(CC2)C3)cc2cnccc2o1 C(C(C)(C)n1cccn1)NC(CN(C(C1CC=CC1)=O)CC)=O N1(C(CSc2n(C(C)C)cnn2)=O)CC(C2CN(C(C3CC3(F)F)=O)C2)C1 C1(C)(CCC=C(C)C)c2nnnn2-c2ccccc2N1.C=C(Cl)COC.C1(C)CC1 CC(C)C(CN(C)C)C(=O)N(C1(CC(=O)NCc2csc(CO)n2)CC1)C Cc1ccc(C(N2CCC(C)(CC(=O)NCC(C)(C)CCO)C2)=O)cc1O N1(CC)CCCC2OCCN(c3nn(C)cc3[N+](=O)[O-])CC12 N1(C(C2(CC)COC2)=O)CCN(C(C2CCOC2)=O)C2COCC12 C1(CC(=O)NCc2c(C(N(CC(F)(F)Cl)C)=O)c[nH]n2)CC2CCC1C2 CCCCCCC(=O)N1CCOCC(NC(=O)CCc2ccsc2Br)C1 c1(NC(CCNC(CC(c2ccc(OC)cc2)C)=O)C)ncc([N+](=O)[O-])c(=N)[nH]1 C1CCCN(NC)CC1.C1(C=O)CC(OCC(=O)NC2CC2)C1.C(COCCO)OC C=CCC(C)(CC)C(=O)N1CC(C(=O)NCCN2CCC2)C(C)(C)C1 C1(NC(C(CNC(Cn2nnc(C)n2)=O)O)=O)CCCN(C)CC1 c1(C(N2CC(O)(CNC(c3cc[n+]([O-])cc3)=O)C2)=O)cc(O)ncc1F Cc1cccc2c(-c3nc(Cn4cncn4)nn3-c3cccnc3)n[nH]c12 S(=O)(=O)(c1cccnc1NC(C)(C)CO)NCc1ccc(CC(C)C)cc1 c1(OC)cc(CNC(=O)N(c2ncc(C=O)s2)C)ccc1C#N C1(O)(CNC(=O)C=CC=C(Cl)Cl)CCCN(C(=O)C(CO)NC(=O)C(F)(F)F)C1 C(CCCCN=C(NCCC1OCCC1(C)C)NC1CCOCC1)N(CC)CC S(=O)(=O)(c1ccc(Br)cc1Cl)NC1CN(Cc2ncc(CC)s2)CC1(F)F c1(C(C(=O)NCC(C)NC(CCc2ccc(OC)nc2)=O)C)ccc(F)c(F)c1 N1(C(=O)Nc2n(Cc3c(F)ncc(C)c3)nc(C)c2Cl)CC2(C)CC1CCO2 c1(C(N2CC(N(C(Cn3c(N)cc(C)n3)=O)C)C2)=O)c[nH]cc(C)c1=O CC(C)(C)C(CNC(=O)CC(F)(F)C(F)F)C(=O)Nn1nnc2c1CCCC2 N(C1CCN(C)c2ccccc21)C(C1CCC(CC)CC1)=O Cc1ccc(F)c(C(N2CCCCC2c2ncc(C)s2)C(=O)NCCC#N)c1 c1(NC(C(=O)NC2CC(N)C(O)C2)=O)cc(Br)c(F)cc1F C1(NC(=O)C(F)C2CCCC2)CCC12CN(C(=O)C=CCCCCCCO)C2 C=CCCC(O)CNC(=O)C(C)(C)C1CCCN1C(=O)C(C)CN(C)C C1(CCC(=O)NCC2CC3(CCC3)C2)CCCCN1C(=O)CC1CCCO1 C12(CCCSC1)CS(=O)(=O)N2.C1(OC)COCC1CC(C)C c1(CC(=O)NC2CC2CNC(=O)CN2CCCC2)nc2ccccc2s1 CC(C)C(CNC(=O)Cc1cnns1)NC(=O)Cc1cnsc1 c1(COC)nc(=N)[nH]cc1C(=O)OC(C)(C)C(C)OC(F)F Cc1[nH]nc(C(=O)NCc2cc(C(=O)NCC3CCCS3)n(C)n2)c1O c1(C(CNC(C2(CN(C)C)CCCC2)=O)NC(CCCSC)=O)ccc(F)cc1 C(=O)(C(C)(C)CF)NC(C1CCC(NC(=O)Cc2ccccc2Br)C1)C C1(NC(CNC(C2CCN(C(=O)OC(C)(C)C)C2)=O)=O)CCc2ccccc2O1 c1(C(=O)NC2(C(N3CCC(CO)CC3)=O)CCCCC2)ccc(C(F)F)cc1F C1(CNC(=O)OC(C)(C)C)CCC2(CC1)CC(NCCC(COC)O)C2 C(=O)(C1CSc2ccccc21)N1CC(CNC(C2Cc3ccccc3CO2)=O)C1 C1(NC(CC)=O)CC2COCC(C1)N2C(=O)C(=O)NCC1(C(C)(C)OC)CC1 C1(CNC(C2CC(CC)OCC2)=O)CCCN(C(=O)CC(C)c2ccco2)CC1 c1(NC(=O)C(N2CCCCC2CC(N)C(F)(F)F)=O)cc(O)c2ccccc2c1 N1(C(COCCC=C)=O)CCC(O)(C(=O)NCc2cn(C3CC3)cn2)CC1 N1(C(N2C3CC(N)CC2CC3)=O)CCc2[nH]c3c(F)cccc3c2C1 C1(C(=O)NC(C(=O)NC)C2CC2)CCC(CNC(c2ccccc2OC)=O)CC1 C(CC(F)F)(C(=O)NC(c1cnsc1)C)NC(COCC)=O N1(C(C2N(C)CC(O)C2)=O)CC(CO)C2(CCN(C(C3(C4CC4)CC3)=O)CC2)C1 c1(NC)ccccc1C(N1CCC(C(C)(C)C(=O)NC(C2CCCC2)CO)C1)=O C1(CN(C(C2CC(CCC)C2)=O)CC)CCN(C(=O)CCc2ccc(C)o2)CC1 C1(C(=O)NCC(C)NC(=O)CCc2cncs2)CC1C1(C)CCOCC1 C1(CNC(C)=O)CN(C(c2ccc(F)c(N)c2)=O)CCC1C CC1=C(C(=O)NC2CC(F)(CNC(c3ccnc(O)c3)=O)C2)CCO1 C1(NC(=O)CCc2ccc(F)cc2)CCCCC1NC(c1nn[nH]c1Cl)=O C1(C)(C(=O)OC)CC(O)CN1C1(CNC(C2CC2C(=O)NCCO)=O)CC1 C1(C(N2CCC(C)(NC(CC(COC)C)=O)CC2)=O)CCCC2(CCOCC2)O1 N1(C(C(CCC)CC2CCCC2)=O)CC(C2CN(C(=O)C(C)O)C2)C1 C1(NC(=O)C=CBr)COC2C(NC(C3(O)CCSC3)=O)COC12 c1(C(C(=O)NCC(C)N(C(=O)C#CC2(C)CC2)C)O)cc(F)cc(F)c1 c1(CC)cc(F)ccc1C(=O)NCC1CN(C(c2cc[nH]c(=N)c2)=O)CCO1 C1(CCNC(=O)NCC(COC)(C)COC)CC(C)CC(C)C1 N1(C(c2cc(CC)no2)=O)CC2CC(NC(c3ccn(C(C)C)c3C)=O)CC1C2 N1(C(C(C)N2CCC2)=O)CCN(C(c2ccc(Cl)c(Cl)c2)=O)CC1C1CCCC1 N1(C(C(CC#C)C2CC2)=O)CCCN(C(=O)C(O)C2CC2)CC1 C12(COC(C(C)(C3CCOCC3)NC(=O)OC(C)(C)C)=O)CCC(CC1)C2.CCO CC1C(C(=O)NCC(C)(CO)CO)CCN1C(=O)Cc1ccc(F)nc1 c1(C(=O)NCCOC(CNC(C2CN(C)C(=O)C2)=O)(C)C)nn(C)c(Cl)c1Cl c1(CC(N2CCC(NC(C=CCCCCC)=O)CC2C)=O)ccc2c(c1)OCO2 c1(C(N2CC(NC(CCOCC)=O)C2)=O)cn(C)nc1C1CCOC1 Cc1cc(CNC(CN(CC(N2C3CN(CC(C)C)C(C3)C2)=O)C)=O)c(O)nn1 CC1CCc2ncc(C(N3CCCN(C(=O)C#CC4CCC4)C(C)C3)=O)n2C1 CC1COCCN1C(C1CCCC(NC(c2ccnc(Cl)c2)=O)C1)=O c1(N)cccc(C(F)(F)F)c1.C(CC)(C1CCNC1=O)C.O=C(CSC)NC CCS(=O)(=O)c1cccc(CNC(=O)NCc2cc(F)c(F)c(F)c2F)c1 N1(C(C2C(C)(C)CCO2)=O)CCCCCCC1C(=O)NCc1ncc(CO)o1 Cc1ccc(C(=O)NCCCC2(NC(c3cc(C4CC4)[nH]n3)=O)CC2)cc1C CC1CC(N=c2[nH]c(Cl)ncc2Cl)CN1C(=O)Cn1nnc(-c2ccsc2)n1 C1(F)(C(=O)NC2CCC2O)CCC(C(=O)O)C1 c1(C(=O)NCCOC(CNC(C(C)=CC)=O)(C)C)ccc(CSC)cc1 N1(C(CCCOC(C)=O)=O)CCC(O)C(NC(=O)C(C2CCCCCCC2)O)C1 Cc1cc(NC(C2CN(C(C3(C#N)CC3)=O)CC2(F)F)=O)c(O)cc1F N1(C(C23CCN(C(c4c(C)ncs4)=O)CC2C3)=O)CCC(S(=O)(=O)C(C)C)CC1 C(N=c1cc(C)n(C)[nH]1)(c1ccc([N+](=O)[O-])c(C)c1)c1n(CCOC)nnn1 C12(CNC(CC(CC)C)=O)CCC(NC(c3ccc(F)cc3C)=O)(CO1)C2 C(=O)(CCCC(CC)NC(c1ccccc1F)=O)NC1CCN(CC=C)CC1 N1(C(c2n(CC)ccc2)=O)CCCCC1C(C)NC(=O)Cc1ccns1 c1(C(N2CCC(C(C)NC(c3cnc(=N)[nH]c3)=O)CC2)=O)ccc2[nH]ccc2n1 c1(C(=O)NCC(CC)(CC)NC(=O)CNC=O)cc(Cl)c(F)cc1F N1(C(CCC(=C)Cl)=O)CCC(C2CC2)(CNC(c2cnc(-c3cccs3)o2)=O)C1 c1(CCC)ccc(C(=O)NCCC(C)NC(=O)C(C)(C)C2CCOC2)cc1 C1(CC(=O)NCC2CCN(CC)C2)CCN(C(c2ccnn2CC)=O)C1(C)C c1(C2(CNC(N3CCCC(C(N)=O)C3)=O)CC2)ccc(Cl)cc1F C1(CNC(c2c(CC(N)=O)occ2)=O)CCCN(C(C2CCSCC2)=O)C1 Cn1ncc2cc(NC(C3(C)CCCN(Cc4cccc(O)c4Cl)C3)=O)ccc12 Cc1noc(C)c1C(=O)NCCN(C(=O)C(C)N1CCC1)CC1CC1 C1(NC(CNC(C)=O)=O)CCN(c2cc(F)ncn2)CC12CCC2 C1(C(=O)NC(CC)CNC(C23COCC2C3)=O)CC2(CSC2)C1 c1(C(N(CC2N(C(CCCCOCC)=O)CCC2)CC)=O)cccc(N)c1CC Cc1ccc(C(N2C3CCC2CN(C(C2(O)CCSC2)=O)C3)=O)cc1C#N C1(CC)CCN(C(=O)Cc2ccc(F)cc2)C1CNC(c1cncc(NC)c1)=O N(C1c2ccccc2CC1NC(=O)C(F)(F)CO)C(Cc1cnc(C)s1)=O C1(CNC(C(c2ccccc2Br)(C)C)=O)COCCN1C(=O)COCCF Cc1nn(C)c2ncc(C(=O)NC(C)CCCCNC(c3cnoc3)=O)cc12 c1(C(=O)NC(CNC(COCCCC#C)=O)(C)C)cc(C)c(S(N)(=O)=O)cn1 c1(CNS(CCSCCOC)(=O)=O)ccnc2cc(C(F)(F)F)ccc12 CC1=C(C)CC(C)(NS(NC(c2ccccc2)=O)(=O)=O)CC1 Cc1cc(N2CCC(C3CC3)C2)nc(=NC(C)CS(C)(=O)=O)[nH]1 C1(CCC)(C(=O)NC(C)C(=O)N(C(C)C(=O)N(C)C)C)CCC1 Cc1ccc(C(C)C(=O)NCC2CN(C(=O)C(c3ccnn3C)C)C2)s1 C1(CC(=O)NC2C(CC(=O)NCC3CN(CC)C3)C2)CCOCC1 c1(C(N(C)CC2N(C(COCCC)=O)CCOC2)=O)ccc(Cl)cc1[N+](=O)[O-] C1(NC(C(C)SC(C)C)=O)CCN(C(C2CCC(C(N)=O)CC2)=O)CC1 C1(OC)CCCCC1C(=O)NCc1nc(C)c(C(=O)NC(c2noc(C)n2)C)o1 c1(C(=O)NCC(C)CN(C)C(c2n[nH]cc2Cl)=O)cncc2ncccc12 N1(C(c2ccc(C(C)(F)F)nc2)=O)CC2(CC(S(C)(=O)=O)C2)C1 Cc1cc(C(=O)NC2CC3CCC2(C(=O)NCCN(C)C2CC2)C3)ccc1O CC(C)CN=C(NCC1=NOC2COCC12)NC1CCNC(=O)C1 C1(CNC(c2nc(C)nc(O)c2)=O)CCN(C2CCCc3ccc(F)cc32)C1 C1(NC(CN(C(C)C)C)=O)CCCC(CN(C)C(C23CSCC2C3)=O)C1 C=CC(C)C(C)C(=O)N(CCCNC(c1ccc(C(=O)OC(C)(C)C)s1)=O)CC N1(C(C(CC(F)F)N(C(CC(C)C)=O)C)=O)CCOC(C)(C)C1C C(=O)(CC(C)C(C)C(C)C)N(CCNC(C1=C(C)CCC1)=O)Cc1ccccc1 N1(C(C2(C(=O)OCC)CC2)=O)CC2CC1CN(C(=O)CCc1cc(Cl)cs1)C2 C1(NC(=O)C=CBr)CN(C(c2ncccc2C(F)F)=O)CC1O C1(NC(CCOCC#C)=O)CC2CC1CN(C(=O)CCC1CCCN(C)C1)C2 C1(NC(=O)CCC2=CCCCC2)CC2(CCN(C(=O)COCC(F)F)CC2)C1 C(=O)(C(C)CCCCCC)NC(CNC(c1cccc(OCCC)c1)=O)CC c1(OC(CC)C)cc(C(N2CCC(NC(c3conc3CC)=O)CC2)=O)ccn1 CCCC(CCCNC(=O)CC1(N2CCCC2)COC1)NC(=O)CCS(C)=O Cn1ccc(CC(=O)C(CONC(C2CC(CC(C)(C)C)C2)=O)=O)n1.N C1(CCC(=O)NC(CNC(COCCOCC#C)=O)CC)CCC(=O)NC1 c1(C(N(CC(O)CN(C)C(c2cnc(Cl)s2)=O)C)=O)ccnn1C1CCCC1 C(=O)(C(F)(F)C1=CCOCC1)NC1CC(CNC(C2CC3C=CC2C3)=O)C1 Cc1c(Br)noc1C(=O)NCC1(CN(C)C(C23CCC(C2)C3)=O)CC1 C1(NC(C2(C)CCNC2=O)=O)CC2CCC1C(NC(=O)COCC1(F)CC1)C2 CC(C)CC(CC(C)C)C(=O)NC(CNC(c1nc(Cl)c(Cl)s1)=O)C(C)(C)C n1(CCC)nc(C)cc1C(=O)NC(C)C(C)NC(=O)CC1(OC)CCOCC1 CCCC(CC)C(=O)NC(C)(CC)CC(=O)NC(COCC)CC CC1(C(N2CC(C(F)(F)F)C2)=O)CC(O)CN1C(c1ccc(Cl)cn1)=O C1(NC(=O)C=CCN2CCCC2)CCCN(C(c2c[nH]nc2C(F)F)=O)CC1 c1(C(=O)NCC(c2ccccc2F)NC(C(C)(C)F)=O)cc(NC2CC2)nc(Cl)c1 C12(CNC(C3(C)CCCO3)=O)CCC(CNC(=O)CC3CC34CC4)(CC1)CO2 N1(C(C2CC(SC)C2)=O)CC2CCC1C(CNC(c1ncsc1C)=O)C2 N1(C(CCCc2onc(CC)n2)=O)CCCC(CN(C)CCc2ccon2)C1 N1(C(c2ccc(SC)cc2)=O)CCC(CC(=O)Nc2cc(Cl)ccc2F)C(O)C1 c1(C(=O)NC2CCN(C(CCCCCC)=O)CC2C)cc(F)cc(S(N)(=O)=O)c1 S(=O)(=O)(c1ccc(=NCCc2ccc(OC)cc2)[nH]c1)NC1(CC)CC1 C1(CC=C)(NC(=O)CCC2OCCO2)CCOC1.C1=CC(=O)NC1(C)C N1(C(CNC=O)=O)CCCC2(CC(NC(C34CCCC(CO3)C4)=O)C2)C1 N1(C(C(C)OCC)=O)CCC(CCCNC(=O)C(C)(O)Cc2ccccc2)CC1 c1(C(=O)NCC(C)(C)OCCNC(C2CCCC2(F)F)=O)ccc(F)c(Cl)c1F Cn1nnc(C(=O)NCCC2CN(C(=O)C(F)(F)C3(O)CCC3)CCO2)c1N N1(C(c2c(C)c(N)n(C)n2)=O)CC2CN(C(c3sccc3C3CC3)=O)CC2C1 C1(F)(CNC(c2c(C(C)C)con2)=O)COCCN(C(=O)C(C)CC(C)(C)C)C1 c1(CC)ccc(F)c(C(=O)N(CC)CC2CCCN2C(=O)CC(C)C(F)F)c1 N1(C(C(c2cccc(Cl)c2)C)=O)CCN(C(=O)Cn2cnc(C(N)=O)n2)CCC1C C1(O)(COC)CCCN(C(C)=O)C1.C1(c2nnnn2C2CC2)CC(C2CC2)N1 N1(C(c2cnn(C3CC3)c2)C(=O)NCCC2CC2)CCSCC1C1CCCCC1 CCC(CC(=O)NCc1nc(C(=O)NCCc2cc(C)n(C)n2)c(C)o1)OC CC1CCC(NC(=O)Cc2cc(Cl)ccc2Br)CN1C(=O)CNC(N)=O c1(CC(=O)NCCCN(C(c2occc2Cl)=O)C2CC2)cccc2cccnc12 O=C(CN=c1cc[nH]cc1)NCC1OCCC1C(N1Cc2ncsc2C1)=O CCC(CCOC)C(=O)N1CCOCC(CNC(c2conc2C2CCC2)=O)C1 C12(CNC(C(C)(O)C3CCC3)=O)CC(CN1C(=O)C(C)(C)n1cnnn1)C2 C(=O)(N=c1c(Br)c[nH]cc1Br)C1N(C(c2ccc(C)c(Cl)c2F)=O)CC(O)C1 c1(C(N2CC(C(N(C3CCN(C(N)=O)C3)C)=O)OCC2)=O)noc2c1COCC2 CC1(CC(=O)NCC2(O)CCOC2)CCN(C(c2cn(C3CC3)cn2)=O)C1 C1(C(=O)NCc2cncs2)(CNC(C2N(CCC)CCC2)=O)CC12CCC2 c1(C(N2CC(C)N(C(=O)C=Cc3ccoc3)CCC2)=O)cc2c(n1C)CCOC2 CCCCC(CNC(=O)C1=CCN(C(c2cnnc(C)c2)=O)CC1)CCC Cc1nccn1CCC(=O)NC(CO)C(=O)NC(c1ccco1)C c1(C(N(CCNC(c2c(OC)ncc(CC)c2)=O)C)=O)cc(Cl)c(Cl)cc1N c1(NC(N2C(C)CC(CC(=O)OC)C2)=O)ccc2c(c1)C(=O)NCC2 c1(CS(CCc2c(C)ncs2)=O)cccc(-n2cccn2)n1 c1(N2C(CC#N)CN(C(C3CCSCC3)=O)CC2)ncnc2cccnc12 C1(NC(C(C=C)O)=O)CCC2(CC1)CN(C(c1csc(Cl)c1OC)=O)CCO2 c1(CN(CCCC)C)n[nH]c(C2CNC2)n1 c1(C(=O)NC(CC(C)NC(c2cn(CCC3CC3)nn2)=O)C)ccc(Cl)c(F)c1 CC1OCCCC1C(=O)NC1(C)CCN(C(=O)CCC2CCC(=O)NC2)C1 N1(C(C)=O)CC2CC2(CO)C1.c1(CN(C(C)C(=O)O)C=O)coc(Cl)n1 CCCCC(O)C(C)C(=O)NC1CN(C(=O)OC(C)(C)C)CC1(C)C c1(OC)nc(=NCC2CCCCN(C(=O)C(C)C)C2)cc[nH]1.C(=O)OC c1(NC(c2ccc(CS(C)(=O)=O)o2)=O)cccc(F)c1C(F)F Cc1cc(C)nc(SCC(N2CCN(C(c3cccnc3)=O)C(C)C2)=O)n1 CCC(C)CCC(=O)N1CC(NC(=O)CNC(=O)C(O)c2ccco2)C1 C(CCCCCC(=O)NC(c1ncc[nH]1)CO)NC(c1ccc(C)nc1C)=O c1(C(C)=O)cc(C(=O)NC(Cn2cncn2)C(=O)N2CCC2C(=O)N(C)C)no1 C1(C(N2CC(CC(C)C)OCC2)=O)CC(C)CCN1C(=O)C(O)C1CC1 CC1CC(C)(C(=O)NCC(C)CNC(C2CCCC(C)(C)O2)=O)CCO1 C(C(=O)N1CCOC(CNC(c2cn(C)cc2C)=O)C1)(C(C)C)SC c1(C(=O)NC(CC)(CNC(=O)C(Cl)=CCl)CC)ccc(N)c2ncccc12 n1(CCC)ccc(=NC(=O)C=C(C)CNC(c2cc(CO)c(C)o2)=O)[nH]1 N1(C(C(C)C(F)F)=O)CC2CCCN(C(=O)CC(F)(F)F)C2C1 C12(CNC(c3cccc(C(F)(F)F)n3)=O)CCC(CC1)N2C(c1ccon1)=O C1(CC(N2CC3CCC(C2)N3C(C2CC(C(F)F)C2)=O)=O)CCCCC12CC2 C1(NC(CC)C(=O)NC(C)C)CCC(C(N)=O)CC1 c1(C(=O)NC2C(NC(CCC3(C)CC3)=O)C2)nc2ccccc2cc1C1CC1 N1(C(C2CC(C)SCC2)=O)CCC(NC(c2cccc(N)c2)=O)C(CO)C1 C1(C)(CCC(=O)NCC(C)OC(F)F)CCCN1C(=O)Cc1ccsn1 N1(C(C(C=C=C)C)=O)CCC2(C(=O)NC(c3cnn(C)c3)CC)CCCC12 Cc1ccc(-c2noc(-c3csc(-c4[nH]cnc4C)n3)n2)c(C#N)c1 CC1CC=C(C(=O)NC2(C3CC3)CCN(C(=O)Cc3csnn3)C2)CC1 N1(C(C(C)(F)F)=O)CC2(CC(NC(=O)C(CO)c3ccccc3)C2)C1 c1(C(=O)NCC2N(C(c3ccc(CC)nc3)=O)CCOC2)ccc2ocnc2c1 C1(NC(c2nn(C)c(Cl)c2)=O)CCC12CCN(C(=O)C=C1CCOCC1)CC2 Cc1ccc2nc(N3CCCC4(NC(C5CCC6CC6C5)=O)CCCC34)sc2n1 C#CCCCCCC(=O)N1CCOCC1C1(NC(=O)CN2CCC(=O)NC2=O)CC1 c1(N(C(C(n2ccnc2-c2ccccc2)C)=O)C2CC2)cnc2c(O)cccc2c1 C1(CC)C(C(=O)NCCCOCC(F)F)CCN1C(c1cnc(C)cn1)=O c1(C(=O)Nc2ccc(NC(C(C)OC)=O)cc2C)c(C)nc2ccc(Br)cn12 N1(C(c2cc(C)[nH]n2)=O)CCN(C(=O)Cc2ccccc2Cl)C(C)CC1C C1(C2CC2)(CNC(C(C)c2ccsc2)=O)CCN(C(C2CC(F)C2)=O)C1 C1(CC)CCc2sc(C(=O)NC3CCCN(Cc4cn(C5CC5)nn4)C3)cc2C1 CCC(CC1CCCC1)C(=O)NC1(Cc2ncc(C)s2)CCO1 S(=O)(=O)(c1cc(F)cc(Br)c1)NC1C(C)CN(Cc2cc(C3CC3)on2)C1 C(=O)(C(C)C(C)O)N(C1CCN(C(c2ccnn2C2CC2(F)F)=O)CC1)CC Cc1cc(C(N2CCCC(C(C)Nc3cc(O)ncn3)C2)=O)nc(C)n1 C1(NC(C2N(CC)CCC2)=O)COCCN(C(=O)C(C2(O)CCCCC2)(F)F)C1 c1(C(=O)NC2CC(CNC(=O)C(F)C(F)(F)F)C(O)C2)csc([N+](=O)[O-])c1 Cc1ccc(C#N)cc1NC(=O)CNC(C1CCCC(F)C1)=O CCCCC(CC)CC(=O)N1CCCC1Cc1cn(C2CCCC2O)nn1 C1(CS(=O)(=O)N2CCCC2)CCCS1(=O)=O.c1(CC(CN)CO)ccc(Cl)cc1 c1(C(=O)NC2(CNC(CCCC(C)=O)=O)CC2)cnc2ncnn2c1N c1(C(=O)NCCC2N(C(C3COC(=O)O3)=O)CCSC2)ccc2sccc2c1 c1(C(NOCC=CC)=O)c(OCC)cccc1C.C1(=O)CC(CC)N1 C(=O)(C(C)CC(=O)N1CC(C(=O)NC(CC2CC2)CC2CC2)C(F)(F)C1)OC N1(C(CN(C2CC2)CC)=O)CCC(CNC(c2c(C)csc2C)=O)C(C)C1 N1(C(c2cc(CC)[nH]n2)=O)CCC2CCN(C(=O)CCc3cccs3)CC2C1 C=C=CCCC(=O)NCCC(C)(C)CNC(=O)C(C)C(=O)OC Nc1ccc(C(=O)NC2CN(C(=O)CO)CC2n2ccnn2)cc1O c1(C(=O)NCCCC(C)NC(c2nc(Cl)sc2Cl)=O)ccc(-c2cnc[nH]2)cc1 S(=O)(=O)(c1ccccc1Cl)NCCCNC(=O)Cc1ccc(F)cc1F C1(CC(N2CCC(N(C)C(c3cnc(S)nc3)=O)C2)=O)CN2CCN1CC2 C12CCN(CC1)C(=O)CCC2C.C1(CN(C(C(F)OC)=O)C2CC2)CCOC1 c1(CNC)cccc(-c2ccnc(C(=O)Nc3nc(O)cs3)c2)c1 Cc1noc(C)c1S(=O)(=O)NCC(=O)Nc1n[nH]c2ccc(C(F)(F)F)nc12 n1(CC(=O)N(C2CN(C(=O)CCCN(C)C)CC2O)C)ncc(O)nc1=O c1(SC)nccc(N2CCC(C3CCCN(C(c4cnc(C(C)O)s4)=O)C3)C2)n1 C1(C(=O)NC2CCC(CC(=O)N(CC=C)CC=C)C2)NC(=O)OC1(C)C CN1CC=CCC1CC(=O)NC1(C)CC(NC(C2(F)CC=CC2)=O)C1 Cc1nc(CC(C)C)oc1C(=O)NCC1CN(C(=O)CCc2cncs2)CC1C N1(CC=C)CCC(NC(C2COC(CNC(C3CCCN3C(N)=O)=O)C2)=O)CC1 C1(C(=O)NC2CC(CNC(C3CCN4CCCC4C3)=O)C2)CCC([N+](=O)[O-])CC1 C1(C(=O)NCC(C)(O)CNC(=O)Cc2ccccc2)(OC)CCSCC1 C1(CCCOCCN(C)C)CN(C(C2CN(C(C)=O)C2)=O)CCO1.C(=O)(CC)N.OCCC c1(OC)cc(CCC(=O)NCCNC(C23CCC(F)(CC2)C3)=O)cnc1Br c1(OC(C(=O)NC(C)CCNC(C2(C)CCCCC2)=O)C)ccc(C#N)cc1 C1(O)(CN(C(=O)CC(C)n2cccn2)C)CCN(C(=O)C(C)(C)CF)C1 c1(N(C(C)C)C)ccc(C(=O)NCC(CO)NC(C2(C(F)F)CCCO2)=O)cc1 C1(C(N2CCC(F)(CO)C2)=O)(OC)CCN(C(c2ccccc2CC#N)=O)CC1 C(CC(=O)NNc1cccc(Br)c1F)c1c(C)cccc1 N1(C(C2C(C=C)CC2)=O)CCN(C(c2cc(CC)cc(Cl)c2)=O)CC(O)C1 CC1C(NC(C2COC(C)(C)O2)=O)CCCN1C(=O)CCc1cccc(Cl)c1 c1(C(N2CCC(N3CCN(C(C=CSC)=O)CC3)CC2)=O)cccc2c1OCC2 c1(NCO)ncc2c(n1)CCOC2.C12(COC1)C(=O)CCO2.C(CCNC(N)=O)O C1(CNC(Cc2ncc(CC)[nH]2)=O)CC2CCC1N2C(=O)Cc1cc[nH]c1 O=C(C(CCC1CCC1)NC(C1CCOC1)=O)NC1CC(F)C1 CCCC(O)CC(=O)N1CCN(C(c2ccc(OC)cc2Cl)=O)C(CCO)C1 Cc1c(N2CCC(NC(=O)Cc3cnn(C(C)(C)C)c3)C(F)C2)ncnc1Cl c1(C(N2CC(OCCC(=O)NC3CC3)C2)=O)cnc2sccn12.C12(CC1)CN2 C1(CN)CC2(CC(NC(c3scnc3C(C(CC=CCC)=O)CC)=O)C2)C1 N1(C(Cc2nnc(C)o2)=O)CC(C)C(NC(c2ncc3ccccn23)=O)C(C)C1 C1(C(=O)NCC=CCCCCC)CC2CCC1N2C(=O)CC=CC(=O)O c1(OC)cc(C)ccc1NC(N1CCC(NC(=S)NC(C)C)C1)=O CC1CC(C(=O)N(CCCN(C(=O)Cn2ccc(C(F)F)n2)C)C)=NO1 C1(CN(C)C)CCC2(CC1)CN(C(C1CC1)=O)CCO2.C1(C)C(=O)N1.C(C)(=O)OC C1(Nc2nccc(SC)n2)CN(C(=O)CCc2cnn(C)c2)CCC1C.C1(=O)CN1 NS(=O)(=O)C1(C(=O)NCCC2CCC(NC(=O)Cn3cc(Br)cn3)C2)CC1 C1(C(=O)NC2(CNC(CCC(C)(C)F)=O)CCOC2)CCS(=O)(=O)C12CCC2 C(C(C(=O)NCC1CNC(=O)C1)C(C)(C)C)NC(c1cnc(CC)s1)=O C1(C(=O)NCC(CC)NC(=O)Cn2nnnc2C2CCOCC2)(CC)CC1(F)F c1(C(=O)NC2CN(C(C3CC(OC)C(OC)C3)=O)C(C)C2)cnc2cc[nH]c2c1 c1(C(=O)NCCN(C2CCN(C)C2=O)CC)cc(C)c(Br)s1 CC(F)CC(=O)N1CCC(C(C)NC(=O)CC2CC(F)(F)C2)C1 Cc1nc(C(C)NC(C2CN(C(=O)C(C(C)C)N(C)C)CC2F)=O)c(C)o1 c1(C(N(CCC(C(C)C)NC(C=CCOC)=O)C)=O)cc(C)ccc1C C1(NC(c2cccnc2)=O)CCCN(C(C2CC2c2cccnc2)=O)CCC1 C1(NC(c2c(C)cccc2Cl)=O)CCC2(CCCN(C(=O)CC#N)C2)C1 c1(C(=O)NCC(CNC(C2CCCN(CC)C2)=O)F)cc(F)c(F)cc1F N1(C(c2ccc(OC)nc2)=O)CC(OC)CC(NC(c2cnc(SC)n2C)=O)C1 C1(C(N2CC(C)(COC)C2)=O)CCN(C(C2CC(C(C)C)=NO2)=O)CC1(C)C N1(C(c2c(CNC(C3(CC)CC3)=O)ccs2)=O)CCCN(C)CC1C C1(C(=O)NC2CC(C(=O)OC)C2)(NC(=O)N(C)C)CCCC1C.C1CO1 C(C(COC)C(=O)NC1(F)CCN(C(=O)COc2cc(C)on2)C1)OC COn1cnc(C)c1C(N1CC(OC)C(C(=O)NC2CCCC2CN(C)C)C1)=O C(=O)(C(O)C(F)(F)F)NC(C)CC(=O)NCCC1CCCC1 C(=O)(CCC(=O)OC(C)(C)C)N1CC(N(C(=O)C(F)n2ccnc2)C)C1 c1(CC)ncccc1C(=O)NC1CCC(C)(CNC(C2CC(=C(F)F)C2)=O)C1 c1(C(=O)NC2C(NC(c3nc(NC(C)=O)sc3)=O)CC2)cc(C)c(C)nn1 C1(N(C(=O)Cc2ccco2)C)CCCN(C(=O)CCc2ccccc2)C1 C(CC(C)C)(C(=O)NCC1(CSC)CC1)N(C(CC=CC)=O)C CC(C)C(F)(F)CC(=O)NCCC(C)N(C)C(C1CCCCC1(F)F)=O N1(C(C2SC3C=CC2CC3)=O)CCC2OCCN(C(c3cccc[n+]3[O-])=O)C2C1 c1(-n2cc(-c3cc(=NC)[nH]cc3)nn2)ccc2c(c1)N(C)CCC2 N1(C(CCN(CCCCC)C)=O)CCN(C(=O)C(N2CCSCC2)C)CC1C N1(C(c2n[nH]cc2C(F)F)=O)CCOC(c2cn(CCC3CCOC3=O)nn2)C1 CCC(C)(C)C(O)C(=O)N1CC2CCCC2(C(N2CC(N3CC(F)C3)C2)=O)C1 c1(CCC(=O)NCC(F)CNC(c2cccc(O)c2F)=O)ccc(O)c(F)c1 c12ccc(c(Br)c1)-c1nnnn1CCCC(=O)N2.C1(OC)(CO)CCNCC1.C(C)(C)O c1(OC(C)C)ccc(C(N2CCC(N(C(=O)CC(C)(C)O)C)C2)=O)nn1 c1(C(=O)NC2CCCC2)cccc(-c2nnco2)c1.c12cnc(s1)[nH]c2=O c1(C(=O)NC2CN(C(Cc3ccc(N)cn3)=O)C2)cc2c(nc1O)CCSC2 O=C1C(CN2CCCC2)CCN1c1cccc(Br)c1.N12CCCC1NC2=O N1(C(c2c(C)c[nH]n2)C(=O)NCSc2ccccc2)CCCC1C1Cc2ccccc21 n1(CCNC(=O)CC2(Cc3c(C)nco3)CCSC2)cc(C2CC2CO)nn1 c1(C(=O)NC2C(CNC(=O)CCC3OCCO3)CC2)cccc(Cl)c1F C(=O)(C1=C2CCCN=C2NN1)NCCC(C)N(C(=O)Cc1ccc(Cl)nc1)C Cc1c(F)ccc(CNC(=O)C(CCN(C)C)NC(=O)C(O)C2CCC2)c1F CCCC(CC(=O)N1CCN(CCO)CC1)NC(=O)CN1CCCCC1C N1(CC)C(=O)c2ccccc2N2C(=O)CCC12C(=O)OCc1sc(Br)cc1OC c1(C(N2CC(COC)(NC(c3ccc(O)cc3F)=O)C2)=O)ccc(C)c(Cl)c1F C1(CNC(C2(C#C)CCC2)=O)CCC2(CO1)CC(NC(=O)C(F)CC(C)C)C2 C(=O)(CCCCN1CCOCC1)NC(C)(CNC(=O)C(F)(F)OC(C)(C)C)CO Cc1cc(C#N)cnc1C(N1CC(C)(NC(C2CC2(C)Br)=O)C1)=O C1(C(N2CC(C(N(C)C)=O)C(N(C3CCCC3O)C)C2)=O)CC2(CCO1)CC2 N1(C(CCC(=C)C)=O)CCC2CCN(C(=O)Cc3cc4ccccc4s3)CC2C1 N1(CC)CCCC(C(N2CC(N(C)C(c3ncccc3O)=O)C2)=O)C1 CCCCCC(F)C(=O)NC1CC(N(C)C(c2ccc(CO)cc2)=O)C1 C1(C(=O)NC(CC)C)C(NC(c2csnc2C)=O)C1(C)C Cc1scc(C(=O)N(CC(C)NC(C2CCN(C(N)=O)CC2)=O)C)c1N Cc1ncccc1C=CC(=O)NC1(C)CCC(NC(C2(C)C=CCC2)=O)CC1 c1(C(N(CCCNC(c2cc(C)sc2)=O)C(C)C)=O)nc(C(F)(F)F)oc1C N1(C(c2c(Cl)cc(C)nc2)=O)CC2CC(O)C1C2NC(=O)CCCCCN(C)C Cc1c(C(N2CCC(N(C)C(c3ccc(CCF)cc3)=O)C2)=O)cnn1CCO O=C1Nc2ccccc2C1C1CCN(c2ncnc3cc(Br)ccc23)CC1 N1(C(C2(CC)CCC2)=O)CCC(CN(C(C2CCCCO2)=O)CC2CC2)CC1 C1(NC(CCC(C)SC)=O)CCCN(C(=O)CC2(C)CC(F)(F)C2)CC1 CCC(CC(F)(F)F)C(=O)NC(CNC(c1ccnc2ncnn12)=O)C(C)(C)C C1(C(N2CC(C)CC(NC(COCCOC)=O)C2)=O)C2(CCC2)C12CCC2 c1(NC(=O)NC(c2nc(C3CC3)cs2)(CC)C)cnc(C(C)C)nc1 N1(C(c2c(C)nns2)=O)CC2CCCC1(CNC(c1cnn(C)c1)=O)C2 CCC(C)CCC(=O)N(CC(C)O)CCNC(C1CC12CC2)=O N1(Cc2scc(C)c2)CCN(c2ccc(OCCCO)cc2)CC1 c1(C(N2CCC(CNC(C(C(C)C)O)=O)(CO)CC2)=O)cc(Br)c(F)c(F)c1F c1(C(=O)NCC(CC)NC(c2c(C)cc[nH]c2=N)=O)ccc2nc(O)n(C)c2c1 Cc1cc(F)cnc1C(=O)NCC1(NC(=O)COCCN(C)C)CCC1 c1(CC(C)NC(=O)NCC(c2ccc(Cl)cc2)C)ccc(N)c(F)c1 N1(C(C(CC(C)C)OC)=O)CC2C3CCC(C2C1)N(C(=O)C1=CCCS1)C3 C1(N(C(=O)COC2CC=CC2)CC)CCCN(C(=O)C=Cc2ccc(Cl)s2)C1 C(=O)(C(CCC(C)C)N(C)C)NC(CCC#C)C(=O)NCCCOCCC(F)(F)F C1(CN(C(CCSC)=O)C)CC2(CCN(c3ccnc(C(N)=O)n3)C2)CO1 N1(C(c2n(CCC)ncc2)=O)CCCCC1CNC(c1nn(C)cc1N)=O C1(CNC(c2c(CC)cccc2)=O)CN(C(=O)COC2CCCOC2)CC12CC2 Cc1[nH]nc2c1CC(C(=O)NC(C)(C)CCNC(C1CCN1S(C)(=O)=O)=O)CC2 C(=O)(CCP(C)(C)=O)NCC(CC)NC(C1(N(C)C)CCCOC1)=O CC(C)C(O)C(=O)N1CCC(C(F)C(=O)NCCC23CC(CCO2)C3)C1 N1(C(CC2CCC(C)C2)=O)CCCN(C(c2cnc(F)c(F)c2)=O)C(C)C1 C1(C(N(CCCC=C)C)=O)CN(C)CCN1C(c1cc(F)n(C)n1)=O C1(C(C(=O)NCC(=C)C)N(C2CCCCC2)CCN(C)C)C2CCOCC12 CC1CC(C)N(n2c(-c3nc(C4(C(F)(F)F)CCCC4)sc3)ccn2)C(C)C1 C1(NC(c2n(CC)cc(Cl)c2)=O)CN(C(C2CC2OC)=O)C2(CCCCCC2)C1 C1(C)(C=CC)CC=CCC1.C1(O)(C2C(=O)N2)CCCCC1.C12(CCC1)CC(=O)N2C CCC(C)C(O)C(=O)NC1CC(CNC(c2cc(OCC)ns2)=O)C1 c1(C(=O)NC2C(NC(C3CC(C)(C)OCC3)=O)CC2)ncc(F)c2ccccc12 c1(OC)cc(CN2CCC(NC(C3CCN(C)CC3)=O)C(O)C2)c(Cl)cn1 C1(NC(C(C)NC(N)=O)=O)CN(C(c2sccc2OC(F)F)=O)CC(F)(F)C1 n1(CCOC)cc(C(=O)NCC(O)CN(C)C(C2CN(C)C(=O)N2)=O)ccc1=O N1(CC23CC(C(=O)NC(CC#N)=O)(C2)C3)CCCCC1C#N c1(CCC)cc(C(=O)N(C(C)CN(C)C(C)=O)C(C)C)n(C)n1 Cn1cncc1C(=O)NCC(CO)NC(=O)CN1CCNC1=O CC12CCC(C(N3CCCC3CNC(=O)C(C)(C)Cc3cnn[nH]3)=O)(CC1)CO2 c1(C(C)N(C)C(c2cnn(C(F)(F)F)c2)=O)cn(Cc2ccc(C(N)=O)o2)nn1 CC1(C)CCCOC1CC(N1CC2C=CC1C(C(N1CCC1CO)=O)C2)=O C1(NC(CC(C)CN(C)C)=O)CN(C(c2ccncc2)=O)CCC12CCOCC2 Cc1cc(S(N)(=O)=O)sc1CN1CCOC(C(=O)NC)C1 C1(C(=O)NCC2(NC(C(C(CC)O)(F)F)=O)CC2)Cc2ccccc2N(C)C1=O CCCCCC(O)CC(=O)NCC1C2CN(C(=O)Cn3c(C)csc3=O)CC12 Cc1cncc(C=CC(=O)N(C(C)CN(C)C(C2CCN(CC(C)C)C2)=O)C)c1 c1(C(=O)NC2C(C(=O)NC(C#C)C(C)OC)CC2)nc(=N)cc[nH]1 c1(CC)nc(Cl)c(F)c(=NC(C)CNC(=O)COC2CCC(C)CC2)[nH]1 CCCC(C(O)C(=O)Nc1cccc(C(C)F)c1)NC(=O)CCCn1ccnc1 CN1C(C(N2C3CCC2(CNC(C24CCCC2C4(F)F)=O)CC3)=O)CCS1(=O)=O CC(C)C(O)CC(=O)N1CC(F)(F)CC1CCNC(c1ccnn1C1CCC1)=O C(=O)(CC(C)C(C)C(C)C)N1CCCC2(NC(C(C)CCO)=O)C(C1)C2 Cc1nc(CCO)oc1C(=O)N(C(C)(C)C)CC=CC(N1CCCC1(C)CO)=O CC1(C#CC(=O)N2CCC(CO)(CNC(C3CC4(C3)CC4F)=O)CC2)CCCO1 C1(C(N2CCC(N(C(=O)C(O)C(C)(C)C)CC#C)C2)=O)CC(=O)NC1(C)C CC(C)C(F)(CNC(=O)C(C)NC=O)C(=O)N1CCC(O)C(C)(O)C1 Cn1nc(C(N2CC(CNC(C3CC3F)=O)C3(CC3)C2)=O)c(Br)c1Cl CCC(C)(C)C(O)C(=O)NCC(C(=O)NCCCn1ccnn1)C(C)C CCCC(C(=O)N(C)C(c1ccncc1)C)NC(=O)OC(C)(C)C.C1CN1 c1(C(=O)NCCC2CCCCN2C(=O)CCOCC2CC2)cnn2cccnc12 c1(C(=O)NCC2(NC(C3C(OC)CC3)=O)CCC2)cnc(C)o1 C1(C(=O)NCC=CC(=O)NCCNC)CC1(C)C(C)C c1(C(N2CC(CCO)(NC(C(CC)=CCCC)=O)C2)=O)cccc(F)c1C C=CCC(C)(CC)C(=O)N(CCC(=O)N1CC(=O)OCC1(C)C)OC C12(NC(C(C)(F)F)=O)CCC(CN(C(=O)C(C)(C)c3cncs3)C1)C2 c1(CCNC(C(CO)NC(C(C2CCCCC2)C)=O)=O)ccc(O)nc1 N1(C(CN2C(=O)NCC2)=O)CCC2(NC(c3ccc(Cl)c(F)c3)=O)CCCC12 Cc1cncc(C(N2CCCCC2C2CCCN(C(=O)CO)C2)=O)n1 Cc1c(C(N2CC(NC(=O)Cc3cnc[nH]3)C(F)C2)=O)ccc(F)c1F c1(NCCOC(C)C)cc(N2CCC(c3cnccn3)C2)nc(C(C)C)n1 c1(OC)cc(Cl)c(Cl)cc1CC(=O)NC1CN(C(c2ccc(C)cc2)=O)CC1F C1(NC(c2cccc(C3C(=O)CCC3)c2)=O)CNCC12CCOCC2 C1(N(C)C)CCC(NC(c2cscc2NC(=O)Cc2cc(C3CC3)no2)=O)C1 S(=O)(=O)(c1c[nH]c(C(=O)NC(C)CNC(=O)C(C)Cc2ccnn2C)c1)NC C1(OC)CCCC(CC(=O)NC(C2CC(NC(c3ncc(C)cn3)=O)C2)C)C1 C1(NC(CCC2(C)CN(C(CCCCSC)=O)C2)=O)CCCCC1(C)O c12ccc(cc1Cl)S(=O)(=O)NC2.c1(SCC)nnc(CN2CCOCC2)n1C c1(CC)nn[nH]c1C(=O)NC1C=CC1C(=O)N(CCC(C)(C)C)CCO C(C(C(=O)N(CCC(c1nn[nH]n1)NC(=O)OC(C)(C)C)C)C(C)C)SC C1(C(=O)NCC(C)C(=O)N(C(C)CC(F)(F)F)C)CC2(CCC2O)C1 N1(C(C2CCC2C(F)(F)F)=O)CCC(C(F)(F)F)C(NC(=O)CC2CCOC2)C1 Cn1nc(O)cc1C(N1CCC2CC12C(N1CCCC1CC(N)=O)=O)=O C#CCCC(=O)NC1C=CC(CNC(=O)CSc2cccs2)C1 C1(OC(F)F)(CC=C)CCN(C(C2CCOC2)=O)C1.c12ccc(cc1)[nH]c2=O N1(CC(S(C)(=O)=O)C2CCOCC2)CCSC2CCCC12.c12ccccc1C2 C1(CC#C)(C(N2CCC(C(N)=O)CC2)=O)CCN(C(=O)Cn2ccnc2C)C1 C(=O)(CCCCC1CC1)N(CCNC(C1(c2ccccc2F)C(C)C1)=O)C1CC1 c1(NC(=O)C=CC(C)(C)C)ccc(C(=O)OC)c(C)c1.C1(CC)CC1C(=O)N C(=O)(C1=CCCC1C)N(CCCNC(C(CC)C#N)=O)C c1(C(=O)NCCC2(O)CN(C(c3coc(Cl)n3)=O)C2)ccc2ccncc2n1 Cc1cnc(C(=O)NC2CCC23CN(C(=O)CC2OCCO2)C3)cc1Br C=CCCC(C(=O)NC1(C)CC(O)(CO)C1)NC(=O)C(=O)NCC1CC1 C1(NC(C=CCCC)=O)CCCN(C(c2ccccc2-c2ccncc2)=O)C1 Cc1nnn(CC(=O)NCC(c2ccccc2)CNC(=O)C=C2CCC2)n1 C1(NC(Cc2nc(C)sc2)=O)CN(C(c2cc(C#N)[nH]c2C)=O)CC1(C)C N1(C(C2CC(C#C)(O)C2)=O)CC=C(C(=O)N(C(C)CSC)C)C1 C1(C(N2CCC(CNC(C3(C)CSC3)=O)CC2)=O)CC(O)c2ccccc2O1 C1(CNC(C=C2CCN(C)C2)=O)CC2CCC1N(C(C1(C)CCN(C)C1=O)=O)C2 CC1NC(=O)C2=C1N(Cc1nnn(C)c1C(F)F)C(=S)NC2c1cnoc1 c1(NC(c2c(-c3ccc(OC)c(F)c3)cncn2)=O)c(Br)ccc(F)c1F C1(CNC(C2CCCCS2)=O)CCCN(C(c2ccoc2Cl)=O)CC1 N1(C(c2n(C)ncc2Cl)=O)CC(NCc2ccncc2)CC(C(F)(F)F)C1 C(=O)(C(CC(C)(C)C)NC(=O)CN1CCNC(=O)C1)Nc1c(C(C)C)cccc1 C(=O)(N=c1ccc(Cl)n[nH]1)C1CC1.c12ccc-1cc2.c1(CCC)ncc(CN)o1 c1(C(=O)NC2CCCC(NC(CCCOC)=O)C2)cc2n(n1)CCCNC2=O c1(CC)nncn1NC(=O)CCC1CCN(C(c2cnn3ccccc23)=O)C1 c1(C(=O)NCc2nc(CNC(CCCOC)=O)sc2)ccccc1C c1(NC(C2C3N(C(C(CC(C)C)O)=O)C(CC3)C2)=O)ccc2c(c1)N(C)C(=O)C2 c1(OCC)cnc(CN2CC(O)CC2C(=O)NCc2ccc(C(N)=O)cc2)nc1 CC1CN(C(=O)CSC(F)(F)F)CCCN1C(=O)CC1OCCC1(C)C c1(C(N2C3CC(NC(C4CC4F)=O)CC2CC3)=O)cn2c(Cl)cccc2n1 c1(COC)ccc(C(=O)N(CC(C)NC(c2cc(-c3csc(C)n3)c[nH]2)=O)C)s1 c1(NC(C2C=CC(NC(c3ccc(C)c(Br)c3)=O)C2)=O)c(F)cc(C#N)cc1F C1(C(=O)NCC(C)C(C)(F)F)CCN(C(=O)C(CO)C(C)(C)C)O1 c1(C(N2CCC3(C(NC(c4ccc(CO)cc4)=O)C3)C2)=O)nccc2ccsc12 c1(C(=O)Nc2cnc(CC)nc2)ccc2c(n1)CN(C(C1(C#N)CCC1)=O)CC2 N1(C(COCCCCCC)=O)CCN(C)CC1CNC(=O)C(C)C1CCC1 C(CCC(=O)N(CCCNC(c1cc(-c2ccco2)[nH]n1)=O)C)NC(C)=O C1(C)(C(=O)NCCOCCN(C)C(C2CCCS2)=O)CCCCO1 C(=O)(C(CN=[N+]=[N-])NC(=O)C(O)CC(C)C)N(CC#C)CCO C1(C(=O)NC2CN(C(CC(=O)OC)=O)CC2C)CC2CC(O)CC(C1)C2 C1(NC(c2c(C)n(C)cc2)=O)CN(c2ncccc2C#N)Cc2nccn2C1 C1(C(=O)NCCCCNC(=O)CC(C)OC(C)=O)(CC)CCOCC1 C(=O)(CCCCC(F)F)NCC1C(C)CCN(C(c2cccnc2)=O)C1 N1(CC(=O)NCC2(NC(c3cncc(Br)c3)=O)CCCC2)CCC(F)CC1 C1(C(=O)NC(C(C)C(=O)N2CC(n3cnnc3)C2)C)CCC(C)(C)OC1 Cc1ccc(C(N2CCC(F)(C(=O)NC3CC(C)C3)C2)=O)cc1C CC1CN(C(C23CC(F)C2C3)=O)CC1CNC(c1ccc(OCC2CC2)cc1)=O Cc1ccc(-c2n[nH]cc2SC(C(CN2CC(CS(N)(=O)=O)CC2=O)C)=O)cc1 CC1(CNC(=O)C=CC2CC2)CCCN(C(=O)CSC(F)(F)F)C1 N1(C(CNCCc2c(C(=O)OC(C)(C)C)ocn2)=O)CC2CC(O)CC2C1 N1(C(c2c(C)cc(C)s2)=O)CCC(N=[N+]=[N-])(C(=O)NC(CC2CCCC2)CO)C1 C(=O)(C1=CC2(CCOCC2)C1)N1CCC(CNC(C(C=C)(C)CC)=O)C1(C)C c1(C(=O)NC2C(NC(C(C)NC(CC)=O)=O)CC2)cn(CCC(C)(C)C)nn1 c1(SCC(c2ccccn2)OCC)cc(S(C)(=O)=O)ccc1C c1(OC)ccc(I)cc1C(N1CC(N(C)Cc2cncc(Br)c2)C1)=O C(=O)(CCC(C)(C)F)N1C(C(N(C)CP(C)(C)=O)=O)CCC1 CCC(CNC(c1ccn(C)n1)=O)(CC)C(=O)NCCCN(C)C(C)=O C1(CC)CN(C(=O)COC(C)=O)CCN1C(c1sc(CC(C)C)nc1C)=O N1(NS(c2c(C)cc3c(c2)OCO3)(=O)=O)CCOC2(CCCS(=O)(=O)C2)C1 C1(CNC(C2N(C(CCC3(C)CC3)=O)CC=C2)=O)CCC(=O)NC1 C1(C(=O)OCC)(C(=O)NC2CC(C)OC2=O)CCOCC1 C(C(C(=O)NCC(CO)C1CCC1)NC(=O)Cc1nocc1CC)SCC CC1(C)CC(NC(c2cc(C3CC3)on2)=O)CN(C(=O)CCN2CCOC2=O)C1 CCS(=O)(=O)CCNC(C1(NC(c2cc(CO)oc2C)=O)CC(O)C1)=O C(C(CC(C)C)C(=O)N(C1CCN(CCC2(C(=O)NCC=C(C)C)CC2)C1)C)OC CC(C(=O)NCCOC1CCN(C(=O)CCN2CCCCCC2)C1)C(F)F c1(C(=O)NC(CNC(C2ON=C(C)C2)=O)C2CC2)scc(Br)c1Cl Cc1ccc(F)c(C(N2CCCC2C(=O)N(C(C)CCN(C)C)C)=O)c1 c1(C(N2CCC(OCC(=O)NCC(=C)F)C2)=O)ccc(C2CC2)cc1 c1(CS(=O)(=O)N(N2CC(C3CC3)C2)C(C)=O)cc(-c2cccs2)nc(C)n1 N1(C(C(C2CCOCC2)C)=O)CCOC(CC(=O)NCCc2ncon2)C1 N1(C(=O)CC2CCC3CC23)CC2(C(=O)NC34CC(CO)(C3)C4)CC1CO2 CN1CCN(C(c2cc(Cl)ccc2N)=O)CC1CNC(=O)C(CO)C(F)(F)F N1(C(c2c(Cl)cn(CCC)n2)=O)CCCCCC1CNC(=O)CCF c1(CC)oc(C(=O)NC2CN(C(c3cnc(C(N)=O)s3)=O)CC2C)cc1C C1(OC)CCC(N=c2[nH]c(=NC(C)c3ccnc(O)c3)[nH]c3c2CSC3)CC1 N1(C(C(C=CCCC)O)=O)C2CCC1CN(C(=O)Cc1nnc(OC)s1)C2 C(COc1ccccc1)(C(=O)NC1CCC1N(C(c1ccncc1)=O)C1CC1)OC C1(C(=O)NCc2n(CC)ncn2)CCC(C2CC2)N1C(c1sccc1C)=O c1(C(C(=O)NCCC(=C)CNC(c2cc(=O)cc(Cl)[nH]2)=O)C)cc(F)cc(F)c1 N1(C(C(=O)NC2C(CC)CCCC2)=O)CCC2(CC1)CCN(C)C2=O C1(C(=O)NCc2c(C(N(C)OCC(F)(F)F)=O)n[nH]c2)CCCC12CCC2 C=CCCCN=C(NC(C)CNC(=O)C(C)C)N1CCN(CC2CCCO2)CC1 C(=O)(CC1CCc2ccccc21)NC(C)(C)CCNC(C1CCCO1)=O c1(C(C(=O)NCC(C(C)C)NC(c2ccccc2)=O)C)cccc(C(F)(F)F)c1 C1(C)(C(=O)OCC)CC(NCCC(N)C2CCC2)C1 N1(C(C(CN(C)C)O)=O)CCC(O)(CNC(C2CC23CCSCC3)=O)CC1 CCN=c1[nH]c(C(=O)NCC(C)(O)CNC(=O)C(C)(C)C2CCOCC2)cs1 c1(C(=O)NC2(CC=C)CCN(C(c3c(F)cccc3Cl)=O)C2)cccn2nccc12 C(=O)(CC1OCc2ccccc21)N1CC=CC(NC(C(C)(C)SC)=O)C1 N1(C(C2CCN(C(C3CCC(=O)N3)=O)CC2O)=O)CC2CCCC(C2)C1 c1(OCCNC(c2occ(C(=O)NC3CCC4(CC4)C3)n2)=O)cc(F)ccc1F c1(OCC(N2CCC(CC)(CO)C2)=O)cc(F)ccc1F.C12CCN(C1)C2=O CCCCC(C(=O)N1CCC2CC2(C(=O)NCC2(CC(C)C)CC2)CC1)C(C)C c1(SCC)cnc(O)c(C(=O)NC2CCC(C)N(C(c3ccccc3F)=O)C2)c1 CON=Cc1ccc(C(N2CCC2CNC(=O)C(C)CC(=O)OCC)=O)cc1 Cc1ccc(-c2nnc(NC(=O)NC3CCN(c4ccc(C)c(F)c4)C3)s2)c(C)c1 C1(NC(C(C)OCC(F)(F)F)=O)CCCCC1NC(c1cnc(O)o1)=O CCC(C)CCCCC(=O)N1CC(NC(c2cnc(C)c(N)c2)=O)C2(CCC2)C1 c1(CC)ccc(-c2nc(-c3ccc(C)cc3)n(CC3COCCO3)n2)cc1 C#CCCC(=O)NC(Cc1cc[nH]n1)C(=O)N1CC(c2ncccn2)C1 N1(C(c2scc(COC)c2)=O)CCC2CCCN(C(=O)C=C(Cl)Cl)C2C1 c1(NCc2nonc2NC(N(CC)CC)=O)cccc(C(C)C)c1F c1(COC)cc(C(C(=O)NCc2nccs2)N(CCOC)CC2CC2)no1 C(=O)(CCOCC(C)C)NC1CC1.C1(=O)CN1CC.C(CCO)OCC(C)N c1(CC(=O)NC(CNC(C2CC(C)(O)C2)=O)(C)C2CC2)c[nH]c2cc(F)ccc12 CN1CCC(C2(C(N3CCC(C)(CNC(=O)Cc4ccsn4)C3)=O)CC2)CC1 c1(-c2n(CC=C)c(N3CCCC3CCOC)nn2)cccc(C#N)c1 C=C1CC2(C1)CC(C(=O)NCC(CC(F)(F)F)NC(=O)COCCC)C2 C1(CCC(=O)NC2(O)C(C)OCC2)CCCCN(C(=O)CN2CC3CC3C2)C1 N1(C(c2c(C)nsc2N)=O)CCC(NC(c2cc(CO)c(C)o2)=O)C(C)(C)C1 C1(NC(C2CCCS2(=O)=O)=O)CCN(C(C2(CO)CC2)=O)C1Cc1ccccc1 c1(C(=O)NC(C(=O)NCc2c(C)nccn2)Cn2cncn2)ccn(C)c(=O)c1 C(=O)(C#CC1CCCC1)NCC12C(CN(C(C3(CC=C)CCC3)=O)C1)C2 c1(OC)cccc(C(=O)NCCOC(C)(C)CNC(C2(C)COC2)=O)n1 C1(NC(=O)C=CC2CC2)CC2(CCCN(C(=O)C=CCOC3CCOCC3)C2)C1 C1(C)(CNC(C(C2CCN(C(c3n[nH]c(C)c3Cl)=O)CC2)C)=O)CCCCCC1 Cc1ccc(C=CC(N2CC(NC(c3ccnn3C(C)(C)C)=O)C2)=O)s1 N1(C(=O)CC2CCCC(F)(F)C2)CC2(CCCCN2C(=O)Cn2nccn2)C1 c1(CNC(c2ccc[nH]2)=O)cc(O)nc(CNC(C2CC3(C2)CC3F)=O)n1 Cc1cccc(C(=O)NCC2(NC(=O)CC3(C)CC(F)(F)C3)CCOC2)c1 CC1(C)C(c2ccccc2)CCN1C(=O)NC12CCC(C1)OC2 N1(C(CC2(N(C(C3C(C)C3C)=O)C)CC2)=O)CC2CCC1CC2 C1(C(N2C(C)(C(=O)NC(COCC)C)C=CC2)=O)CCC(O)CN1C C1(C2(N(CC#C)C)CC2)CCCSC1 N1(C(c2cccc(C)c2)=O)CCC2CCC(C1)N2C(c1cccc(F)c1O)=O CC(CC(N)=O)C(=O)NCC1(F)CCN(C(c2cc(N(C)C)ccc2F)=O)C1 c1(NCCCCNCC(CSC)O)ccc(C(C)C)cc1F CC1CC(=O)NC1C(=O)NCC(C)(F)CNC(=O)CCCN(C)C C1(C)(CCC)CC12CCN(C(=O)CCCn1cc(-c3cnc(C)o3)nn1)CC2 N1(C(C(N)=O)=O)CCC(CCN2CCN(C(=O)CCCc3nccs3)CC2)CC1 c1(OCCC)ccc(C(=O)NC2CC2NC(C2CC2c2cccs2)=O)cc1 C=CC(C)(C)C(=O)NCCCCNC(c1cn(C)nc1C(C)(C)C)=O.C(C)(=O)O Cn1ccc(=O)c(C(=O)NC(C2CCCC2)CNC(c2ncc(Cl)nc2Cl)=O)c1 c1(NCCN2C(CC)COCC2)ccc(S(=O)(=O)NCC2CCCCO2)cc1Cl CC1CCN(C(c2ccc(C3COC3)cc2)=O)CC1CNC(=O)C1=CCCC1 CC1(C)COCC(NC(=O)C(CC2CC2)NC(=O)CCP(C)(C)=O)C1 n1(CC(C)C)ccc(=NC(=O)CC(C)C2CCN(C(=O)C(F)(F)C(C)O)C2)[nH]1 C1(C(=O)NCC2CCN(C(c3n(C)c(O)nc3)=O)C23CC3)CC2(CCCCC2)C1 C12CC13CCN(CC3)C2=O.C1(c2cccc(Br)c2)(CNC(C)=O)CCCCC1 N1(C(C)=O)CC(CNC(C2CC(F)(CC3CCS(=O)(=O)C3)C2)=O)OC(C)(C)C1 Cc1ccc(F)c(OCC(=O)NC(CNC(=O)CSC2CC2)C2CC2)c1 C1(C(=O)NC2(C)CCN(C(C(C)CN3CCOCC3)=O)C2)SC2C=CC1CC2 C(=O)(CCCCCn1cccn1)NC(C1CCOCC1F)C c1(C(=O)N(c2cccc(Cl)c2)C2CC(O)(C(=O)O)C2)ccc(F)c(I)c1 c1(C(=O)NCC2(NC(C3C(OC)COCC3)=O)CCCC2)cccc(Cl)c1F C=C(C)c1ccccc1C(=O)N=c1nc(CN)[nH]s1 C1(C(=O)NC2C(NC(CN3CC(=O)NC3=O)=O)C2)CC2(CCC2)CO1 C#CCC(C(=O)NCCCN1CCOCC1)NC(=O)C(c1ccccc1)C C1(O)(C(C)NC(CC(C)CF)=O)CCN(C(C2CCOCC2)=O)CC1 C(=O)(C(=O)N=S(C)(C)=O)NC(C1CCN(C(=O)Cn2cnc(C(N)=O)n2)C1)C C1(C(=O)NCC(CC(=O)Nc2cc(C(C)C)ncc2)O)C2CCC(F)(F)C12 N1(C(C(Cc2ccccc2)OC)=O)CC2CC(N(C)C(C3CC(F)(F)C3)=O)C1C2 C1(NC(C2C(C)(C)C2)=O)CCN(C(=O)Cn2cc(Cl)cn2)C12CC2 C(=O)(C(F)CC(C)(C)NC(=O)CCc1nncs1)N1CCC(N(C)C)CC1 N1(CCC(=O)NCC=CCNC(C2C(C)(C(F)F)C2)=O)CCc2ccccc21 c1(CNC(CCN(C(COCCCCC)=O)C)=O)c[nH]nc1CC C1(NC(=O)NC2(C(N)=O)CCC2)CCC(n2cc(-c3ccns3)nn2)C1 C1(C)(C(N(CC(C)O)C(C)CO)=O)CC12CCN(C(=O)CCC1CCC1)CC2 CCCC(CC)CCC(=O)NCC(C)(F)CNC(c1cnn2c1OCC2)=O C(=O)(C(CC1CCCO1)C(F)(F)F)NCCN(C(=O)OC(C)(C)C)CC C(=O)(CC(C)C(C)(C)C)NCC(C1CCC1)NC(c1c(C)n(C)nc1C(F)F)=O C(CC(C)(C)CC(=O)NC1CCN(C(c2cc(OC)ncc2Cl)=O)C1(C)C)OC C1(CC(=O)NCC2(CC)CCCCC2)CCCCC1NC(=O)C(C)N=[N+]=[N-] c1(OC)ccc(C=CC(=O)NCCC(O)CNC(=O)C(C)(C)CC2CC2)nc1 CC(C)CC(CNC(=O)CCN1CCOCC1)NC(C1CN(C)C1)=O O(NC(=O)C(CC1CCCC1)NC(=O)C(C)CC1CCCC1)CC=C c1(N2CCCC(CSC)C2)nc(=NCc2ccc(N)c(Cl)c2)[nH]c2c1CSC2 c1(NCC(=O)NCC(C)(C)NC(C2CCSC2)=O)cccc(C#N)c1 c1(OC)ccc(C(=O)NC2CN(C(c3ccc(C)o3)=O)CC2C)c2sccc12 c1(C(N(CCCNC(=O)C=CCOC)CC)=O)c[nH]c2c(Cl)cccc2c1=O C(c1cc2ccccc2n1C)=CC(=O)N(CCNC(C(C)=C(C)C)=O)C(C)C CC1CN(C(C2CCC2(C)C)=O)CCCN1C(c1ccnc(C(F)(F)F)c1)=O C1(CNC(C2(CC)CCNC2=O)=O)CC2CCC(C1)N2C(C1CC=CC1)=O Cc1cnc(C(=O)NCC(C2CC2)N(C)C(c2ns[nH]c2=O)=O)c(C)c1 N1(C(CCN2CC(=O)NCC2)=O)CCC2CN(C(c3ccoc3)=O)CCC12 CC1COCCN1C(N1CCN(C(=O)Cc2cc(Cl)sc2Cl)CC1)=O C(C(C(=O)NCCN(C(=O)C(C1CCCC1)OC(C)C)C)N(C)C)OC(C)=O C#Cc1ccc(C(=O)NCC2(C(=O)N(C)CCc3ccco3)CCC2)cc1C C1(NC(C(C)(Cl)Cl)=O)CN(C(C2CC2c2cccnc2)=O)CC1C(F)F N1(C(CSCC)=O)CC2C3CCC(C2C1)N(C(C1(C)C=CCC1)=O)C3 C(C(C)(C)C(=O)NCCCCC(=O)NC1CN(C(C)C)CC1C)NC(C)=O C1(NC(C(C(=O)OCC)OC)=O)CC2CC(NC(=O)CC3(OC)CC3)CC2C1.CN N1(CCNC(=O)N(C2CCCC2)CCO)CC2CCC1CC2 C#Cc1cnc(C(=O)NC(C)(C)CC(N2CC(S(C)(=N)=O)C2)=O)c(C)c1 C1(COC)(CNC(c2cc(Br)no2)=O)CCN(C(=O)Cc2nc[nH]n2)C1 C1(C(=O)NCCCNS(CC)(=O)=O)C(CC)CCCN1C(=O)C=Cc1cocn1 c1(OCC)cccc(C(=O)NC)c1N.C1(CCOC)(NC(C2COC2)=O)CCCC1 N1(C(C(CC)CCOC)=O)CCC2(CC1)CC(C)N(C(=O)CC(CC)C1CC1)C2 C(CS(=O)(=O)CC(=O)NC1CN(C(=O)CCc2cncnc2)CCC1CO)OC C(N=c1nc2scnc2c(N2CCC(C)(F)C2)[nH]1)c1cc(C(CC)CC)no1 CC1C(CC(=O)NC2CCN(C(=O)COCCc3ccccc3)C2)C1(F)F N1(C(C(=O)NCCC2CCC(C)(C)O2)=O)CCC12CCC(F)(F)CC2 C1(CN2CCN(Cc3c(-c4cn(C)nc4)n[nH]c3)CC2)CCC2(CCC2)CC1 C(=O)(C(C)C(O)CC)NC(CC=C)CNC(c1ccc(OCC(F)F)cc1)=O C(C(C(=O)N(CC1COc2ccccc21)C(C)OC)C(C)C)OC N1(C(C(C)C2CC2)=O)CCC2(C1)CN(C(=O)CCc1ccc(O)c(O)c1)CCO2 C=CCCCCCCC(=O)N(CC(C)(C)C(N1CCC(O)C(F)C1)=O)C C(c1csc(C)n1)=CC(=O)NCCC1(C(=O)NC(C2CC3C=CC2C3)C)CN(CC)C1 C1(C(N2C(CNC(C=Cc3c(C)ccs3)=O)CC2)=O)CCC(=O)N(C2CC2)C1 Cc1cnn2ccc(C(N3CCC4(CC(NC(=O)CCC(N)=O)C4)C3)=O)nc12 C1(O)(C2N(C(CCOC)=O)CCC2)CCN(C(=O)C=C(C)C)C1 CC(C)C(F)C(=O)N1CCC(C)C1CNC(c1ccccc1CC(C)(C)C)=O c1(-c2nc(-c3n(C)ncc3Cl)on2)ccc(F)cc1F C(CC(C)C)(C(=O)NCC1(C)CCC(=O)N1)N(C(c1c(C)ncnc1)=O)C N1(C(C(OC)OC)=O)CCN(C(=O)CC2COCCOC2)C2(CCC2)C1 n1(CC)nc(C(C(=O)NCC2CC2)N(C)Cc2ncoc2C)c(Br)n1 c1(C(N(C2CC(NC(C3CCCCC3)=O)C2)C)=O)cc(F)cc(Br)c1F c1(C(N(C2CN(C(Cc3nc(C)sc3C)=O)C2)C)=O)ccc2c(c1)C(C)(C)CO2 c1(OC)ccc(SCC(N2CCC3C(NC(c4cc(F)n(C)n4)=O)C23)=O)cc1 N1(C(C(COC)C)=O)CCC(O)C1C(=O)NCCCCC(N)=O c1(CC=C)cccc(C(=O)N(C(C(=O)N(C)CCOCC(C)C)C(C)C)C)c1 N1(C(COC(CC)(C)C)=O)CC(NC(c2ncccc2F)=O)C(O)C1 C(CCO)(C(=O)NCCn1cnnn1)NC(C1CC(OC)C1)=O.C(CO)CCO C1(CNC(c2scc(COC)c2)=O)CN(C(=O)CC2CSC2)CC1C(F)F Cc1cc(CCC(=O)NC2CC2C(=O)NCCSCc2ccc(Cl)cc2)nn1C C(=O)(C(CO)C(C)(C)C)NC(CNC(c1c(C)nc(C(C)C)o1)=O)(C)CC(C)C CC1CC(NC(C2CC=CC2NC(=O)Cn2cccc2)=O)C(=O)O1 C1(C(=O)OCC(N2CC(C)(OCC3CC3)C2)=O)COCCN1S(C)(=O)=O CCC(C(=O)NC(C)(C)C=CC(=O)N(C)C)n1ccnc1 c1(C(=O)NCC(=O)NCCC)ccc(CNC(=O)CCC2CCC(C)O2)cc1 CC(C)C(C(C)NC(c1cnc(C2CC2)[nH]1)=O)NC(c1coc(Br)n1)=O Cc1ccc(C(=O)NC23CC(C2)N(C(c2cn(C)nc2C(C)(C)C)=O)C3)c(C)c1 N(C(=NCCNc1ccccn1)NCc1cc(Br)cs1)CC1(C=C)CCC1 N1(C(C2C(COC)CC2)=O)CCOCC(CNC(c2c(C(C)C)n[nH]c2C)=O)C1 Cc1cc(CC(C(=O)O)NC(=O)C(C)C(C)c2ccc(Cl)cc2)ccc1C(=O)O c1(OC)ccc(CC(=O)NCCCCC(C)NC(C2(O)CC2(C)C)=O)c(OC)c1 C1(CC)CCN(C(C2CN3CCC2CC3)=O)C(C(N2CCCC2CC(N)=O)=O)C1 Cc1ccc(C(=O)NCC2CN(C(=O)CCn3cncn3)CC2O)c(Br)c1 N1(C(C2(C(=O)NC)CC2)=O)CCC(C)(CC(=O)Nc2cncn2C(C)C)C1 C=C(Cl)CC(C(=O)N(CC(O)C(F)(F)F)C)NC(c1cccc(COC)n1)=O O=C1CC(=O)CC(C(N2CCC2CNC(=O)CN2CC3C=CC2C3)=O)C1 C(C(F)(F)C1CCC1)C(=O)NCCOCCOC S(=O)(=O)(CCC(C)(F)F)NCC1CC(C)(C)NCC1 c1(C(=O)NCC(CNC(CCSCCOC)=O)O)cc(OC)cc(Br)n1 C1(O)(CN(C(=O)CC2CC=CCC2)C)CCN(C(=O)C(F)OC(F)(F)F)CC1 CCC(C)(CC(=O)N1CCC(NC(c2ccc(OC)s2)=O)C(F)C1)C(=O)OC Cn1cc(CO)c(COC(c2ncccc2C2CC2)=O)n1 C1(CC(=O)NCC2(NC(C(C)c3ccon3)=O)CC2)CCCCCC1 N1(C(C(CC)OC)=O)CC(C)Oc2cc(Br)ccc21 CC1CN(C(C2CN(C(=O)COC3CC3)CC2F)=O)C12CCOCC2 c1(N2CCC(N(C(C)C)C(c3ccc(Cl)o3)=O)CC2)cc(=O)n(C)c(O)n1 C1(CNC(c2cc(C)nn2C)=O)CCCN(C(c2ccc(F)cc2C)=O)CC1 C1(CNC(C(COC)C)=O)CCCCN(C(c2cn(C(C)C)nc2C)=O)CC1 c1(OC)cnccc1C(=O)N(C1CCCN(C(=O)CC2CC3CC3C2)C1)C CCC(CC(=O)NCCC1CCN(C(=O)CC(C)C(C)C)CC1)C(C)C N1(C(c2c(C)cc(SC)o2)=O)CC2(CCC(CNC(=O)COCCN(C)C)O2)C1 C1(CC(=O)NCCN(C(c2cncs2)=O)CC)CCC(C)(C)CO1 C(F)(F)(C(F)(F)F)c1scc(C(N(C(CNC(C(CC)NC(C)=O)=O)C)C)=O)c1 C(=O)(C(COC)CC)N(CCSc1ccc(Cl)nc1)CC.C1(F)(C(=O)N)CC1C Cc1ccn2nc(C(=O)NCC3CC4CN(C(C5C(C)C5(F)F)=O)CC34)nc2n1 C1(CCNC(=O)COC2CCOC2)CC(F)(F)CN1C(C1CCC(F)(F)C1)=O N1(C(C)C)CC(C(=O)N(CCCNC(=O)CC(C)F)C2CC2)CC1=O C(CCC(=O)NCC1CC1C(N1CCC(C(C)(C)C)C1)=O)=CC c1(C(N2CC3OCC(NC(c4occ(C)c4)=O)C3C2)=O)ccc(F)c2c1CCC2 C1(S(N)(=O)=O)(C(=O)NCC(CC)(CC)NC(=O)Cn2cncc2C)CCCC1 N1(C(C(Cc2c(C)nc[nH]2)O)=O)CC2(CCCC2NC(=O)CC2(CO)CC2)C1 C(=O)(C(c1cccs1)=Cc1ccccc1)NC(CC=C)CNC(=O)CC1CC=CC1 C1(C(=O)NCCCC(=C)C)COCCN(C(c2csc(C)n2)=O)C1 CC1(C)CC(NC(c2cscc2SC2CC2)=O)CN1C(=O)CCF N1(C(CCCC#C)=O)CCC2(CC(NC(c3n[nH]c4ccc(F)cc34)=O)CO2)C1 C1(NC(C(C2CCCCC2)C)=O)CN(C(=O)CCc2cnn(C)c2)CC2(CC2)C1 c1(C(=O)NC(CNC(C2(OCC)CCOC2)=O)CC)cc(Cl)n(C)n1 n1(CC(N2CCCC(N(C(COCC#C)=O)C)C2)=O)ccc2ccccc12 N1(C(c2ccc(C(C)=O)o2)=O)CCOCC(C(=O)NC2COCCN(C)C2)C1 Cc1nc2cc(C(=O)NCC(C3CC3)NC(C3CCCO3)=O)cc(O)c2o1 c1(C(=O)NC2CC(SC)C(O)C2)cc(OC)nc(F)c1.C12(CCCC1)C(=O)NC2 C(C(=O)NOCC(N1CCCC(N(C)C)C1)=O)(C(C)C)OC c1(-c2nc(C)n(-c3ccc(Sc4nnc(S)nc4O)cn3)n2)ccc(N=[N+]=[N-])cc1 CC(=O)C(C)CCC(=O)N1CCC2(CCCC2)C1 C(C(C)(C)C#CC(=O)N1CC(O)(C(F)(F)F)C1)NC(C(C)SC)=O c1(C(C)NC(C2CC2c2cccs2)=O)ccc(CNC(C2CC=CCC2)=O)cc1 C1(NC(CC2N(C)C(=O)CC2)=O)CC12CCN(C(c1nccnc1N)=O)CC2 c1(C(N2CCOC(Cn3cccn3)C2)=O)csc(=NC2CCSCC2)[nH]1 C1(C)(C(c2nnnn2-n2cccn2)NCC(C)(C)CNC(N)=O)CC=CCC1 C1(NC(C(C)(C)CO)=O)CC2CN(C(c3nonc3N)=O)CC12 c1(C(N(CC(C)N(C(CCOC(CC(C)C)C)=O)C)C)=O)nc(Cl)cc(N)c1Cl N1(C(c2c(OC)c(C)sc2)=O)CCC(NC(c2sccc2C#N)=O)C1(C)C c1(OC)ccc(C(=O)NC2CCCN(C(=O)C=CSC)C2C)cc1OCCO c1(CC(=O)NC2CCN(C(c3c[nH]ccc3=O)=O)CC2)ccccc1C(F)(F)F c1(N2CCC(C#C)C2)ccncc1S(=O)(=O)NCC(c1cccnc1)O CCCC(C)CC(=O)N1CCC(F)(CNC(=O)CCc2nc(C)no2)C1 Cc1cc(Cl)cc(C(N2CC=C(CCNC(C3COC(C)(C)C3)=O)CC2)=O)c1N c1(C(N2CCC(CCNC(C3CC(C)N(C)C3)=O)C2)=O)c(F)cc(O)cc1F N1(C(C(n2c(C)ncc2)C)=O)CCCC(C(=O)NC(CO)CCC2CC2)C1C Cc1nc2ncc(C(N3C4CCCC3CC(NC(=O)C(N)=O)C4)=O)c(=O)n2[nH]1 N1(C(c2c(C(C)(C)C)noc2)=O)CCC(C(F)F)(CNC(c2cnccn2)=O)C1 N1(C(C(C)OCCC=C)=O)CC(CNC(C23CSCC2C3)=O)CC(C)(C)C1 c1(OCC)oc(OCC)nc1N(C(=O)Oc1cccc(N2CCC(C)C2)c1)C.CC N12CCC(CC1)N1CCC(CC1)C2=O.Cc1cnc(C(=O)NC2CCOC2C)s1 c1(NC(=O)NC2CN(C(C3(OCC)CCOC3)=O)C2)c[nH]c2ccc(Br)cc12 N1(C(C2(C)CCC2)=O)CCC(C)(C)C(C(=O)NC2CCCSC2)C1 C(C)(C(C(=O)NOCCCF)C(C)C)NC(Cn1c(C)cc(C)n1)=O C(c1cc[nH]c1)=CC(=O)NC(C(=O)N(CC)CC1CCCCC1)C CC12CCC(C(=O)NC3CCCC3NC(c3cnc(C4CC4)o3)=O)(CO1)C2 C1(C(N(CC#CC)C)=O)CCN(C(=O)C(N2CCOCC2)C)C12CCC2 c1(C(N(CCN(C(C)C)C(c2ccc[nH]2)=O)C)=O)cc(C(F)(F)F)c[nH]1 c1(NC(C2CC2)=O)cc2c(nc1O)CCN(C)C2.Cc1ccc2cc1CNC2 C(=O)(C(CC(F)F)N(C(=O)CC1CCOC1C)C)NCC(C#C)C(C)C c1(C(CCOC)NC(=O)NC(C#C)(C)C)nc2ccccc2[nH]1 Cc1cc2n[nH]cc2cc1C(=O)NCCCCC(C)NC(=O)C(C)OCC(C)C c1(-c2nc(COCC)nn2Cc2ccncc2)ccc2[nH]ccc2c1F CCC(CCC(=O)NC1CSC1)NC(=O)Cc1cnn(C)c1C c1(NC(c2n(CCCC)nnn2)(CC)C2CCC2)ccc(OCC)nc1C N1(C(C2C=C(C)CS2)=O)CCCCC(NC(c2ccc(OC(C)C)cc2Cl)=O)C1 c1(C(N2C3CC(NC(c4ccc(C)s4)=O)C2CC3)=O)ccc(Cl)c(F)c1F C12(NC(c3cccc4nonc34)=O)CCC(CC1)N(C(=O)CC1CCCCO1)C2 C1(C(=O)NCCC(C)C)Cc2cccc(OC(C)(C)C)c2O1 C(CCN=C(NCC1CC(OC(C)C)C1)N1CC(O)C2(CC2)C1)OC C1(C)(CNC(c2n(CC)ccc2)=O)CCCN1C(=O)CCc1conc1C n1(CC(N2CC(CNC(=O)OC(C)(C)C)C2)=O)cc(CC2CC2(Br)Br)cn1 Cn1cncc1C(N1CCC1(C)C1CCCCC1)C(=O)NCCC1(C)CC1 c1(CN2CCOCC(C(=O)NCCCOC)C2)cc(Br)c(C)cc1F C1(NC(C2N(C(C)=O)CCC2)=O)CC2CC1N(C(c1cnccc1C)=O)C2 C12(C(N3CCCC(N(C(CCC#CC)=O)C)CC3)=O)CCCCC1NC(=O)C2 c1(N2C(CNC(c3c(C)nc(C(C)C)s3)=O)C=CC2)nc(N(C)C)nc(CO)n1 c1(C(=O)OC)cnn2ccc(N(CCCNC3CCC4CC4C3)C)nc12 N1(C(C(C=C)CC)=O)CC(NC(c2ccc(C)c(O)n2)=O)C2(CCC2)C1 CC(C1=CCN(C)CC1)NC(C1(CCNC(C2CCCCCC2)=O)CC1)=O C(C)(C(C)(C)C(=O)N(C)Cc1cncn1C)NC(C(COC)C)=O C1(C(C)C)(C(=O)NC2CC(N(C)C)C2)CCN(C(c2cccc(CCO)c2)=O)C1 c1(NC(C2(N(C(C(C)=CCC)=O)C)CC2)=O)cnc(C(C)C)nc1 CC1(C)CCCC(O)(C(=O)NN2CCCC2)C1.C1(=O)CCNC(=O)C2CC2N1 N1(CCC)C(=O)NC(c2nn(C)cc2S(C)(=O)=O)C2=C1C(C)(CC)NC2=O C(=O)(CCC(C)(C)C(=O)NC1CCCCC1CNC(=O)C(O)C(F)F)OC C(=O)(CS(=O)CCC(F)(F)F)N1CCN(C(CSCC#C)=O)CC1C(F)F C#CCCC(O)C(=O)N1CC2CC(C1)C2NC(c1cc(Br)cn1C)=O N1(C(C2(C)CCN(C)C2)=O)CC(C2CCN(C(=O)CCF)CC2)C1 C1(CC)CN(C(=O)CNC(=O)C(F)(F)C(F)F)CCC1NC(c1ccc(C)s1)=O C(C)(CCC(=O)NCC(=O)NCCOC1(CO)CC(C)(C)C1)OC C1(CNC(Cc2c(C)cccc2)=O)CC2CCCC2N1C(c1nnc(S)n1C)=O C1(CNC(C(C)OCC(C)C)=O)CCCCN(C(c2cnc(C(F)(F)F)s2)=O)C1 c1(NCc2c(OC)cccc2C)nc(=N)[nH]c(=NC2CCCN(CC(F)F)C2)[nH]1 C#CCCC(C(=O)OCc1csnc1OC)NC(C1C=CC(N)C1)=O N1(C(=O)NCc2nccc(Br)c2Cl)CCN(C(=O)C(F)(F)F)CC12CC2 c1(CNC(=O)NCCCc2cc(F)cc(Br)c2)cc(F)ccc1Cl c1(C(N2CCC(C(=O)NC)C2C)=O)cc(Cl)c(F)cc1N N1(C(CC=CC)=O)CC2CCCC1C2CNC(c1ncn(C(C)C)n1)=O c1(C(=O)OCC(=O)NCC(c2ccccc2)C)ccc(-n2cccc2)c(Cl)c1 c1(C(N2C(C(C)NC(C3(CO)CC3)=O)CCC2)=O)ccc(C#N)c(Cl)c1 N1(C(C2C(CCOC)C2)=O)CC(O)CC1C(=O)NCc1ncc(C)o1 C12(COC)CC(NC(c3cnc(O)cc3C)=O)(CN1C(=O)CC1=CCCC1)C2 CS(=O)(=O)C1(C(=O)NC2CC(CNC(=O)CC3CC4CC4C3)CC2O)CC1 c1(C(=O)NC(CC2CNC2)CO)cccc2c1COC2 Cn1nc2c(c1C(N1CC3OCC(NC(C4(Cl)CC4(C)C)=O)C3C1)=O)CCCC2 CCCC(C(=O)N(C)CC1CCCN1CC)NC(=O)CC1CC(C)=NO1 c1(C(=O)NCC2CCN(Cc3n(CC)ncn3)C2)ccc(F)c(S(C)(=O)=O)c1 C(C(C)(C(=O)NCC1(C)COCCO1)NC(c1ccn(C)c1C)=O)SC C(=O)(C1OCCc2ccccc21)N1CC(N(C)C(C2CC23CC3)=O)C1 C1(OC)CCN(C(=O)CCCCNC(C2CCCC(NC)C2)=O)C12CCC2 c1(C(=O)NCCOCCN(C(=O)CCC2(C)CC2)C)cc2ccccc2[nH]1 C1(CC=C)(C(=O)NCC2CC(NC(=O)CCn3ccnn3)C2(C)C)CCOCC1 C(=O)(C(C)(C)CN(C)C(C1CC(CCO)C1)=O)NCCN(C)CC c1(C(=O)OC)coc2cc(C(=O)NC(CNC(C3CCCN3C)=O)C3CC3)[nH]c12 c1(N2CCN(CC3(CC)CC3c3ccccc3)CC2)cnc2nc(C)cnc2n1 c1(C(N(CCCNC(=O)C=CC(=O)N(C)C)CC)=O)cc2cnccc2cc1F c1(C(=O)NCc2cc(C(=O)NC(C)Cn3ccnc3)sc2)cnc(O)c(F)c1 c1(C(=O)NCC2CCN(C(C3(CCF)CCC3)=O)C2)cnnc2ccccc12 c1(C(=O)NC2(CNC(C3CN(C)C3)=O)CCOC2)cc2occc2n1C N1(C(C2CC(OC)C2)=O)CCCCC1CCCNC(=O)CN(S(C)(=O)=O)C N1(CCNC(C2CCC=CCC2)=O)CCCN(C(C2(C3CC3)CCC2)=O)CC1 C1(NC(c2ncnc(C)c2C)=O)CC2CCC1CC2NC(C1(C)CC1(C)C)=O Cc1cccc2nc(NC3C4CN(C(C5CC56CCC6)=O)CC34)sc12 C(CCC(=O)NC1(C)CC(C(=O)N(C)CCOC(F)F)C1)C1C(C)C1 C#CCC(C(=O)N1CCC(O)(CC)C1)NC(=O)C(CC#C)NC(C)=O C(=O)(C(CN(C)C)C(C)C)NCc1scc(CNC(C(C)=NOCC#N)=O)n1 C1(CNC(C(C)CF)=O)CN(C(=O)C=Cc2ccc(Br)cc2)CC1(C)C c1(C(C(=O)N(CCOCCCF)C2CC2)N(C(=O)CO)C)cccnc1 CCCC(C(=O)NCC(=O)OC)NC(=O)CC1CCCO1 N1(C(CCC2C(C)(C)C2)=O)CC(CNC(=O)CSc2cccnc2)CC12CCC2 O=c1oc2cccc(C(c3nnnn3C3CC3)NC3CC34CCCC4)c2[nH]1 C1(NC(C2CC(COCC)C2)=O)CC2(C1)CC2NC(CSC1CC1)=O.C(CC(=O)N)OC CC1(NC(c2cnc(O)s2)=O)CCCN(C(C2(F)CCOC2)=O)C1 C(C)(C(C)(C)C(=O)N1CCC(F)CC1)NC(C(CC)NC(N)=O)=O N1(C(C2(C)CC(C)C2)=O)CCCC2(C1)CN(C(=O)C(C)C(=O)N1CCCC1)C2.OCC CC1=C(C(=O)N(C2CN(C(=O)C(O)CC3CCOCC3)CC2(C)C)C)CCCO1 C(=O)(C1CCCc2ncc(C)n21)N(CC)CC1CCCN1C(=O)CN(C)C CC1CCC(NC(=O)Cn2nnnc2-c2ccsc2)CN1C(=O)CC(C)(C)C c1(CC2C(CNC(N3CCC(C(C)(C)C)C3)=O)C2)cccc2ccncc12 CC(CS(C)(=O)=O)C(=O)N1CCC(NC(=O)CCC2OCCO2)C(C)(C)C1 c1(C(=O)NCCC(C)NC(C(C)N2CCC2)=O)cc([N+](=O)[O-])cnc1O c1(CCC(=O)NC(CNC(C(C)SC(C)C)=O)C(C)(C)C)cnc2ccccn12 O=C(CCCCCCCCCO)NCCC1(NC(c2cn3c(n2)SCC3)=O)CC1 N1(C(CC2N(CC)CCOC2)=O)CCOC(C)(CNC(=O)CNC2CCCC2)C1 CC1=C(C)CC(C(N2CCC(O)C(NC(=O)C(F)(F)CN(C)C)C2)=O)CC1 C1(NC(c2c(CC)nco2)=O)CCCN(Cc2ccc(Cl)cc2C)CC1 CC1(C)CCN(C(=O)Cc2cnccn2)CC1CNC(=O)Cn1ccnn1 N1(C2C(CC)C2(C)C)CCN(C(=O)C(F)CCCNC(=O)OC(C)(C)C)CC1=O N1(C(C(C)=CC)=O)CCCn2nc(C(=O)NC(c3ccccc3F)CC)cc2C1 C1(NC(C2CCC(NC(C)=O)CC2)=O)COCCN(C(C2CSC(C)=N2)=O)C1 C(=O)(CCC(C)(C)C)NCC1C(C(=O)Nc2c(OC)nn(C)c2)CCO1 C(CC(O)C(=O)NCC(C)(C1CC1)NC(=O)COCc1cc(C)no1)NC(C)=O C1(NC(C2CC(=C)C2)=O)CCCN(c2cncc(C(=O)OC)n2)CC1 Cc1n[nH]c(C)c1C(C)C(=O)NCCCCCN(C)C(c1ccncc1)=O Cc1cc(C(CNC(C2COCCO2)=O)NC(c2nccnc2O)=O)cc(F)c1 C(=O)(CCC(=O)NN(C)C)N1CCN(CC2CC(C(=O)OC)CC(CN)C2)CC1 C1(C(C(C)C)NC(=O)CN2CC(C)C2)CCN(C(=O)C(C)n2ccnc2)CC1 N1(C(C2(CCC=C)CC2)=O)CC(CC(N2C(CO)CC2C)=O)C2(CC2)C1 N1(C(CC(C)OC)=O)C2CCC1CN(C(C1(n3cccn3)CC1)=O)C2 C(=O)(C(C)N=c1cc[nH]cc1)N1C(C)CCCCC1.C12C3CC4C(C3)C14C(=O)NO2 n1(CCC(C)C)cc(C(=O)NC2CC(N(C)C)C2)nn1 Cc1cc(NC(C2CC(F)CN(Cc3cc(O)cc(F)c3)C2)=O)c(I)cc1F N1(C(C2C(SCC)CCCC2)=O)CCN(C(=O)Cc2ccc(Cl)c(F)c2)C(C)C1 c1(NC(N(C2CCN(C(c3ccc(C)cc3)=O)C2)C)=O)cc2c([nH]1)CCCC2 Cc1[nH]c(=N)sc1C(=O)NC1CCCC1NC(c1ccccc1C1CC1(F)F)=O c1(C(=O)NC2C=CCN(C(C(CC(C)C)O)=O)C2)ccc([N+](=O)[O-])cn1 C1(NC(c2cnn(CC)c2C)=O)CC2CC1CN(C(C1CC1C(F)F)=O)C2 C12(NC(C3C(C)(C(C)C)C3)=O)CCOC(CNC(c3cnc4n3CCS4)=O)(C1)C2 C(C)(CN=c1nc(N(C)C(=O)OC(c2ccccc2)C)c2[nH]ccc2[nH]1)OC C(CN=C(NCC(c1cccc(Br)c1)(C)O)NC1CCCC1(F)F)SC N1(C(C=CC(C)(C)NC(c2cnn(C(F)F)c2)=O)=O)CC2(CCCC2)C1 c1(C(=O)NCC(C)N(C)C(C2CCC2C)=O)cc([N+](=O)[O-])n[nH]1 c1(C(=O)NC2CC(NC(C3(CC4CC4)CC3)=O)C2)ccc(-c2cn[nH]c2)s1 N1(C(CNC(=O)NC)=O)CCC(C(C)NC(=O)Cc2c[nH]nc2C)C1 C1(CCNC(=O)CCOC2CC2)(C(=O)NCC2CCCCC2)CCOC1 C1(NC(c2ccn(C(F)F)n2)=O)CCCCCN(C(c2ccnn2CCF)=O)C1 C1(CNC(COCCCCC)=O)CC(O)CN1C(c1cscc1C)=O C1(C)(CC)C=C(C(=O)N2CCOC(C(C)NC(=O)CCN3CCC3)C2)C1 C1(CC)CN(c2ccccc2)CCN1C(c1[nH]cnc1C)C(=O)NCC c1(NC(c2c(CC)scn2)=O)cccc(NC(C2C3CCCC23)=O)c1 C1(O)(C(C)NC(CCOCC)=O)CN(C(C2CCC(COC)O2)=O)C1 C(CC1CC1)(C(=O)NCC1CCCC1O)NC(=O)CSC1(c2cc[nH]n2)CC1 N1(C(CCC(C)(C)C)=O)CCN(C(=O)CNc2ccccc2)CC(O)C1 N1(C(c2cc(COC)[nH]n2)=O)CC(CO)C2(C1)CN(C(c1cc(OC)ns1)=O)C2 c1(C(=O)NC2CCC(C)N(c3ccnc(C4CCC4)n3)C2)ccc([N+](=O)[O-])cn1 Cc1cc(C)c(C(=O)NCC2CCCC2NC(=O)CNC(=O)CN(C)C)c(O)n1 NS(=O)(=O)c1cccc(NC(C2C3CN(C(C4(Br)CC4)=O)CC23)=O)c1 C1(CC)(CO)CCN(C(=O)C(CCC)NC(=O)C(CO)N(C)C)C1 C(C1CCOC1)=CC(=O)NC(C1CCCC1)CNC(C1CC1C1CCCCC1)=O c1(OC)ccc(C(=O)NC(C2CCCN2C(c2cnoc2C2CC2)=O)C)cc1F CN=c1nc(N(C2COCC2N2CCOCC2)C)[nH]c(=NCCNCC2CC2)[nH]1 c1(C(C)NC(CN(C(=O)OCC)C)=O)nocc1C(N1CC(N(C)C)C1)=O CC(CC(=O)NC12COC(CNC(C3(O)CCCC3)=O)(C1)C2)C(F)(F)F C(c1ccc(F)cc1F)=CC(=O)NC1CCCC1NC(C1CN2CCC1CC2)=O c1(C(=O)NCC(CNC(C(N2CCOCC2)C)=O)CO)ccc2c(c1)OCCN2 C(=O)(CC1=CCN(C(C2(C)C=CCC2)=O)CC1)NC(C1(CO)CC1)C N1(C(CC2N(C(C3CCN(C)C3=O)=O)CC2)=O)CC2C=CC1CC2 N1(C(Cc2c(C)nn(C)c2)=O)CCC2(CCN(Cc3nn(C)cc3Br)C2)C1 N1(C(c2c(CC)noc2C)=O)CCN(C(C2CC(=O)N(C)C2)=O)C(C(C)C)C1 N1(C(C(=O)NC(C(=O)OC)C)COCc2ccccc2)CCCC(N(C)C)C1 c1(NCC2CCC2)ccc(S(=O)(=O)NCC(c2ncccc2F)C)cc1F C1(NC(C2(C)CC(C)(C)C2)=O)CCN(C(c2cnn(C3CC3)c2)=O)CC1O c1(CC)cncc(C(=O)NCC(C)N(C(=O)Cc2ccon2)CC)c1 C1(C(=O)NCCC(CC)C)CN(C(C2CCC(=O)C2)=O)CC1C C1(NC(=O)NC(c2csc(C3CC3)n2)C)CCCN(CCN2C(=O)CCC2=O)C1 C1(NC(=O)Cc2cncnc2O)CN(C(c2c[nH]ccc2=O)=O)CCC1O C1(C(=O)NC(C2CCN(C(=O)C(C)(C)SCC#N)CC2)C)CC2CCC1C2 c1(C(=O)OC)c[nH]ccc1=NC(CNC(c1cnn2c1OCC2)=O)C(C)C(C)C c1(C(=O)NCC(CC)NC(c2ccc(C(C)(C)C)[nH]2)=O)ccc(Br)s1 CC1CN(C(c2c[nH]nc2Br)=O)C(C)CN1C(c1cc(F)n[nH]1)=O c1(C(=O)NCCC2N(C(CCSCC)=O)CCCC2C)cc(C)c(F)cc1N c1(C(N(CCCCN(C)C(C2(C)C=CCCC2)=O)C)=O)c(Cl)cnn1C Cc1cccc(CNC(C2C=CCN2C(=O)COC2(C)CCC2)=O)c1F C(=O)(C(C)C(=O)N1CCC(C(=O)N(C2CCCCCC2)C)(CF)C1)OC N1(C(CCCOCCOC)=O)CCN(C(c2cn(C)nc2Cl)=O)C(CO)C1 C1(NC(CN(CC)CC)=O)CC2CCC1CN(C(=O)C=CCO)C2.c1(N)ccccc1 C1(C(=O)NCCC(C)OC)CC1C1CN(C(c2ccc(C)c(F)c2)=O)C1 N1(C(C2OCCC2C(=O)O)=O)CCC(CCC(=O)NCCOC2CCC2)C1 Cn1ccnc1C(N1CCC(CNC(=O)Cn2cc(Cl)cn2)C1)=O c1(CC(=O)NCCN(c2ccccn2)C(CC2C(C)(C)C2)=O)cc2ccccc2s1 Cc1ccc(CC(=O)NCC(C2CC2)NC(C2CCC2C(F)F)=O)cc1Br C12=NC=CC(=NCN1)N2.c1(OCC2(CN(C)C)CC2)ccccc1 c1(OC)ccc(C(N2CC(O)(C(C)NC(c3csc(C)c3)=O)C2)=O)c(F)c1F c1(C(=O)NCc2ncoc2C2CC2)ncc(Br)cc1I C(C(C)(C)CC(=O)N1CC2(CCOC2)C1)NC(C(COCC)C)=O Cn1ncc2c1CC(CNC(=O)CC1CCCO1)CC2 c1(OC)cc(C)nc(NC23CC2CN(Cc2nc[nH]c2C(C)(C)C)C3)n1 C1(CC(C)(C)C)CN(C(c2ccoc2)=O)CC1NC(C1CC1c1ccccc1)=O C(N=c1[nH]c2ccc(Br)cc2s1)C1(N2CCOCC2)CCCC1.O=C1C=CCN1 c1(OCC)cc(CN2CCNCC2COCC(C)C)ccc1OC Cc1cc2[nH]c(C(=O)NC3CN(C(c4ccoc4)=O)CC3C3CC3)cc2s1 CC1OC2CCC1(C(=O)NC1CC3(C(N4CC5CC4CC5O)=O)COC1C3)C2 C1(CNC(c2n[nH]cc2[N+](=O)[O-])=O)CCN(Cc2cc(F)ccc2O)CC1(F)F C1(CNC(C2(C)C(C(=O)OC)C2)=O)CCN(C(=O)Cc2ccc(Cl)nc2)CC1 Cc1cc(C(=O)NCC2CCCCC2NC(=O)COCC2CC2)ncc1Cl CC1CN(C(=O)CCC2CCC(=O)N2C)CC1CNC(=O)COc1ccccc1Cl c1(C(=O)NC2C3CN(C(c4cccc(CC)c4F)=O)CC32)cccc2nonc12 CC1(NC(C2CC(NC(=O)CC3CC4(CC4)C3)C2)=O)CCC(O)CC1 c1(CNc2ccc(C(N(CCOC)C)=O)nc2)cc(N)c(OC)cc1F C1(NC(c2cnn(C)n2)=O)CCCCCN(C(c2cccc(NC(N)=O)c2)=O)C1 c1(C(=O)NCC2(NC(CCC3CCC(=O)N3)=O)CCOCC2)csc([N+](=O)[O-])c1 C1(CNC(C=CCN(C)CC)=O)CCN(C(=O)C=CSc2nc[nH]n2)CC1O C1(CN(C(C(C2CCC2)OC)=O)C)CCCN(C(=O)COCCCF)C1 C=CCC(C)NC(=O)CC1CCN1C(=O)C(C)OC(C)=O C(CO)(C(C)NC(c1sccc1OC(F)F)=O)NC(C(C)OCCC(C)C)=O C(C(C(C)C(C)C)NC(=O)CCCC(OC)OC)NC(CCCC)=O C1(C(N2CC(OC)C(NC(C3CC3C#N)=O)C2)=O)CC2(C1)CC(O)C2 N1(C(C2N(CC)C(=O)CC2)=O)CCC(NC(=O)Cc2ccns2)C(C)C1 C#CCCCC(=O)NC1(CNC(c2ccn(CCC)n2)=O)CC1 N1(C(c2c(C)cccc2O)=O)CC2CCC1C(NC(=O)Cc1cc[nH]n1)C2 c12ccc(nc1N)CNC2=O.C1(CN)CC2C=CC1C2 N1(C(C(n2ncc(C)c2)C)=O)CCC(C=CC(N2CCCC(C)C2CO)=O)CC1 Cc1nc[nH]c1CNC(C1CN(C(=O)C(C2CCOCC2)O)C1)=O Cc1cc(Cl)ccc1C1CC1NC(=O)C(N)c1ccsc1 c1(C(=O)NC2CCCC2C(=O)NCCN2CCNC(=O)C2)cc2ccccn2c1 Cc1ncc(CCCC2(C)CCCC2)o1.C1(C2(CN)CC2)CC1(C)C Cc1cccc(OCCC(=O)N(CCC(c2cccs2)NC(=O)C(C)(C)C)C)c1 N1(C(C2CCC(OC)C2)=O)CC2CC(C1)N(C(=O)CCC1=CN1C)C2.C(=O)(CO)N c1(OC)ccc(CC(=O)N(CC(C)NC(=O)C(C2CCCCC2)O)C)nc1 CC1c2cc(F)ccc2CCN1CC1CCC(C)C1 c1(C(N(C(C)(C)C)C(C)Cc2cnc[nH]2)=O)cnc(C2CN(C)C2)o1.Cc1ccc[nH]1 Cc1ccc(CCC(=O)N2CC(NC(=O)CN(C)C3CC3)C2)c(C)c1.CC=O O=S(=O)(c1nc2ccccc2n1C1CC1)NCc1cccc2c1COCC2 C(=O)(CC(C)C(F)(F)F)N1C2CN(C(Cn3c(C)nnn3)=O)C(C2)C1 N1(C(C=C(CC)CC)=O)CCCC(O)(CNC(c2cc(Br)cnc2O)=O)C1 Cc1cccc(CC(=O)NCC2(CNC(c3csc(CO)n3)=O)CCC2)c1 c1(CCC(=O)NC2C=CC(CNC(C3CC(C)C3)=O)C2)cccc(F)c1F C1(C(N(CCC)OC2CCCC2)=O)CC2CN(C(C34C=CC(CC3)C4)=O)CC2C1 c1(N(C2CCCN(C(=O)C(F)F)C2)C)nc2cc(F)ccc2o1 C(=O)(NNc1ncccc1C)C1(C(=O)OCC)CNC1 C1(C(=O)NC2C(OCC)CCC2)C(C)CCCN1C(C1(C)CCOC(C)C1)=O N1(C(CCC(=C)C)=O)CCC2CCCN(C(=O)Cc3nccn3C)C2C1 c1(C(=O)NCC#CCNC(C2C(OC)C2)=O)cc(Br)c2[nH]cnc2c1 c1(SC)cccnc1C(=O)NC(CNC(C1CSCCS1)=O)C1CCC1 C1(C(=O)NC(C)CO)CCCN(C(=O)CCCc2ccccc2Cl)C1 c1(C(=O)NCC(C)(C)NC(CC(CCCC)O)=O)ccc2c(c1)CN(C)C(=O)N2 C1(NC(CCOCCOC)=O)CCN(C(C2(CO)CCCCO2)=O)CC1O O=C(C(=O)NCC1(COC)CCC1)NCC(=O)C1CC1.C1(CC(N)=O)(N)CC1 C1(c2n(-c3cc(C)cc(C)c3)nc(C3CC4CCC3C4)n2)CC(=O)CC12CCC2 C1(C(=O)Nc2cncc(C#N)c2)CC2(CCN(S(=O)(=O)CCCCCl)CC2)C1 C#Cc1cc(NC(=O)NN(C)CCOC(C)C)cc(F)c1 C1(CNC(C2CCN(C(C)=O)C2)=O)CCCCN(C(C2(F)CC=CC2)=O)C1 C1(C(=O)NC(CN(C(C(C(=O)NC)(C)C)=O)C)C)CCc2ncncc2C1 C(=O)(CC(C)C(C)(C)C)N(C(C(=O)NC(CCCC)C)CCC)C c1(C(=O)NCC(C2CC2)NC(C(C)OC2CC2)=O)cccn1C1CCCC1 CCC(CCC(=O)NCCC(=O)OC)NC(C1CC1CCCOC)=O c1(C(=O)NC2CN(C(C3(C#N)CC34CCC4)=O)C2)cnc2c(c1)CS(=O)(=O)CC2 NCCCCCN(c1ccccc1)C(C1CCCSC1)=O C(=O)(CC(O)CC(C)(C)C)N1CCN(C(c2cncc(SC)c2)=O)C(C2CC2)C1 N1(C(c2c(CC)nn(C)c2CC)=O)CCC2(CC1)CC(NC(=O)C1=CCC1)C2 C(N=c1[nH]c(=NCCC(F)(F)F)[nH]c2cccnc12)C1COCC(C)O1 N1(C(c2cncc(C)c2)=O)CC(O)CCC1C(=O)N(C)Cc1ccsc1 C(=O)(CCC(C)(C)NC(C1CN2CCC1CC2)=O)NC(CCOCC)C c1(C=O)ccc(F)nc1F.N12CC(C(C)(C)C1)N2C.C1(C(F)(F)F)(C=O)CCC1 c1(CN2C(C)CCC2C(=O)Nc2c(O)cccc2Cl)ccc(I)c(F)c1F C1(NC(CCOCCOC)=O)CC(CC(=O)N(C2CC(C)(C)C2)C)C1(C)C N1(C(=O)COC2CCOCC2)CCOC2(C1)CN(C(c1ccc(=O)n(O)c1)=O)C2 C#CC1(C)CCN(C(C2CC(OC)CN2C(=O)CSC(F)F)=O)CC1 N1(C(Cc2ncn(C)c2)=O)CCC(C(=O)NC2CN(C(N)=O)C2)CC1 N1(C(c2c(C=C)cccc2)=O)CC(C2CCCN(C(c3cscc3Br)=O)C2)C1 N1(C(C2C(C)(C)CC2)=O)C2CCC1CC(NC(=O)CN1CCn3ccnc3C1)C2 N1(C(=O)Cc2cccnc2Cl)CCC(CF)(NC(=O)C(c2cccc(F)c2)O)C1 c1(C(=O)NC(C(=O)NCC(C)OC(F)F)CCF)cn(C)c(=O)n1C c1(C(N(C2CN(C(C3OCCN(C)C3)=O)C2)C)=O)ccc2[nH]ccc2n1 Cc1cc(C(N2CCC(O)(C(C)CNC(=O)COCC(C)(C)C)C2)=O)cn1C N1(C(CSc2ccc(C)c(C)c2)=O)C2CCC1CN(C(C1(C)CC1(C)C)=O)C2 C1(CC)C(NC(C2CCC(C)C2)=O)CCCN1C(=O)CNC=O N1(C(C(CC(C)C)NC(c2n(CC)ccn2)=O)=O)CCC(F)(F)C(O)C1 Cc1ccc(C(C)C(=O)NCCCNCC2CSCCS2)cc1 CC(C)C(C)(CNC(=O)CCCc1ccccc1)NC(c1cc(C2CC2)on1)=O Cc1ncc2c(n1)NCCNC2.C1(C(=O)NC)CCNCC1 c1(C(=O)OC)ccc(CN2CCC(O)(C(=O)Nc3cncnc3Br)C2)cc1 Cc1cn2ccnc(C(=O)N(C(C)CNC(c3cccn3C)=O)C)c2n1 C12(CNC(c3n(CC=C)nnn3)c3ccn(CCF)n3)CCC(CC1)CC2 c1(C(=O)NCC(C)C)cc2ccc(-c3ccc(CO)nc3)nc2[nH]1 C1(NC(c2cnc(CC(C)C)nc2)=O)CN(C(=O)Cn2cnc(=N)[nH]2)CCC1C c1(C(=O)NCCOCCN(C(=O)C#CC2CC2)C)cc(Cl)nc(Cl)c1 c1(C(N(CCC)CCNC(c2cn(CC)nn2)=O)=O)c(O)cc(Br)cc1F C1(NC(c2csnn2)=O)CCOC(C(=O)NCC2CCCCC2)C1 c1(C(=O)NC2CCC(CNC(c3ccc(OC)nc3)=O)C2)cc2c[nH]cnc-2n1 C1(CNC(=O)CC2CC2)CN(C(C2CN(C3COC3)C2)=O)CCO1 c1(CNS(N)=O)ccc(N2CCC(c3cccnc3)CC2)cc1 C1(C(=O)NCC2(F)CCN(C(CCNC(=O)NC)=O)CC2)CCC2(CCC2)CO1 S(=O)(=O)(c1cc2sc(=NC3COC(C)(C)C3)[nH]c2cc1Cl)NC1(CC)CCOC1 c1(C(=O)NCC2CCC(NC(C(C)(C3CC3)OC)=O)C2)ccccc1SC(F)F Cc1ccnnc1C(N1CCCC(C(=O)NCCc2noc(C(C)(C)C)n2)C1)=O c1(C(=O)NCC2C3CN(C(CC(C(C)C)C)=O)CC32)cc(F)c2ncccc2c1 c1(C(N2C(C)CC(NC(c3c[nH]c(=O)cn3)=O)C2)=O)cc2ccc(O)cc2n1C N1(C(C(C(C)C)NS(N)(=O)=O)=O)CC2(C1)CN(C)C(=O)CO2 C1(C(N2CCC(OC)C2C)=O)CN(C(=O)CC2CC(C)C2)CC(C)(C)C1 N1(C(COC)=O)CC2CC(NC(C3CC(=O)N(C)C3c3ccccc3)=O)CC2C1 O=C(C1=CCCC1)OCC(N1CCC(N2CCOC2=O)CC1)=O C#CCCCC(=O)N(CC(C)NC(=O)Cc1cncc(Br)c1)CC c1(C(=O)NC(COC)C)csc2c1CCN(C(c1ccncc1F)=O)C2 c1(C(N2CCC(C3N(C(C(C)OCCCC)=O)CCC3)C2)=O)cccnc1O C=CC(C)CC(=O)N1C(C(=O)NCC2(F)CC(CO)C2)CCC1C(C)C C1(N(C(CC2(N(C(C(CC)OC)=O)C)CC2)=O)C)CCCC(C)C1C C1(C(=O)NCCNC(=O)CCC2OCCO2)CC2(CC2)C1 C1(NC(CCCCSC)=O)CC12CCC(NC(=O)Cc1ncc(C)[nH]1)CC2 C(CCC(C)C(=O)N1CCC(OCCNC(=O)C(C(C)(C)C)N(C)C)C1)OC C(=O)(CC(C)F)NC(COC)C(=O)NC1CC1C1CC1 C1(C(N(C2CCCCC2)CC)=O)CC(NC(=O)CCC2CC2)CCO1 N1(C(C)=O)CCCC(C(C(=O)CNS(=O)(=O)C2CC2)=O)C1.C1(N)CCC(NC)CC1 CC(C)C(C(=O)NCc1noc(-c2ccccc2)n1)SCc1ccccc1 c1(SCC#C)cccc(C(=O)N(C2CC2)CC2(O)CC(C(=O)OC(C)=O)C2)c1 N1(C(c2c(C)ncs2)=O)CCCC2C1CCN2C(=O)C1=COCC1 c1(C(=O)NCC=CCNC(=O)C(F)CC2CC2)ccc2ccoc2c1 C1(NC(C2CC(OC)C2)=O)COCCC1NC(c1ccnc(-n2cncn2)c1)=O c1(OC)c(C(=O)Nc2ccccc2)cccc1C(N1Cc2c[nH]nc2C1)=O C(=O)(C(C)CC(N)=O)N1CCN(CC(=O)NCCC(C)OC)CC1 C(=O)(C(O)CC(C)(C)C)N1CCC(C)N(C(=O)Nc2cnn3c2C(=O)NCC3)CC1 c1(C(=O)NC2(CNC(C3C(C)(CC)C3)=O)CCOCC2)cc2n(n1)CCCCO2 c1(OC)ccc(CCNC(c2cc(-c3ccc(C)c(N)c3)[nH]n2)=O)c(C)c1 C1(CNC(Cc2cccc(OC)n2)=O)CC(N=c2[nH]c3c(C)cccc3o2)C1 C=CC(C)N=c1nc(N2CCC(N3CCCCC3)C2)c2c([nH]1)CSC2 C1(CNC(C(c2ccc(Cl)cc2)(C)O)=O)CN(C(c2ccoc2)=O)CCC1(F)F C(=O)(C(C)(C)CCS(C)(=O)=O)NC(C)C(CO)NC(c1cc(N)c(F)cn1)=O C1(CC(=O)NC(CC)CO)C2CCC1CN(C(=O)NCCCCc1cncs1)C2 C(=O)(C1=NNC(=O)C1)NC(C(CO)NC(Cc1cccc(OCCC)c1)=O)C C1(COC(C2N(C(=O)OC(C)(C)C)CCC(O)C2)=O)CC2(C1)CC1CCC2C1 C1(C(=O)NCC2(C)CCN(C(C3C(C)(C)C3(F)F)=O)C2)CC2C(C1)C2(F)F C1(NC(=O)C(C)(C)F)CCCC(CN(C(=O)CC(C)(C)C2CC2)C)C1 N#Cc1cc(C(N2CC(O)CC2C(=O)Nc2c(F)cc(Br)cc2F)=O)ccc1O C1(CC)CC(C(=O)NCC(CNC(c2sccc2C(F)F)=O)OC)CCO1 N1(C(c2cnn(CC)n2)=O)CCC2(C1)CN(C(=O)CCCCC(=O)NC)C2 CN1C(=O)c2c(N3CCC(NC(=O)C(N)=O)C3)ncnc2C1=O N1(C(c2c(OC)nn(C)c2)=O)CCCC(C)C1CNC(c1ccc(N)cc1F)=O c1(C(N(C2CN(C(C(CN(C)C)(C)C)=O)CC2O)C)=O)cccc2cccnc12 N1(C(C2CCC(C)(F)CC2)=O)CCCN(C(C2CC3(CC3)CO2)=O)CCC1 C1(C(=O)NC2CC(CNC(C(CCC)OC)=O)C2)CCCCC1C1CC1 c1(OC)nc(C)cnc1C(=O)NC(CO)CCCCNC(=O)C(C)SC CN=c1[nH]c(C(N2CC3CC3(NC(c3cc(C(C)C)on3)=O)C2)=O)cs1 c1(C(N2C(CNC(C3(O)CCOC3)=O)CC(C)(C)C2)=O)nsc2c(Cl)cccc12 C1(CNC(c2cnc(SC)s2)=O)CC(C)(C)CN1C(=O)Cc1coc(C)n1 C1(C(=O)NCCCNC(C(C)OCC#C)=O)CCCCN1C(=O)OC(C)(C)C CN1CCc2nc(C(=O)N(C3CCCC(NC(=O)Cn4ncnn4)C3)C)sc2C1 N1(C(CSc2cn(C)nc2)=O)CCC(C)(NC(=O)C(F)C(C)(C)O)CC1 c1(OC)ccc(Br)nc1C(c1nnnn1C1(C)CC1)NCC1CCCCC1C Cc1cc(F)c(Cl)cc1C(=O)NC1CCN(C(C2CC23CCOCC3)=O)CC1F C(=O)(CCCCCF)NC(CCCC)CNC(=O)C(c1ccccc1)C1CCCC1 c1(CC)ccc(NC2(c3nnnn3CC3CCCO3)CCC(CC(C)C)C2)cc1 N1(C(C2C(C)(C)CCN2C(c2ccc(F)c(F)c2)=O)=O)CCC2(CCCC2)C1 c1(C(=O)NCc2cn(C3CCN(C(C4CC4F)=O)C3)nn2)cc2c(=O)cc[nH]c2s1 c1(OC)cccc(Cl)c1C(=O)NCC1CCN1C(c1ccsc1C#N)=O CC1CN(C(=O)COc2cn(C)cn2)CCCN1C(=O)CC1CCC(F)(F)CC1 C12(C(=O)NCCN(C(C3CN4CCC3CC4)=O)CC)CC3CC(C1)CC(O)(C3)C2 CCC(C)CCC(=O)NC1CN(C(c2c(C)coc2C(C)C)=O)CC1SC C1(NC(CC(=O)N(C)C)=O)CN(C(=O)CCC(F)(F)F)CCC12CCOCC2 c1(C(C)C(=O)NC2(CO)CCCN(C(=O)Cc3ccoc3)C2)ccc2c(c1)OCO2 c1(C(=O)NCC2N(C(C3C(CC)CCC3)=O)CC(C)(C)C2)cc2ccncc2o1 C(=O)(C(CCCOC)NC(=O)CC1(C)CC1)N1CCC(CCC)(CO)C1 C#CCCCCCC(=O)N1CC2C(CNC(c3cc(S(C)(=O)=O)cs3)=O)C2C1 c1(C(=O)NC2CCC2NC(c2csc(F)c2)=O)cnn2c1CCC2 Cc1c(C(N2CCCCC2CNC(C2CC3CCC2O3)=O)=O)cnn1CCC#N N1(C(C(=O)NCC(c2cccc(OC)c2)(C)C)C(C)C)CCOc2ccccc21 C1(N(CC(=O)N(CC(=O)NCCC)C)C)CCN(C(C2CCCC2)=O)CC1 c1(C(=O)OCC)sccc1S(=O)(=O)N1CCCCC1C(CO)CO Cc1cc(NC(C2CC2[N+](=O)[O-])=O)ccc1NC(c1nn(C)c(Cl)c1Cl)=O N1(C(c2ccc(OC)nn2)=O)CCC2(CCCC2NC(=O)CSCCC(C)C)C1 C(C)(C)(CC(=O)NCCC(C)CCNC(c1cscc1C)=O)SC c1(C(=O)NCCCN(C)C(c2c(F)cc(F)cc2Cl)=O)cc(Cl)cc([N+](=O)[O-])c1 c1(C(=O)NC23CC(NC(CC(C)C4CCCO4)=O)(C2)C3)ccc(Cl)cc1F C(=O)(C1=CCS(=O)(=O)C1)N1C(CN(C(=O)CCC2CC(C)(C)CO2)C)CCC1 O=S(=O)(N1CCC(OCC(F)F)CC1)N1CCc2cc(Br)c(F)cc2C1 c1(C(=O)NC(CC)CNC(c2csc(-c3cccnc3)n2)=O)cc(OC)ccc1F c1(C(=O)NC2CN(C(=O)CC3CCSCC3)CC2O)ccn2c1CSCC2 CN1CCC(N)(C(=O)NCC2CCCC2C(C)(C)C)C1 N1(C(c2cnnc(Cl)c2)=O)CCC2(CCCC2CNc2cc(O)ncn2)CC1 c1(OC)ccc([N+](=O)[O-])c(N2CCCC2c2ccc(F)cn2)n1.C1CC1 Cc1ccc(C(=O)NC(C2(O)CN(C(C3CCC(C)(O)CC3)=O)C2)C)nc1C C1(N)(CN2CC(CCn3cc(C(C4CCCCO4)C)nn3)C2)CCCS(=O)(=O)C1 C(C(=O)N(CC(=O)NCC(c1ccncc1)C)CC)(C(C)C)OCC CC(CCNC(N)=O)C(=O)N1CCCC(Cc2cn(C3(C)CC3)nn2)C1 Cc1cc(C(=O)NCC(C(C)(C)C)NC(=O)C(c2ccncc2)C)c(C)o1 C1(NC(c2cc(CC)ncc2)=O)CN(C(=O)C(C)(O)CC)CC1N=[N+]=[N-] C(CCC(=O)NCC(O)Cc1cccnc1)NC(CNC(CNC(C)=O)=O)=O C1(CC(=O)NCC(CNC(C2(COC)CC2)=O)O)CCCCC12CC2 C(CCCCC(=O)NCC(C)C)N(C(C(CC)(C)C)=O)C Cc1cc(NC(C2CC3(CC3)CN2Cc2ccnc(Cl)c2Cl)=O)ccc1O c1(C(C)C)cccc2c1CCC2NCc1cc2c(O)nn(C)c2s1 C1(NC(CN(C)CC)=O)C2CN(C(c3ccc(-n4cccn4)nc3)=O)CC12 C(=O)(C1Cc2ccc(Cl)cc21)NC(C(C)NC(C1CCC(C)(F)CC1)=O)CO Cc1cc(N2CCCC2CS(N)(=O)=O)nnc1C Nc1ccc(C(=O)NCC2CCCC2NC(=O)CC2CC(=O)C2)cc1N c1(C(=O)NCC(CCOC)NC(C2C3C4CCC(C4)C23)=O)cnn2c1OCC2 c1(C(=O)NCC(C)N(C(c2c(COC)nn[nH]2)=O)CC)nc(OC)ccc1Cl c1(C(=O)NCCC2CSCCN2C(C2C3CCC23)=O)ccc2n[nH]cc2c1 N1(C(C(CCC)NC(=O)CC2(O)CCCOC2)=O)C2C=CCC1CCC2 C1(C(N(CCN(C)C(C2(C)CCNC2=O)=O)C)=O)COC2(CCC2)C1.CCO Cc1ccc(NC(C2C3CC2N(C(c2c[nH]c(C(N)=O)c2)=O)C3)=O)cc1Cl N1(C(C2(COC)COC2)=O)CCC(C2CC2)C1Cn1cc(CC(C)(C)O)nn1 C(C(C(C)C)NC(c1cc(F)c[nH]1)=O)NC(C(C)OCCOC)=O c1(N2CCN(C(CC(COC)(C)C)=O)CC2CCO)nc(C)nc(O)c1C C(=O)(CC(F)(F)F)NCCC(C)N(C)C(c1ccc(C(F)(F)F)cc1)=O C(C(=O)N(O)Cc1cn(C2CC3CCC2CC3)nn1)(C(C)C)OC(C)=O C1(C2CCOCC2)(C(N2CC(NC(Cc3cnc(C)o3)=O)C2)=O)CC1(F)F c1(C(N2CCN(C3CCC3)CC2)C(=O)NCC(=C)C)ccc(CC)cc1F c1(N(C)C)ccc(CNc2cc(C(=O)NCC(C)(C)CO)n(C)c2)cn1 N1(C(C2ON=C(C)C2)=O)CCCC(OCCN)C1 CC1COCC(C(=O)NCCN2CCN(C(c3ccc(C(F)F)s3)=O)CC2)O1 C1(NC(C=CC)=O)CC2CC(C1)N(C(c1cc(C(C)CC)no1)=O)C2 C=C(C)CC(C(=O)NCCOc1ccncc1)NC(C1COCCN1C)=O c1(C(=O)NC2CC(NC(C(CCC)CC3CCCC3)=O)C2)cn2ncccc2n1 C1(NC(Cc2c(C)nsc2)=O)CCCC(C(=O)NCCCCN(C)C)CC1 C(C)(CCC(=O)NC(c1cnn(C)c1)C(=O)NCCC1(C)CC1)OC C1(NC(C2(CC=C)CC2)=O)CN(C(c2nncn2CC2CCC2)=O)CC1C(F)F C1(NCc2cc(C(N3CCC(CN(C)C)C3)=O)sc2)CC2CCC1O2 N1(C(=O)CCc2ccc(F)cc2)CC2CC(C1)CN(C(=O)C(F)(F)C(F)(F)F)C2 C(=O)(C1=C(C)OCCC1)NC(CCOC)CNC(c1n[nH]c(C)c1C)=O c1(OC)csc(C(=O)NCC2CN(C(C3CC(C)=NO3)=O)CCO2)c1OC c1(NC(C2CCC(NC(C(C)S)=O)C2)=O)ccccc1CC#N N12CCC3(CCCC13)N2.C(=O)(C1=CCCCCC1)C(c1scc(C)c1)=O C1(N(C(C)(C)C2(C)CC2)C)CCC(NC2CCOC2C)CC1 C(C)(C)(CC(C)(C)C)OC(C1CCN(C(C(C)C)=O)CC1)=O.N1(C)CC(C(=O)O)C1 C1(NC(c2n(CC)nnn2)C(C)(C)OCC)C2CCOC2C1(C)C C(N=c1[nH]c(=N)[nH]c(=NCCN(c2ccccn2)C)[nH]1)C1CCN(C)CC1 c1(C(N2CC(O)CC(NC(c3cnc(OC)s3)=O)C2)=O)ncnc2c1CCC2 C(=O)(C1=NNC(=O)C1)N1CC(NC(c2nccc(CC)c2)=O)(CF)C1 C(=O)(C(F)CCCC)NC1(CC=C)CCN(C(=O)CCc2ccoc2)C1 c1(C(=O)NCC(C)(C)NC(CS(CCOC)(=O)=O)=O)cc2n(n1)CCCC2O N1(C(c2c(CC)nns2)=O)CC(NC(C2(C#N)CCOC2)=O)CCC1C C(=O)(C(C(C)c1ccccc1)N(C(C)C(=O)N(C)C)C)NCCCOC N1(C(c2cc(C)sc2)=O)CCC(C)(C)C1C(=O)N(C)OC C1(C)(C(=O)NC(CC(F)(F)F)C)CCCN(C(=O)C(=O)NCc2nccn2C)C1 CC(N=c1ccnc(NCc2cc(N)ccc2Cl)[nH]1)c1nc[nH]n1 CC1CN(C(=O)C(CNC(C2CC(C3CC3)=NO2)=O)CC2CCCC2)CCN1C CC1C(O)CCCN1C(=O)Cc1csc(NC(c2ccccc2F)=O)n1 c1(C(C(=O)NC(C2CN(C(C3CN(C(C)C)C3)=O)C2)C)C)ccc(C#N)cc1 Cc1cc(C(=O)NC2CN(C(=O)CCc3ncco3)CCC2C)nc(O)c1 CCCC(CC)CCCC(=O)NCCCN(C)C(C1CC(=O)N(C2CC2)C1)=O Cc1noc(C)c1C(C)C(=O)NC1CC1NC(c1cnc(C)n1C)=O c1(C(N(CCC(C(C)C)NC(C(CC(=C)C)C)=O)C)=O)cc2cnn(C)c2s1 c1(NC(c2n(C)cc(Nc3cc(COC)ncn3)n2)=O)ccc([N+](=O)[O-])cc1 c1(C(=O)NC(C(=O)N(CCCC)CCCC)C)ccc(CC)s1 CCCC(CC)C(=O)N1CCCCCC1CNC(c1ncc(C(F)F)s1)=O CCCCCCC(=O)N1C(C(=O)Nc2cc(O)c(C)cc2C)CC2CCCC12 C=CCCC(C(=O)NC(c1cnc[nH]1)C)NC(=O)CCCCC N1(C(C(CC)COC)=O)CCCC(O)(CCNC(C2(CC(C)C)CC2)=O)C1 c1(NC(C2CCC(n3cc(C4CC4)nn3)C2)=O)cc(COC=CCl)ccc1F C1(NC(=O)OC)CCN(C(=NCC(C)(C)C2CCCCC2)NC(C)C)CC1 c1(CC(=O)NCC(C2CC2)NC(=O)CCC2CC(F)(F)C2)nc2c([nH]1)CCCC2 C1(CNC(Cn2c(C)cc(C)n2)=O)CN(C(=O)C(C)C(C)(C)C)C2(CCC2)C1 n12ccc3nc(ncc13)N1CC(C(C)C1)C2.c1(SCC)cc(Cl)cnc1Cl C1(NC(CCCn2cc(C(COC)(C)O)nn2)=O)CC(C)CC(C)(C)C1 N1(C(C(CCC)C#N)=O)CCC2CCN(C(c3oc(C)nc3C)=O)CC12 c1(OC)cc(Br)ccc1CC(=O)NCCN(C)C(c1cc(C)nn1C)=O N1(C(C(C)C2CCC2)=O)CC2C3CCC(C2C1)N(C(c1ncoc1C1CC1)=O)C3 c1(C(C(=O)NCCN(C(c2cc(OC)no2)=O)CC)C)cccc(S(C)(=O)=O)c1 N1(C(CN(C)C)=O)CC(NC(=O)CCCc2nncn2C)C(C)(C)C1 c1(CC(=O)OCC(=O)NCC(C)Sc2ccccc2)ncncc1Cl C(C1CCCCC1)=CC(=O)NCC(CNC(c1c(OC)csc1)=O)(C)F C1(C)(C(N(CCN(C(C(CO)NC(C(C)C)=O)=O)C)C(C)C)=O)CC2C=CC1C2 CC(C)C(CNC(C1CC1(F)F)=O)NC(=O)CC(C)n1cccn1 N1(C(c2cc(C#C)c(C)cc2)=O)CCC(C(=O)NC(C)(C)C)CC(C)(C)C1 c1(CC)cc(C)c(C(=O)NCC2CC(F)CN2C(=O)CCC2CC2(F)F)o1 N1(CCCN(C(=O)CCC2CCOC2)CCO)CCN(c2cc(F)ncn2)CC1 N1(C(C(C)CC(F)F)=O)CCC(C2CCOCC2)(CNC(C2(F)CCC2)=O)C1 C(N=c1[nH]c2c(c(=NCc3ncccc3N)[nH]1)SCC2)C1CC(C(C)(C)C)C1 C1(C(=O)NCC2(CNC(C(C)(C(C)C)OCC)=O)CC2)CC(C)CC(C)(C)C1 C1(O)(C(C)NC(c2c(C)nn(C)c2)=O)CCN(C(c2ccn(C)n2)=O)CC1 CC1=C(C(=O)NC2CC2CNC(c2ncc(Br)cc2N)=O)CCCC1 C1(OC)CC2C1CCN2C(=O)C(CCSC)NC(=O)C=C=C(C)C N1(C(C(C(C)C)C)=O)CC2(CO)CC1(C(=O)NCc1ncc(CO)[nH]1)C2 N1(C(=O)CCCCn2cc(-c3ccns3)nn2)CCC2CCCCC2C1 Cc1nnc(OC(F)F)c(C(=O)Nc2cc(Br)ccc2NC(=O)CSC(F)F)c1C C(CC(F)F)(C(=O)NCCC1(C)CCOCC1)N(C(c1nc(COC)sc1)=O)C Cc1cnc(F)cc1NC(C1CC1NCc1cccc(F)c1I)=O N1(C(=O)NCc2nc(COC)sc2)Cc2cccc(Br)c2CC1C N1(C(c2cccc(N(C)C)c2)=O)CC(N(C)C(c2nnsc2N)=O)C2(CC2)C1 C1(CC)CN(C(C2(C#N)CCCO2)=O)CC1NC(=O)COCc1cccc(C)c1 CC1CC(NC(C2(F)CN(C(c3ccnc(O)c3)=O)C2)=O)CN1C1CC1 N1(C(C(C2CCCO2)NC(c2cc(C)sn2)=O)=O)CCC(CCF)CC1 N1(C(CCCCCOC)=O)CCC2(CC1)CC2CNC(C1CCC(C(N)=O)O1)=O CC(C(=O)NCC(CC(F)(F)F)NC(c1ccc2c(c1)CC2)=O)C(C)(C)C c1(C(N2CC(C)C(CNC(=O)COC3CCCOC3)C2)=O)cc2cccnn2c1 C1(NC(C2CC(CC3CC3)C2)=O)CC2CCCC(C1)N2C(=O)CCC(F)F C=CCCCCC(=O)NCCCNC(C1OCC2CCCC12)=O c1(C(=O)NCC(CC)NC(=O)C(F)(F)C2CC2)ccccc1-c1nc[nH]n1 C(C)(C(CC(=O)NOCCCCCO)NC(=O)C(F)F)OC N1(c2ncc(C(=O)NCc3c(CC)nccc3)cn2)CCC(F)(F)C(C(C)C)C1 N1(C(CC=CC(C)(C)C)=O)CCC(NC(=O)Cc2ccsc2)CC(C)(C)C1 C(=O)(C1=C(C)OCC1)NCC1(NC(C2(COC)CC(F)(F)C2)=O)CCCCC1 N1(C(COCCC)=O)CCC(C)C(NC(c2n[nH]c(CC)n2)=O)C1C c1(C(N2C(C(=O)Nc3c(OCC)cccc3)CC(O)C2)=O)ccc(C)c(I)c1 C(=O)(CC1=NN(C)C(=O)C1)NCCC(=O)NC(CC)C(C)CN(C)C Cc1cc(C)cc(N=c2scc(-c3ccc(C)s3)n2CC2CCC2(F)F)c1 C1(NC(=O)C=Cc2cncc(O)c2)CC2CCC1N(C(=O)CC1CCCCO1)C2 C(=O)(CC(C)CC(F)(F)F)N1CC(F)CC(NC(=O)NC(C)C(=O)N)C1.C(=O)NC C1(C)(C(=O)NC(C(CC)O)c2ccccc2)CCC(C(=O)OC)C1(C)C N1(CC(C)OC(C)C)C(=O)CCN(Cc2ccc(CCC3CCOC3)cc2)C1=O c1(SC)ccc(C=CC(N2CCC(CN(C(=O)COCCF)C)CC2)=O)s1 c1(NC(Cc2c(F)ccc(NC(C(C)OC)=O)c2)=O)csc2ccncc12 N1(C(c2c(C)ccnc2C)=O)CC2CCC(CNC(=O)C(C)C3CC3)C2C1 C1(O)(C(C(=O)NC2C(CN(C)C)CCC2)F)CN(C(c2cc(C3CC3)on2)=O)C1 C1(CNC(=O)NCC2CCC(=O)C2)CCCN(Cc2ccccc2)C1 CCC(CC)(C(=O)N1CCCC(CCNC(=O)C(C)(C)CC#N)CC1)OC c1(Cn2cc(C(C)(C)NC(C3NCC(C)(C)C3)=O)nn2)ncnc2sccc12 CC1CCN(C(c2ccccc2NCC(F)(F)F)=O)CCN1C(C1CC=CC1)=O c1(C(N2CCCCC(CO)C2)C(=O)NCC=C)cc(Cl)cc2cccnc12 c1(C(N(CCCCNC(=O)CC(=O)NC2CC2)C)=O)c(F)cc(F)cc1F N1(C(C2CN(C(C)=O)C2)=O)CC(O)C(O)C1CNC(=O)CC1CC2C=CC1C2 C12(NC(C3CC3(Cl)Cl)=O)CCCC1N(c1ccnc(C3CC3)n1)CCC2 c1(NC(=O)NCCc2cccc(Cl)c2C(F)(F)F)ccc(Cl)c([N+](=O)[O-])c1 c1(C(N(C)CC2(NC(C3CC(C#N)C3)=O)CC2)=O)cc(F)c(F)c(F)c1F C1(Cn2cc(CCCCNC(c3c(C)nncc3)=O)nn2)CC(C)(C)NC(=O)O1 c1(C2N(C(=O)NCC3CC34CCOC4)CCC2)nnc2n1CCOC2 O=C(C1=CC2C=CC1C2)NC(CC1CCCC1)C(=O)NC1(c2ccsc2)CC1 O=S(=O)(c1ccc(NCc2csc(C(F)F)n2)cc1Br)NCCc1ccoc1 C(=O)(C(C)(CO)NC(CCC=CC1CCCC1)=O)N(c1ccccn1)C c1(C(N2C(CCNC(C3(O)CC(C)(C)C3)=O)CCC2)=O)ccc2n[nH]cc2c1Cl C(CCCCCN=c1[nH]c(C)cc(=NCC(C)c2cnn(C)c2)[nH]1)SC C1(CNC(c2ccc(Cl)cc2O)=O)CC2CN(C(=O)C=CCC3CCCC3)CC12 CCC(CC(=O)NCCC(O)C(=O)N(C1CCOC1)CCO)C(F)F c1(C(=O)NC2CC(CNC(C(C=C=C)C)=O)C2)ccc(S(=O)(=O)N2CCOCC2)o1 n1(CC)nc(C(N2CCC2CNC(=O)C(c2cccc(Cl)c2)C)=O)cc1O C1(CN(C(CC2(OCC)CCC2)=O)C)CCCN1C(=O)C(O)CSC C1(C(=O)NC2C=CCN(c3cc(COC)ncn3)C2)CCc2n[nH]cc2C1 N1(C(C(CCC)CC(C)C)=O)CC2CN(C(=O)Cn3nncn3)CC2(C)C1 N(C(=NCCC1CCCO1)NC(C)CNC1(COC)CC1)C(CC)C C1(C)(C(=O)NC2C(C)CN(C(c3cc(Cl)c(Cl)[nH]3)=O)C2)CCN(C)C1=O N1(C(CCNCC(C)(C)C)=O)CCC(CO)CC1(C)C C=CCN=C(NCCC(C)(C)C1CC1)NCc1cc(Cl)ccc1OC C(C)(C)(C(=O)NCc1cn(CC2CCCN2C(=O)CCN(C)C2CC2)nn1)SC N1(C(c2c(C(C)C)c(F)ccc2)=O)CCN(C(=O)C=CC(C)(C)C)CC12CC2 C1(C(F)(F)F)(C(=O)NC(C2CCN(C(=O)CCN(C)C)C2)C)OC2CCC1CC2 c1(C(=O)NC2(C)CCCN(C(C3(CO)CCCO3)=O)C2)cnn2cccc(Cl)c12 CC1CC(CSC)CCO1.C1(=O)CCCn2cc(nn2)CN1.C(C)(C)(C)NC(=O)OC C(=O)(CCC(=O)c1ccccc1N)N(C)CCN1CCSCC1 CC1CC(c2ccccc2)(C(=O)NC2CC(CNC(=O)CC3CCCO3)C2)C1 c1(C(=O)NCC(CO)NC(CCCCC(N)=O)=O)cnc2ncnn2c1O C1(C(=O)NC2CCC(CNC(c3c(CC)ocn3)=O)C2)CS(=O)(=O)CC12CCC2 c1(OC)csc(C(=O)N(C2CN(C(C3C4CC5C(C4)C35)=O)C2)C)c1OC c1(OC)ccnc(C(=O)NC(C)C(C)(C)NC(=O)CCCC(C)=O)c1OC C1(NC(C2CS(=O)(=O)C2)=O)CCN(C(=O)CC(F)(F)Cl)C1C1CC1 C12(CNC(=O)NCc3ccc(C(C(C)C)C)cc3)CC3CC(C1)CC(C)(C3)C2 N1(C(C(Cc2c(C)nn(C)c2C)C)=O)CCC(C2CCN(c3nncs3)C2)CC1 C(=O)(C1=COCCC1)NC(C(=O)N(C1CCOCC1)C)C1(O)CCC1 CCCC(C#N)C(=O)NCC(CC1CCCC1)C(N1CC(F)(C2CC2)C1)=O C#Cc1ccc(F)cc1C(=O)NCCCCN(C(=O)C(C)CC(C)C)C N1(C(C(Cc2ccc(Cl)c(F)c2)N(C)C)=O)CCC(O)CC12CCCC2 C(=O)(C(C)C(C)(F)F)NCC1(CNC(CCCOCC=C)=O)CCCC1 C1(N=[N+]=[N-])(C(=O)NC(C2CCCCC2)C#C)CCN(C(C2CC(C(C)C)C2)=O)C1 c1(CC)nocc1-n1cc(CNC(c2ccsc2)=O)nn1 N1(C(CCCOC)=O)CC(NC(=O)COC2CCN(C)CC2)CC(C)(C)C1 c1(C(N2CC(CN)OCC2)=O)cc(F)cc(C(F)(F)F)c1N CC1CCC(NC(=O)C(C)(C)OCC(F)(F)F)CN1C(c1ccc(=O)n(C)n1)=O C1(NC(CC2CN(C)C2)=O)CC2CC(NC(=O)C(C)(C)F)CC2C1 c1(C(=O)NCC2N(C(C3C(C)C3)=O)CCCC2)cc(N)c(F)cn1 N1(C(CCC2CCN(C)CC2)=O)CCN2CC(F)(F)CC2C1 N1(C(C2N(CC(C)C)CCC2)=O)CC2C(C(=O)NC3(CF)CCCC3)C2C1 N1(C(CCC(C)C)=O)CCCC12CCCN(C(=O)Cc1ccccc1S(C)=O)C2 C(CCCCC(=O)N1CCN(C)C(CNC(=O)CC2CCC(C)(C)C2)C1)N(C)C c1(OC)cc2c(cc1NC(N1CCCC(C(=O)NC3CCN(C)C3)C1)=O)OCO2 C1(C)(NC(=O)NC2N(S(CCC)(=O)=O)CCC2)CCCN(C(=O)OC(C)(C)C)C1 c1(CC(=O)NCC(CN(C(c2c(C)noc2N)=O)C)C)cccc(Cl)c1Cl c1(COC)nc2n(n1)CC(N1CCC3(CCCNC3)C1)CC2 C(=O)(C1CCCc2cncn21)NC(CN(C(CCCC#CC)=O)C)C Cc1cn2c(n1)CC(C(N1CCC(CNC(c3cnc4[nH]ncc4c3)=O)C1)=O)C2 C1(C(=O)O)(NC(=O)NC(C2(C(C)(F)F)CC2)C2CC2)Cc2ccccc2C1 N(C(=NCCNc1ccccc1)NCCSc1ccccc1F)C(C)C.S(C)(=O)(=O)N Cc1cc(=Nc2cnn3c2C=CC(COC(C)CSC)CC3)nc(-n2ccnc2)[nH]1 c1(C(N2C(CC)CN(C(c3ccn(CC#N)n3)=O)CC2)=O)ccc2c(n1)CCC2 N1(CC(=O)NCC=CCNC(C(CC)Oc2ccccc2)=O)CCCNS1(=O)=O c1(C(=O)NCC(C)(C)NC(C2CC3(CCC3)CS2)=O)cccc(C#CC2CC2)c1 c1(CC(=O)NCC2=CCN(C(CCOC(C)=O)=O)CC2)c(C)nc(O)nc1C N1(C(C(C)OC2CCCC2)=O)CCC(N(C)C(c2ccc(C(F)F)o2)=O)C1 Cc1ccc2c(c1)C(=O)N(CC(=O)N(CCC(O)C1CCC1)C1CCCC1)C2=O C(=O)(CC(CC)CC(C)C)N1CCC(CCNC(CCCCC=CC)=O)C1 C(=O)(C1CSc2ccccc21)NCC=CCNC(C(CCC)CC)=O c1(C(N2CCC2CNC(=O)C(C2CC(F)(F)C2)O)=O)c[nH]nc1C1CCCO1 C12(CNC(CCc3c(C)nccc3)=O)CC(CO1)N(C(C1COC(=O)N1)=O)C2 C1(C)(CNC(C2(COC)CCC2)=O)CCN(C(C2CCCC2C#N)=O)CC1 c1(-c2n(C3C(C)C(C)CCC3)nc(CCC(C)(C)C)n2)cn2cccnc2n1 C(=O)(C(CN=[N+]=[N-])NC(=O)CC1CC2C=CC1C2)NC(CCN(CC)CC)C c1(NCCC2CCN(C(=O)CCC3CC3(F)F)CC2)c(F)cccc1[N+](=O)[O-] CCCCCCC(=O)NCC1CCCN(C(C2SCCS2)=O)C1 c1(C(=O)NC(C(C)NC(CC(=C)C)=O)C)cccc(OC(F)F)n1 CN1CCOC(C(N2CCC23CN(C(=O)C(c2ccccc2)O)C3)=O)C1=O Cc1cc(C(=O)CN2CCN(C(C3CC3F)=O)CC2C)ccc1F c1(C(=O)NC(CNC(CN(C(=O)NC)C)=O)C2CC2)cccc(OC)c1 C1(NC(CCNC(C)=O)=O)CCN(c2nc3ccc(OC)nc3s2)CC12CCC2 c1(C(N2C(C(C)(C)NC(C3CC4CC4C3)=O)CCC2)=O)cc(O)cc(Cl)c1 c1(C(=O)NCC2CCC(C)CN2C(=O)CC2(C)CC2)cc2ccc(F)cc2o1 N1(C(CC(CC)C2CC2)=O)CCC(C)(C)C1CNC(c1sccc1C1CC1)=O N12CCC(CC1)C2.CCC(CONC(c1ccncc1Cl)=O)CO C1(NC(CCc2ncc(C)[nH]2)=O)CC12CC(NC(c1cc[nH]n1)=O)C2 n1(CC)cnnc1CCNC(=O)CSCCNC(=O)C(c1cncn1C)O CC1(C)Cc2cc(CNC(c3c(Cl)cc(C#N)cc3Cl)=O)ccc2O1 C1(CNC(C2(NC(C3CC(OC)(OC)C3)=O)CC(O)C2)=O)CCC(O)CC1 c1(OC)ccc(CC(=O)NCCN(CC2(N(CCC)C)CCCC2)CC)cc1 C1(NC(C=C)=O)CN(C(C2(C(F)F)CC(=C)C2)=O)CC1C(F)F c1(NC2(c3n(CCC)nnn3)COC3(COC3)C2)ccc2nc(O)n(C)c2c1 C(=O)(C(C)(C)C(O)CC)N1CCC(CC=C)(NC(c2cc(C)n(C)n2)=O)C1 C1(C(N2CC(CNC(c3ccn(CCOC)n3)=O)C2)=O)C2CC3C(C2=O)C13 CC(CC(=O)NC(C(=O)NCc1nnc(O)o1)c1ccco1)N(C)C C1(CC)CN(C(=NCCC23CC4CC(CC(C4)C2)C3)NC2CCCCC2C)CCS1 CC(=NO)C1CC(C(N2CCC(C)C(NC(=O)C=CBr)C2)=O)C1(C)C Cc1nnc2n1CC(C(N1CCN(C3CN(C(c4cnoc4)=O)C3)CC1)=O)C2 CC(C)(CC(=O)NC1CCC(NC(c2cnc(Br)s2)=O)C1)C(F)(F)F Cc1c(C(=O)NCC(C)N(C(=O)CC2CCC(C)(O)CC2)C)cccc1O N(C(=NCCCc1c(Cl)cccc1Cl)NCC1OCCC1(C)C)CC(=C)C Cc1nn(C)c(C)c1OCC(=O)NC(C)CN(C)C(C1CCNC(=O)C1)=O c1(OCC)cccnc1C(=O)NCCCCNC(=O)CC(C)SC1CCCCC1 C(CCCCCNC(=O)CC1CCC(O)C1)N(C)C(C1(Sc2ccccc2)CC1)=O N1(CC(=O)NC2CCC(NC(C3(OC(C)=O)CC3)=O)CC2)C(=O)C(C)C(C)C1=O C1(CC(=O)NCc2ccc(C)o2)C2CCC(C2)N1C(c1nnsc1N)=O C1(C(N(CC(=O)OCc2ccccc2)CC)=O)CNCC1C1CCCC1 C(CC(C)(C)C(=O)NC1CCC(NC(c2scnc2C2CCCC2)=O)C1)SC c1(C(N2C3CC(NC(CCCOCC=C)=O)C2CC3)=O)cc2oc(Cl)cc2[nH]1 C1(C(=O)NCCC2CCCCN2C(c2ccc(Cl)s2)=O)CC(C2CC2)=NO1 c1(C(=O)NCC(C)NC(C2CC=CCC2)=O)c[nH]c(=N)s1 N1(C(C2(C(=O)OC)CC2C)=O)CCC(C2CC2)(CNC(=O)CC(C)(C)OC)C1 CC1CCC(CCC(=O)NCCN(C(c2cncnc2)=O)C2CC2)O1 N1(C(CCn2cnc(=N)[nH]2)=O)CC2CCC(C(=O)NOC3CCCCC3)(C2)C1 C=CCN=C(NCCOc1cccnn1)NC1CCCC(c2ccc(Cl)cc2)C1 c1(OC)cc(CNC(C(C)(C)CO)c2nnnn2-c2ccc(F)cc2)ccc1C C(=O)(CC(C)C(F)F)NCC(CNC(CCOc1c(OC)cccc1)=O)C O=S(=O)(c1ccc(NCCC2CC=CC2)c(Br)c1)N1CC(CO)CC(CO)C1 N1(C(c2nc(C(=O)OC)sc2)=O)CC2CCN(C(C3CCOCC3)=O)CCC2C1 c1(C(N2C(CC)C(C(=O)NCc3cnc(C)[nH]3)CC2)=O)cnn2ccccc12 c12cnccc1C(=O)N2.N1(C(C)=O)CC2CC2(C(=O)NCCCCC2CC2)C1 c1(C(=O)NCCOC2CCN(C(c3cn(C)nn3)=O)C2)cccc(Br)c1O N1(C(C2(SC)CC2)=O)CCCC(C)(CNC(=O)Cc2cccnc2)C1 C=CC(CC)CC(=O)NC1CCCCC1NC(=O)CC1(c2ccon2)CCC1 c1(C(N2C(C)(C(C)C)CC2)C(=O)NC2CCN(C)CC2)cnn(C)c1Cl C1(C(=O)NCC2OCC(CNC(C=CCOC)=O)C2)CC(C)(C)CC(C)(C)C1 N1(C(=O)OC(C)(C)C)CCN(C(=O)OC(c2cccnc2)=O)CC(C)(F)C1 c1(C(=O)NCC(CC)NC(C2CC2C)=O)ccc(CN(C)C)c(F)c1 N1(C(C(C)NC(CC)(C)C)=O)CCC(C(C)NC(=O)C=CCF)C1 C(C(CNC(=O)C(O)C1CCC1)C(F)(F)F)NC(=O)CCSc1ccccc1 C1(NC(C=COCC)=O)(CNC(C2CC2c2ccnn2C)=O)CCCCC1 c1(CC)cnc(O)c(C(=O)NCCSC2C3CCCC23)c1.C12CCCN(C1)C2=O N1(C(C(C)N(C)C)=O)CCCC(C)(CNC(=O)N)C1.C1(OCC(=O)N)CCCCC1 N1(CCOC(C2CCC(C(C)(C)C)CC2)=O)CCC(C)(F)CC1 CCCCCC(F)C(=O)N(C(C)=O)CC1CC1C1CCOC1 C1(C(=O)OC)(NC(C2CCC2COC)=O)CCCN(C(C2CCN(C)CC2)=O)C1 C1(C(=O)NC2C(C)CCN(C(C3CC4CCC3O4)=O)C2)CCC2CCCCC2C1 C(=O)(CC(C)C(F)F)NC(C(C)OC)C(=O)NC(c1ccc(C)nc1)C n1(CC(=O)NCC(C)NC(c2c(C)csc2)=O)cc(C#N)c(O)nc1=O C(Cc1ccccc1)(CCNC(C1CCCC1C)=O)NC(C=C(C)Cl)=O c1(C(=O)NCCNC(c2cn(CCC)nc2)=O)c(F)cc(F)cc1Cl N1(C(c2cn(C(C)C)nn2)=O)CC2(CCC2)CC1CNC(c1c[nH]nc1F)=O c1(-c2n(CC)nc(CC(C)CC)n2)ccnc2[nH]c(C(F)F)nc12 C(=O)(C1=NOC(C)(C)C1)NC(C(C)NC(c1cc(C(F)F)no1)=O)(C)C C(=O)(CC(CC)C(C)C)NCC1N(C(c2cccc(CCC)c2)=O)CC1 N1(C(=O)CC(O)Cc2ccccc2)CC2(C(=O)NCC34CC(C3)C4)CCC1CC2 c1(C(=O)NC(C(CO)NC(c2ccc(C)c(C)c2)=O)C)cnc(P(C)(C)=O)cn1 c1(CCC(=O)OC)nc(CCC(F)(F)F)nn1-c1ccc(C(C)(C)C)cc1 c1(CNC(C2CCCOCC2)c2n(CCCOC)nnn2)ccc(C)cc1 N1(C(CCCCOCC)=O)CC(C(N2CC(F)(C3CC3)C2)=O)CC(C)C1 CCC(C)C(C(=O)NCCN(C(c1ccc(-c2ccc(F)cc2)s1)=O)CC)OC C1(O)(CNC(c2ccc(Oc3ncccn3)nc2)=O)CCS(=O)(=O)C1 Cc1cc(Cl)ccc1OCC(=O)NCC1CCN1C(c1n[nH]c(=N)s1)=O c1(CCCC)cc(NC(CNC(=O)C=Cc2cn[nH]c2)C2CC2)n2ncnc2n1 Cc1c(CNC(=O)CN2Cc3nc(Br)sc3C2)sc2ccccc12 C12(C(=O)NC34CC(CNC(C(N5CCOCC5)C)=O)(C3)C4)CCCC1CCC2 N1(c2ncnc(C)c2F)CC2CC1CN(C(C1Cc3ccccc3CO1)=O)C2 CCC(O)C(F)(F)C(=O)NC1CCN(C(=O)CNC(=O)CC(C)C)C1C n1(CCC(N2CCC(NC(c3c(OC)n[nH]c3)=O)(CF)C2)=O)nc(C)c(C)c1C c1(C(C)NC(c2ccsc2Cl)=O)ccc(CNC(=O)C(C)n2ccnc2)cc1 C(=O)(C1=CCCSC1)N1C(CN(C(C2C(c3cccc(C)c3)C2)=O)C)CC(F)C1 C=CC(C)(C)CC(=O)NCC1(C)CCCN1C(=O)Cc1nn(C)cc1Br C(N=c1ccn2nccc2[nH]1)C1C(N)CCCC1.C(=O)(CCCOC)C(C(F)=CCC)=O S(=O)(=O)(C1CCC(C#N)C1)NCC(C(=O)OCC)Cc1ccccc1 C1(CNC(c2n(C(C)C)ccc2)=O)CN(C(C2(C)CC2(Cl)Cl)=O)CC1(F)F N1(C(CCOC(C)C)=O)CCC2CCN(C(c3ccc4nnnn4c3)=O)CC12 Cc1ccc(O)c(C(=O)NC2CCCCC2NC(=O)CC2OCCCC2(C)C)n1 C(C(C)(C)C(C)(F)F)NC(CC1(C=C)CN(C(C2CCOC2C=C)=O)C1)=O c1(C(=O)NCCN(C(c2occc2Cl)=O)CC)cnc(C(F)F)c(F)c1 C(=O)(C(C)N=[N+]=[N-])NC(C(=O)NC(C=C)C1CC1)CC1CCC1 c1(COCCCNC(c2cc(OC(F)(F)F)cc(Br)c2)=O)nc(Cl)ccc1F N1(C(C(C)c2cccs2)=O)CCC(C(=O)NCc2nccn2C)(CF)C1 N12CC(CCC1C)NC(=O)CC2=O.c1(OC)ccccc1OCCOC.C1(CO)CC1 N1(C(C2(COCC)CCC2)=O)CCN(C(C)C(=O)NC2CCCN2N=O)CC1 n1(COC)nccc1C(=O)NC(C)CCCNC(c1ncoc1-c1ccon1)=O c1(C(C)NC(=O)C(=O)NCc2ncc(C(F)F)o2)cccc(F)c1F c1(C(=O)NC(C(C)C)(C)C)ccc(CNC(c2cn(CCO)nn2)=O)cn1 c1(C2(C(=O)NCC(C)CNC(=O)C=CCO)CCC2)ccccc1Br C1(C(=O)NCCCOCCNC(=O)CC2(CO)CC2)CCC2C(C1)C2(F)F C1(NC(C(N2CC(C)N(C(=O)CCOC3CC3)CC2)C)=O)CCCC(C)(C)CC1 C12(CNC(C3(F)C(C)OCC3)=O)CC(CO1)N(c1nccc(CO)n1)C2 C1(CN(C(=O)CC2CCC(F)(F)C2)C)CN(C(C2CCCN2C)=O)CCO1 N1(C(CC)=O)CCCCC1C(=O)N(C)CC1CCCN1C(c1cnc(CC)[nH]1)=O N1(c2cc(C(=O)NCc3cnccn3)ncn2)CC2(CCCC(CO)O2)C1 C(CCC(C)C)(C(=O)NCc1cncc(C)n1)NC(CCCCCSC)=O C1(C(=O)NC2CN(C(C)=O)C2)(COC)CCN(C(=O)C(C)C)C1 C=CC(C)(C)CC(=O)N1CCCC1CN(C(=O)CCOCC(F)F)C N1(C(c2c(CC)ncs2)=O)CC2(CCC(NCc3ccc(N(C)C)cn3)C2)C1 c1(C(=O)NC(CN(C)C(c2cc(O)nc(Cl)c2)=O)(C)C)cnc2n1CCS2 C12(C(=O)NCC3C(NC(COCCN=[N+]=[N-])=O)C3)CC(C(F)F)(C1)C2 C1(C(N2C(COC)CC(NC(C(CC)n3ccnc3)=O)C2)=O)CC(=O)NC(=O)C1 Cc1[nH]c(C)c(C(=O)NCC2CC(C(N3CC=CC(O)C3)=O)CO2)c1C Cc1ccc(CC(=O)NC(C)(CNC(c2ccnn2CCF)=O)CO)cc1C c1(CC(N2CC3CC(NC(c4ccnnc4Cl)=O)C3C2)=O)ccn2cncc2c1 C(=O)(CC(O)C(C)C)NCC1C(NC(c2c(C)n(-c3cccc(Cl)c3)nc2)=O)C1 c1(C(=O)NCC2C(NC(C3CCN(C(C)=O)C3)=O)C2)ccnnc1O c1(NC(C2CN(C(=O)CC3COCCO3)CCS2)=O)ccc(F)cc1Br N1(C(COC)=O)CCOC2CCN(C(=O)NC3CCC(=O)NC3C)CC12 C12(C(N(CCCN(C)C)C)=O)CC(CN(C(=O)COCC3CCCO3)C1)C2 C1(C2CCN(C(=O)Cc3c(F)cccc3F)C2)(NC(c2c(C)nn(C)c2)=O)CC1 CN1CC(CNC(=O)C(c2ccnn2C)NC(=O)CCCn2cccn2)CC1=O C(=O)(C#CC1CCC(=O)CC1)N1CC(=C(CNC(CSc2nc(C)[nH]n2)=O)F)C1 C(=O)(CS(=O)(=O)C1CCCC1)NC1CC(O)(CNC(C=CC)=O)C1 N1(c2c(C)c(N(CCCN(C)C3CC3)C)ncn2)CCc2ccccc2C(C)(C)C1 C1(CC(=O)NCC2(C)CCN(C(c3ccc(OC)s3)=O)C2)CC(=O)NC(=O)C1 c1(NC(c2c(C3CN(C(C(C)SCC)=O)C3)noc2)=O)ncc(F)c(OC)n1 c1(C(N2CCN(C(C(CC=C)C)=O)C(CF)C2)=O)[nH]c2ccc(C)cc2c1C C1(NC(CCC(N)=O)=O)CC2CC(NC(=O)Cn3ncccc3=O)C2C1 N1(C(c2ncn(C)n2)=O)CC2(CNC(c3cc(C(F)(F)F)cs3)=O)CC1CO2 c1(CC2C(C(N(CCCNC(=O)C(=O)NCCC(N)=O)C)=O)C2)ccccc1 C(=O)(CC1=CCCCC1)NCC1C(NC(C2(C#N)CCCO2)=O)COC1 N1(C(C2CC3(C(=O)OC)COC2C3)=O)C(C)CCC(OC)C1C.CO N1(C(C(C(C)C)n2cnnn2)=O)CCC(CNC(=O)CCc2cccs2)C12CC2 c1(CN(CCNC(=O)CCn2cncn2)CC2CC2)ccc(F)cc1Cl Cc1ncncc1C(=O)NC1CN(Cc2ncccc2Cl)CC1O CCC(C(=O)NCC1CC(NC(c2ccoc2CC)=O)C1)n1ccc(C2CC2)n1 C(C)(C(C(=O)NC(c1ccc(C)nc1)C)NC(=O)C1=NOCC1)OC C1(CNC(C(CC)SC)=O)CCC2(CN(C(c3c(F)ccc(F)c3O)=O)C2)O1 c1(CC)nc(C)oc1C(N1CCC(C)(NC(c2ccc(CCO)cc2)=O)C1)=O C12(NC(c3cscn3)=O)COCCC1CN(C(=O)CCOCC(F)F)C2 C1(CNC(CCOCC(C)C)=O)CCCCCN1C(=O)C=CCN1CCCC1 c1(CNC(C2(C)N(C(CC3(CC)CCC3)=O)CCC2)=O)ccc(F)cc1F CC1OC2(C(=O)NCC(C)CN(C)C(c3cnc(N(C)C)cn3)=O)CCC1CC2 C1(C(N(CC(F)Cl)C)=O)CCOCCN1C(=O)COCCOCCO C(C(=O)N1N=C(c2ccco2)CC1c1ccco1)Sc1ccc(OC)cc1 N1(C(CC)=O)CCCC12CCCN(C(=O)Cc1ccc(-n3cnnn3)cc1)C2 N1(C(=O)OC(C2C(C)C2)=O)CCCC2(NC3(CF)CC3)CCCC12 N1(C(c2nncc(CCC)c2)=O)CC2(CC(NC(C3CCCC(OC)C3)=O)C2)C1 N1(C(C2CC(CC)C2)=O)CCC(CNC(=O)Cc2cccc(C)c2F)(OC)CC1 c1(-c2ccn(C)n2)ccc2[nH]nc(NC(=O)Cc3cccc([N+](=O)[O-])c3)c2c1 C1(CC(N2CC(N(C(c3c(C)cccc3)=O)CCO)C2)=O)CCCC(F)(F)C1 C1(NC(C(CCC)N(C)C)=O)CC2(CCCN(C(c3cn(C)c(O)n3)=O)C2)C1 C(C)(C)(C(=O)NCCC1CC(NC(=O)Cc2cc[nH]n2)C1)OCCC c1(NCCc2ccc3cnn(C)c3c2)ccc(S(=O)(=O)N2CCCOC2)c(Cl)c1 N1(C(C(=O)NC2C(NC(c3c(OCC)scc3)=O)CC2)C)CCN(C)CC1 C1(NC(C2CC(CC)(CC)C2)=O)CCN(C(c2cnn(C(F)F)c2)=O)CC1F c1(C(=O)NC2C3CN(C(C4CCN(C(C)=O)C4)=O)C(C3)C2)ccc2c[nH]nc2c1 Cc1cc(C)n(CC(=O)NC2(CNC(=O)CCCCC(N)=O)CCOC2)c(=O)n1 CC(C)CCC(=O)C(=O)NC1(CN(C)C)CC1.C1C(CC(C)C)C(=O)N1 c1(C(C)NC(=O)NC2CCC(NC(=O)OC(C)(C)C)C2)cccc2nc[nH]c12 N1(C(N2CC3CC3(CNC(COC(C(=C)C)=O)=O)C2)=O)CC2COCC2C1 C12(NC(C3(C#N)CC34CCC4)=O)CCC(CN(C(c3cc(C)c(C)o3)=O)C1)C2 C1(C(=O)NC2C(SC)CN(C(=O)C3=COCC3)C2)CCC2CCCCN12 c1(NC(CC)C(F)F)nc(Cl)cc2c(N)cccc12 C(=O)(CCCCCN(C)C)NCCC1(NC(c2cnc(OCC)s2)=O)CC1 C1(NC(CSC)=O)CCN(C(c2cnn(Cc3ccccc3)c2)=O)CC1CC#N S(=O)(=O)(c1ccc(Cl)cc1)N1CCC(C(=O)O)C(O)C1 C#CC1(NC(C2C3CC4C(C3NC(=O)C(C)N(C)C)C24)=O)CCC(C)(C)C1 c1(COC(C2C=CCCCCC2)=O)ccc2c(c1)CCCS2 C=CCC(C(=O)NCC(C(N1CCC(C#N)(CCC)CC1)=O)OC)C(C)C c1(C(c2n(CCOCC)nnn2)NCCS(C)(=N)=O)cccc(Cl)c1Cl c1(C(C)=O)ccc(C(=O)NCC(CNC(=O)CCCN(C)C)CO)o1 C1(NC(C(C)c2cccs2)=O)CC(F)(CNC(c2cnn(C)n2)=O)C1 C1(N=[N+]=[N-])(C(=O)NCCCOCCOC)CCN(C(=O)C(C2CC2)SC)C1 C1(N(C)C(c2cncc(Br)c2)=O)(CO)CCCN(C(=O)CC(C)(C)C#N)C1 CCCC(C(=O)N1CC2C(CN(C(=O)Cc3cscn3)C)C2C1)S(N)(=O)=O N1(C(C(C)S(N)(=O)=O)=O)CCCC2C1CCCCN2C(c1n[nH]c2c1CCC2)=O c1(C(=O)NCCCOCC)c(O)nnc(CCNC(C)=O)c1OCC C1(C(N(C)Cc2cnn(C)c2)=O)CN(C(=O)CCc2nc[nH]n2)CC1(F)F C(C(=O)NCC1CCC(NC(=O)CCc2ncccn2)C1)(C(C)C)OCC N1(CC(=O)NCC2(CN(C(C(C3CCCCC3)OC)=O)C)CC2)CCC(=O)CC1 c1(OC)cc(O)ncc1C(=O)NCC1C=CCN1C(=O)C(C1CC1)OC C1(CC#C)(C(=O)NC2(CO)CN(C(=O)C(C(C)O)N(C)C)C2)CCOCC1 C1(CNC(=O)CCN2CCOCC2)CCCCC1NC(=O)C=CCN1CCC1 n1(CC)ncc(Cl)c1C(=O)NCC1CCCN1C(=O)CN1CC(C)(C)C1 C1(c2ccccc2)(C(=O)NCCNC(=O)CN2CCCC2)CC(O)C1 Cc1nc2ccnn2cc1C(=O)NCC1CC(CNC(C2CCCC2C)=O)CO1 N1(C(c2c(CC)nccc2)=O)CCC(O)(CNC(c2cc(C)cc(F)c2)=O)CC1 Cc1ccc(C(=O)NC2CC(O)CN(C(=O)CC3(O)CC3)C2)c(C)c1 Cc1ccc(OC(C)C(=O)N(CCCNC(C2C(C)(C)C2(F)F)=O)C)cc1 C1(NC(CCCOCCOC)=O)CN(C(=O)C(C)=C2CCC2)C2CCCC12 N1(C(C2COCCN(C(c3c(C)nncc3)=O)C2)=O)CC2(C1)OC(=O)NC2C N1(C(C=C(C)C)=O)CCCC2(CCC(NC(=O)Cc3ccc(F)c(Br)c3)C2)C1 C1(C)(CNC(C(C=C)(F)F)=O)CCN(C(c2cncnc2C(C)C)=O)CC1 c1(C(=O)NC(C2N(C(C(CCC)OC)=O)CCC2)C)ccc(S(N)(=O)=O)cn1 C1(C(=O)NCCCCCC)CCCN(C(c2ccn(CC)n2)C(=O)NCCC)C1 C1(CCC)(C(=O)N(CC(C)CNC(=O)Cc2cccc(Cl)c2)C)CCNC1=O N1(C(C2C(NC(Cc3c(C)ccc(Br)c3)=O)C2)=O)CCc2c(O)noc2C1 C1(N(C(C(C)(C)N2CCCC2)=O)CCO)CCCCN(C(C2(O)CCC2)=O)C1 c1(CNC=O)cc(C(N2CCCC2(C)C2CC2)=O)nn1C.c1(CC)ccc(N)o1 c1(C(=O)NCCNC(C2C(C(=O)OC)C2)=O)cc(N)ccc1Cl C1(CNC(c2cccc(CF)c2)=O)CCCCN1C(C1CN(CC(F)(F)F)C1)=O C(C(=O)N(C)CCN(C)C(c1nccc(C)n1)=O)(C(C)C)OC C1(CNC(CC2CC(C(C)(C)C)C2)=O)CC2CCC1N(C(C1C=CCC1)=O)C2 C(CCCC(F)(F)F)N1CCOCC(C(=O)NCC(C2CCCCC2)O)C1 CC(=O)CCN=C(NCC1CN(CC)Cc2ccccc21)NC1CC(C)OC(C)C1 c1(NC(c2ccccc2)COC)cccc(OCC(=O)NCCC2(C)CC2)c1 CC1Cc2cc(C(=O)NCC(c3c(F)cccc3F)(C)CO)ccc2N1 C1(NC(c2cc(CCCC)oc2C)=O)CCC(C)N(C(=O)CC(F)(F)F)C1 c1(CC)c[nH]nc1C(=O)NCc1cc[nH]c1C(=O)NCC1CCCN1C(C)C c1(C2(C(=O)NCC3(F)CC(NC(c4ccc[nH]4)=O)C3)CC2)ccc(F)cn1 c1(C(=O)NCC2N(C(C(N3CCSCC3)C)=O)CC2)ccnn2ccnc12 Cc1nn(C)c(=O)c(C(N2CCC(C)(NC(c3cc(Cl)no3)=O)C2)=O)c1C Cc1ccc(C(N2CCN(Cc3cn(CC(C)(C)C)nn3)CC2C)=O)cc1C C1(NC(Cc2c(C)nn(-c3ccc(C)cc3)c2C)=O)CCn2cc(C)nc2C1 C1(C(=O)NCC(=C)Cl)CCCCN1C(=O)C(F)C1CCCC1 c1(C(=O)N)cccc2c1C(=O)N(CC1CCC3CCC1O3)C2=O.c1(SC)ccccc1 C(C(C)(C)CC(=O)N1CCCC(C)(CNC(C2CCC23CCC3)=O)C1)OC N1(C(C(C)CC2CCC2)=O)CCOCC1CN(C)C(C1CC(F)C(=O)N1)=O N1(C(CCCOCCC)=O)CCN2C(=O)C(NC(=O)CNC(=O)OC)CC2C1 N1(c2cc(N)ncn2)CCCC2(CCN(N(C)CC)C2)C1.c1(C=O)c(C)cnn1C CC12CC(C(N3CC4=C(C3)CN(C(C3CC3Cl)=O)C4)=O)(C1)C1(COC1)O2 C1(NC(c2cc(CC)[nH]n2)=O)CCN(C(=O)CC2(NC(C)=O)CC2)CC1(C)C C(=O)(C1=CC(O)C(NC(=O)CCC2CC2(F)F)C1)NCCC(C(C)C)C C1(C(=O)NC(c2cccc(Br)c2)CC(N)=O)CCC2(CC1)CNC2 c1(C(=O)OC)ncc(NC(=O)C(C(C)(C)C)N2CCCC2)cc1F C1(C(=O)NCC(C(F)(F)F)NC(C2(CC)CCOCC2)=O)CC2CCC(C1)N2C c1(C(N2CC(OCCNC(c3cccc(C)c3F)=O)C2)=O)ccc2nsnc2c1 N1(C(c2c(C)nc(C)o2)=O)CCC(C)C(NC(c2c[nH]nc2C(F)(F)F)=O)C1 c1(OCC(N2CCN(C(CCSCCC)=O)CC2CO)=O)cccc([N+](=O)[O-])c1 C1(CNC(CNC(CC)=O)=O)CN(C(C2CCS(=O)(=O)CC2)=O)CC2(CCC2)O1 CC1CCN(C(=O)CN2CCCCCC2)CC1CNC(=O)Cc1ccon1 CC1(CNC(=O)Cc2cn[nH]c2)CCN(C(=O)CCc2ccsc2)CC1 c1(C(N2C(COC)(COC)CCC2)=O)ccc(Br)cc1F.C1(=O)CCCN1 CC1(CNC(c2csc(=N)[nH]2)=O)CCCN1C(c1cc(C(F)(F)F)n[nH]1)=O c1(C(=O)NCC2CCN(C(=O)CSCc3ccccc3F)C2)csc2cncn12 C(=O)(C1=CCS(=O)(=O)C1)N1CCC(CC2OCCN(C(C)=O)C2)C1.C1C(=O)N1 N1(C(c2nn(C)cc2SC)=O)CCC2CCC(C1)N2C(C1CCOC1C(=O)OC)=O c1(C(N2C3CCC2COC3)=O)cnc(C(=O)N(C2CCCC2)CC)c2cccn12 C1(F)(CNC(C=CC(CC)=CC)=O)CC(CNC(=O)CN2CCC(CO)C2)C1 CC(CCCNC(=O)CN1CCSCC1)NC(c1cnn(C2CC2(F)F)c1)=O C12(C(=O)NC3CC4C(NC(c5cccc(CC)n5)=O)C4C3)CCCCC1CCC2 c1(CC(N2CC(C3CN(C(C45CC(F)C4C5)=O)C3)C2)=O)ccc2cnccc2c1 Cn1nc(O)c2c(C(=O)OCCc3ccc(Br)o3)cc(C3CC3)nc12 N1(C(C(=O)C2CC2)=O)CCC2(CC1)CC2C(N1CCCC(CO)C1)=O C1(C(N2C(CNC(C3CCC4(CC3)CC4)=O)CCC2)=O)CN2CCC1CC2 Cc1ccc(C(N2CCN(C(=O)CC3CC(F)C3)C(CCO)C2)=O)c(F)c1Cl C1(C(N(CC(C)CNC(C23COCC2C3)=O)C)=O)CCC(=C(F)F)CC1 C1(N(C(c2ccc(Cl)cc2)C(=O)NCCOCC)C)CCCC(C)C1C c12cc(O)c(cc1Br)[nH]c2=O.C1(Cn2cc(C(C)(C)OC)nn2)CC2C=CC1C2 N1(C(C(CCC)OC)=O)CCC(CO)(CNC(c2[nH]c(O)nc2C)=O)CC1 C1(CC)CCN(C(=O)Cc2cn[nH]c2)C1CNC(=O)CCOCC1CCC1 C1(NC(CC(=O)NC)=O)CCC2CN(C(C3CCC(C)=C(C)C3)=O)CCC2C1 Cc1cn(Cc2ccc(F)c(Cl)c2)[nH]c1=NC(=O)C(C)c1nc2ccccc2s1 Cc1ccc(C(=O)NCCC(C(C)C)NC(c2csnc2C)=O)c(Br)c1 C1(=CC(=O)NC2CC(CNC(C(C)OC3CCCC3)=O)C2)CCCCC1 C1(C(C)(C)C)CC(c2nnnn2C(C)(C)C)(NCCCC2CCCCC2)C1 N1(C(C2CCN(C(C3(F)C(C)OCC3)=O)CC2)=O)CC2CC2C2CC12 c1(N(CCC)CCNC(C2COC3COCC23)=O)ncnc2scc(C)c12 C1(NC(Cc2c(OC)cccc2)=O)CCCCN(CC(O)COC(C)C)C1 CCN(OC)C(=O)CNC(C1CCC(NC(=O)CC2CC(C)=NO2)C1)=O CC1c2cc(Cl)cc(F)c2CCN1C(=O)C(=O)NCc1cccc2cnccc12 N1(C(CCOCC#C)=O)CC(C)C(NC(C2CS(=O)C2)=O)C(C)C1 C1(NC(c2c(C)coc2)=O)CC2CCC1N2C(=O)CN1CCSCC1 Cc1cccc(CNC(=O)CCC(C)NC(=O)CCc2nccs2)c1C c1(SC)ccc(-c2nc(-c3ccncc3)nn2-c2cccnc2)nc1 C1(CCNC(c2n(CC)ncn2)=O)CCCN(C(c2cccnc2Cl)=O)CC1 c1(C(C)N(C)CC2CCN(C(=O)C=Cc3ccco3)C2)ccncc1 C(CC(=O)NC1CCNC(=O)C1)(C(F)(F)F)NC(COCCCOC)=O C(=O)(C(C(CC)CC)OC)N1CCC(C#C)(C(=O)N(C)Cc2cn(CC)nn2)C1 C1(OC)(CNC(c2nc(C(C)C)oc2C)=O)CCN(C(C2CC2[N+](=O)[O-])=O)C1 C(=O)(C(F)C(C)(F)F)N1CC(C)(NC(C2=CC(C)C2)=O)C1 c1(C(CC)NCCC2CC2C(=O)OC(C)(C)C)cn(-c2ccccc2)nn1 C1(O)(CN(C(C2(OC)CCOCC2)=O)C)CCCN(C(C2(C)CCCS2)=O)C1 c1(OC)ncccc1C(=O)NCC1C=CCN1C(C1CCCC1SC(F)F)=O c1(C(=O)NCC(CNC(c2c(COC)noc2)=O)O)cc(O)cc([N+](=O)[O-])c1 C1(C(=O)NCC(CCC)OCC)N(C(=O)CSCCC)CCC1(C)C CC(C)CS(=O)(=O)CCC(=O)Nc1ccc(N2CCCCCC2)nc1 c1(C(=O)NCc2ccc(C(N(C)Cc3ccco3)=O)[nH]2)cccc(=O)n1C CCC(C)(O)CNC(=O)CC1(NC(=O)C(C)O)CCC1 C#Cc1cc(NC2CN(C(=O)C(=O)NC)C(C)(CC)C2)ccc1C C1(C)(OC)CCCN(C(=O)CCC(C)(C)NC(=O)CC2CC(=O)C2)C1 c1(OC)cccc(C2CC(O)CN2C(=O)Cn2cc(CN3CCNC3=O)nn2)c1 Cc1cc(=NCC#Cc2cccnc2)[nH]c(N2CCOC3(CCSC3)C2)n1 C1(CNC(C(CC(=C)C)OC)=O)CC2CCC1N(C(=O)CNC(N)=O)C2 c1(C(=O)NC(CCOC)CNC(c2cc(C(N)=O)ccn2)=O)ccn2c1CCC2 c1(C(N2CCC(N(CCC)C(c3cc(SC)c(C)o3)=O)C2)=O)cc(C)cc(N)c1 C1(NC(C(C)NC(=O)Cc2ccccc2)=O)CCN(c2ccccc2)C1=O C1(=CC(N2CC(CCO)(NC(c3c(C)con3)=O)C2)=O)CCC(C)CC1 C(CC1CCC1)(C(=O)NC1CC(CNC(C2CCCC2O)=O)C1)OC CCC(C(=O)N1CCOC(C)C1C(=O)NCC1C2CCCOC12)C(C)(C)CC c1(CCC(=O)NC2CN(C(CC(C)c3ccco3)=O)CC2C)cc(Cl)cc(Cl)c1 Cc1cc2c(cc1C(=O)NC1CC(F)(CNC(=O)Cc3ccoc3)C1)OCO2 Cc1cc(C(N2CC3CC3(CNC(c3sc(C#N)cc3Cl)=O)C2)=O)cc(C)c1F c1(C(N2CCC(N(C(C3C(C)OCC3)=O)C)CC2)=O)ccc2c(c1)NC(=O)CS2 Cc1ccc(C(=O)CCC(=O)N2CCCCC2CNC(=O)C(C)CO)cc1C c1(OC)cc(C(N2CC(OC)CC2CNC(=O)CC(C)CF)=O)cc(OC)c1O C1(CCC(=O)NCC=C)CCN(C(=O)Cc2scnc2C)C1 N1(C(c2cc(C(C)(C)O)on2)C(=O)NCCCC)CCS(=O)(=O)C2CCCC12 C1(C(=O)NCCOC2CN(C(C(C)N(C)C)=O)C2)OCCOC1C c1(C(=O)NCC2CN(C(C=CC(CC)C)=O)CC2O)c(C)n(C)c2ccccc12 N1(C(CC2CCN(C)C2)=O)CC2CC1C2NC(=O)CNC(=O)CC1CCCCC1 CC1CN(C(C(C)(C)C)=O)CC1(C)CO.c12csc(n1)C1CCCN1C(=O)C2 c1(C(=O)NC(CCNC(c2c(C#C)c[nH]n2)=O)C)ccccc1S(=O)CC CC1(C(N2CCN(C(=O)COCC(F)F)CC2CO)=O)CC2(CCC2)C1 C(=O)(C(C(C)C)NC(=O)CN=[N+]=[N-])NC(c1c(C)nns1)C C1(CS(=O)(=O)CC(=O)N(C)C)CCN(Cc2ccc(Cl)s2)CC1 Cc1cnc2c(C(N3CC(N(C(=O)C(C)O)C)C(C)(C)C3)=O)cnn2c1 c1(OCC)cnc(C(N2CCC(CC(=O)NCCCC(F)F)CC2)=O)cn1 c1(C(C)NC(c2cc(I)cn2C)c2n(CCC)nnn2)cc(F)cc(F)c1 N1(C(=O)NC(c2cc(C)sc2C)C)C2CCC1CC(CC(F)(F)F)C2 c1(C(N2CC(F)CC(NC(c3ncn(C)n3)=O)C2)=O)cccc(P(C)(C)=O)n1 c1(C(=O)NCC2C(NC(c3oc(CC)c(C)c3)=O)C2)cnc2n1CCCCC2 N1(C(c2c(C)cc(C)o2)=O)CCC(F)(F)C(CNC(C2(C)CCC(=O)N2)=O)C1 CC1CC(CNC(=O)CC(=O)NC2CC2)CN1C(=O)CSc1ccccc1O N1(C(C(C)OC(C)=O)=O)CCC(CC(N)=O)(C(=O)NCC2(F)CCOCC2)CC1 c1(-c2n(C)cnc2)ccc2c(c1)CN(C(=O)N=c1[nH][nH]cc1Br)C2 C1(CC)CN(C(C2CC(C)=NO2)=O)CCN1C(C1CCCN(S(C)(=O)=O)C1)=O C1(N(C(c2cc(C(C)=O)nn2C)=O)C)CN(C(=O)C=CC2CCOC2)CC12CC2 c1(C(=O)NC2C(NC(C(CC)N3CCCC3=O)=O)COC2)cnc2ccnn2c1 Cc1cccc2cc(C(=O)Nc3ccc(-c4ccc5ocnc5c4)cc3F)sc12 C1(CC)CN(C(C2CCCC(F)C2)=O)CCN1C(c1scc(C)c1OC)=O Cn1cc(S(N)(=O)=O)cc1C(=O)NC1CN(C(C2CC2(F)F)=O)CC1F Cc1ccc(C=CC(N2CC(CC(C)NC(C3(C)CCC(=O)C3)=O)C2)=O)s1 c1(NC(C2C(OCC)CCC2)=O)ccc2c(c1)CN(C(c1nc(Br)cn1C)C)C2 Cc1csc2ncnc(N3CCOCC3C(=O)Nc3cc(Cl)ncc3Cl)c12 C1(NC(CC)=O)CCC(C(N2CCOC(CCNC(=O)C(=O)N(C)C)C2)=O)CC1 C12(C(=O)NC3CC(N(C(Cc4cnc(C)s4)=O)C)C3)CCC(CC1)OC2 N1(C(CCSC)=O)CCC2(CC1)CC(CNC(C1CCCC(O)C1)=O)C2 C1(C(C)C)CN(C(=O)C(C2(O)CCC2)NC(=O)CN2CCC(C)C2)CCCO1 C1(n2cc(CC(C(=O)OC)O)nn2)CCCN(C(=O)Cn2[nH]nnc2=N)C1 N1(CCOCC)C(=O)NC(c2cc(C(C)C)n[nH]2)C(C(=O)OC)=C1CCCC C1(C)(NC(C(C)N(C(=O)Cc2ccc(O)cc2)CCC)=O)CCCCC1(C)C C(=O)(C(O)CCC(C)C)N1C(C)(CC(=O)Nc2c(O)ccc(C)c2)CC1 c1(OC)cnc(F)c(C(=O)N(C2CN(C(c3ccnc(OC)c3)=O)CC2O)C)c1 O=S(=O)(c1ccc(NC(c2ccsc2)CO)c(F)c1)NC1CCCS(=O)(=O)C1 C1(C(=O)NC(C)(C)CNC(C2CCC(F)C2)=O)CC2CC1CC2(F)F CN1C(=O)CSC1=CC(=O)N1CC(NC(c2ccc(Cl)nc2O)=O)CC1(C)C N1(C(Cc2ccc(OCC=C)cc2)=O)CCC2CN(C(=O)CC3(CO)CC3)C2C1 C(=O)(C(C(C)C)n1cc(C)cn1)NCCCC1(NC(C=CCC)=O)CC1 C(C)(C)(CCC(=O)N1CCC=CC1CC)NC(c1c(CC)nns1)=O c1(OC)cc(C(=O)NC2CN(C(C3CC3C(C)C)=O)CC23CC3)cc(N)c1O c1(OC)ccc(CCC(N2CC(F)CC2C(=O)NC2CC(F)C2)=O)cc1 CN1CC(C)(C(=O)NCCN(CC(C)O)C(c2occc2CN(C)C)=O)CCC1=O c1(SC)ccc(C)c(C(=O)NC2(CNC(=O)Cn3cnnn3)CCOC2)c1 C(=O)(C(F)(F)C(C)O)NC1(F)CCN(C(CSCC=CC=Cc2nnc(C)s2)=O)C1 C(c1ccccc1)=CC(N1CC(C(C)NC(C2(c3cc(C)no3)CCC2)=O)C1)=O n1(CC)cc(C2(O)CN(C(=O)CN(C(=O)N(C)C)C(=O)NCC(C)C)C2)nn1.C(C)(C)C C1(CCCNC(c2nc(COC)sc2)=O)CCCCN1C(=O)Cc1cnc[nH]1 C1(C2CC2)(CNC(CC(CC)CC)=O)CCN(C(c2ccccc2C(C)C)=O)C1 N(C(=NCCC(C#N)N1CCOCC1)NCC1(CC)CCC1)C(C#C)C(C)C C1(CN(C(=O)CN2CCOCC2)C)CCCN1C(=O)CC1CSCCS1 N1(C(C)C)CCOC(C(=O)NC(C)(CNC(C2CC2(C)Br)=O)C2CC2)C1 c1(OCC)ccc(NC(=O)CN2CCOC(CN(C)C)C2)cc1Br C=C(CNC(c1cnsc1C)=O)CCNC(=O)C(C)COC C1(CC(=O)NC(c2ccnn2C)C(=O)NC(c2nn(C)cc2O)C)CC2C=CC1C2 c1(C(=O)NC(C2(C)OCCO2)(CC)C)ccc(C)cc1-n1cc(C2(C)CC2)nn1 c1(C(=O)NCCOCCNC(C2CC2(Cl)Cl)=O)cccc2cccnc12 C1(CNC(CC(C(C)C)O)=O)CC12CCN(C(=O)CCN1CCOCC1)CC2 C1(NC(c2cnc(OC)s2)=O)CN2CCCN1CC2 CCC(CNC(=O)CN1CCC(C)C1)(CC)NC(=O)CCN(CC(F)(F)F)C n1(CC)nnc(C)c1C(=O)N(C)CC1CCCN1C(c1scnc1Cl)=O c1(C(=O)NC2(C)CN(C(C(C)OCC#C)=O)C2)ccc(SCC)c(F)c1 N1(C(C(C(COC)C)C)=O)CCCCCN(Cc2ccccc2)CCC1 C1(CC)C(C(=O)NC2COC(=O)C2)CCN1C(=O)Cc1cc(C)nn1C c1(CCC(=O)NC(CC)CNC(=O)C(C)(C)C2CCOC2)ccc(O)cc1 c1(C(N(C2CCCCC2)CCNC(C2CC(F)(F)C2)=O)=O)cn2cccnc2n1 O=[N+]([O-])c1cnc2cccnc2c1N1CCc2ccc(-c3ccccc3)cc2C1 Cc1noc(C)c1OCOCC(=O)Nc1ccc(-c2ccnn2C2CCC2)nc1 C(=O)(C(C)(C)C(O)C(C)C)NCC(CNC(c1ccc(CC)nc1)=O)O C(=O)(C(C)CCCC(C)=O)NC1CCC(CN(C(c2c(CC)nn[nH]2)=O)C)CC1 N=c1[nH]ncn1CC(=O)NCc1nc(CNC(=O)CC2CC2)cs1 c1(C(=O)NC)ccc(S(=O)(=O)N2CCC(CO)C(F)(F)C2)cc1.C12CC1C(=O)N2 N1(C(CNC(CCCCC)=O)=O)CCCN(C(c2cc3ccccn3c2)=O)C(C)C1 c1(C(=O)NC2(C)CN(C(CCc3nn[nH]n3)=O)C2)ccc(O)nc1 c1(C(=O)NCC(C(=O)N(C(COC)C)C)N(C)C)ccc(C)cc1 C(=O)(CCCC(=O)NCC(N)=O)NCC(CNC(c1c(C(C)=O)cccc1)=O)C N1(C(C(CC#C)C(C)C)=O)CC(C2CCCCN(C(C3CCN(C)C3=O)=O)C2)C1 c1(C(C(=O)NC(CC)(C)C)N(C)Cc2ncco2)noc2ccccc12 C1(C(N2C(CCC(=O)N(c3ncc(Br)cc3Cl)C)CCC2)=O)CCC(=O)N(C)C1 C1(C(=O)NCCCC(C)NC(c2cnnn2C2CC2)=O)CC(=O)N(C)C1 C1(C(=O)NC2CCC(N(C(=O)CC(F)(F)Cl)C)C2)C(C)(C)C1(C)C C1(C(=O)NCC(=O)OCC)CC=CC(NC(c2c(C#N)cnn2C)=O)C1 c1(NC(C2CCC(CNC(=O)CN3CC4CC4C3)CC2)=O)ncn2c1CCC2 C1(C)(C(=O)NCC2(OC)CN(C(C3(C)CS(=O)(=O)C3)=O)C2)CCN(C)C1=O O=C(CCc1cn[nH]c1)NCC1CN(C(=O)C2CC2)C1.C1(C(=O)N)CC1C(F)F Cc1ccc(-c2cccc(C(=O)NC(c3ccc(F)cc3F)CC(=O)O)c2)c(N)c1 CCC(C)(C)CC(=O)N(C(C)(C)CC(=O)N1CCOC(CC(N)=O)C1)C C=C1CC(C(=O)NCC(C)C2CCC2)(COC)C1.C12CCC(C1)C(=O)N2 c1(Nc2c(C(=O)Nc3n(C)nc4c3CCC4)n[nH]c2)ncnc2ccc(F)cc12 c1(CC(=O)NCC2CCN(C(C3CC(N(C)C)C3)=O)C2)cn2cccnc2n1 C1(CNC(CN(C(C)=O)C)=O)(CO)CCN(C(=O)CC(C)CF)CC1 N1(C(COC(CC)C)=O)CCCCC1CN(C(=O)CC1CC(C)C1)C CCCC(C)CN=c1[nH]c(=NCCS(=O)(=O)N2CCCC2)[nH]c2c1COC2 C(=O)(CC1=CCOCC1)NCCCOCCCNC(C(C)CN1CCCCC1)=O N1(c2nc(O)cc(C)n2)CCC2(CC1)CC2C(N1CCCC1CNC(N)=O)=O C1(C(N(CCC#C)CCOC)=O)CN(C(=O)CC(C)C=C)CC(C)(C)C1 c1(C(=O)NC2CCCC(CC(=O)NCC=CC)C2)cnc(C)nc1C Cc1[nH]c(=N)nc(O)c1CC(N1CCCC(C)C1CNC(=O)CNC=O)=O N1(C(CC2CC(NC(CC(CC)O)=O)C2)=O)CCCC(O)C1C C1(CNC(CC=C=C)=O)CN(C(c2nc(OC)ccc2C)=O)CCCO1 CS(=O)CCC(=O)NC(Cc1ccccc1)CCNC(=O)Cc1cc[nH]c1 C1(C#N)(CC)CCCN(C(=O)CC2CCCN2C(C2CCC3CC3C2)=O)C1 c1(C(=O)NCC2CCCN(C(CCOCCC)=O)CC2)cc2cnc(Cl)cc2s1 c1(C(=O)NC2CCN(C(CCC(C=C)C)=O)C2)nc2ccccc2nc1O N1(CC)CCN(C(c2cc(NCc3cc(F)ccc3Br)cn2C)=O)CC1=O C1(NC(CC)=O)COC2(CCN(C(=O)C(C(C)C)NC(=O)NC)CC2)C1 C1(NC(C(CCC)(C)C)=O)CCN(C(c2ccc(C)c(F)c2)=O)CCC1CO C1(C(=O)NC(C=C)CO)CN(C(C2CCCCC2(C)C)=O)CC12CCC2 C=CCCCCC(=O)NC(C)(C)C(C)NC(c1cc(O)nc(N(C)C)n1)=O c1(C2(C(=O)NC(CNC(CCOCC)=O)(C)C(C)C)CC2)cncc(N(C)C)c1 N1(C(C2C(C)C2C)=O)CCN(C(=O)C=CCO)CC1c1ccc(F)c(F)c1 CC1CC(NC(C2(C)CC2(F)Cl)=O)CN1C(=O)COCC1CCOC1 c1(C(OC)OC)nc(CSCCNC(C2CCCC2c2ccccc2)=O)no1 N1(C(C(C)C)=O)CCC(F)(CNC(c2cn(-c3ncccn3)cn2)=O)C1 N1(C(C(C)(C)c2cc[nH]n2)=O)CCOC2(C1)CN(C(=O)C1=C(Cl)CCOC1)C2 C1(CN2C(NC(=O)NCC(c3ccccc3)N(C)C)CC2)CCCNS1(=O)=O CC1CCN(C(=O)CSCc2cccs2)CC1CNC(c1ccc(=O)n(C)n1)=O C1(CNC(C2C(SC)CCC2)=O)CC2CCCC2N1C(c1coc(C(F)F)c1)=O C1(CCOC)(NC(c2ccc(CO)nc2)=O)CCN(C(=O)C=C(C)C)C1 CCCCCCCC(F)C(=O)NCCOC1CCN(C(C2(F)CCCN(C)C2)=O)C1 C=CC(C)(C)CCCNC(=O)C(C1CCOC1)NC(C1CNC(=O)C1)=O c1(C(=O)NCC2(NC(c3c(CC)c[nH]n3)=O)CCOC2)ccc(C2CC2)nc1O c1(C(=O)NC(C=C)COC)cc(OCC)c(C)c([N+](=O)[O-])c1 c1(C(=O)NC(C)C(C)C(=O)Nc2ccccc2)cc2cccn2cn1 C(=O)(C(C)C(F)F)NCCN(CCC)C(c1cnn(CC(F)F)c1)=O c1(OC)ccc(C(N2CC(CNC(=O)CC(C)C(C)C)OCC2)=O)cc1N c1(C(=O)NCC2CCC(NC(c3ccc(O)nc3)=O)C2)nnc(O)nc1O C1(CNC(CC(C)C)=O)CCC(CC(=O)NC2CCN(c3ccncn3)C2)CC1 Cc1cc2sc(CNC(N3CCN(CC(N4CCCC4)=O)CC3)=O)cc2s1 C1(S(N)(=O)=O)(C(=O)NCC(N2CCN(C(C=C(COC)C)=O)CC2)C)CCCC1 CC1(C)C(NC(c2cc[n+]([O-])cc2)=O)CC1C(=O)NCC1CCNC1=O N1(C(C2CNC(=O)N2)=O)C2CCC1C(CNC(c1coc3c1COC3)=O)C2 C1(CC)CC(C(N2CCN(C(=O)COC3CC=CC3)CC2CO)=O)CC(=O)N1 N#Cc1nc(Cl)ccc1NC(C1CCCC(NCc2ccc(Cl)cn2)C1)=O C1(O)(CN(C(=O)CC2(CO)CC2)C)CN(C(=O)CCCC2CCC2)C1 c1(C(N(C(CNC(C2N(CC)CC2)=O)C)CC)=O)oc(Br)cc1C N#Cc1cncc(-c2cncc(C(=O)NCc3cc(Cl)ncc3Br)n2)c1 CC(C)(F)C(C)(F)C(=O)NC1(CC(=O)Nc2cnc(O)c(F)c2)CC1 N1(C(CCOC(C)=O)=O)CC2CC3CC2C1C3NC(=O)Cc1c(Cl)cccc1Cl Cn1nc(C(=O)NCc2ccc(C(=O)NCC3(C)CCOC3)o2)cc1F C(=O)(C1COc2ccccc21)NCC1N(C(c2nc3cccc(C)n3c2)=O)CC1 Cc1c(C(N2CC(CC(F)C(N3C4CCC3CC(O)C4)=O)C2)=O)cccc1C#N C1(C(=O)NCC2(C(C)NC(CCOCC)=O)CC2)CN(S(=O)(=O)N(C)C)C1 c1(C(=O)NCC(C)(C2CC2)NC(=O)CP(C)(C)=O)cc([N+](=O)[O-])cnc1O c1(CC(=O)OCC)ccc(CC(=O)C(=O)CC2CCC3CC23)cc1.C12CC1CNC2 C1(CNC(c2cc(OC)nn2C)=O)C(C)CCCN1C(=O)CS(=O)(=O)N(C)C C(=O)(C1=CC(C)(C)C1)NCC=C(C(=O)NCC(CSC)(C)O)C c1(NC(CN(C(C(CCC)C#N)=O)C2CCC2)=O)ccc(N=[N+]=[N-])cc1 C=CCC(C(=O)N1CC2CC2(CNC(=O)CC(CC)OC)C1)NC(C)=O C(=O)(C1=NNC(=O)CC1)NCCCC(CCC)NC(c1nnc(O)cc1O)=O C(CCCCCN(C(=O)CC(C)c1ccco1)C)NC(C=CC(=O)OCC)=O C(=O)(CCC(=O)NN(C)C)NCC(C(=O)NC(C)CC1(O)CCC1)(F)C(C)C C(c1ccc(C2CC2)cc1)=CC(=O)NC1CC(NC(c2ccccc2C2CC2)=O)C1 c1(NCCCCC2(NC(CCNC(=O)OC)=O)CC2)ccc(C#N)c(F)c1 c1(C(=O)NCC2(C)N(C(C(C)S(C)(=O)=O)=O)CCC2)c2ccccc2nn1C Cc1cc(C(=O)NCC2(C)CCCN2C(C2C(C3CC3)C2(F)F)=O)ccc1O N(C1CCOc2c(C)cccc21)c1c(C)c(N2CCC(CC#N)C2)ncn1 C1(C(=O)NCCc2nc[nH]n2)CC2CC2N1Cc1ccccc1I c1(CN(C(=O)C(F)NC2CC(Oc3ccccc3)C2)N(C)C)cccnc1 c1(C(N2CC(NC(CCc3cc(C)on3)=O)C(O)C2)=O)ccc2sc(C)nc2c1 c1(OC)ccccc1C(CNC(c1sc(C)cc1Cl)=O)NC(=O)CCC1(C)CC1 c1(C(=O)NC2C(CNC(C3(C#C)CCC3)=O)C2)cc(N2CCC(C)CC2)ccn1 C(C1CCCN1C(C1CCCCCC1)=O)=CC(N1CC(CC(C)(C)C)C1)=O C12(CNC(C(N)=O)=O)CCC1CCN2C(C1CC(O)C1)=O CN1CCC(C(=O)NCCN(C(c2ncsc2C(F)(F)F)=O)C2CC2)C1 c1(C(N2CCC(N(C(C3CNC(=O)C3)=O)CC)C2)=O)cc(C)c(C#N)cn1 C(=O)(C1=C(F)CN(C(=O)CC2CSCCO2)CC1)N1C(C)(C(=O)OCC)CCC1 N1(S(CC)(=O)=O)CCC(C(=O)Nc2nnc(-c3ccccc3)s2)C(O)C1 c1(OC)cccc(CC(=O)NCC2CC(NC(=O)COCc3ccc(Cl)s3)C2)n1 C1(OC)CC(C(=O)NCC(CO)NC(=O)Cc2cc[nH]c(=N)c2)CC1OC Cc1cnnc(O)c1C(=O)NCCCC(C)NC(C1CCC=CCC1)=O [N-]=[N+]=NC1CN(C(C2CCCCCC2)=O)CC1NC(C12CCN(CC1)CC2)=O S(=O)(=O)(c1cc(F)cc(F)c1)N1CCC(CC(=O)Nc2ccnc(Br)c2)C1 c1(N(C2CCNCC2O)C)ncc(Br)c(SNCC2(C(=O)OC)CC2)n1 N1(C(C(C(=O)OC)OC)=O)CCOC(C(N2CCSC(C)C2)=O)CC1 N1(C(c2cc(OC)ns2)=O)CCC2(CC1)C(NC(=O)CCCC(F)F)CS2(=O)=O C(=O)(C1=CCCCCC1)N1CCC(C(C(=O)NC(C#C)CC(C)(C)C)C)CC1 c1(C(N(C)CC2CN(C(=O)Cc3cc(Cl)no3)CCO2)=O)ccn2ccnc2c1 c1(OC)cncc(CC(=O)NCC2(C(N)=O)CN(C(c3ccc(CO)o3)=O)C2)c1 c1(CC(=O)NCCNC(c2n(CC)ncn2)=O)ccncc1Cl N1(C(C(=O)Nc2c(COC)cccc2)C2CCOC2)CCCCC12CCOC2 C1(=CCNC(CN(CCC)C)=O)CCN(C(C2COCCC2C(C)=O)=O)CC1 Cc1ccc(C(=O)NC2CCC2CNC(c2n[nH]cc2[N+](=O)[O-])=O)c(N)c1 Cn1nc(C(F)(F)F)cc1NC(=O)NC(c1ccccc1F)C(F)(F)F N1(C(C2(C=C)CCC2)=O)CC2CCC2(CNC(c2ccc(N(C)C)nc2)=O)C1 c1(CC(CNC(=O)CSc2nccn2C)N(C)C)ccccc1 C1(C(=O)NCCC(=O)NC(C2CCN(C(C=NOC)=O)C2)C)CCCCC1(F)F c1(CC(CSc2cscn2)NC(=O)CSCC2CC2)ccccc1 CC1CCC(CNC(=O)CCCC2CCOCC2)CN1C(=O)CC1CSCCS1 c1(CN(CCC(F)(F)F)CCOC)occc(=O)c1OC CCC(C(=O)OC)C(=O)NC(CNC(=O)CCC1(C)CC1)C1CC1 CN1CC=CCC1CC(N1CCC(C(O)CNC(c2ncncc2Cl)=O)CC1)=O N1(C(C(CCC)CNC(=O)C(C)CC2CCCC2)=O)CC2(CCC(O)CC2)C1 C(CO)(CCCCNC(c1cnc(C(C)C)s1)=O)NC(C(CC)n1ccnc1)=O C1(CC=C)(NC(C2CC2(C)C)=O)CN(C(C2(Cl)CC2(C)C)=O)C1 c1(OCC)cccc(C2CC2CN2CCN(CCc3ccc(C)cc3)CC2)c1 C(=O)(CC(C)C(C)(C)C)NCC1C(NC(c2nc(N(C)C)nc(O)c2)=O)CCC1 C1(C(=O)NCc2c(CC)n(C)nc2)CCCN(C(=O)CC2CC(=O)NC2=O)CC1 N1(CCNC(C2(CCC)CC2)=O)CCCN(C(c2sc(C#N)cc2Cl)=O)CC1 C1(C(=O)NC2CCN(c3sc(C(=O)OC)c(Cl)n3)C2)CCc2nccn2C1 C1(CC)CN(C(=O)C2=COCCO2)CCC1NC(=O)Cc1cc(C2CC2)on1 CN1CC(CCNC(C2(CCNC(C3CC=CCC3)=O)CCC2)=O)CC1=O C(=O)(C(=O)N=S(C)(C)=O)NCC1(OC)CCN(C(CCOCC)=O)C1 N1(C(CC2CC(=O)C2)=O)CC2CC(C(N3CC4CC4(CO)C3)=O)C(C2)C1 c1(-n2cc(CCC(=O)OCC)nn2)cccc2c1CN(C(=O)CC(C)C)C2 C1(C2CCN(C(=O)CC(C)CN(C)C)CC2)(NC(C(n2ccc(C)n2)C)=O)CC1 c1(C(=O)Nc2cc(OC)cc(Cl)n2)cc(-c2cnn3c2CCC3)c(C)cc1F c1(CN(C)C(C2COC2)=O)cccc(CNC(c2c[nH]ccc2=O)=O)c1 CCCC(C)(C)CC(=O)N1CCCC(C)C1CNC(=O)C1=COCCC1 C(CC(C)(C)C)(C(=O)NC(CNC(=O)CNS(=O)(=O)N(C)C)C1CCC1)OC N1(CC2(N)CC3(CCCC3)C2)CCc2c(Cl)cc(Cl)cc2C1 C=C1CCC(C(=O)NC2CCCCC2CNC(c2cncnc2)=O)CC1 Nc1c(C(=O)NC2CCC2NC(c2ccc(Cl)cc2Cl)=O)ccc(Cl)c1Cl C(=O)(C1=CCCCC1C)NC1C(NC(CN(C(COC)=O)C)=O)CCCCC1 Cc1nc(NC(C2CCN(Cc3cc(Cl)ncc3Br)CC2O)=O)nc(C)c1Br C1(N2CC(N(CCNC(C(=O)NCC)=O)C)C2)CCc2ccccc2NC1=O C=CCC(CC=C)C(=O)N1CC(NC(=O)C(CC)CCOC)CC2(CC2)C1 N1(C(C2C(C3C(C)C3)C2)=O)CCCC(C2CN(C(C34CCC(C3)OC4)=O)C2)C1 C1(CNC(C(CC(=C)C)C)=O)CCC(C)(C)CN1C(c1cnc(OCC)cn1)=O C(=O)(CCCCCF)NC1CCC(NC(C2(OC)CC(F)C2)=O)CC1 C1(NC(C(CC)F)=O)CC2CC(NC(c3cc4n(n3)CCCC4)=O)CC2C1 C(=O)(C1=C(Cl)CC1)NCCC(C)NC(C1C(c2ccccc2)C1(F)F)=O c1(C(N2CC(C(=O)NC3C(C(C)(C)C)C3)C(C(N)=O)C2)=O)cc2nc(=O)ccn2[nH]1 N1(C(c2c[nH]c(=NCC)s2)=O)CC2CCC(C1)N2C(c1cnn2ccccc12)=O CCC(C)C(C(F)F)NC(c1cc(CC(C)C)nc(O)c1)=O C=CCC(C(=O)NCC(C)(C)CC=C)NC(c1sc(C)nc1C)=O C1(COC)CN(C(=O)CC2CCCC2)CCN1C(=O)C(O)Cc1cnc[nH]1 c1(CN(C(=O)CC2OCCN(C)C2c2cnn(C)c2)C)cc(C)c(N)cc1F C=CC(C)(O)C(=O)NC1CCC(CCNC(c2c[nH]cc2-c2csc(C)n2)=O)C1 c1(C(=O)NCC(c2ccc(F)cc2F)NC(C(CC)OC)=O)ccc(C#N)cn1 C(=O)(C(F)(F)C(F)(F)F)N(CC(C)(C)CNC(C1CCCC(=O)N1C)=O)C c1(C(N(CCCNC(=O)CC(C2CC2)C2CC2)CCC)=O)cc(C#N)c[nH]1 N1(C(C2CCC3CC23)=O)CCC(C(=O)NCC2CCC2)(CO)C1 C1(C(=O)NCC2C(NC(c3ccc(CC)cc3)=O)C2)(CC)CCC(O)CC1 Cc1ccsc1CNN(CCN(C)C)C(N1CCCC1c1ccccc1)=O c1(CCC(C)C)nc(-c2ccc(N3CCCC3)nc2)nn1C(C)C(F)(F)F C12(CNC(C3COCCO3)=O)CN(C(=O)Cc3ccnc(O)c3)CC1CCO2 c1(OC)cc(C2CCN(C(=O)C(=O)NCCCNC3CCC3)C2)ccc1C1CC1 N1(C(C2(C)CN(C(CC(CC)OC)=O)C2)=O)CC2CCCC2C1 C1(C(N(C(CC)CNC(c2cc(CO)[nH]n2)=O)C)=O)CC(O)C1(C)C C1(O)(CNC(C(C)N(C)C)=O)CCN(C(c2ccc(CC(C)C)cn2)=O)CC1 Cc1ccc2c(c1)CC(C(=O)NC1CC3(CCCN(C(c4cnsc4)=O)C3)C1)O2 c1(-n2cc(C(N(C3CCN(C(CC4C(C)C4)=O)C3)C)=O)nn2)ccc(Cl)cc1 c1(C(=O)NCc2nccc(C)c2)csc2c1CCN(C(=O)C(O)CC(C)C)C2 c1(C(N2CCC(N(C(CCC(C)OCC)=O)C)CC2)=O)n[nH]c2c1COCC2 CC(C)CCCCC(=O)N(C(CC(F)F)C(=O)N1CCS(=O)CC1C)C CC(C)C(F)C(=O)NC1CCCC1Cn1cc(Cn2cc(C(=O)O)cn2)nn1 C1(NC(CSCCOC)=O)CC(C)(C(=O)N(CC(F)F)CCO)C1 C(CCCCC(=O)NC1CCCCN(C(=O)CC2CC(=O)NC2=O)C1)NC(N)=O c1(CNC(C2(CNC(C(C)CC#N)=O)CCCO2)=O)cccc(F)c1O C1(NC(c2ccc(NC)cc2)=O)CCC2CCN(C(=O)CC3CCN(C)CC3)C12 Cc1cccc(C(N2CCCCC2CNCc2ccc(Br)c([N+](=O)[O-])c2)=O)c1C#N c1(C(=O)NCCNC(CC(C)N(C)C)=O)ccc2occc2n1 c1(CNC(CC2N(C(C(c3ccccc3)C)=O)CCC2)=O)cc(O)ncn1 Cc1ncc(C(N2CCN(CCNC(=O)CC3CCC3)CC2)=O)n1C C12(C(N3CC(NC(c4cc(Cl)c(Cl)[nH]4)=O)CC(C)C3)=O)CCC(C)(CC1)OC2 C1(C(N(CC(C)NC(C=CC)=O)C)=O)COCCN1C(=O)OCC.C(C)(C)(C)OCC C1(C(N2CCCC(c3cn(Cc4ccno4)nn3)C2)=O)CCCC2(CCC2)C1 c1(-c2cn(CCC(N3CCC(COC)C3)=O)nn2)cccc(CC(=O)O)c1 c1(OC)cccc(C(C)CC(=O)NCC(C)(C)CNC(c2c[nH]ccc2=N)=O)c1 C(=O)(CC(C)(C)C1CC1)N(C1CC(NC(C2CC2(F)F)=O)C1)C C=C(C)CC(C(=O)NC(C(=O)NCC(C)OCOC)C1CC(OC)C1)OC C1(C(CNC(CCCNC(C)=O)=O)C)CCN(C(C2(C)CC2C)=O)CC1 C(=O)(C1=CC2CCCC12)N1CCC(CNC(=O)CCc2cnc[nH]2)CC1 CCS(=O)(=O)CC(=O)NC1N(C(C2CC3(CC(C(=O)OC)C3)C2)=O)CCOCC1 N1(C(CNC(C)=O)=O)C2CCC1CN(C(c1cccc(F)c1C(F)F)=O)CC2 c1(CN(CCC)C)ccc(C(=O)NC(C)CNC(C2CC(CCO)C2)=O)o1 c1(C(=O)NC2CN(C(CCC(C)C#N)=O)CC2F)cc2n(n1)CCNC2=O C(=O)(C(C(=O)N1CC(CNC(C2SCCCS2)=O)C1)OC)OC C(=O)(CCCC(C)(C)NC(=O)CCC(C)OC)NCC(CC)CC CC1CN(C(=O)CSc2nnnn2C2CC2)CC(C)C1NC(=O)CC1CC1 Cc1cc(=O)c2ccccc2n1CCCCC(=O)N1CCOC(c2ccc(Br)s2)C1 CC(C)CC(C)CC(=O)NCC1=CCN(C(c2ccc3cccnc3c2)=O)CC1 CC1(C(=O)NCC(C(=O)NC(CO)C(N)=O)N(C)C)CC2CC2C1 Cc1c(F)cc(C(=O)NC2CCCN(C(C3CC(O)C3)=O)CC2F)cc1F c1(C(N(C2CCC(NC(CCCOC)=O)C2)C)=O)scc(Br)c1C c1(C(=O)NC(CNC(CCC#CC)=O)(C)C2CCC2)cc(C(N)=O)cc(C)c1 C(=O)(C1CCc2cccnc21)N1C(CNC(C2CC=CC2)=O)CC2(CC2)C1 C1(C(N(C)CC2(NC(C=CSC)=O)CC2)=O)CCc2nncn2C1 CC1(C)OCCC1(O)C(N1CCN(C(=O)C(O)COCc2ccccc2)CC1)=O N1(C(c2csc(C)c2Br)C(=O)NC(C(=O)OC)C)CC2CC3CCCN3C2C1 c1(CCC(=O)N(C2CCN(C(=O)CSC(F)(F)F)C2)C)cc(C2CC2CO)on1 N1(C(c2c(CC)cco2)C(=O)NCCC#N)CCn2ncc(C3CC3)c21 c1(N(C)CCC2CCCN(C(=O)OC(C)(C)C)C2)ccccc1S(C)(=O)=O c1(OC)ncccc1S(=O)(=O)N1CC2(CC(NC(c3cc(Br)c[nH]3)=O)C2)C1 c1(C(N(CC(C)NC(COCCC)=O)C)=O)ccccc1-n1ccnc1C N1(C(CCN(C)CC)=O)CCC2(CC1)C(NC(C1CCCC1(C)C)=O)CS2(=O)=O N1(C(c2nc(CC)[nH]n2)=O)CC2(CC(CNC(c3cccc(CCO)c3)=O)C2)C1 CC(CCCCN=c1cc(C(C)(C)C)nc[nH]1)NC(C1CCCS1(=O)=O)=O c1(C(=O)NC2CC3CN(C(CN(CCC)C)=O)CC32)nccc2ccsc12 CN1CCCC1(C)CNC(=O)C(N1CCN(CC(c2ccc(F)cc2)O)CC1)=O c1(NCc2nc(C)sc2)ccc(S(=O)(=O)Nc2cnc(CC#N)nc2)cc1F c1(C(N2CC(CNC(c3coc(Br)n3)=O)OCC2)=O)cc(O)nc(Cl)c1 N1(C(c2cnc(CC)s2)=O)CC2CC2(CNC(=O)Cc2cc(C)sc2C)C1 Cc1cc(Cl)cc(C(=O)NC2CN(C(C3CCCNS3(=O)=O)=O)CC2C)c1N c1(C(N2CC3(CN(C(c4cc(C)cc(Cl)n4)=O)C3)C2)=O)nn(C)cc1S(C)(=O)=O C(C)(CCC(C)(C)C)NC(C(CCC1CCC1)NC(c1c(C)nccc1)=O)=O C1(NC(COCC(=O)NC)=O)C2CC3C1C3C2C(=O)NC1(O)CCCC1(C)C C1(CCNC(c2c(CC(N)=O)occ2)=O)CCCN(C(C2C=CCS2)=O)CC1 CC1c2ccccc2CC1NC(C1CCN(C2COC2)C1)=O c1(OC)cccc(NC(N2CC3(CC3C(=O)NC(C)C3CC3)C2)=O)c1Cl CC(C)(CNC(=O)CC12COCC(C1)C2)CCNC(C1CC12CCC2)=O N1(C(=O)OC(C)(C)C)CC(n2cc(CC(=O)O)nn2)CC1C(=O)OC N1(C(c2cccs2)=O)CCN(C(C2(C3CCC3)CC2)=O)C2COCC12 C1(C)(CNC(c2n(CC=C)ccn2)=O)CCN(C(C23CCCC2C3(F)F)=O)CC1 Oc1cc(Cl)ccc1CNC(=NCCF)NCC1CN(C2CC2)C(=O)O1 N1(C(=O)Cc2ccc(O)cc2Cl)CC(C2CCCN(C(=O)C(O)C(F)(F)F)C2)C1 N#Cc1ccc(CC(=O)OCc2ccc(Cl)c(Br)c2)c(Cl)c1 C1(CNC(C2(C)CC2(F)Cl)=O)CC2COCC2N1C(c1cc(Cl)ccc1Cl)=O c1(C(N)=O)coc(C(N2CC(CNC(C3OCCO3)=O)C2)=O)c1 c1(-c2onc(C(C(c3ccc(F)cc3)C)C)n2)cccc(O)c1 C(=O)(CCCCCSC)NCC1CC(O)(CNC(C=CC=CCC)=O)C1 C1(C(=O)NC(C)C(N)=O)(CNC(CC(C)F)=O)CC12CCC2 C=C=CC(C)C(=O)NCC(c1ccccc1F)NC(=O)CCSC1CCCC1 C(=O)(CCC(O)C(C)(C)C)NCC(C)CNC(=O)C=C1CCSCC1 C(C(C(=O)NC1(CO)CCOC1)OC(C)=O)NC(c1cn(CC=C)nc1)=O CC(=O)CCN=C(NCC1SCCS1)N1CCC(Oc2cccc(F)c2)C1 Cc1ncc(C(=O)NC2CC(CCNC(C3(CC4CC4)CC3)=O)C2)c(C(C)C)n1 C1(CNC(CCc2cnc(C)o2)=O)CCCCN(C(=O)C(F)C(C)C)C1 c1(CC(=O)NCC(CNC(c2cnc(CC)s2)=O)F)ccc([N+](=O)[O-])cc1Cl c1(C(=O)NC2CC3CC(NC(CCCC#C)=O)C2C3)nnn2c1C(=O)NCC2 c1(C(=O)NCC(O)CNC(C23CSCC2C3)=O)cccc(F)c1 C12(C(=O)NC3C(C)(C)COC3=O)CCC(CN(C(=O)C=CC(F)(F)F)C1)C2 C1(C(=O)NCC(O)CF)(CC)C=CCN1C(=O)CCC.C(=O)(CN(C)C)NCCOC N(C(=NCCC(C)C)NC(C)C1CC1)Cc1ccc(C)cc1OC(F)F c1(CNC(CNC(CCN(C)C)=O)CCO)ccc(OC)cc1 c1(OC)ccc(Cl)cc1C(=O)N(CCCN(C)CCNC(=O)CCC(C)C)C c1(OCC)ccc(C(N2CC3CC2CN3C(=O)CC2CCC(=O)O2)=O)cc1C C(=O)(C(F)(CNC(=O)OC(C)(C)C)C(C)C)NCC1C(NC(CCC=C)=O)C1 CN1CC2C(C(N3CC=CCC3C(=O)NCC(C)(O)C3CC3)=O)C2C1 C(=O)(C1(C)CCn2c(C)nnc21)NC1CC(OC)CN(C(=O)CNS(C)(=O)=O)C1 N1(CC)C(=O)NC(c2cccn2C)C(C(=O)OC)=C1C1(C)CC1 c1(C(=O)NCC2CN(C(=O)NCC(C3CC3)OC)C2)cnn(C2CC2)c1 N1(C(c2c(N(C)C)ccnc2)=O)CCC2CN(C(C3SCCCS3)=O)C2C1 c1(C(=O)NC(CCCC)CNC(=O)CN(C)C(N)=O)ccc(OCC)c(C)c1 N1(C(CC(C)NC(=O)COC2CCC2)=O)CC(N(C)C)C1 N1(CCC)CCC(C(N2CC=CC2CNC(c2cnsc2C)=O)=O)CC1 C12(NC(CCC#C)=O)CCOCC1CN(C(c1ccsc1Cl)=O)C2 c1(C(N2CC(NC(=O)CCc3cc(Cl)no3)C2)=O)cc2c(F)ccc(F)c2[nH]1 C12CN(CC13CC3)C(=O)C(C)N2.C(C(C)C)NC(=O)OC CCCCCCCCC(C)C(=O)NCCN(C)C(C1CCCCC1)=O C1(NC(CCC)=O)CCC(CNC(c2ccc(NC(=O)NC)s2)=O)C1 C1(NC(CC2C(CC)C2)=O)CC2CC1N(C(c1cc(N)cnc1C)=O)C2 C1(=O)CC(C)C(=O)O1.c1(CNC(C(c2ccco2)OC)=O)ccnc(F)c1 C1(F)(CNC(c2c(COC)ncs2)=O)CCC(CNC(C2(C)CCCS2)=O)CC1 Cc1cc(C)c(C(N2CC=C(CNC(C3CC(C)CCO3)=O)CC2)=O)c(=O)o1 c1(C(N(CCCN(C)C)CCNC(=O)CC2(O)CCCOC2)=O)ccc(O)c(Cl)c1 O=C(C1=Cc2ccccc2C1)NCC1CN(C(C2(F)CCC2)=O)C2COCC2O1 c1(C(=O)NCC(CC)c2cccnc2)cc2ccccc2oc1=O c1(OC)cccc(CN(C)CCNc2cnc(-c3ccccn3)s2)c1O c1(NCC2C(C)CCCN2C(=O)C2=C(Cl)CC2)ncc([N+](=O)[O-])c(=N)[nH]1 c1(C(c2n(CCSC)nnn2)NCc2snnc2C)nc(C)c(C)o1 c1(CC)cc(C(N2CC3(C(=O)NC4CCN(CC)C4)CC2CO3)=O)cc(Cl)n1 N(C1CN(C(=O)CC2CC2)CCc2ccccc21)C(C1CC2CCCC(C1)C2)=O N1(C(CCCC(C)O)=O)CC2CCCC(NC(=O)C(c3ccccn3)C)C2C1 N1(C(C2C(C)(C)CCO2)=O)CC=C(CCNC(c2cnco2)=O)CC1 c1(CC)onc(C)c1C(=O)NC1CN(C(=O)C=CCOC)CC1C N1(C(CNC(=O)NC)=O)CCC(O)(CN(C)C(c2ccnc(C(N)=O)c2)=O)CC1 C(=O)(CCCCCCCBr)NCC1(C)CN(C(C2CCc3nc[nH]c3C2)=O)C1 O=C(C#CC1CCOC1)NCC1CN(C(=O)Cc2cccc(C3CC3)c2)C1 c1(C(=O)NC2C(NC(c3n(C)ccn3)=O)CC(F)(F)C2)ccc2c(c1)ncn2C c12nc(cs1)CN2C1CC1.C(C(=O)O)=CCCC.SC c1(-n2cc(-c3c(C)nsc3)nn2)cc(F)c(O)cc1F.C12(C)CCCN(C1)C2=O n1(CCC)nccc1C(N1CC(O)(CNC(=O)CSc2ccccc2)C1)=O C1(CC=C)(NC(=O)Cc2cncc(C)c2)CCN(C(C2CC3CC3C2)=O)C1 Cc1cccc(C(F)(F)C(=O)N2CC(CCNC(c3cscc3C#N)=O)C2)c1 c1(C(C(=O)NC(CC)C)N(C(CN(C)C)C(C)C)C)nn(C)cc1Br N1CCCCC1C1CCCN1C(=O)CCC(=O)c1cc(C)sc1C.CC1CC1 c1(C(=O)NC2CC(OCC(N3C(C#C)COCC3)=O)C2)cccc2ccoc12 c1(C(N2C(CNC(=O)CC(F)F)CC3CC32)=O)nc(C(F)(F)F)n2ccccc12 c1(OC)ncnc(OC)c1C(=O)NCC1(NC(=O)C(C)CSC)CCCCC1C c1(CC(=O)N(CCNC(=O)CCCF)CC2CC2)cccc(OC(F)(F)F)c1 c1(C(N(C(C)C(=O)NCCc2ncc[nH]2)CCC)=O)ccncc1CC CC1CN(C(C2CCC3(CCC3)CO2)=O)CCCN1C(=O)CCC(N)=O C(=O)(CC(CC)CCC)NC(CCNC(c1cn(CC=C)nc1)=O)(C)C N1(C(C2C3CCC(F)(F)C23)C(=O)NCCC)CCC2(CC1)CC(O)C2 c1(OC)ccccc1C(O)CNC(=O)C(N1CCOC(CS)C1)=O C1(C(=O)NCc2occ(C(N3C(CC(=O)NC)CC3)=O)n2)CCCCCCC1 c1(CSC)cc(CNC(N2CCCC(CS(N)(=O)=O)C2)=O)sc1Br Cc1cc(C)c(C(=O)NCC2(NC(=O)CC3C=CS(=O)(=O)C3)CCC2)c(C)c1 c1(C(=O)NC(C2OCCN(C(COCC=C)=O)C2)C)[nH]nc2c(=O)n(C)cnc12 CC1CN(C(c2c[nH]c(=N)o2)=O)CCC1N(C)C(c1ccccc1Cl)=O c1(C(N2CC(F)CC(NC(C(C(C)(C)O)F)=O)C2)=O)cccc(S(N)(=O)=O)c1 C=CC(CCC)CC(=O)N(C)CC1Cc2ccccc2O1 C1(C(N(C)CC2CCN(C(c3ccn(CC)n3)=O)C2)=O)CN2CCCC2CO1 Cc1cc(CC(=O)OCCOC2CCCCCC2)ccc1Cl C(CC(CC)C(=O)NCC1CCN(C(=O)C2=CCCSC2)CC1O)=CC c1(C(N2CC(CNC(c3ncc(CC)s3)=O)C2)=O)ccc2ocnc2c1 Cc1[nH]cc(C(=O)NC2CC3CC(NC(c4cc(Cl)cn4C)=O)CC23)c(=O)c1Cl CC12CCC1CN(C(C1(NC(=O)CC3CC4(CC4)C3)CCCC1)=O)C2 c1(OC)cccnc1C(=O)NCC1CC(C)N(C(c2csc(Cl)c2Cl)=O)C1 C(CC(O)C(=O)NC1CC(CO)N(C(C2CCC(C(N)=O)CC2)=O)C1)N(C)C C12CCCCN1C(=O)OC(C)C2.C1(C)(C(=O)NC(C)(C)C)CCOC1C C1(NC(C2C(C)CN2C(c2scnc2Cl)=O)=O)CC2(CCCCC2)C1 N1(C(C2C(C)OC(=O)N2)=O)CC2CCC1C(NC(=O)CCC1CCCCN1C)C2 N1(C(C(C(=O)OCC)OC)=O)CCN(C)CC1C(=O)NCC(C)(CO)OC c1(OC)ncc(C(C(=O)NCC2CCOCC2)N2CCC2C(C)C)cc1Cl N1(C(=O)C(c2cc(Cl)cc(Cl)c2)O)CC2OCOC2C1 C(CC(C(=O)NCc1ccc(C#N)s1)NC(=O)C(F)C1CCC1)OCC c1(C(C)C(N2CCC(N3C(=O)CCC3=O)C2)=O)nc2ccccc2o1 Cc1nc2cc(C(N3CCOCC(NC(c4cc(Br)n[nH]4)=O)C3)=O)cnc2[nH]1 N1(C(C2(C)CCN(C(C(C=C)O)=O)C2)=O)CCC(F)(C#N)C1 C1(CNC(NC(CC)C)=NCCOC2CCC2)CCn2cncc2C1 CCC(CNC(c1ncc(CC(C)C)nc1)=O)(CC)NC(=O)C(C)C1CC1 c1(C(=O)NC2(CCNC(c3ccc(CO)nc3)=O)CCC2)ccc(O)c(Cl)c1 N1(C(C2C(CC)OCC2)=O)CC(NC(c2n[nH]cc2C(C)C)=O)CC(F)C1 CCC(CCCC(=O)N1CCC(OCC(N)=O)C1)N(C)C(C)=O c1(COCCCC(=O)NC(C)(C)CNC(=O)CCC2CCOC2)ccc(F)cc1 N1(C(=O)COc2ccc(Cl)cc2Cl)CCN(C(c2ccncc2F)=O)CC(O)C1 c1ccc(S(=O)(=O)NC2(C)CCCN2C)cc1[N+](=O)[O-].C(CN(C1CC1)CC)OCC C1(OC)(CNC(=O)Cc2ncc(C)o2)CCN(C(c2ccncc2)=O)C1 C1(CN(C(c2cc(CC)on2)=O)C)CCCC(NC(c2cc3n(n2)CCC3)=O)C1 C=CCC(C(=O)N1CCC(C)(CCn2cc(C(O)CC)nn2)CC1)C(C)C C1(NC(c2cc(C(C)(C)C)on2)=O)C(C)CN(C(C2(C(=O)OC)CC2)=O)CC1C C(=O)(N=c1[nH][nH]c2cc(Cl)ccc12)C12CN(Cc3c(C)n[nH]c3)CC1(F)C2 C1(CC(=O)Nc2cccc(CNC(CC3CC(CC)C3)=O)c2)CCCC(C)(C)O1 C1(C(=O)NC(CN(C(=O)CCSc2ccccc2)CC)C)Cc2nccn2C1 C(=O)(C1=C(Cl)CCOC1)N1C(CNC(c2ccc(-c3ccccn3)o2)=O)CC1 Nc1c(C(=O)NC2CC(O)CN(C(c3cccc(CO)n3)=O)C2)cc(F)cc1F c1(N2CC(CN(C(=O)C=CC3(C)CCOCC3)C)C2)ncnc(Cl)c1C#N c1(C(N2C(C)(COC)CC(NC(c3cnn(C)n3)=O)C2)=O)cc(C)c(F)cc1F CCC(CC(=O)N(C)CC1CN(C(C23CC(C(C)(C)C)(C2)C3)=O)CCO1)SC C1(CC)C(=O)NCCCN1C(=O)C(C1CCN(C(=O)C=C(C)C)CC1)CC N1(C(c2c(OC)c[nH]n2)=O)CC2(CC(NC(c3cc(C)c(C)[nH]3)=O)CO2)C1 C1(CNC(C2ON=C(C)C2)=O)CCC2CN(C(c3cc4c(ncn4C)[nH]3)=O)CC12 C1(O)(CNC(COCCC(C)C)=O)CCCN(C(C2CC(C3CC3)C2)=O)C1 n1(CC(=O)NC2COCCC2NC(c2ccc(CO)nc2)=O)cnc([N+](=O)[O-])c1 N#Cc1nc[nH]c1NC(c1ncc(F)cn1)=O N1(C(C=CC(C)C)=O)CCN(C(=O)CC2CC2)C2CCC12 C1(NC(C(=O)N(C)C)=O)CCC12CN(C(C1COC3(CCC3)C1)=O)C2 C1(CC(=O)N(C2CCCC2)CCCC)CCC(=O)N1C.C12CCN(C1)C2=O Cc1nc(CCCC(=O)N2CC(C)(NC(=O)CN(C)C(=O)OC(C)(C)C)C2)cs1 CN(C)C(=NCc1cccs1)NCc1cccnc1N1CCOCC1 C1(CCC(=O)N(C2CCN(C(c3cocc3C)=O)C2)CC)CCCOC1 N(C)(C1CCCc2cccnc21)Cc1ccc(OC)nc1 C1(C(=O)O)(C(=O)NCCOCCOCCNC(=O)C2CC2)C2CCC12 CC1CN(C(=O)CCn2cnnn2)CC1C(N1CCC(C(=O)NC2CC2)C1)=O c1(C(=O)NC2CC(N(C)CC3N(C(C)=O)CCC3)C2)c(C)noc1C(F)(F)F N1(C(CC2(C(=O)OCC)CC2)=O)CC2CC(CNC(C3CSCCS3)=O)CC1C2 c1(C(N(C(C)CNC(=O)CCS(N)(=O)=O)C)=O)cc2c(ccn2C)[nH]1 c1(C(=O)NCCCN(C)C(C2CCC(C)(O)CC2)=O)ccc2c(c1)CCO2 c1(C(=O)NC(CC)CNC(C2CC3C(C2)C3(F)F)=O)c[nH]c2nc(F)ccc12 N1(C(=O)C(CC(C)(C2CCCC2)NC(=O)CCc2ccc[nH]2)=O)CCNCC1 C(C)(CNC(=O)CCc1ccc(N)cn1)(C(C)C)NC(C(C)=C1CCCC1)=O N1(C(c2cc(COC)no2)=O)CCC(NC(C2CC(C)CO2)=O)C(C)(C)C1 C(=O)(C(C)(C)C(=O)OC)N(CCCNC(C1N(CC)CC1)=O)CC C(=O)(C1=CCCCC1C)NCC(c1ccccc1)CNC(CN(C1CC1)CC)=O c1(C(=O)NCCN(C(=O)C=C(CC)c2ccccc2)CC)cccc([N+](=O)[O-])c1Cl C1(NC(=O)CO)CC2CN(C(=O)CCC(=O)c3ccc(Cl)cc3)CC2C1 c1(C(=O)O)cc(F)cc2c1CCN(C(=O)CCc1cscn1)C2 c1(C(N(C)CCOCCCNC(=O)CSCC(F)F)=O)cnc[nH]1 N1(C(=O)CS(=O)C(F)(F)F)CCC(C2CCN(C(c3ccoc3Cl)=O)CC2)C1 c1(C(=O)OC)cnc(Nc2cccc(NC(=O)C(C)n3ccnc3)c2)c(Cl)c1 C#Cc1cn(C)nc1C(=O)N(CCC(=O)NC1(c2ncc[nH]2)CC1)C1CC1 c1(C(N(CCNC(c2cncn2C(C)C)=O)CC)=O)cnc(O)c(Cl)c1 C1(C)(C(N2CC(O)(C(C)(C)CNC(=O)Cc3cnc[nH]3)C2)=O)CC2CC2C1 c1(NC(Cc2nc(C(c3ccc(F)cc3)OC)sn2)=O)ccc(C)c(Cl)c1 C(C)(C)(C(=O)NC1(C(=O)NCC2CC2(F)F)CC1)OC(C)C c1(OC)nccc(C(=O)NCC(C)C(=O)NCC(O)C(C)O)n1 N1(C(c2ccc(C(=O)NC)cc2)C(=O)N)Cc2cccc(C)c2C1.CCCN(CC)CC c1(SCC)ccc(C(N2CC(C)(NC(=O)CNC(=O)NCC)C2)=O)cc1 c1(CC(=O)Nc2c(CC(=O)NCCC)cccc2)cc(C)ccc1OCCC c1(-n2c(SC)ncc2)ccc(-c2ccc(-c3ccc(C=O)s3)cc2C)cc1C C(=O)(C(C(C)NC(c1ccnc(C)c1C)=O)C(C)C)NCC1CC(C(=O)OC)C1 N1(C(C2CN(C(C)C)C(=O)C2)=O)CCOC2CN(C(=O)CCCS(N)(=O)=O)CC12 c1(OC)ccc(F)c(CN2CC3CCN(c4ncc5c(n4)CCC5)C3C2)c1F Cc1cc(C)c(C(N2CC3CC3(NC(=O)CCn3cncn3)C2)=O)c(=O)o1 C1(C(=O)NCC2N(C)CCC2)CCCCCCN1C(=O)CCCc1cnn[nH]1 CC1(C)C(C(N2CCCC(C3CCCCN3C(C3CSC3)=O)C2)=O)C1(F)F N1(C(C(c2c(C)n[nH]c2C)C)=O)CC(C)(C)OCC1CNC(c1cnsc1C)=O c1(CC)ccc(C(=O)NC(C)CCNC(c2cnn(C3CCC3)c2)=O)[nH]1 c1(CC)ccc(C(=O)NCCCC(C)NC(c2c(C)cnn2C)=O)cc1Cl N1(C(c2c(C)n(C(C)(C)C)nc2)=O)CCC2CN(C(=O)Cc3nccn3C)C2C1 c1(C(=O)N(CCOCc2ccccc2)CC)ccc2nc3n(c(=O)c2c1)CCCC3 S(=O)(=O)(c1ccc(NCCc2ccccc2)cc1I)NCC(CC)n1cccn1 c1(CC(=O)NC2(COC)CCNCC2)ccc2c(Cl)ccnc2c1 C1(NC(C(C)SCC)=O)CCC(C(=O)NCc2sccc2-c2ccccc2)CC1 C1(CCC(=O)Nc2ccc(C(=O)NCC3(SC)CC3)[nH]2)CCCN1C(C)=O c1(C(N2CCC(CNC(C3CCC(F)(F)C3)=O)C2)=O)cc(Br)ccc1Cl N1(NC)CCOC(C2CCCCC2)C1.c1(C(Cc2ccccc2)C)ccn(C)n1 N1(C(C2(C)CC2)=O)CC(C2CC2)(C(=O)NCC2CC2(Cl)Cl)C1 c1(N(C2CCN(C(COc3cc(C)on3)=O)C2)C)ccc(C#N)nn1 C1(C)(NC(C(=O)NCCc2ncc(C)cc2C)=O)CCCC(C)(C)C1 c1(C(C(=O)NC2COC2)N(C)CCC2CCCCO2)cnc2sc(Br)cn12 N1(CC)CCN(CC(=O)NC(C)CCNC(=O)CC2CC2)CC1 CCCCCCCCC(C)C(=O)N1CCN(C(c2cc[nH]c3nccc2-3)=O)CC1 c1(OC)c(C(=O)NC(C)(CNC(C2CC(F)(CO)C2)=O)C2CCC2)ccnc1Cl c1(CC(=O)N(C2CCC(NC(=O)C3=CSCS3)C2)C)cc(Cl)ccc1Cl C1(C(N(CC(F)(F)F)CCOC)=O)CC12CCN(CCc1ccccc1)CC2 CC(C)CC(C(=O)N1CCCC(C(=O)Nc2cnccc2C2CC2)CC1)C(C)C C1(C(=O)NCCCN(C(C(CC)CC(C)C)=O)C)Cc2ccccc2C1(C)C c1(C(=O)NCCC(C)NC(=O)C2=CCSC2)c(Cl)cccc1Br C(=O)(C1CCc2c(Cl)cccc21)N1CC(CNC(CC=CC)=O)OC(C)(C)C1 C1(CC)CN(C(c2oncc2C)=O)CCN1Cc1ccc(Br)o1 Cc1sc(O)nc1C(=O)NC(C)CN(C(=O)C(c1ccccc1Cl)C)C C(=O)(C(CC)CC(F)(F)F)N(CC1CC(NC(CCCC(=O)N(CC)CC)=O)C1)CC CC(C)(CC(F)C(=O)NC1CCCC(C(N)=O)C1)NC(=O)CC=Cc1ccccc1 Cc1ncsc1C=CC(=O)NCC1CC(NC(C2(C)CC(C#N)C2)=O)C(O)C1 N1(C(C2C(CC(C)C)C2)=O)CC23CCC2(COC3)C1.c1(C2C(C=O)C2)cccnc1 CCC(CC(=O)NCCC(=O)OC)N(C)C(C1CCCN1CC)=O N1(C(c2c(OC)nc(C)cc2)=O)CC2CCC1CN2C(=O)CC(C)SC CC1(C)CN(C(C23CCC(O)C2CC3)=O)CCC1NC(c1cnc(C2CC2)o1)=O c1(C(=O)NCC(=O)NC2(CN(C(C3CC(C)C3)=O)C)CC2)ccc(N)cc1 C1(NCC(C2CC2)SC)CCN(C(=O)C(C)CCc2ccccc2F)CC1C C12(N(C3(CS(C)(=O)=O)COC3)C(Cc3cnc(OC(C)=O)s3)=O)CCC(CC1)C2 C1(CNC(c2ccc(C(=O)OC)o2)=O)CN(C(=O)C(c2ccncc2)C)CC1O Cc1cn(C)nc1C(=O)NCC12CC1CN(C(=O)CSCc1ccc(F)cc1)C2 N1(C(CC(=O)NCC#C)=O)CC(NC(=O)CC2CCSCC2)CC12CCC2 c1(N2CC(NC(C3C(C)C3)=O)CC(C)(C)C2)ncnc2c1ncn2C N1(C(CC2CC(=O)OC2)=O)CC2(C1)CN(C(=O)CC1CCCCC13CC3)C2 CC1(C)OCCC1n1nc(-c2cccc(Cl)c2)nc1C1C2CCCCC12 c1(C(N(C2CCCN(C(=O)C3=CCCS3)C2)CC2CC2)=O)ccnc2[nH]ncc12 C=CCCC(C(=O)NCCC1CCCC1(C)C)NC(C12CC(CO)(C1)C2)=O c1(C(=O)NC2CC(F)(CNC(CCS(=O)(=O)NC)=O)C2)cc(C)cc(C)c1N CC(C)C(CCN(C)C(C1CCCOC1)=O)NC(=O)CCCc1cnn[nH]1 CC1CC(NC(=O)CN(C2CCC2)C)CN(C(C2(C3CCCO3)CC2)=O)C1 N1(C(C2N(C(=O)CCCCC#N)CCN(C)C2)=O)CCCCC(C)(F)C1 Cc1ccc(F)c(C(=O)N(C2CCN(C(=O)C(C3(O)CCCCC3)(F)F)C2)C)n1 Cn1ccc2c(C(=O)NC3CC3C(=O)Nc3nccc(Cl)c3Cl)cccc12 Nc1cc(C(=O)NCC2(C(N3CCC4CC4C3)=O)CC3(CC3)C2)cc(F)c1 C1(NC(C(CC=C)C)=O)CC2CCC1CN2C(C1(Cc2ccccc2)CCC1)=O c1(C(N2CC(NC(c3ccn(C)c3)=O)C(C#N)C2)=O)ccc(C#N)c(F)c1 C1(C#N)(OC)CC(C(=O)NC(CCN(C(=O)CN2C(=O)CNC2=O)C)C(C)C)C1 c1(CN(C(Cc2cccc(OCC)n2)=O)C2CCC2)ccc(F)c(Br)c1 C(=O)(CCC(F)(F)C(F)(F)F)NC1CCOCC(C(C(CC(C)C)N(C)C)=O)N1 C1(NC(C(P(C)(C)=O)O)=O)CCN(C(c2cc(Cl)nnc2O)=O)CC12CCC2 N1(CC(=O)NCCO)CCN(CC(c2ccc(F)cc2)=O)C(c2ncc[nH]2)C1 N1(C(c2c(C)nc[nH]2)=O)CC2(CC(CNC(c3ccc(O)c(N)n3)=O)C2)C1 c1(NC)ccc(CN=c2[nH]c(CC(=O)NCC(C)(C)C(N)=O)cs2)cc1[N+](=O)[O-] N1(C(c2n(CC(C)C)ncc2)=O)CC(NC(=O)Cn2ncnn2)CC(O)C1 C(CC(COC1CCCC1)(c1nnnn1C(C)(C)C)Sc1ccccc1Br)OC C1(NC(C(COC)C)=O)CCCCC1CN(C(=O)CCC1CCCC1)C O=C(C1=C(F)CN(C(C2CC23CCCC3)=O)CC1)NCC12CCC(CC1O)C2 N1(C2CC3(CN(C(=O)Cn4cnnn4)C3)C2)CC2CC(F)CC2C1 Cc1cc2c(cc1C)OC(C(N1CCn3c(Cc4nn[nH]n4)nnc3C1)=O)C2 CC1=C(C(=O)NC(CC2CC2)C(=O)NC(C)(C)C(C)(C)C)CCC1 C12CCN(CC1)C2=O.c1(SCCNC(=O)Cc2nc[nH]n2)ccc(F)cc1 C(=O)(CC1=CCCC1)N(CC(O)CN(C)C(C12CCC1CC2)=O)C CCC(C)CC(C(=O)Nc1ccc(C)cc1CO)NC(=O)CCc1cc(C)on1 c1(SC)ccc(C(=O)NCC2(O)CC(C(=O)N(CCC(=O)OC(C)C)C)C2)cc1 CC1(C)CC(NC(=O)CC2(C)CCN(C(=O)C#CC3CC3)C2)C(C)(C)O1 N1(C(CC(C)C2CC2)=O)CC2CCC1C(CNC(c1cn3cnnc3cn1)=O)C2 CN1Cc2cc(CN3CCc4c[nH]nc4C3)ccc2C1=O N1(CC(C)C)CCN(C(=NCC2CCCO2)NCC(F)(F)CO)CC1=O C(=O)(CCS(C)(=O)=O)NCCn1cc(C(c2ccc(OC3CC3)cc2)C(C)C)nn1 C1(NC(=O)Cn2ncccc2=O)CC2CC1CN(C(=O)C=CC1CCCCC1)C2 N1(C(CCC=C)=O)CCC2(CC1)CC(C)N(C(=O)CCCc1ncco1)C2 N1(C(C(C)N2CCCC2)=O)CC2CCCC2(NC(C2CC2(Cl)Cl)=O)C1 C=CC1CN(C(=O)CN2CCCS2(=O)=O)CC1NC(=O)C(=O)N(C)C c1(C(c2n(CC=C)nnn2)NCC2CCOC2)c(Br)n[nH]c1Br C(=O)(C(C)S(C)(=O)=O)NC(CCSC)C(=O)NCc1nccn1C(C)C N1(C(C(CCOC)C)=O)CCC(C)(C)C(CNC(=O)CC(C)CC(C)C)C1 Cc1cc(C(N2CCC(NC(=O)CC(C)C)C(O)C2)=O)c(F)c(F)c1 C(=O)(C1=Cc2ccccc2C1)NC(CNC(c1c(O)ncc(CC)c1)=O)C(C)C CC(C)C(C(=O)N1CCC(NC(=O)C=Cc2ccccc2)C1)C(C)C c1(OC)ccc(OCC(=O)N(C(C)CC(=O)OC(c2cnc(O)n2C)=O)C)cc1 C1(C(C)C)OCCCC1C(=O)NC1CN(C(=O)CN(C)CCO)CC1C N1(C(C2CCN(C)CC2)=O)CC=C(C(=O)Nc2cncc([N+](=O)[O-])c2)CC1 c1(C(OCC)OCC)cn(CC(C)C(=O)NC2CCSCC2)nn1 CCC(C)(C(=O)N1C2CCC1CC(CNC(c1c(Br)nnn1C)=O)C2)C(N)=O CC1(C)CCN(C(=O)CCCNC(N)=O)CC1NC(=O)CC1CCCS(=O)(=O)C1 C(=O)(CCC(=O)N1CC(F)CC1C(=O)NC(CO)C1CCC1)NCC O=C(CCC(F)(F)C(F)F)NC1CCCCN(C(C2CC2C(F)F)=O)C1 CC1CN(C(c2ccncc2)=O)CC1CCNC(C1(C)CCOCC1)=O C1(CNC(C(CNC(=O)CCc2cn(C)cn2)N(C)C)=O)CCCC(C)(C)O1 CC(CN(C)Cc1ccccc1)C(=O)N1CCC1CNC(=O)C(C1CC1)SC N1(C(CN2CC(C)(OC)C2)=O)CCC(C)(NC(C2CN(CC(C)C)C2)=O)C1 N1(C(C=CC)=O)CCCC(CN(C(C2CCCC(=O)N2)=O)CC)C1 C1(NC(=O)COCC(F)(F)F)CCC2CN(C(c3cc(O)nc(O)n3)=O)CC2C1 C1(C(=O)NC(c2cccc(-c3ncccn3)c2)C)CC12CCN(C(C1CCC1)=O)C2 C#Cc1cccc(C(=O)NC(C)CN(C)C(C2CCN(C)C2)=O)c1F c1(NC(c2c(C(C)C)csc2)=O)ccnc(OC2CC2)c1 C(C)(C)(CC(=O)NC(C1CCCN1C(=O)C(CO)N(C)C)(C)C)SC C1(CC(=O)NCC(C2CC2)NC(C(C)Cc2ccccn2)=O)OCCC1(C)C c1(C(N2CC(NC(c3cncc(NC)c3)=O)C(F)C2)=O)ccc2nnc(S)n2c1 C(=O)(C(C)(C)C1CCCN1C(=O)C(N1CCOC1=O)C)N(CCC=C)CC N1(C(C(CC=C)C)=O)CCC2CCN(C(C3CC(C)(C)CO3)=O)CC2C1 C(=O)(CC1=CCOCC1)NCC(CC)NC(c1nc(Br)[nH]c1Cl)=O C1(C)(NS(C2(C(=O)OCC)CC2)(=O)=O)CCN(c2ccc(F)cc2)CC1 N1(C(C2(CCC)CC(=O)C2)=O)CC2(C(=O)NCc3ccnn3C)CCC1CC2 C(=O)(C1=CCC(F)(F)CC1)N1CCN(C(=O)CNC(=O)CC2CC3(CC3)C2)CC1 C1(C(F)(F)F)(C(=O)NC(C2CN(C(C3CC34CCC4)=O)C2)C)CC=CCO1 c1(C(N2CC3CCC2CN3C(C2CC3CC2C2CC32)=O)=O)cc2n(n1)CCCC2O CC1COC(C)(C)CN1C(C1CN(C(c2c[nH]c(=S)cn2)=O)CC1(C)C)=O S(=O)(=O)(c1ccc(Br)cn1)N1C(C(=O)Nc2ccc(OCC(F)(F)F)cc2)CC1 C12(CC(=O)NC3CCN(C(c4nocc4Cl)=O)C3)CCCCC1C2(F)F C1(C(N(CCC(=O)NCCCP(C)(C)=O)C2CC2)=O)CCCC1C1CC1 c1(C(N2CCCC(C3(C)CC3)C2)C(=O)NCCC)cc(=O)n(C)c(=O)n1C C(=O)(C1=COCCC1)N1C(CCNC(CC(C)SC)=O)CCC1 C1(C2(O)CCN(C(C3CC(O)C3)=O)CC2)(NC(COCCC=C)=O)CC1 C1(NC(C(N2C(CC)CCC2)=O)=O)CCN(C(c2ccc(C(N)=O)o2)=O)C12CC2 n1(CC(N2CC(O)(C(C)NC(CC(C)C)=O)C2)=O)cc(F)ccc1=O C1(NC(=O)COc2ccsc2)(CNC(=O)C(F)(F)C2CC2)CCCCC1 N1(C(C(=O)Nc2cccc(C)n2)=O)CCc2cc(F)c(F)cc21 c1(CC)c(C(=O)NCC2(C)CCN(C(c3ccc(CCF)cc3)=O)C2)ccn1C C1(C(N2CC(O)(CC)C2)=O)CCCCN1C(c1cc(CO)ccn1)=O N1(C(C2C(C)CC=CC2)=O)CCOC(C)(CNC(c2cnc(O)c(F)c2)=O)C1 C1(CN(C(=O)CSCc2ccccn2)C)CCN(C(C2(C)COCCO2)=O)CC1 C1(CN(C)C(c2cocc2Br)=O)CN(C(C2CCC(O)C2)=O)CCO1 CC1(C)CN(C(=O)Cc2ccc(Cl)s2)CC1NC(=O)CCc1cncc(O)c1 C#Cc1cccc(C(=O)N(C)CC2CCCCN2C(=O)CSCCN(C)C)c1F C1(NC(CSC)=O)CC2CCC1CN(C(c1c(OC)cc(OC)cc1N)=O)C2 N1(C(C(F)=C(C)C)=O)CCC2CCN(C(=O)CCc3cc(Br)cs3)CC12 CC1C(NC(c2cc(Cl)sc2Cl)=O)CCN1C(c1ccc(C(N)=O)nc1)=O N1(C(C2N(CC)CCC2)=O)CC(NC(=O)C=CC(C)C)CC(F)C1 C(=O)(C1CCCc2c(O)cccc21)NCC1N(C(CCC(=C)Cl)=O)CC(C)(C)C1 c1(N2CCC(C(=O)Nc3ccc(CCC)cc3)CC2)ccc([N+](=O)[O-])cc1Br CON1CCC(CC(N2CC3(CCN3C(C3CCOCC3(C)C)=O)C2)=O)CC1 S(=O)(=O)(c1cccnc1NCC1COC(C)(C)OC1)NC(C(C)CO)C C1(C(=O)NCC2C(NC(=O)COCc3cscn3)C2)CCCCO1 C(=O)(C(C)(C)CC(=O)N1CCOCC1CC(N1CC(C)(C)C1C(=O)OC)=O)OC N1(C(C(CC)N(C)C)=O)CC2(C1)CN(c1ccc(OCCN(C)C)nn1)CCO2 c1(C(N2CCC(N(C(=O)CCc3cnn(C)n3)C)C2)=O)csc2ccc(F)cc12 c1(OC)cc(C(=O)NC2CC2CNC(C23CC(C2)C(C)O3)=O)sc1Cl c1(SC)ccc(CCCC(=O)NC2CCC2CNC(c2cc[nH]c2)=O)cc1 c1(NC(C(C)NC(C(C)OC2CCCCCC2)=O)(C)C)ncnc(Cl)c1F C(CNC(C1(C)CNC(=O)C1)=O)(CC)(CC)NC(CSCCCC)=O Cc1cc(CC(=O)NC2(C)CCCN(C(C34CC(CO3)C4)=O)C2)ccc1F C1(C(=O)NCCC2(C(=O)NCCn3cnnc3)CCC2)CCS(=O)(=O)C1 O=S(=O)(c1ccc(NCCC2CCS(=O)C2)cc1Br)NC1COC1 CC1(CNC(C2CCCOC2)=O)CCCN1c1ncnc(=N)[nH]1 C1(C(=O)Nc2cc(C)no2)CCC2(CN(Cc3cc(I)c[nH]3)C2)O1 c1(C(N2CCCC(N(C(=O)Cc3cccnc3O)C)C2)=O)ccnn(C)c1=O C1(NC(c2nc(COC)sc2)=O)CN(C(=O)CC(C)C(C)C)C2(CCCC2)C1 c1(C(=O)NC2CC(F)(CNC(C3C(C)(C)CC3)=O)C2)ccc(S(=O)(=O)N(C)C)o1 C1(CNC(=O)C(C2CCNCC2)C2CCOCC2)CCN(c2ccccc2)CC1 C1(C(N(CC(=C)C)C)=O)CN(C(c2ccnc(CC)c2)=O)CCC1(C)C Cc1ccccc1C=CC(=O)NCC1CN(C(=O)CN2CCC2C)C(C)(C)C1 c1(CC)ccc(C(N2CC(O)CC2C(=O)Nc2cncnc2OC)=O)c(F)c1 c1(C(C)C)cnc(O)c(C(=O)NCC2CC2NC(c2cc(C(F)(F)F)c[nH]2)=O)c1 C(=O)(C(C)C1=CCCC1)NC(C1CN(C(=O)CCS(N)(=O)=O)C1)C C1(CNC(Cc2c(C)nccc2)=O)CN(C(C2CCCN2CN)=O)CC12CC2 C1(CNc2ccc(-c3c(C)nccc3)s2)CCc2ccccc2N1C(=O)CC#N c1(CC)nc(C)[nH]c1C(=O)NC1CCCC(NC(C2CCCCO2)=O)C1 C(C(C(=O)N(C1CCC1)C1CC1)C(C)(C)C)NC(C1C(OCC)CC1)=O C1(C(=O)NCCCOC(C)C)CCN(C(c2ccc(C3CC3)nc2)=O)CC1O Cc1cnc2n1CCC(n1cc(-c3ccc(C#N)c(N)c3)nn1)C2.C1(N)COC1 C#CC1(CN(C)C(C)=O)CCN(C(=O)CC23CCCC2C3)C1 CC(C)(C(=O)NCC1CCN(C(C2COCOC2)=O)CC1)C(N)=O N1(C(Cc2nnc(C)s2)=O)CCC(C)C1CNC(c1nc(Br)c[nH]1)=O Cc1nc(CC(=O)NC(C)(C)C(C)NC(=O)CCCNC(N)=O)c(C)s1 N1(CC)CCCC(C(=O)NCC(C)CNC(=O)C(c2cscn2)N(C)C)C1 c1(C(=O)NC(CC)(C)CNC(c2ccnnc2S)=O)cc2cccc(C)n2n1 C(CS(=O)(=O)CC(=O)N1CCC(CN(C(c2ccccc2)C#N)C)C1)OC Cc1nc(C2CC2)ncc1C(=O)NC(C1CN(C(C2CCC2)=O)C1)C C1(CNC(CC2(C)CCC2)=O)CC(F)CN1C(c1ccc(C#N)s1)=O C1(C(=O)NCC2CCN(C(c3c(Cl)cc(C)s3)=O)C2)CC12CCOC(C)C2 C1(C(=O)NCc2ccc(C(N3CC(NC(=O)OC)C3)=O)o2)OCCOC1C N1(C(=O)NC(c2cn(C)nn2)C)CC2CCCCC2C1C(=O)N(C)C c1(OCC(=O)NCCCCCCNC(C2C(C#C)C2)=O)cccc(C(C)=O)c1 Cc1cccnc1C=CC(=O)NCC1CCN(C(=O)COc2ccsn2)C(C)C1 c1(NC2CCSC2)ccn2ncnc2c1.O=S1(=O)CC2CN1C2 C1(OC)CN(C(=O)C=Cc2ncc[nH]2)C(C)(CNC(=O)CSCC(F)F)C1 CC1CCN(C(=O)CCC(=O)Cc2ccccc2)CCN1c1cc(O)nc(O)n1 Cc1cccc2c1OC(C(N1CCCOC(CNC(C3CCCCC3)=O)C1)=O)C2 N1(C(C(CCC)S(N)(=O)=O)=O)CCC2(CC1)CC(N=c1cc(Cl)c(O)n[nH]1)CO2 N1(C(C(CCC)N(C)C)=O)CC(C)(C)CC1CNC(C12CCCC(CO1)C2)=O c1(C2(C)COC2)nocc1C(=O)NC1CCC1NC(C1CCCC1C(F)F)=O N1(C(C)C)C(=O)COCC1C(=O)NCC1CN(C(=O)Cc2ccc(O)nc2)C1 CC(C)C(=O)C(=O)NCCC(=O)NCc1cccc(O)n1 CN1CCCC(NC(C2(C)CNC(=O)C2)=O)C1.C12CCCN1CCC(=O)OC2 N1(C(c2cc(OC)ns2)=O)CCC(CN(C)C(C2(OC)CCCOC2)=O)CC1 c1(-c2c(-c3cn(CC(C)C)nc3)n(C)nc2)ccc(F)c(CC(=O)NCCF)c1 c1(C(N(CC(CNC(CCc2cc(C)nn2C)=O)C)C)=O)cnc2occc2c1 C12(C(N3CC(O)(COCC)C3)=O)CC(CO1)N(C(=O)CCCC(C)C)C2 C1(C(=O)NCC#CCNC(COCC(=O)NC)=O)CC(C)(C)CC(C)(C)C1 c1(CCC(C)O)cn(CCC2CCCN2C(=O)CCOC2COC2)nn1 C1(C(=O)NC(CCCCNC(c2nc(C)sc2)=O)C)CCc2nncn2CC1 C#CCC(C)(C(=O)NC(CN(C)C)CC(C)C)NC(=O)CC1C=CCCC1 C(=O)(C(C)CC(N)=O)N1C(C(=O)NCc2nnc(C)o2)CC=CC1 N1(c2ncnc(=N)[nH]2)CC2CCCC(NC(=O)CC3C=CCC3)C2C1 N1(Cc2c(C)n[nH]c2)CC(C(N2CCC3(CC3)C2)=O)C(O)C1 C(CC(CNC(C1CCC1(F)F)=O)NC(=O)CSc1ccncc1)OC c1(CN2C(C(=O)NCC3CCCCC3)CSCC2)ncc2ccccn12 C(=O)(C(CCC1CC1)NC(=O)CNC(C)=O)NCCCC(C)=O CC1(C)CC(CNC(c2cccs2)=O)N(C(=O)CCCc2cc[nH]n2)C1 N1(C(CCC(C)(C)O)=O)CCC=C(C(=O)N(C(C)(C(F)(F)F)c2ccccc2)CCO)C1 c1(-c2cccc(C3(C(=O)NCCCCC#C)CC3)c2)cccn2ccnc12 c1(OC)cc(NCc2c(O)cccc2Cl)cc(C(=O)OC)c1Cl C1(CC)C(NC(=O)Cc2cnoc2)CCN1C(c1cncc(C(C)C)c1)=O n1(CC)c(C(=O)NC(C)(CNC(C2CCCN2CC)=O)CO)nc2ccccc12 c1(C(=O)NCC2CN(c3ccncn3)CCC2(F)F)ccc2[nH]cc(Br)c2c1 c1(OCC)ncccc1CNC(=O)C(C)OC1CCC(CC(=O)OC)C1 c1(CN(CC(=O)Nc2ccccc2)C)cccc(Cl)c1 N1(C(c2scc(C#N)c2)=O)CC2(CCC2)CC1C(=O)NCC(N1CC=CC1)=O n1(CCC)ncc(C(=O)NCC2(F)CCN(C(c3cc(C)cs3)=O)C2)c1C N1(C(=O)CC2CCSCC2)CCN(C(=O)CCC23CCC(CC2)C3)C2COCC12 c1(OC)cccc(C)c1C(N1CCCC(NC(c2cnn(C)c2Br)=O)CC1)=O CCCS(=O)(=O)CC(=O)NC(C)(C)CCCNC(C1(C(F)(F)F)CC(F)C1)=O c1(C(=O)NCC=CCC(N2CC=CC(OC)C2)=O)[nH]ccc(=O)c1C c1(C(N(C2CCCC(NC(CCC=C)=O)C2)C)=O)cccn(CC(C)C)c1=O CN1Cc2ccc(-c3ncc(C(F)(F)F)cc3C(=O)NC3CNC3)cc2C1=O C1(C(N2CCCCCC(NC(CC=C)=O)C2)=O)CC(c2cccc(Br)c2)=NO1 N1(C(C(C=CC)O)=O)CC(C2CC2C(=O)NC2CC3(C2)CC(C)C3)C1 C(=O)(C1=CC2(CCOC2)C1)NC(CNC(c1c(C)c(Br)cnc1)=O)(C)C C1(C(=O)Nc2c(C)ncc(C)n2)CC(N=c2[nH]cnc3cc(I)sc23)C1 C1(CC(=O)NC(CNC(Cc2c(CC)con2)=O)(C)C)CCCN(C)C1 C12(C(=O)OC)CC(NC(c3cnc(C)o3)=O)C1C2 c1(C(=O)NCC=CCNC(C2(F)CCN(C(C)=O)C2)=O)cc(F)cc2cc[nH]c12 C1(N(C)C)CN(C(=O)CCC(=O)N(C)C)CC1C(=O)NC1C=CCOC1 Cc1ccc2c(c1)nc(Cl)n2C#CC(=O)NC1CCCC2(CN(OC(C)(C)C)C2)O1 Cc1cnc(C(=O)NC(C2CCN(C(=O)Cc3ncc(C)o3)C2)C)c(O)c1 C(=O)(C1=COCCO1)N1CCCC(CNC(CC2(C)CCOCC2)=O)C1 C1(C(=O)NCCCCCNC(Cc2c(C)n[nH]c2C)=O)OC2CCC1CC2 C(=O)(C(F)C(C)CNC(=O)CSCc1cccnc1)Nc1ccc(SC)cc1 Cc1ccc(S)cc1.c1(CCNC(CC(=O)NCCCN)=O)cc(C2CC2)[nH]n1 c1(CC(=O)N(CCN(C(=O)CCCS(N)(=O)=O)C)C)ccc(S(C)(=O)=O)cc1 C(CC(=O)NC1CC2CCC1N(C(c1cccc(F)c1O)=O)C2)(C(F)(F)F)OC C(=O)(CCCCCF)NC1(CC(C(=O)NCc2cnc(CC)[nH]2)F)CC1 C1(C(=O)Nc2c[nH]nc2C2CCNCC2)CCC2(CCC2)CC1 CC(CC(=O)NCCCc1ccccn1)N(C(=O)C(F)C1CCCC1)C c1(C(=O)NCCN(C(c2ccc[nH]2)=O)C2CC2)cccc(C#CC2CC2)c1 C(=O)(C#CC(C)(C)C)NC(C1CCCCN1C(=O)COC1(C)CCOCC1)C C1(C(=O)NCC(C)(C)NC(=O)COCCCOC)CC2CCCCC12 CCCCCCCCC(C)C(=O)N1CCC(N)(Cc2cccnc2OC)CC1 C1(NC(C(C(=O)OC(C)(C)C)c2ccccc2)=O)CC(C)(C)OC1=O c1(C(=O)NC(C2(CC)CC2)=O)cnn(CCC2CC2)c1C.C=C1CC1CN(C=O)C CCC(CC)(C(=O)N1CCN(C(=O)CNC(C2CNC(=O)N2)=O)CC1)OC C=C(F)CN=c1nc(N(CC(c2ccc(Cl)cc2)C)C)cc[nH]1 C12CCN(C13CC3)C2=O.c1(OCC)cnc(C(=O)NCC2CC2NC)cn1 N1(C(c2c(CC)scc2)=O)CC(CNC(c2[nH]c(=N)sc2CC)=O)C(C)C1 C1(N(C(=O)CN(C)C(C)C)CC)CCCN(C(c2ncsc2C)=O)CC1 C(=O)(CCCCC(F)(F)F)N1CCCC(C(C)NC(C2CCOCC2)=O)C1 C1(C(N(C)Cc2cn(CC3CC(C4CC4)C3)nn2)=O)NC(=O)C2CC12 c1(-c2cn(CCC(N3CC4C(C3)C4(F)F)=O)nn2)cc2cnc(F)cc2[nH]1 CCCCC(C)C(=O)NC(CNC(c1cccc(-c2cc[nH]n2)c1)=O)CC Cc1ccc(C(N2CCCCC(N(C)C(c3ccc(O)c(F)c3)=O)C2)=O)cc1F C(=O)(CCCC(F)(F)CO)NC1CN(C(c2c(C)ccnc2)=O)CC1O C1(C(=O)NCCN(C(=O)C=CCO)CC2CCCC2)CC2C=CC1CCC2 C1(NC(=O)CC2CCCC2(F)F)CN(C(=O)CCOC2CCCCC2)CCC1F c1(NCC(CC=C)NC(c2ccc(C)nn2)=O)ncc(Br)cc1C#N c1(C(N2CCOCC(NC(COCC=C)=O)C2)=O)ccc2c(c1)CN(C)C2 c1(C(N2C(C=CC(=O)NCC(CC)(C)Cl)CCC2)=O)ncc(C#N)cc1C C1(C(N2CCC(F)(COC)C2)=O)COc2ccc(Br)cc2C1 CC(Cc1cnc[nH]1)C(=O)N(C)CCn1cc(C(N2CCCC2)C2CC2)nn1 C1(NC(C2(C)CC2c2ccccc2)=O)CC2(C1)CC(CNc1cc(Cl)ncn1)C2 C1(CC(=O)NC(C(N2CCOC2c2cccs2)=O)C2CCOC2)CCCC1N C1(c2n(Cc3c(C)cccc3)nnn2)(NC2CCOC2)CC2COCC2C1 CC(CNC(C1CC=CC(O)C1)=O)C(F)C(=O)N1CC2(CC2)CC1CO c1(OCCC)nc(C)ccc1C(=O)N(CC(O)CN(C)C(C1CC1C(=O)OC)=O)C CCC(C)(CCNC(=O)COC(C)C)NC(=O)COCC(=O)N(C)C C1(C2CC2)(CNC(c2c(C#C)c[nH]n2)=O)CCN(C(C2(C(=O)NC)CC2)=O)C1 N1(C(c2ccc(C)o2)=O)CCCC(C)C1CNC(c1nn(C)cc1C)=O c1(C(N2CCCC(Nc3ncnc4ccsc34)C2)=O)ccc2n[nH]cc2c1 C1(N(C(C2C(C)C2)=O)C)CCN(C(C2CCCN(C(=O)OC(C)(C)C)C2)=O)CC1 Cc1nc(O)sc1C(N1CCC(OCC(=O)NC2CN3CCC2C3)C1)=O C1(NC(=O)NCCc2cnc(C)[nH]2)CCC2CC2CC1 N1(C(C=C(COC)C)=O)CC2CCC(C1)C2NC(=O)CC1CCCC(O)C1 C(=O)(C1COCc2ccccc21)NC(C)(C1CC1)C1CC1 C1(OC)CC2(CN(C(=O)CC(CNC(c3cc(F)c[nH]3)=O)C3CCC3)C2)C1 C1(NC(CC(C(C)OC)NC(c2nc(CC)oc2)=O)=O)CCOCC12CCC2 C(=O)(CCC(C)(C)C)N1CC(CNC(C(COC)(F)F)=O)C(C)C1 C1(NCCCO)CCc2onc(C(=O)NS(Cc3cccc(C)c3)(=O)=O)c2C1 c1(C(N(C(C)C2CC2)CC)=O)ccc(CNC(=O)CC2CCCN(C)C2)cn1 C(=O)(C1=CCCCCC1)N(C)CC1CCN(C(c2c(O)ccc(CC)c2)=O)CC1 N1(C(C2(NC(c3ccc(CC)o3)=O)CCCC2C)=O)Cc2ncsc2C1 c1(C(=O)NC2CCC(CCNC(COCCOCC)=O)C2)cc(C)oc1Br C1(C(=O)NC(CCN(C(CN(C(C)=O)C)=O)C)C)CCCC12CCC2 c1(C(=O)NC(CCOC)CNC(C2(n3cccn3)CCC2)=O)nc(Cl)oc1C C(=O)(C(C)S(=O)(=O)C(C)C)NCC1(OCC)CN(C(=O)C(CO)C(C)(C)C)C1 c1(C(=O)NC2CCC(C)N(C(c3c(O)ncnc3O)=O)C2)c[nH]c2nccc-2c1 C1(C)(CC)CCC(C(N2CC(CNC(=O)C(C)NC(C)=O)C3CC23)=O)O1 c1(C(=O)NCC(CC)NC(c2oc(COC)cc2C)=O)ccc(C#N)cc1 C1(C(=O)N(CCC(=O)NCCn2cnnc2)C)(CC)CCOCC1 N1(C(CC2(CC=C)CCCC2)=O)CCN(C(C2CC(F)C2)=O)C(CC(F)(F)F)C1 Cc1ocnc1CNC(=O)CN(C(c1cn(C2CC2)cn1)=O)CC1CC1 C1(CCN(C)C(C2CCC(O)CC2)=O)CCN(C(C2CC2(C)C)=O)CC1 c1(C(N2CC(NC(c3c(CCC)nns3)=O)C(O)C2)=O)cc2cccc(C)n2n1 C1(CC)CN(S(=O)(=O)C2CC(OC)C2)CCCO1 N(C(=NCc1cc(C2CC2)on1)NC1CC1)CN(C(=O)CN1CCCC1)CC(F)F C(=O)(C1=CC2(CCOCC2)C1)N1CC(C)C(CNC(C23CC(C)(C2)OC3C)=O)C1 C(CC(C)N=c1[nH]c2c(c(=NCCCc3cnn(C)c3)[nH]1)CCC2)SC Cc1ccc(C2(NC(C3(n4cnnn4)CCN(C)C3)=O)CCC2)cc1Cl C(=O)(C(C)(C)Cc1ccccc1)NCCC1N(C(C(=O)N(C)C)=O)CCC1 c1(C(C)C)c(C(=O)NCCCCN(C)C(C2CCCS2)=O)cnn1C N12CCCC(C)C(=O)NC1=CC=C(Cl)C=CN(C)C=CC=CC2 n1(CCn2c(C3CCC(=O)NC3C3CC3)nc(C)n2)c(C)nc2ccccc12 C1(CNC(C2(CC(C)=O)CC2)=O)CC(O)C(O)CC1C(=O)NCc1occc1C C1(CNC(=O)NCc2ccc(NC)cc2)CCCC(C)(C)C1 c1(C(N)=O)cc(C(N2CCC(NC(C3CCCC4CC34)=O)CC2)=O)cc(F)c1 N#Cc1ncc(Cl)c(N2CC3CCCC2C3CNC(C2CC3(CCCC3)C2)=O)n1 C1(NC(C(C)(C)C)=O)CC(NC(=O)C=CCN2CCCC2)C12CCC2 C(=O)(C(C)(C)CC)N1C(CN(C(c2c[nH]c(=NC)s2)=O)CC)CCC1 c1(C(=O)NC2CN(C(C(=O)NC(C)C)=O)CC2C)ccnc(F)c1F C1(C(=O)NCC(C(C)C)NC(=O)Cc2cccc(C3CC3)c2)CCC(C)(C)OC1 CC(O)C(C(=O)N1CCC(NC(C2CC3(CC3)C2)=O)C1)NC(=O)C(C)(C)C Cn1cc2c(C(N3CCC(C)(C)C(NC(C4CC(F)C4)=O)C3)=O)cccc2n1 C(=O)(CCCN=C1NCCSN1)NC.C1(CN2CCCC2)CCCN(C(C)=O)C1 CC1(C)CCCC(C(=O)NCC(C)(C2CC2)NC(=O)C=Cc2ccccc2Cl)C1 C=CCCC(CCC)(c1nnnn1CC1CCOCC1)NC1CC12CC(O)C2 Cc1ncc([N+](=O)[O-])cc1C(=O)NCC(C(C)C)NC(=O)C1=NOC2COCC12 CCC(C)(COC)C(=O)N1CC2C(CNC(=O)CN=S(C)(C)=O)C2C1 c1(N2CCC3(C(F)(F)C3)C2)nc2cc[nH]c2c(=NC2CC3C(C2)C3(F)F)[nH]1 N#Cc1cccc([N+](=O)[O-])c1NC1CN(C(C2CC2(Cl)Cl)=O)C1 N1(C(C(C)NS(CCCC)(=O)=O)=O)CCC(CO)(NC(c2[nH]nnc2C)=O)CC1 c1(C(=O)NCC2(CC)CCOC2)ccc(CNC(=O)Cc2cn[nH]c2)cc1 N1(C(c2ccc(C(C)=O)o2)=O)CCC(CNC(=O)CSc2nncn2C)CC1C c1(C(N(C)CCC2CCN(C(=O)C3=NOCC3)CC2)=O)cccc2ncn(C)c12 C=C(C)CC(C(=O)NOCC(N1CC(N(C)C)C(O)C1)=O)OC(C)=O C1(C(=O)NCC(CCCC)NC(=O)CC2CCC(F)(F)C2)CC2(CC(C)=NO2)C1 C1(NC(C2C(NC(C3CCOC3)=O)CCO2)=O)CCn2nnnc2C1 Cn1cc(Br)c(CC(N2CC=CC(NC(=O)CSc3ccccc3)C2)=O)n1 C(=O)(C(CC#N)c1ccccn1)N(C)CC1C(c2ccccc2)C1(F)F C1(NC(CC=C)=O)CC(Nc2ccc(CNC(=O)CSC3CC3)cc2)C12CCC2 O=C1CC(C(=O)NC2CCCC(NC(C3(n4cccn4)CCCC3)=O)CC2)=NN1 C=Cn1ncc(C(=O)NCC(C)C(=O)NCc2nnc(CC)s2)c1N C1(C(C)C)CCOC1C(=O)NC(c1cccnc1)C(=O)NCc1cnc(O)o1 c1(C(=O)OC)ccc2c(c1)C(CNC(=O)Nc1[nH]cc3c1CCC3)CCC2 c1(C(=O)NCC(CN(C(CN(C(C(C)C)=O)C)=O)C)O)ncoc1C1CC1 N(C1CCCc2ccc(Cl)cc21)C(c1c(-n2cccc2)sc(C)c1C)=O C(C(F)(F)C(=O)N1CCC(C(C)NC(c2[nH]ncc2C#N)=O)C1)OC C1(C(C(=O)N(C2CNC2)C2CC2)N(c2ncc(Br)cn2)C)C2CCCCC12 C1(NC2(CC)CCC(O)CC2)CCC2CN(C(=O)CC34CCCC3C4)CC2C1 C(CC(C(=O)N)NC(N)=O)c1cccc(-c2nn[nH]n2)c1.CS c1(C(=O)NCCNC(c2coc(O)n2)=O)ccc([N+](=O)[O-])cc1Br CC(C)CCCCC(=O)NCCNC(c1cnc2sccn12)=O N1(C(CC(C)F)=O)CCN(C(c2c[nH]nc2-c2cccs2)=O)CC1C1CCC1 CCC(C)C(C)(O)CNC(C1C(CC)CCN1C(c1sc(C)cc1C)=O)=O c1(C(=O)NC2CCC(CCNC(c3c(CC)n[nH]c3)=O)C2)c(C)nn(C)c1Cl N#Cc1ccc(C(=O)NC2CC(C(N3CCC(F)(CO)C3)=O)C2)s1 c1(CNC(CCCOC(C)=O)(C)c2nnnn2C2(C)CC2)cc(C)cnc1F N1(C(Cc2cc(C)no2)=O)CCC(C(=O)NCC(F)C2CCC2)C12CC2 C1(CNC(Cc2nnc(C)o2)=O)CCN(C(C2CCCN2C(C)C)=O)C1(C)C Cc1[nH]cc(C(=O)NCCCCC(C)(C)NC(c2ccc(C#N)s2)=O)c(=O)c1Cl N1(C(C(C(=O)OC)OC)=O)CCC2(CC1)CC2CNC(c1cncc(N)c1C)=O Cc1nc2cc(C(N3CC(NC(C4CC5CCC(C4)O5)=O)C(C)C3)=O)ccc2s1 Cc1ccc2nc(CNC3CCN(C4CCCC4O)CC3)cn2c1 C1(CC)CN(C(c2c(OC)cccc2F)=O)CCN1S(=O)(=O)C(C)C CC1=C(C(=O)N(CC(C)(C)NC(=O)C(C)n2cccn2)C)CCC1 c1(C(N(CCCN(C(=O)C(C2CCCCCC2)F)C)C)=O)nccnc1C(N)=O C12CCC(CC1)NC(=O)C(=O)N2C.C1(O)(C(N2CCCC2)=O)CC1(C)C N1(C(C23CN(C(C4CN(C(C)C)C4)=O)C(C2)CO3)=O)CCn2ncc(O)c2C1 CC(=O)C(C)CC(C)C(=O)N1CCC(C)(C)C(CNC(C2(C(C)C)CCC2)=O)C1 C1(CNC(C2C(C)OCC2)=O)CN(C(c2ccn(CCF)n2)=O)CC(C)(C)O1 c1(C(C(=O)N(CCN(C(=O)C(C)n2ccnc2)C(C)C)C)C)ccc(O)cc1 C(=O)(CS(=O)(=O)CCOC)NCC1(NC(C=CCC)=O)CCCCC1 C(=O)(CCC(=O)N1CCC(N(C(=O)Cc2ccsc2Cl)C)C1)N(C)C c1(OCC=C)ccc(Cl)c(C(=O)NC2CCN(C(=O)CSC(F)F)CC2O)n1 c1(C(=O)NC2(C(=O)NCCCOC=C)CCCC2C)cc(C)cc(O)n1 N1(C(C(C(C)C)OCC)=O)CCC2CN(C(c3c(C)nnn3C)=O)CC2CC1 Cc1ccc(C(=O)NCC2CCC(CNC(=O)C(C)C3CCC3)CC2)c(N)c1 C1(O)(CC#C)CC(C(=O)NCc2cn(CC(N3CCC3CF)=O)nn2)C1 C(=O)(C(C(C)(C)C)NC(C1CC1NCc1ncc(C)cc1Br)=O)OCC N1(C(c2cnc(C)c(N)c2)=O)CCC(C)N(C(=O)C(N2CCSCC2)C)CC1 C1(C(N(CCSc2ccccc2)CC)=O)C=CCN(C(=O)C(C)(C)C)C1 c1(OCC)ccc(CCC(=O)NCC(C2CCC2)NC(c2cnn[nH]2)=O)cn1 N#Cc1cc(C(=O)NCC2CCCCN2C(=O)CC(F)(F)Cl)cc(Br)c1 Cc1ccc(CC(=O)NC2CC(CO)N(C(c3cnc(C4CCC4)s3)=O)C2)cc1 C1(NC(C2N(C(c3cc(CC)on3)=O)CC2)=O)CC(N(C)C)C1(C)C Cc1cc(C(=O)NCC2CN(C(=O)C=CBr)CC23CC3)cc(Cl)c1 N1(C(c2cc(OC)ncn2)=O)CC2(NC(c3cccc(C(F)F)c3)=O)CCC1C2 N(C(=NCCC1CC1)NCc1ccnc(N2CCCC2)n1)CC(C)OC c1(C(N2CCCC(N(C(=O)C(C)OCCOC)CC)C2)=O)ccc(C#N)nc1O n1(CCC(=O)NC2C(CNC(=O)CCn3cnnn3)CC2)cc(Cl)cn1 C1(C)(CNC(C2(Cl)C(C)C2)=O)CN(C(=O)CC2(C#N)CC2)C(C)(C)C1 N1(C(COc2c(CNS(C)(=O)=O)cccc2)=O)CCC(NC(=O)CCSC)CC1 CCC(CC(=O)N(C)CC1CCCN(C(c2cnc(S)n2C)=O)C1)OC c1(N2C(CC)CN(C(c3ccc(Cl)cc3)=O)CC2)nc(C#N)nc2ccccc12 C1(C(N(CC(CC)NC(=O)CCc2ncc(CC)[nH]2)CC)=O)CCCC(C)(C)C1 C(C(CNC(=O)CCn1nc(C)c(C)c1C)C(F)(F)F)NC(C1(C#C)CC1)=O O=C(C1CCCc2scnc21)NCCNC(C1(c2ccco2)CC1)=O n1(CC)cnc2c(NCC(C)N(C)C(C3(C(=O)NC)CCC3)=O)ncnc12 CN1Cc2ccc(C(N3CCCCC(NC(C4CCS4(=O)=O)=O)C3)=O)cc2C1 c1(C(C(=O)NC2CCN(CCNC(CC=CCC)=O)C2)O)cccc(C)c1 c1(NC(CNS(CC)(=O)=O)C)cc2c(cc1N(C)C)OCO2 C12(C(N3CC(CC=C)(NC(c4coc(C(F)(F)F)c4)=O)C3)=O)CCCC1C2(F)F c1(C(N2CC3(C2)CN(C(c2ccnn2CCF)=O)C3)=O)cc2c(Cl)cccc2[nH]1 c1(C(C)NC(=O)C(O)CC(N)=O)ccc2nc(O)[nH]c2c1 c1(C(=O)NCC(=C)CCNC(=O)CC(C)c2ccco2)cc(C)nc2ncnn12 N1(C(C=C(C)C)=O)CCC(O)(CC(=O)Nc2cncnc2Cl)CC1 Cn1c(C(N2CC(F)(F)CC2CCNC(C2CCO2)=O)=O)cc2sccc12 c1(C(N2CCCC(N(C(Cn3c(C)ncc3)=O)C)C2)=O)nnn2c1CCC2 C1(NC(C(C)CS(C)(=O)=O)=O)CN(C(=O)C(F)C(F)(F)F)CC2(CCC2)C1 N1(C(C(C)OCC#C)=O)CCC(C)(CCNC(=O)Cc2c(C)cccc2F)CC1 C12(CNC(c3n(OC)cnc3C)=O)CCCCC1N(C(=O)C(C)SC)CC2 c1(OC)cc(C#N)ccc1CNC(=O)NCCC12CCCC1C2 N1(C(C(C)(C)C2CCC2)=O)CCN(C2CCCN(C(=O)Cn3cnnc3)C2)CC1 CCCC(C(=O)N1CCN(C(C2(CC(F)F)CCC2)=O)CC1)NC(N)=O Cc1ccc(C(=O)NC(C2CCCN(C(=O)CC3(C)CCOCC3)C2)C)nn1 c1(OC(C)C(N2CCCC2C2(NC(=O)C(O)C3CCCC3)CC2)=O)ccccc1 N#Cc1cc(C(N2CCC(CCC(=O)NC(C3CCCCC3)(C)C)C2)=O)c[nH]1 N(C(=NCCCCF)NC(c1ccccc1)C)Cc1cc(OC)cc(F)c1 C1(NC(=O)CN2CCCCC2)CC(NC(C2CCC23CCC3)=O)C(O)C1 N1(C(C=C(C)C)=O)CCC(CO)(CNC(=O)CC2CCN(CCF)CC2)C1 N1(C(C(C)N(C(=O)CCCC(=O)C2CC2)C)=O)CCCC2C(=O)NCC12 c1(C(N2CCC(N(CCC)C(c3nc(C)nn3C)=O)C2)=O)cncc2ccsc12 C1(CNC(=O)C2=C(Cl)CC2)CCC2(CCC2)CN1C(=O)CC1CC2(CCC2)CO1 c1(C(N2CCCC(N(c3nc(CC)nc(=N)[nH]3)CC)C2)=O)cccc2c1OCC2 C(CCC(O)C(=O)NCCN1CCC(C)(C)C1)NC(CCNC(=O)OCC)=O CC(O)(CC(=O)NC1CC12CC(NC(=O)CCN1CCC1)C2)C(F)(F)F c1(CC)cncc(C(=O)NCC2(NC(c3nc(CC)oc3C)=O)CC(F)(F)C2)c1 C(C(C(C)C(C)C)NC(c1cc(OC)cnn1)=O)NC(c1c(C)nc(CC)s1)=O c1(CC)cc(OCC(=O)NC2CCCC2NC(C23CC4CC2C3C4)=O)ccc1Cl C(C(C)(C)C(=O)OCC1CC(C(=O)OC(C)(C)C)C1)OC(=O)C(C)(C)C C(CCC(C)(C)C(=O)N(CCC(N1CCCCC(C)(F)C1)=O)CCO)OC C(=O)(CC(C)C)NC(CC)CNC(=O)CCOC1CC1 CON(CC1CC1)C(=O)CCC(C(C)C)NC(C1CC(C#N)(OC)C1)=O C1(NC(=O)COCCF)C2CC3CN(C(c4ccc(Cl)c(Cl)c4O)=O)C1C3C2 C(c1ccc2c(c1)OCO2)=CC(=O)OCC(C1(F)CCCC1)=O C(=O)(CC(C1CC1)NC(C1CC(F)(F)C1)=O)NC(CCN(CC)CC)C C1(c2cccc(NCc3c(OC)cccc3C)c2)Cc2ccc(OC)cc2O1 C(=O)(CC1=CCN(C(c2cc(=N)[nH][nH]2)=O)CC1)NCC(CC)(C)C(C)O c1(NC(CC=C)CO)ccc(S(=O)(=O)NC(COCC)CC(C)(C)C)c(Cl)c1 c1(C(N(CC(=O)O)CC)=O)cc(SC)n(C)n1.C1(=O)CCCn2cc(nn2)CN1 C(C)(C)(CC(=O)NC1(C)CCSCC1)NC(C(CO)N(C)C)=O CCC(CC(=O)N(C)CCN(C(=O)Cc1cnnn1C)C)C1CC1 C1(C(N2CC(C)C(CCNC(=O)COCCCF)C2)=O)CCC2(CCC2)O1 C1(NC(=O)C=Cc2ccco2)CCOCC1C(=O)Nc1cnc(C2CC2)o1 C1(NC(C2(C)CCOC2)=O)CCN(C(C2CC2OC(C)(C)C)=O)C1(C)C N1(C(C2C(CN(CC)CC)OCC2)=O)Cc2cccc(O)c2C1.C1CC(=O)N1 c1(NC)cnncc1C(=O)N(C(C)C(=O)NCc1coc(C)n1)C1CC1 c1(NC(N2CC3CCC3(CF)C2)=O)ncnc2c1COC2 Cn1nc(Br)nc1C(c1nnnn1C1(C)CC1)NCc1ccncc1Br c1(C2N(C(c3cnn(C)c3C3CC3)=O)CCC2)ccc(Br)cc1Cl n1(CC(=O)NCCCN(C(=O)C(C)n2ccnc2)C(C)C)ccnc1 N1(C(=O)OC(C)(C)C)CCc2cc(S(=O)(=O)NCC(F)C3CCC3)c(F)cc21 C1(OC(C2(C(=O)OC)CC2C)=O)CN(Cc2ccncc2)CCC1C(=O)OC N1(C(CC23CC(C)(OC2)C3)=O)CCC2CCC(C1)N2C(C1(C)CCNC1=O)=O Cc1ccc2cc(C(=O)NC(C)(CNC(C3CC34CCC4)=O)C3CCC3)cn2c1 N1(C(c2c(OC)cncn2)=O)CC(C(=O)NCC(C)CO)C(F)(F)C1 CN1CC(F)CC1C(N1CC=CC1CNC(=O)CC(C)(C)C)=O C12(NC(Cc3ccc(C)c(Cl)c3)=O)CCCN(C(C3CN(C)C(=O)N3)=O)CC1C2 n1(C(CC)C)nc(C(N2CC(NC(c3c[nH]ccc3=N)=O)C2)=O)cc1C C(=O)(C(C)(O)C(F)(F)F)N1CCC(=C)CC1C(=O)NCC1CCOC1C(C)C Cc1cccc(COCC(=O)NC(CNC(c2ccncc2)=O)C(C)(C)C)c1 c1(C(N(C2CCN(C(c3c(OC)nsc3)=O)C2)C)=O)csc2ccc(F)cc12 CCS(=O)(=O)CC=CC(N1CCC(C(=O)Nc2ccccc2C(=O)OC)CC1)=O C1(CNC(C=CSC)=O)CC2CCC1N(C(=O)C(C)Oc1cccnc1)C2 c1(CN(C(=O)Cc2cnnn2C)C)cc(Cl)ccc1OC(F)F C1(CC)CCCC2(CCN(Cc3ccc4c(C)noc4c3)C2)O1 c1(CNC(c2c(CNC(=O)CC3COCCO3)ccs2)=O)ccc(F)cn1 N1(C(CC(C)CN(C)C)=O)CCCC12CCN(C(c1cc(CN(C)C)on1)=O)C2 C1(C(C(=O)OC)C)CCCN(C(=O)C(=O)N(c2ccccc2OC(F)F)C)C1 CC1CCC(C(=O)N(CC(C)(C)NC(=O)C(C)(C)Nc2ccccn2)C)C1 C1(NC(=O)CCc2cn[nH]c2)CN(C(C2CC2c2ccccc2)=O)CCC1O c1(C(N2CC(C)C(CNC(=O)CC3CCCC3)CC2)=O)cc2ncccc2[nH]1 N1(C(CC(CC)O)=O)CC2CCN(C(c3ccc(C(F)(F)F)cc3O)=O)C2C1 c1(C2CC(C(=O)OC)C2)cccc(Cl)c1.C12CC(C1)N2 O=C(N=c1[nH]onc1C1CC1)C1CCN(Cc2ncc(Cl)s2)CC1O c1(CCC(N2CCOC(CNCc3cncs3)C2)=O)cc(Br)ccc1Cl C=CC(F)(F)C(=O)N1CCN(CC(C)NC(c2ccc(C(C)C)cc2)=O)CC1 C1(C(=O)NCCN(C(=O)C(C)(C)C(F)F)C)Cc2cc(F)cc(F)c2O1 N1(C(CNC(=O)OCC=C)=O)CC(NC(=O)CC2CC=CC2)Cc2ccccc21 C(=O)(C1Cc2ccc(C)cc21)NCCC(=C)CNC(c1cc(OCC)no1)=O N1(C(c2ccc(C)s2)=O)CC2CCCC2(C(N2CC3(CCC3(C)C)C2)=O)C1 c1(CC)onc(C)c1CNC(c1occc1CNC(c1cocn1)=O)=O N1(C(C2CCCOC2)C(=O)NCC=C)CC(F)(F)CC1(C)CN(C)C c1(-c2n(C3CCCN(CC)C3)nc(C)n2)cc2cccc(OC)c2o1 c1(CC)onc(C(=O)N(C2CCN(C(C3CC(OC(C)=O)C3)=O)CC2)CC)c1C CCCC(C)(C)C(=O)N1CCOC(C)(CNC(C2CC3(CC3)CN2C)=O)C1 CCC(CC(=O)NOC(=O)CCO)NC(C)=O.C(C(C)(C)C)OCCOC(C)=O N1(C(C(C=C)(C)C)=O)CC2CC(NC(=O)Cc3cn4c(C)csc4n3)CC(C2)C1 CN(CCCC(=O)NCCC1CCN(C(c2cccc(F)c2)=O)C1)N=O CC(CCC(C)(C)C)C(=O)NCC1CC(NC(=O)C=Cc2ccc(Cl)cc2F)C1 C(=O)(C1CS(=O)(=O)c2ccccc21)NC(CCNC(C1OCCN(CC)C1)=O)C C#CCCCCCC(=O)N(CCCNC(=O)Cc1csc(C)n1)CC c1(C(N2CCN(CCOC(C)(C)C)CC2)=O)cc2ncsc2[nH]1 CC1CN(C(c2ccc(C#N)[nH]2)=O)CC1CCNC(C1(N2CCOC2=O)CC1)=O c1(OC)ccc(C(=O)NCC(C2CCOCC2)C)c2cnccc12 C1(C(=O)NCCCCC=C)CCCC(NC(C2C3CCCC23)=O)C1 C1(CNC(c2c(C)ncs2)=O)CN(C(=O)C(C)C2=CCCC2)CCC1(C)C C1(C)(C(=O)NC(C2CCOC2)CC)CC(NC(=O)COCCOC)C1 C1(NC(C(CNC(=O)OC(C)(C)C)(F)F)=O)CCC2CC1CO2 O=C1C2=CC3=C(Cl)N=CNC3=NC2CCOCCC2(CC(C)(NC(=O)CO)C2)N1 CC1CC(NC(=O)COc2ccc(Cl)c(F)c2)CCN1C(c1cnns1)=O C1(N(C(C2CC2C(=O)Nc2ccccc2C(N)=O)=O)CC)CCCCCC1 c1(C(CNC(=O)CC23CCC(CC2)C3)NC(c2cn[nH]c2)=O)ccc(F)cc1F c1(C(N2CC3(CN(C(c4cc(COC)[nH]n4)=O)C3)C2)=O)cc(F)c(CO)c(F)c1 c1(OC)cc2c(cc1C(=O)NC1CN(C(C3CCCC3OC)=O)CC1C)OCO2 c1(CNC(CC(CNC(C(C2CCCO2)OC)=O)C)=O)nn(C)c(=O)n1C C1(NC(C2CS(=O)(=O)C2)=O)CCC2CCN(C(c3ncccc3C3CC3)=O)C1C2 c1(CN(C(C(=O)OC)C#N)C)ccc(COC(C)C)cc1 C1(CS(=O)(=O)N(C2CCN(C(CC)=O)CC2)C(C)=O)CC2C(O)CC2O1 C(=O)(C1=C(Cl)CCC1)NC(CNC(CC1C(C)(C)CCO1)=O)CO Cc1cncc(CCC(=O)NC2CCCC2(C)CNC(=O)Cn2cc(Cl)cn2)c1 C1(C)(CC=C)CN(C(c2cc(CNC(=O)CC=CC)no2)=O)C1 C1(NC(=O)NC(C)CC(=O)NC2CCCC2)CN(C)CC12CC2 N1(C(C(CCOC)C)=O)CC2(CC(NC(C3(C)CCN(C)CC3)=O)C2)C1 C1(NC(COC2CCC(C)CC2)=O)COCCN(C(c2cocc2Br)=O)C1 Cc1nc[nH]c(=NCC2(CNC(c3coc4c3COC4)=O)CC2)c1F c1(OC)ccc(C(=O)NC(C)CN(C)C(c2cccnc2C)=O)c2ccccc12 Cc1nc(CC(=O)OCc2cnc(C3CCC3)o2)cs1 C1(CC(=O)NCC(CNC(COCc2n(C)ccn2)=O)(C)C)CCCC(C)(C)C1 Cc1cc(O)ccc1CC(=O)NCCC1CC(NC(C2CCCCC2)=O)C1 N1(C(c2cnn(CC)c2C)=O)CCC(C2(NC(c3occ(C)c3C)=O)CC2)CC1 C1(CC(=O)NCCC2CC(C(=O)NCc3cc(C4CC4)on3)C2)CC=CCC1 c1(CC(N2C(C(N3CC(C)OCC3)=O)CC(F)C2)=O)cc(Br)ccc1Br O=C(C1=C(Cl)CCCC1)NC1CC2(CCN(C(=O)Cn3cc(CO)nn3)C2)C1 Cn1c(=O)c2cc(N(C(=O)Cc3ccc(OC(F)F)cc3)CCl)cnc2n(C)c1=O n1(C(CC)CC)nc(C(=O)NC(C)CCNC(=O)CC23CC(C2)C3)ccc1=O C(C(CC1CC1)C(=O)NC1(C)CCOC1)NC(c1cnc(C)s1)=O N1(C(C2(C)COC2)=O)CC2CCC(C1)C(NC(=O)C(F)(F)c1ccccn1)C2 C1(C(=O)NCCCC(C)CO)CC2CCC1N2C(C1CN(C2COC2)C1)=O C=C1c2ccccc2C(=O)N1CC(=O)NC1C2CN(C(=O)Cc3cncs3)CC12 C1(F)(C(=O)NCCOC2CCN(C(C(c3ccc(C)o3)C)=O)C2)CCS(=O)(=O)C1 C(=O)(C1CCCc2ncnn21)NCC(C)(C)OCCNC(C(C)C1CC1)=O c1(C(N(C2CCN(C(C(C)OC)=O)C2)C)=O)ccc(-n2cncn2)cn1 c1(C(=O)NCC2(O)CN(C(C(C)NC(=O)NC)=O)C2)c(O)ccc2ccccc12 N1(C(c2ncc(C)cc2C)=O)CC2CN(C(=O)CSC(F)F)CCC2(CO)C1 c1(OC)c[nH]nc1C(=O)NC1CCCC1NC(=O)C(C)Sc1ccccn1 c1(C(N2CC3C(CN(C(c4[nH]cc(CC)c4)=O)C)C3C2)=O)cc(F)c(F)cc1Cl N1(C(COC2CC(C#N)C2)=O)CC2CC1CN(C(c1cc(O)cnc1Cl)=O)C2 c1(SC)c(C(=O)NC(C)CC(C)NC(C2(C)CCC(=O)C2)=O)cccc1F Cc1cc(N)c(F)c(C(N2CCCC(CNC(C3CC3C(C)C)=O)C2)=O)c1F Cc1nc(C(=O)NC2CC(C)CN(C(C3CC3CF)=O)C2)c2n1CCCC2 CCC(C)(C)C(O)C(=O)N1CC(CC(=O)Nc2cccc(C)c2C)(OC)C1 c1(NC(c2sc(I)cc2Cl)=O)csc2ncccc12 N1(C(C=NOC)=O)CCC(C(=O)N(C2CCCC(C)C2C)CC)C(C)C1 c1(N2CC(C)C(NC(c3ccc(C(F)F)nc3)=O)CC2)nc2cccc(Br)c2o1 C#Cc1ccc(C(=O)NCC(C)(C)NC(c2nn(C)c(N)c2C)=O)cc1 N1(C(C(C)(C)C(F)F)=O)CCC(CNC(=O)C(O)C(F)(F)F)C(F)(F)CC1 Cc1ccc(C(=O)Nn2cccn2)c2c1CCC2 c1(C(=O)NC2C(C)CCN(C(=O)CN(CC(C)(C)C)C)C2)ncn2ccccc12 Cc1nnsc1SC1CCCN1C(=O)C(=O)OC(=O)C(F)(F)F N1(C(C(Cc2ccoc2)NC(C2CC3(CCC3)C2)=O)=O)CCN2CC(O)CC2C1 c1(C(=O)NC2CC(C)N(C(c3cc(N)c(Cl)c(O)n3)=O)C2)cc2cnccc2[nH]1 C(C(C)(C)CNC(=O)Cc1ccoc1)N(C(=O)CN(C)C(C)=O)CC C(=O)(CC(F)(F)C(F)(F)F)N(C1CCCCC1)CCNC(C(C)C#N)=O c1(C(NNC(Cc2nc(-c3ncc(C)cc3F)sc2)=O)=O)ccc2c(c1)CCC2 N1(C(C2N(C)C(=O)NC2)=O)C2CCCC1CC(NC(c1cc(C(N)=O)c[nH]1)=O)C2 Cc1c(CNC(=O)NCC23CCCC2CNC3)cccc1C(F)(F)F C=C(CNC(=O)C(CC)c1ccccc1)CCNC(=O)CCSc1ccsc1 Cc1cc(NCc2nnnn2C2CCOCC2)cc(C)c1O N1(C(c2c(CCC)[nH]cc2)=O)CCCC(CCN(CCOC)CC)CC1 C(CS(=O)(=O)CCCN1CCC(NC(c2cnccc2Cl)=O)C(C)C1)OC C1(C(=O)NC2(CNC(CC(C)n3cccn3)=O)CCCC2)CC2CC1CC21CC1 CC1Oc2cc(F)ccc2C1NC(C1CCCN(C)C1)=O C1(C(=O)NCC2(NC(CC(C)N(C)C)=O)CCOCC2)CC12CC(C)(C)C2 N1(C(c2c(OC)ccs2)=O)CCC(C)(CCNC(=O)COCc2ncccn2)C1 c1(CCC(=O)NC2CC3CC2N(C(c2c[nH]nc2F)=O)C3)c[nH]c2ccccc12 N1(C(CS(=O)(=O)NCC)=O)CC(NC(C2CCC2COC)=O)CC12CCC2 c1(C(=O)NCCN(C(C)C)C(=O)CNS(=O)(=O)C2CC2)cc2ccccc2n1C c1(CS(N2C(C)(C(N3CCC(N(C)C)C3)=O)CCC2)(=O)=O)cccc2cc[nH]c12 N1(C(C(CC)OCC)=O)CCN(C(c2cnoc2C2CCC2)=O)CC1CCO N1(C(c2n[nH]cc2Cl)=O)CCC2(CCCC2Nc2nc3ccc(Br)cc3s2)CC1 C1(C(=O)NC2C(NC(c3c(C)nc(CCC)s3)=O)CC2)CC(=O)NC1(C)C C(=O)(CC1CN(C)c2ccccc21)N1CCC(N(OC)C)CC1 C12(NC(CC(C=C)CCC)=O)CCCC(CN(C(=O)C(C)(C)O)C1)C2 C(=O)(C(O)C(C)(C)C)NCC1CC(F)(CNC(c2c(C)nc(C(C)C)o2)=O)C1 n1(CC)c(CN(C(=O)C(N)C2CCCO2)CC(C)C)cnc1C N1(C(CC=C=C)=O)CC2(CC2)CC1CNC(c1ccnn1C(C)CC)=O N1(C(C(C)N=[N+]=[N-])=O)CCOCC(NC(C2CC3C(C2)C3(C)C)=O)C1 C1(C(N(C)CC2CCCC2)=O)CCCCCCN1C(c1sccc1C#N)=O Cn1ncc2c1CCCC2C(=O)NC(C1CCOCC1)C1CCCC1 N1(C(C(C)=O)=O)CCC2(CC1)CC(NC(c1scnc1C(F)F)=O)C2 Cc1cc(C(=O)NCCC(C)N(C)C(C23CCC2C3)=O)c(C)n1-c1ccccc1 C#CC1(C(=O)NC(C)(CC)CC=C)CCN(C(C2CCC3(CCC3)C2)=O)C1 C1(C(N2C3CN(C(c4n(C)ncc4Cl)=O)CC32)=O)CCCOC1(C)C Cc1cccc(OCCC(=O)NC23CC2CN(C(=O)C(C)SC(F)(F)F)C3)c1 c1(C(=O)NC2CN(C(C3NC(=O)CC(=O)C3)=O)CC2F)cc2cc(Cl)ncc2[nH]1 n1(CC(=O)NC2CC(OC)CN(C(C=C(CC)C)=O)C2)ncc2ccccc12 C=C(Cl)CCC(=O)NCCSCC(=O)NCc1cncc(CC)c1 Cc1cc(C2(F)CCN(c3cncn(C)c3=O)C2)cc(F)c1 C(=O)(C(C)(C)CCSC)N1C(CNC(c2c(CC)noc2)=O)CCC(C)C1 CC1CN(C(c2nccc(Cl)c2F)C(=O)NCC2CCOC2)CC(=O)N1C Cc1c(F)ccc(C(N2CCN(C(C3CC3C(N)=O)=O)C(C3CC3)C2)=O)c1F Cc1ccc(NC(=O)C(C)(C)C2CCCN2C(C2CCCC3(CC3)C2)=O)c(O)c1 CSC=CC(=O)NC1(CNC(=O)C(C2CCOCC2)C)CCOC1 c1(NC(C2(c3cn(CCC(=O)NCC)nn3)CC2)=O)ncc(CC)s1 CCCC(C)(C)CC(=O)NC(CC(C)C)C(=O)NCc1cnn(CC(=O)OC)c1 CC(C)CC(C(=O)N1CCN(CC2CCC(F)C2)CC1C)c1ccccc1 C(=O)(C(C)CCC)N1CCC(C(=O)NC(c2nccs2)CC)C1 CC(C(C(=O)NCC1CCOC1)N(C1(c2ccccc2Cl)CC1)C)C(C)(C)C c1(C(N(CCC(C)C)CCNC(=O)N)=O)ncnc(NC)c1F.CO c1(C(=O)NCC(CCCC)NC(=O)C(C)CCO)occ2c1CCOC2 c1(C(N(CC(C)NC(C2(F)C3CCCC23)=O)CC)=O)cccc(Br)c1F c1(NC(C2(C)N(C(C(CC(C)C)OC)=O)CCC2)=O)cc(O)c(C)cc1C C(C(=O)N1CC(NC(=O)CCc2nncs2)C1)(N(C)C)C1CC1 C(CCC(=O)N1CC(c2ocnc2CNC(=O)CC2CCCCO2)C1)OC Cc1nc(C2CC2)nc(S)c1C(=O)NCC1(C)CC(NC(=O)C(C)CF)C1 c1(C(N2C(CNC(c3ccccn3)=O)COCC2)=O)cc(O)nc(Cl)c1 n1(CC(C)N(C(=O)COC2CCOC2)C2CC2)cc(C2CCC=CO2)nn1 c1(CC(=O)NCC2C3N(C(CC(CC)C)=O)C(CC3)C2)ccc(F)cc1[N+](=O)[O-] CCC(C(=O)NCC12CCC1CN(C(c1[nH]ccc1COC)=O)C2)C(C)(C)CC N1(C(c2cc(C)ncc2)=O)CCOC2(CCCN(C(=O)C(C)C3CCOC3)C2)C1 c1(C(N2CC(NC(c3c(F)ccc(C)c3)=O)C(C)C2)=O)cc(N)c(C#N)c(F)c1 C=CC1(CC(=O)NC2CC(C(C)NC(=O)C(C)C(O)CC)C2)CCOCC1 O=C(C1Cc2ccccc21)N1CC2CCCC(C1)N2C(=O)C1=NOCC1 c1(N(C2CCN(CC(=O)NCCCF)C2)C(=O)C2CC2)cc(F)c(F)cc1O N1(C(C(N2C3CC(N(C)C)CC2CC3)=O)=O)CC2(C1)NC(=O)NC2=O c1(CNC(CN2C(CNC(=O)Cc3ccc(Cl)cc3)CCC2)=O)ccc(O)cc1 C1(C(=O)NC2CCC2N(C)C)(CC)CCCN(C(=O)C(n2nccc2C)C)C1 c1(C(N2CC(O)(CNC(=O)CC3CC3(Cl)Cl)C2)=O)cncc2c(F)cccc12 c1(NC(C(C(C)OC)N2CCC(OCCN(C)C)CC2)=O)ccc2c(c1)OCO2 C1(N=[N+]=[N-])(C(NOCCOCC)=O)CCN(C(=O)Cn2cc(C)cn2)C1 C1(NC(CC)=O)CC2(CCN(C(c3ccn(C4CCCC4)n3)=O)CC2)C1 C1(NC(C(C)Cc2ccnn2C)=O)CC(F)CN(C(=O)C=CC2CC2)C1 c1(C(N(C2CN(C(COC(C)=O)=O)CC2O)C)=O)cn(C(C)C)c(=O)nc1O N1(C(Cc2ncc(C)s2)=O)CC=CC(NC(=O)C(O)C2CCCC2)C1 C(=O)(C1=CS(=O)CCC1)N1CC2C(NC(C(c3c(F)cccc3F)C)=O)C2C1 C1(NC(c2cc(O)cc(O)c2)=O)CN(C(C2(F)CCCC2)=O)CCC1C(F)(F)F C(C)(CC(C)(C)OC)NC(C(C1CN(C(c2cc(CC)no2)=O)C1)O)=O c1(N2CCCC(CS(C)(=O)=O)C2)nc(NCC2(CF)CCC2)c2ccsc2n1 c1(C(CNC(c2cc(CSC)no2)=O)NC(C2CCC(C)O2)=O)ccc(C)cc1 N1(C(C(C)SC)=O)CCC(C2CCCN(C(=O)COC(F)(F)F)C2)C1 c1(C(CNC(C(N2CCN(CCO)CC2)CC)=O)=O)cccc(=S)n1O N1(C(c2c(CCC)nco2)=O)CCC2(CC1)CN(C(=O)CC1COCC(C)O1)C2 N1(C(=O)CC2CCCC2)CCC2CN(C(=O)C3Cc4ccccc43)CC2C1 c1(C(=O)NCC(C2(O)CN(C(C3CCOCC3)=O)C2)(C)C)ccn(C2CC2)n1 c1(OC)cc(C(=O)NC23CC2CN(C(=O)Cc2cccs2)C3)ccc1C c1(CN(CC(C)(C)F)CC#C)cc2c(cc1OC(F)F)OCO2 c1(N2CC(C)C=C(C)C2)nc2c(c(=NCc3ccc(C)c([N+](=O)[O-])c3)[nH]1)SCC2 C1(C(=O)NC2CCC(NC(c3cc(CC)no3)=O)CC2)Cc2cc(C)ccc2O1 CC1(C)CCN(C(=O)CCc2ccc[nH]2)CC1C(=O)NCC(C)(O)CO CCCCC(C)C(=O)N1CC(CNC(=O)Cc2ccc(COC)cc2)CC(C)C1 N1(C(c2c(C)scn2)=O)Cc2ccccc2C1CNC(=O)Cc1ccon1 N1(C(CC(C)c2cccnc2)=O)CCC(NC(=O)CCSC(F)(F)F)C(O)C1 c1(C(=O)NCC2C(CNC(c3cncc(C)n3)=O)C2)coc(S(N)(=O)=O)c1 S(=O)(=O)(c1cc(Cl)ccc1OCC(N)=O)N1C(C)CCC(CC)C1 C#Cc1cccc(C(N2CCCC(C(=O)NCC3CCCN3C)C2)=O)c1 N1(C(c2cc(C)c(C)nc2O)=O)CCCC2CN(C(c3ccoc3)=O)CCCC12 c1(C(=O)NC23CCC(C2)N(C(=O)C(C2CC2)C2CC2)C3)cc([N+](=O)[O-])ccc1O C1(CCC)CN(C(=O)Cc2cscn2)CCN1C(=O)CN(C)CCO c1(OC)ncccc1C(=O)N(C1CCC(CNC(c2ccc(C)o2)=O)CC1)C C12(C(=O)NCCCNC(CC3ON=C(CC)C3)=O)CCN(C1)S(=O)(=O)C2 N1(C(C(CCCC)O)=O)Cc2ccccc2CC1CNC(C1(C)CC1(F)F)=O Cc1c[nH]cc(C(=O)N(C)CC2(NC(C3CSCCS3)=O)CC2)c1=O C1(C(N2CCC(CNC(CC3(C=C)CC3)=O)C2)=O)CCCC(=O)N1C c1(C(N2CCC3(NC(=O)CC4=CCCC4)C(C2)C3)=O)cc(Cl)cc(Cl)c1O CC(C)C(C(=O)N(CC(N)=O)C)C(C)NC(c1cnn(C)c1N)=O CC1(C)OC(=O)c2c1ccnc2N(CCNC(=O)C(N)=O)C1CC1 c1(C(C)(F)F)nc(NCC2CC2)cc(=NCC2C=CCCC2)[nH]1 N1(C(C)=O)CCCC1(C)C(N1CCC(CCN(C)NC(=O)C=CCO)CC1)=O N1(C(C(CC(C)C)NC(C)=O)=O)CC2CC(NC(=O)CCOCC(C)C)C(C2)C1 N1(Cc2c(OC)ccc(F)c2F)CCc2cc(C(=O)NCCC(C)C)ccc2C1 CCCCCC(F)C(=O)NC1(CF)CCN(C(c2cc(C(F)F)n(C)n2)=O)C1 Cn1cc(C(=O)Cc2csc(NC(C(=O)OCCCC3CC=CCC3)=O)n2)cn1 Cc1nc(O)sc1C(=O)NCC#CC(=O)N1CCC(N2CCCC2)C1 O(N(C)C(=O)CNC(=O)C(CCF)NC(=O)C(C)C1CCC1)CC CC1CCC(C(C)(CCCO)NCc2ccc(OC(F)(F)F)cc2)C1(C)C c1(C(N2C(CNC(=O)CC3CSCCS3)CC2)=O)ccc2[nH]ccc2c1 c1(C(N2CC(N(C(=O)CC34CCCC3C4)C)C(O)C2)=O)coc2cccc(O)c12 c1(SCCC)ccc(C(=O)NCC2(CO)CN(C(=O)CC3CNC(=O)O3)C2)cc1 c1(C(=O)NCCCC(C)NC(=O)CNC=O)coc2c(Cl)cccc12 Cc1cccc(C(=O)N(CC(C)CNC(=O)Cc2csc(CN(C)C)n2)C)c1F c1(C(=O)NC2CC(NC(C3CC34CCCC4)=O)C(O)C2)ccc2c(c1)CC2 C1(CNC(CC(C)C2CC2)=O)CCCCN1C(c1coc(Cl)n1)=O C1(C)(C(=O)NCCCC(CO)NC(CC2N(C(C)=O)CCC2)=O)CCC(=O)NC1 C(=O)(CC(CN(C)C)C(F)(F)F)NC(C)CCNC(=O)C(c1ccc(O)cc1)=O c1(SC)ccsc1C(=O)NC1CC1NC(c1cocn1)=O Cc1nccnc1C(=O)NCC1(CNC(C2CCS2(=O)=O)=O)CCCC1 c1(C(=O)NC2(C)C(NC(C(n3c(C)ncc3)C)=O)CCC2)ccn2nccc2c1 C1(C(=O)NCC(CCOC)O)COCCN1C(C1(C(=O)N(C)C)CC1)=O C=CCCCCCCC(=O)N(C1CCN(C(C2(C)C(C)C2C)=O)CC1)CCC N1(C(c2cc(OCC)no2)=O)CC(OC)CC(NC(=O)C(O)CSC)C1 c1(OC(C)C(N2CC3(CCCC(NC(N)=O)O3)C2)=O)cnc2ccccc2n1 CN1CC(C)(NC(C2(F)CCN(C(c3cccc(F)c3F)=O)C2)=O)CCC1=O c1(C(=O)OC)ccc(OC)cc1NC(=O)Nc1cnn(-c2ccc(Br)cc2Cl)c1 C1(CNC(C(C)OCCCC)=O)COCCN1C(c1cc(C(C)C)sn1)=O c1(C(=O)NCC2CCN(C(C3CC(CC)(CC)C3)=O)C2)cc(C(C)C)n(C)c1C c1(C(=O)NCC2OCCCN(C(c3cc(C)oc3)=O)C2)ccc2sccc2c1 C1(C(=O)NCCNC(C)=O)CCCCC1NC(c1cncc(Cl)c1)=O.NCO CC(c1ccccc1)=CC(N1CCOCC1CO)=O.C12(CC1)C(=O)NC2=O c1(C(N(CCCN(C)C(C23CCC2C3)=O)C)=O)cc2cnccc2cc1F C1(CC(=O)NCC(C)CNC(=O)C=C2CCC2)CCCC(=O)N1 c1(NC(C2CCC(NCc3cc(OCC)ncc3)C2)=O)ncc(Br)cc1F C1(NC(=O)C(F)=CCCF)COCCN(C(=O)Cn2ccc(Br)n2)C1 CC(CCC(=O)NC1(CCN2CCCC2)CC1)NC(C1(SC2CC2)CC1)=O C12(CC(=O)NC(C3CCN(C(CCOC)=O)C3)(C)C)CCCN1CCC2 N1(C(C2(C(=O)OCC)CC2)=O)C(C(N2CCSCC2)=O)CC1C Cc1cnn(CC(C)NC(=O)COCCC2CCCC2)c1.C1(=O)CN1 c1(SC)scnc1C(=O)NC(c1ncc(C(=O)N(C)C)s1)C.C1C(=O)N1 C1(CNC(C2CC(NC(=O)COCC(F)F)C2)=O)CCC(O)C1 c1(CCCC(=O)NC2(CF)CCN(C(C=CC(N)=O)=O)C2)c[nH]c2ccccc12 c1(C(=O)NCCOC2CCN(C(C3(c4cc[nH]n4)CC3)=O)C2)cc2c(F)cccc2s1 C1(C(=O)NC(c2nocc2C(=O)NOCC2CCCO2)C)CNC(=O)C1 CS(=O)(=O)c1ccccc1SCc1ccc(NC(N)=O)cc1 c1(COC(C2(C)CCCN(c3nnc(C)s3)C2)=O)noc2c1CCCCC2 c1(CC(=O)NC(CN(C(C=CC(C)C)=O)C)C)ccc2c(c1)CCOC2 c1(CCOC(C(C2CC2)OC)=O)nc2ccccc2s1 c1(C(=O)NC2CC(C)SC2)ccc2c(c1)CN(C)CCC2 N1(C(C(C)N(C(C)=O)CCO)=O)CCCCC(CCC=O)C1.C(CCC(C)C)O C1(NC(COC)=O)CCCC(CNC(C2CCC2(C)C)=O)C1 C1(C(=O)NCCCC2(O)CCCC2)CC12CCN(C(=O)C(O)C1CCC1)CC2 C(CCC(=O)NC(c1ccccc1)C(C)NC(=O)CC=C(C)C)NC(C)=O N1(c2ccc(C)nn2)CCc2c(c3ccccc3n2CCOC(C)C)C1 C(CN=c1[nH]c(=NC2CCCn3cnnc32)c2c(ncn2C)[nH]1)(C1CCCC1)OC C(N=c1cc(-c2cccs2)nc[nH]1)C1CN(C(C(C)CC(N)=O)=O)CC1(C)C c1(C(N(C2CN(C(c3cccc(CO)c3)=O)C2)C)=O)ccc2ncnc(O)c2c1 c1(C(=O)NC2(C)CCCC2NC(=O)CC2=CCCC2)c(O)cnc2ccccc12 CCCN(OC)C(=O)C12C(NC(C3CC(C)CCO3)=O)C3CC1C2C3 C(=O)(CCCCC1CC1)NCC(c1ccccc1)NC(CSCC=C)=O c1(C(=O)N(CC(=O)C(C)C)C2CC2)ccc(F)c(-c2csc(COC(C)=O)n2)c1 c1(CNC2(C)CC(O)C2)cnc2c(c1)CCC2 c1(CCC=C)cccc(S(=O)(=O)NCC2(CCCO)CCOCC2)c1 c1(C(=O)NC2CN(C(CSCC)=O)CC2C)nn(C)cc1S(N)(=O)=O Cc1cc(OCC(N2CCN(C(C3CC(F)(CO)C3)=O)C(CO)C2)=O)ccc1Cl C1(C(N(CC(O)CN(C)C(C2COCCO2)=O)C)=O)Cc2ccncc2C1 Cc1[nH]c2ccccc2c1CC(=O)NCC(CO)Nc1ncnc2c1SCCC2 C12(CNC(=O)CCc3ccon3)CC1CN(C(=O)CCc1nc(C)no1)C2.CO C(C(C(C)OC)N=c1cc(C(C)=O)nc(Cl)[nH]1)OC C1(C#N)(C(=O)NC(CC(=O)NC(C=C)C)C)CC12CCC2 N1(C(C(C)Oc2cccnc2)=O)CC2CN(C(C3CN(C4CCC4)C3)=O)CCC12 N1(C(C(=O)ONC(=O)C2(NC3CC(=C)C3)CC2)CC)C(=O)c2ccccc2C1=O CC1CCN(C(=O)C(C2CCCO2)NC(C2COCC2C(N)=O)=O)CC1 C#CCC(C)C(=O)NCC1CC(NC(c2cnn(C(C)(C)C)c2N)=O)C1 Oc1ncc(CC2(NCc3ccc(Br)cc3I)CC2(F)F)c(O)n1 C(=O)(CC(C)(O)C1=CCCC1)NCC1C(CNC(c2n(CC)ncn2)=O)C1(F)F C1(C(=O)NC(CNC(C(N2CCNC2=O)C)=O)CO)CC(=O)N(C2CCCC2)C1 C1(CCC)CC2CCC(C1)N2C(c1cocn1)=O.C(=O)(CCC1(C)CC1)NCC C(=O)(CCC(N)=O)NCCC1CC(NC(c2[nH]cc(C(C(C)C)=O)c2)=O)C1 N1(CC(=O)NCC(C)CN(C)C)CCCCCC1.C123CC(CO1)(C2)NC(=O)CC3 C(CS(=O)(=O)CC(=O)NC1CC(NC(=O)CCc2ccc(SC)cc2)C1)OC C1(CNC(C(N2CCCC(O)C2)C)=O)CC12CCN(C(C1CCCC1)=O)CC2 c1(N2CCC(C)(NC(c3ccn4nccc4n3)=O)C2)nc2ccc(F)cc2s1 c1(-c2ccc(CNC(C)C(=O)O)cc2)ccc(O)c(F)c1 C(=O)(C(C)(C)CCNC(=O)CC1CCCC2CC12)N(c1ccc(Cl)cc1)C c1(OC)ccc(Br)cc1C=CCSC1CC2(CCC2)CN1C(=O)OC(C)(C)C C1(C(=O)NC(C)CCCNC(=O)CC2C(C)(C)C2(C)C)CC12CCCCCC2 C1(C(=O)NC2CSC2)CCN(Cc2cccc(Cl)n2)CC1O C(=O)(CCCC(C)NC(c1nsnc1O)=O)NC(C#C)CC(C)C N1(C(C)=O)CCC(C)(C(=O)NC(C2CCCN2C(=O)C(C)C(C)O)C)CC1 Cc1nc(CC(=O)NC2CN(C(=O)Cn3cnc(=N)[nH]3)C2)co1 n1(CC(N2CCC(CNC(C3(CC)CCC3)=O)C2)=O)nc(C(F)(F)F)c(Cl)c1C Cc1oc(Cl)nc1C(=O)NCC1CC(C(=O)N(C)CC2(O)CCC2)C1 Cc1cc(C(=O)NC2CCN(C(c3cccs3)=O)CC2F)cc2[nH]ccc12 N1(C(CCOC(C)=O)=O)CCCCCC(NC(=O)COCC(F)(F)F)C1 C(=O)(C1CCCc2nc[nH]c21)N1CC(NC(CN2CCN(CC)CC2)=O)C(F)C1 CCC1=NOC(CC(=O)NC2COCCC2C(=O)N(CC(C)O)CC)C1 C(CC(C)(C)C(=O)NC1CC12CCCC2)NC(C(C)NC(=O)C1CC1)=O CC1CCN(C(c2cc(CO)[nH]n2)=O)CC1NC(=O)CCCc1cccnc1 c1(NC2(C)N(C(=O)OC(C)(C)C)CC=C2)cc(C(F)(F)F)ccc1Cl C1(NC(CSC(C)C)=O)CC2CCC1(NC(c1c[nH]nc1-c1ccsc1)=O)C2 c1(C(N(CCCN(C(=O)C(F)(F)CC2CC2)C)C)=O)nccc2ncccc12 c1(C(=O)NC(CCOCC)C(=O)NCCCn2nccn2)ncc(F)cc1F C1(NC(C2C(OC)CCCC2)=O)CC(CCl)C12CCC2 N1(C(c2cc(C)oc2)=O)CC2C3CCC(C2C1)N(C(=O)C(C1CC1)C1CC1)C3 c1(C(N(C(CNC(c2cncc(SC)c2)=O)C)C)=O)c[nH]c2ccccc2c1=O c1(C(=O)Nc2c(C)c(C(=O)N(C)C)ccc2)csc2c1CCC(C)(C)C2 CC1(C)CN(C(c2cc(Cl)sc2Cl)=O)CCC1NC(=O)CCCCCc1cccs1 C(=O)(C(F)NC(=O)CC)NCCCOCCCN.S(C(F)F)C(=O)NC c1(C(=O)NCCOC)ccc(N)cn1.C1(OCCN(C)C(=O)C2CC2)CSC1 C(C)(C)(CC(F)C(=O)N1CC2(COC(C)C2)C1)NC(c1noc(CC)c1C)=O c1(-c2nc(C(C)C)nn2-c2cnn(C)c2)[nH]nc2ncnc(O)c12 N1(C(c2c(C)nc(O)s2)=O)CC(NC(C2CCCCC2(C)C)=O)CC(O)C1 CC1(C)CN(C(=O)COC2CCCC2)CC1N=c1nc(C(F)(F)F)[nH]s1 C(=O)(C1=C(Cl)CCC1)N(CC(C)N(C)C(c1cnc(C(C)(C)C)[nH]1)=O)C C(=O)(C(C)C(O)CC(C)C)NC1(C(=O)OC)CC1.C1CCCC(=O)N1C Cc1cc(C(=O)NCC(C(=O)N(CC(C)N(C)C)C)N(C)C)cc(F)c1 c1(OCC(=O)NC2CN(C(C3CCC4CC34)=O)CC2(F)F)cc(Cl)ccc1Cl N1(C(C2C(C(=O)OC(C)(C)C)C2)=O)CCC(C)(CNC(c2cccnn2)=O)C1 Cc1ccc(CN2CCC3(CC3C(=O)Nc3cncc(O)c3)C2)cc1C#N c1(N(C)CC2CCCN2C(C2CCC(C)(C)OC2)=O)ncc2c(c1C#N)CCC2 C1(SC)CN(C(c2cc(CN(C)C)c[nH]2)=O)CC1NC(=O)C1=CCCO1 C1(C(N2CCC(N)C2)=O)(CNC=O)CCN(C)C1.C1(=O)CN1.C(=O)(C(=O)OC)OCC c1(C(=O)NC2(CCNC(C3CC3c3cccs3)=O)CC2)coc(Br)n1 c1(C(=O)NC2(CO)CCCN(C(C(CC(N)=O)O)=O)C2)cnc2cccnn12 CC1CCN(C(=O)C(=Cc2ccccc2)NC(N)=O)CC(C)O1 c1(C(C)C)ncsc1C(=O)NC1CNCC1C(=O)O C(=O)(CC(C)(C)C#N)NCC(CCC)NC(C1(C)CC(C)=NO1)=O C1(C(N2C(CNC(c3nocc3C3CC3)=O)C=CC2)=O)CCC(=O)N1C1CC1 C1(C(N(CC(O)C2CC2)C)=O)CC2CCC(C1)N2C(C1CCCC(=O)CC1)=O N1(C(CC2CC(C)C2)=O)CC2(CCOCC2)CC1CNC(=O)CCSC(F)(F)F c1(C(=O)Nc2ccc(NC(c3cn[nH]c3)=O)nc2)ccc2c(c1)COB2O C1(NC(C=CCCC)=O)COCC1NC(C1SCC=C1C)=O C12(Nc3nccc(C)n3)CCC(CC1)N(C(c1cc(N(C)C)ccn1)=O)C2 C#CC1(C(N2CCC(CO)C(C)C2)=O)CCN(C(=O)CCc2cnc(C)s2)CC1 C(=O)(CCCC(=O)NC1CC1CNC(c1ccnc(CO)c1)=O)OCC c1(C(=O)NC2CCC(C)(NC(C3CC3C#N)=O)CC2)cccc2c1CCO2 CCCCC(C)CCC(=O)N1CC(C2CN(C(c3n[nH]cc3CC)=O)C2)C1 C1(C(N(C2CCN(C(=O)CC3C(C)(C)C3(C)C)C2)C)=O)CC2(CCOC2)C1 N#Cc1c[nH]c(C(=O)NC2CC2C(=O)Nc2cncc(Cl)n2)c1 C#CCC(C(=O)NC(CC)C1CCC1)NC(c1nnsc1N)=O C=CC1(CC(=O)N(C2CCCC2O)C)CN(C(=O)C(C)C2CCC2)C1 CN1C2CCC1CC(C(=O)NC1CN(C(=O)C3=CCS(=O)(=O)C3)CC3(CC3)C1)C2 N1(C(C(COC)C)=O)CCN(C(=O)CCCOC(=O)N(C)C)C(C(C)C)C1 C1(CNC(C(C)(Cl)Cl)=O)CN(C(=O)CC2(C#N)CCC2)C2(CCC2)C1 C(=O)(C(F)(F)CCn1cc(-c2ccccc2Br)nn1)NC(C)C(F)F C1(C(=O)NC2C(OC)CN(C(=O)C=Cc3ccccc3)C2)CC2(CCCC2)C1 c1(C(=O)NC(CCN(C(=O)CC(C)(F)F)C)C(C)(C)C)nnn2c1CSCC2 CC1CN(C(=O)CC2OCCC2C)CCC1CNC(=O)CSC(F)(F)F c1(OC)ccc(C(N2CCN(C(c3cc(O)cc(O)c3)=O)CC2)=O)cc1O CC(C)CC(C)C(=O)NC(C(=O)NCc1c(O)cccc1Cl)C(C)(C)C C(N=c1[nH]cc(C#N)cc1C)C1C(C(F)(F)F)CCN(C(CC=C)=O)C1 Cc1sccc1CNC(=O)NCc1nnsc1C1CC1 N1(C(c2cccc(C(=O)NC)c2)=O)CC(C)(C)OCC1CNC(C1(F)CC1C)=O C1(NC(C(C2CC(F)(F)C2)OCC)=O)CC12CCN(C(C1CCC(=O)O1)=O)CC2 CN1C(=O)CC(NC(=O)C(C2(O)CCC2)NC(=O)CN2CCCNC2=O)C1=O c1(C(=O)NC2(CCNC(C(C)N(C(C)=O)C)=O)CCCC2)ncc(C)cc1F N1(C(CCCCCC#C)=O)CCC2CCC(C1)N2C(C1CCC2(CCC2)O1)=O C1(CC(=O)NCC2CCC(C(C)(C)C)C2)CCCC(NC(c2cnccn2)=O)C1 CCCC(C(=O)N1CCC(C(C)NC(=O)C(Cl)=CCl)CC1)NC(N)=O C(=O)(CCCC(C)=O)N(CC(N1CCC(CC=C)C1)=O)CC(C)C C1(NC(=O)CCCF)CC2CN(C(c3cncnc3C3CC3)=O)CC2C1 C1(C(=O)NCCCCNC(c2[nH]c(=N)sc2)=O)CCCCC12CC2(F)F C(=O)(CC1=NNC(=O)C1)NCC1C(NC(C2CCCN(CCC)C2)=O)C1 c1(OC)ccc2c(c1)CCCC2C(=O)NCCNC(c1ccc(C)nc1O)=O N1(C(C=C)=O)CCC(C2CC2)C1CNC(=O)C(O)CCSC C(CN=c1[nH]c(N(C2CC2C)C)nc2cc[nH]c12)N(CC)CC CC(O)(C(=O)N(CCNC(C1CNC(=O)C1)=O)C1CC1)C(F)(F)F c1(CC(C)(C)C(=O)NC(=O)NC(C)(C)C)cccnc1.CC1C(=O)NCC(C)N1C CC1CN(C(c2cc(Cl)ccn2)=O)CC(C)CN1C(c1ccc(S(C)(=O)=O)s1)=O O=C1NCCCC1n1cc(C2CCN2C(c2ccsc2-c2nn[nH]n2)=O)nn1 C(C)(CC(=O)NCC(=O)NCC(=O)NC(CO)C1(O)CC1)SC c1(OCC)ccc(C(=O)NCC(O)CNC(c2occc2C)=O)cc1OC C1(C(=O)NC(CCOC)CNC(c2cc(OC)n[nH]2)=O)CNC(=O)C(C)(C)C1 N1(C(c2cc(C(C)=O)c(C)o2)=O)CC(CNC(=O)C(C)(C)CO)CC12CCC2 c1(C(=O)NC(CNC(C2(COCC)CC2)=O)C)ccc(O)nn1 O=C(CC(F)(F)C(F)(F)Br)NCCNC(C1CC12CC2(F)F)=O Cc1cccc(C)c1CC(=O)NC(C)Cn1cc(-c2cc(F)cc(F)c2)nn1 C1(NC(C(C(C)C)F)=O)CCSC12CN(C(=O)C#CC(C)(C)C)C2 C1(NC(CSCC(=O)OC)=O)CCN(C(=O)C=CCOCC(F)(F)F)C12CCC2 N1(Cc2ccc(C)cc2)CC(NC(=O)C(C#N)Cc2ccccc2)C(C)(C)C1 C1(C(=O)NCCC(C)NC(=O)COc2cccc(Cl)c2)Cc2ccccc2S1 C(=O)(CC1OCc2ccccc21)NC(C(C)(C)C)CNC(c1ccnc(O)c1)=O C(N=c1ccnc(NC2CCCC(C(N)=O)C2)[nH]1)C1N(C(N)=O)CCC1 C12(COC)CN(C(=O)C=Cc3cocn3)C(CNC(=O)C(=O)Cc3cccs3)(C1)C2 Cc1cc(F)ccc1C(=O)NC1(CCCC(=O)NC23CC(C)(C2)C3)CCC1 C1(C(=O)NC(CC)C(=O)NC)CCN(C(C2CN3CCC2C3)=O)C1(C)C O=CN1CCCN(C(C2CSCCN2C(C2CCSC2)=O)=O)CC1 c1(C(=O)NC2C(NC(C3C(C(=O)OC)C3)=O)CCCC2)cccc2c1C(=O)NC2 c1(C(=O)OCCNC(=O)C(F)CC2CCC2)ccc2n[nH]cc2c1.C12CCN(C1)C2 c1(C(N(CC(C)O)CCNC(C2(C#C)CCC2)=O)=O)cc2c(C)ccc(C)c2[nH]1 N1(CC2CNC(=O)N2)CCc2ccc(Br)c(F)c2C1 C1(NC(=O)C=Cc2ccccc2)CN(C(c2cc(C3CC3)ccn2)=O)CC12CC2 Cc1ccc(C(=O)C(=O)NCC2(NC(=O)COc3cccc(Cl)c3)CCC2)cc1 N1(C(C(C)CS(C)(=O)=O)=O)CC2(CCCC2N=c2ccnc(Cl)[nH]2)C1 C(C(COC)CC(=O)NCCN(CCCCC1CCCCC1)CCO)OCC N1(C(C(C)(O)Cc2ccccc2)=O)CC2CC(C1)N(C(=O)CCn1ccnc1)C2 c1(OC)cc(C(N2CCCCC2Cc2cn(C3CCC3)nn2)=O)cc2ccoc12 CCCCC(C)CCC(=O)N1C2CCC1c1ncccc12 C1(C(=O)NC(CN(C(=O)C(c2cccnc2)O)CC)C)CC(C#N)C1 c1(NC2CC(CNC(c3c(C(N)=O)csc3)=O)C2)nc2ccccc2o1 O=C(C#CC1CCCCC1)N1CC(NC(C23CCC2CC3)=O)C(F)C1 C1(C2CCCC2)(C(=O)NCC2CN(C(C(C)=CC)=O)C(C)(C)C2)CCNC1=O C1(c2nnnn2C2CC2)(NCc2scc(C)c2)CCOC1C C#Cc1cc(F)c(C(N2CC3(CCN(C(=O)C(C)NC(N)=O)C3)C2)=O)cc1F c1(C(N2CC(O)(C(C(=O)N(C3CCC3C(C)(C)C)CC)F)C2)=O)ncc(C)[nH]1 C1(NC(=O)Cc2ccco2)CCCN(C(c2ccc3cccnn23)=O)CC1F C(CN=C(NCC1CC(C)OC(C)C1)N1CCN(Cc2ccccc2)CC1)OC N1(C(c2cc(CC)sn2)=O)CC(C(=O)N(C)CCC2CCCCC2)OC(C)C1 N1(C(C(C)SCCCC)=O)CCC2(C1)CN(C(=O)CCCCCSC)CC(C)O2 C1(NC(c2ccc(C)nc2)=O)CCc2nncn2C1.N12CCC(C1)COCC2=O C1(F)(CNC(C(F)=CC)=O)CCCN(C(=O)C(C(C)C)c2nonc2C)C1 C=CCCCCN=c1[nH]c(=N)[nH]c(=NCC2(OCCOC)CCC2)[nH]1 CC1CC(CNC(c2ncc(Cl)cc2F)=O)CCN1C(C12CSC(C1)C2)=O N1(C(CCN(C(CCC)C)C)=O)CCCC2(NC(=O)C(=O)NC(C)C)CC2C1 C1(CNC(c2c(C#C)c[nH]n2)=O)CN(C(=O)C(=O)NCCNC(C)=O)C2(CCC2)C1 N1(C(c2ncn(CC)n2)=O)CCOc2cccnc2C1 c1(C(=O)OC)ccc2c(c1)CN(C(=O)Nc1nsc3nn(C)cc13)CCO2 N#Cc1n[nH]cc1NC(c1cn(C2CCN(C(c3cnc(Cl)cn3)=O)C2)nn1)=O N1(C(C2C(OC(C)=O)C2)=O)CCCC1C1CCN(C(=O)CSCC(F)(F)F)C1 C1(C)(SC2(C(=O)NCCNC(CCC(=O)c3cn(C)nc3)=O)CC2)CCNC(=O)C1 C(=O)(C(C1=NOC2CC12)N(CCN(C)C)Cc1cnn(C)c1C)NC CC(=O)C(C)CC(C)C(=O)NC1CC(C(=O)NC2CCCCCC2C)C1(C)C c1(OC)ccc2c(OC)cc(NC(=O)N=c3cnc(C(F)(F)F)c[nH]3)nc2c1 C(=O)(C#CC1CCOC1)NC(CCNC(c1cnc(C(C)(C)C)o1)=O)(C)C C1(CNC(C=CC)=O)COC2(COCCN(C(=O)C(C)(C)F)C2)C1 Cc1ccc([N+](=O)[O-])cc1C(N1CC(NC(C2CSCC(=O)N2)=O)C(O)C1)=O c1(C(N2C(C(=O)NCc3ncc(C)s3)CCC2)=O)cc(C)c(O)c(C)c1 c1(C(N2CC(N(C(CC(C(C)C)C)=O)C)C(O)C2)=O)ccc(C#N)nc1O C1(=O)C(C)(C)CC(=O)NCCCN1C(C)C.n1(CC)cc(C(=O)OCC)nn1 C=CC1(CC(=O)N(CC(C)C)C(C)C)CN(C(C2CC(CC3CC3)C2)=O)C1 C(=O)(CCCCC(C)C)NCC1(C)N(c2nnc(C(=O)OC)s2)CCC1 C#Cc1cccc(CC(=O)NC(CNC(=O)C(CC(C)C)OC)CCOC)c1 c1(NC(C2N(C(c3cc(C)c(C)o3)=O)CCOC2)=O)cc(C)c(F)c(C)c1 N1(C(c2c(C)occ2)=O)CC2(C1)C(NC(=O)C(O)CC(C)C)CCS2(=O)=O c1(OC)cc(Br)c(CNCC2CCCCC23CCC3)c(F)c1F N1(C(C(C)(c2ccccc2)OC)=O)CC2CCCC(C1)N2C(=O)C(C)C#N C1(NC(=O)CN2CCSCC2)CN(C(=O)C=C2CCCCC2)C2CCCC12 CN1CCCC(F)(C(=O)NC(C2CCN(C(C3CS(=O)(=O)C3)=O)CC2)CO)C1 C1(OC)CN(C(C2CC2c2cnn(C)c2)=O)CC1NC(=O)CC1(N(C)C)COC1 N1(C(C2(OC)CCN(C(C(C)SCCCC)=O)C2)=O)CC2(CCC2(C)C)C1 C1(C(=O)NCC(C)N(C(c2cc(CCOC)on2)=O)C(C)C)CCN(C)CC1 Cc1ccc(C(N2CCC(CO)C(NC(C3(F)CC3)=O)C2)=O)c(C2CC2)n1 Cc1nc(NCC2(CO)CCN(C)C2)cc(N2CCSC(C(F)(F)F)C2)n1 C1(C(c2ccc(C(N3CC4CC4C3)=O)cc2)=O)CCn2ccnc2C1 C1(C#N)(C(=O)NCC(C)(C2CC2)NC(c2ccc(C(F)(F)F)[nH]2)=O)CC12CCC2 C(=O)(CCC(C)(C)[N+](=O)[O-])N1C(C)CC(CNC(=O)Cn2ccsc2=N)C1 c1(CC)cc(N2CC(NC(=O)CC3CCCC3)CC2C)ncn1 C(=O)(C1Cc2ccc(Cl)cc21)N(CCC(C(C)(C)C)NC(C1CC(F)(F)C1)=O)C N1(C(CCCOCCC)=O)CC=CC(NC(c2ncnn2C(C)C)=O)C1 C1(C(=O)NC(CC(C)NC(C(C)NC(C)=O)=O)C)CC2(C1)CS(=O)(=O)C2 Cn1ncc(C2CC2)c1C(=O)NCC(C1CC1)NC(c1cc(C(C)(F)F)n[nH]1)=O C(N=c1ccnc(NCc2ccc(CN3CCNC(=O)C3)cc2)[nH]1)C1(C)CSC1 N1(C(c2cccc(C#N)n2)=O)CC2CCC(C1)N2Cc1cccc2c1OCO2 c1(CCC(=O)N(CCNC(c2cn(CC)nn2)=O)C)ccc(F)nc1 C1(C(=O)NCCC(C)N(C(=O)CC2CC=CC2)C)CCn2nccc2C1 CC(C(=O)N1CCC(C(C)NC(c2cnoc2C2CCC2)=O)CC1)C(C)O C1(OC)CN(C(=O)CCc2cnc(C)s2)CCC1NC(c1cnc(O)o1)=O N1(C(CC2C(CC)C2)=O)CC(CO)C2(C1)CN(C(=O)CC1COCC(C)(C)O1)C2 CCC(C(=O)N1CC(CNC(=O)C=C(C)Cl)(OC)C1)SC N1(C(c2c(C)nc(CNC(=O)C(C)C(C)(C)C)o2)=O)CC(C)C(C)(CN(C)C)C1 CC1CCCn2cc(C(N3CCCCC3CCNC(=O)Cn3cccn3)=O)nc21 c1(C(=O)NC(CC)CNC(=O)Cn2cccnc2=O)sc(S(N)(=O)=O)cc1C N1(C(CNC=O)=O)CCC2(CCCCC2NC(c2cc(F)c3c(c2)CCC3)=O)C1 N1(C(c2oc(C(=O)OC(C)(C)C)cc2Br)C(=O)NC(C)C)CC2CCC(C1)N2C c1(C(=O)NCC(C)N(C)C(C2CC2c2nncn2C)=O)ccc2nc(O)oc2c1 C(=O)(CS(=O)(=O)Cc1cccs1)NC(C(C)(C)NC(C(C(C)C)SCC)=O)C C1(C(N2CCC(CCC(=O)NCCC34CC(CCO3)C4)CC2)=O)CCCN1C=O Cc1cc(Cl)c(CN(CCC(c2cccs2)NC(c2cncnc2)=O)C)c(Cl)c1 c1(NC(C(C)OC(=O)CCC(O)CN(C)C)=O)c[nH]c2ccccc12 C1(C)(CNC(C2ON=C(C)C2C)=O)CC(F)(F)CN1C(=O)CCn1cncn1 c1(OCC)cnc(C(N2CC=CC2CNC(=O)C(C)CC2CCCCC2)=O)cn1 C(C1CCCCC1)=C(C(=O)NC(CC)CNC(=O)COCC(C)C)C c1(C(=O)NCC(CCOC)NC(=O)C(F)=CC2CC2)c[nH]c2cc(OC)ccc12 C=CCC(C)(CC=C)NC(C1C(O)CCN1C(c1cccc(O)c1)=O)=O CCC(CC(=O)NC(C(N1CC(O)(CN(C)C)C1)=O)c1ccco1)SC c1(CC(=O)N(C(CNC(C2C(CCOC)C2)=O)C)C)sc2ccccc2c1C C1(NC(c2c(C)cc(CC)o2)=O)(COC)CCCN(C(c2ccsn2)=O)C1 N1(C(CC(CN(C)C)O)=O)CCC(CNC(=O)C2=CSCS2)C1(C)C n1(CC)nc(C)cc1CN=C(NC1CCN(CC2CC2)CC1)NC1CC1C.C(=O)OC Cc1ccnnc1C(N1CCCC1C1CCN(C(C2CCOCC2C)=O)C1)=O C(=O)(C1=CCN(C)C1)NCC1(C(=O)NCc2nc(C)c(C)s2)CC1 C1(CCOC)(C(=O)NCC(C)NC(C2CC2C2CCCO2)=O)SCCCS1 N1(C(C2(OC)CCSCC2)=O)CC(C2CN(C(C3CC4CCCCC4O3)=O)C2)C1 C(=O)(C(O)CN1CCCC1)NCC1CC(C(N(C)CCn2cncn2)=O)C1 c1(C(c2nnnn2C(C)(C)C)NCCOCC)cc(Cl)cc(Br)c1F C1(Nc2nc(C)c(C(C)(C)C)s2)CC2(C1)CC(NC(=O)CC(C)N1CCC1)C2 c1(OCC)cc(C(=O)NC2CCC(F)(CNC(=O)C3CC3)C2)c2ccccc2n1 c1(C(C(N2CC(NC(C3(C)CC3)=O)C(C)C2)=O)=O)ccc(Cl)cc1[N+](=O)[O-].CCCC c1(C(=O)Nc2c(Br)ccnc2Cl)cc(-c2cncs2)c2[nH]ccc2c1 c1(CC)nc(C(=O)NCC(C2CCCC2)NC(=O)COC2(C)CCCC2)cs1 c1(OC)ccc(C(=O)NC2CC(C)(NC(C3CCOC(C)(C)C3)=O)C2)nc1OC c1(C(=O)NCC2(C)N(C(C3C(C4C(C)C4)C3)=O)CCC2)ccc2[nH]ccc2n1 C(=O)(CCC(C)CN(C)C)N(C)CC1N(C(c2nc(OC)c(C)s2)=O)CCCC1 C(c1ccc(C)cc1)=C(C(=O)N(CCCNC(C1(COC)CC=CC1)=O)C)C c1(CC(=O)NC2(CNC(=O)CSCC(F)F)CCCC2)ccccc1Cl C1(CN(C(=O)CCSc2ccccn2)Cc2cccnc2)CCCC(C2CC2)O1 C(=O)(C1=CCC(NC(c2cn(C)nn2)=O)C1)N(CCC(=O)OC)C(C)C C1(CNC(Cc2c(Cl)cn(C)n2)=O)CCCN(C(=O)C(C)(C)n2cnnn2)CC1 C1(c2cn(C(CC(=O)OC)(C)C)nn2)CCN(C(C)=O)CC1(F)F.C1(=O)CCCN1 C(=O)(C#CC1(C)CCCO1)NCC(C(=O)N(CCCc1ccco1)C)OC C1(CNC(C2SCCS2)=O)CCCC1C(=O)NC1CCCC1O C1(C2CCN(C(=O)CN3CC4CC4C3)CC2)(NC(C2(S(C)(=O)=O)CCC2)=O)CC1 N1(C(C(C2CC2)SC)=O)CCC2(C)CN(C(=O)CCC3NC(=O)NC3=O)CC12 N1(CC(=O)NCCC(CNC(=O)C(O)Cn2cncn2)OC)C(=O)NC(C)(C)C1=O N1(CCNC(C2(C)CCCO2)=O)CCN(C(c2ccsc2)=O)CC12CCC2 Cc1cc(C(F)F)oc1C(=O)NC(C)(C)CNC(c1ccc(C2CC2)cn1)=O C(CO)(CC(F)(F)F)c1nnc(NC(C2CC3(C(C(=O)O)C3)C2)=O)o1 CN(OC1CCCC1)C(=O)CCOC1CN(C(=O)C(O)C2CC2)C1 C1(C(=O)NC23CC(NC(=O)CC4CC4)(C2)C3)CC2OC(=O)OC2C1 CCC(CC(F)F)C(=O)NCCC1CCN(c2nc(=N)cc(C(=O)O)[nH]2)C1 c1(C(c2n(C3(C)CC3)nnn2)NCC2CCSCC2)cccc(C(F)F)c1 c1(-c2cc(OCC)ncc2NCC(C)C)cn2cc(C(=O)NCCC#N)ccc2n1 O=C1CC(C(N2CCC(O)(CNC(C3(c4ncco4)CC3)=O)CC2)=O)NC(=O)N1 N1(C(CCc2cc(C)on2)=O)CC(NC(=O)Cc2sc(O)nc2O)C2CC2C1 C1(C(N2C(C3(C(=O)NCC(CO)OCC)CC3)CCC2)=O)CCCC(C)CC1 C1(CC)CCC(C)CN1C(=O)CC1N(C(=O)C2=CC(C)(C)C2)CCC1(C)C C1(C(=O)OC(C)(C)C)CC(O)CN1C(N1CCC(C(COC)C)C1)=O C1(NC(c2n(C=C)ncc2)=O)(CC)CCCN(C(c2n[nH]c(C)c2O)=O)C1 c1(OC)ccc(F)cc1C(=O)NC(C1CCCC1)CNC(C1CCC1F)=O N1(CC(=O)NCCN(C(=O)CC2CC2C(F)(F)F)CC)CCCCC1=O c1(C(=O)NC2CCCN(C(c3cc(C)no3)=O)C2C)cc2ncccc2cc1Cl c1(C(=O)NCC23C(CN(C(C(CC)(C)CO)=O)C2)C3)cc(N)c(C)cc1Cl C1(CC(C)C)CN(C(=O)C(C2CCCC2)NC(=O)OC(C)(C)C)CCO1 c1(C(=O)NCC2(O)CN(C(c3c(C)nsc3)=O)C2)cc2occ(Br)c2[nH]1 C1(NC(C(C(C)O)(F)F)=O)CC2(CCC(Nc3ncc(Br)cn3)CC2)C1 c1(C(=O)OCc2ncc(I)s2)ccc(S(=O)(=O)N2CCCCC2)cc1 C=CCCN=C(NCc1cccc(Cl)c1OC)NC1CCN(C(=O)OC)C1 c1(C(=O)NCCCCCNC(C2CC(C)OC2=O)=O)cnc2ccccc2c1 C1(NC(c2c(SC)scc2)=O)CCN(C(c2cc(F)n[nH]2)=O)C(C2CC2)C1 Cc1ccccc1CCC(N1CC=CC1CNC(=O)C(C)NC=O)=O Brc1cnc[nH]c1=NCc1ccc(C2CCOC2)cc1 c1(C(=O)NC2CC(NC(C(C)SCC)=O)C2)cc(F)cc(F)c1N N1(C(c2c[nH]c(=N)o2)=O)CCCC(C2CCCN(C(c3cnco3)=O)C2)C1 c1(C(N2CCC(C#N)(NC(C3CCCCC3N(C)C)=O)C2)=O)cc(O)c(O)c(Cl)c1 c1(C(=O)NC23CCC(CN(C(C4(F)CCC4)=O)C2)C3)ccc2c(c1)CCCCN2.C N1(C(C(CC)=CC)=O)CCC(NC(c2ccoc2Cl)=O)C1C(C)(C)C CC1CN(C(=O)C=Cc2cccnc2)C(C)CN1C(=O)CCC1(C)CC1 c1(C(N2CC3C(C(=O)OC)C3C2)C(=O)NC(C)C)nc2c(s1)CCCC2 Cc1c(CC(=O)NC2CC23CC(NC(=O)CCC2CCCO2)C3)cnn1C N1(C(CCCC)=O)CCN(C(=O)C(O)C(C)C)C(CO)C1 N1(C(CCC=C)=O)CCN(c2nc3cc(Br)cnc3s2)CC(C)(F)C1 CC1(C)CCC(C)(NC(C2CCCCN(C(c3cccc(F)c3O)=O)C2)=O)CC1 Cc1cccc(CCC(=O)N(CC(C)(C)CNC(C2CCC2F)=O)C)c1Br c1(-c2cccc(CN(C(C)CC#N)C)c2)ccc2cnccc2c1 N1(C(c2c(CC)ccc(F)c2)=O)CC2CN(C(=O)C(C3CCC3)OCC)CC2C1 CCCCCCC(C)CC(=O)N(C12CCCC1N(C(=O)C(C)(C)C)CC2)C c1(CN(C(CCc2ccc(C)s2)=O)CCC#N)c(C)cccc1C CC(C)CC(C)CC(=O)N1CC(NC(=O)C(CC(C)C)n2ccnc2)C(C)(C)C1 N1(CC)CCC(N=c2nc3sccc3c(NC3CCN(C)C(C)(C)C3)[nH]2)C(C)C1 CC1CCc2ncc(C(=O)NCC3CCC(NC(=O)CN(C)C)C3)n2C1 N1(C(C(COC)C)=O)CCCCC1CNC(c1noc(SC)c1C)=O CCC(N=c1cc(C)nc(NCC2=CCCC2)[nH]1)c1csc(C)n1 C1(CNC(=O)C(C2CC2)C2CC2)CC2(CC2)CN1C(c1ccc(C2CC2)o1)=O C1(C(CC)C)CCN(C(C2CCN(C(=O)CCCOC)C2)=O)CC1 c1(CC(=O)NC(C)C(C)NC(=O)C2=CCCCC2)ccc2[nH]ccc2c1 N#CC1(C(=O)NC2(CNC(c3c(Cl)n[nH]c3C3CC3)=O)CC2)CCOCC1 c1(C(=O)NC2CN(Cc3c(F)ccc(OC)c3F)C2)c(C)nc2ncccn12 Cc1cccc(F)c1CC(=O)NC1CC(C)(CNC(=O)C(C)C(C)C)C1 CN1CCC(C(=O)N(C)CC2(O)CCN(C(c3ccnc(Br)c3)=O)C2)CC1 C(=O)(C1=NN2CCCN=C2N1)N(CC(C)NC(C1CC2(C1)CC2F)=O)C C1(NC(c2cnc(C)o2)=O)CCN(C(=O)Cn2cnc(C#N)n2)C(C)C1 N(C(=NCCC(C(F)(F)F)N(C1CC1)CCOC)NC1CCCC1(F)F)C(C=C)C c1(C(=O)NCCSc2ccc(C(N3CCNCC3)=O)cc2)cc(Cl)c(F)c(Cl)c1 C12CCC3CC1CN3C2=O.C1(Br)(C(=O)NC(=O)C(Cl)(Cl)Cl)CCCCC1 N1(C(c2cn(CC)nn2)=O)CCC(NC(=O)C(c2cccc(C)c2)C)C12CC2 c1(CNC(c2nc(C(=O)N(C3(CC)CCC3)C3CC3)co2)=O)ccc(Cl)cn1 C(=O)(CS(=O)(=O)CC(=O)NCC1(O)CCCN(C(=O)Cc2ncoc2C)C1)OC C1(C(=O)NCC2N(C(c3c(C#N)cn[nH]3)=O)CC(F)(F)C2)CCn2nnnc2C1 C12(NC(C(C)(C)SC)=O)CC1CN(C(c1nc(C)sc1C)=O)C2 c1(C(=O)NCCC(C(CC)(C)C)C)cnn2cc(C#N)cnc12 C(=O)(C#CC1(C)CCCO1)NC(C1OCCN(C(C(C(C)C)C)=O)C1)C C1(O)(C(N2CCC(N(C(=O)C(C)(C)NS(C)(=O)=O)C)C2)=O)CN2CCC1CC2 C12(NC(c3cc(CCCCC)[nH]n3)=O)CCCN(C(C3CCC=CO3)=O)CC1C2 Cc1cccc(C(=O)NCCN(C(C23CC(C2)C(C(=O)O)CO3)=O)C(C)C)c1F C1(C(=O)N)C2C3CC4C1C1C2CC3C41.N1CCCC(NC(c2[nH]n(C)c(=O)n2)=O)C1 c1(C(N2C(CN)CC(OC)C2)=O)ccc(C(=O)ON2CCC(C)CC2)cc1O C(c1ccc(C(=O)N(C)C)cc1)=CC(=O)NCCN(C(C(CC=CC)C)=O)CC c1(NCC(=O)NCCC(C)NC(=O)C(c2ccnn2C)O)cc(O)nc(CO)n1 n1(CC(=O)NC2CCC2c2cncc(Br)c2)cc(F)ccc1=O c1(ONC(=O)CC2C3CN(C(C4CCCSC4)=O)CC23)ccc([N+](=O)[O-])[nH]1 c1(NC(COc2c(OCC)cc(Cl)cc2)=O)ncc2n1CCCC2 C12(C(N3CC(CC)N(C(=O)C=Cc4ccoc4)CC3)=O)CC(C)(C1)OC21CCC1 c1(OC)c(NCC(=O)NC2CCCC2N=[N+]=[N-])ccc2[nH]ccc12 C1(CCCCC)CCC(C(=O)NCCC(C(C)C)NC(c2cc(C)[nH]n2)=O)CC1 C1(CSCCOC)CCCCC1NC(C1CCN1C(=O)OC(C)(C)C)=O CC1CCCC(C(=O)NCC2CN(C(c3cc(Cl)ns3)=O)C2)CC1 Cc1cc([N+](=O)[O-])cc(C(N2CCC3(NC(=O)CCC4CC4)CCCC23)=O)n1 c1(CCC(=O)N(CC(CC)NC(=O)C(O)C(C)C)CC)nc2ccccc2s1 CCCCCC(CC)C(=O)NC(C)CN(C(c1ncc(CC)cn1)=O)CC C(=O)(CC1=CCN(C(=O)CC(C)SC)CC1)NCc1cnc(CC)[nH]1 CCCC(C)(C)CC(=O)NCC1CC(O)(CNC(c2ccc(SC)s2)=O)C1 C1(NC(C2CC(C)(C)O2)=O)C2CN(C(=O)Cc3cncnc3)CC12 CC(=O)CCCC(=O)NC(c1cn(C)nn1)C(=O)N(C1CN(C(C)C)C1)C c1(C(=O)NCCOCCCN(C(c2cnc(CC)[nH]2)=O)C)cn(C)c(O)n1 C(=O)(C(C(C)NC(=O)CC1(C)CCOC1)C(C)C)N(C)Cc1cnc(C)s1 c1(OC)cccc(Cl)c1C(F)(F)F.C(C(C(C)C)NC(C1(C(=O)N)CC1)=O)NC=O C1(O)(CC(C(=O)NCC2C(C)OCC2)NC(=O)COCC2CC2)CCCCC1 CC#CCC(C(=O)NCCN1CC=CCC1)NC(c1cc(OC)cnn1)=O c1(C(=O)NCC(CNC(CCC(=C)Cl)=O)(C)F)cc(C)c(F)cc1F N=c1[nH]c(NCCc2cc(Cl)ccc2Br)cc(=NCC2CC2F)[nH]1 N1(C(c2cnc(N(C)C)o2)=O)CC2CN(C(c3csnn3)=O)CC(C1)O2 N1(CCN2CCCC(F)(F)CC2)CCC2(CC1)CC2(C)NS(C)(=O)=O CC1CC(NC(=O)CC2COCC2O)CCN1C(c1ccn(C(F)F)n1)=O C1(NC(CNC(C(C)(C)C)=O)=O)COCCC1NC(=O)CC1(C(F)F)CC1 c1(C(=O)NCC2(CNC(C=Cc3c(C)cco3)=O)CC2)n[nH]c2ccc(F)cc12 Cc1cc(C(N2CCN(C(=O)CCc3ccncc3)C(CF)C2)=O)c(C)nc1C C1(CNC(CC(C)(C)C2CCCCC2)=O)CC2(CC2)CN1C(C1CCNC1=O)=O c1(NC(N(C(C)Cc2ccccc2)CC)=O)cncc(Cl)c1 C12(C(=O)NCC3C(NC(CCCN(C)C)=O)CCC3)CCC(CC1(F)F)C2 C1(C(C)C)CN(C(C2C3CCC(C3)C2NC(=O)C(F)C(F)(F)F)=O)CCCO1 C1(C(=O)NCCN(C(Cc2c(C)n[nH]c2)=O)C)CCC(C)(C)CC1 c1(-c2cn(CC(=O)NC(c3n(C)ccn3)C(F)(F)F)nn2)cccc(C#N)c1 Cc1sc2cncn2c1C(=O)NCC(n1cc(CCCC(C)O)nn1)C C1(NC(c2c(C)cc(CC)o2)=O)CS(=O)(=O)CC1NC(C12CC(C)(C1)C2)=O N1(C(Cc2c(C)nc[nH]2)=O)CCC2(CCC2)C(NC(=O)CC2CCCC(=O)N2)C1 C1(CNC(c2c(OC)scc2)=O)CCN(C(=O)CN2CCOC2=O)CC1C n1(CC(N2CC(C)N(C(c3cnc(S)nc3)=O)CC2)=O)ncc2ccc(F)cc12 C1(NC(CCCC=C)=O)CCN(C(=O)C(C2CCOCC2)F)CC(C)(C)C1 CC(C)CC(C(=O)NC1CC1)ONC(=O)CC1CCC(C)CC1.C(CCC(=O)O)SCC C=CC(CCC)CC(=O)NCC1CCCCN1C(c1cn(CC)nc1C)=O C1(C(N(CCCNC(C2CC(O)C2)=O)C(C)C)=O)CCCNS1(=O)=O c1(OC)cnc(Br)cc1C(N1CCN(C(=O)C(O)C2CC2)C(C2CC2)C1)=O c1(C(=O)NCC2CCCN(C(C(C)N(C)C)=O)C2)cnc2cc(Br)ccn12 c1(OC)ccc(C(=O)NC2COCCC2NC(c2cn(C3CC3)nn2)=O)nn1 C1(NC(C2CCN(C(C)=O)CC2)=O)C(C)CCN(C(=O)CSC2CC2)C1C C12(CNC(c3n(C(C)(C)C)ccc3)=O)CCCC1N(C(C1CC(=O)N1)=O)CCC2 Cc1nnc2n1CCCC2C(=O)N(C)CCN(C)C(C12CC3CC1C2C3O)=O N1(C(C(C)(C)OC(C)=O)=O)CC2(C1)SCCC2NC(c1cnn2c1CCC2)=O N1(CCCNC(CCC)=O)CCCCCC1.N12CCC(C1)CCNC(=O)C2C c1(OC)cc(OC)c(CNC(N2CCCC2CS(C)(=O)=O)=O)cc1OC O=S(=O)(c1ccc(NC(C2CCCC2)CO)c(F)c1)NC(CO)C1CCC1 c1(C(N(CCC(=O)NC)C)=O)cc2ccc(-c3ccc(C(C)OC)cc3)cn2n1 CC(C(=O)OC)C(=O)N1CC(CC(C)(C)CC(C)(C)C)C1.C1(C)(C(=O)N)CSC1 C1(C(=O)NCC(=O)N(C)C)CC(C)(C)CCN1C(=O)Cc1ccon1 C#Cc1ccc(CC(=O)NC(C)(C)C(C)NC(=O)Cc2c[nH]ccc2=O)c(F)c1 C1(CNC(c2cncc(C)n2)=O)CN(C(=O)C(C)C(C)O)CCC1C C(=O)(C(Cc1cnc[nH]1)OC(=O)OC(C)(C)C)NC(CC)C1CC1 N1(C(CC)C(=O)NCC(=O)NCC(C)C)CCc2ccccc2C1 N1(C(c2cnnn2C2CC2)=O)CC2(C(N3CCOCC(O)C3)=O)CC1CO2 C1(C(=O)NC2CN(C(C3(Br)CC3)=O)CC2C(F)F)CC2C=CCC(C1)C2 c1(CC(=O)NC)ccc(Cl)c(C(N2CC(CNC(=O)CCC(C)C)CC2C)=O)c1 c1(OC)ccc([N+](=O)[O-])c(N)c1.c1(C)cncn(C)c1=O.C12CN(C1)C2=O c1(C(=O)NCC(CC)(C)NC(C2(C#N)CCOCC2)=O)cccc(OC)c1F c1(C(C)C)cc(C(N2CCCC(Oc3ncc(Br)cn3)C2)=O)nc2ncnn12 C12(CNC(c3n(CC)nc(C)c3)=O)CCC(C1)N(C(=O)C(C)CCCOC)C2 c1(OC)cc(C(N2CCC(C(C)NC(=O)Cc3cocn3)CC2)=O)c(N)c(C)c1 n1(CC)nnc2c(NCC(C)(C)NC(=O)Cc3cc(C)no3)ncnc12 C(=O)(CC(C)(C)CCOC)N1CCC(C(=O)NC(CC)(C)CC)OCC1 Cc1nnc2n1CC(C(N)=O)N(CCc1cccc3c1OCCO3)C2 CC(C)C(CC(=O)NCC1(CNC(=O)C(O)C2CC2)CCC1)NC(=O)OC(C)(C)C N1(C(C2CCN(C(C)=O)C2)=O)CC2CN(C(=O)C=CC3CC3)CC2C(F)(F)C1 C1(C(N2C(CNC(C3C(C)(C)CCO3)=O)CC(O)C2)=O)CCC2CC1CO2 c1(CN2CCN(C3CCN(C(C4(C(N)=O)CC4)=O)C3)CC2)ccc(F)cn1 C1(C)(C(N2CCCC(c3cncn3C)C2)C(=O)NCC)COC(=O)C1 Clc1ccnc(CCSC2CCC23CNC3)n1 N1(c2nnc(C(=O)OCC)s2)CCC(C2CC2)(CNC(=O)CCc2cncnc2)C1 C1(C(=O)NCC(COCC)C)C=CCN(C(C2CC=CC2)=O)C1 N1(C(C=CCN(C(C)C)C)=O)CCC(C)(CNC(C2(CC3CC3)CCC2)=O)CC1 C1(C(N2CC(O)(CC=C)C2)=O)CN(C)CCN1C(=O)CCCOCC N1(C(c2ccc(O)cc2)=O)CCC(C(=O)Nc2cc(C3CC3)no2)(CO)C1 N1(C(CC(CCC)O)=O)CCN(C(=O)C(C)NC(=O)NCC)CCC1C c1(COC(C)=O)ccc(C(C2C(CC)CCC2)=O)cc1.C12(CC1)C(=O)NC2 c1(OC)ccc(NC(C)=O)cc1S(=O)(=O)Oc1ccc2c(c1)N(C)CCO2 C#CC12CCC(C(N3CCC(C)(CNC(C4(COC)CCC4)=O)C3)=O)(CC1)CC2 C(Cc1cc[nH]n1)(C(=O)NCCCCCNC(C1C=CCC1)=O)NC(=O)OC C=CCCCC(C(=O)N1CC(NC(c2cn(C)nc2CC)=O)C1)c1ccccc1 C=C=CCCC(=O)N(C(C)C(=O)NCC(=O)NC(C)CC)CCC c1(OC)cnc(C(=O)NC(Cc2cnc[nH]2)C(=O)N2CCC(C(N)=O)C2)cn1 C1(C)(C(=O)NCC(C)CNC(=O)CC2COCCO2)CC2CCC(C1)S2(=O)=O c1(CC)cc(C(N2CC3CC3(NC(=O)C(N3CCCC(O)C3)C)C2)=O)nn1C CCCCC(CC)NC(C1CC(N(C)C(c2csc(CC)n2)=O)C1)=O C(C(N=[N+]=[N-])C(=O)NCCN(C(=O)C(C)(CC)CO)CC1CC1)OCC c1(C(=O)NCC2C(C)CCN(C(=O)CSCC(N)=O)C2)cccc2ccn(C)c12 C1(CC(=O)NC2CCCN(C(c3nc(C)sc3C)=O)CC2)CCCC2(CCC2)O1 c1(C(=O)NC(CNC(c2cnsc2)=O)CO)csnc1Br C(CCCC(=O)N1CCCCC1CCCNC(=O)CN(CC(C)C#N)C)OC c1(C(=O)NCC2N(C(C3=NOC(C(C)(C)C)C3)=O)CC2)cc2cc(O)ccc2[nH]1 N1(Cc2ccc(C)s2)CCNCc2cccc(Cl)c21 Cc1c(Cl)ccnc1C(N1CCC(CF)(NC(c2ccnc(S)c2)=O)C1)=O C1(CN(C(C2(C)CC2)C)C)NC(=O)CC1(C)C C1(NC(c2c(CC)occ2)=O)CS(=O)(=O)CC1NC(=O)C=Cc1ccc(Cl)s1 Cc1cccc(C(=O)NC2(CC(=O)NCC3(C(C)C)CC3)CC2)c1N CCC(CC)(CO)C(=O)NC1CC(CNC(c2nc(C)sc2C)=O)C1 c1(C=O)ccc(N)c(O)c1.C1(NCC2(C)CC2)CC2CNC1C2 c1(CC(=O)NC2CCCN(C(C3(C#N)CC=CC3)=O)CC2)cc2ccccc2s1 c1(OCC)ccc(C(=O)NC(CNC(C2CC2F)=O)C(C)C)c(F)c1F C1(C(=O)NCCCN(C)C)(NC(CCCCSC)=O)CC2CCC1C2 c1(C(=O)NCCC2(NC(c3sccc3CO)=O)CC2)nc(C(F)(F)F)n[nH]1 c1(CC(CN(C(=O)C=CC2CCCO2)C)NC(c2csc(Cl)n2)=O)ccccc1 n1(CC)ncc2c(N3CCC(F)(CNC(C4CC5CCC4O5)=O)CC3)ncnc12 Cc1ccc2[nH]nc(C(=O)N(C3CCN(C(=O)C(F)(F)C4CC4)CC3C)C)c2c1 c1(C(C)(C)NC(=O)NCc2ccc(C)cc2)ccc2cc(F)ccc2c1 N1(C(C=CCC2(NC(=O)C(C3CC3)C3CC3)CCC2)=O)CC2C=CC2C1 c1(NC(=O)Cc2ccccc2NC(C2(O)CCCC2)=O)nc2ccccn2n1 c1(C(N(C2CN(C(C3CC(C)(C)CN3C)=O)C2)C)=O)cc2c(cc1O)CCCC2 C(=O)(CCC(CF)CF)N1CCC(CC#C)(C(N2CC(n3ccnn3)C2)=O)C1 N1(C(C2(C)CC(C)(C)C2)=O)CCCC(F)(CNC(c2cc(Cl)no2)=O)C1 c1(C(N2CCC(N(C)C(c3cc4c[nH]nc4s3)=O)C2)=O)ccc([N+](=O)[O-])cc1O Cc1ccc(F)cc1S(=O)(=O)NC1CC(F)CN(c2ncc3ccccc3n2)C1 Cc1cnc(C2(NC(=O)CC3CCCN3C(=O)CCOC3CCCC3)CC2)[nH]1 c1(CN2CC(CNC(=O)Cn3cc(Cl)cn3)OCCC2)cccc2c1CCOC2 NCC(C(=O)NCCC1CC1(Cl)Cl)c1ccccc1 C(CCC(O)C(=O)NCc1conc1C1CC1)NC(C(C)SC(C)C)=O C1(CC=C)(C(N2CCCCC2COC)=O)CCCN1C(c1cnsc1)=O c1(CC)cnc(Cl)[nH]c1=NCC1(CC(=O)NC2CC(C(=O)NC)C23CCC3)CC1 C(=O)(C1CCc2ccccc21)NCC1C(CC(=O)OCCCCC2CC2)C1 N1(C(CSCC#C)=O)CC2(CNC(c3ccc(NC(N)=O)cc3)=O)CCC1CC2 c1(C(=O)NC(CCNC(C2C(CC)N(C)CC2)=O)C)occ2c1CCCC2 N1(c2nccc(N3CCC(O)CC3)n2)CC2CCCC(C1)C2O Cc1cc(F)ccc1-n1ccc(NC(=O)C(=O)NC2CSCC2C)n1 c1(NC(C2C(CNC(C3(C(N)=O)CCC3)=O)CCC2)=O)cccc2c1CCC2 Cc1nnc2n1CC(C(=O)NC1CC(F)CN(C(=O)Cc3cncs3)C1)N(C)C2 c1(C(=O)NC2CCCC2NC(c2ccc(Br)nc2)=O)ccc(Cl)c(F)c1 C1(C(N2CCC(CN(C)C(c3cc[nH]c(=N)n3)=O)C2)=O)CC2(CCO1)CC2 C(C1CCCCCC1)=CC(=O)NC1CC1CNC(C1COC2(CCC2)C1)=O CCCCC(C(=O)O)n1nnnc1N1CCCC1C(C)(C)CO N1(C(C(C)(C)C2CN(C(=O)CC#N)C2)=O)CCC(C2(O)CC2)CC1.C1C2CC12CC NC1(C2CCN(C(C3(O)CCCOC3)=O)CC2)CC1 N1(CC)CCC(NC(C2(C)CCN(Cc3nnc4n3CCC4)C2)=O)C(C)C1 C(C(O)CC(=O)NC(C1CSC1)C)NC(C(C)SC(C)C)=O c1(NC(=O)NC2CC(n3cc(-c4ncsc4Cl)nn3)C2)ccc(C2CCC2)cc1 N1(C(C(c2cccnc2)C)=O)CC2(NC(=O)COc3cccc(F)n3)CC1C2 C(c1ccc(Cl)cc1F)=CC(=O)NCC1CN(C(CCSCCC)=O)C2C1C2 Cc1cc(C(N2CCN(CC3(C4CCC4)CCC3)CC2)=O)c(C)n1C c1(C(=O)NC(CC)CNC(c2csc(O)n2)=O)cc(C2CCCC2)n(C)n1 O=C1CCC(CC(=O)NCC2(C(=O)NOCCO)CC(=O)C2)C1 C(=O)(CC(F)(F)F)N(CCCNC(C)=O)CNC(C1CCCN1C(=O)C(C)C)=O C1(NC(CC2(COC)CC2)=O)(CNC(=O)CCc2cc(Cl)cs2)CCCCC1C S(=O)(=O)(c1ccccc1F)NC1CN(C(=O)CSc2ccccn2)C1 c1(OC)cscc1C(=O)NCCC1CC1C(=O)NC(c1cnn(C)c1)CO C12CN(CC(C)(C)C1)CC1CCCC21.c1(C2(C)CC2)c(C2OCCO2)cnn1C n1(CCCC(=O)NC(c2nnc3n2CCC3)C)cc(C#CCN(C)C)nn1 c1(C(=O)CN2C3C(C(N4CCC(OC)C4)=O)C(C3)C2)cccc2ccccc12 c1(CC)ccccc1-n1cc(COCC2CCCN(C(C3CCOC3)=O)C2)nn1 C(c1cnccn1)=CC(N1CC(CCCCNC(C(C)(C)c2ccccn2)=O)C1)=O C1(NC(CCc2onc(C)n2)=O)CCC(C(N2CC3CC2CS3)=O)CC1 c1(CC)conc1C(=O)NC1CC(C(=O)N(C)CCOC(F)F)C1 C(=O)(C(C1CC(OCC)C1)NC1(Cl)CC1)NCC c1(C(N(C2CCN(C(C3C(C=C)C3)=O)C2)CCO)=O)cc(C)c2sccc2c1 C1(CCC)(NC(=O)CCN(C)CCO)CCCN(C(=O)CN(C)C)C1 c1(C(=O)NCC(CC)N(C)C(C2C3CC(=O)CC23)=O)cc(C)nc(C)c1 C1(C(=O)NC(C2(CNC(CC(C)OC)=O)CCN(C)C2)c2ccccc2)CCC(F)(F)C1 c1(C(=O)NC(CCNC(c2sc(C)c(O)n2)=O)C)c2c(nn1C)CCCC2 C1(NC(c2nc(C)nc(O)c2)=O)CCC2(CC1)CN(C(c1ccncc1N)=O)C2 C12(C(N3CC4(N(C(C5C(C)(C(C)C)C5)=O)CC4)C3)=O)CCC(N=[N+]=[N-])C1C2 c1(C(N2CCC(NC(c3ccc(C)nc3)=O)C2C2CC2)=O)cc(F)c(C)cc1Cl c1(CNC(CCSc2n(C)nnn2)=O)nc2ccccc2n1CC(F)(F)F N1(C(C2C(CC)C2)=O)CCC(CCNC(C2CSCCS2)=O)C1 c1(CCC(=O)NC2CC(NC(CC(C)(C)O)=O)C23CCC3)cnc2ncccn12 C1(C(=O)OC(c2cc(Cl)cc(Br)c2)CC)CC2CCC(C1)N2CC(C)C C1(CNC(Cc2scc(C)c2)=O)(NC(=O)C(Cl)=CCl)CC2CCC1C2 N1(CC(=O)N(C(CCNC(Cc2cc(OC)no2)=O)C)C)CCCNS1(=O)=O C1(C(C(=O)NCCCCCC)(C)C)CCCN(C(=O)C=Cc2cnccn2)C1 C=C(C)CC(C(=O)NC1CCN(C(C2CC(C)=NO2)=O)CC1F)OC N1(C(=O)OC(C)(C)C)CCC(C2CCCC2)(C(=O)NCCC2CC(O)CN2)C1 N1(C(C(C=C)O)=O)CC2(C1)CN(C(=O)C(F)CCCC)CCO2 N1(C(c2cc(C)nc(C)c2)=O)CCC(C(=O)NC2CCC2(C)C)=C(F)C1 c1(C(=O)OC)cc(Cl)c(N2CCC(C(C)NC(c3ccc(C(N)=O)[nH]3)=O)C2)nc1C N1(C(CNS(CC)(=O)=O)=O)C2CCC1(CNC(c1ccc(CCO)cc1)=O)CC2 C[S+](C)CCC(O)C(=O)N1CC(CCNC(=O)CCn2cccn2)C1 CC1=NOC(C)(C(=O)N(C)CC2CN(C(=O)Cc3sc(S)nc3C)CCO2)C1 N1(C(=O)Cn2cnc(C(F)(F)F)c2)CCC2(CC1)CN(C(C1CC3CCC1O3)=O)C2 C1(NC(=O)CCC2CCCCO2)CC2CC1CN(C(=O)CC(Cl)Cl)C2 CC(=O)CCCC(=O)NCC(CO)NC(=O)CC1CSCCS1 c1(NCc2n(C)cnc2)ccc(S(=O)(=O)NCC2(CO)CC23CCC3)c(Br)c1 c1(C(=O)NCC(CNC(c2cn3ccsc3n2)=O)OC)cnc2ccncc2c1 c1(-c2scc(C(=O)NCC3C(NC(Cc4ncc(C)o4)=O)C3)n2)cccc(Cl)c1 c1(C(=O)OC)nccnc1CN(c1nocc1C(=O)OC)CCC(N)=O C(=O)(CCCCC(C)CC)N1CC(C(N(C(C=C)C2CC2)C)=O)C(C)(C)CC1 Cc1c(C(N2CCC(C)C(NC(=O)CSC(C)C)C2)=O)oc2ccc(F)cc12 c1(C(c2n(CCCOC)nnn2)NCC2CC(F)(F)C2)nc(Br)c2ccccn12 O=C(C1CCCn2cnnc21)N1CCN(C(c2onc3ccccc23)=O)CC1 N1(C(C(C)=C(CC)C)=O)CCC2CCC(C1)N2C(C1CCC(=C2CCC2)CC1)=O c1(CC(=O)NCC2CC(CCNC(=O)C3=CCCCC3)C2)cc(F)cc(Cl)c1 CC1(C#CC(=O)N2CCCC3(NC(c4cc(C(N)=O)c[nH]4)=O)CC3C2)CCCO1 c1(OC)ccccc1Cn1nc(-c2ccnc(Cl)c2)nc1C(CC)C1CC1 c1(NS(N)(=O)=O)cccc(C(=O)NC2CCCN(C(c3cnccn3)=O)C2)n1 c1(NC(COC)=O)ccc(C(N2CCN(c3ccnc(C4CC4)n3)CC2)=O)cn1 C(c1cccc(C#N)c1)=CC(C(=O)OCC)=O C(=O)(C#CC(C)(C)O)NCC(c1ccc(C)nc1)O.C1CCC2(CC2)C(=O)N1 C(c1ccnn1C)=CC(=O)NCCN(C(C1COCCN1)=O)CC C(CCN=c1[nH]c(=NCC(F)(F)Cl)c2[nH]ccc2[nH]1)ONC(=O)OC(C)(C)C c1(SC)ncc([N+](=O)[O-])c(=NCC2CN(C(=O)C(C)C(C)(F)F)CC2(C)C)[nH]1 C1(C(C)C(=O)N(C)C(c2cccs2)C)CCN(C(c2ccsc2)=O)C1 c1(OC)cc(O)c(C(=O)NC2CN(CC34CCC(CC3)OC4)C2)cc1OC N1(C(C=C(Cl)C=C)=O)CC2CCC1C1CN(C(C3(SCCC)CCC3)=O)CC21.C(C=C)=CC C1(NC(C(CCC2CC2)NC(C2CC(OC)C2)=O)=O)CCC12CCCC2 C1(N(C(CC(CC)C)=O)c2cnccn2)CCC12CCNCC2 C1(C(N(CC(O)CNC(=O)COCC(C)(C)C)C)=O)CCCCN1C(=O)C1CC1 C1(NC(C(COC)C)=O)CN(C(c2ccnc(C(N)=O)c2)=O)CC1C1CC1 c1(C(N2CC3(C(C(N4CCC(CC)C4)=O)C3)C2)=O)cc(C(F)(F)F)ccc1C C1(NC(c2cccc(Cl)n2)=O)CCCC12CN(C(c1sccc1Cl)=O)C2 c1(C(N2CCC(C(=O)NC(c3nnc(C)s3)C)C2)=O)ncn2ccccc12 c1(N2C(C)CC(NC(C3(c4ccccc4)CCC3)=O)C2)nc2cc(F)ccc2o1 C1(CNC(C2CCOC2)=O)CCCN1C(c1cc(C2CC2)no1)=O C12(CNC(C3C(C(C)NC(C4(C=C)CC4)=O)C3)=O)CCC(CC1)C2 c1(C(N2C(C)CCC(CNC(=O)CCC(N)=O)C2)=O)cc2c(nn1)CCCO2 N1(C(CCNC(=O)NC)=O)CCC(NC(c2cc(Cl)cc(Cl)n2)=O)CC1C c1(OCC)nccc(C(=O)NCC2CC2CNC(c2nn(C)c(C)c2Cl)=O)c1F Cc1nc(C(N2CCC(C)(NC(C34COCC3C4)=O)C2)=O)c(C)o1 N1(C(C2C(C)C2c2ccccc2)=O)CCN(C(c2nncn2C)=O)CC(C)(F)C1 C1(C(=O)NCC(C2(O)CN(C(C3C(C)(C)C3(F)F)=O)C2)(C)C)CCCC1(F)F n1(CC(=O)NCC23CC2CN(C(C2CC4(C2)CC4F)=O)C3)cc2ccccc2n1 C1(C(=O)NC2C3CN(C(c4cc(Cl)cnn4)=O)CC32)CCCC12CCOCC2 N1(C(=O)NC(CCC(C)C)C)CCC2NCCC2C1 N1(C(CN(c2ccncc2)C)=O)CC2(CCN(C(c3cnco3)=O)CC2)C1 c1(COCCC(=O)NCC(C)(C2CC2)NC(CCCC2C(C)C2)=O)ccccc1F C1(C(=O)NCc2ccc(C(C)NC(CC(C)O)=O)cc2)CC(S(C)(=O)=O)C1 C1(C(=O)NC(CC)CNC(c2cc(C)cc(F)c2)=O)CCc2cc(C)ccc2O1 c1(-c2cc(C(N(CCCNC(=O)CC3CC34CC4)C)=O)on2)ccccc1Cl CCCCC(CC)C(=O)NCCCCN(C)C(c1ccnn1C(C)C)=O C(=O)(C(F)C1=CCCCC1)NCC(C(N1CCC(=CCC)C1)=O)N(C)C CC(N=c1nc(NC2CC(N3CCC3)C2)c2ncccc2[nH]1)c1cccc(O)n1 c1(C(=O)Nc2scc(C(=O)Nc3c(C)ccc(OC)c3)n2)cc(C)c(C)cc1C N1(C(CC(CC)C)=O)CCC(NC(c2ccc(OC)s2)=O)C(CC)C1 C1(C2CCN(C(=O)C(O)c3ccsc3)C2)(NC(c2cc3c(s2)CCCC3)=O)CC1 c1(C(N2CCC(N(C(c3cnn(C)c3SC)=O)CC)C2)=O)cc(C)nc2ncnn12 C(=O)(C(C)(C)CC(=O)NC(CCC1CC1)C(=O)N1CCC(SC)CC1)OCC c1(C(N2CC(COC)N(C(=O)C=C3CCC3)CC2)=O)nn(C)c2c1CCC2 C#CC(C1CCC1)N(C(=O)CN(C)C(C1CC1C(F)F)=O)CC(C)C c1(CC)nc[nH]c(=NCCNC(=O)COc2cc(Cl)ccc2C)c1F C=CC(CCC)CC(=O)N1CC(OCC(N2CCCC(CC)CC2)=O)C1 N1(C(c2cnc(C(C)OC)s2)=O)CCC(NC(=O)CC2(C)CC(F)(F)C2)C(F)C1 c1(C(=O)NC2(CO)CN(C(CC3(C=C)CC3)=O)C2)cccc(C)c1C(F)(F)F c1(C(=O)OC)sc(C(=O)NC(C)CNC(c2ccc(C(F)F)cn2)=O)cc1N N1(C(C2CC=C(C)CC2)=O)CCC2CN(C(c3cc4occc4s3)=O)CC2CC1 Cc1nnc(CCNC(=O)CC2(NC(=O)CN3CCCC3)CCC2)n1C c1(C(=O)O)ccnc(-c2cn(CC3CN(c4ccccc4)CCO3)nn2)n1 c1(C(=O)NC(C)C(=O)NCCC2CCCO2)c[nH]c2ccccc12 c1(-c2nc(CN)on2)ccccc1C(=O)NCc1cncn1C1CC1 N1(C(c2scc(OC)c2)=O)CCC2(CC1)CC2NC(C12CCCC1C2(F)F)=O C1(CC(=O)N(C(C)CCNC(=O)CC2CCC3CC23)C)CCCC(=O)N1 C1(CC)(NC(c2nn(C)cc2C)=O)CCN(C(=O)Cc2nocc2C)CC1 C(=O)(C(C)C(O)C(C)C)N(CCCCCCNC(c1cc(OC)ncc1F)=O)C C1(Cn2c(C(COC)NCc3nnn(C)n3)nnn2)CCC2CC2C1 N1(C(C2COCC(C)(C)O2)=O)CCC2CN(C(c3cncc(N)c3)=O)C2C1 C12(C(N3CCN(CC#CC)CC3)=O)CC(CO1)N(C(C1CNC(=O)N1)=O)C2 C1(CCNC(CC23CC(C)(OC2)C3)=O)CCC(=O)NC1=O N1(C(c2c(OC)cccn2)=O)CCCC(C)C1CNC(=O)CC(Cl)Cl N1(C(CN(C2CC2)CC)=O)CC(CNC(c2sc(CC3CC3)nc2C)=O)C(C)C1 C=CC1OCCC1C(=O)NCc1ccccc1CN(C(=O)Cc1cc(C)on1)C N1(C(CC(CC=C)NC(c2ccn(C)c2C)=O)=O)CCc2cccc(C)c21 c1(N2C(C)CCC2C(=O)Nc2ncc(Br)cc2F)ncc2c(n1)CCC2 c1(NC(C2CC(C)S(=O)(=O)CC2)=O)ccc(-c2ccco2)cc1[N+](=O)[O-] C12CCCN(C1)C2=O.c1(C(=O)NC(C2(C(=O)OC)CCC2)C)cc(C)sn1 C(=O)(CC(=O)N1CCC(C(=O)NC(C)(C)CCNC(N)=O)O1)OCC N1(C(CCN(C(=O)CC2CCCOCC2)CC=C)=O)CCC(O)(COC)CC1 N1(C(C(CNC(CC(C)C(C)(C)C)=O)C(C)(C)C)=O)CCc2cc(F)ccc21 C(=O)(NN1CC2CCCC2C1)NCC(CO)OC(C)=O N1(C(C(C)C)=O)CC(NC(=O)COC2CC=CC2)CCC1C C(C)(C(C)(C)C(=O)NC(c1nc[nH]n1)CO)NC(c1c(C)cccn1)=O C1(C(=O)NC2CC3CC(NC(CCC#N)=O)C2C3)CCCCC12OCCO2 Cc1cc(=NC2CC3CN(C(=O)CCc4ccc(Cl)s4)CC23)[nH]c(C(C)(C)C)n1 c1(C(N2CCC(OC)C2)C(=O)Nc2ccccc2)cc(F)ccc1Br CC(C)C(O)(C(=O)NC1CCN(C(=O)CC(C)(C)O)C1)C(F)(F)F C12(CCC(N3CCC(Cc4cn(C5COCC5O)nn4)C3)=O)CCC(CC1)C2 C1(CNC(C(CC)NC(N)=O)=O)CC2(CCC2)CN1C(=O)C(C)=C1CCC1 Cc1cc(COC(c2ccc(C(c3ccccc3)=O)[nH]2)=O)cnc1C Nc1cncc(C(=O)NCC2(F)CC(Cc3ccc(F)cc3)C2)n1 c1(C(N2CC(NC(C3C(C=C)OCC3)=O)C(O)C2)=O)ncnc(O)c1F C1(C(N(C)CC2CCN(C(=O)Cc3ccsc3)C2)=O)CCCN1S(=N)(=O)N(C)C C(=O)(C(CC(C)C)N(C(C12CC(C1)S(=O)(=O)C2)=O)C1CC1)N1CCC(CC)CC1 c1(OC)ccc(CC(=O)OCC(F)(F)C(C)(C)O)cc1F CC(C)CC(=O)N(C(C(=O)NCCNC(N)=O)C1CC1)C c1(C(NC(NCC)=NCC2CCN2C(C)=O)C(C)C)cc(C(=O)OC)ccc1F C(CC(O)CC(=O)N1CCC(CC(=O)NC(C)(C)CN2CCCC2)C1)C(=O)OCC C(=O)(C(CNC(=O)C(C1CC1)OC)C(C)(C)C)Nc1cnc(OC)c(Cl)c1 C1(C(=O)NCCC2CC(F)C2)CCCC(NC(C2(c3cc[nH]n3)CC2)=O)C1 C1(n2c(C(=O)N(C3CC3)CC3CCC3)nc(-c3nccs3)n2)CCS(=O)(=O)CC1 C(C1CCCN1C)=CC(=O)N(CC(C)C(=O)NCC1(O)CC(O)C1)C N1(C(C(C)Oc2ccccc2)=O)CC(F)(F)CC1CNC(C1(C(=O)OC)CC1)=O Cn1nccc1-c1n[nH]cc1CNC(=O)NC(C1(C)OCCO1)C1CC1 c1(C(=O)NCCCC(C)NC(c2[nH]nc(OC)c2Cl)=O)cn(C)c(=O)cc1C c1(N2CCCC(COC)(NC(=O)CC3CC3C)C2)ncnc2sccc12 N=c1[nH]cc(C(N2CC(N)(c3nn[nH]n3)C2)=O)c2cc[nH]c12 C(CCCCCNC(C1(COC)CCC1)=O)NC(Cc1cn(CC)nn1)=O CC(F)(CNC(=O)Cn1cccc1)CNC(c1sccc1Cl)=O C1(CCC)CN(C(c2cc(Br)n(C)n2)=O)CC1NC(=O)CN(C)C(C)=O Cc1nccc(C(N2CC(NC(=O)C(C)(C)c3ccn(C)n3)C(C)(C)C2)=O)c1N CC1(C)CCc2[nH]nc(C(=O)NCC3CCCN(C(=O)C(C)(C)C(F)F)C3)c2C1 C1(CNC(c2ccc(CC)[nH]2)=O)CCCCC1NC(C1CC2(CSC2)C1)=O c1(C(N2C(C(=O)NCc3ccccc3Cl)CC(OC)C2)=O)c(C)cccc1C C#Cc1ccc(C(N2CCN(C)CC2CNC(=O)CN2CCCCC2=O)=O)cc1 c1(C(=O)NCCC(CNC(=O)CC23CCCC2C3)O)ccc(O)c(F)c1 C(=O)(CCC(C)NC(c1cnn(C(F)F)c1)=O)NC(CCOC)CO C1(CNC(CNC(=O)NC(C2CC(NC(C)(C)C)C2)C)=O)CCC=CCCC1 c1(C(=O)NCC2C(NC(CCCC(=C)C)=O)COC2)c(C)cc(Cl)cc1C N1(C(c2ccc(C)s2)=O)C2CCCC1CN(C(c1n[nH]c(C)c1F)=O)CC2 c1(CNc2ccc(-n3c(C)cc(C)n3)nc2)cncc(F)c1C C(=O)(C(C)(C)C(C)NC(=O)CC1C=CCC1)NCC1(C(=O)OC)CC1 c1(C(=O)NC(CNC(C(CC(C)C)O)=O)(C)C2CCC2)ccc2occc2c1 CC1CCN(C(=O)CCc2cccnc2)CCC1N1CCC(O)C(C)(C)C1 C1(C(=O)NCCOCC2CC2)CC(C(=O)NCC2CCSC2)C1 c1(NC(C2CC2c2ncc(CN3CCC(O)C3)s2)=O)ccc(O)cn1 c1(CNc2ccc(-c3cc(OCOC)c(O)cc3)s2)n[nH]c2ccc(Cl)cc12 CCC(C)C(C)C(=O)NCC1CCCN1C(c1sc(-c2cnn(C)c2)nc1C)=O CC(C)S(=O)(=O)CC(=O)NC(CNC(=O)CCN1CCNC(=O)C1)CO c1(C(=O)OC)nc(NC(=O)C=CC(=O)NC(C2CC2CSC)C)co1.C1CC1 Cc1nc2ccc(C(N3CCN(C(=O)COc4ccccc4)C4CC34)=O)cc2o1 CC(CC(C)(C)C)C(=O)NC1CCCC1CNC(c1c[nH]cc1C1CC1)=O N1(Cc2ccc(Cl)cn2)CC(=O)N(Cc2ccc(C#N)cn2)C1=O c1(NC(C(C2CC2)NC(C2C(=C)C2)=O)=O)cc(C)c(F)c(C)c1 Cc1ccc(O)c(CC(=O)NCC(C)(O)CNC(=O)CNC(C2CCC2)=O)c1 CC1CCC(C)(C)CN1C(C1C=CCN1C(=O)C1=CCCC1C)=O C1(C(N2C(C)(C)C(CO)C2)=O)CC2C=CC1N(C(C1(C#N)CCOCC1)=O)C2 N(C(=NCCCOC1CCCCC1)NCC1COCCO1)CC(C(C)C)CO CCS(=O)(=O)CC(=O)N1CC2(CC(CNC(=O)CCC(F)(F)F)C2)C1 c1(C(=O)NC2CC3CN(C(C(C4CC4)OCC)=O)C2C3)cnn(C)c1S(C)(=O)=O Cc1ccc(C(N2CC(NC(c3cnc(C4CCOCC4)s3)=O)C3CC23)=O)nn1 n1(CC)c(CNC(=O)C(c2ccco2)NC(=O)CCc2ccncn2)cnc1C Cc1cccc(C(=O)NC2CCC(NC(C3CCC(CN(C)C)CC3)=O)C2)c1C c1(C(N(CC(C)CNC(=O)C(O)C2CCC2)C)=O)cc(O)cc(Cl)c1 c1(OC)c(Cl)cc(C(=O)NC2(C)CC(NC(C3(C)CCC3)=O)C2)c2ncccc12 n1(CC)nc(C(=O)N(C)CC=CC(=O)NC2CCOC2)cc1O N1(C(c2ccc(CC)o2)=O)CCC2(C(=O)N(C3CCCC3)C3CC3)CCCC12 c1(CC(C)N(C)C(=O)NCCN)ccc(Br)cc1OC(F)F CCC1=C(C(=O)Oc2ccccc2)C(c2n[nH]cc2C)NC(=O)N1CC c1(OC)ccnc(NC(C2CC2OCc2ccccc2)=O)c1I c1(CC(=O)NCCCN(C(c2n(CC)ccc2)=O)C2CC2)cccc(C)c1 C1(CNC(c2cc(C(C)C)on2)=O)CC(C(=O)NCCn2cc(CO)nn2)=NO1 c1(C(=O)NCC2CN(C(=O)C=CCO)CC2O)ccc2nc(S)oc2c1 c1(NC(=O)NCC2CC(OC)C2)cnccc1S(C)(=O)=O [N-]=[N+]=NC1CCC(C(N2CCC(CCNC(=O)C(O)C3CCC3)C2)=O)CC1 N1(C(CC(C(C)OC)NC(C2(C)CNC(=O)C2)=O)=O)CC2CCC(C1)N2C Cc1cc(C(=O)N(CCCN(C)C(C2(F)CC2(F)F)=O)C)c(N)c(C)c1 C12(NC(c3cnn(C(C)C)c3Cl)=O)COC(C1)C(NC(=O)CCCCN(C)C)C2 N1(C(Cc2n(C)cnc2)=O)CC2(CCC2)CC1C(=O)N1CC(O)CCO1 c1(CN(C(c2c(NC(COCCOCC)=O)c[nH]n2)=O)C)cccc(C)c1 c1(C(N2CCC(CNC(=O)CNc3ccccn3)C2)=O)cc2cccnn2n1 c1(C(=O)NCCCN(C)Cc2coc(Br)n2)cc(C(F)(F)F)nc(C(C)(C)C)n1 N1(C(C(CCC)OC)=O)CC2CCC2(C(=O)NC2C3CCC2CC3)C1 C(=O)(C(CC(=C)C)NC(=O)CCN(C)C)NC(C1CCOC1)C#C N1(C(=O)Cc2ccccc2)CCC(C2CN(C(C3(O)CCC3)=O)C2)CC1 Cc1ccnc(C(=O)NCCOCCN(C)C(c2ccccc2)c2ccn(C)n2)c1 C(=O)(C1=NN2CCCN=C2N1)N1CC(C2(NC(C3C4CC4C4CC34)=O)CC2)C1 C1(CCNC(C=CC(C)C)=O)CN(C(C2CC2C2CC2)=O)CCO1 Cc1cc(NC(N2CC(F)(F)CC2c2nn[nH]n2)=O)c2nccn2c1 c1(CC(=O)NCC(C(C)C)NC(C23OCC(CC)(C2)C3)=O)ccc(OC)c(F)c1 c1(CCCC(=O)Nc2ccc(SCCO)cc2)ccccc1Br CC(CC(C)(C)C)C(=O)NCC1CC(O)(CNC(c2cccn3nccc23)=O)C1 C(=O)(C(C(C)C)N(C(c1ccccc1SC(F)F)C(=O)NC1CCC1)C)NC C#CC(CC(C)C)NC(=O)C(C)C.C(=O)C(C)CC=CC N1(CC(=O)NC2C(C(N(CC(C)C#N)C3CC3)=O)CCC2)CCCCCC1 C=CCC(C)(C)C(=O)N1CCC(CC(N2CCC(CC(=O)NC)C2)=O)C1 c1(C(N2C3(CN(C(CS(CC)(=O)=O)=O)C3)CC2)=O)cc2n(n1)CCCC2 C1(NC(CC(C)OC)=O)CCN(C(c2c(Cl)c(C)nn2C)=O)CC12CCC2 c1(C(=O)NCC2(F)CC(CNC(=O)Cc3ccncc3)C2)cnn2c1NCCC2 C1(CN(C)C(c2cc(-c3ccncc3)[nH]n2)=O)CCCN(C(=O)CCF)C1 N1(C(C2CCN(CC)C2)=O)CCCCC1C(N1CCC(C(N)=O)C1)=O C1(C(C)C)CCC(C(=O)NC(c2cscn2)CO)N1C(=O)CCc1ncccn1 c1(C(N2CCC(O)(CNC(c3nc(C)n(C(F)F)c3)=O)C2)=O)nnc(O)nc1O N1(C(COCCC)=O)CCN(C(=O)Cc2nccn2C)C(C)C1 C=CCC(C)C(=O)N1CCC1CNC(c1nnc(C)s1)=O CC(N=c1[nH]c(N2CCC(C)C(F)(F)C2)nc2ccsc12)c1ccc(C#N)cc1 N1(C(C(CC)(F)C(=O)OC)=O)CCCC2(CCN(C(=O)C#CC(=O)N(C)C)C2)C1 N1(C(C2C(C#N)C2)=O)CCN(C(c2ccnc(C(F)(F)F)c2F)=O)C(CF)C1 C1(C(N2CCCC(NC(C3CCC(SCC)CC3)=O)C2)=O)CCCC(=O)N1C c1(N2CCN(C(C)=O)CC2)nc2ccc(Cl)cc2c(=NC2CCCCC2CC)[nH]1 c1(-c2nc(C3CC3n3ccnc3)on2)cccc(CO)c1F.CCS CCCC(CC)C(=O)NCC1CCC(N(C(=O)CC2CCNC(=O)C2)C)CC1 c1(C(N2CCC(CCOC)(NC(c3oc(C)nc3C)=O)C2)=O)ccc(O)cc1F C1(NC(c2c(CC)[nH]cc2)=O)CC=C(C(=O)NC(C)(C)CO)C1 C12CCCC3(CN(C3)C(=O)c3ccc(c(OC)c3)NC1=O)O2.C(=O)(C1CC1)OC c1(C(N2CCN(C(C=CCCC)=O)C3C2C3)=O)ccc2c(c1)CCC2 N1(C(CCCC)=O)CCC(C)(C)C1CC(=O)NC1(C2(C)CCCO2)CC1 c1(C(N(CCCCNC(C(C)C2CCCO2)=O)C)=O)cc2n(c1)CCSC2 Cn1nc(CC(=O)NCCNC(c2coc(Cc3ccccc3)n2)=O)cc1Cl.C c1(NCC(N(C(=O)CC(O)C2CCCC2)C)C2CC2)ncncc1I C(CC(C)C)(C(=O)NCC1CN(C2CC2)C1)ONC(COCCOC)=O N1(C(c2ccc(COC(C)C)cc2)=O)CCC(F)C(NC(=O)C2=NOCC2)C1 C(=O)(C(C)=Cn1ccnn1)NC1(CC(Cc2c(C(=O)OC)ocn2)OC)CC1 S(=O)(=O)(C1CC1)CNC(=O)NOCC1(c2ccon2)CCC1 CCCC(C(=O)NCC(C)NC(=O)Cc1conc1C)NC(=O)OC(C)(C)C c1(C(N2C(CC)CN(C(c3oncc3C)=O)CC2)=O)n[nH]c2ccccc12 c1(C(=O)NCC2CN(C(c3ccc(C)n3C)=O)C(C)(C)C2)ncnc2sccc12 Cc1cc(C(=O)NC(C)C=CC(=O)N(CCc2ccccc2)C(C)C)nc(O)c1 CC1(C)CC(CC(N2CC(O)(C3CCCN3C(=O)C=Cc3ccco3)C2)=O)CO1 c1(N2CC(CCNC(C(C(C)C)OC)=O)(OC)C2)[nH]nc2c1c(C)nn2C N1(C(CNC(CCSCCC)=O)=O)CCCN(C=O)CC1 c1(CC)ccc(C(=O)C(=O)N(C)CC2CCN(C(=O)Cc3csc(C)n3)C2)s1 c1(NC(CC(C)OC)=O)ccc(NC(c2cnn(C)c2C(C)(F)F)=O)c(C)c1 CC1CN(C(C2(C(=O)NC3CC3)CC2)=O)CC(C)C1CNC(C1CC(O)C1)=O CCC(C(=O)N(CCNC(=O)CCCC1(OC)CCCC1)CCOC)OC c1(C(c2n(CC=C)nnn2)N(CCC2CCO2)C2CC2)c(C)noc1C C=CCC(CC)C(=O)N1CCOCC(NC(=O)CNC(c2cccc(C)c2)=O)C1 C=CCCCC(C(=O)N1CCC(c2ncco2)C1)NC(c1csc(CC)n1)=O C1(CCNC(CN(CCCCCC)C)=O)CCCN(C(=O)CC2(O)CCOC2)C1 c1(NC(C2N(C(C(C(C)C)O)=O)CCCC2)=O)cc(Br)ccc1C#N C1(NC(N(CC(=O)OCC)CC2CC2)=O)CCC(NC(C)(C)C)C1 c1(C(=O)NCC(C)N(C)C(C2CCOC3(CCC3)C2)=O)cccn2c(O)nnc12 Cc1cc(-c2nc(C(C)CNC(=O)CC3(C)CC3)no2)c(C)n1C c1(CN(CCCC2CN(C(=O)OC(C)(C)C)C2)C)cc(F)c(F)cc1Cl C1(C(N2C(CC)C(C(=O)NC3C(O)CC3O)CC2)=O)CC2CC(=O)C1O2 C12(C(N3CCC(CC=C)(NC(=O)Cc4cscn4)C3)=O)CCCC1OCC2 C1(SCCOC)COC2(CCCN(C(=O)COCC(=O)NC3CC3C(=O)OC)C2)C1 c1(NCC2N(C)CCN(C(C3CCCO3)=O)C2)ncnc2c1CCCC2 C1(C(=O)NC(CCSC)CO)CCN(C(=O)CC2CC3CCC2C3)C(C)C1 C(C(C)(C)CNC(=O)C(C)Cn1ccc(C)n1)N(C(C1C(C(=O)OC)CC1)=O)C C(=O)(CCCc1nc(C2CC2)no1)NC1C(CNC(CNS(N)(=O)=O)=O)CC1 C(C(F)C(=O)NCC(N1CCOC1=O)(C)C)C1N(C(C=CCOC)=O)CC1 c1(C(N2C3C(NC(=O)Cc4cnns4)C(C3)C2)=O)ccc2c(c1)CC(=O)N2 N1(C(COC(CC)C)=O)CCCC2(CNC(=O)C(F)=C3CCC3)CC12 Cn1ncc2ccc(CC(N3CC(F)(F)CC3Cn3cc(C4CC4)nn3)=O)cc12 C1(C(N2CCCCC(N(C(C(CC)CC)=O)C)C2)=O)CC2(CC(C)=NO2)C1 C12(NC(c3cc4ccccn4n3)=O)CCCCCC1N(C(=O)Cn1ccnn1)CC2 C1(CCC)(NC(c2nn(C)c(Cl)c2Cl)=O)CCN(C(c2n[nH]c(C)c2O)=O)CC1 C=CCC(C(=O)NC1(CNC(=O)C(C)C(=O)OC)CCCCCC1)C(C)C C(CC(C)C(=O)N(CC(=O)N(C1CCCCC1C)C)C)=CCC C1(CN(C)C(c2cc(-c3ccccc3)c[nH]2)=O)CCCN1C(=O)CC1C=CCC1 c1(NC(=O)NC2C(c3onc(COC)n3)OCC2)cccc2cc(Br)cnc12 c1(OCCOC)cccc2[nH]cc(C(=O)NCCC(O)CNC(=O)C(C)=C(C)C)c12 C(=O)(CN=S(C)(C)=O)N(C1CN(C(C2CN(S(=O)(=O)C(F)F)C2)=O)CC1F)C C(=O)(CC(C)CC(C)C)NCC(C(C)(C)C)NC(c1c(C)nco1)=O C1(NC(CC(CC)C2CC2)=O)CN(C(=O)C(F)C2CCCC2)CC12CCCC2 c1(CC)cccc(NC(C2CCCC(NC(=O)C(C)(C)CF)C2)=O)c1C Cc1cn(C)cc1C(=O)NCC(C1CCOC1)NC(c1c(C)coc1C1CC1)=O C1(C(C)NCC(C)C)CCN(Cc2cccs2)C1=O S(=O)(=O)(c1ccc(CN)cc1)Nc1cccc(C(N(CC(C)NC(N)=O)C)=O)n1 C1(C#N)(CC(=O)NCC(CC)NC(=O)CCc2ccc(C)nc2)CCOCC1 C(=O)(C(O)CC(C)(C)C)NC1C2(C(=O)NCCCCC3(CO)C(C)C3)CCC(C1)C2 N(C(=NCC1CCOC1)N1CCC(O)C1)C.OCC(C(F)(F)F)c1ccccc1 c1(C2(O)CN(C(=O)NC(c3ccc(Cl)cn3)C)C2)ccccc1Br C=CCC(C(=O)NCC(CO)NC(=O)C(C)C1CCOC1)c1ccccc1 CCCC(C(=O)N(C(C)CC)C(C)C)NC(=O)C=CC(=O)N(C)C C1(NC(COCC#C)=O)CN(C(c2cnc(C)nc2C)=O)CCC1CO Cc1nc(SCC(=O)NCC(CNC(=O)C(C)(C)N2CCOCC2)CO)n[nH]1 N1(CC)CCC(NC(c2cnn(CCNC(=O)CN3CCC(O)CC3)c2)=O)CC1 N1(C(Cn2nc(C)c(Cl)c2)=O)CCC2CC1CN(C(=O)CCC(C)N(C)C)C2 N1(C(CCOCCC)=O)CCN(C(=O)CN(S(=O)(=O)CC)C)C(C(C)(C)C)C1 c1(NC)ncccc1C(=O)NCC1CCN(C(=O)CC(F)(F)Cl)C1 N1(C(CS(CC)(=O)=O)=O)CC2(CCCC2)C1C(N1CCC(CO)CC1)=O c1(C(N2C(CNC(=O)CNC=O)CC(C)(C)C2)=O)ccnc2cc(Cl)ccc12 CCC(C#N)C(=O)NC1CCCCC1CNC(=O)CCc1cnc(C2CCC2)o1 N1(C(C2CN(C)C(=O)C2)=O)CCC2(CCN(C(c3cccc(CO)n3)=O)C2)C1 C(C(C)(C)CC(=O)N1CCC(CCNC(=O)CCC2CC2CC2CC2)C1)N(C)C C1(=O)C(C(C)C)N1.C1(C)(NC(CN(CC)CC)=O)CC(C(=O)OC)C1 O=C(CC1CCc2ccccc21)NCC1CCN1C(=O)CCCc1cccs1 C1(CNC(C2CCN(C(C3(NC(C)=O)CC3)=O)C2)=O)CCOCC1(C)C C=CC(C)(C)C(=O)N1CC(O)(CCNC(C2CCN(C(C)=O)C2)=O)C1 C1(NC(c2n[nH]c(CO)c2Br)=O)C(OCC2CC2)C2CCCC12 CCC1=C(C(=O)NC2(CF)CCN(C(c3csc(C)c3)=O)C2)CCCO1 c1(N(CCCC=C)C)nc(C)cc(=NCC2(C3CCOCC3)CC2)[nH]1 N1(C(c2cc(C)c(C)nc2)=O)CC2CCC(N(C)C(c3ncc[nH]c3=O)=O)C2C1 C(=O)(CC(C)(C)C(F)F)NCC1(F)CCCN(C(=O)OC)C1.N12CCCC1C2=O COn1cnc(C)c1C(N1CCC1CNC(c1cccn(C2CCC2)c1=O)=O)=O C1(Br)(C(N(CC(C)NC(C2(CCOCC)CCC2)=O)C)=O)CC12CCC2 c1(CC(=O)NC(CNC(CN(CCC#C)C)=O)CC=C)ccccc1Br n1(CC(=O)N(CC(C)NC(c2cn(C)nc2C(F)F)=O)C)nnc2c1CCCC2 C(=O)(C(C(C)(C)C)NC(c1csc(C)c1)=O)NCCSCC N1(C(C(C)O)=O)CCC(N(C(=O)C=C2CCC2)Cc2ccccn2)CC1 N1(C(c2cc(C)on2)=O)CC2CCC2(NC(c2ccnc(S)c2)=O)C1 C=CCC(CC)C(=O)N1C(CC(=O)NCCC2CCSC2)C2CCCC12 CC(C)CC(CNC(c1cc(C(C)C)[nH]n1)=O)NC(C1CN(C(N)=O)C1)=O c1(OC)ccsc1C(N1CCC(N(C(=O)CN2CC=CC2)C)C1)=O C12(CNC(c3c(C)cc(SC)o3)=O)CN(C(c3ccn(C)c3)=O)CC(F)(C1)C2 c1(C(N(C(C)C(=O)NC(c2ccncc2F)C)CC)=O)c[nH]c2nccc-2c1 C1(F)(C(=O)NCC(C2CCC2)NC(c2cnc(SC)s2)=O)CCCOC1 N1(C(C2C3CCN(C(C(COC)N(C)C)=O)CC32)=O)CCS(=O)(=O)CC1 N1(CCC2C=CC(C(=O)NC(c3ccc(Cl)cc3C)=O)C2)Cc2ccccc2C1 C(C(O)CCCCC)NC(C1(CC=C)CCN(C(=O)CC2CSCCO2)C1)=O C1(NC(C2(CCCC)CC2)=O)C=CCN(C(c2cc(C)nn2C)=O)C1 c1(C(C)NC(c2c(C(=O)NC(CC=C)CO)cccn2)=O)ccccc1[N+](=O)[O-] N1(C(C2CC(C)=C(C)CC2)=O)CCC(CNC(=O)Cc2cncnc2)C(F)(F)C1 N1(C(C(=O)Nc2ccc(C(=O)NCC(CC=C)NC(C)=O)s2)C)CCC(O)CC1 c1(C(=O)NC2C(CO)CCN(C(=O)NCCC(N)=O)C2)cc(S(N)(=O)=O)cs1 c1(C2C(C(=O)NCCC3(NC(CSCCCC)=O)CC3)C2)cnn(C(C)C)c1 N1(C(CN(C)CC)=O)CC=CC(NC(c2cn(CC(F)F)nc2C)=O)C1 C(N=c1nc(CC)cc(C)[nH]1)C1(F)CCN(C(C2CC3(CC(=C)C3)C2)=O)CC1 C1(C(=O)NCCN(C(=O)C#CC(C)(C)C)CCOC)CCCCC(=O)N1 c1(C(=O)OC)ccc(N2CC=CC(NC(c3ccc(F)cc3F)=O)C2)c(C#N)n1 C1(CN(C(=O)Cc2cnc(O)[nH]2)CC)CCCN1C(=O)CC1COCC1O C1(NC(C(C=CC)O)=O)CCN(C(C2CCCCN2S(=O)(=O)CCC)=O)CC1 C=CCC(CNC(C1CN(C(=O)C(C2CC2)SC)CCC1(C)C)=O)CC(C)C c1(NC2(C)CC2)ncccc1S(=O)(=O)NC1(NCC(c2ccc(F)cc2)O)CC1 N1(C(c2cc(C)ncc2)=O)CCCC(NC(=O)CCC2CCC(=O)N2)C1C N1(C(C(CC)OCC)=O)CCC2(CC1)CCN(C(c1cnn(C(F)(F)F)c1)=O)C2 N1(C(C2CC(CC)C2)=O)CCC2(CCN(C(=O)CC3CC4CCC3CC4)CC2)C1 CC1CN(C(=O)C(O)CN2CCCC2)CCC1C(=O)NC1CCC2CC12 C1(CC(=O)N(CCCCCNC(=O)C(C)n2cccc2)C(C)C)SC(=N)NC1=O Cc1cc(C(=O)NC(C)CCNC(=O)CSCc2ccncc2)c2nccn2c1 C1(N(C)C(c2cccc(-c3ccncc3)c2)=O)CN(NC)CC1O.c1(C)ccc(CO)o1 O=C1CC(=O)CC(C(N2CCOCC2Cc2cn(C3COCC3O)nn2)=O)C1 CS(=O)C=CC(=O)NCC=CCNC(c1ccc(C(=O)NC2CC2)s1)=O N1(C(c2cc(C(C)=O)n(C)c2)=O)CCCOC(CCNC(C2CCCCS2)=O)C1 C1(N(C(=O)C(F)n2ccnc2)C)CC2CCC(C1)N2C(C1(C#N)CCCC1)=O C1(NC(c2ccc(OC)s2)=O)CC(CC(=O)NC2(C)CCSCC2)C1(C)C c1(OC)ncc(F)c(=NC(=O)c2ccn3ncc(SC)c3n2)[nH]1 Cc1cc(C#N)cnc1C(N1CCCCC1CCNC(C1(NC(C)C)CC1)=O)=O Cc1sc(Br)nc1C(=O)NC1(CCNC(C2C=CCC2)=O)CCCC1 c1(-c2onc(-c3ncc(C(F)(F)F)s3)n2)cccc2cccc(Br)c12 c1(NC2CC(F)(CNC(c3n(C)nc(C)c3Cl)=O)C2)ncnc2c1cnn2C c1(N2CC(F)C(F)C2)nc(=NCc2conc2C2CC2)[nH]c2c1CSC2 C(CC)(C(=O)NCCC1CCN(C(=O)COc2ccccc2)C1)OCC N1(C(c2cccnc2)C(=O)OC)CCN(C(=O)C2CC2)CC1 c1(C(N2CC3CN(C(=O)Cc4cncs4)CC32)=O)cc2ncccn2n1 c1(C(=O)OC)ccc(CNCC2(O)CN(C(=O)CO)C2)o1 N1(C(C(CO)NC(C)=O)=O)C(C(=O)NCCCC(C)C)CCC1C CCC(C(=O)N(CC(C)N(C)C(c1ccoc1C1CC1)=O)C)OC C1(C(C)NC(C2CC2F)=O)CCCN1C(c1ccc(C(F)(F)F)s1)=O CC1(C)CCC(C(N2CC(CCNC(C3(C4CCCO4)CC3)=O)C2)=O)CC1 c1(CNC(=O)C(=O)NC2CC2)ccc(C(=O)NC2C(OC(C)C)CC2)cc1 C1(F)(CNC(c2cccc(F)c2O)=O)CCN(C(=O)C(F)(F)c2cscn2)CC1 N1(C(C2CC(C)OC2)=O)CCC(CNC(c2cn(Cc3cccs3)nn2)=O)CC1 N1(C(c2c[nH]c(=N)s2)=O)CC2ON=C(CNC(=O)CN3CCCCC3)C2C1 C1(C(=O)NC2C(CNC(C(c3ccc(C)cc3)(F)F)=O)CC2)CCC(C)(C)CC1 c1(CC)cc(CNC(N2CCC(CO)(Cc3ccccc3)C2)=O)n(C)n1 C(CC(=O)NCC1CN(C(=O)CN(C)C)C2(CCC2)C1)(C(F)(F)F)OC Cc1nc2ccccc2n1CC(=O)NC1(CNC(c2n[nH]cc2Cl)=O)CCOC1 C(=O)(C1=NN(C)C(=O)CC1)NC1CCCCN(C(C(C(C)C)F)=O)C1 N1(C(CCSCCC)=O)CC2CC(C(=O)N(C)CCOCCO)(C2)C1 c1(C(=O)NC(CCNC(C(c2cnn(C)c2)OC)=O)C)c(C(F)(F)F)n[nH]c1C C1(=O)C(C)(C)C(=O)NN2CCN1CC2.c1(SC(C)C(=O)OC(C)(C)C)ccccn1 C1(C)(C(N2CCC(c3cn(C)nc3)C2(C)C)=O)CCCNS1(=O)=O Cc1sc(-n2cnnn2)c(C(=O)NC(CNC(C2CC2F)=O)C2CC2)c1C C(=O)(C1=NOC(C(C)(C)C)C1)N1CC(N(C(c2cnc(C)[nH]2)=O)C)C1 N1(C(C(C(CC)CC)F)=O)CCCC2C(=O)NCC12 N1(C(c2cccc(C)c2Cl)=O)CCC2C(CCN2C(c2ccc(O)cc2Br)=O)C1 N1(C(CCC=C(C)C)=O)CCCC2(CNC(c3cc(Cl)ccc3C)=O)CCCC12 CC1=C(C(=O)NC2COCCN(C(=O)COCC3CCCO3)C2)CCC1 C1(C(N(CCNC(c2cc(C3CC3)ncn2)=O)C2CC2)=O)CCCCC1F Nc1c(F)c(F)c(C(=O)NCC2(NC(C3CC=CCO3)=O)CCC2)c(F)c1F N1(C(=O)CC2CCSC2)CC(N(C(C2CCOCC2)=O)C2CC2)CC2(CCC2)C1 Cc1c(C(=O)NC(CNC(=O)C(C)C2CCCO2)C(C)C)noc1C1CC1 Cc1cccn(CC(=O)NCC2COCCN(C(c3cc(F)n(C)n3)=O)C2)c1=O N1(NC(C=C(C)CSc2nc[nH]n2)=O)CC(O)(C2CCC2)C1 c1(OC)cc(NC2(C(N)=O)CCNCC2)ccc1CC(=O)Nc1ccc(F)cc1 Cn1cc(C(=O)NCCC2CN(C(C3(F)CC3)=O)CCO2)c(Br)n1 C=C(C)C(O)CC(=O)N1CCCC(N(C(=O)CCSCC(C)C)C)C1 C1(CNC(C=NOC)=O)CN(C(c2cccc3nccn23)=O)C2(CCC2)C1 CC1(C)C(C(=O)NCC2CCN(C(C3CC(n4cnnc4)C3)=O)CC2)C1C#N N1(C(CC2(C=C)CCC2)=O)C2CCC1C(F)C(NC(c1cc(OC)c(Cl)s1)=O)C2 C1(C(=O)NCC2N(C(c3c(C)n(CC(C)C)nc3)=O)CC2)CC(=O)NC1(C)C c1(CNC(C2(N(C)C)CN(C(CCNC(C)=O)=O)C2)=O)cnccc1Cl C(=O)(CCS(C)(=O)=O)NC(C(C)NC(c1cnn(C(C)C)c1Cl)=O)(C)C c1(C(=O)NC2CC3CN(C(CS(CC)=O)=O)C2C3)ccc([N+](=O)[O-])n1C c1(C(N2C3CCN(C(CC=C)=O)CC2CC3)=O)ncc2ccccc2c1O c1(NCCc2n(C(C)C)ccn2)[nH]c(=NC(C)C2CC2)nc2sccc12 c1(C(=O)NCCN(C(CSC)=O)CC(C)O)ccc2c(n1)CCC(C)C2 C1(NCC(=O)NCC(C)(C)NC(CC2CCN(C)C2)=O)C=CC(C)(C)CC1.CCC=O c1(NC(C(=O)NC2CC(CC(=O)OC)C2)=O)ccc(CO)cn1 N1(N2CC(C(C(=O)N3CC(CCS(N)(=O)=O)C3)OC)C2)CCOCC1.C=O C1CC(C)(C)C(=O)NCCC(C)(O)C(=O)N1.C(CC1CC1)(CO)OC n1(CC(=O)NCC(C)(C2CCC2)NC(C(COC)C)=O)ccc2c(N)cccc12 C1(CC(=O)NCCCCC#C)CN(C(c2ns[nH]c2=O)=O)C(C)(C)C1 C1(C2CC2)(CNC(C2CC(OCC)C2)=O)CCN(C(C2(OC)CCCOC2)=O)C1 C(N=C(NCCF)NCC(C)(C)C)CCC=C.C(=O)NC N1(C(Cc2cn(C)nc2Cl)=O)CCCOC(CNC(C2(C)C=CCC2)=O)C1 CCCC(CNC(c1ccnn1CC)=O)NC(=O)CCCc1ccsc1 c1(OC)ccc(F)c(C(=O)NC2CN(C(=O)CCc3cnc[nH]3)CCC2C)c1F c1(N(C(COc2c(OC)ccc(Cl)c2)=O)C)ccc(Br)c2cccnc12 N1(C(C=CC)=O)C(C(=O)Nc2ccnc(Br)c2)CC2CC12 c1(NC(C2CC(O)CN2Cc2cccc(F)c2O)=O)ncc([N+](=O)[O-])cc1Br Cc1ccc(C2CCCN2c2nnc(C3CC3)n2CC(=O)NCCO)n1C C1(=O)CCCN(C(=O)CC)CC(C)N1.C1(C(N(CC)CC)=O)CC(OC)C1 CC(CC1CC1)C(=O)N(CCCCNC(C1CS(=O)C1)=O)C c1(C(=O)NCC(CO)NC(CC2(OC)CCC2)=O)cnc2ccnn2c1 c1(C(C)=O)ccccc1C(=O)NCC1CC1NC(c1nc(C)oc1C)=O c1(C(N2CCN(C(C(COCC)(C)C)=O)CC2CCO)=O)ccc(C#N)cc1O c1(NCC2(NC(C3CCCCC3(F)F)=O)CC2)cc(=O)n2ccccc2n1 C#CCCCC(C)C(=O)NC1CC12CCC(NC(c1c(C)ncn1O)=O)CC2 C(=O)(C(C)CCCOC)NC(CNC(c1c(CC)n(CC)nn1)=O)(C)CC CC(C)(C)C(CNC(c1[nH]ncc1C#N)=O)NC(c1cccc(O)n1)=O c1(C(=O)NCCCNC(C2C(C)OCCC2)=O)cnn2c(Br)cccc12 c1(C(C(=O)NCc2nccs2)N(C2CCN(C(C)=O)CC2)C)cccc(F)c1F n1(CC(=O)NC2CCCC2CNC(C2(CF)CC2)=O)ccc([N+](=O)[O-])n1 N1(C(CC(C)N(C)C)=O)CC(CNC(C2(C)CC3(CC3)C2)=O)CC(C)(C)C1 N1(C(c2nc(C)c(=O)n(C)c2)=O)CCCC2CN(C(c3nc(Cl)oc3C)=O)CC12 c1(C(=O)NCC(CC)NC(C2CC3CCC(C2)S3)=O)ncncc1C#N N1(C(C(C2CCN(C(COCC#C)=O)C2)(C)C)=O)CC2C(CO)C2C1 Cc1ccc2cc(-c3nc(C(N4CC5COCC5C4)=O)cs3)ccc2n1 c1(C(=O)NC2CN(C(C3CCC(F)C3)=O)C2)nc(Cl)sc1Cl N1(C(c2scc(C)c2)=O)CC=CC(NC(=O)CCc2ccc(CO)cc2)C1 CCCC(C)(CCC)C(=O)N1CC2CCCC2(CNC(=O)COC(C)C)C1 N1(C(Cn2c(C)ccn2)=O)CCC2C(CCCN2C(=O)COc2cnn(C)c2)C1 C(CS(C)(=O)=O)N(C(c1cc(C(F)F)cs1)C(=O)NCSC1CCC1)C C1(C(C2C(C(=O)NCCCN(C(=O)CCC=C(C)C)CC)C2)=O)CCCC(=O)N1 N1(C(C2C(OCC)C2)=O)CCCCC1CCNC(=O)Cn1c(C)ccc1C N1(C(C2(CC)CCCCO2)=O)CC2CCC1CC2NC(=O)C(C1CCCC1)OC N1(C(C(C)C(F)F)=O)CC(C(=O)NC(C)CC(C)(C)O)CC(C)(C)C1 c1(CC(N2CCN(C(C(C)c3ccsc3)=O)CC2C)=O)ccc2nn(C)cc2c1 CCCCCCCCC(=O)NC1CC(CNC(=O)CC2OCCOC2(C)C)C1 c1(NC(C(c2ccoc2)NC(C(CC)CCOC)=O)=O)cccc(N=[N+]=[N-])c1 N1(C(CC=C)=O)CCCCC1C(=O)N(c1ccc(NC(=O)CCCF)nc1)CC CCC(C(=O)NCC(C1CCCCC1)NC(=O)Cc1cnn(C)c1)NC(N)=O C1(CNC(c2cc(OC)ns2)=O)CC(NC(=O)CCc2cnc(O)[nH]2)C1(C)C C(=O)(C(O)CC(C)(C)C)NCC(C1CCC1)NC(c1cc(N(C)C)no1)=O N1(C(C2CC(C(C)C)C2)=O)CC(NC(=O)C(=O)NC(C)C)CC1(C)C c1(OC)ccc(CCNC(=O)C(C)(C)C2CCCN2C(=O)CS(C)(=O)=O)cc1 N1(C(C(CC)C#N)=O)CCN(C(c2cccc(F)c2C(F)(F)F)=O)CC1CO C12(NC(C(CCSC)NS(CC)(=O)=O)=O)CCCC1N(C(=O)CSC(F)F)CC2 N1(C(C(C2CCC2)OC)=O)CC2CCC1C(NC(=O)Cc1ccc(C)s1)C2 N1(C(c2c(C)cc[nH]2)=O)CC(C(=O)NCC(C)(C)CCO)C(C)(C)C1 C1(N(CCS(C)(=O)=O)C(c2scc(C)c2Cl)=O)C2CCC1CNC2 C1(C(N2CCC(N(C(=O)Cc3cnsc3)C)C2)=O)CCCCC(C)(C)C1 N12CCC(CC(F)F)(CC1)C2=O.C1(C(N)=O)CCN(CCC2CCCO2)CC1 C1(NC(C(CC)C)=O)CN(C(=O)CN2CCC(O)CC2)CC12CCSCC2 N1(C(C)C)CCC(NC(c2ccc(C(N)=O)cn2)=O)C(C)C1 N1(C(=O)Cc2ccccc2)CCN(C(C2CCCN2C2CC2)=O)CC(CO)C1 C(C1CN(C(C2CCOC2=O)=O)Cc2ccccc21)NC(=O)CCc1cnco1 c1(C(N2CC3C(NC(C4CCC(=O)NC4)=O)C3C2)=O)ccc2ncnc(O)c2c1 C(=O)(CC(C)(C)Cc1ccccc1)NCCC(=C)CNC(=O)COC(C)CC c1(C(=O)NCC2(O)CCN(C(C3CC=C(C)CC3)=O)CC2)cc(C)c(=O)n(C)c1 C(=O)(CC(C)(C)CC(=O)N1CCCC1C(C)NC(=O)C(C(C)O)N(C)C)OC c1(C(N2CC(C)N(C(=O)CCCn3ccnn3)CC2)=O)cc2c(cn1)OCCC2 c1(C(=O)NCCc2cnc[nH]2)ccc2[nH]nc(-c3ccn(C(F)(F)F)n3)c2c1 n1(CC(N2CC(O)CC(NC(c3nocc3Cl)=O)C2)=O)ncc2cccnc12 C1(C(=O)NCCCS(C)(=O)=O)CC2C=CC1N(C(C1(C3CC3)CC1)=O)C2 CCCC(C(O)C(=O)NOCC=CCl)NC(=O)CN=c1cc[nH]cc1 c1(OC)cc(C)cc(C(N2CC3(C2)CN(C(c2cnc(OC)nc2)=O)C3)=O)c1N N1(C(C(CC)C)=O)CCN(C(c2cn(CC)c3ccccc23)=O)C2(CCC2)C1 CC(C)CC(C(=O)NCC1CCC1NC(=O)CCC1CC1)N1CCCCCC1 c1(C(N2C(CNC(C3CCN(C(C)=O)C3)=O)CCCC2)=O)ccnc(F)c1O N1(C(CC(C)(C)OC)=O)CC2C3CCC(C2C1)N(C(C1CC2CCC1O2)=O)C3 S(=O)(=O)(c1csc(CNC(c2ccc(C3(C)CC3)cc2)=O)c1)NC c1(C(=O)NC2CCC(F)(CNC(=O)CCC(F)F)C2)cnc2nccn2c1 c1(CN2C(C(=O)N(C(CO)CO)CCO)CC2)cc(Br)cc(C(F)(F)F)c1O c1(C(=O)NC2CCCN(C(=O)CC(F)F)CC2)cc(O)cc([N+](=O)[O-])c1 N1(C(Cc2c(C)ocn2)=O)CC(CO)C2(CCN(C(=O)CN3CCC3C)CC2)C1 C(CC(F)F)(C(=O)N(C)CC1CCOC1)N(C(c1c(C)nncc1)=O)C C1(C(=O)NCCC2(NC(CS(N)(=O)=O)=O)CCC2)Cc2cccnc2C1 C1(NCCNC(C(=O)OC)CC2CC(F)(F)C2)CCCC(O)CC1 c1(C(C(=O)N(C)CCN(C)C(C2(Cl)CC2(F)F)=O)O)ccc(C#N)cc1 C(=O)(C#CC1(C)CC1)NCC(c1ccccc1)N(C)C Cc1c(CN2CCC(NC3CC34CC4)CC2)cccc1F C(C(C)(C(C)C)NC(C1CN(C)C(=O)N1)=O)NC(COC(C)=O)=O CN1CCC(C(=O)NCC(C)(C2CC2)NC(=O)CCc2ccncn2)C1=O c1(CN(c2cc(OCC)nc(C)n2)C2CCNCC2F)c[nH]c2cc(C#N)ccc12 C1(NC(c2c(C)cco2)=O)CCN(C(=O)Cc2cccc(C#N)c2)CCC1CO C1(CNC)CCN(C(c2nc(-c3cccc(Br)c3)no2)C)CC1 C(=O)(CS(=O)(=O)CC(=O)Nc1cccc(CNC(C2CC23CC3)=O)c1)OC CCC(C)(O)CC(=O)N(C)CCOCCCNC(c1cccc(CN=[N+]=[N-])c1)=O c1(OC)ccc(C(=O)NCC(C)(C)NC(C2CC=CCC2C(F)(F)F)=O)c(F)c1 C1(C(=O)NC2C3CN(C(c4ccc(NC)cn4)=O)CC32)Cc2ccccc2CO1 C1(CNC(CN2C(C)CC2)=O)CN(C(c2cc3[nH]ccc3s2)=O)C2(CCC2)C1 C1(C)(CNC(CCCOC(C)=O)=O)CCCN1C(c1cccc(F)c1)=O C(CN=[N+]=[N-])(C(=O)NCc1ccccc1C)NC(CSCC#C)=O N1(C(C23CCC(OC)C2C3)=O)CCC(NC(=O)CC2OCCC2(C)C)C1(C)C Cc1cc(C2(C(=O)NCC(O)CNC(=O)CC3CC34CC4)CC2)on1 C1(C(N(CCCNC(C2(OCC)CCCCC2)=O)C)=O)OCCOC12CCC2 CC1(NC(C2CC3CCC2N3C(=O)C2=C(Cl)CC2)=O)CN2CCC1CC2 c1(C(=O)NCC2CN(C(CN(CCCCCC)C)=O)C2)cnc(N)c(N)c1 CC(CC1=CCCCC1)NC(C1CCC=CC1NC(C1CCSC1)=O)=O N1(C(=O)OC(C)(C)C)CCCC1(C)C(N1C(CN)CC1)=O.c1(C)ccc(F)cc1 n1(CCNC(=O)NC(c2cccnc2)CO)cc(CC2(F)COC2)nn1 CCC(C)(CCNC(C1CCC1C)=O)NC(=O)CCC1CCC(=O)N1 c1(C(N2CCCC(C)(C(=O)Nc3cncnc3O)C2)=O)cc2ccccc2o1 N1(C(C2CC(O)(CC#C)C2)=O)CCCC(CNC(C2(C(F)F)CCOCC2)=O)C1 C#CCCCCC(=O)N1CC(CN(C)C(c2cncc(-n3cccn3)n2)=O)C1 C(=O)(C(C)(C)N=[N+]=[N-])N1CCC(CC(=O)N(CC(=C)CC)CC)CC1 c1(CCC(=O)NC(CC)CN(C(=O)Cn2cnc(=N)[nH]2)C)c(C)n[nH]c1C n1(CC)cc(C(=O)NC2CCC(NC(=O)Cc3csnn3)C2)c2ccccc12 N1(C(C2C(=C)CC2)=O)CCC(C(C)NC(=O)COc2cccnc2Cl)CC1 n1(CC(=O)Nc2ccccc2)cccnc1=O.C1(=O)C(NC)CC(C(N)=O)N1 C1(C(N2CC(NC(C3CC(F)C3)=O)C2)=O)C2CCOCC12 c1(C(=O)NC2C(C)CN(C(C3CC4(C3)CC3(CC3)C4)=O)C2)cccc2c1CCN2 C1(NC(=O)CN(C(c2ccc(O)cn2)=O)C2CC2)CCN2CCCC12 c1(CC(=O)N(Cc2ccccc2)CC2(C(C)(C)C)CNC2)ccc(Cl)cc1 c1(CCC)ccc(C(=O)NCCCN(C2CCCC2)C(=O)CO)[nH]1 C(=O)(C(CC(C)C)C(N)=O)N1CC(NC(c2cc3sccc3[nH]2)=O)CC(OC)C1 C(C)(C(C(C)C)NC(c1ccoc1Br)=O)NC(CN(C)CC)=O N1(C(C2C(C)C(=O)C2)=O)CCCC(N)(C(=O)O)C1 c1(OC)ccc(N(C)C)cn1.c12scnc1C(=O)N1CCCC1CN(C1CC1)C2 N1(C(C2N(C(COCC=C)=O)CC2C)=O)CCC(C)(CO)C1 N1(C(C2CC(NC(C3CC(=O)C3)=O)C2)=O)CCOC(c2cn[nH]c2)C1 C(=O)(C(C(C)C)C(C)C)N1CCC(O)(CNC(c2nccc(C)n2)=O)C1 C1(C(=O)NCn2cc(NC(C3C(C(=O)OCC)C3)=O)nn2)C2CCC3C(C2)CC13 C1(COC)(NC(=O)CC(C)N(C)C)CN(C(C2(OC)CCCC2)=O)C1 C1(C(=O)NC(CCC)c2ccco2)CCOC1C(=O)N(C)Cc1conc1CC c1(C(c2n(CC=C)nnn2)NCCC(O)C(C)C)ccc(C)c(F)c1 CCCCC(C(=O)NCC1CCCC1C(=O)NCc1cc(F)ccc1F)N(C)C C(=O)(C1CCCc2ccnn21)NCCC(C)NC(c1cc(C)c(N)cn1)=O CCCCC(CC)CC(=O)NC(C)C(C)(C)NC(c1cc(CC2CC2)ncn1)=O c1(C(=O)NCC(CN(C(C2N(C(C)=O)CC(O)C2)=O)C)O)cc2ncccc2[nH]1 c1(C(=O)NC(CNC(C(C)n2cnnn2)=O)CO)cc(F)ccc1N N1(C(COCCOC)=O)CC2CCC(C1CO)N2C(c1cccc(F)c1)=O N1(C(=O)NCC(CC)C(C)C)CC(O)C(O)C1CF C1(NC(=O)COCCCF)CC2(CCN(C(c3ccsc3C(F)F)=O)C2)C1 C(=O)(C(O)Cc1ccccn1)NCC(CC)NC(c1ncsc1Br)=O CC1CCC(NC(=O)C(C)(C)c2cccs2)CN1C(C1CC(O)CN1C)=O c1(C(=O)NCCC(C)NC(=O)CC2CCCC23CC3)cc2c(s1)CC(C)(C)C2 CCC1=NOC(C(N2CCC(C(CO)NC(=O)Cn3ncccc3=O)CC2)=O)C1 C1(CONC(CCC2C(C)(C)C2)=O)CC(C(=O)NC(C2(C)CCCC2)=O)=NO1 C(=O)(C(C(C)C)n1cccc1)N(C1(CC(=O)NC2(CC)CC2)CC1)C N1(C(c2n(C=C)ncc2)=O)CC2CCN(C(=O)C(O)(C=C)c3ccccc3)CCC2C1 N1(C(CCOCCC)=O)CC(F)CC1C(=O)N(C1CC(O)C1)C C1(CC(=O)NCCN(C(C)C)C)CCCN(C(c2cn(C)nn2)=O)C1 N(C(=NCCn1cccn1)NCC(C)(C)C)C(C1(O)CCOCC1)(C)C1CC1 N1(C2CN(C(C(CC3CC3)OC)=O)C2)CC(NC(=O)C=CC(=O)NC)CC1=O C1(CC(NOCC=C(C)C)=O)CCCCN1C(=O)CC(C)n1cccn1 c1(CN(C(c2coc(Br)n2)C(=O)NCC2CCOC2)C)ccccc1Cl C12(C(N3CC(C)(C)C(NC(=O)C(O)C4CC4)C3)=O)CC(CO)(C1)OC21COC1 c1(CN2CCC(C#N)(Nc3ncc(F)cn3)C2)ccc2[nH]ccc2c1 Cc1sc(O)nc1C(=O)NCC(C(=O)NC(C)CN1CCCCC1)N(C)C N1(C(C2CC3(CC3)CO2)=O)CCc2nc(O)cc(C(N3CCOC4CC34)=O)c2C1 CCC(C(C)(C)C#N)NC(=O)NC(c1nnc2n1CCC2)C CCCC(C)(CCC)C(=O)N1CCC(O)C(NC(=O)CCc2ccsc2)C1 C(=O)(C#CC1CCCCC1)N1CC(OC)C(NC(=O)C(C)C(F)(F)F)C1 O=c1c(I)cn(CN2CCC(F)(F)C(F)C2)c2ccccc12 Cc1ccc(O)c(NC(=O)CC(C)CNC(=O)C(C2CCCCC2)=O)c1 c1(C(=O)NCC2CCCCN(C(C3C(C)C3)=O)C2)cc2c(F)cc(F)cc2o1 C1(C(=O)N)CC(CC(=O)NCC)C1.C1(C(=O)N(CC(C)OC)CCN(C)C)(CO)CC1 c1(C(=O)NC(C)CNC(c2c[nH]c(C#N)c2)=O)ncc(Br)cc1C(F)F N1(C(C2C3CCCCCC23)=O)CCN(C(C2CC3CCC3C2)=O)C2(CC2)C1 c1(CN2C(c3n(C)ncc3)COCC2)cn(C)c(=O)c2cnccc12 c1(CC)cccc(C(=O)NC2(CC(=O)NCC(O)C(F)(F)F)CC2)n1 c1(NC(C2CCCCN(C(C(C)(O)C3CC3)=O)C2)=O)ccc2c(c1)OCC2 c1(NC(C2CC(NC(c3ccc(O)nc3Cl)=O)C2)C)cc(O)nc(=O)n1C N1(C(C(C#N)C2CC2)=O)CCS(=O)(=O)C(CCNC(c2cnc(C3CC3)[nH]2)=O)C1 N1(C(c2cnc(OC)s2)=O)CC2(CC2)CC1CNC(=O)CC1CCN(C)C1 C(C1c2ccccc2CCN1C(c1ccc(Cl)o1)=O)NC(COC)=O [N-]=[N+]=NCCCC(=O)N1CCN(C(=O)CNC(=O)CSc2nncs2)CC1 C1(C(=O)NCCN(CCOC)C(C2Cc3nncn3C2)=O)CCCC1P(C)(C)=O N1(C(c2occ(C)c2C)=O)CCC2CCC(NC(=O)C(C)(C)C(F)F)C1C2 Cc1n[nH]cc1C=CC(N1CCC(C)(NC(c2ccncc2F)=O)C1)=O C1(C)(C(=O)NCC2(C(C)NC(c3c(C)cc(C)nc3)=O)CC2)CCCCC1(F)F N1(C(c2cc(C(C)C)[nH]n2)=O)CC2CCC1CC2NC(=O)CCn1ccnc1 CS(=O)C=CC(=O)NC1CCC1NC(c1c[nH]nc1-n1cnnn1)=O C(=O)(CCCCCN(C)C(=O)NC1CC1C(C)(C)C)N(CC(C)(C)O)CCC c1(C(=O)NC2(CNC(C3CC(CC)(CC)C3)=O)CCCC2)cc(O)nn1C c1(C(=O)NC(C2CC(NC(CC(=O)OC)=O)C2)C)cc2c(nn1)CCC2 N1(C(C2CCCN(CC(C)C)C2)=O)CC2(C1)SCCC2NC(=O)CNC(N)=O N1(C(C(C=C=C)C)=O)CC2CC(NC(=O)CC3(O)CCCCC3)C(C2)C1 c1(C(N2CCCC(CCNC(CCCCOC)=O)CC2)=O)cc2cccnn2c1 N1(C(CCC=C=C)=O)CC(C(=O)NCCC(O)C(C)CC)CC1(C)C C1(C(=O)NCC2(CC)CCC2)CN(C(=O)C2=CCCSC2)CC12CC2 c1(NCC2C(C)OCC2)cc(F)c(C(=O)O)cc1Cl S(=O)(=O)(CC(=O)N1CCCC(NC(=O)C(F)C2CCCC2)C1)N(C)C N1(C(Cc2cccc(OCC)n2)=O)CCC(C)(C)C1CNC(=O)C#CC(=O)NC c1(CCNC(C2CCC(NCc3csc(Br)n3)C2)=O)ccccn1 CC1(C)CC(CNC(C2CSCCS2)=O)N(C(c2ccc(=O)n(C3CC3)c2)=O)C1 CC(C)CCCCC(=O)N1CC(C(C)NC(=O)Cc2cncc(O)c2)C1 c1(-c2nnc(C)o2)cccc(C(=O)NC2CN(C(c3occc3C)=O)CC2C)c1 N1(C(c2cc(C)c(F)nc2)=O)CCC=C(C(=O)Nc2ccc3c(c2)CCC3)C1 c1(NC(C2CCC(CCNC(=O)CCc3ccco3)C2)=O)ccc(O)c(Br)c1 C1(C(=O)NC2CCC2NC(c2ccc(-c3ccccc3)[nH]2)=O)(OC)CCCCC1 C1(NC(Cn2c(=N)nc[nH]2)=O)CC=C(C(=O)NC2CCCN(C3CC3)C2)C1 c1(C(N(C2CCN(C(c3sc(COC)nc3C)=O)C2)CC)=O)cc(C)cc(F)c1 N1(C(C(C)n2cccn2)=O)CCn2nc(CC(N3CC4CCC(C3)O4)=O)nc2C1 C(CCCC(C)(C)NC(=O)CCc1ccccc1)NC(Cc1nc(C)c(C)[nH]1)=O C(c1cnc(O)nc1O)=CC(=O)NC1CN(C(CN(C)CC)=O)C(C)C1 c1(C(=O)NC2CN(C(CCNC(=O)NC)=O)C3C2C3)cccc2c1OCC2 C1(C(=O)NC(CNC(C2N(CCCC)CCCC2)=O)CO)CCC2(CC1)CC2 CN1CCN(S(=O)(=O)CC(=O)NC2CC2CNC(C2C3CC4C(C3)C24)=O)CC1 c1(CCNC(N(CC(F)F)CCC)=O)c(F)cccc1Cl C(=O)(CS(=O)C(F)(F)F)N1C2CN(C(C=NOC)=O)C(C2)C1 c1(NC(C2(C)COC2)=O)ccc2c(C(N3CCC4CCCC4CC3)=O)ncn2c1 CC(C)(C)C(CNC(c1ccn(C(F)F)n1)=O)C(=O)NC(CO)C(N)=O Cc1nc(CCCC(=O)NC(c2cn(C(c3ccccc3)C)nn2)(C)C)cs1 Cn1nccc1C(O)C(=O)N1CCC1CNC(=O)CCCNC(N)=O C12(OC)CCC(C(=O)NC3CCC(C(=O)NC4CC(CC(N)=O)C4)C3)(CC1)C2 C(=O)(CCC(C)CC)NCC(c1ccccc1)CNC(C(C#C)(C)C)=O CC1(C)CC(NC(=O)CC2(NC(=O)CC3(C)CCOCC3)CC2)CCO1 CC1CCCC(O)C1.C1(=O)CC(C)N1C.C(CCN=[N+]=[N-])NC(C)=O C=CC1(CC(=O)N(C(C)CNC(c2cc[nH]c2-c2ccccc2)=O)C)CCC1 C1(CCN(C(C(CC)O)=O)C)CCN(C(=O)CC(C)n2cccn2)CC1 N#CC1(C(=O)NC2CCCC(NC(=O)C=Cc3cscn3)C2)CC2CC2C1 CC1CC(NC(c2cnsc2)=O)CN(Cc2cnc(Br)s2)C1 C(=O)(C(CN=[N+]=[N-])NC(C1CN(C2COC2)C1)=O)NCc1ccc(SC)o1 c1(SCC)cn(CC2CCN(C(=O)COC(=O)CCOC3CCOC3)C2)nn1 Cc1noc(C)c1CCCNC(C)(CCC#N)c1nnnn1Cc1ccccc1 Cc1ccc2oc(C(=O)NC3CN(C(=O)COc4ccsn4)CCC3C)cc2c1 c1(OC)ncc(C(N2CC3C(C2)N3C(C2CC3(CC3)CN2C)=O)=O)cc1Cl C1(NC(c2ccc(CO)o2)=O)CC(F)(CO)C1.C1(C(=O)NCC2CCCO2)(CF)CCC1 C1(N(C(C=CCCC(C)C)=O)CCF)CCCN(C(=O)C=Cc2cnc[nH]2)C1 CC(C)(C)C#CC(=O)NCC1CCCCN1C(=O)CCCCCN1CCCC1 N1(C(C(C)Cc2ccccc2)=O)CC2CC2C1CNC(c1ccsn1)=O CCC(F)(F)CC(=O)NCC(CC1CC1)C(N1CCSCCC1C)=O C1(CCNC(C=CCC)=O)CN(C(C2(COC)CCCC2)=O)CC(C)O1 C1(NC(CC2ON=C(C)C2)=O)CC2CCC1N2C(=O)CCC(=O)c1ccc(C)cc1 c1(C(=O)NCC2N(C(CC3C(OC)CC3)=O)CCC2C)ccc2sccc2c1 CC1CC2(CCN(C(=O)C(C3CCN(C(c4cncs4)=O)C3)C)C2)CO1 C(CC(C)(C)NC(=O)C(c1cncn1C)O)NC(CN(C)C(c1ccoc1)=O)=O c1(NC(c2cc(C)oc2Br)=O)cc(Cl)ccc1OCc1ccccc1 c1(-n2cc(C3CCCN(C(C(CC)C(C)O)=O)C3)nn2)cccc2n[nH]cc12 C1(C(=O)NCC(C)(C2CC2)NC(c2cccc(C(F)(F)F)n2)=O)OCCC1(C)C C=CC(CC(=O)N1CC(CNC(C2CCC2)=O)CC1CC)c1ccc(OC)cc1 CC1=C(C(=O)NC(C2CCCCC2)CNC(C2CC3CCC2O3)=O)CCO1 C1(NC(c2ncoc2C2CCC2)=O)CCC2CN(C(c3ccoc3)=O)CC2C1 C1(NC(C(CCC)N(C)C)=O)CCN(C(c2ncoc2C(F)(F)F)=O)CC1O c1(CC(=O)N(CCN(C)C)Cc2ccc(Br)o2)c(F)cccc1C#N C1(CNC(C(c2ccccc2)OC)=O)CC(NC(=O)C)C(O)C1.C1(O)CCCC1 C12(NC(CCS(C)(=O)=O)=O)CCCN(C(c3snc(Cl)c3Cl)=O)CC1C2 N1(C(C2(COC)CC(=O)C2)=O)CC2CC1(C(=O)N(c1cccc(OC)c1)C)C2 C(CCCCN=c1nc2scnc2c(NC2CN3CCC2CC3)[nH]1)N(C)C N1(CC(C(C)(C)O)O)CCCCC12CCC2 n1(CC)ncc2c(C(=O)NCC3CC(NC(C4C(C)C4C)=O)C3)cc(C)nc12 C(C(=O)N1CCC(NC(c2cccc(NC(C)C)c2)=O)C1)(C(C)C)NC(C)=O N1(C(C(C)S(C)(=O)=O)=O)CC(C2CCCN(C(C3CC4(CCC4O)C3)=O)C2)C1 c1(NC(C2CC2NC(C2C(=C)C2)=O)=O)ccccc1NC(C1CCC1)=O C(=O)(CCC(C)(F)F)N(CCCC(=O)NCC(=O)OCCCC)C(C)C c1(CC(C(=O)N(CCCCC=C)C)N)cncc(Br)c1 c1(NC2C(C)NC(=O)CC2)ccc(C#N)c(F)c1C#N c1(CNC2CC(CCS(N)(=O)=O)C2)cc(F)c(Cl)cc1F CC1CN(C)CCN1C(=O)CC1CCC(NC(C2CC3(CCC3)C2)=O)CC1 c1(C(=O)NCCC2(O)CN(C(Cc3c(C)cnn3C)=O)C2)nnc(O)cc1O C1(NC(CC=CC=C)=O)CCCN(C(=O)Cn2cc(Br)c(C(F)(F)F)n2)C1 C#CC1(O)CC(C(N2CCC(C(=O)NCCc3cnccc3C)(CC)C2)=O)C1 c1(N)cccc2cnccc12.N(C(=NCc1cccs1)NC1CCOC1)CCOCC c1(COC)ccc(NC(=O)NC(CCF)C(=O)OC)cc1 C1(NC(=O)C=C2CN3CCC2CC3)CC2(CCCN(C(=O)CSc3nncs3)C2)C1 CC1CNc2ccc(C(=O)NCCCNC(=O)Cc3ccon3)cc21 C1(C(=O)NCC(CC)NC(c2ccn(C)c2)=O)CCC2(CCOCC2)CO1 c1(C(N2CC(CNC(c3cc(C(C)=O)on3)=O)C2)=O)cc2scc(Cl)c2[nH]1 c1(OC)ccc(CN2C(=O)NC(c3ccc(C4CC4)s3)C2=O)c(C(=O)OC)c1Cl c1(-c2cn(CCC(=O)N(C)C)nn2)ccc(N(CC(=O)NCCO)S(C)(=O)=O)cc1 c1(C(N2C(CNC(C3C(OC)(OC)CC3)=O)CCC2)=O)csc2cncn12 C=CCCCCCCC(=O)N1CCN(CCNC(=O)C(C)(C)OCC)CC1 c1(CC(N2CC(CC(C)NC(c3ccc(Cl)o3)=O)C2)=O)c[nH]c2ncccc12 C1(NC(CSCCOC)=O)CCCC1NC(=O)CCNS(=O)(=O)CC Cc1cc(C(=O)N(CCC(=O)NC(C2CSC2)C)CCCO)c(O)nn1 c1(CN(c2ncc(OCC)cn2)C2CCCNC2)cc(C)nc(C)c1 c1(OCC)cccc(NC(C)CN(C)C(c2ccc3cncn3c2)=O)c1[N+](=O)[O-] c1(C(N(C)C)=O)ccc(NC(=O)C(N)Cc2ccc(Cl)cn2)cc1Cl c1(OC)c(-c2cn(CC(=O)NC3CCCCO3)nn2)cnn1C C(=O)(CCC(C)C(C)(c1ccc(F)cc1)NC(CC1OCCO1)CO)OC c1(C(=O)NCC2(CNC(C(C3CC3C)OC)=O)CC2)noc(CC2CC2)n1 c1(C(N(CC(CNC(Cc2cccc(OCC)c2)=O)O)C)=O)cccc(F)c1C Cc1nn(-c2ccccc2)cc1-c1nc(CO)nn1CC(c1ccccc1)(C)C C(C)(C)(C(=O)NC1CC1CNC(=O)CCN1CCCCC1)NC(=O)OC c1(C(N2CC(CC)C(NC(C3CCCC3O)=O)CC2)=O)cnc2cc(C)nn2c1 CN1CC=C(CC(=O)NC2CN(C(c3cc(O)ncn3)=O)C3CC23)CC1 C(=O)(C(C)CC(F)F)N1CC(C(C)NC(CCc2cc(C)sc2C)=O)C1 Cc1cc2[nH]c(C(N3CCC4(CC4NC(=O)CNC(=O)C4CC4)C3)=O)cc2o1 Cc1ccc2cc(C(=O)NC3C4CC3N(C(C3CC5(CC5)CO3)=O)C4)cn2c1 C1(C(N2C3CC(NC(=O)CN4CCS(=O)CC4)(C3)C2)=O)CCCCC1(F)F N1(C(CCC2C(C)=NNC2=O)=O)CCC2(C1)CN(C(=O)C1=CCOCC1)C2 c1(OC)cccc(S(=O)CC(=O)N2CC(OC(=O)CCC3CCC3)CC(F)C2)c1 C(=O)(C1=Cc2ccccc2C1)NC(C1CC=CCC1)C(=O)NCCC(C(C)C)OC c1(C(N2CC(CC)N(C(=O)CC3CCCC3O)CC2)=O)ccc2ncn(C)c2n1 N1(C(CC2(C(=O)OC)CC2)=O)CCC2CCN(C(=O)C(C)CC(C)(C)C)CC12 Cn1ccc2cccc(CNc3cnc(F)cc3C(=O)NCCF)c12 C(=O)(C(CC(F)F)NC(c1ccc(Cl)cc1)=O)N(CC(C)S(N)(=O)=O)C N1(C(c2onc(C)n2)=O)CC(NC(C2CCn3ccnc3C2)=O)C2CCCCC12 Cc1cnc(CNC2CC(C(=O)NCC3CCCO3)C2)cn1 N1(CCOC)CCC(COC(=O)CN2CCC(OC(C)C)C2)CC1 CCCC(C)CCCC(=O)N1CCCC1C(C)NC(=O)C(F)(F)c1nc(C)cs1 C1(OC)CCCCC1NC(C1C2CC1N(C(=O)C(C1CCCCC1)C)C2)=O Cc1ccc(C(=O)N(CC(O)CN(C(=O)CC(C2CC2)C2CC2)C)C)cc1Cl CCC(O)CC(=O)N1CCCC(CCNC(c2cc(C(N)=O)co2)=O)C1 C=CC(C)CCN=c1ccnc(NCC2CCCC(F)(F)C2)[nH]1 N1(C(c2c(CNC(C(C(C)C)SC)=O)n[nH]c2)=O)C2CCC1CN(C)CC2 C(=O)(C(C(C)O)N(C)C)NC1CC(C(C)NC(c2c(C(C)C)noc2)=O)C1 c1(CCC)nc(=NC(C)C2CCN(C(c3cn(C)nc3COC)=O)C2)s[nH]1 C1(NC(CC(COC)COC)=O)CC2CCCC(C1)N2C(=O)CC(C)OC C1(NC(Cc2n(C)nc(C3CC3)n2)=O)COCCN(c2ncnc(O)c2Br)C1 N#Cc1ccncc1C(N1CCC(NC(c2cc(Cl)ccc2Br)=O)C(O)C1)=O N1(C(C(=O)NCC)C2CN(C(=O)OC(C)(C)C)C2)CCC(O)(CNC(C)=O)C1 C(C(C)(O)CNC(c1coc(-c2ccsc2)c1)=O)NC(COC(C)C)=O c1(N2CCC(N(C(c3nc(C)sc3C)=O)CC)C2)ccc(C#N)c(C(F)(F)F)n1 Cc1nc(C(=O)NC2CC(CCNC(c3cc(CCO)on3)=O)C2)co1 C1(CC(=O)NC2(C)CN(C(=O)CC3CC4CC4C3)C2)COc2ccccc2O1 N1(C(c2n[nH]c(C)c2Cl)=O)CCC(NC(=O)C(F)C2CCCC2)C(O)C1 N1(C(C2(CCC)CCC2)=O)CC2C(NC(=O)CCCc3ncc(C)o3)C1C2 CN1CCOC(C(=O)NC23CC(NC(C4(C)C=CCCC4)=O)(C2)C3)C1=O N1(C(CC2(COC)CC2)=O)CCN(C(c2cncc(SC)c2)=O)CC1CCO N1(C(CCc2cc(C)on2)=O)CC2CC(C1)N2C(C1(C)CCCCC1C)=O c1(NCCCN(C)C(c2cc3ncccc3s2)=O)ccccc1[N+](=O)[O-] C1(NC(C)C(=O)NCC2CN(C(C3CCC3)=O)C(C)(C)C2)CCC(F)(F)CC1 N1(CC(=O)NCCCNC)CCOc2ccc(Cl)cc21 C12(C(=O)NC3C=CCN(C(C4C(C(=O)OC)COC4)=O)C3)CC=CC(C1)OC2 C(=O)(CCCCCSC)N1C(COC)(CNC(C2(CO)CCCO2)=O)CCC1 N1(C(C2N=C(C)SC2)=O)CCOC2(CCC(NC(C3CCC(=O)N3C)=O)CC2)C1 CC1Cc2ccccc2N1C(c1ccc2nccn2c1)C(=O)NCC1CCCO1 c1(C(N2CCC(CN(C(=O)C(F)C3CCC3)C)C2)=O)ncc(F)cc1F c1(C(=O)NC2CCCN(C(=O)CC3CC=CCC3)CC2)cccc2c[nH]nc12 c1(C(=O)NC2CN(C(C3C(C(C)O)C3)=O)C2)cccc(C(N)=O)c1 N=c1ccc(CCC(N2CCC(C3CCN(C(=O)C=CCO)CC3)C2)=O)c[nH]1 N1(C(CCC2CCCCN(C(CC=C)=O)C2)=O)CCC2(CNC(=O)O2)C1 C(c1ccc(F)c(F)c1)=CC(=O)NCCCN(C)C(C1CCCC(C)(C)C1)=O CN1CC2(CN(C(=O)C(C3CCN(C(C4CCC4Cl)=O)C3)F)CCO2)C1 S1(=O)(=O)c2ccc(cc2Cl)CN1.CC1CC(C)N(CCN(C)C2CC2)C1 CCC(C)C(=O)NCC(N1CCCC1C(=O)N(C1CC1)Cc1nnn(C)n1)=O N1(C(CC(CC)Cc2ccccc2)=O)CC2CCCC2C1CNC(=O)C(N)=O c1(CN2CCN(C(c3c(OC)cccn3)=O)C3C2C3)c[nH]c2ccc(Cl)cc12 N1(C(C(C)C#N)=O)CCN(C(c2cn(C(F)F)cn2)=O)CC1CC(F)F Cc1cc(C(=O)NC2CC(NC(=O)CC(F)(F)C(C)C)C2)c2c(c1)CCO2 N1(C(C=CC=CC)=O)C2CCC1C(F)CN(C(=O)C=Cc1ccc(OC)cc1)CC2 CC1(C)CC(=O)NC1CC(=O)C1CC1.C12CCC(C(O)C1)NC2=O N1(C(CCc2cnc(C)s2)=O)CCCC2C1CCCN2C(=O)CN(C)C1CC1 C(=O)(C(C)(C)CN(C)C(c1occc1C1CC1)=O)NCC(C#C)CC N1(C(CC=CC)=O)CC2(CCCC(CNC(=O)C=Cc3sccc3C)O2)C1 Cc1cc(C(=O)NC2CC(C)N(C(C3CC4(CC4)CO3)=O)C2)c(O)cc1F C(CN=c1cc(C2CC2)nc(C2CC2)[nH]1)=CC(=O)NCc1coc(CF)n1 C1(CC(=O)NCC2CC(C(=O)NCC#CC(F)(F)F)C2)CCC2(CC1)CC2 c1(C(=O)NCC2(F)CCN(C(=O)Cc3ccoc3)C2)cc2c(cc1Cl)NCC2 C1(C(N(CC(CC)NC(c2c(C)ncn2O)=O)C)=O)CCC(C)(C)C1 c1(C(N2CC(C)CC(C)C2)C(=O)NC2(C)CC2)cc(Cl)c2c(c1)OCCO2 S(=O)(=O)(c1cccc(N(C)CCOCCOCC)c1)N1C(CCCC)CCC1 Cn1cncc(C(N2CC(O)(CNC(C3CCCCC3O)=O)C2)=O)c1=O Cc1c(C(=O)NC2C=CCN(C(c3c(Cl)nsc3Cl)=O)C2)ccc2[nH]ccc12 CC1(C(=O)NC2CC(NC(C3CS(=O)(=O)CCO3)=O)C2)CCCNS1(=O)=O C1(CC=C)(NC(=O)Cc2ccn(CC(F)(F)F)n2)CN(C(=O)C(F)OC)C1 C1(C(=O)NC(C)CC2CCC2)CC2(CC(NC(C3CC(O)C3)=O)C2)C1 c1(C(N2CCC(OCCNC(CCNC=O)=O)C2)=O)cnc2ccccc2c1 C(=O)(C(C)(C)N(C)C(C)C)NCCC(C)NC(=O)NC.C(N)(=O)OCC CCC(C)C(O)C(=O)NCC1CC2(C1)CN(C(=O)Cc1cncn1C)C2 CCS(=O)(=O)c1cccc(C(=O)NC2COC3CN(C(=O)CO)CC23)c1 CCC(F)(F)C(=O)NCC(C)(F)CNC(c1cc(C)no1)=O c1(C(=O)NCc2ccc(C(=O)NCC(CC)C)nc2)ccc(F)c(C)c1 C1(NC(C=CCC)=O)CCC(CNC(=O)C(CC)NC(C)=O)C1 N1(C(CN2C(=O)CCC2)=O)CC2COCC(C1)C2NC(=O)C(F)CC1CCCC1 CCCC(C)(CC)C(=O)NC1CC2CN(C(=O)C=Cc3ccncc3)CC2C1 c1(C(=O)OC)oc(C(=O)NCCCNC(=O)CC(C)(C)O)cc1C N1(C(c2[nH]ccc(=N)n2)=O)C2CCC1CN(C(=O)C=CCN1CCCC1)CC2 N#Cc1ccc(O)c(NC(c2ncoc2CCNC(=O)C(F)OC(F)(F)F)=O)c1 c1(NCc2cccc(C(=O)NCC3C(CO)C3(F)F)c2)cc2cc(F)ccc2o1 N1(C(C2C(OC)C2)=O)CCN(CC(=O)Nc2ccc(OC)cc2Br)C(=O)C1 c1(COCC(=O)NCC(F)(F)F)cn2cc(Cl)cc(Cl)c2n1 C1(C(=O)NCCCN2CCCC2)C=CCN(C(=O)CC23CCCC2C3)C1 c1(CC(=O)OC)ccc(Br)cc1C.C1(=O)C(OC)O1 C1(NC(c2n(C(CC)C)ncc2)=O)CC12CCN(C(c1n[nH]c(C)c1Cl)=O)CC2 N1(C(C(c2ccc(C)s2)C)=O)CC2C3CCC(C2C1)N(C(=O)CN(C)C)C3 c1(C(=O)NC(CN(C(c2c(C)n(C)nn2)=O)C)C)cc(O)c2sccc2c1 [N-]=[N+]=NC1CC(CN(c2cccc(F)c2)N2CCCC2C=O)C1.N1(CC2CC2)CCCC1 N1(C(C(C)CC(N)=O)=O)CC(C)(C)OCC1CNC(=O)CC1CCSCC1 C1(CC(=O)N(CC(C)CNC(C2CC(N3CCCCC3)C2)=O)C)CCCC12CC2 C1(CC)CN(C(c2csc(C3CCCN3C(=O)CCCF)c2)=O)CCO1 C1(CNC(Cc2ccc(C)s2)=O)(NC(=O)COC2CCN(C)CC2)CCOCC1 c1(SCC(N2CC(N(C)C(C3(F)CCOC3)=O)C2)=O)ccc(F)cc1 C1(C(N(C)CC)NCc2cc(-c3cccnc3)no2)CN(CC)C(=O)O1 c1(CCC(N2CC(CNC(c3cnc(C)s3)=O)C3C2C3)=O)cccc([N+](=O)[O-])c1 C1(CNC(c2ccc(CC)s2)=O)C2CN(C(C3CCC3(C)C)=O)CC12 c1(C(N(C2CC(NC(=O)COCP(C)(C)=O)C2)C)=O)c[nH]c2ccc(Cl)cc12 N1(C(C(CC)N(CC)CC)=O)CCCC12CCN(C(=O)C(C)(C)CC(C)C)C2 c1(OC(C(=O)NC(C)CCNC(c2c[nH]c(C(F)(F)F)c2)=O)C)cccnc1 c1(NC(c2onc(-c3cccc(OC)c3)n2)=O)cccc2c1OCC2 N1(C(n2cc(C=O)nn2)=O)CCc2cc(CN3CC4CC4C3)ccc21.CC(F)(F)C1CC1 CCCC(C(=O)NC1(CCOC)CCN(C(=O)CCOCC(C)C)C1)OC C1(C(C)(C)C)CC(C(=O)N(C2CCCN(C(C3CSCCS3)=O)C2)CCO)=NO1 C1(N(C(c2ccccn2)=O)Cc2c(C)cccc2)CCCN(C(=O)C(C)C)CC1 c1(C(N2CCC(NC(c3cncc(Br)c3)=O)C2)=O)c(Br)ccc2c1OCO2 CC1(C)CC(C)(CNC(C2C(C)(C)C2(F)F)=O)CN1C(C1CC2CCC1CC2)=O n1(CCC)ncc(C(=O)NC2CC2NC(=O)C(c2ccc(N(C)C)cc2)C)c1C N1(C(CCCOC)=O)CC(C)(C)OCC1CNC(=O)CCN(CC(F)(F)F)C CC(CO)C(=O)NC1CC(NC(C2CC(CCNC(=O)OC(C)(C)C)C2)=O)C1 C1(CNC(c2ncccc2CO)=O)CC12CCN(C(c1cncc(Cl)c1)=O)CC2 C1(C(N2C(C(=O)OC)CCCC2)=O)CC2(C1)CN(C(=O)Cc1ccc(Br)cn1)C2 c1(C(N(CC(C)(C)CNC(C2CSCCS2)=O)C)=O)cn(C)nc1C1CC1 C=C(C)CC(C(=O)NCC1(C(=O)N(C)CC2CCCS2)CCCC1)OC C(=O)(CCCCCF)NCC(C(C)(C)C)NC(c1ccc(C(=O)NC)nc1)=O N1(C(c2cccc(OC)n2)=O)C2CCC1CC(O)(CNC(C1CCSCC1)=O)C2 C12(NC(=O)OC(C)(C)C)CC(CNC3CCCC(C(F)F)CC3)(C1)OC2(C)C C(C1CCCCC1)=CC(=O)NCCC1CCC(C)(C)C1.C1(OC)CC2N(C1)C2=O C(CO)(CCC(C)C)C(C1CC1)NC(N1CC(c2ccc(C)o2)OCC1)=O N1(C(C(CC=CCC)C)=O)C2CCC1C(F)C(NC(C1CN(C)CCN1C)=O)C2 c1(OC)cc2[nH]cnc2cc1NC(c1cc(I)c(Br)cc1Cl)=O N1(C(c2nc(C)[nH]n2)=O)CCN(C(c2ncn(-c3ccccc3)n2)=O)CC1CF c1(NCc2ccccc2C(N2CCC(C)C2)C(=O)OC)c(C)cc(C)cc1C C1(C(N2CCC(=C)CC2)=O)C2CCCC1CN(Cc1ccncc1C(F)(F)F)C2 N1(CCC)CC(C(N2CCOC(C3CN(C(=O)CNC(=O)CC)C3)C2)=O)CC1=O N1(C(CC(CC)C)=O)CCCOC(CNC(=O)CCc2ccccc2OC)C1 c1(SC)nc(O)c(C(=O)NCC2CN(C(c3cc(Cl)c[nH]3)=O)CCO2)cc1C#N c1(C(=O)OC)cn(CC(=O)N(C)CCN(C)C(c2ccsc2SC(C)C)=O)nn1 N1(C(C2C(SCCOCCOC)CCC2)=O)CC(c2ccccc2)OC(C)(C)C1 N1(C(c2cc(C3CC3)no2)C(=O)NCc2cccc(OC)c2)CCC(C)C(C)(C)C1 c1(C(N(CCN(C(=O)C(O)CC2CCOCC2)C(C)C)C)=O)cncc(C#N)c1 c1(C2C(C(=O)NC(C)CN(C(=O)C=CSc3nc[nH]n3)C)C2)cc(Cl)cn1C Cc1ccc2sc(N3CC4CCCC(NC(C5CCC=CO5)=O)C4C3)nc2c1 c1(C(=O)NC2CN(C(C3(C(=O)NC)CC3)=O)C(C)(C)C2)n[nH]c2ccc(F)cc12 C1(NC(=O)CC2CSC2)CCCCC1NC(C1C2CCC1(c1ccco1)C2)=O S(=O)(=O)(c1ccc(N(C)Cc2cccc(-c3ncco3)c2)cc1)NC C1(C)(CNC(CSCC=C)=O)CCC(NC(=O)C(c2cccc(Cl)c2)O)CC1 C1(COC)CN(C(c2ccc(N3CCCC3)cn2)=O)CCC1(F)F N1(C(c2ccc(CC)s2)C(=O)NC(C)(C)CC)CCC2(CC1)C(F)(F)C21CCC1 c1(OC)ccc(CC(=O)NCCCC2CCN(C(=O)C(=O)N)C2)nc1.C(F)F N1(C(C2C(CCC)CCC2)=O)CCC2CN(C(C)=O)CC2CC1 CC(C(C)(C)NC(c1csc(O)n1)=O)NC(=O)C=Cc1ccco1 C12(C(=O)NC(C3(O)CCN(C(C(CCC)NC(N)=O)=O)C3)C)CC1COC2(C)C C(C(C(C)(C)C)NC(=O)CCCF)N(C(CCN(CCCCC)C(C)C)=O)C N1(C(CN2CC(C)(OC)C2)=O)CC2(NC(=O)C(C(C)C)NC(N)=O)CC1C2 N1(c2nnc(C)s2)CCc2c(c(CNC(=O)C(F)F)nn2C)C1 CCC(CC(F)F)C(=O)NCCC1CN(C(=O)C(C)Sc2ccc(Cl)cc2)C1 CN1CCOCC1C(=O)NCC1OCCC1C(N1CC(C)(C)C1C1CC1)=O C=C=CCC(=O)N(C1CCC(C(=O)N(C2CCOC2)C)C1)C1CC1.CC(C1CC1)C1CC1 CCC(O)C(C)C(=O)NC(C)(CC)CCNC(=O)Cc1ccc(OC)nc1 CN1CCN(C(C2CC(F)C(=O)N2)=O)C(C(=O)NCc2cscn2)C1 CC1OC2(C(=O)NCCCOCCNC(=O)CCCCN(C)C)CCC1CC2 c1(OC)cc(NC(=O)C(N2CC(OC)CC2C)=O)cc([N+](=O)[O-])c1 C(=O)(C=CS(C)(=O)=O)N1C(C)CC(NC(c2ccc(CC)[nH]2)=O)C1 C(=O)(CC1OCc2ccccc21)NCC1CCN(C(C(C)(C)O)=O)C1 C#Cc1nccnc1NC(=O)CC(c1ccc(F)cc1)NC(=O)C(C)CC C(=O)(C(CC(C)(C)C)NC(=O)CCc1ncccn1)NC(c1csnn1)C O=C1CC(CC(=O)NC2C=CC(CC(=O)NCC(F)(F)C(F)F)C2)C(=O)N1 c1(C(C)C(=O)N(C(C(=O)O)C2CC2)C)cccc(Br)c1 Cc1cccnc1C(=O)NC(C(=O)NCC1CCC(C)(C)O1)C1(O)CCC1 C1(C(=O)NCC=CCNC(C2CC(C)(C)C2)=O)C2CCC1(c1cnco1)C2 C(=O)(C#CC1CCCO1)N1CCC(CNC(c2ccc(OC)cc2C)=O)(OC)C1 N1(C(c2cn(CCF)nn2)=O)CCCC(C2CCCN2C(=O)CCC(F)F)C1 C(=O)(C(O)C(F)(F)F)NC(C)CC1CN(C(C2CCC(O)C2)=O)C1 c1(C(C)C(=O)NC2CC(N(C)C(C3C4COCC34)=O)C2)ccc(F)c(Cl)c1 Clc1nc2cc[nH]c2c(=NCCC2CN(c3ncccn3)C2)[nH]1 C1(C)(CC(N2CC(NC(C=CCCC)=O)(COC)C2)=O)CCCCC1 Cc1nc(C)c(C(=O)NC2C3CCC2N(C(c2c(C)noc2C)=O)C3)c(C)n1 N1(C(c2ccc(CNC(C=CC)=O)s2)=O)CCN(c2cccc(Cl)c2)CC1 c1(N(C(C(=O)N2CCC2NC(=O)CCNC(N)=O)C2CCC2)C)cccnc1 N1(C(c2cc(C)sc2C)C(=O)NC)CCN(c2cncc(F)c2)CC1C c1(C(N(C)CC2(CNC(=O)Cc3csnn3)CC2)=O)ncsc1S(N)(=O)=O c1(C(=O)ON)cnc2[nH]cnc(N3CC4CC(C3)N(Cc3ccccc3)C4)c1-2 C1(COC)CCCN(C(C2CN(C(=O)CCCNC(C)=O)CCO2)=O)CC1 C1(C(N(C)Cc2cc(Cl)no2)=O)COCCC1NC(=O)CCc1ccn(C)n1 C1(C)(CNC(CN(C2CC2)CC)=O)CCN(CCCC2(C)CC2)CC1 N1(C(C(CC)C)=O)CCC(C(=O)N(C)CCNC(c2nc(Cl)cs2)=O)CC1 CC1CCN(C(c2cn[nH]c2)=O)CC1N(C)C(c1cc(C(N)=O)ccn1)=O C(=O)(C(C)(C)C(=O)NC1CCCC(NC(=O)CSCc2ccc(Cl)cc2)C1)OC C(CC(=O)NCC1CN(C(c2cc(N)ccc2F)=O)C2CC12)(C(F)(F)F)OC CN1CCC(NC(c2cc[n+]([O-])cc2)=O)C12CCCN(C(=O)C(C#N)=CC(N)=O)C2 Cc1ncc2n1CC(NC(C1CC3CCC(C1)N3C(c1ccccc1)=O)=O)CC2 c1(N(C)Cc2ccncn2)ccncc1S(=O)(=O)NCC12CC1Cc1c[nH]nc12 C1(O)(CCNC(C2(CC#C)CCCC2)=O)CCN(C(=O)CCNS(C)(=O)=O)CC1 C1(C(=O)NC2C(N(C)C)COC2)COC(C)(C)CN1 C1(C(N2C(C)(C(=O)NC)CC2)=O)CCC(CNC(=O)CC2(NC(C)=O)CC2)CC1 C1(CC(=O)OC)CCCN1C(=O)C(c1ccnn1C)NC(=O)Cn1cnnc1 c1(OC)ccc(C(=O)NC2CC(C(=O)Nc3c(F)cccc3Br)C2)c(Cl)c1 Cc1cncc(C(N2CCC(CO)(CNC(=O)CCN3CCC3)C2)=O)n1 N1(C(C2CCCN(CCC)C2)=O)CCC2CC1CN2C(C1CC(=O)NC(=O)N1)=O C1(OCCC)CCCN(C(=O)C(N2CCOC(c3ccccc3Br)C2)=O)C1 CC1(C)C2CCC(CC(=O)NCC34CC(CN3C(C3CN5CCC3C5)=O)C4)C1C2 C1(NC(CC2(C=C)CCOCC2)=O)C2CCN(C(c3cnsc3C)=O)CCC12 C(=O)(C1=CCCC1(C)C)N1CC(NC(c2cnc(C)n2C(F)F)=O)C(C)CC1 N1(C(C(CCCC)N(C)C)=O)CCC2(NC(=O)CC(CC)C3CC3)CCCC12 N1(CC)N=C(C(=O)NC(C)C(C)(C)NC(C2CCn3ncnc3C2)=O)CCC1=O C1(O)(CN(C(=O)CC2CCC2(F)F)C)CCCN(C(=O)CC2(C)CC(F)(F)C2)C1 N1(C(=O)CC2CSCCS2)CCCC2(CCCN2C(=O)COC(F)(F)F)C1 c1(NC(C2C(C(=O)OC)C2)=O)nc(C)c(C(=O)Nc2ncccc2O)s1 C1(NC(CC(C)N(C)C)=O)CCCCC1N=c1cc(Cl)nc(S(C)(=O)=O)[nH]1 O=C(C(CC(F)F)N(C(=O)CC1CCCC12CC2)CC)NCCC1CCCCC1O N1(C(C(C)C2(O)CCC2)=O)CCCC1(C)CNC(C1(C)CCCS1)=O N1(C(C(CC(C)C)N(C)C)=O)CCOCC(C)(CNC(c2ccnnc2O)=O)C1 n1(CC)ncc(C(N2CCC(NC(c3cnc(N4CCCCC4)s3)=O)C2)=O)c1C [N-]=[N+]=NCC(C(=O)NCc1cccnc1)NC(C1CC=CCO1)=O N1(C(c2nc(C)c(C)s2)C(=O)NCc2ccccc2I)CCC(O)C(F)C1 CCC(CC(=O)NCC1CN(C(C2CCCCC2OC)=O)CCC1C)C(C)C N1(C(c2onc(C)n2)=O)CCN(C2CCN(c3cn(C)c(C)n3)C2)CC1 c1(OC)cc(N(C)C)ccc1C(=O)NCC1CN(C(=O)C2=C(C)CCC2)CC1O CN1C(=O)COc2ccc(C(=O)Nc3cccc(-c4cnco4)c3)cc21 N1(C(C)C)C(=O)COCC1C(=O)NC1(C)CCN(C(C2(O)CCOC2)=O)CC1 C1(NC(C2OCCN(CC)C2)=O)CC2CC(NC(c3cc(O)n(C)n3)=O)CC2C1 c1(SC)ccc(CN2CCC(CNCc3sccc3Br)CC2)cc1 C1(C(=O)NC2C(C)(C)C(O)C2)C2CC3C(C2NC(C2C=CCS2)=O)C13 c1(C(=O)NC(CN(C(CCC=CCC=C)=O)C)C)ccc(O)c(C)c1C C1CCCCCC(=O)NCc2cn1nn2.c1(C(C)COCC(=O)O)nccs1 C1(NC(c2cccc(OC)n2)=O)CCN(C(=O)CC2CCN(C)C2)C(C)C1 c1(C(=O)NC(C(C)C)CNC(=O)Cc2cnoc2)cc2cccnc2[nH]1 C1(OC)CCC12CC(C(=O)NCC1C3CN(C(c4cncnc4)=O)CC13)C2 C1(CC(=O)Nc2cn(CCC#C)nc2)CN(C(=O)CCCC(C)=O)C(C)(C)C1 c1(N2CC(C)C(NC(=O)CC(C)(C)C3CC3)CC2)ncnc2ccccc12 c1(C(N(CCCNC(C(C)Cn2ccnc2)=O)C)=O)nc(Cl)c(Cl)s1 N1(C(C)C)CCCC(NC(c2cnc(C3CC3)nc2)c2nnnn2CC2CC2)C1 N1(C(C=CC(CC)=CC)=O)CCC(C)(CNC(=O)C(C)(F)c2ccccc2)C1 C1(C(=O)NCC(C)NC(c2csc(C(F)(F)F)c2)=O)CC(=O)N(C(C)(C)C)C1 c1(CC(=O)N(CC(O)CN(C)C(C2CCCC23CC3)=O)C)csc2nccn12 N#Cc1ccc(NC(=O)NC(=O)NCCOCC2CC2)cc1C(F)(F)F c1(NC2CC(C(N3CC(C(=O)OCC)(CC)C3)=O)C2(C)C)cc(CO)ncn1 c1(CNC2C(C(=O)Nc3c(C)cnc(O)c3)C2)cc2cnccc2[nH]1 C1(C(=O)NCC(c2nncn2C)C)CN(C(C2(C)CCC3CC3C2)=O)CC1(C)C N1(C(C=C(CC)CC)=O)CCC2(NC(c3coc(C(=O)OC)c3)=O)CC2C1 C(COC1CCN(C(=O)C(N(C)C)NC(=O)C2CC2)C1)(CCN(C)C)OC.C1(S)CC1 C=CC(C)(C)CC(=O)N1C2CCC1C(CNC(C1(CO)CCCO1)=O)C2 CCC(C)(C)C(=O)C(=O)N1CCC(C(C)NC(=O)C=CC(=O)N(C)C)CC1 c1(C(N2CCC(CNC(CCCCC#C)=O)(OC)C2)=O)ccc(F)cc1[N+](=O)[O-] c1(SC)cccc(F)c1C(=O)NC1CCC1NC(c1cnc(C)[nH]1)=O c1(OCC)cc(NCC(C2CC2)NC(c2cc(=O)cc[nH]2)=O)nc(C)n1 c1(OCCNC(C2C(c3c(OC)ccc(C)c3)C2)=O)cc(=O)n(C)c(O)n1 c1(C(=O)NC2(CNC(C3ON=C(C)C3C)=O)CC2)cc2c(C)c(F)ccc2[nH]1 N1(c2nnc(C)o2)CCC2(CN(C(=O)Cc3ccc4n[nH]cc4c3)CCO2)C1 c1(COC)cc(C(=O)NC2CCCN(C(=O)CN(C)C(C)=O)C2C)ccc1OC C=CC1(C(=O)NC2CC(Cl)(Cl)C2)CCN(C(=O)CC2(O)CCC2)C1 Cc1nc(C(=O)N(CC(C)CNC(=O)C=Cc2cnc[nH]2)C)nn1C Cc1nc(CO)oc1C(=O)NC1CCC(NC(c2cnn(C(C)(C)C)c2)=O)CC1 c1(CNC2CC(C)CN(C(c3cc(I)ccc3O)=O)C2)cc(O)c(O)c(Cl)c1 Cc1ccc(C#N)cc1C(N1CCC(C(N2CCC(C)CC2C)=O)C12CC2)=O C1(CC(N2C(CN(C)C(c3ccc(-c4ccco4)[nH]3)=O)CCC2)=O)CCC(O)C1 N1(C(C2CC3(C)OCC2C3)=O)CC2CCC(C1)N2C(C1C2CC3C(C2)C13)=O Cc1cc(CC(=O)N(C)C(c2cn(-c3cnnn3C)nn2)C)cc(Br)c1 c1(C(=O)NC2C(OC)CN(C(COC(CC)C)=O)C2)nc2cccnc2s1 c1(CN(C(c2n[nH]cc2Br)C(=O)NCC=C)C)ccc(C(N)=O)cc1OC CCC(C)(O)C(=O)N(CCC(=O)NCc1ccncn1)CCCO C(=O)(C1CC(=O)N(C)c2ccccc21)NCC(c1coc2ccccc12)C(=O)OC C1(F)(CNC(C(C)n2ccnc2)=O)CCN(C(C2CCCO2)=O)CC1 Cn1cc(OCC(=O)N(CC(=O)NCC2C3COCC23)C2CC2)cn1.CCl N1(C(CCN(C(CCC)C)C)=O)CCCC(CO)(CNC(c2cncs2)=O)C1 C1(C)(C(=O)NCCCN(C(=O)C(=Cc2cscn2)F)C(C)C)CC(C2CC2)=NO1 C12(NC(CNC(C)=O)=O)CCOCC1CN(C(c1sc(=N)[nH]c1C)=O)C2 CCCC(C(=O)N(C)CC1CCCCO1)NC(C1(C)CC(C)(C)C1)=O C(CC(C)P(C)(C)=O)NCC1C(C(=O)OC)CCCC1 N1(CC(=O)NCC2N(C(c3cc(C)sc3)=O)CC=C2)C(=O)CN(C)C1=O c1(C(=O)NCC2(F)CC(NC(c3cnc(COC)s3)=O)C2)cc(C#N)no1 c1(SCCC(=O)NCC(C)NC(C(C)n2cncn2)=O)nnnn1C1CC1 C(=O)(CC(CCCCCC1CC1)N1CC(O)CC1C(C)=O)NCCCOC c1(CCC(=O)NCC2N(C(Cc3scc(C)c3)=O)CC2)cccnc1F C1(OC)CC2CC(C1)N(C(C1(C(=O)NCc3cnnc(O)c3)CCC1)=O)C2 c1(C(N2CC(N(C(c3cncc(C)n3)=O)C)C2)=O)c(O)ncc2c1CCC2 N1(C(c2ccc(C)cn2)=O)CCC(NC(c2coc(N(C)C)n2)=O)CC(O)C1 c1(CN(C)C(C2CCS(=O)(=O)N2)=O)ccc(CNC(C2(C)CCC2)=O)cc1 CC(C)C(C(=O)NCC1CCN1C(N)=O)NC(=O)COCCCOC(C)(C)C c1(C(=O)NCC(C)N(C(c2ccco2)=O)CC)cc2c(cc1Cl)OCO2 CCN=c1[nH]cc(C(=O)N(C2CC(NC(=O)CC(C)CNC(C)=O)C2)C)s1 c1(C(=O)NCC(C2CC2)Nc2cc(C(F)(F)F)ncn2)ccc(C2CC2)cn1 CC1CCN(C(c2ncc(F)cc2N)=O)CC1CC(=O)NC1CC1C1CCC1 C(=O)(CCS(=O)(=O)Cc1cccc(C(=O)O)c1)NC(C(CC)O)(F)F Cc1cccc(C(C)NC(C2CCC(C3CC3)N2C(c2nnn(C)c2N)=O)=O)n1 C1(CNC(C2(CC=C)CCCC2)=O)CCCN(C(c2cccnc2F)=O)C1 CC(C(=O)NCC(C)(C)CN(C)C(c1cnn(C)c1-c1cn[nH]c1)=O)C(C)(F)F C1(CNC(C2C(OCC)CC2)=O)CN(C(C2CCC(C)(C)CC2)=O)CC1(C)C C1(CCCNC(C2CC2F)=O)CCN(C(c2ccnn2CC(F)F)=O)CC1 c1(OCC)cc(CNC2CC(NC(C3(F)CC3)=O)C2)ccn1 N1(C(CS(=O)(=O)NCC)=O)CC2CCCC1C2CNC(=O)Cn1cc(Cl)cn1 c1(C(N2CCC2CNC(C23CC4CC2(CO)CC4C3)=O)=O)ccc2cnsc2c1 O(S(=O)(=O)c1ccc(F)cc1)c1ccc(-c2nc(C)c(C(F)(F)F)s2)cc1 CC(C)CC(C(=O)NOC1CCN(C)CC1)N(C(=O)C(C)c1ccsc1)C N1(C(C(CC)CC)=O)CCCC(NC(=O)CC2CC(OC)C2)C(F)C1 C(=O)(CC1COc2ccccc21)N1CC=C(CNC(C23CC(C)C2C3)=O)CC1 C1(NC(C(c2ccccc2)OC)=O)CC(C)(NC(=O)COC(C)=O)C1 N1(C(C(C2CCC2)OC)C(=O)NC2CCCC2)CC(C)Oc2c(Cl)cccc21 CC1(CC(=O)NC2CCCN(C(c3cc(C4CC4)cs3)=O)C2)CCOCC1 S(=O)(=O)(c1cc(Cl)ccc1F)N1C(CNCc2ccc(C(=O)O)cc2)CC(F)C1 C1(NC(CN(C(=O)OC)C)=O)C2CCC(C2)C1C(N1CCCC(N(C)C2CC2)C1)=O N1(C(C=C(C)C(C)C)=O)CCCCC1CNC(=O)C(c1cn(C)cn1)O C1(C(=O)OCC)CCCC(CNC(c2nn(-c3cnn(C)c3)nc2C)=O)C1 c1(C(N2CCC(c3ccc(Br)cn3)C2)C(=O)NCC)ccncc1Cl c1(C(=O)OCC)nn(C)c(NC(C2CCCN(C(=O)Cn3ccnn3)C2)=O)c1Cl Cc1cccc(C(N2CC(NC(c3nnccc3C)=O)C(C)C2)=O)c1Br O=C(CC1=CSC2=NCCN12)N1CCCC(CNC(C2(CO)CC2(F)F)=O)CC1 CC(F)(F)C(C)(C)C(=O)N1CCCC(CCNC(=O)CCCNC(=O)C2CC2)C1 c1(C(=O)NC(CN(C(c2ccc(CSC)o2)=O)C)(C)C)ccc(P(C)(C)=O)nc1 CC1(C)CN(C(=O)CC2CC=CC2)CC2(CN(C(c3cc(O)ccc3Cl)=O)C2)O1 N1(C(c2c(Cl)cn(C)n2)=O)CCC2CN(C(C3CCCC3)=O)CC2C1 C(=O)C(CC(C)C)ONC(c1cncc(C)n1)=O.C(C)(C)(C(C)NC(=O)CO)OC c1(CN2CC(C)C(NC(=O)C(F)(F)F)CC2)ccc2ccsc2c1 C12(NC(c3c(C)nc(C(C)C)s3)=O)CCN(C(=O)C=CCO)CCC1C2 C1(CC(N2C(c3c(C(=O)OC)c[nH]n3)CCCC2)=O)CCCNC(=O)C1 c1(C(N2CC3C(C(=O)NCc4c(C)ccs4)(CCC3)C2)=O)ccc2ccoc2c1 C(=O)(CCC(CC)NC(C1(OC)CCOC1)=O)NC(CC#CC)CC N1(C(c2c(C)ncc(N)c2)=O)CC2CC(NC(c3n[nH]cc3Cl)=O)CC2C1 C12(C(=O)O)CCC(n3cc(CN4CCCC4=O)nn3)(CC1)C2.N#Cc1nc[nH]c1 C1(N(C(c2cc(CC)nn2C)C(=O)NCCCOC)C)CCC2CC1C2(C)C CC1CC(NCC(=O)NC(CN2CCOCC2)C(C)(C)C)c2ncnn21 c1(C(=O)NCCC(C)NC(=O)C=Cc2cc(Br)cs2)cccc(O)c1Cl C1(OC)CCC2(C(=O)N(CCCC(=O)NCc3nc(COC4CC4)n[nH]3)C)CC12 Cc1c(Br)c(C)n(NC(=O)C(C)Oc2cccc(Cl)c2)c(=O)c1C#N C(=O)(CCC(C)(C)[N+](=O)[O-])NCC(CC(C)C)NC(C1(C)CCN(C)C1=O)=O C1(C2C(NC(C3CCN(C)C3)=O)CCO2)CCN(C(=O)Cc2cc[nH]n2)CC1 Cc1nc2cccnn2c1C(=O)NC1CN(C(=O)C#CC(=O)N(C)CN(C)C)C1 c1(NCc2cnc(CC)[nH]c2=N)cc(S(=O)(=O)N2CCCC3CC23)ccc1C#N N1(C(CSC(C)C)=O)CCC(NC(C2CC2(F)F)=O)C1(C)C C1(CNC(C=CCC)=O)CN(C(c2cc(-c3cccs3)on2)=O)C2CC12 C12(C(=O)NCC(CC=C)NC(=O)C3=CC(C)CC3)CCC(C(F)F)(CC1)C2 N1(C(c2cc(CC)n(C)n2)=O)CCCC12CCN(C(=O)Cc1conc1C)C2 C1(C(N2CCC(CN(C(C3(CC=C)CCCCC3)=O)C)C2)=O)CCCCNC1=O Cc1cc(O)nc(CNC(=O)C(CC(C)C)NC(=O)C=C2CCC(C)CC2)n1 C1(CNC(C2(OCCn3cc(NC(=O)C4CC4)nn3)CCC2)=O)CN(OC)CC1C.CO Cc1c(C(=O)NCC2CCCN2C(C2CCC3(C2)N=N3)=O)cccc1[N+](=O)[O-] CCN=c1ccc(C(N2CCOCC(NC(C34CC(CC)(CO3)C4)=O)C2)=O)c[nH]1 CC(C(=O)Nc1ccc2c(Cl)cc(Cl)cc2n1)S(=O)(=O)C1CCOCC1 c1(C(=O)NC2CCC(NC(=O)C(C3(O)CCCC3)F)C2)ccc2c(c1)CCC2 C12(NC(CP(C)(C)=O)=O)CCCCC1CN(C(=O)Cn1nnc(=O)[nH]1)C2 c1(OC)cccc(C(N2CC3C(CNC(=O)C(n4ccnc4C)C)C3C2)=O)c1O c1(C(=O)NC(CC(C)Nc2cc(C(C)C)ncn2)C)ncc([N+](=O)[O-])n1C c1(C(=O)NC2C(NC(CC(=O)OC)=O)CCCC2)c(C)[nH]c2ncccc12 N1(C(C(C2CC2)OCC)=O)CCN(C(c2cc(C)n(CC3CC3)c2C)=O)C2CCC12 CCCCCCC(C)C(=O)NCCc1csc(C=O)c1.C1CCN(C)N1C.C(=O)OC C1(C(N2CC3C(C(=O)NC4CCN(CCC)C4)(C3)C2)=O)CC12CCOCC2 c1cc(=NCc2cn3c(n2)SCC3)[nH]c(NC2COC3(COC3)C2)n1 c1(C(N(CC(CN(C(=O)CC2CCCO2)C)O)C)=O)nnc(O)c2ccccc12 CC(C(C)C(=O)NCC1(O)CN(C(=O)CC2CCC(=O)N2)C1)S(C)(=O)=O C1(CNC(CC=C(C)C)=O)COCCN1C(C1CC2CC2C1)=O n1(CC)ccc2cc(C(=O)NCCCC(C)(C)NC(=O)C(O)CC(C)C)ccc12 CC1(C(N2CCCC(F)(CNC(=O)C(C)(F)c3ccon3)C2)=O)CC2(CCC2)C1 C1(C(=O)NC(C(C)C)(C)CNC(=O)COC(F)(F)F)CCC(C)(F)CC1 c1(C(N2C3CN(Cc4nc(C)sc4C)CC32)=O)cccc([N+](=O)[O-])c1C CN=c1[nH]c(=NCC2CCN(C)CC2)[nH]c(=NC2COc3ccccc32)[nH]1 CC(N=c1cnc(F)c[nH]1)C(c1ccccc1)NC(=O)CCc1c(N)cnn1C c1(N2CC=CC(NC(C(C=CC)O)=O)C2)ncnc2cc(C3CC3)nn12 c1(C(N2CCCCC(N(C(=O)CC3COCCO3)C)C2)=O)ccncc1N=[N+]=[N-] c1(CNCc2ccc(C(c3nnnn3C)OC)cc2)cccc2c1CCC2 Cc1csc(C)c1S(=O)(=O)N1CCC2(CC1)CC2(F)Br CC(C)C(CNC(c1cc(O)n(C)n1)=O)C(=O)NCCC1CCCCO1 c1(C(N2CC(C3CN(C(C(C)N4CCC4)=O)C3)C2)=O)ccc2c(c1)C(C)(C)CO2 N1(C(C2(CC=C)CC2)=O)CCN2CCOCC2(CNC(=O)COCCC)C1 c1(C(=O)NC)cc(NC(N2CC3CSCC3C2)=O)cc(C(=O)OC)c1 c1(C(N2C(CC(C)(C)C)CC2)=O)cc(Br)c2c(c1)OCCCO2 Cc1ccc(C(=O)NCC2CN(C(=O)C=CCO)CC23CC3)c(C)c1Br CCC(C#CC(=O)NCC(S(C)(=O)=O)C1CC1)NC(=O)OC(C)(C)C Cc1cc(Br)cc(S(=O)(=O)N2CCC3(CCN(Cc4c(C)nn(C)c4Cl)C3)C2)c1 N1(C(C(C)S(C)(=O)=O)=O)CCCC12CCN(C(C1CCCS1)=O)C2 Cc1cnc(C(N2CCN(C(=O)COC3CCC3)CC2CC2CC2)=O)cc1C C(c1ccc(C)cc1)=CC(=O)NCC(c1ccc(F)cc1)NC(C(OC)OC)=O CC(C)CC(O)C(=O)N1CC(C)CCC1CNC(=O)CCCc1n[nH]c(=N)s1 C1(NC(c2c(CC)noc2)=O)COC2CN(C(=O)C(C)Cc3ccco3)CC12 N1(C(CN(C)C)=O)CCC(F)C(NC(c2cccc(CN3CCOCC3)c2)=O)C1 c1(C(N(C(CNC(c2c(C)ncn2C)=O)C)C)=O)c(F)ccc2[nH]ccc12 C1(CC(C(=O)NCC2CC2)N(c2ccn(C)n2)CC)CCCC(C)(C)C1 c1(OC)cc(C(N2CC3CC2C(=O)N3)C(=O)NC2(C)CC2)cc(Cl)c1OC C=CCCC(CC(C)C)C(=O)NCC1COC(CNC(C2(COCC)CC2)=O)C1.OCC C1(NC(CC(C)OC)=O)CCN(C(c2cc3n(n2)CCC3)=O)C1(C)C N1(C(C(n2cc(CNC)nn2)C)=O)CCN(Cc2ccc(F)cc2)CC1 CC(CCC(=O)NNc1cc(F)nc(F)c1F)NC(=O)OC(C)(C)C N1(C(C(C2CC2)SC)=O)CC2CC1(CNC(C1(C(=O)N(C)C)CC1)=O)C2 N1(C(C(c2n(C)ncc2)(C)C)=O)CCN(C(C2C(C#N)C2(C)C)=O)CC1 n1(CCC)cc(CN2CC(CC(=O)NC3CCCCO3)C2)cn1 c1(C(N2CC(NC(C(=O)NC)=O)C(c3cncn3C)C2)=O)ccc(OC)cc1Cl c1(CN2C(C(N(CC)Cc3cccnc3)=O)CSCC2)cc(C#N)ccn1 c1(C(=O)NCC2N(C(C3C(OCC)C3)=O)CCCC2)nc(C)ccc1Br CC(C)CC(C)CC(=O)NCCC(C)NC(c1nc2n(c1Br)CCC2)=O c1(C(N2CCCC(NC(c3cccc(C(F)F)c3)=O)C2)=O)cc2sccc2[nH]1 c1(CC)nccn1C(C)CC(=O)NC(C)(C)C(C)NC(C1CC(OC)(OC)C1)=O C(N=c1cc(C(=O)NC)nc(CC)[nH]1)C1CC(NC(c2n(CC)ncc2Cl)=O)C1 C(=O)(N=c1cc(C(C)C)n(C(=O)c2nc(-c3ccc(C)o3)sc2C)[nH]1)OC C12CCN(CC1(F)F)CC(O)c1nc(no1)C2.c1(C(C)(C)C)ncon1 c1(C(N2CCC(CCNC(C(C)OCC#C)=O)CC2)=O)cc([N+](=O)[O-])n[nH]1 Cc1cc(NC(C2CC2NC(=O)CCc2ncc[nH]2)=O)cnc1C c1(N2CC(C)(C)C(NC(=O)C(F)(F)CO)C2)ncc([N+](=O)[O-])cc1Br N1(C(CC2(C)CC2)=O)CC(NC(C2(C)CCCOC2)=O)C2CCCC2C1 CCCCC(O)CC(=O)NC1CCCCCC1C(=O)Nc1cccc(C(N)=O)c1 N1(C(C(CC=CC)NC(c2cc(C)nc(C)n2)=O)=O)CC(F)(F)CCC1C C(=O)(CCCC(=O)N(CC(CO)(CO)NC(=O)C=Cc1ccco1)C)NCC N1(C(C(C)Cn2ccnc2)=O)CC2CCCC2C1C(=O)N(CCCO)CCCO CCC(C)(C)C(O)C(=O)NCC1(C(=O)NCCCC(C)(C)CO)CC12CCC2 C(=O)(CCCC(F)(F)CO)NC1C(C)CN(C(=O)CN(C)C(=O)C2CC2)CC1 c1(N(CCSC)CC)ccc(NCC(O)Cc2cnn(C)c2)cc1[N+](=O)[O-] c1(C(=O)NC(CC#C)CC)coc2c1CN(C(=O)C(F)C(CC)CC)C2 c1(C(=O)NC2CCCN(C(c3c(CC)ccs3)=O)C2CC)c(Cl)ccc(F)c1F c1(N(C)Cc2cnccn2)nc(=NC2CCOC2)[nH]c2ncn(C)c12 CC1=NOC(C(=O)NCC2COCC2NC(=O)C(c2cscc2Br)=O)C1 C(=O)(C(C)(C)CCC#N)NC1C(N(C(c2c(C)ccnc2)=O)C)CCCC1 CC1OC2(C(=O)NC3(c4cccc(F)c4)CC3)CC1(N)C2 Cc1cc2n[nH]cc2cc1-c1c[nH]nc1C(=O)Nc1ccccc1F c1(SC)cccc(C(=O)NCC2(CNC(c3ccc(=N)[nH]c3)=O)CC2(F)F)c1Cl C#CC1(C(N2CCC(CC(C)NC(c3cnn(C(F)F)c3)=O)CC2)=O)CCCC1 n1(CCC(=O)NC2CN(C(C3(C)CCOC3)=O)C2)cc[nH]c(=O)c1=O c1(NC2CN(C(C(C(C)C)CCc3ccccc3)=O)C2)nc2cc(Br)cnc2s1 CC1(C)CC(NC(=O)CC2CCNC2=O)CCN(c2ncnc(Cl)c2Br)C1 CC1CC(C(=O)N(CC(C)CNC(c2ccnc(C(F)(F)F)c2)=O)C)CC(C)O1 c1(C(=O)NC(CCN(C(c2ncc(CC)nc2)=O)C)C)cnn2cc[nH]c(=O)c12 N1(C(=O)OCC(CSc2c(OC)cccc2)O)CCCc2ccc(N(C)C)cc21 c1(C(=O)NCC(CN(C(CC=CCC)=O)C)O)cc2cccc(Cl)c2o1 O=S(=O)(c1ccc(NC2Cc3ccccc3C2O)c(Cl)c1)NC1CCC(O)C1 CN1CC=C(CC(=O)NCC(C(=O)Nc2cccnc2)N(C)C)CC1 C(=O)(C(C)(C)C(=O)N1CCC(C(=O)NC2CCCCC2C(C)C)CC1)OCC C(c1cccc([N+](=O)[O-])c1)=CC(=O)NCC(CNC(c1c(C)nn(C)c1C)=O)F C1(NC(CCCCSC)=O)C2CCCC1CC(NC(c1nnsc1C)=O)C2 C1(NC(C2OCCO2)=O)C2CN(C(c3ccoc3C(n3cncn3)C3CC3)=O)CC12 N1(C(c2c(C)nncc2)=O)CC(NC(=O)CCc2ccc(Cl)cc2)CC(C)C1 C1(CCNC(c2cnncc2O)=O)CCCN(C(C23CCCC(CO2)C3)=O)CC1 C1(NC(C2Cc3nnsc3S2)=O)CCCN(C(C2CCCCC2)=O)CC1 CC(Cc1ccc(Cl)cc1)CC(=O)NC1C=CC(CNC(C23CC(C2)C3)=O)C1.C1(C)CC1 O=C(C#CC1CCC1)NC1CC(F)(CNC(c2n[nH]c(C3CC3)c2Cl)=O)C1 c1(NC(C(COC)NC(c2nc(CC)oc2)=O)=O)ccc2nncn2c1 N1(C(COC)=O)CCN(C2CCCC2CNC(c2cc(C3CC3)cs2)=O)CC1 N1(C(CC2(OC)CCC2)=O)CCCN(C(c2cc(F)c(O)c(F)c2)=O)C(C)C1 c1(CCC(=O)NC2(CNC(C3CC(=C)C3)=O)CCOC2)cncc(Br)c1 N1(C(C(n2cc(C3CCC(=O)CC3)nn2)C)=O)CCC(n2cccn2)(CO)CC1 c1(C(N2CC(F)CC(NC(C3CC(=C)C3)=O)C2)=O)cccc2nonc12 c1(C(=O)NC2C(NC(=O)Cc3cncs3)C2)ccc(Cl)c(Cl)c1 c1(C(N2C(C(C)(C)NC(C(C)OCC(C)C)=O)CCC2)=O)ncnc2c1CCC2 c1(CN=C(NC(CC)CC)NCCC2CS(=O)(=O)C2)cc(F)c(N)cc1F CC(O)(C(=O)N1CCCC1Cc1cn(-c2cncnc2)nn1)C1CCC1 C=CC1(C(=O)N(CC(C)C)CC(C)C)CN(C(C2CCN2C)=O)C1 c1(C(=O)NC2C(OCC)CN(C(=O)CN(C3CCC3)C)C2)cc(C)c(Cl)cn1 Cc1cc(CN(C(=O)C=CC(C)NC(C2(C)CC3CC3C2)=O)C)nn1C CCC(CCOC)C(=O)N1CC=CC(NC(C2(c3ccnn3C)CC2)=O)C1 CCC(C)C(C(=O)NC1CC2(C1)CN(C(c1nccn1C(C)C)=O)C2)OC C1(NC(CC=CC=C)=O)CN(C(C2(C#N)CC(=O)C2)=O)CCC1C(F)(F)F Cc1ccc(F)c(C(N2CC(CNC(=O)C=Cc3cccnc3)C(F)(F)C2)=O)n1 c1(OC)cc(C)ccc1C(N1CC(NC(=O)C=Cc2ccc(Cl)s2)C2CC12)=O C1(NC(CN(C(=O)Cc2cn(C(C)(C)C)nc2C)CC)C)CC2CCC(C1)S2 N1(CCNC(=O)Cc2n[nH]cc2Br)CCN(C(=O)C(N2CCCC2)C2CC2)CC1 c1(CC(=O)NC(C2CN(C(c3occ4c3CCC4)=O)C2)C)cn2c(n1)CCCC2 c1(C(=O)NCCC2CC(OC)CN2C(c2coc(C)c2)=O)ccc(F)c(C)c1F N1(C(C2C(OC(C)(C)C)C2)=O)CCC(C(O)CNC(C2CCOC2)=O)CC1 c1(CCNC(c2cc(O)no2)=O)cc(C(N2CCCC2)=O)no1 C1(C(N2CC(C(CC)CC)C2)=O)CN(C(C2COCC(C)O2)=O)CC1CC c1(C(N2CCC(N(CCC)CCC)CC2)=O)cc(C(C)(C)C)ccc1O c1(C(N2CC(CCNC(=O)CSc3ccccc3Cl)C2)=O)csc([N+](=O)[O-])c1 C1(NC(C2OCCN(CC)C2)=O)CCN(C(c2nn(C)c(C)c2Cl)=O)CC(O)C1 c1(C(=O)NC2CCCC(CN(C(=O)CSC(F)F)C)C2)ccc(F)c(F)c1F N1(C(C2C(=O)NCC2)=O)CC(C2CN(C(=O)CC3CC4(CC4)CO3)C2)C1 c1(N2CC3C(NC(CC(CC)O)=O)C3C2)ncnc2cccc(C)c12 Cc1ccncc1C(=O)NCc1nnn(C)c1C(=O)NC(c1nncs1)C Cc1cc(=O)c(C(N2CCC2CNC(=O)C(N2CCNC2=O)C)=O)cn1C C1(NC(C=CCOCCOC)=O)CCOC(C(=O)NC(C2CCC2)C)C1 c1(C(N2CCCC(NC(=O)CN3CC4C=CC3C4)C2)=O)ccc2c(c1)NCC2 C(=O)(C(O)C(F)(F)F)NCc1cccc(C(=O)NC(C#C)(C)C)c1 c1(C(CC(=O)NCC(CC)NC(c2cc(O)nc(O)n2)=O)C)ccc(F)c(F)c1 CN1CCOC(C(=O)NC2CCC2NC(C2CN(S(N)(=O)=O)C2)=O)C1=O C1(C)(CC(=O)OCCSC)CCCO1.c1(CCCN2CC2=O)ccccc1 Cc1ccc(F)cc1CN1CCC1C(=O)NCCCBr C1(NC(CSCCCC)=O)CCN(c2ccc(C(=O)OC)cn2)CC1C C1(C(=O)NC2C(CNC(C3(C(C)C)CC3)=O)CCC2)CC12CCCCC2 C1(OC(C)C)CCC(N(C=O)CCNc2ccsc2C)CC1 CCC(C)CC(C)N(C(=O)C#CCNC(C1CN2CCC1C2)=O)C Cc1cc(C(=O)NCC2(NC(=O)CCCC3CC3)CCOC2)c2c(O)n[nH]c2n1 N1(S(CC)(=O)=O)CCOCC(C(=O)NC2CC2C(=O)NS(C)(=O)=O)C1 C1(CC)CCCCC1C(=O)N(C(C)(C(=O)N(C1COC(C)(C)C1)C)C1CC1)C C=CCC(C)(CC)C(=O)N(CCC(=O)NCC(CSC)OC)C1CC1 CCN=C(NCCF)NC1CC(OC(C)(C)C)C(c2ccc(OC)nc2)C1 C=CCC(C)(C)C(=O)NCC(C)(C)CNC(C1(CC)CCOC1)=O N1(C(Cc2nc(C)oc2)=O)CCC(CF)(NC(c2ccc(-c3cccs3)[nH]2)=O)C1 c1(SCC(=O)NC(C(C)C)CNC(C2CC3CC3C2)=O)nnc2ccccn12 c1(N(C)Cc2nnn(C)n2)cc(P(C)(C)=O)ccn1 N1(C(c2c(CCNC(C3CC(O)C3)=O)n[nH]c2)=O)CC(O)(C2CC2)C1 CCN=C(NCC1CCC1C)N1CCN(c2ncnc(N(C)C)c2C)CC1 c1(CC)nc(C)c(C(=O)NC(COC)CNC(c2cc(O)ncn2)=O)s1 c1(CC2CCOC2C(C)(C)C)ccccc1.CN1CCN1CC1CC1.C(=O)(C)O C(=O)(CCCCCOCC(N)C(=O)OCc1ccccc1)OC N1(C(CN(C(C2C=CCC2)=O)CC)=O)CCC(C)(C)C1C CCC(C)(CC(=O)OC)NC(=O)C(F)(Cl)c1ccccc1.C(C)(C)(C)OC=O c1(CCNC(C2CC(NC(C(C)OCC3CC3)=O)C2)=O)cccnc1 C1(CNC(=O)C(N2CCCc3n[nH]cc32)=O)CCSC2(CCC2)C1 N1(C(Cc2ccc(NS(C)(=O)=O)cc2)=O)CC2CN(C(C3CCC3)=O)CC2C1 c1(N2CC(NC(c3c(OC)ccs3)=O)C(C#N)C2)cc2ncnn2cn1 C(=O)(CCC(=O)NC1CCCC1)NCC(CNC(c1c(SC)ccs1)=O)(C)O C1(C(N2C(CC)C(NC(c3cc(C)c[nH]3)=O)CCC2)=O)CC2C=CCC(C1)C2 C(C(C(=O)N1CCC(OC)C1)NC(=O)C(C)n1cccn1)SCC c1(C(=O)NCCC2(OC)CN(C(C3CC4CC4C3)=O)C2)ccc(F)c(F)c1 C1(CC(N2CCC(N(C(=O)CCC3CC3CC3CC3)C)C2)=O)CCC(=O)CC1 C1(N(CCC)CCNC(=O)C2CC2)CCN(C(=O)NC2CC(C)CO2)CC1 c1(C(N2C(CN(C(=O)C#CC3CC3)C)CCC2)=O)cccc2sccc12 C12(C(=O)NCc3n(CC)nc(C)c3)CCC(CC1NC(C1CCC(O)C1)=O)C2 N1(CC=CC)CCCN(C(=O)C(=O)Nc2cc(N)ccc2SC)CC1 c1(OC)ccc(CN2CC(n3cc(C4CC5(CCCC5)C4)nn3)C2)c(Cl)c1OC c1(C(N2CCC(CCNC(C(C3CC3)OC)=O)C2)=O)cc(OC)cc2c1OCC2 c1(C(=O)Nc2c(C)nc(-c3ccc(C)c(C#N)c3)s2)ccc2ncoc2c1 CCCC(C(=O)OC)NC(C1CN(C(=O)C(C)N=[N+]=[N-])CC1C(C)C)=O C1(C(N2C(C(N(C)C)=O)CCC2)=O)COCCN(C(C2CCCCC2(C)C)=O)C1 c1(CCC(=O)N(CC(C)OC2CCOC2)C)ncccn1.C1(C)CN1 Cc1nn(C)c(C)c1CC(=O)NCC1CCN(C(c2c(Br)noc2C)=O)CC1 N1(C(C(n2c(C)ncc2)C)=O)CC=CC(C(=O)NCC2CCC3(CC3)C2)C1 C1(C(=O)NCC(C(=O)NCC)(C)C)CCCN(C(C2CCCC(=O)N2C)=O)CC1 c1(NCCCNC(C2CCC(C(CC)(C)C)CC2)=O)ncnc2cccc(Br)c12 c1(C(=O)NC2CC(CNC(C3CC(C)OCC3)=O)C2)ccc2oc(O)nc2c1 c1(C(N2CC(NC(CC(CCC)C)=O)C(SC)C2)=O)cc(OC)ccc1[N+](=O)[O-] C(=O)(C(O)CSC)N(CC(=O)N(CCOC)CC)C(C)C c1(C(N2CC(C(=O)OCC)C(C)(C(F)(F)F)C2)=O)ccn2nnnc2c1 c1(NC(C2(CC=C)CCCN2C(=O)CCC)=O)cc2c(s1)CCC(C(=O)OCC)C2 n1(CC(=O)NC2C(NC(C(N)=O)=O)CC2)cc(Br)c(C2CC2)n1 c1(C(=O)NC(C(=O)NCCc2ccn(CC)n2)C2CCOC2)ccc(F)cc1F C(=O)(C(O)CC[S+](C)C)N1C(CCNC(c2cc(C(C)(F)F)ncc2)=O)CCC1 Cc1cc(C(=O)N(C2CCC(NC(=O)CCc3cocn3)CC2)C)cc(N)c1Cl N#CC1CN(CC(c2ccc(CC3CCCC3)c(C(F)(F)F)c2)=O)CCO1 N1(C(C(C(C)C)NC(C)C)=O)CCC2(CCN(C(C3CCCSC3)=O)C2)C1 C1(C(=O)NCC(C)C(F)F)(CF)CCN(C(=O)CCCF)C1 c1(CNC2CC(CC(=O)N(C(C(C)C)CO)CCO)C2)cc(Br)ncc1Br N1(C(c2cn(C(C)C)nn2)=O)CCN(C(=O)Cc2csc(S)n2)C2CC12 C12(NC(CC3C=CC(NC(c4n(CC)ncc4)=O)C3)=O)CC1COC2(C)C n1(C(C(N2CCC(CCNC(COC(C)C)=O)C2)=O)C)cnc2c(N)ncnc12 CCC(C)CCC(C)(C)NC(=O)C(C)CCC#N N1(C(C(C)NC(=O)NC)=O)CCC(O)(CN(C)C(c2cnn(C)c2OC)=O)C1 c1(C(=O)NCCN(C(=O)CCc2ccc(F)cc2F)CC)c(C)cc(C)oc1=O Cc1ncc(C(=O)NCC2CCC(NC(c3ccon3)=O)C2)n1C(F)F c1(NC2CCN(C(CNC(CC)=O)=O)CC2O)c(C)c(C)nc2ncnn12 Cc1ncc(C(=O)N(C)CC2CCCCN2C(=O)CCCOC(C)(C)C)cc1Cl N1(C(CC2(OC)CCC2)=O)C(C(=O)Nc2ccnc(Cl)n2)CC2CCCCC12 N1(C(C(CO)N(C)C)=O)CCC(O)(C(c2ccccc2)NC(c2cnc[nH]2)=O)C1 N1(C(=O)OC(C)(C)C)CC2CC(F)(F)CCC2(NCCC2CC2(F)F)C1 N1(C(c2[nH]cc(C(N)=O)c2)=O)CCCN(C(c2cnccc2Cl)=O)CC1CO Cc1ccc(C(=O)NCC(O)CNC(=O)Cc2ccccc2O)c(C)n1 c1(CC)nc(O)c(C(N2CC(NC(c3cnnn3C)=O)CC2C)=O)cc1C c1(C(N2C(C(=O)NCC3CCCC(CO)C3)CC2)=O)n[nH]c2ccccc12 N1(C(C(=O)Nc2ccc3c(c2)OCO3)C2C(C)C2)CCSC2COCCC12 CN1CC(C(=O)NC2CC(NC(=O)CC3CCC3)C2)C(c2ccc(F)cc2)C1 C=CC(O)C(C)(C)C(=O)N1CCOC2CN(C(=O)COC3CCCC3)CC12 CC1CCC(NC(=O)Cc2ccccc2CO)CN1C(c1cncn1C)=O C12(CNC(c3cnn(C4CCC4)n3)=O)CCC1CCN2C(C1CC(O)C1)=O N1(C(C(C2CC2)SC)=O)CCCCC(CCC(=O)NCCCc2ncco2)C1 c1(CNC2C(C)N(C)CC2)cc(Cl)c2c(c1)OCCO2 c1(CCC(=O)NC2(NC(=O)Cc3ccn(C4CC4(F)F)n3)CC2)ccccc1 Cc1c(Cl)cnn1CC(=O)NCc1ccccc1CN(C(=O)CC(C)CF)C C=CCN=c1[nH]c(C(=O)NCC2(O)CCCN(C(=O)CCCS(C)(=O)=O)C2)cs1 N1(C(CSCC#C)=O)CCN(C(=O)C(C)n2ccnc2)C(C2CCCC2)C1 N1(C(CNC(c2nc(Cl)sc2Cl)c2n(C3(C)CC3)nnn2)C(C)C)CCN(C)CC1 C12(NC(C=Cc3n(C)cnc3)=O)CC3CC(C1)CC(CNC(C1CCCS1)=O)(C3)C2 C(c1ccccc1[N+](=O)[O-])=CCNC(C(C)OC(=O)Cc1cn(C)nc1C(F)F)=O Cc1cc(=NCC(F)=C2CCN(C(=O)OC(C)(C)C)CC2)[nH]c(C)n1 C1(C(=O)NC(c2ncccn2)C)(CC)CN(C(=O)C(C)Sc2nncn2C)C1 C(=O)(C1=CC2CC(C1)CC2O)NC(CNC(COC(CC)(C)C)=O)C N1(C(Cc2c(C)ccnc2)=O)C2CCC1CN(C(C1CCC(F)(F)CC1)=O)C2 C1(C(N2CCC(C)(F)CC2)=O)CN(C(=O)C(O)CC(N)=O)CC12CCC2 N1(C(C2N(C(c3c(CC)nns3)=O)CC(F)(F)C2)=O)CC2C=CCC(C2)C1 c1(C(=O)NC(CNC(CC2(C=C)CCC2)=O)C2CC2)cccc2nc(O)oc12 C1(CC)CCCN(Cn2cc(CCSC3(c4ccc(Cl)cc4)CCC3)cn2)C1 c1(C(N(CC(C)N(C(C(CC)SC)=O)C)C)=O)cc2ccc(Cl)cc2[nH]1 c1(NC2CCCN(Cc3cc(C)c(Br)c(C)c3)C2)ncc2c(Cl)cccc2n1 c1(C(=O)NCC(CNC(C2N(C(=O)OC)CCC2)=O)C)cccc(C)c1F c1(C(N2CCC(NC(C3(C)CC(C)C3)=O)C2C)=O)cc2c(F)ccc(F)c2[nH]1 N1(C(c2nn(CC)nc2C)=O)CC(C)OC2(CCN(CCCCCF)C2)C1 c1(C(N2CCC(Cc3cc(Br)nn3C)C2)C(=O)NC)ncc(Cl)n1C C#Cc1cc(N(C(=O)C(=O)NCc2ccnn2-c2ccc(C#N)cc2)CC)ccn1 N1(C(c2cccc(C)c2O)=O)CCC2CN(C(C3CCC4CCC3O4)=O)C2C1 C(=O)(C(C)(C)CSC)N(CC(CC)(C)NC(c1cnn(C(C)C)n1)=O)C N1(C(C2C(NC(CSCCC)=O)CCO2)=O)CCCCC(COC)C1 Cc1ccccc1-c1nc(C(=O)NCC2CCC2NC(c2cc(Cl)ns2)=O)cs1 N1(C(C(c2ccccc2)=O)=O)CC(NC(c2nocc2Br)=O)CC(O)C1 C#Cc1ccc(C(=O)NC2CC(C)N(C(=O)C=Cc3ccn(C)c3)C2)cc1C N1(C(CC2(NC(CCn3ccc(C)n3)=O)CCC2)=O)CCC(F)C(O)C1 c1(C(=O)NC(C)CC2CN(C(C3CC3C)=O)C2)ncc(Br)cn1 C1(C(=O)NC2(C(N3CCCOCC3)=O)C(C)(C)C2)CC2CC1CC2O C1(CC)(NC(C2C(C#N)C2(C)C)=O)CCN(C(C2C3CNC(=O)C23)=O)CC1 C12(C(=O)NC3C(CNC(c4ccn(CCF)n4)=O)C3)CC3CC(CC(C3)C1)C2 CC(=O)C(C)CC(C)C(=O)NC1(CC(=O)N(CC(O)C(F)(F)F)C)CC1 C1(C(=O)NC(C(C)OC)C(=O)N2CC(SC)C2)CCC2(CCC2)O1 C1(NC(c2cccc(C)c2N)=O)CCN(C(=O)C(O)C(F)F)CC1(C)C C#CC1(C(N2CC=CC2CF)=O)CN(C(=O)C(CC2CC2)OC)C1 N1(C(c2c(C)nncc2)=O)CCC(C(=O)NCc2n[nH]cc2C2CC2)C12CC2 C12(C(=O)NCC(CNC(C3(COC)CC=CC3)=O)O)CC(C1)C(C(F)(F)F)O2 C1(CC(N2CCN(C)C(CNC(=O)C(C)(C)CF)C2)=O)CCn2cncc2C1 C1(C)(C(=O)NCC(CCOC)NC(=O)CCc2ncc(F)cn2)CCCOC1 N1(CC)CCN(C(=O)C(F)CC2CN(C(=O)CCOC(C)COC)C2)CC1C C1(NC(C(c2nc(F)ccc2Cl)C)=O)CC(F)CN(C(=O)Cn2cncn2)C1 C1(Cl)(C(=O)NCCC2C(=O)N2)CC2CCC1O2.C(C)(C(=O)OC(C)C)SC C(=O)(C=CS(F)(F)(F)(F)F)N(C1CCN(C(=O)Cc2cccs2)CC1)CC(C)O Cn1c(C(N2CC3CC3(NC(c3coc(C(C)(C)C)n3)=O)C2)=O)nnc1S C1(CCNC(COCCCOC)=O)CC12CCN(Cc1ccccc1N(C)C)CC2 c1(C(N2CC(CNC(C(C)(C)c3ccns3)=O)OCC2)=O)cc(O)cc(C#N)c1 C=CC(C)(C)C(=O)N1CC(CCNC(c2n[nH]cc2C(F)(F)F)=O)C(C)C1 c1(C(=O)NC(CCNC(CSCCC)=O)C)cc(S(=O)(=O)NC)ccc1F Cc1nc2c(C(N3CCC(NC(=O)CC4CCCC4O)C34CC4)=O)cccc2o1 N1(C(CCC(C)OC)=O)CCCC(C2(NC(c3ccc(C)s3)=O)CC2)C1 c1(C(C(=O)NCSc2ccccc2)N(C2CCC(C)(C)C2)C)ccc(F)c(Br)c1 N1(C(C2CN(C(C)=O)C2)=O)CCC2(COC(CNC(C3(Cl)CC3(C)C)=O)C2)C1 N1(C(=O)NC(C2(NC)CCOCC2)COCC)CCN(c2ccc(F)cc2)CC1 C(c1cccc(F)c1)=C(C(=O)NC1CCC(NC(c2n(CCC)ncc2)=O)C1)F N1(C(C(CC)n2cccn2)=O)CC2CCC(CCC(=O)N(C(N3CCCC3)=O)CC)(C2)C1 C1(NC(c2n(C(C)C)ncc2)=O)CCCN(C(=O)Cc2ccns2)C1 c1(CC(N2CC(CNC(CC(CC)O)=O)NCC2)=O)c[nH]c2cc(C)ccc12 N1(C(c2c(-c3cn(CC)nc3)n[nH]c2)=O)CCCC(NC(C2(C)COC2)=O)CC1 C12(C(N3CCC(CNC(C(CC(C)C)N(C)C)=O)C3)=O)C3CC(CC13)C2(F)F C(CCCN=c1[nH]cc([N+](=O)[O-])cc1C(N)=O)NC(c1c(C(C)(C)C)c[nH]c1)=O c1(C2(C)CCCN(C(C(C)N(CC(=O)O)C)=O)C2)nc2ccccc2s1 N1(C(C(C(C)C)OCC)=O)CCN(C(C2CC23CCSCC3)=O)CC2(CC2)C1 c1(C(=O)NC2C(N(C(=O)COC3(C)CCCC3)C)COC2)ccc(O)nn1 c1(C(C)NC(=O)CC2CN(C(=O)C=Cc3ccco3)C2)ccc([N+](=O)[O-])cc1 c1(C(=O)NCC2(O)CN(C(C3CCN(C(=O)NC)C3)=O)C2)nc(C)ccc1Br c1(C(=O)NC2C3(CC(NC(c4scc(C)c4)=O)C3)C2)cc(F)cc(Br)c1 C1(C(=O)OC(C)(C)C)C(NC(c2cocc2Br)=O)C1(C)C N1(Cc2c3ccc(C(=O)OC)cc3[nH]c2)CCN2C(=O)NCCC2C1 c1(NC(C2C(CNC(CNC(C(CC)C)=O)=O)OCC2)=O)cn(C)nc1C#N C1(C(=O)NC2CN(C(CC3(OC)CC3)=O)C3(C2)CCC3)Cc2cc(Cl)ccc2O1 N1(C(c2c(C)noc2N)=O)CCC(C)C(NC(=O)CC2CC2C(F)(F)F)C1 c1(CN(C)CC2(C(F)(F)F)CCC2)csc2cc(Cl)ccc12 N1(C(c2conc2CC)C(=O)NCC(=C)C)CC=C(c2cccc(OC)c2)CC1 CCC(CC(=O)NCCOCC(=O)Nc1cc(C)nn1CC)C1CCC1 C=CC1(O)CCN(C(=O)C(C)CNC(c2c(C)coc2CC)=O)C1 c1(C(C)SC)nnc2n1CCC(=O)NCCC1CN2CC1OC.C(C)(=O)OC C1(NC(=O)CCCc2ccc(Br)cc2)CCN(Cc2c(Br)ccnc2Br)CC1F c1(C(=O)NCCCCC(C)NC(CC2CC(CC)C2)=O)cc2nc(C)ccc2o1 N1(C(=O)NC(c2cnn(-c3cccc(Cl)c3)c2C)C)CCC(CO)C(O)C1 c1(CC(C(=O)N(CCC)CCNC(C2CC2CCOC)=O)C)ccccc1Cl N1(C(CCSCCC)=O)CCCC(C2CN(C(=O)CCCCCN(C)C)C2)C1 c1(C(N2CCC(F)(CNC(=O)C=CC3CC3)C2)=O)cc(F)c(C(F)F)cc1F CCCCC(C(=O)N1CCC(CCC(=O)N(C)CC2(N(C)C)CC2)C1)N(C)C CC1COCC(C(=O)NC2CC(C(=O)Nc3ccccc3CCO)C2)O1 Cn1cnc2nc(=NC3CC(CC#N)C3)[nH]c(NCC3CC4CCC3C4)c12 c1(C(=O)NCC(C)N(C(c2c(NC(=O)OCC)scn2)=O)C)cc(O)cc(O)c1 c1(C(N2C3CN(C(C4(COC)CCC4)=O)C(CC3)C2)=O)ccc(F)c2ccsc12 C(CC1=CCCCCC1)NC(C1CN(C(COC(CC)C)=O)C2(C1)CC2)=O CC1(CNC(C2COC2)=O)CN(C(c2c[nH]nc2-c2cccs2)=O)CCO1 c1(C(=O)NCC(CCOC)NC(c2ccc(Cl)o2)=O)cc(C2CCC2)n(C)c1C N12CCC(C1)C(=O)N1CC(C1)C2.c1(CCN(c2ccccc2)C)cc(CO)no1 c1(NC(C2CCCN(CCNC(=O)CC3COCC3O)C2)=O)cnn2ccsc12 Cc1cc(CC(N2CCC(CCNC(C3OCC3(C)C)=O)C2)=O)c(C)s1 n1(CC=C)cc(NC(=O)C=CCC(C)(C)NC(=O)C(C)c2cccs2)cn1 N1(C(C(C)NC(CC)=O)=O)CCC(C)(NC(C2CC2(C)C)=O)C1 c1(CN(c2ncc(CC)o2)C(=O)CN(C(C)CC)C)ccc(C)cc1 Cc1cc(C(=O)NC(C)C(C)NC(=O)CCNC(c2ccoc2)=O)ns1 N1(C(CC=CCNC(C(C2CCC(=O)N2)C)=O)=O)CCC2(CC2)C1 CS(=O)(=O)c1cc(C(=O)NCC2CC(NC(c3cncc(Cl)c3)=O)C2)co1 C1(NC(c2c(C=O)cccc2)=O)(CO)CCN(c2nc(Cl)c(C#N)s2)CC1.CN Cc1c(C(N2CC(NC(=O)CCc3c[nH]c(=N)[nH]3)CC(O)C2)=O)cccc1F N1(C(C=Cc2c(C)ncs2)=O)CCCC(C2CC2NC(C2(O)CCOCC2)=O)C1 C1(C)(C(=O)NCCC2N(C(C(C)(C)c3cscn3)=O)CCCC2)COC(=O)OC1 C=CCC(C)(C)CCNC(c1ncoc1C1CC1)c1nnnn1CC1CCOC1 c1(C(N2CC(NC(CCC=C(C)C)=O)C(C)C2)=O)cccc(Br)c1F c1(CC(=O)N(CCC(F)(F)F)CCN(C)CCO)c(C)nc2n[nH]cc2c1C.CO N1(C(C2CCCCN(C(CCC=C=C)=O)C2)=O)CCC2(CCC(O)C2)C1 c1(NCc2c(NC(=O)NC(c3cn(C)nc3)CO)cccc2)cc(O)c(Br)cn1 C1(CC(=O)NCCC2CC=CCC2)CC2(C1)CN(C(c1cnc(O)o1)=O)C2 CC1CCCC1(C)C(=O)NC1(CO)CN(C(c2ccc(CF)cc2)=O)C1 N1(c2ncc(C#N)cc2F)Cc2ccccc2C(CNC(c2cc[nH]n2)=O)C1 N1(CC(=O)NCC#CCNC(C2CCC(c3ccccc3)C2)=O)CCCCCC1 c1(COC(N2CCC(CN)C2)=O)nnnn1CCCSc1ccccc1 C1(CCOC)CN(C(C2(F)CCC2)=O)CCN1C(=O)Cc1ccc(C)nc1 Cn1cc2c(n1)CCC(C(N1CC(F)(CNC(c3ccc[nH]3)=O)C1)=O)C2 C1(CC)CN(C(=O)NC2CCN(S(=O)(=O)CC(C)C)CC2C)CC(C)S1=O C(=O)(C(C)CC(C)C(C)=O)N1CCCC(C)(C(N2CC(C(=C)C)OCC2)=O)C1 N1(C(CNC(C)=O)=O)CCN(C(=O)CC(C)(C)c2cccs2)CC2CCCCC12 CC1=CCC(C(=O)NCCCCCCNc2ncc(C3CC3)cn2)CC1 c1(C(N2CC(N(C)C(C3CCCN3C=O)=O)C(O)C2)=O)cc2c(Cl)cccc2s1 C1(CC(=O)N(C)CCN(C(=O)C(C)(C)C(F)F)C)SC2=NCCN2C1=O CCC(CC(=O)NCCCC(C)NC(c1cnc(C2CC2)[nH]1)=O)C(C)C N1(C(c2nnc(C)s2)=O)CC2(CNC(=O)CCc3cccc(Cl)n3)CCC1CC2 C(=O)(C1=CC2(CCOC2)C1)NCCC(CC)(CC)NC(C(CCCC#C)C)=O C(=O)(CCC(C)(C)N(C)C)N1CCC1.Cc1ocnc1CC(=O)NC1CC1 Cc1c(C(N2CC(CC(C)NC(C3CCOC(C)C3)=O)C2)=O)ccn1CCO N1(C(CCC)=O)CC(NC(c2cn3c(C)cccc3n2)=O)CC12CCCCC2 C(=O)(CCCC(=O)NC1CC(C)(NC(=O)CC2CCC2C)C1)OCC Cc1cnc(C(N2CCC(C)(C(N3CC(n4cccn4)C3)=O)C2)=O)c(F)c1 C1(C(=O)NCCN(C)C(c2cnn[nH]2)=O)CNC(=O)CN1C(C1CCCC1)=O c1(C(N(C2CCC(NC(C3CCOC3)=O)C2)C)=O)ccnc2ccnn12 C(=O)(CCCCCC(C)(C)C)N1CC(OCCC(=O)N(C2CCC2)C)C1 N1(C(C2(C#C)CCC2)=O)CC(O)CC1CC(N1CCCCC1C1CC1)=O C(C(C)(C)C(=O)NC1CCCC1CNC(=O)CSc1ccccc1OC)OC C1(CC(=O)N(CCNC(=O)C(C2CC2)C2CC2)CC)CCC(C)(C)CO1 c1(C(N2CC(CNC(c3c(OCC)ccs3)=O)OCC2)=O)cc(OC)ccc1Br C1(CN2CC(C3OCCN(c4cccc(C)c4)C3)OCC2)CCCNCCCC1 c1(C(=O)NCCC(C)(C)NC(=O)CNC(=O)N(C)C)c(Br)nc2n1CCOC2 C(=O)(CCCC(=O)NN(c1cc(=O)c(O)c[nH]1)C1CCN(C=O)C1)OC.C1(C)CC1 c1(CC(=O)N(C2CCN(C(C3CC(C)(C)CN3C)=O)C2)CC)cc(F)ccc1C c1(OC(=O)CCNC(N2CCCC2c2ncccn2)=O)ccccc1 C12(CNC(CCOCC(C)C)=O)CC(CO1)N(C(c1cnc(C(F)(F)F)s1)=O)C2 c1(CN2CC(C#N)C(NC(c3nc4ccccn4n3)=O)C2)cc2ccccc2s1 C(=O)(C(C)S(C)(=O)=O)N1CC(C(N(c2ccc(C(=O)OCC)cc2)C(C)C)=O)C1 CC1CCC(CC(=O)NCC(O)CNC(=O)C(O)CN(C)C)OC1 N1(C(c2occ(C(N)=O)c2)=O)CCCN(C(=O)CCCC(F)(F)F)C(CO)C1 c1(C(N)=O)ccc(C(=O)NC2CCCCC2NC(=O)CC2CC3CC3C2)cc1 C(=O)(CC1=CCN(C(C2CC(O)CN2C)=O)CC1)N1CC(C)OC(C(N)=O)C1 N1(C(c2cccc(C)c2)=O)CC(C)CCC1CNC(c1ccc2c(c1)CC2)=O N1(C(C(CC)C(C)O)=O)CCN(C(c2ccc(Br)c(OC)c2)=O)CC(C)(C)C1 Cc1ccc2c(C(N3CCC(NC(=O)Cn4ccc(C)n4)C34CC4)=O)coc2c1 C1(NC(C(CCC)CC)=O)CN(C(c2cnc(OC)cn2)=O)CC1N=[N+]=[N-] C1(N(C(c2c(C)coc2)=O)C)CS(=O)(=O)C12CCN(C(=O)CC1C=CCC1)CC2 N1(C(=O)NCCN(C)Cc2ccccc2)CCC(F)(F)C(F)C1 CCCCCCCCNC(C12CC(CN1C(=O)C(C)(O)C(C)C)C2)=O c1(C(=O)NCC2C(CNC(CCSCC(C)C)=O)C2)n[nH]c2c1COC2 c12ccc(cc1)OCCc1[nH]ccc1NC(=O)N2CCC=O.C(C)(C)(C)OC.CC N1(C(CC)C(=O)N2CCC(NC(c3cc(CC)oc3C)=O)C2)CCCC(CO)C1 C(C(F)(F)C(F)(F)Br)NC(=O)Nc1ccc(=O)n(Cc2cccc(F)c2)c1 CS(=O)(=O)c1ccccc1C(N1CCN(C(=O)CC(F)(F)C(F)F)C(=O)C1)=O c1(C(C(=O)NCC2C(CNC(COCCC=C)=O)C2)C)ccc(C)cc1 Cc1ccc2sc(C(=O)NC3CC3NC(c3cc(F)c(F)cc3F)=O)cc2c1 N1(C(c2c(C(C)C)cnn2C)=O)CCC2CN(C(=O)COC3CC=CC3)CCC12 Cn1cnc2cc(C(=O)NC(CNC(=O)C(C)(C)CC(C)(C)C)CO)ccc12 c1(C(=O)NC2C(NC(=O)CCc3cnc[nH]3)COCC2)nnn2c1COCC2 c1(OC)ccc(Cl)c(C(=O)NC2CCC2NC(C2CCC(C(N)=O)O2)=O)n1 N1(C(c2nccc(C(N)=O)c2)=O)CC2(CCCC2NC(=O)C#CC2CCOC2)C1 N1(C(c2cc(C(C)C)n[nH]2)=O)CC2CC1C2CNC(C1CCCN1C)=O n1(CC(N2CC3C(NC(=O)CCOCC(F)F)(C3)C2)=O)ccc(O)nc1=O C(CC(F)F)(C(=O)NC(c1cccs1)C)NC(C(CSC)OC)=O N1(C(CC(CC)SC)=O)CC(NC(c2ccc(C)cc2C)=O)CC12CCC2 CS(=O)(=O)C1CCCCC1NC(=O)C(=O)NCCc1c[nH]c2cccc(Cl)c12 N1(C(C=C(C)C2CC2)=O)CCC2(C=C(C(=O)NC3CCOCC3(C)C)C2)C1 c1(C(CC)C)nc(-c2cc(CC)n(CC)n2)n(-c2ccc(F)nc2)n1 c1(OCC)cc(C(=O)NCCCNC(c2ccc(C(=O)NC)cc2)=O)oc(=O)c1 n1(C(C)C)ncc2c(N3CCC(NC(C4CC4C4CC4C)=O)C3)ncnc12 C(C(=O)N(C)CC1CN(C(c2ncccc2C2CC2)=O)CCO1)(C(C)C)SC Cc1ccc(O)c(CC(N2CCN(C(c3cccn(C)c3=O)=O)C(CF)C2)=O)c1 c1(SCC(C2CCCCC2)C)nc(-c2cncc(F)c2)nn1C1CSC1 CC1CSCCCN1Cc1cc(C(C)(C)C)ccc1Br c1(C(=O)NCC2C(C(=O)NC(CCC)C3CC3)CC2)cccc(F)c1F c1(OCC)ccc(C(=O)NCC(C)N(C)CC2CCCN(C)C2)cc1C1CC1 CC(CN(C)C)CCC(=O)NCC1(F)CCC(NC(C2(CN(C)C)CC2)=O)C1 C1(C)(C(N2CC(CNC(C(COC)OC)=O)C(C)C2)=O)CC2(CCC2)C1 C1(NC(c2cc(C)nn2C)=O)CS(=O)(=O)CC1NC(C1(C#N)CCC1)=O C1(C(=O)NCC=CCNC(C2(CCCC)CCCC2)=O)CCc2nn[nH]c2C1 c1(NC(C(c2ccc(Cl)cc2)N2CCC(NC)C2)=O)ccc(Cl)c(C)c1 c1(OC)ccc2c(C(=O)NCC3(F)CCCN(C(=O)C(C)C)C3)ccnc2c1 c1(CNC(c2cc(C(CC)C)no2)=O)ccc(I)c(O)c1 C1(C(N2CCC(NC(c3ccnc(C(F)F)c3)=O)(CO)C2)=O)CC(C2CC2)=NO1 O=C(C1c2ccccc2CN1)N(C1CC1)Cc1ccc2c(c1)[nH]c(=O)n2C1CC1 C(=O)(CS(=O)(=O)CCOCC)NCCCNC(C1(C=C)CCOCC1)=O CCS(=O)(=O)CC(=O)N1CCCC1(C(N1CCOC(C#N)C1)=O)C(C)C O=C(C1=C(F)CNCC1)NCc1ccc2cc[nH]c2c1 c1(C(N2CCOCC(CNC(CC(CC)OC)=O)C2)=O)cc2ncccc2[nH]1 C12(C(N(C(C)CNC(=O)CC3CC4(CC4)CO3)C)=O)CCC(C#N)(CC1)CC2 C(=O)(C(C)CC(N)=O)N1CCCC(CN(C(C(C)=C2CC2)=O)C)C1 CCC(C)C(CC(=O)NCCc1ccc(O)cn1)NC(=O)Cc1cccnc1F c1(C(N(CC(C)NC(C(CC)N(C)C)=O)CC)=O)cc(OC)c(O)c(OC)c1 c1(C(=O)NCC2C3CN(C(c4cc(OC)nn4C)=O)CC32)c(Cl)ccc(F)c1F Cn1cc(C(=O)C(=O)NC2(C)CC(NC(N3CCC3c3ccccn3)=O)C2)cn1 CCCCC(=O)COC(F)(F)F.C12C3CN(CC13)C(=O)c1ccc(cc1)NC2=O C1(C)(CNC(CN2CCC(C)C2)=O)CN(C(=O)CCN2C(=O)CCC2=O)CCO1 C(=O)(C1=NOC(C)C1C)NC(C1CCN(C(C2CCN(C(C)=O)CC2)=O)C1)(C)C N1(C(COCC)=O)CCCC1C1CCCN1C(c1c(Cl)cnn1C)=O c1(C(=O)NC2CC(NC(c3ncn(C)c3)=O)C2)cc2c(Cl)cncc2s1 CC1(C(=O)NCc2ccccc2CNC(C2(F)CC=CC2)=O)CC2(CC2)C1 C(C(C(=O)N1CC(CF)C1)C(C)C)NC(=O)N.Cc1cccc(C(=O)N(C)C)c1 c1(-n2cc(-c3sc(OC)c(C(=O)OC)c3)nn2)ccc(Cl)c(C)c1OC N1(C(C(C=C)O)=O)CC(N=c2cnc3cc(F)c(F)cc3[nH]2)C(C)(C)C1 C1(CNC(CCS(C)=O)=O)CCCC2(CN(C(C34CCOC(C)(C3)C4)=O)C2)O1 C1(CCNC(C2(NC(=O)CC3C=CCC3)CC2)=O)(SCC)CC1 CC1(C)CCOC(CNC(=O)C(O)C2CN(C(=O)C=Cc3cncs3)C2)C1 N1(C(C(C=C)C)=O)CCC2(C1)CN(C(c1cc(OC)cnn1)=O)C2 C#Cc1ncc(F)cc1NC(C1(C2=CCOC2)CCC1)=O C#Cc1c[nH]nc1C(=O)NCC(C)(C)OCC(=O)NCC(C1CCCC1)C N1(C(C2CCN2C(C2CCCCCC2)=O)=O)CC(Oc2snc(O)c2Cl)C(F)C1 c1(SCCC(N2CC(F)CC(NC(=O)CO)C2)=O)ccccc1[N+](=O)[O-] C1(c2cn(C(C(=O)NC3(CC(=O)OC)CCCC3)C)nn2)CCCCNC1=O N1(C(c2c(C)ccs2)=O)C2CCC1CN(C(C1CCC1C(F)F)=O)C2 C1(C)(NC(CC(=O)OC)=O)CCCCC1C(=O)NCC1CCn2cnnc2C1 c1(C(=O)NCC(N(C(C(C)n2cccn2)=O)C)C2CC2)nccnc1N C1(C(N(CC(CN(C)C(C23CC(C(C)(C)C)(C2)C3)=O)O)C)=O)CC2(CCCO2)C1 C1(NC(C(C=C)CC)=O)CC2(CCN(C(c3ccc(N)cc3C)=O)C2)C1 C12CCN(CC1)N(C1CC1)C2=O.C12CCCC1N2.C12(C=O)CCC1C2.C(O)SC CCCCCCC(F)C(=O)NCC(CNC(=O)C1=CCCCC1)C(F)(F)F CC1CCCN(C(=O)CC2CCCC(C(=O)O)N2)CC1 c1(C(N2CC(C=C)C(NC(C3(Cl)CC3)=O)C2)=O)cc2ncccn2n1 C(=O)(C(C)(O)C(F)(F)F)NC1CCCC(NC(c2cccc(C#C)c2)=O)C1 c1(C(N2CC(c3cccc(C)c3)C2)=O)cnn2cc(C(=O)N(C)C)cnc12 CC1(C)CC(C(N2CCCC2CF)=O)(CNC(=O)Cn2cnnc2O)C1 c1(C(N(CC(=O)NCCCC(O)CO)CC2CC2)=O)cccc2cncn12 c1(C(=O)NC2CN(C(C(C)C3CCCO3)=O)C2)c[nH]cc1C(F)(F)F N1(C(CC2C(CC)C2)=O)CC(C2CCCN(C(c3cnsc3)=O)C2)C1 C1(NC(C=Cc2n(CC)ncc2)=O)CN(C(=O)CCc2nc(C)cs2)CCC1F C1(CNC(C(C)(C)C2CCCCC2)=O)C2CN(C(C3(C)CCC3)=O)CC12 C(=O)(C(C(F)(F)F)C(F)(F)F)NC1(C2CN(C(Cc3cnc(C)[nH]3)=O)C2)CC1 N1(CNS(=O)(=O)NC)CC(=O)N(CCCCSC2(N(C)C)CCC2)C1=O N1(C(C(C)NC(C)=O)=O)CC(NC(c2ccc3n[nH]cc3c2)=O)CC2(CCC2)C1 c1(C(=O)NCC(CNC(=O)C=C2CCCCC2)O)cc2n(n1)CCC2 N1(C(C(C)CC(N)=O)=O)C2CCC1CN(C(C1CCc3ncncc3C1)=O)CC2 CC1CN(C(=O)CC2(C)CCN(Cc3cnc[nH]3)C2)CCO1 C1(CCC)CCC(C(=O)NCC23CC(NC(=O)C=CC4CCCO4)(C2)C3)CC1 N1(C(c2cn(C3CN(C(=O)CC4CC5(CC5)C4)C3)nn2)=O)CCCCC1C1CC1 c1(C(N2CCC3C(CCN3C(=O)C(F)F)C2)=O)cc2ccccc2nc1O c1(C(=O)NC2C(CNC(Cc3c(OC)nccc3)=O)C2)nc(C)n2ccccc12 C1(C(=O)NC2CC3CN(C(COC(C)C)=O)CC32)CC2(COC(=O)N2)C1 N1(CC(C(c2ccccc2)OCC)=O)CCC(C(C)(C)C#N)CC1.C(=O)OC C1(NC(N2CCC(C(C)O)C2)=O)CCN(C(c2ncnn2C)=O)CC1 C(C)(c1ccccc1F)=CC(=O)NCCOCCNC(CN(CCC)C)=O C1(CNC(C=CCN(CC)CC)=O)CCC(C)N(C(=O)CCc2scnc2C)C1 N1(C(C(C)CF)=O)CCC2CCCC12CNC(=O)C=Cc1cccc(C#N)c1 c1(C(=O)NCC2(O)CN(C(c3ccc(OC)s3)=O)C2)ccc(C(N)=O)cc1 N1(C(CCNC(=O)OC)=O)CCC(NC(c2cc(C(C)C)on2)=O)C(CO)C1 N1(C(CC(COC)NC(c2cc(=N)[nH][nH]2)=O)=O)CCn2nncc2C1 N1(C(c2c(CC)cno2)=O)CCCC2(CCCN2C(=O)COCCCF)C1 C1(C(=O)NCC(CC(=O)N2CC(F)(F)C2C2CC2)OC)CC2C(C1)C2(C)C N1(C(CCC)=O)CCN(C(c2c(C)noc2C(F)(F)Cl)=O)CC1CO CCC(C)(C(=O)NCC1(C)CCN(C(=O)C(C(C)(C)C)SC)CC1)C(N)=O C(CC(=O)N1OC2CCC1CC2)C1CCN(C(Cn2ncc(C)c2)=O)CC1 Cc1cc(Cl)c(Cl)cc1C(N1CCN(C(c2cc(=O)n(C)o2)=O)CC1CO)=O Cc1[nH]c(=NCC(Cc2ccncc2)CO)ccc1[N+](=O)[O-] C1(N(C)CC2CCCO2)CCN(C(C2CC(=O)N(C3CCCC3)C2)=O)CC1O C=CCCCCCCC(=O)NCC12CCCCC1N(C(c1nocc1C)=O)CC2 C(CCCC(=O)N1CC(C)(C(=O)NCC(C)(C)n2cccn2)C1)(OC)OC c1(C(=O)NCC2CCCN(C(c3nnc(CC)o3)C)C2)cccc(Cl)c1Cl N1(C(=O)Nc2ccc(Sc3ncccn3)cc2)CCOc2c(Cl)cc(Br)cc21 c1(C(N2CCC(F)(CNC(c3cccc(OC)n3)=O)C2)=O)ccc(OC)cc1F C1(NC(C2N(C)CCC2)=O)CCC2CN(C(c3cccn3C)=O)CC2C1 Cn1c(C(N2CC=C(CNC(C3CN4CCC3CC4)=O)CC2)=O)cc2sccc12 c1(CC)nnc(O)c(C(=O)NCCCCC(C)NC(=O)C(C)=CC2CC2)c1CC c1(OC)cc(O)ncc1C(=O)NCC(C)CNC(c1ccc(SC2CC2)cc1)=O N1(C(C(C)C(F)F)=O)CCC2(CC1)CC2NC(=O)CC1CCC(F)(F)CC1 C1(CC)CN(C(C2CN(C)CCO2)=O)CCN1C(c1oc(C2CC2)nc1C)=O c1(OC)ccc(F)c2c1CN(C(c1ccn3c(C)cc(C)nc13)=O)CC2 C(=O)(C(CNC(=O)OC1CCS1(=O)=O)(CC)CC)NCC(C)OCC=C C12(C(=O)NC(c3nc(C)sc3)C)CCCC1CN(C(=O)CC1CC=CC1)C2 CCC(CC(=O)NCc1n[nH]cc1C(=O)NC(C12CCC(CC1)C2)C)CC(C)C c1(OC)cc(COC(c2nnc(C(F)(F)F)n2C)=O)cc([N+](=O)[O-])c1C c1(C(C(=O)NCCOCC)N(CC(C)OC)C2CC2)cc2ccc(Cl)cc2o1 CC(C)(C)CCC(F)C(=O)NCC1OCCC1C(=O)Nc1cnc(O)c(F)c1 C(C(=O)NCC(O)CCNC(=O)C(F)(F)C1CCOCC1)(C(C)C)SCC c1(C(N2C(CN(C)C(C3CC=CCO3)=O)COCC2)=O)cc2cc(Cl)ncc2[nH]1 c1(C(N2C(C(CNC(C(C)(C)OCC)=O)(C)C)CCC2)=O)cc(C)ccc1C C1(C2(O)CN(C(c3cc(-c4ccco4)c[nH]3)=O)C2)(CNC(C23CC(C)C2C3)=O)CC1 CCCCC(CC(=O)N(c1cccc(C)c1)C)NC(=O)CCNC(C)=O CN1CCCC(C(=O)N(CC(=O)NCC2CC3CCC2C3)CCO)C1 N1(CC(C)C)N=C(C(=O)NCCN(C(=O)COC(F)(F)F)C)CCC1=O.C1COC1 c1(NC(=O)NC2CCN(CCCOC(C)=O)CC2)ccc(C(F)(F)F)nc1N N1(C(c2n[nH]c(CC)c2Cl)=O)CC(CNC(=O)CC(C)CN(C)C)OC(C)(C)C1 c1(C(N2CC(CC(C)NC(=O)CSCC(N)=O)C2)=O)cc2ccccn2c1 CC1(C)CCN(CC#N)CCS1=O.C(CC(=O)C1(S(C)(=O)=O)CC1)N C1(C(=O)NCC2C(CC(=O)NCC3CCCC3O)C2)CC2(CCC2=O)C1 c1(C(=O)NC(CCOC)CNC(c2cc(C3CC3)no2)=O)c[nH]cc(C)c1=O C1(CN(C)C(C2CCCCO2)=O)CN(c2cc(-c3ccccc3)ncn2)CCO1 C1(C(=O)NCC2CCCN(C(=O)CC3CCCCC3O)C2)Cc2ccccc2O1 C1(NC(C(CC)NC(N)=O)=O)C2CC3C1C3C2C(N1CC(C)(C)C1C(N)=O)=O C1(NC(Cc2c(C)cccc2F)=O)CC2CCC(C1)N2C(C1C=CCS1)=O c1(OC)ncc(C(N2CCC(C(C)(C)NC(=O)CCn3ccnn3)C2)=O)cn1 c1(C(C)C(=O)NCC2CCC(NC(c3cnco3)=O)C2)ccccc1C(F)(F)F c1(C(C(=O)N(C(CCNC(CCSCCCC)=O)C)C)C)cccnc1 C1(C(=O)NC(C2CCCN2C(c2cccc(CO)c2)=O)C)CCCS(=O)(=O)C1 C1(C2CN2)CCC(F)(F)CC1.CC(C)(C)OC(=O)N(CC(N)=O)C1CC1 c1(CNC(C2CCN(CCCc3ccccc3Cl)C2)=O)cc(Br)cc2[nH]ncc12 C#Cc1cccc(C(N2CCCC(NC(=O)CCOC(C)C)CC2)=O)c1F CC1CC(C(=O)NCC(C)(C)C(=O)N2CCOC(C(C)(C)C)C2)CN1C C12(C(=O)NC3CCC(CNC(c4ccc(N)c(O)c4)=O)C3)CCCN(CCC1)C2 C(=O)(CC(CNC(=O)COCCNC=O)OCCO)N(C(C)C)C C(=O)(CCCC(=O)NCc1cc(SC)oc1C)NCC N1(C(=O)CS(=O)(=O)C2CC2)CC2CCC(C1)N(C(=O)CN1CCCCC1)C2 c1(OC)nc(C)cc(=NC(=O)C2C=CCN2C(c2ncc(Cl)cc2F)=O)[nH]1 N(C(=NCCF)NC(C1CC1)C1CC1)CC(C)(F)F.C12(C)CCCN(C1)C(=O)N2.C(C)(C)(C)O Cc1ccc(NS(C)(=O)=O)c(C(=O)NCC(O)CN(C(=O)C(C)C2CCC2)C)c1 CC1(C(=O)NCCCn2nccn2)CCCN(c2ncc(F)c(=N)[nH]2)C1 N1(C(c2ccc(CC)o2)=O)CC(CNC(C2CC23CCCC3)=O)CC1(C)C c1(C(N2CCCC(NC(c3cncc(OC)c3)=O)CC2)=O)cc(C)c(N)c(C)c1 CC(C(C)NC(C1(CN(C)C)CC1)=O)NC(C1(C#N)CC1)=O c1(C(=O)NCCC2CCN(C(C34CC(C)(C3)C4)=O)C2)ccnc(Cl)c1N N1(C(C=C(C)C)=O)CC=C(C(=O)NC(c2nccn2C)C2CC2)CC1 C12(NC(Cc3nccc(OC)n3)=O)CCCC1CN(C(=O)C(C)(C)NC(C)C)C2 CN1CCS(=O)(=O)CC1CC(N1CC(O)CC1CNC(=O)C=CS(C)=O)=O C1(C(N(C2CN(C(=O)C(C)(C)CC#N)C2)C)=O)C2CCCCCCC12 c1(C(=O)NC2C=CCN(C(CC(C=C)(C)C)=O)C2)ccc2c(c1)C(=O)N(C)C2=O C=CCCCCCC(=O)NCC1CC1CC(=O)Nc1ccc(F)cc1C#N C1(C(C)NC(C2CS(=O)(=O)C2)=O)CCN(C(=O)CCc2ccc(Cl)cc2)CC1 c1(N2C(CNC(c3c(C)nc(C)[nH]3)=O)CCC2)nc2cc(Br)ccc2o1 C12(NC(c3c(C)nn(CCO)c3C)=O)CCCN(C(=O)C(C)C3CC3)CC1C2 C1(NC(C2C(C)(C)C2NC(=O)CCc2cn[nH]c2)=O)CC2(CCCCC2)C1 C(CCN(C)C)(C(=O)NOCCC1CC1)NC(C=CCOC)=O c1(C(C(N2CC(C(C)NC(C3C(C)(C(C)C)C3)=O)C2)=O)O)cnn(C)c1 C(C(CC(C)C)C(=O)NC(C)CN(C(=O)CCNC(=O)CO)C)OC N1(C(c2csc(Cl)c2)=O)CCC2(CCN(C(c3ncc(Cl)cn3)=O)C2)C1 c1(C(C)C(=O)NCC2CCN2C(=O)COC(F)F)ccc(Br)cc1 N1(C(c2c(C)c(O)ccc2)=O)CCN(C(=O)CC2C=CCCC2)CC(C)(F)C1 Cc1ccc2ncc(C(N3CCC(C)C(CNC(=O)C(C)(C)CC#N)C3)=O)n2c1 N1(C(=O)C=Cc2cccs2)CCC2C1CCCN2c1ncc(F)cn1 CCCCC(C)C(=O)N1CCC(CF)(NC(=O)CCc2ccc(C)c(C)c2)C1 O=C(CCS(=O)(=O)c1ccc(F)cc1)NCC1CN(C(=O)C2=COCC2)C2CC12 C1(C(=O)NCC(C2CCCC2)NC(C(CC)OC)=O)CCN(OC)CC1 c1(C(=O)NCCCC(C)NC(C2N(CC)CC2)=O)oc2ccccc2c1OC c12cccc(c1)C(=O)NC2.N1(C(c2c(CC)[nH]cc2)=O)CCOCC1C1CC1 C1(NC(c2nc(CC)sc2N)=O)CC2CC1CN(C(=O)C(O)C1CCCC1)C2 Cc1ncc(Cl)cc1CC(=O)NCC1CC(F)CN(C(=O)CC2CC=CC2)C1 N1(C(CCCCc2cn(C(C)CO)nn2)=O)CCC(O)(c2cccc(F)c2)CC1 c1(C(N2C(CNC(C3CCC3(F)F)=O)CCCC2)=O)cccc2nc(CO)[nH]c12 C=CCCCCCC(=O)NCC(C)(Cn1cccn1)NC(c1cccnc1C)=O c1(CC)ncc(Cl)c(C(N2CCOC(CNC(=O)C(=Cc3ccco3)C)C2)=O)n1 C=CC(C)C(C)C(=O)NCC(C)(C)NC(c1cc(OC)cc(N)c1)=O C(C)(CC(=O)NC(CC1CCOCC1)C(=O)NCCN1CCC(CO)C1)=C(C)C C1(CC)(OC)CN(C(=O)C(C)CNC(c2ccncn2)=O)C1 N1(C(COCCOCC)=O)CC2CC1CN(C(=O)Cn1cc(C(F)(F)F)nn1)C2 C1(NC(CCOC(C)C)=O)CCCN(C(=O)C(C)S(C)(=O)=O)CC1 N1(C(CC(C(C)OC)NC(=O)Cc2ccc[nH]2)=O)Cc2ccc(C)nc2C1 C1(NC(C(CC2CCC2)NC(=O)Cn2cnnc2O)=O)CCC2(CCC2)C1 C(=O)(CC(O)CC(C)(C)C)NC1CC2(C(NC(CN(C(CCC)=O)CC)=O)C2)C1 N1(C(C(C)(C)SC)=O)CC2(CCN(C(=O)C=Cc3ccc4c(c3)CCO4)CC2)C1 N1(C(CC(C)=O)=O)CC(NCc2cc(Cl)cnc2F)C(C#N)C1 C1(C(N2CCC(NC(c3c(C)onc3)=O)C23CCC3)=O)Cc2cc(Cl)ccc2O1 N1(C(c2c(C)[nH]c(C#N)c2)=O)CC2(CCCC2NC(=O)CC(Cl)Cl)C1 N1(C(=O)Nc2c(OCC(=O)NC)cccc2)CC2(CCO)CCCC2(F)C1 CC1CN(C(=O)COc2ccc(Br)cc2)CC1NC(=O)CC1CCCO1 Cc1cc(CCC(=O)NC2CC(N(C)C(C3(C#N)CC4CC4C3)=O)C2)ccc1Cl Cn1cnc2cnc(N3CC=CC(NC(c4cc(C(F)(F)F)ccn4)=O)C3)nc12 C1(NC(=O)COc2ccccc2F)CCC12CCCNC2 C(c1cncc(F)c1)=CCN(c1cncc(Cl)c1)CCC(C)(C)C1CC1.C1=NC1 C(N=c1nc(C2CC2)[nH]s1)C1C(C(F)(F)F)CN(C(c2cccc(OC)n2)=O)C1 N1(C(c2cn(C)c(=O)cc2)=O)CCC2(C1)CN(C(C1CC3CCC13)=O)C2 C1(NC(c2ncn(CC)c2)=O)CC(SC(C)(C)C)CC1O CCC(CC(F)F)C(=O)NC(C)CNC(C12CC(C1)C(C(F)(F)F)O2)=O C(=O)(C1=C(C)S(=O)(=O)CC1)N1CC(C)CC(CNC(CC(C)OC)=O)C1 N1(C(C(c2cccs2)SC)=O)CC(C2CN(C(=O)CC3COC(C)(C)C3)C2)C1 Cc1ccc(O)c(NC(c2csc(-c3cnn(CC#N)c3)n2)=O)n1 N1(C(C(N2CCC(C)(C(N)=O)C2)=O)=O)CC(C(=O)O)C2(CCCCCC2(F)F)C1 N1(C(C)=O)CCCN(CC(=O)N(C(C)C)CC2CCC(OCCO)C2)CC1 C(=O)(C(C)CNC(c1coc(NC(=O)CNC(=O)C(C)(C)C)n1)=O)NC C1(NC(C(=O)NCCNC(C)=O)=O)C2CCN(C(c3ccc(C(C)C)s3)=O)C12 c1(C(C)SCc2ccc(C(F)(F)F)s2)ccccc1.C(=O)(CSC(C)(C)C)NC C1(CC)C(NC(=O)CCCN2CCCC2)CCCN1C(C1CC1c1nc[nH]n1)=O C(=O)(C(F)C(C)(C)O)N(C1CC(NC(c2ccc(C(F)F)cc2)=O)C1)C C=CCCC(=O)NC1CC(C)(NC(=O)CCSc2nccn2C)C1 N1(CC)CCC(NC(C2C3CC4C(C3NC(=O)C(C)SC)C24)=O)C(C)C1 Cc1cc(C(=O)NC2CCCC2CNC(=O)CC2CCCN2C)c(Cl)cc1N c1(C(=O)NCCN(C(c2cc(CC(C)C)on2)=O)C)ccnn(C)c1=O C1(NC(C(C)(C)OC)=O)CN(C(=O)C(F)(F)c2csc(=N)[nH]2)CC1C CC1(C)CCc2cc(C#N)c(N3CC(CC(C)NC(=O)CCC4CC4)C3)nc2C1 CCC(C)C(C(=O)NC1(CNC(c2ccc(O)c(C(C)(C)C)c2)=O)CC1)OC n1(CC)ncc(Br)c1C(=O)NC(C)C(C(C)C)NC(=O)C#CC1CC1 S(=O)(=O)(c1cccc2c(N(CCC#N)C(C)=O)cccc12)N1C(C)(CC)CC1 c1(OC)nc(C)cc(=NC2CC3CN(C(c4ccccc4C)=O)CC23)[nH]1 N1(C(C2C(C=C)CC2)=O)CCC(CN(C)C(c2cc(CS(C)(=O)=O)on2)=O)CC1 c1(OCC)cc(C(N2CCSC(C)(C)C2)C(=O)NCC2CC2)cc(Br)c1OC C(=O)(C(O)CC(F)(F)F)NCC1CCC(CN(C(Cn2ncc(C)c2)=O)C)CC1 Cc1nc2c(C(N3CC4CC(NC(C5(CF)CC5)=O)CC(C4)C3)=O)ccnc2[nH]1 CCCCCCC(C)C(=O)NCC1(C)CN(C(=O)CN(C)CC)CCO1 Nc1c(C(N2CCC(CCNC(=O)C(F)=C3CCCC3)C2)=O)ccnc1Cl c1(C(=O)NC2(CNC(C(C(C)C)O)=O)CCOC2)cnn2c1OCCC2 C1(OC)CC(C(=O)NCCc2ccncc2)N(C(C2CCCN2C2CC2)=O)C1 c1(C(N(C)CC2CCN(C(CCCCCC)=O)C2)=O)cc2c(C)cccc2[nH]1 c1(C(N2CC3CN(C(c4c(Cl)ccc(O)c4Cl)=O)C3C2)=O)cnc2ncccn12 C1(O)(C(=O)NC(C(N2CCC(SC)C2)=O)COC)CCCCC1 C(=O)(C(O)C(F)(F)F)NCCCCC(C)(C)NC(C(c1ccc(C)cc1)C)=O c1(CC(=O)NC(C(C)NC(C2(S(C)(=O)=O)CCC2)=O)CO)c[nH]c2cnccc12 C1(CC(=O)NC2CCC3(CCC3)C2)CCCN(C(=O)Cc2nc(O)n[nH]2)CC1 Cc1cc(Br)cnc1C(N1CCC(C(=O)Nc2cccc(Cl)c2C)C1)=O c1(C(N2CCCN(C(C3CC=C(C)CC3)=O)C2CO)=O)ccc(Cl)c2occc12 C1(CNC(C(C)OC)=O)CC2(CO1)CN(c1ncnc3ccsc13)C2 N1(C(c2[nH]cc(C(C)=O)c2C)=O)CC(NC(=O)C(C#N)C(C)(C)C)C2(CCC2)C1 C1(NC(C(c2ccco2)NC(=O)C=CCN2CCC2)=O)CCCC12CC2 C(=O)(CC(C)(O)C1CC1)N(C)CC1CN(C(=O)C=C2CCCC2)C1 N1(C(CC(CC#C)c2ccccc2)=O)CC(NC(c2cnns2)=O)CC(C)(C)C1 c1(CC(=O)NCCNC(=O)C=CCOCC(F)(F)F)cc(F)ccc1Cl c1(CC)cc(C(=O)NC(C)CC(C)NC(=O)CC2(CO)CC2)on1 c1(OC)ccccc1CN(C)S(=O)(=O)Oc1cnn(-c2ccc(F)cc2)c1 C1(C(F)(F)C(=O)NCC(C)(C(C)C)NC(=O)COC(C)=O)(OC)CCOCC1.C(C)(=O)O C1(COC)CCCN(c2cc(NCc3cccc(F)c3)ncn2)C1 Cc1cc(Cl)cc(N)c1C(=O)N(C)CCNC(c1ccnc(OC(F)F)c1)=O N1(C(CC2C(CC)C2)=O)CC(C)CCC1C(N1CCC(SC)CC1)=O C1(C)(CNC(c2sc(C)c(O)n2)=O)CC(F)(F)CN1C(c1ccc(C(F)F)o1)=O CCCCC(CC)C(=O)N(CCC(=O)N(C)CC1(O)CCCC1)C Cn1c(=O)ccn(CC(=O)NC2CC(NC(=O)CC3CC(C)(C)OC3=O)C2)c1=O c1(C(N(CCNC(=O)C2=CC3CCCC23)CC)=O)cc2sc(=O)n(C)c2s1 c1(OC)cc(C(=O)NC2CC(=O)N(OC(C)C)C2)ccc1[N+](=O)[O-] c1(NC(c2ccc(Br)o2)=O)cncc(C2CC2C(=O)O)c1 C1(CN(C(C2(OC)CCOC2)=O)C)CCCN(C(=O)C(C)(C)c2ccno2)C1 C1(C)(NC(COCCN(C)C)=O)CCCCC1C(=O)NC1CC(C)(C)OC1=O c1(OC)cccc(C(N2CC=CC2CNC(c2sncc2C)=O)=O)c1N CC1CC2(CCN(C(c3ccc(N)cn3)=O)CC2)CN1C(=O)CCc1ccsc1 N1(C(c2ccn(CC)c2C)=O)CCC(NC(=O)CCn2cccn2)C(O)C1 c1(C(N2CC=CC(NC(c3cccc[n+]3[O-])=O)C2)=O)ccc(=O)n2c1COCC2 C(=O)(CC(CC)C(C)C)NCC1N(C(CC(=C=C)C)=O)CC(C)C1 C1(C(=O)NCC(CN(C(C(C)(c2ccccc2)OC)=O)C)C)CC2(C1)CC2(F)F C1(CN(C(=O)CC2CC(OC)C2)CC)CCCCN1C(C1CS(=O)C1)=O n1(CC)c(CNC(=O)C(C)N(C(=O)Cc2cnoc2)C2CC2)nnc1O c1(C(=O)NCCCN(C(CNC(C)=O)=O)C)ccc(S(=O)(=O)NC(C)=O)s1 C(=O)(CC(F)(F)C(F)F)NC1C2(CN(C(C(C)OCC(F)(F)F)=O)C2)CC1 CCC(CC)CC(=O)NCC1CCN1C(=O)C(C1(O)CCCC1)F CN1CC2COC(CNC(=O)C(=O)NCC(N3CCOCC3)(C)C)C2C1 c12sc3c(c1C(=O)N2)CCCC3.CC1CCCN(C(C2CCC(F)(F)C2)=O)C1 C#Cc1ccc(Cl)c(C(=O)NC2CCN(C(=O)CSC3CCCCO3)CC2)c1 CCCCC(O)C(C)C(=O)N1CCC(OCCNC(C2CCCO2)=O)C1 N1(C(c2ccc(C)s2)=O)CC(C(=O)NCCS(C)(=N)=O)C(F)C1 c1(CN2CCCC(NCCn3ncc(C#N)c3)CC2)[nH]nc2c(F)cccc12 c1(C(=O)Nc2c(CC)cc(F)cc2)cc(N(C)C)ccc1F.C12CC(C1)NC2=O CCCCCCCC(=O)NCC1C(CC)CCN1C(=O)CCN1CCC(F)C1 C(=O)(C(C)CC(C)C)N1CC(CC(=O)NC2(CCC)CCC2)OCC1 N1(C(C23CC(OC)C2C3)=O)CC(NC(c2nc(C)ncc2Cl)=O)C2(CC2)C1 n1(CCC)nnnc1CC1CCCN1C(N(CCOCc1ccncc1)C(C)C)=O c1(C(=O)NCC(COC)NC(=O)CN2CCC(CO)CC2)c(C)ncn(C)c1=O CC(C)C(C#N)C(=O)NCC(C1CCCC1)NC(C1CCN(C(N)=O)CC1)=O c1(OC)ncc(C(N2CCC(C)(NC(=O)Cc3nnc(C)o3)CC2)=O)cc1Br c1(CC)c(C(=O)NC(c2nocc2C(=O)NCC(C)(O)CO)C)ccn1C N1(C(c2cnc(C)nc2C)=O)CCC2(CC1)CN(C(=O)CCSCC(N)=O)C2 c1(CC(N2CC3C(CNC(=O)COCC(F)F)(C3)C2)=O)ccnc(F)c1F CC1CN(C(c2ccc(-c3nc[nH]n3)nc2)=O)CC1NC(=O)CCC1(C)CC1 CC(=NO)c1cc(C(N2CC(O)(CNC(=O)COCCN(C)C)C2)=O)cnc1O Cc1cc(C(N2CC(NC(=O)CC3CCC3)C2)=O)nn1C(C)C1CC1 CC1(C)CC(NC(c2cnco2)=O)CCN(C(C23CCCC2C3Br)=O)C1 S(=O)(=O)(c1cc(Cl)ccc1F)NC1CCC(C(N2CCCC3(CCOC3)C2)=O)OC1 N1(C(C(C)CC2CC2)=O)CCC2(CC2C(=O)NCc2cccc(Cl)c2)C1 CC(C)C(C(=O)NCC1CCN(C(=O)CNc2ccsn2)C1(C)C)C(C)C C1(C)(C(=O)NCC(CNC(CC(=O)NCC)=O)C)CC(C#N)C1 c1(C(=O)NC2CC3N(C(CCCC#CC)=O)C(CC3)C2)cc(S(C)(=O)=O)oc1C C1(C)(C(N2C(CNC(CCCn3ncc(C)c3)=O)CC2)=O)COC(C)(C)CO1 c1(CN2C(CC(=O)Nc3ccc(OC)nc3C)CCC2)cccc2[nH]ncc12 C(=O)(C(C)(C)CN(C)C(c1cccc(CO)c1)=O)NCC(C(=O)NC)C Cc1ccc(C)c(C(=O)N(C)CC2CCCN2C(C2CC3CCCC3C2)=O)n1 c1(C(=O)NCC(CNC(c2cc(CC)oc2C)=O)C)cnc(O)c(C(F)(F)F)c1 C1(NC(C=CCN(C)C(c2cc(Cl)ns2)=O)=O)CCC(O)C(O)C1 C1(CC(=O)Nc2ccc(C(C)C)s2)CCCOCC1.C12CC1C(=O)NC2 C1(COC)(NC(C2COCC2C(N)=O)=O)CCN(C(=O)C(C)CS(C)=O)CC1 N1(C(C2C(C(=O)OC)C2(C)C)=O)CCC(NC(=O)C(C)NC(N)=O)CC1 c1(CCNC(N2CCOC(CN3CCOCC3)C2)=O)ccc2sccc2c1 CC1(CNC(=O)CCCn2ccnc2)CCC(NC(=O)C(F)F)CC1 C1(CC)CN(C(=O)CSc2nnc(C3CC3)o2)CCN1C(=O)C(CO)NC(N)=O C1(NC(c2ncn(C)c2)=O)CCCN(C(=O)CN2CCSCC2)CC1F c1(CC(=O)NCC2(NC(CS(CC)(=O)=O)=O)CCOC2)cc2ccccc2s1 c1(C(N2CCC(N(C(=O)COCC)CCC)C2)=O)oc2ccccc2c1C c1(C(C(=O)NCC2C(C(=O)NCC#CCOC)OCC2)O)ccc(Cl)cc1 c1(NC(C)=O)nc(C)c(S(=O)(=O)NC2CN(C(c3ccc(C)nc3)=O)C2)s1 C(CS(=O)(=O)CC(=O)N(CCCOCCNC(c1cocc1C)=O)C)OC c1(OCC)ccc(F)c2c1CCN(CC(F)(F)C(F)(F)F)C2 C=C(Br)CCC(=O)NCC(c1ccccc1)NC(C12CCC(CC1)C2)=O C(N=c1[nH]c2c(c(=NC3CCC4(CCC4)CC3)[nH]1)SCC2)C1(C)CC(C)C1 c1(C(N(C)CC2CCN(C(C(CC)F)=O)CC2)=O)cccc2nc[nH]c12 c1(NC(=O)NC(C)CCC2CCC2)nnc(SCO)s1.C(=O)(C(Cl)Cl)N c1(C(=O)NCCC2CC(C(=O)NCC(CO)n3cccn3)C2)cc(C2CC2)no1 C1(CC)C(C(N2CCC(OC(C)=O)CC2)=O)CCCN1C(=O)C(C1CC1)OC N1(C(c2c(C(C)C)c[nH]n2)=O)CC2CC(NC(=O)C3=CCCOC3)CC(C2)C1 CCC(C(=O)NCC1COC(CNC(=O)CC2CC=CC2)C1)C1CCC(=O)N1 CC1Cc2cccc(C(N3CC=CC(NC(=O)Cc4cnc[nH]4)C3)=O)c2O1 C1(NC(CC=C(C)C)=O)CCN(Cc2cn(C)nc2C)CC1F C12(CNC(C(C)SCC)=O)CC(CC)(CN1C(=O)COC1(C)CCOCC1)C2 Cc1cc(C(N2C(C)C3CC2C3NC(=O)C(O)CCN(C)C)=O)c(C)c(C)c1 C1(C(=O)CN)CCC2(CCC2)O1.c1(OC)c(C(=O)NCC2CC3CCC2O3)cnn1C c1(C(=O)NC2CN(C(c3cc(C4(C)CC4)on3)=O)C2)c[nH]c2ncc(Br)cc12 c1(CC)ccc(F)cc1C(=O)N(C)CC1CCCN(C(=O)COC2CC2(F)F)C1 c1(CNC(CC2(C)CC2)(C)C(=O)O)cc(C(=O)O)ccc1F n1(CC)cc(C(=O)NCC(O)CCNC(C2CCC2)=O)c(C(C)(C)C#N)n1 c1(COC(=O)NCCc2ccc(C)cc2)ccc(C(F)(F)F)c(C)n1 C(=O)(C1=CCCCCC1)NCC1C(CC(N2C(C)(C(=O)OC)CC2)=O)C1 N1(C(C2(OC)CC2)=O)CC(NC(=O)CC=C(C)C)C2CCCC2C1 Cc1ccc2c(c1)SC(C(=O)N(C)CC1(O)CCN(C(C3(C)CC3)=O)CC1)C2 C1(C(=O)NC2CC(C)CN(C(=O)C(C)(C)n3cnnn3)C2)CC2(C1)CC1(CC1)C2 CCCCC(=O)C(=O)NC1COCCC1NC(c1cn(C)nc1CC)=O N1(C(C=CC(CC)=CC)=O)CCCC(NC(=O)Cc2ncoc2C)C1C C1(CNC(c2nc(CC)sc2N)=O)CN(C(c2c[nH]nc2C(F)F)=O)C(C)(C)C1 c1(CC(=O)N(CCC=C=CC)CC)cnc(-c2ccccc2)nc1 N1(C(CCCC)=O)CC2(CNC(C3(Cl)CC3)=O)CCC1CC2 C#Cc1cc(C(=O)NCC(CNC(=O)C(C(C)C)NC=O)C(F)(F)F)cc(N)c1 Cc1cc(C)n(CC(=O)NCCC2CC(C(=O)NC3(CCN=[N+]=[N-])CC3)C2)n1 C1(C(=O)NCC(C)CN(C)C(c2cnsc2)=O)CC2CCC(C1)N2C C1(NC(CN(C(C)=O)C)=O)CCCN(C(c2cn(C(C)C)nc2Br)=O)C1 N1(C(CC)CC)CC(C(=O)NCC(C)NC(c2cc(C3CCC3)on2)=O)CC1=O c1(CNC2C(C(N3C(CC)CCC3)=O)C2)cc(O)cc2ccccc12 Cn1[nH]c(C(=O)NC2(C)CCN(C(C3(C)CCCO3)=O)C2)nc1=O c1(NC(CN2CCN(Cc3c(CC)cc(O)cc3)CC2)=O)c(F)cc(Br)cc1Br CN=c1[nH]c(=NCCOC(C)C)[nH]c(=NCC2CC2C2CCCCC2)[nH]1 c1(C(=O)NC(CCCNC(C2CC=C(C)CC2)=O)C)cc2ccccc2s1 c1(OC)cnc(C(N2CCOCC2CNC(c2conc2C2CCC2)=O)=O)nc1 Cc1cc(CN2CCC(C(=O)Nc3ncc(C)cc3C(F)(F)F)C2)cc(F)c1 C1(CCC)CN(C(C2CC2c2cnc[nH]2)=O)CCN1C(=O)C=CC(C)(C)SC N1(C(CNC(C=C)=O)=O)CC2CCN(C(c3cc(Cl)c(Cl)cn3)=O)CC2C1 C12(CNC(C3OCCC(C)C3)=O)CCC(CN(C(c3ccc(O)nc3)=O)C1)C2 c1(C(=O)NCCN(CCCN(C)C)C(C23CCC(CC2)O3)=O)nc[nH]c2nccc1-2 C1(C(N2CC=CC2)=O)(CO)CC12CCC2.N1(C(CN(C(=O)OC)C)=O)CCCC1CN N1(C(C(CC)n2cccn2)=O)CCC2(CNC(=O)CN3CC=CC3)CCCCC12 C(=O)(C(C(C)CC)N(C)C(c1snnc1CC)=O)NC(C#C)C(C)(C)C CC1(CC(=O)NC2CCC2NC(C2(C)CCCO2)=O)CC1(F)F N1(C(CC=C)=O)CCC2(CC1)CN(C(=O)COc1cc(C)ccc1C)CC2O c1(C(=O)NC(CC)CNC(=O)Cc2ccsn2)cc(C2CCCO2)n(C)n1 c1(OC)cc(NC(C2(NC(=O)C(c3ccccc3)C)CC2)=O)cc(Cl)n1 C1(C(N(OC)C)=O)CC(NC(=O)CCc2cc(C)[nH]n2)C1(C)C CCC(CN(C)C)CC(=O)NCC1(F)CCN(C(=O)CCC2OCCO2)C1 c1(-c2ccc(C)c(C)c2)ccc2oc(=O)c(C(=O)N(C3CCC3)CCO)cc2c1 Cc1ccsc1CC(=O)NC(Cc1ccoc1)C(=O)NC(C(O)CO)C1CC1 c1(-c2cn(C(C)CNC(c3c(I)cnn3C)=O)nn2)ccncc1C c1(NC(C(C(C)O)NC(CCCCC=C)=O)=O)ccc2ncccc2c1 C(N=c1[nH]c(=N)[nH]c(=NC(C)c2cnc(Cl)c(Cl)c2)[nH]1)c1cccc(OCC)n1 N#CCCCCC(=O)N1CCCC(CN(C(C2CCSC2)=O)Cc2cccnc2)C1 N1(C(C2=CN(C(=O)OCC(C)(C)C)CC2)=O)CC2OC(=O)N(C)C2C1 N1(C(C2(C)CC(NC(C3(C)CC=CCC3)=O)C2)=O)CC(C)(C)C1c1ccccc1 c1(OCC(=O)NC2COCC2NC(c2cc(O)cs2)=O)cc(F)cc(Cl)c1 C(c1ccc(F)nc1)=CC(N1C(CNC(c2ccn(CCOC)n2)=O)CCC1)=O C(=O)(CC(C(F)(F)F)NC(c1cccc2c1CCC2)=O)N(C(C(C)SC)C)C C1(NC(COCc2cccc(C)c2)=O)C2CC(O)C1N(C(c1cc(C)co1)=O)C2 CC1(C)CN(C(C2CC(F)CN(C(c3cccc(=O)n3O)=O)C2)=O)CCCO1 C(=O)(C(COC)CC(C)C)N1CC(C=C)(CC(N2CCS(=O)CC2C)=O)C1 N1(CCCC)C(=O)NC(c2c(Cl)ccnc2Cl)C(C(=O)OC)=C1c1ccc(F)cc1 Cc1[nH]c(=N)ccc1C=CC(N1CCC(C2CC2)C1CNC(c1cnc[nH]1)=O)=O c1(C(=O)NC2C(NC(C3N(C(C(C)C)=O)CCC3)=O)C2)ccc(Cl)c(N)c1 C(=O)(CCCCC(C)=O)N1C(C(=O)N(CCN=[N+]=[N-])C)(COC)C=CC1 CC1CCN(C(=O)C(C(C)(C)C)NC(c2ccc(S(C)=O)o2)=O)CC1(F)F C(=O)(C(C)(C)CS(C)(=O)=O)NCc1nc(CNC(CCCC(=O)OCC)=O)sc1 N1(C(CN2CCC(C)CC2)=O)CCC(NC(c2cc(O)no2)=O)CC1C c1(OC)cccc(F)c1C(=O)NCCC1CC(NC(=O)CC2CC(C)=NO2)C1 N1(C(C(CCF)NC(C2CC(SC)C2)=O)=O)CCC(C2CC2)C1 c1(N(C)CCN(C)CCOC(C)(C)C)nc2cc[nH]c2c(=NCCOC)[nH]1 C1(c2nnnn2C)(NC2CCC(c3n(C)ncn3)CC2)CC2C=CCC12 Cc1ccc2c(c1)CC(C(=O)NCC(O)CNC(c1cc(Br)nn1C)=O)S2 C(CC1=CCOCC1)N1CCCC(C(=O)NC2C(c3ccccc3F)(C)C2)C1 C1(C(N(CC)Cc2cncn2C)=O)CC=CCN1C(=O)C1=COCC1 CC(C)C1=NOC(C(=O)NCC(=C2CN(C(=O)Cc3ccc(CO)cc3)C2)F)C1 C(=O)(C1=C(C)CCOC1)N1CCC(N(C(=O)CC2CCCCC2(C)C)CCC)C1 c1(C(N(C2CCN(C(C(c3cnn(C)c3)OC)=O)C2)C)=O)ccc(C)n1C CN1CCC(NC(N2CCCC(C(=O)NCc3nccc(O)n3)C2)=O)CC1 N1(C(C(c2cnn(C)c2)C)=O)CC(C)C(C)(CNC(=O)CN2CCCCC2=O)C1 C(=O)(CC(C(F)(F)F)n1ccnc1)NC(CNC(CNC(CCCCC)=O)=O)(C)C C(=O)(CCC(C)(C)N(C)C)N1CC(CC(C(=O)NC2CCC(=C)CC2)F)C1 C12(NC(CC=C)=O)CC1CN(C(C1CCN(C3CC3)CC1)=O)C2 Cc1cc(C(N2CCC(C)(CC(=O)NCC3(C)CCN(C)C3)C2)=O)nc(C)n1 C=CCCCC(C(=O)NCCCC1CCOC1=O)NC(C1OCCC1CC)=O N1(C(CCCC(=C)C)=O)CCCC2(CC(NC(=O)CSc3ccncc3)CO2)C1 C(=O)(C1CCc2nccn21)NC1(C(=O)NCC#CCC)CCCC1C N1(C(C2CCC(=O)N2)=O)CCC(CO)(NC(c2ccc(C3CC3)nc2O)=O)CC1 c1(OC)ccc(C(=O)NC2CC(N(C(=O)C(O)CC(C)C)C)C2)c(Br)c1 C(=O)(C1OCCc2c(-c3nc(C4CC4)nn3-c3ccnc4[nH]ccc34)cccc21)OC N1(C(C(COCC)NC(c2cccc(CC)c2)=O)=O)CC2(CCC2(C)C)C1 CCCC(CC)CC(=O)NCCC(C)(C)NC(=O)C=Cc1nccn1CC CCCC(CC(C)C)C(=O)N1CC2(C(=O)NCC3CC(=C4CC4)C3)CC1CO2 c1(C(=O)NC2(CCO)CCOC2)ccccc1S(=O)(=O)NCc1nc[nH]n1 c1(C(N2CCC(C3(C)N=N3)CC2)=O)cnc2c(c1)NCCO2 C(C(C)(C)C(=O)C(C)C)N(C1C(O)CCN(C(Cc2scc(C)c2)=O)C1)C CCN=c1[nH]cc(C(=O)N(CC(C)CNC(=O)C(C)(C2CC2)OC)C)s1 C1(CNC(C(C)OCCC#C)=O)CCN(C(c2c(N)cccc2F)=O)CC1C C(=O)(CC(C)CC(=O)N(C)CCN(C(=O)CCCOc1ccccc1)C)OC c1(NC(c2cc(C)oc2C)c2n(CCCC)nnn2)ccc(Br)c(C(F)(F)F)c1 C1(NC(c2c(C)cccc2F)=O)CC2CCC(C1F)N2C(=O)CC1(O)CCOC1 N1(C(c2ccc(C3CC3)o2)C(=O)NCCC#N)CCCC(N2CC3CC3C2)C1 Cc1cc(I)c(F)cc1C(=O)NCCC1CCCN(C(c2ccncc2)=O)C1 N1(C(Cn2c(C)nnn2)=O)CCC2(CC1)CCN(C(C1CCCC(F)C1)=O)C2 c1(C(=O)NC(C)CNC(=O)CCn2cnc(=N)[nH]2)c(S(C)(=O)=O)cnn1C C1(NC(CCC=CC)=O)CC2(NC(c3ncc(Br)cc3C)=O)COC1C2 c1(CN2CC(CC)N(C(C3CC(C)(C)C3)=O)CC2)ccc2c(c1)CCCO2 C(C(=O)Nc1ccccc1C)(C(C)CC)N(C(CCC)CCO)C1CC1 c1(NC(C)=O)cccc(C#N)c1.C1(CNC=O)C=CCN1C(=O)C(C)c1cc[nH]n1 CC(C(=O)NCC1CC(NC(=O)CCc2cnco2)C1)C(C)S(C)(=O)=O CC(CC(C)(C)O)NC(c1cc(N(C)CCO)ccn1)=O c1(C(=O)NCCN(C(c2n(CC)ncn2)=O)C2CC2)cc2c(s1)COCC2 C1(COC)CC(C(=O)NCC(C)(CO)SC)N(C(=O)COc2cnn(C)c2)C1 CN1CCN(C(c2cc(O)cc(Cl)c2)=O)CC1CNC(=O)C(F)n1cccn1 C1(C)(C(=O)NCC(C(=O)NC)O)CCN(C(=O)C(C)=C(C)C)CC1 c1(CNC(C2CC(OC)CN2C(=O)C(C)(C)CCF)=O)cc(C)cc(C)n1 c1(CN(C(C2CCCO2)C)C(c2ccccc2)=O)nnc(S)nc1O Cc1[nH]nc2c(C(=O)N(C)CC3C4CN(C(C5COC(=O)N5)=O)CC34)cccc12 N1(C(C2CNC(=O)N2)=O)CCN(C(c2ccc(C(F)(F)F)cn2)=O)CC1C(F)F C(=O)(CS(=O)(=O)C1CC1)NCC1CN(C(C(CC=C)(C)C)=O)CC1C c1(C(=O)NCC(C)N(C(=O)CCc2ncco2)CC)n[nH]c2c1CC(C)CC2 CC1CN(C(c2cc(=NS(C)(=O)=O)cc[nH]2)=O)Cc2ccc(Br)cc2O1 c1(C(=O)NC(CN(C(c2c(C)nc(C)o2)=O)C)C)c(C2CCCC2)cccc1F C1(NC(c2cc(CC)nnc2C)=O)(CO)CCN(C(C2SCCC2C)=O)CC1 C(=O)(CCCC#CC)NC(C(=O)NC(C1CCOC1)C#C)CCF C1(NC(c2ncc(OC)nc2)=O)CCN(C(=O)CC2CC2(Cl)Cl)CC1F N1(C(C(CC)NC)=O)CCC2CN(C(c3cc(Cl)on3)=O)CC2CC1 c1(C(N2CC(O)(CCNC(CC(CCCC)O)=O)C2)=O)cnc2ccnn2c1N c1(CNC2C(C(=O)Nc3nc(O)cc(OC)n3)C2)cc(C#N)ccc1Cl C(=O)(CC1=CCCCC1)N1C(CC(=O)N(CC(F)F)CCO)CC(O)C1 N1(C(Cc2c(C)non2)=O)CCCC2C(NC(=O)CCC3CCCC3)C(C)(C)C12 CCCC(CNC(=O)C(CCSC)NC(=O)Cn1c(C)ccc1C)CCO N1(C(C23CC(C)C2C3)=O)CC(NC(C2NC(=O)OC2(C)C)=O)CC12CCC2 N1(C(C(C)SCC)=O)CCN(C(=O)C2=NN(CCOC)C(=O)CC2)CC2(CC2)C1 c1(CC(=O)NC2C3CC4C(C3=O)C24)cn2ccsc2n1.C1CCN(C)N1C c1(OC)cc[n+]([O-])c(C(=O)NCCN(C)C(c2ccc(-n3ccnc3)cc2)=O)c1 C#CCCCCCCC(=O)NC1CCCC1C(=O)NCC1CC(C(=O)OC)C1 c1(C(=O)NC2CCC(NC(C(CC#C)O)=O)C2)ccnc2ccc(O)cc12 CC1CCN(C(=O)CCc2ccccn2)C(C)C1NC(c1cnc(S)n1C)=O N1(C(c2c(C)n[nH]c2)=O)CCCCC(NC(C2C=CC=CC=C2)=O)C1 C(=O)(CS(=O)(=O)CCO)N1CC(NC(C2(CCC=C)CCCC2)=O)C(C)CC1 c1(C(N(CC(C)NC(C(C)CC(F)F)=O)C)=O)cn2c(n1)CCCC2 C1(C(=O)NC2CC(F)(F)C2)(CNC(=O)CN2C(=O)CNC2=O)CCCCC1 C1(C(=O)NC(C2CCN(C(C3(F)CCOC3)=O)CC2)C)CCC(C)(C)CC1 c1(-c2c(NC(N3CCN(c4ccn(C)n4)CC3)=O)ccs2)cc2ncccc2[nH]1 C1(NC(C(C(C)O)(F)F)=O)CCN(C(=O)Cn2ccc(=O)n(C)c2=O)CC(O)C1 C1(F)(C(=O)NC2C(NC(C3CCN(C(=O)NC)C3)=O)CC2)CCCOC1 N1(C(CC(C)(C)C#N)=O)CCCC2(CCN(C(c3ccn4c3CCCC4)=O)C2)C1 C(=O)(C(c1ccccc1)=CC(C)(C)C)NC1(C)CN(C(C2C(C(C)O)C2)=O)C1 Cc1cc(Cl)ncc1S(=O)(=O)N1CCC(NC(c2ccc(F)c(F)c2)=O)C1 C1(C2CCN(C(=O)Cc3nccs3)CC2)(NC(C(CC(C)C)F)=O)CC1 C1(N(C(=O)C=CC=C(Cl)Cl)C)CCC(NC(=O)CCSC(F)(F)F)C1 C12(CCCC1)C(=O)O2.c1(C(N(CCC(=O)N(C)C)C)=O)ccccc1 c1(C(=O)NCC2(CC(=O)NCC(C#C)CC)CC2)cnn2c1OCC2 c1(OC)cc2c(cc1Cl)CN(C(c1ccc(C)nc1C)=O)CC2 C(=O)(CCCC(=O)NC1CC(O)CN1C(=O)CNC(=O)OC(C)(C)C)NC(C)C C(=O)(C(O)CC(C)C)N1CC(F)(C(N2CCN(CCC)CC2)=O)C1 CCCCC(C)(CC)NC(=O)C(O)C1CN(C(C2CCC(CC)O2)=O)C1 N1(C(C(c2cnn(C)c2)OC)=O)CC2CC(NC(c3cc(=O)cc[nH]3)=O)C2C1 C12(C(=O)NCC(C)N(C(=O)C3=C(Cl)CCCC3)CC)CCCCC1NC(=O)C2 N12CCC3CN(CC3C1)Cc1ccccc1C=C(C#N)C(CC)(COCC)C2=O CON(C(=O)C(C)NC(C1CCCC(=O)N1C)=O)C1CCC1 c1(NC(C2(O)CCN(Cc3c(C)n(C)nc3)C2)=O)cc(Cl)ccc1I N1(C(C(C(CC)C)N(C(=O)CC2CC2)C)=O)CC2(CCNC(=O)O2)C1 CCC(CC)(CC)C(=O)N1CC(=C(F)CNC(=O)CC2CC(F)C2)C1 CCC(CC(=O)N(C)CCC1CCN(C(C2CCC2(C)C)=O)CC1)OC Cc1cc(F)c(CC(N2CC3(NC(=O)C=Cc4cocn4)CCC2C3)=O)cc1F C(CC(CC)C(=O)NC(C)CCNC(c1cccc(-n2cncn2)c1)=O)=CC C(CCCC)(CCC)NC(c1n(CCCCCC)nnn1)c1cnn[nH]1 C=CC(F)(F)C(=O)NCC1CCCC(NC(=O)CN2CCCCC2C)C1 N1(C(C(C)SCC)=O)CCOC2CCN(C(c3cc(Br)ccn3)=O)CC12 C1(CC(=O)NCCCC=CC)CC(C)N(C(=O)CCSCC)C1 C=CCCCCCC(=O)NC(CNC(=O)CCn1cnccc1=O)C1CC1 O=C(CC1=CCOCC1)NCCN1CCN(C(C2CS(=O)(=O)CC23CC3)=O)CC1 C(=O)(C(O)CC(F)(F)F)N1CCC(C2C(NC(C(C)(C)CCC)=O)CCO2)CC1 Cc1ccc(Cl)c(F)c1C(=O)NCC1CN(C(=O)Cc2ccno2)CC12CC2 c1(C(=O)NC(C)CCN(C)C(C2CC(F)(F)C2)=O)cc2c(cn1)OCCO2 N1(C(CC(C)(C)NC(CCC(C)OCC)=O)=O)CC2CCCC2C1 N1(C(CCc2onc(C(C)C)n2)=O)CC2CCC(NC(=O)CCS(C)=O)(C2)C1 C=C1CCN(C(C2CCCC3(CC3)C2)=O)C(C(=O)NCC2CC(O)C(O)C2)C1 c1(C(=O)NC(C(C(C)C)NC(=O)CN2CCSCC2)C)cc(F)c(F)c(F)c1 c1(C(C)(F)F)cncc(C(=O)NCC2CCC2NC(C2CC23CCC3)=O)c1 C#CCCCC(=O)N(CC1Cc2c(cnn2CC)C(=O)N1)C.C(F)(F)F.OC C(=O)(CCCCCS(N)(=O)=O)NCC(CCNC(C(C)CO)=O)O CS(=O)c1ccc(CC(=O)NCC2(NC(c3cc(C(F)(F)F)c[nH]3)=O)CC2)cc1 N1(CCN(C(c2c(C)nc(C)[nH]2)C(=O)NCC(F)F)C)CCS(=O)(=O)CC1 Cc1ncc(C#N)c(NC(c2cc(Cl)ncc2Nc2ccncc2Br)=O)n1 c1(N2CCN(C(=O)NC3CCc4cnnn4C3)CC2)cccc2ccccc12 c1(NC2CCCC(NC(c3ccc(N(C)C)cc3)=O)C2)ccc([N+](=O)[O-])cc1 C1(CC(C)C)(C(N(C(CNC(C(CC)N(C)C)=O)C)C)=O)CCNC1=O c1(NCC)cncc(C(=O)NCCC2CCCCN2C(=O)CN2CC=CC2)c1 C1(NC(c2c(C)nsc2)=O)CCCCN(C(c2cccc(N)c2C(F)F)=O)C1 C1(NC(CC(CC)CC)=O)CC12CCC(NC(C1CCC(O)CN1C)=O)CC2 CCCC(C)(CC)C(=O)N1CCC(CCCNC(c2cn(CCO)nn2)=O)CC1 c1(C(C(=O)Nc2cccc(Cl)c2)N(CC#N)Cc2ccc(C)s2)cc(Br)ccc1Cl C12(NC(C(C)Sc3ccc(OC)cc3)=O)CCC(CC1)N(C(=O)C(C)(C)CO)C2 CCCCCCCC(=O)N1CCC(C)C1CNC(=O)Cc1ccc(OC)cn1 C1(O)(CCC)CCN(C(=O)C(C2CC2)N(C(=O)CCC2N=N2)C)CC1 c1(C(=O)NCC2(F)CCC(CNC(=O)CC3C=CCCC3)C2)cc2occc2[nH]1 C1(NC(C=C)C)CCC(=C2CCC2)CC1.c12ccc(cc1)NC(=O)c1nnnn1-2 C1(CNC(=O)C=C2CCC2)CN(C(=O)Cc2cnc3ncccn23)CC12CCC2 c1(CC(=O)OC2CCCCC2)cn2cc(F)ccc2n1 N1(C(C(=O)NC(C2(C)OCCO2)C)=O)CC(C(F)(F)F)C(F)(F)C1 C(=O)(C(CCC1CCC1)NC(C1CC1C(C)(C)C)=O)N1C(C)(COC)CC1 c1(OC)cc(C(=O)NC(C(=O)NCC2(CCO)CN(C)C2)C2CCCC2)sn1 c1(C(=O)NC2CCC(CC(N3CC(=O)NCC3)=O)CC2)cc(F)cc(F)c1F C=CCCCC(C(=O)N1CC(n2cccn2)C1)NC(c1cc(O)ncn1)=O c1(CNC(C(C(C)NC(CCCSC)=O)C)=O)nc(C)cc(C)n1 C=CC(C)(CC)C(=O)NC1(CNC(C2CCCC(C)(C)O2)=O)CCCC1 c1(C(C)C)nc(NCCn2cc(Br)cn2)cc(N2CC(NC(C)C)C3(CC3)C2)n1 c1(OC)cc(F)ccc1NC(C1(CF)CCC1)=O.C(C)(C)SCC.CC1CC1 C(=O)(CS(N)(=O)=O)NCC(c1cn(C)nc1)NC(c1cnnn1C1CC1)=O Cc1nc(-c2cccs2)sc1C(=O)NCCC1CC(NC(C2(N(C)C)CC2)=O)C1 C1(C(=O)NCC(CCOC)NC(C2(C)CCC2)=O)CCc2cnn(C)c2C1 C12(C(N3CC4C(NC(c5c(C)n6c(s5)ncc6)=O)C4C3)=O)CCC(CC1)C(C)O2 C(=O)(C(CCS(N)(=O)=O)NC(C)C)NCCOCCNC(Cn1nnc(C)n1)=O N1(C(CC(=C)C)=O)CC(NC(c2cncc(C(N)=O)c2)=O)C(C2CC2)C1 C1(SCC(=O)Nc2ccsc2Cl)CCN(Cc2cn(CCCC(=O)O)nn2)CC1 C1(C(=O)NC2(CN(C(CN(C(COC)=O)C)=O)C)CC2)C2CCCCCCC12 c1(CCC)nnsc1C(=O)N(C1CC1)CC1CCCN1C(C1CC1[N+](=O)[O-])=O c1(C(=O)NCC(CC)NC(=O)NC2(CC(F)(F)F)CC2)cc(-c2ccccc2)cs1 Cc1c(C(=O)N(C)CCNC(=O)CCOC(C)C)c(C)n2ccncc12 N1(C(c2cc(C(F)F)ccc2F)=O)CCC2CCCN(C(=O)CC=C(Cl)Cl)C2C1 N1(C(CN(C(C)C)C)=O)CCCC2(C1)CN(C(=O)C(c1ccc(Cl)c(Cl)c1)C)C2 C#Cc1ccc(NC(C2CCN(C(=O)CC3C(C)(C)C3(C)C)CC2)=O)cc1 c1(N2CCN(C(C(=O)NCC)=O)CC2)nc(N2CCSC(C)C2)nc2ccsc12 Cc1cc(C(N2CCC(C(C)NC(=O)C=CCn3cncn3)C2)=O)ccn1 c1(C(=O)OC)n[nH]c(=NC2(CNC(C3(C)CCC(C)C3(C)C)=O)CC2)s1 C(C(C)(C)CC(=O)NC1CC2CC1CC2NC(=O)CCOCC1CC1)N(C)C CC#CCCC(=O)NC(C1CCCCN1C(=O)CC1OCCCO1)C C1(CNC(CC(=O)NC)=O)CN(C(c2ccoc2Cl)=O)C2COCC2O1 c1(CC(=O)N(C)CC2CCCC2)ccco1 c1(CC(=O)N(CC(C)NC(C2CCC(OC)C2)=O)C)cccc(C(C)C)c1 C(C(=O)NCCCCC1CN(C(c2cc[nH]c2C(C)C)=O)C1)(C(C)C)NC(C)=O Cc1cnc2cc(C(N3CC4C(CNC(=O)C(C)(F)F)C4C3)=O)nn2c1 c1(C(=O)NC2C(NC(c3cc(C)ncc3)=O)CCC2)cncc2c1CCNC2=O Cn1nnc(C(=O)N(C2CCCCC2)CCNC(=O)CC2CCCCC2F)c1N CCC(C)(C)C(C)CC(=O)NCC1CCCN(C(c2cocc2C)=O)C1 C1(N(C)C)CC(F)(C(N2CCC(N3CC(O)C3)C2)=O)C1 C(=O)(C(F)CCC(C)C)NC1CN(C(c2c(OC)noc2C)=O)CC(C)C1 Cc1cccc(C(=O)NCC(C)(F)CNC(c2ccc(C3CCCO3)[nH]2)=O)n1 C1(CN(C(CCC2CC(NC(CCNC(=O)OC)=O)C2)=O)C)CCCCO1 c1(OCCC(=O)NCC2CCC(NC(CCOCC)=O)C2)ccc(F)cc1Cl C1(CC(=O)NCC(CNC(Cn2c(C)ncc2)=O)CO)CCC2(CCC2)O1 C1(CC=C)(NCCC2CCCN(C)C2)CCCNCC1 N1(C(C2C(C)(C)C2(F)F)=O)CC(NC(c2ccc(F)cc2N)=O)C2(CC2)C1 c1(C(=O)NC2CC(F)(CNC(c3ccc(CC)o3)=O)C2)cccc2occc12 C(CC(C(=O)N(C)CC1CC1(C)C)NC(c1cc(C)oc1C)=O)SC N12CC3(CCC(CC3)NC(=O)C1CC)C2.N1(C(C)C)CCc2nc[nH]c2C1 Cc1nn(C)c(C)c1CCC(=O)NC1CCCC1NC(C1CC(CCO)C1)=O c1(C(=O)NCC2(OC)CN(C)C2)n[nH]c2c1CN(C(c1ccc(F)cc1O)=O)C2 C(C(C(=O)N1CCOC(CCF)C1)C(C)(C)C)NC(CC1(NC(C)=O)CCC1)=O C1(CC)CCN(C(c2ncccc2N)=O)C1CNC(C1CCCC1F)=O C1(NC(C2C(CC)N(C(=O)Cc3cc(C)nn3C)CC2)=O)CCOC2(CCC2)C1 N1(C(c2cnn(CC)n2)=O)CC2(CC2)CC1CNC(c1cn(C)nc1C)=O c1(C(N2CCC(Nc3cn(CCOC)nc3)C2)=O)ccc(Br)c(OC(C)C)c1 C1(C(=O)NCC2N(C(c3ccc(COC(C)=O)cc3)=O)CC2)CC(C)OC(C)C1 C(=O)(CC(C)(C(F)F)N(C)C)N1CC(CNC(c2c(NC)cccn2)=O)C(O)C1 N1(C(c2c(C)scc2)=O)CC2(CCC2CNC(C2CN(C)CCN2C)=O)C1 N1(C(c2cc(CC)no2)=O)CCC2(CC1)CCN2C(=O)Cc1cncnc1 C(Cc1ccccc1)(CC(C)C)NC(C(Cc1ccccc1)OC)=O CCC(C)C(O)C(C)C(=O)N1CCC(C(=O)N2CC3CCC(C2)O3)=C(F)C1 C1(C(=O)NC(C)(C)CNC(C2(C(C)(F)F)CC2)=O)CCc2nnc(O)n2C1 Nc1ccccc1CC(N1CCC(CN2CCCCC2)C1)=O N1(C(COCCCCCC)=O)CC(CNC(C2COC(=O)O2)=O)C(F)(F)C1 C1(CCNC(=O)Nc2c(C(C)C)cncc2)COc2ccccc2O1 N1(C(Cc2noc(C)c2C#N)=O)CCN(C(C2CCCC2O)=O)CCC1C C1(C(=O)NCC2CCN(C(C3N(C)CC(O)C3)=O)CC2)CCCCN1N=O C1(C)(CNC(CCn2c(C)ncc2)=O)CCCN1C(=O)Cn1cnc(Br)c1 C(C)(N=c1[nH]c(=N)c2[nH]cc(Br)c2[nH]1)c1c(C)noc1C c1(C(=O)NC23CCN(C(C(CC)(C)C)=O)CC2C3)csc2cc(Cl)cnc12 N1(C(C(C=CC)O)=O)C2COCC1CC(NC(C1(COC)CC=CC1)=O)C2 CCC(C)C(C(=O)NCc1c[nH]ccc1=O)N(C)C(c1sccc1C)=O C1(C(=O)NC2C(CNC(CCN(CC)CC)=O)CCC2)COCCN1C CC1CC(C(=O)NCC=CCNC(=O)CC2(N3CCCC3)CC2)C(=O)O1 C1(CC)(CC)CC(NC(C2SC3C=CC2CC3)=O)CN1C(c1sc(C)nc1C)=O C(=O)(CC(C)C(=O)N1CCOC(CCCNC(=O)C=Cc2cnc[nH]2)C1)OC C=CCCCCCCCCCNC(=O)NCC1CCCC1CC N1(C(CN2C(C)CCC2)=O)CCC(N(C(=O)C(O)C2CC2)CCO)CC1 C1(C)(CC(=O)NCC(C)N(C)C(C2CSC2)=O)CC1(F)Cl n1(CCC#C)ccc(=O)n(C(=O)CCC(=O)c2ccccc2)c1=O N=C(NOCc1ccc(OCCC(F)(F)F)cc1)C1COC1 C(=O)(CC(CC)CC)N1CC(CNC(C(CC#C)O)=O)OCC1 C12(COC)CC(CNC(C3CC3(C)C)=O)(CN1C(=O)CSCCC(F)(F)F)C2 C1(C(=O)NC(C)CCNC(=O)C(C)(C)N(C)C)CC2(C1)CC1(CC1)C2 c1(C(N(CC(CN(C(C(F)=CC)=O)C)O)C)=O)ccc(C)nc1C1CC1 N1(C(=O)Nc2cccc(C)c2)CCC2(CC1)COC(CNC(=O)C1=CCC1)C2 N1(C(C2(C)CC2c2cccc3ccccc23)=O)C2CCCC1CC(F)(F)C2 n1(CC(=O)NCC2C(NC(c3nccc(C(=O)OC)c3)=O)C2)cc(C)ccc1=O C1(CCC)(NC(=O)C(CC)OC)CCCN(C(c2nccc(OC)c2O)=O)C1 C1(C(=O)NCC(C)(C2CC2)NC(=O)CCCc2ccsc2)CCC(C(N)=O)O1 Cc1ccnc2sc(C(N3CC(C4CN(C(c5ccn(C)n5)=O)C4)C3)=O)c(C)c12 Cc1cc(C(=O)N(CCCCCNC(C2(C#N)CC23CCC3)=O)C)cc(C)n1 CC1C(C)N(C(=O)NCCF)CCS1(=O)=O.S1(=O)(=O)CCN1 c1(C(=O)NC(CNC(Cn2c(C=C)ncc2)=O)C2CC2)cc(C)c2n[nH]cc2c1 N1(C(c2c(CC)cc[nH]2)=O)CCN(C(C2CC(CF)C2)=O)C(CCOC)C1 N1(C(CC(C)SC)=O)CCC(CNC(c2cccc3c2CCC3)=O)C(F)(F)CC1 c1(C(N2CCn3c(cc(C)n3)C2)=O)ccc2nc(C)n(C)c2c1 N1(C(C(C(C)C)S)=O)CCOCC(C(=O)NC(c2ccccn2)CO)C1 c1(C(=O)NC2C(NC(C3(C)CSC3)=O)CCC2)c(Cl)cccc1Cl C1(NC(=O)Cc2nc(C(F)(F)F)cs2)CN(C(=O)COC2CCCC2)CC12CC2 c1(-n2c(CCCOc3ccccc3Cl)nc(CC(CC)C)n2)cccc(Cl)c1C C1(CCOC)(NC(C)=O)CCN(C(C2CCC(c3ccccc3)O2)=O)C1 C(=O)(CCCCC#N)N1CC(C=C)(CC(=O)NCC2CCCSC2)C1 c1(C(N(C(CNC(CCC(C)O)=O)C2CC2)C)=O)cccc(C(N)=O)c1F C1(NC(COCCOC(=O)CCOC(C)CC(C)C)=O)CC2CC(NCC)C2C1 Cc1cc(C)c(C(=O)NC(C)C(C)NC(c2ncoc2C)=O)cc1Br C#CCCN=C(NCCC(C(C)C)N1CCOCC1)NCC1CCOC(C)C1 N1(C(C(C(=C)Cl)(C)C)=O)CC(C)CN(C(=O)C=C2CC3CCC(C2)N3C)C(C)C1 c1(C(=O)NC(CC=C)CNC(=O)CCC2CCCO2)cccnc1OCCOC C(C(=O)NCCOC1CN(C(=O)CC2CCCOCC2)C1)(C(C)(C)C)SC C(CCC(=O)Nc1ccccc1C(C)C)(C(C)C)OCC.C12(CCC1)C(=O)N2 N1(CCCC)CCCCC1C(=O)NCc1nccnc1OC C(C)(C)(C(C)CC(=O)N1CC(=O)NC2(CC2)C1)NC(C(C)OCC=C)=O C1(C(N(CC=C)CC=C)=O)(OC)CCN(C(C2CC23CCC3)=O)C1.c1cccnc1 c1(C(=O)NC(CNC(CCOCC)=O)(C)Cn2cccn2)cc(OC)ncc1Cl c1(COC)nc(C(=O)NC(C)C(CO)NC(=O)C(C)(C)c2sccc2Cl)cs1 N1(CC=C)CCCC(COCCOCCOCC)C1.C(=O)(CC)N(C)CCOC N1(C(C2(C)CCCC2)=O)CCC(C(=O)NOC2CC3CCC2C3)C(O)C1 c1(C(=O)NCCOCCCNC(c2cc(C)nc(C)c2)=O)cccc2c[nH]nc12 Cc1cnc(C(N2CCC(C3CCCN3C(=O)CC3CCOCC3)C2)=O)c(C)c1 c1(C(=O)NCCN(C(C(C)C)=O)C(C)C)cc2sc(Br)cc2s1 C1(NC(=O)NC2CC(CC(=O)OC)C2(C)C)CCn2c(O)nnc2C1 n1(CCC)ccnc1CNC(c1[nH]ccc1CNC(C1CC1C(N)=O)=O)=O C1(OC)CN(C(=O)CC2C3CN(C(=O)COC4CC=CC4)CC23)CC1F N1(C(C(C(C)(C)C)=O)=O)CCCC2(C1)CN(C(c1cnc3ccsc3c1)=O)C2 c1(C(N2C(CCNC(=O)COc3ccncc3)CSCC2)=O)cc(F)cc(F)c1 C1(CCOC)CCCC(NCC(C)OCC2CN(C)C2)C1 CC1CCc2nc(C(N3CC(C4(NC(C5COCCO5)=O)CC4)C3)=O)cn2C1 N1(C(C=C(CCC)C)=O)CC(C)CC1C(=O)NCC(O)CO C1(N(C(CCSCC)=O)C)CCCC(N(C)C(c2ccc(C(C)(F)F)cn2)=O)C1 C=C(C)CC(C)C(=O)N1CCC1CNC(=O)CCN(CCCCC)C c1(C(=O)NC2C(OCC(C)C)COCC2)cccc2c(Br)coc12 N1(C(C2(CC=C)COC2)=O)CCC(C)C1NC(=O)CCCOc1ccccc1C c1(CNC(C(CC=C)(C)C)=O)cnn2c1CN(C(C1CC(=O)N(CC)C1)=O)CC2 CC(O)CCCCCC(=O)NCC1C2CN(CC3CCOC3=O)CC12 C1(CNCc2ccc(OC(CC)C)cc2)Cc2cccc(C)c2O1 C1(O)(CNC(=O)C(=O)NC2CC2)CC(CO)C1.c12n[nH]cc1CN2 CC1CC=C(C(=O)N2CC(CCNC(C3CC(C)(C)CO3)=O)C2)CC1 c1(CCC(=O)NC2(C3CCCN3C(c3ccncc3O)=O)CC2)ccc(O)nc1 CCCC(C)(CCC)C(=O)NCCC1CC(OC)CN1C(c1csc(CO)n1)=O C(CCN=c1[nH]c2cc(F)ccc2o1)NC(c1ccc(C)nc1O)=O C1(C(=O)NCC(C)C)COC2(C1)CN(C(=O)C(C)CC1CCCC1)C2 Cc1nn(C)c(C)c1S(=O)(=O)N1CC(CNC(=O)CCC(F)(F)F)C(C(F)(F)F)C1 C#CC1CN(C(C2CN(C)CCN2C(=O)CN2CCCCC2C)=O)CC1O c1(C(=O)NCCCOCCCNC(CC(C)C)=O)cc(-n2cccc2)ccc1Cl c1(N2CCC3(C(OC)C3)CC2)nc(=N)[nH]c(=NC(C)CCN(C)C)[nH]1 c1(CC(=O)NCC2CCCN2C(=O)CC2=CCCC2)ccc(O)cc1Cl c1(C(=O)NC(C)CNC(c2cnc[nH]2)=O)ccc(O)nn1 S(=O)(=O)(c1cnn(C)c1)NCC(N1C(CNC(c2c(C)noc2N)=O)C=CC1)=O Cc1cnc2c(C(N3CC(C)C(NC(c4cnsc4)=O)C(C)C3)=O)cccc2n1 N(C1COc2cc(Br)ccc21)C(C)Cc1cccc(S(N)(=O)=O)c1 Cc1cc(CC(=O)NCCNC(c2cnn(C3CCC3)c2)=O)on1 c1(C(=O)Nc2c(C#N)cccc2)cn2ccc(C3=CCC(O)CC3)cc2n1 C1(C(C)(C)NC(C(N2CCCC2=O)C)=O)CN(C(=O)C(F)=CCCF)CCO1 C1(NC(C(C)Cc2cnn(C)c2)=O)C=CCN(CC(=O)NCC2CCCC2)C1 C1(NC(c2c(CCC)nco2)=O)CN(C(c2cc(Cl)ccc2C)=O)CC1(C)C Cc1ccc(NC(C)(C)CNc2cnn(CCl)c2)c(C)c1 C(=O)(C1=CS(=O)CCC1)N1CCCC(CCCCNC(c2c(Cl)cn(C)n2)=O)C1 C(=O)(C(O)C(C)C)NC(c1ccccc1)CNC(CCNS(CC)(=O)=O)=O N1(C(CC2(CC(=O)OCC)CC2)=O)CCc2ncccc2C1 CC(C)(C(=O)NC(CC1CC1)CO)C1CCCN1C(=O)C=Cc1ccco1 CCCCC(C(=O)N(CC(=O)N(C)Cc1cccnn1)C)C(C)C C1(C(=O)NCC#CCNC(CCc2cccc(OC)c2)=O)CC2(CCCO2)C1 N1(C(CC2N(C(C(C)CO)=O)CCOC2)=O)CC(N(C)C)CC1(C)C c1(NCCC(C)NC(=O)CCCC2CCCCC2)ncc([N+](=O)[O-])cc1F N1(C(CC(=O)OC)=O)CCc2[nH]nc(C(N3C4CCC3CC(=O)NC4)=O)c2C1 C1(O)(CC(=O)NC(CN(C(CCc2ccc(C)nc2)=O)C)C)COC(C)(C)C1 N1(C(C(CC2CCCC2)NC(c2ncn(CC)c2)=O)=O)CC2(CCCO2)C1 c1(C(=O)NCCC2CC(C(=O)NC3(COC)CC=CC3)C2)nc(C(C)C)oc1C C=C(C)c1cccc(NC(=O)CC(C2CC2)NC(=O)COCC2CCCO2)c1 CCC(C)CCC(O)CC(=O)N1CC(NC(c2cc(C)cc(O)n2)=O)CC1C CN1CC(C)(NC(=O)C(O)CCCNC(c2cccc(O)c2)=O)CCC1=O CC1CC(CNC(=O)CC2CCCCC2)CN1C(c1coc(C(C)(C)C)n1)=O CCCC(CCC)=CC(N1CCCC1C(N1CCC(C)CC1)=O)=O c1(C(N2CCC(SC)C2)C(=O)NC2(C)CC2)cccc(C(F)F)c1F.C1(CN)CC1 c1(C(=O)NCC2CC(NC(c3c(SC)cn(C)n3)=O)C2)cn2cccc(Cl)c2n1 c1(C(N2CC(NC(Cc3cc(CC)no3)=O)C2)=O)ccc(SC(C)C)cc1 c1(N(C)C)ccccc1C(=O)NOCC1CCC1c1cn(CCNC(N)=O)nn1 C1(C(=O)NCc2conc2C)(CNC(CCCOCCOC)=O)CC12CCC2 CC1C(NC(c2ccc(C3CC3)cc2)=O)CCCN1Cc1cccnc1N(C)C c1(COC)cc(C(N2CC(O)(CN(C(=O)CC3CC3(C)C)C)C2)=O)c(C)o1 C(=O)(CCCCC(F)F)NCC1(OC)CN(C(=O)Cn2c(C)cc(O)cc2=O)C1 c1(CN2C(CNC(c3c(C)noc3C)=O)CCC2)ccc2ccn(C)c2c1 c1(C(=O)OCC)nc(CNC(C2(CCOCC(C)OC)CCC2)=O)oc1C C1(NC(c2cnsn2)=O)CN(C(c2csc3nccn23)=O)CCC1C(F)(F)F C1(OC)CN(C(c2c(Br)ncn2C)C(=O)NC(c2ccccc2)C)C2(CCC2)C1 O(NC(=O)CN=c1nc(N(CC(F)F)C)c2c([nH]1)CCC(C)C2)CC c1(CC(=O)NCC2CC2NC(=O)CC2CCC3CC23)ccnnc1O N1(CC(=O)NCC(CNC(c2ccc(C(F)(F)F)nc2)=O)CO)CCOCC1=O CCC(C)C(O)C(=O)N1CCC(NC(=O)C=Cc2cccc(CO)c2)C(C)C1 C1(CNC(C(C)=C2CCCC2)=O)CC(F)(F)CN1C(c1cc(Br)cs1)=O C12(NC(C(C)=CC)=O)CC(CO)(C1)OC21CCN(C(c2cn(CC)cn2)=O)CC1 C12(C(=O)OC)CCCC(C(N3CCN(C(C4(SC)CC4)=O)CC3C)=O)(CC1)C2 CC1CCC(OCC(N2CCCC2CNC(=O)CCc2ccc(N)cn2)=O)CC1 C(=O)(C(CO)C(C)(C)C)NCC1CCN(C(CC2CC(SC)C2)=O)CC1O CC1(C)OCC(C=CC(N2CC(C)(NC(C3CC3(C)Br)=O)C2)=O)O1 C1(C(=O)NCc2cccc(I)c2)CC12CCN(C(=O)C(O)CCl)CC2 C(=O)(C(CC1CCC1)C(C)C)NCC(C(=O)NCC(=O)OC)N(C)C O=C(CCC(F)(F)F)NCC1CCCN(C(=O)Cc2ccc(OC(F)F)nc2)C1 O=C(NNc1ccc(Cl)nn1)Nc1cc(Br)nn1-c1ccc(F)cc1 C(=O)(C1=CCCC(C)(C)C1)NCC1CC(OC)CN1C(c1cnc(O)o1)=O c1(CC(=O)NC2C(NC(Cc3c(C)ocn3)=O)COC2)cnccc1Cl c1(C(=O)NCC(C)NC(c2c(C)ccc(F)c2O)=O)nn2cccnc2c1Cl CC(C(=O)NC1CCCN(C(=O)CCSc2nnnn2C)C1)C1=CCCC1 C(C(C)(CO)CO)NC(C(c1cnn(C)c1)N(c1c(C)ncs1)C(=O)CSCC(C)C)=O c1(C(=O)NC2(CCNC(CC3ON=C(C)C3)=O)CC2)c(N)cc(Cl)cc1Cl c1(C(=O)NCc2ccc(C(N3CCCC(C(C)(C)O)C3)=O)s2)c(F)cncc1F N1(C(C2(CCOC)CC2)=O)CCCOC(CNC(=O)C(c2ccc(Cl)cc2)C)C1 C(=O)(C1CCCc2cncn21)NC1CCN(C(Cc2scc(C)c2)=O)CC1O C(c1cnc(O)nc1O)=CC(=O)NC1CCN(C(c2c(C)noc2C)=O)C(C)C1 Cc1c(Br)ccnc1C(=O)NCC(C1CCNCC1)C c1(NS(CC#N)(=O)=O)ccnc(NCCC2CCCNC2=O)n1 C1(OC)CN(C(=O)C=Cc2ccc(Cl)s2)C(C)(CNC(C2CC(C)(C)C2)=O)C1 C=CC(CCC)CC(=O)NCC1CCCCC1C(=O)NC(c1ncc(C)o1)C C(C(C)(CC(C)C)NC(c1cc(C(=O)OC)ncc1F)=O)NC(C(F)=CC)=O CC(C)(C)C(C#N)C(=O)N1CC2(CC(NC(c3c[nH]cc(F)c3=O)=O)CO2)C1 c1(NCC23CC(C)(OCC2)C3)cc(S(N)(=O)=O)c(Cl)cc1Cl CC1C(NC(c2ccc(F)o2)=O)C(C)CCN1C(c1cnn(CCO)c1)=O c1(CN(C=O)CC2CCC3(CC2)CC3)cc(=O)c(OC)cn1C C1(C(=O)NC2C(NC(c3c[nH]c(=N)s3)=O)C2)CCC(=O)NC1 Cn1ccnc1C(c1ccccc1)SCC(N1CC(NC(=O)COC(F)F)C1)=O C1(=CC(=O)N(CCC(=O)NC(CC)C)CCOC)CCCCC1 C1(C(=O)NCC(C2CCC2)NC(Cc2ccc(C)nc2)=O)CC2CCC1CC2 N1(c2cc(C(C)=O)ncn2)CC2CC1CN2C(=O)CCc1ncc(C)[nH]1 C(=O)(CC(F)(F)C(F)(F)F)NCC1CCC(NC(C=C(CC)CC)=O)C1 N1(C(c2nc(CC)sc2)=O)CCCCC1CN(C)C(c1cnc(Cl)s1)=O c1cnc2cccc(CNC(=NCCCC3CCC4CC3C4)NC3CCC3)c2c1 C1(CC(=O)NCCN(C(C2CCC=CCCC2)=O)C2CC2)CCC(F)(F)CO1 c1(CC(C)C(=O)N(CCCCCNC(c2cc[nH]n2)=O)C)ccc(F)cc1F CC(C)(C)C(C(=O)NCCCn1cc(C2CCCCO2)nn1)C1CCCCC1 C=C(Cl)CCC(=O)N1CCC(CO)(NC(c2cc(O)ncn2)=O)C1 N1(C(C(F)OC)=O)CCCC(N(C(=O)COc2ccc(C)cc2)C)C1 N1(C(C(CC)OC2CCCCC2)=O)CC(NC(=O)C2=CCOC2)C2CCCC2C1 N1(C(CC(CNC(C(C)(C)NC(C)=O)=O)C)=O)CC2(C1)NC(=O)NC2=O c1(C(N2C(CNC(C(C)n3ccnc3)=O)CC2)=O)ccc(CC(N)=O)cc1 N1(C(=O)C(CO)c2ccccc2)C2CCC1CN(C(C13CCC(F)(CC1)C3)=O)C2 c1(C(N2CC(NC(C3CC34CC4)=O)(CO)C2)=O)c(Cl)cccc1Br C1(OC)CN(C(c2cnn(C(C)C)c2)=O)CCC1NC(c1cc(C(C)C)no1)=O C1(C)(C(=O)OCc2occ(C(N(C(C)=O)C)=O)n2)COC(=O)N1 c1(C(=O)NCCCNC(c2ncn(CC)c2)=O)ccc(F)c(F)c1C C1(CC(=O)NCC(c2ccco2)O)CCCN(CC(O)COC(F)F)C1 C(=O)(C1COc2ccc(Cl)cc21)NC1(C2CCN(C(CC(C)C3CC3)=O)C2)CC1 c1(N(C(COC)C)C)ccc(C(F)(F)C(=O)OC)cc1 N1(C(C(F)=C(C)C)=O)CCC2(CC1)CN(C(=O)CSCc1ccc(Cl)cc1)C2 N1(CC(N2CC(CC(C(=O)N(C(CC(C)C)C)C)F)C2)=O)CCN(C)CC1 C=CC1(C(=O)NCC(O)CN(C)C(C2CCc3cnnn3C2)=O)CCCCC1 C1(NC(Cn2c(C)ncc2)=O)CC2CC1CN(C(C1CC(C(C)C)=NO1)=O)C2 c1(COc2cccc(OCCOC)c2)ccnc(Cl)c1SCc1cscn1 N1(C(CCNC(C)=O)=O)CC2(CNC(=O)COC3CC(F)(F)C3)CCC1CC2 N1(C(C2(OC(C)C)CCOC2)=O)CC2(CCCN(C(C3CC3F)=O)C2)C1 C=C(C)C(C)(O)C(=O)N(C)CC1CN(C(=O)C(=O)NCCSC)CCO1 CCCCC(C)C(C)(c1nnnn1CC1CCOCC1)Nc1cc(O)ccc1C CC12COCC1CN(C(=O)C1=CCC(NC(C3OC4CCC3C4)=O)C1)C2 Cc1ccc(CC(=O)NCC(C)NC(=O)C(C)N)c(C)c1.C(C)(C)C1CC1 c1(C(=O)NC2C3N(C(CC(CCC)C)=O)C(CC3)C2)n[nH]c2cccnc12 CCC1=NOC(CO)C1.O1NC(=O)CC2(C)CCN2C(=O)CCC1 C(=O)(C1=NOC2(CCC2)C1)N1CC(C)N(C(c2cnn(C3CC3)c2)=O)CC1 c1(C(N(CCC(C)(C)NC(c2c(C)n[nH]c2)=O)C)=O)ccc(CO)cn1 Cc1cccc(Cl)c1S(=O)(=O)N1CC2C(C1)N2C(C1CC(=O)NC(=O)N1)=O c1(C(c2nnnn2CC2CCCO2)NC(C(=O)NC)C)sc(Br)nc1C c1(C(N2CCCC(NC(=O)CC3CCC3)CC2)=O)ccn2c1CCCC2 C(=O)(CC(C)CC(C)NC(CN)C(F)F)OC C1(CC(=O)OCc2c(C(N)=O)nns2)CSC2CCCC12 C1(C(N2CCC(OC)(CNC(=O)CC3CC(F)(F)C3)C2)=O)CC12CCCCC2 c1(C(N2CC(O)(C(C)NC(C(CC)n3cncn3)=O)C2)=O)cnc(N)cn1 CCC(CN(C)C)CC(=O)NOCC(=O)N(C1CCC1)CCN(C)C Cc1cc(C)n(CC(=O)NC2CC(N(C(=O)C(C)NC=O)C)C2)n1 c1(OC)ccc(OCC(=O)NC2CCN(C(=O)C(C)(C)C3CCCC3)C2)cc1 c1(C(=O)OC)cc(NC(=O)OCC)ccc1Br.C(=O)(CCP(C)(C)=O)O c1(OC)cc(C(N2CCC(NC(=O)C=C3CCCC3)C2)=O)cnc1OC CCCC(C(=O)N1CCC(NC(=O)C(CC)OCC2CC2)C1)NC(N)=O C1(SCC(=O)NCC(C)N(C(C2C(=C)CC2)=O)C)CCCCO1 N1(C(C2CC2F)=O)CC2CC(C1)N(S(=O)(=O)c1cn[nH]c1)C2 n1(CC)ccc(C(=O)NC(CC2CCCC2)C(=O)N(C)Cc2cc[nH]n2)n1 N1(C(C2CC(C)OC2)=O)CCC2CCCC12C(=O)NCCCF n1(CC)cc(C(=O)NCc2ccoc2C(=O)N(CC(C)C#N)C2CC2)c(C)n1 C1(F)(C(=O)NCCCNC(c2c(CCC)n(CCO)nc2)=O)CCCCCC1 C(=O)(NNC(=O)C(C)N(C)CCc1ccccc1)C(=O)Nc1nc(C)sc1 c1(NC(=O)OCC)ccc(NC(C2(N)CCCOC2)=O)cc1C c1(C(=O)NCC(C)NC(=O)Cc2ccccc2CC#N)cccc(O)c1F c1(NC(C23C(CN(C(c4ccc(CC)nc4)=O)C2)C3)=O)c(Cl)ccnc1Cl CCCC(O)C(=O)NC1CCCC(Cn2cc(COC3CCOCC3)nn2)C1 CCCCC(CC)C(=O)NCC1CN(C(=O)CCCC(=O)N(C)C)CCCO1 C#CC1(C(=O)N(CC(O)CN(C(=O)COCCC(C)C)C)C)CCCC1 c1(C(=O)OC)cc(N=c2nc(C)[nH]n2-c2ccccc2Cl)cnc1F c1(C(=O)NC(C2CCCC2)CNC(C2(SC)CC2)=O)cccc2nccn12 C1(C(=O)NC2CN(C(c3nc(C)sc3C)=O)C(CO)C2)CCCC12CCOCC2 C#Cc1ncc(F)cc1NC(=O)Cc1cn(-c2ccc(OCC)cc2)nn1 C1(NC(C2(N(C(c3c(C)n(C)cc3)=O)C3CC3)CCC2)=O)CC2CC1C(O)C2O c1(OC)cccc(S(=O)CC(=O)NCC=CCNC(C2(C)CCCOC2)=O)c1 C1(NC(c2coc3c2COC3)=O)CCCC12CCN(C(C1CC3CC3C1)=O)CC2 N1(C(C=Cc2nc(C)sc2)=O)CCC(C2(NC(C34CC(C)C3C4)=O)CC2)CC1 C12(C(N(C)CCN3CCOC3=O)=O)CC(NC(=O)C(O)C3CCCC3)(C1)C2 c1(C(=O)NC(CC)CN(C(=O)CSC)C)cnc(Nc2nccs2)s1 C(=O)(C(F)CCC(C)(C)C)N1CCCC(CCC(=O)NCc2cn(CC)nc2)C1 N1(CC(N2CC(Cn3cc(SCCOC(C)(C)C)nn3)C2)=O)CCCCCC1 C(N=c1[nH]c2cc(Cl)c(S(N)(=O)=O)cc2[nH]1)C1CCC(C)C1 N1(C(CSC)=O)CCC(C2(O)CN(C(=O)C3CSc4ccccc43)C2)CC1 Cc1ccc(CNC(N2CC(Oc3cccc(F)c3F)C2)=O)c(F)c1C C1(COC)(CO)CC(NCc2ccncc2Cl)C(O)C1 C12CC3CCC(C1)N3C(=O)c1cn2nn1.c1(CNC(N)=O)ccnnc1O c1(CC(=O)NC(C2CCCN2C(=O)CCOC2CCCCC2)C)c[nH]nc1O c1(OC)ccccc1CCC(N1CCCC1CNC(C)=O)=O c1(NCCN(C2C(C=C)OCC2)C)cc(Br)ccc1S(=O)(=O)NC C1(C(=O)NCC2(CC)CCCCC2)CCN(C(c2ccncc2O)=O)C12CCC2 C(=O)(NNc1ncc(Br)cn1)Nc1c(OC(C)C)cc(F)cc1 C(CCCCC(=O)N(C)CC1CCCC2CC12)N(C(CCc1onc(C)n1)=O)C CCC(CN(C(=O)COCC)C)NC(=O)COC1CC=CC1.C(CCC)O C12(NC(c3c(C(C)C)ocn3)=O)CCCC1N(C(c1ccn(C)n1)=O)CC2 CC1C(C)N(C(c2ncc(O)cc2Br)=O)CCS1=O CN1CCc2cc(C(=O)NCCC3CCCN(CC4CCCCCC4)C3)sc2C1 C1(NC(C2CC(NC(CCCSC)=O)C2)=O)CCC(=O)NC1(C)C N1(C(Cc2nc(=N)[nH][nH]2)=O)CC2(CCCC2NC(C2CCCC2O)=O)C1 C1(CNC(c2cccc(OC)c2)=O)CC2(CCC2)CN1c1nccc(SC)n1 C(=O)(CS(=O)(=O)CC(C)C)NCC(CC=C)NC(=O)C(C)CS(C)(=O)=O c1(N(CCC)Cc2ccc(C(=O)NCC)o2)ccc(Cl)cc1 C=C(C)CCCC(=O)N1CC(n2cc(CN(C)C(C)C)nn2)C(C)C1 N12CCOC(C1)C2=O.CCC(CCOC)NC(C1CN(C(C)C)C1)=O c1(C(N2CCCN(c3snc(CC)n3)CC2)=O)cc2c(F)c(C)ccc2[nH]1 n1(CC(=O)NCC(C)N(C(=O)C=CCNC(=O)OC(C)(C)C)CC)cnnc1O Cc1ccc(OCCC(=O)NCCNC(c2ccc(C#N)[nH]2)=O)c(C)c1 Cc1cc(Cl)ccc1OCC(=O)NCC1(C)CCN(C(C2CCOC(=O)N2)=O)C1 C12(NC(=O)C(O)CC3CCCC3)CCN(C(=O)CC3CCOCC3)CC1C2 C1(C(C(=O)N(CC(CC)(C)OC)C)C)CCCN(C(=O)CN(C)C(N)=O)C1 c1(C(N2CC(F)CC(C(=O)Nc3ccc(CC)nc3)C2)=O)ccn2nccc2c1 CC1CCC=C1C(=O)N(CC(C)N(C)C(c1cnn2ccsc12)=O)C c1(C(=O)NCC2OCCCN(C(c3nnc(C)s3)=O)C2)ccc2c(c1)CC(C)O2 N1(C(CN(CC)CC)=O)CCC2C(C1)OCCN2C(=O)CCOC Cc1cc(Cc2nc(-c3ccccn3)nn2C2CCCCCC2)n(CCO)n1 c1(C(N(C2CCCN(C(=O)NC3CC3)CC2)C)=O)ccnc2ccsc12 Cc1cc(C(N2CCC(C(F)C(=O)NCC34CCCN3CCC4)C2)=O)cc(O)c1 Cc1cc(NC(C2CC2c2ccccc2C)=O)sc1C(=O)Nc1ccc(Br)cc1 C1(CC(=O)NCCN(C(=O)CCc2ccc(C)nc2)CCC)CCC(=O)N1C C1(C)(C(=O)NC2C3CC(NC(CCN(C(CC)CC)C)=O)CC32)CCN(C)C1=O N1(C(c2occ(C)c2)=O)CCCC(C2CCN(C(=O)CS(=O)(=O)CCO)CC2)C1 CC1CCn2cc(C(=O)NCCC3CCC4(CCC4)O3)nc2C1 c1(C(N2CCC(O)(C(C)NC(C(C(CC)O)C)=O)C2)=O)cc(F)c(F)cc1Cl c1(C(N(CCNC(c2c(C)cc(F)c(F)c2)=O)C)=O)cc2c(F)ccc(F)c2[nH]1 C(=O)(C(CC(C)C)NC(C1CC1CO)=O)N1CC(NC(=O)OC)C1 C1(C(=O)NC(CC#C)C)(CNC(=O)C(C(C)C)C2CCC2)CC12CCC2 C12(CNC(=O)Cc3cc(Cl)no3)CCCC1CCN2C(C1CCCNS1(=O)=O)=O c1(SC)cc(C(=O)NCC(C)(C)CN(C)C(c2cscc2C)=O)oc1C N1(C(C2C(C)C2C)=O)CC2CC3CC2C1C3NC(c1cnc(-c2cccs2)o1)=O CC1(C)CN(C(C2CCC3CCC2N3C(=O)C2=CCSC2)=O)C12CCC2 N1(C(COCCOCC)=O)CC2CC2C1C(=O)NCC(C)OC(F)F C1(NC(CCOCC)=O)COC2(CCCN(C(c3csc(=N)[nH]3)=O)C2)C1 S(=O)(=O)(c1ccc(=NCCN2CC(C)CC(C)C2)[nH]c1)NCc1c(C)cccn1 C(=O)(C(C)CCCc1ccccc1)NC(N(CC(=O)NCC)C(C)C)=O N1(C(COCCC)=O)CC(NC(C2Cc3nccn3C2)=O)CC12CCCCC2 N1(C(c2ccc(C)s2)=O)CC2CCC2(C(=O)Nc2ccc(Cl)cc2)C1 CN1C(=O)CN(CC(=O)NC2CN(C(C3(O)CC3)=O)CCC2C(F)(F)F)C1=O C(=O)(CCCCCF)NCc1c(C2CCN(C(C3C(=C)CC3)=O)C2)n[nH]c1 C=CCCCCCCC(=O)NCc1nc(CNC(C2CC2(C)C)=O)cs1 n1(CC(N2CCCC(CC=C)(NC(c3cnn[nH]3)=O)C2)=O)cnc2ccccc12 c1(COC)nc(C(=O)NCC=CCC(=O)NCCCc2ccco2)co1 C1(c2nc(-c3n(C)ncc3)nn2CCc2cccc3sccc23)CCCCC1C1CC1 N1(C(C2N(C(C=C(CCC)C)=O)CC(O)C2)=O)CC2CN(C)CC2C1 C(=O)(C1=CC2(CN(C(c3ccc(Cl)o3)=O)C2)OC1)NC1CC(C)SC1 C1(CC(=O)N(C2CCN(C(C3(COC)CC=CC3)=O)C2)CCO)COCC1(C)C C(=O)(C1Cc2ccc(C)cc21)NCCC(C)NC(c1ccc(OC)cn1)=O C1(C(=O)NC2C(C)CN(C(c3cc(Cl)c(Br)[nH]3)=O)C2)CCC(C)(C)CC1 C12(CNC(c3cccc(CC)n3)c3n(CCOCC)nnn3)CC(C)(CCO1)C2 N1(C(c2cc(CCOC)on2)=O)CC(F)CC1CN(C(=O)C=CC(C)(C)C)C c1(C(N2CCC(C)(O)C2)=O)c(-c2ccc3ncsc3c2)ccc2c1OCO2 C(=O)(C(=O)N=S(C)(C)=O)NCC(CO)NC(c1c(C)nn(-c2ccccc2)n1)=O c1(C(=O)Nc2c(C(=O)NC3C(C#N)CCC3)cc(Cl)nc2)ccc(Br)c(F)c1F c1(C(=O)NC2C(C(N3CC(OCCOC)C3)=O)COC2)cnc2n1CCC2 c1(COC(c2c(C(C)=O)ccc(OC(F)F)c2)=O)ccc(C)c(F)c1O N12CC3CCC(C3C1)C(=O)NC1(CC1)C2=O.Cc1occc(=O)c1OCCN(C)C CC(C)(C)CCC(F)C(=O)N1CCC(CCNC(=O)CSC(F)F)CC1 c1(NC(C(CCC)NC(=O)C(C)CSC)=O)ccc(O)c(F)c1 N1(C(=O)CC2(n3ccnc3)CC2)CCCN(C(C2CCCC2F)=O)CC1 Cc1cc2sc(C(N3CCOC(CNC(C4C=CCC4)=O)C3)=O)cc2s1 CCC(C)(C)C(C)CC(=O)N1CCC2(CC1)CC2NC(=O)CCCCC#N c1(OCC(=O)N(CC(CNC(C(C(C)SC)O)=O)C)C)ccccc1NC(C)=O C1(C(=O)NCCCCNC(c2c(C(C)C)nns2)=O)CCCC2CCCN12 c1(C(=O)NC(CC)CN(C(=O)CC2CCSC2)C)oc(C)cc1C C1(C(=O)NC2CCN(C(CC(C)F)=O)CC2O)Cc2ccccc2C1 N1(C(C=CC(C)C)=O)CCCN(C(=O)C(C)n2cccc2)CC1 c1(C(N2CCCC(CNC(C(CC)n3ccnc3)=O)C2)=O)c2c(nn1C)CCC2 Cc1c(NC(C2CCC=CC2NC(=O)Cn2cnc(=N)[nH]2)=O)cccc1C(N)=O CC(C(=O)NCC(C1CC1)N(C)C(C1CC(=O)C1C(C)(C)C)=O)C(C)(C)C C1(CNC(C2(OC)CCOC2)=O)CN(C(=O)C(C)CC2CCCC2)CCC1(C)C c1(NCC2(C)COCC3CCCN23)nccc(=NC2CSCc3ccccc32)[nH]1 N1(C(c2c(CCCC)ocn2)=O)CC(NC(=O)Cn2cccnc2=O)C(O)C1 Cc1[nH]cnc1CC(=O)NC1(CF)CN(C(=O)CC2COC(=O)C2)C1 C12(CNC(CS(CC)=O)=O)CC(CC)(CN1C(c1cccc(COC)c1)=O)C2 Cc1c(Br)ccc(N2CC(CNC(C3CNC(=O)N3)=O)CC2C)c1[N+](=O)[O-] C(=O)(C1=CC2CCCCCCC12)NCCCN(C(CCC(=C)C)=O)C1CC1 N1(C(C(Cc2c(C)noc2C)C)=O)CCCCC(NC(=O)Cc2cncn2C)C1 c1(C(=O)OC)ccc(C(=O)N(C)CCN(C(=O)CC2CC3COCC23)C)cc1Cl N1(C(C2(n3cc(-c4ccc(C#N)cc4)nn3)CC2)C)CCc2ccccc21 C1(C)(CNC(C(C)(C)OCC)=O)COCCN(C(C2(COC)CC2)=O)C1 c1(CC(N2CCCC(CNC(C(C(C)C)(C)C)=O)C2)=O)ccc2c(c1)CCCC2 c1(C(N2CCCN(C(CC=CC)=O)C(C)C2)=O)oc2c(F)cccc2c1C C1(C)(CNC(C2CCN(OC)CC2)=O)CC(F)(F)CN1C(c1cc(F)c[nH]1)=O C1(C(=O)OCC)(C(=O)NCc2cc(NC(=O)NC)[nH]c2C)CC1S(C)(=O)=O C=CC1CN(C(=O)CCCC(C)NC(=O)CC2(COC)CC2)CCO1 Cc1cc(F)c(C(=O)NCc2ccc(CNC(c3cncn3C)=O)cc2)cc1Br c1(NC(C)=O)cccc(CNC(c2ccc(-n3cncn3)nc2)=O)c1 c1(NC(C2CC3CCC2O3)=O)cc(N2CCCS2(=O)=O)cc(F)c1 C(C)(N=c1cc[nH]cc1S(=O)(=O)NC1CCCC2(CC2)C1)c1ncc(C)cc1C c1(OC)c(C)csc1C(=O)N(CCNC(c1ccnc(C)n1)=O)C1CC1 C(=O)(C#CC1CCC1)NCC1CCC(F)(CNC(C(c2ccccc2Cl)C)=O)C1 Nc1cc(F)c(C(N2CCC(NC(c3cnc(C(F)F)o3)=O)C(F)C2)=O)cc1F N1(C(c2cccc(F)c2)C(=O)Nc2ccc(OC)cc2)CCN2CCCCC1C2 CC(C)(C(=O)NC1CCc2ncnn2C1)C1=CCN(C(C2CSCCS2)=O)C1 c1(NC(c2ccc(CC)c(C)c2)=O)ccc(CC)cc1C c1(OC)cc(C)ccc1C(N1CCC(NC(C2COC(=O)N2)=O)C(C)C1)=O c1(C(=O)NC2C=CCN(C(c3ccc(NC)c(F)c3)=O)C2)cnn2c1CCCC2 C1(C)(CNC(c2cn(CC)nc2C)=O)CC(OC)CN1C(=O)CC1CCC1 O=C(N=c1[nH]oc2cc([N+](=O)[O-])ccc12)c1coc2ccc(Cl)cc12 c1(C(=O)NC(CN(C(c2cnc(CCC)s2)=O)C)C)nccc(Br)c1O C1(CCNC(c2ccc(Cl)o2)=O)CCCCN1C(C1C2CCOCC12)=O N1(C(C2CCN(C(c3c(C)c(F)ccc3)=O)C2)=O)CCc2cc(C#N)ccc21 N1(C(C(C(C(C)C)OC)OC)=O)CC(O)C2(CCCC2)C1 S(=O)(=O)(c1cnc(Cl)nc1)N1Cn2c(C(=O)NC(c3ccno3)C)cnc2C1 C1(C)(C(N2C(C=C)CC2)=O)CCCN1C(=O)C(C)=CC(C)(C)C C(=O)(C1CCOc2ccccc21)NC1(CC)CCN(C(=O)Cc2nonc2C)C1 c1(C(=O)NCC2CCN2C(C2(C(F)F)CCCO2)=O)ccc(-c2cscn2)nc1 c1(C(=O)NC(C)CCCNC(=O)C(C)(C)C2CCCCO2)cn2c(n1)CCCC2 c1(C(=O)NCCC(C)NC(C(C(C)C)OCC)=O)c(C)ccc(F)c1Br CC(C)C(F)C(=O)NC(C(=O)NCc1cn(C)nn1)C1CCCC1 C1(C2(O)CN(C(c3cnc(C)o3)=O)C2)(CNC(CC2(OC)CCCCC2)=O)CC1 c1(C(=O)NC2C(CNC(=O)C=CC3CC3)CCC2)cc(F)c(CO)c(F)c1 N1(C(C2CCC(CC)O2)=O)CCC=CC1C(=O)NCCc1cccnc1F C(=O)(C(F)(F)c1nc(C)cs1)NCCN(C(=O)CC1(CO)CC1)CC C12(NC(C(COC)C)=O)CCC(CN(C(c3csc4nnsc34)=O)C1)C2 N1(C(C2C(OC)C2)=O)CCCC1C1CCCCN1C(c1ccnc(C)c1)=O N1(C(CC(C(F)F)NC(C(CCC(C)C)=O)=O)=O)CCc2nncn2CC1 N1(C(CN2CC(C)C2)=O)CC(F)(F)CC1(C)CNC(C1CCC(F)CC1)=O c1(C(=O)NC(C(=O)N(C(C)CC2CC2)C)c2cccs2)nnc(S)n1C c1(OC)ccc(CCC(=O)NCCCCNC(=O)CC(C)C2CC2)cc1Cl c1(CNC(C2CC2C(=O)NCC2(C3CC3)CC2)=O)ccc(C2C(C)C2)o1.COC CS(=O)(=O)CCC(=O)N1CCC(OCc2cn(-c3cc(F)ccc3F)nn2)C1 Cc1c(CN2CCC(CNC(c3cc(Cl)sc3Cl)=O)C2)cncc1Br c1(OC)cc(C(=O)NCc2n[nH]cc2C(=O)NCCC(F)=C(F)F)ncn1 C1(NC(c2cc(C)nc(C)c2)=O)CN(C(C2CC23CCCCC3)=O)CCC1(C)C Cc1cccc2cc(C(=O)NCC3CC(CNC(c4ccoc4Cl)=O)CO3)oc12 CC(C(C)(C)C(=O)N1CC2(CC=CC2)C1)NC(=O)CC1CC=CCN1C C1(C(=O)NCC2CCCN(c3ccnc(C4CC4)n3)C2)CNC(=O)CC12CCOC2 c12ccc(nc1C)[nH]2.C1(C(=O)OCC)CC12CN(C(=O)CBr)C2 N1(C(CCN(C(C)=O)C)=O)CC2CC(NC(C3CC(C)CC(C)(C)C3)=O)C(C2)C1 N1(C(C(C)NC(=O)C(c2ccc(Br)cc2)(C)N)=O)CC(=O)NC(C(F)(F)F)C1 c1(C(N2CCC(NC(C(c3ccccn3)C)=O)C(F)C2)=O)cc(O)cc(N)c1C c1(OCCCC(N2CCC(F)(CNC(C(C(C)C)O)=O)C2)=O)ccc(F)cc1Cl N(C(=NCC1CC(C(F)(F)F)(OC)C1)NCC(C)(C)C)C1CCN(CC)C1 c1(CC)cc(C(=O)NC2CCC(NC(=O)CCCc3nc(C)cs3)C2)cc(N)c1 C1(C(=O)OC)(CC)CCN(C(=O)NCCc2cccc(N)c2F)CC1 N1(C(C(C2CCCC2)OCC)=O)CCCCC1CNC(c1cccs1)=O C1(CNC(C(N2CCOCC2)C)=O)C(C2CC2)CCN1C(=O)CCc1cscn1 C1(NC(c2c(OC(C)C)cccn2)=O)CN(C(=O)CCOCC2CCC2)CC1(C)C CC(C)C(CNC(C1CCC2CC1CO2)=O)C(=O)N1CC(c2nn[nH]n2)C1 c1(CNC(c2cn(C)nn2)CC)ccc(F)nc1 c1(OC)nccc2c(C(=O)NCCCNC(c3ccc(C)c(C)c3N)=O)c[nH]c12 c1(C(N2CCC(O)(CN(C(=O)Cc3cnoc3)C)C2)=O)cc(Cl)ncc1N C(CC(C(=O)NCC1(C(C)C)CCCC1)NC(=O)Cc1c(C)noc1C)OC N1(C(C2(OC)CC2)=O)CCC2C(CCCN2C(=O)C(CO)C(F)(F)F)C1 c1(C(=O)NCCN(C(c2cc(Br)cs2)=O)CC)ccc(C)c(C)c1N N1(C(C(C)OCCCC)=O)CCCC(F)(CNC(c2ncnn2C2CC2)=O)C1 C(=O)(C(C)P(C)(C)=O)NC(C(CO)NC(C(CO)NC(=O)OC)=O)C C1(NC(C2C(CC(C)(C)C)C2)=O)CCC2(CCN(C(=O)CCF)CC2)C1 c1(C(=O)N(CCN(C(C(C(C)C)OCC)=O)CC(C)O)N2CC2)cc2ccccn2n1 C(C)(C)(CCC(=O)N1CCC=CC1C(=O)Nc1ccc(F)cc1C)OC n1(CC(N2C(CC(=O)NC3(C(=O)OC)CC3)CCC2)=O)c(C)cc(O)cc1=O C1(C2CCN(C(c3ccn4ccnc4n3)=O)CC2)(NC(CC(CCC)O)=O)CC1 n1(CC)nc(C(=O)N(C(C)CNC(c2cnc(O)c(F)c2)=O)C)ccc1=O c1(CC(=O)NC2CCC(NC(CCOCC)=O)CC2)cc(F)c(C)cc1F C1(NC(=O)CCc2nc(O)n[nH]2)CC2CC1N(C(=O)COCc1ccccc1)C2 c1(C(C(=O)NCCCN(C(C2CCCC2OC)=O)CC)C)ccncc1C CS(=O)CCC(=O)NC1(CO)CCN(C(=O)C=CSc2nc[nH]n2)C1 C(=O)(CCCC(=O)NCC1C=CC(NC(=O)CCSC(F)(F)F)C1)NCC c1(C(=O)NCCC(=O)OC(C)(C)C)cc(Cl)nn2c(I)cnc12 CC1(C)CN(C(=O)Cn2cccn2)C(CNC(=O)CN2CCOCC2)CO1 c1(C(N2CC(C)C(CNC(C3C4CCCC34)=O)CC2)=O)cc2cc(F)ccc2[nH]1 Cc1nccc(C(=O)NC(CNC(c2cccnc2NC(C)C)=O)C(C)C)n1 c12ncnc3c1ncn3CC1CN2C1.Cn1cc(SCCOCCN)cn1 c1(OC)cccc(C(=O)N(CCCCN(C(=O)CCOCC2CC2)C)C)c1N C(CC(C)(F)F)NC(C(C1CCOC1)NC(C1C(C)C1)=O)=O C1(C(C)C)CN(C(C2CCC3CCCCC23)=O)CCCN1C(=O)CN(C)C C1(C(=O)NCC(c2ccccc2)CNC(C(C2CC2)SC)=O)CCOCC1(C)C C1(N(C(C(CCSC)O)=O)C)CCC2CN(C(c3[nH]cc4c3CCC4)=O)CC12 N1(C(c2c(C)nn[nH]2)=O)CCCC2(NC(=O)Cn3c(C)csc3=O)CCCC12 C1(CC(=O)NCCN(C(=O)C2=CCOC2)CC(C)O)(OC)CCOCC1 c1(C(=O)NCC2OCC(CNC(c3c(CC)ocn3)=O)C2)cc(C)c(Cl)c(N)c1 CC1(C)CC(NC(=O)C=CC2CCC2)CN1C(=O)CCOc1ccc(N)cc1 N1(C(c2cc(CC)n(C)n2)=O)CCC2CC2(C(N2CC(N(C)CC)C2)=O)CC1 S1(=O)(=O)CC(=O)NCCC(C(C)C)NC(=O)CN1C.C(C(=O)N(C)C)SCC.CN c1(C(N2CC(NC(=O)CCC3(C)CC3)CC(C)C2)=O)cc(Cl)c(F)cc1O C1(NC(CNC(CC)=O)=O)CC2CN(C(C3(CC)CCNC3=O)=O)CC2C1 c1(C(=O)NC(CNC(C(C=C)O)=O)C)cc(C)cc(Br)c1F c1(OC)ccc2c(=NC(=O)C3CCC(C(=O)Nc4cnoc4)CC3)[nH]ccc2c1 C1(CC(=O)N(CC=C)CC2CC2)(OC)CCN(C(=O)Cc2ccc(C)nc2)C1 N1(C(c2n(CC)ncn2)=O)CC(C)CCC1CNC(C1CC12CCCCC2)=O c1(CC)onc(C)c1C(=O)NCCCC(C)NC(=O)CCC1CCCC1OCC C12(NC(C3CCN(C(CCC)=O)C3)=O)CC1CN(C(=O)CCCc1ccsc1)C2 C1(C(=O)NC2C(NC(CNC(=O)OC(C)(C)C)=O)C2)(CO)CC(F)(F)C1 N1(C(CNC(C2CCCO2)=O)=O)CCCOCC1 Cc1cnc(C(=O)NC2C3CC2N(C(=O)Cc2cnc(C)[nH]2)C3)c(Br)c1 N1(C(C(C=C=C)C)=O)CC2(CCCC2)C1C(=O)NCCCCCOC Cc1ccc(C(=O)NCC2(C)CN(C(=O)OC(C)(C)C)C2(C)C)cc1CO c1(N(C(CN(C(CC)C)CC(C)C)=O)C)ccccc1 c1(C(=O)OCC(CNCC)OCC)nc(C(C)C)no1.C1C(=O)N1 C12(C(N3CC(C(N)=O)(CNC(c4ccc(CC)s4)=O)C3)=O)CC3CC1C2C3O N1(C(c2c(C#C)cnn2C)=O)Cc2ccnn2CC(NC(C23CCCC2C3)=O)C1 N1(C(c2c(CC)nns2)=O)CC2CCC1CC2NC(C1(NC(C)=O)CCCC1)=O C1(CNC(=O)NC(CC)COC(F)(F)F)(CF)CC12CCOCC2 CCC1=NOC(CC(=O)NCC2(CCNC(=O)CC(C)c3ccccc3)CC2)C1 c1(C(N(c2cccc(C)c2)C(=O)CN2CCC3CC23)=O)cncc2ccccc12 c1(C(=O)OC)cccc(C(=O)NC2(CO)CN(C(=O)C(F)CC3CCCC3)C2)n1 c1(C(=O)NC(CC)CNC(=O)C(C2CCCCCC2)C)c(F)cc(Cl)cc1F CC(C(=O)NCC1CC(C)CN(C(=O)CCN2CCCCC2)C1)C(F)(F)C(F)F C1(C(N2CC(OCCOC)C2)=O)C2CCN(C(=O)C(CO)N(C)C)CC12 N1(C(CC2(C=C)CCC2)=O)CC2COCCC2(NC(=O)CN2C(=O)CCC2=O)C1 C1(C(N(C(C=C)C)C2CC2)=O)C(C)CN1C(=O)CCOC(C)=O c1(CN(C)C(C2CCCN(Cc3ccccc3)C2C)=O)cc(F)ccc1C(=O)O c1(C(=O)NC2CC(CNC(C3CC(CC)OCC3)=O)C2)cc2c(C)cccc2o1 c1(CC(=O)NC2CC(NC(c3[nH]n(C)c(=O)n3)=O)CC2O)ccccc1S(C)=O C1(NC(C2(NC(Cn3c(C)ccn3)=O)CCC2)=O)CC(N(C)C)C1(C)C CC1CN(C(c2n[nH]cc2F)=O)CCCN1C(=O)C(N1C(=O)CCC1=O)C Cc1cc(C(N2CCC(C)(CNC(C34CC3CNC4=O)=O)C2)=O)nc(O)n1 n1(CC(=O)NCCCCN(C(C(C=C)O)=O)C)cc(S(N)(=O)=O)cc1C(F)(F)F Cc1cc(Cl)ccc1C(=O)NCC(O)CCNC(=O)CCn1cncn1 N1(C(c2cc(=N)[nH][nH]2)=O)CC=CCC1C(=O)NCC1COCCO1 Cc1ccc(C(N2CCC2C(N2CCCC(CC3CC3)C2)=O)=O)c(O)c1 CC(C(F)C(=O)N1CC(CNC(=O)Cc2cc[nH]n2)OC(C)(C)C1)C(F)(F)F N1(C(C=Cc2c(C)cccn2)=O)CC(C)C(NC(=O)C(C#N)=CC2CC2)C(C)C1 N1(C(C2C(C(C)C)OCC2)=O)C(C(=O)NCC(C)CC(C)O)C2CC(O)C1C2 C1(CN(C(=O)CC2CC2)C)CCCCN1C(C1CC(O)C1)=O n1(CCC(=O)NCC(CO)NC(C2CCN(OC)CC2)=O)ncc2c1CCCC2 c1(NC(=O)Cn2cc(C3COCC3O)nn2)cc2cccnc2c2ncccc12 C1(CNC(c2ccc(C)nn2)=O)CN(C(=O)CC2OCCO2)CCC12CCC2 C(=O)(C(C(C)C)C1CCC1)NCc1ccc(C(=O)NCc2cc(CC)no2)s1 C(=O)(C(C)(C)CCCO)NC(C1N(C(CC2C(C)(C)C2)=O)CCC1)(C)C C(CC(N)=O)(C(=O)N1CCC(OCCF)C1)NC(c1c(CC)nc(C)o1)=O N1(C(C(C(C)(C)C)n2cc(-c3cccc(OC)c3)nn2)=O)CCN2CC(O)CC2C1 C#Cc1ccc(C(=O)NCCN2CCN(C(=O)CC3CCC(C)O3)CC2)cn1 N1(C(C(C)OCC)=O)CCN(C(c2ccn(CC(F)(F)F)n2)=O)C2COCC12 c1(CC(=O)N(CC(CC)NC(c2cn(C)nc2OC)=O)C)ccc(C#N)cc1 CCCC(C(=O)NC1CCCC1(C)CN(C)C(c1cc(CC)n(C)n1)=O)C(C)C C12(F)CCCN(C1)C2=O.c1(CNC(=O)CNC(=O)C2CC2)cccc(F)c1Cl N1(C(CONC(c2ncccc2O)=O)=O)CCC2(CC1)N=N2 CC(C)C(C(=O)N(C)CCNC(=O)CCCC1CCCC1)c1ccn(C)n1 CCCC(C(=O)NC(C)(CNC(c1cccc2ccnn12)=O)C1CCC1)C(C)C C#Cc1cnc(C(=O)NC2CC2CNC(=O)C(C)(C(C)C)NC(C)=O)c(C)c1 C=C=CCCC(=O)NC.C12CCC(C1)CNC(=O)C(CC)NC2=O.C(C)=C C(N=c1[nH]c(N2CCOC(CS(C)(=O)=O)C2)nc(=N)[nH]1)C1CCCC(C)O1 c1(CNC(C23N(C(CC4(C)CCOC4)=O)CC(C2)C3)=O)[nH]ccc(=O)c1O c1(C(N2CC(OC)C(NC(=O)CC(C)CN(C)C)C2)=O)cccc(=O)n1C CC1(c2cn(-c3cccnc3F)nn2)CCN(C(=O)CCOC2CCC2)C1 c1(C(=O)NC(CCCNC(c2cnc(SC)nc2O)=O)C)cc2cccnc2s1 C=CCCCCC(=O)N1CCCC(C)(CNC(c2ccc(C(C)=O)c(O)c2)=O)C1 CC(C)CCCCC(=O)NCCC1CCN(C(c2cc(Br)ccn2)=O)C1 C(C)(C)(CCC(=O)NC(Cn1cncn1)C(N1CCC(C)(C#N)C1)=O)OC C1(N(C(=O)CCCn2ccnc2)C)C2CCN(C(=O)CCOCC3CCCO3)C12 N1(C(C2(CC)CCCO2)=O)CCC(C(C)C(=O)NCCn2nncc2C)CC1 c1(CCC(=O)NCCC2CCCC(NC(CC)=O)C2)cc(F)ccc1OCC N1(C(CS(CCC)(=O)=O)=O)CC2(C1)CN(C(=O)CC1NC(=O)NC1=O)CC2CO c1(CC)ccc(C(N2CCC(CO)C(NC(=O)Cc3csc(C)c3)C2)=O)c(F)c1 N1(C(=O)NCC(COC2CCOCC2)OC)CC2C3COCC3C2C1 n1(CC)nc(C(=O)NCC2(CNC(C3CCCCC3)=O)CC(F)(F)C2)c(C)n1 C1(N(C(C2C(=C)C2)=O)CC2CC2)CCN(C(=O)CCC(=O)N(CC)CC)CC1 N1(CC(=O)N(CCC(C)C)C)CCC2CN(C(=O)Cc3cccc(C#N)c3)CC12 c1(CC(=O)OC(CC=CC)C)n[nH]cc1NC(=O)OCC.C(C)(C)C CON(CCC(=O)NC(CCO)c1ccco1)C(=O)Cc1ccnc(O)c1 N1(C(=O)OC)CC2C=CC1C(C(=O)NCCNC(c1cnc(C3CCOC3)s1)=O)C2 c1(C(N2CCC(N(C(c3nc(CCC)oc3)=O)C)C2)=O)c(C(F)(F)Cl)n[nH]c1C c1(C(=O)OC)ccccc1CC(=O)NCC(O)CNC(=O)C(C)c1ccsc1 c1(C(N2C(CNC(c3c(C)onc3)=O)CCCC2)=O)cc(F)ccc1O c1(SC)ccc(CCC(=O)NC(C)(CNC(c2sccc2F)=O)C(C)C)cc1 c1(C(=O)N(C2(C(C)C)CCNC2)C2CC2)cccc2ccccc12 Cc1nc2c(s1)CN(C(C1CN(C(=O)CC3(C)CC3)CC1(C)C)=O)C2 c1(CC)csc(C(=O)OC(C2CCCOC2)C(=O)N2CCCC2)c1 N1(C(COCC#C)=O)CC2CC2(NC(c2cnn(CC)c2Cl)=O)C1 N1(C(C(C)OCC)=O)CCCC1C1CCN(C(c2oncc2C)=O)C1 Cc1cncc(C(N2CCCC(CNC(c3cn(C(C)(C)C)nc3C)=O)C2)=O)n1 C(=O)(CC(C)(C)C(C)=O)NCC1C(CNC(c2cnc(CC)nc2)=O)C1(F)F c1(NC(C2CN(C(C3CC4C(C3)C4(F)F)=O)CC2F)=O)cnn2c1CCCC2 CC1(C)C(NC(=O)CNC=O)CCN1C(=O)CC1CCCCCO1 CCCC(CCNC(C12CC(CN(C(=O)C(C)CC(C)C)C1)C2)=O)CCC n1(C(C)C)cc(C(F)(F)C(=O)NC2CC2C(=O)NCC(=O)NC2CC2)cn1 c1(C(=O)Nc2ccnc(OCC)c2F)onc2c1CN(C(=O)C=CC1CC1)CC2 c1(-n2cc(CC(=O)N(C)C)nn2)cc(C(F)(F)F)cc(C(F)(F)F)c1 N1(C(COC(C)C)=O)CC23CCCC2(C1)CN(C(=O)C(C)Oc1ccccc1)C3 c1(CNC(CCN(C(CCC(C)=O)=O)C2COC2)=O)ccc(F)cc1F Cc1nn(CC(N2C(C(=O)NC(C3CCCCC3)C)CC2C)=O)c(=O)o1 C(=O)(C1=NOC(C)C1C)NC(C(=O)Nc1ccc(OC)cc1F)CCC1CC1 CCCCCC(C)(C)CNC(=O)C(CCC)NC(=O)C(C1CC1)OCC C1(CNC(C2(CCOC)CCC2)=O)CC(C)CCN1C(=O)CC1CC1(C)C c1(C(=O)NC2CC(C(C)NC(=O)CC3CCC(=O)N3)C2)cc(CO)on1 C12(CC(=O)NCC3=CCCOC3)CCC1CN(C(=O)Cn1ccnn1)C2 c1(-n2c(C)nnn2)ccc(C(N2CCCC2C(C)NC(=O)CC2(O)CC2)=O)cc1 Cc1nonc1CC(=O)NC1COCC1CNC(c1cn(C2COC2)nn1)=O CC(C)C(C)CC(=O)N1CC2CC(NC(=O)COCCOCCO)CC2C1 C(=O)(C1=C(C)OCCC1)N1CC(NC(c2cnn(C(CC)CC)c2C)=O)C1 c1(C(=O)NC2CN(C(C(C)(O)C3CC3)=O)CC2C(F)(F)F)cc2sc(Cl)cc2s1 CC(CNC(c1csc(F)c1)=O)C(F)C(=O)Nc1cccc(N(C)C)c1 N1(C(c2ncc(C)cc2F)=O)C2CC=C(C(=O)N(CC(O)CO)CCO)C1CC2 c1(NC(C2CCC(NC(C(C)(C)O)=O)CO2)=O)c(C(F)(F)F)cc(Br)cc1Br CC(C)P(=O)(CC(=O)NC1CCC1CNC(=O)C(C)(C)OCC(F)(F)F)C(C)C C1(N(C(C2CCCC2F)=O)CC)CCCN(C(C2CCC3(CC3)C2)=O)CC1 C1(NC(C2(OC)CCCC2)=O)CCC(C)(CNC(=O)CO)C1.c1(NC)ccncc1 c1(C(N2CC3CCC2CN3Cc2ccc(O)cc2Br)=O)c(O)ccc(F)c1F N1(C(COc2c(C)occc2=O)=O)CCCCC12CC(Nc1ncccn1)C2 c1(C(=O)NC(CC)CN(C)C(c2cocc2C)=O)nc2ccc(Br)cn2n1 CC1(C(=O)NCCOCCNC(C2CC2CF)=O)CC2CC2C1 N1(C(C=C(COC)C)=O)CCC(CNC(c2ccc([N+](=O)[O-])s2)=O)C(F)(F)CC1 N1(C(COC(C)=O)=O)CCC2(C)CN(C(=O)CC3CCC(C)C3)CC12 c1(C(N2CC(CC)N(C(C3CNC(=O)N3C)=O)CC2)=O)cn2c(n1)CCCC2C c1(C(CF)N(C(C)(C)C)C(=O)N(CC(O)CO)C2CC2)ccc(Br)cc1 N1(C(C=C(C)C)=O)CCN(C(=O)CCCC(F)F)C(CCC)C1 c1(-c2cn(C(C)CNC(C3CNC(=O)C3)=O)nn2)ccc2[nH]ccc2c1 C(=O)(C1=CC2C=CC(C1)C2)N1CC=CC(C(=O)Nc2c(OC)cccc2)C1 C1(NC(CC2CC(=O)NC2)=O)CCC2CC1CN2C(c1ccc2c(c1)CCO2)=O c1(C(N2C3C(C(=O)NC(c4ncc[nH]4)CC)C(C3)C2)=O)cccc(C#N)c1 Cc1n[nH]c(C)c1S(=O)(=O)Nc1ccc(C(=O)Nc2cccc(C#N)n2)cn1 Cn1nc(I)cc1C(N1CCC(C#N)C1)=O C12(NC(C(CC)OC)=O)CCCC(NC(=O)CNS(=O)(=O)CC)(C1)C2 Cc1ccc2c(CNCC3CCC(C4CC4)O3)cnn2c1C c1(C(N(C(CN(C(C(C=C)(C)C)=O)C)C)C)=O)cc2c(Cl)cc(Cl)cc2[nH]1 C(=O)(C(C(F)(F)F)C(F)(F)F)N(CCCNC(C1CCC(C(C)C)CC1)=O)CC N1(C(c2c(OCC)cccc2)=O)CC2(C)CC1C2NC(C1CC1CC)=O CCS(=O)(=O)CC(C(=O)NCCOC)N1CC(CO)CC1C(=O)OCC1CC1 C(=O)(CCCCC(N)=O)NC(C1CN(C(C2CCC2(F)F)=O)CCO1)C C1(NC(C(CC#C)C2CC2)=O)CCN(C(=O)CC2CCN(CCF)CC2)CC1O Cc1nc2cncc(C(=O)NC3CN(C(=O)CN(S(C)(=O)=O)C)CC34CC4)c2[nH]1 N1(C(CC2(N(C)C)CC2)=O)CCCCC1CC(N1CC(N2CCCC2)C1)=O S(=O)(=O)(c1cc(Br)c(Br)s1)Nc1ccc(-c2c(OCC)nccc2)c(F)c1 CC1CN(C(C2(CC3CCC3)CC2)=O)CCC1NC(=O)C=Cc1cccc(O)c1 C1(CCNC(C(C)n2cccc2)=O)CSCCN1C(=O)COC1CCC1 C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)NC1C(NC(C(C=C)(C)O)=O)COC1 Cc1oc(C)c(C(N2CC3CC3(CNC(=O)C(c3cccnc3)C)C2)=O)c1C C(CC(C)(C)C(=O)NCCN(C(=O)CC(C)c1ccncc1)CCCSC)OC Cc1cccc(OCC(=O)NCC2CC(C)N(C(c3ccns3)=O)C2)c1 N1(C(c2nc(CCC)oc2)=O)CCCCC1C(C)(C)CNC(C1(O)CC1)=O C(=O)(CC(CNC(C1C=CCS1)=O)C1CCC1)N(CC=C)C1CC1 c1(C(N2CCC(NC(c3c(C)noc3)=O)C2(C)C)=O)cc(F)cc(Br)c1F Cc1ccccc1C(=O)NCCOCCCN(C)C(C1NC(=O)CC1C)=O C=CC1(C)COCCN1C(C1CCCN(S(=O)(=O)c2ccc(C)s2)C1)C(=O)NCC CCC(O)C(F)(F)C(=O)NCC1CCC(C(=O)Nc2cccc(C)c2)CC1 C1(NC(c2csc(C)c2C)=O)CCC2CC1CN2C(c1ccnc2[nH]nnc12)=O CC1CN(C(C2C3CN(C(=O)CNC=O)CC23)=O)CCC1O c1(NCCc2c(C)nc(C)nc2O)ncccc1S(=O)(=O)N1CCCCCC1C c1(CCC(=O)N(CCC)Cc2ccn(C)n2)ccc(C(=O)OC)cc1 CC1CCCCCN1C(=O)CN(C(=O)CCc1ccn(C)c1)C S(=O)(=O)(c1ccc(F)c([N+](=O)[O-])c1)N1C(C)(C(=O)NCC)CC1 c12cc(nc(C)n1)NC1CCCN2C1.C=CCN(C)CCN(C)C(=O)C1CC1 C1(C(N(C)CC2CCN(C(=O)CSC(F)F)C2)=O)Cc2cc(F)cc(F)c2O1 c1(C(N(CC(C)SC)C)=O)coc2c1CN(C(=O)C(C)(F)C(=O)OC)C2 c1(N2CC(CC(C)NC(C(C=C)(C)CC)=O)C2)ccc(C#N)c(C)n1 C=CCC(C)(CC)C(=O)N(CCCCCC(=O)NCc1ncoc1C)C C1(C(=O)NCC2CC(C)N(C(=O)CNC(C3CCCC3)=O)C2)CCC2(CCC2)C1 C1(C(N2CCN(C(C=C(CC)CC)=O)C(CO)C2)=O)CCCC(C)(C)CC1 c1(CCCC)ocnc1C(=O)NCC1C=CCN1C(C1CC(=C2CCC2)C1)=O c12n[nH]c3c1CN(CC3)CCN1CCC1C(=O)N2.c1(CN)cc(C2CC2)on1 CCC(F)(F)C(C)(C)C(=O)NC1CC2CC(C1)N(C(=O)C(C)(C)NC(C)=O)C2 N1(C(c2cc(C)sn2)=O)CCC2(CC2)CC1C(=O)NCc1cc(F)ccc1F c1(CNC(C(CC)NC(C(F)=CCC)=O)=O)ccncc1Cl C(CCO)(C(F)F)NCc1cn(CCC(=O)OC2CCN(C)C2)nn1 c1(C(N2CCC(C(C)NC(c3cnnn3C)=O)CC2)=O)cc(F)cnc1Cl N=c1cc(C(=O)NC2CCC(CNC(C3CCC(F)C3)=O)C2)[nH]c(=N)[nH]1 c1(OC)cccc(OC)c1CC(N1CCC(c2cn(CC=C(C)C)nn2)C1)=O c1(C(=O)NC(c2cncnc2)C)ccnc(CNC(=O)Cc2ccn(C)n2)c1 C#CC(CC(C)C)N1CCOCC1.c12cccc(n1)N2.C1(C)C(=O)N1 c1(NC(C(=O)NCC(C(=C)C)C)=O)ccc(C)nc1N(C)C C(=O)(CN=[N+]=[N-])N(C1CCN(C)C1)C(C)C(=O)NCC(O)C1CC1 c1(C(CC)CC)nc(CC(C2CC2)OC)nn1-c1ccc(-c2ccccc2)cc1 Cc1ccc(CC(N2CC(NC(C3CC4(CCCC4)C3)=O)C3(CC3)C2)=O)c(C)c1 C(CCCCCNC(C1CCSC1)=O)N(C(=O)CC1CCC(C(F)(F)F)O1)C c1(C(C)=O)ccc(S(=O)(=O)NC2CCC(NC(c3ccc(NC)s3)=O)CC2)cc1 Cc1oc(C(=O)NCC2CC2NC(c2ccsc2Cl)=O)cc1S(C)(=O)=O c1(CC2N(C(=O)Nc3nnn(C(C)(C)C)n3)CCC2)cnc(O)nc1O C(=O)(C(O)CCC(F)(F)F)N1CC2C(CNC(C3CC4(CC(=C)C4)C3)=O)(C2)C1 N1(C(COCC)=O)CCC(CCCNC(C2CCC2n2cccn2)=O)CC1 Cc1cc(C(N2CC3(CC(NC(=O)C(C)n4ccnn4)CO3)C2)=O)c(Cl)cc1N C1(NC(c2nccc(C)c2)=O)CN(C(=O)CCCn2ccnc2C)CC2CC12 c1(CC(=O)NCC(CNC(C2CCC(CC)C2)=O)C)cccc2c1OCCO2 c1(C(=O)NC23C(CN(C(c4c(C)cc(CC)o4)=O)C2)C3)nnn2c1C(=O)NCC2 c1(CC)ccc(NC(=O)N(C2CCCN(C(=O)C(=O)NCCSC)C2)C)c(Cl)c1 CS(=O)(=O)c1ccccc1S(=O)(=O)NC1(Cc2ccccc2F)CCC1 C=CCCCC(C(=O)NCC12CCC(CC1)O2)NC(c1ccc(CO)nc1)=O C(=O)(CCC(=O)c1ccc(Cl)cn1)NCC(CNC(CN(C(=O)OCC)C)=O)F C1(C(N(CCC#C)CCOC)=O)CN(C(=O)CCc2ccc(C)nc2)CC12CC2 N(C(=NCCCC(F)F)NC(C)CC1CCCCC1)CC1N(CC)CCC1 C1(NC(c2cc(COC)no2)=O)CN(C(c2coc3c2COC3)=O)CC2(CC2)C1 C(c1cn(C)nn1)=CC(=O)NCC1(OC)CC(OC)C1.c1(C)ccccc1 CC(C)(CC(F)(F)F)C(=O)NCc1ccc(CNC(=O)Cc2cnco2)cc1F CC(C)C(C(=O)NC1CC1NC(c1occc1Br)=O)N1CCCC1=O c1(CN(C)C)ccc(C(N2CC(O)(CCNC(C3CC4CCC3C4)=O)C2)=O)cc1 c1(-c2cn(C3N(C(=O)OC(C)(C)C)CCC3O)nn2)cc2cc(Br)ccc2c(=O)o1 C1(C(=O)NC2CC(NC(C3C(OC)C3)=O)CC2O)CCN(C)CC1c1ccnn1C N1(C(C2C(NC(C3=NNC(=O)C3)=O)CC=CC2)=O)CCC(C2CCC2)CC1 c1(C(N2CCCC(CCNC(C(N)=O)=O)C2)=O)cc(N)cc2ccccc12 c1(C(=O)NC(CNC(c2c(Br)cc(OC)nc2)=O)C)cc(C)c(C)cc1N S(=O)(=O)(c1ccc(Nc2ccc(Br)cc2)c(F)c1)NCC1CC(OC)C1 C1(NC(=O)C=CC(=O)OCC)(CO)CCCN(C(C2CC3CCC2CC3)=O)C1 C(=O)(C1CCCc2ncnn21)N1C2C(CNC(CC(C)N(C3CC3)C)=O)C(C2)C1 c1(SC)cc(N2CCOC(C(=O)NCC3CC3C)C2)ncn1 C1(NC(c2c(C)cc(F)cn2)=O)C2CC3CN(C(=O)C(C)CN(C)C)C1C3C2 c1(OC)[nH]c(=N)ccc1C(=O)NC(CCNC(C1(c2ccsc2)CC1)=O)C(C)C c1(OC)ccc(C(=O)NC2CC(NC(=O)C3CC3)C(O)C2)cc1C(F)(F)F c1(C(N2CCC(C)C2CNC(=O)CC2(C(F)(F)F)CC2)=O)cc(O)cc(Cl)c1 N1(C(C(c2cccnc2)NC(c2cc(C)on2)=O)=O)CCC2CCCC12 C1(C(=O)NC23CC(NC(=O)COCC4CCOCC4)(C2)C3)CCC=CCC1 C1(C)(C(=O)NC(C)Cc2nn[nH]n2)CCCN(C(c2cccnc2)=O)C1 C1(CC=C)(C(=O)NC2COCC2CNC(c2cc(C(C)C)on2)=O)CC=CC1 c1(CNC(C)(CO)C2CCOC2)ccc2c(c1)NC(=O)C2 C1(C(C)NCc2c(C)noc2)CCN(C(=O)OCCCCCl)CC1 C1(NC(c2c(CSC)cccn2)=O)CN(C(=O)C(C)C2CC2)C2CCCCC12 c1(CNC2C(NC(C(C(=O)OCC)(C)C)=O)C2)ccc2nnnn2c1 N1(C(Cc2c(O)nc(=N)[nH]c2)=O)CCC(C2CC2)C1CNC(=O)C1=CCCCC1 C1(CC(=O)OCC)CCCCN1C(c1sc(Cl)nc1C)=O.C1CC(=O)N1 CCC(C(C)CN(C)C)NC(=O)C(C1CCCC1)NC(c1ccc(C(C)=O)o1)=O N1(C(C2(C)CC2Br)=O)CCN(c2nnc(CO)s2)CC(O)C1 c1(C(=O)NCC2CN(C(=O)C(F)(F)C3CCCC3)C2)cccc2c1C(=O)NC2=O c1(OC)ccc(C(=O)NCC2(C(N)=O)CN(C(c3coc(C)n3)=O)C2)c(F)n1 N1(C(c2c(C)con2)=O)CCCC(C2CN(C(C3(C)CC(C#N)C3)=O)C2)C1 Cc1ccc(CCC(=O)NCCC2CC(NC(=O)CN3CC=CC3)C2)cn1 C(=O)(C(C(C)O)N(C)C)N1CC(C(=O)NCCc2ncoc2C)(CC)C1 N1(CCC(=O)NC23CC(CNC(CSCC#C)=O)(C2)C3)CCc2ccccc2C1 Cc1sc2ncc(C(N3CCC(O)(CNC(c4cnccn4)=O)C3)=O)n2c1C CCC(C)CC(C)C(=O)N1CC2C(CC(N3CCCSCC3C)=O)C2C1 CCCC(C)C(=O)N1CCC(CCNC(=O)CNC(N2CCCC2)=O)CC1 CC1(C)CC(NC(C2CCS(=O)(=O)N2)=O)CN(C(=O)C(F)(F)CO)C1 C1(NC(=O)C2=CCC2)COCCC1NC(c1c[nH]nc1C1CCCC1)=O N1(C(c2nc(C)sc2)=O)CCC(NC(C23CSCC2C3)=O)C(CO)C1 C1(NC(C(C)OCCOCC)=O)CCCCC12CCCN(C(=O)CNC(C)=O)C2 C1(C(C)C)CN(C(=O)OC(C)(C)C)CCN1C(c1ccc(C2(C)CCO2)cc1)=O c1(C(N(CC(CN(C(C(C(C)C)SCC)=O)C)O)C)=O)ccc([N+](=O)[O-])cn1 Cc1cnc(O)cc1C(N1CC(n2cc(Cc3cccnc3O)nn2)C1)=O N1(C(C=COCC)=O)CCN(C(=O)COCC2CC3CCC2C3)CC1C1CCC1 CC1CC(NC(=O)CNC(=O)CNC(=O)CCc2cncn2C)CS1 CC1CSCCN(C(C2(CF)CCN(C(c3cnc(Cl)n3C)=O)C2)=O)C1 N12CC=C(COC(C)C(=O)NC(CC)CC1=O)CC2.C(=O)(C(C)(C)C)NC CN1N=C(C(=O)N2CCCCCC2C(=O)NCCC2CCCCC2O)CCC1=O C=CC1OCCC1C(=O)N(C)Cc1cccc(CNC(=O)Cn2nccc2C)c1 Cc1cc(F)sc1C(N1CCCCC1C1CCN(C(=O)CC2(CO)CC2)C1)=O c1(C(C(=O)NC2C(CNC(=O)CCc3cccs3)CC2)(F)F)cccc(F)c1Cl N1(C(Cn2c(C)ccn2)=O)C2CCCC1CN(C(=O)C(C)(C)NC(=O)C=COC)C2 c1(C(N2CCCC(CN(C(CCC=CC)=O)C)C2)=O)cc2c(nc1O)CCOC2 Cc1cc(-c2ccc(C(N3CCC(O)(c4cnn[nH]4)C3)=O)cc2)oc1C CCCCC(C(=O)NC1CC(F)(F)C1)N1CC[Si](C)(C)CC1 Cc1ncc(CCC(N2CCC(N(C)C(c3cncc(Cl)c3Cl)=O)C2)=O)c(O)n1 N1(C(c2c(C)sc(Br)n2)C(=O)NC2CCC2)CCOC(C2CCCO2)C1 c1(CC=CC)ccc(C(=O)NCC(C)CN2CCN(C)CC2)cc1 Cc1ncc(C(N2CCN(C(C3CC3c3cccc(F)c3)=O)CC2)=O)cn1 c1(CC(=O)N(C2CCN(C(C(C)C3(O)CCC3)=O)CC2)C)ccc2occc2c1 C(=O)(CCC(C)S(C)(=O)=O)NC(CN(C(C(C)(C1(C)CC1)OC)=O)C)(C)C N1(C(CN(C)C(=O)C2CC2)=O)CCC(NC(=O)Cc2cnccc2Cl)C(CO)C1 c1(NC(C(C=C=C)C)=O)cccc2cccc(Cl)c12 C1(C(=O)NCCNC(C2CN(C(C(C)C3CC3)=O)C2)=O)CCCN1C=O c1(OC)cc(N)c(C(N2CCN(C(=O)CCC3CC3)C(CF)C2)=O)cc1Br C1(NC(CCCCCC)=O)CN(C(c2cc(OC)n[nH]2)=O)CC2(CCC2)C1 C12(NC(c3cccc(F)n3)=O)CCCC1N(C(=O)Cn1cncn1)CC2 C(=O)(CCCCCN=[N+]=[N-])NC(c1c(C(N2CC(C=C)C2)=O)con1)C N1(C(C(N2CCCCCC2)C)=O)CC(NC(=O)C(C)c2ccco2)C2CC2C1 c1(C(N2CCC(C(C)(C)NC(C(C(C)C)NC(C)=O)=O)C2)=O)cncc(Cl)c1Cl c1(CNC(CCN(C(c2c(CC)c[nH]c2)=O)C(C)C)=O)cc(Cl)ccn1 C(F)(C(=O)NOCC1(C)CC1)C1CCN(C(C2(CC=C)CC=CC2)=O)C1 c1(CNC2(C(=O)OCC)CC(CO)C2)cc(S(=O)(=O)N(C)C)cn1C c1(OOCC(=O)OCc2nnc(CCC)s2)ccc(O)cc1O.OC C(CCC(=O)NC1CCCC1NC(c1nscc1Br)=O)N(C)C c1(CC(=O)NC(C=CC(=O)N(CCC#C)C)C)cn(C)nc1C C(=O)(C1=C(S(=O)(=O)CC)CC1)NCC(C)(CNC(=O)CCF)OC C1(C(N(C)CCNC(c2c[nH]c(C#N)c2)=O)=O)CC2(CCC(F)(F)CC2)C1 c1(N2CC(CN(C)C(c3ccnc(Cl)c3Cl)=O)C2)nc(C#N)ncc1Cl N1(CC)CC2CCC1C1CN(N3CCCC(C(F)(F)F)C3)CC21.C(C)(C)(C)OC=O C1(CCNC(C(c2ccccc2)SC)=O)CCCN(C(=O)CC2CC(C)=NO2)C1 c1(CNC2CC(CCC(N)=O)C2)cc(Br)c(Br)cn1 C(=O)(CCC1=CCc2ccccc21)NCC1(C)N(C(CC(C)C(F)F)=O)CCC1 N1(C(C2ON=C(C)C2)=O)CCOC2CCN(C(C3(C)CC(F)(F)C3)=O)CC12 c1(C(=O)NC2C(C)CN(C(c3ccccc3O)=O)C2)c[nH]c2cc(F)ccc12 c1(CNC(=O)CN(CCCOCC(F)(F)F)CC)ccccc1OCc1ccccc1 C1(CNC(=O)Nc2ccc(OC)nc2Br)CCCn2cc(C)nc21 CS(=O)CCC(=O)NC1CCC(NC(C2CC23CCCC3)=O)CC1 c1(C(=O)NC(C)C(N)=O)cc2n(n1)CCN(C(c1cnc3c(Cl)cccn13)=O)C2 c1(CN2CC3(CC(NC(c4cccc(Cl)c4)=O)C3)C2)ccc2c(c1)CCCC2 C1(NC(CC(C)(C)OC)=O)CC2CN(C(c3snc(Cl)c3Cl)=O)CC2C1 N1(C(CC(C=C)CC)=O)CCC=C(C(=O)Nc2cc(C#N)cnc2C)C1 c1(OC)cc(C(=O)NCC2CC2NC(=O)C(c2cccs2)C2CC2)cc(Cl)c1 C1(C(=O)O)(NC(=O)CNC(c2ccc(C(=O)NCC3CC3)o2)=O)CC12CC2 c1(OC)cc(C)c(C(=O)NC2(C3CN(C(=O)C4=CCCCC4)C3)CC2)cc1Br CCC(CC(=O)NC1(C)CC(C(=O)OC)C1)NC(=O)C(CN(C)C)CC c1(SC2(CNC(=O)NCc3cc(-c4ccccn4)ns3)CC2)ccc(F)cc1 c1(C(N(C2CCN(C(=O)COCC(F)(F)F)C2)CC)=O)cc(C(F)F)cc(F)c1 c1(OC)ccc(C)cc1CCC(N1CCOC(CCP(C)(C)=O)C1)=O C(CCCC(C)(C)C(=O)NNC(=O)C1SCCCS1)NC(C1C(C)CC1)=O C(CC1=CCN(C(c2ccc3sncc3c2)=O)CC1)NC(C1CCC(CC)O1)=O n1(CC)c(CNC(N2CCN(C(N3CCN(CC)CC3)=O)CC2)=O)nnc1C Cc1cc2c(C(=O)NCC#CCNC(c3snc(O)c3Cl)=O)nccn2n1 c1(C(C(=O)NCCOC)N(CC=CC(=O)NC)C)ccc(OC)c(C(F)(F)F)c1 CCC(CC)C(F)C(=O)N1CC2(CC(C(N3CCOC(C)C3CO)=O)CO2)C1 c1(NC(CNC(c2c(CC)cccc2)C(=O)NC)C2CC2)ncnc(Cl)c1CC CC(N=c1[nH]c(N2CCC3(CSC3)C2)nc2ccsc12)C1CSC1 c1(C(=O)NC2CN(C(C(=O)NCC)=O)C(C)C2)cnc2[nH]ncc2c1 Cc1cnc(C(=O)NC2CCCC2NC(C2CCCCC2)=O)cc1Cl CC1(NC(C2CCOC2CNC(C2CC3CC2CC3O)=O)=O)CCCCCC1 C(c1ncc(C)[nH]1)=CC(=O)N(CCC)CCNC(c1cnc(SC)[nH]1)=O C(=O)(CC(Cc1ccccc1)SC)N(C1CC(NC(C2(CCC)CCC2)=O)C1)C Cc1ccc(N)cc1C(=O)NC1CC2(C1)CN(C(=O)CCN1CCC1)C2 c1(C(N(c2c(C)cnc(SC)n2)C2CCCNCC2)=O)ccc(Cl)c(Cl)c1Cl N1(C(CN2C(C)CC2)=O)CCCC1CN(C)C(c1cnn(CC(F)F)c1)=O c1(NC2CN(C(c3nn(C)c4c3CCC4)=O)CC3(C2)CC3)c(F)cccc1[N+](=O)[O-] c1(C(N2CC(CN(C(C(C)n3ccnc3)=O)C)C2)=O)cn(CC(N)=O)nn1 CC(C)(C)C#CC(=O)OCC(=O)NC1CC2(c3ccccc3)CC1C2 c1(C(=O)NCC2CC(NC(C(C)CF)=O)C2)c(F)cccc1Br Cc1ccnc(CCC(=O)NC2CC2NC(C2(C(F)(F)F)CC=CC2)=O)c1 c1(C(N2CC(CNC(CCC(=C)Cl)=O)C(N(C)C)C2)=O)ccc(NC)c(F)c1 N1(C(COCCC#C)=O)CCC(=C)CC1C(N1CC(C)CC1CC)=O C1(NC(=O)Cc2cnc[nH]2)CC2(CCC(NC(C3(Cl)CC3)=O)CC2)C1 c1(C(N2CC(O)(C(C)NC(c3cc(Cl)on3)=O)C2)=O)nc(O)[nH]c(=O)n1 c1(CC)nncn1NC(=O)CCC1(C)CCN(C(C2=CC(CC)C=C2)=O)C1.OC c1(C(N2CCCC(F)(CNC(CN3C(C)CC3)=O)C2)=O)cc(O)cc(N)c1Cl N1(CCC)CCCC1C(=O)N(CC(=O)NCC1CCCN1CC)C1CC1 n1(CCC)c(C(=O)NCC23CCC(C2)N(C(=O)C(C)SC)C3)cc2ccccc12 C12(NC(C(C)(F)CNC(C3CCO3)=O)=O)CCCC1OCC2 c1(-c2nc(Cc3c(C)nn(-c4ccncc4)c3)on2)cnn2ccncc12 C1(C(N2C(C#C)CCC2)=O)COCCN(C(C2CC(C)C2)=O)C1 N1(C(C2CC(SC)C2)=O)CCC(N(C(=O)CCCSC)CC2CC2)CC1 c1(C(=O)NC(C(c2c(OC)cccc2)OC)C)ccn2nnnc2c1 C(=O)(CCS(C)(=O)=O)NCC1C(NC(Cc2c(C)ccnc2)=O)C1 C(C(C)N=c1[nH]c(N2CCc3cc(C)cc(C)c3C2)nc2cc[nH]c12)OCC N1(C(C2C(OC)CCC2)=O)CC2CCC1CN2C(=O)C1=C(C)CCC1 C(c1ccccn1)=CC(N1CC=CC(NC(C2(n3cnccc3=O)CC2)=O)C1)=O c1(CCC)nc(C)c(C(=O)N(CCNC(c2ccc(C(C)F)cc2)=O)CC)s1 c1(C(=O)OC)ccc(C(=O)NC2CC(NC(c3ccsc3Cl)=O)CC2O)cc1 N1(C(C(c2ccoc2)NC(CC(C)SC)=O)=O)CCC(C2CCCC2)C1 N1(C(C2(COC)CC=CC2)=O)CC=CC(NC(=O)CC2NC(=O)NC2=O)C1 C=CC(O)(C(=O)NCC(C)CNC(C1(CCc2ccccc2)CC1)=O)C(F)(F)F c1(C(=O)NC2CCCCN(C(C3=NOC(C)C3C)=O)C2)ccc(P(C)(C)=O)cn1 N1(C(C(C)OCCCC)=O)CC2(CCCCN(C(C3CC(SC)C3)=O)C2)C1 C1(C(N(C(C)CNC(=O)CCSCc2ccccn2)C)=O)CCc2n[nH]cc2C1 N1(C(COCCC(C)C)=O)CCC(NC(=O)CC2CC3CC3C2)C(F)C1 c1(C(=O)NCCC(C)N(C)C(c2c[nH]nc2F)=O)cc(F)c(O)c(F)c1 C(=O)(C(C)(C)C(C)(F)F)NCC1C(C)CN(C(c2cc(N)cnc2Cl)=O)CC1 C1(NC(C(C2CCCO2)NC(C2C(C)CC=CC2)=O)=O)CNC(=O)C12CC2 c1(C(C)NC(C2(CCNC(C(C)OCCCC)=O)CC2)=O)cccc(F)c1 C1(CNC(=O)NOCC2CCC2)CCCC1c1ccccc1 C1(C(=O)NC(CN(C(=O)C=C(C)C(C)C)CC)C)CCCN(C(c2ccsc2)=O)C1 CC(C)(C(=O)N1CCC2C(C(=O)NC3CCN(CCCO)C3)C2C1)C(N)=O.C=O C1(CNC(N2CCCC2c2ccc(OC(F)(F)F)cc2)=O)CC2CC(C1)C2 c1(C(C(=O)NCC=CCNC(c2cc(CCC)on2)=O)O)cccc(C)c1 c1(NC(C(=O)NC(c2ccc(OC)cn2)C)=O)cnc(N(C)C)cc1C C(=O)(C1CCc2nccn21)N1CC(Cc2ccc(C)s2)C1.C1(C(=O)N)(C)CCCCC1 Cc1cccc(C(=O)NCC2(C)CN(C(c3csc(C(C)C)n3)=O)CCO2)c1Cl c1(C(=O)NCC2CC2)cc(O)nc2c1CN(C(=O)CC1CCC1)CC2 c1(OC)cccc(C(=O)NCCC2CC(NC(C3(C)CCC(=O)N3)=O)C2)c1 c1(CN(CCC(CC)(F)F)C)ccncc1[N+](=O)[O-] O=C(N=c1nn[nH]n1-c1ccncc1)c1ncccc1O.CCC(F)(F)F CCCCCCC(F)C(=O)N(C)CC1(O)CN(C(C2CC3C=CC2CC3)=O)C1 c1cc2c(cc1CCCn1cc(-c3cc4ccccc4s3)nn1)OCCO2 N1(C(=O)CCC2CCC2)CCCC2CN(Cc3cnsn3)CCC12 c1(C(CC)=O)cccc(N(C(=O)CN2CCSCC2)CC(F)F)c1 Cc1cc(C(N2CCN(C(=O)CNC(=O)CCCCO)C(C)C2)=O)c(O)c(C)c1 C1(CNC(C(CC#C)C)=O)(COC)CCN(C(=O)C=C(C)C2CCCCC2)CC1 CC(CC(C)(F)F)C(=O)N(C)CC1CCCCN1C(=O)CNC(=O)CC(C)(C)C c1(CC)ccnc(C(N2CC(n3ccc(C(=O)N(C)C(C4CCC4)C)n3)C2)=O)c1 c1(C(N(C(CNC(c2nc(C(C)OC)sc2)=O)C)C)=O)cnc2c(ccn2C)c1 CC1CCC(C(N)=O)CN1C(c1ccccc1)=O.C12COCC1N2 C1(CC=C)(C(=O)NC23CC(CNC(c4cnsc4)=O)(C2)C3)CCCC1 c1(OC)c(C)cc(NC(C2(C)CCN2)=O)cc1I C1(C(=O)NOC2CCC2)CCN(C(=O)C2CCCC2CF)O1.C1(CC=O)CCC1 Cc1cc(C(N2CCC(NC(=O)CC3(O)CCC3)C2C)=O)sc1-c1cccs1 c1(NC(C2CC(Nc3ncc(CC)cn3)C2)=O)cc(C)c(F)cc1Br c1(C(=O)NCCC(CCNC(C(CC#C)CC#C)=O)C)cc2c(nn1)CCCC2 Cc1cc(CC2(C(=O)NC3CC(NC(c4cc(O)n(C)n4)=O)C3)CC2)ccc1F c1(NC(c2ccc(-c3nn[nH]n3)cc2)=O)ccc(Br)c2c1CCCC2 c1(NCCS(=O)c2ccccc2)[nH]c(=NC2CC(CO)C2)nc2scnc12 c1(NC(C)=O)ccccc1CC(=O)NCC(O)CN(C(=O)COC1CC=CC1)C c1(CNC(C2CNCCCO2)=O)c(Br)cccc1[N+](=O)[O-] N1(C(c2cc(C)on2)=O)CCC2(CCC2)C(NC(=O)CCCN2CCOCC2)C1 C1(NC(C2(CC)CCC2)=O)C(C)CN(C(c2cnc3ncccn23)=O)CC1C c1(CCC)nnc(S)n1CC(=O)NC(C)CN(C(=O)CC(C)CC)CC c1(CNCC2(NC(c3ccc(Cl)nc3)=O)COC2)cnc2ccccn12 CC(CC(=O)N(C)CCOCCCN(C)C(C1CC1(C)C)=O)c1cccnc1 c1(C(N2CC(CNC(C3CC(=O)CC34CCC4)=O)C2)=O)ccc2c(n1)CCCN2 n1(CC(=O)NC(COC)CNC(c2sc(C)cc2C)=O)cnc([N+](=O)[O-])n1 N1(C(C(=O)NCc2c(OC)cncc2)=O)CCC(CO)C(NC(=O)C(F)(F)F)C1 C(=O)(C(CCCC)OC(C)=O)N1CCC(C(C(N2CCC(CC)CC2)=O)O)CC1 N1(CC(=O)NCCOCCCNC(c2nc(OCC)sn2)=O)CC2C(CC)C2C1 C1(NC(C(C=C)(F)F)=O)CCN(C(c2ccc[nH]2)=O)C(C)C1 C1(NC(=O)OC(C)(C)C)CCCC(C(=O)Nc2cccc(O)c2Cl)CC1 c1(CSC)nnc(C(c2nnnn2C(C)(C)CC)NCC(C)CCO)n1C c1(CC(=O)NCC(C(C)C)NC(=O)CCc2nccn2C)nc(F)c(F)cc1F C(CN=c1cc(C)nc(-c2cccnc2)[nH]1)OC.c1(C2C(=O)N2)cnn(C)c1 c1(CC(=O)Nc2cccc(CNC(C3C(C)(C)C3)=O)c2)ncn2c1COCC2 C(=O)(C(C)(Cc1ccccn1)OC)OCC.C(C(=O)OC)NC(N)=O c1(OC)cccc(C(=O)NCCCCC2CN(C(=O)COC(C)=O)CCO2)c1N CCCCCC(O)CC(=O)N1CCC2CC12C(=O)NCCC1CCCC1 Cc1ccc(C(=O)NC(C(C)NC(c2c(C)noc2C(F)F)=O)C(C)C)c(C)c1 C1(NC(C(CC)NC(C)=O)=O)CC(N=c2nc(C#N)[nH]cc2Cl)C12CCC2 C1(CNC(C(C)NC=O)=O)C2CN(C(c3ccc(C4CC4)cn3)=O)CC12 C=CCC(COC(C1CC1C(F)F)=O)O.C(=O)(CCOCCN(C)C)NCC Cc1nnc2n1CC(C(=O)N(C)CCN(C(=O)C(C1CCCCC1)F)C)CC2 c1(CCC)cc(C(N2CC(OCCNC(=O)C3=C(Cl)CC3)C2)=O)ccc1Cl C(=O)(C(C)(C)C(N)=O)NCC1(C(=O)NCC(C2CCC2)OCC)CCC1 CCCC(CC(C)C)C(=O)NCC1CC(F)(F)CN1C(=O)C=Cc1ccnn1C c1(C(=O)NC(C2(O)CN(C(=O)CC3CCC(C)(C)C3)C2)C)[nH]nc2ncccc12 Nc1ccc(C(=O)NCC2CC(O)CN2C(c2ocnc2C2CC2)=O)c(O)c1 C1(NC(c2ccc(C)o2)=O)CC2CCC1CC2NC(=O)CC1CC(O)C12CCC2 c1(C(N2CCC(c3ccc(C(=O)OC)cc3)C(O)C2)=O)cc([N+](=O)[O-])cn1C CC(C(=O)N1CCC(C(C)(C)CNC(=O)C(C)O)CC1)C(C)(C)C N1(C(c2c(OCC)ccs2)=O)CC(CNC(C23CCC(CC2)C3)=O)CC1C CC(C)C(C(=O)N1CC(N(C)C(C2CN(C)C(=O)N2)=O)C1)Sc1ccccc1 CC(C)C1=NOC(C)(C(=O)NC2CC3CC2N(C(c2ccncc2F)=O)C3)C1 N1(C(C(CCF)NC(=O)Cn2cc(C3CC3)cn2)=O)CCOC2C(O)CC12 Cc1ccc(CNC(C2(NC(C3C(C)(C)C3(C)C)=O)CCSC2)=O)cn1 C1(NC(C2(C)C(CSC)C2)=O)(CO)CCC(C)(C)CC1 c1(CC(N2C(CC(=O)NCC3CC=CCC3)CCC2)=O)ncccc1F CC1CC(CC(=O)N(C2CC2)CC2CC2)CN1C(c1ccn(C)n1)=O C1(C(N2CCC(NC(Cc3c(C#C)cccc3)=O)C2C)=O)CCC2(CCC2)CC1 C1(C(N(CC(=O)OC)C2CC2)=O)CC1C1CN(C(C2(C)CC3C=CC2C3)=O)C1 C(c1ccc(OCC)nn1)=CC(=O)NCC(C)N(C(CSCC=C)=O)C c1(C(N(CCN(C(=O)C=Cc2cscn2)C)C)=O)cc(C2CC2)nc(O)c1 C1(Cl)(C(N(CC(CN(C(=O)Cc2nc(C3CC3)cs2)C)O)C)=O)CC1(C)C c1(C(=O)NCCCOCCNC(C2CCNC2=O)=O)cccc2cnccc12 N1(C(c2scc(C)c2)=O)CCCCC1C1CCCN1C(=O)CNS(=O)(=O)C1CC1 Cc1oc(C#N)cc1C(N1CC(CNC(=O)CCSc2ccccn2)C(O)C1)=O c1(C(C)=O)cc(C(=O)NCCN2CCN(C(=O)CC3CCC(C)C3)CC2)c(C)o1 N1(C(CNC(C2C(CCOC)CC2)=O)=O)CCN(C)C(CO)C1 N1(C(C2N(C(CC)=O)CSC2)=O)CCCC(N(C(=O)CCc2cnn[nH]2)CC)C1 C(CC(C(=O)N(C)Cc1cncnc1)NC(=O)CC1CC=CC1)OCC C12(NC(=O)C=CC3CCCO3)COC(C1)C(NC(=O)Cc1ccccc1)C2 C1(NC(c2cncc(CC)n2)=O)COC2(CCN(C(c3ccnn3CC)=O)C2)C1 CN1CC(C(=O)Nc2cccc(NC(=O)CC(C)(O)C3CC3)c2)OCCC1 c1(C(N2C(CNC(CC(C)(C)OC)=O)CC2)=O)cc(N)cc(O)c1 c1(C(=O)OC)n[nH]cc1CNC(=O)CN(C1CCC1)C.C1(Cl)(C(=O)N)CC1 c1(C(C)(C)C)c(C(=O)NC2CC(NC(=O)COc3ccccc3F)C2)cccc1F Cc1c(C(=O)NCCC2CN(C(c3coc(C(F)F)n3)=O)CC2C)cccc1N C(=O)(C(CNC(c1cn(C2CC2)nn1)=O)C(C)C)NCC(C=C)(C)C c1(OC)ccc(C(N2CCC(C(F)CNC(=O)C(C)(C)C(C)O)CC2)=O)cc1O c1(NC(C(=O)NC(C)C(C)(C)N)=O)nc(Cl)nc2c1c(I)cn2C CS(=O)c1ccc(NC(c2nnnn2CCCF)(C)CC2CC2)cc1 C1(CC)OCCC1C(=O)NCC1(F)CC(CNC(c2ccn(C(F)F)n2)=O)C1 C(=O)(N=c1cc[nH]cc1F)N(CC(COC(C)C)O)C Cc1cncc(C(=O)NC(c2nocc2C(=O)NCC2(C)CNC(=O)O2)C)n1 c1(C(=O)NCC(CNC(CCc2cc(OC)no2)=O)O)nccc(Cl)c1Cl N1(C(C(CO)N(C)C)=O)CCC2(C(=O)NC3CNC(=O)C34CC4)CCCC12 C1(NC(c2ccc(Cl)c(F)c2)=O)CCCC(C(N2CC3CC2C3)=O)CC1 C12CN(CCO1)CCc1cn(nn1)CCNC2=O.c1(COC)cccnc1 CC(C(=O)NCC1CN(C(c2cncc(F)c2Cl)=O)CCO1)P(C)(C)=O C(C)(C)(CCC(=O)NC(C)CCCC(=O)NC)NC(C(NOC)=O)=O CCC(CC(=O)NC1(CNC(c2ccc(C(C)C)c(C(C)C)c2)=O)CC1)C(C)C C(=O)(CCCCC(C(F)(F)F)NCC1(C)CCCS1(=O)=O)OC C(=O)(CS(=O)(=O)C(C)C)N1CC(NC(c2cc(C)c(O)nc2)=O)CC1(C)C c1(C(=O)NCCCN(C(Cn2ncc(C)c2)=O)C(C)C)cnn2cccnc12 n1(CC(=O)NCC2(NC(CC=C)=O)CC3CCC2C3)nc(C)c2cccnc12 Cc1c(O)ccc(C(N2CCN(CCNC(C3CC3(F)Cl)=O)CC2)=O)c1C C1(C(=O)NCC2(O)CN(Cc3nc(C)on3)C2)CCCC(C)C1 c1(CC)oc(C(=O)NC2CCN(C(=O)C(c3ccc(Cl)cc3)N(C)C)C2)cc1C N1(C(C2(C)CCC2)=O)CCN2CCN(C(=O)Cc3cccnn3)CC2C1 Cc1cc(F)c(C(=O)NC2COC3(C2)CN(C(=O)CC2OCCCO2)C3)cc1F N1(C(C=C2CCC(C)C2)=O)CCCC(C)(CNC(=O)Cc2ccc(Cl)s2)C1 CC1CN(C)CC(C(=O)NCC2(C)CCN(C(c3cn(C)c(=O)n3C)=O)CC2)O1 C1(NC(=O)CCN(C(c2ccc(O)nn2)=O)CC2CC2)(CO)CC2CCCC12 C1(NC(CN(CC(C)C)C(=O)CC2(C)OCCO2)=O)CC(C)OC1=O c1(NC(C2C(=C)C2)=O)cc2nnc(C(C)C)n2cn1.N12CCOC(C1)C2 C1(NC(C2CC23CC3)=O)CN(C(=O)CCc2ccc(Cl)c(F)c2)CCC1F c1(CNC(c2cncc(Cl)c2Cl)=O)nc2c(s1)CN(C(C1CC(O)C1)=O)CC2 C(CCCCC(=O)N(C)N(C(=O)C=CSc1ccccc1)CC1CC12CC(O)C2)SC N1(Cc2c(O)cc(F)cc2)CCC2C1CCCN2c1ncc2cn[nH]c2n1 Cc1sc(C)c(C(=O)NC2CCC2NC(=O)C(O)CC2CC2)c1Br c1(CCC)nc(=NC2CC(F)(CNC(c3ccon3)=O)C2)s[nH]1 CCCCCCCCCCCC(C(=O)NCC1=NOC2(CCC2)C1)N(CC)CC Cc1noc(C)c1C(N1CC(CCNC(=O)CC2CSCCS2)C(C)C1)=O C1(F)(C)CCCN(C(=O)CC2CC(C(=O)O)C2)C1.CN1C(=O)CCC1CC(=O)N C1(NC(=O)C=CC2CCCCC2)CCCCCC1C(=O)NCc1cccnn1 CCC(CNC(=O)Cc1ccn(C)c1)(CC)NC(=O)CNC(=O)C(F)(F)F c1(OC)c(C(=O)NCC2CC(OC)CN2C(=O)C=CC(=O)N(C)C)cc(F)cc1F c1(OC)ccc(F)c(C(=O)NC2CCN(C(c3cccc(N)n3)=O)C2CO)c1F C(=O)(C(C)C(O)C(C)CC)N1CC(F)(NC(NOCCCC=C)=O)C1 C(CCCCC(=O)NC(C1CN(C(=O)Cc2ccc(OC)c(Cl)c2)C1)C)OC c1(CC)ccc(C(=O)N(C(CNC(=O)CCN2CCCC2)CC)C)cc1F O=C(C1CCCc2c(O)cccc21)NCC1CC(O)CN1C(c1csc(Cl)n1)=O C1(CN(C(Cn2c(C)ccn2)=O)C)CC(F)CN1C(=O)CNc1cccc(Cl)c1 Cc1nc(N(C)CC2CCCS2)cc(N2CCC(n3[nH]cnc3=N)C2)n1 N1(CC)CCOCC1NCC1CN(C(=O)Cc2nc(C(C)(C)C)cs2)CC1C CN1CC(NC(C2(NC(=O)C3=CCSC3)CCCC2)=O)C2(CC2)C1=O c1(C(=O)NCCN(C(=O)CC(O)CC(C)C)CCC)ccc(C)c(F)c1N C1(NC(c2cncc(OCC)c2)=O)CC2CCC(C1C)N2C(=O)CCC1(C)CC1 C(=O)(C1=CC2(CCOCC2)C1)NCC(CC=C)NC(=O)CC(F)(F)C(F)F c1(C(N2CC(C=C)C(NC(=O)C(C)CC(F)F)C2)=O)cnc(O)c(C(C)=NO)c1 C1(C(=O)NC(C2(O)CN(C(c3cncc(Cl)c3)=O)C2)C)CN2CCC1C2 N1(C(CCC=C)=O)CC2(C1)SCCC2NC(=O)CCc1ccc(Cl)c(OC)c1 N1(CCNC(C(CSC)C)=O)CCC(NC(=O)C(C2(O)CCCC2)F)CC1 C(=O)(CCC(F)(F)F)NC1(C)CC(NC(C2CCC3(CCC3)O2)=O)C1 C#CC1CN(C(c2ccnc(C)c2N)=O)CCN1C(=O)Cc1cc(COC)no1 C1(CNC(C2C(CC(C)C)C2)=O)CCCCN1C(c1scnc1Cl)=O c1(SC)cccc(CC(=O)NCc2ccnc(N3CCOCC3)c2)c1 c1(C(N2CC(F)(CNC(C(C)Cc3cnc[nH]3)=O)C2)=O)ccc(F)c(Cl)c1 C1(C(=O)NCc2cc(C)oc2)CCCC(NC(C2CCN2C)=O)CC1 N1(C(c2cnn(C(C)C)n2)=O)C2CCC(C2)C1C(=O)NCC1CCN(C)CC1 C1(CC(=O)N(C(C)CO)C)CCN(C(C)CN2CCCC2)C1 c1(C(=O)NCC(CC)(C)NC(=O)Cn2cnnn2)cc(=NS(C)(=O)=O)cc[nH]1 C1(CNC(CN(C(=O)CC2CC3CCC2C3)CC)=O)CCN(CC)CC1 c12cc(cc(F)c1F)C2=O.N1(C(C23CCC(C2)C3)=O)CCC(CCCOC)C1 c1(C(=O)NCCCNC(C(CC)NCc2ncnn2C)=O)cnc2c(c1)CCC2 n1(CCC(=O)NCCC(C)NC(C(CC)C(F)(F)F)=O)c(C)nc2ccccc12 C(C)(N=c1cc(NCc2ccc(Br)cc2F)nc(C)[nH]1)c1c(OC)ccc(F)c1 C1(C(=O)NC2C(NC(C(C)C(=O)OC(C)(C)C)=O)C2)CN2CCN1CC2C c1(CC(=O)NC(C)CC2CCN(C(C3CC(C)C3)=O)CC2)ccc2ccoc2c1 c1(C(=O)NCCCOCCNC(C2C(=C)C2)=O)cc2cc(C)c(C)cc2o1 Cc1c(C(=O)OC(C(F)(F)F)c2ccccc2)sc2ccc(Cl)cc12 C(=O)(C1CCCc2ncc(C)n21)N1CCN(C(C=CCC)=O)CC1CC(F)(F)F N1(C(C(C)CN(C)C)=O)CCCCC1CCCNC(=O)CSc1nncn1C C(c1ccc(Br)cc1Cl)=CC(N1CC(C(=O)NCc2c(C)ncn2C)C(O)CC1)=O C1(C(=O)NC(C)(C)CCF)CN(C(C2(C)CCOC2)=O)CC1(C)C CC(Cc1cnn(C)c1)C(=O)NCC1CC1CNC(C1(c2ccno2)CC1)=O N1(C(CC(C)F)=O)CCCCCC1C(=O)NCCC1CC(C)(C)CO1 C1(C(N2CCCC(C)(CNC(CCC(=C)C)=O)C2)=O)CC2(CO1)CC(F)(F)C2 C1(CNC(CCC(=O)NCCC)=O)CCN(C(c2nn(C)cc2Cl)=O)C12CC2 c1(NC(C2N(C(C3CC4C=CC3CC4)=O)CCC(=C)C2)=O)cc(C)cc(C#N)c1 C12(NC(C(C3CCN(C(CCC(=O)NCCC)=O)C3)C)=O)CCCC1C2(F)F C(CCCC(C)NC(C1CCC1C)=O)NC(C1(SC)CC1)=O N1(C(=O)Cc2cccnc2)CCC(C(=O)NCC2CC(O)C(O)C2)(CF)C1 c1(C(C)NC(CCC)=O)cn(C2COC(CN)C2)nn1 N1(C(=O)NC2C3(CCC(C)OC3)CN2)CCC2(CCC(=O)N2)C1 Cn1c(=O)c2cc(C(N3CCC4(Nc5ncccn5)CC4C3)=O)sc2n(C)c1=O c1(C(N2C(C(N3CCC(OCCC)CC3)=O)CC2)=O)ccc2sncc2c1 Cc1cc(C(N2CCC(CNC(c3cnccn3)=O)C23CC3)=O)c2n[nH]cc2c1 C12(CC3CCCC13)C(=O)N2.c1(COC)sccc1C(=O)OC(C)(C)C c1(C(N2CCN(c3cc(C)ccn3)CC2)C(=O)NC)cnccc1SC C1(NC(C(C)c2cccs2)=O)CCC12CCCN(C(C1CC(=O)NC1(C)C)=O)C2 O=C(C1=CCCC1)NC1C=CCC(C(N2CC(SC(F)F)C2)=O)C1 c1(C(N2CC3C(CNC(c4c(C(C)C)n[nH]c4)=O)(C3)C2)=O)cc(Cl)cc(Cl)c1O CC(C)CCCCC(=O)NC(C1(C(=O)NC2CCCC23CC3)CC1)C N12CC3C(C3C1)C2=O.CC(C)(CSC1CC1(Cl)Cl)Cc1cn(CCO)nn1 O=C(CCC(=O)N1CCCC(CNC(=O)Cc2cscc2F)C1)c1cccs1 N1(C(CC(CC#C)NC(c2ccc(COC)o2)=O)=O)CC2(C)CC1CCO2 N1(C(c2coc(Cl)c2)=O)CCCC2(CCN(C(c3cc(=O)cc[nH]3)=O)C2)C1 N1(C(=O)OCC)CCC(NC(=O)NCC2COC2)CC1 C(=O)(C(C)C(C)(C)C)N1CCC(C(C)C(=O)NCC2(N(C)C)CCC2)C1 Nc1cccc(Cl)c1C(=O)NCCCNC(=O)CC12CCCC1C2 C1(C(=O)NC2(CCCC)CC2)COCC1NC(c1csnc1OC)=O N1(C(C(C=C)OC)=O)CC(NC(C2CC(C(C)C)=NO2)=O)CC1(C)C c1(Cn2cc(C(C)(C)NC(C3CC3C(C)(F)F)=O)nn2)c(F)cc(F)cc1F c1(-c2cncc(C(Nn3c(C)nnc3)=O)c2)n[nH]c2ccc(Cl)cc12 C1(CC)CCN(C(c2cc(CO)on2)=O)C1C(=O)NCn1ccnn1 C1(NC(C(C(C)C)NC(=O)OC(C)(C)C)=O)CC2CCC(C1)N2C(C1(F)CC1C)=O c1(NC(CCOCCCNC(CCc2n(C)cnn2)=O)=O)cccc2c1OCO2 C(=O)(C(F)(F)CO)NC1C(CC(=O)NCC(C)OCC#C)CCC1 c1(CCC(=O)NCC(O)CCNC(c2cccc(N3CCC3)c2)=O)cccnc1Cl N1(C(=O)C=CCO)CCC(O)(COC2CCN(c3snc(CSC)n3)C2)CC1 CCCC(O)C(=O)NC1(CCOC)CCN(C(=O)CN2CCC(O)CC2)C1 c1(-c2onc(C(=O)NCC3N(C(C=C(COC)C)=O)CC=C3)n2)cccc(Cl)c1 c1(CC(=O)NCC2CN(C(CCCOCC)=O)CC(C)O2)ccc2nn[nH]c2c1 C1(NC(C2C(C)CCC2)=O)CC2(C1)CC(CNC(=O)CN1CC(C)(C)C1)C2 c1(C(=O)NC2CC3CN(C(C4CC(OCC)C4)=O)C2C3)cn2ccnc2cn1 CCC(CNC(c1n[nH]c2c1CCCC2)=O)N=c1[nH]c2ccccc2s1 C(CCS(C)(=O)=O)N(CC(=O)OC)C(C1CCCN1Cc1cn(CCCF)nn1)=O C1(NC(CC=C(C)C)=O)CCOC12CCN(C(=O)COC1(C)CCOCC1)CC2 Cc1c(C(N2CCN(C(=O)C(F)C(C)(C)O)C(C)C2)=O)ccc2n[nH]cc12 N1(Cc2cn(CC3(CNC(CCC=C(C)C)=O)CC3)nn2)CCOCCC1=O.SCC C1(C(N(C)CC2CCN(C(c3csc(Cl)n3)=O)C2)=O)CN2CCC1CC2 C1(CC(N2C(CNC(C3(CC#C)CCCC3)=O)CCC2)=O)CCCCC1O c1(C(=O)NCC(CC(C)C)(C)NC(C2CC2C(C)C)=O)cc2cccnc2cn1 Cc1c(Br)ccc(C(=O)NC2C3CCC2CN(S(=O)(=O)CCCCCl)C3)c1F C1(NC(c2ccon2)=O)CN(C(C2C3CC4C(C3)C24)=O)CC1C(F)(F)F Cc1nc(C(=O)NCC2(CNC(C3CCCCS3(=O)=O)=O)CC2)c(C)n1C1CC1 CC1CCC(C(=O)NCC2C(CNC(=O)C(CN(C)C)N(C)C)C2(F)F)CC1 O=C(CC(F)(F)C(F)(F)F)NCC1CC1CNC(=O)C1CC1 N1(C(Cc2ccc(OC)cc2)=O)CC2CCC2(CNC(C2CCCSC2)=O)C1 Cc1nc(CCC(=O)NCC2CCCCN2C(C2CC2(C)C)=O)oc1C C(=O)(C1=CC2(CCOCC2)C1)NCC1CCCN(C(c2c(C)ccnn2)=O)CC1 Cn1nc(C(=O)NC2CCN(C(c3ccsn3)=O)CC2CO)cc1C#N N1(C(c2c(CC)non2)=O)CC(O)CCC1C(=O)NC(C)CCC=C(C)C c1(OC)ccc(CN2CC3(CC3)CC2C(=O)NCCCO)c(Cl)c1 C=C(C(=O)NCC1COC2CCCC2N1)C1CCC1 c1(C(=O)NCCCN(C(=O)CCC(=O)NC)CC)cc(S(N)(=O)=O)c(C)o1 Cc1cc(C(=O)NC2CC(NC(c3cc[nH]c3C3CC3)=O)CC2O)cc(C)n1 N1(C(=O)NC(c2cc(Cl)cc(Cl)c2)C(F)(F)F)CC2(CC(=O)NCC2O)C1 N1(C(CC(C)O)=O)CCOC2(CCN(C(c3c(C4CCC4)cnn3C)=O)C2)C1 c1(C(=O)NC2CC(N(C(C(C(C)C)OC)=O)C)C2)cc2c(s1)CCCC2 C#Cc1ccccc1CC(=O)NCC(C)(C)C(=O)NC(CC)C(C)(C)O N1(CC2(COC)CCC2)C(=O)CCN(Cc2cccc(S(C)=O)c2)C1=O C1(C(C)NC(COCCC#C)=O)CCN(C(=O)C(F)CC2CCCCC2)C1 CCCC(O)CC(=O)NC1CC12CC(NC(=O)CN(C)Cc1ccc(C)cc1)C2 c1(C(C)C(=O)NCCOCCN(C(=O)C(N2CCSCC2)C)C)ccc(F)cc1 C(CC(C)(C)C)(C(=O)NC(C)(C)CN(C(=O)CC1CCCOCC1)C)OC C1(C(=O)NC(CCCC)CNC(=O)CC2CCCN(C)C2)CC2(C1)CC2(F)F c1(C(=O)NCC2(NC(=O)COC(F)F)CCOCC2)c[nH]c2c(Cl)cccc12 Cc1cnc(NCC2CCOCC2(C)C)c(S(=O)(=O)NC(C)CN(C)C)c1 C1(C(=O)NC2CN(C(=O)CSc3cnn[nH]3)C2)CCN(C(N2CCCC2)=O)C1 N1(C(C2C(C(C)C)CCO2)=O)CCC(C2CN(C(=O)C(C)c3cccs3)C2)CC1 Cc1ccc(F)c(C(=O)NC2CC23CC(NC(=O)C(C(C)C)C2CCC2)C3)c1 Nc1c(C(F)(F)F)nsc1C(=O)NC1CCCCC1NC(c1ccnnc1O)=O c1(C(C)C)ccc(N2CCCC(c3nc[nH]n3)C2)cc1[N+](=O)[O-] C1(C(C)C)CN(C(=O)CC2CN(C(=O)CCCC3CCCO3)CCO2)CCCO1 C1(S(N)(=O)=O)(C(=O)NC2CC(N(C)C(c3ocnc3-c3ccccc3)=O)C2)CC1 CC(C)CC(F)(F)C(=O)NC1CCN(C(c2ccc3c(c2)OCO3)=O)CC1F C1(C(C)NC(=O)CCOCCOCCCO)CCCCN1C(=O)CCCF c1(SCCC)ccccc1Cl.C1(C(N2CC(=O)NCC2)=O)COC(=O)C1 N1(C(c2c(C)nn(C(C)(C)C)c2)=O)CC2(CC(NC(=O)C=CS(C)=O)CO2)C1 C(=O)(CC(O)C(C)C)N(C1CCCN(C(=O)COCCF)CC1)CC N1(C(Cc2n(CC)ccn2)=O)Cc2nccn2CC(NC(=O)CCC(C)OC)C1 O(P(=O)(C(C)OC(C1CC1c1cncc(OC)c1)=O)OCc1ccccc1)CC C1(C(N(C2CC(NC(=O)Cn3ncccc3=O)C2)C)=O)CCc2nc[nH]c2C1 CC(C)C(CN(C)C)C(=O)N1CCCC(C(=O)NC(C)(C)CN(C)C)C1 c1(CNc2ccc(C(=O)NCCC)nc2)cc(C)c(Br)c(C)c1 C1(NC(C(C)=CC)=O)CCC(CN2CCCCC2)CC1.C12(CC1)C(=O)N2 C1(N=c2[nH]nc(Cl)c3ccsc23)(c2c(C)cccc2)CN(C(C2(Br)CC2)=O)C1 Cn1cc(C(N2CCC(n3cc(NC(=O)CN4CC5CC5C4)nn3)C2)=O)c(Br)n1 c1(C(N2CCC(CF)CC2)C(=O)NC2CCCC2)cccc(Br)n1 c1(CC(=O)NC2C(O)CCN(C(C(CCCC)C)=O)C2)ccc(S(C)(=O)=O)cc1 c1(CC(=O)NCCCN(C(C2(C)CS(=O)(=O)C2)=O)CC)ccc(Cl)nc1C C1(C(=O)O)(CNC2CC(C)C2)CCCO1.n1(CC(=O)OC)cc(C2(O)CCC2)nn1 C1(C(N2CC(S(C)=O)C2)=O)CN(C(=O)C(C)(Cl)Cl)CC12CCC2 c1(C(N2CC(OCCNC(c3cc(O)cs3)=O)C2)=O)nccc2c(F)cccc12 C(CC(=O)NCC(CC)(CC)SC)(CC(C)C)NC(C=NOC)=O C1(C(=O)OCC)(CC)CCN(C(=O)C=Cc2ccccc2F)CC1 N1(C(C(CC)COC)=O)CC(O)CCC1C(=O)NC1(C(F)(F)F)CC1 c1(OC)cc(Cl)c(C)cc1NC(c1cccc(C(N2CCCCC2)=O)n1)=O Cc1ccc(C(=O)NCCOCCc2ccc(Br)cc2)cc1C N1(CC(CN(CCOCC)C)O)CCN(C(=O)Cc2cnnn2C)CC1 c1(CC)ccc(NC2CON(C(=O)OCCN3CCN(C)CC3)C2)cc1CC C1(CNC(c2ccc(OC(C)C)cn2)=O)C(C)CCCN1C(c1ccc(F)o1)=O c1(C(=O)NC2CCCC(NC(CCCC#CC)=O)C2)ccc(C)c2c1CCCN2 CCC(CC)CCNC(C1CCN(C(=O)CC2CCCOC2)C1C(C)C)=O Cc1cccc2c(C(=O)NCC3(NC(=O)CCC4CC4(F)F)CCOC3)coc12 N12CCOCC(C1)C(=O)NCC2C.c1(-n2cccn2)cc(O)nc(O)n1 C1(NC(N)=O)CCC(C(=O)NCc2nnc(-c3ccco3)o2)CC1 Cc1c(C(N2CC(C)(NC(=O)COC3CCCC(C)C3)C2)=O)cnn1C1CCC1 c1(N(C(c2cccs2)=O)Cc2ccc(OC)cc2)ccc(OC)c(C(N)=O)c1 C(=O)(C(CO)C(F)(F)F)NCc1cccc(C(=O)NCC(C(C)O)O)n1 N1(C(CC2C(C)CCO2)=O)CCOC2(CCC(NC(c3cnco3)=O)CC2)C1 c1(NC(C(C)(Cc2ccccc2)NC(CSC)=O)=O)cn(C)nc1OCC(F)(F)F C(C)(CNC(=O)C(O)CC)(C(C)C)NC(c1nc(C(C)OCC)oc1)=O c1(OC)cc(F)c(C(=O)NCC2CCN(C(c3c(C)nsc3N)=O)C2)c(F)c1 c1(NC(C)=O)ccc(CC(C)C)cc1.C1(CCN(C)C)C(=O)N2CCC(C2)N1 c1(C(=O)NCC(=CC(=O)NC(CC#C)C)C)ccc(O)cc1 Cc1nc(Cl)nc(N2CCCN(C(=O)C(C)NC(c3cccs3)=O)CCC2)c1F C1(NC(=O)C=C2CCC2)CN(C(=O)CCc2nc[nH]n2)C2CCCC12 C1(C)(N)CCSCC1.C12(CC1)C(=O)NCCOCCCNC2=O.COC N1(C(CC(=O)NCC)=O)CCC(C(=O)NCCCCCN=[N+]=[N-])C1C c1(C(N2CC3(CN(C(c4cccc(C)c4F)=O)C3)C2)=O)ccc(F)cc1C#N N1(C(c2ccc(CNC(C(c3ccccc3)C)=O)o2)=O)CC2CC(CO)(C2)C1 C#Cc1cc(C(N2CCC(NC(=O)CC(C)(C)C(F)F)C(C)(C)C2)=O)cc(F)c1 N1(C(C(C)C(C)(F)F)=O)CCCCC(CNC(=O)C=CC2CCCCC2)CC1 Cc1nc2c(C)cc(C(N3CC4CC3CN4C(=O)Cc3cnoc3)=O)cn2n1 C1(C(=O)NOC)CCCC(C)(C)C1.C1(CC2CCC2)C(=O)NCC=CC1 CCC(CN(C)C)C(=O)N(C)CC=CC(=O)NCC(CSC)OC CN(C)S(=O)(=O)NCC(N1CCCC1C1(O)CN(C(=O)CCc2nc[nH]n2)C1)=O CC1CCN(C(=O)Cn2cc([N+](=O)[O-])cn2)CC1NC(c1cn(C)c(=O)n1C)=O c1(C(C(=O)NC2CCCC2)N(C2(C#C)COC2)C)cnc(N(C)C)nc1 N1(C(C2(C#C)CCC2)=O)CC(C2CN(C(C3CC(=O)N(OC)C3)=O)C2)C1 C=CCCCCCC(=O)N1CCCC(C(C)(O)CNC(C2(F)CCC2)=O)C1 C#Cc1cnc(C(=O)NC2CC(C(=O)NCC(CCC)CCCC)C2C)c(C)c1 c1(C(N(CC(C)NC(=O)CC=C2CC2)CC)=O)ccc(CO)o1 C1(NC(CC=[SH]C)=O)CCC(CNC(=O)OC)C1.c1ccccc1 C(N=c1[nH]c2c(c(=NCCc3nc[nH]n3)[nH]1)SCC2)C1(C)N=C(C)SC1 Cc1nnc(SN2CCCSCC2)n1C(c1ccccc1)C c1(C(=O)NC2CCC(NC(C3C4CNC(=O)C34)=O)C2)cccc2c1OCCC2 C1(NC(=O)C(O)CN2CCOCC2)CC2(C1)CC2NC(c1csc(Cl)n1)=O N1(C(C(C(C)C)SCc2ccccc2)=O)CC2(C1)CN(C(=O)C(C)C1CC1)C2 O=C(C1CCOc2ccc(Cl)cc21)NC1CCN(C(C2(C(F)F)CCC2)=O)C1 c1(N(N2CCC(C=O)C2)C)ccc([N+](=O)[O-])cc1C(F)(F)F.C(=O)CNC=O S(=O)(=O)(C(C)CN=c1nc2c(cnn2C)c(NC(C)CCCCSC)[nH]1)NC C12(CC)CN(C(=O)CCOC(C)C)C(CNC(c3nc(=O)n(C)[nH]3)=O)(C1)C2 C1(C(=O)NCC2CCCN2C(=O)C=CBr)COCC(=O)N1C(C)C C(=O)(CCCC(C)O)N1CCCC(C2OCCN(C(c3c(C)nn(C)c3)=O)C2)C1 Cc1cc(C(=O)NC(C)C(C)(C)NC(=O)C=Cc2c[nH]nc2C)ncc1C(N)=O N#Cc1ccc(NC(C2(O)CCN(C(c3nocc3Br)=O)C2)=O)cc1F C1(NC(CC2(C=C)CC2)=O)CC(C)(NC(c2ccsc2-n2cnnn2)=O)C1 c1(C(=O)NCCc2cccc(C)c2)nc(=NC2CC2C(C)C)cc[nH]1 c1(C(=O)NCCN(C(C(C=C)O)=O)C)cc(C)ncn1 c1(C(N2CCC(N)(CC)C2)=O)ccc([N+](=O)[O-])nc1 N1(CC)CC(NC(C2CCN(C(C3CN(C)C3)=O)C2)=O)C(C)C1 c1(OC)c(F)c(C(C)OC(c2cc3ccc(O)cc3[nH]2)=O)cc(F)c1F c1(C(N2CCCC(CC(=O)NC3(COC)CCC3)C2)=O)nc(C)ccc1F n1(CC(=O)NCC=CCNC(c2cc(C)c(Cl)s2)=O)ncn2cccc2c1=O C(C(=O)NCCCN(C(=O)C=C(C)Cl)C1CC1)(c1cccs1)SC C1(C(C)C)CCCN(C(=O)NC(C)C2CC2)CC1 c1(CC(C2CN(N3CCC3C=O)C2)NC(C=CC)=O)cc(N(C)C)cc(Cl)c1.OC CC(=O)C(C)(C)CC(=O)N(CC(C)C(=O)NCC(C)C)C Cc1cc2nc(O)[nH]c2cc1C(=O)OCC1CCC1C(C)(C)C N1(C(C(C)NC(C)=O)=O)CC(O)(C2(CNC(=O)CCCN(C)C)CC2)C1 c1(C(C(N2CC(NC(c3c(C)ncs3)=O)C2)=O)N(C)C)ccc(F)cc1 C1(CNC(c2n(CCC)nnn2)c2ncnn2CC)CCC2(CCCC2)O1 O=C(C(O)C1=CCCCC1)NCCC1(NC(C2(C(F)F)CCCC2)=O)CC1 c1(OC)cc(C#N)ccc1C(=O)NCC1CN(C(=O)C(C(C)C)OC)CC1(C)C C(=O)(C1=C(C)CCC1)NCC(CO)NC(C(c1cccc(OC)c1)C)=O Cc1ccnc(C(=O)NC(C)(CNC(c2cc(C3(C)CC3)n[nH]2)=O)CO)c1N N1(C(CC(=O)NCC#C)=O)CCC2(CC1)CC2NC(c1n[nH]cc1C)=O c1(C(N2CC(NC(C3SCCS3)=O)C(F)CC2)=O)ccc2nc(O)[nH]c2n1 C(=O)(CCC1=NNC(=O)CC1)NC(C(C)NC(=O)CSc1ccccn1)(C)C CC1=C(C(=O)N2CCN(C3CCC(NC(c4occc4F)=O)C3)CC2)CCC1 Cc1nc(C)n(O)c1C(N1CCC(N(C)C(c2c[nH]cc(Cl)c2=O)=O)C1)=O N1(C(C(=O)OC(c2cc(Br)c(F)cc2F)C#C)C)C(=O)c2ccccc2C1=O C(=O)(C1CCCc2nccn21)N1C(CNC(c2ccc(CO)nc2)=O)CC(F)C1 C1(C(=O)NC2(C)CCN(C(CC(CC(=O)OC)C)=O)CC2)CCCC(F)(F)CC1 C#CC1(C(=O)NC2CC=CCC2C)CCN(C(c2nc[nH]n2)=O)C1 N1(Cc2cnc(N(C)C)o2)CCC(O)(CC(=O)Nc2cccc(F)c2Cl)CC1 c1(N(CCS(CC)(=O)=O)C)cc(S(=O)(=O)N2CCOC(C3CC3)C2)ccc1C#N c1(OC)ccccc1COC(C1CC1COc1ccccc1C)=O CC(C)CCC(F)C(=O)N1CCC(NC(=O)C=CCO)C1C c1(NC(=O)NC2C(C)(CC)C2)ccc2c(c1)CCCC(=O)N2 c1(C(C)C)cc(C(=O)NCC(N)C(F)F)nc2ncnn12 N1(C(c2coc(Cl)n2)=O)CC2CCN(CCSc3ccc([N+](=O)[O-])cc3)CC2C1 N1(C(c2cc(OC)cc(F)c2)=O)CC2(CCCC2)C1C(=O)NOCC(C)(C)O Cc1[nH]nc(C(=O)NC2C=CCN(C(C3CCCC(C)C3)=O)C2)c1Cl C1(CNC(CSC)=O)CC2(CCN(C(c3ccc(OC)c(OC)c3)=O)CC2)CO1 N1(C(=O)Cc2cccnc2)CC2CCCN(C(C3CCCCC3O)=O)C2C1 c1(OC)ccc2nc(-n3nc(CS(C)(=O)=O)nc3C3C4CCCC34)c(Br)n2n1 N1(C(CNC(C)=O)=O)CC2(NC(c3[nH]c(C4CC4)nc3C)=O)CC1C2 CC(C)(CN(C(=O)CC1C=CCC1)CCO)C(=O)N1CC(C)(O)CO1 c1(NC(c2c(C)ccc(F)c2)C)nc(=NC(C)c2ncccn2)[nH]c2ncn(C)c12 C(=O)(C(F)CCC(C)C)NCC(C(=O)NCc1ccc(OC)cc1)O Cc1cn(C)nc1C(=O)NC1CCCC1(C)CNC(c1ccc(F)cc1)=O CCC1=NOC(C(=O)N(CCCNC(=O)CC(C)n2ccc(C)n2)C)C1 C1(O)(C(N2CC(NC(=O)C(F)C3CCCC3)C(O)C2)=O)CCCCCC1 c1(C(N2C(C(=O)Nc3c(C)noc3C)CSC2)=O)cccn(C)c1=O c1(CCCOC)nc(-c2cnn(-c3ccccn3)c2)n(-c2ccc(F)nc2)n1 c1(NCC(CCC)OC)nc(N2CCC(C3CC3)C2)nc2c1ncn2CC C1(C)(CC)C=C(C(=O)NC(CC(N)=O)C(=O)NCC2CCOC(C)(C)C2)C1 c1(C(N(C2CN(C(CC3CC(OC)C3)=O)CC23CC3)C)=O)ccn2cnnc2c1 O=C(C1c2c[nH]nc2CN1C(c1cccnc1)=O)NC1CC2CC1CC2(F)F CCC(CC(F)(F)F)C(=O)NC1(c2ccc(F)c(Br)c2)CC1 n1(CC)ncc(C(=O)NC(c2ccccc2)C(=O)NCC(C)COC)c1C N1(C(C=Cc2cc(OC)ns2)=O)CCCC2CCN(C(=O)CC3=CCCC3)CC12 C(C)(C(CC(=O)N1CC2CCCCC12)NC(=O)CCCCN(C)C)OC c1(C(=O)NC2C(NC(C3N(C)C(=O)CC3)=O)CCCC2)cc(F)cc([N+](=O)[O-])c1 c1(C(=O)NCC2(O)CN(C(C(C(C)(C)C)OC)=O)C2)cc(C)cc2ccncc12 CCC(CC(=O)N1CC2CC1(C(=O)NOCC1CCCO1)C2)C1CC1 C(CC(=O)NCC1(C)CCN(C(=O)C(C)(C)n2cnnn2)CC1)(C(C)C)OCC N1(Cc2ccc(C#C)s2)CCC2(CC1)CC2NC(=O)Nc1cnc(C#N)nc1 C#CCC(C(=O)NCCC1CCCN(C(=O)Cc2cscn2)C1)C1CC1 c1(C(N2C(CN(C)C(C3(C)CC4(CC4)C3)=O)CCC2)=O)ccc2c(ccn2C)c1 C(=O)(C(C(CC)C(C)C)N(CCc1ccccc1)CC)NCCC C#Cc1cnc(C(N2CCCC(CC(=O)NCC(C)CCO)C2)=O)c(C)c1 Cc1c(NC(=O)C(CCOCCO)NC(=O)C(C)C(F)F)cnn1C(C)C C(=O)(C(CC1CCC1)NC(=O)C(Cl)Cl)N1C(CC(=O)N(C)C)CC1 C(=O)(C(C)(C)C(C)(C)NC(=O)C(C)C)NCCOC1CCCC(C)C1 C(=O)(C(CNC(C1CNC(=O)O1)=O)CC1CCCC1)NCCc1cn(CC)nc1 C1(O)(CNC(=O)CCOCC2CCCO2)CCCN(C(c2cc(Cl)no2)=O)C1 C1(C(C)NC(C2(CC=C)CCC2)=O)CCCN(C(=O)C=CC(=O)N(C)C)C1 C(=O)(C1=C(Cl)CCOC1)NCC(=O)NC(C#C)CC(C)(C)C.N12C3CCC(C3)C1C2 CC1(C(=O)NCC2(NC(c3ccc(-c4cscn4)nc3)=O)CC2)CC2(CC2)C1 N1(CCNC(CN(CCC#C)C)=O)CCC(NC(c2coc(C(F)F)n2)=O)CC1 CCC(C)(O)C(=O)N1CCC(CCNC(=O)CCc2ccc(Cl)nc2)C1 Cc1cc(C(=O)NCC2C(C)CCN2C(c2ccc(Br)c(F)c2)=O)c(C)cn1 c1(C2(C(=O)NC34CC(NC(C(C)=C(CC)C)=O)(C3)C4)CCCC2)ccc(C)cc1 C1(C(N(C)Cc2cn[nH]c2)=O)CC12CCN(C(C1CC1C#N)=O)CC2 C12C3CC4C(C3N1)C24.C1(CC(=O)NCC(=O)NC(N)=O)CCC2CC12 c1(C(=O)NCCC2(O)CN(C(C3C(SC)CCC3)=O)C2)cc(Br)oc1C C1(C(N2CCC(CC)C2CNC(=O)C(C)C2CCC2)=O)CCCC1C1CC1 c1(CC(=O)NCC2(C)CCN(C(=O)CO)C2)c(F)ccc(Br)c1F c1(OCC)cc(N2CCC(C)(CNC(C3CC3F)=O)CC2)nc(C)n1 Oc1nc(NCc2cc(Cl)ccc2C(F)F)nc2c1ncn2C(F)(F)F N1(C(CS(N)(=O)=O)=O)CC2CCC1C1CN(C(C3(O)CCOC3)=O)CC21 c1(C(N2C(CO)CC(NC(CC=CC=C)=O)C2)=O)nc2cnccc2s1 C1(C(=O)NC(C)C(N2CCN(C)CC2)=O)CC2CN(C(C)(C)C)CC12 c1(C(N2CC(NC(C(C)C(F)(F)F)=O)C(O)C2)=O)c[nH]c2ccncc12 c1(OC)ncccc1S(=O)(=O)NC(=O)CC1COCC(C)(C)O1 c1(C(N2C(C)CC(CCNC(=O)COC3CCC3)CC2)=O)ccc2cncn2c1 c1(C(N2CCCC(CNC(C3N=C(C)SC3)=O)CC2)=O)cccc2c1ccn2C C1(NC(C2C(C)(C(C)C)C2)=O)CCCN(C(c2cnn(C)c2C2CC2)=O)CC1 C(=O)(C(C)C(C)CNC(C1(C(F)F)CC(=C)C1)=O)NCCN(C1CC1)CC C(C)(CNC(=O)COCC1CC1)(C(C)C)NC(C(n1ncc(C)c1)C)=O C1(COC)(NC(=O)Cc2ccc(O)nc2)CCCN(C(=O)C(C)CSC)C1 n1(C(=O)NC2CCC2CNC(=O)C(c2ccc(OC)cc2)C)cc(CC)c(C)n1 CC(C)C(C)C(C)CC(=O)NCCCCCNC(=O)CC1CNC(=O)O1 C1(C)(C(N2CC(NC(CSCCC)=O)C(OC)C2)=O)CC(C(C)C)=NO1 CCC(CC)(C(C)C)NC(c1cc(CNC(C2CC(O)C(F)C2)=O)on1)=O N1(C(CCOCCCNC(c2c(C)non2)=O)=O)CCc2cccc(O)c21 N1(C(c2c(C=C)cnn2C)=O)CCCC2(CC(NC(C3CCC(=O)NC3)=O)C2)C1 c1(C(=O)NCC(CN(C(=O)CC2COCCO2)C)O)ccc2c(c1)C(=O)CCO2 C1(C(N(C(C)CCNC(=O)C(F)C(C)(C)O)C)=O)CCC2(CCC2)CC1 N1(C(C2(CCOC)CCCC2)=O)CCN(C(=O)CN(C)C(C)=O)C(C2CCC2)C1 C(C)(CS(C)(=O)=O)NC(CCN(CCOC)C(c1ncc[nH]1)=O)=O c1(C(N2CCC3C(CCN3C(=O)CC(F)F)C2)=O)c[nH]c2ccccc2c1=O C1(C(=O)NCCC2(O)CCN(C(CC(=O)OC)=O)C2)CCc2cnc(C)n2C1 C(CN=C(NCC(C)(O)CN1CCOCC1)NC(C)COC)c1cccc(CC)c1 c1(NC(=O)NC2CC(CN)C(O)C2)cc(-c2noc(C(C)(C)C)n2)ccn1 n1(C(C)C)ccc(C(=O)NC(C(C)NC(C23CC(C)(CO2)C3)=O)C(C)C)cc1=O n1(CC)nc(C)c(C(N2CC3CC2C3NC(c2cnn(CCF)c2)=O)=O)c1Cl c1(CC(C)NC(C2CCN(C(=O)CC3CCCN3C)CC2)=O)ccc(F)c(F)c1 N1(C(CC=CC(C)(C)C)=O)CC(C)(C(=O)NC2(C3COCCO3)CC2)CC1(C)C c1(C(=O)NCC(n2cc(-c3ccccc3F)nn2)C)ncccc1C(F)F C=C(Cl)CCC(=O)N(C)CC1CCCN1C(=O)CC1(N2CCCC2)CC1 N1(C(C(N2CCC(C)C2)=O)=O)CC(N(C)C(c2nc(=O)n(C)[nH]2)=O)C(O)C1 N1(C(=O)CC=Cc2ccc(F)cc2)CC(NC(C2(C(N)=O)CC2)=O)C(C2CC2)C1 N1(C(CC2CC(OC)C2(C)C)=O)CCC2(NC(=O)CCc3cn(C)nn3)CC2C1 C1(CC(=O)NC2COCCN(C(COCCOC)=O)C2)SC2=NCCN2C1=O N1(C(c2c(C)onc2O)=O)CCC(C)(CNC(C2(C)CCCC2C)=O)CC1 C1(C(=O)NC(CC(=O)NC)C2CC2)CC(C)(C)CCN1C(=O)CNC(N)=O N1(C(CCC)=O)CCC(N(C)C(c2ccccc2)C2CC2)CC1 C=CCC(CNC(=O)CCc1cncn1C)C(=O)NCCC=CCC c1(C(N2CCC(CNC(=O)CCCC(F)(F)F)C2)=O)cnc2cc(O)ccc2c1 CC(C)C(C)CC(=O)N(C1CCN(C(c2ncc(C3CC3)cc2F)=O)C1)C C1(C(=O)NC(C)CN2CCCCC2)CCN(C(=O)c2ccc([N+](=O)[O-])o2)O1 CC(CC(F)F)C(=O)N1CCC(O)CC1C(=O)NCc1cccc(O)c1 C1(CNC(COC(CC)C)=O)CC(C)(C)CN1C(C1CCC(C)=C(C)C1)=O c1(C(N2CC(O)(CCc3cn(CC=C)nn3)C2)=O)cc2c(C)c(C)ccc2[nH]1 C=CCC(C(=O)N(CC(=O)NOCCCCF)C(C)C)C(C)C C12(C(c3n(CC(=O)NC4CC(C(=O)NC5CC5)C4)nnn3)=O)CCCCC1OCC2 N1(C(CNC=O)=O)C2CCCC1CC(NC(C1CC3(CCO1)CC3)=O)C2 c1(CC(=O)NC2(C3CCCCN3CCSCC=O)CC2)ccnc2[nH]ncc12 Cc1cc(Cl)c(C(=O)NC(C)C(C(C)C)NC(=O)CC2CCCC2)s1 C(=O)(C(C(=O)NC1CC(NC(=O)CC(F)(F)Cl)C1)C1CC1)OCC C1(CNC(c2cc(Cl)c[nH]2)=O)CN(C(c2cncc(C(F)F)c2)=O)CCO1 S(=O)(=O)(c1ccc(N)cc1)CN1CCCC(N(S(=O)(=O)c2ccc(Br)s2)C)CC1 c1(C(=O)NC(c2cccnc2)C(=O)NC(CC#CC)C)cccn2ccnc12 c1(NC(C2(NC(=O)CC3CCCCC3O)C(C)C2)=O)ccc(CN(C)C)c(F)c1 c1(NCc2n(CC)nc(Br)n2)ccc(Br)c(N2CCCC2)c1 CCCC(C(O)C(=O)NCc1ccc(C)c(F)c1)NC(c1c[nH]c(C)c1)=O N(C(=NCc1ccnn1C)NC1CCN(C(=O)C(C)C)C1)Cc1ccn(CC)n1 N1(C(C=CC2(C)COC2)=O)CCCC(O)(CCNC(C2CCCS2)=O)C1 N1(C(CCN(C)CC)=O)CCC(O)(CNC(C2(C(C)(F)F)CCOCC2)=O)C1 CC1CN(C(=O)CCC=CC(C)C)CC(CCNC(=O)C(F)(F)C2CCCC2)O1 C1(C(N2CC(C)(C)C(CNC(=O)C3CC3)C2)=O)CC2(C1)C(F)(F)C21CCC1 CC(CC(N)=O)C(=O)NC1(C2CN(C(C3(CO)CC(F)(F)C3)=O)C2)CC1 CCCC(=O)N(C)CC1(NC(=O)CC2CC2(C)C)CC1 n1(CC(=O)NC2C(NC(C=C(C)I)=O)CC2)ncc(Br)n1 C(=O)(CCCC(=O)NCCC1CCCN1C)OCC.n12cc(cn1)C(=O)NCC2 C(=O)(C(C)CCC(C)(C)C)NC1C(CCC)CN(C(=O)CC(C)C(C)C)C1 Cc1ccc(C(N2CC(CNC(=O)Cn3nccn3)C(C)C2)=O)c([N+](=O)[O-])c1 CCC(O)C(=O)N1CCCC1CCC(=O)Nc1ccnn1Cc1ccccc1 c1(C(=O)NCCC(COC)(C)C)cccc([N+](=O)[O-])c1S(C)(=O)=O C12(C(N3CC=CC(NC(c4c(OC)n(C)nc4C)=O)C3)=O)CCC(=O)N1CCS2 Cc1nn(C)cc1CC(=O)NC1CC(C(=O)NC2CCC(C(N)=O)C2)C1(C)C N1(C(c2n(C)ncc2Cl)C(=O)NCc2ccco2)CCn2nc(C3CC3)cc2C1 C1(CNC(C2N(C(CSC(C)C)=O)CCC2O)=O)Cc2ccccc2O1 C1(C(=O)NCC(C(C)C)O)CN(C(=O)CC2(O)CCOCC2)C(C)(C)C1 c1(NCCN(C2CC2)CC)nc(=NC(C)C2CC3(CCC3)C2)[nH]c2ncncc12 C1(C(=O)NCCCN(C(CSCC#C)=O)C)Cc2ccccc2O1 N1(C(c2ccc(C#C)o2)=O)C(C(=O)Nc2ccc(C(C)C)cc2)CCC12CC2 N1(C(c2cc(COC)sc2)=O)CCC(COC)(NC(=O)C(C)C(=O)OC)CC1 c1(CN(CCCCNC)C)cccnc1OC(F)(F)F c1(CC)cccc(C(=O)N(CCCNC(C2CSCCS2)=O)CCO)c1O CN1CCN(C(c2cccn(C)c2=O)=O)CC1C(=O)NCCCn1cnnc1 CCCS(=O)(=O)CC(=O)NC1(CNC(=O)C(C)(C)CC(=O)OC)CCOCC1 c1(OC)ccc(C(=O)NCC(n2cc(CCc3nccs3)nn2)C)nn1 C(CN=c1ncc(F)c[nH]1)=Cc1ccc(C(=O)OC)cc1 c1(CNC(=O)Nc2csc(-c3ccccn3)n2)c[nH]c2ccc(Br)cc12 c1(OCC)ccc2cc1C(=O)N1C(=O)NCC1CS2.C1(C)(CN)CCCC1 CC(C)(C)C(C)(C)C(=O)NCC1CCN1C(c1cnc(-c2ccncc2)s1)=O C1(NC(CCCCC=C)=O)CN(C(c2scnc2Cl)=O)CC2(CCOCC2)C1 c1(-c2n(C(C3(C)CC3)C)nc(-c3ccnn3C)n2)ccc2c(c1)C(C)CO2 c1(OCC=C)ccccc1C(C(=O)NOCC=CCl)N(CCNC(C)=O)CC c1(CN2CCN(CC3(C)CC3Br)CC2CCl)ccc2ccncc2c1 C1(C)(NC(C(=O)NC2C(OC)CCC2)=O)CCCN1C(=O)OC(C)(C)C Cc1ccccc1CN(C1CCOC1)CCNC(=O)CC1CCCCC1O N1(C(C(CC)F)=O)CC(NC(=O)COc2cccc(C)c2)C(n2cccn2)C1 C(=O)(C(C)(COC)OC)NC1CC(C(C)NC(C(C2CCCC2)OCC)=O)C1 N1(C(CCC=C)=O)CCC2(CC1)CC(NC(C1(CC(C)C)CC1)=O)CO2 N1(C(CCC=C)C(=O)NCc2cccs2)CCOc2cccc(Cl)c2C1 c1(-c2cc(CC)c(F)cc2)cccc2sc(C(=O)Nc3ccc(I)cc3Cl)cc12 Cc1ccnc(C(=O)NC2C=CCCC2C(=O)NC2(C)CCOC2=O)c1F C1(NC(C2CCCC(C)CC2)=O)CC2CN(C(C3CC3(Cl)Cl)=O)CC2C1 CC1(C)CN(C(c2cc(CO)on2)=O)CC1NC(=O)CN1CC2CC2C1 C(=O)(CCC(O)C(C)(C)C)N(C(CC)C(=O)NC1CCCCC1)C1CC2CC2C1 c1(C(N(CC(C)N(C(C=C(C)C(C)C)=O)C)C)=O)ccc(CO)s1 c1(C(=O)NCC2(F)CCCN(C(C(F)=CC)=O)C2)ccn2ccnc2n1 C1(O)(C(=O)NCC2=CCN(C(C(C)C3CCC3)=O)CC2)CCc2ccccc2C1 C=C1CCCN(c2ccnc(NCCCOCCOC)n2)C1 C(C(C)(C)CC(=O)NCCCC(C)NC(=O)C(C)C1CCOC1)OC C1(C(=O)NCC(C)N=[N+]=[N-])(CC)CCCN(C(=O)CC2CC3(CCC3)C2)C1 N1(C(c2onc(CC)n2)=O)CCC2CCC(NC(C3(O)CCSCC3)=O)C1C2 C(=O)(C1=CS(=O)(=O)CCC1)NCC1CN(C(C2(C)CC3CC3C2)=O)C1 C1(C(=O)NCC2N(C(c3cnc(C)[nH]3)=O)CCCC2)CC(C2CC2)=NO1 N1(C(C(OC)OC)=O)CC(CNC(c2nc(-c3ccccc3)oc2C)=O)C(O)C1 C1(NC(C2C(C(=O)OC)C=C2)=O)CC(C(N2CC(n3ccnn3)C2)=O)C12CCC2 N1(C(C(C)(F)F)=O)CC2CC(C(=O)NC3(CCO)CCC3)CC2C1 C1(C(CNC(C(=O)NCC)=O)(C)O)CCN(C(=O)Cc2occc2C)CC1 c1(C(N(C2CC2)CC)=O)coc(C(C)NC(=O)C(C)N2CC(C)C2)n1 c1(C(N2CC(N(C(CCC=CC)=O)C)C(O)C2)=O)c(F)cc(Cl)cc1F Nc1cccc2ccc(C(=O)NC34CC3CN(C(C3CC3C(F)F)=O)C4)nc12 C1=CCCOC(c2nnc(N3CCOC(c4cc[nH]n4)C3)n2CCC#N)C1 c1(C(N2CC(O)(CNC(C3(F)CC=CC3)=O)C2)=O)cc2c([nH]1)CCCC2 C1(Cc2ncc(CC)s2)CCN(C(=O)C(c2cccc(Cl)c2)N)CC1 C12(NC(COCC(=C)C)=O)CC3CCC(C1C2)N3C(C1CCCC1C1CC1)=O Cn1c(C(N2CCOC(CNC(C3CCCC4(CC4)C3)=O)C2)=O)cc2sccc12 c1(CC)c(C(=O)NCCC(C)(C)C(F)(F)F)[nH]c2ccccc12 C1(NC(C2CC3C=CC2C3)=O)C2CC1N(C(C1CC13CCCC3)=O)C2 C1(O)(C(C(=O)NCCN(CC)CC)F)CN(C(=O)C(C)N2CC(C)C2)C1 c1(CC(=O)NCCOCCNC(C(n2c(C)ccn2)C)=O)ccnc(O)c1Br C#Cc1cnn(C)c1C(=O)NC1CC2(C1)CC2NC(=O)Cn1nnc(=O)[nH]1 c1(C(=O)NCC(CO)NC(c2nccc(CC)c2)=O)cc(Cl)c(Br)cn1 Cc1cnc(O)cc1NC(c1ncccc1NCc1ccc(O)c(F)c1)=O CCCCCC(O)CNC(=O)C(C)(C)C(C)NC(=O)C(C)CCOC C1(NC(C2C=CC(NC(c3c(C)cc(C)s3)=O)C2)=O)CN(C)CC12CC2 C#Cc1cc(NC(=O)NCc2conc2C(C)(C)C)cc(F)c1 C1(CNC(CNC(C2(C(C)C)CC2)=O)=O)CCC(C)CN1C(=O)Cc1ccncc1 N1(C(CC2C(C)CCO2)=O)CC2(CCN(C(C3(C4CCOCC4)CC3)=O)C2)C1 C#Cc1cc(C(=O)NCC(C2CCCN2C(=O)C2=C(C)OCC2)(C)C)ccc1C S(=O)(=O)(c1cn[nH]c1)N1CC(NC(c2cccnc2Cl)=O)(CO)C1 C1(NC(c2cnn(C3CCC(O)CC3)c2)=O)CC(NC(C23CCCC2C3)=O)CC1O CCC(CC(=O)N1CCOC(CC(=O)NOC2CCC(O)C2O)C1)C(C)C c1(C(N2C(CNC(C(C)C3=CCCC3)=O)CC2)=O)ccc2oc(O)nc2c1 c1(C(=O)NC(C)CC2CN(C(C3(O)CCSC3)=O)C2)ncccc1Br N1(C(CCC2CCC(C)O2)=O)CCC(C2(NC(=O)C(C3CCC3)C3CC3)CC2)C1 N1(C(C(C)C(F)F)=O)CC(NC(c2ccc(CF)cc2)=O)C(C2CC2)C1 CC(C)CC(C)(O)c1cn(CC2CCN(C(C3CCNC3=O)=O)CC2)nn1 C12CCCCN(C1)C2.C1(C(=O)O)CCC(n2cc(CN3CCOC3=O)nn2)CC1 C(=O)(CC1=NN(C)C(=O)C1)NC(C)C(C)C(=O)NCCCCCF C1(OC)CCN(C(=O)C(O)CCNC(=O)C(=Cc2ccco2)C)CC1 N1(c2ncnc(C)c2Br)CCC(C2CCN(C(c3ccc(=O)oc3)=O)CC2)CC1 C(C(C(F)(F)F)N1CCN(C(=O)C=CC(C)=O)CC1)NC(C1C(OC)CCC1)=O C1(CC)C(NC(c2nnsc2SCC)=O)CCN1C(=O)COc1ccccc1Cl C1(C(=O)NCCN(C(=O)C(C2CCOC2)NC(=O)OC(C)(C)C)C)CSCN1C N1(C(CC(C)SC)=O)CC(CO)CC2=CCCC12 CCP1(=O)CCN(C(CNc2ccc(OCCCc3ccccc3)cc2)=O)CC1 N1(C(c2cnc(OC)nc2)=O)CCCC2(NC(c3nc(C)oc3C)=O)CC2C1 C1(N(C(CN(C(c2ccccc2)=O)CC)=O)CC)CC(O)CN1C(=O)CC(F)F Cc1csc2c(N3CC(CC(=O)NCc4cccc(F)n4)C3)ncnc12 C1(NC(c2cc3c(s2)CCC3)=O)CC2CN(C(C3CCCC3)=O)CC2C1 c1(OC)ccc(C(=O)NCC2CC23CC3(F)F)c(OC)c1 C1(CC)CN(C(=O)C(c2ccccn2)C)CCN1C(c1ccc(F)cc1Br)=O N1(C(C(CCSC)OC)=O)CCN(C)C(CNC(c2c(F)cccc2Cl)=O)C1 N1(C(Cc2c(OC)cccc2)=O)CCC(C2C(NC(=O)C(C)=C(C)C)CC2)C1 N1(C(c2cccc(C(C)C)n2)=O)CC(NC(=O)C(C2CC2)N(C)C)C2CC2C1 C(=O)(CC(F)(F)C(F)(F)F)N(CCCNC(=O)CC1CCCC(F)(F)C1)C1CC1 c1(C(=O)NC(C)CNC(C2CCC(C(C)(C)O)CC2)=O)cc2cc(Cl)ccc2[nH]1 C(=O)(C1=NOC2(CCC2)C1)N1C(C)C(NC(c2ccc(CN(C)C)[nH]2)=O)CC1 C1(CNC(C(=O)NC2(C(=O)OC)CCCC2C)=O)CC2CCC1CC2 c1(C(N2CCC(NC(c3c(CC)occ3)=O)C2)=O)cccn2cnnc12 N1(C(CCc2ncc(C)[nH]2)=O)CCC(CO)(NC(c2cnn(C)c2Br)=O)C1 C1(OC)(CNC(=O)CCCC2CCCC2)CCN(C(=O)CSc2nncs2)C1 N1(C(=O)NCc2cc(OCC)ncc2)CCC(O)(C(=O)OC)CC1 C1(NC(C2C(=C)CC2)=O)CC(NC(C2(C(F)(F)F)CCO2)=O)C(O)C1 c1(C(N(CCNC(C2C3COCC23)=O)CC)=O)cccc(OC)c1F C1(NC(C2CCN(C)C2=O)=O)CCN(C(C2(F)CCC2)=O)CC1(C)C C1(C(CN(C)C)OC)CCCN(C(c2cn(C)nc2C2CC2)=O)C1 C1(CC=C)(NC(C2CCC(=O)N2C)=O)CCCN(C(c2nc(O)sc2C)=O)C1 c1(C(=O)NC2CCCN(C(c3ccc(C)s3)=O)C2)ccc2nc(O)oc2c1 c1(CC)cc(NC(=O)C(O)C2CN(C(=O)CN3CCCC3=O)C2)ncn1 C1(CC)CN(C(=O)C#CCNC(C23CCCCC2C3)=O)CCCO1 N1(C(C(C)COc2ccccc2)=O)CCCC(c2ccccc2)CC1 N1(C(CC(C)SC)=O)CC(CN(C)C(c2cc(Br)no2)=O)C2(CC2)C1 Cc1nn(C)c(C)c1C(=O)NC1CCCN(Cc2noc(C(C)(C)C)n2)C1 Cc1sc(S(=O)(=O)Nc2c(F)cc(F)c(F)c2F)cc1[N+](=O)[O-] C1(C(=O)NCC(COC)(C)C)C2CN(Cc3cccc(OC(C)(C)C)c3)CC12 C1(NC(c2n(C)nnn2)c2csc(C(F)(F)F)c2)CC2(C(=O)O)COC1C2 C1(CCn2cc(C(C3CC3)OC)nn2)CCCN(C(c2ccnn2C)C)C1 C12CCCN(C1)C(CO)COC2.Cc1noc(OC(C)=O)n1.C(C)(C)O CCC1=C(C(=O)NCCC2CC(C(=O)NCC3CC34CCC4)C2)SCCO1 Cc1nc(CC(N2CC(NC(c3nn[nH]c3Cl)=O)C(C)C2)=O)c(Cl)s1 N1(CC(=O)N(C(=O)CCCN2CCCCC2)CC)CC=CC(O)C1 CCCCC(C)CCC(=O)N1C2CC1CN(Cc1ccc(Br)c(Cl)c1)C2 C=CCC(CC(F)F)C(=O)N1CC2CCCC(C1)N2C(C12CC(C)(CCO1)C2)=O Cc1cc(=NC(CNC(c2cccc(C3CC3(F)F)c2)=O)C(C)C)[nH]c(Cl)n1 C12(CNC(C=CCC)=O)CCCC1CN(C(=O)CC1CC3CC(=O)C1C3)C2 N1(C(CCOC(C)=O)=O)CCC(O)(CNC(c2cc(C3CCCO3)n(C)n2)=O)C1 c1(C(N2C(C(=O)OC)CCC2)=O)ccc(-c2ccc(C#N)s2)nc1C CCCCCC(CCCCC)CC(=O)NC(C)(CNC(=O)C1=C(Cl)CC1)C(C)C C=CCCCCCCC(=O)NC(C)CC(=O)N(C1COC(C)(C)C1)C n1(CCC(=O)NCC2CN(C(CCC=C(C)C)=O)C3C2C3)ncc2ccccc12 N1(C(C)C)CC2C(C(=O)N3C(C4CC4)CN3C3CC3)C2C1.C1CC1.N(C)C C1(OC)(CNC(=O)CCC2(NC(=O)CSC(F)(F)F)CCC2)CCOC1 C(=O)(C(O)C(O)C(=O)NC(c1ccccc1CCC(F)(F)F)=O)OC(C)(C)C N1(C(C2CC(C)C2)=O)CC(C)C(C)(C(N2C3C=CCC2CC3)=O)C1 C=CCCCCCCN=C(NC(C)C)N1CCN(c2cc(C3CC3)[nH]n2)CC1 C1(OCCCN2CCC(Oc3ccccc3)C2=O)CCCC(F)(F)C1 c1(C(=O)OCC)cc(C)c(CNC(=O)C(=O)NCCC2(N)CCOC2)o1 C=CCCCC(C(=O)NCCOCC)N1CCCC(C(C)(C)C)CC1 C1(CC=C)(C(=O)NCCC2(C)CCOC2)CCCN1C(C1COCCO1)=O C(=O)(C1Cc2c(Cl)cccc21)NC1CC(CNC(C(CO)SC)=O)C1 Cn1nccc1C(C)(C)C(=O)NC1CC1NC(C1(c2ccccc2)CC1(Cl)Cl)=O C1(F)(CNC(C(C)OCCC=C)=O)CCCN(C(=O)Cc2ccc(Cl)nc2)C1 c1(C(=O)NC(C)C(C)NC(C2CCC(CO)CC2)=O)cc(O)cc(F)c1F C1(C(N(CCN(C(=O)C(=O)NC2CC2)C(C)C)C)=O)CCC12CCCO2 c1(CC(=O)N2c3c(C)c(n[nH]3)C(=O)N3CCC(C3)C2)cccc2nonc12.CNC Nc1ccc(S(N)(=O)=O)cc1NC(c1ccc(-c2cnco2)cc1)=O c1(C(N2CC(C)N(C(=O)CCCn3ccnc3)CC2)=O)ccc2ncccc2c1 C1(C)(CNC(COCCOCC#C)=O)CCN(C(=O)CN2CC3CC3C2)C1 C1(C(N(CCCNC(=O)Cc2ccccc2)C)=O)CC2CCC(C1)C2F Cc1c(CC(=O)N(CCNC(=O)C(c2cnccn2)C)C)cnn1C Nc1c(Cl)c(C(N2CC(C(=O)O)OCC23COC3)=O)cc(F)c1Br C1(C(N2CCC(C)C2Cc2ccccc2)=O)CN(S(=O)(=O)N(C)C)C1 c1(C2C(C(=O)NC3CC(F)(CNCC4CC(C)OCC4)C3)C2)cccc(Cl)c1Cl CC1(C)CCC(C(=O)NCC2CC(CF)C2)(NC(C2CC23CCOC3)=O)C1 c1(CN2C(C)C(C(F)(F)F)CC2)cc2c(s1)CCCCC2 C1(NC(Cc2cnc(C)o2)=O)COC2(CCN(C(c3ccc(O)c(F)c3)=O)C2)C1 N1(C(CC2CN(C)C2)=O)CC2CCC(C1)C(NC(C1(CO)CCC1)=O)C2 N1(C(=O)OC(C)(C)C)CCCCCC(C(=O)NCc2cn[nH]c2)C1 c1(OCC#C)ccc(NC(=O)CNC(=O)C(=O)N(CCC(C)O)C)cc1 C1(c2nnnn2C(C)(C)C)(NC2(C)CC(CO)C2)CCN(C(C)(C)C)CC1 C(=O)(CC(C)(C)CNC(=O)C(C)N=[N+]=[N-])NC(C(C)O)(C)C c1(C(N2CCC(N(C)C(C3(C#N)CCCOC3)=O)CC2)=O)csc2ccccc12 c1(N2CCC(NC(=O)C(O)CC3CCCCC3)C2)ncc2c(n1)CCCC2 C(=O)(CC1=CCN(C)CC1)NCCCCC(C)NC(c1cc(C2CCC2)[nH]n1)=O Cc1ccccc1NC(C1CCOC1CNC(=O)C(C)C#N)=O O=C(CC(C(F)F)c1ccc(F)cc1Cl)NC1CN(C(=O)CSC2CC2)C1 Cc1cc(C(N2CC(NC(=O)CC3CC(=O)C3)CC2C)=O)sc1C C1(NC(c2cn[nH]c2)=O)CC1C1CCCN(C(C2CC3CCC(C2)S3)=O)C1 C(=O)(C1SCCc2ccccc21)N1CC(C)C(CNC(C2(O)CCC2)=O)C1 Cc1cc(CN2CCCCC2CNN2CCNC2=O)nn1C Cc1[nH]nc2ccc(C(=O)NCCC3(C)CCN(C(C4CC4(C)C)=O)CC3)cc12 c1(C(=O)NC2CCC(CNC(C(N)=O)=O)C2)ccc(Cl)c(F)c1 O=C(C1=CCCSC1)NC1COCCN(C(C2CC(c3ccc(O)cc3)C2)=O)C1 C1(COC(CC)=O)CCC(C)(C)OC1.C12CN(C1)C(=O)C(C)NC2=O N1(Cc2cn(CC)nc2-c2ccc(C(=O)OC)s2)CCn2ccnc2C1 Cc1cccc(C(F)(F)C(=O)NCC(N2CCN(C(=O)C=CCN(C)C)CC2)C)c1 Cc1c(C(=O)OCC2(Cc3ccccc3Br)CC2)cc(C(F)(F)F)cc1O N1(C(CC=CC)=O)CCN(C(c2ccc(-n3ccnc3O)cc2)=O)CC(O)C1 C(CCC1CCC1)(C(=O)NC1CC1c1ccccc1)NC(c1scc(C)c1)=O N1(C(=O)CC(F)F)CCN(C(C23CC(F)C2C3)=O)CC1c1cccc(F)c1 Cc1ncc(C(N2CCC(CCNC(=O)CCCc3cc[nH]n3)C2)=O)[nH]1 c1(C(=O)NC)ccc(S(=O)(=O)NC2CC2NCc2cccs2)cc1 N1(C(C=C(CCC)CCC)=O)C2CCC1C(C(=O)NC(CO)CCSC)C2 C=CC(CC)CC(=O)NCCC1(C)CCN(C(=O)Cc2nc([N+](=O)[O-])n[nH]2)CC1 C1(C)(CNC(C(C)(C)C2CC2)=O)CCC(NC(=O)Cc2csnn2)C1 Cc1cc(C(=O)NCC2CN(C(c3ccc(Cl)cc3N)=O)CC2C)nc(C)n1 C1(C(N(C(C)C(=O)N(CCSC)CC2CC2)CC)=O)C(C#N)C1(C)C C12(CC(=O)NC3CC(N(C(C(CC)C)=O)C)C3)CCC(CC1)C2 C1(C)(CNC(CC(COC)C)=O)CCN(C(c2cc(=O)c(OC)co2)=O)CC1 C1(C(N(C2(CCN=[N+]=[N-])CC2)CC)=O)CCN(C(=O)C(=O)C(C)C)CC1F c1(C(N2CC(NCc3cccc(-n4ccnn4)c3)C2)=O)cc(O)ncn1 CON(C)CCN=c1nc(NCCOCCC2CC2)c2c([nH]1)CCOC2 C=CC1(C(=O)NC(C)CC2CN(C(=O)C(F)(F)c3cnccn3)C2)CCCCC1 C(=O)(C(F)(F)C(F)(F)C(F)F)NC1C(C)CN(C(c2cn(C)nn2)=O)CC1 C(C(C)(C)C(=O)NC1CCCC(CNC(C2(C(=O)OC)CC2)=O)C1)N(C)C n1(CC)nccc1C=CC(N1CCOCC1CNC(=O)Cc1ccc(F)cc1)=O C12(NC(CCc3ccc(CC)cc3)=O)CCCCC1CN(C(=O)CC(C)O)C2 C(=O)(CC(CN(C1CCCCCCC1)C)C(C)C)OC C(CS(=O)(=O)CC(=O)NCC12CCC(CN(C(c3cc(C)no3)=O)C1)C2)OC Cn1ccc2ccc(C(N3CCCC(NC(=O)C=Cc4ccco4)CC3)=O)cc12 c1(CN2CCC(N)(CO)CC2)cc(F)cc2c1OCOC2 C(=O)(C1=CCCC1)NCCC(C)NC(c1cc(-c2ccco2)[nH]c1C1CC1)=O c1(NC(N2CCC(C(=O)CNC(=O)OC)(CO)C2)=O)ccnc(CO)c1C Cc1ccc(Cl)c(C(=O)N(C(C)CCNC(=O)C=Cc2cncs2)C)c1N C=C1CCN(C(=O)CCN=[N+]=[N-])C(C(=O)NCCOCCCC)C1 c1(OC)ccncc1CC(=O)NC1CCC(NC(=O)C(N2CCOCC2=O)C)C1 C1(CCC)(C(=O)NCC2CCCC(CNC(=O)C3=CCCC3)C2)CCNC1=O C(C)(CNC(c1cocc1C)=O)(CC(C)C)NC(c1cn(CC=C)nn1)=O C1(N(C(CN(C)C)=O)CC(=O)Nc2nnnn2C2CC2)CC(C#N)C1 C1(O)(CNC(CNC(C(CC)CC)=O)=O)CCCN(C(=O)Cc2cnccn2)C1 C1(C(=O)NCC(C2CCN(C(CCSCC(C)C)=O)CC2)O)OCCCC1(C)C O=C(C1CCCc2nc[nH]c21)NCC1(NC(C2Cc3ccc(F)cc3O2)=O)CC1 CCC(C)(COC)C(=O)NCC#CC(=O)NC1(c2ccsc2)CC1 Cc1cc(C(N2CCC(C(=O)NC(C3(CO)CC3)C)C2C)=O)ccn1 N1(C(C(C=C=C)C)=O)CCC2OCCN(C(c3ccn4cccc4c3)=O)C2C1 C(C(CC(C)C)NC(c1cnc(C(C)C)s1)=O)n1cc(C(CC)O)nn1 N1(C(C(CCC(C)C)O)=O)CCOC2CCN(C(c3c[nH]c(=N)s3)=O)CC12 CCCCCCC(=O)NC1CCCCN(C(=O)CC(CC)C2CCCCC2)C1 c1(CN2CCCC(CNS(CCCC)(=O)=O)C2)cccc(Br)c1Br N1(C(c2cc(C)cc(Cl)c2)=O)CCCC2(CC(NC(C3(C)CC3)=O)CO2)C1 c1(C(C)C)nc(=NCCC(C)NC(C2OCC2(C)C)=O)s[nH]1 Cc1cc(CNC(c2occc2CNC(c2cn(C(C)C)cn2)=O)=O)ncn1 c1(CNC(CCN2C(C)CCC2)=O)ccc(CNC(c2cc(Cl)cnn2)=O)cc1 C1(CCC)(NC(C=C(CCC)C)=O)CCN(C(=O)C(C)(C(C)C)NC(C)=O)CC1 C1(C(=O)NC2(C)CN(C(=O)CCCn3ccnc3)C2)CC2(C)CCC1(C)O2 C1(O)(C(N2CC(C(C)NC(c3cnn(CC(F)F)c3)=O)C2)=O)CCCCCC1 C(=O)(C1=CC2(CCOC2)C1)NC1(C(=O)NC(C=C)C2CC2)CC(O)C1 O=S(=O)(c1cncc(Br)c1)N1CC2CCN(Cc3ccc(I)c(F)c3F)CC2C1 C(=O)(CCCCc1cnn[nH]1)NCC(N(C)C(c1cc(Br)cs1)=O)C1CC1 C(=O)(C1=CC2CCC1C2)N1CC(CNC(=O)CSCc2ccccn2)OCCC1 C1(NC(CC(CC)C2CC2)=O)C2CC3C1C3C2C(=O)NCCCc1nc[nH]n1 N1(C(CCC#C)=O)CC(CC)C(NC(C2CCCN(C(C)=O)C2)=O)C1 N1(CCC(=O)NC2CC2NC(=O)CC23CCCC2C3)CCCC1=O CC(O)CCN=c1nc(N2CCC(c3ccncn3)CC2)[nH]c(=NC2CSC2)[nH]1 N1(C(CCNC(=O)NC)=O)CCC(NC(=O)CCc2nccn2C)C1(C)C C12(CC(=O)N(C)CC3CCC(CNC(C(F)OC)=O)CC3)CCC(CC1)CC2 Cc1ccc(O)c(C(N2CC3C(C(N4CC[Si](C)(C)CC4)=O)C3C2)=O)c1 c1(C(=O)OC)cc(C(=O)NCC(C)C(=O)N(C(C)CC(N)=O)C)no1 CCC(C)CN=C(NCCSC)NC1CC(=O)N2CCCCC12 c1(OCCC(N2CC3C(CNC(c4nsnc4O)=O)C3C2)=O)c(F)cccc1F c1(C(=O)NCC(N(C(Cc2c(OC)ccnc2)=O)C)C2CC2)cccc(Cl)c1C N1(C(C2(CC=C)CC2)=O)CC(N(C(=O)CCc2ccc(Cl)nc2)C)C2(CC2)C1 N=c1ccc(C(N2CCCCC(CNC(=O)CC3C=CCC3)C2)=O)c(Cl)[nH]1 S(=O)(=O)(c1c[nH]ccc1=NCCOC)N(CCOCCOC)C N1(C(C2CN(S(CC)(=O)=O)C2)=O)CCOC(C)(CNC(=O)C(C2CCC2)OC)C1 C1(C(=O)NCC2CN(C(CCC(C)(C)OC)=O)CC2C)CN2CCN1CC2C CC(C)CCC(=O)NCC1CC(C)N(C(=O)CCCOc2cccc(F)c2)C1 N1(CCC(=O)NC2CC3C(NC(=O)C=CCN4CCCC4)C3C2)C(=O)CNC1=O c1(OCC(N2C(C(=O)NC3(C)CC=CC3)CCC2)=O)nc(O)nc(O)n1 c1(C(=O)NCCC2CCCN(C(c3nnn(C)c3N)=O)C2)ccsc1S(N)(=O)=O C1(CNC(C(CC)(C)O)=O)CN(C)CCN1C(=O)Cc1cccc(CSC)c1 CCC(C)(C#N)C(=O)N1CC2CC2(NC(c2cscc2C(F)(F)F)=O)C1 c1(C(N(CC(C)NC(=O)Cc2ccsc2C)CC)=O)c(C)nc(C)n1O Cc1cc(CNC(=O)CN=[N+]=[N-])ccc1N1CCN(C(=O)CC2CC2)CC1 N1(C(C(C(=C)C)(C)C)=O)CC(C2CCN(C(=O)C(F)(F)c3ncccn3)CC2)C1 CC(CC(=O)NCC(C)(C)Cn1cc(-c2nc(C(=O)O)cs2)nn1)n1ccnc1 c1(OC)cc(CN2CCC(CN(C(=O)CC(O)Cn3cccn3)C)C2)cc(F)c1 N1(C(CCN(C(=O)Cc2cccs2)CCO)=O)CC2COCC2C1 N1(C(C(CCC)C)=O)CCC(F)(F)C(CNC(c2c(C)ncnc2C)=O)C1 C1(NC(CCSCCCC)=O)CC2CC(NC(=O)CCn3ccnn3)C1C2 C1(CN(C)C(C2CC=CCC2)=O)CC(=O)CC12CCC2 N1(C(Cc2c(C)ocn2)=O)CCC(C)(NC(=O)C=CC2CC2)C1 c12cnc(nc1)NC(=O)Cn1cc-2nn1.c1(OC2CC(CC(=O)O)C2)ccccn1 c1(C(=O)NCC2(CNC(C(C3CC3)OC)=O)CC23CCC3)cc(F)c(C)cc1F n1(CC(=O)N(C2CC(NC(=O)OC(C)(C)C)C2)C2CC2)cc(Br)c(O)nc1=O C(CCCCCC(=O)NC1CCCC1NC(=O)C(c1ccccc1)F)SC O=C(C#CC1CCC1)N1CC(NC(C2(Br)CC2)=O)CC(O)C1 C1(CNC(=O)CC2CCCSC2)C(O)C(O)CN1C(=O)CC1CCOCC1 C1(C2CC2)(C(N(CCCC)C)=O)CN(C(=O)CP(C)(C)=O)C1 Cc1cc(C(=O)N(CC(=O)NCC(c2cccs2)O)C2CC2)cc(C)c1 Cc1cc(CC(N2CCCC(CN(C)C(c3cn(C4CC4)nn3)=O)C2)=O)c(C)s1 Cc1cc(C(=O)NC2CN(C(=O)CC(F)(F)F)CC2CO)c(C)n1C1CCCC1 C(=O)(C(C)(C)CS(N)(=O)=O)NC1CC(C)(C)N(C(=O)CN2CCC(=O)NC2=O)C1 c1(NS(=O)(=O)C2CC2)nc2c(C(=O)NCC3(OC(C)(C)C)CCC3)cccc2s1 C1(C(=O)NCC(C2CCCC2)NC(C2CCCCS2)=O)(CC)CCC(O)CC1 C1(C)(C(N2CCN(C(C#C)C)CC2)=O)CN(C(=O)Cc2ccn(C)c2)CC1C Cn1cccc1C(=O)NC(C(=O)NC1CCCC1CCO)C1(C)CC1 C(=O)(N=c1nc(C(F)F)[nH]s1)C1(C)CCSCC1 C1(NC(C(C)OCCC=C)=O)CN(C(=O)Cc2ccc(Br)cc2)CC1O Cc1ccc(F)c(C(N2CC(NC(C3(C(N)=O)CC3)=O)C(CC3CC3)C2)=O)c1 C1(CC)CN(C(c2ccoc2Br)=O)CC1NC(=O)COC1CCOC1 C1(C)(NC(CN(c2ccccc2)CC)=O)CCCN(C(C2CC2C(F)(F)F)=O)C1 C12(C(=O)NC(C3CCCC3)CNC(C(C3CC3)OCC)=O)CCC(F)(CC1)C2.CC N1(C(C(C)(C)n2cc(Cl)cn2)=O)CC2CCC1CN2C(=O)COC(F)F.C1C(=O)O1 c1(NC(=O)NCCCN(C)CCOC2CCC(OC3CCC3)C2)cccc(F)c1 CC1(C)CN(C(=O)C2=CCC(NC(c3nc(=N)cc[nH]3)=O)C2)C2CCCC12 C1(N(C(CCC(=O)NC)=O)C)CCCCN(C(C2(NC(=O)OC)CC2)=O)C1 N1(C(=O)CCCN2CCCCC2)CCSCC1C1CC1.C12(F)CN(C1)C2 N1(C(c2cc(OC)ns2)=O)CCCC(N(C(=O)CCCF)C)CC1 c1(OC(CCNC2CCCC(C)C2)=O)ccc(N=[N+]=[N-])c([N+](=O)[O-])c1 C(CO)(CCS(C)(=O)=O)NC(=NCC)NCc1ccc(OC(C)C)c(C)c1 N1(C(C2C(C)(C)CO2)=O)Cc2n[nH]cc2C1C(=O)Nc1cccc(CCF)c1 c1(C(=O)NC(CNC(Cc2cc(C)n(C)n2)=O)C(C)C)cc2ccc(Cl)cc2[nH]1 C1(NC(C2CCS(=O)(=O)C2)=O)CCCC(NC(C2(C(F)(F)F)CCC2)=O)C1 N1(C(c2c(C)cns2)=O)CCC(NC(c2cc(C(C)(F)F)n[nH]2)=O)CC1C C1(C(=O)NCC2(O)CN(C(c3csc(C(F)(F)F)c3)=O)C2)CC2CC1CC2(F)F c1(OC)cccc(CNC(=O)CCCNC(=O)C=Cc2ocnc2C)c1 c1(C(=O)NCC(C)N(C(C(C(C)C)n2ncc(C)c2)=O)C)cc2cc(Cl)sc2[nH]1 c1(OC)cc(NC(=O)C(CCC2CC2)NCCO)c(SC)cc1Cl N1(C(C#CC(C)C)=O)CCCC(C2CCN(C(C3CC4C=CC3CC4)=O)CC2)C1 Nc1c(C(N2CC3(CCNC(=O)COC(F)F)CCC2C3)=O)cc(F)cc1Cl c1(C(=O)NCC2(C)OCCN(C(C3=C(C)CCC3)=O)C2)cc(C)c(C)c(Cl)c1 N1(C(C2CSCCS2)=O)CCC2(CCCN2C(c2nn[nH]c2Cl)=O)CC1 CCCCC(C)CCC(=O)NCCOCCNC(c1ccc(=O)n(CCO)c1)=O C(=O)(Nn1cnn(C)c1=S)C12N(C(CN3C(C)CCC3)=O)CCC1CCC2 N1(C(c2c(C)[nH]nc2CO)=O)CC(C(=O)NCC2CN(C)C2)C2(CC2)C1 N1(C(CC2N(C(c3c(C)ccnc3)=O)CC2)=O)CC2(CCC2(C)C)C1 c1(CN2C(C(N(C)C)=O)CC(F)C2)cc(Cl)c(Br)cc1F c1(C(C)C)ccc(C(N2CCC23CC(O)C3)C(=O)Nc2ccc(F)cc2)cc1 c1(C(C)C(=O)NCC2(CNC(C3CC3C)=O)CC2)ccccn1 N1(C(c2cccc(C)n2)=O)CCN(C(c2c[nH]c(=N)s2)=O)CC(CO)C1 N1(C(CC2CCN(C)C2)=O)CCCCC1CCNC(c1nnn(C)n1)=O c1(C(N2CC(NC(C3(CC#C)CC3)=O)C(F)C2)=O)cc(C)ccc1Cl C1(CNC(C(CC#C)NC(c2cncc(OC)c2)=O)=O)CCCCC1(C)C C1(C2CCN(C(C3(CO)CC3)=O)CC2)(NC(C2N(C(C)C)C(=O)COC2)=O)CC1 C=CCC(CC(C)C)C(=O)N1CCN(C(=O)CCC(C)(C)C)C(CC)C1 c1(OC(C)C)ccc(C(=O)NCC(C)N(C)C(c2scnc2Cl)=O)cn1 Cc1ccc(F)c(CC(N2CC(NC(=O)Cc3ccc(Cl)s3)CC(O)C2)=O)c1 CC(C(=O)NCCC1CC1C)NC(=O)COCCCF c1(C(N2C(C(C)NC(C(CCC)OCC)=O)CCC2)=O)cnn2cc(C)cnc12 C1(NC(c2c(C)nc(CC(C)C)s2)=O)CN(C(C2(N(C)C)CC2)=O)CCC1C Cc1ccc(CCNC(=O)C(Cc2cn[nH]c2)NC(C2CC(F)CN2C)=O)cc1 CC1CC(Cc2cccnc2Cl)CCN1C(=O)NCc1ncnn1CCCl CN1CCN(C)C(C(=O)N(C2CC(NC(C3CN4CCC3C4)=O)C2)C)C1 c1(Cc2cn(C3CCC(=O)C3)nn2)ccncc1F.C1CCC(=O)N1 N(C(=NC1CCC1)N1CCC(CC2CCCCC2)CC1)C1CCS(=O)(=O)N1 Cc1nc(CC(=O)NC2CCC2C(=O)NC2CC2c2cncs2)n[nH]1 C(=O)(C#CC1CCOC1)N1CCCC(CNC(COCc2c(C)ncs2)=O)CC1 C#Cc1ccc(C(=O)N(C)CCN(C(=O)CC2NC(=O)NC2=O)C)c(OC)c1 C(=O)(C#CC(C)(C)C)NC1C(NC(CCOc2ccc(OC)cc2)=O)CC1 N1(C(C2C=CCN(C(=O)CCCF)C2)=O)CCCC12CCOC2=O N1(C(=O)NC2CC2c2cc(C)cc(OC)c2C)CCC2(CCCO2)CC1 N1(C(CNC(C2OCC(N)C2)=O)=O)CCCCCC1CCC C1(N=c2nc(C3CC3)[nH]s2)(CNC(c2cnn3ncccc23)=O)CCCCCC1 N1(C(c2cc(C)n(C(F)F)n2)=O)CCC(NC(=O)C=Cc2ccc(Br)s2)C(F)C1 CC(CCCNC(C1COC2CC12)=O)NC(c1ccc(CNS(C)(=O)=O)o1)=O c1(CC(N2CC3(CCN(C(CCC=CC)=O)C3)C2)=O)cn(C)c2ccccc12 C1(CNC2CC(CNC(C3(OC)CCC3)=O)C2)CCC(C)=CC1C C1(OC)CCN(C(C2OCCC2NC(=O)COC2(C)CCCC2)=O)C1C Cn1ncc(C(=O)NCC2(NC(=O)C=CC(c3ccccc3)=O)CCOC2)c1N c1(OC)cc(OC)c(C(=O)NCCNC(C2CN(c3nncs3)C2)=O)c(F)c1 N1(C(C2(F)CCC2)=O)CC2(CCCC(CNC(C34COC(CO)(C3)C4)=O)O2)C1 c1(C(N)=O)cc(C(=O)NC23CC(CNC(C4COCCO4)=O)(C2)C3)on1 c1(C(N2CCC(c3cnn[nH]3)C2)C(=O)NCC)ccc(O)nc1 C#CCC(CC#C)C(=O)N1CC2CC2(CNC(c2cn(C)nc2C2CCC2)=O)C1 N1(C(C2C(c3ccn(C)n3)C2)=O)CCC(CNC(=O)CNS(N)(=O)=O)C1(C)C C(=O)(C(O)C(F)(F)F)N1C(C(N(C2C(C)COCC2)C)=O)CCCC1 C1(C(=O)NC(C(C)O)C(=O)N(C2CCC3CC23)C)CC(=O)CC12CCC2 C1(CNC(C(C)N(C(CCN(C)CC)=O)C)=O)C(C)(C)C1(F)F c1(C(=O)NCC2CCCN2C(=O)CSN2CCCC2)ccc(C2CC2)nc1 C(CCC(=O)NCC(CCc1ccccc1)NC(N)=O)C1C(C)C1 C(CC1CC1)(CC(=O)NC(C)CF)NC(c1cc(CCC)[nH]n1)=O c1(C=O)cc2cc(F)ccc2o1.C1(CC(C)N)CN(C(=O)CCN(C)C)CCO1 CCC(C)(COC)C(=O)N(CCNC(=O)CCSc1ccccc1F)CC N1(C(C2N(C(C(CC)OC(N)=O)=O)CSC2)=O)CC(OC)C(C(F)F)C1 C(=O)(C(F)CC(CC)CC)NCC(CC(=O)NCCOCC#C)C n1(CCOC)c(N(C(C(=O)OC)c2ccsc2)C)nc2ccccc2c1=O CCC(C)(CCNC(=O)Cc1scnc1C)NC(=O)CS(=O)(=O)N(C)C C1(C)(C(=O)NCC(COC)(O)CO)CCN(C(=O)CC(C)C2CCCCC2)CC1 CCC(C)C(C(=O)NCCN(C)C(C1(c2ccccc2)CC(F)C1)=O)NC(C)=O CCC(CC)CCC(=O)N1CCCCCC(CNC(=O)CC2CCCCC2O)C1 C(N=c1ccnc(C(C)C)[nH]1)C1CCCN(C(C(CC)(C)C)=O)C1 Cc1cc(C(N2CCCC2CC(=O)Nc2ncc(C#N)cc2I)=O)cc(C)c1F c1(C(N(CCCNC(C2(C(=O)OC)CC2C)=O)C(C)C)=O)cc2nc(C)sc2[nH]1 C1(C(=O)NCC(=O)OC)CCN(C(=O)C(C)(C)C23CCCC2C3)O1 N1(C(C(C)CO)=O)CC2(CC(NC(=O)COCc3ccnc(O)c3)CO2)C1 C(=O)(CCS(=O)(=O)N(C)C)NCC1N(C(c2c(C)[nH]cc2)=O)CC(O)C1 C=CC(CCC)CC(=O)N1CCC(=C)CC1C(=O)N(C)CC1OCCC1(C)C N1(C(C2CC(OC)C2)=O)CC2CCCC(N(C(=O)CCC3CCC(C)O3)C)C2C1 Nc1ncc(C(=O)NCC(O)CNC(=O)C=Cc2ccsc2)cc1O N1(C(Cc2cncc(C)c2)=O)CCCCC(N(C(=O)CN2CCC(C)(O)C2)C)C1 n1(CC)c(CNCC2CC(F)CN2C)cnc1C C1(C2CCCOC2)(NC(C2C3CCN(C(c4cc(C)c(O)nn4)=O)CC32)=O)CC1 c1(OCC)ccc(F)c(C(=O)N(C(C)CNC(c2cc(OC)ccc2N)=O)C)c1 N1(C(CCCC(C)O)=O)CC2CCN(C(C3CCCSC3)=O)C2C1C C(CCCCC(=O)NC(C)CCCC(=O)NC1CCSC1)OC N1(C(C2C(CC(C)(C)C)C2)=O)CC2(CC2)CC1C(N1CC(O)(c2cc[nH]n2)C1)=O N1(C(c2ccc(OC)cn2)=O)CCN(C(=O)Cc2cccc(O)c2)CC1C(C)C N1(C(c2[nH]c(=NCC)sc2)=O)CC(C)CN(C(C2CCC(F)(F)CC2)=O)CC1C C(C)(N=c1[nH]n2cc(C)nc2s1)c1ccc(C(C)=O)s1.c12cccn(c1=O)CC2 C1(CSC)CCN(S(=O)(=O)Oc2cc(Br)cc(C#N)c2)CC1 n1(CC)cc(NC(=O)CCC2CCN(C(=O)CCc3cc(C)no3)C2)ccc1=O C1(OC)CN2CCCC2(C(=O)NCC2(CCNC(C3(C)CCC3)=O)CC2)C1 C1(NC(C)=O)CN(C(=NCCC(N)=O)NC2CCCC2)C1.C12CCC(OC)(C1)N2 C#CCC(=O)N(C(CC(=O)NCC1CC(n2cncn2)C1)C1CC1)C CN1CCN(C(=O)CC2CCCN2C(=O)COc2ccccn2)C(C(F)(F)F)C1 C(=O)(C1=CCCCC1C)NC(C1CC=CCC1)C(=O)Nc1ccc(OC)cc1 c1(C(=O)NCc2ncoc2CCNC(C2CSC2)=O)ccc(F)cc1 c1(C(N2CC(C3(NC(c4ccnc(O)c4)=O)CC3)C2)=O)cc2ccc(Cl)cc2s1 S(=O)(=O)(c1ccc(NC(N)=O)cc1)NC1(C=C)CCCCC1 c1(C(=O)NCC(CCNC(c2coc3c2COC3)=O)OC)cnc(O)c(F)c1 c1(CNC(C2C(C)(CC)C2)=O)cc(C)c(-c2nn[nH]n2)o1.c12ccc(cc1)OC2 c1(CC)nc(O)c(C(=O)NCCN(C)C(c2cnccc2C)=O)cc1C CC(CN=c1[nH]c(NC2CC2F)nc2ccsc12)c1ccsc1 C1(C)(CNC(c2c(CC)noc2C)c2n(CC=C)nnn2)CCCCC1 N1(C(C2(C)CNC(=O)C2)=O)CCOCC(NC(C2CCS(=O)CC2)=O)C1 CC1(NC(C2CCCCO2)=O)CCN(C(=O)C=Cc2ccc(Cl)s2)C1 Cc1cnn(CC(=O)NCC(C2CCC2N)=O)c1.C1(C(=O)NC)(C(=O)N(C)C)CCC1 N1(C(CC=CC=C)=O)CCOCC1CCNC(c1ccc(-c2ccncc2)o1)=O C1(C(N2CCCC(C)C2)=O)CC2(C1)CN(Cc1ccc(Br)cc1I)C2 N1(C(c2c(C)c[nH]c2)=O)C2CCC1CC(CNC(C1OCCOC13CCC3)=O)C2 C1(CNC(C=C(C)c2cccs2)=O)N(C(=O)CC2CCN(C)C2)CCC1(C)C C(C(CC(C)C)C(=O)N1CCCC1C(C)(C)C)NC(c1c(C)scc1)=O C(CNC(=O)CC(F)(F)Cl)(CCCC)NC(CCN(CC=C)C(=O)OC(C)(C)C)=O CC(C(=O)N1CC(c2ocnc2CNC(=O)CCCC=CBr)C1)S(N)(=O)=O c1(C(=O)NCC(CCC#N)O)cccc(Br)c1Br c1(C(=O)NC(C)CCCNC(=O)CC2CCCN2C)cc2c(cc1Cl)OCCO2 N1(C(c2c(CC)nn(C)c2)=O)CCC(NC(=O)C=CBr)CC(C)(C)C1 C1(C(N2CC(NC(=O)C#CC3(C)CC3)CC(C)C2)=O)CC(C2CCOCC2)=NO1 C#Cc1ccc(C(=O)NC23CCCC2N(C(=O)C=Cc2cncs2)CC3)cc1F C(C)(CNC(=O)CN1CCC(C)C1)(CC(C)C)NC(C=C(CCC)C)=O Cc1ccc(C(F)C(=O)NCC2CC2NC(c2cc(-c3ccoc3)[nH]n2)=O)cc1 c1(N(C(c2c(C)c(O)ccc2)=O)CCC2CCCNC2)ncnc2n[nH]c(Br)c12 C1(CC=C)(NC(=O)C(CC2CCCC2)OC)CCN(C(c2nc(C)oc2C)=O)C1 CCC(CC)CC(=O)N1CC(CC(=O)NC2CCCC2C(N)=O)(OCC)C1 c1(CC=C2CC(O)C2)nc(-c2ccc(-c3ccccc3)cc2)nn1-c1nc[nH]n1 c1(OC(C)(C)C)ccc(C(N2CCSCC2CCNC(C23CCC2C3)=O)=O)cc1 N1(C(c2cc(Br)cc(C)c2N)=O)CCN(C(=O)CCCC(C)C)C2COCC12 C1(OC(C)(C)C)CN(C(N2CCC(C#C)(O)C2)=O)CC(F)(F)C1 C(N=c1[nH]c2cc(Cl)ccc2s1)C1(C(C)(C)C)CCN(C(C2CCCSS2)=O)C1 C1(NC(C)=O)CC2CCC(C1)N2C(C1(C#N)CCCO1)=O C1(C(=O)NCCCN(C)C(C2CC2Cl)=O)CC(C(F)(F)F)C1 C1(NC(=O)C=CC2CCCO2)CC2CN(C(=O)CCc3ccco3)CC2C1 CC1CCCC(C)N1C(=O)C(N1CCCC(C)(NC(=O)CNC(=O)C2CC2)C1)=O Cc1nn(CC(N2CCC3(NC(c4c[nH]ccc4=O)=O)CC3C2)=O)c(C)c1Cl C1(CN(C(=O)COCCCF)CC)CCCCN1C(=O)CN1CCCC1CO C1(NC(COc2c(OC)cccc2)=O)CCN(CC2CCOC2)CC1C C#Cc1cn(C)nc1C(N1CCN(C(C2COC(C)CO2)=O)C(CCC)C1)=O c1(OC)ccc2c(CNC(C3CCC(Nc4cscc4C)CC3)=O)c[nH]c2n1 C(C(C)S(C)(=O)=O)(c1c(C)cccc1)N(C)Cc1nc(-c2ncccn2)no1 C1(C(N2C(C)CCC(NC(=O)C(C)(C)C3CCCO3)C2)=O)CC2(C1)CS(=O)(=O)C2 C(C)(C)(CC(=O)N=c1ccn(C2CCC2)[nH]1)NC(COCCOC)=O c1(OC)ccc(F)c(C(N2CCC(C)C2)=O)c1NC(c1ccnc(OC)c1)=O N1(C(C2C(c3ccn(C)n3)C2)=O)CCC2(C1)CN(C(=O)CN1CC(C)(C)C1)C2 C1(CNC(=O)CCC2CCCC2)CN(C(c2cnc(C3CCC3)s2)=O)CCCO1 CC1(NC(c2cccn2CCc2ccccn2)=O)CCN(C(=O)CC=C(Cl)Cl)C1 c1(C(=O)NCC(C2CCC2)NC(C2C(OCC)CC2)=O)c(Br)noc1C CCCCCCCC(=O)NC1CCC(C(=O)NC2CC(CF)C2)C1 C12(C(=O)NC3CN(C(Cc4cn(C(C)C)nc4)=O)CC3O)CCCC1CCC2 Cc1c[nH]cc(C(=O)NC2CCC(C)(CNC(c3cn(C)cn3)=O)CC2)c1=O O=C(NNc1ccc(S(=O)(=O)C2CC2)cc1)c1cc2cc(F)ccc2[nH]1 c1(C(=O)NC2CC(C)CN(C(=O)Cc3nnc(S)n3C)C2)ccc2ccccc2c1 N1(C(CC2(C=C)CC2)=O)CCCC(C2CN(C(C3CC4C=CC3C4)=O)C2)C1 CSC1=C(C(=O)N2CCOC(CNC(=O)C(c3ccc(F)cc3)=O)C2)CCCC1 C(CC(CC)C(=O)N1CCC(F)(CNC(C2(Br)CC2)=O)C1)=CC N1(C(=O)CSC2CC2)CC2CCC1C2NC(c1cccc(-n2ccnn2)c1)=O C(C)(C(=O)NCCCCN(CCCNC(=O)C(F)=C1CCC1)C)(C1CC1)OC C1(CNC(=O)CC2CNC(=O)O2)CCN(C(C2CCS(=O)(=O)CC2)=O)CC1O C1(NC(CNC(C(C)NC(=O)OCC)=O)=O)COC2(CCC2)C1 c1(C(=O)NC2(CNC(C(CC)N(CC)CC)=O)CC2)cccc(Cl)c1-n1cccn1.CC c1(CC(=O)NCC(C)N(C(=O)C(C)N(C)C)CC)noc2ccc(F)cc12 C1(CC)CN(C(c2cnn(-c3c(Cl)cccc3Cl)c2)C(=O)NC2CC2)C(CC)CO1 N=c1[nH]c(C2CC2)ncc1C(N1CCC(NC(=O)Cc2ccsc2)C(O)C1)=O N1(C(c2ccc(C)n2C)=O)CC2CS(=O)(=O)CC2(NC(c2ncc(F)cn2)=O)C1 CC(CCCCNC(=O)C(F)C1CCCC1)NC(=O)CCS(C)=O N1(C(CC2CC(SC)C2)=O)CCC(F)(CC2CC2(C)C)CC1 N1(C(c2ccc(-c3ccccc3)nc2)=O)CC2CC(C1)N2C(=O)Cc1cccs1 C1(C(=O)NC2(CN(C(C(C)OC(C)C)=O)C)CC2)CCN(S(C)(=O)=O)C1 c1(C(N2CC(CNC(c3ccc(C#C)o3)=O)C2)=O)ccc(F)c2ccccc12 c1(C(=O)NC(CC)CSC)cccc(CNC(C2(C)CCCCO2)=O)n1 C(=O)(CCC(C)(C)C#N)OC1CC(NCC(=O)NCC(CC)(C)OC)C1 c1(N(Cc2ncccn2)CC2CC2)nnc(Cn2cncn2)n1CC(F)(F)F c1(COCC)ccc(C(N2CCOCC2CNC(=O)C2=C(C)CCC2)=O)cc1F CN1CCC(NC(C2(CSc3cccs3)CC23CCC3)=O)C1c1ccccc1 c1(C(N2CCCC2c2ccon2)=O)ccc(Cc2cn(C3CCOC3)nn2)cc1 N1(C(C(COC)NC(N)=O)=O)CCC2(CC1)CC(NC(=O)CSCC(C)C)CO2 CC1CCN(C(=O)CNc2nccs2)CC1CNC(c1ncsc1C(F)(F)F)=O CC1CN(C(c2cnccc2Cl)=O)CCC1CNC(c1ccc(C#N)cc1)=O C(=O)(CS(=O)(=O)C(C)C)CCC(Cn1cc(-c2cccc(OC)c2F)nn1)F N1(C(COCC#C)=O)CC(C(=O)N(C2CCCC2C#N)C)CC1(C)C C1(=CC(N2CC(C(C)NC=O)C2)=O)CCCCC1(C)C.C(=O)(CCC1CC1)NC=O N1(C(C(=O)NC2C(OC)COCC2)=O)CC2CCCCC12c1ccccc1 Cc1ccc(I)c(NC(c2n[nH]cc2NCc2cncc(F)c2)=O)c1 N1(C(c2ccc(OC)c(F)c2)=O)CCN(C(=O)C(=O)C2CC2)C(C)C1C N1(C(c2cc(C(C)C)c(O)cc2)=O)C2CCCC1CC(NC(=O)CC(C)O)C2 c1(CC)c[nH]c2ncnc(NCC3CCN(C(c4ccc(C)nc4CC)=O)C3)c12 N1(C(CC=C=C)=O)CC2(C(N3CCC3(C)C(=O)OC)=O)CCC1CC2 c1(C(N(CCCNC(c2c[nH]cc2Br)=O)C(C)C)=O)cccc2ncccc12 C1(OC)(CNC(C23CCN(CC2)C3)=O)CCN(C(=O)CC(C)C)C1 N1(CC(CC)NC(C)CCC2CCCCC2)C(=O)CCCC1=O N1(C(C2N(C)CCC2)=O)CC2CC1CCC2NC(=O)C(C)(C)c1nccs1 c1(OCC)cc(F)ccc1CNc1ncc(-c2cc(C#N)ccn2)cc1O C1(NC(C(COC)C)=O)CN(C(C2CCCOCC2)=O)CC12CCCC2 Cc1ccc2ncc(C(N3CCCC4(C3)CN(C(C3(C)CCCO3)=O)C4)=O)n2c1 c1(C(=O)NCCNC(Cc2c(F)ccc(OC)c2)=O)cc(C)c2nc(C)cn2c1 N1(CC)CCCN(C(=O)NC)CC1.c12ccc(cc1)C(N1CC=C(C)CC1)CN2 C12(C(N(CC(C)NC(=O)CCc3ccn(C)n3)C)=O)CCCCC(F)(C1)C2 C1(C)(NC(COc2ccc(OCC)cc2)=O)CCN(CCC2CCC(C)CC2)CC1 c1(C(N2C(CNC(c3c(C)nsc3)=O)CC2)=O)cc2ccc(F)cc2nc1O n1(CC(=O)NC(CN(C(C=Cc2n(CC)ncc2)=O)C)(C)C)nc(Cl)ccc1=O C(=O)(C(F)C(F)(F)F)N(C1CC(NC(c2oc(CC)c(C)c2)=O)C1)C c1(C2CC(C(N(CC(C)NC(C(C)SCCCC)=O)CC)=O)C2)ccccc1 CC1CN(C(=O)CCCCN(C)C)CC(C)CN1C(=O)CCNc1ccccn1 N1(C(C#CC(=O)N(C)C)=O)CCC2C(CCCN2C(=O)C=Cc2ccco2)C1 C1(CC(=O)N(C2CN(C(c3ccc(-c4ccncc4)o3)=O)C2)C)OC(C)(C)OC1=O c1(NC(c2ccc(OC(F)(F)F)cc2)=O)cncc2ccc(F)cc12 C(C(C(=O)N(OC(F)F)C)NC(c1cnn(C(F)F)c1)=O)N(C)C c1(CC=C(C)C)ccc(C(N2CCCC2CC(=O)Nc2csc(C)n2)=O)nc1 CC1C(=O)N(C2CCOCC2)CCN1C(=O)Nc1nc(C(=O)NC2CC2)cs1 c1(OC)cnc(C(=O)NCC(C2CCOC2)NC(c2ccsc2Cl)=O)nc1 CCC(C)C(=O)N(CCNC(c1ocnc1-c1ccccc1)=O)CC1CC1 Cc1ccc(C(=O)Nc2ccc(NC(C3CCCC(C)C3)=O)cn2)nc1 N1(C(C(n2cc(CN3CCOCCC3=O)nn2)C)=O)CCC(C2CCC2)C1 c1(C(N2C(C(CNC(C(=O)NC(C)C)=O)(C)C)CCC2)=O)cc(F)ccc1Br CC(CC(=O)NC1CC(F)(CNC(c2cncc(C(F)(F)F)n2)=O)C1)C(F)(F)F CCCCCC(C)CC(=O)N1CCC(C)(NC(C2CC(C(C)C)C2)=O)C1 C1(C(=O)NC23CC(NC(C4CNC(=O)N4)=O)(C2)C3)C2CCCCC12 N1(C(C2(COC)CCC(N)C2)=O)CC2C3C=CC(O3)C2C1.C1C(=O)N1 C1(C2=CCOCC2)(CNC(C2CCN(CC(F)(F)F)CC2)=O)CC1 C1(CNC(C(CC=CCC)C)=O)CCC2(CCC2)CN1C(=O)C(C)CSC c1(N2c3cn(nn3)-c3cc(cc(Cl)c3)NC2=O)ccc(C(C)=O)cc1F.CC.SC N1(C(c2n(C)cc(Cl)c2)=O)CCOCC(F)(CNC(c2cccnc2)=O)C1 N1(C(CC2N(C)CCCC2)=O)CCCCC(NC(=O)Cc2nccn2C)CC1 c1(OC)ccc(Cl)c(C(=O)NC2CCCC2CNC(C2CCCOC2)=O)n1 C1(NC(c2n(-c3c(C)cccc3)nnn2)c2csc(Br)c2)CC(C)(C)C12CC2 CCC(O)CCN=c1cc(C)c(S(=O)(=O)NC2CCCCC2C(C)(C)C)c[nH]1 N1(c2cc(OC)nc(CC)n2)CC23CCCC2(CN(C(=O)C#CC2CC2)C3)C1 C1(C(=O)NC2(CN(C(C3CC(OC)C3)=O)C)CC2)Cc2ccccc2C1(C)C S(=O)(=O)(c1ccc(NC2CCCC2S(C)(=O)=O)c(Cl)c1)N(CCC)CC N1(C(C(Cc2ccccc2)SC)=O)CCC(O)(CNC(c2ccon2)=O)CC1 C1(CC(=O)NCC(CCOC)NC(=O)C=Cc2ccc(C)o2)CCC(=O)NC1 c1(C(C(=O)NC(CC=C)CNC(C2(O)CC2)=O)C)ccc(C(F)(F)F)nc1 C=CC1CN(C(=O)Cc2nccn2C)CC1NC(c1nn[nH]c1Cl)=O c1(C(=O)NC2CC(CC3CN(C(=O)OC(C)(C)C)C3)C2)cc([N+](=O)[O-])sn1 C(CCCOC)(C(=O)N(C1CCCC1(C)O)C)NC(COCC=C)=O N1(C(C2(CCOC)CCC2)=O)CCC(NC(C2CCN(C)C2=O)=O)CC(O)C1 c1(CC(=O)N(C2CCN(C(C3CC34CC(O)C4)=O)C2)CC)cc(F)cc(F)c1 CC(C)CC(CNC(=O)CCC1OCCO1)C(=O)N1CCC(F)(C(N)=O)C1 C1(C(=O)NC(CCCC)C(=O)NC)CCCCCCN1C(c1cccc[n+]1[O-])=O c1(C(N2C(CNC(C3C(C)(C)CO3)=O)CCC2)=O)csc2c1CCCC2 c1(OC)ccc(OC)c(CC(=O)N(C(C)CCNC(c2occc2Br)=O)C)c1 C1(CNC(CCC2C(C)(C)C2)=O)CN(C(c2cc(C3CC3)[nH]n2)=O)CCO1 C1(CNC(C2(OCC)CC2)=O)CC2CC1CN2C(c1nc(Cl)cs1)=O c1(CC(=O)NCC(C)CNC(C23CC(C)(C2)C3)=O)cccc2c1OC(C)(C)C2 C(c1cn(C)nn1)=CC(=O)NC(C(=O)N(C)CCN1CCCC1=O)c1cccs1 C1(CN(C=O)Cc2cnc(-c3ccccc3Cl)s2)CCC(F)(F)CO1 Cc1cc(O)nc(C)c1C(N1CCC(NC(=O)CSc2cccs2)C(F)C1)=O C(C(F)(F)F)(c1nc(CCN2CCOCC2)no1)NCCNC(=O)OC(C)(C)C CC1(C)CN(C(C2CCCCO2)=O)CC1NC(c1cnn(CC2CCCC2)c1)=O C1(NC(c2cncc(C)c2)=O)CC(C(=O)N(C)Cc2cc(C)no2)C12CCC2 n1(C2(C(=O)NC(C)C=CC(=O)NC(=O)C(F)=CC3CC3)CC2)cncn1 c1(C(N2CC(NC(C3CCC(CCC)CC3)=O)C(F)C2)=O)cnc2c(c1)CCC2 C1(CCC(=O)N(CCCNC(c2cnsn2)=O)C(C)C)NC(=O)NC1=O C1=CC(=O)NC(C(=O)N(C)OCCOCC)C1.C1CC12CCC2.CC=C c1(OC)cc(C)c(Cl)cc1C(N1CC2(CCN(C(=O)CC3CCCCO3)C2)C1)=O N1(C(c2c(C)occ2)=O)CCC2(CC1)CC(C(N1CC(=O)NC(C)C1)=O)CO2 c1(SCC(=O)NC(C(=O)NCCCNC(C)=O)C)ccc(F)cc1 C1(C(=O)NCC(C)F)CC12CCN(C(C1CCOCC1)=O)CC2 C#CCC(C)(CC)C(=O)NCC1CCC(C(C)C)N1C(=O)CCOCC1CC1 c1(C(=O)NC2CCC(C(=O)N(C3CC(Br)C3)CCO)CC2)ccc(Cl)cc1CO C(c1ccc(F)c(C)c1)=CC(=O)NCC1=CCN(C(C(C(C)C)OC)=O)CC1 c1(C(N2C(CNC(C(c3ccccc3)C)=O)CC2)=O)ncc(F)cn1 c1(NC2C(NC(CCCCC(=O)NC)=O)CCCC2)nc2cc(F)c(F)cc2s1 C1(C)(C(N2CC(CCC=C)(C(=O)NC3(C(=O)OC)CC3)C2)=O)CCC(C)C1 S(=O)(=O)(CC(=O)NC1C2CN(CC(=O)Nc3cccc(F)c3)CC12)N(C)C C(=O)(C(CC=CC)NC(=O)Cc1ccoc1)N1CCC(CC#C)C1 CC1(C)CC(NC(=O)COc2cccc(F)c2)CN1C(c1cc(C2CC2)on1)=O Cc1nc(CO)sc1C(=O)NC12CC(NC(C3CCCN3C)=O)(C1)C2 O=C(CS(=O)(=O)CCO)NC12CCCN(C(=O)CCSC(F)(F)F)CC1C2 N1(C(C(C)OCC)=O)C2CCC(C2)C1CC(=O)NCc1ccns1 c1(C(N2CC(C(C)NC(C3CCCC(C)(C)C3)=O)C2)=O)cc(N)c(Cl)c(O)n1 CC1(C)C(NC(=O)COC(F)(F)F)CCN1C(=O)CCCCc1ccccc1 N1(C(c2nc(OCC)oc2)=O)CC2(CCC(CNC(=O)C(C)CCCOC)O2)C1 C12(C(N(CCNC(c3csc(C(F)(F)F)c3)=O)CC)=O)CCC(C1)C(C)O2 C12(OC)CCC(C(=O)NC34CC3CN(C(C35COCC(C3)C5)=O)C4)(CC1)C2 C(C1=CCN(C(c2ccc(O)cc2F)=O)CC1)NC(=O)CCc1cccc(Cl)c1 Cc1c(C(=O)NC(C)(C)CCN(C(=O)Cc2ccsn2)C)cnc2ccnn12 N1(NC2CN(c3cc(=N)[nH]c(Cl)n3)C2)CCN(C(=O)C(F)(F)F)C(=O)C1 C1(CN)CN(C(c2cc(C(F)(F)F)ccc2Cl)=O)CCCO1 C(=O)(CC(C)P(C)(C)=O)N1C(CNC(CCOCC(C)C)=O)CC(F)C1 CC1CC(CC(=O)NCCS(C)(=O)=O)CN1C(C1SCCS1)=O N1(C(C2(CSC)CC2)=O)CCC2(CCCN(C(c3cccnc3C(F)F)=O)C2)C1 N1(C(c2ccnc(CC)c2)C(=O)NCCC(=O)OCC)CC(OCCC)CC(C)C1 c1(OC)c(F)cc(C(N2CCC2C(=O)NCCOc2cccc(Cl)c2Cl)=O)cc1F N1(C(C(C)OCCC=C)=O)CCOC(CCNC(=O)C(C)(C)c2cc[nH]n2)C1 C(C(=O)NCCOCCCNC(=O)C(C)c1ccco1)(C1CCC1)OC C1(C(=O)NC2(COC)CC2)CCOC1C(=O)NC1(CC(=O)OC)CCC1 c1(NC2CCC(CCC)CC2)ncc(OCC)cc1Cl C1(C(N2C(C)CC(CNC(CSCC(C)C)=O)C2)=O)CCC2CC1C2(C)C c1(C(=O)NCC(CN(C(c2c(C)cno2)=O)C)O)coc2c(F)cc(F)cc12 c1(C(N(CCCNC(C2CC2(C)Br)=O)CC)=O)[nH]c2cccc(C)c2c1C c1(OC)ccc(CN2CCCC(NC(=O)C(O)C(C)(C)C)C2C)cc1Br c1(C(=O)NCC#CCNC(C2CCC(NCC)C2)=O)ccc(C#N)s1 c1(CC)cc(C)ccc1C(=O)NC1CN(C(=O)C(C)(C)COC(C)C)CC1(C)C Cc1cc(Cl)nc2ccc(NS(=O)(=O)CC3CCCCC3CC(=O)O)cc12 c1(CC)nc(C)oc1C(=O)NCCc1n[nH]cc1C(=O)NCCn1ccnn1 C1(NC(=O)COc2ccccn2)CCC(C)C1.C1(C(N(C)C)=O)CC(C(N)=O)C1 C(=O)(C#CCNC(c1nscc1C)=O)NC(C#C)(C)C1CCC1 C12(C(=O)NCC(CCCC)NC(c3cc(C4CC4)cs3)=O)CCC(O)C1CC2 C1(C(=O)Nc2ccc(SC)o2)CCCC(C(=O)NCC(C)(F)C(C)C)C1 c1(CC(C)(C)C)noc2nc(C3CC3)cc(C(=O)NCC3CC(=O)OC3(C)C)c12 c1(C(=O)NC(CNC(=O)C=CCF)C2CC2)ccc(OCCO)cc1 N1(C(c2ccc(CC)cn2)=O)CC(CNC(=O)C=Cc2cn[nH]c2)C(C)(C)C1 c1(OC)cccc(NNC(=O)C(C(=O)OC)c2ccccc2)n1 CC(CF)CC(=O)NCC1CC(CNC(C2(c3ccc(Cl)cc3)CCC2)=O)CO1 C(=O)(CC(C)(C)C)N(CCNC(C(C)NC(=O)CSCC#N)=O)C C1(C2(O)CCOCC2)(C(=O)NC23C(C)OC(CNC(c4cocn4)=O)(C2)C3)CC1 N1(C(C(CNC(C(C(=O)OC)(C)C)=O)N(C)C)=O)CCC(NC(C)=O)C(C)(C)C1 C(=O)(C(C)CCc1cccc(F)c1)N1CCC(N(C(c2nn[nH]c2Cl)=O)CC)C1 Cc1c(Cl)ccc(C(=O)NCC(C)CNC(=O)C(C(C)C)N(C)C)c1F C1(CC)C(C(N2CCCC2CF)=O)CCN1C(=O)C(C1CCCCC1)C C1(Cn2cc(C(C)(C)C)nn2)CC2CCC1N(C(C1(O)CC3CCC1C3)=O)C2 Cc1ccc(N)c(C(=O)OC(=O)CCc2ccccc2)c1F.C1C(CO)NCC(=O)N1 c1(NC(CC(CC)O)=O)cnn2c1CN(C(=O)NCC(F)(F)F)CC2 C(=O)(C1=NNC(C(F)(F)F)C1)NC(CNC(C(c1ccncc1)C)=O)CC(C)C CC1CCOC(C(N2CCOCC2CNC(c2ccccc2CO)=O)=O)C1 c1(C(=O)NC(CCCNC(C(C)C2CC2)=O)(C)C)cc(S(N)(=O)=O)ccc1F c1(C(C(C)OCC)NC(=O)NC2CC(n3cccn3)C2)ccccc1 C(=O)(C1=Cc2ccccc2C1)NCC1N(C(C(COC)NC(C)=O)=O)CCCC1 c1(C(=O)NC2CC(N(C(CC=CC=C)=O)C)C2)sc(Cl)c(Cl)c1N CC1CCC(F)(C(=O)NC(CC(=O)N2CCC2)C2CC2)CC1 C(=O)(CC(C=C)CCC)N1CCC(C(N(CCCCCC=C)C)=O)(CC)CC1 Cc1cc(CNC2CCC3(CC2)CSC3)c2ccc(F)cc2n1 C#CCC(CC(=O)NCCC1CC(C)(C)C1)NC(C1CCOCC1(C)C)=O C#Cc1cncc(C(=O)NC(CC2CC2)CC(=O)N(CCCO)CC2CC2)c1 Cc1cc(C(=O)N(C2CN(C(c3cc[nH]c3)=O)C2)C)c(O)nc1C C1(OC)CCCN(C(c2cc(Br)c(C(=O)O)s2)C(=O)NCCCSC)C1 c1(OC)ccc(C=CC(=O)NC2C=CCN(C(C3(O)CCCC3)=O)C2)cc1F C(CC1(C)CCOC1)(C(=O)NCCNC(=O)C1CC1)N(C(C(=O)N(C)CC)C)C N1(C(C(C)C2CCCO2)=O)CCC2(CC1)CN(C(c1csc(F)c1)=O)C2 C(=O)(CCN1C(=O)COc2ccccc21)N1CCC(C(C)NC(C=NOC)=O)C1 C1(CNC(C2(COC)CC2)=O)CCC1C(=O)NCC1CCCS1 Cc1[nH]nc(Br)c1C(=O)NC(c1cccc(N2C(=O)CCC2=O)c1)c1ccccc1 C(CN=C(NCC(O)Cc1ccc(F)c(F)c1)NC1CCC1)c1nc(C)sc1 C(=O)(C(C)(F)C(C)(C)F)NCC=CCC(=O)NCCCC=C CCC(C)C(C(=O)NCC1CN(C(=O)CNC(=O)CN(C)C)CC1C)NC(C)=O CC1CN(C(c2cnc(S)nc2)=O)CCC1N(C)C(c1ccn(CCF)n1)=O C(=O)(C(O)CCS(C)=O)NCCCN(C(c1cnc(CC)[nH]1)=O)C(C)C C1(NC2CC2)CCN(C(C2CCCN2C(C2C=CCS2)=O)=O)CC1 CC(CCC(=O)NCC(C)O)NC(=O)C(C)CC1CCC1 C1(CNC(=O)CCc2cnn[nH]2)CC(CNC(=O)C(=O)NCC(F)F)CO1 N1(C(C2C(C)CCC2)=O)CCC(O)(CNC(=O)Cc2cc(Cl)n(C)n2)CC1 C1(F)(OC(C)C(=O)C2CCCC2)CCCN(C(=O)C(N2CC(C)(C)C2)=O)C1 N#Cc1cc(C(N2CCC(N3CCN(C(c4cccnc4O)=O)CC3)C2)=O)no1 C1(N(C(C2CC2c2cncs2)=O)CC)CCN(C(=O)Cn2cccn2)CC1 n1(CC)ncc(C(=O)NCc2cc(C(=O)NC3CCN(CCF)C3)no2)c1C N1(C(c2n(C(C)(C)C)ncc2)=O)CC2(CCCC2NC(C2CC23CCOC3)=O)C1 N1(C(CN2CCC(C)CC2)=O)CCOCC(C(=O)NC2CC(C)(C)C2)C1 c1cn2c(n1)CC(NCC13CCC(CN(Cc4ccccc4)C1)C3)CC2 C1(NC(C(c2cccc(C)c2)C)=O)CN(C(c2ccc(C)o2)=O)CC2(CC2)C1 c1(C(=O)NC2C(C)N(c3ncc(C#N)cc3Cl)CCC2)cc2ccccc2cn1 c1(C(c2n(CCCC)nnn2)NCCSC#N)nnc2nc(C)ccn12 C(=O)(C#CC1(C)COC1)NC1CC(CNC(c2c(OC)ccc(Br)c2)=O)C1 CC1=C(C(=O)NCC(C)CNC(c2ccco2)=O)C(=O)OC1(C)C c1(C(=O)NC(CNC(C(CC)Br)=O)C(C)(C)C)c(O)nnc2c1CCC2 C1(CNC(c2c(C)ccc(F)c2)=O)CC2COCC2N1C(c1cncn1C)=O N1(C(=O)NC(c2cccc(C)c2)C(C)C)CCSC2(CCCC2)C1 C(CCC(O)C(=O)NCCc1noc(C)n1)NC(C(CC)n1ccnc1)=O CC(C(CO)NC(c1nc(C2CCCC2)no1)=O)NC(=O)CNC(C1(C)CC1)=O C(CC(C(=O)NCCC(C)(O)C1CC1)N(C)C)NC(Cc1ccc(C)o1)=O C1(C(N2C(c3ccc(C)c(C)c3)CCC2)=O)CC2(C)CCCN2S1(=O)=O c1(NC(C(=O)Nc2c(OC)cccc2Cl)=O)cccc2c1OCCC2O c1(C(=O)NC2(C)CN(C(C3CCN4CCCC4C3)=O)C2)nc(Cl)cc(N)c1Cl N1(c2nc(N3CCC(F)(CF)C3)nc3c2CCC3)CCOc2ccncc2C1 C1(C(=O)NCc2ccc(F)c(F)c2Br)CC2(CCC(F)(F)CC2)N1 N1(C(C(c2c(C)nn(C)c2)C)=O)CCN(C(=O)Cc2ccc(F)cc2)C2CCC12 C1(C(=O)NC(C2(O)CN(C(c3ccnn3CC(C)C)=O)C2)C)(OC)CCCCC1 c1(C(c2nnnn2C2(C)CC2)NC2CC(C(C)C)C2)ccn(C(C)C)c1 C12(CNC(C#CC3(C)CC3)=O)CN(C(c3ccccc3[N+](=O)[O-])=O)CC1CCO2 CCC(O)C(F)(F)C(=O)N1CCC1(C)CC(=O)Nc1ccccc1C O=C(CC1=CCCCC1)NCCOCCNC(c1cccnc1C(F)(F)F)=O C1(NC(CC2C(NC(C(C)Cn3cccn3)=O)CC2)=O)(CC2CC2)CCCCC1 c1(C(N2CCC(CNC(c3ccc(C#N)o3)=O)C2)=O)ccc2c(O)nncc2c1 N1(C(C2N(C)CCCC2)=O)CC=C(CNC(C2(C3CCCO3)CCC2)=O)CC1 CCCC(CCCNC(=O)CCF)NC(C1(C2CCCO2)CC1)=O Cc1ncccc1C(C)NC(C1CCC1NC(C1CC=CC1)=O)=O CCC(C)(CNC(c1cc(C)nn1C)=O)C(=O)NCCNC(C)=O Cc1ccccc1CCC(=O)NCCC1(O)CN(C(=O)C(n2cc(Cl)cn2)C)C1 N1(C(CC)CC)CCCN(C(c2cccc(-n3cccn3)n2)=O)CC1 C1(C(N(CC(C)N(C(c2cc(C)ncc2C)=O)C)C)=O)CCn2nccc2C1 C1(NC(=O)COc2ccc(Br)cc2)CCSC12CN(C(C1CC1[N+](=O)[O-])=O)C2 c1(CC)nc(O)c(C(=O)NCC2CN(C(C3CC(F)CN3C)=O)CC2O)cc1C Cc1cc(OC2CCCCC2)cc(C)c1CC(=O)NCC(C)C(C)(C)C C1(NC(COC)=O)CCCC12CN(C(c1sc(-c3ccccc3)nc1C)=O)C2 N1(C(COCCC=C)=O)C(C(N2CCCC(C(C)C)CC2)=O)CCC12CC2 c1(C(N2CC3CN(C(Cc4c(C)nc[nH]4)=O)CC3C2)=O)cccc2c1C(=O)CC2 C(=O)(NNc1ccc(Br)c(Cl)c1)NC1COCC(C)(CC)O1 CC1CCC(C)N1CC(N1CC(O)(C(F)C(N2CC3C(N(C)C)C3C2)=O)C1)=O N1(c2snc(C(C)C)n2)CCCCC(CNC(c2ccn(C)n2)=O)C1 CC1CN(C(=O)CCCn2cccn2)CC1CC(=O)N(C1CC1)CC1CCCO1 Cc1ccc(C(N2CCOC(CCNC(C3CCCC3C)=O)C2)=O)c(N)c1 N1(C(C2(C)N(C(C3ON=C(C(C)C)C3)=O)CC=C2)=O)CC2(CCC(=O)NC2)C1 N1(C(=O)NCCCCCOC)CCCC(O)(c2cn(C3CCOC3)nn2)CC1 C1(c2ccccc2)(C(N(C2CCN(Cc3cccnc3)C2)C)=O)CC(F)(F)C1 C1(NC(CN2CC(=O)NCC2)=O)CCC2CC1CN2C(c1ccc(C2CC2)s1)=O c1(C(=O)NCCCC2(CNC(c3nc(CC)oc3)=O)CCCC2)cnc(S)nc1 C1(NC(C(C2CCC2)OC)=O)COC2(C1)CN(C(=O)Cc1ccsc1C)C2 N#Cc1ccccc1OCc1noc(-c2ccc(Br)cc2)n1 C1(N(S(=O)(=O)Cc2ccccc2I)C2COC2)CC2(CCNCC2)C1 CCC(CCC(=O)OC(C)(C)C)S(=O)(=O)NCC(N)C(=O)OC c1(C(N2CCCC(CN(C)C(c3cc(CF)on3)=O)C2)=O)cc(F)ccc1O c1(N(CC#CC)CC)cc(Br)ccc1S(=O)(=O)NC1CC1 C(=O)(C1=CC(O)C(NC(c2cc3cccnc3[nH]2)=O)C1)N(C1CCC2CC12)C O=C(CC(C1CC1)C1CC1)NCc1csc(O)n1.C1(N2CC2=O)CCCC1 N1(C(c2cn(CCC)nc2C)=O)CCCC(NC(=O)CC(C)(C)O)C1C C(c1ccccn1)=CC(=O)NCCCCCNC(C1CCC1c1nc(S)n[nH]1)=O N1(c2c(C)c(NCc3nccc(O)n3)ncn2)CCC2(CC1)CC(O)CO2 C(=O)(C1Cc2ccc(C)cc21)N1CC(C2N(C(C=C(C)C)=O)CCC2)(O)C1 Cc1ccc(CC(=O)NC(c2nc(C)no2)C)cc1.C12(CC3(CC3)C1)C(=O)NC2 C(C(CCC)C(=O)OC(C)C)NC(=O)NCCCCC#C Cc1cc(CN2CCCC(C(=O)NCc3[nH]cnc3C)C2)c(C)[nH]1 c1(SC)c(NC(=O)C(=O)NC2CCC(C)(C)C2)cccc1F N1(C(C(=O)NCCOCC(C)C)=O)CCCC1c1nc(COC)cs1.C(CO)O CN1CCc2nc(C(=O)NCC3(C)CCCN(C(C4CC(C)(O)C4)=O)C3)sc2C1 C1(n2cccn2)(C(=O)OCC)CCN(C(=O)Cn2cc(Br)cn2)CC1 Cn1cnc2c(NCCc3cccs3)[nH]c(=NCC(C)(F)F)nc12 CC1OC23CC1(C2)c1cn3nn1.N1(CCO)CC(C)C1c1nccn1-c1ccccc1 CCCC(C(=O)NCCC(C)NC(=O)CC1CSCCS1)S(N)(=O)=O C1(C)(NC(CC(=O)NCC)=O)CCN(C(C2CCC(CC)O2)=O)C1 C(=O)(C1=CC2CC=CCC12)NC1(C)CN(C(c2cc(C)c(N)cn2)=O)C1 N=c1[nH]c2c(s1)CCCC2C(=O)NC1(CO)CN(C(C2CCC3CC3CC2)=O)C1 N#CC1(CNC(C2CCC(NC(=O)CCOC3CC3)C2)=O)CCC1 N1(C(C(C(C)(F)F)(C)C)=O)CCC2(CCN(C(C34CCCC3(C(N)=O)C4)=O)C2)C1 c1(OC)ccc(C(=O)NCC(CC(F)(F)F)NC(c2ccccn2)=O)c(F)n1 C1(C(N2CCOCC2Cc2ccc(O)cc2)=O)CC2(CCC(F)(F)CC2)C1 c1(CC(=O)NC(C)CCCNC(c2nc(Cl)cs2)=O)ccc(-n2ccnc2)cc1 c1(CC(=O)NCc2cn(CCNC(C3CCOC3)=O)nn2)ccnc(Cl)c1F C1(=O)C(CCSC)CN1.c1(SC)nc(N(C)C)n[nH]1.C(=O)COCC(C)C N1(C(COCCN(C)C)=O)CCC2CN(C(c3ccc(C#N)cn3)=O)CCC2C1 O=[N+]([O-])c1ccc(-c2nc(-c3ccc(O)cc3)nn2-c2cncnc2)cc1 Cc1cn2ccc(C(=O)NCC3CCC4(CN(c5snc(Cl)c5C#N)C4)O3)cc2n1 C(=O)(C1=CCCCO1)NCCC(C)NC(C1CN(C(=O)OCCl)C1)=O.C(C)(C)(C)C Cc1cc(C(=O)NCCC2COCCN2C(=O)C=CCl)nnc1C.C(=O)C(C)(C)C CCC(C)(COC)C(=O)N1CC2CC2(NC(C2CC=CC2)=O)C1 N1(C(C2N(C(c3c(C)nccn3)=O)CC(O)C2)=O)CCC2(CC1)CC2C#N CC1CCCN(C(=O)CSC2CCOC2=O)C1CCNC(C1(CO)CC1(F)F)=O C1(N(C(c2cc(C)sc2)=O)C)CN(C(C2CC(CC(F)(F)F)C2)=O)CC12CC2 C1(CC(=O)N(C(CC(=O)NCC(=C)C)C)C)C(=O)NN=C1C C1(NC(COC2CC(NC(C(C)(C)F)=O)C2)=O)CC12CCOC2 C1(C(N2CC(c3cn(C4CCC4)nn3)C2)=O)CCC(C2CCCCO2)CC1 C1(NC(=O)C(c2ccccc2Cl)O)CN(C(c2ccc(F)cc2)=O)CC1C1CC1 c1(C(N2C(C)C(C)N(C(=O)CCF)CC2)=O)cc2cc([N+](=O)[O-])ccc2[nH]1 c1(C(N(C(C)CNC(=O)COC2CCCC2)C)=O)cncc2cccnc12 n1(CCC(C)(C)OC)nc(-c2ccc(F)cc2)nc1-c1ccccc1O c1(C(=O)NCC2(C)N(C(C(C)CO)=O)CCC2)cc2n(n1)CCOC2 N1(C(C(=O)NCC(CC)(C)C(=O)O)=O)CCC2(CC1)CC2Cc1ccc(Cl)cc1 c1(C(N2CCN(C(C(CC)F)=O)CC(CO)C2)=O)ccc(S(C)(=O)=O)cc1 c1(SCCN(C(=O)CCCn2cnc(C#N)n2)C(C)(C)C)cnc2ccccn12 C1(NC(CCCc2n(C)cnn2)=O)CCN(C(=O)CC2CC(=O)NC2=O)CC1F C(=O)(C(F)(F)C(C)(C)O)NC(CCN(C)C(C1(O)CCCCCC1)=O)(C)C C1(O)(CNC(C(CC(CC)CC)F)=O)CC2CCC(C1)N2C(C1CCC(=O)C1)=O c1(C(=O)NCCN(C(CC2(COC)CC2)=O)C2CC2)cc(C)c(Br)c(Cl)c1 c1(OCC(C)C)nccc(N(C)C)c1O.C12(CCSCC1)C(=O)O2 C1(O)(C(=O)NC2(CCCC)CC2)CN(C(=O)CSCCSC)C1 CN1CCCC(CC(=O)NC2CCCCC2NC(c2n[nH]cc2C2CCC2)=O)C1 O=C(C1=NOCC1)NCCCC1CCCN1C(=O)CSCC(F)F CCC(C)CC(C)C(=O)N1CCC(N(C(=O)CC(C)C2CCCO2)C)CC1 N#Cc1ccc(C(=O)NC2CCCC(CNC(=O)C=CSCc3ccco3)C2)s1 C(=O)(C(C)CC(N)=O)N1CC(OCC)(CNC(C2SC3C=CC2CC3)=O)C1 n1(CCC)nccc1C(=O)N(CC(C)CNC(c1nocc1Br)=O)C c1(C(N(C2C(C)CCN(C(CC(C)F)=O)C2)C)=O)ccn2nnnc2c1 C1(N(C(=O)C=Cc2nn[nH]n2)CC)CC2CCC1CC2 C1(CCNC(=O)Cn2cnc(C(F)(F)F)n2)CSCCN1C(=O)CCF N1(C(c2c(C)cc(N)cc2)=O)CCC2(C1)CN(C(C1CCn3nncc3C1)=O)C2 N1(C(Cc2ccn(C)n2)=O)CC2CCC1CN2CCNC(=O)NC1CC1 C#Cc1cnn(C)c1C(=O)NCc1occc1C(N1CC(=O)NC(C)C1)=O C1(N(C(=O)CC(F)(F)c2ccccn2)C)CC2C(O)C(O)CC12 c1(C(=O)NCCN(CCN2CCC(CC)C2)C)cc(C(F)(F)F)cnc1C c1(C(N2CCC(NC(c3ncc(NC)nc3)=O)CC2C)=O)ccc2ncsc2c1 c1(OC)ccc2c(c1)CCCN2C(c1cc(C)c(Br)c(Cl)c1)=O c1(C(N(CC(C)N(C(C2(CC#C)CC2)=O)C)CC)=O)cccc2sccc12 c1(C(=O)NC(CC)CN(C(=O)C(c2ccnn2C)C)C)ncc(C)cc1F c1(N2C3CN(Cc4c(C)c(F)c(F)cc4)CC32)ncnc2[nH]cc(C#N)c12 C1(C(=O)NCCCN(C(c2nc(C3CC3)cs2)=O)CC)CCC(F)(F)C1 C(=O)(C1CCCc2c(Br)cccc21)NC(COC)(C)C(=O)OC c1(CC(C)NC2(c3n(CC)nnn3)CSC2)ccccc1OC CC1CC(CC(=O)N(C)CCN2CCOCC2)CN1C(=O)CCCCC1CC1 C(=O)(CC(C)CC(=O)N1C2CCC1CC(NC(C1CCCN(C(N)=O)C1)=O)C2)OC C=CCCCC(C(=O)NC1CCOC1=O)NC(=O)CC(C(=C)C)OCC c1(C(N2CC(COC)(CNC(=O)CCC(C)=O)C2)=O)cccc(C)c1F C1(CC(=O)NCC(CN(C)C(c2ccc(Cl)[nH]2)=O)O)CCCN1C N1(CC)C(C)CN(C(=O)C(c2cccnc2)NC(=O)CN2CCCNC2=O)CC1C c1(OC)c(NC2CN(C(c3ccc(N(C)C)c(F)c3)=O)C2)ncnc1Cl N1(C(CC(C)C)=O)CCCC(C)C1CCNC(c1coc(C(N)=O)c1)=O CC1(C(=O)NCC2CCC(NC(C3CC4CCCCC34)=O)CC2)CCCNC1=O C(=O)(C#CC1CCOCC1)NCC(C)C(=O)NCCN1CCOC1=O C1(NC(c2ccc(C)c(N)c2)=O)CC2(CCC(NC(C3CC3(Cl)Cl)=O)CC2)C1 C(=O)(C(C)(C)CCCF)NCC1(O)CCCN(C(C)=O)C1.N12CCCC1C=CC2=O C(=O)(CCC(=O)NCC(C(C)(C)C)NC(=O)CCCn1ccnn1)OCC O=C(C#Cc1ccc(Cl)cc1)N1CCC2C1CCN2C(c1cc(Br)ccc1O)=O CC1Cc2cccc(C(=O)NC(CNC(=O)CN3CC4CC4C3)C(C)(C)C)c2O1 CCCCCCC(=O)N1CCCC(C(=O)Nc2cncc(C)n2)CC1 c1(C(N2CCC(C)C(CNC(=O)C(F)(F)C3CC3)C2)=O)cc2ccc(F)cc2s1 CC(C)(C)C#CC(=O)N1CC(C)(C(=O)NC2(CO)CC2)C1 CN1N=C(C(=O)N2CCC2CNC(c2nccc3[nH]ccc23)=O)CCC1=O CCCCC(C)C(=O)NC1CC(F)(CNC(=O)CN2CC(=O)N(C)C2=O)C1 c1(NC2CCN(C(c3cnc(C)[nH]3)=O)C2)c(C)noc1C c1(CNC2CCC(C(=O)Nc3c(N(C)C)nccc3)C2)cccc2occc12 N1(C(c2ccc(C(=O)OC)c(C(F)(F)F)c2)C(=O)NCC)CCC2(CCSC2)C1 c1(CC(=O)NC2CC(CO)N(C(C3CC34CCCC4)=O)C2)c[nH]c2ncccc12 C1(CCCNC(C23CC(CC)(C2)C3)=O)CCCCN1C(=O)Cc1ccc(O)nn1 C1(CC(N2CC(C)C(NC(c3coc(C4CCC4)n3)=O)C2)=O)CCCCC(=O)N1 c1(N2C(C)CC(NC(c3ccc(OC)cc3C)=O)C2)nc2cccc(F)c2o1 C(C(C)(C)CC(=O)NCCOCCN(C)C(c1conc1C1CC1C)=O)OC.COC c1(C(C(=O)NC(c2ccccc2)C)N(C(CC)C)C)nc(Br)nn1C N1(CC)C(=O)NC2C(=C1c1ccn(C)n1)C(=O)OC(=O)c1ccc2s1.OCC C1(C)(NC(c2cccc(CC)n2)=O)CCCN(C(=O)CC(C)COC)C1 C(=O)(CCCC(=O)N1CCC(C2CCCN2C(C2(CC3CC3)CC2)=O)C1)OCC C1(CNCC2(OC)CN(c3nnnn3C3CCCC3C(=O)O)C2)CC12CCCC2 c1(C2(NCC3(C(F)(F)F)CC(O)C3)CC2)c(F)ccc(Cl)c1F c1(CNC(=O)NCC(=O)NC(C(C)OCC)NC(CCC)=O)cc2cccnc2s1 CCC(C#N)CNC(=O)C(C)N(C)C(C1CC(N(C)C)C1)=O c1(C(=O)NCC2CC(F)(CNC(c3c(CC)nc(C)[nH]3)=O)C2)ccc(Cl)c(N)c1 C1(C(=O)NCC(CNC(COCCOC)=O)OC)CN(C)CCO1 CCCC(CC)CCC(=O)N(CC(C)C(=O)NCCN1CCCC(O)C1)C S(=O)(=O)(c1cccc(=NCc2cccc(Cl)c2Br)[nH]1)NC(C(C)(C1CC1)OC)C C(CC(=O)NCC(O)CC)(C(F)F)NC(c1c(CC)cccn1)=O C1(CNC(C2(NC(C3C(C)(C(F)F)C3)=O)CSC2)=O)CC2(CC2)CO1 CN1CCC(OCCC(=O)OCc2ncncc2Cl)CC1 c1(C(N(C(CC(=O)N(CCCC)CC)C)C)=O)nnc(S)n1C C(=O)(CC(C(F)F)NC(c1ccccc1)=O)NCCN(CCC)C1CC1 CCCCC(C(=O)N1CC(N2CC(NC(C3(C(N)=O)CC3)=O)CC2=O)C1)C(C)C C1(CC(=O)NC(c2cn(C)nc2)C(=O)NC2CC2(C)C)CCCCCC1 c1(C(=O)NC2(CC=C)CN(c3ncc(C)cn3)C2)ccc2c(c1)CCC2 C1(C(N2CC(O)(CC=C)C2)=O)CN(C(C2(OCC)CCC2)=O)CC1F O=C(CCn1cnnc1-c1ccccc1)N=c1cc(Sc2ccccc2O)[nH][nH]1 C1(C(N2CCC(C(C(=O)N(CC(F)F)CCC)F)C2)=O)CC2(CCC2)C1 C1(C(=O)NC2C=CCN(C(C(OC)OC)=O)C2)COc2ccc(O)cc2O1 C1(NC(C(CO)NC(C2C(C)C2)=O)=O)CC(F)(F)C1(C)C.C1C(=O)N1 CC1(C)CCC2(CC1)CC2C(=O)NCCN(C(c1ncc(F)cc1F)=O)C1CC1 c1(C(=O)NCC2(F)CN(C(C3C(C)C3(F)F)=O)C2)cc(N(C)C)nc(Cl)c1 C=C(C)c1ccccc1NC(C1C2CC2CN1C(=O)C(CCSC)NC(C)=O)=O C1(C(N(C(CNC(C2CN(CC)C(=O)C2)=O)C)C)=O)CCc2ncnn2C1 CON1CCC(C(=O)NC(C)(C)CNC(=O)CCc2ccco2)CC1 C1(C(=O)NCC2C(NC(Cc3c(C)ocn3)=O)C2)CCC2CC2CC1 C(CO)(CCCCNC(=O)CCC1CCC(=O)N1)NC(Cc1c(C)ccs1)=O c1(CC)ccc(NC(C2CC(NC(c3cnncc3C)=O)C2(C)C)=O)c(C)c1 c1(C(=O)NC2CCCN(C(COCCCOC)=O)C2)cccn2cncc12 C1(CC)CN(C(c2csc(COC)n2)=O)CCN1C(c1cc(OC)nc(Cl)c1)=O CCC(CCOC)C(=O)NCC1CC1NC(c1cccc(NC)c1)=O C1(CC)(NC(C2CCCCN2C(=O)Cn2cccn2)=O)CCCCC1 CC1(C(=O)NC2CC(CCC(N)=O)C2)CC(O)CN1C(=O)Cc1ncccc1F Cc1cc(C(=O)NC(C)CNC(=O)C(C)OC2CCCC2)nn1-c1ccccn1 c1(C(=O)NCC2(CN(C)C(c3cnsc3)=O)CC2)cc2c(o1)CCCC2 CC(C)C(O)C(F)(F)C(=O)N(C)CC1CC(NC(=O)C(C)C2CC2)C1 C1(C)(NC(C(CNC(C=C(C)C(F)F)=O)CC2CCCC2)=O)CN2CCC1CC2 N1(C(CCc2ccc(CC(C)C)cc2)=O)CCC2(NC(C3CCC3)=O)CC2C1 N1(C(CCCCN(C)C)=O)CCC2(CC1)CC2C(=O)NC(CO)CCF C=CC(CC)CC(=O)NC(c1ccccc1)C(=O)NCc1nnn(C)n1 N#CC1CC(NC(=O)C=CCNC(=O)CCCC2CCCO2)C1 C#CCC(O)C(=O)NCCC(C)N(C(=O)CCOc1ccc(Br)cc1)C c1(CC(C(C)=O)OC(c2nc(Cl)sc2Br)=O)ccc(Br)cc1F c1(C(N2CC(NC(C(C)NC(C)=O)=O)C(C)C2)=O)c[nH]cc(Br)c1=O C(CC(O)C(F)F)NC(c1cc(CCNC(C2COCCO2)=O)on1)=O n1(CC(=O)N(CCC(C)NC(C2(C(C)C)CC2)=O)C)cnc(C(F)(F)F)c1 C1(C)(OC)CCCN(C(=O)COC23CCC2CN(C(=O)Cc2cn[nH]c2)C3)CC1 N1(C(C(C)(C)F)=O)CC2CCCC(C1)N2C(=O)CCC(=O)c1ccccc1 CC(O)CC(=O)NCC(C)(F)CNC(c1sccc1Cl)=O C1(COC)(NC(=O)CC2COCC2O)CCN(C(=O)C=CBr)CC1 C(C)(C(=O)N1CC(NC(=O)COCC)C1)SCC CCCC(CC)C(=O)NC1(CN(C)C(c2c[nH]nc2Br)=O)CC1 N1(C(C(F)OC)=O)CC2CCC1C(NC(=O)C=C(C)c1ccccc1Cl)C2 c1(C(CN(C(=O)Cc2cnoc2)CCO)O)cccc2ccccc12 C(C1COC(C)(C)O1)=CC(=O)NC.C1(NCC=CC(=O)OC(C)(C)C)CC(C(=O)N)C1 C1(NC(C(C)OC2CCCC2)=O)CCC2(CCN(C(c3cncc(Cl)c3)=O)C2)C1 C(=O)(C1=NOC2(CCC2)C1)NCC1CCC(C)N(C(C2CC2C(N)=O)=O)C1 N1(C(CC(COC)C)=O)CCC(C)(C)C(CNC(=O)CC2CC2)C1 CCCCC(C(=O)NC1CN(C(=O)Cc2ccc(CO)cc2)CC12CC2)C(C)C C12(C(=O)NCCCN(C(C)=O)C)CCC(NC(C3CC3C(F)F)=O)(CC1)C2 N1(C(C2CCN(C)C(=O)C2)=O)CC2CCOC2(CNC(=O)C(=O)NCC(F)F)C1 C12(NC(C(CC=CC)C)=O)CCOC(CNC(c3cc(C(N)=O)ccn3)=O)(C1)C2 c1(C(N2CC(NC(C(CC#C)O)=O)C3(C2)CC3)=O)cc2ccccc2[nH]1 CC1C(C)N(C(C2CCC3CC2CO3)=O)CCN1C(=O)Cc1cc(F)ccc1F Cc1cnc2scc(C(=O)NCC(C)(O)CNC(=O)CCn3cnnn3)c2c1 N1(C(Cn2c(C)ccn2)=O)CCCCCC1CNC(=O)C(c1ccc(Cl)s1)C N1(C(c2cc(-c3ccccc3)ns2)C(=O)NCCC#N)CC(O)C(O)C1 c1(C(N2CC(F)CC(NC(CN3CCC(OC)C3)=O)C2)=O)ccc(C#N)c(C)n1 Cc1cc(Br)cnc1C(=O)Nc1cccc(C(=O)OC(C)(C)C)c1 C1(C(=O)NCC(CCOC)(C)C)CC2(CC2)CN1C(=O)C(C1CCC1)OC N1(C(c2c(C)cco2)=O)CCC(C2CC2)(CNC(c2ncc(Cl)n2C)=O)C1 C(=O)(C(CCC(C)C)NC(c1cnn(CC)c1)=O)N(CC=C)CC C1(C2CC2)(CNC(c2n(C)c([N+](=O)[O-])cn2)=O)CCN(C(=O)COC(F)F)C1 c1(C(N(CCNC(c2conc2C(C)C)=O)CC)=O)cc(C2CC2)nc(Cl)c1 Cc1nc(C)c(CCC(=O)NCC2CCN2C(c2cccc(C)c2Cl)=O)c(O)n1 CCC(CC)C(C)C(=O)NC(C)C(C)(C)NC(=O)CN1CCC(O)CC1 O=C(CCCCC(F)F)NCC1CCCN1C(C1(c2ccccc2)CC1(F)F)=O c1(C(N(CC(C)NC(=O)CC2(CN(C)C)CCOCC2)C)=O)cc(=O)n(C)cn1 CC(C)(C)S(=O)(=O)CC(=O)N1CC2CCN(C(C3C=CCCC3)=O)C2C1 C(=O)(CC(F)(F)C(F)(F)F)NCCC1N(C(c2[nH]cc(CC)c2)=O)CCOC1 C12(COC)CN(C(c3cc(C)cs3)=O)C(CNC(C34CCCCC3C4)=O)(C1)C2 C1(C(N(C(CN(C(CCC=C(C)C)=O)C)C)C)=O)CCCOC1C C(=O)(C(F)CC(C)(C)C)NCCCCN(C)C(c1ccncc1F)=O c1(C(N(CC(C)N(C(c2n(C(CC)C)ncc2)=O)C)C)=O)ccc2c(c1)CCO2 c1(C(N2C(C)CCC(NC(c3cnc(OC)s3)=O)C2)=O)ccc(F)c(F)c1C C(CCCCNC(C1(NC(N)=O)CC1)=O)N(C(=O)CC1CCN(C)C1)C C1(CNC(c2c(C)noc2)=O)CN(C(c2coc(CO)c2)=O)CC1N(C)C C(=O)(C1CCOc2ccccc21)N(C)CCN(C(=O)C(C)(C)O)C N1(C(C(=O)NC(C)C)=O)CCC(NC(C23CCC(C2)C3)=O)C1(C)C C(C(C(C)C(C)C)NC(=O)CCNC(=O)C=CCl)NC(Cc1c(C)ccnc1)=O CCCCC(CC(=O)N1CCC1C(N)=O)NC(c1cccc(C)c1O)=O C12(CNC(CC3CC(=O)C3)=O)CN(C(c3cccc(O)n3)=O)CC1CS(=O)(=O)C2 c1(C(=O)NCC(CC(C)C)NC(CC2(OC)CCC2)=O)cc2cccc(C)c2s1 C1(NC(=O)CC2CC(C3CC3)C2)CCN(C(=O)C(F)C2CCCC2)C12CC2 C1(CNC(C(c2c(C)cccc2)(C)C)=O)CCC(C)(C)CN1C(=O)C(C)C1CC1 c1(C(=O)NC2(CO)CN(C(CCOCC#C)=O)C2)ccc2c(c1)nc(CO)n2C N1(C(C(C)CN(C)C)=O)CC2(CC(NC(c3cnccc3Br)=O)CO2)C1 C1(C(N(CC(C)NC(c2ncc(C)cc2C)=O)CC)=O)CCN(S(N)(=O)=O)CC1 N1(C(C2CN(C)C(=O)C2)=O)CCC2CN(C(c3ccnn3C3CCC3)=O)CCC12 C1(NC(c2nc(CCCC)sc2)=O)CN(c2nccc(C#N)n2)CCC1C C(=O)(CC(C(F)(F)F)P(C)(C)=O)NC1CN(C(c2c(CC)nc[nH]2)=O)CC1O CC1CC(=O)NN1C(=O)CC(CC(=O)Oc1ccc(Cl)c(Cl)c1)C=O c1(C(=O)N)cc(C)c(C)nc1O.Cc1cc(O)cc(C)c1.C1C(=O)NCC2C1C2 C1(NC(=O)NCC(Br)=C(C)CN(C)C)CCOC(c2cnn(C)c2)C1 n1(CCC(=O)OC)nnc2c1CCN(C1CC(n3cccnc3=O)C1)C2 C1(C(=O)NCC(COCC)C)COCCN1C(=O)COC1CCCC1 C1(C(=O)NC(C=C)C(F)(F)F)CC2(CC2)CN1C(c1cc[nH]c1CC)=O C1(CC)CCC(C)CN1C(C1(NC(c2cncn(C)c2=O)=O)CC1C)=O C1(CNC(c2c(C)nc(C3CC3)o2)=O)COCCN(C(c2cc(C(N)=O)cs2)=O)C1 c1(C(=O)NC2C(CC)N(C(=O)C(C)n3cncn3)CC2)cc(C)c(Cl)cn1 c1(C(=O)NC2CC(O)CN(C(=O)CN3CCCCC3)C2)cc2ccc(F)cc2s1 c1(C(=O)NCC(CC=C)NC(=O)COCC(=C)C)sc(C)cc1OC Cn1ncc(CCN(C(N2CCC(C3CC3)C2)=O)C2CC2)c1O Cc1nc(N(C)C)sc1CC(=O)NCC1CC1NC(=O)C(C)(C)c1cscn1 C(C(C(=O)N1CCCC1CC(C)(C)NC(=O)CCCF)NC(C)=O)OC c1(CN2CCC(CNC(c3ccc(Cl)cc3O)=O)C2)cc(Cl)ccc1[N+](=O)[O-] C1(CNC(C(C2CCOCC2)C)=O)CCCCN1C(=O)CN1CC2CC2C1 N1(C(c2ccc(C=C)cc2)=O)CCC2C(CCN2C(=O)CC(C)F)C1 C1(NC(C=Cc2cc(C)no2)=O)CCCN(C(c2cnnc(O)c2)=O)C1C C=CCC(F)(F)C(=O)N1CCC(N(C(=O)C(n2ccc(Br)n2)C)C)CC1 C(=O)(CC1=CCN(C)CC1)N1C(C(N2CCCC(C#C)(C)C2)=O)CC=CC1 c1(Cc2c(C)n(C)nc2)ccc(CN2CCOCC2)c(F)c1.C1(=O)C(=O)NN1 CCCC(C)(CCC)C(=O)NCC1CCCN1C(=O)C=Cc1cccc(Br)c1 C1(NC(CCCOCC)=O)CCC2(CC1)CC(NC(=O)CCN1CCCCC1)C2 CN1CCN2CCN(C(=O)NC3CCC(C#N)(c4ccncc4)CC3)CC2C1 C(C)(C(=O)NC)NC1(C)CNC(=O)C1CC.CC(C)COC(C)(C)C C1(C(=O)NCC2(F)CC(NC(=O)CC3CCOCC3)C2)CCC2C(CC1)C2(F)F N1(CC(=O)NC(C(C)(C)NC(C(C)N(C(C)=O)C)=O)C)CC(=O)N(C)C1=O C1(CNC(CCN(C(CC)CC)C)=O)C2CN(C(C3(CF)CC3)=O)CC12 Cc1c(C(=O)NC(C)CCNC(C2(Br)CC2)=O)cnn1C(C)(C)C CCCC(C(=O)NC(C1CCCCC1)CNC(c1cc(C(=O)OC)c[nH]1)=O)OC C12(CNC(C3C(CNC(C(C(C)C)SC)=O)C3)=O)CCCN1CCC2 c1(OCC)cc(C(=O)NC(C2CCCC2)CNC(C2CC2C2CC2)=O)[nH]n1 N1(C(C2(C(C)C)CC2)=O)CC(CNC(=O)CCCc2cccnc2)CC(C)(C)C1 N1(C(C(F)=C(C)C)=O)CC(F)CC1C(=O)NC(c1ncc(F)cn1)C c1(C(=O)NCC2N(C(C(CC)OC)=O)CCC2)cc(C)nn1C C(=O)(C(C(=O)OC)OC)NC(C1CC=CCC1)C(=O)NCC(=C)F c1(C(=O)NCC2(NC(c3cocn3)=O)C(C)CCCC2)cc2ccc(Cl)cn2c1 c1(C(=O)NCC(C(C)(C)C)NC(=O)CN2CCCC2)cc(S(N)(=O)=O)co1 c1(C(N2C(C(N(C)Cc3ncco3)=O)CC2C)=O)cc(O)cc(F)c1 C1(CNC(c2cc(C)no2)=O)CN(C(c2cscc2C(F)F)=O)CCC1(F)F N1(C(C=CCC)=O)CCCCC(NC(=O)C(c2ccc(C)cc2)C2CC2)CC1 C1(C(N(C(c2ccccc2)CNC(C2(OC(C)=O)CC2)=O)C)=O)CCC(=O)N1C C1(C(N2C3(c4nc(C)c(C)o4)CCC2CC3)=O)COC2(C1)CN(C(=O)C=C(C)C)C2 c1(OC(C)CNC(C2(CNC(c3cc(CC4CC4)on3)=O)CC2)=O)ccncc1 C#Cc1ccc(OCC(=O)NC2CC3C2CCN3C(=O)C(O)C(C)C)cc1 N1(C(CC2(C)CCCN2C(c2c(F)cccc2F)=O)=O)CC2CCC(C1)C(=O)O2 C1(NC(=O)COCc2cccc(Cl)c2)CC2CCC1N2C(c1ccon1)=O Cc1c2c(nn1C)CCC(N(C(=O)C(CNC(c1ccccc1)=O)N(C)C)C)C2 CCN=c1[nH]c(C)c(C(N2CC3CCC3(NC(c3ccns3)=O)C2)=O)s1 c1(N2CCN(C(CN(CC)CC)=O)CC2)oc(CC(C)C)nc1C#N CC1CCCC=C1C(=O)N1CCC2C(NC(=O)COC(C)(C)C(F)(F)F)C2C1 C1(NC(c2c(C)nc(CO)o2)=O)(CO)CCCN(C(c2cnco2)=O)C1 CC1CCN(CC(N2CCSCC2C(=O)NCCCC2CCOC2)=O)CC1 c1(C(N2CC(C)(C(=O)Nc3cncnc3)C2)=O)n[nH]c2ccccc12 c1(CN(c2ccc(Cl)cc2)C)nc(CC2CCC2)nn1-c1cccc(F)c1 c1(C(N2C(CNC(C=CCN(CC)CC)=O)CCC2)=O)cccc2nc(Cl)cn12 C1(CNC(C2C3CC4C(C3)C24)=O)CN(C(C2(OC)CC2)=O)CCN1C.c1(O)ccc(F)cc1 c1(CN2C(C(=O)NC3CC(c4ccccc4)C3)COCC2)ccc(F)c(F)c1 C(=O)(C(C)(C)CS(C)(=O)=O)NC(C(C)NC(c1cccc[n+]1[O-])=O)CO C(=O)(C1=CC(C)(C)C1)N(C1CC(NC(=O)CCc2ccccc2C#N)C1)C Cc1ccc(Br)c(Cl)c1C(=O)NC(CO)C(C)NC(C1CCCS1)=O C(=O)(CCCC(=O)NCC1CCCCC1NC(=O)CCC=CC)NCC=C C1(C(=O)NC(C(=O)NCCC2COCC2O)c2ccoc2)CCC2CC1CO2 c1(CC)noc(C)c1C(=O)NCC1CCCN1C(=O)CCC1CC1(Cl)Cl Cc1ccc(C(N2CCCC(C)(NC(C3CC(C)CO3)=O)C2)=O)c(C)c1 N1(C(C(CC#C)C)=O)CC2(CCN(C(c3ccc4cnccc4n3)=O)CC2)C1 c1(NC(C(C)NC(c2c(C(C)C)sc(Cl)n2)=O)C(C)C)cc(C(N)=O)nc(Cl)n1 N1(C(c2ccc(C#C)cn2)=O)CC2(CC(NC(=O)CC3C=CCCC3)CO2)C1 CCCCC(O)C(=O)NC1CCN(C(C2(c3ccc(C)cc3C)CC2)=O)CC1O S(=O)(=O)(c1cccc(N2CCC(N3CC(C)(C)C3)C2)n1)NCCSCC=C N1(C(C(CCOC)OC)=O)CCC(C(=O)NCC(N2CCOCC2)=O)CC1C C(CC(=O)N(c1ccccc1O)C)(C(C)C)NC(C(COC)(C)OC)=O N1(C(c2cn(C3CCOCC3)nn2)(C)C2CC2)CC(c2ccccc2)C(C)CC1C c1(C(N2CC(CNC(C3C(C)C3C)=O)OCCC2)=O)c[nH]c2cc(F)c(F)cc12 N1(C(c2c(C)nn(CCO)c2)C(=O)NCc2cccc(Cl)c2)CCNC(=O)CC1C n1(CC)cnc2c(N(CC(Cl)Cl)C)[nH]c(=NCCC3CN(C)C3)nc12 c1(OC)cc(O)ccc1-c1cn(C2CN(C(c3cc(F)cnc3Br)=O)C2)nn1 Cc1c(C(=O)N(CCCNC(=O)C(C2CC2)C2CC2)C)nn(C)c1C1CC1 Cc1cc(NC(C2(C)CC(NC(C3CC3(Cl)Cl)=O)C2)=O)cc(C)c1F N1(C(c2nc(OCC)oc2)=O)CC(C(=O)NCC2CCCC(C)(C)C2)C(C)(C)C1 c1(NC(CCN(C(c2csnn2)=O)CC)=O)ccc(Cl)nc1C C1(NC(C(C)CC2CCC2)=O)CC2CN(C(C3CC(C4CC4)=NO3)=O)CC2C1 CCC(CC(=O)NCC(O)CNC(c1csc(-c2ncccn2)n1)=O)C(F)F C(=O)(C(C)(C)S(C)(=O)=O)NC1(CC)CCCN(C(=O)C(C)CCN(C)C)C1 c1(CNC(c2n(C3CC(C(F)F)C3)nnn2)CCC2CC2)cc(Br)cc(Cl)c1F CN1CCCC(c2cccc(NCC(N3CCN(CCC(=O)O)CC3)=O)c2)C1 c1(C(N2CCCC(NC(CC)=O)C2)C)cccc2cccnc12 C1(C(C)(C)NC(CCSCC)=O)CCN(C(C2CSCC(=O)N2)=O)CC1 CC1CC(NC(=O)Cc2cnoc2)CCN1C(c1ccnn(C)c1=O)=O Cc1cc(C(=O)N(CC(C)N(C(=O)Cn2nc(C)cc2C)C)C)c2n[nH]cc2c1 c1(C(N(CCC(C)NC(=O)CC2CC=CCN2C)C)=O)cc2cccnc2s1 C1(C(=O)NC(CNC(=O)CC2CCCC(C)C2)C(C)C)(CC)CCNC1=O c1(OCC)ccccc1C=CC(=O)NC(C1CCCCC1)CO C1(NC(C2(OCC)CCC2)=O)CC2(NC(c3cn(C)nn3)=O)COC1C2 N1(C(CN(C)CC)=O)CC(NC(=O)CCOc2ccc(F)cc2)C2CC2C1 c1(C(=O)NCC(C2CC2)NC(C(C=C)(C)CC)=O)cc2nccn2c(O)n1 C1(C(N2CCN(C(c3ns[nH]c3=O)=O)C(CF)C2)=O)CCc2ncsc2C1 C1(NC(C(N)=O)=O)CC2CCC(C1)N2C(C1COC(=O)N1)=O CCCCCC(O)C(=O)NC1CCOC1C(=O)N(CCC)OC N1(C(C(C2CCCN(C)C2)(C)C)=O)CC2(CC(NC(=O)C=CC3CCCO3)C2)C1 CCC(CC)C(C(=O)NC1(CC=CC(=O)NCc2cc(C)ncn2)CCC1)OC C12(C(=O)NC(C3CN(Cc4ccc(C(C)(C)C)cc4)C3)C)CCC(C1)C(C)(C)O2 CC1CN(C(=O)CCN2CCCC2)CCCN1C(=O)C(C)n1ccnn1 C1(C(N(C)Cc2cc(C)no2)=O)COC2(C1)CN(C(C1CCNC1=O)=O)C2 C=CCCC(C)NC(=O)CCCc1ccccc1 c1(OC)cc(Br)c(C)cc1NC(=O)CC1CCN(CC2CC2C2CC2)C1 CC1=NNC(=O)C1CCC(N1CC=CC(NC(C2CC(F)(F)C2)=O)C1)=O C#CC1CCCCN1C(=O)C(C)(CO)NC(=O)CCc1cncnc1 CC1CN(S(=O)(=O)c2cccnc2NC(CF)CF)CC2(CCC2)O1 C(C(=O)O)(C(=O)NCCO)OC.N1(CCC(C)(C)C)CCSCC1C C=CCCCC(C(=O)NCC(CC)CC(C)C)NC(c1cc(F)ccc1C)=O N(C(=NCCCF)NCC1CCC(F)(F)C1)CC(c1ccccc1)(C)C N1(C(CCn2cc(CCN(C(C)=O)C(C)C)nn2)=O)CCc2scc(C)c2C1 c1(NCC(CCC)(C)C)nc(=NC2CN(CC)CC2C)[nH]c2c(C)nn(C)c12 C1(CNC(c2cncc(C)c2)=O)CC2CC(C1)N(C(=O)C(C)(F)F)C2 CC1CC(CNC(=O)C(C)(C2CC2)N(C(=O)C(C)C)C)=NO1 C(=O)(CCP(C)(C)=O)c1nsc(-c2cn(CC(C)N(C)C)nn2)c1Br CC1(C)CC(CO)(O)CN1C(=O)COCCCl.c1(CNC(=O)OC(C)(C)C)ccsn1 CC1(NC(=O)CCS(C)(=O)=O)CCCN(C(=O)Cn2cc[n+](C)c2)C1 C1(N)CCOC1C.C1(C2CN(C(C3CN(CC)C3)=O)C2)CCCN1C.C O=S1(=O)CCC2CNC(c3cc(-c4ccncc4Br)n[nH]3)CC12 C1(C(=O)NCCCC(CCC)NC(c2ccoc2CC)=O)CC2(CCCC2)CO1 c1(NC2C(C)C2)nnc(C(F)F)n1C N1(C(C2(C=C)CCC2)=O)CC2(CCC(CNC(=O)C(c3ccccc3)C)O2)C1 Cc1nc(O)ccc1C(=O)NCC1CC(C(N2CCC(C)(CO)CC2)=O)C1 c1(N(CCCNC(CCCn2ncc(C)c2)=O)C)nc(C(F)F)nc(=N)[nH]1 N1(C(c2c(CC)cco2)=O)CCCC(NC(c2cn(CC)cn2)=O)C(F)C1 C=CCC(CC=C)C(=O)NCC1(CO)CCCN(C(C2(O)CCCCC2)=O)C1 c1(COCC(=O)NCC2CC2NC(c2cncn2C2CC2)=O)ccccc1Cl CC1CCN(C(=O)CC2(O)CCCOC2)CCN1C(=O)CC1CCCOC1 N1(C(C2C(C)=CCS2)=O)C2CCCC1CN(C(c1ccc(F)cn1)=O)C2 C(CCCCC(=O)N1CCCC1C1CCN(C(=O)Cn2cc(CO)nn2)C1)OC c1(C(=O)NC(CC(C)NC(C2(S(C)(=O)=O)CCC2)=O)C)ccc2[nH]c(=N)[nH]c2c1 c1(CC)nc(C)c(CC(N2CC3C(CNC(C4(N(C)C)CC4)=O)C3C2)=O)c(C)n1 N#Cc1ccc(C(=O)NC2C3CC4C(C3)C24C(=O)NCCc2csnn2)cc1 N1(C(C2CN(C(C)C)C2)=O)CCOC(CC(=O)N)C1.N1(CCC2CC2)CC=CCC1 N1(C(C(C)=CC)=O)CCC2CCCC12CNC(C1(C)CSC1)=O C1(NC(C(CCC)N(C)C)=O)CC2(C1)CC(CNC(C1CC1C(N)=O)=O)C2 C1(NC(C2CC(=O)NCC2)=O)CN(C(c2c(Cl)cc(Br)cc2Cl)=O)CC(F)(F)C1 C(C(N=[N+]=[N-])C(=O)NCC(Cn1cc(-c2ccccc2Cl)nn1)OC)OCC N1(C(CN(CC)CC)=O)CC2(C1)SCCC2NC(=O)Cc1cnc2ncccn12 C#Cc1cc(C(=O)NCCC2CCCN2C(c2cscc2C(F)F)=O)ccc1C c1(C(Cc2ccccc2)=O)ccc2c(c1)C(C(=O)N1CCCCC1)CC2=O.CO C1(CNC(c2c(C)cncc2)=O)CC12CCN(C(C1CCCN1C)=O)CC2 C1(C(=O)NCC(C(CC)C)CO)CCN(C(=O)C(C)n2ccnn2)C(C)(C)C1 CCC(CNC(=O)C(c1cncc(F)c1)OC)(CC)NC(=O)Cc1scnc1C C12(C(=O)OC)CCCC(C1)N(C(c1ccccc1)CCc1ccccc1)C2 c1(CCC(=O)NC2CCC(C(=O)NCC(F)CO)C2)nc2ccccc2s1 C1(CC(=O)NC2CCCC(C)C2)OCC2CCN(C(c3ccc(Cl)nc3)C)CC12 c1(OC)ccnc(O)c1C(=O)NC1CC(C)(NC(C2CC=CC2)=O)C1 c1(C(N2CCC3(CNC(=O)C3)C2)C(=O)NC)cn2cc(Cl)ccc2n1 c1(NC(C2CCCN2Cc2sc(Cl)nc2Cl)C)ccc2c(c1)ncn2C C(=O)(CCCCCCN=[N+]=[N-])N1C(C(C)C)CN(C(=O)CCCC2CC2)CCC1 Cc1ccc(CC(=O)NC(C)C(C2CCCCC2)NC(c2cnn[nH]2)=O)cc1 N1(C(C(CC)CC2CC2)=O)CCC2(CC1)CN(C(=O)C(C)(C)C(F)F)CCO2 C1(C)(CC)CC(C(=O)N(C)CCOCCCNC(=O)CCCN(C)C)CCO1 N1(C(c2nc(C(C)OC)sc2)=O)CCN(C(C2CC23CCC3)=O)CC2(CC2)C1 C1(C(C)NC(c2c(C(=O)OC)coc2)=O)CCCN(C(c2cc(C)no2)=O)C1 C1(CNC(c2snc(Cl)c2Cl)=O)CC2CCC(C1)N2C(c1cccc(O)n1)=O CCCCC(O)CC(=O)NCC(O)CNC(=O)COc1ccc(Br)nc1 C(C(O)CCNC(c1ccnnc1)=O)NC(C(C)OCC(C)C)=O N1(C(=O)C2=CCCSC2)CCC2(CC1)CC(N=c1[nH]nc(O)s1)CCO2 c1(C(=O)NC2CCCC(NC(c3c(OC)scc3)=O)C2)cc2cccc(C)c2o1 N1(C(c2noc(C)c2C)=O)CCC2(CCCN(C(=O)C(C)NC=O)C2)C1 C1(NC(C(C)(C)Cc2cnn[nH]2)=O)CCCCN(C(c2cnco2)=O)C1 C(CNC(=O)CCCc1cnccn1)(C(C)(C)C)NC(CC1(C)CC1)=O N12CC3CC(C1)CN(C3)C(=O)CCNCC2=O.N12CCC(CC1)C2=O.CN.CO CCCCC(CC)CCC(=O)N(C1CCCN(C(C2CCCC2)=O)C1)CC1CC1 C(=O)(CC1=CCCCC1)NCC1N(C)CCN(C(C(C(C)C)NC)=O)C1 c1(C(N2C(C)CC(NC(c3cnns3)=O)C2)=O)c[nH]c2cc(O)ccc12 C(=O)(CCC(C)CC)N(CC1CCN(C(C2CCC(CC)O2)=O)CC1)CC c1(CNC(=NCCC=C)NC2(C)CN(C(=O)OC)C2)coc2c(C)cccc12 Cn1cc(-c2ccoc2C(=O)NCC(O)CNC(=O)C(F)C2CC2)cn1 CC(C)CCCCC(=O)NC1COCC1NC(=O)CN1CCCCCC1 CCCC(F)C(=O)N(C1CCCCCC1)CCNC(C1CCCC1)=O c1(OCC)nccc(C)c1C(=O)NCC(O)CNC(c1ccc(CC)cn1)=O c1(NC(=O)CCC=CBr)ccc2cc[nH]c2c1.C12CC(F)(C1)CNC2=O C=CCC(C)(C)C(=O)N1CCC(CN(C)C(c2occc(=O)c2OC)=O)C1 c1(OC)cc(OC)cc(C(=O)NC2(C)CCN(C(=O)CCC(C)C)C2)c1 c1(OC)ccccc1CC(=O)NC1CCCN(C(=O)C(C)(C)C2CCCC2)C1 CCC(C(=O)N1CC(O)(CC)C1)N(C(=O)CCc1nccn1CC)C C=CCC(CC(=O)N1CC2(CC(O)C2)C1)NC(c1ccc(C)nc1O)=O CC(C)CC(C)C(=O)N1CCC(C(=O)NCCCSCC2CC2)O1 C#Cc1ccc(C(=O)NC2CCN(C(C3CC(=C(F)F)C3)=O)CC2O)nc1 Cc1cc(C(=O)NCCCN(C(=O)CC2CCCC(C)(C)O2)C)cc2c1CCC2 C=CC(CC)CC(=O)NC1CCOC1C(=O)NC1(CC=C)CCOC1 C1(C(=O)NC2C(NC(CCc3ccn(C)n3)=O)C2)CC(c2cccc(F)c2)=NO1 c1(CNC(C2(OC)CN(c3ccnc(C)n3)C2)=O)c(Cl)sc2nnsc12 c1(NCC2N(C(C3C(OC)CCC3)=O)CCCC2)cc(C(C)C)nc2ncnn12 N1(C(C)C)CCC(C(N2CC(NC(C3CCCCC3O)=O)CC2CO)=O)CC1 N1(C(C=CC(c2ccc(CO)s2)=O)=O)CCC(C(=O)NC2(CO)CCCC2)CC1 CC1c2nccn2CCN1C(=O)C(CC(F)F)NC(c1cc(F)cnc1O)=O C12(NC(C3CN(C)C(=O)N3)=O)CCC(NC(C3CCCC(C)(C)O3)=O)(CC1)C2 c1(C(N2CC3CC3(C(=O)Nc3cncc(Cl)n3)C2)=O)cc2cc[nH]c2cc1Cl CCC(CC)(CC)C(=O)N1CCC(C)N(C(c2noc3c2CCCC3)=O)CC1 C1(NCC(CC#N)O)CC2CC1CC21CC1 N#Cc1cc(F)ccc1CN1CC2CC(C1)N2C(=O)Cc1ccc(Cl)s1 Cc1ccc(C(C)C)c(C(=O)NCC(C)(C2CC2)NC(=O)CC2CCC(C)O2)c1 Cc1ccc(NC(c2ocnc2C2CC2)=O)cc1NC(=O)CN(C1CCC1)C Cc1c(N)ccc(C(N2CC3(C2)CN(C(=O)C(c2cncnc2)C)C3)=O)c1C N1(C(c2c(F)ccc(OC)c2)=O)CCC2(CCCN2C(=O)CSCC(N)=O)C1 C1(CN(C(=O)CC2CC2)C)CCCCN1C(C1CCN(C)C1c1ccccc1)=O c1(NC(C(C)(C)OCC)c2nnnn2Cc2ccncc2)ccc(C)c(C)c1 C1(CNC(CCOCC)=O)C2CC1N(C(C1CC(OC)C1)=O)C2 c1(C(N2C(C)CN(C(c3cc(Cl)ncc3Cl)=O)CC2)=O)c[nH]c2ccccc12 c1(NCC(C2CC2)NC(C2(CC#C)CCCCO2)=O)ncc(Cl)cc1[N+](=O)[O-] C1(C(=O)NC(CCNC(Cc2c(CC)con2)=O)C)CCC(C)(C)O1 C1(NC(C(C)S)=O)CN(C(C2CCCC(C)(C)C2)=O)CC12CC2 C(C1c2ccccc2CCN1C(c1ccc(C(N)=O)c(Cl)c1)=O)NC(CCC)=O N1(C(C=Cc2cncc(C)c2)=O)CCC(C)N(C(C2CCCCS2)=O)CC1 N1(C(c2nn(CC)c(C)c2)=O)CCC(F)C(NCc2ccc(C(C)(F)F)cc2)C1 S(=O)(=O)(C1Cc2ccccc2C1C)N1CCC(CS(CC)(=O)=O)CC1 Cc1cc(C(=O)NC2CCC(CCC(=O)N3CC(CC(C)C)C3)C2)cnc1O N1(C(=O)NC(CCC)C2CC2)CCC(C)(c2cccc(C(F)(F)F)c2)C1 C(=O)(C#CC(C)(C)C)NCC(C)(CNC(=O)C(C1CCCC1)OC)OC C1(C(=O)Nc2cccc(CCC(=O)NC)c2)CC12CC(C)(C)Oc1ccccc12 C1(c2c(SC)c(F)ccc2)NC(=O)N(C)C(C2CCc3c(Cl)cccc32)=C1C C(=O)(CCC(F)(F)C(F)F)N(CC(CNC(c1occ(C)c1)=O)O)C CC1(C(=O)NCC2CC3(CC3)CN2C(=O)CCn2cccc2)CC2(CCC2)C1 c1(SCC(=O)N(CCCNC(=O)C2=C(Cl)CC2)C)ccc2c(c1)CCCC2 C12(C(=O)NCCC3C(C)CCC3)CC(CO)(CN1C(C1CCCO1)=O)C2 C#CCCN=c1scc(-c2cccc(C=C)c2)n1CC1CCN(CC)C1 Cc1cc(I)c(C(N2CCCOC(C(=O)O)C2)=O)cc1C c1(OC)ccnc(Br)c1NC(c1cncc(-c2ccnn2CC2CCOC2)n1)=O Cc1c(C(=O)N(C)CCNC(C2CC2(Cl)Cl)=O)c(C)n2ccncc12 C(=O)(CC(C)(C)N(C)C)NCCC1CCN(C(CC2(NC(C)=O)CC2)=O)C1 C1(C(=O)NCC2(NC(C(F)=CCC)=O)CCCCC2)CC2CCC(C1)S2(=O)=O c1(OC)ccccc1CC(C)CCN1CCC(COC(F)F)C1 C1(NC(C2CN(C)C2)=O)COC2(CCN(C(=O)Cc3cc(Br)ccc3Cl)CC2)C1 C#CC1(NC(=O)C(CC(=C)C)NC(=O)CCNC(C)=O)CCC(C)(C)C1 CC(C)C(CC(=O)OC(CC(N1CCN(C)C(=O)C1)=O)=O)c1cccc(F)c1 N1(C(c2c(C)nc(O)[nH]2)=O)CCN(C(=O)CC2(C)CC2)C(C)C1C Cc1ccc(Cn2ccnc2CCOC(C)C)nc1.C12CCC(CC1)NC(=O)C2 C1(C(=O)NCCn2cccn2)(CF)CCN(C(c2ccc(CO)o2)=O)C1 C1(NC(CN(S(C)(=O)=O)C)=O)CCC(CNC(C2CCCC2(C)C)=O)CC1 c1(C(=O)OC)cccc2nc(OCCC(N3CCCC3C3CCCNC3)=O)nn12 C1(CC(=O)NC(CCN(C)C)(C)C)CC(NC(c2cnn(C)c2Cl)=O)C1(C)C C1CC(C)(C)C(=O)NC(C)CN1C.C1(N)CN(C(C2CC2(F)F)=O)C1.CS C1(CNC(c2c(COC)scc2)=O)CCN(C(=O)CN2CCCC2)C12CCC2 Cc1ncc(C(=O)NCC2C=CCN2C(=O)CC2CC(F)(F)C2)c(O)n1 c1(C(N2CC(NC(CCCC=C)=O)CC2(C)CC)=O)cc2c(o1)CCCC2 c1(C(N(C2CCCCN(C(=O)C3=COCC3)C2)C)=O)ccc2c(c1)CC(=O)NC2 N1(C(Cc2cc(OC)ncc2)=O)CCCCC(NC(C2CC2(F)F)=O)C1 C(=O)(CCCCCNC(c1nccnc1C)=O)NCc1n(CC)nnn1 C1(C(N2C(C)CC(NC(=O)CC(C)(C)c3cccs3)C2)=O)COCCN1C=O c1(C(N2CCC(CNC(c3ccccc3)=O)C2)C(=O)NC)nccc(Br)c1C N1(c2c(C)cnc(NC(c3cc(C(F)(F)F)cs3)=O)n2)CC2(CCCN2OC)C1 C(=O)(C(CC(F)F)N(C(=O)CC1OCCO1)C)N1CCC(CN(C)C)CC1 C1(CCNC(CCC2(C)CC2)=O)CC2(CCC2)C1.C(C)(C)(CC1CCCC1)OCC(=O)O CC(=O)CCCCC(=O)N1CCC(NC(=O)CC2CCC(=O)N2)C(CO)C1 N1(C(C2C(CN(C)C)C2)=O)CCC(O)(CN(C(=O)CCc2ccnc(Cl)c2)C)C1 C1(CC)CN(C(C)=O)CC1NC(c1nccn1C)=O C1(CNC(=O)C=CCF)CN(C(=O)C=CC2CCCCCC2)CC12CCC2 C(=O)(C1=C2CCCN=C2NN1)NCC1CN(C(C2(C)CN(C)C(=O)CC2)=O)C1 CCCC(CCCNC(c1ccc(SCC(N)=O)cc1)=O)NC(=O)C(F)(F)CO C1(NC(C2CCC(N(C)C(C3COC(=O)C3)=O)CC2)=O)CCCC1C1CC1 c1(CNC(C(C)N(C(C)=O)C)=O)ccc(CNC(=O)CC2CC23CC3)s1 C1(C(=O)NC2(C(=O)NC(c3nn(C)cc3O)C)CCSC2)CCC2CC1CO2 C12(CNC(C=CC)=O)CCC1CN(C(=O)C(F)(F)Sc1cnn(C)c1)C2 C(=O)(C#CC1(C)CCCO1)N(C)CC1CCCN1C(=O)COCCCF C1(C2CCOCC2)(NC(CCCCN(C(=O)CCn2cccc2)C)=O)CC1 C(=O)(C(C)(CC)CC)N(C(CC)CC(=O)NCC1CCOCC1)C c1(C(=O)NC(CC)(CNC(c2ccnn2C)=O)CC)cccc(Cl)c1Cl c1(NC(c2nc(C)c(C)s2)c2n(CC)nnn2)ccc(F)cc1 C(C(C(=O)N(C)CCOCCNC(c1coc(=O)[nH]1)=O)C(C)(C)C)OCC=C N1(C(C=CC(C)(C)SC)=O)CCCC1C1(O)CN(C(c2n[nH]cc2Cl)=O)C1 c1(C(=O)NC(C)(CO)C(=O)NCC2COCCO2)cc2ccccn2n1 C1(CNC(CC2CCN(C)C2)=O)CCN(C(=O)CC#N)C1(C)C C(C(CC(F)(F)F)NC(C1CCC1OCC)=O)NC(CNC(=O)OCC=C)=O CCCCC(CC)CCC(=O)NC1(C)CC(NC(=O)C(C)Sc2nc(C)cs2)C1 CCCCCC(CC)C(=O)NC(C)CNC(c1c(F)cccc1[N+](=O)[O-])=O N1(CCC)CCN(Cc2cnc(OCC)nc2)CC1.c12cccc(c1)NC(=O)N2.OCC CC(C)(CC=CC(=O)N(CCC(=O)NCC(F)F)C1CC1)NC(=O)CC1CCC1 N1(C(CCC=C)=O)Cc2ccnn2CC(NC(c2cc(C)ncn2)=O)C1 CC1(C)C(C(N2CCCC(CCCCNC(c3ccnnc3O)=O)C2)=O)C1(F)F CCC1=C(C(=O)NCC(c2ccc(F)cc2)C(=O)OC)SCCO1 Cc1cnc(N2CC(CO)(NC(C3CCC4CCCCN34)=O)C2)nc1S(C)(=O)=O c1(C(N2CC(N(C(c3ccc(C(C)=O)o3)=O)C)C2)=O)cc2ccccn2n1 C1(C(N2CC(NC(C(COC)C)=O)C(C)C2)=O)CCOC(C)(C)C1 C1(NC(CCC(=O)NCCC)=O)COC2(CCCN(C(C3(COC)CC3)=O)C2)C1 N1(C(CC2(C)CC(F)(F)C2)=O)CCN(C(=O)C(C2CCCCC2)F)C(CCO)C1 c1(OC)c(C(=O)NCC#CCNC(=O)CC2CCC(=O)NC2)c(C)nn1C N1(C(C=CCOC)=O)CC(NC(=O)C(O)Cc2cnn(C)c2)C(F)C1 c1(OC)ccc(Cl)c(C(=O)NCC(C(C)C)NC(=O)C(C)(C)C#N)c1F O=C1CCCC(C(=O)NC2(CNC(=O)CCc3cccnc3)COC2)N1 c1(C(=O)OC(C(c2ccc(CNC(C)=O)s2)=O)C)noc2c1CC(F)(F)CC2 c1(C(=O)NC(C2CCN(C(CCOC(C)C)=O)C2)C)ccc(S(C)(=O)=O)s1 C1(N(C(=O)CCc2nc[nH]n2)C)CCC(NC(C2CCC2C(N)=O)=O)CC1 C12(NC(CCC=C=C)=O)CCOCC1CN(C(c1ccncc1Br)=O)C2 C(C(C(=O)N1CCOC2CC12)C(C)(C)C)NC(CC1(N(C)C)CC1)=O C#CC1CC2CCC1N(C(N1CCC(c3cccnn3)CC1)=O)C2 C(=O)(C(C)(O)CC)NCCC(=C)CNC(c1cocn1)=O CC1(C)CCCC2(CCN2C(=O)NC2CCC3(CC3)C2)C1 Cc1ncc2n1CC(C(=O)NCC(C)(C)CNC(=O)CC1CCN(C)CC1)CC2 c1(C(N2CCN(C(CC(C)(C)F)=O)C(CS(C)(=O)=O)C2)=O)cccc2cncn12 c1(C(N2CC(NC(CC3C(C)=NNC3=O)=O)(CO)C2)=O)ccc([N+](=O)[O-])cc1F C(=O)(CCCC(=O)NC1(CCO)CN(C(C2CCN(C)C2=O)=O)C1)NC CCC(CC)CC(F)C(=O)NCCC1CCN(C(=O)CCc2nccs2)CC1 C1(C(N2CCC(SC)CC2)=O)CC2(CCN(C(=O)C(C)(C)C(C)SC)C2)C1 N1(C(CC)C)CCN(C(=O)CNC(=O)CNC(C2CC2c2ccnn2C)=O)CC1 C(=O)(CC(=O)N(CC(O)CNC(C1CC1CC(C)(C)C)=O)C)OCC c1(C(=O)NCCC23CCC2CN(C(=O)C=CC2CC2)C3)cnc2[nH]ncc2c1 C1(C(=O)NCC(CC)NC(c2cncc(NC)c2)=O)CCC2(CC1)CNC(=O)C2 Cc1cc(O)c(C(=O)NC(C(C)NC(=O)COCCF)C(C)C)cc1Br Fc1cccc(-c2cncc(-c3cn(CSc4cocn4)nn3)c2)c1F c1(CN2CCC(O)(C(N3CCN(CCOC)CC3)=O)CC2)ccc2n[nH]cc2c1 c1(NC(C2CCC(CNC(CN(C)CC)=O)CC2)=O)ncsc1S(N)(=O)=O c1(OC)c(F)ccc(Br)c1C(=O)OCC(c1ccc(F)c(F)c1)N C123CCCN(C1C2)C3=O.c1(NC(=O)CC2CCC2)ccccc1C(F)(F)F C1(NC(CC2CC(NC(C(C)OC)=O)C2)=O)CC(=O)N(C(C)C)C1 N1(C(c2c(C)[nH][nH]c2=N)=O)CCCC2CN(C(=O)CC34CCCC3C4)CCC12 C1(C(C)C)COC(C)(C)CN1C(=O)NC1CC1.c12cc-1n(C1CC3CCC1C3)n2 c1(C(=O)NC(C(c2ccccc2)NC(COCCC#C)=O)C)coc2c1CSC2 C(=O)(CCCC(C)=O)NCC1CC(NC(C(CC)Oc2ccccc2F)=O)C1 c1(C(N2CCC(CC=C)(NC(c3cccn3C)=O)C2)=O)cccc(C)c1N C(=O)(C1CCCc2ccnn21)NC(C(C)NC(C1(CCC)CC1)=O)CO C(CCC(C)(C)C(=O)NCCC(=O)NO)NC(C1CCC(C)O1)=O C(=O)(C(C)(C)C(=O)N1CCN(C(c2ccc(C(F)(F)F)o2)=O)C(C)C1)NC c1(C(=O)OC)csc(C(c2nnnn2-c2ccccc2)NC(C)CCO)c1 N1(C(c2c(CC)nn(C)c2)=O)CC2(CCC2)CC1C(=O)NCc1c[nH]nc1CC c1(C(=O)NCC(CC(C)C)NC(c2ccnc(C#N)c2)=O)cccc(F)c1F c1(C(=O)NC(CCC)CO)csc(=NCc2ccc(Cl)nc2)[nH]1 C1(C(=O)NC2C3CC2N(C(=O)C(=C2CCCCC2)F)C3)CN2CCN1CC2 CCC(C(=O)N(C)CC1(O)CCN(C(c2ccc(C)c(O)n2)=O)C1)C(C)C S(=O)(=O)(c1ccc(C(=O)NCCc2ccc(O)cc2)cc1)NC1C(C)CCCC1 N1(C(CC(COC)NC(=O)Cn2ccccc2=O)=O)CC2(C1)NC(=O)NC2=O N1(C(C2C(C(=O)Nc3ccc(-n4cncn4)cc3)C2)=O)Cc2ccccc2C1 c1(CC(=O)NCC2CCN(C(=O)COCC3(F)CC3)C2)ccnc(F)c1F c1(C(N2C(CC3C(Cn4cc(CN)nn4)C3(F)F)CC2)=O)nccc2cc[nH]c12 c1(C(N(CC=CC(=O)NC(C)Cc2cnn(C)c2)C)=O)ncn2c1CCC2 C(=O)(C(CC(F)F)C1(NC(=O)N(C2CCC3(CC2)CC3)C)CCC1)OCC O=S(=O)(c1cc(F)cc2c1CCC2)N1CCC(n2nnnc2C(F)(F)F)CC1 C1(C(=O)NCC(CNC(C(CC(C)C)N(C)C)=O)C)CC2C=CC1C21CC1 c1(OC)ccc(Br)c(CC(=O)NCCN(C)C(c2ccc(F)c(Cl)c2)=O)c1 c1(C(=O)NC2CC(CNC(C(C3CCC(=O)N3)C)=O)C2)cc2ccc(O)nc2s1 c1(CC)ccc(CCC(=O)NC2CCCC2NC(=O)CCc2csc(C)n2)cc1 c1(OC(C2(c3ccc(Br)cn3)CCC2)=O)ccc2[nH]ccc2n1 c1(OC)ccccc1C=CC(=O)NC1CN(C(c2n[nH]cc2Cl)=O)CC1C N1(C(CC2C(C)(C)C(O)C2)=O)CCCC(N(C)C)CC1.C12CC(C1)OCC(=O)N2 N1(C(c2ncc(C3CC3)cc2F)=O)CCN(C(C2CCC2CF)=O)C2COCC12 C=CCCC(C(=O)NC(C)CCCCCO)NC(C1CC(O)C(F)C1)=O N1(C(=O)CCN2CCC2)CCCC(C2CCN(c3ncnc4cccnc34)C2)C1 Cc1c(Nc2ccccc2C(C)(C)C)nc[nH]c1=NCCSCCCF C1(N(C(C(=O)OC)COC(F)(F)F)C)(OC)CCCC(C)(C)C1 Nc1sc2c(c1C(=O)NCCC1CCN(C(C3(Cl)CC3(F)F)=O)C1)CCC2 c1(C(C(=O)NCc2nocc2CC)NC(CCSCCC)=O)c(C)cccc1Br CC1CN(C(c2sccc2CO)=O)CC(CCNC(C2CC(=O)C2)=O)O1 CCC(C)CC(C(=O)NCC12CCCN1CCC2)NC(=O)CCC=C(C)C c1(NC(CNC(C2CCCO2)CC)=O)cn2ccccc2n1 C1(C(=O)NCCNC(=O)NC)CCN(C(C2CCCOCC2)=O)C1C C(CC(C)C)(C(=O)N1CCC2(CC2NC(=O)CCc2nc(O)n[nH]2)C1)NC(C)=O c1(C(=O)NCCC(CNC(c2n(CC)ccn2)=O)(C)C)c(O)nnc(C)c1C c1(SC)cccc(C(=O)NC2CCN(C(=O)CCc3cnn(C)n3)CC2C)c1Cl N1(C(c2c(OC)oc(C)n2)=O)CCCCCC(NC(C2CC(C)CCO2)=O)C1 c1(C(=O)NC23CC(CNC(=O)C=Cc4ccccc4)(C2)C3)ccc2nonc2c1 N1(C(c2[nH]c3cc(C)oc3c2)=O)CCCC2C1CCCN2C(=O)CC1CCC1 C(=O)(C1=CCCCC1C)NCCC1CC(NC(c2cc(C)n(C(C)C)c2)=O)C1 c1(CC(=O)NCCC2CCCN(C(C(C)c3cccs3)=O)C2)c(F)cccc1Cl C1(N(C(C(C=C=C)C)=O)Cc2ccccc2)CN(Cc2cc(Cl)n(C)n2)CC1(C)C c1(C(N2CCC3C(NC(C4C(CC)CCC4)=O)C32)=O)ccc2sc(C)nc2c1 N1(C(C)=O)CCCC12CCN(C(=O)C=Cc1cccc(C)c1)CC2 c1(-c2c(OCOC)cccc2)ncn2c1CN(C(C1CCCN1C)=O)CC2 Cc1nc(C)c(C(N2CC(CNC(c3cc[nH]c3C3CCCC3)=O)CC2C)=O)o1 c1(C(C)=O)c(Cl)nc[nH]c1=NCC1(NC(C2CC2(C)C(C)C)=O)CCCC1 Cc1ccc(C)c(C(N2CCCCC2CCNC(C2(C(=O)N(C)C)CC2)=O)=O)c1 C1(NC(c2ccc(OCF)cc2)=O)C2CC1CN(C(c1ccc(F)c(O)c1)=O)C2 c1(CNC(C(C)OCC(C)C)=O)cccc(C(=O)NCCC(O)C2CC2)n1 N1(C(C(N2C(C)(CNC(=O)OC)CCC2)=O)CC2CC2)C(=O)c2ccccc2C1=O Cn1cc(Br)c(C(=O)NCC(C)(CO)NC(=O)CCCC2CCC2)cc1=O C1(CC)CCN(C(c2ncccc2O)=O)C(C(=O)NCC(C)(C)C(F)F)C1 c1(C(=O)NCCCNC(=O)CCc2ccco2)cn(C2CCC2)nn1 N1(C(C2CC(O)(CC#C)C2)=O)CCC(C2CC2)C1C(=O)NCc1csc(C)c1 c1(OC)cc(SC)c(-c2ccccc2)cc1OC(=O)Cn1cc(CCCCO)nn1 C1(C(C)NC(c2cn(CCC)nc2)=O)CCCCN1C(C1CN(C2COC2)C1)=O N1(C(C2CCC(C(C)C)CC2)=O)CCN(C(C2(c3ccno3)CC2)=O)CC1CF C(c1cncc(C)c1)=CC(=O)N(C)CC1C2CN(C(CCC(=C)Cl)=O)CC21 N1(C(C2CC(C)(C)OCC2)=O)CC2CCN(C(=O)COC(F)(F)F)CC2C1 c1(-c2onc(NC(C(CCCCC)O)=O)n2)noc2cc(OC)ccc12 c1(N(CCCNC(c2c(C(C)C)nn(C)c2)=O)C(C)C)c[n+]([O-])ccc1[N+](=O)[O-] N1(C(CCN(C(C)C)C)=O)CCC2CN(C(=O)Cn3ccnc3C(C)C)CC2C1 Cc1nc2nccc(N3CCC(NC(=O)CC=CC(C)(C)C)C(CO)CC3)n2n1 C1(C(=O)NCc2ccc(C(NOCCOCC)=O)o2)CCC(F)CC1 c1(C(=O)NC(CCCC)CNC(C2CNC(=O)N2C)=O)cnc2c[nH]nc2c1 C(C(COC)C(=O)NCc1nnn(C)c1C(=O)NCC(N1CC=CC1)=O)OC C(=O)(CS(=O)(=O)CC(F)(F)F)N1CCN(C(C2CCCC(=O)O2)=O)C(CO)C1 Cc1cnc(C=CC(=O)NC2(CO)CN(C(=O)CCC3CCCN(C)C3)C2)[nH]1 CCC(CC)C(=O)NC1(C)CC(NC(c2cccc(N)c2)=O)C1 Cc1c(N)ccc(C(=O)N(C)CCOCCNC(C2CC23CCCCC3)=O)c1F C(C1=CCN(C)CC1)NC(C1(CNC(CC2CCC(C)C2)=O)CC1)=O c1(C(=O)NC2C(NC(C(C)OCCOCC)=O)C2)cn(C)c(C)cc1=O C(=O)(CCCC(C)NC(C1(C)CCCC1O)=O)N1CC(O)(C(C)C)C1 C1(CNC(C(CC)C)=O)CCCCN1C(c1ccc(OC(F)(F)F)cn1)=O S(=O)(=O)(CCC(=O)Nc1nccc(OC)n1)NCCc1ccc(C(=O)OC)cc1 C1(C(=O)NC2CC(N(C)C(c3ccc(COC)nc3)=O)C2)CC(=O)OC1(C)C C(=O)(C1(C)CCn2ccnc21)NCC(C)CN(C)C(c1ccc(=N)[nH]n1)=O c1(N(C)C)cc(C(=O)NC(c2ccccc2F)Cc2ccccc2Cl)cc(Cl)n1 c1(CCNC(C2(OC)CCCCCC2)=O)c(C)oc2cc(O)ccc12 N1(C(CC(C(=O)OCC)(C)C)=O)CCCC2CN(C(C3CC(C)(O)C3)=O)CCC12 c1(OC)ccc(-n2nnnc2C(c2ncc[nH]2)NC2CCCC2C#N)c(C)c1 C(C)(CO)(C(=O)N1CC(C#N)C1)NC(c1c(C)scc1)=O CCC(C)(COC)C(=O)N(CC(C)NC(=O)COCc1cccc(C)c1)C c1(CN2CC(CNC(C=CSC)=O)N(C)CC2)ncc2ccccn12 N1(C(C2(C)CCCC2O)=O)CC2CCC1C(C(N1CCOC(C3CC3)C1)=O)C2 Cc1ccc(C(CCO)NCC(=O)Nc2ccc(CNC(N)=O)cc2)cc1 c1(C(CNC(=O)C(C)Cc2ccccc2)NC(CC(C)O)=O)ccc(F)cc1F C1(NC(CCOCCN(C)C)=O)C=CC(CNC(c2coc(Cl)c2)=O)C1 N1(C(C(Cc2cc[nH]n2)NC(C(C=C)(C)CC)=O)=O)CCC2(CNC(=O)N2)C1 Cc1nc(NCC(N2CCOCC2C)C)cc(=NCc2c(Br)nnn2C)[nH]1 C1(C(N(C(COC)C(=O)OC(C)(C)C)C)=O)CCCC(CC(=O)OC)C1 N1(C(C(C#C)(C)C)=O)CC2CS(=O)(=O)CC2(CNC(c2nccnc2N)=O)C1 N1(C(c2ccc(OCC)cc2C)C(=O)NC2CCOC2)CC2(CCC2)OCC1C C1(C)(C(N2CCC(C(CNC(c3ncc(C)nc3)=O)F)CC2)=O)CCCS1(=O)=O c1(OC)nc(=NC2CCCCC2CNC(=O)Cc2ccc(F)cc2)nc(OC)[nH]1 N1(C(CC(CCC)(C)O)=O)CC2CCCN(C(=O)C=Cc3ccnn3C)C2C1 C1(C(N2C(C)C(O)CC2)=O)C2CC(O)C(C2)N1C(c1ccc2cncn2c1)=O N1(C(c2ccc(Cl)c(Cl)c2)=O)CCC2(CCN(C(c3ccc(Cl)o3)=O)C2)C1 CC(C)(C)CC(C)(C)C(=O)NCC1COCCN1C(c1cnc2c[nH]nc2c1)=O C1(C(N2CC(CCCCNC(c3n(CC)ncn3)=O)C2)=O)C2CCC(C2)C1(C)C S(=O)(=O)(c1c(F)cccc1F)NC(=O)COc1cccnc1 C1(CNC(c2nocc2Cl)=O)CN(C(C2CCCC2)=O)CCO1 C1(C(N(CCCNC(c2ccc(C)s2)=O)CC)=O)CCC2(CCCO2)CC1 C1(NC(Cc2c(C)ccnc2)=O)CC2(CCN(C(=O)C=CCF)CC2)C1 C(=O)(CCC(C)(F)F)N(C)CC1N(C(c2cc(C(C)=O)on2)=O)CC(F)C1 C(=O)(C1=CCOCC1)OC(C1CN(c2cccc(NC(=O)OCC)c2)C(=O)C1)C c1(CC)cc(OC)ccc1C(N1CCCCC1CCN(C)C(C1CC1C)=O)=O CC1CN(C(c2cnn(CCNC(=O)COCCF)c2)=O)CC(CCN(C)C)O1 S(=O)(=O)(c1ccc(Cl)cc1)N1C(NC(C(=O)OCC)Cc2ccsc2)CCCC1 CC1C(NC(c2cncc(F)n2)=O)CCCN1C(c1cc(Cl)nc(=N)[nH]1)=O c1(NC(CC2(C=C)CN(C(=O)CC3CCCC(C)C3)C2)=O)cn(C)nc1C#N C1(CC)CN(C(C2C(C)OC(C)C2C)=O)CCC1N=c1[nH]c2ccc(Cl)cc2s1 N1(c2ncn(C)n2)CCC(F)(c2cn(C3CCNC3=O)nn2)CC1 c1(C(CNC(c2nc(C(=O)OCC)oc2)=O)C)nnc(C)n1C c1(C(=O)NCC(CNC(C(C)(C)C2CCCCC2)=O)(C)O)ccn2cccc2c1 N1(C(c2ncn(C(C)(C)C)n2)=O)CC2CCCC(C1)N2CCOCC1CC1 c1(C(c2nnnn2CCC2CC2)NCCNC2(C)CC(=C)C2)cc(C)oc1C C1(O)(C(=O)NC2CCN(C(C3(CO)CCCCC3)=O)C2)CCCOC1.C1CCC1 CC1CN(C(=O)CSCCC#N)CCC1NC(=O)CCN1CCNC(=O)C1 C12(NC(C(CN(CC)CC)F)=O)CCCN(c3ncnc(Cl)c3F)CC1C2 C(=O)(CCC(F)(F)F)N(CCOCCC(N1CCCC(CCC#C)C1)=O)C C(=O)(CCCN=C(NCC(F)F)NC1CCN(c2ccccn2)C1)NC C(=O)(CS(=O)(=O)C12CC(C1)C2)NCCC1N(C(C(C)OCC(C)C)=O)CCOC1 C12(C(=O)NCC3(C(N4CC(c5nncs5)C4)=O)CC(=C)C3)CCCN(CC1)C2 C(=O)(C1=CCC(F)(F)CC1)NCC1N(C(c2c(CC)cc(N)cc2)=O)CC(O)C1 C1(C(=O)NC2(C)CN(C(c3cc(Cl)cc(F)c3F)=O)C2)COc2ccccc2C1 C(CNC(C1OC(C)CC1C)=O)(C(C)(C)C)NC(C(CSC)C)=O C(=O)(CCCCCNC(C1CCS1(=O)=O)=O)N(C)Cc1cnn[nH]1 C1(C(=O)NCCCC#C)(NC(c2cc(C(C)=O)on2)=O)CCSC1 C1(O)(CNC(C(COC)OC)=O)CCCN(C(c2ccn(C(C)C)c2C)=O)C1 C1(OC)CN(C(=O)CC2CN(C(C)=O)CC2C)CC1NC(c1nc(C)oc1C)=O O=C(C1=C(Cl)CCOC1)NCC1CCC1C(=O)NC1CC2CCCC(C1)C2 c1(OC)ccc(Cl)c(CC(=O)NC(C)(C)CN(C(=O)C(F)CNC2CCC2)C)c1 c1(C(=O)NCC2C(NC(c3n(C)ncc3)=O)C2)c(F)ccc2ccoc12 C(C(C)(C)C(=O)N(C)CC1(C)CCCC1NC(c1ccoc1)=O)OCC c1(C(N2CC(O)CC(NC(CNC(CC)=O)=O)C2)=O)cc(C)nc2onc(C)c12 c1(CC)cc(C(=O)NC(CNC(=O)CC(C)(C)OC)C2CCC2)cc(N)c1 C=CCC(C)(O)C(=O)NC(C)C(C)C(N1CC(N(C)OC)C1)=O N1(C(c2cnc(COC)s2)=O)CCC(CNC(=O)Cn2nc(C)cc2C)C1(C)C CC1(C)CCC(CC(=O)NCC2CN(C(=O)C(N3CCCC3)C3CC3)C2)C1 C1(OC)(CNC(=O)CCC2CC3CCC2C3)CCN(C(c2cnco2)=O)C1 c1(N2CC3C(CNC(c4[nH]cc(CC)c4)=O)C3C2)ccc(C(C)=O)cc1[N+](=O)[O-] N1(C(C2C3(CCN(C(=O)CCc4ccncn4)C3)C2)=O)CC2CCC1C(O)C2O N1(C(C2CCCCC2NC(C2(OC)CCC2)=O)=O)CCCC(C)C1CO C(=O)(C1=CC2(CCOC2)C1)NCCCC(C)(C)NC(CC)=O.N12CCC(C1)C2=O C(=O)(C1=NN2CCCN=C2N1)N1CCCC(O)(CNC(CC(C=C)CC)=O)C1 C(=O)(C1=CCCCC1)N(CC(C)CNC(=O)CC1(C)CC1(F)Cl)C C(N=c1[nH]c2ccc(N)cc2s1)C1N(C(C(CC#C)(C)C)=O)CCC1 C(CC(N=c1nc(C(C)(C)C)[nH]s1)C(C)C)SC.C12(CC1)C(=O)N2C C1(NC(C(C)=C2CCCC2)=O)CN(C(=O)CC2(C)CCCO2)CC2(CC2)C1 c1(C(=O)NC(C2(O)CN(C(C3CCCCC3F)=O)C2)C)ccc(F)cc1F N1(C(C2CC(OC)CN2C(=O)C(N2CCNC2=O)C)=O)CCC2(CNC(=O)O2)C1 c1(OC)ccc(F)c(C(N2CCC(CNC(=O)C3=CCCC3C)C2(C)C)=O)c1 c1(NC2CC3CN(C(=O)OC(C)(C)C)C2C3)nccc2ccc(Cl)cc12 N1(C(CCCC=C)=O)CCC(C=C)(C(=O)NCCN2CCCCC2C)C1 N1(C(CC(=O)NC)=O)CCC(O)(CNC(C2C(C(C)C)C2[N+](=O)[O-])=O)C1 C1(C)(NCc2cc(C(=O)OCC)nn2C)CCOC1C1(C(=O)OC)CCC1 N1(C(COC(C)(C)C)=O)CCC(CCNC(C2CC2F)=O)CC1 C1(C(=O)NCCC(O)C2CC2)CCCCCCN1C(=O)CCN1CCOCC1 c1(C(=O)NC2CCC(N(C(=O)CCCN=[N+]=[N-])C)C2)cc(N)c(F)cc1F N1(C(c2c(C)nn(C)c2)=O)CCCC(NC(=O)C(C(C)C)OCCC(C)C)C1C Cc1nc2ccccn2c1CNC(C1CCCC1C1CC1)=O C1(CNC(CS(=O)(=O)NCC)=O)CC(C)(C)CN1C(=O)CC1CC2CC2C1 C(C)(C)(CCC(=O)NCC(CC(=O)N(c1cccc(F)c1)C)C1CCC1)OC C=CC1(CC(=O)NCC2CCCN(C(C3CCCCCCC3)=O)C2)CCOCC1 N1(C(C(C)n2cnnn2)=O)CCCC(N(C(=O)Cn2ccc(C(F)(F)F)n2)C)C1 C1(C(N2C(CNC(c3ccc(CC)s3)=O)CC2)=O)CCCCC(=O)C1 Ic1cnc(C(c2nnnn2Cc2ccccc2)NCCc2sccc2Cl)s1 c1(C(C(N2CCCC2CCNC(C2CC2[N+](=O)[O-])=O)=O)N(C)C)ccc(Cl)cc1 C1(N(C(CNC(=O)OCC)=O)C)CC2CC1N(C(c1cc(C(C)C)n(C)n1)=O)C2 C1(CNC(=O)C=Cc2cncs2)CN(C(=O)C=Cc2cc[nH]c2)C2CCN1C2 CC1OCCC1CNC(=O)CCN(C(=O)CSCC(F)F)CCO c1(SC)nc(Cl)cc(=NC2CCN(CCCn3ccnn3)CCC2(F)F)[nH]1 CCC(C)CCN=c1[nH]c2c(c(=NCc3ccc(Cl)c(Cl)c3)[nH]1)COC2 C(=O)(C(C)(C)C(C)(F)F)NC(C)C(CCc1ccccc1)NC(c1cc[nH]n1)=O n1(C(C)C(=O)NC2CCN(C(C3(C)CCC(=O)NC3)=O)C2)ncc2ccccc12 N#Cc1ncc(C=Cc2ccccc2)cc1-c1ccc(Cl)cc1 CC1(C)OCCC1NC(=O)C(C)(C)C1CCN(C(=O)C=CC(=O)N(C)C)C1 c1(C(=O)NCc2cccc(O)n2)cnc2ccc(-c3cnn(CCO)c3)cn12 C=C(C(=O)NCCC(C)N(C(=O)CCc1ccc[nH]1)C)C(F)(F)F c1(NC2(C(=O)Nc3cccc(C(CC)(C)C)n3)CC2)ccc2c(c1)OCCO2 C1CCCCCC(=O)N1.C1(F)(NC2CCCC(C(N)=O)C2)CCN(C(C)=O)C1 C1(NC(c2c(C(C)C)cccc2)=O)COCCN(C(=O)C=CC=C(Cl)Cl)C1 C=CCCC(C(=O)N1CCC1(C)CC)NC(=O)C(C)C(=O)OC(C)(C)C CC1(C)CCCC(C)(NC(C2(CO)CCCN2C(C2CCC(C3CC3)C2)=O)=O)C1 C1(C(=O)NC)CCC(C)(C)N(C(=O)C(C)(O)C(F)(F)F)C1 N1(C(C(=O)NC(C)C)=O)CCN(C(C2CCSCC2)=O)CC1C N1(C(CCc2ccc(C)nc2C)=O)CCC(O)(C2(NC(C3CC3F)=O)CC2)CC1 C1(NC(CNC(=O)OC)=O)(CO)CCCN(C(=O)Cc2cncc(C)c2)C1 Cc1ccc(CN2CCOCC2c2nnc(-c3cccnc3)o2)c(C)c1C C1(C(N(CCC(=O)NCC(C)CCCO)C2CC2)=O)C2CCCCCC12 C(=O)(CC(C)(C)NC(=O)Cc1ncccc1F)NCCCC=C N1(C(CC(=C=C)C)=O)CCCC(C)(CNC(=O)CC2OCCCO2)C1 c1(C(=O)NCC2CN(C(C3CCN(c4ccc(Cl)cc4)C3)=O)C2)nnc(O)cc1O c1(C(=O)NCCN(CCOC)C(c2cc(N)ccc2SC)=O)ccc2nc[nH]c2c1 CC12COCC1CN(C(=O)C(CC1CC1)NC(=O)CCC(=O)C1CC1)C2 C1(NC(CC2CC(C)C2)=O)CCCC1CNC(c1ccccn1)=O c1(OCC)ccc(SC2CCCC(C3CCCCC3)C2)cc1O.C1(C=O)CCCN1 N1(C(C=CCCC)=O)CCC(C(=O)Nc2ncc(C(N)=O)cc2Cl)C(C)(C)C1 c1(OC)cccc(C)c1C(=O)NCC1CCCN1C(=O)C(O)CC(C)C c1(C(=O)NC(CCN(C(COCCC)=O)C)C(C)C)ccc(S(N)(=O)=O)cc1N Cc1ccnn1CC(=O)NCCc1n[nH]cc1C(=O)NCc1cocn1 C(N=c1nc(N(CC(CCO)OC)C)c2c([nH]1)CSC2)c1cnn(CC)c1C C1(C(=O)NCCCSC)CC(C)CN(C(C2CC(CF)C2)=O)C1 C(=O)(C(C)CS(C)=O)NCCCNC(COC(C)C)=O C(=O)(CS(=O)(=O)C(C)(C)C)N1C(C(C)NC(CC(C=C)C)=O)CCC1 c1(CC(=O)N(CCN2CCN(C(C3CCO3)=O)CC2)C2CC2)ccc(Br)cc1 C=CCC(C)(CC)C(=O)N(C)CC1CN(C(c2ccccc2CC(=O)OC)=O)C1 CCC(C(=O)NCCCC(c1ccccc1)NC(C1CCCOC1)=O)C1CCC1 C#Cc1ccccc1CC(C)N(C(=O)COc1ccccc1)CC1(F)CNC1 C1(CNC(c2cnc(C(C)OC)s2)=O)CCCN(C(=O)C2=CCCS2)CC1 c1(CNC(C(C)=C2CCC2)=O)cc(C(=O)NCC(C)(O)C2(C)CC2)no1 C(=O)(CCC(=O)NC1CCCC1NC(=O)C(C1CCCN(C)C1)(C)C)NC c1(C(N(C(C)CNC)C(C2CCN(C3CCCC3)CC2)=O)=O)cccnc1C c1(OC)ccc(CC(C)NCC2CCOC2(C)C)cc1F c1(SC)ccnc(C(=O)NCCC(C)NC(c2cocc2C)=O)n1 CCC(CC)(CC)C(=O)NCC(C)CNC(=O)C(c1c(C)noc1C)(C)C c1(C(N(C2CCCN(C(c3c(CC)nco3)=O)C2)CCO)=O)ccc(F)c(N)c1 c1(C2C(C(=O)NC(COC)CNC(=O)CC3OCCCO3)C2)cccc(C)c1 C1(C(N(C2CCN(c3nnc(C(N)=O)s3)C2)CC)=O)CC2(CCC2)CO1 C(=O)(C(C)(Cl)Cl)NCCOCCCNC(C(C)OCCC(C)C)=O c1(-c2cn(CCCOC)nn2)nc(-c2ccoc2)nn1-c1ccnc(Cl)c1 c1(C(=O)OC)cc(C2CCCCC2)[nH]n1.C1(C)CN(C)C(=O)C=CCOCCN1 c1(C(N(C2CN(C(C3N(C(C)=O)CC(O)C3)=O)C2)C)=O)ccc2c(c1)N(C)CC2 c1(NC(CNC(C2(NC(CCC)=O)CCC2)=O)=O)cccc(N(C)C)c1 c1(C(=O)O)nc(C)sc1C(N1CC=CC(NC(=O)NCCCl)C1)=O C1(NC(C2CCCN(C(C)=O)C2)=O)CCN(C(c2ccnnc2O)=O)CC12CC2 C(c1ccc(N(C)C)cc1)=CC(=O)N(c1ccc(C)cc1)S(C)(=O)=O C1(NC(c2c(COC)cccn2)=O)CC2CCC1CN2C(=O)CCCNC(C)=O N1(C(c2nncn2C)C(=O)NC(CC)C)CCOC(C2CC2)C1 C1(C(C)C)CCCC(NC(C2(c3cccs3)CCCC2)=O)C1 c1(OC)cncc(C(=O)N(C2(O)CCN(C(=O)CC(=O)NCC3CC3)C2)C)c1 N1(C(c2csc(C)c2C)=O)CCN(C(C2CCC(C)O2)=O)CC1CC(C)(C)C C(=O)(CC(C)CN(C)C)NC(C)CCCNC(=O)Cc1ccccc1 C1(CCC(=O)NCc2c(CC)nco2)CCCCN(C(c2coc3c2COC3)=O)C1 C1(CC)CC(C(N2CCCC2(CC)CC)=O)CCO1.C12(CC1)C(=O)NC2.C1(C)CC1 C1(C)(NC(c2cccc(CSC)c2)=O)CCC(OC)C1.C12(CC1)C(=O)NC2 c1(NC(C2CC2NCc2ccc(OC(F)F)cc2)=O)cccc([N+](=O)[O-])c1Br Cc1cc(NC(C2CC23CCN(C(c2ccc(Cl)cc2I)=O)CC3)=O)cc(O)c1 c1(CC)cccc(C(N2CC(NC(=O)CCOCC(F)F)CC2C)=O)c1C c1(C(=O)NC(C2CN(C(Cc3cc(C)on3)=O)C2)C)ncc([N+](=O)[O-])n1C C1(C(=O)NCC(=O)NCC(C)C)CCCCN1C(=O)CC1CCCC1C N1(C(C2(CCC)CC2)=O)CCC2CCN(C(c3ccc(Br)o3)=O)C2C1 c12ccsc1COC2=O.C(CC(CC1CC1)NC(=O)OC(C)(C)C)=C(C)C c1(C(N2CCC(N(C)C)C2)=O)cc2ccc(-c3ccc4c(c3)OCCO4)cn2n1 N12CCOC(C1)CCNC(=O)Cc1nc(cs1)CC2=O.C(C)(=O)N.CC C1(C(N2CC3C(CO)C3C2)=O)CC2CCCC2N1C(=O)Cc1ccc(F)cc1 N1(C(c2c(N)ncc(C)c2)=O)CC2(CCC(NC(c3sc(C)nc3C)=O)CC2)C1 C1(C(C)NCCC2OCCC2(C)C)CC12CCSCC2 C1(NC(c2n(C(C)C)ccc2)=O)CN(C(C2CCCC(=O)CC2)=O)CC1C1CC1 Cc1ncccc1-n1nc(-c2ccoc2)nc1CC1CCCC1C N1(C(c2c[nH]c(=N)o2)=O)C2CCC1CC(CCNC(c1ccc(Cl)cn1)=O)C2 C1(NC(CC=CCNC(Cc2ccc(C)nc2)=O)=O)CN(C)CCC1O C(=O)(CCN=c1[nH]c2ccccc2s1)NC(CNC(C1CC(OC)C1)=O)(C)C(C)C c1(OC)ccc(CC(=O)NCC(O)CN(C(=O)Cc2cccnc2C)C)cc1Cl C(=O)(C(C1CCC1)N(C(C)CN(C)C)C)NC(COCC)C c1(C(N2CC(NC(C3CCCN3CC(F)F)=O)C(F)C2)=O)cc2c(o1)CCCC2 c1(C(N2CC3CC(NC(CC(C=C)CC)=O)C3C2)=O)c(F)ccc(F)c1Cl c1(NC(CCNC(C=CSC)=O)C(C)C)cc(C(C)=O)c([N+](=O)[O-])cn1 C(=O)(CC1=CCOCC1)NCC1C(NC(Cc2cccc(OCC#N)c2)=O)C1 N1(C(C(C=C)(F)F)=O)CC2=C(C1)CN(C(c1cc(OC)cc(CC)c1)=O)C2 C12(NC(c3ccc(COC)[nH]3)=O)CC1CN(C(=O)CCC1CC(F)(F)C1)C2 CCC(Cn1cc(CCC#N)nn1)(CC)CO Cc1ccc(C(=O)NCC2CC(F)(CNC(C3CCC(C)(C)C3)=O)C2)n1C CCC(F)(C(=O)NC1COC2CNCC12)C(=O)O CC(C)CC(C)CC(C)C(=O)N1CC2CC(O)C1C2NC(C1COCCO1)=O c1(C(N2CC(NC(CCC#C)=O)CC3(C2)CC3)=O)cc(C)c2c(c1)CCC2 C1(NC(CC(=O)NCC)=O)CC2CC(NC(=O)CC3(OCC)CC3)CC2C1 C1(CNC(CC(C)SC)=O)COCCN(C(c2cn(C(C)C)nc2C)=O)C1 CCCCC(O)CC(=O)NCC(CNC(c1n[nH]c2cccnc12)=O)OC c1(SC(C)C(=O)NC2CN(C(=O)NCC3CC3CO)C2)ccc(F)cc1 N1(C(C23CC(OC)C2C3)=O)CC2CCC(CNC(=O)CSC)C2C1 CCCCCCCCC(=O)NCCCCC(C)(C)NC(C1CC(=O)C12CCC2)=O C(=O)(CCCCC(C)=O)N1CC(C=CC)C(NC(C2COCC2N=[N+]=[N-])=O)C1 C1(C(N2CC(NC(c3ncccc3N)=O)C(C(F)F)C2)=O)(CC)CCOCC1 C1(c2nccc(COC)n2)CC2CCC(C1)N2C(=O)CC(CN(C)C)CC c1(CC)cc(C(N2CCCC2(C)C(=O)N(C)CCN(C)C(C)=O)=O)c(C)o1 C1(=CCNC(c2sccc2CO)=O)CCN(C(=O)CCCCN2CCCC2)CC1 CC1(C)CCCC(CC(=O)NC2CC(n3ccnc3)CC2O)O1 c1(C(=O)NCCC(C)N(C(c2nc(C)oc2)=O)C)cnc2scc(C)n2c1=O C#Cc1ccc(C(N2CCC(C(=O)NC(C)(C#N)C3CCC3)C2)=O)nc1 c1(NC(C)Cn2cc(Br)cn2)ccc(S(=O)(=O)NC(CCO)c2ccco2)cn1 c1(CNC(C(C(C)C)NC(=O)OC)=O)cccc(CNC(C2CCOC2C)=O)c1 C1(NC(C(C)C(C)(F)F)=O)CCCC2CN(C(C3(C4CCOCC4)CC3)=O)CC12 C#Cc1cc(C(=O)NC2CCN(C(c3cc(N)ccc3Cl)=O)C2CC)ccc1Cl C1(C(=O)NC2CCCN(C(=O)Cc3cscn3)CC2)CC2C=CCC(C1)C2 N1(C(C2(C)CCOCC2)=O)CC2CCC1C(CNC(=O)C1=C(C#N)CCC1)C2 CC1CN(C(c2ccc(Cl)nc2)=O)CC(C)C1N=c1[nH]ccnc1F c1(C(N(C2CC(NC(c3snc(C)c3N)=O)C2)C)=O)n[nH]c2c1CCC2 CC1CN(C(c2ccc(CN(C)C)cc2)=O)CCC1NC(=O)CC1CC1 C=Cn1nncc1C(=O)NC1CCCC1NC(c1nccnc1C)=O c1(OCC(=O)NCC(CCNC(c2ccn(COC)n2)=O)O)cccc(Cl)c1 c1(C(N2CCC(NC(C=CC=CC)=O)C23CCC3)=O)cc2c(C)ccc(F)c2[nH]1 c1(C(=O)NC(CNC(CS(=O)(=O)N(C)C)=O)(C)CO)cn2c(n1)COCC2 C(=O)(CCC(C)(C)F)OC.C12CC(CN1CCN(C)C)NC(=O)COC2 c1(CCCC)ncc(C(=O)NCCC(C)(C)NC(c2c[nH]cc2C)=O)s1 Cc1ccc(C)c(CN2C3CCC2CN(C(=O)C=CC2CC2)C3)c1O C(=O)(C1=NN2CCCN=C2N1)NC(C(C)C)CNC(C1C2CC3C(C2)C13)=O C(CCC(=O)NC1CCC(C(=O)NC2C=CC(C(=O)OC)C2)C1)OCC C1(N(C(=O)C(CO)NC(N)=O)CC)CCN(C(=O)C(F)Cc2ccccc2)CC1 C1(NC(CCc2onc(C)n2)=O)CC2CN(C(C3CC(=O)NC3(C)C)=O)CC2C1 c1(CCC)onc(C)c1C(N1CCC(CN(C(c2nonc2CC)=O)CC)C1)=O N1(CC2(NC(=O)Nc3ccccc3)C(C)OCC2)CCSCCC1C C1(NC(C2C(C)CCC2)=O)CN(C(C2CCCC23CCC3)=O)CC2(CC2)C1 C1(CNC(C2C3CCCCC3N2)=O)CN(C(C23CC2CNC3=O)=O)CC1O C(=O)(C1=CCC(F)(F)CC1)N1CC(C)N(C(C2CCCCC2(C)C)=O)CC1 C12(C(N(C)CC3OCCN(C(C=Cc4c(C)ccs4)=O)C3)=O)CC1COC2(C)C Cc1ccc(Cl)c(C(N2CC(C3CN(C(C4CC5CCC4C5)=O)C3)C2)=O)c1O C1(F)(CNC(CC(COC)(C)C)=O)CC2CCC(C1)N2C(=O)C=CS(C)=O C1(CNC(C2CCCS2)=O)CC2(CCN(C(C3C4CC5C(C4=O)C35)=O)CC2)C1 C(C(C)C)(C(O)C(=O)N(C)CC1CCCN(C(=O)CCc2cnc[nH]2)C1)OC C1(CNC(c2cc(C)[nH]n2)=O)(NC(c2cccc(N(C)C)c2)=O)CC2CCC1C2 C1(CC)CN(C(c2cc(C(C)C)ns2)=O)CCC1NC(=O)C=Cc1cncc(O)c1 C(=O)(C1=C(Cl)CCCC1)N1CC(CNC(=O)CC2C=CCCC2)OCCC1 Cc1cc2ncc(C(=O)NC3CC4(C3)CN(C(C3(CF)COC3)=O)C4)cn2n1 C1(NC(C2(CC)CC2)=O)CN(C(c2csc(C(F)F)c2)=O)CC1C N1(CC)CCC(NC(=O)CN(CC(C)C)C(C2C3CC(=O)CC23)=O)C(C)C1 n1(CCN(C(C2(C)CC(OC(=O)NC)CN2C)=O)CC)c(=O)oc2ccccc12 CCC(CCC(=O)N(C)CCOC)NC(c1nonc1N)=O C1(CNC(CN(CCOC)C)=O)(NC(C2CCC2C)=O)Cc2ccccc2C1 C1(C(=O)NC(C2(O)CCN(C(CCC=C)=O)C2)C)CCc2nn[nH]c2C1 c1(C(N2CC(NC(C(C)NS(C)(=O)=O)=O)C(O)C2)=O)cn2cccc(F)c2n1 Cn1c(C(=O)NC2CC3CC2N(C(=O)Cc2csnn2)C3)cc2sccc12 C(C(=O)NCCOCCOCCOCC(=O)NC1CC1)(C1CCC1)OC N1(OC)CC2CC2(CNc2cnc(-c3cnn(C)c3)s2)C1 C1(C)(NC(C=CC(C)C)=O)CCCN(C(=O)Cc2cc(C(F)(F)F)ccc2Cl)C1 C1(CN(C)C(C2(CNC(c3ccc(C(N)=O)[nH]3)=O)CCCO2)=O)COC(=O)N1C Cn1cnc2c1CCCC2C(=O)NC1CN(C(c2cc3scnc3[nH]2)=O)C1 C1(COC)(NC(=O)C(=O)NCC2CCC(=O)C2)CCCOC1 c1(CC(=O)NCC2(NC(C3C(C#N)C3)=O)CCC2)ccc2nonc2c1 c1(CCN=C(NC2C(C)(OC)C2)NC2CC2)cnn(S(C)(=O)=O)c1 N1(CCCOCC)CCCC(CCNC(=O)COc2ccc(F)cc2)C1 CCCC(CCC)=CC(N1CCC(C)(NC(c2cc(C3CC3)cs2)=O)C1)=O C1(C(=O)NCCN(C(c2cccc(OCCOC)c2)=O)CC)CC2C(C1)C2(C)C CC1CC(NC(=O)Cc2cscc2Br)CCN1C(=O)CC1CCOC1 Cn1cc(Cl)c(C(N2CC=CC2CNC(=O)Cc2cncnc2)=O)n1 C(CCCCC(=O)N1CCC(CNC(=O)Cc2ccns2)CC1C)NC(C)=O c1(C(N2C3CC2CN(Cc2cccnc2)C3)=O)cc([N+](=O)[O-])ccc1Cl C(=O)(C(F)CC(C)C)NCCN(CCC)C(C1CCCCC(=O)N1)=O CC(CC(F)(F)F)C(=O)N1CC=C(CCNC(c2n[nH]cc2Cl)=O)CC1 CCC(C(=O)NCCCCCC1CC1)N(C(=O)CCC1OCCO1)C c1(C2CCN(C(=O)N(C(C)(C)C)C34CC3C4)CC2)nc2ncccn2n1 c1(NC(C2CCCC(NC(C3CCCC3)=O)C2)=O)cc(F)cnc1Br C1(C(=O)NC(C2CCCCC2)CO)COCCN1C(=O)C(F)CC1CCOC1 c1(C(C(=O)NCC(CNC(c2cnc(CC)s2)=O)F)(C)O)ccc(F)cc1 C(C1CCCCC1)=CC(N1CCC(CC(N2CCCC(F)C2)=O)C1)=O c1(CNC(C2C(C)COCC2)=O)ccc(CNC(C23CCC2CC3)=O)cc1F C1(C(C)C)C(=O)NC(=O)CNC(=O)C(C2=CC=CC=CS2)N1C.C(C)(C)(C)OCC.CC C(=O)(CC(O)(C(F)(F)F)c1ncco1)Nc1onc(-c2scc(C)n2)n1 C1(C(=O)NCCCCCNC(CSCC=C)=O)CC2CCCCCC12 N1(C(C(CCC)F)=O)CC2(CCCC2)C1C(=O)NC(C)C(=O)NC(C)(C)C c1(CCC(=O)OCc2nc(Br)ccc2Cl)cc(F)cc(Br)c1 C1(C)(C(=O)OC)CCC1(C)C(=O)NCCCCCNC(c1ncsc1C(C)C)=O C1(NC(CNC(c2c(OC)cccc2)=O)=O)CC(C)N(C)CC1C C1(NC(C(C)S)=O)CC2(C1)CN(c1cc(-c3ccccn3)ncn1)C2 C1(CNC(c2cc(CC)c(C)s2)=O)CN(C(=O)CNS(N)(=O)=O)CC12CCC2 c1(COC(c2c(C)c3c(cc2)OCO3)=O)cc(=O)n2[nH]c(-c3cccs3)nc2n1 c1(NC(c2n(CCC)nnn2)(C)COC)ccc2oc(O)nc2c1 c1(C(C(=O)NC2CC(NC(C3(Cl)CC3)=O)C2)OC)cc(F)cc(F)c1 c1(C(N(C2CN(C(C3(COC)COC3)=O)C2)C)=O)coc2cc(F)ccc12 C1(C(=O)NCC2(NC(c3ccc(Cl)s3)=O)CCC2)C2CCC1(c1ccccn1)C2 C=CC(CC(=O)N1CC(CCNC(=O)C(C)CO)(OC)C1)c1ccccc1 C1(C(=O)NCc2c(C(=O)NCCc3n(C)cnn3)n[nH]c2)CC2CCC2C1 n1(C(C)CNC(=O)COCC(F)F)cc(CCC2CCC2)nn1 Cc1cc(C(c2nnnn2NS(C)(=O)=O)C2CCOCC2)ccc1Br.C1CCN1 C1(CC=C)(C(=O)N(c2nc(C(C3CC3)C)cs2)C)CCCC1.SC C(=O)(CCC(F)(F)Cn1cc(CCNS(N)(=O)=O)nn1)NC(CCCC)COC C1(N(C(C2C(C(=O)OC)C2)=O)C)CCN(c2nnc(C3CC3)o2)C1 N1(C(C2CCCN(CC)C2)=O)CC(NC(c2ccc(C(C)C)s2)=O)CC(C)C1 c1(CC(=O)N(C2CCN(C(=O)Cc3cn(C)nn3)C2)C)nc(C2CC2)cs1 Cc1ccnc(C(=O)NC2C3CN(C(c4cc(C(N)=O)[nH]n4)=O)CC23)n1 C(=O)(C(C)(C)CF)NCC(=O)NC1C(NC(C(C)OC2CCCCC2)=O)C1 CCC(C(=O)NCCC1CCCN1C(=O)Cc1ccn(CC)n1)N1CCCC1=O c1(OC)cc(C)cc(C(N2CCN(C(c3ccsc3OC)=O)C3CC23)=O)c1C N1(C(C(CNC(C(C2CCC2)OC)=O)OC)=O)CCCC(O)(CO)C1 Cc1cc(C(N2CCC(C(C)(C)CNC(C3C4CCCC34)=O)CC2)=O)nc(O)n1 C12(NC(c3ncn(CC)n3)=O)CCCC1CN(C(c1cc(F)c(Cl)cc1F)=O)C2 CC1=C(C(=O)N2CCOCC2CCNC(c2c(C)ccnc2O)=O)CCC1 c1(OC)cc(Cl)c(Cl)cc1C(N1CCC(N(C)C(C23CC(C)C2C3)=O)C1)=O Cc1ccccc1C(N1CCOC(CCCCNC(=O)CC2(C)CCCO2)C1)=O c1(CC(=O)NC(CC)CNC(C2CC2F)=O)c[nH]c2cccc(Br)c12 CC1CC(C)CCN(C(=O)C(CCS(C)=O)C(=O)OC(C)(C)C)C1 CC1CCN(C(c2cccc(F)c2)=O)C1C(=O)NCC1(F)CCOCC1 C1(C(=O)NCC(C)NC(C(CC)Oc2ccccc2F)=O)CCn2cncc2C1 C(=O)(CCc1nncs1)N(CCNC(C1(CCCC)CC1)=O)CC1CC1 CC(C)CC(CNC(c1cc(C(C)(C)C)on1)=O)NC(=O)CC12CCCC1C2 CCS(=O)(=O)c1ccc(C(=O)NCCC2CC(NC(=O)C(C)SC)C2)cc1 c1(C(=O)NCC2(O)CC(NC(COCCCCC)=O)C2)ccccc1S(=O)CC C(=O)(CCS(C)=O)NCC(CN(C(C1(Cl)C(C(C)=O)C1)=O)C)(C)C c1(OC)ccc(C(F)F)cc1NC(=O)C(C)ON1CCSCC1(C)C c1(C(N2CC(CNC(C3N(CC)CCC3)=O)OCC2)=O)cc(O)cc(F)c1 c1(C(N(C2CCN(C(C3CC(O)C3)=O)C2)CC)=O)ccc(S(C)(=O)=O)s1 C1(NC(CC(C)(C)CNC(c2cc(F)c[nH]2)=O)=O)CCn2nnnc2C1 CC1CC(NC(C2CCC(F)C2)=O)CN1C(=O)CCCc1ccccc1 c1(C(N(C(CNC(=O)CCCCCF)C2CC2)C)=O)cnc(O)c(F)c1 C(=O)(C(C)C(C)(C)C)NC1C(NC(c2ccc(NC)cn2)=O)CCCC1 O(NC(=O)C(Cc1cn[nH]c1)NC(=O)CN1CCC1C)CCC=C Cc1cc(C(=O)NCC=CCNC(=O)CC2CCC(C)C2)ccn1 C1(NC(c2cc(COC)[nH]n2)=O)CN(C(C2CSCCS2)=O)CC12CCC2 C12(NC(CC(CC)C)=O)CCC(NC(C3CCC(C)=C(C)C3)=O)(CC1)C2 C1(CCC)CN(C(C2C3CC(=O)CC23)=O)CC1NC(=O)C=CBr c1(C(N2C(C(N(C)CCc3cnccn3)=O)CC2)=O)ccc(Cl)cc1Cl c1(NC(C2CC(Nc3ccnc(SC)n3)C2)=O)cc(Cl)c(F)cc1F c1(C(N2CC(C)(OCC(=O)NC3CC=CCO3)C2)=O)cc(O)ncn1 C(c1ccc(OCCC)c(O)c1)=CCN(Cc1ccc(OCCCCC)cc1)CC c1(C(=O)NCCC(O)CNC(c2nccc(Cl)c2O)=O)ccc(F)cc1[N+](=O)[O-] N1(C(C(=O)C2CCCC2)=O)CCCN(C(c2cc(Cl)ccc2F)=O)CCC1 c1(CCC(=O)OC(F)F)ccc(Cl)cc1.N1(C(=O)CC)CCN(CC(O)C2CC2)CC1 Cc1c(NC(=O)NC2CCC=CO2)cccc1COC(C)(C)C C1(CN(C)C(C2C(C)(C)C2(F)F)=O)CN(C(=O)CN2CCOCC2=O)CC12CC2 CC1(C(=O)NC2COCC2NC(=O)CN2CCC(C(N)=O)CC2)CCC(=O)NC1 c1(C(C)NC(c2nc(CC(=O)OC)no2)CC)cccc(OC(F)F)c1 C12(C3C(CC(C)(C)C)C3)CCC(CN(N3CC4CCOCC4(CO)C3)C1)C2 C=CC1CCN(C(c2cncc(CNC(c3ccc(C)n3C)=O)c2)=O)C1 C#Cc1cccc(CC(=O)N2CCC2CC(=O)NC)c1 C1(CC(=O)N(C2CCCN(C(=O)C3=COCC3)CC2)CC)CCCCC1(C)C N1(C(C)=O)CCCC(C(=O)NC2CN(C(=O)CN3C(=O)CNC3=O)CC2C)C1 c1(C(=O)NC2CCN(C(c3cncc(C)n3)=O)C(C)C2)cc([N+](=O)[O-])n(C)n1 c1(C(=O)NC(CN(C(C(C=C)c2ccccc2)=O)CC)C)cccc(NC)n1 N1(C(C23CCC(OC)C2C3)=O)CCC=C(CNC(C2CC2F)=O)C1 C1(CNC(c2c(C)cc(=N)[nH]n2)=O)CCN1C1c2ccccc2-c2ccccc21 c1(CC(CO)NC(=O)CCC2CCCOC2)cccc(Br)c1 c1(C(=O)NC2CC(C)(NC(Cc3ccc(C)s3)=O)C2)ccn(C)c(=O)c1 C1(NC(=O)C2CC2)CCC2CN(C(C3CCCc4ccccc4C3)=O)CC2C1 C(=O)(C1CSc2ccccc21)NCC1CC(C)(C)CN1C(=O)CC1CCCCC1 O=C(CCC(=O)N1CCN(C(c2ccnnc2S)=O)CC1)NC.N1CCOCC1 C(N=c1[nH]nc(C2CC2)o1)c1n(C(C)C)c(C2CCCN(C)C2)nn1 c1(C(=O)NC2CN(C(CSCC(C)C)=O)C2)coc(C(C)C)n1 N1(C(C2CNC(=O)O2)=O)CCCN(C(c2cc(C3CC3)no2)=O)CC1CO n1(C(C(=O)NCCCN(C(C2CCC(OC)CC2)=O)C)C)c(C)cc(O)cc1=O CC(C)C(CCNC(=O)C=Cc1nnn(C)n1)NC(c1csc(CO)n1)=O C#Cc1ccc(NC(=O)C(O)CNC(=O)C(C)N=[N+]=[N-])c(C)c1 C(=O)(C(C)(C)C(F)F)NCc1cc(C(N(CCc2nc(C)on2)C)=O)no1 c1(CNC(=O)OCC)cnn(C(=O)NC2CCCN(Cc3ccccc3)C2)c1 Cc1ccc(-c2nc(CCn3cncn3)nn2C2CCCC2(C)C)c(Cl)c1 CC1(C#CC(=O)NC2CCCC2NC(=O)CCSc2ccccn2)CCCO1 c1(C(N(C2CCN(CC=C)C2=O)CC)=O)c(C)nc2ncnn2c1F C1(N(C(C(CNC(C)=O)(C)C)=O)C)CN(C(=O)CC2CCNC2=O)CC1(C)C C(=O)(CCCn1cccn1)N.CC(C(=O)NC1CC1CNC=O)NC(c1ccco1)=O C(CCC(C)(C)NC(C1CCCC1CNC(c1ccccc1O)=O)=O)OC CC1(NC(=O)C=CC2CCCC2)CCCN(C(c2cc(C(F)(F)F)n[nH]2)=O)C1 N1(C(C(c2ccn(C)n2)C)=O)CC2CC(C1)C2NC(=O)CCc1cnc(O)[nH]1 N1(C(C(C)OCCN(C)C)=O)CCOC(C(N2CC=CC23CCC3)=O)CC1 c1(C(N2CCCC(CC)(NC(C3COC(=O)O3)=O)C2)=O)ccc2ncccc2n1 CC1=CCC(C(=O)NCC2CCN2C(c2cc(C(O)C(F)(F)F)ccn2)=O)CC1 N1(C(c2c(OCC(C)C)cccc2)=O)CCc2cc(C(N)=O)ccc2C1 c1(OCC(N2CC(C)C(CNC(=O)CCC[N+](=O)[O-])C2)=O)cc(F)ccc1F CC1CN(C(=O)OC(C)(C)C)CCC1CNC(=O)Nc1ccc(Cl)n1C c1(Cn2ncc(Oc3ccc(COC)cc3)c2)cc(O)nc(N(C)C)n1 N1(C(C2(SCC)CC2)=O)CCN(C(=O)C=Cc2cncc(C)c2)CC2(CC2)C1 C1(C2CN(C(=O)CC3CC3(C)C)C2)(NC(c2cn(CCCC)nc2C)=O)CC1 CCC(COC)(c1ccccc1)NC(CC(C)SC)c1nnnn1C1CCCCC1 N1(C(C2C(CCOC)C2)=O)CCCC1CN(C(=O)C=CSC)C CS(=O)(=O)C1CCCC1C(=O)NC12CCC(NC(=O)C(O)c3ccsc3)(CC1)C2 Cc1cc(=NC2CCCN(C(=O)C(O)C(C)(C)C)C2)[nH]c(S(C)(=O)=O)n1 CP(C)(=O)CCC(=O)N1CCN(C(C2CCC(=C3CCC3)CC2)=O)CC1CF C1(CC(=O)NC2(C(=O)NCc3cnsc3)CCCC2)CCC2(CC1)CC2 c1(C(=O)NC(C2CN(C(=O)C(F)(F)C3(O)CCC3)C2)C)ccc(F)c(Cl)n1 c1(Nc2c(C)cc(Br)cn2)cc(Br)cc2ccccc12 N1(C(C(CC)(C)C)=O)CCCC(C2CC2NC(c2ccc3[nH]ccc3n2)=O)C1 C1(C)(C(=O)NC2C(NC(C3(CC#C)CCOCC3)=O)CC2)CC=C(C)CC1 C12(C(=O)OCC(C3CCC(CC)O3)=O)CC1CCN2C(C1CC2CCC1O2)=O CCC(COC)C(=O)NCC1CC(C(=O)NCC(O)C(=O)OC)CO1 c1(OC)cc(C(=O)NC2CCCC2CNC(=O)CCC(C)CN(C)C)cc(C)n1 C1(C)(C(N(CC)Cc2csc(NC=O)n2)=O)CCCN(c2ccc(C#N)cn2)C1 N1(C(c2c(C)cc(F)cc2)C(=O)NC2CCOCC2)CCC(CO)C(C)(C)C1 c1(SCC(=O)NC2C(CNC(C=Cc3occ(C)n3)=O)C2)ccc(F)c(F)c1 CC1CCCn2cc(C(N3CC4CC(NC(c5cn(C)nn5)=O)CC4C3)=O)nc21 C(C(C)(C)CC(=O)NC1CC2(C1)CC2N(C)C)NC(COCCSC)=O C=C(C)CC(C(=O)N1CCC(C)(NC(c2ccc(N)c(O)c2)=O)C1)OC C(CCCC(=O)N(C)CC1CCN(C(=O)Cc2ccn(C(F)F)n2)C1)SC Cc1cc(C(N2CCN(C(C3CCOC3C(F)(F)F)=O)CC2CO)=O)cc(N)c1 CC1(C)CC(CNC(C2CCC(=O)O2)=O)CN(C(C2CC3(C2)CS(=O)(=O)C3)=O)C1 C1(CNC(CC2(C)CCCO2)=O)CN(C(C2(C)CCOCC2)=O)CC2(CCC2)O1 C1(NC(c2cc(C(C)C)no2)=O)CCC12CCN(C(c1cn(C)[nH]c1=N)=O)CC2 c1(C(=O)OC)cc2c(C(N3C(C)C(=O)NC(C)C3C)=O)nccc2o1 c1(C(N(C)CC2(O)CCN(C(CSCCCC)=O)C2)=O)ccc2nc(S)oc2c1 c1(C(N2CC(CC)C(CNC(=O)C(C)SC)CC2)=O)onc2ccccc12 C1(C)(CNC(C2CC(C(F)F)(OC)C2)=O)CCCN(C(c2cccn2C)=O)C1 Cc1cc2sc(C(N3CC4CC(NC(=O)C=Cc5ccc(Cl)s5)C4C3)=O)cc2s1 C1(C(N2CC(CC(=O)NC3CCN(C(C)C)CC3)C2)=O)CCCCC(F)(F)C1 C(N=c1ccc(S(C)(=O)=O)c[nH]1)C1CC(NC(c2[nH]cc(CC)c2)=O)C1 C(N=c1[nH]c(=NC2CCCN(C)C2)[nH]c2c1CSC2)C1OCC(C)C1 N1(C(C2(CO)CCN(C)C2)=O)CC2CCC(CNC(c3c[nH]nc3Cl)=O)C2C1 CCC(CC(=O)NCC1COCCN1C(=O)Cc1nncn1C(C)C)OC c12ccc(cc1)C(=O)n1cc(nn1)C(=O)NCCNC2=O.C12(CC1)CC2.CC.OC O=C(C1=C(Cl)CCC1)NC1CCN(C(c2cc3n(c2)CCC3)=O)CC1O C1(c2onc(-c3cc(SC)sc3)n2)CCCCN1Cc1cccc(Cl)c1 c1(NC)cccc(C(=O)NC2CC(NC(=O)CC(=O)NC3CC3)C2)n1 c1(C(N2CC(C)N(C(=O)CCC3CCC3)CCC2)=O)ccnc2c(F)cccc12 CCCCCC(C)CC(=O)NC(CC(C)C)C(=O)N(CC(F)F)C c1(C(C(=O)NC(Cc2nnn(C(C)(C)C)n2)C2CC2)(C)C)ccc(Cl)cc1F C1(C)(CC(c2n(CC)nnn2)NCCc2cccc(C3CC3CO)c2)CC(C)=NO1 c1(C(N(CCCCN(C(CCOCC)=O)C)C)=O)cnc(OC)s1 c1(CCC(=O)NC2CCN(C(C(=O)OCC)C)C2)ccc(NC(C)=O)cc1 c1(CC(=O)NC2C(OC)CN(C(=O)CN3CC(C)C3)C2)cn2cc(F)ccc2n1 c1(CC(=O)NC(CN(C(CCCC(C)=O)=O)C)C)ccc2oc(O)nc2c1 C1(C(C)NC(C(C)C#N)=O)CCN(C(=O)COC2CCN(C)CC2)CC1 c1(C(N2CC3(OCC(NC(C4CC(C)OC4)=O)C3)C2)=O)cc(N)cc([N+](=O)[O-])c1 N(C(=NCCCN1CCCC(C)C1)NC1CSC1(C)C)CCc1ccc(C)cc1 Cc1nccc(C(N2CCOCC(NC(=O)CCC(F)(F)F)C2)=O)c1C C(C)(C(C(=O)NCCC1CCN(C)C1=O)NC(c1cn(C)cn1)=O)OC Cc1cnc(C(F)(F)F)cc1C.C12CC(n3cncn3)C1CN2 C1(CC)CN(Cc2cc[nH]n2)CCN1C(c1ccnc(O)c1)=O c12cc(F)c(F)cc1C(=O)N2.N1(C(C(C)(C)C)=O)CC2(CC(NC(=O)CO)CO2)C1 C[Si](C)(C)C1(C(N2CCOC(c3cccc(O)c3)C2)=O)CC1 C1(C(=O)NCC(C)(C)NC(CN(C)C)=O)CC2C=CC1C2 C1(C)(C(=O)OC)CCN(C(=O)CC2(NC(=O)C(C)=C(C)CC)CCC2)C1 C(N=C(NCC(C)(C)C)NCC1CC1Cl)c1ccn(C)c1 c1(NC)cnccc1C(N1CCCC(C(C)(C)C(=O)N(C)C)C1)=O S(=O)(=O)(c1ccc2cc(C(=O)OC)ccc2c1)NCCCC(=C)C N1(C(C(=O)NC2CCOCC2)C2C(CC)C2)CCC2(CC1)CN(C)C2 C(=O)(C(F)CC1CCOC1)N(C(c1ncon1)C)C1CC1 c1(OC)cnn2c1CN(c1nnc(C3CCOC3)n1CC1CCCO1)CC2 C(N=c1nc(C(C)C)cc(C)[nH]1)C1CC(OC)C1.N12CCCC(O)(C1)C2 C(=O)(C(F)C(F)(F)F)NCC1CCC(CNC(=O)C=Cc2cc[nH]n2)CC1 C1(CCC=C)CCCC1(c1cccnn1)NC(C1(CO)CCC1)C1CC1 c1(OC)ccccc1Cn1nc(Cn2cccn2)nc1-c1cnc(Cl)s1 c1(OC)cc(OC)c(NC(C2CC(F)(F)CN2C(c2csnc2C)=O)=O)cc1Cl c1(C(N2CCC(CCC)(CO)C2)C(=O)NC(C)C)ccc(OC(F)F)c(Cl)c1 N1(C(C2(CNC(c3cc(Cl)no3)=O)CCCO2)=O)CC(O)(C2CC2)C1 c1(C(=O)NCC2N(C(CCNC(=O)NC)=O)CCC2C)cc(OC)cnc1F c1(C(=O)NCC2CN(C(c3cnc(C)o3)=O)C(C)(C)C2)ccc(Cl)c([N+](=O)[O-])c1 c1(C(N(C2CCCC(NC(=O)CC=C(Cl)Cl)C2)C)=O)cccc(OC(F)(F)F)c1 c1(C(=O)NC2CC3CN(C(C=Cc4c(C)nsc4)=O)C2C3)cccc2cncn12 C(C)(N=c1[nH]nco1)C1N(C(c2c(C)nc(CC)s2)=O)CCCC1 c1(OC(C2OCCC(NCc3c(Cl)cn(C)n3)C2)=O)cccc2cnc(Cl)cc12 c1(C(=O)NCC(=C)CCNC(c2ncnn2C2CCOCC2)=O)sc(C)nc1C N1(CCC(N2CCC(CNC(C3N(CC)CC3)=O)C2)=O)C(=O)NC(C)(C)C1=O Cc1cccc(C(N2CCC(C(C)C(=O)NCC=C3CCSCC3)CC2)=O)c1 N1(C(c2n(CC)nc(C)c2)=O)CC(NC(C2CCOC2)=O)Cc2ccccc21 C(=O)(C(C)(C)COCC(F)F)N1C(C(=O)NC2CN(C(C)=O)C2)CC1 C1(C(N2CC(OCCNC(CNS(C)(=O)=O)=O)C2)=O)COCC1C(N)=O N1(C(COCCOC)=O)CCC(F)(CNC(c2c(C3CCCC3)noc2C)=O)C1 Cc1cc(C(=O)NCC2(F)CC(NC(C3(C(=O)NC4CC4)CCC3)=O)C2)on1 C1(OC)CN(C(c2cn(CC(F)F)cn2)=O)C(C)(CNC(=O)COCC(C)C)C1 C(=O)(C(CC(C)(C)C)OCC(F)F)Nc1ccc(C(N(CCC)CCC)=O)s1 C(C(=O)N1CCOC(C(=O)NCC(C)OCCO)C1)(C(C)C)SC c1(CC(N2CC(CNC(C=CC(CC)C)=O)C(C)C2)=O)ccc(C)c(F)c1 C1(C(=O)NCC(C)CNC(C2CC2c2cnc[nH]2)=O)CCC(C)(C)CO1 Cc1noc(C(C)C)c1-n1cc(C(C2CCS(=O)(=O)C2)N)nn1.C12=CC=C(C=C1)C2 Cc1cc(=O)ccn1CC(N1CCC(CCNC(c2ccc(SC)s2)=O)C1)=O Cc1nc2n(n1)CC(C(=O)N(CC(C)CNC(=O)CCn1ccnc1)C)CC2 c1(C(N(CC(CNC(C(=O)NCCOC)=O)C)C)=O)ccn2ccnc2c1 c1(C(=O)NCCCN(C(C2C(C)CC2C)=O)CC2CCCC2)nccc2n[nH]cc12 CN1C2CCC1CC(CC(=O)NCC1CC(F)(CNC(C3C4COCC34)=O)C1)C2 C1(OC)CC(NC(=O)C=C2CCC2)C12CCN(C(c1ccc(O)cn1)=O)CC2 Cc1cc(C(=O)NC(C)CCNC(=O)C(C(C)O)N(C)C)cc2ccsc12 C(=O)(CC(CC(C)C)NC(=O)C(Cl)Cl)NC(C(=O)OC)CO Cc1cncc(CC(=O)N(C)CCN(C)C(c2ncc(F)cn2)C)c1 C1(CC#C)(C(=O)NCC(C)NC(C2CC(c3ccccc3)(CC)C2)=O)CCCC1 CCCCCS(=O)(=O)CC(=O)N(C1CN(C(=O)Cc2cnc(C)o2)CC1F)C c1(CC2C(C(=O)NCC(C)(C3CCC3)NC(c3cnsc3)=O)C2)ccccc1Cl C1(O)(CNC(COC(CC)C)=O)CCCN(C(c2coc(Cl)n2)=O)CC1 C(CCC(C)CC(=O)N1CCCC(CNC(c2ncc(C)cc2F)=O)C1)=C(C)C N1(C(CCC2C(C)C2)=O)CC2CCC(NC(c3cnn(C4CC4(F)F)c3)=O)(C2)C1 C(=O)(C1=NN(C)C(=O)CC1)NC1CC(NC(c2nc(CCC)sc2)=O)C1 C1(CCC#C)CCN(C(C2CCCN(C(c3cc(C)n(CC)n3)=O)C2)=O)CC1 CC(CCCCCO)NC(C12CC(CN1C(=O)CCCF)C2)=O C(=O)(C(O)CC(C)(C)C)NC1C2N(C(c3c(C)n(CCO)nc3)=O)C(CC2)C1 c1(NC(C(=O)NC(C)CCc2cccn2C)=O)ccccc1N1CCCC1=O c1(OCCC)c(OC)cc(C(N)=O)cc1NCc1ncc(NC)cn1 n1(CC(=O)NCC2(O)CCC23CCC3)ccc2ncc(Br)cc12 CCCC(C)CC(=O)NC1(C2CCCN2C(c2cc(C)cnc2C)=O)CC1 c1(C(=O)NC2(CN(C(c3cccc(OC)c3)=O)C)CC2)ccc(=O)n(C)c1 C(=O)(C(=O)C(C)(C)C)N1CCCC(C(C)NC(c2c[nH]nc2C2CCOC2)=O)C1 N1(C(C=CC=CC)=O)CCC(C)(CNC(=O)CCc2ncc(C)[nH]2)C1 c1(C2C(C(=O)NC(CNC(C(CC#C)C)=O)C)C2)ccc(F)c(F)c1 C12(CNCCC(=O)Nc3ccccc3)CC3CC1C2C3.C12CC1CNC2=O C1(C(C)(O)CNC(=O)CC2(C#N)CC2)CCCN(C(C2CCCCCC2)=O)C1 C(=O)(CC(C)C(F)F)NC(CC)(C)CCNC(c1cnc(O)o1)=O C#CC1(C(=O)N(C2CC(O)C2(C)C)C)CCN(C(=O)Cc2cnccc2C)CC1 C1(C(=O)NC2C(C)CC2C(C)C)(NC(=O)Cc2ccc(O)cn2)CCN(C)C1 C1(C(=O)NCC(CCC)OCC)CCN(C(=O)C2=C(C)OCCS2)C(C)(C)C1 N1(C(c2scc(COC)c2)=O)CC(OC)CC1CNC(=O)CN1CCCC(O)C1 C1(N(C(N(C2CCOC2)CC)=O)CCO)CCCN(C(C)(C)C)C1 C(=O)(C1=CC2(CCOC2)C1)N1C2CC(CNC(C3(CC)CCCC3)=O)CC1CC2 O=C1NCC2(CC(NC(C3C4CN(C(C5(CF)CCOCC5)=O)CC34)=O)C2)O1 N(C1CCCOc2ccccc21)CC(=O)NCCOc1ccc(Cl)cc1 c1(CC)nc[nH]c1C(=O)NCC(C)N(C(=O)CC1CNC(=O)O1)C c1(OC)ncc(C(=O)NC(C)CCN(C(=O)CCc2nccs2)C)c(C)n1 c1(C(=O)OC)cc(C(=O)NC2(CNC(=O)C(F)Cl)CCOCC2)ccn1 C(CCC)(C(=O)NCC1(CC)CCCC1)=CCC.C1(NC=O)CCN(C(=O)CC)C1 c1(C(C)OC)nc(C(=O)NCCCN(C(=O)CCCNS(C)(=O)=O)C)co1 CC1C(NC(c2cnc(O)c(N(C)C)c2)=O)CCCN1C(=O)CCSCC(N)=O C1(N(C(c2cc(OC)c(O)nc2)=O)C)CCC2CN(C(c3cc(F)c[nH]3)=O)CC12 N1(C(CC2CCC(OC)CC2)=O)CCN(C(c2cc(C)[nH]n2)=O)C(CO)C1 c1(C(=O)NC2CN(C(C(C)C3CC3)=O)CC2O)cc2c(s1)CCS(=O)(=O)C2 CCCC(C)(C)CC(=O)NC1CC2(C1)CC(C(=O)Nc1cnn(C(C)(C)C)c1)C2 CCC(CC(C)C)C(=O)N1CC(CNC(C2CN(C(N)=O)C2)=O)C(C)C1 O=C(CCCCCc1ccc(F)cc1)N(CC(O)CO)Cc1ccc(O)cc1 N1(C(CNC(C2(OCC)CCCC2)=O)=O)CCN(C(C2CC(C)(F)C2)=O)CC1 c1(OC)[nH]c(=N)nc2sc(C(=O)N(C)CCNC(=O)C(N3CCOC3=O)C)cc12 C1(NC(C(Cc2ccco2)NC(=O)C=CCOC2CC2)=O)CC2CC1C(O)C2O C1(C(N2CC(CCC=C)(C(=O)O)C2)=O)CC12CCc1cc(Br)ccc12 CCCCC(F)C(=O)N(CC1CC1)CC1CCCN1C(=O)C(O)CN(C)C N1(C(C(CC)OC)=O)CCC(CO)C(NC(=O)CCCCCn2cnnn2)C1 C1(C)(CNC(C(CCOC)OC)=O)CCCN(C(c2scnc2C)=O)C1 C1(CNC2C(c3ccc(F)cc3)CCCC2)CC12CCC(F)(F)CC2 C1(COC)(CNC(C2CC2C2CC2C)=O)CCCN1C(c1ccc(C#N)[nH]1)=O N1(C(c2c(C)n(CCO)nc2)=O)CC2CCN(C(C3CC4CCC4C3)=O)C2C1C C1(C(=O)OCCNC(C2CCC(NC(=O)OC(C)(C)C)C2)=O)CCC2(CC2)C1 Cc1nn(CC(=O)N(CCC(=O)NCCCCC2CC2C)CCCO)c(=O)o1 C(=O)(C1c2ccccc2C2CC1C2)NC(C)(C)CNC(c1cc2n(n1)CCO2)=O C#Cc1cncc(C(=O)NC(C)CN(CCCC(=O)NC(C2CCCC2)=O)C)c1 C(c1ccc(OC(F)F)cc1)=CC(N1CC(CNC(c2cc(OC)ns2)=O)C1)=O C12(C(=O)NCC3N(C(C4C5COCC45)=O)CCCC3)CC=CCN1CCC2 c1(C(=O)NC2CC3CN(C(C(CCC)C)=O)C2C3)cn2cc(Cl)cnc2n1 C(=O)(C(F)C(F)(F)F)N1C(CC(=O)N(C2CCC2)CCC)CC1 C1(NC(=O)CCSC(F)(F)F)CCCCN(C(C2CCC3CCC2O3)=O)C1 C1(C(=O)NC2CC(C)(NC(c3n(CCC)ncc3)=O)C2)CCCCC12CC2 c1(C(c2ccncc2)NC(=O)NCC2CC(C(F)(F)F)C2)nnc(S)n1C1CC1 Cc1cc(OCCCNC(=O)CSc2ccc(C)c(C)c2)ccc1F C(=O)(C(C)C(O)CC(C)C)NC(CC)(C)CCNC(=O)C(O)C1CCCC1 N1(CC)CC(C(=O)N(C(C)CNC(c2cc(=O)n(C)o2)=O)C)NC1=O N1(C(c2cn(CCCC)nc2C)=O)CCC(C2CC2)(CNC(=O)C(F)CC)C1 N1(C(c2c(CC)n(C)cc2)=O)CCCC(NC(C2(C)CC=CCC2)=O)C1C CCC(CC)CC(=O)N1CC(C(=O)Nc2cccc(OCF)c2)CC12CC2 N1(C(C(C)c2cncs2)=O)CCC(NC(=O)CCc2cccc(F)c2)C12CCC2 C12CCCC(C1)NC(=O)NCc1cc2n[nH]1.c1(C(=O)OC)cc(C(F)(F)F)c[nH]1 c1(C(=O)NCCC23CN(C(C(C)CN(C)C)=O)C(CC2)C3)nc2ccccc2[nH]1 N1(C(c2c(C)cc(C)[nH]2)=O)CC2C3CCC(C2C1)N(C(=O)CN1CCC1C)C3 CS(=O)(=O)c1cc(Nc2ccc3c(c2)OCO3)ncn1 N1(C(CCC=CC)=O)CCC2(C1)C(=O)N2C.C(C)(C1CC1)OC CC(C(C)(C)NC(=O)CC1CC(C)=NO1)NC(=O)COC1CC(F)(F)C1 N1(C(=O)OC(C)(C)C)CCc2cc(S(=O)(=O)NC3CC(CCO)C3)ccc21 N1(C(CC(C=C)C)=O)CCN(C(=O)Cn2nc(C)nc2C)CC1COC N1(C(Cc2c(C)nn(C)c2Cl)=O)CCN(C(=O)CCN2CCCC2)CC(C)(F)C1 C12(CNC(NCC3(C)ON=C(C)C3)=NCC3CCC3)CCCC1CC(=O)N2 N1(C(c2c(CC)ncs2)=O)C2CCC1CC(CNC(=O)CSc1ccncc1)C2 C1(C(=O)N(C(C)CC2CC2)C)(CC)CCCN1C(c1ccoc1)=O c1(CN2CC(NC(c3ccc(OCC)cc3)=O)C(O)CC2)ccc(F)c(F)c1Cl C1CCC2(C1)C1C(N3CCN4C(=O)CCC4C3)COC2C1 CC(C)C(F)(F)CC(=O)N1CCC(NC(c2ccc3nccn3c2)=O)C(C)C1 c1(OC)cnc(NC2CCCC2C(N2CCC(F)C2)=O)nc1 N1(C(c2ccc(N(C)C(=O)OC(C)(C)C)cc2Cl)=O)CCC(C2CC2)(C(=O)O)C1 C1(F)(C(N(CCOCCCN(C(C2CC(SC)C2)=O)C)C)=O)CCCN(C)C1 C1(NC(C(CCSC)OC)=O)CCC(F)(CNC(=O)C=CC(=O)N(C)C)C1 CC1CN(C(=O)CCCc2cnn[nH]2)CC(C)N(c2cc(C(N)=O)ncn2)C1 Cc1c(C(=O)NCCNC(=O)Cc2cccc(F)c2Br)cc(N)cc1O Cc1cc(Br)c(NC(=O)Cc2cc(-c3ccnc(Cl)c3F)ccn2)cc1[N+](=O)[O-] C1(NC(C(C)C(C)(C)C)=O)CN(C(=O)Cc2cc[nH]n2)C2(CCCCC2)C1 N1(C(c2sc(C)c(O)n2)=O)CCCN(C(C2CC(C)CC(=O)N2)=O)C(C)C1 C1(NC(CCCCCOC)=O)CC2CCC1CC2NC(c1cc(C)c(C)[nH]1)=O C1(C(=O)NC(c2cccnc2)C(N2CCC(C#C)C2)=O)CC12CCOCC2 C(=O)(C1CCOc2ccccc21)NC1C(NC(COCCC(C)C)=O)CCC1 C1(C(=O)NCc2cccc(C(C)(C)O)c2)CC2(CCOCC2)CCO1 c1(NCC(CC(C)C)CCO)[nH]c(=NCc2csnn2)nc2c1ncn2C C(=O)(C1=CC2(CCOC2)C1)NC1(CC=C)CN(C(=O)Cc2cccc(Br)c2C)C1 Cc1nnsc1C(=O)NCC1CC(CNC(C2CCCN2C(C)C)=O)C1 C1(CC(=O)NCC#CCCO)CCCC1NC(=O)CN(CCO)CCO c1(C(N2C(CNC(c3cnn(C)c3N)=O)CCC2)=O)ccc2c(c1)CCC(=O)N2 C(=O)(C1=COCCC1)N1CC(NC(=O)CNC(=O)NCC2CC2)C2C1C2 c1(CCC(=O)N(CCNC(C2CCC(CC)CC2)=O)CC)c(C)nc(O)nc1O Cc1cc(Cl)c(C(=O)N(C)C)cc1[N+](=O)[O-].C1(Cc2cncn2C)C(=O)N1 N1(C(c2cc(C)ccn2)C(=O)Nc2cccc(OC)c2)CCSCC1(C)C CC(C)CCCCCC(=O)NCC1CC2CCC1N2C(=O)CN1CCC1C c1(OC)c(C(=O)NC2CCC(C)N(C(=O)Cc3ccc(C)o3)C2)ncnc1C CCC(C)C(C(=O)N(CCCNC(C1CS(=O)C1)=O)C1CC1)OC c1(OC(C)(C)C)ccc(C(=O)CNC(=NCC)N(C)SC2CC(OCC)C2)cc1 C12(CNC(CC3(C)CCCO3)=O)CC1CN(C(c1cccnc1Cl)=O)C2 N1(C(c2cc(C)no2)=O)CCOc2ncc(-c3ccc(C)c(CO)c3)c(C)c21 N1(C(COCCCC)=O)CCC2(CC1)CN(C(C1(C(C)(F)F)CC1)=O)CC(C)O2 C=C=C(C)CC(=O)NC1CN(C(=O)CN(C(C)=O)C2CC2)C1 C1(C2CCN(C)CC2)(C(=O)NC2CC3(C(NC(c4cnc(OC)s4)=O)C3)C2)CC1 CC1(C)OC2(C(N3CCCC3CNC(=O)CC3=CCCC3)=O)CC1C2 CN=c1nc(N2CCC(OCC(F)(F)F)CC2)[nH]c(=NCC(F)(F)Cl)[nH]1 n1(CC)cnc2c(NCCS(=O)(=O)N(C)C)nc(N3CCC=C(Cl)C3)nc12 c1(C(=O)OC)cnc(C(=O)NC2CCC(NC(=O)CCC3(C)CCC(=O)N3)C2)cn1 Cc1c(C(=O)NC(C)CNC(c2ccc(-c3ccccn3)o2)=O)nnn1C(C)C N1(C(C2N(C)C(=O)OC2)=O)C2CC=C(C(=O)NCC3CC(O)C34CCC4)C1CC2 c1(-n2c(C)nnn2)ccc(NC(C2(c3ccc(CC4CC4)cc3)CC2)=O)cc1 CN1CCc2ccc(NC(=O)C(O)C3CC3)cc2C1.c12ccc(cc1)CN2C CC1CC(=O)NC1C(=O)NCCCN(C(c1ccnn1CCC(F)(F)F)=O)C1CC1 C(CCN(C(=O)C(C)C1CCCC1)C)(C(C)(C)C)NC(C(C)=NOCC#N)=O C#CCC(CC#C)C(=O)NCC1CCN(C(=O)C2=NOC(C)C2)CC1(F)F CCCC(CCC)C(=O)NC1CC(NC(=O)CC(C)C(=O)OC)CC1O C1(C(=O)NCCOCCC)CCN(C(=O)CCCC2CC2C)CC1O C1(NC(C=C(C)C(C)(C)C)=O)CCC(C)(C)CC1CNC(c1occc1Br)=O CCCCCCCCCC(=O)N1CC(NC(C2CNC(=O)N2)=O)CC12CCC2 C(=O)(C1=Cc2ccccc2C1)N1CC(F)CC(NC(=O)Cc2cncs2)C1 C12(C(=O)NC(C#C)C(C)OC)CCC(CC1NC(c1ccncc1)=O)C2 C#CC1(O)CCN(Cc2ccc(I)c(F)c2)C1 Cc1ccc2nonc2c1C(=O)NC(C1CN(C(=O)CNc2ccsc2Cl)C1)C c1(CN2CC3C(CNC(=O)NCc4ccccc4)C3C2)c(F)ccc(Br)c1F C1(CC=C)(C(=O)NCC(c2ccccc2)NC(=O)Cc2cocn2)CCOCC1 c1(C(=O)NCC2C(NC(CCC)=O)CCC2)ccc(N)c(C(F)(F)F)c1 C1(N(C(Cc2cc(C)no2)=O)C)CCC(NC(c2ccccc2Br)=O)CC1 C1(CNC(c2cnn3c2CCC3)=O)CC2(CO1)CN(C(C1CCCC1)=O)C2 c1(CNC(C2C(C)=CCS2)=O)ccc(CNC(=O)C(c2ccccc2Cl)O)cc1 c1(C(=O)NC2C(NC(C3C(COC)C3)=O)C2)c(C)nn(-c2cccc(Cl)c2)c1C c1(OC)ccc2c(c1)NC(=O)C2CC(=O)NCC=CCNC(C1CC(CF)C1)=O N1(C(C2CC(N(C)C)C2)=O)CC2CCN(C(c3ccccc3CC#N)=O)C2C1 C1(F)(CNC(C(C)OCC#C)=O)CCN(C(C2(C)CC2(C)C)=O)CC1 CN1CCNC(=O)C12CCCN(N1CCC(c3cccnc3)C1)C2 C1(C(N(CCNC(C2(COC)CC2(F)F)=O)C2CC2)=O)CC2(C1)CC21CCC1 N1(C(c2n(C(C)C)ncc2F)=O)CCC2(CC1)CN(C(=O)CC1CC13CC3)C2 C1(CCN(CC)CC)CCN(c2ccnc(NCc3ncco3)n2)CC1 CC(C)CCCC(=O)NCC12CC1CN(C(=O)CCC1NC(=O)NC1=O)C2 C1(CC)CC1(C)C(=O)NCCC(C)NC(=O)COCCCC(C)C c1(NC)cnccc1C(=O)NCC1(OC)CCN(C(=O)CN2CCC(C)CC2)C1 C1(N(CCNC(c2cccc(COC)c2)=O)CC)CCS(=O)(=O)CC1 CN1CC(C(=O)Nc2cn(C)c(C(N3CCC(C#N)C3)=O)n2)CC1=O C(=O)(CC(F)(F)CC(=O)N1CCC(C)N(C(=O)CCCCN(C)C)CC1)OC CCC(C)C(C(=O)N1CC2CC1(C(=O)NCc1ccc(CO)o1)C2)N(C)C N1(C(CCC(C=C)C)=O)C2CCCC1CC(NC(c1nc(Br)c(C)s1)=O)C2 c1(CC)cn(OC)cc1C(C)NC(c1coc(C)n1)c1nnnn1C(C)(C)CC c1(OC)ccccc1CC(N1CC(O)(CNC(=O)C(C)OCC(C)C)C1)=O n1(CCCC(=O)N(CC(C)NC(C2CC(C)(O)C2)=O)CC)nc(C)nc1C C(C(C)(C)C(C)(C)O)NC(COC1CC(C(=O)NC2C(CC)(C(F)F)C2)C1)=O C=C(C)C(C)(O)C(=O)N1CCCC(O)(CNC(c2cn(C)nc2CC)=O)C1 CCCCC(C)CCC(=O)NCC1C2CC1N(C(c1sc(C3CC3)nc1C)=O)C2 O=C(C1CCCc2nn[nH]c21)NC1C=CCN(C(c2nc3c(s2)CCCC3)=O)C1 C(=O)(C1=C2CCCN=C2NN1)NC(C)CN(C(=O)C(F)(F)C1(O)CCC1)C N1(C(c2n(C)ncc2Br)C(=O)NC2(C)CC2)CCc2sc(Br)cc2C1 Cc1cc(Cl)cc(C(N2CC3CCCC2C3CNC(c2ccc(F)o2)=O)=O)c1N C1(CC#C)(C(N2CCN(CC)CC2)=O)CCN(C(=O)CCc2c(C)n[nH]c2C)C1 c1(C(N2CC(NC(C=C(CC)CC)=O)C(C)C2)=O)cc(Br)c(O)cc1F CN1CCC(C(N2CC3(NC(=O)CN4CCCCCC4)CC2C3)=O)CC1 C1(F)(C(=O)NCC2(NC(c3n(C(C)C)ccc3)=O)CCCC2)CCOCC1 C1(CNC(CC2(COC)CCCC2)=O)CCCN(C(c2ccncn2)=O)C1 C1(NC(CSCCOC)=O)CCCC(C(=O)N(CCCC(C)(F)F)C)CC1 c1(CC)n[nH]c(=NC2CC(CNC(c3cc(C)nc4ccnn34)=O)C2)o1 CCC(CCCO)NC(C1CC=CCN1C(=O)CCCCNC(N)=O)=O CON(CCC(=O)N(C(C)C(C)C)C1CC1)C(=O)CN1C(=O)CNC1=O N=c1nc(O)c(CC(N2CCC(NC(c3ccsc3)=O)C23CC3)=O)c[nH]1 c1(N2CCC(CCNC(C(CC)Sc3ccccc3)=O)CC2)nc(C#N)c(Cl)s1 c1(C(=O)NC(CN(C(COCCCC)=O)CC)C)cnc(C(C)(C)C)o1 C1(CCC(=O)NCC=C(C(=O)N(CCCOC)CCO)C)CCC(=O)C1 C1(C)(NC(C2C(C)C2)=O)CCCN(C(C2C(C)(C)C2(C)C)=O)C1 n1(CC(C)C)cc(OC(c2n[nH]cc2NC(=O)OC(C)(C)C)=O)cn1 C1(C(=O)NCCN(CC)CC)CCCN(C(=O)C(CCOC)OC)C1 N1(OC)CCC2C1CCCN2C(=O)CCn1cncn1.c1(C)ccccc1CN CCCCCCC(C)C(=O)NC1(C)CC(NC(c2cc3cnccc3[nH]2)=O)C1 c1(CCC)nc(=NCC2(O)CCN(C(=O)C(C)CF)CC2)s[nH]1 Cc1nc(C(N2CCCCC2CCCNC(=O)CN(C)C2CC2)=O)c(=O)[nH]c1C C(=O)(CCCC(=O)NC1CCN(C2CC2)CC1)NCC(C)N(CC(F)F)C c1(C(=O)NCC2(F)CC(NC(c3cc(OCC)n[nH]3)=O)C2)sc2nccn2c1C c1(OC)cc(C(=O)NCCC2CCC(NC(=O)CCC(C)SC)C2)ccc1F c1(C(N2C(CCNC(CC(C)SC)=O)CCC2)=O)ncnc(O)c1Br N1(C(C(C(C)(C)O)F)=O)CCc2c(CNC(C3CCS3(=O)=O)=O)cccc2C1 N1(C(CC(C)OC)=O)CCOCC1C(=O)NCc1nnnn1C1CC1 c1(-c2nnc(N3CCC(C)(CC)CC3)n2CC2CC2)cc2ccc(Br)cc2s1 C(=O)(N=c1ncn(C(=O)OC)[nH]1)c1nc(CCC)nn1C N1(C(c2c(C)[nH]c(=N)s2)=O)CCC2(C1)CN(C(c1ccc[n+]([O-])c1)=O)C2 C(=O)(CC(O)CNC(=O)C1=COCC1)NC(c1cnsc1)C C=CC(C)(C)CC(=O)N1CCOCC1CCNC(C1CC2(CCC2OC)C1)=O C1(C)(C(N2C(CNC(CCc3cnc(C)o3)=O)CCC2)=O)CCC(=O)C1 Cc1cccc(CN2CC(NC(C3CC3c3ccccc3)=O)C(O)C2)c1Cl C1(C(N2CC3C(CNC(C4(COC)CC=CC4)=O)C3C2)=O)CCCCCS1(=O)=O CCC(CC(=O)NC1CC2CCC1N2C(=O)Cc1ccoc1)C(C)(C)C c1(OCC)ccc(N(CC(O)CC)C)c2ncccc12.c1(CN)ccccc1 C#Cc1cccc(CC(N2CCC=CC2C(N2CC(C3CCCO3)C2)=O)=O)c1 N1(C(C2CCC(=O)O2)=O)CCCN(Cc2cscc2Br)CC1 C#Cc1ccc(C(=O)N(C2CCC(NC(c3ccc(N)c(Cl)c3)=O)C2)C)c(F)c1 c1(C(N2CCC(CC=C)(NC(=O)C(C)C(C)(C)O)C2)=O)nc(C)c(C)[nH]c1=O c1(CCC)c(C(=O)NC23CC(NC(C4OC(C)CC4C)=O)(C2)C3)cnn1C c1(N(C(=O)C2=CCCN(Cc3ccccc3)C2)C)nc2ccc(C#N)cc2[nH]1 C1(C(N(C2CN(C(c3c(C)sc(Cl)n3)=O)C2)C)=O)Cc2cccc(C)c2O1 C(=O)(C(C)(C)CCC#N)NC(C(C)NC(C(CC1CCCC1)OC)=O)CO c1(C(N2CC3CN(C(C(c4ccccc4)C)=O)CC32)=O)cc(Br)c(O)cc1O C1(NC(c2c(C)coc2)=O)CCCC(CC(N2CCCCC2C(C)CO)=O)C1 Cn1nc(O)cc1C(=O)N(C1CCCCC1)CCNC(c1occc1C1CC1)=O C1(CNC(CC2(C)CCCO2)=O)CCC2(CN(C(=O)CCNS(C)(=O)=O)C2)O1 C(=O)(C(CCCC)NC(=O)C(C#N)CC)N(CC(CC=C)(F)F)C C(=O)(C(=O)C(F)(F)F)NC(CCNC(Cn1c(C)ncc1)=O)C(C)C Cc1ccc(CC(N2CCCCC2CCNC(c2cccc(F)c2)=O)=O)c(Cl)c1 CCC(CC(F)(F)F)C(=O)N(C)Cc1cn(-c2cc(C#N)c(Cl)cc2F)nn1 c1(C(N(CCC(C)NC(C(CC#C)C2CC2)=O)C)=O)cc2c(C)cc(Cl)cc2[nH]1 N1(CCOc2ccnnc2)C2CCC1CC(C(=O)Nc1ccc(C)c(C)c1)C2 c1(CN(C(C2(C#C)CC2)=O)C)ccc(CNC(c2n[nH]c(C)c2F)=O)cc1 CCC(C)(C)CC(=O)N1CCOCCC1C(=O)NC(CC1CC1)CO C(CC(C)(C)C(=O)N1CCCN(C(c2nccc(OC)c2N)=O)CC1)SC Cc1cc2nnc(CNC3(CC(C)Oc4ccccc4)CC3)n2cc1C c1(OCC)ccc2c(c1)CCN(C(c1ccc(CO)o1)C(=O)NCCCSC)C2 C(CCC1CC1)(C(=O)N(C(CCC)COC)C)NC(c1cc(COC)on1)=O c1(N2CCN(C)C(CO)C2)nc(N2CCOCC(F)(F)C2)c2c(n1)CCCCC2 N1(C(CC2(C#N)CCC2)=O)CCN(C(c2cccc(Cl)c2F)=O)C2COCC12 c1(N2CCC(NC(C)=O)C2)cnc(Cl)cc1NCc1cc(OC(C)C)ncn1 N1(C(c2c(C)cncc2C)=O)CC(O)(C2CCN(C(=O)C(C)CS(C)=O)CC2)C1 CCC(C)(CO)C(=O)NC1CC(CCNC(c2ccnn2-c2cccnc2)=O)C1 c1(C(CC)NC(c2cc(SC)[nH]n2)=O)ccc(NCCOCC2CC2)cc1C C1(CN(c2cnc(C)s2)C(=O)C(C)Br)CC2(CNC2)C1 c1(C(N2C(C(=O)NCCC3(COC)CC3)CC2C)=O)ncc(C)cc1F N1(C(c2nc(CNC(C3C4CCC(F)C34)=O)oc2)=O)CCOC2(CC2)C1 c1(OC)ccc(C(=O)NCCC(C(C)C)NC(=O)CC(C)F)cc1C1CC1 c1(C(=O)NCCCNC(c2cscc2C(F)F)=O)cccc([N+](=O)[O-])c1O Cc1ccncc1C(N1CC(NC(=O)Cn2nnc(-c3ccco3)n2)C2CC12)=O N1(C(COCCCC#C)=O)CCC(CNC(=O)CCC2CCN(C)C2)C1 N1(C(CN(C(=O)OC)C)=O)CCCC2CCN(C(C3CCS(=O)CC3)=O)CC12 c1(N(CCC)Cc2cccc(F)c2)ccc(C(=O)COC(C)=O)cc1 CCC(C)CC(=O)NCC1CCC(F)(CNC(C2(SC)CCC2)=O)C1 C1(C(N(C)CC2N(C(COCCOC)=O)CCC2)=O)CC(C(C)(C)C)=NO1 c1(CCC(=O)NC(c2cn(C)nn2)C)ccc(S(=O)(=O)CCO)cc1 c1(C(=O)NCC2COCCN2C(=O)C2=CCSC2)cc2n(n1)CCCCO2 N1(c2nc(C)cc(N3CCC(NC(CC)=O)C3)n2)CCCC2CNCC12 N1(C(c2occ(C)c2)=O)CC(O)CC1C(N1CCC(O)(C(C)C)C1)=O Cc1nc(-c2cc(-c3csc(NC(=O)C(N4CCC(C5CC5)C4)=O)n3)cs2)cs1 CC(C)(O)C(C)(C)C(=O)N1CCC(C(=O)NCc2ccncc2F)C(C)(C)C1 CN1C(=O)CCC1C(=O)NCc1cccc(CNC(C23CC4CC2C3C4)=O)c1 Cc1cccc(C)c1NC1(C(=O)NOC(=O)C(C(=O)C2=NNC(C(F)(F)F)C2)C)CC1 N1(C(c2c(CC)n(C)nc2)=O)CCC(NC(=O)COCC2CCCOC2)C(C)C1 N1(C(c2c(C(N)=O)nccc2)=O)CC(NC(=O)C=Cc2cocn2)CC(F)C1 c1(NC(C(N2C(CCC)C(=O)NCC2)=O)=O)ccc2cccc(F)c2n1 CC(C)(CC(=O)NCC1CC12CCN(C(c1cn[nH]c1)=O)CC2)C(F)(F)F CCC(CC(C)C)C(=O)NC(CN(C)C(c1ccccc1OC)=O)(CO)CO c1(C(C)=O)ccc2c(c1)CCN(c1cc(NCC(C3CC3)N(C)C)nc(C)n1)C2 Cc1cccnc1C=CCNC(N1CCC12CC(C(F)F)C2)=O c1(O)ccc(F)c(SC)c1.C(=O)(C(CNC(=O)CCCF)c1ccccc1)OC(C)(C)C C1(CN(C(CCCSC)=O)C)COCCN1C(c1cc(-c2ccco2)cs1)=O C1(CC(=O)NCC(CCOC)NC(=O)CCn2cccn2)CCCC(=O)N1 C1(c2onc(-c3nc(C)c(C)s3)n2)CC2(CC(c3nn[nH]n3)C2)C1.C(C(=O)NC)O N1(C(c2cc(CC)no2)C(=O)NCC2CC2)CCC(C2CCCC2)C1 N1(C(=O)NC23C(CC(=O)N2)CCC3)CCC(=O)N2Cc3ccccc3C12 c1(C(N2CC(NC(C(C#C)(C)C)=O)C(C)C2)=O)c[nH]c2cc([N+](=O)[O-])ccc12 c1(C(N(CC(=O)NCCCN(C)C)CC#C)=O)cncc(OCC)c1 C1(CNC(C(C)Sc2ccccc2)=O)CCC(F)(CNC(=O)CC(=O)NCC)C1 C1(COC)(CNC(c2cncnc2)=O)CCCN1C(=O)Cc1ccc(OC)nc1 c1(C(=O)NCC2C(NC(Cc3cc(C)no3)=O)C2)cc(Br)cc(C)c1N c1(C(=O)NCCN(C)C(c2cccn3cncc23)=O)cc2sc(N(C)C)nc2s1 C1(C(N(CCN(C(Cc2c(C)n[nH]c2C)=O)C(C)C)C)=O)OC(C)(C)OC1(C)C C1(CNC(c2c(CC)non2)=O)C2CCC1CN(C(C1CC3(C1)CC(O)C3)=O)C2 c1(C(N2CC(CC)(NC(=O)Cc3occc3C)C2)=O)cc(O)ncc1F C1(O)(NC(CCNC(=O)NC)=O)CCN(c2ncc(Cl)c(C)n2)CC1 c1(OCC(=O)NCC(CN(C)C(=O)NC2COC2)O)cnn(C)c1 C1(NC(c2n(CC)ccc2)=O)COCCN(C(=O)CNC(=O)CN(C)C)C1 C1(CC(=O)NC2COCC2O)CN(Cc2ccnc(C(F)(F)F)c2)CCO1 c1(C(N(C(CC)C)C2CC2)=O)ccc(CNC(=O)C=NOC)nc1 C1(C)(CC)C=C(C(=O)N(CCC(C)(C)NC(c2cc([N+](=O)[O-])c[nH]2)=O)C)C1 c1(CC(CO)N(C(CN(c2ccccc2)C(C)C2CC2)=O)C)cccc(Br)c1 CC1C(=O)N(CC(N2CCC(N(c3ncnc4c3CCC4)C)C2)=O)C(=O)C1C c1(-c2ccc(C(N(C)Cc3cccc(Br)c3)=O)nn2)cc(F)ccc1F C1(NC(C2C=CCN(C(C(C=C)(F)F)=O)C2)=O)CC(C)CCC1O C12(C(=O)NCCCCN(C(c3n(CC)cnn3)=O)C)CCCN1CCC2 CC1CCN(C(=O)CC2(O)CC3CCC2O3)CC1CNC(=O)CCCC1CCC1 CN1C(=O)CCC1C(=O)NC1(CNC(=O)C=CCN2CCCC2CO)CCC1 c1(C(=O)NC2C3(CC(NC(CCS(C)(=O)=O)=O)C3)C2)cnc2cc(O)ccc2c1 S(=O)(=O)(CCC(=O)NC1CCCC1CNC(=O)Cc1csnn1)N(C)C N1(C(=O)NC(C(COC)C)C)CCN(Cc2ccccc2)CC1(C)C c1(C(=O)NC(C(C)NC(c2c(C)scc2)=O)CO)nn(C)cc1Cl Cc1cc(C(N2CCC3(NC(c4cccs4)=O)CC3C2)=O)n2nc(C)c(C)c2n1 C(C(C)C)(C(O)C(=O)NCC1CC2(CC2)CN1C(C1CC(F)(F)C1(C)C)=O)OC C1C(CSC2CC2)C(=O)N1.CC1CCN(CC(=O)NCC2CN(C3CC3)C2)C1 C(C(C)CN=c1cc(CCN(C)C)nc(Cl)[nH]1)Sc1nnc(C)s1 c1(C(C)NCCCOc2cccc(F)c2)cc(Br)c2occc2c1 N1(C(CC(CC)(C)C)=O)Cc2ccnn2CC(NC(c2cccc(CO)n2)=O)C1 C(=O)(CC1C(=O)N(C)c2ccccc21)NCC(C)N(C(C(CCSC)(C)C)=O)C C12(C(=O)NC34CN(C(COC)=O)C(C3)C4)CCCC(=O)N1CCC2 c1(CC(C)C)ccc(C(=O)N(C(c2ccccc2)CNC(C2CC2F)=O)C)[nH]1 N1(C(C2CC(C)C2)=O)CCC2(C(=O)NCC(C)CCCO)CCCC12 c1(C(=O)NC2CN(C(=O)CSC3CC3(F)F)C2)nccc2[nH]ccc12 N1(OC(C(C)NS(CC)(=O)=O)=O)CCC(C)C(C(F)(F)F)C1 c1(C(N(CC(C)O)CCNC(c2cnc(CCCC)s2)=O)=O)cc2occc2[nH]1 CCCCCCC(C)CC(=O)N1CC(O)(CNC(c2ccncc2N)=O)C1 C#CCCCCCC(=O)N1CCC2CC2(NC(=O)Cc2cnc(C)o2)C1 N1(C(C(C)(O)C2CC2C2CC2)=O)CC=C(C(=O)N2CCCC(F)CC2)C1 N1(C(C2CCC(NC(CCC)=O)C2)=O)CCOC(F)C1 c1(C(N2C(CCC#C)CCC2)=O)cc2ccccn2c1 C1(C(=O)NCC(CN(C(=O)CC2CCCCO2)C)(C)C)CC(=O)N(O)C1 c1(C(N2CC(C)(C(=O)NC(C=C)(C)CC)C2)=O)cc(CC)ncn1 c1(OC)cc(C(=O)NCC2COC(C)(C)CN2CC(=O)N(C)C)c2c(c1)CCC2 N1(C(=O)OC(C)(C)C)CC2CC1(C(=O)OCC1COC1)CO2 CC1COC(C(=O)N(O)Cc2cn(-c3ccc4c(c3)OCO4)nn2)c2ccccc21 N1(C2C(NC(C3C(C)OCO3)=O)CCC2)CCC(F)(F)CC1 C1(O)(CCNC(=O)NCCCCSC)CCOC1 C(=O)(C1CCCn2cnnc21)N1C(CC)C(NC(=O)C(C)=C(C)C)CC1 c1(CC)[nH]nc(C(=O)NCC(C2CC=CCC2)NC(=O)C)c1Br.CC(C)(C)C1CC1 c1(NC(CNC(C2CC3CC3C2)=O)CC(F)(F)F)ccc([N+](=O)[O-])cc1F C1(NC(C2(C)ON=C(C)C2)=O)CC2CC1N(C(c1nc[nH]c1C(F)(F)F)=O)C2 N1(C(C2(C)COCCO2)=O)CCC=C(C(=O)NC2CC3(CCC3)C2CO)C1 Cc1ncc(C(N2CCC2CNC(C2(C(F)F)CCCO2)=O)=O)s1 C12(NC(C3CN(C(C)=O)C3)=O)CCC(CNC(C3C4COCC34)=O)(CC1)OC2 N(C(=NCCCOC(C)C)NCC(C)C(F)(F)F)C1CCN(C(=O)OC)CC1 c1(CNC(C2(c3c(Cl)cccc3Cl)CC2)=O)cc(Cl)ccc1[N+](=O)[O-] N1(CC(C)NC(C2C(CC)C2)=O)CCN(C(=O)CC=CCl)CC1 C1(CNC(Cc2ccn(C)n2)=O)CN(C(=O)Cc2cccnc2)CC1O C1(CC)(NC(c2cnoc2-c2ccco2)=O)CN(C(=O)C(n2ccc(C)n2)C)C1 c1(CC)cncc(C(N2CCN(c3ccc(C(N)=O)cn3)CC2)=O)c1 C1(NC(CCOCCCOC)=O)CN(C(C2(Br)CC2(F)F)=O)CC1C C1(NC(C(CCOC)NC(=O)CC2CCCC(=O)N2)=O)CC2(COCCO2)C1 N1(C(CC(CC)C)=O)CC(C)(C)CC1CC(=O)NCC(C)(O)C1CCC1 c1(C(=O)NC2CC(C)(C(=O)NC3CC(F)(F)C3(C)C)C2)n[nH]c2c1CCC2 c1(C(N2CCCC(C)(CNC(c3n(CC)ncn3)=O)C2)=O)csc2c1CCCC2 C(C(C)C(F)C(=O)N1CCC(N(C)C)CC1)NC(Cc1nc(C)[nH]n1)=O C(CC(O)C(=O)NC(c1ccccc1)C(N1CCNC(=O)C1)=O)SC c1(C(C(=O)NCCCC)N(C2CC2C)C)cnn(CCO)n1 N12CCOC(C1)C2=O.n1(C2C(C(=O)NCC3(CSC4CCC4)CC3)C2)cccc1 C(=O)(CCC(=O)NN(C)C)N1CC(O)CC(NC(c2cc(C)n(C)c(=O)c2)=O)C1 C(=O)(CC(C)(C)C(F)F)NCCOCCN(C(c1c(CC)con1)=O)C N1(C(C(CCC)(C)CC)=O)CCn2c(CNC(c3ncnn3CC)=O)nnc2C1 c1(-n2cc(CCCN)nn2)ccc(C)c(F)c1F.C(C)(C(=O)NCCS)SC C1(CN(CCNC(C(CC)C)=O)C)C2C3CC4C1C1C2CC3C41 c1(CNC(C2CCCN2C(=O)CC(O)c2ccccc2)=O)cc(Cl)cc(Cl)c1O c1(CNC(C2(c3ccc(OC)cc3)CC(O)C2)=O)ccc(OC)c2ncccc12 C1(C)(CN(C(=O)CSCC(N)=O)NC(CC(C)N)=O)C=CCCC1.C1(C)CC1 N1(C(C(CCC)OCC)=O)CC2(CCC2NC(=O)C=Cc2cncc(C)c2)C1 c1(C(=O)NC(C)CC2CN(C(=O)C(F)=CC3CC3)C2)cc(C(F)(F)F)ccc1F c1(C(C(=O)NC(CCCC)CNC(c2cnn(C)c2N)=O)O)ccc(F)c(Cl)c1 N1(CCNC(=O)CSC(F)F)CCC(NC(=O)Cc2cnoc2)CC1 c1(C(=O)NCC2N(C(C(F)OC)=O)CCC2)cc(C(C)C)nc2ccccc12 c1(C(N2CC3C(NC(CCc4ccc(C)s4)=O)(C3)C2)=O)cccc(C)c1F CC1(C)CN(C(=O)CC2(N3CC4CC4C3)CC2)CC1NC(C1CC=CCO1)=O C(=O)(C1=C(F)CN(C(=O)C(C)C(F)F)CC1)NCc1cnc(C)n1C C1(CNC(c2n(CCCCCC)nnn2)CCC2OCCO2)CCCOC1C CC(C)CC(O)C(=O)N1CCCC(C)(NC(c2cc(CC3CCC3)c[nH]2)=O)C1 C=C(Cl)CCC(=O)NC1CCCN(C(c2cnc(C)s2)=O)C1 Cn1nnc(CNC(=O)CC2CCCN2C(=O)Cc2cncs2)n1 C1(NC(=O)CC2CCCC2(F)F)CCCN(C(=O)C(c2ccccc2)=O)CC1 CC1=C(C(=O)N2CCC(F)(CNC(=O)CCc3ccccc3Br)C2)CCCC1 C1(NC(c2c(C)onc2)=O)CC2CN(C(C3CCC(OC(F)F)CC3)=O)CC2C1 C1(C)(CNC(C(CCC)CC)=O)COCCN(C(c2cnn(CC(C)C)c2)=O)C1 N1(C(C2CC(C(C(=O)C(F)(F)C3CC3)=O)CCO2)=O)CCn2ccnc2C1.N c1(C(CNC(=O)CSC2CC2)NC(=O)CCc2cc[nH]n2)cccc(Cl)c1 N1(C(c2c(CC(C)C)cccc2)=O)CC2(CCN(C(C3CCC(C)O3)=O)C2)C1 N1(C(CN2C(C)CSC2)=O)CCCC(c2cn(Cc3cnns3)nn2)C1 C(=O)(C1CCCc2nncn21)N(C)Cc1cn(-c2ccc(Br)cc2)nn1 CCCC(C(=O)N1CCC(c2ccccc2)(NC(c2cn(C)nn2)=O)C1)OCC c1(OC)c(N2CCCC(C)(NC(=O)CCc3cncc(C)c3)C2)ncnc1Cl C(C(C(C)(C)C)NC(C1C2CC1(c1ccc(Cl)cc1)CO2)=O)NC(C=C(C)OC)=O N1(C(C(C)(O)C2CC2)=O)CCC(NC(c2ccc3nccn3c2)=O)CC(O)C1 c1(C(=O)NCC(C(C)C)NC(Cn2c(C)cc(C)n2)=O)ccn(C(C)C)c(=O)c1 C1(CC(=O)NC(c2cccc(Cl)c2)C)C2CCCC2N1C(=O)CCc1cnoc1 CC1CNC(=O)CN1C(=O)C(C)(C)NC(=O)CC1CCOCC1 c1(CCC)nc(=NC(C)CN(C)C(c2ccc(C3CC3(F)F)cc2)=O)s[nH]1 N1(C(CCOC)=O)CC(CNC(c2cc(OC(C)C)cc(SC)c2)=O)CC1(C)C n1(CCC)cc(C(=O)NCCC2CCN(C(=O)CC(C)C)C2)cn1 Cc1nc(CC(C)C)c(C(N2CC3CC3(CNC(C3(n4cccn4)CC3)=O)C2)=O)s1 C(C(CNC(C1CCOC1)=O)CO)NC(c1ccc(SC(F)(F)F)o1)=O c12cnc(nc1)[nH]c2=O.C1(C(=O)OC)(CN(C(COCC(C)C)=O)C)CCC1 c1(C(N2CCC2CC2CC(CCC(=O)OC(C)(C)C)C2)=O)cccc(C(F)F)c1 C12(CCCCO1)C(=O)NC1CCN(C1)C2=O.C1(COC)CC(=C2CCC2)C1 c1(CC)ccc(C(=O)NC(C)C(C)NC(=O)C(C)Nc2nc(C)cs2)cn1 N1(C(C2C(C)CC2C)=O)CC2(CCCN(C(=O)Cc3ccnc(F)c3F)C2)C1 C1(OC)CCCN(C2CCc3ccc(Br)cc32)CC1 CS(=O)CCC(O)C(=O)NC1CCN(C(c2cnn(C(C)(C)C)c2)=O)CC1 C1(NC(c2scnc2C(F)(F)F)=O)CN(C(c2ncc(F)cc2F)=O)CC12CC2 N1(C(CCc2ccc(C)s2)=O)CC(CNC(=O)CN2CCCCC2C)C(F)(F)C1 c1(C(N(C2CCN(C(c3cc(O)cc(=O)o3)=O)CC2)C)=O)cnc2occc2c1 C1(C(N)=O)CCCCC1NCCc1ccc(Cl)s1 C1(N(C(CC=C)=O)C)CCC(NC(c2sc(-c3ncc[nH]3)nc2C)=O)CC1 C1(C(=O)NCC2C(NC(c3c(OCC)oc(C)n3)=O)C2)Cc2cc(F)cc(F)c2O1 c1(C(=O)NC(CC)CN(C(=O)CS(=O)(=O)CCOC)C)cn2ccc(C)cc2n1 c1(NC(C2CCCN(C(c3cncc(C#N)c3)=O)CC2)=O)ccccc1C(N)=S C1(NC(CN(C2CC2)CC)=O)CCN(C(=O)CCc2cncc(C)c2)CC1O n1(C(CC)C)nc(C(=O)NC(C)CCCNC(=O)C(C)(C)COC)cc1C C1(O)(CNC(c2c(C)ocn2)=O)CCN(C(c2csc3cncn23)=O)CC1 N1(C(C2CC(N(C)C(C34CCCC3C4)=O)C2)=O)CCc2cncnc2C1 C1(C(=O)NCC2C(OCC)CN(C(C=CCC)=O)C2)CCc2nncn2C1 N1(C(c2c(COC)cc[nH]2)=O)CC2(C)CC1(C(=O)Nc1csnc1OC)C2 N1(C(c2c(C(C)(C)C)cccc2)=O)CC2(CC2)CC1CNC(C1CCCOC1)=O c1(C(N2C3CN(C(C(CC=C)C)=O)CC2CC3)=O)ccc2c(ccn2C)c1 C1(c2cc(C(N3C(C(=O)NC4CC4)CCCC3)=O)on2)CC12CCOCC2 c1(C(N2C3C(c4cn(-c5c(OC)nccc5)nn4)C(C3)C2)=O)cc2sccc2[nH]1 C1(C)(C(=O)NCC2CCC(NC(CC=CCC)=O)C2)COCCO1 c1(NC(C2(F)CCN(C(c3c(C)cco3)=O)CC2)=O)cccc2c[nH]nc12 c1(C(=O)NC2C(O)CCN(C(C(C)CC(F)F)=O)C2)ccc2ccnn2c1 c1(C(N2C(C)(C)CC(NC(c3cccnn3)=O)C2)=O)cscc1S(C)(=O)=O c1(C(C)C)nc(Cl)cc(=NCC=CCNC(N)=O)[nH]1.c12ccc(cc1)NC(=O)C2 CCCCCCCCCCNC(C1CNCCN1Cc1cc(CC)ccc1Br)=O C(=O)(C(C)C(=O)N1CCCC(CC(N2CCC2(C)CC(=O)N(C)C)=O)C1)OC CC(=Cn1ccnn1)C(=O)N1CCN(C(=O)CCC(C)(C)F)CC1CC1CC1 CC(CCNC(C1C(CNC(C2(O)CCOC2(C)C)=O)C1(C)C)=O)C(C)(C)C n1(CC)cc(Cl)cc1C(=O)NC1C=CCN(c2ccnc(C3CC3)n2)C1 CC1(C)CN(C(C2(F)CCOC2)=O)CCC1NC(c1cc(Cl)c(N)cc1F)=O CC1CCN(C(c2cnn(C)n2)=O)C1C(=O)Nc1ccc(N(C)C)nc1 CP(C)(=O)CC(=O)N1CC(OCCC(=O)NC(C(N)=O)C2CC2)C1 c1(NC2CCC(C(=O)NC(c3ccc(Cl)cc3)CC)CC2)nc(C)ncc1Br N1(C(COCc2onc(C)n2)=O)CC(C)(C)CC1CNC(=O)CC1(O)CCC1 c1(-c2ccc(C(=O)NCCN(CC)Cc3nc(C)c(C)o3)o2)ccccc1Cl c1(OC)ccc(Br)c(C(=O)NC23CCN(C(=O)Cc4coc(C)n4)CC2C3)c1 N1(C(CSCCCC)=O)CCCCC(NC(=O)CCc2ccnc(C)n2)C1 Cc1cccc2cc(C(=O)NC(CNC(=O)CC3(C)CC3(Cl)Cl)CO)sc12 CC1CC(C(=O)N(CCCCCNC(=O)C=Cc2ncc[nH]2)C)C1(C)C N1(C(COc2ccc(CC(=O)O)cc2)=O)CCCCC12CCN(S(=O)(=O)CO)C2 c1(CC)cnc(O)c(C(N2CC(OC)C(NC(=O)Cn3cnc(C#N)n3)C2)=O)c1 C1(CCC)CC(C(=O)NCC2(OC)CCN(C(=O)CCCCF)C2)CCO1 Cc1c(NC(=O)C(CNC(C2CCC(C)=C(C)C2)=O)N(C)C)cccc1Cl C1(C(N2C(CN(C(C3(CC)CCCC3)=O)C)CCC2)=O)CCN(C)C(C)C1 c1(CC)cc(C(=O)N(C2CCN(C(=O)CN(C3CCCCC3)C)C2)CC)n(C)n1 CC1(C)C(NC(c2ccnc(C(F)F)c2)=O)CC1CNC(C1CC(C)(O)C1)=O N1(C(C(C)(O)C2CC2)=O)CCC(CNC(c2ccc([N+](=O)[O-])o2)=O)C(O)C1 C1(C(=O)NCCC2CCN(C(CNC(=O)OCC)=O)CC2)CCC(C)(C)CO1 CS(=O)(=O)C1CC(NC(C2CN(Cc3cc(O)cc(Cl)c3)CCO2)=O)C1 N1(C(C(CC)NC(C)=O)=O)CCC2CCN(C(c3cc(F)ccc3O)=O)C2C1 C1(NC(C(C(=O)OC)F)=O)CCCCN(C(c2cnc(C3CC3)[nH]2)=O)C1 c1(C(=O)NC2C(C)CN(C(C3(O)COC3)=O)C2)cc2c(F)ccc(F)c2[nH]1 C(N=c1cc(Cc2ccccc2)n(C)[nH]1)c1n(CCOC)nnn1 C1(C2CC2)(CNC(C2CCCC2O)=O)CCN(C(=O)CC2CSC2)C1 Cc1cc(Cl)c(NC(c2ccc(C(F)C(F)(F)F)cn2)=O)cc1Cl O=C1CCC(C(F)C(=O)NCCNC(C2CC=CCO2)=O)CC1 c1(C(N2CCC(CN(C)C(c3cc(N)cc(O)c3)=O)C2)=O)n[nH]c2c1COCC2 C(CC(C(=O)C(=O)C(C)N(C)C)OC)OC.C(CN)(CC)N C1(C(=O)NCCC2(O)CN(C(CC3CC(=O)NC3)=O)C2)CCC2(CCOCC2)O1 C1(C(=O)NCC(C#C)C(C)C)CCN(C(=O)C=Cc2nccs2)C(C)(C)C1 N1(C(c2ccc(S(=O)(=O)NC)o2)=O)CC(C)CN(C(c2csnc2C)=O)CC1C c1(NC2CC3CN(C(C(COC)C)=O)C2C3)cc2nc(O)oc2cc1[N+](=O)[O-] C1(CC(=O)N(CCCC)Cc2cn(Cc3ccc(Br)cn3)nn2)CCCC(C)C1 C1(CN(C(=O)CC2CCOC2)C)(NC(=O)OC(C)(C)C)CC1(C)C c1(C(=O)NC2(CC)CCCN(C(CCOCC)=O)C2)ccc2cnc(C)n2c1 CC(C)C(O)C(C)C(=O)NC(CC(F)F)C(=O)NC1CCCC1(C)C N1(c2nnc(C)o2)CCC(C2CCN(C(C3C4CCCC34)=O)CC2)C1 c1(CC(N2CCC(c3cn(CCCF)nn3)C2)=O)noc2cc(F)c(F)cc12 C(C(C(=O)NC1CCC1)N(C)C)OCC.C1(=O)CO1 c1(C2N(C(C=CC(=O)N(C)C)=O)CCC2)ccccc1F C1(C)(NCCN2CCCCC2)COC(=O)C1.c12cccc(c1)NC(=O)C(=O)N2C CCC(C(=O)NC)N.c1(C(=O)NCCCN(C(=O)OC(C)(C)C)C)ccc(C)s1 C1(OC)CC(CO)N(C(=O)CCC2CCN(C(c3nccs3)=O)CC2)C1 N1(C(CCCCOC)=O)CC2CCOC2(CNC(=O)C(C(C)C)NC(C)=O)C1 N1(C(CC2CC(NC(C)=O)C2)=O)CC(C)(C)CC1CC(N1CCC(CO)CC1)=O C1(F)(CNC(c2ccc(C(C)C)nc2)=O)CCN(C(c2ccc(Cl)cc2)C)CC1 C1(C(N2CCC(C)(N(C)CC)C2)=O)COCCN(C(=O)CC2COCC(C)O2)C1 C1(NC(COCC(C)C)=O)CCCCC1NC(=O)CCF NC(=O)CC(O)C(=O)N(C1CCSC1)C(c1ccco1)=O c1(C(=O)NCC2(NC(C3CCC(C)(C)C3)=O)CCOC2)cc([N+](=O)[O-])ccn1 C=CC(F)(F)C(=O)NC1CC(N(C)C(c2cc(-c3ccccn3)no2)=O)C1 Cc1cc(C(N2CC(O)CC2CN(C)C)C(=O)NCC(C)C)ccc1I CCCCC(CC(=O)N1C2CCCC1COC2)NC(c1cc(C)n(C)c1)=O c1(C(N(C)Cc2cn(C(C)Cc3ccccn3)nn2)=O)ccnc(C(C)(C)C)n1 CCC(C)C(C)NC(C)=O.C1CCOCCN(C)C(=O)CO1 C(=O)(CCCN(C)N=O)NCC1CN(C(c2n(CC)ccn2)=O)C1 CC1CCC(CNC(=O)CCCCCn2cnnn2)N(C(c2sccc2Cl)=O)C1 C1(OC)CCN(C(=NCCCCl)NCc2cnnn2C)C1 C1(CNC(=O)C(C)CNC(=O)CC2(C(=O)NOC)CCCC2)(C)CCCC1.C(=O)(NC)OC c1(C(N(CCCNC(C2COC(C)C2)=O)C(C)C)=O)ccn2nccc2n1 C1(CCC)(NC(C2CCC(=O)O2)=O)CCCN(C(c2csc(O)n2)=O)C1 C#Cc1ccc2c(c1)CN(C(=O)NCCc1ccccc1)CC2 C1(C(=O)NCCC2(O)CCN(C(c3c(CC)[nH]nc3Cl)=O)C2)COCC(C)(C)O1 C1(C(N(C)CC2CCN(CC)C2)=O)CCN(C(=O)CCOCC2CC2)C1(C)C Cc1oc(C(N2CCC(C(F)C(=O)NCc3ccsc3)C2)=O)cc1CO C1(c2onc(NC(C3C(C)C(=O)N(C4CC4)C3=O)=O)n2)COC2(CCCCC2)O1 N#CC1COCCN1C(c1ccc(CCC(N2CCC(CO)C2)=O)cc1)=O N1(C(C(CCC)F)=O)CC2CCC1CN2C(C1OC(C)(C)OC1(C)C)=O CC(C(=O)NC1CC(NC(c2cnn3ccccc23)=O)C1)C(C)S(C)(=O)=O CC(C)(CC(N)=O)NC(C1CC(F)CN1C(=O)CNC(=O)OC(C)(C)C)=O C(=O)(CC(C(=O)OC(C)(C)C)C(C)C)N1CCCC(CNC(C=CCCC)=O)C1 C=CCCCCC(=O)NC1CCC(C(=O)Nc2cccc(NC(=O)NC)c2C)C1 N1(C(C(C)SC)=O)CCCC1(C)NC(=O)C(N)CN1CCCC1 N1(CCNC(C=CC=CC)=O)CCN(C(C2CC(=O)N(C3CN(C)C3)C2)=O)CC1 C1(NCc2c(C)nc(Br)s2)CCC2(CCCOC2)C1 c1(C(=O)NC2(CC(=O)Nc3cncc(F)c3Cl)CCC2)ccc(F)c(Cl)c1 c1(CNC(=NCC(=C)C)NC(C)CC)cc2cc(Cl)cnc2o1 c1(CCN(C)C)cccc(C(=O)NC2C=CCN(C(c3csc(CO)n3)=O)C2)c1 c1(C(=O)NCCN(CCC)C(C2CC2CCOC)=O)cc(C2CCCN2C)[nH]c1 CCCCC(C)(F)C(=O)NC(CC(=O)N1CC2CC(F)CC2C1)C(F)(F)F C(=O)(CCCS(C)(=O)=O)NC1(C)CN(C(c2nccnc2C(F)(F)F)=O)C1 N1(C(CCC(C)SC)=O)CCC(F)(CNC(=O)CC(n2nc(C)cc2C)C)CC1 C1(C)(NC(C(C)N(C(c2cc(C)oc2)=O)C2CC2)=O)CCSCC1 CC1(C)CCC(CNC(c2cc(Br)cnc2N)=O)N(C(C2COCCO2)=O)C1 c1(CNC(c2sc(C)c(-c3onc4c3CCCC4)n2)=O)c(C)cc(O)nc1C c1(C(N2CC(C=C)C(NC(C3CC4CC4C3)=O)C2)=O)n[nH]c2ccc(C)cc12 Cc1ncccc1C=CC(=O)NC1CN(C(=O)CCc2cncs2)C(C)(C)C1 C1(CCC(=O)NCC(CC)OC)CCN(C(C2(CC)CCCC2)=O)CC1 N1(C(C2(OC)CCCCCC2)=O)CCC2(C1)CN(C(=O)CC1CCCCC1F)C2 N1(C(c2c(C)nc(Br)o2)=O)CC(CNC(=O)CC2CCCCO2)CC(C)(C)C1 c1(C(=O)NC(CN(C(c2cc3ccsc3s2)=O)CC)C)cnc(O)c(OC)c1 CC(c1ccccc1F)=CC(=O)NC(C)(CNC(C1CCCN1C=O)=O)C(C)C CCS(=O)(=O)CC(=O)N(C1CC(C#N)C1)CC(=O)NCCc1cocn1 C#CCCCCC(=O)NC(C)(C)CCC1CCN(C(C2(CCF)CC2)=O)CC1 c1(C(c2n(C(C)C)nnn2)NCCSCCO)cc(Cl)c(Br)cc1F N1(C(C=CCC)=O)CC2CCC(C1)C(NC(c1ncn3cc(Cl)ccc13)=O)C2 c1(N(C2CCN(C(=O)CC3C=CCC3)C2)C)ccc([N+](=O)[O-])cn1 c1(NC(C2C3CN(C(CCc4c(C)cccc4)=O)C2C3)=O)cc(C#N)ccc1Br CC(C)(C)CC(O)C(=O)NC(C1CCCC1)CNC(c1cc[nH]c2nccc1-2)=O N1(C(c2cc(C#N)cc(C(F)(F)F)c2)=O)CCOc2ccccc2C1CO C1(NC(C2CN(CC)C(=O)C2)=O)CC2(C1)CC(NC(=O)C(c1ccccc1)=O)C2 c1(C(=O)NCC(C2CCCC2)NC(C2C(C)CCO2)=O)cnc(N(C)C)c(Cl)c1 CC1=NS(=O)(=O)NC=C1C(=O)NC(CNC(C1CCC(=O)N1C)=O)C(C)(C)C C1(NC(C(CCC)CC)=O)CN(C(c2cc(OC)ncc2Cl)=O)CC1S(C)(=O)=O C(C(=O)N1OC2CCC1CC2)C1CCC(NC(C2C(C)CC(=O)N2)=O)C1 C12(CNC(C3N(CCC)CCCC3)=O)CC(CO1)N(C(=O)C=C(Cl)Cl)C2 c1(C(N2CC(NC(CC(CC)C(F)F)=O)C3(C2)CC3)=O)cnc2ccnn2c1C c12nccc(c1F)C(=O)C(=O)C(CC)O2.C1(C(N(CCO)CCOC)=O)(N)CC1 C(=O)(C1CCCc2n[nH]cc21)N(CC(CNC(C1(COC)CCOCC1)=O)O)C c1(OCC(=O)NCC#CCNC(CC2CCC(C)CC2)=O)ccccc1C#N N1(C(C2(CC(C)C)CC2)=O)CCCCC(C(N2CC3CC(C)C3C2)=O)C1 CN1CCN(C)C(CNC(C2CCN(C(=O)C3CC(=O)N(C)C3)O2)=O)C1 n1(CC(=O)NC23CC(CNC(C4COC(=O)C4)=O)(C2)C3)cnc([N+](=O)[O-])n1 Cc1ncc(C(=O)NCC23CC(NC(c4cnc(C5CC5)s4)=O)(C2)C3)c(=N)[nH]1 Cc1cccc(Br)c1C(C(=O)NCC1CCC2(CC2)C1)NC(c1cccc(=O)o1)=O C1(NC(c2nnn(C)n2)=O)CC2CCC1N2C(c1ccc(C(C)(C)C)cc1)=O CN1CCN(CC(=O)N(C)CCN(C(C2CC2Cc2ccccc2)=O)C(C)C)CC1 N1(C(C(CCCC)F)=O)CCN(C(C2CC2(F)Cl)=O)C(C)C1C CN1CC=C(CNC(C2CC2N2CCOC2=O)=O)CC1 c1(NC(C2C(O)CCN(Cc3c(C)ncs3)C2)=O)cnc(C#N)c(Cl)c1 C1(C(=O)NCC2CCN(C(C(CCC)N(C)C)=O)C2)Cc2c(C)cccc2O1 c1(C(N(CC(C)CNC(c2cnc(N)cn2)=O)C)=O)ccc(N=[N+]=[N-])cn1 N1(C(c2c(C)cnnc2)=O)CCC2(NC(=O)CCn3c(C)c(C)sc3=O)CC2C1 n1(CC(=O)NC(C(C)NC(C2CC(=C)C2)=O)C)cc(Br)c(C)n1 CC1(C(=O)NC2(C(O)C(F)(F)F)CCC2)COCCN(C(C2CCCCS2)=O)C1 C1(NC(c2cnccn2)=O)CCC12CN(C(=O)COCC1CCCCO1)C2 C1(C(=O)NCC(C(=O)NCC2CN(C3CC3)C2)OC)CCCSC1C N1(C(C(=O)N(C)C)=O)CCC2CC(NC(C3OCCO3)=O)CCC2C1 CC1CN(C(=O)CCc2cn(C)nn2)CCC1NC(C1CCC=CO1)=O c1(N2CC3C(CNC(c4snnc4C4CC4)=O)C3C2)ncc([N+](=O)[O-])cn1 N1(C(C(CC=C)CC)=O)CC(C)OC2(CCN(C(c3nnn(C)c3C)=O)CC2)C1 CC1(C)CCC=C1C(=O)N1CCCC(N2CCN(C(c3ccnnc3)=O)CC2)C1 N1(C(C(=O)NC(C(=O)OC)CC(C)C)C2CC2Cl)CCOC2(CCN(C)CC2)C1 c1(C(N2C(C)CN(C(c3cnco3)=O)C(C)C2)=O)ccc2c(n1)NC(=O)CO2 C1(C(N2CC(C)(CC(=O)NCc3c(C)nn(C)c3C)C2)=O)CC(=O)CC12CCC2 c1(C(=O)OC)nccnc1NCc1nnn(C)c1C(=O)NCC1C(C)(C)C1(F)F c1(CC(=O)NC(C2CCN(C(=O)CC3C=CCC3)C2)C)cncn1C Cn1c(Cl)cnc1C(N1CCCC1c1ccc(Cl)s1)=O C1(F)(CNC(C=CCOC)=O)CCCN(C(=O)COCCCCC)CC1 C1(C)(NC(C2CCN(C(C)=O)CC2)=O)CCCN(C(n2cnc(Br)n2)=O)C1 C#Cc1cn(C)nc1C(N1CCC(NC(=O)CC2COCCN2C)C1(C)C)=O Cc1ccc(C(=O)NC(C)CNC(c2cc(N)nc(Cl)c2)=O)c(F)c1 c1(C2CCN(C(=O)NC(C)Cc3cc(Cl)cc(Cl)c3)CC2)cccc2nonc12 S(=O)(=O)(c1cc(C)cs1)N(C(=O)NC1CCCO1)Cc1ccc(OC)cc1OC N1(C(C(C)NC(CC)=O)=O)CCCCCCC1C(N1CC(F)(F)CC1C)=O c1(OCC(C)NC(=O)C(=O)Nc2cc(Br)no2)cccc(C(C)(C)C)c1 C(=O)(CCC1=CCCCC1)N(C)CC1N(C(Cc2cnc(C)o2)=O)CCCC1 C1(CC(N2C(CCNC(CCCC#N)=O)CCC2)=O)CCC(=O)NC1=O Cc1cnn(C)c1C(=O)NCC1(C)CC(NC(=O)C(C)CF)C1 C1(C(=O)NCC=C(C(=O)Nc2cccc(OC)c2)C)CCC(C2CC2)C1 c1(OC2CCN(C(=O)NC3C(C)CC=CC3)CC2)cc(F)c(Br)cc1F c1(CN2CC3CN(C(C4CCC(C(=O)OC)CC4)=O)CC32)cc(F)cc(C)c1O C1(CCC)CCC(C(=O)N(CCCNC(=O)CCC(C)O)CC)CC1 N1(C(C(C(C)OC)NC(c2nnccc2C)=O)=O)CCc2cncnc2C1 c1(COCC)cc(C)on1.N12CCC1CNC(=O)COC2=O.C(C)(C)(C)O C(=O)(C(C)(C)c1nncn1C)NC1CC(CNC(C2(C(C)C)CCC2)=O)C1 S(=O)(=O)(c1ccsc1C(N1CC(NCCCC(=O)c2cccnc2)C1)=O)NC c1(C(=O)N(CC(=O)NC(c2ncc[nH]2)CC)C(C)C)cn(CCO)nn1 c1(C(N2C(C)(C)C(NC(C3OCC3(C)C)=O)CC2)=O)cc2ncccc2o1 C1(NC(c2cn(CC)nn2)=O)COCCN(C(c2cc(C(F)(F)F)c(Cl)s2)=O)C1 N1(C(CC(C)(C)O)=O)CC2(CCC2)CC1CNC(c1cc(C2CC2)[nH]n1)=O CCC(C)C(CC(=O)NC1CCC(C(C)C)CC1)NC(=O)C(C1CCOCC1)O CCC(C)(C#N)C(=O)NC1CCC(NC(=O)COc2ccc(C)cc2C)CC1 CN1C(=O)CC(C(=O)NC2CCN(C(c3c[nH]c(=N)o3)=O)C23CC3)C1=O N1(C(c2c(CC)cno2)=O)CCN(C(=O)C(C2CC2)SC)CC1CO C1(CC(NOC(C)C)=O)CN(C(=O)C(C2CCCCC2)O)CCO1 C(=O)(C(Cc1cc[nH]n1)NC(c1cnco1)=O)NCCCOCC#C C1(N(C(Cc2n(C(C)C)cnn2)=O)C)C2CN(C(=O)CC3CCCO3)CC12 C(c1ccc2c(c1)COCC2)=CC(=O)NCC(F)CNC(C1CCCOCC1)=O N1(C(C2CC(C)CN(C(c3cnn4c3CCC4)=O)C2)=O)C2CCC1CC(=O)NC2 C1(F)(CNC(C2CC(C)N2C(=O)Cc2ccon2)=O)CCN(C)C1 N1(C(C(CC)O)=O)CCC(C)(C)C(C(=O)NCCc2cccnc2O)C1 N1(C(C2C(C)C2C)=O)C2CCC1CC(N(C)C(c1sccc1OC(F)F)=O)C2 c1(C(=O)NCC(CNC(C2(CC=C)CC=CC2)=O)(C)OC)cc(C)cc(C#N)c1 CON(C(=O)C1CCC(C)(C(N2CCCC2)=O)C1)C(C)CC(=O)O C1(CNC(c2cn(CC(C)C)nc2)=O)CCCCC1NC(=O)C=CC1CCC1 c1(CCC(N2CC(NC(CC(COC)C)=O)C2)=O)ccc2ccn(C)c2c1 C1(NC(C(C)(C)NC(C)=O)=O)CC2CCCC(C1)N2C(C1CCCC(=O)N1)=O N1(C(C(COC(C)C)NC(c2c(CC)csc2)=O)=O)CCCC1(C)C c1(C(N2CC(OC)(CNC(=O)Cc3csnn3)C2)=O)c[nH]c(=O)cn1 c1(C(N(C2CN(C(C3CSC3)=O)CC2O)C)=O)cc(-c2cn[nH]c2)ccn1 C1(NC(COCCOCCOC)=O)C=CCC(C(=O)NC(C)CF)C1 CS(=O)C=CC(=O)NCC1CCCC(CNC(C2(C(F)(F)F)CC2)=O)C1 CCC(C)CCCC(=O)Nc1cccc(NC(=O)C(C(C)C)C2CCC2)c1 c1(C(=O)NC(CNC(C(C(CC)(C)C)O)=O)C(C)C)coc2c(OC)cccc12 c1(N(C(C)CN2CCCC2)C)ccc(S(=O)(=O)NC2CCOCC2)cn1 Cc1ccc(C)c(C(N2CC3CC2CN3C(c2ccc3cnnn3c2)=O)=O)c1N c1(C(=O)NCCCCNCC2(O)CCCCC2)ncc(Br)cc1I C1(CC)CN(C(C2CC(C3CC3)=NO2)=O)CCC1NC(c1cccnc1C)=O C=C1CC(C(=O)NOC2CC2)(CO)C1.c1ccc(C(=O)NC2COC2C(C)C)o1 C1(NC(C2(C#C)CC2)=O)CC2CCC1CN(C(C1CCC(C(N)=O)O1)=O)C2 N1(C(C(COCC)C)=O)CC(CNC(=O)CCCSC(C)(C)C)CC1(C)C c1(C(N2CC(CNC(=O)CC3CC3)OCCC2)=O)ccc2n[nH]cc2c1F C12(C(=O)NC(c3ccc(OC)c(F)c3)C)CCOCC1C2(F)F c1(-c2scc(NC(c3c(C)nc(Cl)s3)=O)n2)cc(Cl)c([N+](=O)[O-])cc1Cl CCC(CC)CN=c1[nH]c(=NCc2cccc3[nH]ncc23)c2ncccc2[nH]1 C1(CCC(=O)OCC)CCN(N2CCC(c3cnco3)CC2)CC1O C1(CNC(COc2c(C)cccc2)=O)CC2CCC(C1)N2C(c1ccsn1)=O Cc1nn(C(C)(C)C)c(C)c1NCC(=O)NC(=O)NCC(O)Cc1ccccn1 C1(C(c2nnnn2C2CC(F)(F)C2)NC2CC3CC3C2)(CC)CC(C)(C)C1 C(c1ccc(Cl)cc1F)=CC(=O)NC1C(CC)N(C(C2CC3(CC3)CO2)=O)CC1 C1(CC)CC(C)CN(Cc2ccc(-c3ccccn3)cc2)C1.C12(CC1)C(=O)N2 C(CS(=O)c1ccc(C)cc1)NC(c1n(CCC)nnn1)C1CC=CC1 C1(C(N2CCCC(C)(C(=O)OCC)C2)=O)CC(c2ccccc2)=NO1 c1(C(=O)NC2CCC(NC(C3(C)CC(C#N)C3)=O)CC2)ccc(Br)nc1O N1(C(C2CC(=O)OC2)=O)CCN(C(=O)CN2CCNC2=O)CC1C(F)F C1(NC(c2c(C)nns2)=O)CC(O)CN(C(=O)CC(C(F)F)n2ccnc2)C1 N1(C(c2c(S(=O)(=O)C(=O)NCC3(OC)CC3)ccs2)=O)CC2ON=C(CNC)C2C1 Cc1oc(CO)cc1C(=O)NC1CC(NC(=O)C(F)(F)C2CCCCC2)C1 Cc1cc(C)c(C(=O)NCC(C(F)(F)F)N2CCN(C(=O)CSC)CC2)c(C)n1 N1(C(C2CN(C)C2)=O)CC(C(N2CC(CS(C)=O)C2)=O)C2(CCC2)C1 C#CC1CCN1C(=O)CN(C(=O)C(C)(C)SC)C c1(CN2CC3CN(C(C4(C)COC4)=O)CC3C2)c[nH]c2ncc(Cl)cc12 CC(C)S(=O)(=O)c1ccc(C(N2CCC(C(C)NC(c3cnsn3)=O)C2)=O)cc1 C=CC(CCC)CC(=O)NC1CC(C(=O)NCC(C)CCCO)C1 CC(C)C(C)C(=O)NN1CCCC1C(N1CCC(N2CC(O)C2)C1)=O c1(C(=O)NCC(C2CCOC2)NC(CSC(C)C)=O)cc(Cl)c(F)cc1O N1(C(C2N(N=O)CCCC2)=O)CC(NC(=O)C=Cc2ccco2)CC2(CCC2)C1 c1(CC(=O)NC(CNC(C2C(C=C)C2)=O)(C)CC(C)C)ccc2c(c1)OCO2 c1(OC)ccc2c(c1)CCC2(O)CNC(=O)NCC(O)CS(C)(=O)=O C#Cc1ccc(F)c(C(=O)NC(CNC(=O)CC2(N(C)C)CCCC2)CO)c1 Cc1ncccc1CC(=O)NCC1C2CN(C(=O)C(O)Cc3ccccc3)CC12 C(=O)(CCCC(C)c1ccccc1)NCC(C1CC1)NC(C1(C)CC(C)C1)=O CN1CC(C)(NC(C2C=CCN(C(C3(O)CCOC3)=O)C2)=O)CCC1=O N1(C(C(CN(C(C(CCC)(C)O)=O)C)(C)C)=O)CC2CCC(CO)(C2)C1 N1(C(c2ccc(OC)cc2)=O)CCC(C)C(NC(=O)Cc2csc(Br)n2)C1 C(CCCOC)(C(=O)NC1COC(C(F)F)C1)NC(c1cc(CCC)on1)=O C1(C(=O)NC2C(CC=C)COC2)CN(C(c2cccc(O)c2)=O)CCN1C c1(C(C)NC(CCCC)(C)c2nnnn2CSC2(C)CC2)ccc(F)c(F)c1 N1(C(C2C(C)(C)C(NC(=O)Cn3cccn3)C2)=O)CCC12CC(O)C2 CC1=C(C(=O)N2CCN(C(=O)CP(C)(C)=O)CC(C)C2)C(=O)OC1(C)C N1(C(C=CSC)=O)CCN(C(=O)Cc2ccnc(OC)c2)CC2CCCCC12 C(=O)(C1CCc2nccn21)N(C(CN(C(C1CCC(C#C)CC1)=O)C)C)C c1(C(C)C)ccc(C(N2CC3CC2C3C(=O)NC2CC(F)C2)=O)cn1 C(=O)(C(C(C)(C)C)c1ccccc1)NC1(OCC)CCN(C(C(F)=CCC)=O)C1 c1(CNC2C(C(N3CCC(N(C)C)C(O)C3)=O)C2)cc2ccccc2[nH]1 C1(C(=O)NC2CCC(n3cc(-c4cccnc4)nn3)C2)C2CCCCC12 C1(NC(c2cc(Cl)cc(Cl)n2)=O)CC2CN(C(C34CC(CO3)C4)=O)CC2C1 CCC(CC)C(C)C(=O)N(C(CNC(c1ccn(C(C)(C)C)n1)=O)C1CC1)C N#Cc1ccccc1CC(=O)NC1CN(C(=O)Cc2ccc(F)cc2)CC1F c1(SC)c(C(=O)NC23CC(CNC(c4snc(O)c4Cl)=O)(C2)C3)cccc1F Cc1cc(C)cc(S(=O)(=O)N2CCC(C(N3CCC(CO)C3)=O)C(O)C2)c1 C1(CC)C(NC(=O)Cc2coc(C)n2)CCCN1C(C1C2CCC(=O)C12)=O c1(C(=O)NCC(O)CNC(C2CCC3CC3CC2)=O)cnc2[nH]c(O)nc2c1 CC(C)(C)CC(C(=O)NCC(=O)NC1CC1)NC(c1ncccc1Cl)=O N1(CC(=O)NCCC2CN(C(C(CCC)=CCC)=O)C2)C(=O)C(=O)N(C)C1=O N1(C(C)=O)CCN(C(c2cc(Cl)cs2)=O)C2C1C2(F)F c1(OC)cccc(C(N2CCCC2C(N2CCCC(Br)C2)=O)=O)c1Cl CCCC(C(O)C(=O)NCC1CC1c1ccoc1)NC(c1c[nH]cc1C(C)C)=O c1(C(N(CC(C)NC(=O)C(N)=O)C)=O)c(Cl)cc(Br)cc1[N+](=O)[O-] C(=O)(CS(=O)(=O)C1CC1)N(C(C)CCNC(=O)Cc1ccnn1C1CCC1)C C1(C(N(CCCNC(=O)C(C)(C)c2cnc[nH]2)C(C)C)=O)CCCCN(C)C1=O N#CC1Cc2cccc(C(=O)NCC3(NC(=O)CC4CCCCC4)CCOC3)c21 C1(C(=O)NC2CC(C)(NC(c3c(C)ccs3)=O)C2)CN2CCCCC2CO1 c1(NC(C2N(C(CC3(C)CC3(F)F)=O)CC(O)C2)=O)ccc(Br)cc1Br c1(OC)ccnc(-c2nc(-c3cc[nH]n3)nn2Cc2ccc(C)cc2)c1F n1(CC(=O)NC2C(NC(CCc3c(C)ncs3)=O)C2)ccc(O)nc1=O C(=O)(C1=CCCCC1C)NC(c1ccccc1OC)CNC(CCOC)=O CCC1=NOC(C(N2CCCC(NC(=O)C=Cc3ccsc3)C2)=O)C1 c1(N2CC3(C2)C(=O)N3)nccc(SC(C)C)n1.C1(COC)(CO)CC1 C=C=CC(C)C(=O)N(C)CC1CCCN1C(c1cc(O)n(CC)n1)=O Cc1cc(=NCc2cscn2)[nH]cc1S(=O)(=O)NC1CCOCC1 C1(C(=O)NC(CNC(C(N2CCC(C)CC2)=O)=O)C)CCCC(=O)N1C C1(CNC(c2ccc(OC)s2)=O)CC2(CO1)CN(C(c1cc(Cl)ccc1C)=O)C2 C1(N(C(CCC=CC)=O)C)CCCC2CN(C(=O)CCC3CCCOC3)CC12 C1(NC(c2ccn(CC(C)C)n2)=O)CCC(NC(=O)C(C2CCOCC2)C)CC1 C1(CNC(c2cc(CC)sn2)=O)CCN(C(c2cccn(C)c2=O)=O)CC1O Cc1ccc(C2(C(=O)N(C)CCNC(C3(C)CCCC3C)=O)CCC2)cc1 n1(CC)ncc(C(=O)NCCC(C)N(C)C(c2cnn(C)n2)=O)c1C(F)(F)F CC1(C)CC(C(=O)N2CCN(C(=O)C(C)(C)c3ccns3)CC(O)C2)=NO1 N1(C(c2cc(SC)oc2C)=O)CCN(C(c2cnoc2C)=O)C(C)CC1C c1(NCC(CC)N(C)C)cc(Br)ccc1S(=O)(=O)NCC(CO)C1CC1.OC c1(C(N2CCOCC(CNC(CSCC#C)=O)C2)=O)cnc2cc(O)ccc2c1 c1(CCN2C(c3ccc(Cl)cc3)CCC2)ccc(F)cc1F Cc1cc2ccccc2n1CC(=O)NCC1CC(C)(C)CN1C(=O)CP(C)(C)=O C1(C(N2CC(CC)C(NC(=O)CC3CC=CCN3C)C2)=O)CCS(=O)(=O)CC1 Cn1cc2c(n1)CCN(C(=O)CC1CCN(Cc3cc(Br)c(F)cc3Cl)CC1)C2 c1(N2CCC=C(C)C2)cc(N2CCCC(NC3CCCC3)CC2)nc(C(C)C)n1 C1(C#CC(=O)NCC(F)(C(=O)N(CC(C)C(=O)OC)C)C(C)C)(CC)COC1 C(=O)(C(C)C(F)F)N1CC(C)(C(N2C(C(=O)NC)CC2)=O)C1 C=CCC(C(=O)N1CC(O)(CN(C(=O)CCc2ccn(C)c2)C)C1)NC(C)=O.OCC N1(CC(=C)Cl)CCOC(C(=O)NC2CCCCC2C(=O)O)C1 c1(C(N2C(CN(C)C(C3COC4(CCC4)C3)=O)CCC2)=O)cc(N)c(F)cc1F C1(C(=O)NCCC(=O)OC(C)C)CCCCC1NC(=O)CCc1cccs1 c1(OC)cccc2c(C)c(C(=O)NC3CCN(C(=O)CC(F)F)CC3O)oc12 c1(C(N(C)CCNC(c2c[nH]c3cnccc23)=O)=O)cc2c(cc1Cl)OCCO2 C(=O)(CCCCCNC(N)=O)N(C1CC1)CC1(CNC(C(C)(C)OC)=O)CC1 CC1=C(C(=O)N2CC3(CC(NC(c4ccc(C)nc4)=O)CO3)C2)CCC(C)(C)C1 N1(C(c2cccc(OC)c2)=O)CCC(O)(C2CCN(C(C3CC34CC4)=O)CC2)C1 C1(NC(=O)CCSCC2CCCC2)(CF)CCN(C(c2cc[nH]c2)=O)C1 N1(C(c2ccn(CCC)n2)=O)CCN(C(=O)C(c2cccc(C)c2)F)CC1CF C1(NC(c2cn(C)c(O)n2)=O)CCCCN(C(=O)Cn2ccc(C3CC3)n2)C1 c1(C(=O)NC2(CC(=O)N(C(C)C(F)F)C)CC2)cccc(C2CC2)c1 CCCC(CNC(=O)C(C1CCC1)NC(=O)CC(COC)COC)CCO C1(C(=O)NC2C(NC(=O)Cc3ccnc(F)c3F)CCC2)CCc2ncsc2C1 C1(NC(c2c(C)csc2)=O)CCOCC1NC(=O)Cc1cc(C2CC2)n[nH]1 C(=O)(C1=CCCOCC1)NCc1ccc(C(N2CC(C)C(C)C2C)=O)o1 C12(C(=O)NCCCN(C)C(c3cc(C4CC4)cs3)=O)CCCCC1C2 C1(NC(c2cnc[nH]2)=O)COC2(C1)CN(C(=O)Cn1nc3c(n1)CCCC3)C2 N1(C(CNC(c2nccc(CC)c2)=O)=O)CCN(C(=O)C(C)C#N)CC1C C1(C(N2CC(CNC(C(C)CCO)=O)OCCC2)=O)COc2ccccc2O1 C1(CNC(CCC(C)N(C)C)=O)CCC(F)(CNC(C2(C)CC(C)(C)C2)=O)C1 CCC(CC(=O)NC1CN(C(c2cc(Cl)n[nH]2)=O)CC12CC2)C(C)(C)C CCC(C)(F)C(=O)NCC1CC(NC(c2cc(SC)c(C(C)C)o2)=O)CC1O Cc1cc(Cl)c(C(=O)NCC2CN(C(C3CCC(=O)N3)=O)CC2C)s1 C1(C(=O)NCC2N(C(C(C=C)(F)F)=O)CC2)Cc2ccc(OC)nc2C1 C(=O)(C1=C(CC)OCCC1)NCCOCCC(=O)N(CC(C(=O)OC)C)C.CCO C1(CNC(CNC(c2c(CC)cco2)=O)=O)CN(C(C)=O)CC1c1ccnn1C CC1(C)CC(NC(c2ccncc2C(F)F)=O)CN1C(c1cnn2ccsc12)=O C1(NCC(=O)Nc2cc(C#N)c[nH]2)CC2CCC1N(C(C1N(S(C)(=O)=O)CC1)=O)C2 CC1CCOC2(CCN(C(c3cc(Br)c(Cl)s3)C(=O)NCc3cccs3)CC2)C1 N1(C(C(=O)NC2CCOC2)Cc2ccccc2)CC=CCC2(CCCC2)C1 S(=O)(=O)(c1ccc(NC2CC(n3cncn3)C2)cc1Br)NC1CCN(C)C1 C(C(CC(F)F)C(=O)NN(C)C)c1cn(Cc2cc(CCCCC)no2)nn1 C12(O)CCN(C1)C(=O)CS2.C1(C(=O)OC)CC(C(=O)NCCCN(C)CCO)C1 N1(C(C=CCCC)=O)CC(C)CC1C(=O)Nc1[nH]cnc1C#N N1(C(c2cc(OCC)no2)=O)CCC(C)C1CNC(=O)C(C1CC1)C1CC1 Cc1[nH]c(C(N2CCC(N(C(=O)C(C)OC3CCCC3)C)C2)=O)c(C)c1[N+](=O)[O-] CCCC(CC)C(=O)N1CCCCC1CNC(c1ccnc(OCCN(C)C)c1)=O c1(C(N(C)CC2(CNC(=O)CCc3ccc(Cl)cc3)CC2)=O)c[nH]c(=O)cn1 C1(NC(c2cn3ccsc3n2)=O)CCCCN(C(C2CC23CC3)=O)C1 c1(C(N(CCNC(=O)CC2CNC(=O)C2)CC)=O)ccncc1Cl C12CCCC1N2.C1(OCC(=O)NCCOC)CN(C(C2(C)CC2)=O)C1 C1(CC(=O)N(CCC)CC2CCC2)CN(CC2CCOC2)CC1C C1(C(N2CCC(CC(=O)NC(C)C3CC3)CC2)=O)CCCNS1(=O)=O C(=O)(C1CCCc2c1ncn2C)NC1CC(NC(C=C(CCC)CCC)=O)C1 C1(NC(C2(CC=C)CC2)=O)CN(C(c2ccc(N)cc2Cl)=O)CC2(CC2)C1 C(=O)(CC(C)(C)CC(=O)OC)NC1CN(C(C=CC)=O)C2(C1)CCC2 C1(C(=O)NCc2c(COC)cccn2)CC2CCC1N2C(C1CCCO1)=O C1(NC(c2c(CN(C)C)ccs2)=O)CC2CC1CN(C(C1CCNC(=O)C1)=O)C2 C=C(C)CC(C)C(=O)NCCOCCN(C)C(C12CC(F)(CO1)C2)=O c1(C(N(C2CCN(C(C3(COC)CCOC3)=O)C2)C)=O)cnc(O)c2ccsc12 c1(-c2n(CCCC)nc(Cc3ccncc3)n2)ccc(S(=O)(=O)CCO)cc1 C(=O)(C1CNC(=O)c2ccnn21)NCC(CNC(C#CC(C)(C)C)=O)(C)O N1(NC(=O)OC(C)(C)C)CCC(NC(C2CCC2F)=O)CC1.C12(CC1)C(=O)N2 c1(C(=O)NC(CCNC(c2c(C)onc2O)=O)C)ccc2cc(C#N)ccc2c1 c1(C(N2CC(OC)CC(C(=O)OC)C2)=O)ccc2c(c1)C(=O)N(C)C2 C1(CNC(C(C)(O)C2CCC2)=O)CN(C(c2cc3n(n2)CCC3)=O)CCCO1 C1(C(=O)OCC)(C(=O)OCC)CN(C(c2cc(C)c[nH]2)=O)C1.C12CCC1S2 O=C(CCCC(=O)C1CC1)NCC1CCCN1C(C1CCC2CC1CO2)=O c1(CC(OC)OC)nnc(N2CCOC(Cn3nc(C)cc3Cl)C2)n1CCC#N N1(C(CCC=CC)=O)CC(CCNC(=O)CCCOC(C)C)OC(C)C1 CC1CC(NC(=O)CCc2cnn[nH]2)CN(C(=O)C=CCn2cncn2)C1 C(CC(C)C)(C(=O)N(CC(F)F)C)N(C(CCCCSC)=O)C C(CCCC(=O)OCC)(C(C)(C)C)OC(C)(C)C.CC(C)(C)OC1CC1C(NC1CC1)=O C1(C(N(CC(O)C(F)F)C)=O)CCCN(C(C23CC(C#N)(C2)C3)=O)CC1 Cc1c(O)ccc(C(N2CCCC(O)(CNC(=O)CNS(=O)(=O)C3CC3)C2)=O)c1C C(=O)(C(C)(C)CCC)NCC(CCCC)NC(c1ccc(C)nn1)=O CCC(CCCO)NC(=O)C(C1CCCN(C(C2CC(O)C(F)C2)=O)C1)(C)C C1(CC(=O)NCC(=C2CN(C(C3CC3c3ccsc3)=O)C2)F)CCCCCO1 C1(NC(CC(OCC)OCC)=O)CC2CCC1N2C(=O)COc1ccccc1C N1(C(C(CCC)NC(C)=O)=O)C2CCC1CC(F)(C(N1CCOC(CN)C1)=O)C2 c1(NC(CC2OCCN(Cc3cc(C)nc(C)c3)C2)=O)cnc2[nH]ncc2c1 CCC(C)C(CNC(=O)CCC1CCCN(C(c2nn(C)cc2Cl)=O)C1)CO N1(C(C2(OC)CCC2)=O)CCC(C2CC2)(NC(=O)Cc2nocc2C)C1 c1(NC(N(c2nnc(C)o2)C)=O)cc(Br)cnc1OC(C)C C(c1cncn1C)=CC(=O)NC(C1(C(N2C(CC=C)CCC2)=O)CC1)C C1(NC(CNC(=O)OC)=O)CCCC(C(F)(F)F)C1 c1(C(C(=O)NC(C2CN(C(c3cnc(C)s3)=O)C2)C)C)ccccc1F c1(NCCC(=O)NC2CC(CNC(COC(C)C)=O)C(O)C2)ccc(C#N)cc1 N1(CCCC(N2CCCCC(C)(c3ccccc3)C2)=O)CCCC2(CCCC2)CC1 N1(C(C(C)C#N)=O)CC2CCC1C(NC(=O)C(C)NC(c1ccccc1)=O)C2 c1(C(=O)OC2CC(C(C)(C)C)C2)cccc2cccnc12 C(CNC(=O)COc1cccc(Cl)c1C)(C(C)C(C)C)NC(c1c(C)nco1)=O c1(C(=O)NC2CC(NC(C(COC)C)=O)C2)cc(C)cc2c(C)ccnc12 c1(C(N(CCCN(C(Cc2c(C(=O)OC)csc2)=O)C)C)=O)ncncc1F Cc1cc(C(N2CC(C)C(NC(C3CCOCC3)=O)C(C)C2)=O)c(N)c(F)c1 CC1(C)NC(=O)OC1CNC(C1CCC=CC1NC(=O)CN1CCCC1)=O c1(C(N2CC(O)(CCNC(C3(C(C)C)COC3)=O)C2)=O)cccc(F)c1O C1(NC(=O)CC2CC2)C2CC3C(C2)C13C(=O)NCCN1CCN(C2CC2)C1=O Cc1cc(F)ccc1CC(=O)NC1CC(NC(=O)C(C)C2CCCC2)C1 CCCCCC(C(=O)NC1CC(NC(=O)CC2CC3C=CC2CC3)C1)C(C)C n1(C(CC)C)nccc1C(=O)NCCC(C)NC(=O)C(c1cnn(C)c1)C C1(NC(c2cc(C)nc(O)n2)=O)CC2CC1CN(C(=O)Cc1cnnn1C)C2 CCC(C)(C)C(O)C(=O)N1CCCCC1CNC(C1(C)CCC(O)CC1)=O S(=O)(=O)(c1cnn(C)c1)NCC(=O)NC1(CNC(c2c(C)cncc2C)=O)CC1 c1(C(N2CC3CCCN(C(C4C5COCC45)=O)C3C2)=O)ccc(Cl)c2occc12 n1(CC(=O)NC2CC(NC(c3cncc(C(N)=O)c3)=O)C2)cc(Br)ccc1=O C1(CNC(=O)NCCCCn2cc(C3(C)CCOC3)nn2)CCCC(CC#N)C1 C#Cc1ccc(C(=O)N(C(C)CC(N2CCC(C(N)=O)C2C)=O)C)c(C)c1 C1(C(=O)NCC(C)(C)CCNC(=O)C=CC(=O)NC2CC2)CCC2C(C1)C2(F)F C1(NC(c2c(C)nco2)=O)CCC2CCN(C(c3cnc4sccc4c3)=O)C12 C1(n2cc(C)nn2)CN(S(=O)(=O)CC2(C(=O)O)CCC2)CC1O.CO C1(CC(N2CC(N(C(C=CCC)=O)C)C2)=O)(CC)CCOCC1 N1(C(c2c(C)n[nH]c2)=O)CCC(CNC(c2ccnnc2S)=O)CC1 N1(C(c2c[nH]c(=NCC=C)s2)=O)CC2CN(C(=O)CCc3cccnc3)CCC12 C1(C(=O)NCC2N(C(CC3CC(C(=O)OC)C3)=O)CCC2)CS(=O)(=O)CC(=O)N1 c1(CC(=O)NCCC(C)N(C(C(CC)C)=O)C)c[nH]c2c(Br)cccc12 c1(CC(C(N2CC(C)(NC(C3CCN(C)C3)=O)C2)=O)O)ccc(Cl)cc1 C1(N=c2cc[nH]cc2C#N)(CNC(C(C=C)O)=O)CCCCC1 C(C(N=[N+]=[N-])C(=O)N1CCCC1C=CC(=O)NCC(C)(C)COC)OCC c1(C(=O)NCC(CNC(C2CC3C(C2)C3(C)C)=O)OC)c(C)cc(C)oc1=O CC#CCCC(=O)NC(C1CC=CCC1)C(=O)NCC1(CC)CCC(=O)N1 C1(C(N2CCC(C(C3(NC(c4cncs4)=O)CCC3)C)C2C)=O)C2C3CCC(C3)C12 C(=O)(C#CC(C)(C)C)NC(c1cc(C(N2CC(N=[N+]=[N-])C2)=O)ccn1)C CCC(C(=O)N1CCC(CCNC(=O)COCc2nc(C)no2)C1)N(C)C C1(CCCC)(C(=O)NCCC2CC(NC(=O)CSCC(F)F)C2)CCC1 c1(OCC)ccc(C(N2CC(NC(c3cc(C)co3)=O)CC(C)C2)=O)cc1Cl N1(C(C(C)(C)O)=O)CCN(C(c2cnc(Cl)s2)=O)C(c2ccccc2Cl)C1 N1(C(CN(CCOC)C)=O)CC2CC(C(N3CC4CCN(C)C4C3)=O)CC2C1 c1(CC)ccc(C(=O)NCCC2(NC(=O)C=CC(C)C)CCC2)c(F)c1 C#CC(C)(C)C(=O)NC1CC2(C1)CC2NC(C1CSCC(=O)N1)=O c1(CCC(=O)N(CC(CC)NC(CCC)=O)C)nnc(C)n1C CCCCC(CC(=O)NCc1cc(C)co1)NC(=O)C(C)N1CCCC1 C1(C(=O)NCC(COC)C)CC(C)CCN1C(=O)CN(C)C(=O)C1CC1 N1(C(c2ccc(OC)s2)=O)CC2CCN(C(=O)CC3CC=CCC3)CC2C1 N1(C(CC2C(C)=NNC2=O)=O)CCCC(F)(CNC(=O)Cc2cc[nH]n2)CC1 c1(CNC2CC(NC(c3n(C)ncc3Cl)=O)C2)cc(Cl)c(Cl)cc1O N1(C(C(C)NC(=O)C2CC2)=O)CCN(C(C2CCN(C)C(=O)C2)=O)CC(C)(F)C1 c1(OC)csc(C(=O)NCCCCC2CCN(C(=O)CC(=O)NC3CC3)C2)c1 Cc1nc2ncc(C(=O)NC(CNC(C3CC(O)CN3C)=O)C(C)C)c(=O)n2[nH]1 S(=O)(=O)(c1ccn(C)n1)N1CC2(CC(NCc3c(OC)c(F)ccc3)C2)C1 N#Cc1nc(CN2CCC3(CC2)CC3C(=O)N=c2cc[nH][nH]2)ccc1Cl Cc1cc(NC(C2(C(C)C)CCN(C(=O)CC(C)(C)C)C2)=O)cc(O)c1 C1(CC(=O)N(CC=CC(=O)NCC2(CCCC)CCC2)C)CCCNC1=O c1(C(N2CC3CC2C3C(N2CCN(C3CCOCC3)CC2)=O)=O)ccccc1Cl c1(N2CCC(COC(C=C(CCC)C)=O)C2)ccc(SC)c(C)c1 C1(NC(Cc2cnc(C)s2)=O)CCCCC1CNC(=O)COc1ccccc1F c1(C(=O)NCC2(CCNC(C(c3ccccc3)C)=O)CC2)c(N)cnn1C N1(C(C(c2ccc(Cl)cc2)CC)=O)CCn2c(CCN)nnc2C1 Cc1cc(C(=O)NC(c2ccccc2)C(C)NC(C2(CF)CCC2)=O)cc(C)c1 C1(CC(=O)NC(C)C(F)(F)F)CCCN(C(C2CC(C)(O)C2)=O)CC1 CC1=C(C(=O)NC2CCC3CC2CN3C(C2CN3CCN2CC3)=O)SCCO1 C1(C(=O)NCC(C)NC(C2OCCN(CC)C2)=O)Cc2cccc(C)c2O1 c1(C(=O)OC(c2ccc(C)o2)C)cc2n(n1)CC1(CC1)C2 C(c1cc(OC)c2c(c1)OCCO2)=CC(=O)C(=O)C=CC=C.CCC(C(=O)O)N N1(C(c2cc(C)[nH]n2)=O)CCCC(CCCCNC(=O)C(=O)NCCC(N)=O)C1 O=C(C1=C(Cl)CCOC1)NCC1CCCCN1C(=O)C(c1cccnc1)O S(=O)(=O)(c1cccc(Br)c1)CCNC(N1CCC(O)(CN(C(C)(C)C)CC)C1)=O C1(OCCC)CCC(C(N2CCC(N(C)C(c3ccc(O)nn3)=O)CC2)=O)CC1 C1(CNC(C2(C(C)NC(C3CC(C)(O)C3)=O)CC2)=O)C2CCCCCC12 Cc1n[nH]c(C)c1CCC(=O)NCCC(O)CNC(C1CCC(O)C1)=O C1(NC(C=C(C)C(C)C)=O)CC2CN(C(C3(C)CC3)=O)CCN2C1=O c1(C(=O)NC(CC)CNC(=O)C(CCO)N(C)C)cc2ccc(F)cc2nc1C c1(C(=O)NC(CCCC)CNC(=O)CCCCC(F)F)cc2c(cc1C)OCO2 N1(C(c2c(NCC)cccn2)=O)CCCC(NC(c2cc(Br)n(C)c2)=O)C1C c1(C2(C)CC2)cn(CC2C=CCN2C(=O)CCC2CCCO2)nn1 c1(C(N2C(C=C)CC2)=O)ccc(CNC(=O)C=CC(=O)N(C)C)nc1 c1(NC2C(OC)C(O)C2)nc2c(c(=NC3C4COCC34)[nH]1)CCC2 ONC(=O)CC(C)P(C)(C)=O.CC(C)C(O)COC c1(CC)cc(F)ccc1C(=O)NCCN(C(=O)C(C#N)C(C)C)C(C)C c1(NC(C(C)C)C(C)NC(=O)C(n2cc(Cl)cn2)C)cc2nncn2cn1 CN=c1nc(C(=O)NCCC2CC(NC(c3cc(=O)cc(Cl)[nH]3)=O)C2)cc(C)[nH]1 N1(S(CCCC)(=O)=O)CCC(C(F)(F)F)C(F)(F)C1 C1(C)(C(=O)NC2CCC(F)(CNC(C=C(CCC)C)=O)C2)CCC(C)C1(C)C CCCCC(C(=O)N1CCC(C)C(NC(C2C(OCC)C2C)=O)C1)C(C)C CC(C)(C)CC(F)C(=O)NC(CC(F)F)C(=O)N1CC(O)C(O)C1 c1(C(=O)NC(CNC(c2cnc(SC)s2)=O)(C)C(C)C)cc2ccc(Cl)cn2c1 Cc1[nH]nc(C(=O)NC(C(=O)NC(C)(C)C(C)O)C2CCC2)c1Cl N1(C(C)=O)CCC(NC(C2C=CCCC2)=O)C(O)C1.c12cn(nn1)C2C1(C)COC1 CCC(C)CCCCC(=O)N1C(CC(=O)NC(c2csc(C)n2)C)C2CCCC12 C1(CC)CC(CC(N2CCN(C(=O)C(C)NC(=O)COC)CC2)=O)CC(=O)N1 N1(C(CC=C)=O)CCc2sccc2C1CNC(c1cc(S(C)(=O)=O)co1)=O C1(c2nc(C(C)C)[nH]n2)CCCCN1C(C(C)(C)C)=O CC(C)CC(O)C(=O)NCCN(C(c1ccc(C(N)=O)s1)=O)Cc1cccnc1 CCC(C)CCCC(=O)NC(c1nocc1C(=O)NCCOC(C)=O)C c1(-c2cccc(OCC)c2)cc(N(C)C)ccc1C(=O)NC(C)C#N c1(OCCCNCc2occ(C(=O)OC)c2)cccc(F)c1 Cc1cnc(C=CC(=O)NCC2CCOC2C)[nH]1 c1(C(=O)NCC2CC2)cccc(NCCN(C(C)C)C(c2ccc(CO)cn2)C)n1 c1(CC(=O)NCC23CN(C(C4C(C)CCS4)=O)C(C2)CO3)cn2c(n1)CCCC2 Cc1c[nH]c2ncc(C(N3CC=CC3CNC(c3ccc(Cl)o3)=O)=O)cc12 C1(C#N)(C(N2CC(CC(=O)NC(CC)C(C)C)OCC2)=O)CCCOC1 C1(NC(=O)OC(C)(C)C)CC2CC(NC3(C)COCCO3)CC2C1 CC(C(=O)NCC1(CNC(C2CCC2)=O)CC1(F)F)C(F)(F)F N1(c2cccc(C(=O)OC)n2)CCN(C(C2CC3C(C2)C3(C)C)=O)CC1C C12(NC(C3CC4(CCC4)C3)=O)CCC(CC1)N(C(c1cc(Cl)c[nH]1)=O)C2 N1(C(C(C2CCCC2)NC(c2c(CC)ncs2)=O)=O)CCNC(=O)C1 c1(OC)ccc(C(N2CC3CN(C(c4cn(C)cn4)=O)C3C2)=O)c(Cl)c1 O=C(CCCC(F)(F)CO)NCCC1CN(C(C2CC3CCCCN3C2)=O)C1 C1(NC(CCC(=C)C)=O)(CO)CCCN(C(c2cc(Br)c[nH]2)=O)C1 N1(C(c2n(C)ncc2Cl)=O)CC2COCCC2(NC(C2CCC23CCC3)=O)C1 C(=O)(CS(=O)(=O)Cc1ccccn1)NCC1N(C(C(CC)COC)=O)CCOC1 c1(NC(N2CC(C=C)C(O)C2)=O)nccn2nccc12 c1(C(C(=O)OC(=O)Cc2nc(C3CC3)n[nH]2)O)cccc(Br)c1 C#CC1(C(=O)N(C)Cc2cnn(C)c2)CN(C(=O)CC2CCC(C)CO2)C1 C1(NC(C=C(C)C)=O)CC=C(C(=O)NCCc2cccc(C)c2)C1 N1(C(c2n(C)cnn2)=O)CCC(CNC(C2CCCSC2)=O)CC1 C(C)(N=c1[nH]c2ccc(Cl)cc2o1)C1N(C(C2C(OC)CCC2)=O)CCCC1 C#Cc1cc(C(N2CCCC2CNC(=O)Cn2cnnn2)=O)cc(C(F)(F)F)c1 N1(C(CC2C(C)CCC2)=O)CCC(C)(CCNC(=O)OC(C)(C)C)C1 C1(NC(CNC(=O)Cn2ccnn2)=O)CCCN(C(=O)CCCCC2CC2)C1 C=CC1CCCC(NC(=O)CCCCN(C)C(c2ccn(C)c2C)=O)C1 c1(CCC(=O)NCCC(C)NC(C2CC3CCC2O3)=O)ccc2c(c1)CC(=O)N2 C(C1CN(C(=O)C=CSC)Cc2ccccc21)NC(C(CC)N(C)C)=O c1(C(N2CC(NC(=O)C(O)c3ccco3)CC(OC)C2)=O)cc2cnccc2o1 C1(F)(CNC(C2N=C(C)SC2)=O)CCN(C(C2(C)CC2C(F)(F)F)=O)CC1 c1(CC(C)(C)NC(C=CCC#C)=O)ccc(OC)cc1 O=C(C1Cc2ccc(F)cc21)NC1C2CC1N(C(c1coc(N(C)C)n1)=O)C2 c1(C(N2CC3C(NC(c4cn(C5CC5)nn4)=O)(C3)C2)=O)ccc([N+](=O)[O-])[nH]1 S1(=O)(=O)c2ccc(cc2)CCN1.C1(c2cccc(N)c2)CC(=O)NC(=O)N1 N1(C(C(C)Sc2ncccn2)=O)CC(NC(=O)C(C)N2CCCC2)C(C)C1 C1(NC(C(CC)n2cccn2)=O)CC2C1CCN2C(c1csc(C2CC2)n1)=O C(C(C)CC(=O)NC1(C2CCC2)CC1)NC(C(C)c1ccsc1)=O c1(C(c2nnnn2CCC2(C)CC2)NCCCC(=O)OCC)cc(C#N)cs1 c1(C(=O)N(C2CCC3(C(NC(C4=C(C)OCC4)=O)C3)CC2)CC)[nH]c2c(Cl)cccc2c1C CC1(C)OCCC1CC(N1CCCC1CC(N1CC2CC1CO2)=O)=O NS(=O)(=O)N1CCC(C(N2CCC(C(C)(C)C)(CNC(C3CC3F)=O)C2)=O)CC1 c1(CC(=O)NCC(C)N(C(=O)CN(C)C2CC2)C)cccnc1 C(=O)(CC1OCCc2sccc21)NCCC1(NC(C2OCC(C)(C)C2)=O)CCC1 C1(NC(C2CCN(C(CC3(C#N)CC3)=O)C2)=O)CC2CCC(C1)C2O C1(N(C)C(c2coc(C(C)(C)C)n2)=O)CN(C(C2(NC(N)=O)CC2)=O)CC12CC2 C1(CC(=O)NC(C)CCCNC(=O)Cc2nc(C(C)(C)C)cs2)CCOC1(C)C N1(C(Cc2c(C)cco2)=O)CC(C)C(F)(CNC(c2cnc(C)n2C(F)F)=O)C1 N1(C(C(CCC)F)=O)CCC2CN(C(c3cnc(C)o3)=O)CC12 C1(C(C)NC(c2nc(COC)oc2)=O)CCCN(C(=O)C(C)NC(N)=O)C1 C=CC(C)CC(=O)NC1CCN(C(=O)C=C2CCC(C(C)(C)C)CC2)C1 C(=O)(CCCCN(C)C(C12CC(C#N)(C1)C2)=O)NC(C)Cc1nccn1C CCCC(CCCO)C(=O)NC(C1CCCN(C(c2cc(C)cs2)=O)C1)C C1(=O)C(N(C)C)CN1.c1(=O)c(CCC)n1.C=CCCOCCOCC C=CCC(CNC(=O)Cc1cn[nH]c1)C(=O)N(CCC(F)(F)F)C c1(C(=O)NCC(CNC(CC(C)(C)OC)=O)O)cc(F)c(Br)c(F)c1N N1(C(C(C)OCC#C)=O)CC2CCC(C1)C2CNC(c1ccccc1C1CC1)=O C(=O)(CCCCCCSC)NC1C(CNC(C2N(C(=O)NC)CCC2)=O)CCC1 c1(C(N2C(COC)CN(C(c3ncccc3C)=O)CC2)=O)cc(O)cc(N)c1C c1(C(N2C(C(CNC(C=C(C)Cl)=O)(C)C)CCC2)=O)cc2cc(C)c(Cl)cc2[nH]1 Cc1cc(C)n(CC(=O)NCC2CC(CNC(c3cnoc3C)=O)CO2)n1 c1(OC)ccc(N)c(C(N2CCC(CNC(=O)C=CCN(C)C)(OC)CC2)=O)c1 Cc1csc(C(N2CCCC2C2(C(=O)NCCN3CCC(C)C3)CC2)=O)c1 c1(OC)ncccc1C(=O)NC1CC(O)C1CC(=O)NOCCO C12(C(NOCC(N3CCC(C)(CO)C3)=O)=O)CCCC(CO1)C2 C12Cc3ccccc3N(C1)C(=O)COC2=O.Cc1cncc(NC2=NCCC2)c1 N1(C(CC)=O)CCN(C)CC1CNC(=O)CNC(=O)C(c1cnn(C)c1)OC c1(C(=O)NC2C(NC(c3cc(Cl)c(Cl)s3)=O)C2)cc(Br)cc(F)c1F c1(C(C(C)C)=O)ccc(NC(C2(c3ccccc3)CCOC2)=O)cc1 c1(COC(Cc2ccc(C)o2)=O)ccc2[nH]c(C)c(C)c2c1 c1(C(N(CC(CC)NC(=O)CCCNC(=O)C2CC2)C)=O)ccc(C)c(C)c1F Cc1ccc(C=CC(N2CCCC(C(C)NC(C34CC5CC3C4C5)=O)C2)=O)cn1 N1(C(CCNC(=O)OC)=O)CC2(CCNC(c3cccc(F)c3Cl)=O)CCC1C2 c1(C(=O)NCCC2(CNC(=O)CC3CSCCS3)CC2)ccc2cccnc2n1 C1(C2(O)CN(C(=O)C(O)C3CC3)C2)(CNC(C2CC(F)(F)C23CCC3)=O)CC1 C1(C(C)NC(c2c(C(C)C)c[nH]n2)=O)CN(C(c2cnns2)=O)CCO1 Cc1nn(CC(N2CCC(C3CCCCN3C(=O)CC3CCCC3)C2)=O)c(=O)o1 C1(NC(C(CCC)C)=O)CCN(C(c2conc2C(C)C)=O)CC1CO C1(C(N(CCCO)C)=O)CCCN(CC=CCl)CC1 c1(C(=O)NC2CC3(CCCN(C(C(C)C#N)=O)C3)C2)ccc2ccccc2c1 C1(CNC(=O)Nc2cnc(C(F)(F)F)cn2)CC12CCSCC2 C1(C(C)N(C)C(C2(N3CCC(C(C4CC4)N(N(C)C)C)C3)CC2)=O)CCCOC1.N C1(CC(=O)NC(CCOC)COC)CN(C(=O)C(C(C)C)NC=O)CCO1 C(=O)(CCCCF)N(CCN(C(=O)C(c1ccccc1)C)C(C)C)C CC(C)(O)C#CC(=O)NCC1CC2CCC1N2C(C1CSCCS1)=O CC1(C)CCN(C(=O)CC2CC(NC(c3cc[nH]c3)=O)C2)CC1 N1(C(C(C)N2CCC2)=O)CC(O)(C(C)NC(c2ccc(C3CCCCC3)o2)=O)C1 c1(OC)ccsc1C(=O)NC(C)(CNC(=O)C(C)C1(O)CCC1)C1CC1 c1(C(N(C)CC2CCN(C(=O)C(F)(F)Cl)CC2)=O)ccc(Cl)c([N+](=O)[O-])c1 c1(C(N(CC(C)NC(=O)C(C)(C)CO)CC)=O)ncnc2c1ccn2C1CC1 CCCCC(O)C(=O)N(CCNC(C1CC(O)C1)=O)CC C(=O)(C(CCOCC)NC(=O)CC12CCCC1C2)N1CC(O)(CCC)C1 c1(C(=O)NCC(C)NC(c2cc(Br)cnc2O)=O)cc2[nH]ccc2s1 C1(CC(N2CCC(C)C2)=O)C2CC1N(C(=O)CCC1N=N1)C2.C1(=O)CN1 c1(CC)ccc2c(c1)nc(CN(CC(C)(O)CO)C)n2CC Cc1ccc(CCC(N2CC(F)CC2CN(C(C23CC(C2)C3)=O)C2CC2)=O)cc1C C1(C)(CNC(C2(OCC)CCC2)=O)CCC(NC(=O)Cn2cnnc2O)C1 N1(C(c2ccc3sncc3c2)=O)CC2(CC2)Oc2cc(Br)ccc21 CC1(C)C=C(C(=O)NC23CC(CNC(c4ccccc4C(F)F)=O)(OCC2)C3)C1 c1(CNC(=O)NC2(CC3CCC(C)CO3)CC2)ccc2cn(C)nc2c1 c1(CC(=O)NC2C(C)CN(C(=O)CC3=CCCCC3)C2)ccc2ccccc2c1 c1(C(=O)NC2(CO)CCN(C(CC(CN(C)C)O)=O)C2)cnc2sccc2c1 N1(C(c2cnc(CCCC)s2)=O)CCN(C(=O)CCC(=O)NCCC)C2CC12 N1(C(C(C=C)O)=O)CCCCC2(CCN(C(C)C(=O)N(C)C(C)C)C2)C1 C1(CCN(C(=O)CCCC2CC2)C)CCCCN1C(=O)CN1CCCOC1=O CC(C)(C)C(CNC(=O)CN1CC2CC2C1)C(=O)NCC1C2CCCC12 c1(C(=O)NCC2(CCNC(C3C(CC)CCO3)=O)CC2)cnnc2ccccc12 c1(C(=O)NCC2(NC(c3ccc(C)nn3)=O)CCCC2)ccccc1P(C)(C)=O c1(SCC(=O)NCCCOc2cccc(OC)c2)nc2c(C)cc(Br)cc2s1 c1(C(N2C(NC(=O)NCCN(C)C)CC(O)C2)=O)c[nH]c2cnccc12 c1(C(N2C(CNC(C3CC(F)C3)=O)CC(F)C2)=O)cccc2occc12 C(C(C)(C)CO)N(CCCC)C(C1CCC(n2cc(-c3ccn(C)n3)nn2)C1)=O N1(C(C(CC)OC)=O)CCC(C2OCCCC2NC(=O)CCc2cncs2)CC1 Cc1cc(N)c(C(=O)NCC(C)NC(c2nnc(O)nc2O)=O)cc1C C1(C(=O)NC(C)CCNC(c2ccc(-c3cccnc3)o2)=O)CC2CCC1CC2 O=C(C1=CC2(CCOC2)C1)NC1CC1CNC(C12CCC(O)(CC1)CC2)=O c1(NC(C2(F)CC(N)C2)=O)ccc(CO)c(C(N)=O)c1 CCC(CNC(c1ccc(C)c2c1CCC2)=O)N=c1cc(C#N)nc(C2CC2)[nH]1 c1(OC)ccc(C(=O)NCC2(O)CCN(C(=O)CCc3ccccc3)C2)nc1Cl Cc1ccc(I)cc1N(CCC(=O)OCCCC1(C)CC1)C N1(C(c2c(C)cncc2)=O)CCCC(F)(CNC(c2cnn(CC(C)C)c2)=O)C1 N=c1[nH]nc(Cl)cc1C(N1CC(F)CC1CNC(=O)COc1ccccc1)=O c1(C(=O)NCC2CCN2C(=O)CC2CC2(Cl)Cl)csc(-c2cnc[nH]2)n1 c1(CC)cccnc1NC(=O)NC1CCCN(Cc2cc(C)n(C)c2)C1 C1(NC(Cc2cc(=N)[nH]cc2)=O)CCCC2CN(C(c3ccc(Cl)[nH]3)=O)CC12 c1(OC)c(Cl)ccc(NC(c2csc(-c3cc(F)c(F)cc3F)n2)=O)c1F C(C)(C)(CCC(=O)N1CCn2ccnc21)NC(c1cc(C(C)=O)[nH]n1)=O N1(C(C(COC)C)=O)CCC(C2CCN(C(C3CC34CCOC(C)C4)=O)CC2)C1 N1(C(C2C(C(=O)OC)CC2)=O)CC2CCC2(CNC(=O)CCS(N)(=O)=O)C1 CC1(C)CC(CC(N2CCCC(n3cccc3C(=O)O)C2)=O)CO1 C1(NC(CN)=O)C2CC3C1C3C2C(=O)NCCN1CCCCC1=O.C(=O)NC C1(O)(CNC(c2ncn(C)c2C(F)(F)F)=O)CCN(C(c2cncnc2)=O)CC1 C1(NC(C(C)(C)CCl)=O)COC2(CCN(C(=O)CNC(N)=O)C2)C1 C(=O)(CCCC(C)(C)C)NCCCCC(C)NC(c1c(Cl)cc(Cl)nc1N)=O C1(NC(CCOC(C)C)=O)CCN(C(=O)Cn2cnc(C(F)(F)F)c2)CC1C C12CCC3CN(CC13)C(=O)CC(CO)C(=O)N2.C1(CC(=O)NCC)CCCC2CC12 O=C1CC2(CCN1)CCN(C1CCC3(CC1)CNC3)C2 C(=O)(C(CCC)C(C)C)NC1(CC=C)CN(C(=O)Cc2ccccn2)C1 c1(CN2CC(NC(=O)Nc3cccc(C)c3)C(F)C2)cc(Br)ncc1F c1(OC)cc(Br)ccc1C(N1CC(Cn2cc(C3(C)COC3)nn2)C(SC)C1)=O CC(C)CC(C(=O)NC1CCC1)ONC(=O)COc1cncc(N(C)C)c1 c1(N(C(c2cccnc2)C(=O)N2CC(OC)C2)C(=O)CO)cc(C)cn(C)c1=O.CO N1(C(COCC)=O)C2CCC1CN(C(=O)C(C1CCC(F)(F)CC1)OC)C2 N1(C(c2c(C)ncs2)=O)CC2CCN(C(=O)CCCn3ccnc3)C2C1 C(=O)(CC(CC)OC)NC(C(N1C(C)(C(=O)NC)CC1)=O)C1CC1 C1(N(C(CC)=O)CCNC(=O)Cc2ccc(C)s2)CCCN(CC2CCCC2)C1 c1(C(N2C3CC(NC(c4cc(Cl)ccc4O)=O)C2CC3)=O)cn2c(n1)COCC2 N1(C2CCCN(C(C=C(C)C(C)(C)C)=O)C2)CCN(Cc2cnsc2)CC1=O CC1SCCC1N=c1cc[nH]cc1S(=O)(=O)NCc1ccc(Br)o1 N1(C(c2cc(CC)n(C)n2)=O)CC(C)N(C(=O)CC2C=NN(C)C2=O)CC1C C1(F)(C(=O)NCCc2c(C(N(CC(F)F)CCC)=O)c[nH]n2)CCOCC1 c1(C(C(=O)N(C2CCN(C(c3c(CC)[nH]cc3)=O)C2)CC)C)c(Cl)cccc1Cl c1(COCCC=C)nc(-c2ccc(N)cn2)nn1Cc1ccncc1 c1(C(=O)NCC2N(C(C(CCC)O)=O)CC(OC)C2)cn(CC)c2ccccc12 CC1CN(C(c2ccc[n+]([O-])c2)=O)CCCN1C(=O)Cc1ccc2c(c1)COC2 Nc1nc2ccccc2nc1-c1cccc(CO)c1 CC(=O)CCCC(C)C(=O)NC1CCC(C(N2CCS(=O)CC2C)=O)CC1 n1(CC)nc(C)c(C(=O)N(CCCNC(C2CC3C=CC2C3)=O)C)c1C c1(C(=O)NCCCCCNC(c2c(CC)ncs2)=O)nnn2c1COCC2 C1(CCN(C=O)Cc2ccoc2)CCC2(CC1)CC2 c1(C(N2CC(C)(CCC(=O)NCc3cnc[nH]3)C2)=O)cnnc(O)c1 C1(CCC)CN(C(c2cc(OC)cs2)=O)CCN1C(=O)C=Cc1cccnc1C c1(C(=O)NCC2C(NC(CNS(C)(=O)=O)=O)CC2)ccccc1CC(F)(F)F N1(C(CCC)=O)CC2OCC(C(N3CCN(c4ccc(CC)cc4)CC3)=O)C2C1 n1(C(C)C)nccc1C(=O)NCC1CCN(C(=O)Cc2cnn(C(F)F)c2)C1 C1(CNC(C(CC)=CC)=O)CC2(CCN(C(c3ccc(C#N)c(N)c3)=O)C2)CO1 NC(=NCC1CC1)N1CCN(c2nncs2)CC1.CC(C)CC(CNC)CO.CCC1CC1 Cc1ccc(CC(=O)NCC2(F)CCN(C(=O)CC3CC4CC4C3)C2)c(Cl)c1 c1(OC)ccccc1C(=O)NCC1(C)CN(C(=O)COCC(C)(C)C)C1 Cc1nocc1CC(N1CC(NC(C2CC2c2cnn(C)c2)=O)C1)=O N1(CC=C)CCC(NCC(C2CC2)N(C(=O)CCc2cn(C)nn2)C)C1=O C1(CN(C(=O)CN(c2ccc(CO)s2)C)CC)CCN(C(C2CCCC2)=O)CC1 N1(C(C(CC)C(=O)OC)=O)CC2CC1(C(F)(F)F)C2.c12cn(nn1)C2 CC(=NO)c1cc(C(=O)NC2CC2NC(c2ncnc(C)c2C)=O)cnc1O c1(C(=O)NCC2CC(NC(C3(COC)CC3)=O)C2)cnc(N(C)C)s1 N1(C(C(CCC)n2cccn2)=O)CCC2CC(NC(=O)C=CS(C)(=O)=O)CCC2C1 C1(C(=O)NC(COC)CNC(=O)C(C2CCOCC2)C)CCCCC1C c1(C(N2CC(C(C)NC(=O)CSCC3CCCO3)C2)=O)cc2ccccc2[nH]1 Cc1cc(C(=O)NC2(C(=O)N(C)Cc3nc(C)cs3)CCCC2)cc(C)n1 n1(CC(=O)NCC(C)NC(=O)C(CO)C(C)(C)C)ncc2cccnc12 C(=O)(C(CC(C)C)NC(C)=O)NC1(CO)CN(C(C(C)NC(CC)=O)=O)C1 c1(C(N(C(c2cn(-c3c(F)cccc3Cl)nn2)C)C)=O)cncc2sccc12 N1(C(C(=O)NCCOC)=O)CC(C)Oc2cc(C)c(Br)cc21 c1(C(CC)(C)C)cn(C2CC3(C(=O)N(CC)CC4CCC(=O)O4)CC23)nn1 C(=O)(C(C)S(=O)(=O)CCC)N1CCC(CN(C(C2(CC#C)CC2)=O)CC)C1 C1(NC(C(=O)NCC)CC)CCC(NC(=O)C(C)(C)C)CC1.C1(=O)CCC(=O)N1 n1(CCC)c(C(=O)NCC(F)CNC(C2OCCO2)=O)cc2ccccc12 c1(C(C)C)ccccc1N(C(=O)COCCO)Cc1ccc(OC)cc1.C1(C)(C)CNC1 c1(C(=O)NCCNC(c2cccc3nc(Cl)cn23)=O)cc(F)c2[nH]nnc2c1 C(CC(=O)NCC1CC(C(=O)NCCSC2CC2)C1)C1(C)CC1.C1(C(N)=O)CCC1 C1(NC(c2cc(C(C)(C)C)n[nH]2)=O)CC2CC1N(C(C1C3COCC13)=O)C2 N1(C(c2c(C(C)C)c[nH]n2)=O)CCC(C2CCN(C(c3cnc[nH]3)=O)C2)C1 c1(C(N(c2cn(CC)nc2)Cc2ncnn2C2CCOCC2)=O)oc(C)cc1C Cc1cc(-c2cscc2C(=O)NCc2cccc(F)c2)cnc1OC(C)C N1(C(C2(C)CCCO2)=O)CCOC(CNC(=O)CNC(=O)CC2CCCC2)C1 CC1(CNC(=O)C2=CSCCO2)CCN(C(=O)CNC(c2ccoc2)=O)CC1 C1(CNC(C(CC)N(CC)CC)=O)C(C2CC2)CCN1C(=O)CCC[N+](=O)[O-] C#Cc1cc(F)c(C(N2CCC(O)(CNC(c3c(C)nnn3C)=O)C2)=O)cc1F N1(C(c2onc(C(C)N)n2)=O)CCC(C)C1CNC(c1cnnn1C1CC1)=O CCCS(=O)(=O)C(C)C(=O)NCC(O)CCNC(c1cnn(CCO)c1C)=O N1(C(CC2CC(=C)C2)=O)CCN(C(c2oc(C)cc2Cl)=O)CC1 Cc1ccc(NC(C2CCN2S(=O)(=O)CC(Cl)(Cl)Cl)=O)c(Cl)n1 c1(NC(C2CC3CC3N2C(c2ccc(CO)cc2)=O)=O)cccc2c1OCO2 N1(C(C2C(OC)C2)=O)CCN(C(c2csc3nnsc23)=O)CC(O)C1 C1(COC(=O)C(F)(F)F)CN(C(=O)CCCSc2ccccc2)C2CC12 C=CC1(C(=O)NC(CNC(c2c(F)cccc2Cl)=O)CC(C)C)CCOCC1 C1(CCNC(=O)NC(C(=O)OCC)C2CC2)CCCCC1C C(CCN=C(NCc1ccn(C)c1)NC(c1cccc(F)c1F)C)NCC(C)C N1(C(C2(NC(C)=O)CC2)=O)CCCC12CCN(C(=O)CC(C)C)C2 c1(C(N2CCC(CNC(CNC(CN(C)C)=O)=O)C2)=O)cnn2ccc(O)nc12 N1(C(CCOC(C)=O)=O)CCC(CNC(C2CCCSC2C)=O)C1(C)C c1(C(N2CC(C(C)NC(c3ccncc3F)=O)C2)=O)cc2c(cc1O)OCO2 C1(NC(C2CC(F)CN(Cc3cc(O)ncc3Br)C2)=O)CCC(F)(F)CC1 c1(C(N2C(Cn3cc(C4(C)CSC4)nn3)CCC2)=O)cncn(C)c1=O N1(C(CC(c2ccc(OC)cc2)NC(=O)COC)=O)C(C)C(=O)OCC1(C)C N1(C(Cc2cccc(C)c2)=O)CCC(N(C(=O)C(O)C2CCC2)C)C(C)C1 C1(NC(C(=O)NC2CCN(C3CCN(C)CC3)CC2)=O)CCCC(C2CC2)C1 c1(C(N2CC(CCC=C)(C(=O)NCCCSC)C2)=O)cccc(O)n1 c1(CC)nc(C(=O)NC2(C)CC(NC(=O)CC(C)c3ccncc3)C2)cs1 C(C(C)(CC(C)C)NC(C1CC(F)C1)=O)NC(c1ccc(COC)o1)=O Cc1nc2c(o1)CCCC2CC(=O)N1CCC1CNC(c1cc([N+](=O)[O-])n[nH]1)=O c1(C(N2CCC(C(=O)NCCCC)CC2)=O)cn2ccc(C3=CCOC3)cc2n1 N1(C(C(CC)C#N)=O)CCC(O)C(C(N2CCC(OC)C2)=O)C1 N1(CCCCCNC(c2n[nH]c(O)n2)=O)CCN(C(=O)CC=C(Cl)Cl)CC1 CCCCC(C)C(=O)NC1CC(NC(=O)CC2CCS(=O)(=O)CC2)C1 N1(C(c2c(C)cc[nH]2)=O)CC2(CC2)CC1CNC(c1ncc(C(F)F)s1)=O c1(C(N2C(CCCNC(=O)Cc3ccco3)CCCC2)=O)cc([N+](=O)[O-])c[nH]1 c1(C(=O)NCC2C(C)CCN2C(c2ncccc2F)=O)cc2cccc(Cl)c2[nH]1 C#CCCCCC(=O)NCCC(C(C)C)NC(c1cc(OC)ncc1F)=O N1(C(C(C=C)(C)C)=O)CC2CCCC(NC(c3nc(O)c(C)s3)=O)C2C1 C12(CCCC(=O)NC(C)CN(C(=O)CC3(CO)CC3)C)CC3CC(CC(C3)C1)C2 N1(C(C(C2CCCCC2)C)=O)CC2CCC(C1)C(NC(C1CC1Cl)=O)C2 C1(C(N2CC(OC)C(C(=O)N(CC(C)O)CC(C)O)C2)=O)CC2CC(=O)C1O2 N1(C(C2CCC(C(=O)OC)CC2)=O)CCC(NC(c2cc(Br)c[nH]2)=O)C(F)C1 C(=O)(C(C(C)(C)C)SCCCCN(C(C(CC)C)=O)C)N(CCCN)C.OC C(C(C)(C)CNC(c1nc(C2CC2)cs1)=O)N(C(=O)CCC1CCCOC1)C Cc1ncsc1CC(=O)NC1(C(=O)NC(c2ccno2)C)CCCC1 N1(C(c2ccnc(C)n2)=O)CCOC(C)C1C(N1CC2(CCS2)C1)=O Cc1c(C(N2CCCN(C(C3CC4CC4C3)=O)CC2)=O)[nH]c2cc(F)ccc12 C(=O)(C1=CS(=O)CCC1)N(C1CN(C(C2(CO)CCCO2)=O)C1)C C1(NC(C2SCCCS2)=O)CC2CC1N(C(c1cc(-c3ccco3)on1)=O)C2 CC(CN(C)C)CCC(=O)N1CC(C(=O)NCCc2ccccn2)C2(CC2)C1 C(C(C(F)(F)F)N1CCN(c2nccc(OC(C)C)n2)CC1)NC(CCC)=O N1(CC)CC(C(=O)NC(C)C(C)NC(C2CC(N(C)C)C2)=O)CC1=O c1(SC)ccnc(N2CCC(CC(C)NC(c3coc(C4CC4)n3)=O)CC2)n1 c1(-c2cn(C3C(NC(C)=O)CCC3)nn2)ccnc(CO)c1 c12ccc(C)c(c1)C(=O)N2.N1(C(=O)OC)CCC(O)C(NC(c2ccon2)=O)C1 c1(CSC)cccc(C(N2CCCC2C2(NC(=O)C(O)C(F)F)CC2)=O)c1C C1(NC(C2(C(C)C)CCN(C(=O)CC3OCCCO3)C2)=O)CCN(C)C(C)C1 c1(CNC(c2c(NC(=O)CC3CCCOC3)c[nH]n2)=O)nc2ccccc2s1 CC(C)CC(CNC(c1cc(CNC(C2(O)CC2)=O)no1)=O)CO N1(C(c2c(CC)n(C)nc2)=O)CCC(C)(C)C(C(=O)NC(C)(C)C(O)C(F)F)C1 C(=O)(CCCS(C)(=O)=O)N1CCC(OCCNC(=O)Cn2cnnc2O)C1 c1(C(N(CC(CNC(C=C(C)c2cccs2)=O)O)C)=O)ccnc2nc(C)nn12 N1(C(CN(C(COC)=O)C)=O)CCN(C(=O)Cn2cc[n+](C)c2)CC(O)C1 C1(C(=O)NC2CC(n3cc(-c4conc4C(N)=O)nn3)C2)CCCC(C(=O)O)C1 c1(Oc2c(COC(Cn3cnc(C#N)n3)=O)cccc2)cc(Br)cc([N+](=O)[O-])c1 C(CCCCC(=O)N1CCCC(CNC(c2cccc(N)c2O)=O)C1)SC C1(=CCNC(CC2C(C)CCC2)=O)CCN(C(=O)Cc2c[nH]nc2O)CC1 Cc1ccccc1C1CCCCN1C(=O)Cc1sccc1C(=O)O C(=O)(CC1CCc2ccccc21)NC(CNC(CC(C=C)CC)=O)CCCC c1(SC)nc(C(F)F)cc(=NC(C)CC(C)NC(=O)C(F)=C(C)C)[nH]1 N1(C(C23OCC(C(=O)OC)(C2)C3)=O)CCCC(N(C(=O)Cc2cccs2)C)CC1 n1(CCn2cc(C3(C)CN(C(C4CCC=CCCC4)=O)C3)nn2)cccc(O)c1=O c1(C(N2CCC(n3cc(-c4ccc(O)cc4)nn3)C2)=O)cc(F)c2c(c1)OCCO2 C1(CNC(c2cnc(C(F)(F)F)cn2)=O)COCCN(C(c2ccccc2)=O)C1 N1(Cc2c(F)ccc(C)c2)CC(C(N2CC3CCC2CO3)=O)CC(F)(F)C1 c1(C(N2CCCC(C)(NC(CC3(C)CC3)=O)C2)=O)cc(F)c(Cl)cc1F C1(NC(C2(NC(=O)OC(C)(C)C)CC2)=O)CN(C(=O)CCF)CC1C1CC1 C12(NC(c3c(C)snc3)=O)CCC1CN(C(c1cnn(C(C)C)c1)=O)C2 c1(C(=O)NC2CC(CCNC(C(CC)N(C)C)=O)C2)cc2c(C)cc(F)cc2[nH]1 c1(C(=O)NCC2C(CNC(=O)CNC(c3cccs3)=O)C2)c(F)ccc2occc12 Cn1ccn2ncc(C(=O)NCCOC3CN(C(=O)C=Cc4cn[nH]c4)C3)c12 Cc1occc1C(=O)NCC1CCN1C(c1coc(C2CCCC2)n1)=O c1(C2CCCN(c3ccc(C=C)cn3)C2)ccc(S(C)=O)cc1 C1(NC(C(C2CCOCC2)OCC)=O)CC(S(C)(=N)=O)C1 C=CC1(C(=O)NCC(C)N(C)C(c2cc(C)cc(Cl)n2)=O)CCOCC1 c1(C(=O)NC2CC(CNC(c3c(C)cccn3)=O)C2)ccc(Cl)c2occc12 c1(C(C2CCC2)NC(=O)NCCC=C)csc(=N)[nH]1 c1(C(=O)NC2C3CN(C(COC)=O)C3CC2)c(C(F)F)ccc2ccccc12 C1(C)(C(=O)NC2(CCNC(C(C)OCC(C)C)=O)CC2)CCC12CCC2 C#Cc1cnc(C(N2CCC(N(C(=O)CC(C)CF)CCO)CC2)=O)c(C)c1 O=S(=O)(N1CCN(C2CCOCC2)CC1)N1CCC2(CCCC2)C1 Cc1cc(C(=O)OCc2ncc(-c3cccs3)o2)c(N)c([N+](=O)[O-])c1 CC1(C)CCC(CC(=O)NCC2CCC(C(=O)NCC3CCC3(C)C)CC2)C1 CCC(CC(=O)N1CC=C(C(=O)N2CCCC(CC)CC2)CC1)C(C)C c1(OC)c(Cl)ccc(C(N2CCC(O)C(NC(=O)CC3CC=CC3)C2)=O)c1F C(CCCCCNC(=O)CC1CCCCC12CC2)N(C(C(C)=C(CC)C)=O)C c1(NC(=O)NC2CCNCCC2CO)nc2ccc(Br)cn2n1 N1(C(C(C)C2CCC2)=O)CCC(O)(CN(C(=O)C=CC(N2CCOCC2)C)C)C1 C1(C(=O)NCCCNC(c2ccccc2F)C)(CF)CC(F)(F)C1 CC1=C(C(=O)NC(C)CC(C)NC(=O)C2=CCOC2)Cn2ncnc2N1C c1(OC)cc(OC)c(NC(=O)C(C)NC(c2cccc(F)c2)C(C)(C)C)cc1Cl N1(C(C2C(C=C)CC2)=O)CC(NC(=O)CCc2cccn2C)CC(C)(C)C1 c1(C(=O)NC2CCC(NC(c3cnn4cnnc4c3)=O)C2)n[nH]c2c1CSCC2 c1(CC(CC)NC(C2CC(C(F)(F)F)CO2)=O)cnccn1 C1(CC(C)NC(CC2ON=C(C)C2)=O)CCN(C(C2(C)COC2)=O)CC1 c1(NCc2c(C)cc(Br)cc2C)cccn2ncnc12 N1(C(C=CCOCCOC)=O)CCC(C2(NC(=O)CCC3CCC(=O)N3)CC2)C1 c1(CNCC2(C(N3CCNC(=O)C(O)C3)=O)CC2)ccc2ncoc2c1 C(=O)(C1=C(Cl)CCC1)NCC1C(NC(Cn2nnc(=N)[nH]2)=O)CCCC1 CC1CC(NC(c2cn(-c3ccc(Cl)cc3)nn2)=O)CN(C(=O)COCCF)C1 N1(C(C(CC=C)C)=O)CCC2C(C(=O)NCCNC(N)=O)C2C1 C=CC(CC)C(=O)NCC(CC1CCCC1)C(=O)NC1(C(N)=O)CCOCC1 C(=O)(C#CC1CCOC1)NCc1ccc(CNC(CC2(C)CCOCC2)=O)cc1 CCCCC(CNC(C1CC1c1ccc(C)s1)=O)NC(=O)CNS(=O)(=O)CC CC1CC(NC(C23C(NC(c4cc(O)ncc4F)=O)C4CC2C3C4)=O)CC(C)O1 Cc1cc(C(N2C3CCC2C(CNC(c2c(C)ncn2O)=O)C3)=O)c(N)c(C)c1 c1(N(CCCCl)C(N2CCN(C(C)=O)CC2C)=O)n[nH]c2c1CCC2C N1(Cc2ccc(OC)cc2Br)CCC2(CC1)CC2(C)C(=O)NC(C)C(C)C C1(C)(NC(CC=C=C)=O)CCN(C(=O)COc2ccc(CC#N)cc2)C1 N1(C(=O)Nc2c(C)cccc2)CCN(C(c2cc(O)cc(Cl)c2)=O)CC1C Cc1ccccc1C(C)CC(=O)NC(C)C(C)(C)NC(=O)CN1CCC(O)CC1 C=Cc1cncc(C(N2CCCC(N(C(c3sccc3CC)=O)CC)CC2)=O)c1 Cc1ccc(C(=O)NC2CCCCN(C(C3C=CCS3)=O)CC2)c2ccccc12 S(=O)(=O)(c1cccc(C(N2CCC(C)(NC(C3CC(C)(C)C3)=O)C2)=O)c1)N(C)C CC(CC(C)(F)F)C(=O)NC(C1(CNC(=O)Cc2ccccc2)CC1)C c1(C(=O)NCC2N(C(C(C(C)C)N(C)C)=O)CC2)cccc([N+](=O)[O-])c1 c1(C(=O)NCCC2SCCS2)cc(F)c(F)cc1Cl C1(N(C(c2ncsc2Br)C(=O)NCC(C)C)CCOC)CCCCCC1 C(c1cc2ccccc2o1)=CC(N1C(CNC(c2nc(CC)[nH]n2)=O)CC1)=O N1(C(=O)CC2CCC(O)C2)CCN(C(c2cc(Cl)nnc2Cl)=O)CC(O)C1 C1(NC(c2[nH]cc(C(C)=O)c2)=O)CC12CCC(NC(=O)C1=C(C)CCC1)CC2 CN1C(=O)CCC1CC(=O)NCCNC(C1CCN(S(=O)(=O)C(F)F)C1)=O c1(C(C)C)ccc(C=CC(=O)N(C(C)CNC(c2cc(C#N)no2)=O)C)cc1 Nc1ccc(C(N2CCCC2CCCNC(c2cc(F)ccc2F)=O)=O)cc1O N1(CCCCCOC(C)C)C2CCC1CN(C(=O)CC1CC1C)CC2 N1(C(C=CCC)=O)CCCC(C2CCCN(C(c3ccc4scnc4c3)=O)C2)C1 Cc1cc(C(N2CC(O)CCC2C(N2CCC(C(C)O)CC2)=O)=O)cc(O)c1 C1(C(=O)NCc2c(C(=O)NCc3ccc(CC)s3)scc2)CC2(CCC2)CO1 N1(C(c2c(CC)n(CC)nc2)=O)CCOC2(C1)CN(C(=O)C(C)C(F)(F)F)C2 CCC1c2cccn2CCN1S(=O)(=O)c1ccc(N2CC3CCC(C2)O3)nc1 c1(C(=O)OC)ccc(C=CC(=O)NCC(F)CNC(=O)C=CS(C)=O)cc1 C(C(C)C(=O)NC1(C)CC(NC(=O)C(C)(O)C2CCC2)C1)SC C1(C)(C(=O)NCCCN(C(C2CCCS2(=O)=O)=O)CC)CCN(C)C1 c1(N2CCCN(C)C(=O)C2)nc(=NC2CCC3(CC3)C2)[nH]c2cc[nH]c12 C1(CNC(Cc2nc(COC)sc2)=O)CC2CC2N1C(C1CCSCC1)=O C1(C(N2CC(CC)C(C(=O)NCC(C)(C)C3CCC3)C2)=O)Cc2nccn2C1 C#Cc1cnn(CC(=O)NCC2CCC2NC(c2ccc(CC)[nH]2)=O)c1 c1(C(=O)NC2CCCN(C(C3(OC)CC3)=O)C2)c(O)ncc2c1CCC2 CC(C)(CNC(=O)C(CO)NC(C1(CSC)CCC1)=O)CC1CC1 N1(C(C(C)NC(CC)=O)=O)CC(O)(CNC(C2SCCCS2)=O)C1 CC(C)CCCCCC(=O)NCC1CCCC(CNC(c2nsnc2O)=O)C1 n1(CCC(=O)NCC(C)CNC(c2scnc2Cl)=O)ccc2cccnc12 c1(C(=O)NC2CN(C(c3cc(CC)nn3C)=O)C3C2C3)cnn2c(C)ccnc12 c1(OC)cc(C(=O)NC2(CNC(C3CCN3C(C)(C)C)=O)CCC2)ccn1 c1(C(N2CC3(CC(C(=O)NC(COC)(C)C)C3)C2)=O)c(F)ccc2[nH]ccc12 C1(C(=O)NC2CCN(C(CCC=CC)=O)C2)COCC1(C)C N1(C(COC)=O)CCC2(CC1)CC2C(=O)N(C(CC(C)C)C(=O)O)C1CCCC1 C1(C(=O)NCCNC(c2c(C)oc(CO)c2)=O)CCC(C2CC2)C1 C=CC1(C(N2CC(CCC)C2)=O)CCN(C(=O)CC2CCOC2(C)C)C1 c1(N(C(=O)C(F)(F)F)CC2C(C(=O)O)C2(F)F)cccc2cnccc12 C1(C(=O)NCC(CN(C(=O)CCOCC(F)(F)F)C)O)CC(=O)N(C2CC2)C1 C1(NC(c2n(CC#C)ccc2)=O)C2CC3CN(C(=O)CCC=C(C)C)C1C3C2 c1(C(N2C(CC)CN(Cc3cccc(SC)n3)CC2)=O)ccc2nonc2c1 Cc1cc(CCC(=O)NC2CC(NC(C3CCCC3C(F)(F)F)=O)C2)no1 CCC(C)(C)C(O)C(=O)NCC1C2CN(C(c3cc(OC)ccc3O)=O)CC12 C(CCC(C(=O)NCCC#N)N(CCCC(C)O)CC(C)C)OCC N1(C(Cn2c(C)nnn2)=O)CCN(C(=O)Cc2cc(Br)ccc2F)C(CO)C1 N1(C(c2nc(C)sc2)=O)CCC(C)(CNC(C2CCC(C(=O)OC)CC2)=O)C1 N1(C(CCC(=O)NCC)=O)CCCCC2(C1)CN(C(=O)CC1CCCC1(F)F)C2 c1(C(=O)NC(C(C)NC(c2c(C)cc(CC)o2)=O)C)cccc(C(C)(C)C)c1N c1(CC)cc(C(=O)N(C2CCCCC2NC(=O)Cc2csc(Cl)c2)CC)n(C)n1 C1(NC(CC2CCC(=O)N2)=O)CC2CCC1C(NC(=O)CCN1CCCC1=O)C2 c1(N2CCC2)nc(C#N)c(Cl)s1.c1(CSC)ccc(C(=O)NC(C)=O)cc1 c1(OC)cc(NC(=O)COC(c2[nH]c(C)c(C)c2C)=O)ccc1OC(F)F CC(C)(CNC(=NCc1ccco1)NCC(O)CN1CCCC1=O)C(F)(F)F C12(CNC(C3CC(SC)C3)=O)CC(CCO1)N(C(=O)C(O)Cc1cnc[nH]1)C2 C1(NC(=O)CC2CCC2(F)F)CC12CC(NC(C1(CC(F)F)CC1)=O)C2 C(=O)(CCCCC(C)C)NCC(COC)NC(C(C)OCCCC)=O CC(C(F)(F)F)C1(O)CC(NC(N)=O)C1.C1(=O)CNC(=O)NCCN(CCF)N1 C=CCCC(C)(C)C(=O)N1CCCC1C(=O)NCc1cc(O)cc(F)c1 C1(NC(=O)C=CC2CCCN2C(=O)CCc2cccs2)CCC(C2CC2)C1 c1(C(=O)NC2(CF)CCN(C(CCC(=O)OC)=O)C2)cnc2ccccc2c1 Cc1ccc(Cl)c(F)c1C(N1CCC(c2cn(CCCCO)nn2)CC1)=O C(=O)(C(CCC)CCCO)NC(CCNC(CS(CCC)(=O)=O)=O)C(C)C C1(CC(N2CCC(CNC(c3cn(CC)nn3)=O)C2)=O)COCC(C)(C)O1 C=CCC(C(=O)NCCC(O)CNC(=O)CSc1nncn1C(C)(C)C)C(C)C c1(C(=O)NCC(CNC(c2nc(C)[nH]n2)=O)CO)cc2cc(Cl)cnc2o1 N1(C(COC(C)(C)C)=O)CCC2(CCOCC2)C(CNC(c2ccc(Cl)[nH]2)=O)C1 Cc1cn(C)nc1NC(=O)C(=O)NC1CC(=O)N(C2CNC2)C1 C(=O)(N=c1ccn(CC(N)=O)[nH]1)C1CCC(C(=O)Nc2ccc(OC)cc2)CC1 c1(CC)cnc(Cl)[nH]c1=NC(CNC(=O)C#CC1CCCCO1)Sc1ccccc1 c1(C(N2C(C)CC(NC(=O)CS(=O)(=O)N(C)C)CC2)=O)cnn2ncccc12 c1(C(N2CCC(CCCCNC(c3c(C)nns3)=O)CC2)=O)c(O)cccc1F CCCC(F)C(=O)NC1CC(CC(=O)NCC2SCCS2)C1(C)C c1(NC(C=Cc2ccc(OC)cc2)=O)ccc([N+](=O)[O-])c(O)c1 C(=O)(C1=C(C)CCCC1(C)C)NC1CC(OC)CN1C(=O)CC(F)(F)C(F)(F)F N=c1nc(N2CCC(C(N3CCC3CNC(C3CCCC3C(F)F)=O)=O)C2)[nH][nH]1 C12(C(=O)OC)CC1CCN2C(=O)Nc1cc(C)oc1C C1(N2CCC(CCC)C2)CCCCCCN1C(=O)NCC(C)C Cc1c[nH]nc1C(=O)NCc1c[nH]nc1C(=O)NCC1CCC(C)C1 c1(N(CCC#C)C)ncnc2c1ncn2CC1CCn2nnnc2C1 C12(OC)CCCC1CN(C(=O)Cc1ccsn1)C2.c1(CC(=O)OC)c[nH]nc1C(F)(F)F Cc1ncncc1C(=O)N(CC(C)(C)CNC(C1(C2CCCCO2)CC1)=O)C c1(C(=O)NCCCN(C(C2CC(CCO)C2)=O)C2CC2)ccc(CCO)cc1F C1(C(N(CCNC(CC2(SC)CC2)=O)C2CC2)=O)CCCN1C(C)=O c1(CNCC2CCC(C(N3C4CN(C)C(C4)C3)=O)CC2)nc2ccccc2s1 Cc1cc(NNC(=O)C(C)ON2CC(C)CC(C)C2)ccc1F N1(C(C(C(C)C)OCC)=O)CC2C3CCC(C2C1)N(CCc1ccccc1)C3 c1(OC)cc(C(=O)NC2CCC(CNC(=O)Cc3cn(C)nc3C)C2)c(Cl)cn1 C12(C(=O)NCCCC3CC3)CCC(C(N3CCCC34CC4)=O)(CC1)C2 N1(C(c2c(N)nccn2)=O)CC(NC(C2CCN(S(C)(=O)=O)C2)=O)CC12CCC2 c1(NC(C2CC(=C)CN2C(c2cnc(OC)nc2)=O)=O)cc(F)nc(F)c1 N1(C(c2cnc(OC)nc2C)=O)CC2CC(NC(=O)C(C)CC=C(C)C)CC1C2 C1(C2(O)CN(C(C3CC3c3cccs3)=O)C2)(CNC(c2c(C)[nH][nH]c2=N)=O)CC1 c1(C(=O)NC2CCN(C(C(CC)SC)=O)C2)cc2c(OC)ccc(C(C)C)c2[nH]1 Cc1nc(N2CC(CN(C)C(C3CCC(O)CC3)=O)C2)cc(C(C)C)n1 N1(C(C2(C(C)C)CC2)=O)C2CCCC1CN(C(=O)C(C)(C)Cc1cnn[nH]1)CC2 N1(C(c2c(C)scn2)=O)CCC(CO)C(NC(=O)Cc2ccccn2)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])N1CCN(C(c2ccc3nc[nH]c3n2)=O)CC(C)C1 N1(C(C(C)CF)=O)CCN(C(=O)Cc2cnn3c2CCCC3)C2CS(=O)(=O)CC12 c1(C(N2CC(NC(c3c(C)n[nH]c3C)=O)C(C)(C)C2)=O)csc2c1CCC(C)C2 C1(C(=O)NC(CCNC(COC(C)C)=O)(C)C)Cc2c[nH]cc2S1(=O)=O Cc1ccc(Cl)cc1-c1cn(C2CC(NC(=O)CNS(N)(=O)=O)C2)nn1 Cc1onc(Cl)c1C(=O)N(C)CC1(O)CCN(C(=O)CN(C2CCCC2O)C)C1 N1(C(=O)CCF)CCCN(C(=O)CC2CCC2)CC1c1ccccc1.C1CC1 C1(CNC(CS(CC)=O)=O)CCC2(CN(C(C3(OC)CC3)=O)C2)O1 C12(CNC(=O)C(=O)NCc3nncs3)CCCC1N(C(=O)Cc1cnns1)CC2 CCCCCCCC(=O)N1CCN(C(=O)C(F)CCCCC)C(C2CC2)C1 C1(COCC)CCCN(C(=O)C(Cc2cnc[nH]2)NC(=O)Cc2cc[nH]n2)C1 N1(C(c2ccc(SCc3ccc(C)s3)cc2)=O)CCC2C(O)CCCC2C1 c1(OC)cc(Cl)c(Cl)cc1C(=O)NC1CN(C(=O)C(C)(O)C(C)C)CC1C N1(C(=O)CC2CSCCS2)CCCC2CN(C(=O)CC3=CCOCC3)CC12 c1(C(=O)NCC2(O)CN(C(CC(C)CN(C)C)=O)C2)cccc(C#CC2CC2)c1 N1(C(C(N2CCC(C)C(CO)C2)=O)=O)CCn2c(-c3cccnc3)nnc2C1 N1(C(c2cc(C(C)=O)c(C)o2)=O)CCCN(C(C2CC3(C2)CC3F)=O)CC1C N1(C(C(C(C)(C)C)OC)=O)CCC2(CC2)CC1C(=O)Nc1cc(C)cc(F)c1 N1(C(C(C)S(N)(=O)=O)=O)CCC2CCCC12CNC(c1csc(=N)[nH]1)=O Cc1cc2nc(-c3cn(C4CCC(C5CC5)OC4)nn3)cn2cc1C C1(C(C)C)CN(C(C2C=CCCC2)=O)CCN1C(=O)C1=C(Cl)CCC1 C1(C2CCOCC2)(C(=O)NCCC2N(C(CSCCC)=O)CCSC2)CC1(F)F C12C3CCN(CC13)C(=O)C1(C)C(C1)C(=O)N2.C(COC)(C1CC1)OC N1(C(CC(C(F)F)NC(c2cccc(CC=C)c2)=O)=O)CCC(O)CC(C)C1 C1(NC(C2CC(OCC)C2)=O)CN(C(c2cc(C(C)(C)C)n[nH]2)=O)CCC12CCC2 c1(NC(C2CCN(C(c3cc(C)c(C#N)cc3)=O)C2)=O)c(Cl)cc(C#N)cc1Cl c1(C(CNC(CCN(CCCO)C(c2c(C)n[nH]c2)=O)=O)O)cccc(O)c1 N1(C(CCC2(C)CC2)=O)CC2CCC(NC(c3ccc(C(C)(F)F)cn3)=O)(C2)C1 c1(C(N2CCC(N3CCN(C(C(CC)(F)F)=O)CC3)C2)=O)cncn(C)c1=O c1(C(=O)NCC2(CC(N3CC4(C=CCO4)C3)=O)CC2)cccc(F)c1F c1(C(N(C2CCN(C(C)=O)CC2)NC(C(CC)(C)SC)=O)=O)cc2ccccc2s1 CC1CCN(C(=O)NC(c2nnc(S)n2C)C)CC1F N1(C(C(C)(C)C2CCC2)=O)CCOC2(C1)CN(C(C1CC(n3ccnc3)C1)=O)C2 N1(C(CCSCC)=O)CCC(NC(c2ncccc2C)=O)CC(C)(C)C1 C1(CC(=O)OCCOC)(N(C(=O)COCCC2CC2)CC)CCOCC1 c1(C(N2C(CC(=O)N(C(COC)C)CC)CC(F)C2)=O)ccc(=O)n(C)c1 CCCCCC(=O)NC(C1CN(C(=O)CC(c2cccs2)C2CC2)CCO1)C C(C(=O)NN1CCCC1C(N)=O)=CC(C)(C)CN1CC(CO)C(C)(C)C1 C=CCC(C(=O)NCC1CN(C)CCN1C(=O)COCCCN=[N+]=[N-])C(C)C C1(C(=O)NCCN(C(C(C)C2CCCC2)=O)C)CCCS(=O)(=O)C1 C(C(CN=c1nc(N2CCCC(C)(OC)CC2)c2c([nH]1)COC2)C(C)C)OC c1(CC(=O)NC(CNC(C2C(CC)N(C)CC2)=O)CC)ccc2n[nH]cc2c1 C#CCC(C(=O)NC(c1cncc(F)c1)C)NC(=O)C=C(C)C(=O)NC CC1CCC(NC(=O)C(=O)Nc2ccncc2)CN1C(c1nnn(C)c1N)=O C(=O)(C(C)(C)C(C)(C)O)NC(C)C(C)C(=O)NCC(CO)C(C)C c1(C(N2CC(C)(NC(C3CCCCC(=O)C3)=O)C2)=O)cccc2cnsc12 C1(C(=O)NCCN(C)CCNC(C2CC(O)C(F)C2)=O)CCCC(C#N)C1 c1(C(=O)NC2CC(NC(c3ccc(C(C)C)s3)=O)CC2O)cc2c(s1)CCC2 Cn1ccnc1COCC(=O)NCCC1CN(C(=O)CN2CCSCC2)C1 C#CC1CC2CCC1N(C(c1ncc(CC)s1)C(=O)NCCC#N)C2 N1(C(CN2CC(C)(C)C2)=O)CC2CCCC(C1)N(C(=O)C(C#N)C1CC1)C2 c1(CC)cc(C(=O)NCC(C)CN(C(=O)CC(C)n2ccnc2)C)cs1 N1(C(C2N(CCCC)CCCC2)=O)CC(NC(=O)Cn2nnc(=N)[nH]2)C2(CC2)C1 c1(C2CN(C(=O)CCc3nc(C4CC4)no3)CC2O)nc2ccccc2[nH]1 c1(C(=O)NC2CC(CNC(CCN(S(CC)(=O)=O)CC)=O)C2)c(Cl)ccc(F)c1F C1(c2[nH]cc(C)n2)NC(=O)N(CCN(C)C)C2=C1C(=O)N(C)C2C c1(OC)ccc(CN2CCC(CCNC(c3cccnc3)=O)CC2)c(Cl)c1O C=C1COCCN(C(c2cnc(SC)s2)C(=O)NCc2ccccc2)C1 C(=O)(CCCCCNC(C)=O)N1CC(CNC(C=C(CC)C)=O)C(C)C1 C1(C(=O)NCCCCN(C)C(C2(Br)CC2)=O)CCn2cnnc2C1 Cc1nc(Cn2cc(-c3ccnn3Cc3cccnc3)nn2)c(C)s1 C1(C(=O)NCC(C(F)(F)F)OC)CC2(CC2)C12CCC2 CC1(C)CCC(C(=O)NC(CC2CC2(F)F)C(=O)O)CO1 N1(C2(C(=O)NCCNC(C3(C(F)(F)F)CC3)=O)CC2)CCOCC1 C=CCC(CNC(c1cncc(OC)n1)=O)C(=O)NC(C1CCC1)C Nc1cc(C(N2CCC3CC2CN(C(C2CCOC2)=O)C3)=O)c(F)c(F)c1F C(=O)(CCCC(=O)N(CCCNC(=O)CC(C)CC1CCCCC1)C)OC Cc1cncc2cc(C(N3CC(O)CC3CNC(c3ncncc3Cl)=O)=O)sc12 C1(NC(=O)C=Cc2ncc[nH]2)CC2CC1CN2C(c1cscc1C(N)=O)=O N1(C(c2ccc3c(c2)CCO3)=O)CC2C3C=CC(C3)C2C1 C(C)(CCC(=O)N(C(C)CNC(c1cnc(-c2ncccn2)s1)=O)C)SC c1(C(=O)NC(C2CCN(C(CCOCC(C)C)=O)C2)C)ccc2c(c1)C(C)CO2 N1(C(C2CC(N(C)CC)C2)=O)CCC(C)C1C(=O)N(C)CC1CCCC1(C)C c1(OC)ccnn1OC(C1CC1NC(=O)CCC)=O.C1(OCC(=O)CN)CCCC1 c1(C(N2CCCC(C)(C(=O)Nc3c(Cl)ccnc3Cl)C2)=O)c(Cl)ccc(Br)c1F C(CNC(c1c[nH]c(=O)cn1)=O)(CC(=O)N(C)CC1CN(C)CCO1)OC C(N=c1ccnc(C(C)(C)C)[nH]1)C1(C)CCN(C(CCCNC(C(C)C)=O)=O)C1 CC(C)CC(C(=O)N(CC(O)CN(C)C(C1CCCN1N=O)=O)C)N(C)C N1(C(c2ccc3c(n2)COCC3)=O)CC2(CCN(C(C3CC4CC4C3)=O)CC2)C1 N1(C(c2c(C)nc(C)n2O)=O)C2CCC1CN(C(c1ccc3c(n1)NCC3)=O)C2 c1(CNC(c2cn(C)nc2Cl)c2n(CCOCCOC)nnn2)cnc(C)nc1 C12COCCC1CC(=O)N2.N1(CC)CCCC1C1(C(=O)O)CC1.N(C)(C(C)=O)CC C1(NC(CC(C)SC)=O)CCN(C(=O)CCCc2cncs2)C1C1CC1 C1(OCC(=O)NC2CCOC2)CCN(C(=O)CC2CC(O)C23CCC3)CC1F N1(C(C(F)OC)=O)CCOCC12COCCN(C(C1CCC1(C)C)=O)C2 N1(C(C2CC3(C(OC)CC3)C2)=O)CCCOC(CNC(=O)CCCCN(C)C)C1 c1(CC)c(OC)cccc1C(=O)NCc1c[nH]nc1-c1ccc(OC)cc1 Cc1ccc(C)c(CC(=O)NCC2CCN(C(C3(C)C=CCC3)=O)C2)c1 C1(NC(c2c(OC)c(C)sc2)=O)CCN(C(c2cncs2)=O)CCC1CO C12(C(N(c3nccc(C(=O)OC)n3)C3CNCC3(F)F)=O)CCC(CC1)CC2 C(=O)(CCCC(=O)NC(C)C)N(CCC)CCNC(C1CC(F)(F)C1(F)F)=O C(=O)(CCCNC(N)=O)NC(CN(C(=O)CCN1CCC1)C)CO CN1CCCC(C)(C(N2CC3CCC3(CC(=O)N(C)OCC(F)(F)F)C2)=O)C1 C(=O)(C(CCCOC)NC(=O)CC1CCC(=O)CC1)NC(CC)C(=O)N(C)C C1(NC(C=C(C)C)=O)CC2(C1)CC(NC(c1cc(C(F)(F)F)ncn1)=O)C2 N1(CCNC(CN(C(=O)CC2CCCC2C)CC#C)=O)CC=C(C)CC1 c1(C(=O)NCc2nc(CNC(C3(O)CCCC3)=O)cs2)ccc2[nH]nc(Cl)c2c1 C1(CC)CN(C(=O)Cn2ncc(Br)n2)CCC1NC(c1cccnn1)=O CC(C)(C)CC(O)C(=O)NCC1C(CNC(=O)C(F)n2ccnc2)C1(F)F CC1CCN(C(C2CCCC2F)=O)CCN1C(C1CC2CC2C1)=O C1(N(C)C(c2cccc(-c3cnco3)c2)=O)CC2CCC(C1)N2C(=O)CO C=C(Br)CC(C)(C)C(=O)NC1CC(C)(CNC(C2CC(O)C2)=O)C1 c1(C(=O)NC2CC(C(C)NC(C(C(C)O)(F)F)=O)C2)cccc2cc[nH]c12 C12(NC(c3cccc4ncnn34)=O)CCCC1N(C(=O)CSC1CC1)CC2 C(CC(=O)N1CCNC(=O)CC1)(C(F)(F)F)NC(CC1(C)CCOC1)=O N1(C(CCN(C)C(C2CCCC(=O)CC2)=O)=O)C2CCC1CC1(C2)N=N1 C1(NC(c2occ(C)c2C)=O)CC(F)CN(C(C2CC(=O)N(CC3CC3)C2)=O)C1 C1(NC(c2c(C(C)C)ocn2)=O)CC2CC1N(C(c1cnccc1Cl)=O)C2 N1(C(C2(NC(C)=O)CCCCC2)=O)CC(NC(=O)CCC(F)F)CC2(CCC2)C1 Cc1nc(CN(C(=O)CC2CCCC2NC(c2csc(Cl)c2)=O)CCO)n[nH]1 N1(C(C=C(C)Br)=O)CCCC1C1CCCCN1C(=O)CCCN(C)N=O c1(C(=O)NCCC(C)N(C(=O)CCCc2ccsc2)C)cc2ccc(O)cc2[nH]1 N1(C(COCCCCC)=O)CCC(OCCNC(C2CCC(C)C2)=O)CC1 c1(OC)c(C(=O)NC2C=CCN(C(C3CCCC3(C)C)=O)C2)nc(O)nc1O N1(Cc2ccc(SC)o2)CCC2(CC1)CC2CC(=O)NCCS(=O)(=O)O C#CCCCCCCC(=O)NC1CCCC1CC(=O)NCCc1ocnc1CO C(C)(CCC(=O)NC)OC.N12CCC(CC1)NC(=O)CCCCN(C)CC2 N1(C(c2cc(Br)c[nH]2)=O)CCC2(CCC2)C(CNC(C2(O)CCSC2)=O)C1 CC1CC(c2nnnn2CC(F)F)(NCc2csc(N(C)C)n2)CS1 C=CC1CCN(C(=O)C#CCNC(=O)CC2CC(C)=NO2)CC1 N1(C(COC)=O)CC(F)(C(=O)NC(C2CCOCC2)C)C1 CCC(CCOC)C(=O)NC1CC2CC1N(C(c1ccc(Br)c(O)n1)=O)C2 Cc1ccc(C(=O)C(=O)NC2CC2NC(=O)C(c2ccc(Br)cc2)C)cc1 c1(N2CC3C(NC(=O)CC4(O)CCOC4)C3C2)nc(Cl)nc2c1CCC2 C(CCC(c1ccccc1)NC(=O)CC1COC(=O)C1)NC(=O)C=C1CCCC1 c1(C(=O)NC2(C(=O)NC3C(C)(C)C3)CSC2)ccc(C#N)[nH]1 Cc1cc(C(N2CC3CCC2CN3C(=O)CCC2CC2(F)F)=O)c(C)nc1C Cc1ccc(C)n1CCC(=O)NC1CC(F)(CNC(=O)Cc2csc(Cl)n2)C1 C1(NC(CCOCC#C)=O)CN(C(c2ccc(F)c(OC)c2)=O)C2CCCC12 C(=O)(CC1=CCOCC1)NC(CC(C)NC(CSc1c(C)cccc1)=O)C CCC(C)(C)C(O)C(=O)NCC(CO)NC(=O)Cc1ccc(C#N)cc1Cl c1(C(=O)NC(C(CO)NC(C(C)OCC#C)=O)C)ccccc1N(C)C(C)C C1(CNC(C2C(C3C(C)C3)C2)=O)CCN(C(c2cnccn2)=O)CC1(F)F N12CCCC(C1)CCNC(=O)C2.c1(OC(=O)NCCN)cccnc1 N=c1cc(C(N2CCCCC2C2(NC(c3ncccc3Cl)=O)CC2)=O)cc[nH]1 N1(C(c2ccc(C#C)cn2)=O)CC(C2CN(C(c3c[nH]c(=NCC)s3)=O)C2)C1 C1(C(=O)NC2(CCC=C)CC2)CC2(C1)CC(CC(=O)NCC1CCC=CCCC1)C2 Cc1cc2occ(C(=O)NCC(C3CCCC3)NC(C3(O)COC3)=O)c2cc1C C(C)(CCC(=O)N(C)CCc1ncon1)NC(CC(C)F)=O N1(C(CC2(C(=C)F)CCC2)=O)CCN(C(C2CC(C3CC3)=NO2)=O)CCC1C N1(CC2(CNC(C3CCCOC3)=O)CCCC2)CCCCCC1 C1(C)(CNC(C2CC(C)SCC2)=O)CCCN(C(C23CC2COC3(C)C)=O)C1 c1(OC)c(C(N2CCOCC2CNC(C2CC3CCC2O3)=O)=O)nc(O)nc1O CCC(C)CC(CO)NC(c1c(CNC(C2CC(O)C(F)C2)=O)nnn1C)=O C(C(=O)N1CC(CNC(=O)COc2ccnc(C)c2)C(O)C1)(C(C)C)NC(C)=O Cc1cc(CC(=O)NC2CN(C(c3cncc(C(F)(F)F)n3)=O)CC2O)c(C)s1 CC1CCc2[nH]c3ccc(C(=O)NC45CC(Br)(C4)C5)cc3c2C1 O=S(=O)(c1c[nH]c2cc(Br)ccc12)NCC1CCCn2cc(C(F)(F)F)nc21 c1(N(C)C)cncc(C(=O)NC2CCC2CNC(c2c[nH]ccc2=O)=O)c1 C1(N2C3CC(OCC3)CCC2=O)CCN(Cc2ccccc2)CC1.C(N)=O.CO CCCCC(C)C(=O)NC1CC12CCN(C(=O)CC1CCC(C)(C)O1)C2 c1(CC)nn(C)c(Cl)c1C(=O)NCC(CC)NC(c1cc[nH]c(=NC)c1)=O C(=O)(CCCCCC(C)C)NCC(C)(C(C)C)NC(CC(CC)C)=O N1(C(c2cnc(CCCC)s2)=O)CCCOC(CCNC(C2CCC(=O)N2)=O)C1 CC(CC(=O)NOCCCC(F)(F)F)N(C)C(c1cn(C)nn1)=O Cc1cccc(C(CNC(=O)Cn2nc(C)cc2C)NC(c2c[nH]nc2C)=O)c1 c1(CNC2CC(NC(c3cccc(-c4ccncc4)c3)=O)C2)cc(O)cc(F)c1 N1(C(C2(COC)CC2)=O)Cc2ccccc2C(NC(=O)C(c2ccc(C)s2)C)C1 c1(CC(=O)NC2C(C(N(c3ccc(Cl)c(O)c3)CC)=O)CC2)cnc(O)nc1O C(CCCCC(=O)NC1CC2(NC(C3CC(C)(O)C3)=O)COC1C2)OCC C1(CC(=O)NCCC2(NC(Cc3c(C)non3)=O)CCCC2)CC(C)(C)CO1 C=C(C)C(CC(=O)NCC1=CCCN(C(c2cnc(Cl)s2)=O)C1)OCC C12(C(=O)NCC(=O)OC(C)(C)C)CCN(C(=O)C(c3cccs3)N(C)C)CC1C2 c1(OC)cc(Br)c(F)cc1NC(=O)CC1CCN(S(=O)(=O)c2cccnc2)C1 N1(C(C(C)OCCOC)=O)CCC(C(N2CC3(C2)CN(C)C3)=O)CC1C c1(-c2nc(CC(C)OC)nn2C(C)C)c[nH]c2ccc(Br)cc12 C(=O)(CC(C)(C)n1cc(CCC2CCOCC2)nn1)N(C(=O)C(C)C)CCOC C1(C(=O)NCC2CN(C(c3c(OC)n[nH]c3)=O)C2)Cc2cccc(Cl)c2C(=O)O1 Cc1cccc2c1S(=O)(=O)CC2NC(=O)CC(C)(F)F Cc1cn2c(C(=O)N(C3CCC(NC(=O)Cc4ccco4)C3)C)cnc2s1 C12CCN(CC1)C(=O)CNC1CC(C1)CCO2.C(C(=O)NS(C)(=O)=O)=CCC C1(C(=O)NC2CC(C)(C)N(C(=O)CCc3cnc(O)[nH]3)C2)CCc2c[nH]nc2C1 N1(C(Cc2ncc(C)o2)=O)CCN(C(=O)C(C)CSC(F)(F)F)C(CO)C1 C12(C(=O)NC(c3ccc(C(C)(C)C)cc3)CO)CCCN(CCC1)C2 C1(C(C)C)CCCN(C(c2ncccc2O)=O)C1.C12(O)CN(C1)C2 C(CC(C(=O)NCCc1ccccc1F)NC(=O)CC1COCCO1)SC Cc1cc(N)c(C)nc1C(=O)NCC(=C1CN(C(c2c(F)ccnc2Cl)=O)C1)F Nc1c(C(N2CCOCC(NC(=O)CCc3cn[nH]c3)C2)=O)ccnc1Br c1(C(=O)NC2CCC2CNC(=O)C(c2ccc(Cl)cc2)(F)F)n[nH]c2c1CCC2 n1(CC)ccc(C(N2CCC(O)(CCNC(C34CSC(C3)C4)=O)C2)=O)cc1=O C1(NC(C(C)C2CCCO2)=O)CN(C(=O)CCNC(C2CCC2)=O)C2CCCC12 CCC(C)CC(C)C(=O)NC12CC(CNC(=O)CCOCCOC)(C1)OC2C C(=O)(C(O)C(C(C)C)OC)NC(CC)C(N1CCOC(C(N)=O)C1)=O N1(C(CCC#C)=O)CC2(CCN(C(c3ccc(C(F)(F)F)cc3SC)=O)CC2)C1 c1(CN(CC=C)CCc2ccc(F)cc2)ccc(OC)c([N+](=O)[O-])c1 N1(C(CC2(C)CC2(F)Cl)=O)C2CCC1CC(NC(=O)CCn1ccnc1)C2 c1(CC(N2CCN(C(=O)CCc3cncs3)C3CC23)=O)cnc(O)nc1O Cc1cc2c(cc1C)OC(C(=O)NC1CC(NC(c3cccc(Cl)c3F)=O)C1)C2 CCCCC(CN=c1ncc(C(F)F)c[nH]1)NC(c1ccn(CCO)c(=O)c1)=O C1(NC(C2C(C)(C)OCC2)=O)CN(C(=O)Cc2ccc(F)cn2)CC(F)(F)C1 C(=O)(C(O)C1=CCCCC1)NC(CC(C)C)C(=O)NC1CC(C)N(C)CC1C c1(C(=O)NCCSC(C(=O)N(C)CC)CC)ccncc1NC N1(C(C)C)CCCC(C(=O)NCC(C)CNC(=O)C(C)C2CCCO2)C1 c1(C(=O)NC2CN(C(c3cc(CC)cc(N)c3)=O)C(C)C2)cc(C)c(C)nc1O N1(CC2(NC(c3n(CCC)ccc3)=O)CC2)CCN(C(=O)C(O)C2CCC2)CC1 C1(NC(c2scnc2C2CC2)=O)CC2(C1)CN(C(C1CCOCC1)=O)C2 c1(OC(C)C(=O)NC2CC(N(C)C(c3ccncc3F)=O)C2)cccc(Cl)c1 N1(C(C2(CC#C)CC=CCC2)=O)CC2CC(NC(c3cccc(O)n3)=O)CC1C2 CC1(NC(C2(C(F)F)CCCO2)=O)CCN(C(=O)CS(N)(=O)=O)CC1 C(=O)(C(C)C(=O)NCCCCN(C)C(C1(F)CC1C)=O)OC N1(C(CCCCCOC)=O)CC2(CCN(C(=O)C(O)CCl)C2)C1 c1(Nc2cccc(OC)c2CN2CC(C)NC(=O)C2C)ccc(F)cc1C#N CC1=C(C(=O)N2C3CCC2C(F)C(NC(C2CC2(C)C)=O)C3)CCS1(=O)=O n1(CC)nc(C(=O)NCCC2(NC(C3CCN(CC(F)(F)F)C3)=O)CC2)c(C)n1 C1(C(N(C(c2c(Cl)cccc2Cl)C)C)=O)CCc2nnn(C)c2N1 N1(C(c2c(C)nco2)=O)CC2(CC2)CC1CNC(c1cc(C)[nH]n1)=O C12(NC(CCN(CC)CC)=O)CC(C1)N(C(=O)C(C(C)O)NC(=O)C1CC1)C2 C1(CNC(c2scc(C)c2Cl)=O)(NC(=O)Cc2c(Cl)cnn2C)CCCCC1C c1(C(N2CCCCCC2CNC(C2(CF)CC2)=O)=O)ccn2cnnc2c1 C=CC1(C(=O)N(CC(CC)NC(=O)CCc2cc(C)sc2C)C)CCOCC1 CC1CCN(C(=O)C(=O)N(C)CCN(C(=O)CC(C)CN(C)C)C)CC1 C(=O)(C1Cc2c(Cl)cccc21)N1CC(CNC(c2c3ncc(C)n3ccc2)=O)C1 c1(CC(=O)N(C(C)CNC(=O)Cn2cncn2)C)ccc(OC(F)(F)F)cn1 N#Cc1cc(F)c(NC(C2CN(Cc3cccc(O)n3)CCS2)=O)c(F)c1 C(=O)(C1=CCCCO1)NC(C)CC(C)NC(=O)C=C1CCN(C)CC1 N1(C(C(CC(C)(C)NC(C2C3CCCC23)=O)F)=O)Cc2ccc([N+](=O)[O-])cc2C1 c1(C(=O)NC2C(NC(Cc3c(CC)con3)=O)COCC2)ccc(F)c(C)c1 C1(C(=O)NCC(COC)NC(=O)COCCCCC)CC(F)(CF)C1 CC1(NC(c2coc3c2CSC3)=O)CCCN(C(=O)CCn2cncn2)C1 N1(C(C2C(CC)(CC)CCC2)=O)CCCN(C(c2ccc(C)cc2F)=O)C(C)C1 N1(C(C(C)OC2CCCC2)=O)CC2(COC(CN(C(=O)C3=NNC(=O)C3)CC)C2)C1 CC1CCN(C(=O)C(=O)N=S(C)(C)=O)CCN1C(C1CCCC(=O)N1C)=O C=C1CCC(C(=O)NC2CCC2NC(=O)COc2ccccc2C)CC1 N1(CC(=O)OCC)CCC2(CC1)CC(C)N(C(C1CCCN(C(C)=O)C1)=O)C2 O=C(C1=NOCC1)NCCCOC1CCN(C(c2cn[nH]c2)=O)CC1 c1(NCC2(C(N3CCCC3CO)=O)CCC2)cc(C(F)(F)F)nc2ncnn12 C1(CC)CCN(C(=O)CSC(C)(C)C)C1C(=O)NC1CC(O)C(O)C1 C1(OCC)CCC(C)(C(=O)NC2C3CN(C(=O)CCCC(C)=O)CC23)CC1 C1(CNC(CCC)=O)CC(C)CCN1C(c1cnc(C2CCC2)cc1C)=O c1(C(=O)NCCOC2CN(C(C3(C#N)CC3)=O)C2)ccc2c(c1)C(=O)NCC2 C(=O)(CS(=O)C(F)(F)F)NCCNC(C(c1c(OC)ccc(F)c1)=O)=O C1(F)(C(=O)OCC)CCC(CNC(=O)C(C)(C)C2CCCC2)CC1 CCC(C)(C)CCCC(=O)N1CC2CC(NC(C3C(F)(F)C34CCC4)=O)C1C2 C(CNC(=O)Cn1cncn1)(C(C)(C)C)NC(C1CC(C)OC1)=O C(=O)(C1CC(=O)Nc2ccccc21)NCC1(O)CN(C(Cn2ncc(C)c2)=O)C1 CCCC(C#N)C(=O)N1CCC(O)C(NC(=O)C=Cc2cnn(C)c2C)C1 CCC(Cc1ccccc1C)C(=O)NC1CCCC1CNC(C1CC1C(N)=O)=O C1(C(C)C)CN(C(=O)CCCCCF)CCN1C(C1C(C)C1C)=O O=C(C(O)CC(F)(F)F)NC12CC(NC(=O)CN3CCCOC3=O)(C1)C2 c1(C(CNC(C2CCOC(CC)C2)=O)NC(CC=C=C)=O)ccc(Cl)cc1Cl N(C1CCOc2ccc(Cl)cc21)C(c1n(CCSC)nnn1)(C)CC1CCOCC1 C1(SC)CN(C(c2[nH]ccc2CO)=O)CC1NC(=O)COCc1ccnc(O)c1 CCCCC(C)CCC(=O)NCC(O)CCNC(=O)CNC(c1ccoc1)=O CC1=NOC(=O)C1CC(=O)NCCOCCN(C)C(C1(Cl)CC1(F)F)=O C(=O)(C1=C(SC)CCCC1)N1CC2C(CNC(C=C(CCC)C)=O)(CC2)C1 N1(C(c2ccc(C(C)C)s2)=O)CCCC(N(C(=O)COCC2CC2)C)CC1 C1(N(C(C(C)n2ccnn2)=O)C)CN(C(C2(C#N)CC=CC2)=O)CC1(C)C c1(NC(c2cc(Br)cs2)C)[nH]c(=NCc2cncc(C#N)c2)nc2c1ncn2C C1(C(N2CCC(CN(C(c3c(C)onc3)=O)C)CC2)=O)Cc2nn[nH]c2C(C)C1 C(=O)(C1=CCCC1(C)C)NC1CCCN(C(c2cccc(OC)c2)=O)CC1 C1(NC(C=COCC)=O)CN(C(C23CC4CC(CC(C4)C2)C3)=O)CCC12CCC2 C1(CC=C)(NC(C(C)OCC=C)=O)CCN(C(C2CCCCN2C(N)=O)=O)C1 c1(C(=O)OCC)cc(C(=O)NCC2C(=O)N2)on1.C(=O)(NC1CC1)OC.CCS C(=O)(CCCC(=O)OC)N1C(C(=O)NC2CCN(C3CC3)C2)(COC)C=CC1 N1(C(c2n(C(CC)CC)ncc2)=O)CC(CSCC(C)C)CC1CCNC(=O)CC CCC(C)C(O)CC(=O)NCC(C)(C)CC(=O)N1CC(=O)NC(CC)C1 c1(CNC(c2nccs2)=O)cccc(OC(F)(F)F)c1.C12CCC(C1)NC(=O)C2 n1(CC(N2C(CNC(C3(C(C)(C)C)COC3)=O)CC2)=O)nnc(-c2ccsc2)n1 C(C(F)(F)C(=O)N(CC(=O)NC1CCCC1(F)F)C)N(C)C CCC(CCC(=O)N1CCOCCC1C(N1Cc2ncsc2C1)=O)OC C1(C(=O)NC(C(=O)NCCCN(CC)CC)CCF)CC12CCOCC2 CC(O)CCN=c1cc[nH]cc1S(=O)(=O)N1CCCC(C2(C)CC2)C1 CCC(C(=O)N(CC(C)(C)NC(=O)Cc1ccc(C)c(C)c1)C)C(C)(F)F CCN=c1[nH]c(C(=O)NCC2(F)CC(NC(=O)C(C)(C)C(F)F)C2)cs1 CC(C)C(F)(F)CCNC(=O)C(C1CC1)N(C)C(c1scnc1Cl)=O c1(NC(CC2N(C(c3c(C)oc(-c4cccs4)n3)=O)CC2)=O)cccc(F)c1F c1(C(N2C(C(=O)Nc3nccc(C)n3)CSCC2)=O)ccc(Br)cc1Br C1(CNC(CCNC(C2CCOCC2)=O)=O)CCN(C(c2ns[nH]c2=O)=O)CC1 CC#CCCCC(=O)NC1(CF)CCN(C(=O)CCC2CC(OC)C2)C1 C(N=c1[nH]nc(C(F)(F)F)s1)C1OCC(CNC(COCCOC)=O)C1 C12(C(=O)NCc3nc(COC)sc3)CC(CN1C(c1cnsc1C)=O)C2 c1(-n2c(-c3nc(C)c(C)o3)nc(C3CC3(C)C)n2)ccc(C(F)(F)F)c(Cl)c1 C1(CC(=O)NCC2CC(NC=O)C2)CC2(CCC2)CO1.N12CSCC1C2=O.CCO C12(NC(C(C3CCOCC3)OC)=O)CCCC1N(c1cc(O)ncn1)CC2 c1(C(N2C(CNC(C=C(C)Cl)=O)C(C)CC2)=O)ncnc2c(C)csc12 C1(CNC(N2C3CN(C(C)C)C(C3)C2)=O)CCOCC12CCCC2 N1(C(=O)COc2ccsn2)CC2CCCC2(C(N2CCC(F)(C(N)=O)C2)=O)C1 N1(C(Cc2scc(C)c2)=O)CCC2CCC(NC(=O)Cc3nc(C)sc3C)C1C2 c1(CC(=O)NCCC2CCCCN2C(=O)COC2CCC2)ccc2c(c1)CCC2 C1(SCC)CN(C(C2(c3cccs3)CC2C)=O)CCC1NC(=O)C(O)C(C)C C1(CCNC(CN(C)CC)=O)COCCN1C(c1ccc(C2CC2(F)F)cc1)=O N1(C(c2cc(CNC(C)=O)on2)C(=O)NCCCSCC)CCCC(C(C)C)C1 C(=O)(CCCC(C)(C)C#N)NCC(C)CNC(=O)CCCC1CCCO1 N1(C(COC(C)=O)=O)CCC(C)C(N(C)C(C2C=CC=CC=C2)=O)C1 C1(C(=O)NCC(=O)N(C)C)(CC)CCN(C(C2CN(C)C2)=O)C1 C1(C(=O)NCC2(C(N)=O)CN(C(C(CC)F)=O)C2)CCN(C)C(=O)C1 C12(C(=O)NCC(C)(C)NC(C3CC(C)(C)OCC3)=O)CCOC1CC(=O)NC2 C1(O)(CCNC(c2ccc(C#C)o2)=O)CCCN(C(c2c(C)ncnc2C)=O)C1 C(CCC(F)(F)F)N(C(C1(NC(c2ccn(C)n2)=O)C(C)C1)=O)C CS(=O)(=O)C1CC(C(=O)NCC=CCNC(C2CCc3nn[nH]c3C2)=O)C1 C1(CC=C)C(NCc2ccc(-c3ccccc3)o2)CC1C(=O)OCC N1(C(COC2(C)CN(C(Cn3ncc(C#C)c3)=O)C2)=O)CC2(COC(C)(C)C2)C1 c1(OCC#C)ccc(CN2CC(C(=O)NCC3CCCN(C)C3)C2)cc1 N1(C(C=CC)=O)CCCC(N2CCN(C(=O)C(=C3CCCCC3)F)CC2)C1 c1(C(C2(Cl)CC2)=O)nc(C(F)(F)F)ncc1Cl.c12cn(nn1)C1CCN(C1)C2 CC1(C)CCC(CNC(c2ccc(O)cc2)=O)N(C(c2coc3c2CSC3)=O)C1 N1(C(C2(CC=C)CN(C(c3csc(Cl)n3)=O)C2)=O)C2CCCC1CN(C)C2 C1(C(=O)OC)CC(F)(F)CC1C(=O)NCC(CO)NC(c1cc(C)c(C)o1)=O c1(CC(=O)NC2C(C)CN(C(c3nncn3C)=O)CC2)cccc2c1OCO2 C1(C)(CCC)CCCN(C(=O)CC2CC(C(=O)NC34CCC(CC3F)C4)C2)C1 Cc1ccc(C(=O)NC2CC(C)(NC(=O)CS(C)(=O)=O)C2)c(O)n1 c1(C(N2CC(C)C(CNC(=O)CCF)CC2)=O)cccc2c1CC(=O)N2C C1(C)(NC(C2CCCN(C)C2)=O)CCN(C(=O)COCCO)CC1 c1(CC(=O)NC(CC2CN(C(C3C(C)=CCS3)=O)C2)C)ccc(F)c(Cl)c1F CC(C(=O)N1CCCC1CNC(c1c[nH]nc1-c1ccccc1)=O)C(F)F C1(CC(=O)NCC(c2ccccc2F)NC(c2cnc(C)o2)=O)CCC(C)(C)O1 C1CCCC(C)NC(=O)C2C(COC)(C2)C1.c1(C(=O)NC)cc(C2CC2)ns1.OC Cc1[nH]c(=N)sc1C(N1CCC1CNC(=O)CCC1CCC(=O)N1)=O c1(C(N2C(C)(C)CC(NC(c3csc(Cl)n3)=O)C2)=O)cc(Cl)cc(F)c1N C(CCC(=O)N(c1ccoc1)C(C)C1CC1)(C(N)=O)NC(C(OCC)OCC)=O CC1(C(N2C3CC2CN(C(=O)Cc2cccc(C#N)c2)C3)=O)CCC2CC2C1 C1(C(=O)NCC2N(C(CN(CC)CC)=O)CC2)OCC2CCCC12 CN1CCN(C(=O)NCCc2ccc(Cl)cn2)c2ccc(F)cc21 C(C)(CCCCNC(c1cc(OC)n(C)n1)=O)NC(CC=CC)=O CC(CCC(=O)N1CCCC(NC(C2CS(=O)(=O)C2)=O)CC1)S(C)(=O)=O c1(CC(=O)NC(CN(C(C(C2CC2)OCC)=O)C)C)ccc(SCC)cc1 C(c1ccc2ccccc2c1)=CC(=O)NCC1(NC(C(CC)N(C)C)=O)CCC1 c1(C(=O)OC)cncc(C(=O)NC2CC3CN(C(=O)C(C)NC(C)=O)CC23)c1C N1(C(CNS(NC)(=O)=O)=O)CC2CC(NC(=O)C=Cc3cncn3C)C1C2 N1(C(=O)OC(C)(C)C)CC2CCCC(C(=O)NCC(F)(F)F)C2C1.c1cscc1Cl N1(C(=O)CC23CCCC2C3)CCC2CCC(C1)N2C(c1ccc(CO)c(Cl)c1)=O S(=O)(=O)(c1nc(N2CCC(C)(CO)C2)ccc1Br)N(C)CCc1cn(C)cn1 c1(C(=O)NC(C2N(C(c3cnc(C)[nH]3)=O)CCCC2)C)ccc2cncn2c1C c1(C(=O)NC23C(CN(C(C=COCC)=O)C2)CCC3)ccc(Cl)c2ncccc12 N1(C(c2ccc(C)n2C)=O)CCCCCC1C(=O)NC1CCCC(O)CC1 C(CN=C(NCC1CCC(C2CC2)O1)Nc1ccccc1F)C1CCC(C)(C)C1 C(=O)(CCS(=O)(=O)c1ccc(F)cc1)NCC(C)NC(C(CC)(C)O)=O c1(OC)cccc(C(=O)N(C2CN(Cc3ccc(C(N)=O)cc3)C2)C)c1O c1(NC(CC2(CNC(c3c(CC)[nH]cc3)=O)CC2)=O)cccc(Cl)c1O c1(CNC(C2C=C(C)CS2)=O)cncc(C(=O)NC2(C3CCCO3)CC2)c1 CC1=CCC(C(=O)NCc2nc(CNC(C3CC(=C(F)F)C3)=O)cs2)CC1 n1(CC)nc(C2CC2)cc1C(C(=O)NC1COC1)N1CCC1C1CCCC1 C(=O)(C(C(C)C)NC(C1(NC(c2ccnn2C2CC2)=O)CCC1)=O)OCC c1(C(=O)NCC2C(C(=O)NC(C(C(=O)OC)C)C)C2(C)C)cc(O)nc(C)n1 C12(OC)CCC(C(=O)NCC3(C(C)NC(=O)C(F)C(F)(F)F)CC3)(CC1)C2 N1(C(=O)NCc2ccn(CCC)c2)CCCC(c2ncccn2)C1 c1(-n2cc(C(CC)(C)O)nn2)cccc(C(=O)NCC(C)NC(=O)C2CC2)c1 c1(NC)cccc(C(=O)NCC(C2CCN(C(c3ccns3)=O)CC2)F)n1 CCCCCC(C)(CC)C(=O)NC1CCN(C(c2cccc(C)c2O)=O)C1 CC1(C(=O)NCC2CCN(C(=O)C(F)(F)C3CCOCC3)C2)CNC(=O)C1 N1(C(C2C(C(=O)OC)C2)=O)C(C(=O)NC2(CCO)CCCC2)CC1C c1(C(C)C(=O)NC2(CN(C(=O)CC3CC(C)(C)C3)C)CC2)ccccc1Cl C1(O)(CC(=O)NC2(C)CC2)CCN(C(c2cccc(OCOC)c2O)=O)CC1 C(=O)(C1Cc2c(Cl)cccc21)NCC=CCNC(c1c(N(C)C)cncc1)=O C1(C(N(C)CC2(CNC(C3OCC3(C)C)=O)CC2)=O)CCCNC1=O CC1=NN(C)C(=O)C1CC(=O)N(C1CCN(C(c2sccc2C(F)F)=O)C1)C S(=O)(=O)(c1cc(Cl)c(Br)cc1F)NC(=O)NC1CC(C)NC1 C#CC1(NC(C23CCC(CC2)N3C(c2cccc(F)c2C)=O)=O)CCCOC1 O=S(=O)(c1cccc(Nc2cc(O)nn2C2CCC2)c1)N1CCc2ccccc21 c1(NC(C2CC(F)CN2C(c2ccncc2Br)=O)=O)ccc(O)c(F)c1F C#CC1C(C(=O)NC2(CNC(=O)C3=NOCC3)CCCC2)C1(C)C c1(CC(=O)NC(CNC(C(CC(=C)C)C)=O)CO)ccc(Cl)c2cccnc12 c1(C(N2CC(C)C(CNC(=O)C3=COCCO3)C2)=O)ccc(N)c(N)n1 C1(NC(=O)CNC(=O)C2CC2)C2CC1N(C(=O)Cc1ccc(F)cc1)C2 c1(C(=O)NCCOCCN(C(C2C(CC)C2)=O)C)ccc2cc(F)ccc2n1 N1(C(c2cc(CC(C)C)sc2)=O)CCN(C(c2cnn(C)c2)=O)C(C)C1C C1(NC(c2coc3ccc(C)cc32)=O)CC(N=c2nc(C(C)(C)C)[nH]s2)C1 C1(C(=O)NC(CC)CN(C(C2CC2C(C)(C)C)=O)CC)COCCO1 Cn1sc(C(N2CCCC2CC(N2CCCC2)=O)=O)cc1=O c1(C(N2CCCC(NC(c3ccc(OC(C)C)nc3)=O)C2)=O)ccc(N)c(F)n1 C1(N(C(=O)C(c2cccc(Cl)c2)C2CC2)CC)CCCN(C(=O)C=CCO)C1 c1(OC)ccc(=NC2CCCC23CN(C(=O)CC2CCC(O)C2)C3)[nH]c1C(F)F c1(CC)cc(C(=O)NCC(C)N(C(=O)C(C)(C)C2(O)CCOC2)C)nn1C C1(CCC)(NC(=O)CNC(=O)CCNC(C)=O)CCN(C(c2cccs2)=O)CC1 C(=O)(CCCCCC(C)(C)C)N1CC(O)(CCNC(c2c(C)c[nH]c2)=O)C1 Cc1cc(NC(C23CSCC2C3)=O)ccc1NC(=O)CC(C)C1CCCO1 N1(C(COC(C)C)=O)CCN(C(=O)C(C)C)CC1CCO C1(C)(CC(=O)NC(C2CC=CCC2)C(=O)NCCN(C)C2CC2)CCCCC1 C1(NC(=O)CCC2CCCC2)CCCN(C(=O)CCc2nc(C3CC3)n[nH]2)CC1 C1(CNC(C(C2CCC2)OC)=O)CC12CCN(C(=O)Cc1cccc(F)c1)CC2 N1(C(c2cc(C(C)C)no2)=O)CCC(O)C(C(N2CC(O)C(F)C2)=O)C1 c1(C(N2C(CNC(C(CC)N(C)C)=O)C=CC2)=O)ccc2cc(OC)ccc2c1 C(C(C)C(F)C(=O)N1CCC(O)C1(C)C)NC(c1cc(CC)oc1C)=O C(=O)(C(C)P(C)(C)=O)NCCC(=C)CNC(c1nccnc1C)=O n1(CC(=O)NCC2CCC(NC(c3cc(Br)no3)=O)C2)cccnc1=O CCC(C)(O)C(=O)Nc1cc(-c2cccc(N3CCCC3)c2)cs1 Cc1cccc2cc(S(=O)(=O)OC3CCCC3N3CCOCC3)sc12 c1(C(=O)NCC2(OC)CN(C(c3c(OCC)scc3)=O)C2)ccc(C)c(C)c1O N1(C(c2c(C)sc(O)n2)=O)CCCC(C2(NC(=O)C(N3CCCC(C)C3)=O)CC2)C1 C=CC1(CC(=O)NC(C2(OC)CCC2)C)CN(C(=O)C(O)C(C)C)C1 C(c1cnn(C)c1)=CC(=O)NC1(c2cn(CCCC(=O)OC)nn2)CCC1 c1(CN=C(NCc2ccn(CC)c2)NC(CC)CC)cccc(F)c1C#N n1(CC#C)cnnc1C(=O)NCc1ccc(C(=O)NCC(F)Br)o1 CC1(C(=O)NCc2cccc(NC)c2)CC=CCC1.c1(C(=O)N)csc(Cl)n1 c1(C(=O)NC2CCN(C(CC3(CSC)CC3)=O)C2C)cc2c(C)ccc(F)c2o1 CCC(C)C(C(=O)NCC1(NC(=O)CCCCCOC)CCOC1)N(C)C C1(CC(=O)NC2(CC)CCCC2)CCN(C(C2C(C)C2C)=O)CC1 C1(C(N(C)CC2CCCC2O)=O)(NC(=O)CC2(O)CCOCC2)CCCCC1 c1(CC(N2C(C)(C(=O)NC3CC3O)CC2)=O)ccc(O)nc1 Cc1ccc(C2(C(=O)NC3CC(C)N(C(c4ccns4)=O)C3)CCOCC2)cc1 c1(C(C(=O)NCC(C)(C2CC2)NC(CC2CC(=C)C2)=O)(F)F)cc(Cl)ccc1F c1(C(N2CC(C)(NC(=O)CC3CCCC4CC34)C2)=O)c[nH]cc(Br)c1=N C12(CNC(C(CCN(C)C)NC(c3c(C)cco3)=O)=O)CCC(CO1)C2 C1(C(=O)NCCC2(O)CN(C(Cn3cnc(C#N)n3)=O)C2)CC2C=CC1C21CC1 C1(NC(c2ncc(C)cc2C)=O)CN(C(C2CCN(C)CC2)=O)CC2(CCC2)C1 N1(C(Cc2cc(C)nn2C)=O)CCOCC(NC(=O)COc2ccc(F)cc2)C1 c1(N(C)C)ccc(C(=O)NCC2CC2CNC(=O)Cc2nccn2C)nn1 N1(C(C2(CC(C)C)CC2)=O)C(C(=O)NCC2CC3(CC3)C2)CC2CCCC12 CC1=C(C(=O)NC2CCC(c3cccs3)C2)CCC1.C1(=O)C(=O)CN1C(C)C c1(NC(C=C2CCN(C(C(CCC)C)=O)CC2)=O)cc(C(F)(F)F)ccc1F O(C1CCCc2ccccc21)CC(N1C(CCNC(CSCCC)=O)CCC1)=O CCC(C)CCC(O)CC(=O)N1CC(NC(c2cccnn2)=O)CC2(CCC2)C1 Cn1c(C(N2CCCCC(CNC(c3cnns3)=O)C2)=O)cc(Cl)c1Cl C1(NC(COC2CC(NC(C3NC(=O)NC3=O)=O)C2)=O)CCCC(C2CC2)C1 c1(C(N)=O)ccccc1NC(C1C2CN(C(C3(O)CCSCC3)=O)CC12)=O CS(=O)(=O)C1(C(=O)NCC(=C2CN(C(c3ccsc3)=O)C2)F)CCC1 C(=O)(C1COc2ccc(Br)cc21)N1CCC(CCNC(CN(C)C)=O)C1 c1(C(=O)NC2(CCNC(C3CCC(F)(F)C3)=O)CC2)cc2ccncc2[nH]1 C1(C(=O)NC(C)CNC(=O)CN2CCCC(O)C2)CCC2(CCC2)C1 C1(NC(=O)CCc2cccs2)CCCC2(CN(C(=O)COc3ccccc3)C2)O1 Cc1cc(C(N2CC(F)CC2CC(N2CCC(OC3CCC3)C2)=O)=O)cnn1 CC1CCN(C(=O)CC(=O)N(C)C)C1CNC(C1NC(=O)OC1C)=O c1(CNc2nccc(SC)n2)c2c(cc3c1CCC3)CCC2 c1(C(=O)NCC2CN(C(Cn3ncc(C)c3)=O)C(C)CC2)c(N)cc(Cl)cc1F N1(C(C2CC(NCc3c[nH]c4ccncc34)C2)=O)CCCC2CCCCC12 N1(C(c2ccc(OC)nc2)=O)CC(NC(=O)C(C)C2CCOC2)C(C)(C)C1 N1(C(C(c2ccccc2F)C)=O)CC2(CCCCN2C(c2nn(C)cc2Cl)=O)C1 C(C)(c1ccco1)=CCN1CC(OCCNC(C2(OC)CCCC2)=O)C1 C1(CNC(C(C#C)(C)C)=O)(CO)CCCN(C(=O)Cc2cc(C)ccc2O)C1 C1(CSCCNC(C2(C)CC(C)(C)C2)=O)CC2(CCN(CC(F)(F)F)C2)CO1 C1(C(N2CC(C)N(C(c3ccoc3Br)=O)CC2)=O)CCc2nncn2CC1 c1(C(N2CC(O)(CN(C)C(c3cnnn3C)=O)C2)=O)ccc2cc(Cl)ccc2c1 C(CC(C(=O)NCO)NC(=O)OC(C)(C)C)=CCNC(C1CC1F)=O.C1(=CC)CCSCC1 C1(NC(C(CC=C)(C)C)=O)C2CCC1CN(C(c1cc(F)ccc1O)=O)C2 C1(CC(N2CCN(C(C)C)CC2)=O)C2CCC1CN(S(=O)(=O)c1nccs1)C2 N1(C(C(C=C)(C)CC)=O)CCC2CCN(C(c3c(SC)cnn3C)=O)C2C1 C(=O)(C#CC1CCCC1)NCC1(CNC(c2cc(C)c(C)[nH]2)=O)CCCCC1 N1(C(C(C)NC(N)=O)=O)CC(F)(CNC(C2CC(F)(CO)C2)=O)C1 C(=O)(C(F)CC(C)(C)C)N1C(C(=O)NCC(N(OC)C)=O)CC1C c1(-c2nc(C=Cc3c(C)nccc3)on2)ccc(F)c2cccnc12 C(=O)(CCCCCNC(C1(C#N)CC(C)C1)=O)NC1C(CC=C)COC1 c1(C(N(CC(C)NC(C2CC(O)(CC#C)C2)=O)C)=O)ccc(C(F)F)nc1 c1(CC(=O)NCC(C(C)C)NC(CC2(C=C)CC2)=O)ccc(F)cc1Cl CC1(CNC(c2scnc2-c2cccs2)=O)CCN(C(C2(n3nccn3)CC2)=O)C1 Cn1cc(CCNC(C2(CCNC3CC=CC3)CC2)=O)n(C)c1=O C1(C(=O)OC)CCC(C(=O)NC2CCCC(C(=O)NC(C)(CO)CO)C2)CC1 Cc1c(CNC(=O)CC2CC(NC(C3CC4CCC4C3)=O)C2)cnn1C C=C(CNC(C1CC12CCN(C(=O)C(C)(CC)CC)CC2)=O)c1ccccc1 N1(C(c2nc(OCC)oc2)=O)CCC2CCN(C(=O)C#CC3CCCC3)C2C1 O=C(CNC(=O)CCNC(=O)Cn1c(O)nnc1O)N1CC(O)CCO1 c1(C(=O)NC2C(C(=O)NCC(COC)(C)C)C2(C)C)ncc(F)cc1N CN1CC=CCC1CC(N1CC=CC1(C(=O)N(C1C=CCC1)CCO)CO)=O N1(C(CCC(C)O)=O)CC(NC(=O)CCS(C)(=O)=O)C(C)(C)C1 c1(C(=O)NC(CNC(C2NC(=O)CC(C)C2)=O)C)cnc2c(Br)cccn12 CCC(C(C)C)NC(=O)C(C1CCCO1)NC(=O)CNC(N)=O C1(CC)CCN(C(=O)OC)CN1C(=O)C(F)CC1CN(C(=O)CCCNC(C)=O)C1 Cc1cc(C(=O)NCCOCCN(C(=O)CC2CC3COCC23)C)ccc1Cl C(CCC(C(=O)NCC(C)CC(F)(F)F)NC(c1cncc(O)c1)=O)OC N1(C(C(C)(C)OC)=O)CC2CC2(C(=O)Nc2ncncc2Cl)C1 c1(NC(C2CCN(Cc3cc(Br)ncc3F)CC2O)=O)ccc2oc(O)nc2c1 N1(C(COC)=O)CC(NC(c2n[nH]c3c2COC3)=O)CC2(CC2)C1 C(=O)(CCCC(F)F)NCc1ccc(CNC(c2ccc(C#C)o2)=O)cc1 c1(CC(=O)NC(C2CCN(C(COCCC#C)=O)C2)C)noc(C)c1C#N C1(CCNC(c2cc(Cl)no2)=O)CCCN(C(C2(Cl)CCCCC2)=O)C1 N1(C(c2ccc(C)nc2)=O)CCC(C2CC2NC(=O)CN(C)C(N)=O)CC1 N1(C(C2(C)CC(=C)C2)=O)CCOCC(C(=O)N(c2ccc(C)cc2C)C2CC2)C1 n1(CC(=O)NC(CC2CCCO2)CN)ccc(C(F)F)n1 C(=O)(CCC(F)(F)F)NCCCN(C(c1cc(C)cc(C)n1)=O)CC N#Cc1cc(C(=O)NCC2CCC2NC(=O)C=CCn2cncn2)ccc1Cl C(=O)(C(F)(F)C(F)(F)F)N1CC(NC(c2cccc(OC)c2C)=O)C(C)C1 Cc1cc(C(N2C(C)C3CC2C3NC(c2cc(C3(C)CC3)n[nH]2)=O)=O)ccc1Cl C1(NC(CNC(=O)NC)=O)CCN(C(c2c(C)noc2C)=O)CC1C(=O)NC CC1CCCN1CC(=O)NCC(C)=CC(N1CCCC1CCO)=O C(CCCCNCC1CCC(C)S1)(OC)OC C1(NC(=O)Cc2csc(-c3ccoc3)n2)CCCN(C(=O)C#CC2CCC2)CC1 CON(C(=O)C1C2CN(C(C3CCC=CCCC3)=O)CC12)C1CCCC1 C12(CNC(COCCCCC)=O)CCC(C1)N(C(c1cc(C)nn1CCC)=O)C2 CCC(CC)(CC)C(=O)NCC(C)(C)OCC(=O)NC(c1cncs1)C C1(NC(C(=Cc2ccc(Br)o2)C)=O)C2CCC1N(C(c1ccnn1C)=O)C2 c1(C(=O)NC(CCCC)CNC(c2cnc(C(C)C)[nH]2)=O)n[nH]c2cccnc12 c1(CC)cc(N2CC3CC(NC(c4cccc(F)c4Cl)=O)C3C2)nc(CC)n1 C1(NC(C(C)OC)=O)CC2(CCN(C(c3cc(C#N)c[nH]3)=O)C2)C1 N1(CC(c2cccnc2)=O)CCCCC2(CCCCN2)C1 C(C(N)=O)(C(C)O)NC(COC1CN(C(c2nc(C(C)C)oc2)=O)C1)=O c1(N)ccc(O)cc1C.Cc1cnc(CC2(CO)CN(C(=O)OC(C)(C)C)C2)nc1 c1(C(N2CCC(NC(CC(C)OC)=O)C2C(C)(C)C)=O)cncc(C=C)c1 CC(C)C(CNC(c1cc(F)ccc1F)=O)C(=O)N(CC(F)(F)CO)C C1(C(=O)NCc2cc(C(N(CC(CN(C)C)O)C)=O)n[nH]2)CCCC2(CC2)C1 Cc1c(C(=O)NC2(CO)CCCN(C(=O)CC(C)O)C2)sc2ccccc12 C1(C(=O)NC(CSCC)C(=O)NC(CC2CC2)CC2CC2)CCOCC1(C)C CC1(C)CCOC1CC(=O)NC1CCC(NC(c2cnc(C3CC3)s2)=O)CC1 c1(C(=O)NC2C(CNC(C(CN(C)C)O)=O)CC2)cccnc1N c1(OC)ccc(F)cc1C(N1CCC(O)C(C(=O)Nc2cc(O)ccc2C)C1)=O N1(C(C2(CC#C)CCOCC2)=O)CCCC2(NC(c3occc3Br)=O)CC2C1 C12(NC(=O)CCCc3cccnc3)CCCC1N(C(=O)Cc1cscn1)CC2 c1(C(=O)NCC2(NC(c3c(OC)csc3)=O)CCOC2)nccn2nc(C)cc12 c1(N(CCCCO)C)ccc(N2CCC(Oc3ccccc3F)CC2)nn1 C(CCCC(=O)N1CCCC1CC(=O)NCCS(C)(=N)=O)(OC)OC O=C(C(F)C1=CCCCC1)N1CC2(CCCN(C(=O)CCC(F)(F)F)C2)C1 CC#CCC(C(=O)NCCC1(OC)CCCCC1)NC(=O)CSCC(F)F C1(CC(=O)N(C)CCOCCN(C)C(C2CC2F)=O)CC12CC2 C1(CC(N2CC(C)(NC(c3ccc(COC)o3)=O)C2)=O)CCC2(CC1)OCCO2 C#Cc1ccc(C(=O)N(C(C)(C)CC(=O)NC(C)C)C)o1 n1(CC)nc(C(=O)NC2C3CCC2N(C(c2ccnc(O)c2)=O)C3)ccc1=O c1(CN(c2nccc(C(=O)O)n2)CC(c2ccccc2)=O)c[nH]c2cc(F)ccc12 C(=O)(NNc1cccc2c(Br)cccc12)NCCCCN(C)C1CC1 C1(NC(C)=O)CN(C(=O)COc2cccc(CC3CC=CCC3C)c2)CC1O Cn1ncc2ccc(C(N3CC4(CC(NC(=O)C(O)P(C)(C)=O)CO4)C3)=O)cc12 CCCCC(CC)C(=O)N1CCN(C(=O)CC2(OC)CC2)C(CO)C1 c1(N(CC(c2ccccc2)C)C(N2C(C)CCC2)=O)ccccc1N N1(C(C(=O)OCC)=O)CC(C)(NC(C2=NC=NCCN2)=O)C1 N1(C(CCC#C)=O)CC2CC(NC(c3cnc(-c4ccccc4)[nH]3)=O)C1C2 C1(CNC(c2ccco2)=O)C2CN(C(=O)CCCSCN(C(C=NOC)=O)C)CC12 CC1CCCCC1(CNC(c1coc(C(F)F)c1)=O)NC(C1CCCC1(C)C)=O C(CN=c1cc[nH]cc1S(=O)(=O)N(C)Cc1ccccn1)N1CCC(C)CC1 C(CN=C(NCC(=O)NCC1CN(C)CCO1)NC(C)C)OCC C1(NC(=O)CCN2CCCS2(=O)=O)CN(C(C2CC2F)=O)CC12CC2 c1(C(=O)NCCOCCC(N2CC(O)(CN(C)C)C2)=O)cnn2ccccc12 Cc1cccc(C)c1CC(N1CCCC(CNC(c2ccns2)=O)C1)=O C1(NC(=O)CC23CCCC2C3)CC2CC1CN(C(c1cc3n(n1)CCCC3)=O)C2 C(=O)(CCCCC(N)=O)NCCC1(C)CCN(C(c2nc(Cl)cs2)=O)C1 C(=O)(C(CC(F)F)NC(C1CC(C2CC2)=NO1)=O)NCC(C)N(C)C c1(OC)ccc(F)cc1N(C)C(c1cc(CNc2cnn(C)c2N)ccn1)=O c1(OC)nc(C(N2CC(NC(c3cccc(N)c3)=O)C(CC3CC3)C2)=O)sc1C Cc1ccc2c(c1)C(C(=O)N1CCCN(C(c3cnc(CC4CC4)s3)=O)CC1)C2 C12(C(=O)NCc3cccc(CO)c3)CC1CN(C(=O)C(C)=C)C2.C(C=O)OC N1(C(CCCCNC(CC(C)=O)=O)=O)CCC(F)(F)C(CO)C1 c1(N(C2CCCN(C(C3(CCO)COC3)=O)C2)CCO)ccc2nnnn2n1 c1(C(=O)NCCOCCNC(C2C(OCC)C2)=O)cc(O)nc(O)n1 S(=O)(=O)(c1cc(C(C)C)cc(F)c1F)NCC(=O)N(c1ccc(Cl)cc1)CC C1(C)(NC(c2cn(CC3N(C(C)=O)CCC3)nn2)C2CCOCC2)COC(=O)N1 C1(CNC(c2ccc(C)o2)=O)CC2CCC(C1)N2C(=O)CNc1ccccn1 CC1=C(C(=O)NCC=CCNC(=O)C(O)Cc2ccccn2)CCC1 c1(COC)ccc(C(=O)N(C2CN(C(=O)CN3CC4CC4C3)C2)C)s1 c1(CNC(CC2C(=O)NC(=N)S2)=O)cc(O)nc(CNC(=O)CC2CC=CC2)n1 C(=O)(CC1CCOc2ccccc21)N(C1CN(C(c2c(C)c(O)ccc2)=O)C1)C N1(C(c2cc(C)sc2)=O)CCN(C(c2cc(F)c[nH]2)=O)CC1C1CCCC1 c1(C(COCCOCCN(C(CN)CO)C)N(C)C(=O)OC)ccccc1.OC C(=O)(CC(C(C)(C)C)NC(c1ccc(CO)o1)=O)NC(C)CSC(F)F C1(C(N2CCC(OCCNC(CNC(N)=O)=O)C2)=O)COc2cc(F)ccc2C1 C=CC1(C(=O)N(C)CCOCCCN(C(=O)CC2(CC)CCC2)C)CCCCC1 C(=O)(CCCC(=O)N1CCCC(C)(CNC(c2nc(Cl)cs2)=O)C1)OCC c1(C(N2CC(NC(C=CCC)=O)C(C)CC2)=O)cc(C)c2ccccc2n1 C(=O)(C(CNC(C1CCCNC1=O)=O)CC1CC1)NC1C=CC(C(=O)OC)C1 CC(C)(C)CCCCC(=O)NC(=O)COCc1nc[nH]n1.N12CCC(C1)CC2=O C1(NC(C(C)OCC)=O)CCN(C(c2cccc3cc[nH]c23)=O)CC12CCC2 c1(NCC)cnncc1C(=O)NC1(NC(c2cc(C(F)(F)F)n[nH]2)=O)CC1 C1(NC(c2c(CCC)cccc2)=O)CCCC(NC(C2CC3(CCC3)C2)=O)CC1 CC1(C(N2CCCCC(NC(c3ccc(Cl)cc3)=O)C2)=O)CCCNS1(=O)=O N1(C(C2CN(C(=O)NC)C2)=O)CCN(C(c2cnncc2C)=O)C(C)CC1C N1(C(CCC(C)OC)=O)CCCC(O)(Cn2cc(CC(C)(C)C)nn2)CC1 c1(C(=O)NC2C(CNC(C(CC)NC(C)=O)=O)CCC2)ccn2c(O)nnc2c1 C1(C(N2CCC(CC(C)C)CC2)=O)CCCCCCN1C(C1COCC1C(N)=O)=O CCCCCCCCCC(CC)C(=O)NCC(C)(C)NC(C1CCOC1)=O c1(NC(COCC(C(=O)N(C)C)NC(C)=O)=O)c(C)nc2ncnn2c1C CC1C(NC(C2CCCC3CC23)=O)C(C)CCN1C(C1CC(C)(F)C1)=O C1(C(N2CCC(O)(C(C)NC(COCCCC#C)=O)C2)=O)CCCC(=O)N1C N1(C(CCc2n(C)cnc2)=O)CC2CC1CCC2NC(=O)Cc1csc(Cl)c1 C#CC1CCC(N(c2cc(-c3cnc(COCC4CC4)cn3)on2)CC2CC2)C1 O=C(C(C1=NOC2(CCC2)C1)N1CCOC2CC12)NCC1CC1 C(CCCCCF)c1cn(CCCCCC)nn1.C(=O)(C(C(C)C)O)N1CCC1CO C1(C)(COC)CC(NC(c2cc(N)ccn2)=O)CN1C(=O)CN1CCCC1=O CCCCCC(O)C(=O)NC1CCC1CNC(c1ccc2ncnn2c1)=O N1(c2cc(NCCC3CC3)nc(COC)n2)CCCC2(CCC(=O)NC2)C1 Cc1ccccc1-c1noc(C(c2ccc(Cl)cc2)C2CC2)n1 CCCCCCCC(=O)N1CC(C)(C)CC1CNC(C1CCCC(C)(C)C1)=O N1(C(CCCCOC)=O)CCC(C(N2CCCC(F)(F)CC2)=O)CC1(C)C Cc1cc(C(=O)NC(CCNC(=O)CCc2ncccn2)C(C)C)ccc1C#N c1(C(N2CC3C(CNC(CCC)=O)(CC3)C2)=O)cc2cccc(OC)c2[nH]1 C(=O)(C(O)CCCNC(=O)C(C)(F)c1ccon1)NCCC1CCCN(C)C1 c1(CNC(=O)C(C(CCNC(=O)NC23CC(OC)C2C3)C)=O)cc(C)cc(C)c1 Cc1ccc(C(N2CCN(C(=O)C3CC3)CC(O)C2)=O)c(F)c1F N1(CC(=O)NCC2CCN(C(C3N(C)CCC3)=O)C23CC3)C(=O)NC(C)(C)C1=O N1(C(CNC(CCC)=O)=O)CCN(C)C(C(=O)NC(COC)C(=O)OC)C1 CCC(CC)C(=O)N1CC(O)(C(C)NC(=O)CN(S(=O)(=O)CC)C)C1 c1(NCC2CC(C(C)C)C2)nccc(=NCC(C)CN(C)C)[nH]1 CC1=C(C)CC(C(N2CC(CNC(C3COCCN3C=O)=O)C2)=O)CC1 N1(C(CCCCOCC)=O)CC(C)OC2(CCN(C(=O)C=CC(=O)NC3CC3)C2)C1 CC1(C)C2CCC1(NC(=O)Nc1ccccc1OC1CCOC1)C2 n1(CC)ccc(C(=O)N(C2CCN(C(c3cnc(O)c(C)c3)=O)CC2)C)cc1=O c1(OC)ccccc1C(N1CCCC1C(=O)N(C(C)CO)C)=O C1(NC(c2n(CCC)nc(C)c2)=O)CCCN(C(=O)COCP(C)(C)=O)C1C n1(CC(C)C)cc(NC(=O)CCSCCCNC(=O)OC(C)(C)C)c(C)n1 N1(C(Cn2ncc(CC)c2)=O)CCCC1(C(=O)NC1(C(COC)O)CC1)C(C)C c1(C(N(CCNC(c2nnc(S)n2C)=O)CC)=O)c(O)ccc(F)c1Br Cc1cc(C(=O)NCC2(O)CN(C(=O)CC3CCCOCC3)C2)c(F)cc1F C1(NC(CCc2cnc(C)s2)=O)CCCN(C(=O)CCc2cccnc2Cl)C1C N12CCCC1CN(C)C(=O)C1(CC1)C2=O.C1(C(CO)NC(N)=O)CCCC1 CC1(C)CCCOC1C(=O)NC1C2CCC(C2)C1C(=O)N(C1CCC2CC1CO2)CC N(C(=NCCN1C(=O)COc2ccccc21)NCCc1ccccc1)C1C(C)C1 c1(CSCC(N2CC(C)N(C(=O)OC(C)(C)C)CC2)=O)ccc2ccccc2c1 Cc1ccc(NC(=O)NC2CCCC(C(C)(C)C)CC2)c(F)c1 N1(C(COCC#C)=O)CCC(C(C)(C)C)(CNC(c2occc2COC)=O)C1 C=C(C)CC(C(=O)N1CC(O)CC1CC(N1CCC(C(=O)NC)C1)=O)OC C(=O)(C(F)CC(C)(C)NC(c1cc(C)n(C)c1)=O)NC(CC=C)(C)CC=C C1(NC(CC2(C)CC2(F)F)=O)CC2CCC(C1)N2C(=O)C(O)C1CCC1 c1(C(N2C(CCNC(C(CCCOC)C)=O)CSCC2)=O)ccc2ccnn2c1 N1(C(c2c(CC)cccn2)=O)CC(NC(=O)Cn2cc(F)ccc2=O)CCC1C CP(C)(=O)CN1CC(C(=O)NC2CCCCN(C(C3C4CC5C(C4=O)C35)=O)C2)C1 C1(F)(CNC(c2c(OC)c(F)ccc2)=O)COCCN(C(C2C3COCC23)=O)C1 N1(C(C(C)C(F)F)=O)CC(NC(=O)COc2ccccc2Cl)CC12CCOCC2 CCCCC(C(=O)NC1CCN(C(c2nc(Cl)sc2Cl)=O)C1)NC(N)=O c1(C(N2CCCC(N(C(CCC(=O)OCC)=O)C)CC2)=O)cc2c(nn1)CCC2 C1(C(=O)NCc2cc(C)no2)CC(O)CN1C(=O)CCN1CCCCC1 C(CC(C(=O)N1CCC(O)(CN(C)C)C1)NC(=O)C1=CCC1)=CC C12CN(CCO1)C(=O)C2.C1(C(=O)NC(C)Cn2cnnc2)CN2CCC1C2 c1(C(=O)NCCCC(C)NC(=O)CCC2CC2C)c[nH]c2c(C#N)cccc12 CCC(C)(C)C(C(=O)NC(c1ncc(C)[nH]1)CC)OC CN(C(=NCCCCC(F)(F)F)NCCN(C)CCO)CCn1cc[nH]c(=O)c1=O c1(C(=O)OC)cc(NC(=O)NC2CCCC(C(C)C)CC2)ccc1OC c1(C(N2CCCC(CN(C(C(CC3CC3)OC)=O)C)C2)=O)cccc(N)c1C N1(C(c2cnc(COC)nc2O)=O)C2CCC1CN(C(C1CCCS1)=O)C2 CC(C(C)(C)NC(C1CSCCS1)=O)NC(=O)CSCCN(C)C CC1CCC(=CC(=O)NCC2CC2CNC(C2CCCN2C)=O)C1 C(c1ccc(C)c(Cl)c1)=CC(=O)NC(CCCNC(c1cc(CC)nn1C)=O)C C1(NC(C(C2CCOCC2)OCC)=O)CCOCC1NC(=O)Cc1cnn(C)c1 C(C(=O)NCCC1CC(NC(=O)COC(F)F)C1)(C(C)C)SC c1(C(=O)NCCN(C(CC(=C)C)=O)CCCN(C)C)ncnc(O)c1Cl C(=O)(CC(C)C(=O)NCC1(CNC(c2cc(C(N)=O)n(C)n2)=O)CC1)OC C1(Cl)(C(=O)NC(CC2CCCC2)C(=O)NCC2(Cl)CCC2)CC1(F)F Cc1nsc(C(=O)NC2(CO)CN(C(c3cscn3)=O)C2)c1N c1(NC(C)=O)cccc(F)c1C(N1CCC1CNC(C1CCCCC1O)=O)=O C1(C(F)(F)F)(C(=O)NC2CC(c3c(OC)cccc3)C2)CNCCO1 C1(C(N(C2CN(C(c3cscn3)=O)CC2O)C)=O)CC2(CCC2)CCO1 c1(C(C)C)ccc(F)c(C(=O)NCCCCC(C)NC(C2CC(C(N)=O)C2)=O)c1 Cc1cncc(C(=O)NCCC(C)CCNC(C2CC3CC3C2)=O)c1C N1(C(CC(C(F)F)NC(C(CC)O)=O)=O)CCC2(CC1)CN(C)C2 C1(NC(CCC(C)OC)=O)CCC2CCN(C(=O)C(C)N(C)C)C1C2 Cc1nnsc1C(=O)NC1CC1NC(=O)CSCCc1ccccc1 Cc1cc(-c2ccccc2)nc(=NCCCNC(C2CCN(C)C(=O)C2)=O)[nH]1 c1(C(=O)NCCC2N(C(c3n(CC)cc(Cl)c3)=O)CCC2)noc2c1CCCC2 CCC(C)C(C(=O)N1CC(O)(C(C)NC(c2cc(CSC)on2)=O)C1)NC(N)=O N1(C(CC(=C)C)=O)CC2(CC(NC(=O)C(C)(C)C3(C)CC3(F)F)CO2)C1 Cc1coc2ccc(C(N3CCN(C(c4ns[nH]c4=O)=O)C4CC34)=O)cc12 c1(C(=O)NCC2CN(C(C3N(C(=O)OCC)CSC3)=O)C2)cnnc(C2CC2)c1 C(=O)(C1CCC(NC(c2cc3cc(Cl)ccc3s2)=O)c2ccccc21)OC Cc1cccc(CC(N2CC3(NC(C4CC4(C)C(F)F)=O)CCC2C3)=O)c1Cl C(CCO)(C(F)F)N(C)C(C1CC(F)CN1C(c1cnc[nH]c1=N)=O)=O C(=O)(C(C(=O)N1CCC(F)(C(=O)NCC2(C)CC3(CC3)C2)C1)OC)OCC c1(NC(C=Cc2c(C)nccc2)=O)c(F)cc([N+](=O)[O-])cc1F c1(C(N2CCN(C(C3CC3(F)F)=O)C(C3CCCC3)C2)=O)ccc2nsnc2c1 C12(CNC(COCCOC)=O)CC(CO1)N(C(C1CC1OC)=O)C2 N1(C(C(CCC)C)=O)CCCC(C)C1CNC(=O)CCNC(=O)OC C(C(CN=c1[nH]c2c(c(=NCC3CCCNC3=O)[nH]1)CCC2)OC)OC c1(CC(=O)C(=O)O)cn(C(F)F)c2ccccc12.N1(C(C(C)CO)=O)CCCC12CCC2 C1(C(=O)NCCN(C(C2CCC(CC)O2)=O)C2CC2)CCC(C)=C(C)C1 c1(C(N2CCN(C(c3nc(C(C)C)on3)(C)C)CC2)=O)ccc2c(c1)COCCC2 Cc1cnc(C(=O)NCC(C2CCCN2C(=O)C(C#N)C2CC2)(C)C)cc1C N1(C(c2cnn3ccsc23)=O)CCC2CN(C(=O)C(F)(F)C3CC3)CCC2C1 c1(CCNC(=NCCCOC(C)C)NCC(F)(F)Cl)nn(C)cc1S(N)(=O)=O Cc1nsc(N(CC(C)CNC(=O)CCC2CCC(=O)N2)C)c1C#N C(=O)(CC(C(F)F)n1cccn1)NC1CCN(C(C(F)=CCC)=O)C1C C(C(F)(C(=O)NC1CCOC1=O)C(C)C)NC(Cc1cn(CC)nc1)=O C1(NC(COCC(C)(C)C)=O)CN(C(c2cccc(C(F)F)c2Cl)=O)CC12CC2 C#CCCCC(=O)N(C(C)CN(C)C(c1cc(C)n(-c2ccccc2Cl)n1)=O)C CON1CCC(C(=O)N(CC(=O)NC2CC2C(F)(F)F)C)CC1 C1(CC)CN(C(=O)CCCNC(=O)CCCn2ccnn2)CCN1C(C)=O c1(C(=O)NCC(CCOC)NC(=O)CCS(N)(=O)=O)cn(C)c(=O)nc1O C(C(O)C(C)(C)C)c1cn(C(CNC(C(C2CCCCC2)C)=O)C)nn1 N1(C(CC2C(C)=NOC2=O)=O)C2CCCC1CC(NC(=O)CN1CCC(C)C1)C2 N1(C(CC(C)C2CC2)=O)CCC2CC12C(N1CCC(C(N)=O)CC1)=O N1(C(CC(C(C)C)(F)F)=O)CC(NC(C2(C(C)C)CCC2)=O)Cc2ccccc21 N1(C(C)=O)CSCC1C(=O)N(C)C(c1ccncc1)C c1(C(=O)NCC(=O)NCC(N2CCN(CC=C)CC2)=O)cc(=N)[nH]c(Cl)n1 C12(C(=O)NCCOCCC(=O)NC3CC(C4CC4)C3)CCCC1CCC2 C#Cc1cc(F)cnc1NC(C1CC12CCN(C(c1ccc(O)c(F)c1)=O)C2)=O c1(C(=O)NC2(CCNC(C(C(C)(C)C)N(C)C)=O)CC2)cncc2nc[nH]c12 C1(N(C(COCCC=C)=O)C)CCC2CN(C(=O)CC3CCCCN3C)CC12 C1(OCCCN(C)C)CN(C(C2(C)CCCOC2)=O)CC1CNC(=O)COCC c1(C(N2CCC(NC(c3ncnc(O)c3Cl)=O)(CO)C2)=O)cnc2ncccn12 CC(C)C(C)(O)C(=O)N1CC2CCC2(NC(C23CC(CN2C2CC2)C3)=O)C1 C(=O)(CC(C)N=c1[nH]c2c(c(=NC(C)CCSC)[nH]1)SCC2)N(CC)CC Cc1ccc(C(=O)N(CCC(C)(C)NC(=O)CC2CC3CC3C2)C)s1 CCCCCCCCCCCC(=O)N1CCCN(C(=O)NC2CC2(F)F)C(C)C1 C1(NC(CC(C)NC(N)=O)=O)CN(C(=O)CCCCc2cnn[nH]2)CC1(C)C Cc1cc(C)c(C(=O)NC2(CCNC(=O)COCc3ccnn3C)CC2)s1 N1(C(C=C(COC)C)=O)CC(C)CN(C(=O)C(C)(C)OC(C)=O)CC1C.C(C)(C)(C)O C(=O)(C(C)(C)COCC(F)F)NCC(CCOC)OC.c1(N)cscc1C c1(C(=O)NCC=CCC(=O)N(C(CC)CC)CC)cnc(C)c(C)c1 CN1CCCCC1C(=O)N(C1CCCN(C(=O)CN2CCNC2=O)C1)C c1(NS(=O)(=O)c2c(F)cc(F)cc2Br)cn(C2CCCc3ccc(Cl)cc32)nn1 N1(C(C2CCC(NC(C(C)OCC(F)(F)F)=O)CC2)=O)CC2CC(F)CC2C1 N1(C(c2c(C(=O)OC)noc2)C(=O)NC2CCC2)CCCC(CCC(C)C)C1 C1(CNC(c2cc(Cl)sc2Cl)=O)CC2(CCC2)CN1C(=O)C1=CCSC1 N1(C(c2ccc(C)nc2)=O)CC2CC1CN2C(=O)CN1CC=CC1 c1(OC)ccc(C(=O)NC2CCN(C(C3(C4CC4)CC3)=O)CC2C)cc1Cl Cc1nn(-c2ccccc2)c(C)c1C1CCC1.C12CN(C)CCN1C(=O)NC2 CC1CCN(C(c2cccc(CF)c2)=O)C1CNC(=O)CCCCNC(N)=O C#CCC(C)C(=O)N1CC(CCNC(=O)C2=COCC2)C(C)C1 C1(c2cn(CC3CN(C(c4conc4C(C)C)=O)C3)nn2)(OCC)CCCCC1 C1(C(N2CC(n3cc(CNC(c4ccn(C)n4)=O)nn3)C2)=O)CCOC2(CCC2)C1 C1(C(N(C(C)CCNC(c2c[nH]c(Br)c2)=O)C)=O)CCc2nccn2C1 C1(NC(C(n2cc(Cl)cn2)C)=O)CC2C1CCN2C(C1CC(Cl)(Cl)C1)=O N1(C(C2OCC(=O)C2)=O)CCC2CC(CNc3cc4nncn4cn3)CCC2C1 CC1(C)CCN(C(=O)C2=CC3C=CC2C3)CC1NC(C1CCCC2(CC2)C1)=O CCC(F)(C(=O)OC)C(=O)N1CCC(CCNC(=O)CCCSC)C(F)(F)C1 C1(C(=O)OCC)CCSCN1C(C1CC1c1cnc(C)s1)=O N1(C(C2C(C(=O)OC)C2)=O)CCC2(NC(C3CC4(C3)CC(F)(F)C4)=O)CCCC12 c1(C(N2CC(C)(NC(CCC3CC(OC)C3)=O)C2)=O)cc2ccccc2cc1N C1(O)(C(C)CNC(C2CCNC(=O)C2)=O)CCN(C(=O)CCc2ccn(C)c2)C1 CC1OC2(CO)CC1(C(=O)NCC1(C)CN(C(c3ccncc3Cl)=O)CCO1)C2 N1(C(CC2CN(C(C)=O)C2)=O)CCCC(NC(c2cc(C)cc(C)c2)=O)C1C CC1CCC(NC(=O)CN2CC3C(NCc4cccnc4O)C3C2)CC1 n1(CC(N2CCC(CN(C(c3c(C)ncn3O)=O)C)C2)=O)nc(C)c(Br)c1C C1(C(=O)NC2C(C(N(c3cncc(C)c3)C(C)C)=O)COC2)CCC(C2CC2)C1 c1(C(N2C(CO)CC(NC(C)=O)C2)C)cc(C)c(Cl)nc1Cl C1(CC(=O)NC(C(=O)OC)CSC)CC2(CC2)CN1C(=O)CCOC1CC1.CN c1(C(=O)NC2CCC(C)N(C(=O)Cc3ccno3)C2)cc(C#N)c(O)nc1N C(C(=O)N=c1cc[nH]cc1F)C1CN(C(c2ccc(NC(C)=O)cc2Cl)=O)C1 c1(C(N(CC(O)CNC(c2cc(CO)on2)=O)C)=O)cccc2sncc12 N1(C(C(C)OCC#C)=O)CCC(C)(C)C(NC(=O)Cc2ccc(F)cc2C)C1 C1(C(N2CCC(NC(CCSCCC)=O)CC2C)=O)CCCC12CCOCC2 CCCC(C)CCCC(=O)N(C1CCCN(C(=O)C2=NOC(C)(C)C2)CC1)CC c1(C2C(c3cn(CC(=O)N(CCCC)C)nn3)C2)c[nH]c(Br)c1 C1(CN(C(C2C(CNC(c3cn(CC)nn3)=O)CCC2)=O)C)OCCC1(C)C c1(C(=O)NC2C(Cn3cc(CCCOC)nn3)CCC2)cccnc1S n1(CC)cc(C(=O)NCC(CO)NC(=O)COC2CCCCCC2)c(C(C)C)n1 Cc1nc(C(=O)NCC2CCCCN2C(c2ccc(C(C)F)cc2)=O)ccc1Br N1(C(C)=O)CCC(C)(NC(C2CCN(C(c3cc(C)c(Br)o3)=O)CC2)=O)C1 c1(C(N2C(CNC(COC)=O)(COC)CCC2)=O)ccc2c(c1)NC(=O)CN2C C1(C(=O)NC2(CF)CCN(C(c3nccc(N)c3)=O)C2)CCc2ccnn2C1 C1(C(C(N2CC(CNC(c3cncs3)=O)C2)=O)O)CCCCCC1 N1(C(CC(=C)Br)=O)CCOC(CCCNC(C2C3CC4C(C3)C24)=O)C1 N1(C(c2c(CC)non2)=O)CCN2CCN(C(=O)C(C(C)C)NC=O)CC2C1 C(CC(C(C)(C)C)NC(=O)C1=CCCS1)N(C(C1C(C)OCCC1)=O)C CN1CCCC2(C1)CN(C(=O)CC1CC1)CCN2C(C1CCCOC1)=O C1(C(=O)NC(CNC(COCc2cc(C)on2)=O)(C)CO)CCCC(C)C1 C1(C(N2CC(NC(C3CC4CCC3CC4)=O)C(F)C2)=O)CCC2(CCC2)O1 CC1(NC(C2COCCO2)=O)CCN(C(c2ccc(Cl)s2)=O)C1 N1(C(C=COCC)=O)CCC(CC)(NC(c2nn(C)c(C)c2Br)=O)CC1 c1(C(=O)NC2CC(NC(c3c(OC)nc(C)cc3)=O)C2)cc(C)ccc1[N+](=O)[O-] CCC(F)(F)CC(=O)NC(CC1CCC1)C(=O)NCC1CC1Cl N1(C(c2cnn(CC)c2Cl)=O)CCN(C(c2ncnn2C)=O)CC1C C1(Cc2c(C(C)=O)cccc2)OCCC(N)C1O.n12cc(nn1)CNC2=O C(=O)(C(CC)CC(F)(F)F)N(CCC)CCNC(=O)COCC1CCCOC1 c1(C(N2CCC(NC(c3c(N(C)C)nccc3)=O)C2)=O)c(F)ccc2ccoc12 C1(C(=O)NC(C)COC(F)F)CCCN1C(c1ccc(CO)s1)=O c1(CCNC(=O)NCC2CCC=CCC2)ccnc(O)c1F C1(NC(CS(=O)(=O)NCC)=O)CC2CCC1(NC(=O)CNS(=O)(=O)CCC)C2 C1(O)(C(C)CNC(C2(CN(C)C)CCOC2)=O)CCN(C(=O)OC(C)(C)C)C1 c1(NC(C(=O)N(CCCC)C2CC2)=O)cc(OC(C)C)cc(OC)c1 C1(C(=O)NC(C(C)NC(COCCSC)=O)CO)COCC(C)O1 C1(NC(CNC(=O)OC)=O)CCC2(CC1)CC2C(=O)Oc1ncc(C)c(SC)n1 N1(C(CN(C(C)=O)CC)=O)CCOC2CN(C(c3ccc(F)c(C)c3N)=O)CC12 CCC(C(=O)N(C1C2CN(C(c3c(F)ccc(N)c3F)=O)CC12)C)C(C)(F)F n1(C(C)C)ccnc1C(F)(F)C(=O)NCCN(C(C1CC1C)=O)CC1CC1 C(=O)(CC(O)CNC(=O)Cc1cc[nH]c1)NC(C(=O)OC)(C)C1CC1 N1(C(CN(C2CC2)CC)=O)CC(C)(C)OCC1CNC(=O)C(c1cccnc1)C c1(OC)c(C(=O)NC2CN(C(C3CCC34CCC4)=O)CC2C)csc1C CC(C)CC(O)C(=O)NC12CC(CNC(c3coc(C(F)(F)F)c3)=O)(C1)C2 C1(NC(c2cc(OCC)n[nH]2)=O)CCN(C(C2CN(C)CC(C)O2)=O)CC1C c1(C(N(C2CN(C(=O)CCC3CC3)CC2F)C)=O)ccc(S(N)(=O)=O)cc1 C(=O)(N=c1nc(CNS(C)(=O)=O)[nH][nH]1)c1cccc(-c2cc(=NC)[nH]cc2)c1 C1(N(C(C)C(=O)NC2CC2)S(C)(=O)=O)CCN(C(=O)CC(F)(F)F)CC1 C1(COC)(NC(=O)C(CO)NC(N)=O)CN(C(c2nc(Cl)cs2)=O)C1 C(=O)(C(C)(C)CS(N)(=O)=O)NC(C1CCCN(C(=O)CCS(C)(=O)=O)C1)C c1(OC)cc(C(=O)NC2CC(CNC(c3cc(C(F)F)cs3)=O)C2)ncn1 CCCC(CC)CC(=O)NCCNC(c1sc(CC2CC2)nc1C)=O C1(CCC(=O)N(CC(=O)N(CCOCC(F)F)C(C)C)C(C)C)CC(F)(F)C1 C#CCC(O)C(=O)NC1CCN(C(=O)Cc2csc(-c3ccc(NC)cc3)n2)C1 c1(OCC(=O)NCC2CC(F)(CNC(C3(O)CCOC3)=O)C2)cc(F)cc(F)c1 c1(C(N(CCCCN(C(=O)C(Cl)=CCl)C)C)=O)cnc(C2CCOCC2)s1 c1(C(N2CC(NC(C3CC34CCCC4)=O)C(O)CC2)=O)cnc2ccccn12 C(=O)(CC(C)(C)CCOC)NC1(C)CCN(C(C2N(C(=O)NC)CCC2)=O)C1 C1(CNC(C2CC2[N+](=O)[O-])=O)CN(C(C2N(C)CSC2)=O)CC1N(C)C CCC(C)C(C(=O)NC12COC(CNC(=O)CC(F)(F)F)(C1)C2)NS(C)(=O)=O C1(CNC(=O)C2=COCCC2)CCN(C(c2cc(O)nc(O)n2)=O)CC1(F)F N1(C(C2CC(C)CC(C)C2)=O)C2CC=C(C(=O)NCCN=[N+]=[N-])C1CC2 C(C(=O)NC(C)(C)C(C)NC(=O)CCn1cncn1)(C(C)C)c1cnc(C)s1 C1(OC)(CNC(=O)Cn2nccc2C)CN(C(c2ocnc2C)=O)C1 C1(C(=O)NC(c2n(CC)ncc2)C)CC2CCC(C1)N2C(=O)C(F)CCC(C)C c1(NC)ccc(C(=O)N(C)CC2CCCN(C(c3c(Cl)n[nH]c3C)=O)C2)nc1 c1(C(N2CC(C)(C(=O)Nc3ncc(C)nc3)C2)=O)ccc(-c2cc[nH]n2)nc1C c1(CC(=O)NCCN(C(c2c(CN(C)C)ccs2)=O)C2CC2)cccnc1Cl N12CC3CCC1CN2C3.CC(CC1CCC1)C(=O)NCCn1ccc(C=O)n1 c1(C(N2CC(NC(CC(CC=C)(C)C)=O)(CC)C2)=O)ccc(C)c2c1CCC2 C1(C(N(CC(C)NC=O)C)=O)C=CCN1C(C12CCC(C1)C2)=O.C(C)(C)(C)O c1(OC)ccc(C(=O)N(CC(C)O)CCNC(=O)C(c2ccnn2C)O)nn1 C(CCF)(C(=O)N1CCC(OCCO)C1)NC(C(COC)C)=O c1(OC)cc(C(=O)N(CCCNC(=O)CC2CCN(OC)CC2)C)c(F)c(Cl)c1 C1(NC(C=NOC)=O)CC2CCC1C(NC(c1ccc(C)c(C)c1N)=O)C2 N1(C(C(C)n2cccn2)=O)CC2CCCN(C(c3csc(S)n3)=O)C2C1 C1(C(=O)NCCN(C(=O)CCC2(CO)CCCC2)C)CCC(=O)NC1 C#CCC(C(=O)NC(C1(O)CCCCC1)C)NC(c1cc(OC)n(C)n1)=O Cc1cc(C(C)NC(c2cc(C)n(C3CCCCC3)n2)=O)n(C)n1 C=CCC(C(=O)NC(C1CCCCC1)C)NC(=O)CCn1cncn1 Cc1cc(C(=O)NC2CC(c3cc(-c4cncc(F)c4)on3)C2)nnc1C N1(CCC(=O)N(C2CC(NC(C3(c4ccncn4)CC3)=O)C2)C)CCCCC1=O C(=O)(C1CCCc2nc[nH]c21)NCC1CCCN(C(C=C(CCC)C)=O)C1 C1(NC(C2(NC(C3CC(N(C)C)C3)=O)CC(F)C2)=O)CCC(C)(O)CC1 C1(Br)(CNC(=O)NCC(CCOC)NC(=O)OC(C)(C)C)CC1(C)C C1(NC(CCCn2ncc(C)c2)=O)CN(C(=O)C(=O)NCC(F)F)CC1C1CC1 c1(OC)cnc(C(=O)NC2(C)CCN(C(=O)Cc3occc3C)C2)cn1 C1(C(=O)NCCC(C)OC)CCN(C(c2coc(Cl)n2)=O)CC1O Cc1sc(O)nc1C(=O)NC1CCN(C(C2CC3CC3C2)=O)C1C(C)C c1(C(=O)NC2CC(NC(C(C)(C)OCC)=O)C2)ccc(N)cc1 Cc1ccccc1NC(=O)C(N1CCN(CC(F)F)CC1)C1CCSC1 C1(C(N2CCC(CC(C)NC(=O)C(C)O)C2)=O)CC2CC2CC1C c1(CC)cc(C(N2CC(NC(C3COC3)=O)C(CO)C2)=O)nn1C C1(C(C)(C)NC(CCN(C)C(=O)C2CC2)=O)CCCN1C(=O)Cc1n[nH]cc1Br C(C(=O)NCC1CN(C(c2csnc2Cl)=O)CCCO1)(C(C)(C)C)NC(C)=O Cc1coc(C(=O)N(C)CCN(C(c2ccn(-c3ccncc3)n2)=O)C(C)C)c1 c1(CC(=O)NC2CCN(C(c3n(C)ccc(=O)c3)=O)C2)ccc2ncccc2c1 c1(C(N2CCC(NC(C=CCOC)=O)C2)=O)ccccc1NC1CC1C Cc1cc(C)c(C(=O)NC(CCN(C)C(c2nsnc2O)=O)C(C)(C)C)c(O)n1 O=C(N=c1cc2ccccn2[nH]1)N1CCc2ccccc2CC1 C1(CNC(CCc2n(C)cnc2)=O)CN(C(=O)CSCC#N)CC(C)(C)C1 C1(CNC(c2ncc(C)cc2F)=O)CN(C(=O)C(C)c2ccco2)CC(C)(C)O1 c1(C(=O)NCCOC2CN(C(=O)CCC3CCCC3)C2)cn2ccnc2cn1 N1(C(c2n[nH]c(C)c2[N+](=O)[O-])=O)CCN(C(=O)C2=CCCOC2)C(C)CC1C C1(NC(C(c2ccc(CC)cc2)O)=O)CC2CC(C1)N(C(=O)C=CCOC)C2 C(=O)(C1=C(Cl)CCOC1)N1CC(C(C)NC(c2ncn3c2CCC3)=O)C1 N1(Cc2ccn(C)n2)CCC(C2CN(C(c3c(Br)ccc(F)c3F)=O)C2)CC1 c1(CC(CC)NCC2CCCOC2c2cn(C)nn2)ccc(Br)c(F)c1 c1(C(N2CCCC2C2CCC2)C(=O)NCC(=C)C)ccc(COC(C)=O)cc1 c1(C(N(C)CC=CC2CCC2)=O)ccc(C(C)(C)C)nc1Br C1(NC(=O)C(N2CCOCC2)C2CC2)CCCCC1CNC(C1CC2(C1)CC2F)=O c1(C(=O)NC(C)C(=O)N(C)Cc2cn(CC3(CC)CC3)nn2)cccc(Cl)c1.COC Cc1cn(C)nc1CN(C(C1(CNC(=O)CC2(CO)CC2)CCCCC1)=O)C c1(CC)cc(C(N2CC(NC(=O)C(O)COC)C(C(F)F)C2)=O)ccc1O N1(C(c2c(Cl)cc(C)s2)=O)CCC(NC(=O)C(=O)NCC(F)F)C(C)C1 c1(C(=O)NCCCC(C(=O)NCC(COC)O)O)ccc2nccn2c1 N1(C(c2c(C)oc(C(C)C)c2)=O)CC2CC(NC(=O)CCOC3CC3)C1C2 Cc1c(Cl)cc(NCc2ccnc(CNC(=O)OC(C)(C)C)c2)cc1Cl c1(CC(=O)NCC(C2CC2)NC(C2C(OC(C)=O)C2)=O)ccnc(F)c1F Cc1cncc(C(=O)NC2CCC2C(=O)NCC(CO)C2CCC2)c1 N1(C(COCc2c(C)cccc2)=O)CC2CC1CN2C(c1ccc(=N)[nH]n1)=O c1(C(N2CC(C)(NC(c3nc(C)oc3)=O)C2)=O)cccc2ccc(O)nc12 C#CCC(CC#C)NC(C1(CNC(=O)CCC(N)=O)CCOCC1)=O c1(NC(C2CCN(C(C3CCOCC3)=O)CC2)=O)nc(Cl)c(Br)cc1[N+](=O)[O-] C1(C(N(CC(C2CCC2)OC)C)=O)CCC(CNC(C2CCSC2)=O)CC1 C1(NC(c2ccc(F)c(O)c2)=O)CC2CC1CN(C(=O)C(O)C1CCCC1)C2 C(=O)(CC1=NNC(=O)C1)NC1CC=C(C(=O)N(C)C)C1 C1(NC(C2C(CNC(CC3(CC)CCC3)=O)CCC2)=O)CCC12CCCC2 c1(CC)ncccc1C(=O)NC(CNC(c1cccc(SC)n1)=O)C(C)(C)C C1(C(N2CC(C)C(O)CC2)=O)CCN(C(=O)Cn2ccnc2)C2CCOC12 C1(C(=O)NCC(C)(C)OCC(=O)N(C2CCC2)C)OC2CCC1C2 c1(C(C#N)N(C(CCC2CC(OC)C2)=O)C2CC2)ccc(F)cc1 C1(OCC(N2CCCC2CN2C(=O)CCC2=O)=O)CCCCCC1 C(=O)(CC(C)CC(=O)N1CC(CNC(C2CC2C2CC2)=O)CC(C)C1)OC C1(C(=O)NCC(C)N(C(c2cncc(NC)c2)=O)C)CCC(C2CC2)C1 N1(C(C(=O)N(CC=Cc2ccccc2)C2CC2)=O)CCC(C2CC2(F)F)C1 C1(C(=O)NCC2(F)CN(C(C3(CF)CC(F)(F)C3)=O)C2)CN=C2N=CNN2C1 c1(CCC(N2CC(F)(CNC(C3C(C)(COC)C3)=O)C2)=O)c(C)noc1C N1(C(C(CNC(C2SC(=O)OC2)=O)O)=O)CCCC12CCCC2 C1(C(OC2CC3CN(C=O)CC32)=O)CC(C(C)C)=NO1.C=C1CC2(C1)C(=O)NC2.OC C=CC(C)(CC)C(=O)N1CCN(C)C(CNC(c2ccc(C(F)F)nc2O)=O)C1 N1(C(C(C)(C2CCC2)NC(C(C)c2cc[nH]n2)=O)=O)CCC(N=[N+]=[N-])C1 C1(C(=O)NCC(c2ccccn2)C)CN(C(c2cc(Cl)c[nH]2)=O)CC12CC2 c1(N2CCCC(NC(=O)NCCN(C)Cc3ccco3)C2)cc(=O)n(C)c(O)n1 c1(C(C)=O)ccc(C(N2CCC(CNC(C34CC(F)C3C4)=O)C2)=O)cc1F C(C(C)(C)C(=O)NCC1(O)CN(C(C2CCC2C(C)(C)C)=O)C1)N(C)C Cc1coc(C(C)(C)C)c1C(=O)NC1CC(NC(=O)CCCc2cccnc2)C1 C(=O)(CC(C)C(C)C(C)C)NC(C1CN(C(C2(C)CNC(=O)N2)=O)CCO1)C C1(CNC(C(C2CC(C)=NO2)NC2CC(OC(C)=O)C2)=O)CC(O)C(O)C1 Cc1ccccc1C1=NOC(C(=O)NC2CC(C)(CNC(=O)CSC(C)C)C2)C1 C1(CNC(c2cncc(C)n2)=O)CCN(C(c2cnc(C)s2)=O)CC1O c1(C(N2CCC(NC(CCC(C)C)=O)CC2C)=O)cc2ccc(Cl)c(F)c2o1 C(=O)(CC1=NN(C)C(=O)C1)NC(CC)CCO C(CC(C)C(=O)N1CCC(CCNC(=O)CC2(n3cccn3)CC2)CC1)=CCC C(CCNC(=O)C(=O)NCCC(N)=O)(C(C)(C)C)NC(C(CC)SC)=O c1(C(=O)NC(C(C)NC(c2csc(C3CC3)n2)=O)CO)nccc2n[nH]cc12 N1(CC(CCSCC(=O)Nc2ccc(OC)cc2)O)CCSC(C)C1C C1(C(N(CCC(=O)NCC(C(CC)C)CO)C)=O)CC(=O)CC12CCC2 CC1(C)CC(CNC(C2CCCC3CC23)=O)N(C(=O)COC2(C)CCC2)C1 c1(C(C(=O)N)C)c(F)cccc1F.C1(=O)CC(=O)NC2C(C2)CN1.CC(=O)OC CC(C(=O)N1CCSCC1C(=O)NCCCc1nncn1C)C(F)(F)F c1(CC)nccnc1C(N1CCC(C(C)NC(=O)Cc2cnn(C)c2C)CC1)=O C1(C(=O)Nc2c(C)nn(C)c2)CCCCCCN1C(C1CN(C(N)=O)C1)=O C=CCCC(=O)NC1(C(=O)NCC(C2CCOCC2)C)CCC1 N1(C(C2CC(CC)C2)=O)CCCCC1CN(C(=O)C(C1CCCO1)C1CC1)C N1(C(C(C)OCCC=C)=O)CCCCC(CC(=O)NCCN(C)CCOC)C1 C1(C(=O)NCC(C)NCCBr)CC(F)CN1C(c1ccc(OC(F)F)cc1)=O C1(NC(CCCSCCC)=O)C(C)(C)C(NC(=O)C(C)C(C)(F)F)C1(C)C C#Cc1ccc(C(N2CCC(F)(CNC(=O)CC3CC3(C)C)C2)=O)cc1C C12(NC(=O)CCC(F)F)CC(CNC(c3ncccc3O)=O)(C1)OC21CCC1 C1(C(N2CCC(OC(C)=O)C2)=O)C2CN(Cc3ccnc(C(C)(C)C)c3)CC12 c1(C(=O)OC)ccc(C(N2CCCC2CCNC(=O)CSC)=O)n1C C1(O)(CNC(=O)CCc2ncc[nH]2)CCCN(C(=O)C(c2ccc(Cl)s2)=O)C1 S(=O)(=O)(c1cccc(CO)c1)N1CCC(CCC(=O)Nc2ccc(F)cc2)CC1 c1(C(=O)NC(C)CNC(=O)CN2CCCC(N(C)C)C2)cccc[n+]1[O-] c1(C(=O)NCC(CNC(C2C(C)C2(F)F)=O)OC)cnc(OCC2CC2)cn1 C1(OC)CC(CNC(C2CC(C)N(C)C2)=O)N(C(=O)COCc2ccccc2)C1 Cc1nc2ccccc2n1CC(N1CC(NC(=O)C(C)n2ccnc2)C(C)C1)=O CCC(C)CC(C(=O)NC1CCN(CC)CC1)NC(c1cc(Cl)ccc1Cl)=O C(c1ccccc1)=CC(C)C(=O)NC(C)C(C)(C)NC(c1cnc(C2CC2)s1)=O Cc1nc2cc(Cl)cc(C(=O)N(C(C)CN(C(=O)CCn3cccc3)C)C)c2[nH]1 c1(OCC)ccc(C(=O)NC2CCN(C(=O)CCC(C)(C)C)C2C)cc1Cl O=C1CCC(C(=O)NCC#CCNC(=O)C(c2ccc(CO)cc2)O)CN1 N1(C(C=COCC)=O)CCc2nc(C(=O)Nc3onc4ccccc34)ccc2C1 N1(C(CN2C(C)CC2)=O)CCCC(N(C(=O)Cn2cnc(C#N)n2)C)C1 N1(C(CC2N(C(C(CC#C)O)=O)C3C2CCC3)=O)CC(C)CCC12CC2 C12(CC(=O)NC(CC3CCN(C(c4c(C)nsc4)=O)CC3)C)CCC(C)(C1)OC2 C1(NC(C(C2CCCC2)OC)=O)CN(C(=O)CCc2cnco2)CC1C1CC1 C1(N(C(=O)CC2C=CS(=O)(=O)C2)C)CN(C(=O)CCc2cn(C)cn2)CC12CC2 C1(CC(=O)N(C2CCOC2)CC)CN(C(C23CC2CNC3=O)=O)C(C)(C)C1 c1(C(=O)NCC(CC)Nc2nnc(C3CC3)s2)ccccc1-c1ccc[nH]1 N#Cc1ccc(Cl)cc1N1CCC(C(=O)NC2CCC(=O)NC2=O)CC1 CCC(CC(=O)NCC(C1CCN(C(=O)Cc2cnoc2)CC1)(C)O)C1CC1 C1(C(c2nnnn2CC2(CC(C)C)CC2)NCC2CC2)CC2(CCC2)C1 Clc1cccc(CC2(COCc3ccccc3Br)CC2)c1 C=C1CCC(C(=O)NCCc2n[nH]cc2C(=O)NC(C)CC(F)(F)F)CC1 C(C)(C(C)(C)C(=O)NCC(c1nccs1)C)NC(C1CC(=C)C1)=O CCCCCC(O)CC(=O)NC1(C(N2CCC2C)=O)CC1(C)C C(C(C)(O)CC(=O)NC(CCC1CC1)C(=O)N1CC(N2CCOCC2)C1)OC c1(C(=O)NCCCC(C)NC(c2cn(C3CCOC3)nn2)=O)csc(C#N)c1 c1(CCC(=O)NC2CCCN(CC(=O)Nc3cccnc3)C2)ccc(F)cc1 C(=O)(CCS(=O)(=O)C1CCCC1)NC1C2CN(C(c3c(C)c(F)ccc3)=O)C1C2 C=CC(CC)CC(=O)NCC(C1CCN(C(c2cnc(O)n2C)=O)CC1)(C)O N1(S(C)(=O)=O)CCC2CN(c3cc(-c4ccccc4)nc(Br)c3)CC12 c1(C(=O)NCC(C2CCOC2)NC(c2cc(CC)on2)=O)cccc(C)c1Cl c1(C(=O)NC(C2(O)CN(C(=O)CCc3ccnn3C)C2)C)sncc1Br CC1CN(c2cc(NCc3cc(O)n(C)n3)ncn2)CCC1N(C)C N1(C(C2N(C(C)C)CCC2)=O)CCC(C)(C)C(NC(C2CC(Cl)(Cl)C2)=O)C1 Cc1c(C(N2CCCC2CNC(=O)CCc2ccoc2)=O)ccn1C1CC1 N1(C(C(C)OCC=C)=O)CCN(C)C(C(=O)N(C2CCC2)CC)C1 C(CC(=O)Nc1ccccc1C)(C(C)(C)C)NC(CC(C(=C)C)O)=O C(=O)(C(C)(CC=C(Cl)Cl)c1ccccc1)NCCNC(c1c(C)noc1)=O O(NC(=O)C1=NOC(CNC(=O)C(F)=CC2CC2)C1)C(CC)CC C1(O)(CCNC(C(C)CN2CCCCC2)=O)CCN(C(=O)Cc2ccoc2)CC1 c1(C(=O)NCCCN(C(C(C)NC(C)=O)=O)CCO)cccc2ccncc12 Cc1cc(N2CCC(n3cncn3)CC2)nc(N2CCCC(C)(N(C)C)C2)n1 CCC(C)C(C(=O)NCCCCCNC(=O)COC1CC(F)(F)C1)NCC(C)O c1(C(=O)NC2CC(NC(COCC=C)=O)C2)cc(N(C)CCC)ccn1 C#Cc1c(F)cc(NC(c2nc(CCc3ccccc3)no2)=O)cc1F CC1OC2(CCN(C(N)=O)CC2)NC1=O.c12ccc3c(c1)C(NC2=O)CCC3 c1(CNC(=NCCOC)NCC2CCC(F)C2)nnc2ccc(Cl)cn12 C(C(O)CNC(=O)C(C)n1cncn1)NC(CNC(CNC(C)=O)=O)=O Cc1cc(C(=O)NCC(C)CNC(c2nocc2C2CC2)=O)oc1C c1(CN(C(=O)C(C)C2CCC2)CCCNC(C=C(CC)CC)=O)ccccn1 c1(C(=O)NCC2(CN(C(C(C)CC3CCCCC3)=O)C)CC2)n[nH]cc1[N+](=O)[O-] C(=O)(CC1COc2ccccc21)N(CCCCCCNC(C1CCCS1)=O)C CC1(C)CCc2c(C(=O)NC3CCCCC3c3cccc(Br)c3)n[nH]c2C1 CC(c1cccnc1)=CC(=O)NCCOCCCNC(=O)CCCCCC#N C(CCC(C)(C)C(=O)NC1CCN(CCCO)C1)NC(CCc1n(C)ccc1)=O C12(CNC(C3N(CCC)CCC3)=O)CC1CN(C(=O)CCN1CCC(O)CC1)C2 c1(C(=O)NCC(C2N(C(C(C)C(C)O)=O)CCC2)(C)C)cn(C)c2ccccc12 c1(C(=O)NC(CNC(C(CC=CC)CC)=O)CO)cncc2nc(O)[nH]c12 C1(C(N2CCC(N(C(c3cnc(CC)s3)=O)C)C2)=O)CCCCN1C(=O)C1CC1 c1(SCC(=O)NCC2C(CNC(C3C4COCC34)=O)C2(F)F)ccc(O)cc1 C1(NC(C=C(C)C(F)F)=O)CCN(C(c2csc(-c3cnccn3)n2)=O)C(C)C1 c1(OC)nc2c(cc1NC(=O)C(=O)NC1CC1C1CC1)CCC2 CN1CCC(C(=O)NC2(CC(=O)NCCn3cncn3)CC2)C1=O N1(C(c2cc(C)no2)=O)C2CCC1CN(C(C1CCCCC1(C)C)=O)CC2 N1(C(c2c(C(C)C)ocn2)=O)CCN(C(=O)CSc2n[nH]c(O)n2)CC1C c1(C(C)=O)cnc(N2C3CCC2C(CNC(c2cc(Cl)c[nH]2)=O)C3)cc1C CC(C)C(F)(F)CCNC(=O)C(=O)N1CC(NC(C2CC2C)=O)C1 C1(CNC(c2nc(CC)sc2)=O)CC(C)N(C(C2CCC(=O)N2)=O)C1 N1(C(C2(C(=O)OCC)CCCC2)=O)CCN(C(=O)CC2NC(=O)NC2=O)CC1 CCCCC(C)C(=O)N1CCCC1CNC(C1CSCN1C(=O)CC)=O C1(C(N2CC(N(C(C(C)NC(C)=O)=O)C)C2)=O)CC(C)CC(C)(C)C1 C1(CNC(c2c(CC)onc2)=O)C2CN(C(C3CC3CC(C)(C)C)=O)CC12 CC(CCCC(=O)N1CC(N(C)C(c2cc(N)ccc2O)=O)C1)c1ccccc1 C1(C(=O)NCC(CNC(C=NOC)=O)(C)O)CC2(CCOCC2)C1 C1(NC(CCC=CC)=O)CC(CNC(c2oc(SC)cc2C)=O)C1(C)C c1(CN(CCN(C(c2ccc(CC)s2)=O)C)C)ccc([N+](=O)[O-])cc1C(C)=O Cc1nc2cc(C(=O)NC3CC(F)CN(C(c4cncc(F)c4)=O)C3)cnc2s1 c1(C(N(C(C)CNC(=O)CSN2C(=O)CNC2=O)CC)=O)ccccc1SC n1(CCC(N2CC(C)(NC(Cc3nc(C)oc3)=O)C2)=O)c(C)cc(O)cc1=O CCC(C)CC(C)C(=O)N1CCCC(NC(c2ccnn2CCOC)=O)C1 N1(C(c2n(CC)nnc2)=O)C2CCCC1CN(C(=O)CCCNS(C)(=O)=O)CC2 N1(C(C2CCCN(C)C2)=O)CCCC(F)(C(=O)NC2(CCCF)CC2)C1 c1(C(=O)NCCC(=O)NC2CCCC(CC)C2)cc(C)cc(F)c1 CC(C(=O)N(C)CCc1cccc(Br)c1)C1OCCc2ccccc21 C(C(C)C(=O)N(C)CCNC(=O)CC1CC(C(C)O)C1)SC N1(C(CN(C(C)=O)C)=O)CC(CNC(c2ccccc2CCN(C)C)=O)C(C)C1 CN1CCC(C)(C(=O)NCC2CCC2NC(C23CCC(C2)C3)=O)C1 C1(CCC)(NC(=O)C=CC(C)(C)SC)CCN(C(c2cncn(C)c2=O)=O)CC1 c1(CC)cccc2c(C(=O)NC(CO)C(C)NC(c3nocc3C)=O)c[nH]c12 N1(C(C(C)NC(COC)=O)=O)CCN(C(=O)C(C)(C)CN(C)C)CC1CO CN1CC2CCCC(C1)N2C(=O)NCCC1CC2(CCO1)CC2 CCCC(F)C(=O)NC1CCC(C(=O)NC2CC2)CC1.c12cccc(c1)NC2=O CN1N=CC(CC(=O)NCCn2cnc(C(=O)N(C3CCCCC3)C)c2)C1=O c1(C(N(CCCNC(c2oc(C)nc2C)=O)CC)=O)sccc1S(N)(=O)=O CC1CN(C(C2CCCN(C34CC(C(C)C)(C3)C4)CC2)=O)CCc2ccccc21 CCCCCCCCC(=O)N1CC2(CCCN(C(c3cc(CO)on3)=O)C2)C1 c1(OC)c(CNC(c2cccn2C2CCCC2)=O)cccc1Cl C1(NC(c2c(OCC)ccs2)=O)CN(C(=O)COC2CCCC2)CC1O CC(C)(F)C(C)(F)C(=O)N1CCC1CNC(=O)CCc1c[nH]c2ccccc12 S(=O)(=O)(CCC(=O)N1CCN(C(=O)CNC2(CO)CC2(F)F)CC1)NC CC1C(NC(c2cncc(-n3cnnn3)c2)=O)CCN1C(=O)Cc1ccco1 C(N=c1nc2[nH][nH]cc-2c(O)n1)C1(O)CN(C(=O)CC2CC(O)C23CCC3)C1 N1(C(=O)NCC(=O)NCCN2CCC(O)C2)CCC(O)(C(N2CC=CC2)=O)CC1 c1(C(CC)C)ccc(C(=O)N(CCCNC(=O)CNC=O)C)c(O)n1 N1(C(C(CCCC)O)=O)CCC2(CC2)CC1C(=O)Nc1ccccc1CCO C(=O)(C(C)(C)C(=O)N1CCCC(N(C(=O)CN2CCC2C)C)CC1)OC Cc1cc(N2CCC(N(C)C(c3nc[nH]c3C(C)(C)C)=O)C2)nc(C2CC2)n1 N1(C(CC2C(C)C2)=O)CC=C(CNC(c2ccccc2C2CCOC2)=O)CC1 N1(C(c2c(C)scc2)=O)CC(C(=O)NCCCN(C)C2CC2)C2(CC2)C1 c1(C(=O)OCC)cc2c(nc1N1CCOC(CNC(=O)C=CSC)C1)CCOC2 C1(N(C(=O)CC2(C)CC2)C)CCCCC1C(=O)NCCc1cccc(O)n1 N1(C(c2c(OC)c(Cl)ncc2)C(=O)NC2CCOC2)CCC2CCCCCC2C1 C#Cc1cc(=O)n(C)c(=O)n1CC(F)=C(F)F c1(C(CC)NC(=O)NCC2(C)CCCCO2)cc(Cl)cnc1F CC1=C(C)CC(C(N2C3CC2CN(C(C2(C)C=CCC2)=O)C3)=O)CC1 C1(C)(CNC(C2N=C(C)SC2)=O)CCCN1C(=O)CCCn1nc(C)cc1C C=CC(CC)C(=O)NCc1ncc(C(=O)NC2CCCC2C(C)C)cn1 c1(CC)csc(C(F)(F)C(=O)NCCCN(C(=O)CC(C)N(C)C)C(C)C)n1 C1(CC(N)=O)(NC(=O)CCC(=O)C2CC2)CCN(C(C2CC23CCOCC3)=O)CC1 C1(OC)CN(C(=O)CO)CC1NC(=O)CC(C)(C1CCC1)N(C)C.c1(SC)nncs1 Cc1nc(C(=O)NCC2(O)CCN(C(=O)COCCc3ccccc3)C2)nn1C Cn1cc(C(C)(C)C(=O)NC2CCC(NC(=O)C(O)CN3CCCC3)C2)cn1 N1(C(C(C=C)O)=O)CCC2CN(C(c3ccnc(CC)n3)=O)CCC12 CC1(C)OCc2onc(C(=O)NC3CC(NC(C4SC5C=CC4CC5)=O)C3)c2O1 c1(CC(=O)NC2C(CNC(c3cc(COC)no3)=O)C2)ccccc1OC C1(CCC)CN(C(=O)C(c2ccc(C)s2)C)CCN1C(c1cc(C)ccc1F)=O CC1(C)C(C(=O)NC2CCC(NC(C3CCS3(=O)=O)=O)CC2)C1(C)C c1(C(=O)NC(CC2CN(C(C3(SC)CCC3)=O)C2)C)cncc2sccc12 C(CN=c1nc2sccc2c(NCC2CCC3C(CC2)C3(F)F)[nH]1)c1c(C)noc1 Cc1ccc(NC(=O)C=CC(=O)NCC2CC2NC(=O)C(C)(C)c2ccns2)cc1 c1(OC)ccc(CC(N2CCCC2(C)c2cn(CC(F)(F)CO)nn2)=O)nc1C Cc1cnn(C)c1-c1cn(CC(=O)NCCN(C(C)C(=O)O)C)nn1.OCC N1(C(CCP(C)(C)=O)=O)CC(C2CCN(C(C3CC(F)C3)=O)CC2)C1 c1(C(N2CCC(C3CCOC3)C2)=O)cccc(S(=O)(=O)NC2CCCC2)c1 C1(NC(CCN(CCC)C)=O)CC2CC1N(C(=O)CCCOc1ccccc1)C2 CC1CC(C(=O)NC(Cc2ccccc2)CO)N(C(=O)CSc2nc[nH]n2)C1 n1(CC#C)cnnc1C(=O)NC(Cc1cc[nH]n1)C(=O)N1CCC1(C)C(=O)NC Cc1coc(C)c1C(=O)NC1CC(CNC(=O)CCC2CCCN2C)C1 O(NC(=O)CCCC(C)(C)NC(C1CC(C)CCO1)=O)CC(=C)Cl C1(C(=O)NCCC(C)(C)NC(=O)Cn2ccc(C(F)F)n2)CCn2ncnc2C1 N1(C(C(CC)Cc2ccccc2C)=O)CC(NC(=O)C2=NOCC2)CC2(CC2)C1 CC(C)(C)C1=NOC(C(=O)NCCC2CN(c3ncnc(=N)[nH]3)CCO2)C1 Cc1oc(C(C)(C)C)cc1C(=O)NCCN(C(=O)CCN1CCC(F)C1)C1CC1 c1(C(=O)NC(C(C)NC(c2ncc(C)c(Cl)c2)=O)C)cc2c(C)cc(Cl)cc2[nH]1 c1(CCC(=O)NCC(C)CNC(c2ccc(Br)o2)=O)ccc(F)c(F)c1 C(C(CC(C)C)C(=O)N1CC2CCN(C(c3cnc(O)c(Br)c3)=O)C2C1)OC C=CC(C(=O)NC1CC(NC(c2cnc(O)o2)=O)C1)c1ccccc1 CC(C)(CCF)C(=O)NCC1CCN(C(=O)CC2CCCSC2)CC1O c1(C(=O)NC(C)CNC(=O)C(=O)NCC2CC2)n[nH]c2c1C(=O)CCC2 c1(C(N2CC(COC)(NC(c3ccc(O)nc3)=O)C2)=O)c(C)nn2ncccc12 Cc1coc(C)c1C=CC(=O)NC(C)CCNC(=O)CN1C(=O)NC(C)(C)C1=O C1(CNC(c2c(CC)n(CC)nc2)=O)CN(C(=O)CC2CCCN2C)CCC1C N1(C(C(C)(C)OC(C)=O)=O)CCC(O)(C(C)CNC(c2cc[nH]c2C)=O)C1 CCCC(CCCNC(c1cccs1)=O)NC(c1cscc1Cl)=O C1(C(=O)NCCC(=C)CNC(=O)CN(C)C2CC2)CCCCC1NC C12(C(=O)NC3COCCN(C(c4c(C)cnn4C)=O)C3)CC1COC21CCC1 C(=O)(C(C)(F)C(C)(C)F)NCC1CCCCN(C(c2c(OC)nc(C)nc2)=O)C1 CC(C)C(CC(=O)NCC1CC1CNC(=O)C=CC1CCC1)C(C)C C(C)(CC(=O)N1CC2C(CNC(=O)C(N)=O)C2C1)(C(F)(F)F)N(C)C N1(C(c2cn(CCNC(c3c(C(C)C)noc3)=O)nn2)=O)CCSC(C)C1 CN1C(=O)CSC1=CC(=O)NCC1CCCCC1NC(c1ccnc(CO)c1)=O N(C(=NCCc1ccc(O)cc1)NCc1ccccc1)Cc1c(C)cco1 N1(C(c2c(CCC)[nH]cc2)=O)C2CC1CN(C(=O)CCc1scnc1C)C2 Cc1cccc2c1N(C(=O)CCC1CCCCN1C)CCC2C c1(OC)ccc([N+](=O)[O-])cc1C(N1CC2CCN(C(=O)CCC3CCC3)C2C1)=O c1(CC)cnoc1C(=O)NC1CCC(CNC(C2(CC(C)C)CC2)=O)C1 N1(C(C(CC)N(C)C(c2cc[nH]c2)=O)=O)CCC2CCCC2C1 C=C(C)CCCC(=O)N1CCC(C)C1C(=O)NCCCn1ccnc1 c1(-c2n(CCC)nc(CCCO)n2)cnc2n(c1=O)CCS2 c1(OC)ccc(C(F)(F)F)c(F)c1.c12ccc(F)c(c1)-c1ccc(cn1)NC2=O CC(C)C(C(=O)N1CCCCC1CNC(c1cnn(C)c1Br)=O)NC=O C1(C)(C(=O)NCCCN(C(=O)CN2CCC(F)C2)C)CCCS1(=O)=O C1(C(N2CCN(C(COC)=O)C3C2CCC3)=O)CCc2nc(C)ncc2C1 C1(CC)CCN(C(=O)CCC2CC(OC)C2)C1C(=O)NCC1(C)CC(F)(F)C1 C12(C(=O)NC(C)Cc3ccco3)CC1CN(C(=O)CN1CCOC1=O)C2 C1(C(=O)NCC2CCC(NC(C3(CC)CC3)=O)CC2)CCc2ncnn2C1 C1(NC(c2cccc(OCC(N)=O)c2)=O)CN(C(=O)C(F)C(F)(F)F)CCC1F C1(NC(C2N(CCCC)CCCC2)=O)Cc2n[nH]cc2C(C(F)(F)F)C1 Cc1nc2cccc(C(=O)NC3CCN(C(C4CCCCC45CCCC5)=O)C3)n2n1 C1(N(C(c2ncc(CC)cn2)=O)C)CN(C(C2CCCC2F)=O)CCC1O N1(C(C(=O)NCCOCC)=O)CCN(C(C)=O)C(C)CC1C.C(=O)(C(C)(C)C)N N1(C(c2ccc(CC)[nH]2)=O)CC2CCCC2C1C(=O)NCC12CC(CN1C)C2 C1(CNC(C2(CC)CC2)=O)CN(C(c2cc(C(F)F)nn2C)=O)C2(CCC2)C1 C1(C)CSCCO1.C(C)(C(=O)NCCS)SC.C1CC(=O)N1 C1(CNC(=O)C(=O)NC2CC3(C2)CC3(F)F)CC(C2CCC2)C1 C=CC1(C(N2CC(n3cc(-c4cnn(CCOC)c4)nn3)C(C)C2)=O)CCOCC1 c1(CN2CCC(n3ccc(C(=O)OC)n3)CC2)cccc([N+](=O)[O-])c1F CCC(C)C(CNC(=O)C(CCOC)NC(c1ccn(C2CC2)c1C)=O)CO C(=O)(C(O)CC(F)(F)F)N1CCCC(CNC(C(C(CC)C)NC(N)=O)=O)C1 C1(O)(C(C)CNC(c2ccc(Br)o2)=O)CCN(C(C2(O)COC2)=O)C1 c1(NC(C(N2C(C)(CCO)CCC2)=O)=O)cc(C2CC2)cc(Br)c1 C=CC(C)(O)CC(=O)N1CCC(C(C)C(=O)Nc2cc(C(N)=O)cc(C)c2)C1 CC1CCc2nc(C(=O)NC(C)CCCNC(c3cnc(S)[nH]3)=O)ccc2C1 C1(CN(C(c2cc(C)ns2)=O)CC)CCCN(C(=O)C(c2cccc(Cl)c2)O)C1 N1(CC)CCOC(C(N2CCCC(C(C)(C)C(=O)NC3CC(O)C3O)C2)=O)C1 C(=O)(C1CCc2nnc(C)n21)N(CCOCCNC(C(CC)(C#N)CC)=O)C C(=O)(CC(C(F)F)n1ccnc1)NC1C2CN(C(C(c3ccnn3C)C)=O)C1C2 CC(C)CCC(F)C(=O)N1CCCC(CN(C)C(C2CCCN2C(C)C)=O)C1 C1(c2ccccc2)CC(NCc2ccc(-c3ccccn3)o2)CCS1 Cc1cccc2c1OCCC2N(C)C(=O)C(=O)Nc1ccc(C#N)cc1 C(=O)(C(CC)C(=O)N(C)Cc1ccc(F)c(F)c1)OC.C1(C)C(=O)O1 N1(C(c2ccc(C)o2)=O)CCC(NC(=O)CCC[N+](=O)[O-])C(O)C1 C1(C(=O)NCC(C(N)=O)O)CC2CN(C(=O)CN3CCC(F)CC3)CC2C1 C12(CNC(Cn3ccc(C)cc3=O)=O)CCCC1N(C(=O)C=CCO)CCC2 C1(C(=O)Nc2nccn2C2CC2)CCN(C(=O)CCC2CCCCN2)CC1 c1(CNC(C(OC)OC)=O)ncccc1CNC(=O)C(c1ccc(Cl)cc1)C CC(CCN=c1[nH]c2cc(F)ccc2o1)NC(C1(S(C)(=O)=O)CC1)=O C1(C(NOC(C)(C)C)=O)CCCC1O.N1(C(=O)C=CC(F)(F)F)CC(C)(CF)C1 N1(C(C#CC(=O)N(C)C)=O)CCC2CCN(C(c3coc4c3COC4)=O)CC2C1 C1(NC(C(C)OCC=C)=O)C2CC3CN(C(=O)CSCCC(C)C)C1C3C2 C(N=c1nc(N2C3CCCC2c2c[nH]nc2C3)c2c([nH]1)CCS2)c1c(C)nco1 CC(CN=C(NC(=O)CC1CCOC1)N1CCN(C(C)C)C(=O)C1)N(C)C CC(C)C(O)C(C)C(=O)N1CC(NC(C2(C)CNC(=O)C2)=O)C1 N1(C(C(C#C)(C)C)=O)CCCCC(NC(=O)C(C)NC(=O)NC2CCCC2)CC1 c1(OC(C(=O)NCC2C3CN(C(C(CC)(F)F)=O)CC32)F)ccc(Cl)c(F)c1 C1(SCC(=O)N(C2CCN(C(c3cnsn3)=O)C2)C)CCCCO1 CC1CCC(C(=O)N(CCCN(C(=O)C(C)(C)c2sccc2Cl)C)C)C1 N1(C(C(CC)O)=O)CC2CCCC(C1)N2C(=O)C(F)C(C)(F)F.c1(SC)ccccc1 N1(C(C(C#C)(C)C)=O)CCOC2(CCN(c3ccc(C)cc3[N+](=O)[O-])C2)C1 C(=O)(CCCCCS(N)(=O)=O)N1CC(C(C)NC(c2nc(Br)c[nH]2)=O)C1 c1(OC)cc2c(cc1F)C(C)CCC2NC(=O)Oc1c(C)cc(C(C)C)cc1C CC1CC(C(N2CCCC(F)(CNC(c3c(Cl)n[nH]c3C3CC3)=O)C2)=O)CC(C)C1 c1(C(N2CC3C(NC(=O)C(O)CF)(C3)C2)=O)cc2c(F)c(Br)ccc2[nH]1 C(=O)(N=c1[nH][nH]c2c(Cl)cccc12)C1(C)CCCN(Cc2cnn(C)c2Cl)C1 N#Cc1c(N2CCC3(CC2)CN(C(=O)CC2CC4(CC4)CO2)C3)cccc1C#N N1(C(c2cc(SC)oc2)=O)CC(NC(c2nc(O)c(C)s2)=O)C(O)C1 c1(CNc2c(C)ccc(-c3ncco3)c2)ccc2cncn2c1C C(C(CC(C)C)C(=O)NC(c1ncccc1C)CC)OCC Cc1c(NC(C2CCC=CC2NC(=O)CCC(C)N(C)C)=O)cccc1CO C1(C(=O)NCC(CC=C)NC(=O)C(C)C(F)F)CCC2(CC1)CC(O)C2 C(CC(C)C(=O)N1CC=CC1(C(N1CCC(C(N)=O)C1C)=O)COC)=CC N#Cc1csc(CNC(c2cscc2Br)c2nnnn2CC2CCOCC2)n1 c1(CCCC=C)ccc(C(=O)NCC2CC2NC(=O)CCN2CCCC2)cc1 c1(C(=O)NC2CC(C)(CNC(C(CC)(C)O)=O)C2)cc(C)c(O)nn1 C(CC(=O)NCCC1CN(C(C2CC(C(N)=O)C2)=O)C1)SC N(C1COc2cccc(F)c21)C(N(C1CC1)Cc1cn(C)[nH]c1=N)=O N1(C(C(C)CC(N)=O)=O)CCC2(CCCC2NC(=O)CN2C(=O)CCC2=O)CC1 C1(OCCNC(=O)C(C2CCCO2)C2CC2)CCN(C(c2ccccn2)=O)C1 c1(C(=O)NC2C(NC(C(COC)COC)=O)CCC2)ccc2ccn(C)c2c1 c1(C(=O)NCC2(O)CN(C(C3CC(OC(C)=O)C3)=O)C2)cncc(C(F)(F)F)c1 c1(C(=O)NCC(CNC(CCC=C)=O)C(F)(F)F)coc2ccccc12 c1(OCC(N2CC(C)C(NC(=O)CC3COCCO3)C2)=O)c(F)cc(F)cc1F c1(C(=O)NC(CC)CN(C(C2CC3C=CC2C3)=O)CC)cnc(C)c(N)c1 C(CC1CC1)(C(=O)NCCN(C)CC)NC(COC(CC)C)=O C(=O)(C(F)(CNC(c1cc(O)ccc1F)=O)C(C)C)Nc1ccc(OC)cc1Cl C1(CCCNC(C2C(F)(F)C23CC3)=O)CCCCN1C(=O)C=Cc1cocn1 CN1CC(F)CC1C(=O)NC(CNC(C1CCC(C)(C)C1)=O)CO c1(C(=O)NC2CCN(C(C=CSC)=O)CCC2CO)cnc2ncccc2c1 c1(OC)cccc(F)c1C(=O)NC1CC(C)CN(C(c2cc(C)ccc2Br)=O)C1 c1(C(C)NC(=O)NC(CCN(C(CCC)C)C)=O)ccnn1C C1(C(N2CC3C(CNC(c4cc(C)oc4)=O)C3C2)=O)CCCC2CCCCC12 C1(NC(c2ccc(N(C)C)nn2)=O)CCC12CCN(C(=O)COCCSC)CC2 CC(C)(CCC(=O)NOCCOCCF)NC(C1CCC2(CCC2)C1)=O c1(C(N(C(C)CNC(=O)CC2(C)CC2(F)F)C)=O)cnc(Oc2ccccc2)s1 C1(NC(C#C)=O)CCSC12CN(c1ccc(C(F)(F)F)nn1)C2 c1(OC)ccc(Sc2nnc(CN(C)CCF)n2C2CC2)cc1 C#Cc1cc(F)c(C(N2CC3CCN(C(C45CCC4C5)=O)C3C2C)=O)cc1F N1(C(C(C)N(CCC)C(c2ccc(CC)o2)=O)=O)CCC(N=[N+]=[N-])CC1 CN1C(=O)CC(C(N2CC(NC(c3ccc(F)c(CO)c3)=O)C2)=O)NC1=O N1(CCNC(NCC(F)=C(C)C)=NCCF)CC(C2CCCC2)C1 c1(C(C(=O)NCCOCC)N(C)C)nn(C)c(C)c1Cl.c1(CO)nncn1C(C)C N1(CC2C(C(C)(C)C)C2)CCCCC1CNC(=O)CC=C(Cl)Cl.n12ccc(n1)C2 N1(C(CCC(C)(C)F)=O)CC2CCC(C2)C1CO C1(NC(C(C)(C)N(C(=O)CC2COCC2O)C2CC2)=O)CN2CCC1C2 CN1CCC2(C1)C(=O)N2.C(C1=NOCC1)NC(=O)CCOCC(F)F N1(C(C)C)CCC(N(C(=O)CCCC2CCCS2)C)C1 CC1CC2(CC(C(N3CCC(C(F)C(N4CCOCC4)=O)C3)=O)C2)C1 CC(C)CC(C(=O)N1CCC(CC(F)F)C1)N(C(=O)C(C)(C)CO)C C=C(C)CC(C)C(=O)NCC1CCCC1NC(c1nn(C)cc1CSC)=O CC1(CNC(=O)CCCc2ccccn2)CC(NC(c2cc(Cl)cs2)=O)C1 c1(SC)cc(F)cc(F)c1NCC1(c2nnnn2C(c2scc(Cl)c2Cl)C)CC1 c1(OCCCC)ccc(C(=O)NCCC(C)CCNC(=O)COCCSC)cc1 c1(C(=O)OCCCSc2ccccc2F)c(Cl)sc(Cl)c1Cl C12(NC(C(CC)NC(C)=O)=O)CCC(C1)N(C(=O)C(C)C)C2 C1(COC2CC(C(=O)NCC(=O)NC3CCCCC3)C2)CC(O)CCO1 c1(C(N(C2CN(C(=O)C(N)Cc3cscn3)CC23CC3)C)=O)cc(F)c(F)cc1F C1(NC(C2(c3cc(C)on3)CCC2)=O)CN(C(c2c[nH]c(=N)s2)=O)CC1(C)C C1(C)(C(=O)NCC(CN(C(=O)C=Cc2csc(Br)c2)C)O)CC(C)(C)C1 N1(C(c2c(C)[nH]nc2Cl)=O)CC(NC(c2cnn(C)c(=O)c2)=O)C(C)(C)C1 c1(C2CC(C(N(CC(C)CNC(C3CC3F)=O)C)=O)C2)ccccc1 CC#CCC(C(=O)NCC1COCC(=O)N1C)NC(=O)C(C)CCCC N1(C(c2c(NC)cccc2)=O)CCC2(C1)CN(C(=O)CC(F)F)C2 N1(C(c2cnc(OC)nc2)=O)CCC2C1CCCN2Cc1cc(F)c(F)cc1Br N1(C(C(C)OC2COC2)=O)CCC(CNC(C2CCC=CO2)=O)CC1 N1(CC)C(C)CN(C(C2(CC)CCN(C(c3cccc(C)n3)=O)C2)=O)CC1C CC1(C)CCc2nc(C(=O)NCC(N3CCOCC3)=O)ccc2C1 c1(NC(c2cc(OC)ns2)C)nc(N2CCCCCC2)nc2scnc12 C1(OC)CC(NC(c2c(C(=O)NC3CCC3(OC)OC)n[nH]c2)=O)C12CCC2 n1(CC=C)nnnc1C(C(C1CC1)OC)NCCc1nc(C)cs1 C1(NC(CCc2onc(C)n2)=O)COCCN(C(=O)CCC2CC2C)C1 C1(CCC(=O)NCC2(NC(=O)C=C3CCSCC3)CCC2)CCC(O)CC1 CC(C)(O)CC(=O)NC(C1CCCC1)CN1CCN(C(C2C3CCCCC23)=O)CC1 Cc1ccncc1CNC(=O)NC1CC1.c12ccc(cc1)c(=O)[nH]2 C(C1=CCN(C(c2cc(C3CCCC3)no2)=O)CC1)NC(C(C(C)C)C)=O C12(CNC(C3CCCOC3)=O)CCCCC1N(c1ccc3c(n1)CCC3=O)CC2 C1(C(=O)OCC=Cc2ccco2)CCN(C(=O)Cc2cccs2)C(=O)C1 C1(C(N(CC(C)(C)CNC(=O)C(O)CC(C)(C)C)C)=O)CC2(CCOCC2)CO1 c1(-c2c(C(N3CCCC(NC(=O)CCC4CC4)C3)=O)c[nH]n2)ccccc1F C(=O)(C(C)(C)CN(C(c1cn(C)nc1I)C(=O)NCc1ccccc1)C)OC C1(C(N(C(CSC)C)C)=O)CN(C(=O)C(C)C2CCC2)CC1(C)C C(=O)(N=c1nc[nH]n2cccc12)C1(C)N(c2nc(SC)nc(C)c2Br)CC1 Fc1cc(F)c2c(-c3nc(C(C4CC4)C4CC4)nn3C3CCC3)onc2c1.C1CC1 C1(NC(C=CC=CC)=O)CN(C(=O)Cc2nccn2C)C2CC12 c1(C(C)C)n[nH]c(CNC(=O)C(O)CNC2CCCS2)n1 C1(n2cc(C(CC)O)nn2)CC2CCC(C1)N2C(=O)C(C)NC(=O)CO Cc1c(NCCC(C(F)F)N2CCOCC2)nc[nH]c1=NCc1cnoc1 C1(NC(C(C)Cc2ccccc2Cl)=O)CNCC2(CCC2)C1 c1(NC(=O)C(N2CCC(NC3CCCCC3)C2)=O)csc(C2CC2)c1 c1(C(C)C)nc(CN)sc1C(=O)NC1CCC(NCCn2ccnc2)C1 c1(Cn2c(CCC)nc(-c3ccc(OC)cn3)n2)cc(Cl)ccc1Cl c1(OC)cc(F)ccc1C(N1CC(CNC(=O)CCC2CC2(F)F)CC(C)C1)=O c1(OC)cccc2c1CCCC2NC(c1nc(C)cs1)Cc1ccccc1 C1(C(=O)Nc2ccc(CO)s2)CC2CC1CC2C(=O)NCC(O)C1(Cl)CC1 C1(C(N(C)CCNC(c2ccc(N)cc2F)=O)=O)CCOCC12CCC2 CC1CCC(NC(=O)CC2(O)CCCCCC2)CN1C(=O)Cc1cncs1 n1(CC(C)O)cc(CNC(C2CCC2F)=O)nn1 c1(CC)cc(Cl)sc1NC(c1cscc1OC)=O.C12(F)CN(C1)C2=O C1(C(N2CCN(C(C(C(C)C)(C)C)=O)C(CCO)C2)=O)CC2CCC1C21CC1 O=C1CCN(C(C2(CNC(=O)CCCC3CCCC3)CCCO2)=O)CCN1 C(C(=O)NOCCN1CCC1)(C1CCOCC1)NC(C1CCC(=O)N1)=O N1(C(c2c(C)cc(C#N)s2)=O)CCC2(C1)CN(C(c1cnccc1Br)=O)C2 N1(C(CC2CN(C)C2)=O)CCCC(n2cc(-c3ncccc3Cl)nn2)C1 C=CCN=C(NCC(C)Oc1ccc(Cl)cc1)NCC(C)(O)C1(C)CC1 N1(C(CN(C(c2cc(CC)n[nH]2)=O)CCO)=O)CC(O)CCC1C c1(C(=O)NC2(CC)CCOC2)cc(C)nc2ccc(C(F)(F)F)cc12 C1(CCO)(CC)CC(C(=O)N(C2(CC)CC2(F)F)C)C1.C1(=O)NN1 N1(C(c2c(C)cc(CNC(C3CC(C)(C)CCO3)=O)o2)=O)CCOCCC1C c1(OC)cc(Br)c(CNC(=O)CNC(c2cccc(N=[N+]=[N-])c2O)=O)cc1F N1(C=O)CCCC1.c1(C(=O)NCCCC2(N(C)C)CC2)coc(Br)n1 N1(C(COC)=O)CCN(CC(C)NC(=O)C(c2cccc(O)c2)C)CC1 C1(CC)CCCCC1OCCC(=O)NCC1CCCN(C(=O)CN(C)C(C)C)C1 C1(C(N2CCN(C)C(CO)C2)=O)CN(C(=O)C=CC2CCC2)CC(C)(C)C1 c1(NC(C(=O)NCC(C(C)C)N)=O)ccccc1C(F)F c1(NC(=O)NC2(CCCNC(CC)=O)CC2)ccc(Br)c(OC(F)F)c1 CC1CCC(C)(C(=O)NCCOC2CN(C(=O)CSc3n[nH]c(=N)s3)C2)CC1 N1(C(c2cnc(C)s2)=O)CCC(N=c2[nH]c(C(F)(F)F)nc3[nH]ccc23)C1 CC1(NC(c2ncoc2C2CC2)=O)CN(C(c2ccc(Cl)s2)=O)C1 C=CCCCC(C)N=c1nc(N2CCCC(n3cc(C)cn3)C2)c2c([nH]1)CSC2 C1(NC(=O)CCF)CCCCC1CNC(c1cccc(-c2cscn2)c1)=O C(CS(=O)(=O)C1CCCC1)C(N1C(C(N(OC)C)=O)CC(=O)C1)=O C1(N(C(c2c(C)cccc2)=O)C)CCCC2CN(C(c3cnc(S)n3C)=O)CC12 C1(C(=O)NC2CC(F)(CNC(CCCC(=O)NCC)=O)C2)CCc2c[nH]nc2C1 n1(CCCOC)c(N2CCC(C)(F)C2)nnc1CCN1CCN(C(C)=O)CC1 C1(C(=O)NC(CCC=C)C2CC2)CN(C(=O)C(=Cc2cn[nH]c2)C)CCC1(C)C C=CCCCC(C1CC1)NC(=O)C(c1ccccc1)N(C(=O)CC1CSCCO1)CC C1(C(=O)NCCOC)C(C2CC2)CCN1C(=O)C(CC1CCCC1)OC C1(C(=O)NC(C)CNC(C2(CF)CCC2)=O)CCCCN(C)C1=O c1(C(N2C(c3nc(C)[nH]n3)COCC2)C(=O)NC2CCC2)ccc2n[nH]cc2c1 N1(C(C(C)(C)N=[N+]=[N-])=O)C2CCC(C(=O)NCCC(=O)OCn3cnnn3)C1CC2 c1(OC)ccc2c(C(N3CC(C4CN(S(=O)(=O)CC(C)C)C4)C3)=O)coc2c1C C1(CCNC(=O)OC(C)(C)C)(NC(C2CCOC2C(F)F)=O)CC(F)(F)C1 C(=O)(CCN(CCCF)C(=O)C=CC=C(Cl)Cl)OC C1(CNC(CCc2ccc(C)s2)=O)CCCCC1NC(c1ccoc1)=O c1(NC(=O)NC2(CC)CCCC2)cc(F)ccc1CSc1ccccc1 Cc1cc(C(=O)OC(c2ccc(F)cc2C)C)c(F)cc1Cl c1(C(N2CC(OCCOC)C2)=O)cc(C)nnc1NC.C1CCC(=O)N1 c1(C(N(CCCNC(CC2CC(C)C2)=O)C)=O)ccc2cnn(C)c2c1 C(CN=c1cc[nH]cc1C#N)(C(C)(C)C)NC(C(C(C)C)C)=O N1(C(c2ccc(N(C)C)cc2)=O)CC2CCN(C(=O)Cc3ccc(Cl)nc3)CC12 C(C(=O)N1CC(N(C(=O)C(F)(F)C2CCCCC2)C)C1)(C(C)C)OCC(C)C N1(C(CN(CCC)C(C2CCOC2(C)C)=O)=O)CCC2(CC2)C1 C1(CNC(C=CC(C)C)=O)CN(C(C2CCNC2=O)=O)CC12CCC2 CC1(NC(c2nnnn2C2CCOC2)CC2CCC2)CCSC1 N1(C(CCn2ncc(C)c2)=O)CCC(F)(C(=O)NC(c2cccnc2)C(C)C)C1 CN=c1nc(NCC2CC3(CCC3)C2C(F)(F)F)[nH]c(N2CC3CC3C2)n1 C(=O)(C(C)C(F)(F)F)N1CC(OC(CC)C(=O)NC2CCCCC2)C1 Cc1oc(C)c(C(=O)NC2CCC(NC(c3ccn(C)c(=O)c3)=O)CC2)c1C N1(C(c2c(C)nns2)=O)CCC2CN(C(c3ccnnc3)=O)CCC2C1 Cc1nn(C)c(C(=O)NC2CC3(C2)CN(C(=O)C(O)C2CCCC2)C3)c1Br N1(C(COC)=O)CCCN(C(=O)C=Cc2cc(Br)ccc2F)C(CO)C1 N1(C(C2(C#N)CCC2)=O)CCC2CN(C(=O)C3CCc4c[nH]nc43)CCC2C1 C12CCN(CC1)C(=O)C1(CC1)N(C)C(=O)CNC(=O)CC2.C(C)(C)(C)N(C)C C1(NC(C(C)OCc2ccccc2Cl)=O)CCC12CN(C(C1CC(C)(O)C1)=O)C2 Cn1ccc(=O)c(C(N2CCOC(CNC(C3CC4(CCO3)CC4)=O)C2)=O)c1 c1(NC(C(=O)Nc2ccc(CCOC)c(Cl)c2)=O)cnn2c1OCCC2 C1(C(=O)NC(CC2CN(C(c3c(OC)scc3)=O)C2)C)CC12CCOCC2 c1(C(N2CCC(CCC(=O)NCC(C(=O)NC)O)C2)=O)cccc(O)c1C C1(NC(CCC(C)NC(c2cc(C)ncc2)=O)=O)CCc2nn[nH]c2C1 c1(C(=O)N(C2(c3ncc(C)[nH]3)CCOC2)C2CC2)ccc(Br)cc1F Cc1nc2ccc(C(=O)NC3CCN(C(c4nc(=N)cc[nH]4)=O)C3)cn2n1 C1(C(C)NC(C(C)CF)=O)CCN(C(=O)CC2CCCCN2C)CC1 C1(C(=O)NCCC2(NC(C3CC(CF)C3)=O)CC2)C2COCC12 C1(C(=O)Nc2cccc(F)c2)CC(C)CN(C(c2c(OC(C)C)cccn2)=O)C1 C1(F)(C(=O)NCC(C)N(C(c2cn(C)[nH]c2=N)=O)CC)CCS(=O)(=O)C1 C1(C(=O)NCCCN(C(=O)CSc2ccccc2F)CC)CCCCC1(C)C CS(=O)(=O)CC(=O)NC1CCC(CCNC(c2ccc(CO)o2)=O)C1 c1(C(N2CC(N(C(C(C)Cn3cccn3)=O)C)C2)=O)ccc2[nH]ccc2n1 N1(CC(=O)NCC(C)N(C(C2C(C=C)C2)=O)C)C(=O)c2cccnc2C1=O c1(OC)ccnc(CN2CC3C(NC(=O)CCc4ccnc(Cl)c4)C3C2)c1 CC#CCC(C)N=c1nc2c(ncn2C)c(NC2CCC3(CC3)C2)[nH]1 C(=O)(C(C)(F)C(=O)NCCN1CCC(NC(=O)C(C)(C)CC)CC1)OCC CC(C)CC(CNC(C1CCCS1)=O)NC(=O)C(C(C)C)c1ccccc1 c1(C(N2C(C)(C(N(C3CCN(C4CC4)C3)C)=O)C=CC2)=O)ccc2nccn2c1 C=CCCC(C)NC(c1conc1C(C)NC(=O)C=CC1CCOC1)=O CC(CNC(=O)COC1CCCOC1)N=c1c([N+](=O)[O-])c[nH]c2c(Cl)cccc12 c1(NC(C(=O)N(CCCC)C(C)CC)C)cccc([N+](=O)[O-])c1 CC1C(C(=O)NCCCc2ncco2)CCN1C(=O)C=CC(C)(C)C N1(C(C2N(C)CCOC2)=O)CC2CC(NC(C3CC(=O)NC3(C)C)=O)CC1C2 N1(C2C(C(=O)OCC)C2(C)C)CCN(C)C(CNC(=O)OC(C)(C)C)C1 C1(CN(C(C=CC=CC)=O)C)CCCN(C(C2(C#N)CC(C)C2)=O)C1 C1(C(=O)NC2(C3N(C(C(CC4CCC4)OC)=O)CCC3)CC2)CCS(=O)CC1 CCCC(C)(O)CC(=O)N1CCC(CNC(c2cnc3occc3c2)=O)CC1 Cc1ccc2cc(C(N(C)CC3CN(CCOc4ccccc4)C3)=O)sc2c1 C1(COC)CC(CNC(c2cnn(CCO)c2)=O)N(C(=O)C=CC(C)CC)C1 C1(NC(=O)C=Cc2ccco2)CC(NC(=O)CCOC2CCOCC2)CC1O c1(C(=O)NCC(CC)NC(CC(C=C)CC)=O)nc(C(F)(F)F)n2ccncc12 c1(CCC)cc(C(=O)N(CC(C)NC(=O)CCCOC2CC2)C)nn1C C=CCCCCC(=O)NCc1ccsc1C(=O)N(C)CC1CCOC1 c1(OC)cc(C(C)CC(=O)N2CC(F)(CNC(C3(C)CC(C)C3)=O)C2)ccc1C C=C1CCN(C(c2ccc(C)cc2F)=O)C(C(N2CCCC(N3CCC3)C2)=O)C1 C1(c2nc(C3N=C(C)SC3)on2)CN(n2cc(C3CCCC(O)C3)nn2)CC1C C(c1ccncc1C)=CC(=O)NCCC1CCN(C(C(C)NC(CC)=O)=O)C1 N1(C(C(CCC#C)O)=O)CCC2(CC1)CN(C(=O)CSc1nnc(S)s1)C2 c1(C(N2C(C3CCN(C(CCC=C(C)C)=O)C3)CCC2)=O)ccc(S(C)=O)cc1 Cc1nn(CC(=O)NC2(CC(=O)N(C)C(c3ccccn3)C)CCC2)cn1 C(=O)(C#CC1(C)COC1)NC(C(C)NC(c1sc(C)c(O)n1)=O)C Nc1cccc(C#CC(=O)NCC2CC2(F)Cl)n1 c1(OC)ccc(CC(=O)NC2CC(CCNC(c3ccnnc3O)=O)C2)cc1Cl C(=O)(CC(F)(F)C(C)(F)F)N(CCN(C(=O)CCS(C)=O)C)C c1(C(=O)NCC2CC(F)(CNC(c3sccc3Cl)=O)C2)cc(Cl)c(F)cc1F C1(C#N)(C(=O)NCCC(C)N(C(=O)CCc2c(Cl)cncc2Cl)C)CC2CC2C1 N1(c2cc(NC(CNC(=O)OC)C)nc(C)n2)Cc2cnn(C)c2C1 Cc1nccc(N(C(=O)CCC(C)N(C)C)C)n1 C1(CNC(C(CC)OCC)=O)CN(C)CCN1C(c1ccnc(Cl)c1N)=O N1(C(C2CCN(C)C2=O)=O)CCC(C=CC(=O)NCCC(=O)N(C)C)CC1 C(CC(=O)NC1CCCC(C)(C)C1)(C(C)C)NC(C1(OC)CCOC1)=O CCCS(=O)(=O)C(C)C(=O)N1CC2CCC(C1)N2C(c1c[nH]cc(Br)c1=N)=O Cn1nc2c(c1C(N1CCC(NC(=O)CC3CCNC(=O)C3)CC1)=O)CSCC2 C1(C)(NC(=O)NCCC2(NS(C(C)C)(=O)=O)CCC2)CCOC12CC2(F)F c1(NC(c2c(C(C)NC(C(C(C(C)C)O)C)=O)noc2)=O)ccc2nccn2c1 N1(C(c2c(C)nc(O)cc2)=O)CCC2(CCCN2C(=O)C2=NOC(C)C2C)C1 CC(C)C(O)C(F)(F)C(=O)NCCCC(C)(C)NC(=O)C(C)C(C)(C)C c1(C(N(C(CNC(CCC=CC)=O)C)C)=O)cnc2ncnn2c1O C1(CC(NOCCCC)=O)CN(C(=O)CC(C)C2CC2)CC12CC2 C1(NC(CC)=O)COC2(CN(C(=O)C(C)NC(C)(C)CC)CC)CC1C2 c1(C(=O)NC(C(C)C)CNC(=O)C(C)CO)ccc(OCC(F)F)nc1 c1(C(N(C(c2ccc(O)cc2)C)C)=O)ccc(NCCO)nc1 c1(OC)ccc(C(=O)NCC(O)CNC(C2CNC(=O)N2)=O)c(Br)c1F C(=O)(CCCCC(C)(C)C)N1CCC(CNC(C(CCC#C)O)=O)C1 N1(C(C)=O)CCOCC1C(=O)NCC(C1CCCC1)NC(=O)CN(C)C(N)=O Cc1c(C(=O)NCc2ccccc2CN(C(=O)CC(C)(C)O)C)nn(C)c1N Cc1ccc(CN2CCC(O)C(C(=O)NCc3ccoc3)C2)c(Cl)c1Cl N1(C(C)C)C(=O)CCC1C(=O)N(CCCSc1cccc(F)c1)C CC1(C)COCC(C(N2CCC(NC(c3ccc(C#N)s3)=O)C2)=O)O1 N1(Cc2cccc(C#C)c2)CC=C(CCNC(c2cc3c[nH]nc3s2)=O)CC1 C(=O)(CC(C)C(C)C)N1CCC(CNC(C(C(C)C)C2CCC2)=O)(CO)C1 c1(N(C)C(=O)NC2CC2)ncc(Cc2ccnn2CC2CCCC2)s1 Cc1ccnc2c(C(=O)NCC3(Nc4ncnc(C)c4F)CCC3)cccc12 C(CNC(c1ccc(C2CCC2)cc1)=O)(CC(C)C)NC(C=CC=CCC)=O c1(CC)nc(S(=O)(=O)NC2CC(c3cccc(C)c3)(O)C2)cn1CC N1(C(C2CCCC2)CNC(=O)OC(C)(F)F)Cc2ccccc2C1 C(CN=c1nc(N2CCSC(C)C2)c2cccc(F)c2[nH]1)c1c(C)n[nH]c1 CC(C)CC(C(=O)NCC1CCC(=O)N1)ONC(=O)CC1(C#N)CC1 CC1CCN(C(=O)Cc2ccc(Cl)s2)C1CNC(=O)COCC1CCCO1 S(=O)(=O)(c1c[nH]ccc1=NCCC1CCC(=O)CC1)NC1CCN(C(C)(C)C)C1 C1(NC(CCSc2ccc(C)cc2)=O)CN(C(=O)Cc2nc(C)cs2)CC1(C)C C1(NC(c2ccc(NCCO)cc2)=O)CNCCC12CCC2 c1(C(=O)NC(C2C(C(=O)NCC(COC)O)C2)C)coc(=N)[nH]1 C1(NC(c2c(CC)cccc2F)=O)COc2nccnc2C1 c1(N2C(C)CN(Cc3nccn3C)CC2)ncnc2ccccc12 C1(C(N2CC3(C2)CN(C(C2(CO)COC2)=O)C3)=O)CC2(CCOCC2)CO1 C=CC(CC)C(=O)NC(C1(O)CCN(C(=O)CSCC(N)=O)C1)COC N1(C(CCC(=C)C)=O)CC2(CNC(C3CC(O)(C#N)C3)=O)CCC1CC2 C1(C(=O)NCCNC(C(=O)NCCOCCCC)=O)CCCCCS1(=O)=O Cc1nc2cc(C(=O)NC3CC3CNC(=O)C3=COCCC3)cnc2s1 CC12CN(C(c3nn[nH]c3Cl)=O)CC1CN(C(C1(CO)CC1(F)F)=O)C2 C1(c2nnnn2CCCOC)(NC(c2cccc(Cl)c2)CC)CCN(C)C1 N1(C(Cc2cc(C)no2)=O)CCC2CN(C(c3ccc(F)c(F)c3N)=O)C2C1 C12(C(=O)NCCNC(C(C)OC3CCCCC3)=O)CCCCC(=O)N1CCC2 C1(NC(CC(C2CC2)NC(C(C)(C)Cl)=O)=O)CCOCC1F c1(CCC)cc(C(=O)NCCCC(C)(C)NC(=O)CCOC(C)=O)sc1C c1(CC)cc(C(=O)NCc2nocc2C(=O)NCC2CCCOC2)ns1 N1(C(c2c(OC)ccc(OC)c2)=O)CC2CCC(C1)N2C(C1CSCCS1)=O CC(C(=O)NCc1ncoc1C1CN(C(=O)Cc2ccc(O)cn2)C1)C(C)(C)C CC1c2cc(F)ccc2CCN1C(=O)CNC1CCC(Oc2ccccc2)CC1 C(=O)(CS(N)(=O)=O)N(CCNC(Cc1cc(C)no1)=O)C1CC1 c1(C(=O)NC2CC(NC(CCc3c(C)ncs3)=O)C2)cc(=O)cc[nH]1 CCCC(C)(C)CC(=O)NC(COCC)C(N1CCCCC1C(=O)OC)=O CCCCCCCC(=O)N1CC(OCCC(=O)NCC2CCCSC2C)C1 C12(C(=O)NCC(CC(C)C)NC(C3(CC4CC4)CCC3)=O)CCC(CC1)CC2 c1(C(N2CC(O)(C(C)NC(C(C)CC(F)F)=O)C2)=O)ccc2c(c1)OCCN2 c1(C2CCN(C(c3csc(Cl)n3)C(=O)NC)C2)nc2ccccc2s1 C1(NC(c2ccc(C(=O)OC)o2)=O)COCCC1NC(C1C=CCCC1)=O CC(C)C(O)CC(=O)N(CC(C)CNC(c1ccccc1CO)=O)C C1(NC(C(F)(F)C2(OC)CCC2)=O)CCN(C(=O)CSC2CC2)C(C)C1 N1(C(CC(C=C)C)=O)CC(NC(c2coc(SC)c2)=O)CC2(CC2)C1 C1(C(=O)NC2CC(NC(c3c(COC)nn[nH]3)=O)C2)CCC(CC(C)OC)CC1 C1(C(=O)NC2CC(NC(C3C(C)OCCC3)=O)CC2O)Cc2nccnc2C1 C1(CCNC(C(CC)F)=O)CC(F)(F)CN1C(c1cc(C)cc(Cl)c1)=O C1(C(F)(F)F)(CNC(=O)OC)CCCN1C(C1C2CN(c3ccccc3C)CC12)=O N1(C(C#CC(=O)N(C)C)=O)CCC2CC(CNC(C3CCS3(=O)=O)=O)CCC2C1 C(=O)(CC1=NNC(=O)C1)NCCCC(CCC)NC(C1(F)CC1C)=O C1(NC(=O)C=C(C2CC2)C2CC2)CC2(CCCN(C(=O)CC3CCSC3)C2)C1 C=CCCCN=C(NCc1n[nH]cc1C(C)C)NC1CCOC1 C(CCN=C(NCCC1CC1(F)F)N1CCC(c2cccnc2)C1)OC C1(NC(CCC#CC)=O)COC2(CCN(C(=O)C(O)CC[S+](C)C)CC2)C1 c1(OC)ccc(C(=O)NCCCC2CCN(C(C3CC3(F)Cl)=O)CC2)nn1 C(C(CC(C)C)C(=O)NOCC(C)C)NC(C=CCCC)=O C1(C(N(CC(CN(C(C2CCC(CC)O2)=O)C)O)C)=O)CCc2nccn2C1 C1(C(=O)NCCCN(C(C(CC)n2ccnc2)=O)CCO)CCCC2(CCC2)O1 c1(C(=O)NC2(C)CC(NC(CC3CC(=C)C3)=O)C2)cnn(C)c1Cl n1(CC)cc(CC(=O)NCc2csc(C(=O)NCC3CSC3)c2)cn1 Cc1nc(C)c(C(CC)C)c(O)n1.N12CCOCC1C2=O.C1CC(F)C1.C1C(=O)NC1 CCC(C)(CC)C(=O)NC(C1CCCCC1)CNC(=O)CCc1cn(C)cn1 C1(NC(=O)C(c2ccc(Cl)cc2)=O)CC(NC(C23CC(C2)C3)=O)C12CCC2 Cc1nc(NCC2CCCC(NC(c3ccc(C4COC4)cc3)=O)C2)ncc1Br N1(C(c2cc(CNC(=O)C3=COCC3)no2)=O)C2CCCC1CC2 C1(CNC2CCCN(CC)C2)CC2(CCN(S(=O)(=O)CCC3CCC3)CC2)CO1 C(=O)(C(C)C(C)NC(=O)CNC(c1coc(C(C2CC2C)=O)c1)=O)OCC S(=O)(=O)(c1cccs1)N(C(=O)CCCN1C(=O)CNC1=O)C C1(CC)CCN(C(=O)C=CCC(C)(C)NC(=O)C(C)C2CCCC2)CCO1 c1(C(=O)NCCCC(C)NC(C=CC=CCC)=O)ncnc2c1ccn2C CCC(C)C(O)C(=O)NC1CCCC1CNC(c1cc(C2(C)CC2)on1)=O c1(CC(N2CC(NC(C(C)C)=O)C(C)CC2)=O)csc2c(Cl)cccc12 C(N=c1[nH]c(=NCC2CCCSC2)c2cccc(F)c2[nH]1)C1(C)NC(=O)NC1=O C1(C(=O)NC2C3CN(C(C(C)OCC)=O)C2C3)CC2(C1)CS(=O)(=O)C2 C(=O)(C1CCCc2ccnn21)N1CCN(C(CS(C)(=O)=O)=O)C2C1CCC2 C(CCOCCC)(C(N)=O)NC(CNC(CC1(OCC#C)CC1)=O)=O c1(-c2n(-c3ccc(C)c(C)c3)nc(-c3ccoc3C)n2)coc2c(Cl)cccc12 C=CC(C)(O)C(=O)N1CCN(CC(n2cc(-c3csc(C)n3)nn2)N(C)C)CC1 C1(C(C(C)CNC(=O)C=CC(=O)N(CC(F)(F)F)C)=O)CCCN1C1CCCC1 c1(CC)c(C(=O)NCCCCC(C)(C)NC(C2CC(C)N(C)C2)=O)cccc1F c1(N(C)C)nc(C(=O)N(C2CCN(C(c3cccc(F)c3Cl)=O)C2)C)[nH]c(=N)n1 C1(C2CCN(C(=O)CC3CCCO3)CC2)(NC(=O)CC2CCCCC2O)CCC1 C#Cc1ccc(C(c2nnnn2CC2CCOCC2)NC2(C(=O)OC)CC2)cc1 N1(C(C(C)(C)N2CCNCC2)=O)CCC2(CCCCC2C(=O)O)C1 c1(CC(=O)NC2CC3CC(NC(=O)Cc4csnn4)C2C3)c[nH]c2ncccc12 C(=O)(N=c1[nH]nc(Cl)s1)C1N(C(c2cnccc2OCC)=O)CCC(O)C1 C1(C(=O)NC(CCC)CC)C2CCCC2N1C(=O)CC1CC1NC(=O)CCC C1(C(C)O)COCCN1C(c1ccc(CNC(=O)C(N2CCOC2=O)C)o1)=O CON(C(=O)C1OCCC1CNC(=O)C(C1CCCCC1)O)C1CCC1 CC(C)CCCC(=O)NC(CO)C(N1CCCC(N2CCC2)C1)=O C(CN=c1[nH]c(N2CCCCC3(CCC3)C2)nc(=N)[nH]1)=CCCC c1(C(N(C(C)C)CCN(C)C(C2(S(C)(=O)=O)CC2)=O)=O)cc2ccc(F)cc2o1 c1(C(N2C(CC)CN(C(C3OCC3(C)C)=O)CC2)=O)oc2ccccc2c1Br C1(F)(CNC(=O)CN2CCOCC2)CCCN(C(=O)CCn2cc(Cl)cn2)CC1 c1(CC)c(C(N2CC(NC(=O)CCOCC(F)F)CC(O)C2)=O)cccc1F c1(CNC(=O)NC(c2ccccn2)CC)cnccc1C Cc1cccc(NC(C2(C(=O)NCC3(CNC(=O)C=C4CC4)CCC3)CC2)=O)c1 c1(C(N2C3C(NC(C(C)N(C)C)=O)C(CC3O)C2)=O)c[nH]c2cc(F)ccc12 N1(C(CC)=O)CCC(C(=O)N(CCNC(c2nnsc2C(F)F)=O)CC)C1 CCCC(CCNC(C1CC(C)(C)CN1C(=O)COCCCOC)=O)CCC c1(C(N2CCCC(CCNC(C(CCSC)O)=O)C2)=O)c[nH]c(=N)c2[nH]ccc12 C(=O)(CC1C(=O)Nc2ccccc21)N1CCC(N(C(C2(Br)CC2)=O)CC)C1 N12CCC(C(CC)C1)C(=O)NC(C)C2=O.C12(C(=O)NCC#C)CC(C)(C1)C2.CC#C Cc1cc(C(N2CCC(NC(C3CC(CCO)C3)=O)C2)=O)c(Cl)cn1 N1(C(CC(=O)OCC)=O)CCN(C(=O)Cc2cccc(C3CC3)c2)CC1CO Cc1cc(=N)[nH]cc1C(=O)NC1CC(N(C)C(C23CCC2C3)=O)C1 Cc1nc2cc(C(N3CCC(F)(C(N4CCC(C(N)=S)CC4)=O)C3)=O)ccc2s1 C1(CC(N2CC(N3CCCC3)C2)=O)CC2(C1)CN(C(c1ccc3c(c1)CC3)=O)C2 Cn1nc(C2CC2)nc1CC(=O)NCC1CCCCC1NC(=O)C(O)C1CC1 c1(C(N2C(C)(C(=O)NCc3cccc(C)n3)CCC2)=O)ccc(Br)cc1CO N1(C(c2ccc(O)nc2)=O)CCOC(C(N2CCC(O)C2)=O)C1 CC1(C)CC(C)(CNC(C2CCCN2C(N)=O)=O)C1.O(N)C c1(C(N2CCCC(CCNC(Cc3cn(C)nc3)=O)C2)=O)coc2c1CCCC2 CCCC(C(=O)OC)C(=O)N1CC2CN(C(c3cccc(C(N)=O)n3)=O)CC2C1 N1(C(C2(C=C)CC2)=O)CCC2CCC(NC(C3CCC(=O)N(C(C)C)C3)=O)C1C2 C1(NC(C=CC)=O)CC(OC)C12CCN(C(=O)Cn1nc(Cl)ccc1=O)CC2 C1(CCC)(NC(=O)CC(=O)NC)CCCN(C(C2CN(CC(C)C)C2)=O)C1 C1(C(=O)NCCC2CC=CCC2)(CNC(C(C)=C(C)C)=O)CCCO1 C(=O)(CCC(=O)OC(C)(C)C)NC1CC(C)(NC(C2CC2(C)C)=O)C1 c1(OC)cc2c(cc1CNC(=O)CSCc1ccc(C(C)C)nc1)OC(C)C2 C1(C(=O)N(C2(COC)CCOC2)C)(CF)CC(F)(F)C1 C1(C)(CC(=O)NCC2CC(C(C)C)C2)CCN(C(=O)C(N2CCCCC2)C)C1 CCS(=O)(=O)CC(=O)NC1CC2CC(NC(=O)CC3CCC(C)(C)C3)C1C2 CC(C(=O)NC1CN(C(=O)CCC(C)(C)C)C2(CCCC2)C1)C(F)(F)C(F)F c1(C(=O)NCC2N(CC)CC2)ccnc(CNC(=O)CC(C)(C)O)c1 O=S(=O)(c1ccc(N2Cc3c[nH]c(=N)nc3C2)nc1)N1CC2CCOC2C1 C(C)(c1ccccc1F)=CC(N1CCN(C(C(C)OC)=O)C(c2cn[nH]c2)C1)=O Cc1cccc(S(=O)(=O)N2CCCC2CC(=O)NCc2nccc(Cl)c2F)c1 Cc1ccc(OCCC(=O)NCC(C)NC(c2cccnc2S)=O)c(C)c1 C1(CNC(C2(CC=C)CC2)=O)CN(C(=O)CC(C)O)CCC12CCOCC2 N1(C(c2c(C)csc2)=O)CCCC2(CCN(C(C3(F)CC=CCC3)=O)C2)C1 N1(C(C2(O)CCN(C(c3nn[nH]c3C(F)(F)F)=O)C2)=O)CCCC(F)(F)C(F)C1 c12cc(Cl)cc(c1O)C(=O)N1C(CC(=C)C1)C(=O)N2.c1(COC)cnccc1C C=CC1(C(=O)NCCc2cnc(C)o2)CCN(C(c2cnc(OC)cn2)=O)C1 CN1CCC(C(=O)NCCC(O)C2CCC2)(NC(c2ccc(=N)[nH]n2)=O)C1 N1(C(C(N2C(CCNC(=O)Cn3cnnn3)CCC2)=O)=O)CCC(C)CC1.CC Cc1nn(-c2ccc(F)cc2)nc1C(=O)NCC1CCN1C(c1n[nH]cc1F)=O CC1CCN(C(=O)C=C(Cl)Cl)C1CN(C)C.c1(C(=O)NC)ccc(C)[nH]1 c1(C(N(C)CCNC(=O)CCOC2CCOC2)=O)cccc(-n2ccnn2)c1 N1(C(c2cccc(COC)c2)=O)CCN(C(c2ccoc2Cl)=O)C(C2CCC2)C1 C1(NC(C2(CC#C)CCCC2)=O)CN(C(=O)CC2CC(C)=NO2)CC1C C(CCC(O)C(=O)NCCC1CC(O)C1)NC(C1C(CCC)C1)=O C(=O)(C(C(C)NC(=O)CCCC(C)C)C(C)C)NCC(COCC)O CC(C)CCN=C(NC1CCCC1)NCC1(CNC(=O)OC(C)(C)C)CCC1 n1(CC)ncc(C(=O)NC2CCCC2(C)CNC(C2CC2(C)C)=O)c1Cl C(=O)(CC(C)C(=O)NC(C)CCNC(c1ccccc1C1(C)CC1)=O)OCC c1(COC)ccc(C(N2CC(C(=O)NCCOC(C)CCSC)C2)=O)cc1 N1(C(C2C(C)C2C)=O)CCCC2(NC(c3cccc(C(N)=O)c3)=O)CCCC12 c1(NC(C2N(C(CP(C)(C)=O)=O)CCC(O)C2)=O)cccc2c1CCO2 N1(C(c2cccc(Br)c2OC)C(=O)NCCC)CCOc2cccc(Cl)c21 C(=O)(C(O)C(F)(F)C(F)(F)F)NCC(C1CCN(C(CC=CC)=O)CC1)(C)O N1(C(C2CCC(C(=O)NC3(CC)CC3)C2)=O)CCc2c(O)n[nH]c2C1 N1(C(C)=O)CC2CC3CC2C1C3NC(c1cc(Cl)c(Cl)c([N+](=O)[O-])c1)=O C1(C(=O)NCCCNC(CC)=O)CC(C)(C)O1 C(=O)(C(F)(F)F)NC(C)C(=O)NCC1CC(NC(C2CCCN2C)=O)C1 c1(C(N2C(C)CN(C(C3CC4(CC4)CO3)=O)CCC2)=O)ncnc2c1CCCC2 Cc1cc(C(F)F)oc1C(=O)NC(C)CCNC(=O)C(C)(C)c1cc[nH]n1 c1(C(N(CC(C)NC(CSCC(=C)C)=O)C)=O)ccc(OCC)cc1 C1(CN2CCN(C)CC2)(CO)CCCN(C(=O)Cn2ccc(C3CC3)n2)C1 C1(C(=O)NCC2(C(C)(C)O)CN(C(C(C(C)C)OC)=O)C2)CC2(CCOCC2)C1 Cc1cccc(C(=O)NCC2OCCC2C(=O)NCCC2CC2)n1 C1(CC)CC2(CCC2)CN1C(C(=O)NC1CCOCC1)C1CC1(C)Br N1(C(c2c(OC)c[nH]n2)=O)CCN(C(=O)Cc2c(F)cncc2Cl)CC1CCO N1(C(C2(C)CC(C#N)C2)=O)CCC2(CC1)CC2CNC(c1ccc(=O)oc1)=O c1(NC)ccc(C(N2CCC3(CC3C(=O)NCC3(F)CCCCC3)C2)=O)c(F)c1 C(=O)(C1=CC2(CCOC2)C1)NCC(CNC(C1C(C)(C)CCC1)=O)O C(CC(C)NC(=O)CO)NC(CSCC#C)=O C(=O)(C(C(C)C)C(C)C)NCC1CCN(c2nnc(C)o2)CC1C C1(NC(c2cnc(SC)s2)=O)CCCCC1CNC(c1ccc(C)n1C)=O C1(NC(CC=C)=O)CN(C(c2c(C(F)(F)F)cccc2O)=O)CC12CCOCC2 c1(CNC(c2cc(Cl)c(Cl)[nH]2)=O)cnn2c1CN(C(C13CCCCC1C3)=O)CC2 N1(C(C2C(NC(C)=O)CC2)=O)CCC2C(O)C(C)(C)C12 C1(NC(C2CC(C)SCC2)=O)CC2(CCN(C(=O)CC3COCCN3C)C2)C1 C1C(C)C(=O)N1.N1(CCNC(C(C2CCCC2)OC)=O)CC2CC2C1 c12nnc(n1C(C1CCNCC1)C)SC2C.c1(CN2CC(C)C2)ccccc1 N1(C(c2c(F)cccc2F)=O)CCC2CN(C(=O)C(c3cccnc3)O)CC2C1 C=CCC(CC(=O)NCc1cnccc1Cl)NC(=O)C(C)S(C)(=O)=O c1(CC(=O)NC(CNC(CC=C=C)=O)C2CCC2)c[nH]c2cc(C)ccc12 N1(C(C=CC)=O)CCC(NC(=O)C(c2ccc(C)cc2)C)C(CO)C1 c1(CC(=O)NC2(C)CC(N(C(C(C)=C(C)C)=O)CCCC)C2)cccc(Cl)c1F C1(C(=O)NCCN2CCN(C(CCC(CC)C)=O)CC2)CCn2ncnc2C1 N1(C(C2C(CC)CC2)=O)CC23CCCC2(C1)CN(C(=O)C(C)(C)c1ccn(C)n1)C3 C1(C(=O)NC2CCCN(C(C3(C)CC3(Cl)Cl)=O)C2)CCCS(=O)(=O)C1 c1(C(=O)NCC2(CNC(C(c3n(C)ncc3)O)=O)CCC2)ccc(C#N)o1 N1(C(c2cn(C)cn2)C(=O)Nc2ccc(OC)cc2C)CCn2ncc(Cl)c2C1 N1(C(C(C)C2CCCO2)=O)CCOC2(CCc3ccccc32)C1 C1(NC(C(CCC)OCC)=O)CC2(CCCCN2C(c2ccsc2)=O)C1 N1(C(C2CC(=C)C2)=O)CC23CCCCC2(C1)CN(C(c1ccc(F)cc1Cl)=O)C3 c1(CCC(=O)NCC2CCCCCN2C(C2CCSC2)=O)ccc2ncsc2c1 CC1CCN(C(c2cc(CNC(=O)C(C3CC3)C3CC3)no2)=O)CCO1 CC(CC(=O)N1CCC(O)(CCNC(c2cnc(O)o2)=O)C1)C(C)(C)C C1(CNC(c2n(CC)ncc2C)=O)CN(C(=O)OC(C)(C)C)C(C)(C)C1 N1(S(=O)(=O)c2cccnc2N2CCC=C(Cl)C2)CCC2CC(O)CCC2C1 C1(C)(C(=O)NCCCCC(C)NC(C2CC3C=CC2C3)=O)COC(C)CO1 C(CNC(c1ccc(Cl)s1)=O)(C(C)(C)C)NC(c1ccc(C)s1)=O C1(C(N2CC(CC)N(C(C3CC4(C3)CC(F)C4)=O)CC2)=O)CCCCN(C)C1=O Cc1cc(C(F)(F)F)ccc1C(N1CCOC(CNC(=O)C2=NNC(=O)C2)C1)=O C1(NC(c2cc(C)c(C)nc2)=O)CC(C(=O)NC2CC23CCCCC3)=CC1O CC(CN1CCCC1=O)CN=c1nc(N2CCOCC2)[nH]c2ccccc12 Cc1ccnn1C(C)C(=O)N(CC(N1CC(n2ccnc2)C1)=O)C1CC1 N#Cc1cc(Cl)c(C(=O)Nc2cccc(CNC(=O)CNS(N)(=O)=O)c2)s1 C1(C(=O)NCC2CC(N3CCCC3)C2)CC2CCC(C1)N2C(c1csc(Cl)n1)=O N1(C(C(C)OCC#C)=O)CCC(NC(c2ccncn2)=O)C(CO)CC1 C1(Cc2n(-c3ccc(C)cc3)nc(-c3ccsc3)n2)COCCN(S(C)(=O)=O)C1 C1(N(C(=O)C=CC2CCC2)C)CCN(c2ncccn2)CC1 C12(N(CC(C(=O)OC)C)C(=O)OC(C)(C)C)CCC1CN(C(=O)C1=CCC1)C2 C(C(COC)CC(=O)NCC(C)(O)CNC(c1cnn(C(C)C)c1Cl)=O)OC c1(C(N2CC(CNC(COCCC#C)=O)C2)=O)ccc(Cl)cn1 c1(OCCC(=O)NCCCCCNC(CCCCOCC)=O)c(C)nn(C)c1C N1(C(C(C)N(CC)CC)=O)CCC(CNC(=O)C(C)NC(=O)OC)C1.CF c1(OC)ccsc1C(=O)NCC1CC(CC2CC2)C1.C12CC(C1)CNC2=O C1(CNC(CC(=O)NCC)=O)CC(C(C)(C)O)CN(C(C2(C)CC2)=O)C1 Cc1nc(N2CCCC(C(=O)NCC(F)F)C2)sc1C#N c1(C2(CC(=O)NCC3N(C(C(COC)C)=O)CCC3)CC2)ccc(OC)cc1C N1(C(c2c(Cl)c(C)n(C)n2)=O)C2CCC1CC(CNC(C1C3CCCCC13)=O)C2 O=C1CCCCN1CC(N1CC2CC1(C(=O)NCC1CCCO1)C2)=O N1(C(C=CSC)=O)CC(CNC(c2ccc(C)cc2F)=O)CCC1C C1(C(N2C(CCCC)CCC2)=O)CC12CC(NC(C1COCCC1C)=O)C2 N1(CCC(=O)NCCC(C(=O)NC)(C)C)C(=O)C2CC=CCC2C1=O C1(C=O)Cc2ccccc2N(C(=O)CCC2CC2(Cl)Cl)C1C(=O)O c1(SC)cscc1C(=O)NC1CCCC1CNC(c1cc(C)ns1)=O C1(CC(=O)NCCCCC2C(C)C2)CC(NC(c2cnn(C(F)F)c2)=O)C1(C)C C1(NC(c2cc(C)n(C)n2)=O)CN(C(=O)C(O)Cc2ccccc2)CCC1F N1(C(Cc2nc(C)[nH]n2)=O)CCCC2(C1)CN(C(=O)C(C#N)C(C)C)C2 c1(C(N2C3CN(C(c4c(OC)cccc4OC)=O)CC32)=O)nc2ccccc2s1 c1(C(N2CC(OC(N)=O)C2)=O)ccnc2c1CCO2.N12CCCC1CNC(=O)C2 O=C(C1CCCc2scnc21)NC1CC2CCC(C1)N2C(C1CCCS1(=O)=O)=O Cc1c(C(N2CCC(CCC(=O)NC(C)CC(F)(F)F)C2)=O)ncn1C C1(OC)COCC1n1cc(C(N(CC(N2CCCC2)=O)C(=O)C2CC2)C2CC2)nn1 N1(C(C2CCC(C)(C)C2)=O)CC(C(N2CCC(OC(F)F)C2)=O)C2(CC2)C1 C(C(=O)N1CC(NC(c2ccncc2F)=O)C(F)C1)(C(C)(C)C)NC(C)=O CC1C(=O)CCC1CC(N1CCC1CNC(=O)C(C1COC(C)(C)O1)O)=O C1(C(N2CC(C)NC(=O)C2)=O)N(C(=O)COCC(F)F)CCCC1(C)C Cc1csc(C(=O)NCc2ccccc2CNC(=O)CN2CCC(C)CC2)c1C N1(C(COCCCC#C)=O)CC(NC(=O)CNC(=O)OCC)CC1(C)CC CC1CC(NC(C2CC(CCNC(C3(C4CC4)CC3)=O)C2)=O)CS1 N1(C(CCC)=O)CC(NC(=O)CCc2cccn2C)CC1(C)COC C=C(Cl)CC(C(=O)N1CC(OC)C(C(N)=O)C1)NC(c1ccc(C)nc1)=O Cn1ccc2ccc(NC(C3CC4CC4N3C(c3cnnc(Cl)c3)=O)=O)cc12 N1(C(C2CCC(NC(C(C)N3CCCC3)=O)C2)=O)CCCN(C=O)CC1 Cc1ccc(C(N2CC(NC(=O)CCC(N)=O)C(F)C2)=O)nc1 c1(C(=O)NCC2CC(CNC(C=CCC)=O)C2)ccc(N(C)C)nn1 C1(C(C)NC(=O)CCc2nc(C3CC3)no2)CCCCN1C(=O)CN(C)S(N)(=O)=O CC1CN(C(c2c(Cl)nsc2Cl)=O)CCN1C(c1cnnn1-c1ccccc1)=O C1(C)(C(=O)NCC)CCCN(Cc2cc(O)cc(Br)c2)C1 c1(C(N2CC(CNC(Cc3cccc(C)c3)=O)OCC2)=O)cc(Cl)c(F)cc1N C(=O)(CC(C)(C)C#N)N1CCC(CN(C(Cc2c(C)scc2)=O)C2CC2)CC1 N1(C(C(n2cc(CN(C)C3CC3)nn2)C)=O)CCNC(=O)C1c1ccccc1F C=CCC(CO)CN=C(NC(C)C)NCC1CC(C)(C)CN1C(=O)OCC.C(C)(C)(C)O c1(C2(C(N(C)C)=O)CC2)ccc(C(N)=O)cc1.C1(=O)CC(=O)NCCC2CC(C2)N1 N1(C(C(CC)N(CC)CC)=O)CC(F)(F)CC1C(C)NC(=O)NC c1(C(=O)NC(C2CCN(C(C34CC3C4)=O)C2)C)cnc2ncnn2c1O CCCCC(C)CCC(=O)Nc1cc(O)ncn1 c1(C(=O)NC(C2C(C(=O)OC)C2)C)cc(-c2nn[nH]n2)cc([N+](=O)[O-])c1N c1(C(N2CCC3(CN(C(C(C)CN(C)C)=O)C3)C2)=O)cccc2nc(O)ccc12 S(=O)(=O)(c1ccc(F)c(F)c1F)N1CCOCC(NC(C(C)(F)F)=O)C1 C1(C)(OCC)CC1NC(=O)NCCNC1(CN=[N+]=[N-])CC1 C1(NC(CN(C)CC)=O)CN(C(c2ccccc2-n2ccnn2)=O)CC12CC2 CC1CN2CCN1CC2C(N1CCN(C(C2CC3CCC(C2)C3)=O)CC(C)C1)=O c1(OC(C)C)ccc(C(N2CCC(O)CC2C(N2CCCCC2)=O)=O)cc1I C(CC(CC)(CC)NC(=O)Cc1cc(Cl)ccc1Cl)NC(CC(=O)NC)=O N1(C(c2cc(C)sn2)=O)CCC(C)(C)C(NC(C2CCOCC2(C)C)=O)C1 N1(C(c2cc(C(C)=O)oc2)=O)CC2(CC(NC(C34CCOC(C)(C3)C4)=O)C2)C1 CCC(CC(=O)N1CCC(NC(c2ccnc(COC)c2)=O)C1)C(C)(C)C C1(C(N2CCC(C(C(N3C(C#C)CC3)=O)C)C2)=O)CC2CCC(C1)O2 C(=O)(C1=C(C)CCC1)N1CC(OC)C(N(C(=O)CN2CCCCCC2=O)CC)C1 N1(C(c2ccc(NC=O)cc2)=O)CC2(CC(NC(C34CCC(CC3)O4)=O)C2)C1 CCC(C(=O)NCC1COCC1NC(=O)CC#N)n1ccc(C2CC2)n1 C1(NC(CCN(CCC)C)=O)COC2(CCN(C(=O)COCC(F)F)CC2)C1 C(=O)(C1CCCc2n[nH]cc21)NCC1(F)CCN(C(C(CC)(C)CC)=O)C1 S(=O)(=O)(c1ccc(=NCC2C3COCC23)[nH]c1)NCc1cc(C)c(F)c(C)c1 N1(C(C(C=C)CC)=O)CCC(NC(=O)CCCc2nc(CC)no2)C2(CCC2)C1 N1(C(c2ccc(OC)c(C)c2)C(=O)NC2CCOC2)CCCc2ccccc2C1 C(=O)(C(O)C(C)c1ccccc1F)NCCN(C(=O)CC1(C)OCCO1)CC N1(C(c2ccn(CCC)n2)=O)CC(NC(C2CCN(C(=O)NC)CC2)=O)C2CC12 N1(C(CN(C2CC2)CC)=O)CCC(CNC(=O)C(F)(F)C(C)O)C12CCC2 C1(SC)CN(C(=O)CC2(C)CCCO2)CC1NC(c1sc(N(C)C)nc1C)=O c1(C(N(CCNC(CCNS(CC)(=O)=O)=O)CCOC)=O)ccc2nc(O)[nH]c2n1 c1(NC(C2C(NC(c3ccc(N)cn3)=O)COCC2)=O)ccc2ccoc2c1 N1(C(c2nnn(C(C)(C)C)n2)=O)CCC2CCC(NC(c3cc(Cl)c[nH]3)=O)C1C2 CSC1=C(C(=O)N2CCC2CNC(c2ccc3c(cnn3C)c2)=O)CCCC1 C1(Cc2n(C)nc(CC(=O)OCC(F)(F)F)c2)CC2C=CC1CC2=O c1(N(C)Cc2c(C)cc(C)cc2C)nccc2ncncc12 C1(CC(N2CC(=C(CNC(C(C)Cc3ccnn3C)=O)F)C2)=O)CCCS1(=O)=O c1(OC)cncc(C(=O)N(C)CC2CCN(C(c3cc(N)ccc3C)=O)C2)c1C C1(C(=O)NCCCNC(CC2(C)CC2(F)Cl)=O)CC2(C1)CC(F)C2 c1(OC)cc(N)cc(C(N2CCOC(CNC(C3CCCCC3)=O)C2)=O)c1OC Cc1nc(C)n(CCC(=O)NCC2CC2CNC(=O)CN2CCCC(CO)C2)n1 C(=O)(CN=S(C)(C)=O)N1C(CCN(C(=O)C(O)CCCN(C)C)C)CCCC1 C(C(=O)NCCCC1CCCN1C(C12CCCC1C2)=O)(C(C)(C)C)OC C1(C(=O)Nc2c(C)nccc2)C2CCC(O2)C1C(N1CCN(CCO)CC1)=O c1(CC(Cn2cc(Cn3c(C)ncc3)nn2)O)ccc(F)cc1 c1(SCCC(=O)N(C(C)CN(C(=O)C(C)N2CCC2)C)C)ccc(F)c(F)c1 C1(C(N(C)CC2N(C(C(C(C)C)F)=O)CCC2)=O)COc2ccccc2O1 C1(CNC(C(C(C)C)OCC)=O)CCCCCN1C(c1cnn(C)c1)=O C1(C(=O)NCC2(F)CC(NC(c3cccc(C)c3)=O)C2)CN2CCCC2CO1 c1(C(N2CCC(O)(CC(C)C)CC2)=O)coc2c1CN(C(=O)CN(C)C1CC1)C2 C(CC(C)C)(C(=O)NC(CNC(=O)CCCF)C1CCC1)NC(=O)OC Cc1cccc(C)c1C(=O)NC1CCCN(C(c2ncc(Br)cn2)=O)CC1 N1(C(C=Cc2cc(C)no2)=O)C2CCC(C2)C1C(N1CCCCC(C)C1)=O C1(C2CN(C(C3(C)CCCC3CC)=O)C2)(NC(COCCOC)=O)CC1 c1(C(=O)NC(C(C)(C)C)CNC(c2cccc(N)c2)=O)cc2cccnc2o1 N1(C(=O)NCC(F)F)CCN(Cc2ncsc2C(=O)O)CC1 CC1CC(C(N2CC3CCC(C2)O3)=O)CN(C(C2CCCC2O)=O)C1 C(CCC(=O)NCC(CO)NC(c1n[nH]cc1Br)=O)SC(=N)N C1(C(=O)NCC2(C)CCC(NC(C(C=C)(C)C)=O)CC2)Cc2cc(F)ccc2O1 C(=O)(CC1CCCc2cc(OC)ccc21)NCCN(C(CCOC)=O)CC(C)O O=C1CCC(C(=O)NCCC2CC(NC(c3scnc3C3CC3)=O)C2)C1 N1(C(CCCNC(N)=O)=O)CCN(C(C2CCC3CC23)=O)CC1CF Cc1ccc(CC(N2CC(NC(C3(C)CCSCC3)=O)CC2C)=O)c(C)c1 C=Cn1ccnc1S(=O)(=O)NCc1cccn2ncnc12 C1(C(N(CC(C)N(C(c2ccc(OC)cc2O)=O)C)C)=O)Cc2ccccc2O1 N1(C(C2CC(OC)C2)=O)CCC2(CCOC2)C(CNC(=O)CSCC(N)=O)C1 C1(CC(=O)NC(CC)CSC)CN(C(c2c[nH]nc2C2CC2)=O)CCC1C C1(NC(C2CC(SC)C2)=O)CC2CC1CN(C(=O)CC(C)C1CCCCC1)C2 CC12CCC(C(=O)NCC3(O)CCN(C(=O)C4=CSCS4)CC3)(CC1)CO2 c1(CC)cc(C(=O)N(CC(C)CNC(=O)C(C)n2cncn2)C)c(C)o1 C1(N(CC(=O)NCC(C)C)C)CCCN(C(=O)CNC(N)=O)C1 CCC(C)(C(=O)N1CCC(CCNC(c2cnccc2C)=O)CC1)C(N)=O C(CC(CC)(CC)NC(c1ccc(CN2CCCC2)cc1)=O)NC(CCC)=O C1(CNC(CCCOCC)=O)CCCC(NC(=O)C(C)=C2CCC2)C1 CC1=C(C(=O)N2CC(CF)(NC(c3cn(C)nc3-c3ccoc3)=O)C2)CC1 c1(C(=O)NC2CCCN(C(=O)Cc3cccc(Cl)c3Cl)C2)noc2ncccc12 c1(C(=O)NCC2(C)CCCN(C(C(F)=CC)=O)C2)ccc2c(c1)CCCCN2 CCC(CC(=O)N(C1CN(C(c2cnn(CCCOC)c2)=O)C1)C)CC(C)C c1(C(=O)NCCC2CN(C(C(COCC)(C)C)=O)C2)ccc(F)c(C(F)F)c1 CC1CN(C(=O)CCC2CCC(=O)N2)CC2(CCN(C(C3COCCO3)=O)C2)O1 C1(CC(=O)NC2CC(CNC(c3n(CC)cnn3)=O)C2)COCC(C)O1 c1(CC)nc(CNC(C2(CO)CC(F)C2)=O)sc1C C1(CNc2ccc(C(C)C)cc2C(F)(F)F)CC(C2CCCCC2)C1 Cc1nc(C(C)C)ccc1C(=O)NCC1(NC(C2CN(C)CCO2)=O)CCOC1 C=CCCCCCCCC(=O)N1CC2(C1)CN(C(c1cncc(C)c1)=O)CCO2 N1(C(c2ncnc(C)c2C)=O)CCCC2(CCN(C(=O)C(C)CN(C)C)C2)C1 c1(C(=O)OCC)cc(C)nnc1NC(CNC(C1COC(=O)N1C)=O)C(C)C C=CC1(C(=O)NC2CCN(C(=O)CCn3c(C)ccc3C)CC2C)CCCCC1 CC(C)C(C(=O)NCC(C1CC1)N(C(=O)CN(S(C)(=O)=O)C)C)n1cccn1 N1(C(=O)CN2CCC(O)CC2)CC(C(N2CCC(CCF)CC2)=O)C(F)(F)C1 C1(C(NC2c3cc(C)nn3CCC2)=O)CCc2ccccc2NC1=O Cc1coc(C(N2CCC(CNC(c3ccnc(Cl)c3)=O)CC2)=O)c1C C(C)(CO)(C(=O)NC(CO)C(C)NC(=O)Cn1cnnc1O)NC(C)=O N1(C(C2C=CC(NCc3nc(Cl)ccc3F)C2)=O)CCc2ccsc2C1 C(=O)(C1Cc2ccccc21)N1C(C(N2CC3CC3(C(=O)OC)C2)=O)(CC)CCC1 C12CC3(C1)C(C3(F)F)C(=O)N2.N#CC1(CNCC2CCCO2)CCC1 C1(N(C(C=CC(C)NC(CSCC#C)=O)=O)C)CCN(C)C1=O C1(CN=[N+]=[N-])CCN(C(=O)C(Cc2ccoc2)NC(=O)CO)C1 c1(C(C(=O)O)OC(=O)COCc2cccc(F)c2)cccc(Cl)c1Cl c1(C(=O)NC(CC)(C)CNC(c2cccn2C2CCCC2)=O)ccncc1N N1(C(c2[nH]cc(CC)c2)=O)CCN(C(=O)CC2CC(OC)C2(C)C)CC1COC N1(C(C)=O)CC(C(=O)Nc2ncc(C(C)(C)O)cn2)C(C2CC2)C1 CC(C)(C)C(O)CC(=O)NC1CCCCC1NC(C1(O)Cc2ccccc2C1)=O C1(CC(=O)NCCN(C(=O)CSCc2ccccn2)C2CC2)CC=CCC1 C1(C(=O)NCC2CCCO2)Cc2cc(O)ccc2CN1C(c1cccnc1S)=O Cc1ncc(C(=O)NC(C2CCCN2C(C2CCCN2C2CC2)=O)C)cn1 Cc1ccn(C(C)CC(=O)N2CCCC2C(C)(C)CNC(C2(C)CCC2)=O)n1 c1(C(N2CC(N(C(CCCC)=O)C)C2)=O)cnn2ccncc12 N1(C(c2c(C)csc2)=O)CC2(CCN(C(C3CC4CC4C3)=O)CC2)C1 C12(CC13CCC3)CNC2.c1(C(C)C)cnc(CNc2ncccn2)[nH]1 CCC(C(=O)NC1(CNC(=O)Cc2occc2C)CCOC1)C(C)(F)F c1(C(N2CCN(C(c3c(Br)ccc(C)c3)=O)CC2)=O)cnc2c(c1)CCCO2 c1(C(N2CC(Cn3cc(CS(CC)(=O)=O)nn3)C2)=O)c(O)cccc1F C1(COC)(CNC(C2CCCC(O)C2)=O)CCN(C(C2(C)CC2(F)F)=O)C1 N1(C(C2N(C)C(=O)CC2)=O)CC2CCC1CN2C(C1C(C(=O)O)CC(=O)N1C)=O c1(CNC(C(CO)NC(C(C2CC2)SC)=O)=O)cccc(F)c1C C=C1CCCN(C(C2(c3cn(-c4cnn(C)c4)nn3)CCOCC2)=O)C1 c1(C(=O)NC2(CCNC(=O)CSCC(N3CCCC3)=O)CC2)cc(F)cc(Cl)c1 C12(C(N3CC4C(CNC(C(C)CN(C)C)=O)(C4)C3)=O)C3C4C1C1C2C3C41C N1(c2nccc(OC)n2)CC(NC(C2CCOC(C)(C)C2)=O)CC(C)(C)C1 N1(C(C(C)C(C)(F)F)=O)CC2CCCC(NC(=O)CCCN(C)C)C2C1 C1(S(C)(=O)=O)(CC(=O)N(C(CC)Cc2ccccc2)C)CC1 CC1CN(C(c2c(N)cccc2F)=O)CCCN1C(=O)C(F)CC1CCC1 C(=O)(CCCC(C)(C)C)NCC(CCNC(c1ccnc(OCC)c1F)=O)O CC1OCCC1(C)NC(=O)COC1CCN(C(=O)C(C)(C)n2ccnn2)C1 C#CC1(C(=O)NCCC2(NC(c3csc(O)n3)=O)CCCC2)CCCC1 N1(C(C=CCCC)=O)CCC(C)N(C(C2CCCOC2c2ncc[nH]2)=O)CC1 N1(C(c2n(C)cnn2)=O)CCC(CNC(=O)CC23CCCC2C3)CC1 Cc1sc(C(N2CC(NC(=O)C3=CC4CCC3C4)C(C3CC3)C2)=O)cc1[N+](=O)[O-] N1(C(C(CC=C)C)=O)CCCC(CC)C1C(=O)NC1CCC(=O)N(C)C1 N1(C(C(CC)CC)=O)CC2CC(C(=O)NCc3cnc(O)c(F)c3)(C2)C1 C1(C(=O)OCC)CCC(C(C)C)N1C(=O)COc1cccnc1 C1(C)(C(=O)NCC(n2cc(-c3ccc(C(=O)N(C)C)s3)nn2)C)CCCO1 C1(NC(=O)CC2COC(=O)C2)CC12CCC(NC(C1(CCO)CC1)=O)CC2 c1(CN2CC(NC(c3ccc(OCCOC)cc3)=O)C2)c(Cl)ccc(Cl)c1F CCC1=C(C(=O)NCCCCNC(C2CC2c2cccc(Cl)c2Cl)=O)CCCO1 C1(CC)CCOCCN1C(C1CN(C(c2nocc2C)=O)CC12CC2)=O c1(C(N2CCCCC(NC(C(CO)OC)=O)C2)=O)cc2n(n1)CCCC2O N1(C(c2ccc(CC)[nH]2)=O)CCC(O)C(C(=O)Nc2cnccn2)C1 C(CC1CCOC1)(C(=O)N1CC(Cc2ccsc2)C1)NC(=O)OC(C)(C)C c1(NC(=O)CCC(=O)N2CCCC2)c(C(C2CC2)C2CC2)cc(F)cc1Cl c1(C(c2nnnn2CSc2ccccc2)NCCOCCO)n[nH]c(C2CC2)n1 N1(C(c2c(C)noc2)=O)CCC(NC(C2CCCS2(=O)=O)=O)C(O)C1 C1(CN(C(CSC)=O)C)CN(C(C2(c3ccccc3C)CCCC2)=O)CCO1 N1(C(CCCSC)=O)CCC2(C1)CN(C(C1CC13CCC(F)(F)CC3)=O)CCO2 C1(C(=O)NCCCCCCCC)CN(C(c2ccc(C(C)C)o2)=O)CC1C1CC1 N1(C(CCc2c(C)cccc2)=O)CC(NC(=O)C(Cl)(Cl)Cl)C(C#N)C1 Cc1ccccc1CNC(C1CC(O)CN1C(=O)C(n1nccc1C)C)=O c1(-c2cn(C(C(N3CC(OCCCCC)C3)=O)C)nn2)ccc(=N)[nH]c1 C(C(=O)N(CCC(=O)NCCCN1CCC(OC)C1)CCO)(C(C)C)SC N1(C(c2c(C)c(N)ccc2)=O)CCN(C(=O)CCC2CCC(C)O2)CC12CC2 CC(C)CC(C)(CNC(c1ccncc1)=O)NC(C1CC1(C)C)=O C1(CNC(c2cnc(Br)s2)=O)CCCN(C(C2(F)CCOC2)=O)C1 N1(C(C(c2c(C)ccnc2)(C)C)=O)CCCC(NC(=O)CNC=O)CC1 C(C(C(=O)N1CC=CC1CNC(=O)CCC1CCC1)C(C)(C)C)OCC=C C1(NC(C(C)NC(CC)=O)=O)CCCC2CN(C(=O)CNC(=O)NC)CC12 N1(C(C(CSC)OC)=O)CC2CCC1CC2NC(=O)C(N1CCCCC1)C N1(C(C2(OC)CCSC2)=O)CCC(NC(=O)C2=CCOCC2)C(F)C1 N1(C(C(C=C)(C)CCOC)=O)CCC2(CC1)CC(n1cncn1)CCO2 Cc1nc2cc(C(N3CCCC(CN(C)C(c4cccc(N)c4)=O)C3)=O)[nH]c2s1 C1(CCC)CCCCC1OC(=O)CCCN(C)C(=O)NC1C(C)(C)C1(C)C c1(OC)nccc(NC(C2CC(F)(F)CN2C(C23CC(C2)C3)=O)=O)c1C C(C)(C)(CC(F)C(=O)N1CC(O)C(O)C1)NC(CCC(=O)N(C)C)=O N1(C(=O)C=C2CCOCC2)CC2CCC(Nc3nccc(CC#N)n3)C2C1 c1(C(=O)OC)ccc(C(=O)NC2CCCC(C(=O)NC(CO)C(C)C)C2)cc1O c1(CC(=O)N(CC(CC)NC(=O)C(O)CSC)C)cccc2ccsc12 n1(CCC(N2CC(F)(CNC(C(CN(C)C)O)=O)C2)=O)cccnc1=O Cc1ccc2c(C(=O)NC3CCCN(C(C4CC5CC5C4)=O)CC3)cnn2c1C C1(C(=O)NC(C)Cn2ccnc2)(CN(C(=O)CC2CC23CC3)C2CC2)CCCC1 c1(SC)cc(C(N2CCC(C3(NC(C4CCSC4)=O)CC3)C2)=O)ccc1[N+](=O)[O-] c1(C(=O)NC(CC)(C)CCNC(=O)CN2CCCC2C)ccc(O)c(F)c1 C1(NC(C2C(=C)C2)=O)CN(C(C2CN(C)CCN2C)=O)CC1C=C CCC(CNC(=O)C(CNC(c1cncc(NC)c1)=O)N(C)C)(CC)CO N1(C(C(C)OCCC=C)=O)CCCC2(C1)CN(C(=O)CC1CCC(OC)CC1)C2 CC1=CC=C2C=CC=C1NC(=O)NC1CC2=NN=CNC1 C=CCCCC(C(=O)NC(CC=C)CC)NC(=O)C(C)O N#CC1(C(=O)NC2CC3CC(CO)C2C3)CC2CCC1CC2 C(=O)(C(C)(C)S(C)(=O)=O)N1CCC(OCCNC(c2c(C)ccc(CC)c2)=O)CC1 Cc1c(C(=O)NC2CCCN(c3nnc(C(C)(C)C)o3)C2C)cnc2ncnn12 C1(NC(C(C)SCCCC)=O)CC2(CCN(C(C3CC4C(C3)C4(F)F)=O)CC2)C1 C(=O)(C(F)C(C)(C)O)N(CCC(=O)N(CCCC(=O)OC)C)C1CC1 C1(NC(C(C)OCC)=O)CN(C(=O)CC(C)SC)CC12CCC2 c1(C(=O)NC(CC)CNC(=O)CSc2ccncc2)cnc(C)c(C)c1 c1(C(N(CCCC)CCO)=O)cncc(CNC(C2C(C)C2C)=O)c1 Cc1ncc(F)c(=NCC2CCC(NC(=O)CCc3ccc(F)cc3Cl)C2)[nH]1 c1(C(N(CCNC(c2cnc[nH]2)=O)CC2CC2)=O)ccncc1F C(=O)(C(O)CC(F)(F)F)OC(CCCCCC(=O)N1CC=CC(OC)C1)=O C#Cc1ccc(C(N2CCC(C(CO)NC(=O)CC3(CSC)CC3)CC2)=O)o1 C(=O)(C(C)(C)C(N)=O)NC1C=CCN(C(CSc2cccc(OC)c2)=O)C1 C1(C(=O)NC(c2nccc(O)n2)C)CCN(C(=O)c2cc3n(n2)CCO3)O1 C#CC1(CO)CCN(C(=O)CC2N(C(=O)C=CCN(C)CC)CCC2(C)C)C1 c1(C(=O)NC(CC(C)NC(CCOCCC)=O)C)cc2c(Cl)nccc2o1 C(C(C)C(C)(C)C)NC(c1snnc1C1CC1)C N(C1c2ccccc2C2CC1C2)C(CNC(=O)NC)=O.C12CCCN(C1)C2=O C1(CC(N2C(C(CCC)C)CCC2)=O)CCN(C(=O)CC2(OCC)CC2)CC1 c1(C(=O)NCC2CCCC(NC(C3CCCCC3)=O)C2)cnc2[nH]cncc1-2 c1(OC)cnc(C(=O)NC2CN(C(=O)COC3CCCCC3)CC2OC)c(F)c1 c1(CNC(C(CC)n2cncn2)=O)cc(C)c(C(N2CCC(O)(CC)C2)=O)o1 C#CCC(C(=O)N(C1CC(OC)C1)C)NC(=O)Cn1[nH]cnc1=N C1(C(=O)NCC(CC=C)NC(=O)Cn2c(O)nnc2O)CCCCC1OCC CCC(CC)CC(=O)N1CCC(N2CCN(C(C3CCN(CC)C3)=O)CC2)CC1 C=CC(C)(C)CC(=O)N1CC(C(N2CC3CC3(C(=O)OC)C2)=O)C(F)(F)C1 C1(C)(CNC(C(COC)OC)=O)CCN(C(c2ccc(CC(C)C)s2)=O)C1 C1(NC(c2c(C)ocn2)=O)CS(=O)(=O)CC1NC(C1(C#N)CC2(CC2)C1)=O c1(N(C)C)ncc(C(N2CCC(NC(=O)CCCNC=O)C2)=O)o1 C(C(=O)N=c1cc(-c2ccc(Cl)s2)o[nH]1)OC(N1CC(CN(C)C)C1)=O CC(C)C(CNC(C1(C)CC1(F)F)=O)C(=O)NCCS(C)(=N)=O Cc1ccncc1C=CCNC(N1CCCC1CSC)=O.C1(N(C)C)CC1 N1(CC=C)CCOCC(COC)C1.C12CCN(CC1)C2=O C1(C(=O)NCc2cc(O)c(O)cc2O)CC2CCC(C1)N2C(c1ncsc1Br)=O C1(C(=O)NCCCCN(C(=O)Cn2ccc(C3CC3)n2)C)OCCCO1 CC1Cc2c(Br)ccc(Br)c2CN1C(=O)CNS(=O)(=O)c1ccccc1F C(=O)(CC(F)(F)C(C)C)NC1CCC(CCNC(c2ccc(OC)c(F)c2)=O)C1 N1(C(C2(S(N)(=O)=O)CC2)=O)C2CCC1CC(NC(C1(CO)CCCO1)=O)C2 N1(C(C2N(CCC)CCC2)=O)CC(OC)CC12CCC2.C12(CCOCC1)C(=O)N2 C1(n2c(C3CC(N)CC(C)(C)O3)nc(C3(CC)CC3)n2)CC2(CCOCC2)N1CC c12ccc(cc1)-c1nc(nn1CC(C)C1CC1)C2.c1(SC(C)C)nncs1 c1(C(N2CC(NC(c3cn(CC)nc3)=O)C3C2C3)=O)cc(F)c(F)cc1F C#CC1CCCCN1C(=O)C.c1(C(=O)OCC)cnn(C2CC2(F)F)c1 N1(C(c2n(COC)ncc2)=O)CC2ON=C(CNC(=O)COc3cn[nH]c3)C2C1 c1(NC(C2(O)CCN(C(c3c(C)noc3)=O)C2)=O)ccc([N+](=O)[O-])nc1 c1(C(=O)NC2(C)CC(NC(C(c3nc(C)sc3)=O)=O)C2)cccc2oncc12 c1(CC(=O)NC(C(C)(C)NC(C=CCN(C)CC)=O)C)cn(C)nc1C C1(C(=O)NC(C=C)C)COCCC1NC(c1cc[nH]c1)=O C12(C(=O)NC3C(C(C)C)N(C(=O)CN4CC=CC4)CC3)CCCN1CCC2 C(=O)(CCC(C)(C)C(=O)NCC1(O)CCCN(C(C2(N(C)C)CCC2)=O)C1)OC CCCCC(O)CCC(=O)N1CC(O)(C(C)NC(c2cnc(C)cc2Cl)=O)C1 CC(C)CC(C)C(=O)NCCN(CCOCCO)C(C1CC1C(F)F)=O CC(C)(CC#N)C(=O)N1CC=CC(C(=O)NCC2(C3CC3)CCC2)C1 c1(C(N2CCC(NC(C(C)N(C)C)=O)CC2C2CC2)=O)nc2ccccc2[nH]1 C1(NC(CN2C(C)CCCC2)=O)C2CC3C1C3C2C(N1CCC(n2ccnc2)C1)=O c1(NC(c2c(CC)n[nH]c2)c2nnnn2CC(F)F)cccc(S(C)=O)c1 S(=O)(=O)(c1ccc(Br)s1)N1C(C(=O)NCc2ncccn2)CC2CC21 c1(C(=O)NCCCC2CCN(CC(=O)NC3CC3)CC2)ccc(CCF)cc1F c1(C(=O)NCC2N(C(c3c(C)cc(F)s3)=O)CC=C2)ccc(OC(F)F)c(Cl)c1 c1(C(=O)NC(CC(C)NC(c2c(C)cc(C)[nH]2)=O)C)ccc(S(N)(=O)=O)n1C C(CCSC)(C(=O)N1CC(C(=O)NC2CC2c2ccncc2)(SC)C1)OC N1(C(CC(CCC)O)=O)C(CNC(c2ccc(N)c(O)c2)=O)CC2CCCC12 C1(CNC(C2(CSC)CCC2)=O)CCCC2(CN(C(C3(CO)CCCC3)=O)C2)O1 c1(C(N2CC(C)C(NC(=O)C(C)n3cnnn3)C2)=O)ccc(S(C)(=O)=O)o1 C1(C(=O)NC2(C)CC(O)C2)C2CC(O)C(C2)N1C(=O)C#CC1CC1 N1(C(c2cn(CC)nc2C)=O)CC(C(N2CC(OC)C2)=O)C(C)(C)C1 c12ccc(c(F)c1)CNC2=O.C1(C)(NC)CCCCCC1.C1(OC)CC1C(=O)NC N1(C(C(CSC)C)=O)CCC(CNC(=O)C(CO)OC)C(C2CC2)C1 NC1(NC(N2CCCC2CN2CCCC2)=O)CCCCC1 n1(CCOC)cc(CN(O)C(=O)c2cccn2C2CC2)nn1 N1(C(Cc2ncc(C)s2)=O)CCCOC(CNC(=O)CCC(C)(C)F)C1 c1(-n2cc(C3N(C(COC)=O)CCOC3)nn2)ncc(-c2ccccc2)cc1F c1(C(=O)NC2(CNC(c3cccc(C(C)C)c3)=O)COC2)ccc2nonc2c1 C1(C(=O)NC(CCCC)CNC(c2ccc(N)c(F)c2)=O)C(F)(F)C12CCC2 N1(C(C=CCC)=O)CCC(C2CCCN(C(C3(c4cc[nH]n4)CC3)=O)C2)C1 C=CCCCC(C)(C)CNC1CCCCN(C(=O)CC(C)(O)CCC)C1 Cc1nn(C)c(C)c1OCC(=O)NCCC(C)CCNC(c1cc(Cl)cn1C)=O C1(NC(C2C(C(N)=O)C2)=O)CCCCC1NC(=O)C(C1CCCCC1)O C1(C(N2CC(NC(=O)Cn3ncc4cccnc34)C2)=O)CCn2ccnc2C1 N1(C(C2C(C)=CCS2)=O)CC=C(C(=O)N(C2CCN(C)CC2C)C)C1 N1(C(C(C2CC2)SC)=O)C2CCC(C(=O)Nc3cc(C)c(F)c(C)c3)C1CC2 C(C)(CCC(=O)N1CC(C(N)=O)(CC2(C(=O)NCC(C)=O)CC2)C1)OCC CS(=O)(=O)c1ccccc1NC(C1CC12CCN(Cc1cccc(Br)c1Cl)C2)=O C1(CNC(c2ccc(C(F)(F)F)nc2)C)OCCOC12CCC2 C(=O)(CC1=CCCCC1)NC(CNC(C1(CC)CCCO1)=O)(C)CO Cn1cc2cc(C(=O)NCCNC(C3CN(C(C4(F)CCOC4)=O)C3)=O)ccc2n1 CC1CN(C(c2ccc(C(F)(F)F)nc2)=O)CC1NC(c1ccc(S)cc1)=O c1(CNC(CC2(COC)CCC2)=O)cc(NCN(C(=O)C(F)(F)C2CC2)C)on1.C1CC1 c1(CC)cccc(C(C)=CC(=O)NC(CO)C(=O)NC)c1 C12(C(N(CC(C)C#N)C3CC3)=O)CCCC1CN(C(C1C3CN(C)CC13)=O)C2 CC1CN(C(=O)CSc2cn[nH]c2)CC1CNC(=O)C(C)O c1(C(=O)NCC=CCNC(c2nc(C(C)OC)oc2)=O)ccc(CCF)cc1 OCC1CCc2sc(CNC(c3ccc(C(=O)O)cc3)CO)cc21 c1(NC2CC(C)(C)C2)nc(N(C)Cc2ccc(CC)o2)cc(C)n1 CC1(CNC(C2(CCO)CC2)=O)CCN(C(C2CC3CC3C2)=O)C1 Cc1cnn(CCCCNCC(C)(C)Cn2cccn2)c1 C#CCC(C(=O)NOCCOCCOC)NC(=O)C(CCC)N(C)C N#Cc1cc2cc3[nH]c2cc13.c1(NC(c2ncccn2)=O)ccnc(Br)c1F Nc1c(C(N2CC=CC(NC(=O)C=CC3CCOC3)C2)=O)cc(F)cc1F c1(C(=O)NCC(CN(C(C(CC)C)=O)CC)C)cncc(NS(C)(=O)=O)c1 C(=O)(C(C)(C)CCC(=O)N(C(C)CNC(C)=O)CC)OCCC(C)(C)C N1(c2snc(CCC)n2)CC(NC(c2scnc2CC)=O)CC1C Cc1cc(C)cc(C=CC(=O)NC2CC(NC(=O)C(C(C)C)C(C)C)CC2O)c1 C1(CNC(CC2CCC(NC(=O)OC(C)(C)C)C2)=O)CC2COCC2C1 N1(C(c2c(S(CC)=O)cccc2)=O)CCN(C(=O)COCC2CC2)CC(C)(F)C1 c1(C(=O)NCC(c2cc(C(F)(F)F)n[nH]2)=O)ccc(Cl)cc1 c1(C(=O)NC2(CCNC(C(C)N(CC(F)(F)F)C)=O)CC2)coc(C2CC2)n1 c1(C(=O)OC)ccc2c(c1)CC1(CC1)N2C(=O)CNC(CN(C)C)CO C1(C(=O)NC2CCN(C(C(CC=C)NC(C)=O)=O)C2)CC2CCC1N2C(=O)NC C1(NC(c2nc(OC)c(C)s2)=O)COCCN(C(=O)Cc2ccc(Cl)cc2C)C1 c1(NC(C)=O)ccccc1NC(=O)Cn1nc(C)cc1C(F)(F)F C1(CNC(C2CC23CCOC3)=O)CCCN(C(=O)C=Cc2ccccn2)C1 c1(SCCC(=O)NC2CN(C(=O)CSc3ccccn3)C2)ccccc1 C1(C(=O)NCC2CCCC(NC(C=CCCC)=O)C2)CCc2ccccc2CC1 Cc1c(C(N2CCC(C(F)CNC(=O)CCC(C)C)CC2)=O)c(Cl)nn1C N12CC3(CC1CCO3)C(=O)NC(=O)OC2=O.C(C)(C(C)C)NC c1(SCNC(C(c2n(CCC)ccn2)N(C)C)=O)ccc2c(c1)CCC2 N#Cc1ccccc1OCC(=O)NCCCNC(C1(C(F)(F)F)CCC1)=O c1(C(=O)Nc2cc(C)c(Cl)nc2)ccc2cncn2c1 C(CNC(C1(O)CC1)=O)(C(C)C(C)C)NC(c1c(C)n(-c2ccccc2)nc1)=O c1(C(C(=O)N(CCOCCN(C(C(=O)OC)=O)C)C)C)cccc([N+](=O)[O-])c1C CN1C(=O)CC(N(C2CN(c3cc(Cl)c(O)nn3)C2)C(C)=O)C1=O C1(NC(C=NOC)=O)CCN(C)C12CCCN(c1ncnc3cc(Br)ccc13)C2 Cc1ccc(C(=O)NCCCN(C(c2ccc(O)nc2)=O)C2CC2)c(C)c1 C(C)(C)(CC(F)C(=O)NCc1cncc(Cl)c1)NC(CC(CC)C)=O Cc1cnnc(O)c1C(=O)NC1CN(C(=O)CCOCC(C)C)CC1C c1(OC)ccc(CC(N2CC(NC(=O)C(c3ccccc3Cl)O)C2)=O)cc1OC N1(C(C2C(=O)NCC2)=O)CCN(C(c2cc(C3CC3)nnc2O)=O)C(CF)C1 N1(C(CCCOCC)=O)CC(NC(C2CC(c3ccccc3)O2)=O)CCC1C c1(C(N2CC(NC(C(C3CCC3)OC)=O)C2)=O)cc(Cl)c(N)c(Cl)c1 Cc1cncc(C(N2CC(F)(C(=O)NCC3CC34CC4(F)F)C2)=O)c1 [N-]=[N+]=NC1CCCC2(C1)N(C(=O)CN1CC3CC1(C(=O)O)C3)CCC(=O)N2 C(=O)(C#CC1CCOC1)NCc1nnn(C)c1C(=O)NC1C(=O)OCC1(C)C c1(C(=O)NCC2CC(CCNC(C(COC)C)=O)C2)cnc(N(C)C)nc1 N1(C(CN(C)CC)=O)CCC(C2(O)CC(NC(=O)Cn3c(C)ccc3C)C2)CC1 Cc1ncccc1C(=O)N(C(C)CNC(C1(C)CCCS1)=O)C c1(C(N2C3CC(CNC(CCC#CC)=O)C2CC3)=O)ccc(F)c2c1CCC2 C1(C(=O)NC(C)(CNC(=O)CC2CCOC2)CO)(COC)CCOCC1 C(=O)(C1CNC(=O)c2ccnn21)N1CCN(C(CNC(C=CSC)=O)C)CC1 C(CCCCC(=O)NCC1(COC)CC=CC1)Oc1ccccc1 C1(C(=O)OCC)(C(=O)N(CC(O)CNC(=O)Cc2csc(C)c2)C)CCOCC1 N1(C(C2CC(C#C)(O)C2)=O)CCN(C(c2ccc(OC)c(F)c2)=O)C(CCC)C1 c1(OCC)nc(C(=O)N(C2CC(NC(=O)CC3(C)CCCC3)C2)C)co1 c1(C(N2CCC(CCNC(COCC#C)=O)CC2)=O)c(F)ccc(C)c1F CS(=O)(=O)c1ccccc1CC(=O)NC1CCC1NC(C1CC12CCCC2)=O c1(OC(C(=O)NC(c2cn(CC3CC3C(F)(F)F)nn2)CCC)C)cccnc1 C=CCC(CNC(=O)COCc1cnn(C)c1)NC(C1C=CCS1)=O C(=O)(C(F)(F)C(C)O)NCC1OCCC(NC(c2c(CC)nccn2)=O)C1 C1(N(C(C2CC(Cl)(Cl)C2)=O)CC)CCCN(C(c2cc(C#N)c[nH]2)=O)C1 C1(N(C(c2ccc(CCC)s2)=O)C)CCN(C(=O)CN2CCC(C)CC2)CC1C Cn1cncc(-c2cnccc2-c2nccn2CCN2CC3(C2)CC3(F)F)c1=O C1(CCOC)CN(C(=O)CC2(C#N)CC2)CCN1C(=O)C=C(C)C(C)(C)C c1(C(N2CCC(C3N(C(C(C)C)=O)CC3(C)C)CC2)=O)cc(O)ncc1Br C1(NC(c2cnn(-c3ccccc3)n2)=O)CN(C(C2(CO)CCCO2)=O)CC1F C1(CC(=O)NCC(C)(C)NC(CCOCCOCC)=O)CC(O)C1(C)C c1(C(=O)NC(C)C)ccc(C(=O)NC(CNC(=O)Cn2cnnn2)C2CCC2)s1 CS(=O)CCC(O)C(=O)NCCCN(C1CCCC1)C(=O)CNC=O CC(N=c1[nH]c2ccc(Br)cc2s1)C(O)c1cccc(S(=O)(=O)N(C)C)c1 CC1CN(C(c2cscc2F)=O)CCC1NC(=O)C=Cc1ccsc1 C1(C(C)C)CCOC1C(=O)NCCCC(=O)NCC1CC1c1ccoc1 c1(C(=O)NCCCCCN2CCCCC2)cc(NC(C2CC(=O)N2)=O)n[nH]1 C1(C)(C(N2CCC(CN(C)Cc3cccc(C(N)=O)c3)C2)=O)CCNC(=O)C1 O=C(CCC(CF)CF)NCC1COCCN1C(c1ccc2c(c1)CCO2)=O C1(CNC(C2(OCC)COC2)=O)C2CN(C(C3CC3c3ccccc3)=O)CC12 C(=O)(CCCC(C)(C)C#N)NCC(C)N(C(c1ccc(CC)nc1C)=O)C N#Cc1ccc(NC(C2C3CC2N(C(c2ccc(F)cc2O)=O)C3)=O)cc1 N1(C(CC(C)N(C)C)=O)CC(O)(C2(CNC(C3(CC(F)F)CC3)=O)CC2)C1 CC(C)CCCCCC(=O)NC(CC(=O)NCCC1CCCCC1O)C(F)F c1(OC)nc(N2CC3CC2CN3C(c2c(F)cccc2F)=O)ncc1Br C1(C(=O)NC(CN(C(c2cccc(Cl)c2)=O)CC)C)CCCC2(CC2)C1 C1(CNC(c2c(OC)ccs2)=O)CN(Cc2cnccn2)CCCO1 C1(CNC(CCc2cc(C)[nH]n2)=O)CN(C(=O)CN(C2CCSC2)C)CCCO1 C(=O)(N=c1[nH][nH]cc1I)NC1N(c2ncc(C)c(C)n2)CCOC1 C(=O)(C1CSc2ccccc21)N(C(C)CNC(c1cc2ncccc2o1)=O)C C1(CC(=O)NCCC2CCN(C(C3CCC(=C)CC3)=O)C2)CCn2cncc2C1 C1(NCC(C(C)(c2nnnn2C(C)(C)C)OCC)C)CCCC2CN(CCO)CC12 C1(CC)C(NC(c2snnc2C)=O)CCN1C(=O)C(O)CCSC n1(CCCCCO)nc(C2CCCO2)nc1-c1cc(C2CCCC2)[nH]n1 c1(CC)ccc(C=CC(=O)NC2CC(CCNC(=O)C(C)C(F)F)C2)cc1 C1(C2CCCN(C(=O)C(c3ccc(F)cc3)O)C2)(OCC(=O)NC2COC2)CC1 O=C(C1=COCCC1)NC1(CCCCn2ccnc2)CC1 c1(OC)cc(C(=O)N(C2CCCN(C(=O)C(C)O)CC2)C)cc(OC)n1 CC(C)C(F)(F)CC(=O)OC.C1(OCOCC)CN(C(=O)CCC)CCO1 C(=O)(C(O)C(F)(F)F)NC1C(C)(C)C(C(N2CC(OCCO)C2)=O)C1 CC(C(=O)NCC1CCC1NC(=O)CCF)C(C)(C)c1ccccc1 CC1C(NC(=O)CCCCC2CC2)CCCN1C(c1cc(C2CC2)on1)=O N1(C(C2(c3ccc(C#C)cc3)CC2)=O)CC2(CCN(C(=O)CC3C=CCC3)C2)C1 c1(C(N2CC(C)C(NC(c3ccncc3F)=O)CC2)=O)cc2ccccc2o1 c1(C(N2C(CNC(C(n3cc(Cl)cn3)C)=O)CC2)=O)ccc(-c2ccco2)s1 N1(C(C2CC(C#C)(O)C2)=O)CCN(C(=O)Cc2ccsc2C)C(CC(F)F)C1 N1(C(C2NC(=O)OC2)=O)CC2C(NC(C3(Cl)CCCCC3)=O)C2C1 C=CC(CC)CC(=O)N(CCNC(c1cc(C2(O)COC2)on1)=O)CC C(CCC(=O)NC(C)(C)CNC(C1CC1C(F)F)=O)OC(C)(C)C c1(CNC(C2CCCN2C(c2cccs2)=O)=O)ccnc(Br)c1 C12CCC(CC1)NC(=O)C=CC(=O)N2.N1(C(COCC(=O)OC)=O)CCC1CO CC(C)C(O)C(C)C(=O)NC1CC(CC(N2CCCC2C(=O)N(C)C)=O)C1 N1(C(CSCCCC)=O)CC2CCCN(C(=O)C(C)OCC)C2C1 N1(CCC)CC(CNC(c2c(Br)noc2C)c2nnnn2CC)CC1=O Cn1ccc(C(N2CC(C(=O)NCC(C)(C)OCCO)C(F)(F)C2)=O)cc1=O N1(C(c2c(C)cc(F)s2)=O)CC2(CCCC2NC(c2cn3c(n2)CCCC3)=O)C1 c1(C(c2n(C(C)C)nnn2)NCC(C)CCO)cc(F)cc2c1OCC2 C1(=O)CCCCCCNC(=O)c2ncc(Cl)cc2N1.c1(CC)cc(O)ccc1Cl Cc1cc(C(=O)NC(CO)C(N2CC=C(CN(C)C)CC2)=O)c(C)cn1 c1(C(=O)NCCN(CC(C)O)C(=O)CC2CCCO2)cncc(C(C)(C)C)c1 C1(NC(c2cnn(C(C)C)c2F)=O)C2CC3CN(C(C4C(C)(C)C4(C)C)=O)C1C3C2 C1(C(N2CC(=CCC)C2)=O)CCCCCN1C(=O)CN1CC(C)(OC)C1 C1(c2nnnn2CC2CC2)(Nc2cc(CC)c(C)cc2)CCCCC1CC.C(C)=O N1(C(C2CCC(C)N2C(C2CCCS2)=O)=O)CCc2cccc(F)c21 CCCCCCCCC(F)C(=O)NCCCC1(CNC(=O)COC)CC1 CCC(O)C(C)C(=O)NCCC1CN(C(=O)CSCC(F)(F)F)C1 N1(C(CCCCSC)=O)CCC2(CCCCC2NC(=O)CCc2cc(C)no2)C1 CCC(C)C(CC(=O)NCC1COCC1(C)C)NC(=O)Cc1cnsc1 C(CCC(=O)NC1CCC(CCC(=O)NCc2cscn2)C1)OC(C)C c1(C(=O)NC(=O)CC2SC(=N)NC2=O)cc(F)nc(F)c1.CC12CN(C1)C2 C1(CNC(CCOCCC)=O)CC(C)(C)CN1C(=O)Cc1nocc1C(C)C C(CCCC(=O)N(C)OCC(=O)OC)NC(CCCOC)C(=O)OC c1(NC(C2N(C(c3cc(CC)[nH]n3)=O)C(C)CC2)=O)ccc(Cl)c(Cl)c1 c1(CC2C(NCc3cn(CO)nn3)C3C2CCC3)cc2c(cc1Cl)CCCC2 C1(C(F)(F)F)(OCO)CCCN(C(=O)CCc2c(F)cccc2Br)C1.O=CO N1(C(c2cscn2)=O)CCC(NC(C2(c3ccccc3)CCCO2)=O)C1 N1(CC(N2CC(NC(C3CCN(C)C3)=O)C3(C2)CC3)=O)CCc2sccc2C1 c1(SCN(CCP(C)(C)=O)CC(=O)O)cc(F)c(Br)cc1F c1(OC)ccc(F)c(C(=O)NC2CN(C(=O)Cc3cc(C)ns3)C2)c1 CCC(C)CCC(=O)N(CC(CO)(CO)NC(=O)CCOC1CC1)C Cc1cc(Br)ccc1S(=O)(=O)N1CCC(NC(c2cc(Cl)ccc2Cl)=O)C(F)C1 C12(C(=O)NC3C(C=C)COC3)CCCC1CCN2C(=O)CC(=O)OCC C1(N(C)C(c2ccc(CO)cc2F)=O)CC2CCC(C1)N2C(=O)C(N)=O N1(c2ccnc(CCOC)n2)C2CCCC1CN(C(c1cc(C3CC3)on1)=O)C2 C1(CCNC(c2c(C(C)C)nns2)=O)CN(C(C2CC2(F)F)=O)CCCO1 N1(C(c2ccc(C(C)=O)cc2)=O)CC2CC1CN2C(=O)CCn1ccccc1=O CC1=C(C(=O)NC2CN(C(=O)CC3CCOC3)C2)Cc2ccccc2O1 N1(C(=O)Cc2ccccn2)C2CCC1CC(NC(C1(Br)CC1)=O)C2 N1(C(C)C)C(=O)COCC1C(=O)N(C)CCN(C(=O)Cc1cnn(C)c1)C c1(C(=O)NCC2C(CC)CCN2C(C2CCC2(OC)OC)=O)n[nH]c2c1CCC2 C1(C(N2CC3(CC(CNC(C(CC)(C)O)=O)C3)C2)=O)CC2(CCCC2)CO1 CC1CCN(C(c2sccc2C#N)=O)CC1NC(c1ccc(F)c(C(F)F)c1)=O C1(N(c2c(C)nn(C)c2)C(=O)CC(C)N(C)C)CCC2(CC1)CNC2 C(C)(C)(CC(=O)NC(C1CCOCC1)CO)N(C)C(c1ccc(CO)cn1)=O Cc1cc(C(=O)NC2CC(Nc3nccc(CO)n3)C2(C)C)ccn1 c1(OC)ccc(Cl)c(C(=O)NC2CC2C(=O)NC2(N3CCOCC3=O)CC2)n1 C1(C(=O)NC)(C(=O)NC2CC(C(=O)NC(C)CCN(C)C)C2)CCC1 N1(C(c2c(C)c(C(F)(F)F)n[nH]2)=O)CCN(C(=O)C(O)CC(N)=O)CC2(CC2)C1 C1(NC(c2c(C)oc(Cl)n2)=O)CCC(C)(NC(=O)Cc2ccc(Cl)cn2)CC1.CC N1(C(Cc2cc(OC)no2)=O)CCN(C(c2coc(C(F)F)n2)=O)CC1C CN1CCOCC1(F)C(=O)NC(C)(CCC#N)c1ccccc1 c1(C(N2CCC(CNC(CC3CC(OC)C3)=O)C2)=O)scc(C)c1OC c1(C(N(C2CCN(C(c3cc(OC)no3)=O)CC2)CC)=O)nc(C)c(C)cc1N C1(C(=O)NCc2c(C)cccn2)CN(C(=O)CSCCC#N)C(C)(C)C1 C(=O)(C1=CC2CCCC12)N1CCC(C(N(c2cccc(Cl)c2C)CC)=O)C1 C1(C(=O)OC)CN(N(Cc2cccc(F)c2C)C2CC2(C)C)C1C C1(=CC(N2CC(CNC(CC(CCC)O)=O)C(C)C2)=O)C2CC3CC(C2)CC1C3 C(=O)(C1CCC(=O)c2ccccc21)NCCN(CCC)C(c1ccc(F)cc1)=O c1(SC2CCN(C(C(=O)N(C3CCC3)CC3CCCCO3)=O)C2)ccc(O)cc1 N1(C(CC2(OC)CCC2)=O)CC(C(=O)NC(C)(C(N)=O)C(C)C)CCC1(C)C N1(C(C(Br)=C(C)C)=O)CCCCC(C2CN(C(=O)C(C3CCCOC3)N(C)C)C2)C1 c1(C(=O)NC(C#C)C(C)C)ccc(C2COCCN2C(=O)CC2CC2CC)n1C C1(NC(C(C)OCOC)=O)COCCN(C(=O)C(C)Oc2ccc(Cl)cc2C)C1 Cc1ccc(CNCC2CC23CCN(c2nccc4[nH]ccc24)CC3)cc1C#N c1(C(N2C(CNC(C(C)C)=O)C=CC2)=O)ccsc1C#N C1(C(=O)NCCN(C)C(C2C3CCC23)=O)CCCN(C(N)=O)C1 N1(C(C(C)(C(C)C)NC(C)=O)=O)CCC2(CC1)CC2NC(c1ccnc(O)c1)=O C1(NC(c2c(C)nco2)=O)CC(CC(=O)NCCC2(O)CCC2)C1(C)C N1(C(C(CCC)OC)=O)CCOC2(C1)CN(C(=O)Cn1ccc(=O)n(C)c1=O)C2 Cn1nnc2c1CC(C(N1CC3(NC(=O)CCN4CCC4)CCC1CC3)=O)CC2 C(CC(C)C(=O)N(CCCCN(C(=O)C(C)CC)CCN(C)C(C)C)C)=CC CCN(OC)C(=O)CNC(C1C=CCN1C(=O)CCN(C)CCO)=O C12(C(N(C3CN(C(=O)C=Cc4cccc(F)c4Cl)C3)C)=O)CC(C)(C1)OC21CCC1 c1(NC(N(C(C)C)CCN(C(=O)C(F)CC2CC2)C)=O)ccncc1Cl c1(C(N2C(CNC(C(COC)COC)=O)CCC2)=O)cccc2ncnn12 Cc1ccc2c(c1)OCCN(C(C1CC(=O)C1C)=O)C2 N1(C(C2C(COC)CC2)=O)CC(NC(=O)Cc2ncncc2Cl)C(C)(C)C1 C(CN=c1[nH]c2cc(Cl)ccc2s1)SCCNC(c1cc(CCC)nc(O)c1)=O CCC(CC(=O)N1C(C(=O)NCC(CC)n2cccn2)CCC12CC2)C(F)F C1(C(CNC(CC2CCN(C)C2)=O)F)CCN(C(=O)CCC(F)F)CC1 c1(OC)c(OCCCN2CCCC(CNC(=O)C(N)=O)C2)cccc1C(=O)O c1(NC(C2(O)CCN(Cc3c(F)cccc3I)C2)=O)ccc2[nH]nc(I)c2c1 C(C(C)S(C)(=O)=O)(c1ccccc1)NC(C(=O)NCCCOCCSC)=O Cc1cc2ncc(C(N3CCC(C)(CNC(=O)CCc4ccoc4)C3)=O)cn2n1 Cc1nc(O)ccc1C(=O)NCC(O)CNC(=O)Cn1ncnn1 C(C(C(=O)NCCCc1ncc[nH]1)NC(C1CCS1(=O)=O)=O)OC(C)C Cc1nn(C)c(C)c1CCC(N1CC2CC(NC(C3CCCCC3)=O)CC2C1)=O C(=O)(C(O)CC(F)(F)F)N(C1CCCC(=O)CC1)CCC(N1CC(C#N)C(O)C1)=O c1(OC)ccncc1CNC(=O)C(CNC(c1sc(C)nc1C)=O)N(C)C n1(CC)nc(C(=O)NCCC2CC(NC(=O)C3=COCCO3)C2)ccc1=O N1(C(c2c(C)cc(C)[nH]2)=O)CC2CCC(C1)C2NC(C1CC2(CC(C)=NO2)C1)=O c1(NC(N(CC(=O)N(C)CCC2CCCC2)C2CCC2)=O)ccnnc1O c1(CC(=O)OC)ccc(NC(=O)CCCCC2CCSS2)c(Br)c1 N1(C(C=Cc2cn(C)nc2)=O)CCC2C(NC(c3ccc(CCO)cc3)=O)C2C1 CC1(C)CN(C(c2c[nH]nc2F)=O)CC(C)(C)C1NC(C1CCCCC1F)=O C1(CC)CC(C)CN(C(C2CN(C(=O)COCC3CC3)CCO2)=O)C1 c1(CNC(c2nnnn2Cc2ccco2)(C2CCOC2)C)cc(N)cnc1Cl c1(C(C)C)nccn1CC(=O)NC1CCC1NC(C1(CO)COC1)=O Cc1cc(Br)ccc1C(c1nnnn1C1(C)CC1)NCCCOC(=N)O c1(CC(N2CCCC(C(C)(O)CNC3CC3)C2)=O)c(F)cc([N+](=O)[O-])cc1F c1(NC(C2C(NS(CC#N)(=O)=O)C2)=O)cncc(Cl)c1Cl C1(C(N(CCC(N2CC(F)(F)C2)=O)C)=O)CCC(Cl)CC1 Nc1cc(C(N2CC(NC(=O)CC3CSCCS3)C2)=O)ccc1-n1cncn1 c1(C(=O)NCCN(C(c2onc(CC)c2C)=O)C)ccc([N+](=O)[O-])o1 N1(C(CCCC#C)=O)CCN(C(=O)Cn2cnnn2)CC1c1ccccc1OC C1(c2ncc(C(=O)NCC3N(C(C(CC)OCC)=O)CCC3)[nH]2)CCC(=O)NC1 C1(C(=O)NCC2OCCN(C(C3(COC)CCCCC3)=O)C2)CCOCC1(C)C c1(CC(=O)NC(C)CCNC(C2CCC(=O)N2C)=O)c(F)cc(Br)cc1F CC1CN(C(=O)CC2CC2(C)C)CC1CCNC(c1cccc(C(C)(F)F)n1)=O C(C(F)(F)CO)N(C(=O)CCC1CCC1)CC(=O)NC1CC1c1ccsc1 CC1CN(C(c2ccn(C)c2)=O)CCC1C(=O)Nc1cnn(C)c1C(N)=O C1(C(=O)NC(CCNC(c2c(CC)ncnc2CC)=O)C)CCCCC(C)(C)C1 c1(CC)[nH]nc(C(=O)NCC2CC(OC)CN2C(c2cc[nH]c2C)=O)c1[N+](=O)[O-] c1(C(=O)NC(CCCC)CNC(c2cnn[nH]2)=O)ccc2sncc2c1 c1(C(N(C(C)CNC(C2CCN(C)C2)=O)CC)=O)cc(C)sn1 c1(C(N(C2(CNC(C3CC3(Cl)Cl)=O)CC2)C)=O)ccc(OCCN(C)C)cc1 CN1CC2CCC1CN(C(=O)Nc1ccc3c(c1)CCO3)C2 Cc1nc(C(=O)NCCc2cccc(CO)c2)nn1-c1ccccc1 N1(C(CC2CCC(C)(C)C2)=O)CCC(C)(C)C1CNC(C12CC(F)(C1)C2)=O C1(NC(C(CCN(C)C)NC(C(CC)CC)=O)=O)CCC(=O)N(C)C1=O C(C)(CCC(=O)NCC(C)(C)CN(C)C(C1(F)CCC1)=O)SC c1(C(=O)NCCN(C(CC(CC)(F)F)=O)CC(C)O)ncnc2ccsc12 N1(C(c2cc(C)on2)=O)CCC(CN(C)C(C2OCC2(C)C)=O)CC1 c1(OC)cccc(C(N2CC=CC2C(=O)NCc2cncc(Br)c2)=O)c1Cl N#Cc1ccc(C(N2CCCCCC2C(=O)Nc2ccc(Cl)cc2)=O)c(F)c1 C1(C(=O)NC2(C)CC(NC(=O)C(c3ccc(F)cc3F)O)C2)Cc2nccn2C1 C1(C(=O)NCC2(C(=O)NCC(c3cccs3)C)CCC2)C2CC3C(C2)C13 C1(C(=O)NC(C(=O)NCC(c2cccs2)C)C2CC2)CCOC(=O)CC1 C1(NC(c2n(CCC)ncc2)=O)C=CCN(C(=O)Cc2ccco2)C1 C#Cc1cccc(C(=O)NC2CCC(NC(c3cc(C)co3)=O)C2)c1F CCC(C)C(C(=O)NCC1CC2CCC1N2C(c1cnn[nH]1)=O)c1ccccc1 N1(CCN(C(=O)CCN(C(=O)CC2CCOC2(C)C)C)C)CCOCC1=O c1(C(=O)NC(CCN(C(COCCCC#C)=O)C)C)[nH]c2ccccc2c1CC C1(CCC(N2CC(C(C)(C)NC(=O)C)C2)=O)CCC(=O)NC1.c1(N)nccs1 c1(C(C(=O)NC2(C)CN(C(c3c(C)nn[nH]3)=O)C2)C)ccc(Br)cc1F C1(NC(CN(C(=O)C(O)C(F)(F)F)CCC)=O)CCC(O)CN1C c1(C(N2CCC(CCNC(CC3(C#N)CCC3)=O)C2)=O)cc(F)cc2cc[nH]c12 N1(C(C(C)NS(C)(=O)=O)=O)CC2CC(NC(C3CC(F)(CO)C3)=O)CC2C1 N1(C(c2ccc(N(CC)CC)nc2)C(=O)NCC)CC(COC)CC1(C)C N1(C(CCC2CCC(C)O2)=O)CCCN(C(C2SCCCS2)=O)CC1 C(=O)(CC(C)CC(F)(F)F)OC(C1CCCOC1)CC c1(NC(=O)NCC2N(CC(=O)NCC(F)F)CCC2)cnc(Cl)c(Cl)c1 N1(C(c2cc(C)c(C)s2)=O)CC(NC(=O)C(O)(C2CC2)C2CC2)CC1(C)C C12(C(N(C3CN(C(=O)CSc4cccc[n+]4[O-])CC3O)C)=O)CC1CCC2(F)F C(CCCC(=O)NCC(C1CCCC1)NC(c1cccc(CO)c1)=O)OC c1(CCC)n[nH]c(=NC(=O)N(CC(c2ccc(F)cc2)O)C)s1 N1(C(c2n(C(CC)C)ncc2)=O)CC2(COC(CNC(C3CCCS3)=O)C2)C1 CS(=O)(=O)c1coc(C(=O)NC2C3CN(S(=O)(=O)c4cccnc4)CC23)c1 c1(OC)cc(OC)cc(CN(C)C(=O)NCC2CCOC(=O)N2)c1 C(=O)(C(CC(N)=O)NC(=O)CCC(C)(C)F)NCCCN(C(C(C)C)=O)C(C)C c1(C(N2CCC(N(C(C(CC)(C)OC)=O)C)CC2)=O)c(C)cc(C)nc1C N1(C(CC2C(=O)NC(=O)N2)=O)C2CCC1CN(C(=O)CCC1CC1(F)F)C2 N1(C(C(CO)C(=O)OC(C)(C)C)=O)CCCC(CNC(=O)C2=CCSC2)C1 N1(C2CCC(N(C)C(c3cnn(C)c3)=O)C2)CCN(C(c2ccsn2)=O)CC1 c1(OC)cc(CN2CCCC2CC(=O)NC2CCCN(C(C)=O)C2)c(Br)cc1O c1(CCCSCC(=O)NCC#CCNC(=O)COC2CC=CC2)ccccc1 C12(NC(C3CCC4(CCC4)C3)=O)CCCN(C(=O)CN3CCCCC3)CC1C2 N1(C(CCC)=O)CCCCC1C1CCCN1C(=O)Cc1cn2c(C)csc2n1 N1(C(c2cc(CNC(C=C(CCC)CCC)=O)on2)=O)CCCC2CNC(=O)C12 Cc1nn(CC(=O)NC2(C)CC(NC(C3OCCC3C(C)C)=O)C2)cc1[N+](=O)[O-] C(CC(C(=O)NC(C)Cc1nn[nH]n1)NC(C1CCN(C)C1=O)=O)OC C1(NC(C=CC=CCC)=O)CC12CCN(C(c1cc(CO)ccc1OC)=O)CC2 c1(NC(=O)Nc2cc(F)ccc2O)c(C2CC2)cccc1F N1(C(C(C(C)S(C)(=O)=O)C)=O)CCCC2(CNC(=O)C(=O)N(C)C)CCCC12 Cc1nnsc1C(=O)NC(c1nocc1C(=O)NC12CC(C)(C1)C2)C CCC(CC(=O)NC(CO)C(C)NC(c1cc(C(C)C)n(C)n1)=O)CC(F)(F)F N(C(=NCC1CN(S(=O)(=O)Cc2ccccc2)C1)NC(C)C1CC1)C(C)CF N1(C(C23CC(C)C2C3)=O)CCCC2(CCN(C(=O)CCCC3CCCC3)CC2)C1 c1(C(N2CCCC(C(=O)NCc3cc(CC)on3)C2)=O)cccc(C)c1O Cc1nc(C)c(C(N2CC3(C2)CN(c2snc(Cl)c2C#N)C3)=O)nc1C N1(C(c2cc3c(cc2Cl)OCCO3)=O)CC(C2CCC(F)(F)CC2)C1 C1(CC(=O)N(CCC(=O)N(C)Cc2c(CC)noc2)C2CC2)CC2(CC2)CO1 Cc1nc(=N)[nH]cc1C(N1CCC(NC(=O)C(C)C(F)(F)F)C1C1CC1)=O C=C=C(C)CC(=O)N(CC(C)N(C(=O)CC1CCOC1)C)C N1(C(c2c(C)cccc2)=O)CCN(C(=O)COC2CCC2)CC1c1ccccn1 c1(C(N2CCC(C)(C(=O)NCCC3CCCCO3)CC2)=O)c[nH]c2nccc-2c1 N12CCCCC1CCC(C)(C)SCC2=O.C1(CC(=O)NCC(C)C)CC2CC2C1 CC1=CCS(=O)(=NC(=O)CCCC(=O)NCc2sc(N(C)C)nc2C)CC1 CC1(C#CC(=O)N2CCC(NC(=O)Cn3nnc(=O)[nH]3)C(O)C2)CCCO1 C(C(C(=O)OCc1ccc(OC)o1)c1ccccc1)NC(C)=O.C1CCCC1 c1(CC(N2CCC(N(C(CN(C)CC)=O)CCO)C2)=O)ccccc1C c1(CN(C(=O)CCN2CCC(F)C2)C)cccc(CNC(=O)CC(C)F)c1 c1(C(N(C)CC2(NC(C3C(CC)C3)=O)CC2)=O)cc(Cl)cc2ccccc12 C(=O)(CS(=O)(=O)C1CC1)NCC(CN(C(C1N(C(CCC)=O)CCCC1)=O)C)O C1(Cn2c(C(C)(CCCl)Nc3n(C)ncc3)nnn2)C(C)(C)C1(F)F N1(C(CCn2c(C)cc(C)n2)=O)CC2CCOC2(CNC(=O)CCOC2CC2)C1 CC1CCC(NC(=O)C2=NOCC2)CN1C(=O)CC(n1cc([N+](=O)[O-])cn1)NC1CC1 C1(C(=O)NCCCC(=O)NC2C(OCC)COC2)CC2C(C1)C2(F)F CC(C)C(C(=O)NCC1(NC(c2cnc(O)n2C)=O)CCOC1)N1CCCC1=O C1(NC(CNC(N)=O)=O)CCCC(CNC(c2sccc2C2CC2)=O)C1 C(C(C)(CC)C(C)O)NC(C1(CNC(=O)C(F)F)CC(=C)C1)=O Cc1cnnc(O)c1C(N1CCCC(CCC(=O)NC2CN(C)CC2(C)C)C1)=O c1(N2CC3C(NC(CCCN(C)C)=O)C3C2)ccc([N+](=O)[O-])c(O)n1 C1(C(N(CC(CC)NC(=O)CCc2nnc(CC)o2)CC)=O)CN2CCC1CC2 c1(C(=O)NC2(C3CN(C(C(CC)C)=O)C3)CC2)ccc2c(n1)NCC(=O)N2 c1(C(N2CC(NC(C(C)OCCC=C)=O)C(C)C2)=O)cnc(C)[nH]c1=N CCC(C)C(C(=O)OCC1CCOC1)N(CC)CC.c12nc(C)c(s1)c(=O)[nH]2 CCC(C)CCCCC(=O)N1Cc2ccc(CNC(C3(C)CCC3)=O)cc2C1 C1(F)(CNC(c2scc(C)c2)=O)COCCN(C(=O)C(F)OC(F)(F)F)C1 Cc1noc(C)c1CN1CCNC(C(=O)NCCCO)C1 N1(C(c2cnc(C)n2C)=O)CCCC(CNC(=O)C(c2ccccc2)F)CC1 C(=O)(C1CCOc2c(F)cccc21)NCC(CNC(c1c(COC)ncs1)=O)O N(C1CC2CCCc3cccc1c32)C1CCN(c2cccc(C)n2)CC1 n1(CC)c(N2CCCC2CC2CCCO2)nnc1C1CCC(=O)N1 c1(C(=O)NC2CCC(NC(C3C(c4onc(C)n4)C3)=O)C2)cnn(CCO)c1C N1(C(c2cc3oc(C)c(C)c3[nH]2)=O)CCCC12CCN(C(C1CC(=O)N1)=O)CC2 c1(C(N2CCC(Nc3ccc(OC)cc3)C2)=O)c(S(=O)(=O)NC)noc1C c1(N(C)C)cc(C(=O)NC2CCCC2NC(=O)CCF)cc(Br)c1 c1(C(N2CCC(NC(c3ccc(COC)[nH]3)=O)CC2C)=O)ccc2scnc2c1 N1(C(Cc2c(C)n(C)nc2)=O)CC2CCC(C1)N2C(c1nc2c(s1)COCC2)=O c1(C(CC(=O)O)NC(=O)CSn2cc(-c3csnn3)nn2)ccc([N+](=O)[O-])cc1 Cc1noc(C)c1CNC(=O)CC1CCCC1.C12(CC1)C(=O)N2C1CC1 C(=O)(CC(O)C(C)C)NCc1c(C(N(CCCC)CCOC)=O)occ1 c1(CC)cccc(OCCNC(COCCCN(C(=O)CNS(N)(=O)=O)C)=O)c1 C=CC(C)CC(=O)NC1CC(CNC(c2cn(C)nc2-c2ccoc2)=O)C1 C(=O)(C(CC)C(=O)N(C)CC1N(CC)CC=CC1)OC c1(SCC(=O)N(C2C3CN(C(C4C(C)C4)=O)CC32)C)ccc([N+](=O)[O-])cc1 C12(C(=O)NC3C4N(C(CS(=O)(=O)NC)=O)C(CC4)C3)CCCN1S(=O)(=O)CC2 CC1CC(NC(C2CC(=O)N2)=O)CCN1C(=O)CC1CCC1 c1(OC)ccc2[nH]nc(C(N3CCC(NC(C4CC4C#N)=O)C(CO)C3)=O)c2c1 C(=O)(C1CCCn2ccnc21)N1CC(N(C)C(C23CC(C)(C2)C3)=O)C(O)CC1 C1(CC(N)=O)(C(N(CCN(C)C(C2(CCN(C)C)CCCC2)=O)C)=O)CCCCC1 n1(CCNC2(c3nnnn3C3COC3)C(CCC)CCC2)ncc(O)nc1=O CC(F)(F)CCCC(=O)N1CC2(CC(NC(=O)Cn3ccnn3)CO2)C1 c1(OC)ccccc1CSCC(=O)NC1(CC(=O)OC(=O)CS(C)(=O)=O)CCC1 n1(COCC)c(C(N2CCC(OC)C2)=O)cnc1O.C1(Cc2ccco2)C(=O)N1 C1(CNC(C(C)(O)c2ccccc2)=O)CCCCC1NC(=O)CN1CC=CC1 c1(CNC(CC=CCC)=O)n[nH]c2c1CN(C(C1CC(F)C1)=O)CC2 c1(CC)ccccc1OCC(N1CC(CNC(=O)Cc2csnn2)CC1C)=O Cc1cccc(C(=O)NC2CCC(CO)CC2)n1.C12C3CN(CC13)C2=O N1(C(c2c(CC)n(C(C)(C)C)nc2)=O)CCCC(CNC(=O)C(O)CSC)CC1 Cc1c(CN(C)C(=O)NCCC2(O)CCOC2)ccc2c1CCC2 CC(C(=O)N1CC=CCC1)C(C)NC(=O)CCc1cn(C)cn1 C(=O)(C(C)C(O)C(C)CC)N1CC=C(C(=O)N2C(C=C)CC2)C1 CCCC(C)(C)CC(=O)NC1CCN(C(c2cc3oc(Br)cc3[nH]2)=O)CC1C N1(CC)CCOC(C(=O)N(C(c2ccccc2)CNC(c2cc(C)cs2)=O)C)C1 CC1CC(C(=O)NCC2(O)CCN(C)C2)CN(C(=O)Cc2ccc(O)nc2)C1 N1(C(CN(C(=O)CC2C(C)(C)C2(C)C)CC#C)=O)CC(N(C)C)CC1CO N1(C(c2nc(CC)oc2)=O)CC(O)CCC1C(=O)NC1(C(=O)NC)CC1 c1(C(=O)NC2CCC(NC(C3(CC)CCOCC3)=O)C2)ccc(Cl)c(F)c1 CCCC(C)C(C)NC(=O)CCN(C(=O)CCc1ccncn1)CCN(C)C Cc1nc(Cl)ccc1CC(=O)N(C)CC1CCCCN1C(C1CCSC(C)C1)=O c1(C2C(C(=O)NCC(C)(CC)NC(CCCOCC=C)=O)C2)ccc(OC)cc1 c1(CN2C(C(=O)NCc3cc(Br)ccc3F)CC2)sc2ccccc2c1Cl c1(CC(=O)N(C)CC2(O)CN(C(CSCCCC)=O)C2)ccnc(O)c1 c1(NC(c2nnnn2CCCF)C(C)C2CCCC2)cnc2n1CCOCC2 N1(C(c2ccc(N(C)C)nc2)=O)CC2(C)CC1C2NC(c1ccc(CO)cc1)=O CCCC(CNC(=O)C=CCO)C(=O)NCC1CCC(=O)O1.c12cccnc1N2 C=CC1CN(C(C2C3CC2N(C(=O)C(c2cncn2C)O)C3)=O)CC1O c1(C(CNC(c2csc(O)n2)=O)NC(c2c(C)snc2)=O)ccc(F)cc1 c1(C(N2CCC(NC(c3cncc4c3CCC4)=O)C2)=O)nccc2n[nH]cc12 N1(C(C(CC)C)=O)CCN(C(C2C3CC4C(C3=O)C24)=O)CC1CF.n12cc(nn1)C2 c1(C(=O)NC(C(C)C)CCNC(C2CC3(CCC3)CO2)=O)cccc2c1CCC2 N1(C(Cc2c(OC)nccc2)=O)CCCC2(CCN(C(C3CC(F)C3)=O)CC2)C1 N1(CC#CC)CCN(C(c2cnc(C)o2)C(=O)NCC)CC1 N1(C(C(CC)CC)=O)CC(C)CN(C(=O)C(c2cccc(Cl)c2)O)CC1C C1(CNC(c2cc(CC)no2)=O)CCN(C(c2ccc(C)cc2F)=O)C12CC2 N1(C(C=NOC)=O)CCCC2(CCCN2C(=O)CC(C)C(C)(C)C)C1 C12(NC(c3ccc4ncsc4c3)=O)CCCC1CN(C(=O)Cn1cnnc1)C2 N1(C(C(=C)F)=O)CC2(CCCC2NC2(CC(C)Oc3c(C)cccc3C)CC2)C1 c1(OC)cc(C(=O)NC2CC2NC(=O)C(C)(C)C(C)O)cc(Cl)n1 c1(C(=O)NC2CN(C(C(C=C)O)=O)C(CO)C2)cc(S(N)(=O)=O)sc1Cl c1(C(=O)NCC(CC)NC(C2CCCCC2C(F)(F)F)=O)ccc(OC)nn1 c1(C(C)N)c[nH]ccc1=O.C(CC(=O)NCC)OCCCNC(C=CC)=O C=CCCN=C(NCc1cc(C2CC2)on1)N1CCC2(CCCCC2)C1 c1(SCC)cc(C(=O)NCCC2CCN(C(=O)CCC(N)=O)C(C)C2)ccc1F C(=O)(C1=CCN(C)C1)N(C(C(=O)NCCC)C)C Cn1cc(C(N2CC3CC(NC(C4CC=CCO4)=O)C2C3)=O)ccc1=O c1(C(=O)NCC2C(CNC(c3c(C)cc(C)s3)=O)C2)cc2c(s1)CCCCC2 c1(SC)ccc(O)c(C(=O)NCCCC2CCCCN2C(=O)C2=C(C)CC2)c1 C1(NC(CC(=O)NCC)=O)CN(C(=O)Cc2cc(Br)ccc2O)CC1(C)C N1(CCCCCCC)CCCCC(NC(=O)COC(F)(F)F)C1 CCCC(C(=O)NCCN(CC)CC)OCc1cnn(CC)c1 N1(C(CC(C)N2CCOC2=O)=O)CCCNC(=O)CC1.C1CC(=O)ON1C1CC1 N1(C(c2c(C)cno2)=O)CCC(O)(CCNC(=O)C(C)Cc2ccccc2)C1 c1(C(N2CCC(NC(C)=O)C2)C(=O)NC2CCC2)cccc2c1ccn2C N1(C(=O)NC2CCC=CO2)CCC12CCCN(C(c1c(C)cc(F)cc1)=O)C2 S(=O)(=O)(c1ccc2c(c1)C(C)(C)CC(=O)N2)N1CCC(SC)CC1 c1(C(N(CC(CC)NC(C23CCCN(CC2)C3)=O)C)=O)c(Cl)nc2ccccn12 c1(C(N(C)CC2CCN2C(=O)C(F)(F)C2=CCOCC2)=O)ccc(S(N)(=O)=O)cn1 c1(NC(C)=O)ccc(-c2ccc(C3(C(=O)NC4COC4)CC3)cc2F)cc1O C(CC1CCC1)(C(=O)N(CCO)OC)NC(c1ccc(CC)nc1)=O C12CCCCN1c1nccc(n1)OC2.C(COCCOCCO)OC c1(C(=O)NCCN(C(=O)C(C)C(=O)OC)CCC)cc(F)cnc1OC c1(CC(=O)NCC2C(CNC(c3c(OCC)csc3)=O)C2)cccc(OC)c1Cl c12cc(ccc1C)C(=O)NC2.C1(NC(=O)C=Cc2ccsc2)CC(C)(NC)C1.CC(C)=C Cc1cc(NC(=O)C(O)C(C)(C)C)ccc1NC(=O)C(N1CCCC1)C1CC1 c1(C(=O)NCC(C)(C)NC(=O)Cc2cncs2)ccc(=O)n(CCO)c1 C1(CC(=O)NCCCC(C)NC(c2c(C)ocn2)=O)CC2CCC1C2 C(C(C)(C)C(=O)N1CC(C(N)=O)(CNC(=O)CCNC(N)=O)C1)N(C)C N12CCCC(CC1)CNC(=O)C2.c1(CN(C)C2CC2)ccc(N(S(C)(=O)=O)C)nc1 CC1(C(N2CCCC2CCC(=O)NC2CNC(=O)C23CC3)=O)CCC(=O)NC1 n1(CC)[nH]c(=NCCC(C)c2ccccc2)cc1C C1(C)(CNC(C=CC=CCC)=O)CC(OC)CN1C(C1CC(C)(C)C1)=O c1(NCC2(F)CCN(C(=O)OC(C)(C)C)CC2)ncc(C#N)cc1F C(c1cccc(F)c1)=CC(=O)NC1C(C)CN(C(=O)C=Cc2nccs2)C1 CC1CN(C(=O)C=CC(C)(C)NC(C2CC3(CC3)CO2)=O)CCS1=O C1(C(=O)NCC(CC)NC(=O)Cn2nc(C)oc2=O)CC(C)(C)OC(C)(C)C1 N1(C(COC(CC)CC)=O)CC(C)C(NC(=O)CNC(=O)C(C)(C)C)C(C)C1 c1(C(=O)NC2CC(F)(CNC(c3c(Cl)cc(C)s3)=O)C2)c(C)nc(C)nc1C C(CC(O)C(=O)N1CC(O)CC1C(=O)NCCc1ncon1)N(C)C C1(CNC(C=C(C)C(C)(C)C)=O)CCN(C(C2(CO)CCCO2)=O)CCC1(F)F N1(C(c2[nH]cc(OC)c(=O)c2)=O)CCN(C(C2OC3CCC2CC3)=O)CC(C)(F)C1 Cc1cc(Cl)c(Cl)cc1C(=O)NC(C)CN(C)C(C1CCC(=O)N1)=O N1(C(=O)C2CC2)CCCC(N2CCN(C(c3coc(C4CCCC4)n3)=O)CC2)C1 O=C(CCCCCn1cnnn1)NCC1CCN1C(C12CCC(CC1)OC2)=O c1(C(N2CCCC(NC(c3cc(Cl)c(Cl)c(Cl)c3)=O)C2)=O)ccc2scnc2c1 Cc1ccc(F)c(N(C)C(C2CC(c3ccccc3)C2C)=O)c1 N1(CC2CC(C)OCC2)CCC2(CC1)CN(C(=O)C=Cc1cn(C)nn1)CCO2 C1(CNC(CCC)=O)CCCCN1C(=O)C(O)CF C(C(=O)N(C)OCC)N(C(c1ccnn1CC)=O)CC C1(c2n(C)ccn2)CN(C(C2(O)CCSCC2)=O)CC1NC(=O)C(N)=O C(=O)(C(C)CCCC)NC(CCCC)CNC(C1CC(=O)N(C)C1)=O CON1CC(C(=O)N(C)CC2(O)CCN(C(c3c(C)noc3C)=O)C2)CC1=O c1(C(=O)NC2CCC(CNC(C(C(CC)O)C)=O)CC2)cc2n(n1)CCCC2=O C1(C(=O)NCC2CC(NC(Cc3ncc(C)[nH]3)=O)C2)CCC(C)(O)CC1 N1(CCC)CCN(C(=O)C(C2CCCN(C(=O)Cc3cnn(C)c3)C2)(C)C)CC1 C1(OCC(=O)N(CCCNC(C2CC(C)=NO2)=O)CC)CCCCC1C Cn1ccc2cc(NC(C3CCN3Cc3cc(Cl)cc(Br)c3O)=O)cnc12 C1(CC(=O)NCCC(=C)CNC(c2ncc(C)cc2OC)=O)CC(O)C12CCC2 c1(OC)ccc(NC(=O)CCN2CCCC(CO)C2)cc1NC(=O)C(C)C c1(C(N(C2CC(NC(=O)CNC(=O)C3CC3)C2)C)=O)nn[nH]c1Cl C1(NC(CCN(C(C2(C)ON=C(C)C2)=O)C)=O)CCN2CCC1C2 N1(C(CC2CCN(C)C2)=O)CCN(C(c2ccns2)=O)CC1c1cnn(C)c1 N1(C(C=CC)=O)CC2C3CCC(C2C1)N(C(c1cc(F)cc2cc[nH]c12)=O)C3 N1(C(c2ncc(OC)cc2F)=O)CC2CCN(C(C3SCC=C3C)=O)CCC2C1 C1(c2c(C(=O)OC)nco2)CCN(C(N2CCC2c2nnc(C(C)C)o2)=O)CC1 C1(N(C)C(c2cn(C(F)F)cn2)=O)CCCN(C(=O)Cc2cc[nH]c2)CC1 C1(=O)CC(C2CC2)N1.C1(C)(NC(C2CN(CCC)C2)=O)CCSC1 C#Cc1cccc(C(N2CC(NC(=O)CC3NC(=O)NC3=O)C(C)C2)=O)c1Cl C(=O)(C1=CCC(C)CC1)N1CC(OC)C(NC(=O)C(C)(C)n2cnc(C)c2)C1 N1(CC(=O)NCC(N(C(=O)C=CBr)C)C2CC2)C(=O)CCC1=O C1(NC(c2c(C)nn(C(C)C)c2C)=O)CCN(C(c2ccccn2)=O)CC(O)C1 CCC(O)C(C)C(=O)N(CCC(C)(C)NC(C1CCC(N(C)C)C1)=O)C N1(C(c2c(OC)scc2)=O)CC=C(C(=O)NCCN=[N+]=[N-])CC1 N1(C(c2cnc(S)n2C2CC2)=O)CC(C2CCCN(C(C3CC(CF)C3)=O)C2)C1 C(=O)(C(O)C(C)(C)CC)N(CCCNC(c1cc(C(=O)OC)ccn1)=O)CC Nc1cc2c(cc1C(N1CCCC1CNC(=O)CCOCC1CC1)=O)OCO2 N1(C(C(CC)C)=O)C2CCC1C(CNC(=O)C(C)NC(c1ccoc1)=O)C2 CCCCC(C)CCC(=O)N1CC(NC(C2COCCN2C2CCCC2)=O)C1 C(CC(C(=O)N1CCN(CCO)CC1)NC(=O)Cn1cc(CO)nn1)=CC c1(NC(C(C)OC(C(C2CCOCC2)OC)=O)=O)ccc2ccccc2c1 N1(C(C2C(C)OCC2)=O)CCC(CNC(=O)CCCCN(C)C)C(F)(F)C1 N(C(=NCCF)NCC1(C)CCC(=O)N1)CC1CCC(C(C)(C)C)CC1 N1(C(C2CC(C)N(C)C2)=O)CCCCC12CC(NC(c1ccnc(O)c1F)=O)C2 CP(C)(=O)C(CC(=O)N1CCOCC(F)(CNC(C2CCC2)=O)C1)C(F)(F)F N#Cc1ccc(N2CCC(OCCNC(=O)CC3CCC(C(F)(F)F)O3)C2)nn1 C1(NC(CC=CCC)=O)CCC2CCN(C(c3cc(C4CC4)on3)=O)C1C2 C1(C(=O)NC(CCC)C2CC2)(OC)CCN(C(=O)CC2NC(=O)NC2=O)C1 C(C(O)CN=c1nc(N2Cc3cncnc3C2)c2sccc2[nH]1)OC N1(Cc2onc(C(C)C)n2)CCC2(CC1)CN(C(C1CC(C)CO1)=O)C2 c1(NC(c2cc(CF)on2)=O)c(F)cc([N+](=O)[O-])cc1Br c1(C(N2CC(CN(C(=O)CCc3c[nH]c(=N)[nH]3)C)C2)=O)cc(O)nc(N(C)C)n1 N1(C(c2c(Cl)cn(CC)n2)=O)CC(NC(=O)COC2CC2)CC1(C)CC C12(C(=O)NCc3cc(OC)no3)CC(CCO1)N(C(C1CC1OC)=O)C2 C(CCC(O)C(=O)NCCCCN(C)C)NC(c1c(C)scn1)=O N1(C(c2cnc(C)s2)C(=O)NCC2CCOCC2)CCC2C(=O)NCC2C1 Cc1nc(C)c(C(=O)NCCOC2(CNC(=O)Cc3ccsc3)CCOCC2)s1 C1(C(=O)NC(C)Cc2ccccn2)CC2CCC(C1)N2C(=O)CC1CSCCO1 C#CCCCC(=O)NC1CCCC1CNC(c1nocc1C1CC1)=O C#CCC(CC#C)C(c1ccccc1)NC1CC1c1ccc(F)c(F)c1 CC(C)C(CCN(C(=O)C#CCNC(C1(CO)CCCC1)=O)C)ON c1(C(=O)NC(C)CCCCNC(=O)CCS(C)=O)cc2c(cn1)OCCO2 CC1CN(C(C2CC2F)=O)CCCN1C(=O)C=Cc1cccc([N+](=O)[O-])c1 Cc1c(F)cc(CN2CC3(CCC(NC(=O)C(C)Cc4ccccc4)C3)C2)cc1F C1(COC)CC(CNC(c2ccnnc2S)=O)N(C(=O)CSCCC#N)C1 c1(C(=O)NCC(C)N(C(Cc2nnc(C)o2)=O)C)ccc(O)c(F)c1 C(C1=CCCCCC1)NC(CC=C)C(=O)OC C(=O)(C(C)(C)CC(=O)NC12CC(CNC(C3CCC(NC)C3)=O)(C1)OC2C)OC c1(-n2c(-c3c(C)coc3)nc(C(C3CC3)N(C)C)n2)ccc(S(=O)(=O)N(C)C)cc1 c1(NCC(C(C(C)C)O)(C)C)ccc(S(=O)(=O)NCC2(C)CC2(F)F)cc1C#N Cc1cccnc1CNC(=O)C(C)N(C)C(c1ccsc1C)=O C#CC1(N(C)C)CN(C(=O)C(C2CCCN(C(=O)CC3CSCCO3)C2)(C)C)C1 N1(C(=O)CNC(N)=O)CCC1C(=O)NOCC1CC2CC2C1 c1(C(N(CCC(N2CC(C)CC(CC)C2)=O)C(C)C)=O)ccc2cccnn12 CN1CC(C(=O)NCCOCCOCCNC(C23CCC(C2)OC3)=O)CC1=O c1(C(=O)NC(c2nnc(C)o2)C)ccc2c(c1)C(=O)CCS2 c1(OC)cnc(F)c(C(=O)NC2CC3CC(NC(C4(C)CC(C)(C)C4)=O)CC23)c1 C#CCCCCCCC(=O)N1CCC1(C)CC(=O)NCC1CC(C(C)C=C)C1 N1(C(COC(C)(C)CNC(=O)CC2CC3CCC2C3)=O)CC2CC2C2CC12 C1(CNC(c2ncsc2C2CC2)=O)CCCN(C(=O)CC2CCSC2)CC1 c1(C2CN(C(CC3C(CNC(C(c4ccccc4)C)=O)C3)=O)C2)ccc(O)cc1 C(CC(CC)C(=O)NC1(CCO)CN(C(=O)CSc2n[nH]c(O)n2)C1)=CC n1(CC)c(C)cc(C(=O)NC2CCC2NC(=O)COCC2CCOC2)c1C N1(C(c2c(C)nc(CC)o2)=O)CCC(C)(C)C(NC(c2cncnc2)=O)C1 S(=O)(=O)(c1cccc(F)c1)Nc1c(C)nn(CC(=O)NCC)c1C c1(CC)cc(C(=O)NCC2CC(C)N(C(c3cc(C)c(C)s3)=O)C2)cc(N)c1 C1(C(N(C(c2cn(-c3cc(OC)c(F)cc3)nn2)C)C)=O)CCn2nnnc2C1 N1(C(CC(C)C)=O)CC(NC(=O)COCCF)C(C2CC2)C1 c1(CCCCCC)nc(-c2ccc(C(=O)NCC(C)C)cc2)n(C2CC2)n1 N1(C(C2(F)C(C)OCC2)=O)CC2(CCCN(C(C3Cc4ccccc4C3)=O)C2)C1 c1(CC(=O)NCCCCNC(C2CC2(F)F)=O)sccc1Br C#Cc1cncc(C(=O)NCCC2CCN(C(=O)C(C)(C)n3cc(Cl)cn3)C2)c1 c1(-c2cn(CCC(=O)N(C)C)nn2)ccc(C#N)c(Cl)c1.CC1CC2N1C2=O c1(OC)ccc(CC(=O)NCC2CCCCN2C(=O)CS(N)(=O)=O)nc1OC c1(C(N2CCC(CNC(CCCC#CC)=O)CC2)=O)cc(F)c(O)c(Br)c1 CC1(C)C(C)(C(=O)NCCC(=O)NCC=CCl)C1(C)C N1(C(CCOC)=O)CCCC(C)C1CNC(c1cc(O)nc(OC(C)C)n1)=O C(=O)(C(O)CCCc1ccccc1)NC1CC(NC(CC2(C)CCCC2)=O)CC1O c1(C(=O)OC)c(C(N2CC(CNC(c3coc(C(C)(C)C)n3)=O)C2)=O)n[nH]c1C C1(NC(c2ccc(C(F)(F)F)cc2)=O)CCN(Cc2cc([N+](=O)[O-])cs2)C12CC2 C#CC(CC(=O)N(C(C)CN1CCOCC1)C)c1ccccc1 Cc1nc[nH]c1C(=O)NCCN(C(=O)CC1(C(F)F)CC1)Cc1ccccc1 c1(OC)ccc(C(N2CC=C(CNC(=O)CN3CC(C)C3)CC2)=O)cc1Br CC(CC(=O)N1C2CCC1C(CNC(c1cccc(Br)c1)=O)C2)C(F)F n1(C(=O)NCC(CC2CN(C(c3c(C)noc3)=O)C2)(C)C)nc2c(n1)CCCC2 N1(C(C(N2CCN(C)CC2)C)=O)CC2CC1(CNC(C1CCCCC1F)=O)C2 N1(C(C2CN(C)C2)=O)CCN(Cc2ccnc(Br)c2)CC12CC2 CC1CCCCC1C(N1CCCC1CNC(C1CCC2CC2C1)=O)=O c1(C(=O)NCC(CSc2ccc(OC)cc2)C)cnn2ccc(Cl)c(F)c12 C1(CN(C(c2nc(CC)oc2C)=O)C)CN(C(=O)C(O)c2ccco2)CC12CC2 N1(C(Cc2n[nH]c(=NC)s2)=O)CCC(CNC(c2ccsn2)=O)C(C)C1 C1(C(N(C)CC2(O)CCN(C(c3nn(C)cc3N)=O)C2)=O)CCC2CC2CC1 C=C(C)CC(C)C(=O)N1CCCC(N(C)C(C2CCC(CC#N)CC2)=O)C1 c1(CCC(=O)NCC=CCNC(c2nc(C(C)(F)F)sc2)=O)ccc(Cl)c(F)c1 N1(C(c2c(CNC(c3cc(CC)ncn3)=O)cc[nH]2)=O)CC(CO)C2(CC2)C1 c1(C(=O)NCC(CC=C)NC(c2nnsc2C)=O)cnn(C)c1C(F)F C1(C(N(CC(Cl)Cl)C)=O)CCCCCN1C(c1cn(C)c(=O)cn1)=O C#CCC(C)(C(=O)N1CCC(Cl)=C(Cl)C1)NC(=O)CCC(C)(C)N(C)C C1(C2(C)CC2)CN=C(N2CC(C3CC3)NC2)N1 CC(c1ccccc1)=CC(=O)N(CC(O)CNC(=O)CC12CC(C1)C2)C c1(CC(=O)NC(CNC(c2c(F)ccc(CC)c2)=O)(C)C)nc2ncccn2n1 c1(C(N2CC3C(NC(c4c(=N)cc[nH]c4)=O)C3C2)=O)cnc2ncnn2c1O c1(-c2nnc(N3C(CC)CC(C)CC3)n2CC2CCOC2)ccc2c(c1)OCO2 c1(C(=O)NCC(C)(CNC(=O)CSc2cn[nH]c2)OC)n[nH]c(C)c1O Cc1ncc(C(=O)NC2COCC2CNC(C2(C)CCNC2=O)=O)n1C c1(C(=O)NCC2C(C)CN(C(C3(C#N)CCOCC3)=O)C2)c[nH]c2cccnc12 c1(C(N2CC(N(C)C(C3CNC(=O)N3C)=O)C2)=O)cc2cc(Cl)ccc2[nH]1 C=CCCCCCCCC(=O)NC1CN(C(c2snnc2C2CCC2)=O)CC1O N1(C(N)=O)CC=C(CN)CC1.C1(CNC(=O)OC(C)(C)C)CCNCC1 CC(C(=O)N1CCC(O)(c2cn(C3CCN(C)C3=O)nn2)CC1)S(C)(=O)=O C1(CC(=O)NCC2C(NC(C(C)OCCOCC)=O)C2)CC(F)(F)C1 c1(OC)cc(SC)ccc1C(=O)NC1(C2CCCN2C(c2ccon2)=O)CC1 C1(CNC(C(CC)CCOC)=O)CC12CCN(C(=O)Cc1ncoc1C)CC2 Nc1ccc(C(N2CC3(C2)CN(C(C24CC5CC2C4C5)=O)C3)=O)c(Cl)c1Cl C=C1CCN(C(C23CCCC2C3(F)F)=O)C(C(=O)NCCN(CC(C)O)C)C1 C1(CC(N2CC(Cn3cc(-c4ccc(N)cn4)nn3)C2)=O)CCCCC1(F)F c1(N2CCC3(CC(OC)C3)C2)cc(C)[nH]c(=NCC2CC(C)CC(C)C2)n1 C1(NC(CS(=O)(=O)NC)=O)CCCC12CCN(C(=O)CCc1cnc[nH]1)CC2 N1(C(C(CC=C)(F)F)=O)CC2CCC1C1CN(C(C3CCCS3)=O)CC21 C1(C(=O)NCCN(CC)CC)CCN(C(=O)c2ccncn2)O1 C=CCC(C(=O)NC1(CCCC(=O)Nc2ccc(F)cc2Cl)CC1)C(C)(C)C C1(CNC(=O)CN2CC3CC3C2)CN(C(c2ncoc2C(F)(F)F)=O)CCO1 c1(N2CCN(CC)C(C)C2)nccc(=NCCC2CCCC2)[nH]1 N1(C(C=CC)=O)Cc2ccccc2C(NC(=O)Cc2ccc(OC)c(Cl)c2)C1 C1(CC(=O)N(CCCN(C)C(C2(C#N)CCCO2)=O)C)CCCC(C)(C)C1 Cc1cccc(C(C)NC(c2ccccc2CNC(=O)C(C)OC2CC2)=O)n1 C1(C#N)(C(=O)NCC=C(C(=O)N(CCCC)CC(N)=O)C)CC1C C1(C(N(C2CC2)CC)=O)CCCC(NC(=O)CCOC2COC2)CC1 c1(C(=O)NCCOCCN(c2ccc(S(C)=O)cc2)C)occ2c1CCCC2 c1(C(CNC(C=CC=CC)=O)NC(=O)CCCc2cccs2)ccc(C)cc1 C1(NC(C2(NC(N)=O)CC2)=O)CC(O)CN(C(c2cnc3n2CCC3)=O)C1 c1(C(=O)NCCCN(C(c2cc(OC)nn2C)=O)C)ccc(Br)c2cn[nH]c12 N1(C(c2cnc(C)c(Cl)c2)=O)CCCC(C2CCN(C(C3(C)COC3)=O)CC2)C1 CCCCCC(O)C(=O)N1CC2CCC1C(NC(C1CNC(=O)C1)=O)C2 C(=O)(C(C(C)NC(c1oc(C)cc1C)=O)C(C)C)N1CC(CCC)OCC1 O=C(CCCCCCCNC(=O)C1=CC2C=CC1C2)NOCC1(F)CCC1 CC(C)(C#N)CC(=O)N1CC(C)(C)CC1CONC(=O)COC1(C)CCC1 O=C(CC1CCOc2ccccc21)NCCCC1(NC(C2CCCCO2)=O)CC1 C(CC(C)C)(C(=O)NC)NC(c1n(CC=C)nnn1)CCc1ncn(C)n1 c1(C(N(C(CNC(=O)CCC2(C)CCC(=O)N2)C2CC2)C)=O)ccc(=O)n(C)c1 N1(Cc2c(C)c(Br)cnc2)CCC2(CC1)CC2C(N1CCn2cnnc2C1)=O c1(NC(C23C(CCN(C(C=C(COC)C)=O)CC2)C3)=O)cccc([N+](=O)[O-])c1C CC(C)CC(C)(C(N)=O)NC(=O)CC1C=CC(NC(C2CC3CC(=O)C2C3)=O)C1 N1(C(CC2N(C)CCC2)=O)CCC2CN(C(=O)CCc3cccnc3)CC2CC1 Cc1ccc(CCNC(=O)C(C2CCCCC2)NC(C2CC3(CC3)CO2)=O)nc1 N1(C(C(CC)=CCCC)=O)CCC(C2CC2)(CNC(c2nnc(C)nc2O)=O)C1 c1(C(=O)NC2(CC=C)CN(C(=O)CC(C)n3cccn3)C2)ccc(C2CC2)cc1 C(C(C)CC(=O)N1CCC(CO)(CNC(=O)CCN2CCC(O)CC2)C1)OC C(=O)(C(=O)N=S(C)(C)=O)N(C)CC1CN(C(=O)CC2(C)CC2)C(C)(C)C1 C1(C(=O)NC2(COC)CCOC2)CCCCN1C(c1cccc(F)c1)=O Cc1cc(Cl)ccc1NC(C1CC12CCN(Cc1cc(Cl)cnc1Br)C2)=O c1(NC(N2CCC(=CCO)CC2)=O)cccc(C(F)F)c1Cl N1(C(C(CC(C)C)F)=O)CCN(C(=O)CCCF)C2COCC12 C(C(CC(C)C)C(=O)NCCN1CC=CC1)NC(CCN(CC)CC)=O.C(C)(=O)O C1(CC(=O)NC2CN(C(C(C(C)C)c3ccc(F)cc3)=O)C2)CCC(C)(C)CO1 CC(C)CCC(CO)NC(C1(F)CCN(C(C2CC3CC3C2)=O)CC1)=O N1(C(C)=O)CC2CCCC1C2CNC(c1cnc(C(F)(F)F)c(F)c1)=O Cc1onc(C2CC2)c1C(=O)N(C)CCOCCNC(c1cnc(O)n1C)=O c1(C(CC)C(=O)N2CC(COC)(NC(c3coc(C)c3)=O)C2)cccc(Cl)c1 N1(C(C2CN(c3n(C)nnn3)C2)=O)CCN(C(=O)Cc2cccs2)C2COCC12 C1(C(=O)NCCCN(CC(C)C)C)CC12CCN(C(C1CCS1(=O)=O)=O)CC2 C1(CNC(C2(N(C)C)CCOCC2)=O)CC2CCC1N(C(=O)Cc1cc[nH]c1)C2 C(=O)(CC(C)C(C)C)N(C(C(=O)Nc1ccc(C(C)C)cc1)C1CC1)C c1(C(N(C)CC2N(C(CN(C)C3CC3)=O)CC(F)C2)=O)csc2cc(Cl)cnc12 N1(C(c2cc(C)n(C3CC3)n2)=O)CCC(F)C(NC(=O)C(c2cccnc2)O)C1 c1(C(=O)NC2CC3CN(c4ncncc4Br)CC23)cc2c(F)cccc2[nH]1 c1(C(=O)NC2C(NC(C3N(C)CC3)=O)COC2)cc(I)cn1C CC(CCCCNC(C1CNC(=O)N1)=O)NC(=O)CC1CCC(C)(C)O1 c1(OC)ccc(C)cc1CC(N1CC=CC1CNC(=O)C(F)(F)C(F)F)=O c1(C(=O)NC(C2CCN(C(c3ccn(C)n3)=O)C2)C)cncc(F)c1 N1(C(CSCC#C)=O)CCN(C(c2cc(F)cc3ccoc23)=O)C(C)CC1C N1(CC(=O)NC2CCCC(NC(C(CCCC)O)=O)C2)Cc2ccccc2C1 c1(NC(CC(C(C)OC)NC(c2cc(C)oc2C)=O)=O)ccc2nncn2c1 C#CC1(C(=O)NCC(c2cnn(C)c2)O)CCN(C(C2CC(=O)NC(=O)C2)=O)C1 Cc1[nH][nH]c(=N)c1C(N1CCCC1CNC(=O)C=Cc1ccsc1)=O c1(C(N2CCC(CCNC(C=C(C)Cl)=O)CC2C)=O)ccc2cnnn2c1 C(=O)(C1c2c[nH]nc2CN1C(c1ccnc(O)c1)=O)N(C1CC(F)(F)C1)C c1(NC(C2C(NC(c3cc(Cl)cnc3F)=O)CCC2)=O)ccc([N+](=O)[O-])cc1I Cc1cc(N2CC(F)(C(C3CC3)OC(C)(C)C)C2)c([N+](=O)[O-])c(C)n1 C=C1COCC(C)(C)N(C(C(=O)OC)C2=CCC(CC(=O)NCC(C)C)CC2)C1 C1(C(=O)NCC(O)C(=O)N2CCC(NC(=O)NC)C2)(CC)CCCC1 CN1CCOCC(NC(c2cc(CNC(=O)Cc3ccc(=N)[nH]c3)nn2C)=O)C1 C(=O)(C(C(C)C)N(C)C)N(C1CCN(C(COCc2onc(CC)n2)=O)C1)C c1(CC(=O)NCCCCCNC(C2CC3(CCC3O)C2)=O)cc(Cl)ccc1Cl N1(C(CCOCC#C)=O)CC(N(C)C)C(CNC(=O)C(CN(C)C)CC)C1 C(=O)(CN=c1cc[nH]cc1)NC(C)(C)CC(=O)NC1C=CCCC1 N1(C(CCN(CCCCC)C)=O)CCC(CNC(=O)CN(C)C(C)C)C12CCC2 C1(NC(C2C(C(C)C)C2)=O)CC2CC1N(C(c1c(N)cncc1Br)=O)C2 Cc1cc(C(=O)NC2CCN(C(=O)CN(C3CCCC3)C)CC2F)nc(O)n1 C(CCCC(CO)NC(c1ccc(F)cc1Cl)=O)NC(C1(C(C)(F)F)CCC1)=O C=CCCCCCC(=O)NCC1CC(NC(=O)CCOCCN(C)C)C1 c1(C(N(CCNC(C2ON=C(C)C2)=O)C2CC2)=O)cnn2c(=N)[nH]cnc12 C1(C(=O)NC(Cc2cc(NS(C(C)C)(=O)=O)n(C)n2)=O)CCN(C)C(=O)C1 C1(C(N(CCNC(=O)CC2CCCC2)C2CC2)=O)Cc2nnsc2S1 C12(C(=O)NCCC(=O)N3CC(c4c(C)cccc4)C3)CCC(F)(CC1)CC2 C1(C(=O)NCC2C(C(=O)NCCN(CCC)CC)CC2)CCCC(=O)N1 CCCC(CCC)CC(=O)NCCCC1(NC(=O)CN(C)C(C)=O)CC1 C1(C(=O)NC(C2CCN(C(c3occc3C3CC3)=O)C2)C)CCCN1C c1(CNC(=O)NC2CC(C)C2)nc(C(N)=O)co1 N1(CC(N2C(CNC(c3ns[nH]c3=O)=O)CC2)=O)CC2C=CC1C2 C1(C(N2CCC(CC(=O)NCCSC(C)C)C2)=O)CCC(C)(C)OC1 c1(CC)n[nH]c(=NCC(c2ccccc2C)OC2CCCN(C(C)=O)C2)o1 N1(C(C(CNC(C2C(C)C3CCC2C3)=O)(C)C)=O)CCCC2OCCC2C1 CC(C)(Cc1ccccc1Br)C(=O)NC1CC1NC(c1nsnc1O)=O N1(C(=O)CN2CC3CCC2C3)CCC2CCC(NC(C3CC(F)(CO)C3)=O)C1C2 CC1CN(C(c2ccco2)=O)CCC1NC(=O)CCCc1ccc(O)cc1 N1(C(=O)NC(C)Cn2cccn2)CCN(Cc2ccc(O)cc2)CC1 C1(C(=O)NCCNC(C(C)CN(C)C(=O)OC(C)(C)C)=O)CCCC2CC12 c1(C(=O)NC2(C)C(C)C2)ccn(CCNC(C2(CN(C)C)CC2)=O)c1 C=CC1CN(C(=O)CCc2ccc(CO)cc2)CC1NC(=O)CSC(C)C c1(NC(C2CN(C(CC=C)=O)CC2C)=O)cc(C)c(OC)cc1C C(N=c1[nH]c(=NCc2nccc(O)n2)c2ccccc2[nH]1)C1CC(C)OCC1 C(=O)(C(CCC1CC1)NC(=O)Cn1c(O)nnc1O)N1CC(C(=O)OC)(CC)C1 c1(C(N2C3CCC(CNC(CN4CC(C)(C)C4)=O)(C3)C2)=O)cc(F)cc(F)c1O N1(C(c2n(C)nc(C(F)(F)F)c2)=O)CCC2CN(C(=O)CCCC3CC3)CC12 c1(OC)cc(Br)cc(F)c1CN1CCC(CNc2nccc(C)n2)C1 CCS(=O)(=O)CC(=O)NC1CC(O)CN(C(c2c[nH]nc2C2CCCCC2)=O)C1 N1(C(c2cncc(SC)c2)=O)CC(NC(=O)CSc2cccc(Cl)c2)CC1(C)C C1(NC(CNC(C)=O)=O)CC(O)CN(C(=O)COc2ccc(C#N)cc2)C1 c1(C(=O)NCC2C(NC(=O)CCOCC3CC3)C2)ccc(Cl)c(F)c1 Cc1ncccc1CC(=O)NC1CC(CCNC(c2csc(CO)n2)=O)C1 N(C(=NCC1CCCCC1)NCC1CCC=CO1)CCc1nnc(C)s1 C12(C(N(CC(=O)NC)C)=O)C(NC(c3sncc3C)=O)C3CC1C2C3 C(CN=C(NCCS(C)(=O)=O)NCCCOCCN(C)C1CC1)N(CCOC)C c1(OC)cc(Br)ccc1C(=O)NCC(F)CNC(=O)CC(O)C(C)C C1(CNC(C2CCN(OC)CC2)=O)CC2CCC(C1)N2C(=O)C(C)OC1COC1 CCCC(C)(C)C(=O)N1CC2CC1C2NC(c1csc(C(F)F)c1)=O n1(CC(=O)N(C(CCNC(COCCC)=O)C)C)cc(C)c(O)nc1=O C1(N(C)C(C2C=CCC2)=O)CCCCC1NC(=O)COCC1CCOCC1 CCC(CCCC(=O)NCCN1CCOCC1)NC(C1CC1Cl)=O CCC(CC(=O)NCC1CN(C(=O)C#CC2CC2)CCC1(C)C)CC(C)C c1(OCC)cc(C(=O)NC(C)C(C)(C)NC(=O)C(C#N)C2CC2)ccn1 c1(C(N(C2CCC(NC(=O)CCCCC#N)C2)C)=O)cnc2cc[nH]c2c1 c1(CC(=O)OC)ccc(N2CCCC2c2cccnc2Br)c(C)c1 c1(C(N2CC(CNC(=O)C(c3ccc(F)cc3)O)C2)=O)cccc(F)c1Br N1(C(=O)CSC(F)F)CC2(C1)CN(C(c1sccc1SC(F)F)=O)CC2CO c1(CCCC(=O)N(CCNC(C2(C)CC2(F)Cl)=O)C2CC2)ccc2c(c1)OCO2 c1(OCC(=O)NCC(C)N(C(=O)CCNC2CC2(C)C)C)ccc(F)cc1F c1(C(CC(=O)N(CC(C)NC(=O)CCc2nc(C)no2)CC)C)c(C)noc1C c1(C(N(CCC(C)NC(c2c(C#C)cnn2C)=O)C)=O)cn(C)c(=O)cc1C C1(C(N(CCC)CCC)=O)(NC(=O)Cc2ccccc2C)CCOCC1 c1(C(=O)NC(C)C(C)NC(=O)CN2CCCCS2(=O)=O)csc2nccn12 Cc1cccc2c(C(=O)NCCCC(C)(C)NC(=O)Cc3cccs3)csc12 C1(F)(CNC(CC(C)(F)F)=O)CCCN(C(C2CNC(=O)O2)=O)C1 N1(C(c2cn(CC3CCOC3)nn2)C(=O)NCC)CCC2(CCCO2)C1 C(=O)(CC1=CCOCC1)N1C(CNC(c2nccc(OC)n2)=O)C(C)CC1 N1(C(C2(C#N)CC3(CC3)C2)=O)CC(NC(=O)CCc2cncnc2)CC(F)(F)C1 C1(CNC(c2cnns2)=O)CN(C(=O)Cc2cc(Cl)cc(Cl)c2)CCC1(F)F C(=O)(C(C)C(C)S(C)(=O)=O)N1C(C)C(NC(=O)CN(C)C)C(C)CC1 N1(C(CCC2N(C(c3nc(CCC)oc3)=O)CCC2)=O)CCOC2CCCC12 Cc1[nH]nc2cc(C(=O)N(CC(C)NC(C3CC(=C4CCC4)C3)=O)C)ccc12 c1(CN2CCC(F)(C(N3CC4COCC4C3)=O)C2)n[nH]c2ccc(Br)cc12 C1(CNC(c2c(C)scc2)=O)COC(C)(C)CN1C(C1CC1c1ccnn1C)=O c1(OCC(=O)NCC(C)NC(c2cc(OC)n[nH]2)=O)cccc(F)c1.C1(O)CCCC1 C[S+](C)CCC(O)C(=O)N1CCC(OCCNC(c2cccc(C(N)=O)c2F)=O)C1 C1(C(=O)N(CC(N)=O)C)(NC(C(C)c2cncs2)=O)CCN(C)C1 CCCC(C(O)C(=O)NCCOC)NC(=O)CCOC1CCC1.C1(=O)CCCN1 c1(CC)cccc(ON2C(C)CCC2)c1.C1(C)C(=O)O1.S(C)(=O)(=O)N(S(C)(=O)=O)CC C(=O)(C(C)(C)CC(C)C)N1CCN(C(c2onc(CC)n2)C)CC1 C(=O)(C1CCCn2ncnc21)NCC1CCN(c2cc(OC)nc(COC)n2)C1 C12(C(N(C3CCN(C(c4cncc(OCC)c4)=O)C3)CC)=O)CCC(C)(CO1)C2 CC(C)CCCCCC(=O)NC(C)C(=O)NCC(=O)NCC1CC1 c1(C(=O)NCC2C(NC(c3cccc(C#C)c3Cl)=O)C2)cccc2ncn(C)c12 C(=O)(C(C)(F)CC1CCCC1)NCC(C)(O)CNC(C1(C#N)CC=CC1)=O C1(NC(c2ccco2)=O)COC2(CNC(c3cc([N+](=O)[O-])c[nH]3)=O)CC1C2 CC1CN2CCN1C(C(N1CC(c3cn(C)nn3)C1)=O)C2 CC(C)CCC(=O)NC(C1CCCCC1)C(C)NC(C1(NC(N)=O)CC1)=O C1(CCNC(C(CNC(=O)Cc2ccco2)OC)=O)CC(C)(C)CO1 C1(CCNC(C=CCN(CC)CC)=O)CCCN(C(c2cnoc2C)=O)CC1 C1(CNC(CN(S(C)(=O)=O)C)=O)CC(C)(C)CN1C(c1cc(C(C)(C)C)on1)=O C1(NC(CCCC)=O)CN(C(=O)Cc2c(C)noc2C)C2(CCOCC2)C1 CC(C)(CC(=O)N1CCN(C(=O)C=CC2CCCCC2)C2CCC12)C(F)F C1(N(c2cnn(CCO)c2)C(C)=O)CCN(C(=O)C(C)(C)c2ccno2)CC1 Cc1cc(=NC(=O)N2CC3C=CC2C3)[nH]n1C1CCCCO1 C(C)(C(=O)NCCOCC(=O)NC1CC1O)OCCCC Cc1ccc(Br)c2cc(C(=O)NCC(C)N(C)C(c3cn[nH]c3)=O)[nH]c12 C(CN=c1nc2ncn(C)c2c[nH]1)C1(C)CN(C(Cn2ncc(C)c2)=O)C1 Cc1ccc([N+](=O)[O-])cc1S(=O)(=O)N1CC2CC1CC2N1CCC(C#N)C1 C(C(=O)N1CCCC(C(=O)NCCC(C)(C)C)C1)(C(C)C)OC c1(NCCCSC)cc(S(=O)(=O)NCc2cc(F)cnc2Cl)ccc1C#N N1(C(CCOC(C)=O)=O)CCN(C(=O)CCn2ccnn2)C(CC#N)C1 C1(S(C)(=O)=O)(C(=O)NC2CCN(C(c3n(C)cc(Cl)c3)=O)CC2O)CCCC1 Cc1cc(-c2ccc(C3CCCN3C(C3CCCC(O)C3)=O)cc2)c(C)[nH]1 CC(CC(=O)NOCCCC1CC1)C(C)(C)NC(=O)COCCCN=[N+]=[N-] C12(CNC(=O)C=Cc3cnc[nH]3)CCC(CC1)N(C(C1COCCO1)=O)C2 CC1(C)OCc2ccc(-c3nc(CO)nn3CC3CCCOC3)cc21 N1(C(CN(C(C)=O)C)=O)CCC(C)(C)C1CC(=O)NCCC1=CCCC1 c1(C(=O)NCC2C(NC(C3CCCN(C(C)C)C3)=O)C2)cc2cccnc2o1 c1(C(=O)NCC(C)NC(c2cc(C)ncc2C)=O)cccc(S(C)=O)c1 C(=O)(CCCC(F)(F)F)N1CCC(C(N2C(COC)CCCC2)=O)C1C(C)C C1(CC)(CC)CC(NC(=O)C=C(C)COC)CN1C(c1nccn1C)=O O=C1CCc2cc(C(=O)NC34CC3CN(C(C3CC3F)=O)C4)ccc2N1 C(CC(CC)C(=O)N1CCCC(N(CCO)C(c2sc(F)cc2C)=O)C1)=CC c1(C(C)=O)cncc(C(=O)NCCCCNC(=O)C(C(C)O)N(C)C)c1 c1(C(=O)O)ccc(NNC(=O)NC2COc3c(Cl)cccc32)c(F)c1 c1(C(=O)NCC2CC(OC)CN2C(=O)Cc2cnsc2)ccn2ncccc12 CC1(C(N2CC(C)(C(=O)NCC(O)CC3CCC3)C2)=O)CCOCC1 N1(C(=O)OC(C)(C)C)CCC(O)(CNC2COCCN2CC2CCC2)C1 c1(C(C(=O)NCC(C)CNC(=O)C(C)n2cccn2)C)ccc(O)cc1 c1(C(=O)NCC2CC(OCC)C2OO)ccc2nc(CC)[nH]c2c1 N1(C(CC(C)(C)N(C(=O)CC2CCCNC2=O)C)=O)CCC2C(C1)C2(F)F c1(C(=O)NCC2(C)CCCN(C(c3ccc(C)o3)=O)C2)cc2nc(F)ccc2o1 CCC(C(=O)N1CC(O)(CNC(C2(COCC)CCCO2)=O)C1)N(C)C Cc1cc(C(N2CCC(C(C)NC(c3c(C(F)F)cnn3C)=O)C2)=O)ncc1Cl C(=O)(C(C)(C)CC#N)OCC1CC(OC)CN1C(=O)CC(O)C(C)C c1(CC(=O)NC23CC(CNC(C)=O)(C2)C3)cc(C)sc1C C1(NC(=O)CCc2ncc(Br)cn2)COC2(CCN(C(=O)C3CC3)CC2)C1 c1(N(CC(C2CCCO2)OC)C)cc(NCCCC(F)(F)F)nc(C(F)(F)F)n1 c1(C(=O)NCc2ccc(Br)c(F)c2)cc(-c2ccc(OC)cc2)cn2ccnc12 CC1=C(C(=O)N2CCN(C(=O)C(C)NC3(CO)CCCC3)CC2)SCCO1 c1(C(=O)OCC)c(NC(=O)CC2CCOCC2)ncn1CC1CC1 CC(C(=O)NOCCC1CC1)C1CCCO1.c12ccccc1c(=O)n(C(C)C)o2 C1(C(=O)NC(C=C)C2CCC2)CN(C(c2sccc2C)=O)C(C)(C)C1 N1(C(CC2(CSC)CC2)=O)CCC(C(C)(C)NC(c2occc2Cl)=O)C1 CC(CC(C)(C)C)C(=O)NC(C(=O)N(CC(C)(F)F)C)c1ccco1 c1(C(=O)NCC(C)N(C(C2(C)C(CC)CCC2)=O)C)ccc(C)c(C)c1N c1(C(N2C(CNC(C(C)C3CCC3)=O)CC2)=O)snc2ccccc12 C1(C(N(C(C)CN(C(=O)C(C)(C)N(C)C)C)C)=O)CCCC1(C)C C(=O)(CCC(F)(F)C(F)F)NCC1N(C(CSCCC#N)=O)C2C(C1)C2 C12(NC(CNC(=O)NC)=O)CC(NC(c3csc(C#N)c3)=O)(C1)C2 c1(CCOC)nc(=NCC(C)(C2CC2)NC(=O)CCC2CCCO2)s[nH]1 CN=c1nc(C(=O)NCC(CC(C)C)NC(=O)C=C2CCC(C)CC2)cc(C)[nH]1 C(=O)(C(CNC(c1cccc[n+]1[O-])=O)CC(C)C)Nc1c(OC)ccc(Cl)c1 Cc1cccc(CCC(=O)NC2CC(CCNC(c3cc[n+]([O-])cc3)=O)C2)c1 c1(C(c2n(C3(C)CC3)nnn2)NCC2(C3CC3)CC2)cc2cc(Br)ccc2s1 C(=O)(C(C)(C)F)N(CC1CN(C(C(C)N(C)C(=O)OC(C)(C)C)=O)C1)C1CC1 c1(C(N(CCNC(Cc2c(C)noc2)=O)C(C)C)=O)nn(C(C)(C)C)cc1Cl CC1COCC(C(=O)NCc2c[nH]nc2C(=O)N(C2CC3CCC2O3)C)O1 C(=O)(C(O)C1=CCCCC1)N1C(C(N(C)CC2CCCC2)=O)CC(F)(F)C1 Cc1noc(C)c1C=CC(N1CC(NC(c2ccc(O)c(Cl)c2)=O)CC(O)C1)=O N1(C(C(C)=O)=O)CCCC12CCN(C(=O)COCc1ccccc1)C2 CC(CS(=O)(=O)c1ccc(Br)cc1)C(=O)Nc1ccc(C(F)(F)F)cn1 C1(C(=O)NCC2(OC)CN(C(c3ccc[n+]([O-])c3)=O)C2)C2CC3C(C2)C13 N1(C(CC)=O)CC(C(N2CCC2CO)=O)C2(CCC2)C1 C1(CNC(c2ccnc(CO)c2)=O)CN(C(c2ccnc(OCF)c2)=O)CCO1 C#Cc1cncc(C(=O)NCCC2CN(C(=O)CC3NC(=O)NC3=O)CCO2)c1 N1(C(c2c(OC)ccc(Br)c2)=O)CCCC2C1CCN2Cc1scnc1C c1(CN2C(C(N3CC4CCC3CC4)=O)CCC2)ccc(Cl)c(Cl)c1F N1(C(=O)OC)CCC(NCc2n[nH]c(C(F)F)n2)c2ccccc21 Cc1cc(C(F)F)ncc1C(=O)NC(C)(C)CCCNC(C1CCCC(F)C1)=O N1(C(c2cccn(C(F)(F)F)c2=O)=O)CCC2CN(C(=O)C(Cl)(Cl)Cl)CC2C1 N1(C(C(CN(C)C)NC(CC(C=C)C)=O)=O)CCCCC(F)(F)C1 c1(C(N2CCC(NC(C(N3CCSCC3)C)=O)CC2C)=O)ccnc2[nH]ncc12 C1(NC(c2cnc(CC)s2)=O)CC12CCN(C(C1CC=CC1)=O)C2 C1(C(=O)NCc2c(C)cco2)CCCCN(C(C23CCC(C2)OC3C)=O)C1 c1(C(=O)NC(CCN(C)C(c2cc[n+]([O-])cc2)=O)c2cccs2)c[nH]cc(Cl)c1=O C=CCC(C)(C)C(=O)N1CCC(NC(c2ncccc2CSC)=O)C(O)C1 c1(C(C2CN(C3CC3)C2)OC(C(n2c(C)ncc2)C)=O)ccccc1Br N1(C(C(COC(C)=O)NC(C)=O)=O)CCCC2(C1)CN(C(=O)C(O)C(C)C)C2 N1(C(C2CCCSC2)C(=O)NCCCF)CCCCCC1CCO C(C)(CC(=O)NC(CN(C(COC)=O)C)C)NC(C1CCCCC1)=O c1(CC=CC(=O)NCCN(CCC)C(C2SCCCS2)=O)cccnc1 c1(NC(C(c2cccnc2N2CCCC2)C)=O)nc2c(Cl)cccc2s1 C(C)(CNC(=O)CCOCC(C)C)(CNC(c1cc(C(N)=O)cs1)=O)OC c1(C(N2CCCC(NC(C3(C4CC4)CC=CC3)=O)CC2)=O)c(F)cc(F)cc1Cl N1(C(CC2C(COCC)C2)=O)CCOC(CNC(C2(COC)CCC2)=O)C1 C1(C(=O)NCC(C)=CC(=O)NCc2cncnc2)C2CCC(F)C12 Cc1cc(C(=O)NC2CCCCN(C(C3CN4CCN3CC4)=O)C2)c(C)c(C)c1 CC1(C)CCCCN(C(=O)CCNC(C2CC3(CC3)CO2)=O)C1 C1(C)(C(c2nnnn2C2CCCCCC2)NCC2CCCN(C)C2)CCC(F)(F)C1 N1(C(c2ccn(C)n2)=O)CC2CCC1CN(C(=O)CC#N)C2 CCCC(C(=O)N1CC(OCC)C(NC(=O)CC2(C)CC2)C1)OCC CC1(CNC(=O)C=CC2CCOCC2)CCC(NC(=O)Cc2ccc(O)cc2)C1 C1(NC(=O)C#CC2CC2)COC2(CCN(C(c3ncc4c(F)cccn34)=O)C2)C1 C1(C=O)CCN(c2cccnc2)CC1.C1(CNC2C(CC)CCC2)CN(C)CCO1 c1(Cc2c(C)sc(NC(c3cc(C(C)(C)C)n[nH]3)=O)n2)ccc(Cl)c(Cl)c1 c1(C(N2C(C(C)(C)NC(C3CCCO3)=O)CCC2)=O)cncc2c(O)nccc12 c1(N(CC(O)CC2CC2C)CCC)ccc2ccccc2c1 Cc1oc(Cl)nc1C(=O)NC(C1CCCN(C(C2CC(O)(C(F)F)C2)=O)C1)C N1(C(C(COC)O)=O)CC23CCCCC2(C1)CN(C(=O)Cc1cn[nH]c1)C3 c1(C(=O)NCCN(C(COCCC(C)C)=O)C2CC2)ccnn1C(C)C CC1CCC(C(=O)NCCN(C)CCO)CN1C(=O)CCOC(F)(F)F n1(CCC(N2CC(OC)(CNC(C3CC(F)C3)=O)C2)=O)nc(C)c(C)c1C N1(C(C=CC(CC)=CC)=O)CCCC(NC(=O)Cc2ccn(CC(C)C)n2)CC1 C(=O)(C(CCCn1cncn1)N1CCCC(NC(=O)OC)CC1)NC(CC)(C)C N1(C(COC(CC)CC)=O)CCCC1Cc1cn(CCC2CC2(Cl)Cl)nn1 N1(C(C(CC2CN(C(C(CCC)(C)C)=O)C2)F)=O)CC2CN(C)CC2C1 c1(CCCC)cc(CCNC(=O)COc2cccc(OC)c2)n2ncnc2n1 CC(C)(O)CC(=O)N1CC2CC2(NC(c2ccc(N3CCCCCC3)nc2)=O)C1 C1(CNC(C(CC)NC(=O)Cn2cncn2)=O)CCCCN1CC c1(C(C(=O)NC)N(C(C)COC)Cc2ccccc2)ccc(C(F)(F)F)o1 N1(C(c2cccc(C(=O)NC)c2)=O)CCN(C(=O)C(C)C(C)(F)F)CCC1C N1(C(CONC(C2C(C(=O)OC)C=C2)=O)=O)CCC2(CCCCC2)C1 c1(OC)cnc(C(=O)NCC(C(C)C)NC(c2ccnc(Cl)c2N)=O)c(F)c1 Cc1nn(C)c(C(=O)NCCCC(C)NC(C2CCCCNC2=O)=O)c1Cl c1(C(C)C)cc(NCC23CCC(NC(=O)C4=COCC4)(CO2)C3)n2ncnc2n1 N1(C(c2nnc(C)s2)=O)CC(C)(C)CCC1CNC(=O)C(c1ccccc1)F C(C(C)(C)CN(C(C(C)NS(CC)(=O)=O)=O)C)NC(=O)CN(C)NC(=O)C(C)C c1(CNC(CCC=C(C)C)=O)ccc(CNC(=O)CN2CCCC2CCO)cc1 C1(C(C)NC(=O)C=CCC2(C)CCCC2)CCCN(C(C2(F)CC(CO)C2)=O)C1 C(=O)(C(C)CCCOC)NCCCN(C(C=C(CC)CC)=O)CCO c1(CNCCc2c(C)ccnc2)coc2c1N(C)C(=O)CCC2 C12(CNC(c3c(C)cno3)=O)CCC1CCN2C(c1ccc(CO)o1)=O C1(C(=O)NCCOC2CCN(C(C3CCCCO3)=O)C2)CCCC2(CCC2)C1 N1(C(Cc2c(C)ccs2)=O)CCC2(CC1)CCN(C(=O)C(C)OCC(C)C)CC2 Cn1cc2cc(C(N3CCCOC(CNC(C4(C)CC4(C)C)=O)C3)=O)ccc2n1 c1(C(N(CCNC(=O)CCC2CC2(F)F)CC)=O)ccc2[nH]c(=N)sc2c1 C(CC(F)F)(C(=O)N(C1CSC1)C)NC(=O)OC.C1(C)C(=O)N1C N1(C(CC=CC=C)=O)CC2(CC(CNC(c3cc(Cl)cnc3OC)=O)C2)C1 C1(C(CC)NC(c2c(-c3ccco3)noc2C)=O)COCCC1(C)O c1(C(=O)NC(CC(C)C)C(=O)N2CCCC2CO)ccnc2cc[nH]c12 N1(C(=O)OC(C)(C)C)CC(CNCCCS(N)(=O)=O)C(C)(C)C1 C1(N(C(C2(CC)CCCCO2)=O)C)CCCN(C(=O)Cc2cnn(C)c2C)CC1 C1(NC(=O)NCC2CCCCN2)(Cc2cccc(F)c2)CCCCC1 C12(NC(c3c(C)cc(F)s3)=O)CCC(C(=O)NCC3CN(C)CCN3C)(CC1)C2 C=CC(C)C(=O)NCc1cn(CC(=O)NCC2(C)CCCC2)nn1 CC1(C(=O)NCC(CNC(c2ccnc(C3CC3)n2)=O)CO)CCCCO1 c1(C(=O)NC(C(N2CC(C=C)OCC2)=O)CC#CC)cc2ccccn2n1 c1(OC)ccncc1C(=O)NCC1CC(C(=O)N(C2CCN(C(C)C)C2)C)C1 N1(C(CCC2CCN(C(CCCOCCC)=O)CC2)=O)CC(=O)NC(C)C1 c1(C(N(CCNC(C2(OC)CC2)=O)C2CC2)=O)cn(C)c(=O)c2ccccc12 C1(CNC(c2ccc(C)c(Cl)c2)c2nnnn2CC(F)F)Cc2nnc(C)n2C1 c1(CNC(CCN(C(C(C)OCC)=O)CC)=O)cnn(CCO)c1 C(=O)(CS(=O)(=O)CCO)NC1C(NC(c2n(C)cc(C#N)c2)=O)CC1 N1(C(C23C(C)OC(C)(C2)C3)=O)CC2(C1)CN(C(=O)C1=COCCO1)CC(C)(C)O2 C(c1cc2ccccc2o1)=CC(=O)Nc1c(O)ncc(C(=O)OC)c1 C12(C(=O)NCC(CNC(=O)CCn3cnnn3)F)CCCN(CC1)C2 C1(N(C(c2ncn(C(C)C)n2)=O)C)CC2CC1N(C(C1CC3CCC3C1)=O)C2 N1(CCC(=O)NCC2CN(C(=O)Cc3nncnc3O)CCO2)C(=O)CCC1=O C(=O)(C(CNC(=O)C(C(C)C)NC(=O)CC)CC1CC1)NC(C1CC(=C)C1)C#C CC1(C(=O)NC2C=CC(CNC(=O)CC3CNC(=O)O3)C2)CC1(F)F CC1Cc2cc(Br)ccc2C1NC(=O)NCc1ccccc1-c1ccccc1 N1(C(CC(C)(C)O)=O)CC2(NC(c3cccn3C3CC3)=O)CCC1C2 c12cccc3c(cccc13)S(=O)(=O)N2.c1(C(=O)OC)cn(C)nc1OC c1(OC(N(c2ncc(F)cn2)C)=O)cnc(OC(C)(C)C)nc1 C(=O)(CCC(F)(F)F)N1C(C(=O)NCC(c2cn(C)nc2)O)C=CC1 C(CCCC(=O)NCCC(=O)NC(C)(C)CNC(C1CC1COC)=O)OC c1(CNC(C2(CC=C)CCOC2)=O)cccc(NC(C2CC(NC(C)=O)C2)=O)c1 N1(C(Cn2c(C)nc(C)n2)=O)CCC(C)C(CNC(c2ccc3c(c2)CC3)=O)C1 C1(NC(CCC2C(C)=NNC2=O)=O)COC2(CCN(C(C3CSC3)=O)CC2)C1 O=C(C(Cc1ccco1)NC(=O)C(F)OC(F)(F)F)NCC(F)CO C(=O)(CC(C(F)(F)F)P(C)(C)=O)N(CCCNC(C(CC)F)=O)CC N1(C(=O)OC(C)(C)C)CCC2(C1)CS(=O)(=O)CC2C(N1CC(F)(F)CC1CO)=O C(=O)(C(C)CC(C)CC)NCCN(CCC)C(c1nc(Cl)c(Cl)s1)=O C1(CCOCC)CCCN(N(C)C2CCC(OC(C)C)CC2)CC1 c1(CC(=O)NCCCNC(=O)C(F)(F)c2cncs2)ccc(F)cn1 N1(C(c2onc(COC)n2)=O)CCC(CNC(C2CCCCC2C)=O)C(C)C1 C=C1CCN2C(C1)C2=O.C(C(=O)N(C)C)(C(C)C)NC(C(C1CCC1)OC)=O C(=O)(C(O)C(F)(F)F)N1CC(C)(NC(C(N2CC(C)C2)C)=O)C1 N1(CC23C(CN(C(=O)OC(C)(C)C)C2)COCC3)CCc2cccc(Cl)c21 c1(C(N2C3C(NC(C(CCC)OCC)=O)C(CC3)C2)=O)ccc2c(c1)CCC=C2 C(=O)(CC1=CCN(C(C2(O)CCOCC2)=O)CC1)Nc1cc(C)c(C)c(C)c1 C1(CN(C(CCOCCOCC)=O)CC)COCCN1C(c1ccccc1Cl)=O N1(S(CCC)(=O)=O)CCC2CN(C(c3ccc(F)cc3Cl)=O)CC2C1 c1(C(=O)NCCCCCNC(C(F)=C(C)C)=O)ccc2c(c1)C(=O)N(C)C2 Cc1cccc(CC(=O)NC2CC(NC(=O)C(C(C)(C)C)C3CCCC3)C2)c1Cl C(C)(CNC(c1sccc1Cl)=O)(CC(C)C)NC(C(CC1CCCC1)OC)=O C(=O)(CCCC(C)SC)N1C(CNC(C2(OCC)CC(C)C2)=O)CCCC1 c1(CN2CC(C(=O)NCc3cc(N(C)C)[nH]n3)C2)cnn2c1OCCC2 C#CC1(NC(c2ccc(CNC(=O)CC(C)(C)C)nc2)=O)CCOC1 N1(CC=C)CCC(O)(CC(=O)Nc2ccc(Cl)cc2)CC1 N1(C(C(C=C)(C)C)=O)C2CCC1CC(CNC(c1c(C)nsc1NCC)=O)C2 C(=O)(NNc1ccnc(F)c1)c1c(C(F)(F)F)ccc(C#C)c1 C1(CCC(=O)N(CC(C)CO)C)CCN(C(=O)CCC2(C)CC2)CC1 c1(SC)cc(C(=O)NC2(C3CCCN3C(=O)CSc3ccc(Cl)o3)CC2)oc1C CN1CCCCCC1C(N1CC(CCNC(C2(C)COCCO2)=O)C1)=O c1(C(=O)NCC2OCC(CNC(=O)CCOC3CCCC3)C2)cc2occc2s1 c1(C(N(CCC)CCNC(c2cnc(C)cn2)=O)=O)cc2c(cc1O)CCCC2 C(=O)(C1=NOC2(CCOC2)C1)N1C(C2(O)CN(C(=O)CC3CC3)C2)CCC1 c1(C(=O)Nc2cnn(C3CN(C(c4ccnc(CO)c4)=O)C3)c2)cnc(Br)nc1 c1(CNC2CCN(C(c3ccc(Br)cn3)=O)C2)c(C(F)(F)F)cccc1Cl C(C(C)C(C)C(=O)N1CCC(OCC(N2CCCC(C)C2)=O)C1)OC.C1CO1 Cn1ncc(C#N)c1C(=O)NCC1CC(NC(c2cnc(C(F)F)s2)=O)C1 c1(C(=O)NC2C(NC(C(c3cncn3C)N(C)C)=O)C2)c(Cl)cncc1Cl C(C)(CN=c1nc2[nH][nH]cc-2c(O)n1)N(C(c1ncc(CC)s1)=O)C c1(OC)cccc2c(C(=O)NC3CC3NC(c3ccn4nnnc4c3)=O)cnn12 C#CC1CN(C(C2CC(OC)C2)=O)CCN1C(C1CSC(C)=N1)=O N1(C(c2cc(OC)c(Cl)cc2)=O)CCC(C)N(C(=O)C(=O)NC2CC2)CC1 N1(C(N(C)CC2CCCCC2)=O)CCCC(NC2(C(=O)OC)CC2)C1 CCC(C)(CC)C(=O)NC1CC(C(=O)N(C)Cc2cccnn2)C12CCC2 N1(C(C(CCC(N)=O)N)=O)CCC2(CC1)CN(C(c1sccc1Br)=O)CCC2O C(=O)(CCCC(=O)N1CCN(C(C2CC3CC3C2)=O)C(C)C1)OCC N1(C(c2ncc(C)cn2)=O)CCN(C(=O)CC2COC(=O)N2)CC1C(F)F C(CCC(C)(C)C(=O)NCC1C2CCCC1NC2)OC N1(C(C2C(CC)C2)=O)CC2CC(C(=O)NCCC3CCCC34CC4)(C2)C1 c1(OC)ncnc(N2CCC(C(C)NC(=O)CCCNC(C)=O)C2)c1OC c1(C(C(=O)NCCCN(C(c2cc(C(C)C)[nH]n2)=O)CC)C)ccc(C)s1 CC1(C(=O)NCCCNC(=O)COc2ccc(O)cc2)CC2(CC2)C1 c1(C(N2CC(CN(C)C(C34CC(O)C3C4)=O)OCC2)=O)ccc2c(c1)CCCS2 C1(C(=O)NC2(CC#C)CC2)CN(C(c2ncncc2OC)=O)CCO1 C(N=c1[nH]c(N2CC(CO)C3(CCC3)C2)nc2c1COC2)c1ccc(C)nn1 c1(OCC(=O)NC2(C)CN(C(C(CC=CC)C)=O)C2)ccc(Cl)c2ccccc12 Cc1nc2cc(C(=O)NC(C3(O)CN(C(=O)Sc4ccccc4)C3)C)cnc2s1 N1(CCC(=O)N(CCCCN(C(=O)CC2CC23CC3)C)C)CCOCC1=O C1(C(=O)NC2CN(C(C(C(C)O)N(C)C)=O)C2)CCn2nncc2C1 C1(C(=O)NCC2N(C(C(CSC)OC)=O)CC2)CC(=O)NC(=O)C1 Cc1cc(N2CCCC(C)(F)C2)nc(NC(c2nnc3n2CCC3)C)n1 CC1CCC(C)N1C(C1(F)CCN(c2nccnc2F)C1)=O C1(C)(NC(C2C(c3cccc(C)c3)C2)=O)CCN(C(c2ccnnc2S)=O)CC1 CC(N=c1[nH]c(N2CC3CC2C3)nc2cccc(F)c12)c1ccn(C)n1 N1(C(C(C)OCCCC)=O)CC(NC(c2ccc(=O)oc2)=O)C2(CCC2)C1 C1(C(N2CC3C(NC(c4cncc(C#C)c4)=O)C3C2)=O)CCc2n[nH]c(C)c2C1 C1(C(N2CCC(NC(c3ccc(C)c(C)c3)=O)(CF)C2)=O)C2Cc3ccccc3C12 C1(CNC(c2cc(C(C)(F)F)n[nH]2)=O)C(O)C(O)CN1C(c1ccnnc1O)=O Cn1nncc1CC(=O)NCC1CCN(C(c2ccc(Cl)s2)=O)C1 c1(C(CC(=O)NCCCN(C)CC2(SC)CC2)=O)ncccc1C1(O)COC1.C(N)SC c1(C(=O)NCCCC2CN(C(c3ccns3)=O)CCO2)cc2ncccn2n1 C1(NC(C(C)Sc2nc(C(C)C)oc2)=O)CC(Nc2ccccc2Cl)C12CCC2 N1(CCC(=O)NC(CCC(=O)OC)C)CCC2CCNC(=O)C12 C#Cc1ccccc1NC(C1CN(C(=O)CC(=O)CCCCC)CC1C#N)=O C1(N(C(=O)CC2CC2)C)CCCC(NC(c2cn(CCC3CC3)nn2)=O)C1 N1(C(c2c(C)nc(C(C)C)o2)=O)CC(C2CN(C(=O)CC3(C)CCCO3)C2)C1 c1(C(N(C2CCC(C(F)(F)F)CC2)C)=O)cccc(NC(N)=O)c1 C(CC(C)(C)C(=O)NC1CN(C(=O)CCc2cc(F)ccc2)CC1(C)C)OC C1(C)(CNC(C2N(C(C(C)(C)C)=O)CCC2)=O)CCCN1C(=O)CN1CC=CC1 c1(OC)cc(C=CC(=O)NCC2CCN2C(c2ccccc2OC(C)C)=O)sn1 Cc1cc(C(=O)NCC(C)CC(=O)N(c2ccc(Cl)cc2)C)ncc1N N1(C(CC(CCC)CCC)=O)CCCC12CCCN(C(c1coc(C#N)c1)=O)C2 C(=O)(C1CCc2ccccc21)NCC1CN(C(C=CC)=O)CC2(O1)CCC2 CC(C)CC(CF)NC(=O)C(N1CCOC(C2CCOCC2)C1)=O N1(C(CCn2c(C)ncc2)=O)CCC(CNC(=O)CSC2CCOC2=O)CC1 c1(OCC)cnc(C(=O)N(CCCNC(=O)C(C)CO)CC2CCCC2)cn1 C=CCC(C(=O)NCC1CCCC1C(=O)NC1CCCC(C(N)=O)C1)NC(C)=O c1(C(=O)NCC2CC(COC)CN2C(=O)CC(C)(C)O)cc(C)c2[nH]cnc2c1 C(CN=C(NCc1cc(C)cc(C)c1)NC1CCCC(C(C)C)C1)OCC c1(NC(C2CC(F)CN2Cc2ncccn2)=O)cnc2[nH]ccc2c1 C(=O)(C(C)(C)CCCF)NC1C(n2cc(-c3c(C)cc(F)nc3)nn2)CCC1 c1(C(=O)NC2CC(C)CC(C)(C)C2)cc(F)c(F)c(C#N)c1F c1(CN2CCC(CNC(C(C)(c3ccccc3)OC)=O)C2)cc(Cl)c(Cl)cc1Cl CC1CC1(F)C(=O)NC1CC(CNC(=O)CCC2CC2)C1 c1(C(=O)NCC2CN(C(C3CC(C4CC4)C3)=O)C2)cc2n(n1)CCCC2 C1(C(=O)NCC(C)CN(C)C(c2cc(CC3CC3)on2)=O)CCN(C)C1=O C1(NC(C(C)(C)NC(=O)CN)=O)CS(=O)(=O)CC1Nc1ccccc1 CCCC(C(=O)N(C)CCN(C(=O)Cn1ccc(=N)[nH]1)C)NC(N)=O CC1CN(C(c2conc2CNC(C2CCC3(CC3)C2)=O)=O)CCO1 N1(C(C=CC)=O)CCC(N(CCC)C(c2cnn(-c3nccs3)c2)=O)CC1 c1(NC(C2(CNc3nc(C)nc(O)c3)CC2)=O)cc(S(=O)(=O)O)ccc1O C12(CC)CC1CN(C(c1ccc(C(N)=O)cc1)C(=O)NCCC#N)C2 N1(C(c2c(C)nnn2C)=O)CC(C)CN(C(=O)CCC(C)C)C(C)C1 Cc1cc(C)c(CC(=O)N(C2CCC(NC(=O)Cc3cnoc3)CC2)CCO)s1 C1(O)(C(C(=O)NC(C)CCNC(=O)C(C)C2CCC2)(F)F)CCCCC1 C1(C(=O)NCC2(COC)CN(C(c3cccc(CO)n3)=O)C2)CCCS1(=O)=O N1(C(C(COC)C)=O)CC2(CCOCC2)CC1CNC(=O)CCS(C)(=O)=O N1(C(C2(NC(c3c(C)n(C)cc3)=O)CC2(C)C)=O)CCC(O)C(C)C1 N1(C(CCCC)=O)CCC(NC(c2ccns2)=O)C(c2ccccc2)C1 c1(CCC(=O)NCC2(C)CCN(C(c3c(C)n[nH]c3)=O)C2)c(F)cccc1Cl C(C(=O)NCCN(CC(C)O)C(=O)CSC(F)F)(C(C)C)n1cc(C)nc1 C1(CNC(N2CCC(NCc3ccccn3)CC2)=O)CC2CC(C1)C2 CC1CCN(C(=O)CCNC(=O)Cc2ccon2)C1C c1(C2(C(=O)NCC(CC(CC)CC)O)CC2)ccc(S(=O)(=O)CCO)cc1 c1(C(=O)NCC2CC(C)C2)nc2ccccc2n(C)c1=O CC1CN(C(=O)CP(C)(C)=O)CC1(C)CNC(=O)Cc1ccnn1CC#N N1(C(c2c(N)ncc(Br)c2)=O)CCC2CC1CN(C(=O)CC1CCC3CC13)C2 C12C3CC4C(C3n3cc1nn3)C24.C(=O)(CC(O)CCSC)NC(CCCC)=O c1(OC)cc(Cl)c(C)cc1NC(=O)CC1CCN1C(=O)Nc1ccnn1C c1(NC(=O)CC2CN(C(c3nc[nH]n3)=O)CCO2)c[nH]c2ncccc12 C1(NC(C=CCN(C(C=Cc2cc(C)no2)=O)C)=O)CC2OCCCC12 n1(CC(=O)NC2CN(C(C3C(C)OC(=O)N3)=O)CC2O)ncn2nccc2c1=O C(=O)(CCCC(C)(C)C)NCCCC(C(N1CC(C)C(O)C(C)C1)=O)O N1(C(CCC=CCC=C)=O)CCC(CC)C1CNC(c1ccsc1OC)=O Cc1sc(NC(=O)Cc2cc(O)n[nH]2)nc1C(C)C C1(NC(C2C(C=C)CC2)=O)CC2(C1)CC2NC(=O)CCCN1CCCCC1 c1(C(C)C)ccc(C(=O)NC2CCN(C(=O)CCCNC(N)=O)CC2C)c(F)c1 c1(CC)nc(N(C)CC2CCN(C(=O)C3=CCCS3)C2)c2ccsc2n1 Nc1cc(F)cc(F)c1C(=O)NCC1CC(CNC(=O)C2=CCOCC2)CO1 C1(C(=O)NCCC(CNC(=O)CC(C)OC)OC)(OC)CCCCC1 c1(SCC)ccccc1C(=O)NC1CCC(NC(C2CC(O)CN2C)=O)C1 CC(C)CCC(=O)NCCC1CSCCN1C(=O)COCC1CCOC1 C1(=O)CCCC(=O)c2sc(c(C)n2)C(=O)NCC#CCN1CC.C(=O)(NCC)NC C1(COC)(NC(c2cc(C)oc2C)=O)CCN(C(=O)C2=CCCS2)CC1 O=C(C1=CCCO1)NCCCCC1CCCN(C(=O)CN2OCCCOC2)C1 c1(CN(C(=O)COC(C)(C)CNC(c2cncs2)=O)C)ncccn1 c12cccc(c1)C(=O)NC(C1CC1)C(=O)C2=O.C1(C(=O)NCCNNC)CCCC1 c1(C(N2CC3(CC(NC(C4ON=C(C)C4C)=O)C3)C2)=O)cc2ccncc2s1 C1(CNC(C2ON=C(C)C2)=O)CC2(C1)CN(C(=O)CN1CCN(C(C)C)CC1)C2 c1(C(N2CCC(C)C2CNC(C2CC(OC3CC3)C2)=O)=O)cc(O)ccc1Cl C(=O)(C(C)C(O)C(C)C)NCc1oc(C(=O)NC(CC=C)CC=C)c(C)n1 C1(O)(C(C)NC(C2(CO)CC2)=O)CCN(C(=O)C(C)(O)c2ccccn2)C1 c1(CC(=O)NCCC(C)NC(C2(CO)CCCO2)=O)ccc(Cl)c(F)c1 c1(C(=O)NC(C(c2c(OC)cccc2)NC(=O)C=C(C)C)C)ccc(O)cc1C CC(CCC(=O)NCC(C1CCC1)NC(c1cccc(N)c1)=O)N(C)C N1(C(c2nnc(C)s2)C(=O)NC(C(=O)OC)C)CCOC2(CCCCC2)C1 C(=O)(CC1=NN(C)C(=O)C1)NCC1(O)CN(C(C2CC(CCC)OCC2)=O)C1 N1(C(C2C(OC(C)=O)C2)=O)CCCC1CC(=O)NCCCc1ccsc1 CC1CN(C(C2CC2C)=O)CCC1NC(=O)CCc1cncc(F)c1 c1(C(C(=O)NC)N(CCCN2CCOCC2)C)ccc2c(n1)CCC2 C(=O)(CC1=NNC(=O)C1)NCCNC(c1ccc(Cc2ccccc2)[nH]1)=O N1(C(c2c(C)cc(F)cc2)C(=O)NCCCF)CCCCCCC1C Cc1cc2[nH]c(C(N3CCC4(CC3)CC4NC(c3ccnc(C)n3)=O)=O)cc2o1 C1(CC(=O)O)CCCCN1C(=O)NCc1nc(C2(N(CCCO)C3CC3)CC2)n[nH]1 c1(C(=O)OCc2cccc(C(=O)OC(C)(C)C)c2)cncc2cnccc12 c1(N(C(=O)C(=O)N2CC(c3ccncc3F)C2)C2CC2)cc(F)c(F)cc1I C(C(=O)NCC(C)(C)NC(=O)Cc1cccc(OCC#N)c1)(C(C)C)OC c1(C(=O)NC2CN(C(C(CC(=C)C)NC(C)=O)=O)CC2O)nc(C)c(C)[nH]c1=O C12(CNC(c3c(CC)occ3)=O)CCC1CCN2C(=O)CCc1cccc(Cl)c1 c1(C(N2CC(O)(CNC(C34CC3C4)=O)C2)=O)sc(O)nc1O CC1CCN(C(C2CC3CC2C3)=O)CC1(F)F.CC(C)(CNC(=O)OC(C)(C)C)O C=CCC(CC=C)C(=O)NC(CNC(c1cc(Br)c(Cl)s1)=O)CC(C)C C1(CC)COC(C)(C)CN1C(=O)CC(C)(C)CNC(=O)CN(C)S(N)(=O)=O C1(NC(C2(COC)CCC2)=O)CN(C(c2ccnc(C)c2)=O)CC1OC C(=O)(N=c1ccc(NC(=O)OC(C)(C)C)n[nH]1)NC(CC(=O)NC)CN=[N+]=[N-] CC(C)(C)CC(O)C(=O)NC1CN(C(c2c[nH]nc2-n2cnnn2)=O)CCC1F C1(CNC(c2ncnc(O)c2Br)=O)CCCCC(O)C1 C1(CNC(C=CCCC)=O)CC12CCN(C(C1(N(C)C)CCCC1)=O)CC2 N1(C(CCCC#N)=O)CCC2CCCC12C(=O)NOCCOCCN(C)C N1(CC(N2CC(n3cc(-c4cccs4)nn3)C2)=O)CCOCC1 C1(C)CC=CCN1C.C1C(O)CCNC(=O)C=CC(=O)N1.CC(Cl)=C c1(C(N2CCC3CN(C(C45CCC(CO4)C5)=O)CC23)=O)c(N)ccc(F)c1F Cc1ccc(C2CC2NC(=O)N(CCC2CC2)C(C)C)cc1 C(CC(=O)N(C(C)CC(C)C)C)(C(F)(F)F)NC(c1c(C)nsc1)=O CCCCS(=O)(=O)NCC(=O)NCC1CC1NC(=O)C(N1C(=O)CCC1=O)C N1(C(c2sc(CC)c(C)c2)=O)CCC2C1CCCN2C(C1CC1COC)=O c1(C(N2C(C)CCC(NC(=O)Cc3cc[nH]c3)C2)=O)ccc2nc(O)oc2c1 C(=O)(CCCCCCc1ccccc1)NCC1N(C(CNC(=O)OC)=O)CCC1 CCCCCCCC(=O)NC(C1CCCOC1)C(=O)NCC(C)(C)C(C)(C)C c1(C(N2C(CCC)CN(C(=O)CSC(C)C)CC2)=O)cc2cc(Cl)sc2[nH]1 N1(C2CN(C(CSC(CC)CC)=O)C2)CCN(C(=O)COc2cc(C)no2)CC1 c1(C(N(C2CN(C(c3cc(Cl)cc(Cl)c3)=O)C2)C)=O)ccc(S(C)(=O)=O)s1 O=S(=O)(c1cnc(NCCCn2cnnc2)c(Cl)c1)NCC1CC=CC1 c1(C(=O)OC)cc(=NC(=O)c2ccccc2-c2nc(C)n[nH]2)[nH][nH]1 C1(CC#C)(C(=O)N(C2CC(SC)C2)C)CCN(C(C2(C)CCCCO2)=O)C1 N1(c2ncc(C)cc2Br)CCCC2(NC(c3cnc(Cl)cc3Cl)=O)CCCC12 c1(OC)ccc(O)cc1C(N1CCCC(N(C)C(c2ccc(O)cc2)=O)C1)=O C1(C)(CNC(C(C2CCN(C(C3CC(CF)C3)=O)CC2)C)=O)CC2CCC1C2 S(=O)(=O)(c1cccc(F)c1)N1CCN(C(c2c(Cl)ccnc2Cl)=O)CC1 C1(NC(Cc2ccc(OC)nn2)=O)C(C)CCN(c2ccnc(C3CC3)n2)C1C N1(C(Cc2n(C)ccc2)=O)CCCN(C(C2Cc3nnsc3S2)=O)CC1 N(C(=NCCN1CCCCC1)NCCN1CCCC1=O)CC(c1ccc(C)o1)O C1(N(C)C(C2CCC(=O)O2)=O)CCCC2CN(C(=O)Cc3ccnn3C)CC12 c1(C(N2CCC(NC(c3onc(COC)n3)=O)C23CC3)=O)cccc2nn[nH]c12 C1(CC)CN(C(c2cocc2C)=O)CCC1NC(=O)CCn1ccc(C)n1 Cc1c(C(=O)NC2CCC2NC(c2cnc(C(C)(C)C)o2)=O)cccc1N C1(C)(C(N(CCC#C)CCO)=O)CCCN1C(c1ccc(C(F)(F)F)nc1)=O N1(C(C=CC)=O)CC23CCCCC2(C1)CN(C(=O)C(C)NC(=O)CC)C3 C1(C(=O)NCCOCCNC(C2C(C(C)(F)F)C2)=O)CCCCO1 N1(C(c2nn(C)c(O)c2)=O)CCCC(C2CN(C(=O)C=CC3CCCO3)C2)C1 c1(C(=O)NC(C2CCN(C(c3cc(C4CCC4)[nH]n3)=O)C2)C)ccc(F)cc1Cl C1(F)(C(=O)NC(C)(C)C)CCN(C(C)=O)C1.C(C(C(=O)O)N(C)C)SC c1(N2CC(C(C)C)OCCC2)ccc(S(=O)(=O)NCC(N)=O)cc1F CC(CCNC(C1CC2CCC1O2)=O)CC(=O)N1CC(OCCN(C)C)C1 C1(C)(C(N(CC#CC)C)=O)C=CCN1C(C1CC(C)(F)C1)=O c1(C(=O)NCCC2CCC(NC(=O)Cc3ccoc3)C2)cc(O)ccc1F c1(OC)cnc(C(=O)NC2CC(CCNC(c3cccc(C#N)c3)=O)C2)c(F)c1 C12(C(=O)NCC3C(NC(c4ccc(CCF)cc4)=O)CC3)CC3CC1C2C3O Cc1nc2c(o1)CCCC2CC(=O)N(CCc1cccc(F)c1)C(C)=O c1(CN(CC=CCNC(CSC)=O)C(C2CC2F)=O)ccc(Cl)nc1 N1(C(=O)CCNc2cccc(F)c2)CCCCC1C1CCCN1Cc1cccs1 c1(C(=O)NC2C(C)CN(C(c3coc(Cl)c3)=O)C2)cc2cc(N)ccc2[nH]1 CCCC(C)(CC)C(=O)NCC(F)(C(N1CC2(COC(C)C2)C1)=O)C(C)C C(C(C)(C)CC(=O)NCC(C)CC(C)C)NC(c1nc(C)sc1)=O C12(CNC(C3C(CC)C3)=O)CCC(CN(C(=O)C=C(C)C(C)(C)C)C1)C2 C1(C(N2C(C3CCN(C(c4cc([N+](=O)[O-])c[nH]4)=O)C3)CCC2)=O)CC2CCC1CC2 N1(C(c2n(CC)ccn2)=O)CC2(CC2)CC1C(=O)NC1CN(C)CCC1O c1(CC)cc(F)ccc1C(=O)N(C(C)CNC(c1cscc1F)=O)C CCC(CCCC(=O)N1CCCC(N=[N+]=[N-])C1)NC(c1occc1C)=O c1(CSCC(=O)NCC2CCC(NC(CCCOCC)=O)C2)cccc(C#N)c1 c1(SC(N2C(c3cn(C(C(=O)OC)C)nn3)COCC2)=O)ccc(N)cc1C C12(CC(N3CCC(C(C)(C)C)C3)=O)CCC(CC1)C2.C12CC1NC2=O C1(NC(CC2CCC(C)C2)=O)CC2CCC1N(C(=O)CNc1ccccn1)C2 c1(C(=O)NC2(CNC(C3C(C=C)C3)=O)CCC2)cc(C)nn1C1CCC1 c1(C(C)C)ccc(C#N)c(N2CCN(C(=O)CCc3cnn(C)c3)CC2)n1 c1(CC)ccc(C(=O)NCC2CC3(CC3)CN2C(=O)C(C)(C)C2CC2)cc1CC c1(NC(C2C(CNC(c3cccc(F)c3F)=O)C2)=O)nc(Cl)cnc1Br N#Cc1ccc(C(N2CCC2CNC(C2CC(n3cnnc3)C2)=O)=O)c(F)c1 N1(C(C2=C(C)OCC2)=O)CCC(C2CC2)C1CNC(c1ccc(O)cc1F)=O C#CC(C)(C)C(=O)NCC(=O)NCC(=O)NC1CCCC(SCC)C1 C1(COC)(NC(=O)C2=CCCOC2)CCN(C(c2csc(C(C)=O)c2)=O)CC1 c1(C(c2n(CC)nnn2)NC(c2nc(C)cs2)C)cccc(OC)c1OC Cn1cnnc1CC(=O)NCC1CC1NC(C1C2CCCC12)=O C(=O)(CCCCC(=O)O)N(C(c1cn(Cc2nc(C(N)=O)cs2)nn1)C)C C1(C(=O)NC(C2CCCN2C(c2cnoc2C2CCC2)=O)C)CCC(C)(C)O1 CCCCC(O)CCC(=O)NCC12CC1CN(C(c1cc(C)c(N)cn1)=O)C2 c1(C(=O)NCCCOCCNC(C(C#N)=C(C)C)=O)n[nH]c(C2CC2)n1 Cc1ncc(C(=O)NC(C)(C)CCNC(=O)C(C)C2CCOC2)cc1C#N CCC(C)(C(N)=O)NC(=O)CCN(C(=O)Cc1cnccc1C)C(C)C c1(C(N2CC3C(CNC(=O)C(F)C(F)(F)F)(C3)C2)=O)ccc2c[nH]nc2c1 N1(C(C(CC)n2cncn2)=O)Cc2n[nH]cc2C1C(=O)Nc1cccc(OC)c1 N1(C(c2c(CC)[nH]cc2)=O)CCN(C(=O)CCCCOC)C(CC(F)(F)F)C1 CC(C)(F)C(C)(F)C(=O)NCCCCC(=O)NC12CCCN(CC1)C2 C(C)(CCc1ccco1)(c1nnnn1C1CCCCC1)NCC(C)(C)F c1(C(=O)NCC2C(C)(C)CCN(C(C(C)CO)=O)C2)ccc2cnccc2c1 CCC(CC(=O)N1CCCCC1C(C)(C)CNC(=O)CN(C)CCOC)C(F)F C1(NC(c2cc(COC)no2)=O)C2CC(NC(=O)COC3CC3)CC12 N1(CCCN(CCC)C)CCN(N2CCC(CC(=O)OC(C)C)CC2)CC1 N1(C(c2c(C)cncn2)=O)CCN(C(c2ccc(Cl)s2)=O)C(CO)C1 c1(-c2n(CCOCC)nc(CCO)n2)cnc(C)nc1O C(=O)(C1=C(C)S(=O)(=O)CC1)NCC1C(NC(C2CC(OC)C2)=O)CC1 n1(CC(N2C3C(NC(CN(CCOC)C)=O)C(CC3)C2)=O)ncc2cccnc12 Cn1c(C(F)F)nc2cc(C(=O)NCC3CCCC3NC(=O)C=CCO)ccc12 c1(C(N2CC(CN(C(=O)CC3CC3)C)C2)=O)cc(COCCO)[nH]n1 CCC(C)C(=O)N1CC(C(C(=O)N2CC(c3cccs3)C2)OC)C1 CC12C3C4C1C1C2C3C41C(=O)NC1(C)CCCN(C(=O)CC2CCS(=O)(=O)C2)C1 n1(CCC(N2CCC(N(C(C(C)C)=O)C)CC2)=O)cc(C#N)c(O)nc1=O c1(CN(C)C(c2cnnn2C)=O)ccccc1CNC(=O)C(O)Cc1cnc[nH]1 CCC(C(=O)N1CC(NC(c2ccc(OC)c(Cl)n2)=O)C(C)(C)C1)C(C)(C)CC C1(NC(C(N2CCOCC2)C)=O)CN(C(c2c(CO)cnn2C)=O)CCC1CO CC(C)C(C(=O)NCC(C)(C)CN(C)C(C1(C)CCCOC1)=O)NC(N)=O C(=O)(C1CCCc2nc(C)[nH]c21)NCC(C)NC(c1c[nH]c(=NCC)s1)=O C(CNC(=O)CC1(N(C(=O)CNC(N)=O)C)CC1)(C1CC1)SC C1(CC=C)(NC(=O)CN(C)CC)CCN(C(c2cn(-c3ccccc3)cn2)=O)C1 C(C)(CCCCNC(=O)C(C)(C)c1cscc1Cl)NC(C(C)OC1CC1)=O C1(C)(NC(C(=O)NCCC2(C(=O)OC)CCC2)=O)CCC(=O)N(C)C1 N1(C(Cc2c(C)occ2)=O)CCCN(C(=O)CN2CCn3ccnc3C2)CC1C C(=O)(C1COc2ccc(Cl)cc21)NC(CC)CNC(C1CC1(C)C)=O c1(OC)ccc(C(=O)NC2CCC(CNC(C3(O)CCC3)=O)C2)c(OC)n1 c1(CNCC(O)CN(C)C(c2ccc(Br)cc2OC)=O)ccc2c(c1)CNC2 O=C1CC(C(=O)N2CC(O)C3CCCC23)=NN1c1ccccn1 N1(C(C2C(C)CCO2)=O)CCC(O)(CNC(=O)CCn2cc([N+](=O)[O-])cn2)CC1 Cc1ccccc1S(=O)(=O)CC(=O)N1CCC(NC(c2occc2Cl)=O)C1 C1(c2cn(C3CCCCN(C)C3)nn2)CC2CCC(C1)N2C(=O)Cc1ccon1 C(=O)(C(=O)N=S(C)(C)=O)NC(C)C(CO)NC(=O)C(c1noc2ccccc12)C N1(C(c2c(C)noc2)=O)CCC2(CCC(NC(=O)CCc3cnco3)CC2)CC1 c1(C(=O)NC(c2ccccc2F)CNC(c2cc(C)[nH]n2)=O)ncc2[nH]ncc2n1 C1(CC=C)(NC(C23CCC(OC)C2C3)=O)CCN(C(=O)C=CC(C)(C)C)C1 c1(C(=O)OC)ccccc1NC(=O)CCN(CC1CCC1)Cc1ccccc1F c1(COn2c(Cc3nc(C)sc3)nc(-c3nccs3)n2)cccc([N+](=O)[O-])c1 C1(C)(C(N2CC(C)(CC)C2)=O)CN(C(=O)CCOC(C)CC(C)C)CC1C C(C(C(C)(C)C)NC(=O)Nc1ccccc1)NC(=O)NC(C)CC1(O)CCC1 CN1CCN(C(C2CCN2C(=O)CCc2cnco2)=O)CC1=O C1(CNC(C(C(=O)NC)(C)C)=O)CC2CCC(C1)N2C(=O)C#CC1CC1 Cc1sc(C)c(C(=O)N(C2CCCN(C(=O)CCC3CCCCC3)C2)C)c1C#N C1(CCNC(c2scc(C)c2)=O)CCCN(C(C2CCN(C)C2=O)=O)C1 C1(NC(C2(N(C)C)CCCC2)=O)CC2CCC(C1)N2C(=O)CCCNC(N)=O c1(C(=O)NCC2CCC2C(=O)NCC2CC(F)C2)cccc2cncn12 Cc1cc2c(C(N3CCC(NC(c4sccc4C(F)F)=O)CC3)=O)cccc2[nH]1 n1(CCC)cc(Cl)c(C(=O)NC(C2CCCC2)CNC(=O)CC2CCCO2)n1 c1(CN2CCC(CC)C2)ccnc(C(=O)N(C)NC(C(C2CC2)OCC)=O)c1 C1(C)(C(=O)NCCc2nc(C(=O)OCC)c(C)o2)Cc2ccccc2N1 C1(NC(C(=C(C)C2CC2)F)=O)CCC2CCN(C(c3coc(C4CC4)n3)=O)C1C2 N1(C(CC2OCCN(C(c3ccc(CC)s3)=O)C2)=O)CCC12CCC(C)CC2 c1(C(=O)NCC23N(C(CNS(NC)(=O)=O)=O)CCC2CC3)ccc2ccccc2c1 C1(C(=O)NC(C(C(CC)C)ONC(=O)OC)CC)C2CC3C(C2=O)C13.C(C)(C)(C)O CCC1=C(C(=O)NC(CNC(c2cccnc2SC(C)C)=O)C(C)C)SCCO1 c1(C(=O)NCC2CN(C(C(C)NC(N)=O)=O)C2)ccc(CSc2ccccn2)o1 C12(CCC1)C(C)(C)OC2=O.N1(CC(=O)NCCC)CCC1C1CCOC1 N1(C(c2cc(C(C)=O)oc2)=O)CC2OCCN(C(c3cc(CO)nn3C)=O)C2C1 Cc1cc([N+](=O)[O-])ncc1C(N1CC(O)CC1CNC(c1nnccc1C)=O)=O C1(NC(CC2CC(NC(c3ccc(C(N)=O)[nH]3)=O)C2)=O)CCCCCC1O C1(S(N)(=O)=O)(C(=O)NC2(CNC(c3cnc(C(C)O)s3)=O)CCOC2)CC1 c1(C(N2CC(C)C(NC(=O)CC34CCCC3C4)C2)=O)cc2c(nn1)OCCS2 C1(NC(CCc2ccc(C)o2)=O)CN(C(c2cc(C#N)cn2C)=O)C(C)(C)C1 CN1C(=O)NCC12CN(C(C1CC3(CC3)CN1C(=O)Cc1cc[nH]n1)=O)C2 c1(C(N2CCC(C(F)F)(CNC(COC(CC)C)=O)C2)=O)cncc2ccsc12 N1(C(c2ccc(O)nc2)=O)CCC(NC(C2(Br)CCC2)=O)C(F)C1 c1(OC)ccc(CNC(=O)CCc2c(F)cccc2Cl)c(OC)c1OC c1(C(=O)NCC(CSC)OC)n[nH]c2cc(O)ccc12 N1(C(C2(OC)CCCC2)=O)CCC(F)(C(=O)NCC2CCC=CO2)CC1 C12(C(=O)NCC3(NC(N)=O)CCCC3)CC1CCN2C(=O)C(F)=CC1CC1 Cc1coc2ccc(C(N3CCC4CCN(C(=O)CCCN(C)C)C4C3)=O)cc12 c1(OCC)ccc(C=C(CNCc2cccc(C(F)(F)F)c2F)C(F)(F)F)cc1 c1(C(N2CCC(NC(C(COC)O)=O)C2)=O)cc(C)cc(O)n1 N1(C(C(=O)NC2CC2c2nc3ccccc3s2)=O)CCn2ncc(Cl)c2C1 N1(C(COc2ccc(C#N)cc2)=O)CCC2(C1)CN(C(C1CCC3CCC13)=O)C2 N1(C(c2n[nH]c(C)c2Cl)=O)CCC(F)(CNC(=O)COCC(F)F)CC1 C(C(C)(C(=O)NOCC(O)C(C)C)NC(c1cc(C)nnc1O)=O)SC c1(C(=O)NCC2(NC(Cc3cn(C)nn3)=O)CCOC2)ccc2c(c1)COCO2 Cc1ncc2n1CCC(C(N1CC(C3(NC(C4COC(=O)N4)=O)CC3)C1)=O)C2 CCC(CC)(CC)C(=O)NCC12CC(C1)C(NC(c1cc(C)cc(F)c1)=O)CO2 c1(C(=O)NC2CC(F)(CNC(c3c(NC)nccc3)=O)C2)ccc([N+](=O)[O-])cc1 Cn1nccc1NC(C1CCN(C(=O)CC(=O)N(C)C)C1)=O C1(CN(C(c2ccc(C(C)C)o2)=O)C)CCCN(C(C2(C)CCC(=O)C2)=O)C1 Cn1c(Cl)cnc1CN1CCC(NC(c2snc(Cl)c2Cl)=O)CC1 C(c1ccco1)=C(C)C(=O)N(CC(C)N(C)C(c1ccc(C(C)C)o1)=O)C Cc1cccc(CN2CC3C(C2)N3C(c2cc(C3CC3)no2)=O)c1 C1(CN(CC(N2C(CC)CCC2)=O)C)CCN(C(c2sc(CO)nc2C)=O)CC1 C#Cc1ccc(CN2CCC(C(=O)NC(Cc3ccc(OC)cc3)CO)C2)cc1 C1(O)(CNC(c2sc(C)c(O)n2)=O)CCN(C(=O)CC(F)(F)F)CC1 C1(C(=O)NCC2(C)CCN(C(C3CC(C#N)C3)=O)C2)CC2CC(C1)CC(F)(F)C2 O=C(C1CCCc2nn[nH]c21)N1CCCC1C(C)(C)NC(C1CC(O)C1)=O C12(C(N3C(CCNC(c4ncn(C)n4)=O)CCC3)=O)C3C4C1C1C2C3C41C(N)=O c1(N(C)CCc2cn(CC3CCCO3)nn2)ccc2c(c1)nc(C(F)F)n2C CCCCC(CC(=O)NCC1CCCN(C)C1=O)NC(=O)C(C)COC(C)=O c1(C(N2C(CNC(C3CC=CCC3)=O)CC(F)C2)=O)cnc2[nH]ncc2c1 C12(C(N(CC#C)C3CC3)=O)CCN(C(c3cc(C(N)=O)c[nH]3)=O)CCC1C2 N1(C(C2(C)CC(C)(C)C2)=O)CCC(O)CC1C(N1CCC1c1ccccc1)=O Cc1cc(C(=O)NCC23CC(CO2)N(C(=O)Cn2nccn2)C3)ncc1C(N)=O N1(C(=O)Cc2ncc(F)cc2F)CCC2C(CCCN2C(c2ccc[nH]2)=O)C1 c1(C(=O)NC2(C)CC(NC(C3C(C(C)=O)CCCC3)=O)C2)ccn2cncc2c1 C1(CC(=O)NCCC(CNC(c2c(C)nco2)=O)O)Cc2ccc(Cl)cc2C1=O N1(C(C(COC)O)=O)CCCC2(CCN(c3cc(SC)ncn3)C2)C1 CCC(CC(=O)N1CCN(C(=O)CSS(C)(=O)=O)CC(C)C1)C(C)C CCC(CNC(=O)CC(C)(O)c1ccccc1)(CC)NC(=O)C(C1CC1)N(C)C N1(C(CC(C(F)F)NC(c2c(NCC)scn2)=O)=O)CC2(CCC1CO)CC2 c1(NC(C2CN(C(Cc3ccc(C)cc3)=O)C2)=O)cc(Br)c(C)cc1F N1(C(CCCC)=O)CCC(CNC(c2conc2CC)=O)(OCC)C1 C1(NC(CC(=O)NCC)=O)CCN(C(=O)CCc2ccnc(C)n2)CC1O C1(C(=O)NCc2ccc(-c3ncco3)cc2)CCNC2(CC2)C1 c1(C(N2CCC(F)(CNC(C=COCC)=O)C2)=O)ccc2[nH]c(=O)c(=O)[nH]c2c1 C(CCCCCC(=O)NC(c1n[nH]c(CC)n1)C)NC(c1ccc(C#C)nc1)=O C(C(C)(C)C(=O)NCC1CCC1(F)F)N(C(Cc1c(C)ocn1)=O)C C1(CC)CN(C(c2csc(CC3CC3)n2)=O)CCN1C(=O)CC1(O)COC(C)(C)C1 Cc1noc(C)c1CC(C)C(=O)NCCC1CC(NC(c2c(C)noc2C)=O)C1 CCCC(C)(CC)C(=O)NCCC1(NC(=O)C=Cc2nnc(C(C)C)o2)CC1 C(C(C)N=c1ccc([N+](=O)[O-])c(O)[nH]1)c1ccc2n[nH]c(C)c2c1 n1(CCOC)cnc2c(NC(C)COC)[nH]c(=NC3C4CCC(C4)C3C)nc12 C12(NC(c3cc4scc(Cl)c4[nH]3)=O)CCCC1(F)CN(C(c1cc(F)n[nH]1)=O)C2 C1(C(=O)OC(C2CCCN(C(=O)OC(C)(C)C)C2)C2CC2)CCC(=C(F)F)CC1 c1(C(=O)NCC2(O)CN(C(c3ccc(Cl)cc3I)=O)C2)ccc(C(F)(F)F)cc1F N1(C(c2ccc(CCC)s2)=O)CC2=C(C1)CN(C(c1ncccc1Cl)=O)C2 N1(C(C2CN(C(c3c(C)cc(Br)s3)=O)CC2(F)F)=O)CC2C3CCC(C3)C2C1 Cc1cccc2c1c(CNCC1C(C(=O)Nc3nccc4[nH]ccc34)C1)cn2C N1(C(C(COC)COC)=O)CCCC(CC(=O)N(CC(C)OC)C)C1 N1(CC=C)CCC(N2CCC(N(C)C(c3cc(C)nn3C)=O)C2)C1=O C1(C(=O)NC(CC=C)C)CN(C(c2ocnc2C)=O)CC(C)(C)C1 N1(C(C(C)=C2CC2)=O)CCC2(CC1)CN(C(c1cnc3n1CCC3)=O)C2 c1(CCN2CCOCC2)ccnc(Br)c1.c12cccc(c1)NCC(=O)NCC2C c1(C(N2CCCC(c3ccccc3)CC2)C(=O)NC2(C)CC2)ncc(Cl)cc1F C1(C(=O)NC2CC(CNC(=O)CC3CCCC(=O)N3)C2)CC12CCSCC2 c1(C(N(CC(CC)NC(c2cnn(C3COC3)c2)=O)C)=O)ccc(Cl)cc1 N1(C(C(C)NC(C2CCC2)=O)=O)CC2(CCN(C(=O)C(C)N(C)C)CC2)C1 c1(C(N(C(CNC(c2ccc(C(=O)OC)n2C)=O)C)C)=O)cccc2cncn12 c1(NC(C=CCNC(C(CC)n2cncn2)=O)=O)cccc(CO)c1C c1(CC(=O)NCC2CCN(C(C(C)(C)OC(C)=O)=O)C2)ccc2c(c1)COCC2 C1(OC)CN(C(=O)N(C)C)CCC1CO.c12cccc(c1)NC(=O)N2 CCCCCC(O)CC(=O)NC1C2CC3C1C3C2C(N1CCCC(F)(CO)C1)=O c1(C(=O)NC(CNC(CCCCC#C)=O)(C)CC(C)C)cc(C)c(F)cc1F c1(C(=O)NC2(CCNC(C3CCCC(C)C3)=O)CCC2)ccc2[nH]ccc2c1 N#Cc1cc([N+](=O)[O-])cnc1NC(=O)CN1C(=O)COC(C(F)(F)F)C1=O C1(C(=O)OC)CCC(F)(CN)CC1.c12ccc(C(F)(F)F)cc1NC2=O C12(C(=O)OC)CC(N(C)C(=O)NCC3CC3C#N)(C1)C2 c1(OC)ccc2scc(C(N3CCCC(C)(C#N)C3)C(=O)NC3COC3)c2c1 C1(C(N2C(C(N3CC(n4ncccc4=O)C3)=O)C=CC2)=O)CC2(CCC2O)C1 C(c1ccc(C)nc1)=CC(=O)NCC(C)NC(C(C)Oc1c(OC)cccc1)=O N1(C(C2(C(C)C)CCC2)=O)CCC(CN(C)C(c2cc(Cl)ns2)=O)C1 Cc1cnn2ccc(C(=O)NCC3C4CC3N(C(c3ccnn3C)=O)C4)nc12 C(=O)(CCC(C(C)C)NC(=O)Cc1cnn(C)c1)NC1CN(C(CC)=O)C1 c1(N2CCN(C)C(=O)C2)nc2ccsc2c(=NC2CCC3CC2CO3)[nH]1 c1(C(N2C(CNC(c3c(C)onc3O)=O)CCC2)=O)cc2n(c1)CCOC2 C#Cc1ccc(C(=O)NC2CC(F)CN(C(=O)CC3CCCC(OC)C3)C2)cc1 C1(C(N(C)Cc2ccncn2)=O)CCCN1NC(=O)c1ccccc1 N1(CC)CCC(C(=O)NCC2(O)CN(C(c3sccc3C3CC3)=O)C2)C1 c1(C(=O)NC2CCC(CNC(C3C(COC)C3)=O)C2)cnc2n1CCCC2 C1(C#N)(OC)CC(C(N2CC3C(NC(=O)CCc4ccccn4)C3C2)=O)C1 c1(C(=O)NC2C(N(C(C(C)=CC)=O)C)CCCC2)cc2n(n1)C(C)CCC2 O=C(C1=NOC2(CCN(C(C3CCC=CCC3)=O)C2)C1)NCCN1CCCC1 CCC(=O)CCC(=O)N1CC(C(N2CC(C)(CCO)C2)=O)C(F)(F)C1 c1(C(=O)NC2(CC=C)CCN(C(=O)C(F)CC=C)C2)ncnc2ccsc12 c1(C(=O)NC(CC(C)C)CNC(c2cnn(C)c2N)=O)ccc2cn(C)nc2c1 C1(O)(CNC(c2cc(OCC)ncc2)=O)CCN(C(c2occc2Br)=O)CC1 c1(CC)c[nH]cc1C(=O)NCCC1CCN(C(C2CC23CC3)=O)C1 N1(C(C(CC2CCC2)NC(C)=O)=O)CC2CCCC(C1)N2Cc1cnn(C)c1 c1(-c2cn(CC3N(C(C4C(=C)CC4)=O)CCC3)nn2)c(C)noc1C N1(C(c2c(C)noc2C(C)C)=O)CCC(O)(CNC(=O)CCC2CC2(Cl)Cl)CC1 C(CCC(=O)NCC1CCCC1NC(=O)CNC(N)=O)SC(C)(C)C N1(C(C(CC)N(CC)CC)=O)C2CCC1CC(CNC(c1cncnc1C)=O)C2 C(=O)(C1=NOC(C)C1C)NCCCCC1CCCN(C(CCC#C)=O)C1 c1(NC(CC)=O)ccc2c(c1)CN(C(C)C(=O)NCCOC(C)(C)C)C2 c1(C(N(CCNC(CSc2nc(C)[nH]n2)=O)C)=O)cccc(OC(C)(C)C)c1 Cc1c(C(=O)NCC(C(C)C)NC(C2C=CC=CC=C2)=O)cccc1S(N)(=O)=O CC1(C)COC(CC(=O)NC2CCCCN(C(C3CC(C4CC4)C3)=O)C2)CO1 C=CC(C)(C)C(=O)NC(C)CC1CN(C(C2(C(=O)N(C)CCC)CC2)=O)C1 N1(C(CCCCOCC)=O)CC2CC(C)N(C(C3CCOC3C)=O)C2C1 C(N1CCN(C(=O)COCC)CC1)CCC1N(C(COCCC=C)=O)CCCC1 c1(NC(c2nc(CCC)oc2)=O)cnc(C)c(C)c1C.C1CCC(O)C(=O)N1 C1(C(=O)NCCCCCN(C(=O)C(c2ccccc2)O)C)CC2(C1)CC1(CC1)C2 C1(CNC(c2c(OC)cccc2)=O)CC2COCC2N1c1ncc(C)cn1 c1(C(=O)NC2CC3CC(NC(C(CCC)OC)=O)CC32)cc2cccc(C)c2[nH]1 CCC(CCC(=O)NCC(C(=O)NCc1c(O)cccc1F)N(C)C)OC N1(C(C(C)CCN(C)C)=O)CCCC(C)(NC(=O)CCOc2cccnc2)C1 C1(NC(C(c2cccs2)NC(CCCOCCOC)=O)=O)CCc2nncn2C1 c1(CC(=O)NCC2CN(C(C34CC(C)(C3)C4)=O)CC2O)c(F)cccc1F C1(C(=O)N)CC2CCC1C21CC1.c1(NC(C)=O)ncc(C(=O)NC2(CC)CCCC2)o1 c1(C(=O)NCCOCCCNC(=O)CCF)cc2cccc(Cl)c2s1 C1(NC(C(COC)N(C)C)=O)CN(C(c2ccc(C3CC3)o2)=O)CC12CCC2 Cc1cc(C(=O)NCC2=CCN(C(=O)CC3CCC4CC4C3)CC2)c(F)cc1N C(=O)(CCS(N)(=O)=O)N1CC(C(C)C)C(CNC(C2(C(=O)N(C)C)CC2)=O)C1 CC1CCN(C(C2CC3(CCC3O)C2)=O)CC1CC(=O)NCC(C)(F)C(C)(C)F N1(c2ccc(OC)cc2)CC(N=c2cc(C)nc(N3CCCC3)[nH]2)C(F)(F)C1 c1(C(=O)NCCC2(NC(c3c(C)ccc(C)c3)=O)CC2)cccc([N+](=O)[O-])c1 c1(C(=O)NC2CCN(Cc3cc(-c4ccco4)on3)C2)ccn2c1CSCC2 Cc1c(CCCOC(c2ccc(Nc3ccccc3)nn2)=O)cccc1[N+](=O)[O-] c1(-c2c(CCC)cccn2)ccc(-c2nccn2C(C)(C)CO)cc1OC N1(C(=O)C(O)C2CC2)CC2CCN(C(C3(CF)CCC3)=O)CC(C2)C1 c1(CC)nnsc1C(=O)NC(C)C(C)NC(=O)CN(C)S(N)(=O)=O C1(C2(O)CCC2)(C(=O)NCC23C(CN(C(C(C)NC(CC)=O)=O)C2)C3)CC1 N1(C(CC(CC)N(C(=O)CC(C)n2cccc2)C)=O)CCc2nc(C)[nH]c2C1 n1(C(C2CCOCC2)CC)nc(-c2cncs2)nc1C1COC1 Cc1cccc2[nH]cc(CC(N3CC(NC(c4ccc5nccn5n4)=O)C3)=O)c12 c1(NC(c2n(CCC)nnn2)c2csc(C3CC3)n2)cc(OC)c(Br)c(OC)c1 C(C(=O)N1CC(n2cccn2)C1)(C(C)O)NC(C(C)CC1CC1)=O C(C(CC(=O)NOCC(=O)OC)OC)N(C(C(C(CC)C)=O)=O)C1CC1 c1(C(N2CCC(C)(NC(C3CCCC3)=O)C2)=O)ccc(C2=NOC(=O)C2)cc1 Cc1ccc2[nH]cc(CC(=O)NCC(C)(C)NC(=O)Cn3cncn3)c2c1 C1(C(=O)OC(c2ccc(C#N)cc2)CC)CCC2(CCC2)CN1CC C1(CC(C)(C)C)CN(C(=O)CCNS(C)(=O)=O)CCN1C(C1CC1c1ccco1)=O O=C(N=c1[nH]onc1C1CC1)C1CC2CC2N1C(c1cncs1)=O N1(C(c2n[nH]c(C)c2F)=O)CCCC2(CCN(C(c3cnc(S)n3C)=O)C2)C1 c1(C(N2CCC(C#C)C2)C(=O)NCCC2CC2)nccc(Cl)c1Cl C1(NC(C2CC(C)C2)=O)CN(C(=O)CN2CSCC2=O)CC(C)(C)C1 N1(C(CN(C(c2c(OCC)cccc2)=O)C(C)C)=O)CCNC(=O)CC1C CON1CC(C(=O)N(C)CCNC(=O)C=Cc2cccc(C(F)(F)F)c2)CC1=O C1(C(=O)NCC2(COC)CC2)CC(NC(=O)Cc2nc[nH]n2)C12CCC2 c1(NC(C2N(C(c3n(CC(C)C)ncc3)=O)CC=C2)=O)ccccc1C C(C(C)(C(C)C)NC(C1CN2CCC1C2)=O)NC(c1c(OCC)scn1)=O Nc1cc(F)c(C(N2CC(CNC(=O)C(F)CC3CCCC3)C2)=O)cc1Cl c1(NC(N2CCCC(N3CCCC3)C2)=O)cccc(OCc2ccncn2)c1 N1(C(=O)CC2(OC)CCC2)CC(N=[N+]=[N-])C(S(C)(=O)=O)C1 N1(C(CC)=O)CC2CC(NC(c3ccc(OCCF)cc3F)=O)CC(C2)C1 N1(C(C2CNC(=O)O2)=O)CC2CCC1CC2NC(c1ccnc(C2CC2)c1)=O N1(CC)CCC(NC(=O)CCCNC(=O)C(CC)OC2CN(C(C)=O)C2)C1 C1(CC(=O)NC(CN(C)C(c2ccc(C3CC3)cc2)=O)(C)C)CCC=CCC1 C1(CNC(N2C(C3CCC(=O)NC3=O)CCCC2)=O)CC2(CCCC(N)C2)C1 Cc1nc2ccc(C(N3CCC(C4CC4)C3)C(=O)NC3CCOCC3)cc2[nH]1 C1(CC#C)(C(=O)N(C2CCC(C(C)C)CC2)C)CCN(C(=O)CCCOCC)C1 C1(C(N2CCCC(F)C2)=O)CC(F)CN1c1nccc(C(F)(F)F)n1 N1(C(CC(C)(C)C)=O)CC2CCN(C(=O)C(c3cccnc3)N)CC2C1 N#Cc1ccc(-c2ccc(NC(c3cc(Cl)ccc3O)=O)cc2)c(Cl)c1 c1(C(N2CC(N3C(=O)CC(NC(CN(C(C)=O)C)=O)C3)C2)=O)ncccc1O CCC(C)(C)C(C)CC(=O)NCC1(CNC(C2CCc3c(nnn3C)C2)=O)CC1 N1(C(CCCOCC)=O)CCc2ccccc2C(NC(=O)Cn2ccc(=N)[nH]2)C1 N#CC1(C(N2CC(CC(N3CCC(N4CCC4)C3)=O)C3(CC3)C2)=O)CCCCC1 CC1C(NC(C2(n3cnnn3)CCCCC2)=O)CCN1C(=O)CCCC1CCC1 c1(C(=O)NC2CN(C(c3cn(CC=C)nc3)=O)C(CO)C2)cc(C)c(Cl)cc1C C(=O)(C(C)(F)C(C)(C)F)NCC1CCN(C(C(C)(C)NC(C)=O)=O)C1 c1(C(N(C(C)CNC(C2CC(O)(C#N)C2)=O)C)=O)ccc(Cl)c(Cl)c1N N1(C(=O)C(O)Cc2cnc[nH]2)CC2CCCCC2(NC(C2CC(OC(F)F)C2)=O)C1 c1(C(=O)NC2C(C)(C)CN(Cc3ccc(Br)s3)C2)ccc2c(c1)CCCC2 c1(C(=O)NC2C3CN(C(C=CSC)=O)C2C3)ccc(C)c(O)n1 Cc1cccc(Cl)c1OCCNC(=O)NCC(CO)n1cccn1 c1(C(C)C)cc(CC(N)C(=O)NCc2ccc(C(N)=O)o2)n(C)n1 CC1=NN(C)C(=O)C1CC(=O)NCCCN(C(=O)C(C)SCc1ccccn1)C N1(C(CCc2onc(CC)n2)=O)CC(NC(=O)C(C)n2cnnn2)C(F)C1 c1(SC)ccc(F)cc1.c12cc(co1)C(=O)NC1CC(C1)NC(=O)C(OC(C)=O)C2 C1(NC(c2cnc(C3CC3)[nH]2)=O)CCN(C(c2ccoc2Br)=O)C1 C1(C(=O)NOCC2CCC2)CCC2CCC1N2C(=O)CCc1ccncn1 C1(C(=O)NC2(CNC(c3cncc(OC)n3)=O)CCOCC2)CCC(N=[N+]=[N-])C1 c1(C2C(C)C2)ccc(C(=O)N(C2CCN(C(=O)CCCN(C)C)C2)C)o1 c1(C(N2CCC(C(N(CCC#C)C)=O)C2C(C)C)=O)ccn2ccccc12 C(=O)(C(C)(C)CN(C)C(c1sccc1F)=O)NC(c1ccsc1)C C=C(C)CC(C(=O)N1CCC(O)(C(=O)Nc2nc(C(=O)NC)cs2)C1)NC(C)=O N1(C(CCc2ccc(C(N)=O)[nH]2)=O)CC(N=[N+]=[N-])C1.C12CCC(C1)C(=O)N2 Cc1nnc2n1CC(C(=O)NC1CC3CCC1C(NC(=O)CCCN=[N+]=[N-])C3)C2 S(=O)(=O)(c1cccnc1N1CN2CCC1CC2)NCCS(C)=O c1(OC)ccnc(C(=O)NCCN(C(=O)C(O)CC(F)F)C2CC2)c1OC c1(C(=O)NC2CN(C(Cc3c(C)ocn3)=O)C(CO)C2)cc2nc[nH]c2cn1 CC1=CCC(C)(C(N2CCN(C(=O)COc3c(F)cccc3F)CC2)=O)CC1 C=C(C)C(CC(=O)NCC)OCC.C1(SCC)(CC)CN(CC(C2CCCO2)=O)C1 CC(C)CC(C(=O)NCC#CC(N1CC(O)C(C2CC2)C1)=O)C(N)=O c1(C(=O)NC2(COC)CCN(C(=O)C(C)CSC)C2)c(N)c(C)cc2c[nH]nc12 C1(NC(CCc2c(C)ncs2)=O)CCCN(Cc2noc(C3CCCC3)n2)C1C Cc1nc2c(o1)CCCC2CC(=O)NC(CC(F)(F)F)c1ccccc1 C1(NC(COC(C)C)=O)CCC2CN(C(=O)CC3(C(F)(F)F)CC3)CCC2C1 c1(CCC)csc(C(C(=O)NCC2CC2)N(CCCC(C)O)C)n1 c1(C(=O)NCC2=CCCN(C(C(C)(C)OC)=O)C2)ccc2nc[nH]c2c1F C1(C(N(CCOC)CC)=O)COCCN1C(=O)C(C1CCOCC1)F N1(C(CC(=O)NCC)=O)CCC2OCCN(C(c3cc(COC)nn3C)=O)C2C1 CC1CC(CNC(c2ccncn2)=O)CN1C(=O)CCC(=O)N1CCOCC1 c1(CC(=O)NCC2COCCN2C(c2ccnnc2Cl)=O)ccccc1[N+](=O)[O-] C(=O)(CCCCCCN(C)C)N1CC2C(CN(C(=O)C3=CCS(=O)(=O)C3)C)C2C1 C#Cc1cccc(C(=O)N(C)Cc2ccc(CNC(=O)CCSC)cc2)c1F N1(C(C(c2cccc(Cl)c2)CC)=O)CCC(CNC(c2cc[nH]c2)=O)(OC)CC1 C1(C(=O)NCC=C)CN(C)CCN1C(c1ccc(O)nc1)=O N1(C(c2cc(C)[nH]n2)=O)CCC(C)(C)C(NC(C2CC3C(C2)C3(F)F)=O)C1 C(C(=O)NCCNC(=O)C1CC1)(C1CCCC1)NC(c1cnco1)=O CC1CN(C(C2CCN(C(=O)CC3CCCN(C)C3)CC2)=O)CCO1 N1(C(CNC(C(C)(C)C)=O)=O)CC2(C(N3CCOCC3CC(N)=O)=O)CC1CO2 n1(CC(N2CC3(C(NC(C(C)CF)=O)CC3)C2)=O)ccc2cc([N+](=O)[O-])ccc12 C1(=O)C(C(C)(C)C)c2cn(nn2)CCCN1.c1(C2(COC)CC2)nc(SC)no1 N(C(=NCc1ccc(-c2n[nH]c(C)n2)cc1)NC1CCCC(F)C1)C(CC)CC C(=O)(C1=C(F)CN(CCC2NC(=O)NC2=O)CC1)NC(=O)OCC.CNC C1(C(N2CCC(CN(C)C(C3CC(C(F)(F)F)C3)=O)C2)=O)CC2C=CC1O2 N1(C(C(COC)C)=O)CCCN(C(C2(C)C=CCC2)=O)CC1 C(c1ccncn1)=CC(=O)NC1CC(NC(CC2C(OC)CCC2)=O)C1 C1(C(=O)Nc2c(-c3ccc(OCCC)c(F)c3)scc2)CCCCN(C(C)=O)C1 CC(C(C)(C)C(=O)NCCC1(O)CCOC1)NC(=O)CC1CSCCO1 N1(C(CCc2onc(C)n2)=O)CC(N(C(=O)CCC(=O)N(C)C)C)C(C)(C)C1 c1(OC)cccnc1NC(=O)CC=CCNC(=O)C(C)(CO)OC C1(C(=O)NCC2N(C(c3cc(C(N)=O)no3)=O)CCC2)CCCS(=O)(=O)C1 C(c1ccc(O)cc1)=CC(=O)NC1COCC1NC(c1cc(C(F)F)ncn1)=O N1(C(CC=C)=O)CCC(C2(O)CCN(C(c3cc(Cl)no3)=O)CC2)CC1 N1(C(C2CCN(C(=O)NCC)CC2)=O)CC2(CCCC2NC(C2CCCO2)=O)C1 N1(C(COCCOC)=O)CC2(CCN(C(C34CCC(OCC)(CC3)C4)=O)CC2)C1 CC(CC(=O)c1ccc(Cl)cc1)C(=O)NCCC1(O)CN(C(C2CCCO2)=O)C1 CCS(=O)(=O)CC(=O)NC1CCC(C)(CNC(c2cc(C(=O)OC)nn2C)=O)C1 C1(CNC(Cc2ccc(C)o2)=O)(CNC(C2CCCC2N(C)C)=O)CCCCC1 C(C1=NOCC1)(c1nnnn1Cc1ccco1)NCCCN(C)C c1(C(N2CCC(CNC(C(CC)C#N)=O)C2(C)C)=O)cc(F)c(C)cc1F c1(N2CCC(C(C)(C)C)(CNC(CSC)=O)C2)ccc([N+](=O)[O-])cc1C(F)F C(=O)(C1=NNC(C(F)(F)F)C1)NC1CCC(NC(C(CCC)OCC)=O)CC1 C1(C(N2CCC(CC=C)(NC(c3ncccn3)=O)C2)=O)CCCC(C)(C)O1 c1(NC(C2C3CN(C(C(C)C)=O)CC32)=O)nc2c(s1)CC(N(C)C)CC2 C12(C(N3CC(=O)NC3=O)=O)CCC(CC1n1cc(-c3c[nH]nc3C(F)F)nn1)C2 CC(C)(C#N)CCCC(=O)N1CCOC(C(=O)NCCCSCCO)C1 C1(C(=O)NCCCC#C)CC(F)(F)CN1C(c1ccc(Br)c(F)c1)=O C1(CNC(C2(NC(c3cc(CCC)on3)=O)CCSCC2)=O)(CO)CC12CCC2 N1(C(c2cc(C)oc2C)=O)CC2CN(C(=O)CC3CCS(=O)(=O)C3)CC12 C(C(CC(C)C)NC(c1cc(C(N)=O)co1)=O)NC(CCCOCCOC)=O c1(C(=O)NCC(CC)(C)NC(C2(CO)CCOCC2)=O)ccc(OC)nc1 c1(OC)ccc(OC)c(CCC(=O)NC(CNC(=O)C(=O)N(C)C)C(C)(C)C)c1 C1(NC(CC(CCC)O)=O)CCCC12CN(C(c1sc(CC)nc1C)=O)C2 C(=O)(C1CCCc2cncn21)OC(COC)C(=O)Nc1ccccc1 O=C1CC(C(=O)N2CCCC(CCCCNC(=O)CN3CCCOC3=O)C2)=NN1 C12(C(=O)NC(CC3CN(C(COCCCC)=O)C3)C)CCCC1C2Br c1(C(N(CC(CC)NC(C2CSCCS2)=O)C)=O)ccc(C)nc1 C1(C(=O)NCCC(C)NC(=O)C(C)(C)c2ncco2)(N(C)C)CCCSC1 Cn1ncc(CNC(=O)CC2(C)CCN(C(C3COCCO3)=O)C2)c1O N1(C(CCCSC)=O)CCC2(CCC(NC(=O)CNC(=O)CC(C)C)C2)C1 C(=O)(C(C(C)C)N(C)C)N1CCC(CCC(=O)NC2C(SC)CCC2)C1 C1(C2CN(C(C3(N(C)C)CC3)=O)C2)(NC(C(C)c2ccco2)=O)CC1 C(C(C)(O)C(=O)N(CCC(C)NC(C1(Cc2ccccc2F)CCC1)=O)C)OC N1(C(C=C(CCC)CCC)=O)CC(NC(=O)CCCNC(C)=O)CC(F)(F)C1 C1(C(=O)NC2(CC)CCCN(C(=O)C(F)=C3CCCC3)C2)CC2CCC(C1)C2O c1(C(=O)NCc2cccc(NC(CCCOCC)=O)c2)ncc(F)cc1F c1(NCC)nccc(=NC(=O)CC2COCCN2S(=O)(=O)c2ccc(Cl)cc2C)[nH]1 C1(CCNC(c2cc(CC)[nH]n2)=O)CN(C(c2ccncc2N)=O)CC(C)O1 c1(C(=O)NC(C)CNC(=O)CN2CCOCC2=O)cc(S(N)(=O)=O)ccn1 c1(CC(C(=O)NC(CC)(C)CNC(=O)C(C)(C)OC)C)ccc([N+](=O)[O-])cc1 c1(C(N2CCC(C)C2CNC(=O)C=CBr)=O)c(Br)cccc1Br CC1Cc2cc(CN3CCCC(NS(=O)(=O)C4CC4)C3)ccc2O1 c1(C(=O)NC(C(=O)NCC2(O)CC(C)(C)C2)C2CCC2)ccc2[nH]ccc2c1.NC N1(C(c2c(NC)nccc2)=O)CCC2(CC1)CC2C(=O)N(CCCN(C)C)C C1(CC(=O)NCC(CN(C(c2cc(C(C)=O)on2)=O)CC)(C)C)CCC(=O)NC1 CC(C)C(F)(F)CC(=O)NCC1COCCN1C(=O)CCCNS(C)(=O)=O N1(C(CN(C(=O)CCc2cccnc2)CCOC)=O)CC2CCC1C(O)C2 CCC(C)(C)CCCC(=O)NCC1(F)CCCN(C(=O)CSC)CC1 Cc1cccc(C(F)(F)F)c1C(=O)NC(CNC(=O)Cc1cc[nH]n1)CO C1(NC(=O)Cc2csc(Br)c2)CN(C(=O)C2=CCCC2)CC1n1ccnn1 c1(CCNC(C2(CN)CC2(F)F)=O)c(Cl)cc(Cl)cc1Cl C(=O)(CCC(=O)N1CCC(NC(C2(C)CC(C#N)C2)=O)C1)NCCC c1(CC(=O)NC2C(NC(C=NOC)=O)CC2)nc(C)c(C)s1 Cc1c(C(N2CCC(C)C2CNC(=O)COCCc2cccs2)=O)cccc1O c1(C2C(=O)N2)cccnc1.C1(CNC(=O)COCCF)CCSC1 C=C(C)CCCC(=O)N1CCCC(O)(CNC(c2c(C)noc2Cl)=O)C1 c1(COCC(N2CCC(CN(C(C3(SC)CC3)=O)C)C2)=O)ccc(C)cc1 C(C1Cc2ccccc21)NC(C1(C)CCCN(C(c2c(C)occ2)=O)C1)=O c1(C(=O)OC)ccnc(N2CCC(n3cccn3)(CC(=O)OC)C2)c1Br n1(CCCC)cc(C(N2CC(C(C)NC(c3ncccn3)=O)C2)=O)nn1 Cc1cc(C(=O)NC2CCN(C(C3(C#N)CCCC3)=O)CC2F)c2[nH]cnc2c1 c1(CC)c(C(N2CCC(C(C)NC(C3CN(C)C3)=O)C2)=O)[nH]c2ccccc12 c1(OC(C)C)ccc(C(=O)N(CCC(C)NC(c2n[nH]cc2Cl)=O)C)cc1N c1(C(=O)NCCN(C(C2C(C#C)C2)=O)C)cc(F)cc2cnccc12 C1(C(=O)NCC(C2CC2)NC(c2ccn(C(F)F)n2)=O)(COC)C=CCC1 C1(NC(C(c2c(C)cccc2)C)=O)CN(C(c2oc(Br)nc2C)=O)CC12CC2 O=C(N=S1(=O)CCCC(O)C1)c1cc(O)c(F)c(F)c1 C1(C(=O)NCC2C(CNC(C3CC=CC3)=O)C2)CCC(NC(N)=O)CC1 C(CCNC(C1CSCN1C(=O)CC1CC=CCC1)=O)(C(C)C)OC Cn1[nH]c(C(=O)NC(C)(CNC(=O)C(F)C2CCCC2)Cn2cccn2)nc1=O S(=O)(=O)(c1ccc(NCCc2ccccn2)c(F)c1)N1CCCC(COC)CC1 C12(C(=O)NCCc3cncc(C(F)(F)F)c3)CCCCC1CNC2 C(=O)(CC1OCCc2ccsc21)NC(CN(C(C1(C2CC2)CC1)=O)CC)C CC(CC(=O)N1CC2CC2C1C(=O)N(C)Cc1cnnn1C)C(C)(C)C c1(CC2CCN(C(=O)NC3CSC3)CC2O)cc(Cl)cc(Br)c1O c1(C(=O)NC23CC(CNC(C4C(N(C)C)CC4)=O)(C2)C3)cccn(C)c1=O C(CC(=O)NC1CC12CC2)N(C(c1nc[nH]n1)=O)CC c1(C(N2CC(NC(c3cc(CC)n(C)n3)=O)C(C)C2)=O)nccn2cnnc12 CC1CC(NC(=O)CCNC(C2CCOCC2)=O)CN1C(C1CCCCCC1)=O N1(C(C2=C(C)CC2)=O)CCC2CN(C(C3CC4(CC4)CO3)=O)C2C1 c1(C(=O)NC(C)CCNC(=O)CNC(C2CCCC2)=O)cncn1C N1(C(C(N2C(C(=O)OCC)C(O)C(O)C2)=O)=O)CCc2sc(C)cc2C1 N1(C(c2c(OC)nccc2)=O)CCC(NC(=O)CC2(C)CC2(F)F)C(F)(F)CC1 C1(CNC(c2ccoc2Cl)=O)CCC2(CN(C(=O)Cc3cocn3)C2)O1 Cc1csc(C(N2CC3CC3(CNC(=O)Cc3cnn(C)c3C)C2)=O)c1C N1(C(c2scc(COC)c2)=O)CCN(C(=O)CSS(C)(=O)=O)CC1C1CC1 C(=O)(CCC(=O)NC1C2CN(C(n3cc(Cl)cn3)=O)CC12)N(C(C)C)C c1(C(C(=O)NCC(CNC(CCC(C)C)=O)(C)O)O)ccc(Cl)cc1F c1(CN2CC(C)C(Nc3ncnc(=N)[nH]3)C2)cn(C)c2cc(F)ccc12 c1(C(=O)NC(C)CN(C(=O)C(C)(Cl)Cl)C)cn(C)nc1C(C)(C)C c1(C(N(c2ncc(OCC)cn2)C2CNCCOC2)=O)cc(O)nc(O)n1 CCCCC(CNC(C1CC(O)CN1C)=O)NC(=O)CC1CC(SC)C1 N(C1CCOc2ccccc21)C(C1N(C(CCCC(=C)C)=O)CC(O)C1)=O c1(COC)ccoc1C(=O)NC1CC(F)(CNC(=O)CCCC2(CSC)CC2)C1 C1(C)(C(C)C)CN(C(=O)CC2CC(CF)C2)CCO1 CC1CC(C)N(C(=O)Cc2coc3ccccc23)CCN1C(=O)Cc1ccon1 CCCCC(CC(=O)N1CCOC(C)(CC)C1)NC(c1cc([N+](=O)[O-])ccn1)=O C1(COC)(NC(=O)CC2CCN2C(C2(C)CC(=O)C2)=O)CC(C)(C)C1 c1(NC)cccc(F)c1C(N1CC(CCNC(=O)CSCc2csc(C)n2)C1)=O C(=O)(CC(O)C(=O)Nc1nc[nH]c1C(F)(F)F)NCC(C)(C)NC(=O)C1CC1 C(=O)(C1CC(=O)Nc2c(F)cccc21)N1CCCC(NC(=O)COCC2CC2)C1 C(C1=NOC2CN(C(=O)Cn3cc(C4CC4)nn3)CC12)NC(c1c(C)ccs1)=O c1(C(N(C(C)C(=O)NC(C(O)CO)C2CC2)CCC)=O)ccc(F)c(O)c1 c1(-c2c(C(=O)Nc3nccc4ncnn34)c(F)cnc2)cnc2ccccc2c1 N1(C(C2(C)CC2(Cl)Cl)=O)CCN(C(C2(n3cccn3)CC2)=O)C(CCO)C1 c1(OCCC)cccnc1CNC(=O)COC(c1ccc(SC)cc1)=O.C1CCC1 C(C(CC(F)(F)F)NC(=O)CCCC1CCCCO1)NC(c1c(CC)nns1)=O N1(C(C2(NC(=O)Cc3ccc(O)cc3)C(C)(C)C2)=O)CCC2(C1)COC(=O)N2 c1(NC)ccc(C(N2CCCCC2CN(C(=O)CN=[N+]=[N-])C)=O)cc1 C1(C(N(CCCNC(=O)CC2(C)CCOC2)C)=O)CC2(CCC2O)C1 C1(NC(=O)NCC2CC3CC23)CCN(c2ccc(Br)nn2)CC1 c1(C(N2C(CC)CN(C(c3cnc[nH]3)=O)CC2)=O)ncnc2cc[nH]c12 N1(C(C(C)OC)=O)CCC2(CC1)CC2CNC(=O)COCc1ccnn1C c1(C(=O)NCC2C(NC(C3N(C)CC(C)(C)C3)=O)C2)ccc2oncc2c1 Cc1cccc(C(=O)NCC2CCCCN2CCS(=O)(=O)NC2CCCC2)n1 N1(C(c2nc(CC)oc2C)=O)CC(C(=O)N(CC(O)CO)C(C)C)CCC1(C)C N1(C=O)CCC(F)(F)CC1.C1(C(=O)O)CC(CO)N1C(c1cscc1CO)=O C1(NC(=O)CCSC(F)F)CCCCC1c1cn(C2CCCCC2)nn1 c1(C(=O)NC2CC(NC(c3ccn(C(C)(C)C)n3)=O)C2)cccc2c1CCO2 N1(C(C(C)N2C3(COC3)C2=O)=O)CCCC2(CC2)C1.CCO.NC C(CCCCCC(=O)N1CCC(c2ncccc2Cl)C1)NC(=O)OC(C)(C)C CCC(C)C(C(=O)NCC1(F)CCC1)NC(=O)CCC(=O)N(C)C Cc1cnc(C(=O)N(C2CCCN(C(=O)CC3CCN(C)C3)CC2)C)cc1C C1(=CCNC(C(C)Cc2cnn(C)c2)=O)CCN(C(c2cc(Br)n[nH]2)=O)CC1 C(=O)(CCCC(C)=O)NC(C(=O)NC(C#C)CC1CCCC1)CC1CC1 N1(C(c2c(C)n(C)nn2)=O)CCCC(C)(C(N2CC(c3cnccn3)C2)=O)C1 n1(CCSCC)cc(C2(C)CN(C(=O)C(C)OCCc3ccccc3)C2)nn1 Cc1cc(C(N2CCN(C(C3(F)CCC3)=O)CC2C(C)C)=O)nc(O)c1 c1(C(N2CC(O)(C(C)NC(C3C(C)CC(C)O3)=O)C2)=O)cc([N+](=O)[O-])cnc1O c12c(F)cc(cc1F)CC(=O)O2.c1(NC2CC(C(=O)OCC)C2)cnn(CC)c1 c1(OCC)ccc(N)c(NC(c2cc(C3CC3)no2)c2nnnn2C(C)C)c1 C(C)(CCC(C)C)N(C(COC1CCN(C(C(C2CC2)NC(C)=O)=O)C1)=O)C Cc1cc2[nH]c(C(N3CCC(O)(C(C)NC(c4occ(C)c4C)=O)C3)=O)cc2s1 C1(C(=O)NC(C)CCNC(c2ccoc2)=O)Cc2nncn2C1 CC1CCOCC1Nc1nnc(C(N)=O)s1 C(=O)(CCC(=O)NC1CC(C)(NC(c2ccnc(C)c2)=O)C1)OCC CC(C)(C)C(O)Cc1cn(CCC(=O)NC2CCN(c3ccnc(Cl)n3)C2)nn1 C1(NC(CCOCCC)=O)CCCN(C(=O)C(CC2CCCCC2)CC)C1 C(=O)(CC(C)CC(C)(C)C)NC(CC(=C)Cl)C(=O)N1CCC2C(OC)CC12 C12(CC(=O)NC(c3cccc(F)n3)C)CCC1CN(C(c1nonc1N)=O)C2 C1(C)(CNC(C(C)C2CC2)=O)CC(F)(F)CN1C(=O)Cc1ccc(C#N)cc1 C(=O)(C(C)(c1ccccc1)SC)NCCCN(C(=O)C(C)NS(C)(=O)=O)CC CCC(C(=O)NCC1CCN1CC)NC(=O)CC1(CC)CCC1 c1(CCOC)n[nH]c(=NCC(C)(C(C)C)NC(c2cc(C)cc(F)c2)=O)s1 CC(CC(=O)NCC(C)(C)CC(=O)NC1CCCC(C2CC2)C1)C(F)(F)F c1(NC(c2cnn(C)c2)C(=O)OC)nc(C)c(C)cc1C(=O)N(C)C C1(CC(C)NC(c2cc(O)cs2)=O)CN(C(c2csc(C(F)F)c2)=O)CCO1 C12(CNC(CC3CCN(C)C3)=O)CCC(CN(C(=O)C(C)(F)F)C1)C2 CC(CC(C)(F)F)C(=O)N(C1CN(C(c2cc(CO)on2)=O)CC12CC2)C c1(CN2CC(F)CC(C(=O)NCCOCC#C)C2)cc([N+](=O)[O-])ccc1F CC1CCC(C(N2CC(NC(c3cccc(Cl)c3)=O)C(O)C2)=O)CC1 CC1CCCC1(C(=O)NCCN1CC(C)(O)C1)NC(=O)CN(C)C(N)=O N1(C(C2OCCN(CC)C2)=O)CC2CCCCC2(NC(=O)Cc2ccsc2C)C1 Cc1cc(Br)c(Cl)cc1COC(C1(C#N)CC2(CC2)C1)=O CC(C)C1=NOC(C(=O)NC23CC(NC(=O)Cc4ccc(CO)cc4)(C2)C3)C1 c1(C(=O)NC2(C3CCN(C(=O)CSC(F)F)C3)CC2)cc2ccccc2oc1=O C1(NC(N2C(CC)CC(O)C2)=O)(CC)CC(C)(C)C1 C1(N(C(c2ccn(C)c2)C(=O)NC(C)C)C)CCCCC1 c1(CNC(CN(C)C)=O)nn(C)c2c1CN(C(=O)C(C1CCCO1)C1CC1)CC2 c1(CC)nc(C)ccc1NC(=O)CCCCN(C(=O)C(C1CCOCC1)C)C Cc1ccc2sc(C(N3CCC(C)C(NC(c4c[nH]nc4C)=O)C3)=O)c(C)c2c1 c1(C(N2CC(NC(c3c(CC)c(F)ccc3)=O)C(O)C2)=O)ccc([N+](=O)[O-])cn1 C(N=c1cc(C)nc(N2CCOC(C)(C)CC2)[nH]1)C1C(C=C)OCC1 N1(C(C#CC(C)C)=O)CC(=O)NCC1C(=O)NCC1(O)CCOC1 N1(C(C(c2cccc(C)c2)O)=O)CC2CCC(NC(=O)C(C)O)CC2C1 C(=O)(CCCCCCCCCC1CC1)NCC(CNC(CC(CC)CC)=O)CO Cc1cnc(-c2nc(-c3cncs3)nn2C2CCCSC2)cc1C c1(N)ccccc1Cl.C1(N(CCCO)C(C2(C#N)CC2)=O)CC2CNC1C2 C#CC1CCCN(C(=O)C=CCC2(NC(c3ncn(C)c3C)=O)CCC2)C1 N1(C(c2n(C)ccn2)=O)CC(C2CN(C(=O)CC3COCCOC3)C2)C1 c1(CC(N2C(CNC(c3ccc(CN(C)C)o3)=O)C=CC2)=O)ccnc(O)c1 C(=O)(CCCC(CC)CC)NC1C(NC(COCC)=O)CCCC1 C12(CCNC1=O)C(=O)N1CC(C)(C)C1C2.C1(CC(C)C)CCN(C(=O)CC2CC2)C1 c1(SC)ccc(C(=O)NC(C)(C)CN2CCN(C(=O)CC3CC(=O)C3)CC2)cc1 C1(C(=O)NC(CCC)C(=O)N2CCC3CC23C)CN2CCC1CC2 C1(CC(=O)N(CCCNC(c2ccn(CC#N)n2)=O)C)CC2CCC1C2 CCCC(CCCNC(=O)C(C)C1(O)CCC1)NC(=O)CN(C)CCOC CCC(CC(=O)N(CCCNC(=O)C(N1CCCC1)C1CC1)C1CC1)C(C)(C)C c1(NC2C(CNC(C(C)c3ccco3)=O)CCCC2)ncc(Br)c(O)n1 C=CCCC(F)(F)C(=O)NCC12CCC1CN(C(=O)Cn1ccc(O)nc1=O)C2 CCC(C)(C#N)C(=O)N1CC(C(=O)NC2CC3CCC2O3)C(F)C1 N1(C(C(=O)NCCCSC)C(C)CC2CCCC2)CCC(C2CC2(F)F)C1 c1(Cc2nc(Cc3cc(F)cc(F)c3)on2)c(F)cc(Cl)cc1F N1(C(c2c(CC)oc(C)c2)=O)CCC2(CC2C(=O)NCC(CO)C(F)(F)F)C1 c1(CN2CC(NC(C3CC(F)C3)=O)C2)c(C(F)(F)F)cccc1F Cc1cc(Cl)c(C(=O)NCC2(CNC(=O)C(C)C#N)CC(F)(F)C2)cc1F C1(NC(c2c(C)scn2)=O)CN(C(C2CCOCC2(C)C)=O)CC(F)(F)C1 C(=O)(CC(C=C)CCC)N1CCN(C(C(C)OCCC=C)=O)CC1CC(F)F C(=O)(C1=Cc2cc(C)ccc2OC1)N(CCNC(c1c(OC)noc1C)=O)C C(=O)(C(CC)(CO)OC)NCC(CC)NC(=O)CN1CSCCSC1 CC(=O)C(C)CC(C)C(=O)N1CCCC(C(C)(C)C(=O)NC(c2cc[nH]n2)C)C1 C(=O)(C1Cc2ccc(Cl)cc21)NCCCC(C)(C)O c1(NCC#CC)cc(S(=O)(=O)N(C)CCN2CC(C)OC(C)C2)ccc1C#N c1(OC)c(C(N2CCN(S(C)(=O)=O)CC2C)=O)ccnc1Cl C(CO)(CC(C)(C)C)NC(C(CCC)NC(=O)C(C(C)C)NC(N)=O)=O Cc1cc(NC(=O)NCC2CC2C2CCCO2)n(C2CC2)n1 N1(C(CC(C)(C)C)C(=O)Nc2ccccc2Cl)CCc2ccc(Br)cc2C1 N1(C(c2ccc(C#C)c(F)c2)=O)CC2CC(C)N(C(=O)Cc3cncnc3)C2C1 C1(C(=O)NCCc2cc(C(N(CC(=O)OCC)CC)=O)no2)CCC(O)CN1C C(CCCCCN=c1[nH]c(NC(c2ccccc2)CF)nc(=N)[nH]1)N(C)CC C1(NC(=O)C=Cc2ccsc2)CCC2(CC1)CCN(C(=O)COc1ccsc1)C2 C1(NC(c2csnn2)=O)C2CN(C(=O)CC3CSC3)CC12 C12(NC(c3ccc(SC)o3)=O)CC3CCC(C1C2)N3C(c1cncn1C1CC1)=O N1(C(c2ccc(Br)cn2)C(=O)NCCOCC)CCC(F)(F)C(CO)C1 CCC(C(=O)NC(C1(O)CN(C(=O)CNc2ccccn2)C1)C)n1nccc1C c1(C(C)C)ccsc1C(=O)NCC1(CNC(=O)C(c2ccccc2)O)CC1(F)F C1(CNC(C=CC=CC)=O)CCCN(C(c2cccc(N3CCOCC3)c2)=O)C1 c1(C(=O)NCCCCNC(C=Cc2n(CC)ccn2)=O)cc([N+](=O)[O-])cc(C)n1 N1(C(C)=O)C(=O)CCC1C(=O)OCC1(Oc2cnc(Cl)[nH]2)COC1 c1(CN2CCC(C(=O)NCCn3c(CC)nnc3)CC2)ccc(Cl)nc1Cl c1(C(c2nnnn2C(C)C)NC(CC=C)C)cc(C)c(C)c(Br)c1 c1(C(N2C(C)CN(C(=O)CN3CCC(C)(O)C3)CC2)=O)cc(Cl)c(F)c(Cl)c1 C1(C(=O)NCc2cc(C(=O)NCC(C=C)O)n[nH]2)C2CC3C(C2=O)C13 Cc1cc(C(=O)NC(C(=O)Nc2cccs2)c2ccco2)ccc1C#N C(=O)(C(C)CC(C)(C)C)NCC=CC(=O)Nc1c(C)cccc1C C1(C(N2CC(NC(=O)C(F)(F)C3CCCCC3)C(O)C2)=O)CC2CCC1CC2 c1(C(N(C(C(=O)OC)C2CCOC2)CC)=O)n[nH]c(=N)s1 C1(N(C(C2N(CC)CCC2)=O)C)C2CN(C(=O)CCOC(C)=O)CC12.CC(C)C C(=O)(C(F)CCC(C)(C)C)NCCCC(C)NC(c1cc(C2CCC2)no1)=O C1(CNC(C=CC(CC)C)=O)CC2(CC(NC(c3ccc(F)c(F)c3)=O)C2)C1 N1(C(C=CC(C)(C)C)=O)CC2CCCC(CNC(=O)C#CC3CCCOC3)(C2)C1 CC1CC(NC(c2cncnc2C2CC2)=O)CN1C(=O)C=Cc1cccn1C N1(C(CC2CCN(CC(C)C)C2)=O)CCC(CNC(c2cnc[nH]c2=N)=O)CC1 c1(CC)cccc(C(N2CCCC(N(C(=O)Cc3ccco3)CC)C2)=O)n1 C1(C(N2CCC(NC(CCCN(C(=O)OC)C)=O)C2)=O)CC2(CC2)CN1C C1(C(F)F)(CNC(c2ccc(C)s2)=O)CCN(C(=O)CCc2ccnc(C)n2)C1 C1(NC(CC(=O)NCC#C)=O)CCCC(C(=O)NCc2ncc(C)s2)C1 c1(SC)nc(N2CCOC(CNCc3cccc(C)c3O)C2)cc(C)n1 C(=O)(C(C)(C)Cc1ccc(O)cc1)NCC(C)NC(=O)C(F)C1CCC1 C1(C(N2CCC(C)C(NC(=O)Cc3cc[nH]n3)C2)=O)CCC2CC1C2(C)C CC(CC(C)(C)C)C(=O)NCC1CCCC1C(=O)NCCN1C(=O)CCC1=O C1(CNC(c2n[nH]cc2Cl)=O)CN(C(c2ncccc2Cl)=O)C2CCCC2O1 C1(N)CCC(C(F)(F)F)CC1.c1(C(CC#C)=O)cccc(CNC(C)C(=O)NC)c1 c1(C(=O)NC(CNC(COCC)=O)CC)nn(C)cc1SC Cc1ccc(C)n1CC(=O)N(C)CCC1CCCCN1C(C1CCC(=O)N1C)=O c1(CC)cc(C(N2CCC(CNC(c3cnc(C4CCC4)s3)=O)C2)=O)ccc1F CC1(C)CN(C(=O)CCCCN2CCOCC2)CC1NC(=O)C1=CCCC1 C(=O)(CC(CC)CC(F)(F)F)NC1CCN(C(c2nnc(CC)s2)=O)CC1F C1(O)(C(CNC(C2(CC(C)C)CCC2)=O)C)CCN(C(c2cccnc2N)=O)C1 CC1CCN(C(c2cc(O)ccc2N)=O)CCN1C(=O)C1=CCCCO1 CN1CC2CCC1CN(C(C1CCN1C(c1ccc(N)c(F)n1)=O)=O)C2 C1(NC(N(C)C)=O)CCCC2CCN(C(N3CCC(C(N)=O)CC3)=O)CC12 CC(C)C(C)C(=O)NC1CCOC1C(=O)NC(c1cscn1)C C1(C(N2CCN(CC3CN(C(C4C(OC)C4)=O)C3)CC2)=O)CC(C)(C)OC1(C)C C1(SCC)CCC(C(=O)NCC2(C(=O)O)CC(O)C2)CC1 C(=O)(C(C(=O)NCC1CCCN(C(=O)Cc2ccsc2Cl)C1)C(C)C)OCC c1(CC(=O)N(CCNC(C2(F)C(C)C2)=O)C2CC2)csc2ccc(Cl)cc12 NC1CS(=O)(=O)C2CN(C(C3COCCN(C(c4occ5c4CCC5)=O)C3)=O)CC12 C1(NC(C2CC(SC)C2)=O)CCCCC1CNC(=O)CCCc1csc(=N)[nH]1 C=C(C)C(C)(O)C(=O)NC1CN(C(=O)CC(F)(F)Cl)CC1CC(C)(C)C N1(C(CC(C)C)=O)CCCCCC1CNC(C12CC(F)(C1)C2)=O c1(C(=O)OC)ccc(O)c(C(=O)NCC2(F)CCN(C(=O)C=C(C)Cl)CC2)c1 c1(C(N2C(CN(C(c3cc(C)sc3)=O)C)CCC2)=O)ccc(C(O)CF)cc1 c1(C(N2CCC(N(c3cc(COC)ncn3)C)C2)=O)cccc(C#CC2CC2)c1 CC1CN(C(c2cccc(CO)n2)=O)CCC1CNC(=O)CC(C)(C)O c1(C(=O)NCC2(C)C(C)CN(C(=O)CN3CCSCC3)C2)cccc2sccc12 N1(C(c2c(CC)occ2)=O)CCCC(C2CCN(C(C3CC3C)=O)CC2)CC1 c1(C(=O)NC2CCC(CNC(C3CCCO3)=O)CC2)cc(F)c(O)c(F)c1 c1(CC)cc(C(N2CC(NC(C3(C)COCCO3)=O)C2)=O)oc1CC c1(C(N2C3C(N(C(CCCSC)=O)C)CC(C3)C2)=O)cccc2cccc(O)c12 C(CCC(C(=O)NCCn1nncc1C)NC(=O)C(C)N1CCCC1)OC n1(CC)cc(C(=O)NC2CCN(C(=O)C=Cc3ccoc3)C2CC)c(C2CC2)n1 N1(CCCCCNC(C(C2CC2)OCC)=O)CCN(C(C2(CO)CCC2)=O)CC1 CCC(O)C(F)(F)C(=O)N(C(CNC(=O)CCc1cc(C)nc(C)c1)C1CC1)C c1(OC)cc(CN2CCCC2C(=O)Nc2ncc(C(C)=O)s2)cc(C(C)C)c1O C12(CS(C3(C)CC(O)C3)(=O)=O)C(NC(=O)C(F)F)C3CC1C2C3 N1(C(C2C(C)OCCO2)=O)CCC(C(=O)NCCN(CCCF)C)=C(F)C1 CC1CN(C(C2SCCS2)=O)CCN(C(C2CC3COCC3C2)=O)C1 N1(CC(=O)NC2C=CCN(C(c3cccc(F)c3)=O)C2)CSCCSC1 C(CC(F)F)(C(=O)NOCC(O)CO)N(C(=O)C(OC)OC)C1CC1.CO N1(C(c2c(NC(C)=O)cncc2)=O)CC(C)C(NC(c2cocc2C)=O)C(C)C1 N1(C(C(C=CC)O)=O)CCC(C)(CCNC(c2cn[nH]c2)=O)CC1 CCC(N=c1cc(C)[nH]c(=NCCC(C)(C)C)[nH]1)c1ccc(-c2ccccc2)cc1 c1(C(N2CC(SC)C(NC(=O)CC(C)F)C2)=O)ccc(S(N)(=O)=O)s1 c1(C(=O)NC2CCN(C(Cn3c(C)csc3=O)=O)C2C)c(C)nn(C)c1C C1(CNC(c2n[nH]c(C)c2C)=O)CCCCN(C(c2c[nH]c(C#N)c2)=O)C1 c1(-c2n(C(c3ccccc3)C)nc(-c3cncs3)n2)cnc2c(c1)OCC(=O)N2 Cc1cc(C(N2CCOC(C#N)C2)C(=O)N(C)C)cc(Br)c1C.C1(C)C(=O)N1 N1(C(C(C)OCC)=O)CCC(O)(CNC(=O)C(C)Sc2ccc(C)cc2)C1 N1(C(C2(C#N)CCC2)=O)CCC(CCNC(=O)C(N2CCOCC2)C2CC2)CC1 C1(NC(C(COC)C)=O)CC(C)N(C(=O)CC2(C)CC2(Cl)Cl)C1 CC1OCCN(C(=O)CC2COCCO2)C1C(N1CC(CO)C(O)C1)=O c1(C(C(N2CCC(N(CCC)C(c3coc(O)n3)=O)C2)=O)O)ccc(F)cc1C c1(CC(=O)NCCCCN(C(c2ccc(C)c(C)c2)=O)C)c[nH]c2cccnc12 c1(C(=O)NCCCC(CCC)NC(C2(C)CC2)=O)cc(S(N)(=O)=O)cnc1C O=C(C1=CCCSC1)NCc1cccc(C(=O)NCCc2ccc(O)nc2)n1 CC1(CNC(c2snnc2C2CC2)=O)CCCN(c2nccc(C#N)n2)C1 C1(c2n(CCOC)nnn2)(NC2CCC(=O)NC2C)CCN(C2CCOC2C)CC1 c1(OCC)ccc(Cl)nc1C(=O)NCC(C)CNC(=O)Cc1nnc(C2CC2)o1 CC1CCC(C(N2CC(C)(NC(c3ccc(F)c(CO)c3)=O)C2)=O)C(=O)N1 C1(C(=O)NC2CC(NC(Cn3c(C)ncc3)=O)CC2O)CC2(CCC2O)C1 C1(Cn2cc(C(C)O)nn2)CN(C(=O)CN2CSCC2=O)CCO1 C1(C(=O)NC2CC(NC(C(CCOC)C)=O)C2)CCC(=O)N(C2CC2)C1 N1(C(c2c(C#N)cccc2)=O)CCCC2CN(C(c3cn[nH]c3)=O)CCCC12 CC(C)(C(=O)N1CCN(C(c2cnc(N)c(Cl)c2)=O)CC(CO)C1)C(F)(F)F c1(OC)cc(OC)ccc1-c1cnc(OC)nc1.N12CCN(C(CO)C1)C(=O)C2 C1(CNC(c2nc(CCC)oc2)=O)CN(C(=O)Cc2ccnc(O)c2)CC1C c1(C(=O)NCC2CCCC(NC(c3cnsc3)=O)C2)n[nH]c2c1CCOC2 C(=O)(C1=CCCS1)N1CC(OC)(CNC(=O)C(O)Cc2ccccn2)C1 c1(CC)ncc(C(=O)NCC2CC3CCC2N3C(c2occc2C)=O)c(O)n1 C(CC(C)C)(C(=O)N(C)CCOCCCN=[N+]=[N-])N(C(C(CC#C)C1CC1)=O)C c1(NC)cccc(C(=O)NCCSCC(N2CCCC3CC23)=O)c1 N1(C(c2c(C)ccc(OC)c2)C(=O)NC)CCCC2C1CCN2C C1(NC(C(CC)(F)F)=O)CCN(C(=O)C(O)CCSC)CC1O N1(C(C2(CCCC)CCCC2)=O)CCCN(C(=O)C(C)(CC)OC)CC1 N1(C(c2cccc(CC)n2)=O)CC2CCN(C(c3cc(O)cc(O)n3)=O)C2C1 c1(C2(CNC(=O)NC(C)C(=O)N(C)C)CCC2)cccnc1 C(CC(C(=O)NCC1(F)CCOC1)NC(c1csc(O)n1)=O)=CC c1(C(N2CCC(C(C(=O)NCC(COC)OC)C)C2)=O)cc(C)c(C)cn1 N(C1CCc2c(F)cc(F)cc21)C(C1CC(O)CN1C(=O)C=CCF)=O C1(NC(Cn2ccc(C)n2)=O)CN(C(C2CCCN(C)C2)=O)CCC1(C)C c1(CC(=O)NCC2(CC(=O)O)CCC2)cc(Br)cnc1F N1(C(CC)=O)CCC(C(=O)N(c2cnc3ncnn3c2)CC)CC1(C)C CCC(CNC(C1CC(n2cnnc2)C1)=O)NC(=O)CO Cc1cnc2cc(C(N3CCCC(F)(CNC(C4(O)CCCC4)=O)C3)=O)ccn12 c1(C(=O)NCC2CC(CNC(C3(CCOC)CCC3)=O)C2)cnc(OC)nc1C C1(OC)CN2CCC1(C)CC2.C(CCC(C)C(=O)NCCCOCC(=O)N(C)C)OC C1(C(N2CC(CC(C)NC(C34CCC(CC3=O)C4)=O)C2)=O)CC2CCCC2C1 C1(CCNC(CC2(COC)CC2)=O)CN(C(C2CCC3CC23)=O)CCCO1 C1(C(=O)NCCC(C)OC)(CNC(=O)C=C(C)C2CC2)CCCO1 CC(C)(C(=O)NC1CCc2nncn2C1)C1=CCN(C(=O)CCN2CCCC2)C1 c1(C(=O)NC(CN(C(C)C(=O)NC2CCCCC2)C)C)n[nH]c2ccc(F)cc12 c1(C(=O)NCC2C(NC(Cc3cn(C)nc3)=O)CCC2)cnccc1C(F)F C(=O)(C1=NOC(C)C1)N(C(=O)CN1CCC(C)(Cc2ccc(CC)o2)C1)OCC CCCCC(C(=O)NC1CCCN(C(=O)CSCCC(F)(F)F)C1)C(C)C C1(OC)CC2(CCN(C(=O)Nc3ccc(OOC(F)F)c(C(F)(F)F)c3)C2)C1 c1(C(=O)NCCC2CC(NC(C(C)(C)CC#N)=O)C2)c[nH]c(=O)c2ccncc12 N1(C(Cc2cccc(C(C)C)c2)=O)CCC2(CC1)CC2NC(=O)C(O)C1CC1 N1(C(COC2CC(NC(C3(C)CCCC3O)=O)C2)=O)CCC(F)(F)C(O)C1 c1(C(N2CCC(N(C(C(CC)SC)=O)CC3CC3)CC2)=O)cn(C)c(=O)cn1 C1(OC)CN(C(=O)N(CC(=O)NC(C)C)C)CC1C1CCN(c2ccncc2)CC1 C=CCCCC(c1nnnn1CCCSC)NCC1C=CCOC1.C(C)(=O)O CON1CCC(C(N2CCC(N(C(=O)Cc3cc(F)ccc3Cl)C)C2)=O)CC1 N1(CC(=O)N(C2CCC(NC(=O)COCCCF)CC2)C)CC2C=CC1C2 N1(C(C=C(CCC)C)=O)CC2(CC(NC(=O)C(C)(C)C(C)O)CO2)C1 CCCC(C(=O)NCCC1CC1C)NC(C1CC=CC1)=O C(C(C)(O)C(=O)NC(CNC(=O)Cc1scnc1-c1ccccc1)C(C)C)OC Cc1cccc(C(=O)NC(C2CCCN2C(=O)C=Cc2ccc[nH]2)C)n1 c1(SC(C)C(=O)NC2CC2NC(c2cnnn2C)=O)ccnc2cc(Cl)ccc12 CC1=NC(C(=O)NC(C2CN(C(c3ccoc3)=O)C2)C)CS1 C(C)(C)(CCCNC(=O)C(C)NC(c1ccco1)=O)NC(CCNC(C)=O)=O C1(N(C)C)CC(NC(=O)CCN(C(C2CCNC2=O)=O)C2CC2)C1(C)C c1(N)nc(C)c(Br)c(C)n1.C12(C(=O)OC)CC(C(=O)NC(C3(CO)CC3)=O)(C1)C2 c1(C(N2C(CNC(=O)CCOC3COC3)C=CC2)=O)cccc(SCCO)c1 C(=O)(C(F)C(C)CC(C)(C)C)N1CC(CC)C(NC(=O)C2=NOC(C)C2)CC1 N1(C(CCc2c(C)nccc2)=O)CC2CN(C(C3C4CN(C)CC34)=O)CC(C1)O2 N1(C(CCOC)=O)CCC(C(F)CNC(c2ccccc2C(=O)OC)=O)CC1 C(=O)(CC(C)C1CC1)N1CCC(CN(C(CC2C(CN)CC2)=O)CC2CC2)C1 CC1(C)CCOC1CC(=O)N(c1ccc(OCc2ccccc2)cc1)CCCl c1(C(=O)NCN2CCCC(COCC=C)C2)ccc(Br)c(Cl)n1 c1(C(N(C)C)=O)ccccc1CC1(C)N(C(CCCN(C)C)=O)CC1 C1(C)(C(=O)N(C2(CC=C)CN(C(c3sc(C4CC4)nc3C)=O)C2)CC)CC(C)=NO1 C(=O)(C1OCCc2ccccc21)NCC1(NC(C2CC(CC)OCC2)=O)CC1 N1(C(=O)CCOC2CCOCC2)CCCC2C1CCN2C(C1CC12CC(O)C2)=O Cc1cc(C(=O)NCC2CC(NC(C3CC(Cl)(Cl)C3)=O)C2(C)C)ccn1 C(=O)(C1CCCc2c[nH]nc21)NCC(CC=C)NC(c1n[nH]c2c1COCC2)=O c1(OC)cccnc1C(=O)NCc1cccc(CNC(C2(C)CC(C)=NO2)=O)c1 c1(OC)ccc(CC(O)C(=O)NC2(CNC(=O)C=C3CC3)CCOC2)cc1 C(=O)(C1Cc2c(Cl)cccc21)N1CC2(C(NC(C3(OC)CCC3)=O)CCC2)C1 C1(NC(C2C(C)N(C)CC2)=O)CC2(CCC(NC(=O)CCC3(C)CC3)CC2)C1 CC1CCC(O)(C(=O)NC2CCN(C(c3c(C#N)cnn3C)=O)C2)CC1 c1(CNC(C(C)(C)NC(CNC(C=C)=O)=O)=O)ccc(F)cc1 c1(CC)nc(C)c(C(=O)NC23CC(CNC(C4CCCS4)=O)(C2)C3)o1 c1(C(N2C(CCNC(CN(CC)CC)=O)C(C)CCC2)=O)cc2ccccn2n1 C(=O)(C1CCc2ccccc21)NC(=O)CC1CC1CC1CC2(CCC2)C1 c1(C(=O)NCC(C)(C)NC(=O)CC2CC=CCC2)c(O)nnc2c1CCCC2 Cc1nc(N2CCN(C(=O)CCc3nc[nH]n3)CC2C(C)C)ncc1Br N1(c2c(C(=O)OC)cncc2)CC(NC(C2CC(F)(F)C2)=O)CC(C)(C)C1 c1(C(N2CCC(C3OCCO3)C2)C(=O)NC(C)(C)C)cc2sccc2s1 c1(CNC(C2(CCC=C)CN(C(=O)CC3CC4CCC3O4)C2)=O)ccccc1O C1(CC(=O)NCC(O)C2CCC2)CCN(C(c2scnc2Cl)=O)CC1 N1(C(C=CC(CC)C)=O)CCOCC(C(=O)N(C2CCC2C)C)C1 O=C(N=c1c(Cl)c[nH]cc1Br)c1ccc(NS(=O)(=O)CC2CC2)cn1 CC#CCCCC(=O)N(CCC(=O)N(CC(C1CC1)OC)C)CC N1(C(COc2ccn(C)n2)=O)CC2C3CCC(C(NC(=O)CNC(N)=O)C3)C2C1 C1(CC=C)(NC(c2n[nH]c(COC)n2)=O)CCN(C(C2(C#N)CC2(C)C)=O)CC1 N1(C(CCCc2ccc(C)cc2)=O)CCCN(C(C2CC(F)C2)=O)CC1 c1(C(N(C2CCN(C(C3CC4CC4C3)=O)C2)C)=O)cccc(CO)c1 C1(NC(C(CC)C2CCC(=O)N2)=O)CC(NC(=O)Cc2cccnc2)CC1O C(=O)(CC1OCCc2ccsc21)N(CCNC(c1c(CC)scn1)=O)C(C)C n1(C(C)C(=O)N(C(C)C)Cc2ccncc2)cccc(C(F)(F)F)c1=O c1(C(=O)NC2CC(NC(COC)=O)C2)cccc(C2CCCN(C)C2)c1 O=C(N=c1cc2n([nH]1)CCCC2)C1CC2(CCC2)CN1C(C1CC=CC1)=O C1(CNC(c2c(OCC)n[nH]c2)=O)CN(C(C23CCCC2C3)=O)CC2(CCC2)O1 C1(NC(c2c(CCC)n(-c3cccc(N)c3)nn2)=O)NCCC12CCCC2 Cc1cc(O)ncc1NC(C1CCC(C)CN1C(=O)CNC(=O)CN(C)C)=O c1(C(=O)NCCC2CCN(C(C(C3CCC3)OCC)=O)C2)nc[nH]c2nccc1-2 C1(CC)CCCCC1NC(=O)CCCNC(=O)CSCCOC(C)=O N1(C(C(C)(C)C#N)=O)CC2(CCC2NC(=O)C(O)C2CC2)C1 C=CC1(O)CCN(C(C2(C)CCN(C(=O)C(C)NC(=O)NC)C2)=O)C1 c1(C(=O)NCC(CCOC)NC(C(C)OCC)=O)ccc(-c2ccco2)nc1O N1(C(CNc2ccc(C#N)cc2)=O)CCOCC12CCN(C(=O)CCC(N)=O)C2 C1(CN(C)C)(OC)CCN(C(=O)Nc2nc(C3CCCCO3)cs2)C1 C1(C)(CNC(CC(C)CN(C)C)=O)CCN(C)C1=O.c12cccnc1C(=O)NC2 C(C(F)(F)CCC(=O)OCC1CC2(C1)CC2F)n1cc(-c2ccc(C)cc2)nn1 N1(C(C=NOC)=O)CCN(C(c2ccc(C(C)C)cc2)=O)C(c2ncc[nH]2)C1 C(CC(C)C)(C(=O)NCC1CC(CNC(=O)CCCC2CC2)C1)NC(C)=O N1(C(CC(CC)NC(=O)CCCCCOC)=O)CC(C)(C2CCC2)C1 CN1CCN(C(=O)CC2CC(C3CC3)C2)CC1C(N1CCC(O)(C(N)=O)C1)=O c1(OC)ccc(-c2csc(N)n2)cc1OC.N1(CC)C(C(=O)O)CCC12CCCC2 CCCC(CNC(c1ccnnc1C)=O)C(=O)N1CC(C)C1(C)C c1(C(=O)NC(CNC(c2c(C)nn(C(C)(C)C)c2)=O)(C)C)ccc(F)c(F)c1F Cc1c(C)c(CNC(=O)NCC(c2ccccc2)(C)O)c(C)c(C)c1Br Cc1cccc(Cl)c1C(=O)NC1(C#N)CCN(C(c2ccnc(Cl)c2F)=O)C1 C1(OC)CC(c2nnnn2CC2CCOC2)(NCC2CCCCC2)C1 N1(C(C(C)(CO)OC)=O)CC2CCC(C1)N2C(=O)CNS(=O)(=O)c1ccccc1 C1(OC)CCC2(C(=O)NC3CCOC3C(N3CCC(C)(C)C3)=O)CC12 CCC(C#N)(CC)C(=O)N1CC(CNC(=O)C(C)CCOC)(COC)C1 c1(-c2nc(SCCCCNC(=O)NCC(C#C)O)c(C)o2)ccc(Cl)c(Cl)c1 C1(NC(c2cccc(OC)c2Cl)=O)CN(C(=O)C#CC2CCCC2)CC(C)(C)C1 S(=O)(=O)(c1cccnc1N1CCC(C)C1C)N(CC(C)C)CCCOCCO OC1CN(CC2CCNC2)CCc2ccccc21 N1(C(C(C)SC)=O)CC2(C1)CN(C(=O)Cc1c(C)cccc1F)CC(C)(C)O2 C1(C)(CC(=O)NC(C(=O)OCC)C2CC2)CCN(C(C2CC(O)C2)=O)C1 Cc1cnc(CNC(C2(NC(C3C4CCC(F)C34)=O)CCN(C)C2)=O)cn1 c1(C(N(C(CNC(CN(CC(C)C)CCC)=O)C)C)=O)cnc2ccccc2n1 C(=O)(CC(C)C(F)(F)F)N1CCCC(CCn2cc(CCCC)nn2)CC1 C(=O)(C(C)(C)S(=O)(=O)C1CC1)NC(CN(c1c(C#N)ccc(CC(C)C)n1)C)C C(C(F)C(=O)NC1(CCF)CC1)C1CN(C(CC=CC=C)=O)C1 C1(C(N(C2CCN(C(C3(C)CCC3)=O)CC23CC3)C)=O)Cc2cccc(F)c2O1 C1(C(=O)NC2C(C)(C)CN(C(c3cc(C(N)=O)no3)=O)C2)CNC(=O)CC1(C)C c1(C(=O)NC2C(C#N)CN(Cc3ccccn3)C2)c[nH]c2nccc-2c1Cl Cn1nc(C(F)F)cc1C(=O)NC1CCC(NC(=O)CC2COC(=O)C2)CC1 c1(N(CC(=O)NCC(C2CC2)NC(C(C)OCCN(C)C)=O)C)ccc(Cl)nn1 Cc1cc2ccccc2c(NCC2(CO)CCOCC2)n1 C(=O)(CC(C)(O)C(F)(F)F)NC1CCCN(C(C(C)Sc2ncccn2)=O)CC1 C1(F)(CO)CCC(Nc2cccc(C(F)C(F)(F)F)n2)CC1 N1(C(C(C)CC(N)=O)=O)CCCC2C1CCN2C(c1ccn2ccnc2c1)=O c1(C(C)C(=O)NCC2CCN(C(C3CC(C)(O)C3)=O)C2)cccc(C#N)c1 C1(NC(C(CCCC)O)=O)CCOC2(CCN(C(=O)C=CS(C)(=O)=O)CC2)C1 C(=O)(CCCC(F)(F)F)NC1CCC(CNC(c2cc(C(=O)OC)[nH]c2)=O)C1 C1(NC(C2C(C)OC(=O)N2)=O)C2CC(O)C1N(C(=O)C(F)=C1CCC1)C2 C1(NC(C(COC)(C)C)=O)CCN(C(C2CCOCC2)=O)CCC1CO Cc1cc(=O)n(C)cc1NC(C1CN(C(=O)COC2(C)CCC2)CC12CCC2)=O C1(C2CCN(C(=O)CC3COCC3(C)C)CC2)(NC(CN(C)C(N)=O)=O)CCC1 N1(C(c2nccc(C)c2)=O)CCC(NC(=O)CNC(c2ccco2)=O)C(CO)CC1 N1(C(c2ccc(OCCCC)cc2)=O)CCN(C(=O)C(O)CN(C)C)CC12CC2 C1(NC(C(CCC)N(C)C)=O)CC2CN(C(c3cccc(C4(C)CC4)c3)=O)CC12 C(C(C)(C(=O)NCC1CC1Cl)NC(=O)Cn1cc(C)cn1)SC C1(NC(C(C)OC2CCOCC2)=O)CC(C)N(C(=O)CCc2nc[nH]n2)C1 c1(C(=O)NC(CC(C)NC(C2CC(C#N)C2)=O)C)ccnc2c1CCO2 c1(NC2CC3(C)CC(O)C32)nc(N2CCCC(F)(F)CC2)nc2cc[nH]c12 N1(C(c2ccsc2)=O)CCC2CN(Cc3ccc(Br)cc3F)CC12 C1(C2(NC(CCOCC#C)=O)CC2)CCCN1C(=O)C(F)C1CC1 C1(NC(c2occc2Cl)=O)CC2CC1N(C(=O)CCc1nnc(O)nc1O)C2 C1(C(N2CC(C(=O)NCC3CCC(C)CO3)(SC)C2)=O)(OC)CC(C)(C)C1 c1(CC)ccc(C=CC(N2CC(CNC(c3cn(C4CC4)cn3)=O)C(C)C2)=O)o1 C(CC(C)(O)C(C)(C)C(=O)NCc1cc(OC)cc(CC)c1CC)OC(F)(F)F C1(CC(N2CCC(CC)C2C(=O)N(C(C)C)C2CC2)=O)CN2CCN1CC2 Nc1ccc(C(=O)NCCC2(O)CCCN(C(=O)C=Cc3cc[nH]n3)C2)cc1O Cc1cc(C(=O)NC2CC(O)CN(C(=O)CCC(C)(C)C)C2)c(C)nc1C CC(C)C(CC(=O)NCC1CCN(C(=O)CCN2C(C)CCCC2C)C1)C(C)C Cc1nnc2n1CC(C(=O)N(C1CN(C(=O)CCc3cnoc3)CC1(C)C)C)C2 C1(NC(c2cnn(C(F)F)c2)=O)CN(C(c2cnns2)=O)C2CCCCC12 c1(NC(C2CN(C(C3CC(O)(CC#C)C3)=O)CC23CC3)=O)ccccc1N=[N+]=[N-] CCC(CC)C(O)CNC(=O)C#CCNC(c1cocc1C(N)=O)=O N1(C(c2ccc(CC)cn2)=O)CC2(CCC2)CC1CNC(=O)C(C)n1ccnc1 N1(C(C2(COC)CC2)=O)CCC2(CCC(NC(c3csc(Cl)c3)=O)C2)C1 C1(C)(CNC(c2n(CC)cc(Cl)c2)=O)CCCCN1C(c1scnc1Cl)=O Cc1ccc(-n2cc(C3CCCCN3C(=O)CCCC3CCC3)nn2)c(C)c1 C1(C(=O)NCCCCC(=O)N(C(CSC)(C)C)C)CCC(C2CC2)C1 C(=O)(CCCCCF)NC1C(OC)CN(C(=O)CCOC2COC2)C1 N1(C(C2C3CC(=O)CC32)=O)CCCCC(NC(C2CC23CCCCC3)=O)C1 c1(C(=O)NCC(C(C)C)NC(C2CN3CCN2CC3C)=O)ccc2occc2c1 O(NC(=O)C(CNC(=O)C(C)N=[N+]=[N-])CC(C)C)CCC(C)=O C1(C)(C(=O)NCC2CCC(C(CC)C)CC2)CCCN(CC(=O)O)C1 CC(C)CCC(=O)NCC12COC(CNC(C3CCCC(N(C)C)C3)=O)(C1)C2 c1(CC(N2C(C)CCC(NC(c3cc(Cl)c(Cl)s3)=O)C2)=O)cn2ccccc2n1 c1(CC(=O)NCC(C(C)C)(C)NC(=O)C(O)CC[S+](C)C)cnc2cccnn12 C=C1CC(C(=O)NCCC(C)N(C)C)(CNC(c2ccc(SC)o2)=O)C1 Cc1cc(F)c([N+](=O)[O-])cc1-c1nc2c(s1)CN(c1ccncn1)CC2 Cc1cc(C#N)ccc1C(N1C(C(=O)NC2CCOC(C)(C)C2)CCC12CC2)=O CN1C(=O)CCC1CC(N1CCOC(C(=O)N(C2CCC2)C2CCC2)C1)=O C1(NC(C=CCC)=O)C(C)(C)CN(C(C2(CCF)CCC2)=O)CC1(C)C Cc1nc(CC(=O)NC2CC(C(=O)NC3CC(=O)N(C4CC4)C3)C2)[nH]c1C C1(NC(C(CC)n2ccnc2)=O)CC2CN(C(=O)CCN(C)CCO)CC12 CCC(CNC(c1cncc(C(C)(F)F)c1)=O)(CC)NC(=O)CCCF C(=O)(C(F)(F)C(C)O)N1C(C)CC(NC(=O)COc2cccc(F)c2)C1 C#CCCCC(C)C(=O)N1CCCC(N(C(c2cn[nH]c2)=O)CC2CC2)C1 C1(NC(CS(CC)=O)=O)CCC2CCN(C(c3cc(OC)ncc3F)=O)C12 C1(C(N(CC(F)F)C)=O)CCN(C(=O)CC(O)C2CCCC2)C(C)(C)C1 C1(C(=O)OCC)CN(C(c2[nH]c(C3CC3)nc2C)=O)CCC12OCCO2.OCC C1(NC(C(C2CCOCC2)OCC)=O)CCN(C(c2ccc(C)c(N)c2)=O)CC1F N1(C(c2cnc(C)[nH]2)=O)CCC(C(C)NC(=O)CCN2CCC(F)C2)CC1 c1(C(C2CC2)C(=O)O)nc(C2CC(NC(c3cnn(C(F)F)c3)=O)C2)no1 C1(NC(c2c(C)csc2Cl)=O)CCN(C(c2occ(C)c2C)=O)CC1CO c1(NCC(C2CC2)SC)cc(N2CCOC(C3CCOCC3)C2)ncn1 CCC(Cc1ccccc1Br)C(=O)NCCCN(C(=O)C(C)N(C)C)C C1(C(=O)NCC2CCC(NC(CC3C(=O)OCC3)=O)C2)OCC2COCCC12 N1(C(C(=O)NC)=O)CC(CC(=O)NCc2nc(C3CC3)oc2C)C2(CC2)C1 C#CCC(CC(F)F)C(=O)NCC1CCN1C(=O)CCn1ccnc1C CC(O)C(C)(C)C(=O)NCC(C)N(C(=O)Cc1cccc(O)c1F)C C1(C#N)(C(=O)NCCC2(NC(C3C(C)CC3C)=O)CCC2)CC12CCC2 N1(C(C23CC(NC(=O)CC4COCCO4)(C2)C3)=O)CCOCC2CSCC12 C(=O)(C(C)(C)CC1CCOCC1)N1CC(NC)C1 C(=O)(C(C)(C)CCCN=[N+]=[N-])N1CC(C)(CNC(C(C(C)C)OC)=O)C1 C(=O)(C1=CCN(C(c2ccc(C3CC3)o2)=O)C1)NCCCC1CC(C)C1 c1(C(N2CC3CC3(NC(=O)C(Cl)(Cl)Cl)C2)=O)ccc2c(c1)CCO2 c1(C(N2CC(F)(CNCc3nccs3)C2)=O)ccc(F)c(F)c1 Cc1c(NCCN2CCCC2CO)nc[nH]c1=NCC(=O)N=S(C)(C)=O c1(C(N(C(C(NOC(CC)CC)=O)C)C2CC2)=O)cc(F)cnc1O C1(N(C(=O)CNC(c2ccns2)=O)C)CCN(C(=O)Cn2cccn2)CC1 CCCC(CC)C(=O)NC1CC1NC(=O)C(C)C1CC1 N1(C(COC(C)=O)=O)CCC(C(F)(F)F)C(NC(c2ccc(C)c(F)c2)=O)C1 C=CC1(C(=O)NCc2cccc(O)c2C)CCN(C(=O)C(Cl)=CCl)CC1 Cc1cncc(C)c1C(=O)N(CCCCCC(=O)NCC1CC1(F)F)C C1(OC)CN(C(=O)CC2(C)CC2)C(C)(CNC(C2(F)CCOCC2)=O)C1 Cc1cn2c(n1)CC(C(N1CC(NC(c3cccc(C(F)F)c3)=O)C1)=O)CC2 N1(C(c2cccc(NC)n2)=O)CCN(C(c2cnn(C)n2)=O)C(C)C1C C(=O)(CCC(N)=O)N1C(C(C)NC(CCCOCC)=O)CCC1 N1(S(=O)(=O)CCNC2CCCCNC2)CCCc2cc(Br)c(F)cc21 N1(C(C)=O)CCc2cc(S(=O)(=O)N3CCC4CCCCC4C3)ccc21 c1(C(N2CC(CNC(=O)CC3CCCCC3F)C2)=O)ccc(Cl)c(Br)c1 C1(CC(N2CC(C)(NC(C3C(c4ccc(C)s4)C3)=O)C2)=O)CC(=O)NC1=O C(=O)(C1CNC(=O)c2ccnn21)NC(CC#C)C(=O)NCC1(CC2CC2)CC1 c1(OC)cnc(F)c(C(N2CCC(CO)(NC(c3cc(Cl)cc(Cl)c3)=O)C2)=O)c1 C(=O)(C(CCC)S(N)(=O)=O)NC(C1CC(NC(C(CCC)=CCC)=O)C1)C N1(CCCCC(C)c2ccccc2)CCCC2(CCCO2)CC1 N1(C(C=CC=CC)=O)CCC(F)(CNC(=O)C(F)(F)CC2CCCO2)CC1 N1(C(c2cncc(OC)n2)=O)C2CCC1C(CO)N(C(c1csc(C)n1)=O)C2 c1(C(N(CCN(C(c2c(CC)c[nH]c2)=O)C)C)=O)cc(O)ccc1OC CCC(C)(C)CCCC(=O)NC1CC2CN(C(c3[nH]cnc3C)=O)CC2C1 c1(C(N(CCCCNC(=O)C(F)F)C)=O)n[nH]c2cc(Cl)ccc12 C1(C(=O)NCC(C)CN(C)C(c2cccc(C(F)F)c2F)=O)Cc2cscc2C1 Cc1nn(C(C)(C)C)cc1C(=O)N(C)CC1CCCN1C(=O)CC1CCC2CC12 c1(OC)ccc(C(=O)NC2CC(C)N(C(=O)C(F)=C3CCC3)C2)cc1O N1(C(CSSC)=O)CCC2(CCCN2C(=O)CN(c2ccncc2)C)C1 C(CCNc1cn(C)nc1C)(C(=O)N(C)C(=O)OC(C)(C)C)NC(=O)OC Cc1ccc(C(N2CC(NC(C3CC(F)C(=O)N3C)=O)CC2CO)=O)cc1C C(C(C)(C)CC(=O)NCC1(F)COCCOC1)n1cc(C(CC)O)nn1 c1(NC(=O)NC)ccc2c(c1)CN(C(c1cscc1Br)C(=O)NC1CCC1)CC2 c1(-n2cc(C3N(C(Cn4c(C)cnc4)=O)CC3)nn2)cnnc(O)c1Br C1(C(N(CCN(C(C(C)=C2CC2)=O)C)C)=O)CCOC2(CCC2)C1 Nc1cc(F)c(C(N2CCOCC(NC(=O)CCc3cnc(O)[nH]3)C2)=O)cc1F C1(NC(CCCCOC)=O)CN(C(=O)Cc2nnc(C)s2)C2(CCOC2)C1 C1(C(N(C(CC)CNC(=O)Cc2ccc(OC)nc2)C)=O)CC2CCCC2C1 C(=O)(CC(C)C(C)(C)C)NC(C(=O)NCc1c(CC)nn[nH]1)CCC1CC1 N1(C(C2(C3N(C(C)=O)CCC3)CC2)=O)CCCC(NC(=O)CCC#N)C1 C1(C)(C(=O)NCCCc2ncn(C)n2)CCN(C(C2CC(=O)CS2)=O)C1 c12ccccc1C2.C1(CN(C(C2C(=C)C2)=O)C)CCCN1C(=O)CCSC Cc1cc(C(N2CC(CNC(c3ccc(N)cn3)=O)CC2C)=O)c(F)c(Br)c1 C(=O)(CS(=O)(=O)C1CC1)N1CC(CNC(c2c(C)cncc2C)=O)C(C)CC1 c1(SCNC(C(C2CCCCCC2)N(CCCC)C)=O)ccc(OC)c(OC)c1 CN1C(=O)CSC1=CC(=O)N1CCCC(C2(NC(c3c[nH]ccc3=O)=O)CC2)C1 C1(C)(CC)CC(NC(=O)Cn2cccc2)CN1C(=O)CCc1c(Cl)cncc1Cl C1(C(=O)O)(C(=O)NCc2ccccn2)CC2(CCC2)C1 C=C(F)C1(CC(N2CCC2CNC(C2CCCN2CC(F)(F)F)=O)=O)CCC1 N1(C(c2nnc(C(C)C)s2)=O)CCC(C2CCOCCN(C(=O)CN(C)C)C2)CC1 C(=O)(CC(C)CCCCC)N1CCC(CNC(C(C=C)OC)=O)(CO)CC1 C1(CNC(COc2cc(C)on2)=O)CC(F)(F)CN1C(=O)CC1CCOCC1 N1(C(C(CC=C)CC=C)=O)CCc2ccc(C(=O)NC(C)(CC)CC)nc2C1 C(=O)(CCCCC(=O)NCCCC1CCN(C(C2(C)CCCO2)=O)CC1)NC C(=O)(C1=CC2C=CC(C1)C2)NC1CC(C)(NC(=O)CSC(F)F)C1 N1(C(=O)NCC(C)(C)NC2CCC2)CCCC(F)(c2cn(C)nc2)C1 Cc1cc(C2CCC2)ccc1C(=O)NCC(C)CNC(=O)Cc1ccccc1F N1(C(C2CCN(C)CC2)=O)CCC(NC(=O)C=Cc2cnc[nH]2)C1(C)C Cc1scc(C(=O)NCC2(CNC(C3CC3C(C)(F)F)=O)CC2)c1Br C1(C(=O)NCC2C(NC(=O)CCOCc3ccccc3)C2)CC2(CC(=O)N2)C1 C1(CC)CN(C(=O)C(C)(C)N(C)C)CCC1NC(c1ccc(SC)cc1)=O C(CC1=CCCCC1)NC(C1C(CNC(Cc2c(C)noc2C)=O)CC1)=O CCCC(C)(O)CC(=O)NC1CC(NC(=O)C(c2cccc(Br)c2)C)C1 CCC(CC(F)(F)F)C(=O)NC1CCCC(NC(c2conc2COC)=O)C1 c1(C(=O)NC(C(C)(C)C)CNC(C2CC3(CSC3)C2)=O)cc(F)c(F)cc1Cl CCCCC(=O)C(=O)NCC1CC1.C12CCN(CC1)CC1CCC(O1)C(=O)N2 O=C(CCCS(=O)(=O)N1CCCC1)NC1(CF)CCN(C(=O)C(F)n2ccnc2)C1 CCC(CC)(CO)C(=O)NCC1(C)CN(Cc2nccs2)CCO1 C1(C(=O)NCc2cc(C(=O)NCCC3CC(F)(F)C3)co2)(CC)CCNC1=O C1(NC(=O)Cc2csnn2)CC(NC(C2CC3(CCCC3)C2)=O)C12CCC2 c1(C(=O)NC(C)CCCNC(c2ccncc2O)=O)ccccc1C#CC1CC1 S(=O)(=O)(c1ccc2nc(N3CCOC(C)(C)C3)sc2c1)NCCOC(C)C S(=O)(=O)(c1ccccc1F)NCC(=O)N(C1CCCN(C(C(C)C#N)=O)C1)C CON1CC(C(=O)NC(CNC(c2cc(C)c(CO)o2)=O)C(C)C)CC1=O C(CC(C)(C)CNC(C1(F)CC=CC1)=O)NC(C(CC)n1nccc1C)=O C=CC(C)(O)C(=O)NCC1(O)CCN(C(c2cc(F)n[nH]2)=O)C1 c1(C(=O)NCC=CCNC(C(C(C)C)n2ccnc2)=O)ccc2nn[nH]c2n1 CC(C)(C)CCCC(=O)NC1CC2CC1CC2CNC(=O)CC1C(=O)ON=C1C C1(CCC)CCCC1C(=O)NCC1CCCC1NC(=O)COCc1ncnn1C CC(CC(=O)NCCOC1CN(C(=O)CC2CCCSC2)C1)C(F)F c1(C(=O)NCCC(C)(C)NC(c2ncc(C)c(Cl)c2)=O)cccn2nccc12 C1(OC2CC(NC(=O)CC3COC3)C2)CCC2C(C1)C2(F)F c1(NC(c2ccc(NS(C)(=O)=O)cc2)=O)ccc(F)c(C(N2CCCC2)=O)c1 c1(NC(C2(C)CN(CC3CCC(F)(F)C3)C2)=O)cc(O)ccc1F C(=O)(CCCNC(=O)C1CC1)NC(C1CCN1C(c1cn(CCO)nn1)=O)C N1(C(CCC)=O)CCC2(C1)CN(C(=O)C=CSc1nc[nH]n1)CC(C)O2 N1(C(COCC)=O)CC2CC3CC2C1C3NC(c1ccc(OC)c(Cl)c1)=O CC1(C)CC(N=c2cc(NCc3cc4c(nc3N)CCC4)nc(C(F)F)[nH]2)CO1 c1(C(=O)NC(C(=O)NC(c2nncs2)C)CO)ccc(=N)[nH]c1 c1(CN2CC3C(C(=O)Nc4c(C)c(F)ccc4)(C3)C2)ccc2ccc(Cl)cc2n1 CCCCS(=O)(=O)CC(=O)N1CCC(Nc2cnc(C#N)cn2)C(C)C1 C(CC(C(=O)NC1CC(O)C(O)C1)NC(=O)Cc1cncnc1O)OCC c1(NC(C2CC2NCc2cccc3sccc23)=O)cc(Cl)c(F)cc1F C#CCC(CC(=O)NC1CCC2(CCC2)C1)NC(c1ccsc1C#N)=O C1(C(N2CCN(C(C3CC(C)(C)OC3)=O)CC2)=O)C2CCC3C(C2)CC13 c1(OC)cc(NC(N2CCNC(c3ccnn3C)C2)=O)c(F)cc1C c1(CN(CCC)Cc2ccc(C3CC3)cc2)ccc(C)cc1Br c1(C(=O)NCC2(O)CCN(C(C(C)=O)=O)C2)cc2n(n1)CCCC2 CCC(C(=O)OC)C(=O)N1CCC(C)(NC(c2cnn(C)c2Cl)=O)CC1 N1(C(C2(C)CC(=C)C2)=O)CCC(CNC(=O)C(C)SCCCC)(OC)C1 N#Cc1ccc(CN2CCCC(C(=O)NCC(N3CCOCC3)=O)CC2)cn1 n1(CCN(C(C(C2CCCC2)NC(C)=O)=O)C)cc(C)cn1 c1(OC)ccc(CC(=O)NC2CC(NC(=O)CCCOC(C)=O)CC2O)c(F)c1 N1(CCC#C)CCC(C(N2CC3CC2C3NC(c2nc(O)sc2C)=O)=O)CC1 N=c1[nH]c(N2CC3CC(NC(C4(C(N)=O)CC4)=O)C3C2)ncc1[N+](=O)[O-] Cc1nc2c(cc1NC(=O)NCC(c1cc(F)cc(Br)c1)N)c(C)nn2C C1(C2CC2)(C(N2CCCC(F)(CNC(C(C)n3cnnn3)=O)C2)=O)CCOCC1 CC(CN=c1[nH]c(=NCC2CCCCS2(=O)=O)[nH]c2ccccc12)S(C)(=O)=O C1(OCCN(C)C(=O)NC2(COC)CCOCC2)CC(=O)NC(CC(C)C)C1 C1(NC(CCC(C)O)=O)CCCC12N(C(c1ccc(Cl)c(Cl)c1)=O)CCC2 c1(C(=O)NCC2(C(=O)Nc3c(Br)cnn3C(C)C)CC2)cc(Cl)cc2nc[nH]c12 c1(C(=O)NC2C(NC(C(CC)(C)OC)=O)COCC2)coc2c1COC2 N1(C(C2C(=C)C2)=O)CC(NC(c2ccoc2Cl)=O)CCC1C CCC(O)C(C)C(=O)NC1CCN(C(c2cc(C)[nH]n2)=O)C1C c1(CC(=O)NCC2CC2CNC(=O)C(O)CC2CC2)csc2cccc(F)c12 N1(C(c2c(C)nsc2N)=O)CCCC(NC(=O)C=Cc2ccc(F)cc2)CC1 c1(C(=O)NC(C(=O)Nc2c(C)cccc2)Cc2ccccc2)ncn2c1CCCC2 C(C(C)(C(=O)N(C)Cc1c[nH]nc1C)NC(=O)Cc1cc(C)on1)SC c1(C(N2CC(CCNC(=O)C(C)C(O)CC)(OC)C2)=O)ccc2nc(O)[nH]c2c1 C1(CC(=O)C=O)COCCN1C(=O)CCc1cn[nH]c1.c1(NCCN)cccnc1 c1(C(N2CCC(C)(CNC(C(F)=C(C)C)=O)C2)=O)ccc(C(C)C#N)cc1 N1(C(c2ncc(C)o2)C(=O)NC(CC)C)CCN(C(=O)NC)CC1 c1(C(N(CCC)CCNC(C2CC(OC)C2)=O)=O)nccc2ccn(C)c12 c1(C(=O)NC(CC)CN(C(c2ccccn2)=O)CC)cc(F)c2ccccc2c1 c1(C(c2n(C)nnn2)NCc2ccc(Cl)cc2F)ccc(S(N)(=O)=O)s1 c1(NC(=O)CC2CCN(C(=O)C=CC(F)F)C2)ccc(CSC)cc1 C1(NC(CC(C=C)(C)O)=O)CC2(CCC(NC(=O)C3=CCC(C)CC3)CC2)C1 c1(C(C)(F)C(=O)NCCNC(C2(C(O)C(F)(F)F)CCC2)=O)ccccc1F Cc1cn2c(C(N3CC(NC(C4(CF)CC4(F)F)=O)C(C)C3)=O)c(C)nc2s1 C12(NC(C(N)=O)=O)CCN(C(C3(S(N)(=O)=O)CC3)=O)CC1C2 N1(C(CC(C)(C)O)=O)CCC2CC1CN(C(=O)C1=CC3(CCOC3)C1)C2 c1(C(N2CCN(C(C(CC)C#N)=O)CC2C(F)F)=O)nc2ccccn2c1F C1(C(=O)NC(CSC)(C)C(=O)NC2CCCC2N(C)C)CCN(OC)CC1 C(C(=O)NCCN1CCC(NC(=O)C(F)C(C)C)CC1)(C(C)C)NC(=O)OC c1(C(N2CC(CNC(CSSC)=O)C2)=O)ccc(-c2ccc(C)o2)nc1 N1(C(=O)CC2(CO)CC2)CC2(CNC(C3C=CCC3)=O)CC1CCO2 c1(C(C(=O)N(C2CN(C(COC(C)=O)=O)CC23CC3)C)O)cc(F)c(F)cc1F c1(C2C(C(=O)NC3CC(O)(CNC(CC=C=C)=O)C3)C2)ccccc1F c1(C(=O)NCC(C2CCCC2)NC(C=C(COC)C)=O)cc(C)c(C)[nH]1 c1(N(CCCNC(c2cc(CF)on2)=O)CC)nc2ccc(N)cc2s1 c1(C(N2CC(C)C(CNc3cc(C(F)F)ncn3)CC2)=O)c([N+](=O)[O-])cnn1C N1(C(C(CC(=C)Cl)NC(c2cnsn2)=O)=O)CCC2CCC(C1)N2C c1(C(N2C(C(=O)NC(CC=C)C(=O)OCC)CC=CC2)=O)cccn2ccnc12 c1(C(=O)NC2CN(C(COC)=O)C(C)(COC)C2)c(C)cc(C#N)cc1C C1(NC(CCCOC(C)C)=O)CC(C(N2CC(C)(F)C2)=O)C12CCC2 N1(C(CCNC(=O)OC)=O)CCCC(CCNC(c2cnc(O)n2C)=O)C1 c1(-c2cn(CCCCCNC(CC3CCN(CC)C3)=O)nn2)cccc(F)c1F Cc1c(Cl)nc[nH]c1=NCC1(NC(C2CCN(C(C)C)CC2)=O)CCCC1 C1(CNC(CSC(C)C)=O)CN(C(=O)C(C)CSc2ccccc2)C(C)(C)C1 Cc1ncn(C)c1C(=O)NCC1CC(CNC(=O)C(C(C)C)c2cnn(C)c2)C1 O(CP(C)(C)=O)CCOC(C(C1CC(NC(=O)OC(C)(C)C)C1)F)=O c1(CC)cc(C)c(C(=O)NC2CCC(CNC(c3cnco3)=O)CC2)o1 C(=O)(CCCCC(C)C)NCCCOCCNC(c1cn(CC=C)nn1)=O c1(CF)cc(=NC(Cc2ccc(F)cc2Br)C2CCCCC2)[nH]c(C(F)(F)F)n1 C12(C(N3CC(C)(NC(=O)CC4CCCNC4=O)C3)=O)CCCN1CCC2 C1(CNC(C(C)OC)=O)CCN(C(=O)C(C)(C)n2ccnn2)CC1O c1(CC)oc(C(=O)NCCC2CCC(NC(C3CC4CCC3O4)=O)C2)cc1C C1(C(=O)NC2(C(C)O)CC2)CCC2CCC1N2C(C1CCC(=O)O1)=O CC1(C)COC(CC(=O)NC2C3CC2N(C(=O)C(C)(C)C)C3)C1 C(=O)(N1CCCc2nncn21)C1(CNC(=O)CC2CCC=CCCC2)CC=CC1 c1(NC(C(=O)NCCSCCCC)=O)cccc(-n2cnnc2)c1 C=CCCC(F)(F)C(=O)NC12CC1CN(C(c1cc(Cl)c(Cl)s1)=O)C2 C12(NC(C(C)NC(C)=O)=O)COC(CNC(=O)CCNS(C)(=O)=O)(C1)C2 c1(C(=O)NC2CCC(N(C(C(COC)C)=O)C)C2)ccccc1N=NN(C)C Cc1c(N)ccc(C(=O)NCC2CCCCN2C(=O)C#CC2CCCO2)c1C C1(C(=O)OCC)CC(NC(=O)C(C)NC(=O)CCF)C(O)C1 c1(CCC(N2CCN(c3ccc(OCC)cc3)CC2CO)=O)cccc(Br)c1Cl C1(NC(c2nc(C)oc2)=O)CCC2(CC1)CN(C(=O)C(C)(C)C(C)C)CCO2 C1(CCNC(Cc2ccc(C)cc2)=O)CN(C(=O)Cc2cn[nH]c2)CC(C)O1 CCC(O)(C(=O)N1CC(NC(=O)C=C2CCN(C)CC2)C1)c1ccccc1 c1(C(=O)NCC2CC3CCC(C2)C3F)ccc2c(c1)CCC2=O c1(N(CCC)C)ccc(C(=O)NC2CN(C(c3ccc(F)o3)=O)CC2C)cc1 c1(C(N2CC(CC=C)(NC(=O)C=CCO)C2)=O)cc(Br)c2c(c1)nnn2C c1(CC)c(C(=O)NCC(C)(C)CN(C(=O)Cc2cnccc2C)C)nnn1CC c1(-c2c(C)n[nH]c2C)cccc2c(C(=O)Nc3cccc(Br)n3)[nH]nc12 CC1(C)CCC(O)(C(N2CC3CC2C3CNC(=O)CCc2nc[nH]n2)=O)CC1 c1(CNC(C(CNC(c2nnc(C)s2)=O)OC)=O)cc(C)ccc1O c1ccccc1-c1nc(C)c(C)o1.C1(CN(C=O)OC)CC(C)=NO1 CCC(CC(=O)NCCN(C1CCCCC1)C(c1ccc(OC)nc1)=O)C(F)F c1(C(N2CC(C(C(=O)NC3(CC=C)CC3)O)C2)=O)occ2c1CCC2 c1(OC)cccc(Cl)c1CC(=O)NCC(C1CCC1)NC(C1CCC(=O)N1C)=O c1(C(C(=O)NCCCSC)N(C)CC2COC(C)(C)O2)cc(Cl)cc(Cl)n1 c1(C(=O)NC(CNC(c2ccc(C#C)cc2)=O)C2CC2)cc2n(n1)CCCO2 CS(=O)(=O)c1ccc(N2CCN(C(=O)CCC(F)F)C(C3CCCC3)C2)cc1 c1(C(N2CCC(CNC(c3ccc(CF)cc3)=O)C2)=O)cc(O)cc(F)c1 N12CCCC(F)(C1)C2.c1(SCCNC(CC)=O)cccc(C)c1.C(=O)(C(C)OCC)N C1(C)(CNC(c2c(C)cn(C)n2)=O)CN(C(C2CC3(C2)CC(C)C3)=O)CCO1 CCS(=O)CC(=O)NC1(C(=O)NCc2nn(C)cc2C)CCCC1 N1(C(CSC)=O)CCC(C2(O)CN(C(C3COCC(C)O3)=O)C2)CC1 C(=O)(CCCCN(C(=O)Cn1cc(CNC(C2CC(C(N)=O)C2)=O)nn1)C)NC Cc1ccc2c(=NC(C)CN3CCC3)[nH]c(=NCCCCO)[nH]c2c1 C(=O)(C(C)(CNC(=O)CCc1cncs1)CC)NCC1(CC)CCOC1 C1(CNC(c2nccc(CC)c2)=O)(NC(C2CCN(C)C2)=O)CCC(C)(C)CC1 C1(N(C(c2cnc(CC)s2)=O)C)CC2CC1N(C(c1cc(Cl)ccc1N)=O)C2 N1(C(C(C2CCCC2)OC)=O)CC(C)OC2(CCN(C(=O)CCC[N+](=O)[O-])C2)C1 c1(SCN2C(=O)CC(C(N3CC(N4CCN(C)CC4)C3)=O)C2)cc(Cl)ccc1F C(=O)(C1=CS(=O)CCC1)N(C1CC1)CC1N(C(c2c(C)cc(SC)o2)=O)CCC1 c1(-c2cn(CC3N(C(Cc4nnc(COC)s4)=O)CC3)nn2)ccncc1C C(=O)(CCCCCc1ccccc1)NC(CN(C(c1cnc(CC)s1)=O)C)CC c1(OCC)ccc(OC)c(-c2nc(CNC(C)CC(C)C(F)F)co2)c1 N1(C(C(C)OC)=O)CCCC2(C1)CN(C(=O)C(F)Cc1ccccc1)CCO2 C1(NC(C(C)CC2CCC2)=O)CCN(C(=O)Cc2ccnc(C(F)(F)F)c2)CC1 N1(C(C2(F)CCN(C(CCCOC(C)=O)=O)C2)=O)CCc2ccc(C)cc21 c1(C(=O)NC)ccccc1O.C(C(=O)NCC)O.C(=O)(CN(C)C)N.C1COCC1 c1(C(=O)NC2CC(NC(CCc3ccc(C)o3)=O)C2)ccc(S(N)(=O)=O)cn1 C1(C(N(CCC(C)C)C)=O)CCN(C(c2cnc(C3CC3)o2)=O)C1C(C)C Cc1cc(NC(=O)CC2CC(NC(c3c[nH]c(C(N)=O)c3)=O)C2)c(O)cc1F C1(NC(C2CCC(C)C2)=O)CN(c2nc(Cl)ncc2Br)C2CCCCC12 C1(C#N)(CC(=O)NCC23C(CN(C(c4n(C(C)C)ccn4)=O)C2)C3)CCCCC1 c1(OCC(=O)NCCC(=O)NC)ccc(Br)c2ccccc12 CC1(C)CC(NC(C2CC3CCC(C2)S3)=O)CCN(C(c2scnc2Cl)=O)C1 CC(C)(CC(=O)NCCC1(CNC(C2CCC3(C2)CC3(F)F)=O)CC1)CC(F)F c1(C(N2C(CNC(c3cc(CCC)n[nH]3)=O)CC2)=O)cc2c(cc1O)CCCC2 CCC(C)CCCC(=O)NC(C(=O)N(C)Cc1n[nH]c(C)n1)C1(O)CCC1 c1(CN(C(C(CN(C)C)NC(=O)CC2CCCCO2)=O)C)ccccc1Br Cc1c(C(N2CC(NC(c3sccc3C(C)C)=O)C(C)C2)=O)nn2c1CCCC2 Cc1ncccc1C(=O)NCC1CC(NC(c2cc(-c3ccc(C)o3)[nH]n2)=O)C1 C1(C(=O)NC(C2(O)CCN(C(=O)Cc3ccccc3C)C2)C)CC12CC(O)C2 C1(NC(C(C)N(CCC)C(C2CCOC2C(C)C)=O)=O)CCN(C)CC1(C)C c1(C(N2CC(NC(=O)C=Cc3cnccn3)C2)=O)cccc(S(=O)(=O)C(F)F)c1 C1(C)(C(=O)NCCC(C)N(C(c2ccc(OC)c(C)c2)=O)C)CCC(=O)N(C)C1 c1(C(N2C(CNC(Cc3nc(C)c(C)s3)=O)COCC2)=O)ccc(F)c(C)c1N Cc1csc(C=CC(=O)NC2CC(C)(NC(c3cnc(N(C)C)s3)=O)C2)n1 N1(C(CNC(CC)=O)=O)CCC2(CC2NC(C2CN(C)CCN2C)=O)C1 N1(C(C2(C)CCC(=O)C2)=O)CC2(CCN(C(C3C4CCCCCC34)=O)CC2)C1 c1(C(=O)NC2C(NC(C3C(C)CCO3)=O)CCCC2)cc2nc(F)ccc2o1 CN1CCCC(O)(CC(N2CC3C(CNC(=O)CCc4csc(=N)[nH]4)C3C2)=O)C1 N1(C(CC=CC)=O)CCC(F)C(NC(=O)CCNC(=O)CO)C1 c1(C(=O)NCCC2(O)CCN(C(CC(C(C)C)O)=O)C2)nccc2ccccc12 CC1CNc2ccc(C(N3CCN(C(C4CC4C4CC4)=O)CC3)=O)cc2C1 N1(C(c2cn(C(C)C)nn2)=O)CCN(N2CCCC(C)C2)CC1C1CC1.C(=O)CO CCC(C)(C(=O)N1CCC(N(C)C(c2ccn3ccnc3n2)=O)C1)C(F)F c1(C(N2C(CCNC(C(CSC)OC)=O)CCCC2)=O)c[nH]c2nccc-2c1C c1(C(c2ccccc2)N(CCOC)C)cc(OC)ccc1C(C)OC.c1(S)ccccc1 c1(C(=O)NCC(C)NC(C2(CCOC)CC2)=O)ccc(NC(C)=O)s1 N1(C(CNC(=O)C2CC2)=O)CCN(C(=O)C(Cc2ccccc2)C2CC2)CC1CO c1(CC(N2C(CNC(c3cc(CO)on3)=O)CC(OC)C2)=O)c(C)ncnc1O c1(C(C(=O)NCC)N(C)Cc2cnn(C)c2)csc2ccc(C)cc12 C(CN=c1[nH]c(=NC(C)c2nnnn2C)c2c(ncn2C)[nH]1)(C(C)C)OC C1(NC(c2cccc(C)c2)=O)CC2COCC(C1)N2C(C1CCCC1(F)F)=O CC1(C)CN(C(=O)CCC2CC2(Cl)Cl)CC1CNC(=O)CN1CCSCC1 C(CC(=O)N1CC2C(C1)C2(F)F)(C(F)(F)F)NC(c1ccccc1C1CC1)=O CC1(C)CC(C(=O)N(CCCNC(=O)C2=CCSC2)CCO)CCO1 CC1CCC(C(=O)NC2CSC2)N(C(C2CC=CCO2)=O)C1 C(=O)(CC1=CCCC1)NC(CCCNC(c1c(OC)cccc1)=O)C C1(N(C(c2c(C)noc2)=O)CCF)CCCN(C(=O)CC23CCC(CC2)C3)C1 N12CCC(CC1)C2=O.N1(CC(=O)NCC(C)N(C(=O)NCC=C)C)CCCC1C Cc1ccncc1C(=O)NCC(O)CN(C)C(C1(C)CC=CC1)=O c1(CC(=O)NCCCN(C(c2cc(CC)c(O)cc2)=O)C)ccc2n[nH]cc2c1 c1(C(=O)NCC(C2CCC2)NC(CCc2ccn(C)c2)=O)c(C2CC2)cnn1C N(C(=NCCc1ncnn1C)NC(c1ccc(F)cc1F)C)C(C#C)CC c1(CN2CCC(NC(c3cccc(F)c3Cl)=O)C(F)C2)cc(O)c(O)cc1O c1(C(N2CCC(CN(C(c3cc(C)on3)=O)C)CC2)=O)cc(F)c(Cl)c(N)c1Cl N1(C(CCOCCOC)=O)CC=C(CNC(=O)CNC(=O)C2CC2)CC1 N1(C(c2ccc(OC)c3c2CCCC3)C(=O)NC(C)C)CC2C(=O)N(C)C(=O)C2C1 c1(CC)scc(C)c1S(=O)(=O)N1CC(Cl)CC1c1nc(Cc2ccccc2)no1 c1(CC)cc(C(=O)N(C(C)(C(=O)NC(c2ccc(C)s2)C)C2CC2)C)ccn1 c1(Nc2cccnc2)ccnc(N(C)C)n1.n1(CCCNC)cncn1 N1(C(C(CC)(C)CC)=O)CCC(C)(C)C(NC(=O)CCOc2cccc(C)c2)C1 c1(C(N2CCC(O)(CNC(CSC)=O)C2)=O)cc(Br)cc2nc(O)[nH]c12 C1(C(=O)NC(CCC2N(C(CC(C)C)=O)CCCC2)(C)C)CCN(C)S1(=O)=O C1(C(=O)Nc2cnc(F)nc2)CCCN(C(C2CC=CC(O)C2)=O)CC1 N1(C(c2csc(Br)n2)=O)CCC(O)(CNC(C2(F)CCCOC2)=O)C1 C1(C(N(C)CC2CCCS2)=O)CC(F)CCN1C(=O)COC1CCOC1 C1(C(=O)NC23CC(NC(c4ccc(C)nc4)=O)(C2)C3)C2CS(=O)(=O)CC12 c1(OC)cccc(Cl)c1C(N1CCC(NC(=O)CC2CSCCS2)C1)=O N1(C(c2c(CC)ncs2)=O)CCC2(CCCC2C(=O)Nc2ccccc2I)C1 C(CCC)(CCC)=CC(=O)NC(CC=C)CNC(c1cnn(C(F)F)c1)=O CC1(C)CCC2(CC1)CC2C(=O)NC12CC(NC(c3cc4n(n3)CCO4)=O)(C1)C2 N1(C(C2CCCO2)=O)c2ccccc2CC1CCO.c12cn(nn1)C2 C1(CC(C)NC(c2cc(OCC)n[nH]2)=O)CCN(C(=O)Cc2cnn(C)c2)CC1 c1(C(=O)NC2CCC(NC(c3c(COC)noc3)=O)C2)ccc(C)c(C)c1O C1(C(N(C2CN(C(C3CN(C)C3)=O)C2)C)=O)CCc2nn(C)cc2C1 CCC(C)C(CC(=O)NCc1ccc(OC)s1)NC(C1CC1C1CCC1)=O CC(C)CC(C)CC(C)C(=O)NCC1(C2(O)CN(C(=O)Cn3cnnn3)C2)CC1 C1(CC(=O)N(C)CC2(NC(c3n[nH]c(C)c3Cl)=O)CC2)CCC2(CC2)CO1 N1(C(Cc2ncc(CC)[nH]2)=O)C2CCCC1CN(C(=O)C=C1CCC(C)C1)C2 Cc1ccc(F)cc1NC(c1csc(NC(C2CCS(=O)(=O)C2)=O)n1)=O CC1CN(C)C(C)CN1C(C1CN(Cc2cccc(Cl)n2)CC(F)(F)C1)=O CC(C)(CS(N)(=O)=O)C(=O)NCCNC(C1CCC(C(=O)O)S1)=O CS(=O)(=O)c1cccnc1N1CCC(NC(=O)CCn2cccn2)C(F)C1 c1(NCC2CCC(C(N(CC(C(=O)OC)(C)C)C)=O)CC2)ccc2n[nH]cc2c1 N1(C(c2cnc(CC)s2)=O)CCCC(NC(c2cc(F)c(F)c(F)c2)=O)C(F)C1 c1(C(=O)NCC2(F)CCC(CNC(CC)=O)C2)c(C)sc(C)c1Br N1(C(c2cccc(O)c2)=O)C2CC(F)C(C2)C1C(N1CC2CC(C1)O2)=O Cc1cccc(CC(=O)N(C2CC(NC(=O)CC3CCC3C(=O)O)C2)C)c1F CCCC(C#N)C(=O)N1CC2(CC2)CC1CNC(c1cc(C(C)C)on1)=O C1(CNC(CNC(C)=O)=O)C2CN(C(c3cn(C(F)F)cn3)=O)CC12 c1(NC(=O)NC(C)C(c2ccc(OC(F)(F)F)cc2)C)nc2c(Cl)cccc2o1 C1(C(=O)NCC(C)S(N)(=O)=O)CCC(C)CN1C(=O)C=Cc1ccnn1C C1(C)(CCC(=O)NC(CC)COC)CCCN1C(=O)CC1CCCCO1 c1(C(N2CC(NC(c3ccc(C)cc3Br)=O)C(C)C2)=O)cnn2cccc(C)c12 C1(C(N2CC(N(C(C(n3c(C)ccn3)C)=O)C)C2)=O)COCC(=O)N1C(C)C CCCC(CC)CC(=O)NCC(C1CCC1)NC(=O)C(c1ccc(F)cc1)(C)O C(C)(N=c1cc[nH]c2ccc(OC)cc12)c1c(OC)nccc1 Cc1ccc(C)n1CCC(N1CC2(NC(C3CCCC(CF)C3)=O)CC1C2)=O c1(C(N2CC(C)C(NC(c3cnncc3O)=O)C2)=O)ccn(C)c(=O)c1 C=C(C)C(C)(C)C(=O)N1CCC(CCNC(c2cccc(SC)n2)=O)C1 c1(C(=O)NC2CCCC(N(C(c3cc(C)oc3)=O)C)C2)ccc(N(C)C)c(F)c1 C(=O)(C1=CC(C)(C)C1)NC1CN(C(c2c(OC)nccn2)=O)C(C)C1 C1(CC(=O)NCC(CNC(CCCOCCOC)=O)(C)O)CC2CCC1CC2 N1(C(CCCCCC)=O)CC(OC(CC(=O)NC(C)=O)=O)C2CCCCC12 c1(C(=O)NC2CCN(C(CCc3ccc(C)nc3)=O)CC2)ncc(C#N)cc1C N1(C(CN2CC(C)(OC)C2)=O)CC2CC1CN2C(c1ccc(N)c(Cl)n1)=O C1(C)(CNC(CCC2OCC(C)(C)C2)=O)CN(C(=O)COCC(F)F)C(C)(C)C1 N1(C(C(CC=C)C)=O)CCN(C(c2cccc(COC)c2)=O)C(CCO)C1 N#Cc1c(Cl)c(C(=O)NC2CCC(NCc3scnc3Cl)C2)cc(F)c1Cl N1(C(CCc2nc(C)sc2)=O)CCC(O)(CN(C(=O)C(F)C2CCOC2)C)CC1 NC(=O)CC(C(=O)N1CCCC(C(F)F)C1)NC(=O)Cc1cnsc1 C=CC1CCCN(C(=O)CC(c2cc(F)cc(F)c2)C)C1 N1(C(C(C)CC2CCC2)=O)CC=CC(C(=O)N(CC(N)=O)CC(N)=O)C1 C1(NC(C(CC=C)CC)=O)CCC12CCN(C(=O)CNS(=O)(=O)N(C)C)CC2 Cc1nc(N(CC(O)CN(C)C(c2cnn(CC(C)C)c2C)=O)C)c(C)c(O)n1 n1(CC(C)(C)C)nc(C2Cc3ccccc32)nc1-c1ccc(OC(F)(F)F)cc1 C1(NC(C2CN(C)C2)=O)C2CCC1N(C(=O)CCC1CCCC(=O)N1)C2 Cc1[nH]c(=N)ccc1C=CC(=O)NC1CC(NC(c2ccc(Cl)[nH]2)=O)C12CCC2 c1(CCC(N2C3C(NC(=O)Cc4ccco4)C(C3)C2)=O)nnc(S)nc1O N1(C(c2nccc(N)c2)=O)CCCC1C1CCCN1C(c1cc(Cl)no1)=O CC1CN(C(=O)C(c2ccc(Cl)cc2)=O)CCCN1C(c1nn(C)cc1N)=O N1(C(CCn2c(C)cc(C)n2)=O)CC2(CC(CN3CCC(F)C(F)C3)CO2)C1 c1(NC(=O)Nc2c(C)cc(N(C)C)cc2)cc2nncn2cn1 N1(C(C(CSC)O)=O)CCN(C(=O)Cn2nc(C)cc2C)CC(O)C1 C(=O)(C1CCCn2cnnc21)NCCC1CC(NC(c2cc(C)cc(F)c2)=O)C1 c1(CC)n[nH]c(=NC(=O)NCC(Cc2ccc(Cl)cc2)CO)s1 c1(OCC)cc(C(=O)NCC2CC2NC(=O)CN2CCCC2)[nH]n1 C(=O)(C(CC(F)F)NC(=O)C(C)NC(N)=O)NC(CC)C(C)O CP(C)(=O)c1cnc(C(=O)NC2CC(O)(CNC(c3cnccn3)=O)C2)cn1 c1(NC(N)=O)cccc2c1C1CN(C(c3cc(F)ccc3Cl)=O)CC1O2 C1(CNC(C(C(C)C)SC)=O)CCN(C(C2CC(C(C)=O)C2(C)C)=O)CC1C C1(C(=O)NCc2cccc(C(=O)NC(c3ccc(C)s3)C)n2)CC2CCCC2C1 C=C(C)CCCC(=O)NC1CCCCC1NC(c1cn(C)c(=O)n1C)=O c1(C(=O)NCCCCC2CC2)ccc(Cl)c2occc12 c1(C(=O)NC2CCN(C(C3CCC(C(=O)OC)C3)=O)C2)ccccc1C(N)=O C1(NC(C2(C(=O)NC)CCC2)=O)CCCCN(C(=O)CCc2c(C)noc2Cl)C1 C(CC(C(C)C)NC(=O)C(F)n1cccn1)N(C(CCCSC)=O)C C1(C(=O)OCC)CN(C(=O)NCc2cnc3n2CCC3)CC2(CCC2)O1 c1(CC(N2CC(C)C(CCNC(c3ccco3)=O)C2)=O)coc2cc(F)ccc12 C1(CNC(C2C(OCC)C2)=O)CC2COCC2N1C(=O)CCNC1CCOCC1 CC(C)CC(C)CC(=O)N1CCC(CCNC(C23CCC(C2)C3(C)C)=O)C1 N#CC1(C(=O)NCCCN(C(=O)C(F)n2ccnc2)CCO)CC2CCC1CC2 c1(CNc2c(C#N)nccc2)ccc(S(=O)(=O)N2CCCC2)o1 c1(NC(C23CC(C(=O)NCCc4ccco4)(C2)C3)=O)cccc([N+](=O)[O-])c1 C1(NC(C(C)OCC#C)=O)CN(C(=O)C(c2nc(C)cs2)C)CC2(CCC2)C1 CC1CCOC(C2C(C(=O)NC3CCCC3)C2(C)C)C1.C1CO1 C1(NC(=O)C=CC2CC2)CC2CCC(C1)N2C(=O)CCc1cc(F)ccc1F C1(CNC(CC(=O)OCC)=O)CN(C(C2CC(C)OC2C)=O)CC1C C(=O)(CCCC(C)(F)F)NCC1CCN(C(CSc2cccc(C)c2)=O)C1 CC1CC(C(=O)NCCCNC(=O)CC2CS(=O)(=O)C2)CC(C)C1 CC(C)CCC(F)C(=O)NCCCCC1(NC(c2ccnc(O)c2)=O)CC1 c1(C(=O)NCCCNC(Cc2cnc(C)s2)=O)cc(N)c(O)c(F)c1 N1(C(c2cc(CNC(CN3CCC(C)C3)=O)oc2)=O)CCC2(CCC2)CC1 N(C1CCCc2nc(CC)sc21)C(=O)Nc1ccc(N(CCC)CCC)nc1 C1(NC(C=CC(C)(C)NC(C2CC(OC)C2)=O)=O)CCCC(CO)CC1 N1(C(C(=Cc2cn[nH]c2)C)=O)CCC(C(N2CC3CC2CS3)=O)(CO)C1 N1(C(c2c(CNC(C=CC(CC)C)=O)c[nH]n2)=O)CCc2ccsc2C1 C#Cc1ccc(C(=O)NC23CCCN(C(=O)CCCOC)C2C3)cc1F c1(NC(C)Cc2c(F)cc(F)cc2F)ccc(S(=O)(=O)NC2CC(F)C2)c(Br)c1 C1(CC(=O)NC(CCC=C)C2CC2)C2CCCC2N1C(c1ccc(C)cc1F)=O CCCCCCNC(=O)C(c1nnc(CC(C)C)s1)N(C)CC1CC(C)(C)C1 c1(NC(CCN(CC(N)=O)C2CC2)=O)cc(C(F)(F)F)cnc1O Cc1cc(C(=O)NC2(CNC(c3cccnc3O)=O)CCCCC2C)cc(O)c1 C1(CC#C)(C(=O)NCC(O)CNC(c2cccc(NC(N)=O)c2)=O)CCCCC1 c1(C(=O)NCCCC(C)NC(=O)C2CC2)c(O)ccc(F)c1Br c1(OC)cc(CC(=O)N(CCCCN(C(=O)C(C)OC(C)=O)C)C)ccn1 C1(NC(CC=C=C)=O)CC2CCC1N(C(=O)Cc1ccc3c(c1)CCO3)C2 Nc1c(C(N2CCC(CCNC(=O)C(N)=O)C2)=O)cc(Cl)nc1Br CCC(O)C(C)C(=O)NC1CCCC(C(=O)N(C)CC2(OC)CCC2)C1 O=C1CC(C(=O)N2CCN(C(=O)CC3CCC(C(F)(F)F)O3)CC2CO)=NN1 c1(C(N)=O)cncc(C(=O)NCC2CCN2C(=O)CC2(O)CCOC2)c1 c1(C(N(CCOCCNC(C(C)=C(C)C)=O)C)=O)c(C)ccc2ncccc12 C1(CNC(COCCSC)=O)CC(C)N(C(=O)COCCCC(C)C)C1 c1(CC)cncc(C(N2CCC(N(CC3=NOCC3)C(C)=O)C2)=O)c1 n1(C(CC)CC)ccc(C(=O)N(CCNC(C2CC2=CC(C)(C)C)=O)CC)n1 Cc1ccc(C)c(C(N2CC3(CC3)CC2C(N2CCCC(C)C2C)=O)=O)c1O c1(C(=O)NCC(C(C)C)NC(CCn2c(C)csc2=O)=O)cc2cccnc2[nH]1 C=Cc1ccc(CNCC2CC(Nc3c(Cl)ccnc3Br)C2)cc1 C=C(C)CC(C(=O)NCCOCC(N)=O)NC(=O)CCc1cnco1 C1(C(C)C)CN(C(c2ccc(C(N)=O)o2)=O)CC1C(=O)N(CC(C)(C)CO)C Cc1occ(C(F)(F)F)c1C(=O)NCC1CN(CC(N2CC3C(C)C3C2)=O)C1 Cc1cnccc1CNC(C1C=CCN(C(=O)CCCN(C)C)C1)=O C(=O)(CC(O)CC(C)C)NCc1c(C(=O)NC(C#C)C(C)C)cco1 N1(C(c2cc(OC)n[nH]2)=O)CCCC12CN(c1ccc(C(F)(F)F)nn1)C2 C(=O)(CCCC(F)F)NCCCCNC(=O)COC1CC1(F)F CC(C)(CN=c1[nH]c(=NCc2cn3ccsc3n2)[nH]c2ccsc12)CC(F)F C1(NC(C=CCN(C(C(c2ccccc2)C)=O)C)=O)CC2CC2C1 c1(C(=O)NC(C)C(CO)NC(=O)CC#N)cccc(OC2CCC2)c1 C1(C(=O)NC(CC(=O)OC)(C)c2cccc(F)c2)CC2(CO1)CC(F)(F)C2 N1(C(c2c(C)c(N)ccc2)=O)CCC2CN(C(=O)C=Cc3cn[nH]c3)CCC2C1 Cc1nc(C(N2CCC(C(C)C)C2)C(=O)NCc2cccs2)oc1C N1(C(C)=O)CCC(C2CCN(C(c3cn(CCO)nn3)=O)CC2)CC1 c1(C(=O)NCCCN(C(=O)CCCC2CCOCC2)CC)sccc1Br c1(C(CO)N(C(CC(C)CC)=O)Cc2c(CC)csc2)ccccc1F c1(CN(CC=C)C(c2nc(C(=O)OC)cs2)=O)ccc(OC)c(OC)c1 N1(C(=O)NC2CCC(Oc3ccc(F)cc3)C2)CC2CC(O)CC1C2 c1(C(=O)NCC2(O)CN(C(C3OCC(C)C3)=O)C2)ccc2c(c1)CC2 c1(NC(CN(CC(C)C)C(=O)CN2CCC(C3CC3)C2)=O)ccncc1N C1(C2CC2)(CNC(CCOC)=O)CCN(C(=O)CC2CCNC2=O)C1 c1(C(=O)NCC2(c3nc(=O)[nH][nH]3)CC2)ccc2c(O)n[nH]c2c1 N(C(=NCc1cccc(F)c1)NCCN1CCC1)CC1(CCOC)CCCC1 C1(NC(C2CC(C#C)(O)C2)=O)(CNC(c2cc(OC)n(C)n2)=O)CCCCC1C c12ccc(cc1)-c1nc(cs1)CC=CCOC2=O.N1(CC)CCCCC1C(=O)O Cn1cccc(C(N2CC=CC(C(=O)NC3(C)CC4CCC3C4)C2)=O)c1=O N1(C(=O)CCc2ccco2)CCc2[nH]nc(C(N3CCC(O)C(F)C3)=O)c2C1 C1(OC)CC(NC(=O)Cn2ccccc2=O)CN(C(=O)CC2COCCN2C)C1 c1(CN(CCCO)C)cccc2cc[nH]c12.C123CC1CN(C2)C3=O N1(C(CCCCSC)=O)CCOCCC1C(=O)N(C)CC1COC(=O)N1 n1(CC)c(C(=O)NCC(C(C)C)NC(=O)CC2CCCC23CC3)cnc1O N1(C(C2(CCCC)CC2)=O)CCCC(C2(NC(=O)Cc3cnc(C)o3)CC2)C1 CC1CN(C(=O)CN2C(=O)CN(C)C2=O)C(C)CN1C(=O)COC1(C)CCC1 c1(C(=O)NCC2(C(C)NC(C(C)C3CCCC3)=O)CC2)cc(C#N)c[nH]1 c1(C(=O)NCC(C2CCOC2)NC(C=C(C)Cl)=O)csc(-c2cccnc2)n1 N1(C(CCC2CCC(C)O2)=O)CCN(C(c2cncc(CO)c2)=O)C(CC2CC2)C1 C1(CC#C)CN(C(c2cn(CCNC(=O)CCn3cnnn3)cn2)=O)CCO1 CCC(CC(=O)NC(C1(C(=O)NC(C)C(C)(C)CN(C)C)CC1)C)OC CC1COC(C(N2CC(O)(C(C)NC(=O)CC#N)C2)=O)C1 N1(C(c2n(C3(C)CC3)ccn2)=O)CCC(O)(CNC(=O)CCN2CCCCC2)C1 C1(O)(CNC(C2(CC)CCC2)=O)CCCN(C(C2Cc3nnsc3S2)=O)CC1 Nc1c(NCC2CC(n3cncn3)C2)cc(F)cc1C(F)(F)F C(=O)(C1CCc2cccnc21)N1CC(N(C(C(C(C)C)SC)=O)C)C1 C1(C(=O)NC(CC)C(F)(F)F)CC2(CC2)CN1C(=O)Cc1ccc(C#N)cc1 N1(C(=O)OC(C)(C)C)CC(NC(C(=C)C(C)C)=O)CC(c2cnn(C)c2)C1 CC1CCC(NC(c2ccc(NC(C)=O)s2)=O)CN1C(=O)CCCC1CC1 N1(C(CN(C(=O)OCC)C)=O)CC2CCC1C(NC(=O)CC1CC(F)(F)C1)C2 N1(C(CCNC(N)=O)=O)CCN(C(=O)CC2CCCOCC2)C2CCC12 C1(CCNC(C2(C)CC2)=O)CC2CCC(C1)N2C(=O)CCc1ccc(F)c(F)c1 c1(C(=O)NC2CC(F)(CNC(C(C3(O)CCCCC3)CC)=O)C2)ccnc(C)n1 c1(COC)nn[nH]c1C(N1CCC(N(C)C(c2ccn(C3CC3(F)F)n2)=O)C1)=O C(C)(CC)(CCNC(C1CC(N=[N+]=[N-])C1)=O)NC(C=CCN(CC)CC)=O N1(C(C2CC(C#C)(O)C2)=O)CCC2(NC(c3nnc(C(F)(F)F)s3)=O)CCCC12 N1(C(Cc2nc(C)oc2)=O)CCOC(CN(C(=O)C(C#N)=CC(C)C)C)C1 c1(CCC=CC(=O)N(CC(C)NC(=O)CCSC(F)(F)F)CCO)ccccc1 Cc1cc(O)ccc1C(=O)NCC(C1CCCCN1C(C1C=CCCC1)=O)(C)C C#CCC(C(=O)OC)NC(C1CCCN(C(C2CC=C(C)CC2)=O)C1)=O C1(NC(C2CCCN(C(=O)OC(C)(C)C)C2)=O)(C)CCOCC1.C1(O)CC1F C1(NC(CCCC)=O)CN(C(=O)CN2C(=O)CCCC2=O)C2(CCC2)C1 c1(C(N2CC(N3CCN(C(C(C)OC)=O)CC3)C2)=O)ccnc2ccsc12 N1(C(c2c(C)[nH]c(C(C)(C)C)c2)=O)CC2CC1CN(C(C1CCSCC1)=O)C2 C(CN=c1[nH]c(=NC(C)CCOc2ccccc2)[nH]c2c1CSC2)OCC CC1C(=CC(N2CCCC2C(C)NC(C2C=CCCC2)=O)=O)CCCCC1 CCC(C#N)C(=O)N1CCC(C(C)C(=O)NCCC2CC=CC2)CC1 c1(NC(C)=O)nc2cc(C(N3CCCC(n4ccnc4)C3)=O)ccc2o1 C(=O)(C(F)CC(C)(C)C)N1C(C(=O)N(C)CC2CCCOC2)(CC)CCC1 CC1(C)COCCC1CN1C(C(=O)NCC2CC3CCCC3C2)CC=CC1 C1(C(=O)NCC2(CCNC(c3cc(CO)[nH]n3)=O)CC2)CCc2nnc(O)n2C1 c1(C(N2C(CNC(CC3(COC)CCC3)=O)COCC2)=O)cncc2[nH]ccc12 c1(C(C)OCCOC)nc(CCC(C)C)nn1-c1ccc(CCC(C)C)cc1 N1(C2C(C)SCC2)CC(C(=O)NCc2cc(C(=O)O)c(C)o2)C(F)C1 C(=O)(C(CC)(CC)C(=O)O)N1CCN(CC(N2C(CC)C=CC2)=O)CC1 c1(C(=O)NC(CN(C(C2CC3CC3C2)=O)CC)C)cc(C)n(-c2cccs2)c1C N1(C(CCC)=O)CCCC1(C)CNC(=O)COC1CCOC1 c1(-n2cc(CN(CC(=O)O)C(=O)CN3CCOCC3)nn2)ccc2c(c1)CCO2 N1(C(C(C)OCC)=O)CC2(CCC2NC(=O)CCCOc2ccc(Cl)cc2)C1 C1(CSCCNC(=O)C(=O)NC2CC2)CCCCN1C(=O)C=CBr N1(C(C2(C)CNC(=O)C2)=O)CCCC(F)(CNC(c2sccc2C2CC2)=O)C1 N1(C(c2c(C)nc[nH]2)=O)CC2(CC(CNC(=O)CC3CC3(C)C)C2)C1 N1(C(C2N(C(CCOCC#C)=O)CCN(C)C2)=O)CCC2CCCC2CC1 C#Cc1cc(C(=O)NC2CC2CNC(=O)C2=NNC(=O)C2)cc(C(F)(F)F)c1 C(C(O)C(=O)N)NC(CC(=O)CCN(C)CCO)C(C)C.C(C(=O)NC)SC C=CCC(F)(F)C(=O)NCC1CCN(C(=O)Cc2cc(F)cc(Cl)c2)CC1O C(=O)(CC(C)C(C)(C)NC(c1cscc1Cl)=O)N(C(C)C)CC Cc1ccc(-c2ccccc2-c2ccccc2)cc1C(=O)Nc1ncc(Br)cc1O CC(C)(CNC(c1ccc(NC(N)=O)cc1)=O)CC#N N1(C(C(CCC)O)=O)CC(CNC(=O)C(C)OC)CC12CCOCC2 CC(C)CC(CC(=O)NCC(C)(C)CN(C)C(C1CCC1C(F)F)=O)CC(N)=O c1(C(CC)NC(C2(CCNC(=O)C=CCO)CC2)=O)cn(C)nn1 C1(C(N(C2CN(C(=O)C=CBr)CC2F)C)=O)CCC2CC1C2(C)C N1(C(CC2CC(C)(C)OCC2)=O)CC2CCN(C(=O)COc3ccccc3)C2C1 C(=O)(C(C)OCCNC(C1(N(C)C(C2C=C2C)=O)CC1)=O)OC C(=O)(CCCCN1CCCC1)N(CCCC)CCCC.C(=O)(C(C)C#N)NCCN C(=O)(CCCCN(CC)C)NCC1(C(=O)NC2(CF)CC2)CC1.c1(C)ccc(C)cc1 C1(CC#C)(NC(c2cn(CCNC(C3CCC3)=O)nn2)=O)CCCCC1 CC12CC(C(N3CCC(CNC(=O)Cc4nc(=N)[nH][nH]4)CC3)=O)(C1)C1(CCC1)O2 N1(C(C(CC)NC(C(CC=CC)C)=O)=O)CC(=O)NCC1CC CCCCCC(O)CC(=O)NCCC(C)(C)NC(=O)CC1CC12CC2 C1(NC(C)=O)COCCC1OCC(=O)C(c1cn(Cc2ccc(C)cc2)nn1)C CC(CN(C)C)CC(=O)N1CCCC(C(C)(C)C(=O)NC(C2CCC2)C)C1 C1(C(=O)NC(c2nc(CC)[nH]n2)C)C2CC(O)C(C2)N1C(c1cocc1C)=O C1(NC(c2c(C)[nH]cc2)=O)COC2(CNC(=O)C=CBr)CC1C2 N1(C(CC(=C=C)C)=O)CC(CNC(=O)Cn2ccccc2=O)C2(CC2)C1 C(C)(C(C)(C)C(=O)N1CC=CC(OC)C1)NC(CNC(C(CC)C)=O)=O Cc1nc(O)ccc1C(=O)N(CC(=O)NC1CCC2CC2CC1)C Cc1nc(C)n(O)c1C(=O)NC(CNC(c1ccoc1Br)=O)CC(F)(F)F c1(O)cc(C(=O)C(=O)NC2CC2OCCl)ccc1C.N(CCO)(C1CC1)CC Cc1cnc(CCCC(=O)NCC2(F)CC(NC(=O)C(=O)N(C)C)C2)o1 C1(NC(C2(C)CCCC2)=O)CCCCN(C(C2CCC3(CCC3)O2)=O)C1 C1(C(N2CC(O)(CNC(C(C)OC3COC3)=O)C2)=O)C(C(F)(F)F)C1[N+](=O)[O-] c1(CCC(=O)N(C(CC)C2CC2)C)c[nH]c2ccccc12 N12CCC(C(C)C)(C1)C(=O)Nc1csc(n1)C2=O.C(C(CC1CC1)OC)SC C1(OC)CC(NC(c2oc(C3CC3)nc2C)=O)CN(C(C2CCC2OC)=O)C1 C1(C(=O)NCCCN(C(c2ccc(OCF)cc2)=O)CC)CCCC(C)(C)CC1 N1(C(CC2(OC)CCCCC2)=O)CCC(C)C(NC(=O)CC2CCOC2C)C1 C1(C)(CC)CC(NC(=O)CCNC2CC2)CN1C(c1ccccc1Cl)=O C1(CNC(Cc2cn(C)nc2)=O)CC2CCC(C1)N2C(=O)C1=CCS(=O)(=O)C1 C1(NC(Cc2cc(C)n(C)n2)=O)CN(C(c2cnc(N)c(Cl)c2)=O)CCC1(C)C n1(CCCC)cc(C(=O)NC2CCC(NC(C3CCC3(F)F)=O)C2)nn1 Cc1nc(C(N2CCCC2C2(Cc3cn(-c4cnn(C)c4)nn3)CC2)=O)cs1 c1(NC(c2ccncc2-c2ccsc2)=O)cc([N+](=O)[O-])c(Br)cc1F Cc1cc(C(=O)NC(CNC(c2cc(C(N)=O)[nH]n2)=O)C2CC2)ccc1C(C)C Cc1cc(CC(N2CCCC2CNC(=O)COC(C)(C)C)=O)nn1C CC(C)C(C)(O)CNC(=O)C(CCC1CCC1)NC(=O)COCCF C(=O)(C1=C(Cl)CCC1)N1C(C2CCN(C(C(C(=O)OCC)OC)=O)C2)CCC1 Cc1oc2cc(C(=O)NC3CCC(NC(=O)COC4CCOC4)CC3)[nH]c2c1C n1(CC)c(C(=O)NCC2(NC(=O)C(C)SCC(=O)NC)CCCC2)cnc1O C=CCC(C)(CC)C(=O)NCC(F)(C(=O)NCCC1CC(C)=NO1)C(C)C N1(C(C2CC2F)=O)CCC(C2CCN(C(=O)C(C3CCOCC3)F)CC2)CC1 c1(C(N2CCC(C3CC3)(NC(C)=O)C2)=O)cnc2c(c1)CNC2=O C1(C(N2CC(N(C(c3c(CC)con3)=O)C)C2)=O)CCCN(C(=O)COC)C1 N1(C(c2cnc(SC)s2)=O)CCC(NC(=O)COCC(N2CCCC2)C)C(C)C1 N1(C(C2C=CC(Nc3cc(SC)ncc3)C2)=O)CCC2(C1)CC2(F)F c1(C(=O)NC23CC(NC(c4c(C)cccc4Br)=O)(C2)C3)c(Cl)cc(C#N)cc1Cl c1(C(N2CCC(C#N)(NC(C)=O)C2)=O)ccc2c(CO)n[nH]c2c1.CO c1(C(C)NC(C(C)(C)Sc2nc(C)on2)=O)ccc(Br)cc1[N+](=O)[O-] C1(CCCNC(c2c(C)non2)=O)CN(C(=O)Cc2cccs2)CCO1 c1(C(=O)NCC2N(C(CCc3cc(C)cc(C)c3)=O)CC2)ncc([N+](=O)[O-])n1C c1(C(N2C(C)(CNC(Cn3nnc(C)n3)=O)CCC2)=O)cnc2c(c1)COCC2 N1(C(CC2N(C(c3c(CC)cno3)=O)CCC2(C)C)=O)CCC2(CC1)CC(O)C2 c1(CCOC)ccc(C(N2CC(OC)C(CNC(=O)C=CCN(C)C)C2)=O)cc1 Cc1nc(S)sc1CC(N1CCC(CO)(NC(=O)CC2(C)CC2)C1)=O N1(C(c2ccc(NC(c3c(CC)cccc3)=O)nc2)=O)CCC(C)(COC)CC1 C1(NC(C2N(C(=O)COC3CC3)CCN(C)C2)=O)CCn2ccnc2C1 c1(N2CC3C(CNC(C(C)C(C)(C)C)=O)C3C2)ncnc2scc(Br)c12 N1(C(CN=[N+]=[N-])=O)CCC2(CCN(C(c3cnnc(O)c3)=O)C2)C1 C1(N(C2C(C)CC2)C(=O)CN(C(c2ccsn2)=O)C2CC2)CCCCC1 Cc1ccc(O)c(C)c1NC(C1CCCCN1C(=O)C1=CCOCC1)=O C(CS(=O)(=O)CC(=O)N(C1CN(C(=O)C(C)(O)CC(C)C)CC1(C)C)C)OC N1(C(C(F)=CC)=O)CC(NC(=O)C(C)Sc2ccc(Cl)cc2)CC12CCC2 N1(C(C(C)O)=O)CC2CC(NC(c3cnn(-c4ccccn4)c3)=O)CC1C2 c1(OC)cnc(C(=O)NCC(C)NC(C2CC2c2nccn2C)=O)c(OC)n1 CC1C(NC(C2(C)CNC(=O)C2)=O)CCN1C(=O)Cc1nc(C2CC2)nn1C C1(C(=O)NCCN(C(c2c(SC)nc(O)nc2C)=O)C)CCC2CC1C2(C)C O=C(C1=C(F)CN(C(=O)CC2CCCC(O)C2)CC1)NCC1CN2CCC1CC2 c1(C(=O)NCC2N(C(C=C(C)C)=O)CCCC2(C)C)c([N+](=O)[O-])c(C)nn1C C(=O)(C1CC(=O)Nc2ncccc21)N(C)CCNC(C1(S(C)(=O)=O)CCCC1)=O C1(C)(C(N2C(C)C(NC(=O)CCC3CC3(Cl)Cl)CC2)=O)COC(=O)OC1 C(=O)(CC(C(F)(F)F)NC(=O)Cc1n[nH]c(C)n1)NC(COC)C(C)C C1(NC(C(c2cscn2)N(CC)CC)=O)CNCC(C)(C)C1 N1(C(C2(OC)CC2)=O)CCC2(CC1)CC2NC(=O)C(C(C)C)SC c1(CC(C)(C)NC(=O)Nc2nc(C)c(C)n2C)nnc2n1CCCC2 N1(C(c2[nH]cc(C)c2)=O)Cc2ccc(-c3ccc(N4CCOC4=O)cc3)cc2C1 CC1CN(C(=O)CCOCC2CC2)CC1(C)CNC(=O)CC1CCOCC1 C1(CNC(C(CCC)O)=O)CN(C(c2cc(Cl)ns2)=O)CC(C)(C)C1 C(=O)(C(C)=Cn1ccnn1)NC1CN(C(C2C(OCC)CC2)=O)CC1C N1(C(C23C(CN(C(=O)NC(c4ccccc4)C)C2)C3)=O)CC2CCCCC2C1 c1(NC(C)=O)ccc(N)c(C(=O)NC2CCCC2NC(c2cocc2C)=O)c1 C1(COC)(NC(c2ncn(C)c2C)=O)CCN(C(c2c(C)nsc2NC)=O)CC1 C1(F)(CNC(c2csc(-c3ccco3)n2)=O)CCN(C(C2(CF)CC2)=O)CC1 C1(C(=O)OC)CC12CCN(C(c1cc(C#N)n(C)c1C)C(=O)NCCC#N)CC2 C1(CC=C)(NC(=O)C(C)CC(N)=O)CCCN(C2CCCN(C)C2=O)C1 C(C)(C)(C(=O)N(C(C)CCNC(=O)C(n1ccc(C2CC2)n1)C)C)OC c1(NC)ccc(C(=O)N(CCCCCNC(=O)C(O)Cc2cnc[nH]2)C)cc1F C1(CC(=O)N(CCNC(C2(C)CC2(F)F)=O)C2CC2)(COC)CCOCC1 N1(C(C(=O)NCC=C)C2CC2(C)Br)CCN(C(=O)C(C)OC(C)=O)CC1 c1(C(=O)NCC2N(C)CCN(C(C(C)c3ccco3)=O)C2)cccn2ncnc12 C1(F)(CNC(C(C)Sc2nncn2C)=O)CCCN(C(C2CCCC(=O)CC2)=O)C1 N1(C(c2c(COC)scc2)=O)CC(NC(C2C3C4CCC(C4)C23)=O)CC2(CC2)C1 C(=O)(C(C)(C)CS(C)(=O)=O)NCC1(NC(C(CCOC)C)=O)CCOCC1 C1(NC(C2(SC)CCC2)=O)COC2(C1)CN(C(c1ccc(N(C)C)nc1)=O)C2 N1(C(CC=C(C)C)=O)CCC(Cn2cc(-c3ccc(CO)s3)nn2)CC1 c1(CC)cc(C(c2nnnn2CC(C)CCCO)NC)ccc1C CCS(=O)(=O)CCNC(=O)C=CCC(C)(C)NC(C1CCOC1C)=O Cc1[nH]nc(C(N2CCC(C(F)C(=O)NCc3ccnn3C(C)C)C2)=O)c1Cl C(=O)(C1=NOC2(CCC2)C1)C(COCCN)=O.CC1(C)C(N)CCS1(=O)=O c1(C(=O)NCC(C)NC(c2cc(C)[nH]n2)=O)cc(N)nc2ccncc12 C1(C)(C(N2CCCCC(NC(CCCC)=O)C2)=O)CCC(F)(F)CO1 C1(NC(CSCC=C)=O)(CC)CCN(C(c2ccc(CC#N)cc2OC)=O)CC1 C12(C(=O)NCC=CCNC(c3cc(C(C)(F)F)on3)=O)CCCCC(=O)N1CCC2 C1(C(=O)NCC2CC(NC(c3c(OC)csc3)=O)C2(C)C)CCOCC1(C)C c1(C(C)C)c(C(=O)NCC2CCCC2NC(C2(CO)COC2)=O)cnn1C Cc1cc2c(C(=O)NCCc3cc(Br)sc3Br)cccc2o1 c1(C(N(CCCC(=O)N(CC#C)C)C)=O)cc(Cl)ccc1C N#Cc1ccc(F)c(S(=O)(=O)N2CCC(F)CC2C(=O)O)c1 C1(C)(C(=O)NCc2cncc(CC)c2)CCN(C(C2CCCC(C)CC2)=O)CC1 CC1CCOC(C(=O)NC(CCF)C(=O)NCc2cc(C(C)C)n[nH]2)C1 CCC(CC(=O)N1CCOC(C)(C)C1)C(C)(C)C.C12(CCOCC1)C(=O)NO2 c1(CC)nc(C)n(C)c1C(=O)NC(C)C(CO)NC(=O)C=C(C)c1ccccc1 C1(C(N2CCC(N(C(=O)CNc3ccccn3)CC)C2)=O)CCC(C)CC1 C(c1ccc(O)cc1)=CC(N1CC(CNC(c2ccc(F)o2)=O)C1)=O C1(NC(c2cc(CC)[nH]n2)=O)CC(CC(=O)NCC(CC)N(C)C)C1(C)C c1(C(=O)NC2CCN(C(C3(OC)CC(CF)C3)=O)CC2)cccc(C2CC2)c1C C1(NC(Cc2ccc(SC)cc2)=O)CN(C(=O)CCCF)CCC1C C(=O)(CC(C)(C)NC(C1CC2CCC2C1)=O)NCCC=C N1(C(C(C)=CC=C)=O)CC=C(CC(=O)NC(C)C(C)SC)CC1 CC1(C)CN(C(C2(N(C)C)CC2)=O)CC(CNC(C2CC2C#N)=O)O1 c1(O)ccc(F)cc1F.N1(CCC(=O)C(=O)Cc2ccccc2)CCC(O)C1=O N1(C(C(CCC)OC)=O)CCCN(C(c2cc(C#N)no2)=O)C(CO)C1 C1(CCC)CN(C(C2CC2F)=O)CCN1C(C1CSC(C)=N1)=O C1(NC(C2N(C(C(CC=C)OC)=O)CC(O)C2)=O)CC2CCC(C1)O2 CC1CCC(NC(c2ncccc2C(F)F)=O)CN1C(C1CC12CCC2)=O c1(NC(CNC(=O)CC2CCCCC2(F)F)CC2CC2)ccc([N+](=O)[O-])cc1Cl C1(NC(C2C(C=C)CC2)=O)CC2CC(NC(=O)COc3cc(F)ccc3F)CC12 c1(C(=O)NCCN(C2CCCCC2)C(C(C)OCC=C)=O)cccc(F)c1N c1(CC)ccc(F)c(C(=O)CCCC2CN(C)CC2O)c1.C12C=CC(C1)C(=O)N2 N1(C(Cn2c(C)ncc2)=O)CC(NC(=O)CC2COC(C)(C)O2)CC12CCCC2 C(C)(CCCNC(c1nnn(CC(F)(F)F)n1)=O)NC(CC1(COC)CC1)=O Cc1c(C(=O)NCC(C)(C(C)C)NC(=O)CC2(O)CCOCC2)ccn1CCO N1(C(C(CC#C)(C)NC(c2sccc2CC)=O)=O)CCCC2CCCCC12 C#CC(C)(C)C(=O)N(C)CCN(C(=O)C(C)(F)F)C C1(CS(=O)(=O)NC)CCCN(C(C2CCC(NC(=O)OC(C)(C)C)CC2)=O)C1 N1(C(C(CCC)C)=O)CCC(NC(=O)C=Cc2cn(C)cn2)C(C)C1 c1(C(=O)NC(C)CNC(C2CCCN2C2CC2)=O)cc2c(c([N+](=O)[O-])c1)OCO2 N1(C(c2cnn(C3CC3)c2)=O)CCC2(CCCN2C(=O)CC2COCC2O)C1 N1(C(CC=CC)=O)CCCN(C(c2cccn(CC(C)(C)O)c2=O)=O)CC1CO N1(C(CCN(C)CC)=O)CCN(C(c2cc(C)c(Br)cn2)=O)C2CC12 CN1CCc2[nH]nc(C(=O)NCC(C3CCC3)NC(c3ccco3)=O)c2C1 C1(O)(CNC(CN(S(C)(=O)=O)C)=O)CCN(C(=O)CCCC2CCCO2)CC1 N1(C(=O)NCC2(CO)CCCCO2)CC2CN(C3CC3)CC2C1 CC1CCCCN1CC(=O)NCCN1CCN(C(=O)C=CCO)CC1 CN1CCC(C)(C(N2CC3CC3(NC(=O)C(=O)NCC(F)F)C2)=O)CC1 CC(C)(C(=O)NC1CN(C(c2cnccn2)=O)CC(F)(F)C1)C(F)(F)F OC1CC2(CCC2)C1C(c1nnnn1C1CCC1)NC(c1ccnc(F)c1)C1CC1 Cc1nc2cc(C(=O)N(C3CCN(C)C3)C3CC3)ccc2n(C)c1=O N1(C(C2(C)CC2C(F)(F)F)=O)CC2(CCOCC2)CC1CNC(=O)COC(F)F C1(CC)C(NC(=O)CCc2c(C)noc2Cl)CCN1C(=O)Cn1nc(C)oc1=O N1(CCN2C(c3ccc(O)c(F)c3)CCC2)CC(=O)c2ccccc2C1=O N1(C(c2c(I)ncn2C)C(=O)Nc2n(C)ccc2)CCS(=N)(=O)C2(CCC2)C1 C1(N(C(CN2C(C)CCC2C)=O)C)CCCN(C(C2(O)CCOCC2)=O)CC1 c1(C(N2C(c3n(C(C)C)ncc3)CCC2)=O)ccc2c(c1)OCC(=O)N2 CN(C)N(C(=O)Nc1ncc2c(n1)OC(=O)C2)C1CCS(=O)(=O)C1 c1(CNC(C=NOC)=O)cccc(CNC(=O)C(C)O)c1.c1(C)ccncc1 c1(C(N(C2CCN(C(CCCC)=O)C2)C)=O)cccc2c(C)csc12 c1(CNC(Cc2scc(C)c2)=O)nc(C)c(C(=O)NCCC2CC(=O)N(C)C2)o1 CC(C)(CCNC(=O)COc1ccsn1)NC(=O)CC1CC1C(F)(F)F C12(CCC(=O)NC(C3CC(NC(c4cc(Cl)c[nH]4)=O)C3)C)CCC(CC1)C2 c1(SC)cc(C(=O)NC(C)CN(C(=O)CN2CCC2C)C)ccc1N C1(OC)(OC)CC(C(=O)O)CN(C(OC(F)(F)F)=O)C1.C12CCCC(C1)N2 N1(C(CCOC)=O)CCCC2(C1)CN(C(c1ccc(-c3cccs3)[nH]1)=O)C2 N1(C(CC(CCC)(C)C)=O)CCCC(C2CCN(C(=O)C(C)(C)OC)C2)C1 c1(OC)ccnc(O)c1C(N1CC2CC2(CNC(C2CNC(=O)N2)=O)C1)=O C(CCCNC(=O)CCN(CCCO)C(C1CC1Cl)=O)N(C)C C(=O)(C(F)CC1CCCC1)NCCOCCNC(c1cnn(CCF)n1)=O c1(C(=O)NCC2(O)CCN(C(CSC)=O)C2)cc(F)cc2ccncc12 C(=O)(C1=C(C)OCCS1)N1CC(N2CCN(C(C3(COCC)CCC3)=O)CC2)C1 c1(C(=O)NCC2CC(NC(CCc3cc(C)no3)=O)C2)ccc2nc(O)sc2c1 C1(CNC(N(CC#C)C(C)C)=O)CCN(C(=O)CC=CCC)C1 CC(C)C(CCNC(=O)CC(C)n1ccnc1)NC(=O)CSCc1ccccc1 S(=O)(=O)(c1c[nH]ccc1=NCCCCC(=O)N(C)C)NCc1n(CC)ccn1 Cn1cnc2c(N3CCCC3CCN(C(=O)CC(C)(O)C3CC3)CC)nc(Cl)nc12 N1(CCC)CC(C(N2CCCC2CNC(=O)Cc2ccccc2F)=O)CCC1=O c1(C(N(C)CC2N(C(C3(CCCC)CCC3)=O)CCCC2)=O)cc(N)cc(O)n1 CC1CCc2[nH]nc(C(N3CCC(C)N(C(=O)CC=C(Cl)Cl)CC3)=O)c2C1 C1(C(=O)NCCCCCC=C)(CCOC)CCN(C(=O)CC2CCOC2C)CC1 C1(NC(c2nc(CC)sc2)=O)(CNC(=O)CC2(O)CCCCC2)CCCCC1C Cn1cc(S(C)(=N)=O)c(CN2CCC(O)(CN3CCOCC3)CC2)n1 C(C(CC(C)C)C(=O)NCC(N1CCCC1)C)NC(C1(CC=C)CC1)=O C(=O)(NNC(=O)C(=O)Nc1ccccn1)C1C(C)(C)C1 C(N=C(NC1CCOC1)N1CCC(C(O)C(F)(F)F)CC1)c1cnn(C)n1 C(CCC(N)=O)(C(=O)N(CC(C)NC(c1cccc2oncc12)=O)C)NC(C)=O C(=O)(CC(C)C(C)C(C)C)NCC1N(C(CC)=O)CCC1C N1(C(C2(C(=O)OCC)CCO2)=O)CCC2C(CCCN2C(=O)C(C)(F)CC)C1 c1(NCCCc2cn(C(C)CNC(=O)CC(C)F)nn2)ccccc1C#N c1(OC)ccc(F)c(CC(=O)NC2CCC(F)(CNC(=O)C(C)(C)C(N)=O)C2)c1 c1(C(=O)NC2CN(C(c3coc(Br)n3)=O)CC2F)ccc(C(F)F)c(F)c1 c1(NC(C)=O)cccc(C(N2CC(C(C)NC(=O)COCC3CCC3)C2)=O)n1 C1(NC(C(COC)C)=O)CN(C(=O)Cc2cccc(C(N)=O)c2)CC1NC(C)=O C(CCC=C)(C(=O)NC1CC(F)CN(C(=O)C(F)OC(F)(F)F)C1)NC(CC)=O C(=O)(CC1=Cc2ccccc2C1)N1CCC(C(CNC(C=CSC)=O)O)CC1 C1(CNC(C(=O)NCC)=O)COCCN1C(c1ccccc1F)=O N1(CC(=O)NC(C2(O)CCN(C(=O)C(O)C3CCCC3)C2)C)CCOCC1=O C1(C)(C(N(CC(C)N(C(=O)C(C)(F)F)C)C)=O)CCC2(CC1)CC2 C1(C2CC2)(NC(=O)CCc2cnc(O)[nH]2)CCN(C(=O)CC2CCSC2)C1 CC1(n2cc(CC(O)C(=O)NC)nn2)CCN(C(C2CC3(CCC3)CO2)=O)CC1 Cc1cnc(C(=O)NC2(C3CN(C(C4CCCC(C)(C)C4)=O)C3)CC2)cc1C#N c1(C(=O)NC2(CNC(c3c(C)nc(C(C)C)s3)=O)CC2)cc2n(c(=O)c1)CCS2 C1(C(N(C)Cc2onc(CC)n2)=O)CSCCN1C(=O)CCc1cc(C)on1 CC1CCN(C(=O)C(C#N)=CC2CC2)CCN1C(c1nncn1C1CC1)=O N1(C(c2c(SC)nn(C)c2)=O)CCC(NC(C2(C3CC3)CCC2)=O)C(C)C1 C=CCC(CC=C)C(=O)NCC1CCN(Cc2c[nH]c3ccccc23)CC1 C1(C(=O)NC(c2ncn(C)n2)C)CC12CCN(C(=O)C(C)CC1CC1)C2 C(CC(=O)N1CCC(F)C(O)C1)(C(F)(F)F)NC(c1cc(C)nn1C)=O CC1(C)CCCC(CC(=O)NC(c2ccccc2)CNC(c2ncccc2F)=O)O1 c1(OC)cc(-c2ccc(C3(C(=O)Nc4cncs4)CC3)cc2F)ccc1F CC1CN(C(c2ccc(C3CCCO3)[nH]2)=O)C(C)CN1C(=O)CCCCCC#N N1(C(C=CS(CC)(=O)=O)=O)C2CCC1C(C)C(NC(C1CC(=O)NC1(C)C)=O)C2 c1(C(N2CC3C(NC(=O)CC4=CCCC4)C3C2)=O)n[nH]c2ccc([N+](=O)[O-])cc12 C(=O)(C1Cc2ccccc21)N1CC(NC(CCC=C=C)=O)C(C)(C)CC1 N1(C(C(c2cccc(OC)c2)C)=O)CCC(CNC(=O)C=C(Cl)Cl)C12CC2 C(CCC(C)(C)C(=O)N1CC2(CCC2O)C1)NC(c1c(C)csn1)=O n1(CC(=O)NCC2N(C(C(C3CC3)OCC)=O)CCC2)c(C)cc(C)nc1=O C1(NC(CSCc2cccc(C)c2)=O)CCC(N=c2nc(C)nc3[nH][nH]cc2-3)CC1 N1(C(=O)OC(C)(C)C)CCCC2C1CCCN2C(=O)OCC1CC1c1cccs1 C1(SCC(N2C(CCCNC(CN(C3CCSC3)C)=O)CCC2)=O)CCS(=O)(=O)C1 Cc1cc(=NC(=O)c2cscc2-c2occc2N2CC3(CCC3)C2)[nH]o1 C1(NC(C(CC)Cl)=O)CC2(CCCN(C(=O)CCc3cncnc3)C2)C1 CC1=NS(=O)(=O)NC=C1C(=O)N1CC(NC(=O)CS(=O)(=O)C(C)(C)C)C(CO)C1 N1(C(c2ccc(F)c(C)c2N)=O)CCC(C2CCN(C(c3cnccn3)=O)C2)C1 c1(C(N(C(C)CNC(=O)Cn2nc(Cl)ccc2=O)C)=O)ccc(Cl)c(F)c1F c1(C(N2CC(C)C(NC(C3CC(C#N)C3)=O)CC2)=O)ccc2ncccc2c1F CCC(C(=O)NC(C)(C)CN(C(c1ncoc1C(C)C)=O)CC)OC1CCCC1 c1(OC)cc(NC(=O)NC2(C(F)(F)F)CC(NC(=O)C(O)C(C)C)C2)ccc1O N1(C(c2cc(COC)no2)=O)CCC(CN(C)C(c2cscc2C)=O)CC1 Cc1cnccc1C(C)C(=O)N(C(C)CN(C)C(c1snc(C)c1N)=O)C c1(CCNC(=NCC=C)NC2CCC(C(C)(C)C)CC2)c[nH]c2ccc(F)cc12 N1(C(C2CC(NC(=O)C=CCn3cncn3)C(O)C2)=O)CCN2CCCC2C1 c1(CNC(C2CN(C(=O)CCC3NC(=O)NC3=O)C2)C)cc(S(C)(=O)=O)co1 N1(CC)CCC(NC(N2CCOC(c3ccccc3)C2)=O)C1=O C12(NC(c3occ(C)c3C)=O)CCCN(C(c3cnc(C(F)F)s3)=O)CC1C2 C1(C(=O)OC)CCNCCC1NC(c1c(C)nn(C)c1-n1nccn1)=O c1(C(N2CCC(N(C)CC#N)C2)=O)ccc2nc(Cl)nn2c1 CC1(NC(=O)CCc2ncccn2)CCCCC1C(N1CCCC(O)C1)=O c1(OC)nc(OC)nc(NC(CC(C)C)C(=O)N2CCCC3(CC3)C2)n1 C(C(CCOC)NC(=O)C(C)(C)OC)NC(C(C)OC)=O CC1(C)CN(c2c(C3(C(=O)O)CC3)ccc(Cl)c2F)CC(CCO)O1 CC(C)(F)CC(=O)NC1CCN(C(=O)CSCCc2ccccc2)C1 C1(C(=O)NCCOC(CNC(c2ccc(OC)cc2)=O)(C)C)CC(C)CC(C)C1 c1(OC)ccc(C(N2CCC(NC(=O)C(=O)NC3CCNC3=O)CC2)=O)cc1OC C(CCCC(=O)NCC1CCN(C(=O)C(C)(O)C2CCC2)C1)OCCC=C CC(C)C1=NOC(C(=O)NC2COCC2C(=O)NCC2(Cl)CCC2)C1 c1(N2CCCC(COC)C2)cc(NCC2(C)CCCS2)nc(C(F)(F)F)n1 N1(C(COCCC=C)=O)CCC(C(C)(C)C)(CNC(c2cc(CC)c(C)s2)=O)C1 Nc1ccc(-c2cn(CCNC(=O)CCCC3CC3)nn2)cc1 N1(C(c2cc(C(C)C)n[nH]2)=O)CC(C)(C)C(NC(=O)Cn2cccn2)C(C)(C)C1 C1(C(N2CCC(C(N3CCC(F)(CO)C3)=O)C2)=O)(CO)CCCCC1 c1(C(=O)NCC(CNC(c2cc(CC)n(C)n2)=O)O)coc2ccc(OC)cc12 C1(C(N2CC3C(CNC(COc4ccc(C)cc4)=O)(C3)C2)=O)CC2(CCOCC2)C1 C1(CCNC(C(CC=C)C)=O)CCCC(C)(C)O1 C1(CNC(C(C)NC(C2CCCC2)=O)=O)CCCCCN1C(=O)CN(C)C.C1(S)CC1 CC1CCC(O)(Cc2ccc(Cn3ccnc3)cc2)C1 C12(C)CC(C1)NC2=O.C(=O)(CC(C)C)NC.C(C(=O)NC)N(CC)CC c1(C(=O)OC)cnc(NCC(C)NC(C2(O)CCOC2)=O)c([N+](=O)[O-])c1 c1(OC)cc(C(N2CCCC(N(CCO)C(c3ccco3)=O)C2)=O)sc1Cl C(CC(C)C(=O)NC1CCC(NC(=O)CC2CCC2NC(=O)COC)CC1)OC c1(C(N2CC(CC)N(C(c3cc(=N)[nH]c(Cl)n3)=O)CC2)=O)ccc2c(c1)CCO2 c1(C(C)=O)c(NC(C2CCCN(C(c3cc(C#N)c[nH]3)=O)C2)=O)cccc1F c1(C(=O)NC)cccc(NC(=O)C(C2(O)CN(C(c3nncs3)=O)C2)F)c1 C(=O)(C(C(C)(C)C)NC(C1CCC1)=O)NCC(C)N(C(CCCOC(C)C)=O)C c1(C(=O)NC(CN(c2ncnc(CC)c2F)C)C)ccc2nccnc2n1 C1(NC(c2nc(Cl)cs2)=O)CN(C(c2cc(F)c(F)cc2F)=O)CC12CCC2 Cc1c(Br)c(C(N2CC(NC(=O)CCSCC(N)=O)C(F)C2)=O)nn1C C1(CCNC(C2C3CCCOC23)=O)CCN(C(=O)C(O)CC2CCCCC2)CC1 C1(NC(CC2CC(C(=O)OC)C2)=O)CCC(=O)NC1CSc1cccc(Cl)c1 c1(OC)cncc(C(=O)N(CC(C)(C)C(=O)NCCN2CCCOC2=O)C)c1 C1(C(=O)O)(CNCCCCSC)CC2(CC2)C1 CC1C=C(C(=O)NC2CC(NC(=O)Cc3nc[nH]n3)C(O)C2)CC1 c1(CCN2CC(CC(=O)N(CC(N)=O)CC)C2)cccc(-c2cn(CC)nn2)c1 c1(C(=O)NC2C(CNC(c3csc(C)c3C)=O)CC2)cccc(OC(F)F)c1F c1(C(=O)NCC(CC)NC(=O)CCCC2CCCC2)cn(C(C)C)c(=O)nc1O c1(C(=O)OC)nn(C)cc1NC(=O)Nc1cccc(C(C(F)(F)F)OC)c1 N1(C(C23CC2C3)=O)CCCC(O)(CNCC=CC(F)F)C1 Cc1nccc(CCNC(C2(C)C=CCN2C(=O)CC2CCCN(C)C2)=O)n1 C12CC1=CC=C(Br)C=CC(C)CCN(C)C(=O)CCS2 C#CC1(C(N2CCCOC(CC)C2)=O)CCN(C(c2cnn(CCC)c2)=O)C1 CCCC(CCCNC(=O)CN1CCCC1CO)NC(c1ncccc1N)=O C1(O)(CNC(Cc2cnc(C)[nH]2)=O)CCN(C(C2CCCN2N=O)=O)CC1 C(=O)(CC(C)(C)N(C)C(C1CC12CCC2)=O)N(CC(C)C)CCO C(=O)(N=c1[nH]nc(-c2ccc(F)c(F)c2)s1)N1CCN(C(COC)C)CC1 c1(C(=O)NC(CSCC)C(=O)NC2CCCCO2)c[nH]c2cccc(C)c12 C1(C(C)NC(CCCC)=O)CCN(C(=O)COC(C)(C)C)CC1 C(=O)(C(CCOCCO)NC(=O)CCC1CCCN1C)NCC(=O)OC C(=O)(CS(=O)(=O)C(C)(C)C)N(CCN(C(C1(CC)CCC1)=O)C)C(C)C CC1CCCCCN1C(C1CC(C)N1C(=O)C1=C(Cl)CCC1)=O c1(NC(C(C(C)(C)C)c2ccccc2)=O)ccc(Cl)c(S(=O)(=O)N(C)C)c1 c1(C(=O)OC)cccc2c1C(=O)N(SCCNC(=O)CCC1CCOC1)C2=O c1(CC)cc(NC(C23CC2CN(C(C2CNC(=O)O2)=O)C3)=O)cc(F)c1 c1(C(=O)NCCN(C(c2nc(C)ncc2Cl)=O)CC)cc2ccc(Br)cc2o1 c1(C(=O)NCC(CC(C)C)NC(c2c(C)ncnc2O)=O)nc2cnccc2s1 N1(C(CC(CC)C2CC2)=O)CC=C(CNC(c2cc(OC)ncc2F)=O)CC1 c1(C(N2CCC(SC(CCC)CCO)CC2)=O)cccc2nnnn12 c1(C(N2CCCC(NC(CN(C)CC)=O)(COC)C2)=O)csc2c1CCC(C)C2 Cc1ccc(-c2csc(C=O)n2)[nH]1.C1(C(=O)N)CCC(NC(=O)OC(C)(C)C)C1 N1(C(CCCCC#N)=O)CCN(C(=O)CC2CC=CCC2)C2COCC12 C1(CCNC(C2C(=O)NCC2)=O)CN(C(c2cc(C3CC3)[nH]n2)=O)CCO1 CC(C)(C(=O)NC1CCC(F)(CNC(c2nnc3n2CCCC3)=O)C1)C(F)(F)F c1(CC)cccc2ccc(C(N3CC(NC(C4CC(=O)NC(=O)N4)=O)C3)=O)nc12 C#Cc1ccc2c(=NC(=O)c3ccc4c(c3)CNCCC4)nc[nH]n12 C(CCN=c1ccc(S(=O)(=O)NCC(O)CF)c[nH]1)N1CCS(=O)(=O)CC1 c1cc2c(C3CC3)[nH]nc2cc1-c1nc(C2CC2)nn1C1CCCCS(=O)(=O)C1 c1(C(N2C(C(C)NC(C3CCCCNC3=O)=O)CCC2)=O)[nH]nc([N+](=O)[O-])c1Cl c1(N2C(C(C)(C)SC)SCC2)[nH]c(=NCc2cnccc2Cl)nc2sccc12 CCCCC(CC)CC(=O)NC(C)(C)CCNC(=O)C(Cc1cccs1)N(C)C S(=O)(=O)(c1cnn2ccc(=NC(C)c3nccs3)[nH]c12)NC(c1c(C)nns1)C N1(C(C2C(C)(C(C)C)C2)=O)CC2(CCN(C(=O)CC)CC2)C1.c1(C=O)cccs1 c1(C(=O)NC(CCC)CNC(c2csc(O)n2)=O)c(F)ccc(F)c1F c1(CC(N2C(CNC(c3c(C)nn(C(C)C)c3)=O)CC2)=O)ccc([N+](=O)[O-])cc1 N1(C(Cn2nc(C)c(Cl)c2)=O)CCCCCC(NC(C2CCC(F)(F)C2)=O)C1 C(=O)(C(CNC(c1ccc(OC)cn1)=O)CC(C)C)N1CC(CC)C1 C1(NC(C(C)N(CCC)C(c2ccc(SC)o2)=O)=O)C2CCCCC12 C1(N(C(=O)Cn2ccnc2C)CC)CCCN(C(c2c(C)ncnc2C)=O)CC1 c1(C(N2CC3N(C(C=COCC)=O)C(CC3)C2)=O)n[nH]c2c1CC(F)(F)CC2 c1(C(N2CCCC(Cn3cc(-c4n(C)ccn4)nn3)C2)=O)ccnn(C)c1=O C1(NC(CCOCCOC)=O)CC(N=c2cc[nH]cc2C#N)C1(C)C c1(C(=O)NCCNC(C2Cn3c(C)ncc3CC2)=O)cc2c(o1)CCCNC2=O S(=O)(=O)(c1ccccc1C#N)N1CCC2(CN(C(c3cccc(C)c3)=O)C2)CC1 c1(CC(=O)NC2C(NC(CNC(CN(C)C)=O)=O)C2)csc(-c2nc[nH]n2)n1 c1(CC)cc(Br)ccc1C(=O)OC.C1(=O)C(C)N(CC)CC(C)N1 Cn1c(O)nc2cc(Br)c(NC(C3CCOC(C)(C)C3)=O)cc12 N12CCC(CC1c1ccccc1)C2=O.C(=O)(CC=C(Cl)Cl)NCC1C(C(C)(C)C)C1 c1(C(=O)NC(CC)CNC(C2CCCN(CC)C2)=O)ccc2c(c1)OCCO2 N1(C(c2cccc(N)c2F)=O)CCC2(CC=CCO2)C1 c1(SCCN(C(CC)CC)C)ccc(Cl)cc1 c1(C(=O)NC2CCCCC2NC(C2CC(CF)C2)=O)cc2sccc2s1 C1(C(=O)NCC(Cn2cc(CCN3CC4CC4C3)nn2)OC)C2COCC12 C1(O)(CCNC(=O)CCCC2CC2)CCCN(C(=O)C(=O)NCC(F)F)C1 c1(CNCc2c(OC)c(C)cc(C)c2)cc(=O)oc2cc3c(cc12)CCC3 c1(C(=O)NCC23C(CN(C(C=C(CC)CC)=O)C2)C3)ccc2cc[nH]c2c1 C1(CCN(C(=O)C(=O)NCCC(N)=O)C)CCN(C(C2CC2C(C)(F)F)=O)CC1 N1(C(C=CCCC)=O)CC(NC(c2ccc(NC(C)=O)s2)=O)CC(F)C1 c1(CN(C(=O)C(C)c2ccco2)CC)ccc(C(F)(F)F)cn1 C12(C(N3CCC(F)(CNC(=O)C(F)=C4CCC4)CC3)=O)CCCCCC1OCC2 C1(NC(c2ccc(COC)[nH]2)=O)CN(C(c2cc(OC)ns2)=O)CC1N=[N+]=[N-] c1(OC)cc(C(=O)NCC2(O)CN(C(c3cn(CCO)nn3)=O)C2)ccn1 c1(C(=O)NC(C(=O)NCCSC)Cc2cnc[nH]2)ccc(C)n1C N1(C(CCNC(COC)=O)=O)CCN(C(=O)CCc2ccccc2Br)C(C)C1 c1(OC)ccc(C(N2CC(F)CC2CNC(=O)CCC2CC(C)(C)CO2)=O)cc1 O=C1CC2(CCC(C(N3CCCC3C3(NC(c4n[nH]cc4F)=O)CC3)=O)CC2)CN1 c1(C(C)CN(C)C(=O)NC2CC(C(=O)OC(C)(C)C)C2)cccc(Br)c1 N1(C(N)=O)CCOC(CNCC2CCSC2)C1 c1(C(=O)NCC2(O)CN(C(CCN(CC)CC)=O)C2)cc2ccncc2o1 C1(SC)(Cn2cc(CC3C(NC(C4CCC(C)C4)=O)C3(C)C)nn2)CCOCC1 C(C(O)C(=O)N(CC(CC)NC(c1ccc(C)s1)=O)C)=CC C(=O)(CC(COC)COC)N1C(CC=C)(C(=O)NCC2CCCC2CC)CCC1 Cc1cc(Cl)c(C(N2CC(O)(CN(C)C(c3cnc(C(C)C)[nH]3)=O)C2)=O)s1 C#Cc1ccc(C(=O)NCC(CO)NC(C2CCCC(C)(C)C2)=O)nc1 c1(C(=O)NC2C=CCN(C(=O)C(O)(C3CC3)C3CC3)C2)cccn(C2CC2)c1=O CCC(C)CCCCC(=O)N1CCOCC1CN(C)C(C1(CC)CCOC1)=O c1(C(=O)NC(CN(C(c2cc(C)n(C3CC3)n2)=O)C)C)ccnc(F)c1F CN(C1CCOc2cc(F)ccc21)C(Cn1ncc(CNC(N)=O)c1)=O C1(C)(CNC(CC2(C)CC2)=O)CCC(NC(c2ccc(CCF)cc2)=O)C1 c1(CC)cnc2cccc(C(=O)Nc3cc(Br)cc4cc(C(=O)OC)[nH]c34)c2c1 Cn1cc2cccc(C(N3CC4CC4(C(=O)NCC4(CCO)CCC4)C3)=O)c2n1 C1(CNC(CN(C)C(N)=O)=O)CCCN(C(C2CCCCN2C(C)C)=O)C1.CC(N)=O C1(CC(=O)N(CC=C(C(N2CC(C)(OC)C2)=O)C)C2CC2)C=NN(C)C1=O N1(C(c2ccc(C)[nH]2)=O)CC2CCN(C(C3Cc4nccnc4C3)=O)CCC2C1 c1(C(=O)NC(C)CCCNC(c2cnc(C#N)s2)=O)cc2ncccc2cc1Cl CC(C)(C)CC(O)CC(=O)N1CC(CNC(c2nnc(C(N)=O)s2)=O)C2(CC2)C1 C(CCCCCC(=O)N(C(C)C(C)S(C)(=O)=O)C(C)(C)C)SC c1(C(N(CC(C)NC(C2CC2C2CCC2)=O)C)=O)ncnc2ccsc12 Cc1ccc(C#N)cc1NC(C1CCN(C(=O)C(F)CC(C)(C)C)CC1O)=O C(=O)(CC(=O)N(C(C)CNC(=O)CCCNC(c1ccco1)=O)C)OC O=C1CCC(C(N2CCC(CNC(=O)Cc3nnc(S)s3)CC2)=O)CN1 C(N=c1cc(C)[nH]c(=NCCOc2ccccc2)[nH]1)C1CCCC(OC)C1 C#Cc1ccccc1CC(=O)NC12CC(NCc3cccc(OC)c3OC)(C1)C2 C(C(O)C(=O)NCC(C(=O)NCc1nnc(C)s1)N(C)C)SC CCCCCCCC(=O)NC1CC(F)(CNC(C2COCC2C(=O)OC)=O)C1 c1(C2(C(=O)NCCCCCNC(C(C)CN(C)C)=O)CCC2)ccnc(Cl)c1 C1(NC(=O)CCC2CCCCO2)CC2CC(NC(C3CC(O)C3)=O)CC12 C1(NC(C(C2CN(C(=O)C3=CCCC3C)C2)OC)=O)CCN(C)CC1(C)C N1(C(c2cc(Cl)cc(Br)c2)=O)CC(c2ccccc2)C2COCCC12 C1(NC(CCc2n(C)ccc2)=O)CCC2(CC1)CN(C(C1CCCOC1)=O)C2 CC(C)CCCC(C)C(=O)N(CCCCNC(C1(F)CCCN(C)C1)=O)C c1(-c2ccc(C(N3C(CC)C(=O)N(CC)CC3)=O)cc2)cccc(F)c1C#N Cn1cccc(-c2ccc(NC3CCC(=CF)CC3)cn2)c1=O CCC(CC)CCCN(C)C(c1ccc(-c2cnc(N3CCCCC3)nc2)s1)=O C(=O)(CCCCO)NC1C(NC(c2cc(CC)[nH]n2)=O)C1 C1(C(=O)NCCCC(C)NC(=O)Cn2cccnc2=O)Cc2c[nH]cc2S1(=O)=O Cc1ncc(C(=O)NC2CCCC2(C)NC(c2nccnc2C)=O)c(C)n1 C1(NC(C2CC2(F)F)=O)CN(C(c2ncc[nH]2)=O)CCC12CCOCC2 c1(CC2C(C(=O)NC3CCCN(c4ncccn4)C3)C2)ccnc2c(Br)cccc12 Cc1cc(F)c(C(=O)NCC2(O)CCN(C(c3coc(Cl)n3)=O)C2)cc1F C12(CC=CCC1)C(=O)NC2.c1(N2CC(C(C)OCC)C2)cncc(Cl)n1 N1(C(c2c(CC)[nH]nc2Cl)=O)C2CCC(C(N3CCn4nccc4C3)=O)C1CC2 c1(C(CNC2(CC=C)CCC2)F)nnnn1C1CC1C(=O)OC C1(CNC(CN(CCOC)C)=O)CCN(Cc2ccc(Cl)o2)C1 c1(CC(N2CCC(CN(C)C(C3CC(O)CN3)=O)C2)=O)n[nH]c2ccccc12 N1(C(CC2(C)CC2)=O)CCNC(c2ccc(OC(F)(F)F)cc2)C1 c1(C(=O)NCC2CCN2C2CCCC2)cc2cc(Br)cn2cn1 C(=O)(C(CC(=C)C)NC(c1cc(CC)on1)=O)NC(C#C)CC1CC1 c1(OCC(=O)NCC2(NC(C3C(CCC)C3)=O)CCC2)ccccc1C c1(C(=O)NCCCC(CCC)NC(=O)C(C)NC=O)ccc2c(c1)nnn2C C(=O)(C1=NNC(=O)C1)N(C1CCN(C(C2CC(=O)N(CC(F)(F)F)C2)=O)C1)C c1(C(=O)NC(C)CCCCNC(=O)CN2CCCCC2=O)cc2n(n1)CCCC2 C1(C(N2CCC(NC(c3ccc(CC)[nH]3)=O)(CF)C2)=O)Cc2ccccc2C1 N1(C(C(N2C(CC)CCC2)=O)=O)CC(C)Oc2ccc(C(F)(F)F)cc21 C(=O)(C1=CN2CCN=C2C=C1)NC(C)=O.c12ccc(c(Cl)c1)C(=O)OCC=CC2 C1(NC(C(C=C)O)=O)C2CCN(C(c3cc4ccsc4s3)=O)CC12 C1(NC(C2CC(C)CN2C(C2CC(CF)C2)=O)=O)CCC(O)C(O)C1 N1(C(C(CNC(COCCCC)=O)CC2CC2)=O)C(CO)CCC12CCC2 Cc1cc2[nH]c(C(N3CC=CC(NC(=O)C(C)C4CCCC4)C3)=O)cc2s1 c1(C2(C(=O)NCCCNC(C3N(C(CC)=O)CSC3)=O)CCC2)ccccc1Br C=CCC(CCCCC)C(=O)N(C)CCN(C)C(c1ccn(CC)n1)=O c1(NC(Cc2c(C)nn(C3CCOCC3)c2C)=O)ccc2c(c1)N(C)C(=O)CO2 C1(CC)CCN(C(=O)CC2(C)CC2)C1CNC(c1nn(CC)nc1C)=O C1(CC)C(C(=O)NC2(CC)CC2)CCN1C(C1CC(CF)C1)=O C1(N(S(C)(=O)=O)C(C)C)CCN(C(=O)C(=O)NC2CN(C)CCO2)CC1 C1(C(=O)NCCOCCN(C)C(C2(O)CCSC2)=O)Cc2c[nH]cc2S1(=O)=O N1(C(c2c(CC)scc2)=O)CCN(C(c2ccc(C3CC3)cc2C)=O)CC1CC CC(C)(C)CC(O)CC(=O)NCC1CCCCN1C(=O)COC1CCOCC1 CC1CCN(C(C2CC3CC3C2)=O)C1CNC(C1CNC(=O)N1)=O C1(NC(CCCOC)=O)CC(CO)N(C(c2c[nH]nc2-c2cccc(O)c2)=O)C1 C(=O)(CCCCC(F)F)N1CCCC(NC(Cc2c(C)noc2C)=O)CC1 N1(C(c2c(CC)[nH]c(=N)s2)=O)CC(NC(C2CCCSC2)=O)CC12CCCCC2 N1(C(C(C)(C)C2CCCO2)=O)CC2(C(=O)NCc3cnn[nH]3)CC1CO2 N1(C(C(C2CCC2)OCC)=O)CCC(N(C)C(c2cc(CC)nn2CC)=O)CC1 CCCCC(C(N)=O)n1ccnc1-c1cccc(-c2ccccn2)n1 C1(CNC(Cn2cc[n+](C)c2)=O)CCCCN(C(c2ccc(O)nn2)=O)C1 N1(C(c2c(CC)[nH]nc2Cl)=O)CCN(C(=O)CC2CCC3CC23)CC2(CC2)C1 CC(C)C1=NOC(C(=O)N(C2CCN(C(=O)COCC(C)(C)C)CC2)C)C1 c1(N2CCC(CC(C)NC(=O)Cc3ncc[nH]3)CC2)nc(C#N)c(Cl)s1 c1(C(=O)NCC(C(=O)NC(c2nc(CC)on2)C)O)cc(C)c(N)cn1 C1(CNC(C2(CSC)CCC2)=O)CCC(N(C)C(C2CCC3CC23)=O)CC1 c1(C(=O)NC(CC=C)CNC(=O)CC2CCOC2)ccc(CS(C)(=O)=O)cc1 N1(C(C(C=C)(C)O)=O)CC(NC(C2(n3cc(Cl)cn3)CC2)=O)C(C)(C)C1 C#CC1(CNC(=O)CCOCCNC(C23CCCCC2C3)=O)CCOCC1 O=C(CC(F)(F)c1ccccc1)NCC1CCN(C(C2(c3cc[nH]n3)CC2)=O)C1 N1(C(C(=O)NC2(CCNC(CCC=CC)=O)CC2)C)CCCC(O)C1 c1(C(N=S(CCOCCOC)C)=O)ccnc(C2CC2)c1 c1(C(=O)NC2CC(NC(c3cccnc3)=O)C23CCC3)ncn2c1COCC2 O=C(C(O)CC(F)(F)F)N1CCC(CO)C(NC(C2(O)COC2)=O)C1 N1(C(C(OC)OC)=O)CC2CC(NC(=O)Cc3c(CC)noc3CN)C1C2 N1(C(c2sccc2F)=O)CCC(O)CC1.O=C1CC2(CC2)N1 N1(C(C2C(NC(CCc3c(C)cccc3)=O)C2)=O)CC2(C1)CC1(CCC1)C2 C(C)(C)(C(=O)NCC(C)(C)NC(=O)CCC1OCCO1)OC(C1CCCCC1)C c1(CC)nc(SC)ncc1CNC(=O)C(C)n1cc(-c2ccc(C)cc2N)nn1 CCCC(CCC)C(=O)NC12CC(C1)N(C(=O)CC(C(F)F)N1CCOCC1)C2 c1(C(=O)NC2CC(NC(c3c(C)c[nH]c3)=O)CC2O)noc2c1CCCC2 c1(NC(c2c(O)ccc(CCC)c2)=O)ccc(S(C)=O)c(F)c1 c1(C(CC)NCC2CCN(C)C2C2CCCCC2)ccc(C)c(Cl)c1 c1(C(N2CC3CCC(C2)N3C(=O)CCc2cnc(O)[nH]2)=O)ncc([N+](=O)[O-])cc1Br O=C(C1=CCCOC1)NCC1(F)CC(NC(C2C(C3CC3)C2(F)F)=O)C1 C1(C(=O)NCCCOCCCC)(NC(=O)COC2CCC2)CC(F)C1 c1(COC)nc2ccccn2c1C(=O)NCC(C)N(C)C(C1CC2CCC1C2)=O Cc1cc(NC(=O)CN2CCN(C(C3(C)CCCCO3)=O)CC2)cc(C)c1O N1(C(C2(CCCCCC3CC3)CC2)=O)CCC(F)(c2cn(C3CCCC3)nn2)C1 C12(CO)CC1CN(C(=O)Cc1cnc[nH]1)C2.C12(CCC1)CC(=O)N2 C1(C(=O)NCc2ccc(Cl)cn2)CC2(CCC2)CO1.C12CC(C1)C(=O)N2C CC(C)C(C)(CNC(=O)CNC(c1ccoc1)=O)NC(C1CCC(F)C1)=O CCCCC(C(=O)NCc1cccn1CC)NC(=O)C(C)N(C)C.CC C(=O)(C#CC(C)(C)C)NC(C(N1CC(OC)C(O)C1)=O)CC1CCC1 N1(c2nc(C)c(F)cn2)CC2(CCN(C(c3cc(F)c(Cl)c(Br)c3)=O)CC2)C1 N#Cc1cccc2[nH]c(CNC(=O)C(F)(F)C3CCOCC3)nc12 N1(C(C(C(C)OC)O)=O)CC(NC(C2(O)CCOCC2)=O)CC1(C)C N#Cc1c(C(=O)O)cnn1-c1ccccc1.n12cc(nn1)CNC(=O)C2 C1(NC(c2c(C)[nH]cc2)=O)C(C)CCN(C(C2CCCCN2C)=O)C1C C1(COC(C2CC23CC3)=O)CCCCCC1O Cc1cc(C(N2CCC(N(C(=O)C(C(C)O)N(C)C)CCO)CC2)=O)ccc1O c1(C(=O)NC2CC(CNC(c3c(C)con3)=O)C2(C)C)ncc(C)cc1F Cn1nccc1C(O)C(=O)NCC(C)(C)NC(C1COC(=O)C1)=O CCC(C(=O)N1CCC(OCCNC(=O)CC2CC2(Cl)Cl)CC1)C(C)C c1(C(=O)NC2(C(N(CCC#C)CCO)=O)CCCCC2)ncc(C#C)cc1C c1(OC)ccc(CC(=O)N(C)CCNC(=O)CC2CC3CCC2C3)c(Cl)c1 CC1(C)CCCOC1C(=O)NC1(C2CN(C(C3SC4C=CC3CC4)=O)C2)CC1 N1(C(C(=O)NCCC)C)CCN(C(=O)Nc2cccc(SC)c2)CC1 C1(CNC(C(CC2CC2)OC)=O)CC(O)CN1C(=O)CCC1CCOCC1 C1(NC(C(CC)COC)=O)CCC2CC1CN2C(c1cnc2n1CCCC2)=O C1(C(C)C)CN(C(=O)CN2CCCOC2=O)CCC1NC(c1cnns1)=O c1(CNC(=O)NCC(CNC(=O)OC(C)(C)C)OC)ccc(Br)c(F)c1F C=C1COCCN(C(c2cc(CNC(c3c[nH]cc3C)=O)on2)=O)C1 CC1(C)CCCOC1C(=O)NC1CC(NC(=O)Cc2ccc(F)c(F)c2)CC1O CCC(CC)CC(=O)NC12CCCC(NC(=O)C(C3CCCOC3)OCC)(C1)C2 C(C(CNC(c1scc(C)c1C)=O)C(F)(F)F)NC(Cn1ccc(C)n1)=O CC(C)(C(=O)N1CC2CN(C(C3(n4cnnn4)CC3)=O)CC12)C(F)F Cc1cc(C(=O)NC(C)CN(C)C(C2CC(F)C(=O)N2)=O)ncc1Br N1(C(Cc2n(C)cnc2)=O)CCC(C(=O)NCCCCC2CC2)C(C)(C)C1 C(=O)(C1c2c[nH]nc2CN1C(c1n(C)cc(Br)c1)=O)OC(C)(C)C C1(CNC(C(F)OC)=O)CCN(C(C2CN(C(C)C)C2)=O)C12CC2 N1C(NC2CCCC2)=NCc2nc(cs2)C1.c1(C(F)F)cc(C2OCCO2)no1 c1(CC)cccc(C)c1NC(=O)C(c1cn(C)nn1)NC(=O)CC1CC(=O)NC1=O C(c1ccnn1C)=CC(=O)NC1(C2N(C(C3ON=C(C)C3)=O)CCC2)CC1 C1(C(NOCC)=O)(CNC(c2ccnc(CC)c2)=O)CC12CCC2 CC(C)(C)CCCC(=O)NC1CN(C(c2cc(C3(C)CC3)on2)=O)CCC1CO Cc1cc(C(=O)N(CC(C)(C)CNC(C2CC3(CCCO3)C2)=O)C)ccc1Cl C(CC(C(=O)NCCOC(C)=O)NC(=O)Cc1cn(C)cn1)OCC c1(CCC)cc(C(=O)NC2CCCCC2CNC(=O)C(C)=C2CCC2)nn1C c1(C(N2CCCC(C(CNC(CC(=C)C)=O)(C)O)C2)=O)ccc(C(N)=O)c(Cl)c1 c1(C(N2C(C)(C(=O)NCCCC3(C)CC3)C=CC2)=O)cc2ccccn2n1 C1(C(N2CC(C)C(NC(c3ncn(C(C)(C)C)n3)=O)C2)=O)CCc2nn[nH]c2C1 C1(NC(C2(C#N)CC23CCC3)=O)CC2CCC1CC2NC(c1ccc(Cl)s1)=O CCC(CCCC(=O)NCC(c1cnn(C)c1)C)NC(=O)CN(C)CC c1(OC)ccc(C)c(OC)c1C(N1CCOC(CNC(C2CC2OC)=O)C1)=O c1(C(=O)NC(CC(C)C)CNC(=O)Cn2cc(Cl)cn2)ccc2cnccc2c1 c1(CC(=O)NCCN2CC=CC2)cc(C(F)(F)F)cc2ncnn12 C1(C)(OC(C)CNC(=O)NCC2CCOC2(C)C)CCC(C)(C)CC1 n1(CC(=O)NC(C2(O)CCN(C(c3nncs3)=O)CC2)C)ccc(=O)n(C)c1=O c1(C(=O)NCC(C(C)C)NC(c2cc(OC)c(F)cc2)=O)cccc2cnnn12 c1(C(C)=O)ccc(NC(c2nc(NC(C3CC3C3CC3)=O)cn2C)=O)nc1 c1(OC)cc(CNC2CCC(CC(N3CCCC(O)C3C)=O)CC2)cc(Cl)c1 C(C)(CCC(=O)NC(C)CC(C)NC(c1cnnn1-c1cccc(F)c1)=O)SC c1(OCCCNC(C(=O)OC)C)cccnc1Oc1cccc(Cl)c1 C(=O)(C1=NOC(C)(C)C1)N1CC(CNC(c2c(C)n[nH]c2)=O)C2C1C2 Cc1ccsc1C(=O)NCC1CC(NC(c2cscc2C)=O)C1 c1(C2(NCC3N(C(C4C(=O)OCC4)=O)C(=O)CC3)CC2)ccc(F)cc1F C1(NC(c2ccn(C(OC)OC)n2)=O)CCSC12CN(C(=O)C=C(C)Cl)C2 C1(CC)CCOC1C(=O)NCCC=CC(N1CCCC1CN(C)C)=O Cc1nc(CCC(=O)NCCC2(O)CN(C(=O)CCc3ccoc3)C2)cs1 N1(C(C(C)(C)CF)=O)CCC2CN(C(=O)CNC(=O)C3CC3)CCC2C1 c1(C(=O)NCC(CC)NC(=O)CC2CN3CCN2CC3)cccc2nc(O)[nH]c12 N1(C(Cc2ccc(C)o2)=O)CC2CC1CCC2NC(c1ccc(N(C)C)nc1)=O N1(C(c2c(COC)noc2)=O)CCC(NC(=O)Cc2cc(F)ccc2O)CC1C CN1CCNC(=O)C12CCCN(C(C1CC1c1ccc(Br)s1)=O)C2 C(=O)(C(COC)CC(C)C)NC(CC=CC)C(=O)NCc1ncc(CO)o1 c1(C(=O)NC2CCC(NC(C(CC)C)=O)CC2)nccc(C)c1Br Cc1nsc(C(=O)NC2CCOC2C(=O)NCCc2ccnn2C)c1N c1(C(=O)NC23CC2CN(C(c2ccoc2)=O)C3)cc2c(s1)CCCNC2=O CC1(C)CN(Cc2c(F)cccc2Cl)CC(C(C)(C(=O)O)c2ccccc2)O1 C=CC(C)(CC)C(=O)N1CCCCC(C(=O)NCc2cc(C)on2)C1 C(C)(CCC(=O)N1CC(C)(CCC(=O)N(C)Cc2cnccn2)C1)OC c1(C(=O)O)ccc(-c2cccc(Cn3cccn3)c2)nc1 C(=O)(C(C)S(N)(=O)=O)N(CCCNC(C(c1ccc(F)c(Cl)c1)C)=O)C CC1(C)C2CC(C(=O)NCCOC3CN(c4nc(-c5ccccc5)ns4)C3)CC12 c1(C(N2CCC(F)(CNC(=O)CCc3ccoc3)C2)=O)cc(O)cc(Cl)c1 C(=O)(C(C)CC(F)F)NC(CNC(c1c(C)nn(C2CC2)c1)=O)C CCC(O)C(C)C(=O)Nc1[nH]c(-c2cnn(C(F)F)c2)nc1C Cc1cc(C(=O)N(CC(C)O)CCNC(c2ccsn2)=O)c(C)cc1Cl c1(NC(C2(C)CCN(Cc3cncc(OC)n3)C2)=O)ccc(Cl)cc1F CC1CN(C(=O)CN2CCCCS2(=O)=O)CC(C)C1NC(c1cnc(=N)[nH]c1)=O N1(C(c2cccc(C)c2C#N)=O)CCN(C(c2ccc(F)cc2)=O)C2COCC12 C[S+](C)CCC(O)C(=O)NC(c1ccccc1)CNC(C1CSC1)=O N1(C(C(C)OCC=C)=O)CCC2(CC1)CC(NC(C1CNC(=O)S1)=O)C2 C(C(C)(C)CNC(=O)CCc1ccn(C)c1)N(C(C(C)OCC1CCCO1)=O)C N1(CCC(N2CCCC(CSC)C2)=O)C(=O)C2CCCCC2C1=O c1(OC)ncc(C)cc1NC(C1(NC(C2CC(=O)CC(=O)N2)=O)CCC1)=O C#CCCC(=O)NCC1(C(=O)NCC2(F)CC2c2ccccc2)CC1 N1(CC(C)C)CCC(C(=O)NCC(C)(C)OC(c2nc(C)on2)C)CC1 CC1CC(c2cccc(F)c2)N(C(c2ccnn2CCF)=O)C1 c1(C(N2C(C(N3CCN(C(C)C)CC3)=O)CSCC2)=O)cnc2ccccn12 c1(C(=O)NC(C(C)NC(C2CC2(C)C)=O)(C)C)cc(O)c2ccsc2c1 c1(C(C2CC2)NC(=O)Nc2cccc(N3CCCNC3=O)c2)cc(Br)ccc1Cl C1(NC(=O)Nc2cc(S(C)(=O)=O)oc2)CN2CCC1c1ccccc12 C1(F)(CNC(C2ON=C(C)C2)=O)COCCN(C(c2ccc(Br)c(N)c2)=O)C1 C1(NC(CCCN(C)C)=O)CC2(CCCN(C(C3CCOC3(C)C)=O)C2)C1 C=C(Cl)CC(C(=O)N(C)CCN(C)CCO)NC(c1cc(CC)[nH]n1)=O c1(OC)cc(C(n2c(C)cc(CO)c2C)C)cc(OC)c1OC C1(C(=O)NCC2(O)CC(NC(C3CCN(C)CC3)=O)C2)CC(C)(C)OC1=O CC#CCCCC(=O)N1CC(N(C)C(c2cccc(Cn3cccn3)c2)=O)C1 CC1CCOC1C(=O)NC1CC(CCNC(=O)C(F)=CCCF)C1 c1(OC(C(=O)OC(C2(C)CC(=C)C2)C)C)ccc(F)c(F)c1 CCC(C)C(O)C(C)C(=O)N(C)CC1COCCN1C(=O)C(N1CCSCC1)C N1(C(CCCOCCC)=O)CCN(C(=O)C(CC)SC)C(C(F)F)C1 C1(CCCNC(C2(CC#C)CCCO2)=O)CN(C(=O)Cc2cscn2)CCO1 CC1CN(C(=NCC2CCC(C)C2)NCc2ccnn2C)c2ccccc21 N1(C(C=CCCCCC)=O)CC(NC(c2ccc(C(N)=O)c(Cl)c2)=O)CC(F)C1 Cc1c(C(N2CC(NC(c3cc(F)n[nH]3)=O)C3(CC3)C2)=O)cccc1S(N)(=O)=O Cc1cnc(C)nc1.c1(-c2n(CCC)ccn2)cc(-c2nccn2C)nn1C C1(NC(CCCC(=O)NC)=O)CN(C(C2CC(C)CO2)=O)C2CCCCC12 CC(CC(C)(F)F)C(=O)NC(C1CCN(C(=O)CC=Cc2ccccc2)CC1)C C12(NC(C3CC(=C)C3)=O)CN(C(=O)Cc3ccc(F)cc3F)CC1CS(=O)(=O)C2 N1(C(C(C)OC)=O)CCC2(CC1)COC(CNC(=O)CSCc1csc(=N)[nH]1)C2 C1(NC(c2c(C)cco2)=O)CC2(CCN(C(c3scnc3C(C)C)=O)C2)C1 c1(CC(N2CC(NC(c3ccc(CCC)s3)=O)C2)=O)c(C)nc(O)nc1O N1(Cc2c(C(=O)NCc3ccccc3)scn2)CCCCCC1C1CCNCC1 C#CCCCC(=O)NCC1CC(CNC(c2cnc(N(C)C)o2)=O)CO1 C1(NC(C2C(C)OCC2)=O)CCC2(CC1)CN(C(=O)C=Cc1cnc[nH]1)CCO2 C1(CNC(CN(CC)CC)=O)CN(C(=O)CCNC(c2ccsc2)=O)CCO1 c1(C(N(CCCCNC(C(C)n2ccnc2)=O)C)=O)cc2c(O)ncnc2cn1 c1(OC)cccc(CCC(=O)NCC(C)N(C(=O)CC2CC(=O)NC2=O)CC)c1 N1(CC)CCOCC1CC(=O)NCC(=C1CN(C(=O)C(C)c2cccs2)C1)F c1(C(N2CCC(C(C)NC(c3c(CC)cccc3)=O)C2)=O)cc(C)ncc1C N1(C(C2(NC(C3CCCCC3F)=O)CC2)=O)C2CCCC1CC2 N1(C(c2ccc(C)c(F)c2)=O)CC2CCN(C(C3CC=CC3)=O)CC12 c1(SCC)ccccc1C(N1CCC(C(C)NC(c2ccc(C#N)s2)=O)C1)=O C1(F)(C(=O)NC2CCCN(c3cnccn3)CC2)CNCC1C1CC1 N1(C(C(CSC)OC)=O)C2CCCC1CN(C(c1nocc1C(C)C)=O)C2 C12(C(N3CC(c4c(C)nn[nH]4)C3)=O)CCN(C(C3(O)CCC(C)CC3)=O)CCC1C2 C1(C)(NC(CN(C)Cc2ccccc2)=O)CC(C(=O)NC2(C(C)(C)C)CCC2)C1 Cc1ccc(CCC(N2CC(CCNC(=O)CN3CCC3)C(C)C2)=O)cn1 c1(NC2CC(C)N(C(=O)Cc3cnco3)C2)ncnc2cccc(F)c12 Cc1onc(CC(N2CCCCC2CNC(=O)C(O)C2CC2)=O)c1C#N CN1CCN(C2=NCC(C(F)F)N2)CC1=O c1(C(N2C(C3(O)CN(C(C(CC=C)(F)F)=O)C3)CCC2)=O)ncn2ccccc12 Cc1oc(C#N)cc1C(=O)NCC1CCC(C(N2CC(c3ncc[nH]3)C2)=O)CC1 C1(C(N2CCN(C(c3c(C)cc(Br)s3)=O)CC2)=O)CC(C2CC2)=NO1 C1(CN(C2CCN(C(=O)OC(C)(C)C)CC2)C)CCC(C2CC2)C1 C12(C(N3CC(C)(C(=O)NCC4(CCCO)CC4)C3)=O)CCCC(CO1)C2 c1(C(=O)OC)c(N)sc2c1CCN(C(c1ccn(-c3cc(C)cc(Br)c3)n1)=O)C2 c1(C(=O)NC(CC(C)NC(c2ccc(C)nn2)=O)C)ccc(F)c2ccccc12 N1(C(C(C)OCCOC)=O)CC2CC1C2NC(c1c(OC)cccc1)=O N1(C(CCCOC(C)C)=O)CC2(CC(C(=O)N(c3ccncc3)C)CO2)C1 N1(C(C(C=C)(C)O)=O)CCC2(CCCCC2NC(c2csc(C3CC3)n2)=O)CC1 C=CCC(CNC(=O)CCCC1CC1C)C(=O)N1CC(c2nn[nH]n2)C1 c1(C(=O)OC)cnc(CCN2CCCCC2)nc1.C1(=O)CCCN(C)CCN1C N1(C(C(COC)C)=O)CC(NC(c2csc(C)c2)=O)CC2(CCC2)C1 CC1(C)C2CCC(C(N3CCNC(CNc4ncc(I)cn4)C3)=O)C1C2 c1(OC)ccc(CNC2CN(C(=O)C(c3cccc(C)c3)=O)C2)cc1Br c1(C(=O)NCC2(CC)CCOCC2)cc(F)cc(I)c1 N1(C(C(=O)OCC)=O)CCn2c(nc(C(N3CC4C(C3)C4(C)C)=O)c2Cl)C1 C1(C(=O)NCc2cn(C(c3cccc(C)c3)C)nn2)CCC12CCOCC2 C(CC(=O)N1CCC(C(N2CCC(c3ncco3)C2)=O)O1)OC CS(=O)(=O)c1cccc(=NCc2cc(C(F)(F)F)cc(Br)c2)[nH]1 N1(C(COC2CN(C(C(C)C3CCCC3)=O)C2)=O)CCCCC1C(C)(C)O n1(CCOC)nnnc1C(c1cc(OC)ns1)NCC1CC1c1nc(C)cs1 C1(O)(CNC(Cc2nc(C)sc2)=O)CCCN(C(=O)Cc2ccc(Cl)nc2C)C1 c1(C(N(CC(F)(F)F)CCCNC(Cc2cn(C)nn2)=O)=O)cc(F)ccc1O c1(-c2ncn(C)n2)ccc(C(=O)OC(Cc2ccccc2Cl)C(N)=O)cc1 C=C1COc2c(C(=O)NCC(C)(C)CN(C)C(C3CCCCS3)=O)cnn2C1 c1(C(N(C)CC2CCCN(C(C(CC)C)=O)C2)=O)cccc2nccn12 c1(CC)cc(C(=O)NCc2ncccc2C(=O)N(C)Cc2ccncn2)nn1C c1(OC)cc(F)c(C(N2CC(N(C(=O)C3=CCC3)C)C3(CC3)C2)=O)cc1N c1(C(=O)NCC2CCCCCN2C(c2n[nH]cc2F)=O)nccc2ncncc12 N1(C(C(CC)NC)=O)C2CCCC1CC(NC(c1ccc(OC)c(F)c1F)=O)C2 C1(C(N2CC(C)(CNC(C=CC=CCC)=O)OCC2)=O)CCn2nnnc2C1 C1(NCc2cncc(N(C)C)c2)CCC=CCCC1 c1(OC)ccccc1CN1CCOC(CNC(c2cn(C(C)C)nc2C)=O)C1 N1(CC)CCOC(C(=O)N(C(C)C(=O)NCC(c2nccc(O)n2)C)CC)C1 C1(C(=O)NC2CC(NC(CNS(NC)(=O)=O)=O)C2)CCc2[nH]nc(C)c2C1 CCC(CC)(CN=c1[nH]c2cc(Cl)cc(Cl)c2o1)NC(c1cnn2c1CCC2)=O c1(C(N2CCC3CCN(C(CCCC#C)=O)CC32)=O)ncc2ccccc2c1O C1(C(N2CC3(C2)CN(C(C2CC2c2ccco2)=O)C3)=O)CN2CCCN1CC2 c1(C(=O)NCC(C2CC2)NC(c2c(C)cc(N)cc2)=O)c(C)cc(F)cc1C N1(C(C(c2cncnc2)C)=O)CCC2CC(NC(C3(F)CCC3)=O)CCC2C1 c1(OCC)cccc(F)c1Cl.C(CCCC(=O)N(C)CCOCCCN(C)CC)O C#CC1(O)CC(C(=O)NC(CC2CCC2)C(=O)NCc2cccc(Cl)c2)C1 N1(C(c2ncoc2C2CC2)=O)CCN(C(c2cc(F)cc(F)c2F)=O)CC(O)C1 Cc1ccc(C(=O)NCC(C(C)(C)C)NC(c2ccoc2)=O)c(N=[N+]=[N-])c1 c1(OC)ncccc1CC(=O)NC1(CCNC(=O)CCC2CCCO2)CCC1 CCCCCC(C(=O)N1CC2(CCN2C(=O)C2=CCCSC2)C1)C(C)C C1(CNC(Cn2c(C)cnc2)=O)CC2(CC2)CN1C(=O)COCc1cccnc1 C(=O)(C(O)CC(F)(F)F)N1CCC(CC(=O)NC(COC)CCO)CC1 c1(CNCC2CCC(C(=O)NC(CC)C)C2)cccc(Br)c1Cl C(CCCCC(=O)N1CC(N)C1)n1cc(C)nn1.c1(OC)ccccc1C(=O)OC N1(C(CCOCCC(C)C)=O)CCC2(CC(NC(C3(C(F)(F)F)CC3)=O)CO2)C1 c1(CCC(=O)NCC(CC)(CC)NC(C2SCCCS2)=O)c(Cl)cccc1Cl Cc1cc(C(=O)NC(C)CCCNC(=O)CC2CSCCS2)c2ncccc2c1 Cc1nc2ccccn2c1NC(C1CC1C(=O)Nc1cc(F)c(F)cc1I)=O N1(C(C=Cc2cn(C)nc2)=O)CCC2CCCC12C(N1CC(C2=NOCC2)C1)=O C(=O)(CN(C)N1CCC(C)(c2ccccc2F)CC1)NC(C)C N1(C(C(C)(C)OC)=O)CCC2(CCCN(C(C3CC3c3nc[nH]n3)=O)C2)CC1 C(N=c1[nH]c2c(c(=NCC3(CO)CCC3)[nH]1)COC2)c1c(C(F)(F)F)cccc1 c1(C(=O)NC(C(C)C)CNC(=O)Cc2ccc(Cl)s2)cc(O)n(C)n1 c1(C(=O)NCC2C(C)CCN(C(CSC)=O)C2)cc(O)nc2c1c(C)nn2C c1(C(N2CC(=C(CNC(c3cnc(C4CC4)nc3)=O)F)C2)=O)nnn2c1CCC2 C1(C)(c2cn(-c3c(C)n(C)nc3)nn2)COCCN1C(c1ccc(F)c(Br)c1)=O c1(OCCO)c([N+](=O)[O-])ccc(CNC2CCCCC2)c1O C(=O)(C(CC)C(C)(C)CC)N1CC(NC(C(CC=C)(C)C)=O)C(C2CC2)C1 c1(C(N(C2CCN(C(C3CC3C(=O)OC)=O)C2)CCC)=O)cc(C(N)=O)c[nH]1 CC1CC(C(=O)NC2CC(N3CCOCC3)C2(C)C)CCN1C C(=O)(C1=NN(C)C(=O)CC1)N1CC(C)C(CNc2nccc(C#N)n2)C1 N1(C(C(CCC)OC)=O)CCN(C(=O)CCSC)C(c2cc(F)ccc2OC)C1 C1(=CC(=O)NCC2CN(C(=O)C=C3CCSCC3)CC2O)CN2CCC1CC2 n1(C(C)C)ccc2c(N3CCCCC(C(=O)OCC4CC4)C3)nc(Cl)nc12 c1(NC(=O)CN2CCCC2CCNC(c2ccsc2)=O)ccccc1Cl C(=O)(C1CCCc2nn(C)cc21)NCC1CC(NC(c2c[nH]c(=NC)s2)=O)C1 C1(CNC(=O)C=Cc2nccs2)C2CC1N(C(=O)Cc1cccnc1)C2 c1(C(=O)NC2CN(C(C3N(C)C(=O)CC3)=O)C(C)(C)C2)cc(F)cc(Cl)c1O c1(CC(N2CCC(NC(Cn3nc(C)oc3=O)=O)(CF)C2)=O)cccc(F)c1Cl N1(C(C2CC3(C2)CC3(F)F)=O)CCC(F)(C(=O)NC2CCC(O)CC2)CC1 C12(C(=O)NCC(CNC(c3c(C)coc3C3CC3)=O)(C)O)CCC(CF)(C1)OC2 C1(NC(CSCc2cn(CC(C)O)nn2)=O)(COCCO)CC(C)(C)C1 c1(C(N2CC(NC(=O)CCN3CCCC3)C(C(F)F)C2)=O)cnc2ccccn12 c1(C(=O)NCC2(C)OCCN(C(C(CC)F)=O)C2)nn(CC)cc1[N+](=O)[O-] Cc1nccs1.C(C(C)C(=O)N(C1CNC1)C)C(=O)C(F)(F)c1ccccc1 N1(C(Cc2cc(C)no2)=O)CCC(C)(N(C)C)CC1.c12ccc([nH]1)CNC2=O C1(CC(=O)N(CC(O)CN(C(=O)C(C2CC(F)(F)C2)O)C)C)COCC1(C)C C(CO)(C(=O)NC(C(=O)NCc1nc(C2CC2)n[nH]1)C1CCC1)OC O=C1NCCCC1CC(N1CC(CCCc2cn(-c3ncc(Br)cn3)nn2)C1)=O C1(O)(CCNC(c2c(CC)occ2)=O)CCN(C(c2cnc(C(C)OC)s2)=O)C1 C(=O)(C1CCCn2cnnc21)NCC(C1CCOC1)NC(=O)COCC1CC1 CCC(C)N(OC)C(=O)c1cc(CNC(=O)NC2CCC(N=[N+]=[N-])C2)cs1 N1(C(C2OCCN(C(C)C)C2)=O)CCN(C(=O)Cc2cccnc2)CC1C C1(C(=O)OC(C(CC)CC)C(=O)OC)CNCC12CCOCC2 c1(OC(C(=O)N(CC(C)NC(=O)Cc2nc(C)no2)CC)C)cccc(CO)c1 Cc1c(C(=O)NC(C2(O)CN(C(=O)C(C)C(F)F)C2)C)cnn1C(C)(C)C C1(C)(c2cn(CC(COC)O)nn2)CCCN1C(C1CCC(=O)NC1)=O c1(N2CC(OC)C(F)C2)nc2cc(C)ccc2c(=NCCC#CBr)[nH]1 c1(NC(=O)NC2C(SC)COC2)cnc[nH]c1=NC c1(-c2cn(CCC(=O)N(C3CC(=O)NC3=O)CCC)nn2)ccc(CO)cc1 C(C)(C(C(C)C)NC(=O)CSc1ccccc1)NC(CCCOC(C)C)=O N1(C(c2ccc(C)o2)=O)CCCCC2(C1)CN(C(=O)C=CC1CCCC1)C2 CC1COCCCN1C(C1CCN(C(C2CC3CCCC3C2)=O)CC1)=O c1(C(N2CCC(NC(C3CC3C(F)(F)F)=O)C2)=O)c(F)ccc(OC(F)F)c1F CC1CCN(C)c2ccccc2N1C(c1cc(C2(Cl)CC2)n(C)n1)=O c1(COCCNC(C(C)NC(=O)CC2CC2)=O)csc(Cl)c1 c1(NCC(=O)NCC(C)N(CS(C)(=O)=O)C)ccc(Cl)cc1Cl N1(C(COCC)=O)CC2C(C(=O)NC3CCNC3=O)C2C1 N1(C(C(=O)NC(CNC(CCC(=C)C)=O)C)C)C(=O)NC2(CCCC2)C1=O c1(C(N2C(C(CNC(CN(C3CC3)CC)=O)(C)C)CCC2)=O)cc(C)ccc1F C1(C(=O)NCCC2N(C(C(C)OCC)=O)CCC2)CCCC(=O)O1 C=CCC(C(=O)NCC1CCC(C(N2CCCCCC2)=O)O1)OC C#Cc1ccc(CC(N2CCC(N3CCC(=O)NC3=O)CC2)=O)c(F)c1 C1(C(=O)NC2CN(C(C(C)O)=O)CC2C)CCC2C(C1)C2(F)F N1(C(c2cc(C)sc2)=O)CC(CNC(c2sccc2Br)=O)CC12CCC2 CC1(O)CC2CC1CC2NC(=O)CC1CCCCN1C(C1OC2CCC1C2)=O CC(C)C(C)C(CNC(=O)C=CSc1ccccc1)NC(c1cnc(S)nc1)=O C(CC(=O)Nc1ccc(Cl)cc1C)(C(C)(C)C)NC(C(CCC)C)=O N1(C(CN(c2cccc(O)c2F)C(c2c(CC)n(C)nc2)=O)=O)CCCC(F)CC1 c1(C(N2C(CN(C)C(C3CC3c3cccs3)=O)CCC2)=O)cccn2nnnc12 N1(C(CCCOC)=O)CCCC2C1CCCN2C(C1CC2(CCO1)CC2)=O C1(CNC(c2cn(CC)nn2)=O)CN(C)CCN1C(c1c(Cl)c(C)nn1C)=O C12(NC(N3CCN(c4cccc(F)c4)CC3)=O)COCC1C2(F)F c1(SC)cc(C(=O)NC2(CN(C)C(C3C(C)(C)C3(F)F)=O)CC2)oc1C Cc1ccc2sc(C(=O)NCc3ccc(CNC(=O)CC4CC4C)cc3)cc2c1 C1(CC(N2CC(C(=O)OCC)C2)=O)C2CCCC2N1C(=O)CC1(O)CCOCC1 C(=O)(C1CCc2c[nH]nc21)NCC(CN(C(CCCC=C)=O)C)C C(=O)(C(F)C1CCCC1)N(CCOCCN(C(=O)CCn1cccc1)C)C1CC1 c1(CS(C)=O)cccc(C(=O)NCCC2CCN(C(C3(C)CC3(C)C)=O)C2)c1 C1(OC)CC2CC(NC(=O)C(C3CCCC3)NC(c3sccc3C)=O)CC12 N1(C(C2CCCC3CC23)=O)CCC(C2CC2)(NC(=O)C(F)(F)CO)C1 Cc1ccc(C(=O)NC2CC2CNC(c2sccc2C)=O)cc1N1CCOCC1 CCCC(CC)CC(=O)NCC1CN(C(c2c(C)cnn2CC)=O)CCC1(F)F N1(C(=O)Nc2cncc(C(N(C)C)=O)c2)CC2(CCC1CO)CC2 CC1(C)CCCCC1C(=O)NC1CCC(CNC(c2cnc(O)c(F)c2)=O)C1 CC(C)C(CC(=O)N1CCCC1CNC(=O)C(F)(F)C(F)F)c1ccccc1 c1(C(=O)NCC2(CC(=O)OC)CCOC2)cc2c(=O)[nH]ccn2n1 c1(C2CCN(C(C(C)(F)c3ccccc3)=O)C2)ccc(C(=O)NC2CC2)cc1 Cc1cc(C(=O)N(C)CC2CCCCN2C(=O)CC(O)CC2CC2)cc(N)c1 CC(C(=O)NCC12CC(NC(=O)Cc3csc(S)n3)(C1)C2)C(C)S(C)(=O)=O C(CC1CCC1)(C(=O)NCCc1ncc(C)o1)NC(C(C)NC(=O)NC)=O c1(C(N(C2CC(NC(C3C(C)C3C)=O)C2)C)=O)cc(S(N)(=O)=O)ccn1 C1(C(=O)NCC(C(C)C)NC(c2cn(CC)nc2)=O)CCc2c(n[nH]c2C)C1 C1(NC(C2CCC(F)CC2)=O)CCN(C(=O)C=Cc2ccncn2)CC1 Cc1cccc(C)c1OCC(=O)N(CC(CC=O)NC(=O)C(C)CO)C N1(CC2CC(OC)OC2OC)CCOC(C)(C(=O)OC)C1 C1(NC(C(CC(=C)Cl)NC(=O)Cc2cc(C)cs2)=O)Cc2ccccc2C1 N1(C(CCCC(=O)NCC)=O)CCN(C(=O)CCCn2ccnc2C)CCC1C C1(C(=O)NC2(C)CN(C(C3CC4(CSC4)C3)=O)C2)CSC(c2ccccc2)=N1 c1(C(N2C(CNC(c3cn(C(C)C)nc3)=O)C=CC2)=O)ccnc(S)c1 c1(C(=O)NCCC2CCCN2C(c2ccn(CCF)n2)=O)cnc2c(c1)CCC2 C1(C(N(C2CN(C(c3nccnc3N)=O)C2)C)=O)CCCC(O)C1 Cc1cc(C)c(C(N2Cc3c(C(=O)NC4CC(=O)CS4)coc3C2)=O)cc1C c1(CNC(c2ccc(NC)nn2)=O)ccc(-c2cncc(NS(C)(=O)=O)n2)c(C)c1 c1(C(=O)NC(CNC(CC(C)N2CCCC2=O)=O)(C)C2CC2)cc2n(n1)CCO2 C1(NC(=O)C(=O)C2CCCC2)CCC(NC(C2CCCCC2)=O)CC1 C(CC(F)F)(C(=O)O)N(C(C1C(CC)C1)=O)Cc1cn(Cc2ccccc2)nn1 C1(OCC(=O)NC(CNC(c2ccsc2C(F)(F)F)=O)CO)CCCOC1 C12(NC(C3(C)CC3)=O)CCC(CC1NC(=O)CCn1cc[nH]c(=O)c1=O)C2 C1(CNC(CCC(C)OC)=O)CC2CCC1N(C(c1ccc(N)c(C)c1Cl)=O)C2 N1(C(COCC(C)(C)C)=O)CCN(C(=O)CC2CC2)C(c2cccc(F)c2)C1 CS(C)(=O)=NCC(=O)NC1CCCN(C(c2ncccc2C(F)(F)F)=O)CC1 N1(CC(=O)NC2CC(Nc3cc(O)ncn3)C2)CCC2(CCC(O)C2)C1 N1(C(C=CCCC)=O)CCC2(CC1)CN(C(=O)CC1CCC(F)(F)C1)CC2CO CC1CN(C(C2(C)C=CCC2)=O)CCN1C(c1cn(C)nc1C(=O)C(F)(F)F)=O N1(C(C(=O)NCC(CC)NC(CC=CC=C)=O)CC)C(=O)c2ccccc2C1=O n1(CC)cc(C(=O)NC(C)CC2CN(C(c3cnc(C(C)OC)s3)=O)C2)cn1 CC(C(=O)NCc1cn(C2CCN(C(C3CC34CC4)=O)CC2)nn1)C(C)O CCC(CC)CCCC(=O)N1CC(C)(C)CC1CNC(c1cc(=O)n(C)o1)=O N1(C(c2c(OC)oc(C)n2)=O)CCC(NC(c2sc(C)cc2Br)=O)C(O)C1 c1(C(=O)NC2C(NC(C(C)OCCC=C)=O)C2)ncn2cc(Cl)ccc12 Cc1cc(Cl)ncc1NC(=O)NC(c1ccnc(-n2cnnc2)c1)C1CC1 c1(CC(=O)NC(CCNC(Cn2c(C)ccn2)=O)C)ccc(Br)cn1 C1(CNC(=O)NCC(C)SC)C2CCC(C2)C1C(=O)NCC1CC1F O=S(=O)(c1cccc(NC2(NCC3CCCO3)CCNCC2)c1)N1CCOCC1 CC(C(C)NC(=O)Cn1cnnc1)NC(=O)CSC(F)F CC1(C)CCN(C(=O)C=CC2CC2)CC1C(=O)NCC(O)CF c1(CNC(C2CC2Cl)=O)ccc2c(c1)CN(C(=O)CC(O)C1CCCC1)C2 Cc1ccc2cc(C(=O)NCCC3CCN(C(=O)CN4CCC4C)CC3)nn2c1 Cc1nc2cc(Cl)cc(C(=O)NCC(CO)NC(C3CCCN3C3CC3)=O)c2[nH]1 C1(NCCN(C(CCCC)=O)C(=O)CC2(C)CC2)CCCC(OC)C1 C1(N(C(C(=O)NC(COC)C)CCc2ccc(F)cc2)C)CC2(CCCCC2)C1 CCCCS(=O)(=O)NC(C)C(=O)N(C)CCNC(=O)C=CS(C)=O c1(C(N2CCC(CNC(C3C=CCC3)=O)C2)=O)noc2ccccc12 CC1(C(=O)NCC2(O)CCN(C(c3cc(C#N)cs3)=O)C2)CCCC1(F)F C1(CNC(c2cnc(CC)o2)=O)CC(C)(C)CN1C(c1cc(C(F)F)n(C)n1)=O C1(C(N(CC(C)(C)NC(c2ccc(Br)cc2)=O)C)=O)CCCC(=O)N1C C1(C#CC(=O)NC2(C)CCCN(C(c3cccc(Cl)c3C(F)F)=O)C2)(CC)CC1 c1(NC(C2CCCN(S(C)(=O)=O)CC2)=O)ccc(S(=O)(=O)N)cc1.CCO Cn1cnnc1C1(NCCCSC2CCCO2)CC1 O(NC(=O)C(C)(CNC(c1cc(CO)n(C)n1)=O)CC)C(C=C)C C1(CC(=O)O)CC=CCC1.C1(=O)C(C)N(CC)C(C)CN1CC.C(C)=O N1(C(C(CSC)(C)NC(c2cc(C3CC3)on2)=O)=O)CCc2ccccc21 C1(C)(C(=O)OC)CCC1(C)C(=O)N(C)CC1CN(C(C2CCOC2)=O)CCO1 C1(C(=O)NCC2CN(C(Cc3nc(C)[nH]n3)=O)CC2C)COC2(CCC2)C1 c1(C(N2CCC(NC(C3CC(OC)C3)=O)C2C)=O)ccc2cnccc2n1 C1(C(N2CCC(N(CCC)C(C)=O)C2)=O)CCc2nc(CC)ncc2C1 C1(NC(CN(C)CC)=O)CN(C(=O)C=CCN2CCCCC2)CC1(C)C N1(C(c2c(C)[nH]nc2CO)=O)CCC(O)(C2CCN(C(=O)CNC(N)=O)CC2)C1 c1(N(CCC)C)n[nH]c(C(=O)N(C)CCNC(c2ccc(C(C)C)o2)=O)n1 c1(COCC(=O)NC(CNC(CN(CCCC)C)=O)CCC)ccccc1C c1(C(=O)NC2C=CC(CNC(C(CCCCC)O)=O)C2)ccc2sc(C)nc2c1 C(C(C)(C)SC)(C(F)(F)F)OC(c1c(-c2ccncc2)nc(OC)s1)=O CC1CCC(Cl)=C(C(=O)NCC=CCNC(=O)C(C)NC(=O)OC(C)(C)C)C1 C1(CNC(=O)CCCc2cccs2)CCCC(NC(=O)Cc2ccco2)C1 C1(C(=O)NC2(CC(N3CCC(OC)CC3)=O)CC2)CCC(=O)N(C)C1 C=C(C)C(C)(C)C(=O)N1CCOC(CN(C)C(C2CCC(=O)NC2)=O)C1 c1(CC)n[nH]c(=NC(C)C2CCN(C(c3cc(CC4CCC4)c[nH]3)=O)CC2)s1 C(=O)(C(F)C(C)CNC(c1nonc1C)=O)NCCCC(=O)OCC S(=O)(=O)(c1cncc(N)c1)NC(=O)NC(C(C)C)C(=O)Nc1ccc(F)cc1 C(C)(C(C(=O)N1CCC(CN=[N+]=[N-])C1)NC(=O)Cc1cc[nH]c1)OC N1(C(c2c(CC)ocn2)=O)CCC2(NC(c3cnc(O)c(C)c3)=O)CC2C1 N1(C(C(C2CC2)SC)=O)CCN(C(=O)CCCCN(C)C)CC1c1nccn1C C(=O)(CCCC(C)=O)NC(C(CO)NC(CCCCOCCC=C)=O)C C1(NC(C(COC)OC)=O)CC2CN(C(=O)C3=C(C)OCC3)CC12 c1(OC2CCN(C(C(=O)NC3C(CN)CCC3)=O)C2)cc(F)c(Cl)cc1Br CCCC(C)(CCC)C(=O)NCC1COCC1NC(C1SCC=C1C)=O C1(C(=O)NC(C(=O)NC)C2CC2)CCC(C)(C)N(C(=O)COc2ccsn2)C1 C1(F)(CNC(C=CC(C)NC(C)(C)C)=O)CCN(C(=O)C(F)CC2CC2)CC1 c1(OCCC(=O)NS(=O)(=O)CC2OCCO2)ccccc1F c1(C(N2CC(NC(CCc3cc(C)on3)=O)C(O)C2)=O)c(F)ccc2[nH]ccc12 c1(C(=O)NCC2(O)CC(C(N3CCC(=CCC)C3)=O)C2)cc(O)nc(N(C)C)n1 C1(C(=O)NCC(C(=O)NCCN2CCOC(C)C2)OC)CC2CCCC2C1 C=Cn1nccc1C(=O)NC(C)CNC(c1cc(-c2cccc(F)c2)ccn1)=O C1(OC)CCC12CC(C(N1CCOCC1CCNC(C1CCC1)=O)=O)C2 C1(CCNCC(=O)NCCC=CC=CC)CC(O)CN1C(=O)OC(C)(C)C CCC(C)CC(=O)N(CC(C)O)CCNC(=O)CN1CCN(c2ccccc2)CC1 c1(C(=O)NC(C)(C)CCNC(C2C3CCC(F)C23)=O)ccc(O)nc1Cl c1(NC(C)=O)cccc2cc(C(N3CC4CC3CN4C(=O)CC3CC3C)=O)[nH]c12 C(C1c2ccsc2CCN1C(c1cn[nH]c1)=O)NC(C(C)(C)C1CCOC1)=O N1(C(=O)NC(c2ncccn2)C)CCNCC1c1cccc(F)c1 Cc1ccc([N+](=O)[O-])c(C(=O)NCC2CC2CNC(C2CCCCCCC2)=O)c1 CC(C)CCC(=O)NC1CCC(CCNC(=O)CN(c2ccccc2Cl)C2CC2)C1 C1(NC(C2CCCCC2O)=O)CC2(C1)CC(C(=O)NCC1CC1CO)C2 c1(CC(N2CCC(CNC(C=C(CC)C)=O)C23CC3)=O)nccc2ccccc12 C1(NC(CC2(OCC)CCC2)=O)C=CCCC1C(=O)NCC1CCSC1 c1(CC)ccc(NC(c2nnnn2CCCOC)c2cnc[nH]2)c(C)c1 c1(C(N2CC(F)(C(N3CC(C)OCC3)=O)C2)=O)c[nH]nc1[N+](=O)[O-] c1(C(=O)NC(c2ccnn2C)C(=O)OC)nc(C)no1 C1(CC)CN(C(C2CCCC(F)C2)=O)CCN1C(=O)CCc1ncccc1C c1(C(=O)NCC(C2CCC2)NC(CC2CC(=C)C2)=O)ccn(CC(F)(F)F)n1 N1(C(C2(CC)CCC2)=O)CCC2(C1)CN(C(=O)Cc1ccc(C#N)nc1)CCO2 C1(C(=O)NC2(C)CCC2)CC=CC(NC(C2CCC2C(C)(C)C)=O)C1 c1(C(=O)NC2CCC(N(C(=O)Cn3cccn3)C)C2)cccc2ccncc12 C1(C)(CC)CCC(C(=O)N(C)CCOCCC(=O)NCCC=CC(C)(C)C)O1 C1(CNC(C(C)C(C)(C)C)=O)CCCC2CN(C(=O)Cn3ccccc3=O)CC12 c1(C(=O)NC2C(NC(Cc3nc(C)sc3)=O)CCC2)cc(O)cc(=O)o1 CC(C)(C)C#CC(=O)N1CCC(CF)(NC(=O)CC(C)(C)c2cccs2)C1 N1(C(c2n(CCC)ncc2)=O)CCC2CC12C(=O)NC(C)CCC(C)C C(=O)(C1=CCCCC1C)N1C(CNC(c2c(C)cccc2O)=O)CCCC1 C#CC1(C(=O)N(CC(C)COC)C)CN(C(C23CCCC2C3)=O)C1 c1(N2CCN(C(C(C)OCCC=C)=O)CC(O)C2)cc2nnc(C(C)C)n2cn1 C(CC(C(C)(C)C)NC(=O)Cc1cnnn1C)N(C(=O)CCC1CCC(=O)C1)C N#Cc1ccccc1NC(N1CC2C(CNC(c3ccc([N+](=O)[O-])[nH]3)=O)(C2)C1)=O c1(C(=O)NCC(F)CNC(C2CCCO2)=O)[nH]cc2c1CCS2(=O)=O c1(CNC2(CO)CC(CC(C)C)C2)ccc(I)cc1F CCC(C)CCC(=O)NC(C)CC(C)NC(c1csc(CC(C)C)n1)=O N1(C(CC=CCC)=O)CCC(N(C)CCn2ccnc2C)C1 C1(CC(=O)NCCC(C)CCNC(=O)C(Cl)=CCl)SC2=NCCN2C1=O C(C(C(=O)NCC(c1ccncc1)C)NC(=O)CCC1CC1(F)F)OCC C(CCC(C)(C)C(=O)NC1CCC1(C)C)NC(C1=C(C)CC1)=O C(=O)(C(CC(C)C)C(C)C)NCC(C)(C(C)C)NC(c1cc(C)nc(O)n1)=O C1(COC(=O)NCC(C)(C)CNC(=O)OC(C)(C)C)CCC2COCC2O1 C1(CCNC(C=CCN(C(=O)OC)C)=O)(CNC(=O)N)CCOC1.C1(CO)CC1 CC(Cn1ccnc1)C(=O)NCCNC(=O)Cc1csc(Br)c1 CCC(C)CCCCC(=O)N1CC(OC)C(C(=O)NCCc2ccon2)C1 C(=O)(CCC(C)CC)NCCOC.CCCC(C(=O)N1CCCC1)NC(N)=O N1(C(C2C3CN(C(c4cc(C)c(O)nc4)=O)CC32)=O)CC2(CCC(=O)O2)C1 O=CCCCCC(F)F.C1(c2cccc(C3CC3)c2)CN(C(=O)CO)CC(F)(F)C1 C(=O)(C(C)(O)C(F)(F)F)NC1C(NC(c2nn(CC)c(C(F)(F)F)c2)=O)CCC1 n1(C(c2ccncc2)C)nc(C2CCCO2)nc1-c1cc(C(F)F)no1 c1(NC(C2N(C(c3c(OC)nc(C)cc3)=O)CC(F)C2)=O)ccc2[nH]ccc2n1 c1(C(N2CCC(F)(CNC(C(C)(C)N(C)C)=O)C2)=O)ccc([N+](=O)[O-])cc1N c1(CNC(C(c2ccccc2)C)=O)ccc(NC(=O)OC(C)(C)C)cc1 C1(CCNC(c2n(C)cc(Cl)c2)=O)CC(F)(F)CN1C(C1CCOC1=O)=O C1(Cn2cc(C(C)C)nn2)CCCN(C(=O)CCc2ccc(C(C)(C)C)cc2)C1 c1(CN(CC(=O)NCCCCCNC(C(CC)SC)=O)C)ccc(O)cc1 C1(C(N2CC(OC3CCN(C(C(C)(C)N(C)C)=O)CC3)C2)=O)CN2CCN1CC2 C(=O)(CC(CNC(C1(OC)CCC1)=O)NC(C)=O)N1CC(C(=O)NCCCC)C1 Cc1nn[nH]c1CNC(=O)C(=O)Nc1cccn1C C1(C(N(C(C)C)CCC2CCC2)=O)C2CCN(C(N3CCOC3=O)=O)CC12 c12ccc(cc1NC)C(=O)OCC(=O)N2.C=C(C)C(C)COC N1(CCOC(=O)OC(C)(C)C)CCCC(COCC(N)=O)C1 c1(C(N(C)CCOCCNC(C2(CS(C)(=O)=O)COC2)=O)=O)nn(C)cc1Br CCCC(CC)CCC(=O)N(C(C(N1CCC12CC(C)(CO)C2)=O)C1CC1)C C(C(C)C(C)(F)F)NC(CCN(C(C(C)OC)=O)CCO)=O Cc1ccc(C(=O)NC(C)CCN(C(=O)CCn2cc(Cl)cn2)C)c(Cl)c1C Cc1cc(Cl)ccc1-n1cc(C(C2CCC2)NC(N)=O)nn1.C1(=O)CCCCCN1 c1(C(=O)OC)csc(=NC2CC(F)CN(C(=O)C(C)(C)F)C2)[nH]1 C1(CNC(CCc2c(C)noc2)=O)CC2(CC2)CN1C(=O)CC1CNC(=O)C1 N1(C(c2c(C)nc(O)[nH]2)=O)CC2CCC1C(NC(=O)CSCC1CCCCO1)C2 C(=O)(CCCC(F)(F)CO)N1CCC(NC(C(CC)OC)=O)C(CC)C1 CCC(C)(C(=O)NCc1ccc(CNC(=O)C(C)(C)c2cnc[nH]2)cc1)C(F)F N1(C(c2c(C)scn2)=O)CC2(C(=O)NCC=C(Cl)Cl)CC1CO2 CC1CN(C(=O)C=CCN2CCCC2)CC1NC(C1CCC(C(N)=O)N1C)=O Cc1ncc(N)cc1C(N1CC(N(C)C(C2OCCOC2(C)C)=O)C1)=O C=CCC(CNC(=O)C(Cl)Cl)C(=O)NOCCC(C)O C1(NC(C2CCOC2)=O)CCOC2(CCN(C(=O)CCC3CC3(Cl)Cl)CC2)C1 C1(NC(c2c(C)scc2)=O)CCC2(CCN(C(C3(F)CC=CC3)=O)CC2)C1 c1(C(N2CC(NC(C3(C(C)C)CCCC3)=O)C(C)C2)=O)ccc(Br)cc1O C(=O)(CC(C1CC1)C1CC1)NCCCNC(C1C(CC)C1)=O Cc1ccn2cc(C(N3CCCC(NC(=O)C(C)CC(C)(C)C)C3)=O)nc2c1C c1(C(=O)NC(C)CNC(c2cncn2C2CC2)=O)cc(Cl)c(F)cc1Br CC(C(C)(C)C(=O)NCC(=O)OC(C)(C)C)NC(c1ccnn1C1CCC1)=O n1(CCCCC)ccc(=NC(=O)OS(=O)(=O)CC2(C)CC2)[nH]1 N1(C(C(C=CC)O)=O)CCC(C(=O)NC(CC)C(C)CN(C)C)CC1 CC1(C)CCN(C(=O)N(C2CC2(Cl)Cl)C(=O)C2CC2)C1C.CCCCCc1cn[nH]c1 C12(CC(=O)NC(C(=O)OCC)C)CCC1CN(C(c1cc(C)n(CC)n1)=O)C2 c1(NC(c2c(NC(C(c3ccccc3)C)=O)c[nH]n2)=O)cnc(SCC#N)nc1 c1(NC(c2nnnn2C2CCCCC2)C2C(C)C2)ccc(Br)cc1N(C)C N1(C(C2C3(CC(NC(CC4(OCC)CC4)=O)C3)C2)=O)CCC2(CCC(O)C2)C1 C1(NCc2c(OC)ccs2)CCC(C(=O)NC2(C)CCOCC2)CC1 C1(NC(c2cc(CC)on2)=O)CCCN(C(=O)CC2(C)CC2(Cl)Cl)C1C N1(C(C(CO)NC(c2c(CC)nccc2)=O)=O)CCC(O)C(C)C1 c1(C(N2CC(N(C(=O)C=Cc3ccsc3)C)C(C)(C)C2)=O)cnn2c1OCCC2 C1(NC(c2ccc(N3CCC(O)CC3)cc2)C)C(C(=O)O)C2CCCC12 c1(CCN(C)CC)cn(CCCCNC(C2CC(C)=NO2)=O)nn1 CC#CCCCC(=O)N1CCC2(NC(=O)CCOC3CCOCC3)CC2C1 C1(NC(CNC(C)=O)=O)CCN(C(C2CC(C)CO2)=O)CC1 C1(CNC(=O)CCC(F)(F)F)CCCC2CN(C(c3cncnc3)=O)CC12 C1(CC)CC2CCC(C1)N2C(C1CC2(CC(NC(C3CCC(C)O3)=O)C2)C1)=O C1(NC(C(F)=CC)=O)CN(C(=O)COc2ccccc2)C2(CCOCC2)C1 C(C1=CCN(C(C2CCCCC2CNC(=O)C(F)=CC2CC2)=O)CC1)OC N1(C(c2ncc(C[SH2]CC)nc2)=O)CCN(C(C2CN(C(C)=O)C2)=O)C(C)CC1C.CC C1(NC(c2ccc(OC)o2)=O)C=CCN(C(=O)CCCOC(C)=O)C1 Fc1cc(Cl)ccc1-n1nc(C(F)F)nc1-c1ccnc(F)c1 N1(C(C(C)N(C(=O)Cc2cccc(O)c2)C)=O)CCC(C2=NOCC2)C1 c1(OCC(C)C)ccc(C(=O)N(CCNC(C2CCN2C(C)C)=O)C(C)C)cn1 Cc1nc2ccccc2cc1C(N1CCN(CCC(=O)O)CC1)=O C(=O)(CCCC(C)(C)C#N)NC1(C(N(CC(F)(F)CO)C)=O)CC(O)C1 Cn1c(NC(N2CCCC(Cn3ccc(O)nc3=O)C2)=O)nc2ccccc12 c1(C(=O)NCC(c2ccccc2)CNC(CC=CCC)=O)ccc(Cl)c(F)c1 C1(C(C)C)CN(C(C2CCCCC2CNC(C2CCOC2(C)C)=O)=O)CC(=O)N1 C(=O)(C1=C(F)CN(C(=O)CCC(N)=O)CC1)N1CCCC(CC#C)C1 Cc1cncc(CCNC(C2(C)CN(C(=O)CC3OCCC3(C)C)C2)=O)n1 c1(C(=O)OC)ccc(CC(=O)NCC2CCCN2C(=O)C(C)CC(F)F)c(C)c1 CN1CC(=O)N(CC(=O)NCC2(C)CCCN(CCN3CCOCC3)C2)C1=O c1(C(C2(N(C(c3scc(OC)c3)=O)CC3CC3)CCOCC2)C)cc(C)nc(O)n1 C=C1CCN(C(C2CC(=O)OC2(C)C)=O)C(C(=O)NCCCOCCCC)C1 Cc1ccc(C(=O)NCC(F)CNC(=O)C=CCCc2ccccc2)c(C)n1 C(N=c1nc(O)c2c(ncn2C)[nH]1)C12OC(C)C(NC(=O)C(C)N3CCC3)(C1)C2 C12(C(=O)OC)CN(Cc3cnc(OC)c(Cl)c3)CC1CCO2 CCC(CNCCOCC)N=c1nc2c(cnn2C)c(NCCCF)[nH]1 N1(C)CCCC2(CNC(=O)CN(CC(=O)Nc3c(C)c[nH]n3)C)CCCC12.C(C)C N1(C(c2cnc(N(C)C)o2)=O)CCC2CCN(C(=O)CN3CC=CC3)CC2C1 C1(N2C(C)C(C(F)(F)F)OCC2)CCc2ncccc2C1 Cc1cncc(C(=O)NC2CC(C)N(C(c3ccc(C(=O)N(C)C)cc3)=O)C2)c1 CC(C)CC(C(=O)NCCNC(=O)C1CC1)ONC(C1CCCCC1(C)C)=O C1(C(N(C)CC2(O)CCOC2)=O)N(C(=O)CC2CC=CC2)CCCC1(C)C O=C(C(F)CC1CCC1)NCC1(O)CC(C(=O)NCC2CC2Cl)C1 N1(C(Cc2cn(CC)nc2)=O)CC(O)CC1CC(=O)Nc1ccnn1C1CC1 c1(OC)ccc(-c2nc(CN(C)C)nn2-c2nnc(C3CC3)n2C)cc1OC c1(CC(=O)N(CC(CNC(CCC=CC)=O)C)C)nsc2ccccc12 Cc1cc(C(=O)NC2C=CCN(C(=O)CCc3ccccc3O)C2)c(C)s1 CCC(F)(C(=O)OC)C(=O)NCCC(C)N(C)C(c1cnsc1C)=O CCC(N=c1nc2scnc2c(N2CCC(C)C2)[nH]1)C1CCC1 N1(CC)CC(C(=O)NC2CN(C(c3occc3C)=O)CC2O)CC1=O C1(C(=O)NCC(COC)NC(=O)C=Cc2ccc(C)cc2)CCC(C2CC2)CC1 c1(C(N2CCCC(CNC(C(CC)(C)OC)=O)C2)=O)cc2c(s1)CCS(=O)(=O)C2 C1(CC(=O)NCCN(C(=O)C(O)Cn2cncn2)CCO)CCSCC1.C1(N)CC1 S(=O)(=O)(c1ccc(N2CCn3ccnc3C2)c(F)c1)NC(COC)C(C)C c1(C(=O)NC(CNC(C(F)=C(C)C)=O)(C)C2CC2)ccc(C(C)(C)C)[nH]1 c1(CNN(c2cc(OC)ncn2)C(=O)Nc2ccccc2)cnc2c(c1)CNCC2 c1(OC)ccc(F)cc1CNCCCOCCC(F)(F)F Cn1cnc2cc(C(=O)NC3CC3NC(=O)COc3ccc(F)c(F)c3)ccc12 N1(C(C(CC2CCCC2)SC)=O)CCC(C)(C(OC)OC)C1.C12CCN1C2=O N1(C(C=CC(=O)N(C)C)=O)CCN(C(C2CCC2)=O)C2CC12 C#CCCCCC(=O)NCC(C)(F)CNC(C1CCCCC1CC)=O Cc1cc(NC(=O)CC(F)(F)Cc2ccc(Br)cc2)cc(C#N)n1 c1(OC)ccc(Cc2nc(-c3ccc(Cl)cn3)nn2CC2CC2C)cc1 C1(C(C)(C)C)(C(=O)N)CCCCC1.c1(C(C(C)CN(C)C)=O)c[nH]c(Br)c1 c1(C(N(C)CC2(O)CN(C(C(C=C)C)=O)C2)=O)ccsc1C#N C1CC(O)C(O)CC1C(=O)NCCCCCSC.CC(=NOCC#N)C(=O)NC1CC1 C1(C(=O)NC2(C)C(C)C2)C2CC1N(C(=O)Cc1ccon1)C2 C(CC(=C)Cl)(C(=O)N(CC(C)O)C)NC(COCC#C)=O C1(C(=O)NCC(C#C)OC)CN(C(c2cn(C(C)C)cn2)=O)CC1CC CCCC(C)C(=O)N1CCC(C)(CNC(c2cncc(OC(F)(F)F)c2)=O)C1 C(C(C(F)(F)F)OC)NC(C1(NC(C2CC(O)(CC#C)C2)=O)CC(F)C1)=O C1(C(N(CCCNC(CC=C)=O)CCO)=O)CCOC2(CCC2)C1 C1(CNC(=O)C=Cc2cc[nH]n2)CN2CCCCC2CN1C(c1cc(O)cs1)=O N1(C(C(=O)NCCCC(=O)OCC)C2CC2Cl)CCOc2cc(C(N)=O)ccc21 C1(C(=O)NC2C(NC(c3cc(C)ncn3)=O)COC2)CCOC2(CCC2)C1 c1(OCC)nn(C)cc1NC(c1nc(Br)nn1C)c1nnnn1C1CCCCCC1 C1(F)(C(N(C(C)C)C)=O)CCN(C(=O)CCC2CC2C)C1 C1(C(C(=O)NCCCCC)C)CCCN(C(c2sccc2Br)=O)C1 c1(C(=O)NC(C(C)C)CNC(=O)CN2C(C)CCC2C)cnn(C)c1S(N)(=O)=O N1(C(C(C)CF)=O)CCOCC(NC(C2(CF)CCC2)=O)C1.c1(N)ccc(CF)cc1 N1(C(CC2C(C)=NN(C)C2=O)=O)Cc2ccc(C#N)cc2C1 c1(C(=O)NCCCOCCNC(C2C(C)CCS2)=O)ccccc1-c1ccccc1 c1(OC)cc(O)ncc1C(N1CCC(NC(C2CCCS2(=O)=O)=O)C(F)C1)=O C1(NC(=O)Cn2nnc(C3CC3)n2)CC(O)CN(C(C2C=CCC2)=O)C1 C12(C(=O)NC3CCC(NC(=O)CCc4ncco4)CC3)CC=CC(C1)OC2 C1(C(N2CCC(NC(CC(=C=C)C)=O)(COC)C2)=O)CCC(C)(C)CO1 C=C(C)CCCC(=O)NCC1(NC(=O)Cc2csc(C(C)(C)C)n2)CC(F)(F)C1 C1(C)(CC(=O)NCC(CNC(=O)C(=Cc2cn(C)cn2)F)OC)CC(F)(F)C1 C(=O)(CC(O)C(Cl)(Cl)Cl)N(CCCNC(c1ccc(=NC)[nH]c1)=O)C c1(OC)ccc(CCC(N2CC(NC(c3coc(C(C)=O)c3)=O)C(O)C2)=O)cn1 c1(OC)cccc(C(C)(C)C(=O)N2CC(CO)(NC(=O)CC3CNC(=O)C3)C2)c1 C1(CN(C(Cc2c(C)non2)=O)C)CCCN(C(=O)C(C)(C)c2cc[nH]n2)C1 c1(NS(CC)(=O)=O)cccc(C(=O)NC2CN(CC(F)F)C2)n1 C1(NC(C(c2n(C)ccc2)=O)=O)CCCN(C(c2csnc2C2CC2)=O)C1 c1(C(=O)NC2CC3(CC(NC(C(CC)C(C)O)=O)C3)C2)nccc2n[nH]cc12 c1(-c2nn(CCC)c(-c3ccc(C4CCO4)cc3)n2)cc(C)c(C)c(Br)c1 c1(OC)ccc2[nH]c(=NC3CC(C)N(CO)C3)[nH]c(=NCCOCCF)c2c1 CCCCC(CNC(=O)COCc1nccn1C)NC(c1cnc(SC)n1C)=O C1(CC(=O)NCCC2(O)CCN(C(CCC=C)=O)C2)COCC2(CCC2)O1 n1(CCC)ncc(C(=O)NC23CC2CN(C(=O)CCC2CC2(C)C)C3)c1C N1(C(c2nnc(CC)s2)=O)CCC2CCC(C1)N2C(C1CC(C(C)(C)C)=NO1)=O c1(C(N2CCC(C)N(C(c3cc(O)ccn3)=O)CC2)=O)cccc2c1OCCC2 N1(CC)CCC(NC(=O)C(C)(CO)NC(=O)C=Cc2nccs2)C(C)C1 Cc1nc2ncnn2cc1C(N1CCC(C)N(C(=O)C=CCn2cncn2)CC1)=O c1(CC)n[nH]c(=NC2CN(C(c3ccc4cc[nH]c4c3)=O)Cc3ccccc32)s1 C(=O)(C(C#N)C(C)(C)C)NC1(C)CCN(C(C2(COC)CCOC2)=O)CC1 c1(C(C(=O)NC2COC2)N(C2CN(CC)C(=O)C2)C2CC2)noc2c1CCCC2 C1(NC(=O)C=CC2CCOC2)CCCC12CN(C(C13CC(F)(C1)C3)=O)C2 CC(CC(=O)N1CC2C(NC(C34CC(CC5CC5)(CO3)C4)=O)C2C1)C(F)F O=S(=O)(c1c[nH]ccc1=NC1CC2CCC(C1)O2)NC1CN(C2CCC(O)CC2)C1 C(C)(CCC(=O)N1CCOC(CCC(=O)NCc2nc(C3CC3)no2)C1)OC Nc1cc(F)cc(F)c1C(=O)NC12CCN(C(C3(c4cccs4)CC3)=O)CC1C2 N1(C(c2ccc(OC)nc2)=O)CC2(CCC2)CC1CNC(=O)C(C)C1CCCC1 C#CC1CCC(NC(C2C3CN(C(C4(c5ccccc5)CC4)=O)CC23)=O)CC1 C(C(=O)NNc1c(F)c(F)cc(F)c1F)c1n(CC(C)(C)C)ncc1 Cc1ccc(C(=O)NC2CN(C(c3ccc(I)cn3)=O)CC2F)cc1Cl O=C(C1CCCn2cncc21)N1CCC2CCN(C(C3(F)CC3)=O)C2C1 N1(C(C2C(OCC)C2)=O)CC(NC(c2cnn(C(C)C)c2)=O)CC2(CC2)C1 c1(OC)cc(Br)c(C(C)NC(=O)NC2(CO)CCOC2)cc1OC c1(OC)cc(CO)ccc1C(N1CC=CC(NC(=O)CCC2CCCOC2)C1)=O N1(C(c2nc(C(=O)OCC)sc2)=O)CCC2CCC12CNC(c1sccc1C)=O N1(C(CCc2cncc(C)c2)=O)CCC2(CCCC2C(=O)NC2(CO)COC2)C1 Cc1ncc(C(=O)NCC2CN(C(=O)Cc3nncn3C(C)C)CCO2)cc1N C1(NC(C)C(=O)NC(C)CC(=O)NC2CCCCC2)CCCCC1=O O=C1CCOC(C(=O)NC2CCN(CCNC(C3(CF)CC3)=O)C2)C1 c1(OC)ccc(F)cc1C(=O)NCCN(C)C(C1CC2CCC1NC2)=O c1(C(=O)NC2C(NC(C=C(C)C3CC3)=O)CCC2)nn2c(c1C)CCCC2 C(CCC(=O)NC(c1ccccc1)CNC(C1CC(C)=NO1)=O)N(C(C)=O)C C(=O)(C1Cc2ccc(F)cc21)NC1CCCN(C(C=C(C)C)=O)C1C C(CC(C)C)(C(=O)N1CC(NC(c2ccc(CNS(C)(=O)=O)s2)=O)C1)NC(C)=O C1(C(=O)NCC2CN(C(C=CCCC)=O)C(C)C2)CCC(=O)CC1(C)C c1(C(=O)NC2C(NC(CNC(CC)=O)=O)CCOC2)cncn(C)c1=O c1(C(N(C2(CC(=O)N(CC=C)C)CC2)C)=O)ccc(CC2CC2)cc1 c1(C(c2nnnn2C2(C)CC2)NCCS(CC=C)(=O)=O)ccc(Cl)c([N+](=O)[O-])c1 C1(NC(CCSCCCC)=O)CC2CCC1CN2C(=O)CSCCSC C(=O)(CCCC(=O)N1CCC(CNC(c2ncc[nH]2)=O)C1(C)C)N(C)C N(C)(S(=O)(=O)N(C)C)CC(=O)N(CC(CNC(C(C(C)C)F)=O)C)C C#CC1(C(N2CC3CC3(C(=O)OC(=O)CONC(=O)OC(C)(C)C)C2)=O)CCCC1 C(=O)(C(C)S(=O)(=O)C1CCOCC1)N1CC(NC(C(C)(C(C)C)NC(C)=O)=O)C1 N1(C(=O)CC2CCCC23CC3)CCC2(CC1)CN(C(C1(CO)CCC1)=O)CCO2 Cc1nc(CN(C(C2CC=CCC2Sc2ccc(F)cc2)=O)C(C)=O)n(C)n1 N1(CC)CCN(C(=O)Nc2ccccc2OC(c2ccc(O)nc2)=O)C(CO)C1 C1(C(=O)NCC2(NC(C(COCC)C)=O)CCOCC2)CCCCN(C)C1=O C=C1COCC(C)(C)N(C(C2CCCCC2)=O)C1.C1C(=O)N1 Cc1noc(N)c1C(=O)NC1CCCC1NC(C1C2CCC1(c1ccco1)C2)=O CCS(=O)(=O)c1ccc(C(N2CC(C(=O)Nc3cc(O)ccc3Cl)C2)=O)c(Cl)c1Cl CC1CN(C(C2CCCC2)=O)CC1CC(=O)NC(C)C1CC1 c1(C(=O)NCC2N(C(c3cnc(C)s3)=O)CC(O)C2)cc(Cl)ccc1F C1(C(=O)OC)COCCN(C(=O)Nc2ncc(Cl)nc2Br)C1 c1(NCc2c(-c3c(C)cccc3)cccc2)ccccc1N=c1ccn(C)[nH]1 C1(N(C)C)Cc2ccccc2N(Cc2cn(C(C)(C)C)nn2)C1 C1(OCC=C)CCN(C(C2CCCSC2)=O)C1 C1(CC(N2C(C)(CNC(c3c(C)[nH]cc3)=O)CCC2)=O)CCOC(C)(C)C1 N1(C(c2n(CCC)ncc2)=O)CCN(C(C2(C)CNC(=O)C2)=O)CC1CC(F)F N1(C(CC=CC=C)=O)CCCC(CN(C)Cc2nnc(C(C)(C)C)s2)C1 c1(OC)c(C(N2CCC(CNC(C3COC3)=O)C2)=O)cnc2ccccc12 c1(COCC)cccc(NCC)c1.N12CCC(CC1)NC(=O)C(=O)C1(CC1)C(=O)O2 Cn1nc(CO)c2c1CN(C(=O)OCC)CC2.c1(N2CCC(CO)C2)cccc(F)c1 N1(C(=O)CC2(CO)CCC2)CC2(CNC(C3CC3)=O)CC1CCO2.C12(C)CC(C1)C2 C1(C2CCCOC2)(NC(C(Cc2cn[nH]c2)NC(c2c(C)snn2)=O)=O)CC1 N1(C(c2nc(C)c(Br)cc2)=O)CCC2CCN(C(C3(CC4CC4)CC3)=O)CC12 N1(C(CCC)=O)CCOC2(CCC(NC(=O)C(C)(C)CC(C)(C)C)CC2)C1 c1(C(C)C)ccc(OCC(N2CCC(CNC(C3CC3C3CCC3)=O)C2)=O)cc1 COn1cnc(C)c1C(=O)NC1CC(CCNC(C2OCC3CCCC23)=O)C1 c1(C(N2CC(F)CC(NC(c3c(C)nsc3)=O)C2)=O)ccn2ncccc12 Cc1cc(C(=O)NC2CN(C(C3(c4ncccc4F)CC3)=O)CC2C)ncc1Cl CCC(C(=O)NCC#CC(=O)NC1CCCCN(C)C1=O)C(F)(F)F C1(C(=O)NC(CNC(c2c(COC)cco2)=O)C(C)(C)C)CCC(C)=C(C)C1 c1(N)cc(C)ccc1.C1(SC)CN(Cc2ccccc2)CC1N(C)C C1(NC(CCCC)=O)CCOCC1C(=O)NCC(N1CC=CC1)=O c1(N(C(=O)CN2CCCC2C)CCC)ccc(F)c(F)c1 CC1CN(C(c2nnc(S)n2C)=O)CCCN1C(=O)CCc1nc(C2CC2)no1 c1(C(N2CC3N(C(c4cccc(OC)c4Cl)=O)C(C3)C2)=O)nc2cccnc2s1 Cc1cc(F)c(C(N2CC(c3cn(Cc4ccc(Cl)cn4)nn3)C2)=O)c(Br)c1 Cc1ccoc1C(=O)NCC(=O)NC1C=CCC1 c1(C(=O)NCC(CO)NC(c2cnc(O)c(Br)c2)=O)ccc2c(c1)CCC2=O N1(C(CCS(N)(=O)=O)=O)CC2CCCC2(NC(=O)Cc2cc(C3CC3)no2)C1 c1(C(=O)NCC(C)N(C(CCC(CC)C)=O)C)ccc2nc(C(F)F)[nH]c2c1 C1(NC(C(c2c(OC)cccc2)=O)=O)CCCN(C(c2cc[nH]n2)=O)CC1 CC(C)(CNC(C1CC12CCN(C(C1C=CC=CC=C1)=O)C2)=O)C(F)(F)F N1(C(CC(C)C(C)(C)C)=O)CCn2c(CNC(=O)C=CC=C(Cl)Cl)nnc2C1 CSC=CC(=O)N1CCCC1CN(C(=O)C=CSCC(F)(F)F)C C1(C(=O)NC(c2ccc(C)cc2)C)C2CCC(C2)N1C(c1ccc(F)c(Br)c1)=O CS(=O)CCC(=O)NC1CC2(C1)CC2NC(C1(CF)CC1)=O C(=O)(CCS(C)(=O)=O)N.CC(C(=O)NCCC)C(F)F C1(C(=O)NCC2(NC(C3CC3F)=O)CCCCC2)C2CCC3C(C2)CC13 C(=O)(C(F)(F)CO)NCC(C)CN(C)C(c1c[nH]c(C(N)=O)c1)=O c1(C(N2CC(N(C)C)C(O)C2)C(=O)NC(C)C)nn(C)nc1Br.C(C)(C)(C)SC c1(C(=O)NCC(C)=CC(=O)NCc2cccc(CO)c2)c[nH]nc1[N+](=O)[O-] c1(C(N2CCC(CCNC(C(C)OCC(C)C)=O)C2)=O)ccn2ccccc12 c1(C(N2CCC(NC(COCCOC)=O)(CO)C2)=O)cn2cccnc2n1 N1(C(c2cccc(CS(C)=O)c2)=O)CCC(NC(=O)CC2CC3(CC3)C2)C12CC2 N1(C(C=CC=CC)=O)CCCCC(CNC(c2nc(C)ccc2CC)=O)C1 N1(C(CCC)=O)CCN(C(c2cc(C)cc(O)n2)=O)C(CO)C1 C(=O)(CCCn1ccnc1)N(CCN(C(=O)CCn1ccccc1=O)C(C)C)C C1(C#N)(CCC(=O)NCC(CC)NC(=O)CN(C)CC)CCC1 C1(O)(CNC(C2N(CC)CCC2)=O)CCCN(C(=O)CCC(F)F)C1 c1(NCCCN(C2CCCO2)C)ccc(S(=O)(=O)N2CCCC2CO)cc1Cl C(C1CCOC1)=CC(=O)N(CCN(C(=O)CCC1CCC1)C)C c1(C(=O)NCC(CNC(CNC(CN(C)C)=O)=O)F)cnc(P(C)(C)=O)cn1 c1(C(N(C2CCCN(C(C3C4CC5C(C4)C35)=O)C2)C)=O)c[nH]c(=O)cn1 C(CCN=c1ccn2c(Br)cnc2[nH]1)SCCNC(=O)CC1(C(F)(F)F)CC1 C1(NC(C(CCC)NC(C)=O)=O)Cc2ccccc2C1NC(=O)C=CC(F)(F)F c1(OCC)ccc(CC(=O)NC2CC2NC(c2cnn(CCF)c2)=O)cn1 N1(C(Cc2c(C)non2)=O)CCC(C(=O)N(C2CCCC2)CC(C)C)C12CCC2 c1(C(C(=O)NC2(C)CC2)N(C2(N(C)C)CC2)C)ccc(Cl)cc1OC(C)(C)C c1(C(N2CC(C)(C)C(CNC(=O)C(O)C(F)(F)F)C2)=O)cc(C#N)c(O)nc1N C1(C2CCN(C(=O)Cc3cccnc3O)CC2)(NC(C=COCC)=O)CCC1 CC1CC(NC(=O)CCC(=O)c2ccc(N)cc2)CN1C(=O)Cc1cncn1C c1(C(N2CCC(NC(CNC(CC)=O)=O)C2)=O)cnc(S)n1C N1(C(C2CC(N(C)C)C2)=O)CCC2(CC1)CC(NC(=O)CC(O)C1CC1)C2 C12(C(=O)NCC3C(NC(C4C(C)(C(C)C)C4)=O)COC3)CC(C#N)(C1)C2 C1(C(N2CC(CN(C(C(C)CO)=O)C)OCC2)=O)CCC2(CCCCC2)CC1 c1(C(=O)NC2CC2C(=O)NCCc2ccc(Br)cc2)c[nH]c2cccc(Br)c12 CC(C)C(C(C)NC(=O)Cc1n[nH]cc1Br)NC(=O)C=Cc1ccccc1 CC1(C)COCC1CC(N1CCCCC1CCNC(c1ccc[nH]1)=O)=O CCS(=O)(=O)c1ccc(C(=O)N=c2ccn(-c3ncccc3F)[nH]2)c(N)c1 Cc1ncc(C(=O)NCC2CCN(C(=O)CN3CCCCCC3)CC2)c(=N)[nH]1 C(CN=[N+]=[N-])(C(=O)NCCC1CCCC1(C)O)NC(c1ncc(OC)nc1)=O S(=O)(=O)(c1cccc(Cl)c1Cl)NC1CCN(Cc2ccccc2C(=O)OCC)C1 CC(C)(CNC(C1(C(C)(F)F)CCC1)=O)CC1CN(C(C2CNC(=O)N2)=O)C1 C=CCC(C)(C)CC(=O)NC12CCC(CC1NC(=O)C(=O)NCC)C2 C1(CSC)CC(C)CCN1C(c1cn(-c2ccc(Cl)cc2)nc1C)=O C1(C(=O)NC2C(C)CN(C(=O)C=C3CCCCC3)C2)CCCC(F)(F)C1 C(CCCCCC(=O)NCCSC)NC(C(CC)(C)C#N)=O C12(CNC(CC(C(C)C)(F)F)=O)CCCCC1N(C(=O)CSC(F)F)CC2 N1(C(c2cccc(F)c2)=O)CCN(C(C23CCCN(CC2)C3)=O)C2(CCC2)C1 C=CC1CC(N=c2ccc3c([nH]2)CCC3=O)CCO1 c1(CN2CC3(C(C(=O)Nc4c(C(N)=O)ccc(Cl)c4)C3)C2)ccc2occc2c1 C12(NC(c3cc(Cl)ns3)=O)CCCC1CN(C(=O)CCOc1ccc(F)cc1)C2 c1(NC(CCCC)CO)nccc(=NCCN(CCO)Cc2ccccc2)[nH]1 c1(NC(c2ccc(-c3cccnc3N3CCC3)o2)=O)ccc2c(c1)CCCN2 CC(C)(C)C(CNC(c1ccc(N)cn1)=O)C(=O)NCC(O)C1(Cl)CC1 C1(C(N(C(C)CNC(c2cc(O)cc(=O)o2)=O)C)=O)C2CCC1(C)C2(C)C C1(C(C)NC(c2c(OC)nsc2)=O)CCCN(C(=O)CC2CC(C3CC3)C2)C1 N1(C(COCCN(C)C)=O)CCC(C2CCC2)(CNC(=O)C(F)C(F)(F)F)CC1 c1(OC)ccc2[nH]c(=NCCCN(C)C)[nH]c(=NCCCN(C)C3CC3)c2c1 c1(CNC(C2C(Cl)(C(=O)OC)C2)=O)ccccc1CN(C(=O)C(C)O)C CC(=O)C(C)CC(C)C(=O)N1CCC2CC2(C(=O)NC2CCCC2N=[N+]=[N-])CC1 C1(CNC(=O)CCn2cc(C3CCC3)nn2)CN(C(C2C3CCCC23)=O)CCO1 c1(C(N(CCNC(C2CCC(SCC)CC2)=O)C)=O)ccc2nnc(C)n2c1 C1(NC(CC2(C)CC2(Cl)Cl)=O)CCOCC1C(=O)Nc1cncc(Cl)n1 CN1CCOC(C(=O)NC2CC3C2CCN3C(=O)CCc2csc(=N)[nH]2)C1=O Cc1nn(C)c(C(=O)NC2CCN(C(C3CCN3S(C)(=O)=O)=O)C2)c1Br CCCC(C)(O)CC(=O)NC(C(=O)NC1CN(C)CC1(F)F)C(C)C c1(CC(N2CCN(C(C(C)=C3CCC3)=O)C3C2C3)=O)cn2c(C)csc2n1 C1(C(N(CCCCN(C(=O)C=CC(C)(C)C)C)C)=O)CCCC(=O)O1 N1(C(C(C)N(CC)CC)=O)C2CCC(C2)C1C(=O)NCC1C2(CC2)C12CC2 CN1CCCC(C(=O)NC2(CCCNC(=O)C(O)C3CC3)CC2)C1 c1(C(=O)NCC2CCCN2C(C2(n3cc(Cl)cn3)CC2)=O)cccc(C2CC2)c1 N1(C(Cc2c(C)cco2)=O)CCOCC1CNC(=O)C(C)(C)OCC(F)(F)F c1(C(=O)NC2CC(C(=O)NCCC(=O)N(C)C)C2)cc2ccccn2n1 N1(Cc2cc(OCC)ns2)CCCC(C(=O)NCCC2CCCO2)CC1 N1(C(CC(C=C)CC)=O)CC2CC(C1)N(C(c1ccc(C3CCCCC3)s1)=O)C2 c1(OCC)cccc(C)c1C=CC(=O)NCC1CC(NC(c2cocc2C)=O)C1 O=C(N=c1[nH]c(Br)cnc1Br)C1CC1C(F)(F)F c1(OC)c(C2CCN(C(CC)C(=O)N(C)CC3CCOC3)CC2)ccnc1F CCCC(O)CC(=O)NCC1CCCN1C(=O)C=Cc1cncn1C C(=O)(C(F)C(C)(C)O)NCC(C)N(C(COCc1cc(OC)ncc1)=O)C c1(NCCCc2c(C)cccc2)nc(=NCCc2ccc(Br)s2)[nH]c2c1COC2 c1(OC)ccc2c(c1)C(C(=O)NCCN(C(=O)CN1CCOC1=O)C)CCC2 c1(CCCC)ccc(CC(=O)NC(CNC(C2CC2C)=O)C(C)C)cc1 c1(C(=O)NC2C(CC)CN(C(=O)COC3COC3)CC2)cn2cccc(C)c2n1 c1(C(N(CCNC(=O)Nc2ncn(C(C)C)n2)C2CC2)=O)c(F)cc(F)cc1F C1(CNC(c2cnn(C)n2)=O)CCCCC1NC(=O)COc1ccsc1 Cc1c(CC(=O)NC2CCNC(C)(C)C2)cccc1Cl Cc1ccc(CNC(C2CC3CC3N2Cc2cnc(C)nc2)=O)c(C)c1 C1(C(=O)NCC2(NC(CC(C)(F)F)=O)CCCC2)CCn2c(cnc2Br)C1 C12(CNCC3(O)CN(C(CCCN(C)C)=O)C3)CCC(CO)(CC1)CC2 Cc1ccc(C(=O)NCC=CCNC(C23CC(C2)C(c2ccccc2)O3)=O)cc1F N1(C(C(C)n2cccn2)=O)CCN(C(=O)CCCCC2CC2)CC1CCN(C)C C1(C(N2CCC(N3CC(O)C3)C2)=O)CN(C(C2(CO)CC2)=O)CCO1 C1(C(N(CCC)CC)=O)CCC2CCC1N2C(c1cc(Cl)n[nH]1)=O CCCC(F)(F)C(=O)NCC1CC(F)(CNC(=O)C(C)CC2CC2)C1 CCCC(C(=O)OC)C(=O)N1C2CCC(C(=O)NN3CC4C(C)C4C3)C1CC2.O N1(C(c2ccc(O)nc2Cl)=O)CCOC(C)(CNCc2c(OCC)cccc2)C1 Cc1ccc2c(c1)CC(C)N(CC(=O)Cc1cccc(Cl)c1)C2 c1(C(=O)NCC2CCC(F)(CNC(C(CC)O)=O)CC2)ccc2c(c1)NC(=O)C2 N1(C(COC(C)=O)=O)CC(NC(=O)CC2(CSC)CC2)C(c2nccn2C)C1 C=CCCCC(C)(C)C(=O)N1CC2CC1C2NC(c1cc(C)ccc1C)=O c1(C(=O)NCC2CCCCN(C(C(COC)O)=O)C2)c(F)cccc1[N+](=O)[O-] Cc1nc(C(C)C)ccc1C(N1CCOC(Cn2cc(-c3cn[nH]c3)nn2)C1)=O C1(CC(=O)NCC2CC(NC(C3CC4(CC4)C3)=O)C2)Oc2ccccc2NC1=O N1(C(c2ccoc2C(C)C)=O)CCCCC1C1CC1.CC1=CC(=O)NC1 C1(C(=O)NCC2N(C(COCC(C)C)=O)CC3(CC3)C2)CC2(C1)CC1(CC1)C2 c1(C(N2CC(CNC(COC(CC)C)=O)OCC2)=O)cc(N)c(F)cc1C Cc1ccc(-c2cn(CCCONCCC3CCc4ccccc43)nn2)c(C)c1 C1(NC(=O)Cn2cc(I)nn2)C2CN(C(c3cnccc3N(C)C)=O)CC12 c1(C(N2CC(NC(C3CCC(=O)N3)=O)CC(C)C2)=O)ccc(=O)n2c1COCC2 CC1(C(N2CCN(C(c3cnc(N)c(O)c3)=O)C(CO)C2)=O)CCS(=O)(=O)CC1 c1(NC)cnc(C(=O)NCCCCCNC(=O)CSCCN(C)C)cn1 c1(C(=O)NCC(C2CC2)NC(C(C)OC(F)(F)C(F)(F)F)=O)cnc2n1CCS2 N1(CC(C2CC2)OCC)CCC(NC(c2cc(C)ccc2F)=O)C(C)(C)C1 N12CC(F)(F)CC1(C)NC2=O.c1(SC)nc(C(=O)OC)cc(C(F)F)n1 N1(C(C2CN(C(CC(COC)C)=O)CC2C2CC2)=O)CCc2c(F)cccc21 C1(C(N2CC(NC(c3c(C)cno3)=O)C(C)C2)=O)C2CCCCCC12 CC1(C(=O)NCC2=NOCC2)CCCC1O.C12CCCC(C1)C(=O)N2CCO C(=O)(CC1=NNC(=O)C1)N(C)CC1COCCN1C(=O)C(F)C(C)(C)O Cc1ccc(F)c2c1CCN(Cc1cc(Cl)c3ncccc3c1)C2 C(C)(CCC(=O)NC1(c2ccnn2C)CC1)N(C(C1C(C(=O)OCC)C1)=O)CC N1(C(c2cc(C)[nH]c2)=O)C2CN(C(c3cc(Cl)sc3Cl)=O)CC12 N1(C(C=CC)=O)CCN(C(=O)CCc2ccc(O)cc2)C(C)C1 N1(C(CNC(C)=O)=O)CCC(C2CCCN2C(=O)Cc2n[nH]cc2Br)CC1 CC(C)C(C(=O)OC(C)(C)C)C(=O)N(CC(N1CCS(=O)(=O)CC1)O)CCO N1(C(C=CC(C)NC(CC(CC)OC)=O)=O)CC(C)C(F)(F)C1 c1(CC(CO)OC(=O)NC2CC2)ccccc1 C1(C)(C(=O)NC(C)CC2CCN(C(=O)CCCF)CC2)CCC(F)(F)C1 c1(SC)ccc(CCCC(=O)NC2CN(C(c3cncc(C4CC4)c3)=O)C2)cc1 CCCCCS(=O)(=O)CC(=O)NC1CCC12CN(C(=O)C(c1cccnc1)O)C2 C1(CC(=O)NCCCN(C(C2CCCN2C(C)=O)=O)CC)CCCS1(=O)=O CN1CC(C(N2CC(N3CCCC3)C2)=O)CC1=O.C1C(=O)N1CCO N1(C(=O)OC(C)(C)C)CCOC(C)(C)C1C(=O)NCC(F)(F)Cl C#CCCCC(C)(c1nnnn1Cc1nnn(C)n1)NC(C1(CO)CC1)C CCC(C)C(C)C(=O)NC1(C(=O)O)CC(F)(F)C1 C1(C(N(CCN(C(=O)CC=C(Cl)Cl)C(C)C)C)=O)CC2(CO1)CC(F)(F)C2 c1(C(N(C(C)C(=O)NCC2CC=CC2)CC)=O)n[nH]c2c1CCC2 N(C1CCc2c1ccc(F)c2Br)C1CC(CCC)OCC1 Cc1ccc(=NCCC(=O)NC2CN(C(c3ccc(Cl)[nH]3)=O)CC2C)[nH]c1 C1(C(=O)NC(c2nc(C(C)(C)C)no2)C)(COC)CCCO1 c1(C(=O)OCC)c(N(CC(C)NC(=O)CCF)C)nnc2c1COCC2 c1(C(=O)NCCn2cc(COc3ccc(F)cc3)nn2)[nH]nc2ncccc12 c1(C(N2C(CNC(C=Cc3occ(C)n3)=O)CC2)=O)noc2c1CC(F)(F)CC2 c1(C(=O)NCCC2CC(NC(c3cc(C)oc3C)=O)C2)coc2c1COC2 CN1CCN(c2cccc(C(=O)NC3(C)CN(C(C4CCCS4)=O)C3)n2)CC1 N1(C(=O)Cc2cscn2)CCCC1C1CCCCN1C(=O)CN1CCSCC1 N1(C(CN(CCC)C)=O)CC2(CC1CNC(C1(COC)CC1)=O)CC2(F)F C1(CCc2cn(CC(=O)OC)nn2)CCN(C(C2CCC(C)CC2)=O)CC1 CC(CS(C)(=O)=O)C(=O)Nc1ncc2ncnc-2[nH]1 C1(N(C(c2cc(OC)no2)=O)C)CN(C(c2c[nH]c(=N)o2)=O)CCC1C C1(CC(=O)NC(CC(C)C)(C)CNC(=O)CC(F)F)Cc2ccccc2O1 N1(C(C2CCN(CC)C2)=O)CCN(CC2CN(C(=O)CC#N)C2)CC1 c1(CC(=O)NC(CCCCNC(c2c(C)cco2)=O)C)cccc2nsnc12 c1(C(=O)NC(C(N2CCCC(CC=C)C2)=O)C2CCC2)cc(F)cc(F)c1 N1(C(=O)CC2CCCCC2O)CC2CC(C1)N2C(c1n[nH]cc1Cl)=O Cc1cc(CNC(C2C(CNC(=O)CCCC3CC3C)C2(C)C)=O)cc(C)n1 N1(C(C(CCC(N)=O)n2cc(C(C)(C)CO)nn2)=O)CC(=O)N2CCCCC2C1 c1(C(=O)NCC2C(NC(c3c(CC)cno3)=O)CCCC2)cc2ncccc2s1 C(C(C)(C(=O)NCC1(O)CN(C(c2ccc(C3CCOC3)cc2)=O)C1)OC)OC c1(NCCCCNC(=O)CSC2CC2)c([N+](=O)[O-])cnc2c(F)c(F)ccc12 C1(NCC(=O)NC(C)C)CCN(CC(F)(F)F)C1=O c1(CC(C(C)C)NC(=O)NOCc2ccccc2)ccc(Cl)cc1 C1(N(C(C(C2CCCC2)OC)=O)C)CCN(C(=O)CCn2cccn2)CC12CC2 c1(OC)ccc2[nH]c(C)c(C(=O)N(c3cccc(NC(C)=O)c3F)C)c2c1 CC(C)C(C(=O)N(C1C2CNC1C2)C1CC1)n1nccc1-c1cccc(F)c1 C1(C(C)C)CN(C(=O)CCc2ccc(Cl)cc2Cl)CCN1C(=O)CCCF c1(C(N2CCC(OC(C)=O)C2)=O)nn(-c2ccccc2)c(=O)cc1O c1(C(=O)NCC2C(NC(Cn3c(C(C)C)nnn3)=O)CC2)ccc(N)c(Cl)n1 C1(C)(C(=O)NC(c2ccccc2)C)CN(C(c2cc[nH]c2)=O)C1 Cc1c(C(N2CC=C(CNC(=O)CC3CNC(=O)C3)CC2)=O)sc2nnc(S)n12 c1(C(N(C(CNC(CCC=CC)=O)C)CC)=O)cncc(N(C)C)c1 n1(CC(C)O)cc(C(=O)NCC(C)(C)NC(c2cc(CCO)on2)=O)ccc1=O N1(C(CC2(C)CCCO2)=O)CCC2CCC(C1)N2C(C1CC2CCCCN2C1)=O c1(C(=O)NCC(C)N(C(c2cscc2C(N)=O)=O)CC)c(C(F)F)cnn1C C1(CC(=O)NCCC(C)(C)O)CC(F)CN1C(C1C(C#N)C1(C)C)=O C1(CNC(C(c2cnn(C)c2)NC(CNC(=O)NC)=O)=O)CC12CCC2 N1(C(c2cc(CC)on2)=O)CCC(N(C(=O)CSCC(F)(F)F)CCO)CC1 N1(C(C(CC#C)O)=O)CCC2(CC1)CCN(C(=O)Cc1sc(O)nc1O)C2 N1(C(c2c(Cl)c(C)n(C)n2)=O)CC2=C(C1)CN(C(=O)C(C1CCCCC1)N(C)C)C2 c1(C(N2C(C)(C(=O)NCc3cc(C4CC4)no3)C=CC2)=O)c[nH]c2cccnc12 c1(C(N(CCC(=O)N(C(C#C)CC2CC2)C)C)=O)cnsc1C C1(CNC(COCCC#C)=O)CCC(NC(C2(C(O)C(F)(F)F)CCC2)=O)CC1 CC#CC1CCN(C(=O)C(c2cnn(C)c2)NC(=O)C(O)C(C)C)C1 N1(C(CCNC(C(C(c2ccccc2)C)O)=O)=O)c2ccccc2CCC1C C1(NC(C(F)=CC)=O)CC12CCN(C(=O)CC1OCCCC1(C)C)CC2 c1(C(=O)NCCN(C(CCSCCC)=O)CC(C)O)cnc2c(c1)N(C)CCO2 c1(C(C)(C)NC(=O)NC(CCOC)COC)cc(Br)ccc1C c1(NCCN(C)Cc2ccc(C)cc2)sc2nccnc2c1N C#CCCCCC(=O)N(C)Cc1ccc(CNC(=O)CC(C)(C)C)cc1 c1(C(=O)OC)c[nH]c2c(OC)nc(NC(C3CC4CCC3O4)=O)cc12 C1(C(=O)NCC(=O)OCC(C)(C2CC2)OC)CCCN1S(C)(=O)=O C=C1CCN(C(=O)CCOCCCNC(c2nc(Cl)cs2)=O)CC1 c1(OC)cc(CNCC2CCC3C2C3(F)F)c(N)c(C)c1.c1(C)cn(C2CC2)nn1.O C1(C(C)C)CCC(NC(=O)CC2CC(C)N(C(c3cnns3)=O)C2)CC1 C1(CC)OCCCC1C(=O)N(C)CC1(NC(=O)COCc2ccccc2F)CC1 C1(C(=O)NC2C3CN(C(Cc4c(C)nc(C)[nH]4)=O)CC2C3)CCC2(CCCC2)CC1 c1(C(=O)NOCCCO)ccc(Br)c(Cl)c1F.c12cn(nn1)C1COCC1C2 C1(NC(C2CC(NC(C)=O)C2)=O)CC2CCC1CC2NC(C(C)(C)OC(C)=O)=O C1(N(C(CN(C2CCCC2)C)=O)C)CCN(C(c2cnn(CCO)c2)=O)C1 N1(C(C2CCC(C)CC2)=O)CCCCC2(C1)CN(C(=O)CCc1csnn1)C2 c1(C(=O)NC2CCN(C(COC(CC)(C)C)=O)CC2F)ccc2snnc2c1 c1(C(=O)NC2(c3n(C)cnc3)CC2)ccc(C#N)cn1.C12OCCC1NC2=O CC(C)(C)CCC(CO)OC(=O)CCNS(C)(=O)=O N1(C(c2c(C)sc(Cl)n2)=O)CCN(C(=O)CN(C)C)C2COCC12 CCC(C)CCCCC(=O)N1CCC(N(C)C(C23CC(C(F)(F)F)(CO2)C3)=O)C1 Cc1nc2cccnn2c1C(=O)N(C(C)CCNC(=O)CCC(C)CC(C)C)C C(=O)(C(CC(C)C)C(C)C)NCC1(O)CN(C(CC2(COCC)CC2)=O)C1 O=C1Nc2cc(Cl)c(Br)cc2C1CCl.c12cc(F)ccc1C1CCCN21 N(C1CCCc2cn(C3CC3)nc21)C(C(N1C(C(C)C)C(C)CCC1)=O)=O c1(C(N2C(C(NOCCOC)=O)C(C)(C)C2)=O)cc(O)cc(=O)o1 n1(CCC)nc(CCc2ccccc2)nc1-c1cn(C2CCOCC2)nn1 c1(C(=O)NC(C)CCCNC(c2csc(C3CC3)n2)=O)coc2ccccc12 C1(C)(CCNC(C(CSC)OC)=O)CCN(C(=O)CCc2cnn(C)c2)C1 C(C(C)C)(C(O)C(=O)N1CCC1Cn1cc(CCCC(C)O)nn1)OC Cc1sc(C(=O)N(CCNC(C2CC(F)(c3ccccc3)C2)=O)C(C)C)nc1O c1(OC)cccc(C(C(=O)Nc2ncccc2OC)N(C)CC2CCCO2)c1 C(N=c1nc(-c2ccccc2)[nH]c(=NCc2cc[nH]n2)[nH]1)c1cncc(CC)c1 N1(C(CCC2N(C)CCC2)=O)CCCCC(NC(=O)CC2CCCS(=O)(=O)C2)C1 N1(C(c2n(CCC)ccc2)=O)CCN(C(c2oc(C)cc2C)=O)C(CCC)C1 C1(C(N2CCC(CCNC(c3n[nH]c(C)c3F)=O)C2)=O)CC2(CCCC2)C1 C=CCN(OC)C(=O)C(C1CCCC1)NC(=O)Cc1cccnc1C Cc1cc2[nH]c(C(N3CCCC(N(CCO)C(C4CC(N(C)C)C4)=O)C3)=O)cc2o1 C1(NC(c2cc(C)oc2C)=O)CCC2CCN(C(=O)CC3CCC(=O)N3C)C1C2 c1(C(=O)NC(CC=C)CNC(=O)C=Cc2ccc(C)o2)c(C)cccc1F N1(C(CCCC(C)=O)=O)CCCC2(NC(=O)CC(O)C3CC3)CCCC12 C=Cc1ccc(C(=O)NCC2(F)CCN(C(c3cccnc3S)=O)CC2)cc1 Cc1ccc(CN2CCCC(C)(C(=O)Nc3ccnnc3C)C2)c(F)c1 C=C=CC(C)C(=O)N1CC(N(C)C)(CNC(C2CC3(CC3)CO2)=O)C1 c1(C(N(C2CCN(C(CSCC#C)=O)CC23CC3)C)=O)cc(F)c(F)c(Cl)c1F c1(C(=O)NCC2(O)CN(C(C3(CC4CC4)CCCCC3)=O)C2)cc(F)cc(N)c1F C1(CC(=O)NC2COCC2NC(C2(CF)CCC2)=O)CC2CC2C1 N1(C(c2cc(C)n(C)n2)=O)CC(NC(=O)CCCN(C)N=O)C2CCCC12 c1(C(=O)NC2C3CN(C(C4CN(C(C)=O)C4)=O)CC32)ccc2c(c1)CN(C)CC2 N1(C(c2nc(CC(C)C)sc2)=O)CC2C(CNC(C3(CCF)CC3)=O)C2C1 C(C(=O)N(C)CC1(CNC(=O)COc2ccsc2Cl)CC1)(C(C)C)SC C1(C(=O)OCC)C2CN(C(=O)NC3CCN(CC#N)C3)CC12 C1(NC(c2n(CC)ncc2)=O)(CO)CCCN(C(c2csnc2Cl)=O)C1 C1(NC(C(C(C)(C)C)O)=O)CCC2CCN(C(c3cnc4ccnn4c3)=O)C1C2 N1(C(CC2CC(C)(C)C2)=O)CCOC(CNC(C2CCC2(C)C)=O)C1 c1(C(=O)OC)cccc(CNC(=O)N(C2(C(C)C)CCC2)C)c1F C1(NC(CC2(COC)CC2)=O)CCC12CCN(C(=O)CC1CCCOC1)CC2 C(=O)(C1CC=Cc2ccccc21)NCCC(C)N(C)C(C1CC(F)C1)=O CCCC(C(=O)N1CC(C(=O)OC)CC1C)C(C)C.c12nc(cc(C)n1)CN2 C(C(CC(C)C)NC(c1scnc1C1CCCC1)=O)NC(C(C)=C1CCC1)=O c1(C(N2C(COC)CC(=C)C2)C)c(F)cc(F)cc1F C(=O)(C(O)CC(C)(C)C)N(CC(N1CCC(O)(CC=C)CC1)=O)C(C)C C1(C(=O)NC(CC(=O)OC)C)CCC(CNC(=O)C(F)n2cccn2)CC1 c1(NC(N(C(C)C2CC2)CC2CCCOCC2)=O)nn(C)cc1S(N)(=O)=O c1(OC)ccc(C(CNC(=O)C(=O)Nc2cscc2C(F)F)OC)cn1 C1(C(N2CCCC(CNC(=O)CN3CCOCC3=O)C2)=O)(COC)CCOCC1 c1(C(=O)NCCCN(C)C(C2CCCC(F)C2)=O)ccccc1OCCF N12CC3CC(CC1C3)Nc1nccc(n1)C2=O.C(=O)CCc1cncs1.CO N1(C(C(C)n2ccnc2)=O)CC2CCC2(NC(=O)Cc2ccc(CO)cc2)C1 CCCC(C)(CC)C(=O)NCCC1CC(C(N2CCOC(CCC)C2)=O)C1 c1(OC)ccc(C(O)C(=O)N(CCCCCNC(c2ccoc2)=O)C)cc1 C(=O)(C(C)C(O)CC(C)C)N1CC(n2cc(CNC(C3=C(C)CCOC3)=O)nn2)C1 C1(C)(C(=O)NCC(C)CNC(C2C3CC4C(C3=O)C24)=O)CCC(F)(F)CC1 c1(C(=O)NC2C(OC)CN(C(=O)C(C)(O)C3CC3)C2)nccn2nccc12 c1(OC)cc(C(=O)NC2CN(C(=O)Cn3ccc(O)nc3=O)CC2F)cc(F)c1 C1(OC)CN(C(=O)C(C)C2(O)CCC2)CC1C(N)=O.C12(CCC1)C(=O)NC2 Cc1c(SC2CCCN(CC34CC(n5cc(C6CC6)nn5)C3C4)C2)cccc1F c1(SC)cc2c(NCc3conc3C(F)(F)F)nc(C)nc2s1 c1(OC(C)C)cccnc1C(=O)Nc1ncccc1-c1ccn(CCl)n1.C(C)C Cc1ccc(C#N)cc1C(=O)N(C(C)(C(=O)NC1CC(=O)N(C)C1)C1CC1)C C12(NC(c3cc4[nH]ccc4s3)=O)CCCN(C(=O)CSc3ccccc3)CC1C2 C(=O)(C1Cc2ccc(C)cc21)NCC1CCN(C(c2c(CC)cco2)=O)CC1 C(=O)(CC(C)(C)CNC(N)=O)NC(C1CCN(C(C2(SCC)CC2)=O)C1)C CC1CCC(C)(C(=O)NCC2CN(C(=O)CCc3ccc(F)cc3)CC2O)CC1 c1(C(C(=O)NCC(CNC(C=CCCC=C(C)C)=O)C)C)cccc(Br)c1 C1(C(N2CC3(CC(NC(C4=C(C)OCC4)=O)C3)C2)=O)CCc2ccccc2C1 S(=O)(=O)(c1ccc(Cl)c(C(C)NC(=O)CNc2ncc(C(F)(F)F)[nH]2)c1)NC c1(C(=O)NCCCC=C)ccccc1Cn1cc(C(C2CCOC2)C)nn1 C#CCC(CC(F)F)C(=O)NCCN(C)C(C1(n2cccc2)CCOCC1)=O N1(C(C)=O)C2CCCC1CN(C(C1CCCC1Nc1n[nH]cc1F)=O)C2 C1(CC(=O)NCCN(C)C2CC2)CCC(C(=O)NC2CC(O)C2)C1 c1(C(N(C2C(N(C(CCC(=C)Cl)=O)C)CCCC2)C)=O)cc2cccnc2cn1 C1(S(N)(=O)=O)(C(=O)NCCOCCCNC(c2c(C)cn(C)c2)=O)CCC1 C#CCCCC(C)C(=O)N(C(C)CNC(c1ccc(CO)s1)=O)C C#CCC(CC#C)NC(C1COCC1NC(=O)C(C)Cn1ccnc1)=O c1(CC)cccc(C(=O)NC2CC(C(N3CCC(C)(C(N)=O)C3)=O)C2)n1 Cc1ncc(C)c(N2CCCC(NC(C3CCCN3C(N)=O)=O)CC2)n1 c1(C(C(N2CC(O)(CCNC(C3C=CCCC3)=O)C2)=O)OC)ccccc1Cl N1(C(c2c(CC)csc2)=O)CCCC(C(=O)Nc2cnc(N(C)C)nc2)(CC)C1 c1(C2(CNC(=O)NC3CC(Cn4nccn4)C3(C)C)CC2)cc(Cl)ccc1F CCC(CC(F)(F)F)C(=O)NCC(C1CC1)N(C(=O)C=Cc1cc(OC)ns1)C C(=O)(C1=CCCCC1P(C)(C)=O)NCCCC(C)NC(CC(C(=O)OC)(C)C)=O CC1CN(C)CC(C(N2CC(F)(CNC(=O)Cc3ccnc(Cl)c3F)C2)=O)O1 C12CCCCN1S(=O)(=O)CCOC2=O.C(=O)(C(C#N)c1nccs1)OCC N1(C(C(CSC)C)=O)CC(O)CC1C(=O)NC1CC=CCC1C c1(C(C(=O)NCC(C)N(C(C(c2c(C)noc2C)CC)=O)C)C)ccccc1F C(=O)(C#CC(C)(C)CNC(C1(C)CCCCC1C)=O)NC(C#C)CC(C)C C1(O)(CNC(C2ON=C(C)C2)=O)CCN(C(=O)C(C)(C)C2CCOC2)CC1 c1(C(=O)NC2CC3(CN(C(=O)CSC4CCOC4)C3)C2)ccc2nc[nH]c2c1 C1(C(=O)NCC(CO)NC(=O)CCC2CCCC2)CCN(CC(F)F)CC1 C1(CC(=O)NC2(C)CC2)CCC(C)O1.C1(C(=O)OC)CC1C(=O)NCC1CC1 C1(NC(C(CC=C)C)=O)CC2CCC1CC2NC(=O)C(=Cc1cn[nH]c1)C C(=O)(CCCCC1CCCCC1)N(CCCCNC(=O)C(C)(C)c1cnc[nH]1)C CC1(C)CN(C(C2C=CC(NC(C3CCNC3=O)=O)C2)=O)CCC1CO C(=O)(CC(C)(C)NC(C1(C#N)CCOC1)=O)N(CCN(C)C(=O)C1CC1)C c1(C(N2CC(N3CCN(C(CCSC)=O)CC3)C2)=O)cc2n(n1)CC1(CC1)C2 CC1CCN(C(C2CC=CCC2)=O)CC1CNC(c1cc(Br)cs1)=O c1(C(=O)NC2(CC(=O)N(CC)CC3CCC3)CC2)ccc(COC)o1 Cc1cnc(N(CCNC(=O)Cc2cn(C)nn2)C2CC2)nc1O C1(CNC(C)=O)CN(C(c2ccnc3c2CCO3)=O)CCC12CCC2 N1(C(CN(CC)CC)=O)CCC2C(C(=O)NCc3ncccc3C)C2C1 C1(C(=O)NC(CC#CC)C)CC(O)CN1C(c1cccc(C(=O)C2CC2)c1)=O N1(C(C2(C)C=CCC2)=O)CC2CC(C(N3CCOC(CO)CC3)=O)(C2)C1 N1(C(c2nc(C)oc2C)=O)CCCC(NC(c2snnc2C2CC2)=O)C1C O=C(C#CC1CCC1)NCC1CC1NC(c1ccc(-c2cccs2)s1)=O CC1CCCN(C(=O)C(=O)NCC2CC3CC3N2C(=O)CCN2CCCC2)C1 c1(OC)cc(C(=O)NCC(C)NC(=O)CCC(C)O)ccn1 CC1CCC(C(=O)NCCC(C)O)N(C(C2CC23CC3)=O)C1 n1(CC(N2CCN(CC(O)CC(F)(F)F)CC2)=O)nc2n(c(=O)c1=O)CCC2 c1(C(=O)NCC(CN(C(C(C=C)(C)O)=O)C)(C)C)cc(S(=O)(=O)NC)ccc1C Cc1ccc(O)c(CNC(C2CC(C)N2C(C2CC(=C3CC3)C2)=O)=O)n1 N1(C(C2C(CC)C2)=O)CCC(F)(F)C(NCc2cccc(-c3ncco3)c2)C1 c1(CN2CC3CN(C(COC(CC)C)=O)CC32)ccc2ccccc2c1Br c1(C(N2C(C(=O)NCCc3cccc(OC)c3)CSCC2)=O)cc(O)nc(O)n1 n1(CC(=O)OC)ccc(CN2CCCC2c2cccnc2)n1 CC1CC(C2CN(C(=O)CCC3CCCO3)C2)=NO1.C1(=O)CC2CC2CCN1 c1(SC)cc(C(N2CCC(C)(NC(c3ccn(CC(C)C)n3)=O)C2)=O)c(C)o1 c1(C(N2CC(CNC(C(C(C)C)SC)=O)C2)=O)cccc2[nH]ncc12 C12(NC(=O)Cc3cnc(C4CC4)[nH]3)CCCC1N(C(c1cccc(O)c1)=O)CCC2 C(=O)(CCCCCCn1cc(CCCCO)nn1)NCN1C(C)CCCCC1 CCC(COC)(CC)C(=O)NC(C1(O)CN(C(=O)C(C2CCCO2)C2CC2)C1)C C1(C2CN(C(C3CSCN3C(N)=O)=O)C2)(NC(C2C(C)C2)=O)CC1.C1(=O)CN1 Cc1cccc(F)c1CC(=O)N(CC(C)NC(c1cc(C#N)cn1C)=O)C CN1CCCC(C)(C(N2CC(O)(CNC(C34CCC(CC3O)C4)=O)C2)=O)C1 c1(OC)ncc(C)cc1NC(C1CCN(C(=O)C(n2ccnc2C)C)C1C)=O C1(C(N2CC(CNC(c3c(C)cc[nH]3)=O)OCCC2)=O)Cc2cncn2C(=O)N1 C#CCCCCC(=O)NCc1ccc(CC(C)NC(c2[nH]nnc2C)=O)cc1 C1(NC(=O)C(C2(O)CCCC2)F)C2CN(C(c3ccc(C4CC4)cn3)=O)CC12 N(C)(C(=NCCC(C)=O)NCCN1CC23CCC2(COC3)C1)Cc1c(OC)nccc1 C1(C(=O)NCCN)(NS(C)(=O)=O)CCN(CCc2cc(Br)ncc2F)CC1 C(CC(C)C)(C(=O)NC1(CO)CCN(C(C2(C)CCN(C)CC2)=O)C1)OC CC1(C)OCCC1CC(N1CCCC1(C)C(=O)NC12CCC(CC1)C2)=O C(=O)(CCCC(C)(C)NC(=O)CN(C)C)NC1CCCC(C)C1 C(=O)(C1CCc2ccccc21)NC1CCCCN(Cc2cc(C)c(O)cc2)C1 Cc1ccn2ncc(C(=O)NC(C)CN(C)C(C3CCCCO3)=O)c2c1 C1(C(N2C(CCCNC(C3(CC)CCCCC3)=O)CCC2)=O)=CC2=NC=CS2=N1 Cc1cc(NC2CCC(NC(=O)Cc3csc(C)n3)CC2)n2ncc(C)c2n1 C1(NC(C(C)NC=O)=O)CN(C(=O)COc2ccccc2C#N)CC12CC2 N1(C(C(CC)N(CC)CC)=O)CCC2(CC1)CN(C(c1ccc(Cl)nc1)=O)C2 C(C(C)(C)CCNC(C1(NC(C2CCCCO2)=O)CCCCC1)=O)OC c1(C(=O)NC2C(NC(C3(COC)CC(=O)C3)=O)COCC2)ccc(O)cc1F c1(C(N(CCCC)OC2CCCC2)=O)cccc2c1CN(C1CC1)C2=O C(=O)(C(C)C(C)(C)C)NCC1(NC(CCc2onc(CC)n2)=O)CCOC1 S(=O)(=O)(c1c[nH]c(C(=O)NCC(CNC(C2CCCN2C)=O)OC)c1)NC C(CCC(C)C(=O)NC1(CCCNC(c2sccc2Cl)=O)CCCC1)OC C=C1c2ccccc2C(=O)N1CCNS(=O)(=O)c1cncc(CC)c1 n1(CC)ncnc1C(C)Nc1ccn(CNC(=O)C(F)(F)F)n1 N1(C(c2ccc(C)[nH]2)=O)CC(C)(C)CC1C(=O)NC12CC(F)(C1)C2 c1(C(=O)NCCOCCNC(=O)C(=O)NCCO)ccc2c(c1)COC2 N1(CCC(=O)N(C(CN(C(C(C)NC(N)=O)=O)C)C)C)CCC(O)CC1 Cc1ccc(O)c(C(=O)N(C(CC(C)C)C(=O)NC(C)Cn2ccnc2)C)c1 C1(C(=O)NCC(=O)OC)(C(=O)N(C)CCN(C)C(C2CCCS2)=O)CCCC1 C1(NC(C(C)OC)=O)C2CC1N(C(=O)CCCc1ccc(C)cc1)C2C C1(CC(=O)NCC(C(=O)NCC(CC)N(C)C)O)COCCOC1 N1(C(C(C=C)(C)C)=O)CCC(F)(F)C(C(=O)NCC2CC(F)(F)C2)C1 c1(CC)ccsc1C(=O)NC(C1CC(NC(=O)C(CC2CC2)OC)C1)C c1(C(N2C(CNC(c3c(C)n[nH]c3)=O)C=CC2)=O)ccc(O)nc1 c1(OCCNC(c2ccc(C(F)(F)F)nc2)=O)ccc(CNc2nc[nH]n2)cc1 N1(C(=O)OC(C)(C)C)CC(C(=O)O)CC12CCCOC2.c12cnc(nc1)NC2 C=C1CC2(C1)CC(C(=O)NCCc1ccc(C)s1)C2 C1(CNC(C2(c3c(C)cccc3)CC2)=O)CN(CC2(N(C)C)CC2)C(C)(C)C1 C(C)(COCc1cnc(OCc2ccccc2)nc1)(C(F)(F)F)NC1C(C)C1 N1(C(C(P(C)(C)=O)O)=O)CCOC2(C1)CN(C(C1CCC13CCC3)=O)C2 c1(C(N2C(CC(=O)Nc3scc(C)n3)CCC2)=O)cc(C(=O)O)cc(N)c1 C(=O)(C1CCc2ccccc21)N1CC2(OCC(NC(C3CNC(=O)N3)=O)C2)C1 N1(C(c2n(CC#C)ccc2)=O)CCCN(C(=O)C(F)CN(CC)CC)CC1 CCC(C)CCC(=O)N1CCOCC1CNC(=O)C(F)(F)c1nccs1 N1(C(C(C)(C)OC)=O)CCC(NC(=O)CC2CCCS2)C(CO)C1 C=C(C)CC(C)C(=O)NC1CCC(F)(CNC(=O)CCCCc2ccccc2)C1 C(CC(C)C)(C(=O)NC12CCC1CN(C(=O)C(=O)Nc1cccnc1)C2)NC C12(NC(CCCC)=O)CCC(F)(F)CC1CN(C(C1(C)CC=CCC1)=O)C2 C(=O)(C(O)P(C)(C)=O)NC(CC)CNC(c1cc(C2(C)CC2)n[nH]1)=O C1(C(N(CCOC)CCNC(c2cn(C3CC3)nn2)=O)=O)CCC=CCCC1 C12CCN(S(=O)(=O)NCCS(=O)(C(C)(C)C3CC3)=NC1=O)C2.C(C)(C)(C)OC(=O)O.O O=C1CCN(Cc2ccc(Br)cc2F)C(=O)N1CC1CC(n2cncn2)C1 c1(N2C(=O)CC(C(N(CC)Cc3cccc(Cl)c3)=O)C2)ccc2ncccc2c1 C1(CCO)(CNC(c2nnnn2CC2CC2)CC2CC2)CCCC1 Cc1nc(C(N2CC=CC(C(=O)NOC(c3ccncc3)C)C2)=O)sc1C C=CCCC(C(=O)N(CCNC(=O)CC1CSC1)C(C)C)c1ccccc1 C1(NC(C2CCSC2)=O)CCCCN(C(C2CCNC2=O)=O)C1 N1(C(C(c2ccccc2)OC)=O)CC2(C1)CN(C(c1cscc1F)=O)CC2CO c1(C(=O)NC(C)C2CC2)cncc(OCC(F)F)c1 N1(C(c2c(Br)cn(C)n2)=O)CCC(CO)C(NC(=O)C(F)=CC2CC2)C1 N1(C(COC)=O)CC2(CCCN(C(c3cccc(N4CCCC4=O)c3)=O)C2)C1 c1(OCC)nc(C(=O)NCC2CCC(NC(C3CC(C)(C)O3)=O)C2)ns1 C(CCCCCCNC(=O)COC1CCN(C)CC1)n1cc(C(C)O)nn1 C1(C(NOCCC#C)=O)CCN(C(=O)C(N2CCOC2=O)C)C1C(C)C CC(CN)S(=O)(=O)c1ccc(F)c(C(N2CCC(C)(O)C2)=O)c1 c1(OC)c(C(N2CCCOC(CNC(C3C=C3C)=O)C2)=O)cccc1[N+](=O)[O-] C1(C(=O)NC2CN(C(CSC(C)C)=O)CC2CO)CCCCC1(C)C c1(CC(C)Nc2c(C)nn(CC)c2C)c[nH]c2cccc(Br)c12 c1(C(=O)NC2CC(C(C(=O)N(CCN(C(C)=O)C)C)F)C2)cc(N)cc(F)c1 CN1CCN(c2cc(NC(C)(CNC(=O)OC(C)(C)C)CO)[nH]n2)CC1(C)C C=C(C)CCC(=O)N1CC(O)(C2CCCN2C(=O)C(C)CC)C1.C(=O)(CCCCCCN)O c1(NC(C(c2ccc(Br)cc2F)(C)C)=O)cccc(S(C)(=N)=O)c1 c1(C(=O)NCC2(CNC(c3n(CC)ncn3)=O)CCCC2)ncccc1CO C1(C(N(CC#C)C(C)C)=O)CN(C(C2CCSC2)=O)CC1CCC N1(C(N2CCC(CC(=O)O)(C(=O)NCC)C2)=O)CC(OC(C)(C)C)CC1(C)C n1(CC)nc(CNc2csnc2C2CC2)c(Br)n1 C1(=CC(=O)NCC2CN(C(=O)Cc3cc(CF)on3)C2)C2CC3CC(C2)CC1C3 C1(CNC(c2nc(C(C)C)sc2)=O)COCCN(C(=O)CSc2nnnn2C)C1 C1(C(NOCCC#C)=O)CCC(O)CN1C(=O)CC(CC)OC C1(NC(c2scc(C)c2)=O)CC2CCC1CN(C(=O)COc1cccc(Cl)c1)C2 c1(C(=O)NCCc2cn(CC3CCOC3)nn2)nn2cc[nH]c(=O)c2c1CO c1(C(C(=O)NCCC#N)N(CC)Cc2cocn2)cc(OC)ccc1OC c1(CC)ccc(C)c(C(=O)NC(C2(O)CN(C(=O)CC3CC(F)C3)C2)C)c1 C1(NC(C(CCOC)C)=O)CCCN(C(c2c(OCC3CC3)cccc2Cl)=O)CC1 C1(NC(=O)CCCn2cc(-c3c[nH]nc3C(=O)O)nn2)CCC(CCO)CC1 c1(C(=O)NC(CC)CNC(C2CC3C=CC2C3)=O)cnn2c1CC(C)CC2 Cc1cc(C(F)F)n(CC(=O)NCC2CCCCN2C(c2cnco2)=O)n1 c1(CC(=O)NCCN(C(C2CCCC(OC)C2)=O)C2CC2)c(Cl)cccc1Cl c1(C(=O)NCC(CC=C)NC(=O)C(C(C)C)NC(N)=O)ccc2oc(C)nc2c1 N1(C(c2cn(CCCC)nn2)=O)CCCC12CCCN(C(c1cn(C)cn1)=O)C2 c1(OCC)ccc(C(N2CCCOC(CNC(=O)CN(C)C(C)C)C2)=O)cc1Cl CCCC(CC)CC(=O)NCC12CCC(CC1)N2C(=O)CCCC(=O)NCC c1(C(=O)NC2C(CNC(c3nc(CC)oc3)=O)CC2)ccc(O)c(C)c1C CCCCCCC(C)C(=O)N1CC(C(=O)NOCCF)C(C(C)C)C1 CC1CN(C(c2ccc(O)cc2)=O)CC1NC(c1cccc(C2COC2)c1)=O C(=O)(CC(C)(O)COC)NC1(CC)CN(C(C2CC2(Cl)C(=O)OC)=O)C1 Cn1cc(C(=O)NC2CC3CC2N(C(=O)CSC(F)F)C3)c2ccccc2c1=O C1(NC(C(C)CN(C)C)=O)CCCC1(C)NC(=O)C(=O)C(C)C CON(CCC(=O)N1CCSCC(C)C1)C(=O)C(C(=O)OC)NC(C)=O c1(OC)cc(C(=O)Nc2ccc(C(=O)Nc3ncc(Br)nc3Cl)cn2)ccc1C C(=O)(C1=Cc2cc(F)ccc2OC1)NCC1(C)CCN(C(c2cc(F)c[nH]2)=O)C1 C1(CCC(N2C(C(=O)OCC)CS(=O)(=O)C2)=O)C2CC3CC(C2)CC1C3 C1(NC(C2CCCCC2O)=O)CC2(C1)CC(C(N1CCCC(F)(CO)C1)=O)C2 C1(NC(CCCOC(C)C)=O)CCN(c2ccccc2)CC1 C1(C(=O)OC)CCCC1C(=O)NCC(O)CN(C)C(C1CC2(CC2)C1)=O c1(C(=O)NC2CC(NC(C3C(C)C3)=O)C2)c(F)cc(Cl)cc1Br c1(C(N(CCn2cc(C3(CC#N)CC3)nn2)CC)=O)cc2ccncc2o1 N1(C(C(C=C)C)=O)CCOC(C)(CNC(=O)C(CC)=CC)C1 S(=O)(=O)(c1ccc(NCc2c(O)noc2C)nc1)NCC(CCCCC)CO Cn1nc(C(N2CCC(CCNC(c3ccc[nH]3)=O)C2)=O)c(Cl)c1C(F)(F)F C12(C(N(CCN(C(c3c(CC)oc(C)c3)=O)C)C)=O)CCCN1CC(O)C2 N1(C(c2nc(CCCCC)sc2)=O)CC2(CC(NC(=O)C=C(CC)CC)CO2)C1 C1(CC(=O)N(C2CCCN(C(=O)C=CC(C)(C)C)C2)CC)CCCNC(=O)C1 C(=O)(CCC(C)NC(c1ccc(OC)s1)=O)NC1CC(C=C)C1 N1(C(C(n2cc(-c3c(C)n(C)nc3)nn2)C)=O)CC2ON=C(c3cccs3)C2C1 Cc1ccc(C)c(CNC(c2ccccc2-n2cc(-c3cnc(C)s3)nn2)=O)c1 C1(NC(c2c(C)nc(O)nc2C)=O)CCCC2CN(C(=O)C#CC3(C)CC3)CC12 C1(CC(=O)NC2C(C(=O)NCC=C)COC2)(CN)CCCCC1 c1(C(=O)Nc2ccc(Cl)o2)cccc(COCC2CC(=O)N2)c1 N1(C(C2(CCC=C)CC2)=O)CC2CCC1CC(NC(=O)Cc1cc(C)sc1C)C2 C1(C(N2CC(C(CC)C)C2)=O)CC(C)CN1C(C1CC(N(C)C2CC2)C1)=O CC1CC(C(=O)NC2CCC2NC(c2cc(Cl)ccc2F)=O)CC(=O)N1 N1(C(C23CSCC2C3)=O)CCC(c2cn(Cc3ccccc3)nn2)CC1 CC1(C)CC(C(=O)NCc2nccs2)CN1C(c1ccc(CO)cc1)=O N1(C(c2c(=O)cc(C)[nH]c2)=O)CC=C(CC(=O)NC2CC(=O)N(C)C2=O)CC1 N1(CC)CCC(CC(=O)NC(C)C(C)SC)C(C(F)(F)F)C1 N1(C(C)=O)CC2CC3CC(C2)CC1C3.c12cccc(c1)OCC2 c1(SC(c2ccc(F)cn2)CC)ccc(-c2ncc[nH]2)nc1 c1(C(=O)NCC(CNC(CC=CC=C)=O)(C)C)ccc(OC2CCOCC2)cn1 N(C(=NCCc1ncnc(-c2ccccc2)n1)NCC(F)F)C1C(OCC)C1 c1(CC)cc(C(=O)N(CC(C)(C)CNC(c2ccoc2C(F)(F)F)=O)C)c(C)o1 C(=O)(C1=CC2CC(C1)CC2O)N1C(CNC(c2ncn(CC)n2)=O)CCCC1 C(=O)(C1CCCc2nncn21)NCCC1OCCN(C(C=CC(CC)=CC)=O)C1 N1(C(C(C#N)=CC(C)C)=O)CC(NC(c2cc(CO)[nH]n2)=O)CCC1C c1(N2CC(C)OC(C)(C(F)F)C2)nc(C(F)(F)F)nc2ncn(C)c12 c1(C(N2C(CCC)CN(C(=O)CC(C)(C)N(C)C)CC2)=O)cnc(S(C)(=O)=O)s1 N1(c2nnc(CC)o2)CC2CC1CCC2NC(=O)Cn1nc(C)n(C)c1=O C(=O)(CCCCC(=O)NCC1(CN(C(=O)C(C)N(CC(F)(F)F)C)C)CC1)OC Cc1c[nH]cc(Br)c1=NC(=O)N(CC(F)F)CCC1COC1 N1(C(C(C(=O)OC)C)=O)CC=C(CC(=O)N2CC3(CCC2CO)CC3)CC1 C#Cc1cc(C(=O)NCC2(Cl)CCC2)cc(F)c1.C12(CC1)C(=O)N2 N1(C(CC#N)=O)CCN(C(=O)Cc2ccc(OC(F)F)cc2)C(c2ncc[nH]2)C1 C=C(C)CC(=O)NC(C)CC1CN(C(=O)C(N2CCOCC2)C2CC2)C1 Cc1cc(N2CCN(C(c3cc(C(F)(F)F)cnc3C)=O)CC2)n2ncnc2n1 C(=O)(C(C)CCCOCC)Nc1cccc(C(=O)OCCSCC=C)c1 Cc1cc(C)c(N2CCC(C(=O)NCC(C)(O)c3cccs3)C2=O)c(C)c1 c1(-n2ncc(NC3C(C)COC3)c2)ccc(Cl)cc1 Cn1nnc2c(N3CC4CC(NC(=O)CC5CC5(C)C)C4C3)ncnc12 CC1(C)CCN(C(=O)CCCC#N)C1CC(=O)NCC1CC2(CCC2O)C1 N1(CCCn2cc(CC=C)nn2)CC(C)Cn2nc(C)cc21 Cc1cccc(=O)n1CC(C)(O)C(=O)NC1C2CN(C(=O)CCCNC(N)=O)CC12 c1(C(N(CCCNC(c2cnc(C(=O)OC)cn2)=O)CC)=O)nnn2c1CSCC2 Cn1nc(C(=O)NCCn2ccccc2=O)c2ccc(-c3ccnc(F)c3)cc12 CC(CNC(c1cnnc(O)c1)=O)C(=O)NOCC1(C)CCC1 CCC(C)(C)C(C)CC(=O)NCC(C1CC1)NC(=O)CCc1ccccc1 C(=O)(C(CCSC)NC(C1CCC(=O)C1)=O)NCC1(OCC)CC1 Cc1ccc(-c2nc(CCOc3ccccc3)nn2-c2cccnc2)nc1 C1(C(=O)NCC(C)Cc2cn[nH]c2)CN(C(c2ncc(F)cc2F)=O)CC1(C)C C1(N(C)CC=CC(=O)N(C2(Cl)CC2)C2CC2)CC2(C1)CC21CCC1 N1(C(CS(=O)(=O)NC)=O)CCC2CCCN(C(c3cccc(N)c3F)=O)C2C1 c1(CC(N2C(CNC(CN(CCC)C)=O)CC(OC)C2)=O)ccc(F)cc1OC c1(CNC(c2c(F)cncc2Br)c2n(C(C)C)nnn2)ccc(F)c(Cl)c1 Cc1c(OCC(=O)NC2CN(C(C3(CCF)CCC3)=O)CC2(C)C)cccc1Cl c1(-c2nc(-c3n(C4C(c5ccccc5)(C)C4)ccc3)on2)ccccc1I C1(c2ccc(F)cc2)(NC(C=C(C)Cl)=O)CCN(C(=O)CCOCC(F)F)C1 c1(C(=O)NCCCN(C(C2OCC2(C)C)=O)CC)sc2ccc(F)cc2c1C C1(CNC(C2(CC)CCOC2)=O)CN(C(c2ccnc(S)c2)=O)CC1O n1(CCOCCCC)cc(C(=O)NCC2(NC(=O)C=C(C)C)CCC2)cn1.OC CC1(C)CCCN(C(=O)C(C2CC2)NC(C2CS(=O)(=O)C2)=O)C1 CC(C)(CC(F)(F)F)C(=O)N1CCN(C(c2cccc(N)n2)=O)C(CC(F)F)C1 c1(C(N(C(C)C(=O)NCC(C)(O)CO)CC)=O)cccc(C)c1N c1(OC)c(Br)c(C)nn1C.c1(OC)cccc(CN2C(=O)N3C(CCCC3)C2)c1 Cc1c(N)cc(C(N2CCCCC2CCNC(c2cnn(C)n2)=O)=O)cc1N C1(C)(CNC(CSCCOC)=O)CCCN(C(C2CC2c2ccncc2)=O)C1 C#Cc1ccc(OC)c(C(=O)NCC(O)CNC(=O)Cc2ccc(O)c(Cl)c2)c1 C(=O)(CC(C)C(C)(C)NC(=O)CC1CCCOC1)Nc1cnc(SC)nc1 CCC(CC(=O)NC1CC2CC(NC(=O)COCC3CC3)C2C1)C(C)(C)C c1(C(=O)NC2CCC(NC(=O)C(=Cc3cccnc3)F)CC2)cc(Cl)nnc1O Cc1nn(C)c(C)c1CC(=O)OC1CNC1.CC(C)(C)C c1(N2CCC(OCCN(C)C(c3cccc(F)c3)=O)C2)ccn2ncc(Br)c2n1 N1(C(C(C2CCN(C(C3CCCN3C=O)=O)CC2)C)=O)CCC(F)C(F)C1 c1(OC)cc(CNC2CC2C(=O)NCc2ncccc2OC)ccc1[N+](=O)[O-] N1(C(C(C)n2ccnn2)=O)CCC(CF)(NC(=O)C(F)=CCCF)C1 c1(N2CC(CC(=O)NC(c3ccns3)C)OCC2)nc[nH]c2ncc(C(N)=O)c1-2 c12c(ccc(Cl)c1Cl)C2.N1(CCN)CCN(Cn2nc(C)cc2CC)CC1=O.SC N1(C(C2(C)CC(=C)C2)=O)CCCC(CCC(N2CC(O)C(O)C2)=O)C1 CCC(CC)(CC)C(=O)N1CC(C(=O)NC2CCC(C)(F)CC2)C2(CCC2)C1 C1(CNC(c2ccc(CC3(C(=O)NCCCCl)CC3)s2)=O)C2CN(CC(F)F)CC12.N.CO C(CC(=O)NC1CCC1CC(N1CCC1C)=O)OCC#C c1(CN2CCC(NC(c3ccc(OC)cc3C)=O)CC2C)cc(O)c(F)c(F)c1 CC1CCCN1C(=O)C(CNC(=O)CCN(C)C)N(C)C c1(OC)ccc(Br)c(C(=O)NC2C3CC2N(C(C2CC(C)C2)=O)C3)c1 Cc1cc(C(=O)NCC2CCC2C(=O)NC(c2ccns2)C)c(C)s1 c1(C(N2C(CN(C(C(C)SC(F)(F)F)=O)C)CCC2)=O)cnnc(O)c1 N1(C(Cn2ccc(C)n2)=O)CC2CC(NC(=O)CSc3cccc(Cl)c3)C1C2 C1(CCOC)(C(=O)NCC2CC2CNC(=O)CC2CCCCO2)CCCC1 Cn1ccc(CC(N2CC(C(C)(C)CNC(=O)CC3CCOC3)C2)=O)c1 c1(C(=O)NCC(CC)NC(c2cccc(F)c2C(C)C)=O)ccc(F)c(F)c1F C1(NC(c2cnc(N(C)C)o2)=O)CCC(NC(c2n[nH]c(C3CC3)c2Cl)=O)CC1 CN1CCCCC1C(=O)NC(CNC(C1CN(c2ccc(Cl)cc2)C1)=O)CO C(=O)(N=S(C)(=O)c1ccc(C#N)cc1)NCCC1(C)COCCO1 C1(NC(CCCCC)=O)COCCN(c2cc(C3CCCCC3)ncn2)C1 NS(=O)(=O)CC(=O)N1CC(NC(=O)Cc2cccnc2)C2CC12 Cn1cc(-c2cc(C(N3CC(CCNC(C4C=CCCC4)=O)C3)=O)no2)cn1 C1(N(C2CC3(CNC3)C2)C(CCN(c2ccccc2)C)=O)CCN(C(N)=O)CC1 C1(CCNC(C2C(COC)C2)=O)CN(C(=O)C(F)(F)c2ncccn2)CC1C C(=O)(C(CC(C)C)CC(C)C)NC1C(CNC(c2n[nH]c(C)c2[N+](=O)[O-])=O)C1 c1(OC)ccc(C(c2nnnn2C2(C)CC2)NC2CC23CCCCC3)c(Br)c1O N1(C(C(C=C)OC)=O)CCCN(C(=O)CCC(=O)c2ccccc2)CC1 Cc1nc(C)c(C(=O)NC(C)C(C)C(=O)NCC2CCC2CO)o1 Cc1c(F)cc(CN2CCCCC2CNC(=O)Cn2nccn2)cc1F C1(CC(=O)NC(CC)C(=O)NCC(=O)NCC2CCC2)CCCOCC1 N1(C(CSCCCC)=O)CC(CNC(=O)Cc2cc(F)ccc2Cl)C(C)(C)C1 CCC(COC)C(=O)NC(C(C1CCCCC1)NC(c1cnn(C)c1)=O)C(C)C c1(C2(C(=O)NCC3N(C(=O)C(F)=C4CCCC4)CC3)CC2)ccc(Br)cn1 C12(CNC(=O)CCn3cncn3)CC(NC(c3ncccn3)=O)(CCO1)C2 CC1CCCN(C(c2nncn2C2CC2)=O)C1CNC(c1cc2ccsc2[nH]1)=O S(=O)(=O)(CCC(=O)NCC1CC2CN(C(=O)C(F)C(C)(C)O)CC12)N(C)C N1(C(C23OCC(C(=O)OC)(C2)C3)=O)CCC(NC(=O)C(CC)C(C)C)C(F)C1 C=CC(C)C(=O)NC(Cc1cc[nH]n1)C(=O)NCc1csc(CC)n1 N1(C(=O)Cc2ccsn2)CC2CCC1CN(C(C13CC(F)(C1)C3)=O)C2 C1(C)(CNC(C(c2ccccc2)C)=O)CN(Cc2cccc(F)c2Cl)CCO1 C12(C(=O)NCc3c(CCNC(C(N)=O)=O)ocn3)CCOC1CCOC2 C#CCCC(O)C(=O)N1CC(N(C)C(c2ncn(C)c2C)=O)C1 CCCCC(C)CCC(=O)N1CCCC(CC(=O)NCC2CCC2C)CC1 C(C)(C(C(=O)N(C)CC1(O)CN(C)C1)NC(=O)C(C)C1(O)CCC1)OC c1(C2(C(=O)NCCn3cc(-c4ccnc(F)c4)nn3)CC2)cc(F)c(F)c(F)c1 C1(CC)CN(C(=O)CS(=O)(=O)NCCOC)CCN1C(=O)C(F)CCC CCCC(C)C(=O)NCC1CCC(NC(=O)CN2CCP(C)(=O)CC2)C1 c1(C(=O)NC2(COC)CN(C(c3sc(F)cc3C)=O)C2)cnnc(C)c1 N1(C(C(C)OCCCC)=O)CCCN(C(C2(C(F)F)CC2)=O)C1C C1(CC)CN(C(=O)CCc2ncccc2C)CCN1c1ccnc(SC)n1 C1(CCNC(=O)C(C2CCCO2)C2CC2)CCCN1C(=O)CCn1cccc1 N1(C(C(CCSC)NC(C2CCC(=O)O2)=O)=O)CCc2sccc2C1 N1(C(=O)OC)CCCC(CNC(=O)NC(c2cn(-c3ccccc3C)nn2)C)C1 CCC(CCC(=O)NC1CCCC1NC(c1nc(O)c(C)s1)=O)OC C#CC1CN(C(c2ccc(C)c(C)c2)C(=O)NCCCNC(=O)OCC)CCO1 C(=O)(C1=NOC2(CCOC2)C1)N(CCCNC(C1CNC(=O)N1)=O)CCO N1(C(c2cccc(CC(=O)OC)c2)=O)CC2=C(C1)CN(C(=O)CNS(=O)(=O)NC)C2 c1(C(=O)NCC2C(NC(CN(C3CC3)CC)=O)COC2)ncc(C)cc1OC c1(C(=O)NCC2CC(F)(CNC(CCNC(N)=O)=O)C2)cc2ncccc2o1 CC1CC(=O)Nc2ccccc2N1C(=O)CCC(C)(C)C#N Cc1ccc(C(F)F)cc1C(=O)NC(C)(C)CCNC(=O)C(C)OCCC(C)C C(CCC(O)C(=O)NCCS(N)(=O)=O)NC(c1c(C)nccn1)=O c1(CC)ccc(F)cc1C(=O)NCC(C)NC(=O)Cc1nc(Br)sc1C C1(NC(C(CC)C)=O)C2COCC1CC(NC(=O)C=CC1CCCCCC1)C2 C(=O)(C1CCCc2nncn21)N1CCC(CNC(=O)C#CC2CCOC2)CC1 c1(C(=O)NCC(C2CCC2)NC(C2CN3CCN2CC3)=O)cc2cccn2cn1 c1(SCC)cncc(C(=O)NC2CC(NC(=O)C=C(C)C)C2)n1 N1(C(C(COC)C)=O)CC(C)(C)CC1CC(=O)N(C)Cc1cnco1 C1(C(=O)NC2(C(NOCCOC(C)C)=O)CCSC2)(CF)CCOCC1 N1(C(C2CCC(C)O2)=O)CCC(C(N2CCC(C)(C(N)=O)C2)=O)C(C(N)=O)C1 C1(Cl)(C(=O)NCC2CCN(C(c3c(CC)ccs3)=O)C2)CC12CCC2 C12CCC3CCC1N3C2=O.C12(COC1)CC1(CC1)C(=O)NC2.C1(CO)CCC1 C1(C(N(CCC2CN(C)C2)C)=O)C2CCCC2CN1C(C1CCS1(=O)=O)=O c1(C(N2C(C)(CNC(CC(C=C)C)=O)CCC2)=O)nc(F)ccc1Cl C1(C(=O)Nc2cccc(NC(c3n(C(CC)C)ncc3)=O)c2)CCC(C)(C)OC1 c1(C(c2ncccn2)NCC(C2CCCO2)OC)ncc(Br)cn1 N1(C(c2c(C)coc2)=O)C2CCC1CN(C(c1csc([N+](=O)[O-])c1)=O)CC2 Cc1cc(C(C)NC(c2cccc(-n3cnnn3)c2)C)nc2ccccc12 c1(OC)ccc(C)c(C(=O)NCC(C2CCN(C(C3CC(SC)C3)=O)CC2)O)n1 C1(CC)CN(C(c2cc(C)[nH]n2)=O)CCC1NC(c1ccc(C(C)(C)C)[nH]1)=O N1(C(CCCOCC)=O)CC(C)CN(C(c2cc(=N)[nH]c(Cl)n2)=O)C(C)C1 N1(C(C(c2cccc([N+](=O)[O-])c2)C)=O)CC(NC(=O)C(C)(C)O)CC12CCOC2 C(=O)(C(C)CS(C)(=O)=O)N1C(C(C)NC(c2c(C)nn(C)c2F)=O)CCC1 N1(C(Cn2c(=N)nc[nH]2)=O)CCC(C2CC2)C1C(N1CC(F)C(F)C1)=O N1(C(=O)CC2CC(F)C2)CCN(C(c2cc(SC(F)(F)F)c[nH]2)=O)C2(CCC2)C1 CCC(CCC(=O)N1CCC(CN(C)C)C1)NC(=O)CN(C)C(C)C C1(CCNC(C(=C(C)C2CC2)F)=O)COCCN1C(=O)Cc1cnc(C2CC2)[nH]1 C(CCCC(CO)NC(c1scnc1CC)=O)NC(CNC(C(CC)CC)=O)=O c1(CNC2COCCN(C(CC=CCC)=O)C2)c(F)cc(C)cc1F N1(C(=O)NCCCC(F)F)CCC1c1cccs1 N1(C(C(C)OC)=O)CC2(CO)CC1(CNC(=O)C(O)C(C)(C)C)C2 N1(C(C2C(COC)C2)=O)CCC(C)(NC(=O)C(C(C)O)NC(=O)OC)CC1 c1(C(N(CC(C)NC(C2CC2(Cl)Cl)=O)C)=O)c(C(F)F)cccc1N N1(C(C2CCN(CC3CC(C)OC3)C2)=O)CCc2nc(C(C)(C)C)ncc2C1 C1(CNC(c2c(C)cc[nH]2)=O)(CO)CCN(C(=O)CC2SC(=N)NC2=O)CC1 C(=O)(C(N)CCC(F)(F)F)N(C(COC)C)C CN1CCC(C(N2CCCCC2CNC(=O)CN2CCCNC2=O)=O)CC1 C(=O)(C1=CC2CCCC12)N1CC(C)N(C(=O)CCC(=O)c2ccncc2)CC1 C12(CNC(C3C(c4cc(C)no4)C3)=O)CN(C(c3cnnn3C)=O)CC1CCO2 CC(C)C(F)(CNC(=O)Cc1cnn(C)c1)C(=O)NCCCOC(=N)O C1(N(C)C(=O)OC(C)(C)C)(CC2N(Cc3scc(C)n3)CCC2)CCOCC1 c1(C(N2C(C(N(CC(C)SC)CC)=O)CC(OC)C2)=O)cc2cccnn2c1 N1(C(c2c(CC)nns2)=O)CC(NC(=O)CSc2cccc[n+]2[O-])CC1C CC(CC(=O)NC1(C2CCN(C(c3ccc(F)cn3)=O)C2)CC1)CC(C)(C)C c1(C(=O)NC2(CNC(c3n(CC)ncc3)=O)CCC2)cc2occ(Br)c2[nH]1 C#Cc1ccc(CCC(=O)NC2CCCCN(C(c3cc[nH]c3)=O)C2)cc1 C1(CC=C)(NC(=O)CNS(=O)(=O)C2CC2)CN(C(=O)C(O)CC2CCOCC2)C1 Cn1ccc(=NC(=O)C2CC(NC(=O)CNS(=O)(=O)C3CC3)CCO2)[nH]1 c1(C(=O)NCCC2CCN(C(c3cncn3C)=O)C2)ncccc1O.C1CC1 c1(NC(C2(C)OCCCO2)c2n(CCSC)nnn2)cn(C)c2c(C#N)cnn12 CN1CCC(CC(N2CC(O)CC2C(=O)NCCC2CCCC3CC23)=O)CC1 c1(OC)c(Cl)cc(C(=O)NCC(C)NC(=O)COc2ccc(Cl)c(C)c2)nc1Cl N1(C(c2n(C)nc(C3CC3)c2)=O)CCCC(C)(NC(C2C3CC(F)(F)CC23)=O)C1 c1(C(C(=O)NCC2C(CNC(Cc3ccn(C)n3)=O)C2)(F)F)c(F)cccc1F c1(C(N2CC(C(NOCCOCC)=O)(CF)C2)=O)cnc2n1CCC2.C(N)=O Nc1cccn(CC(N2CCCC2CCNC(=O)CC2CCC3CC23)=O)c1=O c1(CSC)ccc(C(=O)NC(C2CCCCC2)CNC(C2(C)CCCO2)=O)o1 C1(C(N2CCCC(OCC)C2)=O)CC2CCC(C1)N2C(c1cscc1C)=O n1(CCC(=O)NC2C(C)CN(C(c3cnc[nH]3)=O)CC2)ccc2cccnc12 C1(C2CN(C(c3ccsc3Cl)=O)C2)(NC(C(C)OC2CCOC2)=O)CC1 N1(C(C=CC(C)NC(=O)CCC2OCCO2)=O)CCC(C)C2(CCC2)C1 C1(C(N(CC(CC)NC(=O)CCc2csnn2)C)=O)(CCN(C)C)CCCC1 c1(CC(=O)NCC(=O)NC2CC(OCCC(C)C3CC3)C2)cc(F)cc(F)c1 C(N=C(NCC1CCOC1)N1CCC(C)(CC)C1)c1ccc(OCCC)c(F)c1 O(NC(=O)C(CNC(C1(CN)CC12CCC2)=O)N1CCOCC1)C(C)(C)CO CC1C(NC(=O)C(C)Cc2ccc(F)c(F)c2)CCCN1C(=O)C1=COCCC1 N1(C(c2n(C(CC)CC)ncc2)=O)CC2CN(C(=O)C(C(C)C)OC)CC2C1 c1(SCC(=O)NC2C(NC(C(C(=O)OC)OC)=O)C2)ccccc1[N+](=O)[O-] c1(C(=O)NC2CCN(C(C3(CC)CC3)=O)C2)cc(OC)nc(C)c1 C(CCC(=O)NC1CC(C(F)(F)F)C1)NC(=O)NCC#C.C12(CCC1)C(=O)NC2 C1(CNC(c2ccccc2O)=O)CCC2CN(C(c3ccon3)=O)CCC2C1 C(=O)(C(F)C(C)C)NCC1CC1.C1(CC#C)CCN(C(C2(C)CC=CC2)=O)C1 Cc1ccc2[nH]c(C(N3CCC(C(=O)Nc4ccc5ccnn5c4)C3)=O)cc2c1 N1(C(C(C)=C2CC2)=O)CCC(C)C1C(=O)NCCCF c1(C(=O)NC2C(C)CN(C(=O)CC3CCN(C)C3)C2)ccc(P(C)(C)=O)cn1 Cc1ncnc(C)c1N(C(=O)CCCCSCC(N1CCCC1)=O)C N1(C(CCN(CCC)C)=O)CC2(CCN(C(=O)CC3(N(C)C)CC3)CC2)C1 c1(C(=O)NC(C2CCN(C(=O)C(C)C3CC3)C2)C)cnc2ccnn2c1O N1(C(CCN(CC)CC)=O)CCC(CO)C(NC(=O)CCCC(=O)NC(C)C)C1 C(=O)(CC1=CCOCC1)Nc1ccccc1.C1(C)(OC)COCCC(C)NC1=O CC1CN(C(C2CCO2)=O)CC1CCNC(c1ccc(-c2cnc[nH]2)cc1)=O CC1CC(C(=O)NCCC2(C(=O)Nc3ccc(F)cc3F)CCC2)=NO1 C(=O)(CCC(C)(C)OC)NC(CC)CN(C(=O)C(C)CC1CCCCC1)C c1(C(N2C(CNC(C(CC)C(C)C)=O)CC2)=O)cc2nccc(C(F)F)n2n1 Cc1nc(C#N)ccc1NC(C1CCN1Cc1cccc(Cl)c1F)=O N1(C(c2cn(CC)nc2)=O)CCCC(C2CCCN(C(C3COC(=O)N3)=O)C2)C1 C1(NC(CS(=O)(=O)N(C)C)=O)CCCN(Cc2cccc(C(F)(F)F)c2F)CC1 S(=O)(=O)(c1ccc(C(N2CCCCCC2CNC(=O)CC2CC2(C)C)=O)o1)NC N1(C(C(C=C)(C)CC)=O)CCC(C)(C)C(NC(c2cnccn2)=O)C1 C1(N(CC#C)C(c2sc(C)nc2C)=O)CCN(C(=O)COCC2CCC2)CC1 CC(C)CC(CNC(=O)C(C)(C)OC(C)C)NC(c1cccc(C(F)F)c1)=O Cc1ccc(O)c(CNC(C2CC(NC(c3cncn(C)c3=O)=O)C2(C)C)=O)c1 C1(CNC(c2c(SC)ccs2)=O)CCN(C(=O)C(F)=C2CCCC2)C12CC2 c1(CCC(N2CCCC(NC(=O)COc3cn[nH]c3)C2)=O)coc2ccccc12 c1(C(=O)NCCN2CCC(C3(C(F)(F)F)CC3)C2)nc2cnc(Cl)cc2s1 C(C1=CCN(C(c2nccn2C(C)C)=O)CC1)NC(C(C(C)C)OCC)=O c1(NC(C(n2cc(C(C)(C)C)nn2)C)=O)nc2ccc(I)cc2s1 N1(C(=O)CC=C(Cl)Cl)CC(CNC(C2(C(F)F)CCCC2)=O)C2(CCOCC2)C1 Nc1ccc2[nH]c(=NC3CCC(NC(C4CC45CCCOC5)=O)CC3)sc2c1 c1(NC(C2C(CNC(C3C(C)(CC)C3)=O)C2(C)C)=O)ccc(OC)cc1C c1(C(C)=O)ccc(C(=O)NCC2CC2NC(c2c[nH]cc(Cl)c2=O)=O)cc1C C(=O)(C1CCCc2c[nH]nc21)NC1CCN(C(C23C(C)OC(CO)(C2)C3)=O)C1 c1(C(=O)NC2C(C(C(=O)NCc3c(C)nccn3)C)CC2)c[nH]c2cccnc12 C1(NC(=O)NCCSCCCC)COc2ccccc2OC1 CCCCC(CC(=O)NCCN(C)CCF)NC(C1CC=CCC1)=O c1(NC(C2N(C(Cc3cn(C)nc3)=O)C3CCC2C3)=O)ccc(C#N)cc1F Cc1cccnc1CCC(=O)NCC1CCC1NC(=O)CC1CCCCC1C c1(CN2CCN(C(C3=C(C)OCCS3)=O)C(C)C2)nc2cccc(F)c2[nH]1 c1(C(=O)NC2CC3(CC(NC(c4c(OC)scc4)=O)C3)C2)ncn2c1COCC2 N1(C(Cn2c(=N)scc2)=O)CCC2(CC1)CCN(C(C1(C(F)F)CCCO1)=O)C2 Cc1cc(CCNC(C2(CCNC(C3CC=CC3)=O)CCC2)=O)n[nH]1 C1(C(=O)NC(COC)C)CCC(C)(C)N(C(=O)CSc2nc[nH]n2)C1 C1(NC(C2(CNC(COC(CC)C)=O)CCCC2)=O)CCOCC1CC Cc1cccc2[nH]c(C(=O)NC3CN(C(=O)Cc4cc[nH]c4)CC(C)(C)C3)cc12 c1(OC)cc(C(=O)NC2CN(C(=O)CCC3OCCO3)CCC2C)ccc1C c1(OCC#C)ncccc1C(=O)NC1(NC(=O)CCSCC)CC(F)(F)C1 N(C1CCCn2cc(CNC(=O)OC(C)(C)C)cc21)C(=O)NC1(CC)CC(C)C1 S(=O)(=O)(c1ccc([N+](=O)[O-])c(Cl)c1)N(C1CN(S(=O)(=O)c2nccs2)C1)C CCC(C)C(O)C(=O)NCCC1(NC(c2cc(F)cnc2O)=O)CCCC1 CC1C(NC(=O)CCCc2ccsc2)CCCN1C(=O)CCP(C)(C)=O N1(C(c2c(C)cccc2)=O)CCC(CC(N)=O)(NC(=O)C(C)CC(C)C)CC1 C1(C)(CCC(=O)N(CC(C2CC2)OC)C)CN(C(c2cn[nH]c2)=O)C1 c1(CN)ccc2nccn2c1.c1(CC)ccc(CC(C2CSCCN2)=O)cc1 Cc1cn2c(CC(=O)N(C)Cc3cn(Cc4ccccc4Br)nn3)csc2n1 c1(NC(C2C(NCc3ccc(CC)cc3OC)C2)=O)cc(Cl)cc(Cl)c1F c1(OC)cc2c(cc1C(=O)OC1CNS(=O)(=O)C1)CCC2 Cn1cc(Cl)c(C(N2CC(NC(=O)CC3CCCCC3)C(O)C2)=O)n1 CC(C)C1C(=O)N1.C1(=O)CC(=O)OC(=O)CN1.C1(NC(C)(C)C)CCCC1 C1(NC(=O)NC2C(OC(C)(C)C)COCC2)CCC2(CCOC2)C1 C1(NC(c2c(C)n(C)cc2)=O)CCN(C(=O)C(C(C)O)N(C)C)CC1CO C(=O)(C(C)(CSc1ccccc1)CC(F)(F)F)NCc1onc(CC(=O)NC)n1 c1(C(N)=O)cccc(NC(C2CC2C(=O)NCc2cc(Cl)sc2Cl)=O)c1 c1(C(=O)NCC2C(CNC(=O)CC3CCOC3)C2)ccc2ncnn2c1 N1(C(CSCCOC)=O)CCC2(CC1)COC(CNC(=O)CCc1cc[nH]n1)C2 C1(N(C(c2cccc(C3(C)CCO3)c2)=O)C(C)C)CCCN(C(C23CC2C3)=O)CC1 c1(CN(C)C(C2(NC(=O)Cc3ccccc3)CSC2)=O)cnnn1C C1(CN(C(=O)CCCC2CCC2)C)CN(C(c2cc(C(C)(C)C)n[nH]2)=O)CCO1 CCCC(CCc1ccccc1)C(=O)N1CCCC(N(C)Cc2cncn2C)C1 CCCC(C)CC(=O)NCc1nc(C(=O)N(C(C)C(C)SC)C)c(C)o1 N1(C(C(COC)OC)=O)CCC2(CC1)CN(C(C1(F)CCCOC1)=O)C2 N1(C(c2ccc(C(C)=O)cc2F)=O)CCCC(NC(c2csc(C)c2)=O)C(F)C1 c1(C(C)(C)C)cn2c(n1)CCC(CN1CCC(c3cccc(O)c3)C1)C2 C(CCC(=O)NCC(Cc1ccccc1)NC(=O)C(C)=CC(C)(C)C)OC(C)=O C1(NC(CSCCCC)=O)C=CCN(C(C2(C)CC(C#N)C2)=O)C1 c1(N(C(=O)C2CC2)Cc2ccc(C)o2)nc2cccc(F)c2c(=NC2CC(C)C2)[nH]1 c1(C(=O)NCC(CO)NC(=O)COCc2ccncc2)cc(Cl)cc2c1OCC2 O=S(=O)(c1[nH]c(=NCC(O)C2CCC2)ccc1Br)NCC1COCCO1 C1(N(C(C)=O)C)CCN(C=O)CC1.N1(CCC(C2(O)COC2)C)CCCCC1 N1(C(C(CC)NC(N)=O)=O)CCC12CN(C(C1CC(OC)C1)=O)C2 N1(C(=O)Cc2cccnc2)CCC(C(=O)N2CCC(O)C23CCC3)=C(F)C1 CC1OC2CCC1(NC(C1CCN(C(c3cc(O)nc(O)n3)=O)CC1C)=O)C2 c1(CN2C(C(=O)Nc3cncc(C(N(C)C)=O)c3)COCC2)cccc(F)c1I C1(CCC)(NC(C2CC(N(C)C)C2)=O)CCCN(C(c2cn(CC)nn2)=O)C1 C1(C(=O)OCc2cc(O)cc3c2OCOC3)CCc2ncccc2C1 CC1(C)CCCN(C(c2ccc(C(F)F)o2)=O)C1CNC(C1CCCSC1)=O N1(C(c2cc(C)no2)=O)CC2CCC(Nc3ccc([N+](=O)[O-])cc3)CC2C1 N1(C(=O)CCN2CCOCC2)CC2CCN(C(=O)C(O)Cc3cnc[nH]3)C2C1 C12(C(=O)NC3CCC(N(C)C(c4cc(CO)on4)=O)C3)CC(C1)S(=O)(=O)C2 N1(C(C=CC=CC)=O)CCC(C(=O)Nc2cc(C(N)=O)sn2)(COC)C1 C1(CNC(C=C(C)C)=O)CC2CCCC2N1C(c1cccc(C(N)=O)c1)=O Cn1[nH]c(=NC(=O)C2CCN(c3ccccc3C#N)C2)cc1C#N C1(CNC(=O)Cc2ccccn2)(CNC(C2CNC(=O)O2)=O)CC12CCC2 C1(n2cc(C(C)OCC)nn2)CCCN(C(c2ccc(C(F)F)o2)=O)CC1 C1(C(N2CCC(C(=O)NCCC(C3CCC3)OC)(CO)C2)=O)CC2C=CC1CC2 C(C1=CCN(C(=O)CCCn2ccnn2)CC1)NC(CCNS(CC)(=O)=O)=O c1(OC2CCCOC2)ccc(NC(C(C)(C)NC(=O)CO)=O)cc1.C1(S)CC1 C1(NC(C2CCCSC2)=O)CN(C(=O)COc2cc(F)cc(F)c2)CC2(CC2)C1 N1(C(c2c(CC)con2)=O)CCC(NC(=O)Cc2ncn(C)c2C)C(F)C1 c1(CC)cc(CNC(=O)C(=O)NC2CCCC2CNC)cs1 C#CC1(C(N2CCC(CF)C2)=O)CCN(C(=O)CCOCCOC)C1 N1(CC(=O)N(CC)CC)CCN(S(=O)(=O)N(C)C)CC(CO)C1 C(=O)(C1CCCc2nccn21)N1C2CCC(CCNC(C(C)(Cl)Cl)=O)(C2)C1 c1(SCCOCCNC(c2c[nH]c(=N)s2)=O)ccc(OCC(N)=O)cc1 c1(CC(=O)NC(C(=O)NC(C#C)CC2CCCO2)C(C)C)cnc2ccccn12 C1(NC(c2ccns2)=O)CC2CCC1C(NC(c1ccc3c(c1)CC3)=O)C2 C1(O)(CNC(CC=C(C)C)=O)CCCN(C(C2CC(N(C)C)C2)=O)C1 C1(OC)CCC2CN(C(=O)CCC3(C)CN(C(=O)CCCN(C)C)C3)CC12 c1(C(N2C3(CN(C(C4(COC)CCOC4)=O)C3)CC2)=O)ccc(F)c(C)c1N c1(CNC(c2ccc(C)nc2O)C)nc(O)c2ccc(C(C)C)cc2n1 N1(C(C(COC(C)C)NC(C)=O)=O)C2CCC1C(C(=O)Nc1cc(C)n(C)n1)C2 c1(C(=O)NCC(C)(C)OCCNC(c2ncc(C)nc2)=O)cccn(C)c1=O C1(CNC(=O)COC2CC=CC2)CN(C(C23CC(C2)C3)=O)CCCO1 C1(OC)CC2(C1)CC2C(=O)NCC1CCCN(C(=O)COCc2ccccc2)C1 CC1CC(C)(C(=O)N(C)CC2CCCN2C(=O)C2=CSCCO2)CC(C)O1 c1(C(=O)NC(C2CN(C(CCNC(=O)OC)=O)C2)C)ccc2occ(CO)c2c1 C1(NC(C(C2CCOCC2)C)=O)CCC(N(C)C(c2cnc(O)n2C)=O)CC1 c1(CC)ccc(C(=O)NC(C2CCN(C(c3sccc3C(C)=O)=O)C2)C)cn1 c1(OC)cc(C)ccc1C(=O)N(C1(C(=O)NC2CC2CC(C)C)CC1)C C1(C(C)NC(=O)Cn2ccsc2=N)CN(C(c2cscc2C(F)(F)F)=O)CCO1 N1(C(C2(C)CCCS2)=O)CCN(C(c2ccc(C3CC3)s2)=O)C(CC(F)F)C1 C(CC)(C(=O)NC(C(=O)NOCCC1CC1)C1CC1)=CC CC1CC2CN(C(=O)C(C)(C)C3CCCC3)CC2N1C(=O)CCOCC1CCC1 n1(C(C)C(=O)NCCOCCC2CC2)cc(C2(C)CCCO2)nn1 N1(C(C2(C)CCNC(=O)C2)=O)CC(O)(C2(CNC(C3(O)CC3)=O)CC2)C1 N1(C(c2c(C)nc(C)o2)=O)CC(NC(=O)CCCC(N)=O)CC12CCOCC2 C(=O)(CCC(F)F)N1CCC(n2cc(-c3cn(C)nc3)nn2)C1.C12CN1C2 C(=O)(C(C(C)C)NC(=O)OC)NCC=C1CCN(C(c2cc(CCC)on2)=O)CC1 c1(CC(=O)N(CCC)CCNC(c2n[nH]cc2CC)=O)ccc(Cl)cc1Cl CCC(C(=O)N(C)CCN(C)C=O)NC(c1cscc1SC)=O.c1(S)ccccc1 c1(C(N(CCC(N2CC(CCC#C)C2)=O)C2CC2)=O)cc(C)cc(O)c1 c1(NC(N2CC(Oc3ccc(SC)o3)C2)=O)ccc(N2CCCNC2=O)c(Cl)c1 Cc1cccc(C2(F)CC2NC(N2CCN(c3ncccc3Br)CC2)=O)c1 NC(=O)CCCCC(=O)NC1CCCCCC1NC(C1CC1(F)F)=O n1(C(C)C)ccc(CC(=O)NCC2CC(F)(CNC(=O)C=CC3CCOC3)C2)n1 [N-]=[N+]=NC1(C(N2CC(n3cccn3)C2)=O)CCN(C(=O)CCc2cnco2)C1 CC(C)CC(C)C(=O)N1CCC(CNC(c2cccnc2)=O)C(O)C1 c1(NC(Nc2cc(OC)cc(F)c2)=S)ccc2c(c1)CCC(=O)N2 C(=O)(C(C)CC(=O)N1CCCC1(C)CNC(c1ncc(C)cc1F)=O)OC C1(C(N2CC(NC(C3(CC4CC4)CCCCC3)=O)C2)=O)CCC2(CCC2)O1 [N-]=[N+]=NC1CN(C(C)=O)CC1NC(=O)Cc1cc2ccccc2o1 C1(CNC(C2(SC)CCC2)=O)CN(C(c2cc(O)cc(F)c2)=O)CCCO1 n1(CC)ccc(C(N2CC(CNC(C3CC4CC3CC4O)=O)CC2C)=O)cc1=O C(=O)(C1=C(Cl)CCC1)NCCN(CCOCC)C(C1(CCN(C)C)CC1)=O c1(CN(C2CC(O)C2)C=O)cccc2occc12 C1(C(=O)NCC(N(C(c2cccc(CC)n2)=O)C)C2CC2)CCC(C)(C)CC1 c1(C(=O)NC2CC(CNC(C(CC#C)O)=O)C2)ccc(=O)n(CCO)c1 c1(OCC)ccc(Cl)c(C(C)NC(=O)CN(C2CCC2)C)c1 N1(C(C(C)NC(c2ccco2)=O)=O)CC(C)C(C)(C[NH+](C(=O)C2=CSCS2)[O-])C1 c1(OC(C)C)ccc(C(C)(C)C(=O)N(CC(N2CCOCC2)C)C)cc1 C12(C(N(C(C(=O)OC)C)C)=O)CCN(C(c3cn[nH]c3)=O)CCC1C2 c1(C(=O)NCC(C)(F)CNC(C2CC3C(C2)C3(F)F)=O)cc2c(Cl)nccc2o1 c1(C(=O)NCCN2CCN(C(c3c(COC)scc3)=O)CC2)ncn2ccccc12 N1(C(C(CCCC)=O)=O)CC2CN(C(=O)Cc3cc(Cl)n(C)n3)CC2C1 C(C(C)C)(C(O)C(=O)N1CCC2(C1)CN(C(=O)C(F)(F)C(F)F)C2)OC C(=O)(CCCCCCC(=O)N1CC(C(N2CC(C)Nc3ncccc32)=O)C1)OC c1(CCCC(=O)NC2CN(C(CCC(C)=O)=O)CC(O)C2)ccc2c(c1)OCO2 c1(C(N2C(C)CN(C(=O)Cc3ccsn3)CC2)=O)cc(=O)n2nccc2[nH]1 c1(C(CC)C(=O)NC2CCCC2NC(=O)CN2CCCC2=O)ccc(F)cc1 C1(CNC(CN(S(CC)(=O)=O)C)=O)CCCN1C(c1ccc(C(C)=O)o1)=O N1(C(c2c(CC)n(C)cc2)=O)CCC=C(C(=O)NCC2CN(C3CC3)C2)C1 N1(C(C(COCC)n2cc(-c3[nH]cnc3C#N)nn2)=O)CCCC(C)(O)CC1 N1(CC)CCCC1C(=O)NC1(C)CC(C(=O)N(C(C)CC(N)=O)C)C1 C(c1ccc(Cl)cc1F)=CC(=O)NCCCCC(CO)NC(C(CC)N(C)C)=O N1(C(C2CC(OC)C2)=O)CCC2(CCC2NC(=O)CC(C)(C)C(F)F)CC1 c1(OC)ccc(-c2cc(=N)[nH]c(N3CCCC(C)(C(C)C)C3)n2)c(Cl)c1 c12ccc3c(c[nH]c3c1)CC2=O.C(=O)(N=c1cc(C)n(CCO)[nH]1)OC C(=O)(CCCC(N)=O)N(C)CC1CCC1.C1(C)(c2ccccc2)C(=O)N1 c1(N2CC(S(CC)(=O)=O)C2)[nH]cnc2nc(Br)cc1-2 c1(C(=O)OC(C2CCC2CNC(C)=O)=O)cnn(C)c1OC C1(C2CCCN(C(=O)CN=S(C)(C)=O)C2)(NC(C(n2c(C)cc(C)n2)C)=O)CC1 n1(CC(=O)NC2C(CNC(C(C=C)CC)=O)CCCC2)ccc(=O)cc1C N#Cc1c(F)c(C(=O)NCC2CCCN2C(C2CCC3CC3C2)=O)cc(F)c1F C1(C(=O)NC2C(C)CN(C(c3ncoc3C(F)(F)F)=O)C2)CCOCC12CCC2 C1(C(=O)NC2CCC(N(C(CC=C(C)C)=O)C)C2)CC2C=CC1CC2 C1(NC(c2ccc(C(C)(C)C)[nH]2)=O)CC2(C1)CN(C(=O)CCc1ccoc1)C2 C1(C2CCN(C(=O)C(CC)Sc3nc(=N)[nH][nH]3)C2)(NC(c2ccc(CC)[nH]2)=O)CC1 C#Cc1cccc(NNC(=O)C2(CNc3ccccc3)CCCC2)c1C N1(C(C(C)OCCOCC)=O)CCCC(CN(C(=O)Cc2c(C)n[nH]c2C)C)C1 c1(C(N2CC(CNC(C(C(C)OC)O)=O)C2)=O)ccc(Cl)c(S(N)(=O)=O)c1 CC(C)C(C)CC(=O)NC1CCCC1CC(=O)NCCc1ncon1 c1(C(=O)NC2(CN(C(c3ccc(C#C)cc3)=O)C)CC2)nc(Cl)c(=O)[nH]c1N c1(C(=O)NC2CC(C)N(C(c3cnc[nH]3)=O)C2)cc(N)c(F)c(F)c1F Cc1ccnc2sc(C(=O)NC3(CO)CCN(C(C4CCSC4)=O)C3)c(C)c12 c1(C(=O)NCC2CCN2C(C2CNC(=O)N2)=O)ccc(-n2ccnc2)nc1 n1(COC(=O)CC2CCC(F)(F)C2)nnc(C(N2CCCC(C)C2)=O)c1N.CCOC N1(C(CSCC)=O)CCC2C(CCCN2C(c2cscc2OCCC)=O)C1 c1(OC)ncc(Cl)cc1C(=O)NC1CC2(C1)CC(C(=O)NCCOc1cccnc1)C2 C(CN=[N+]=[N-])(C(=O)N(C(C)C(C)C)C1CC1)NC(CC1(OCC)CC1)=O C(=O)(C(CCC(N)=O)N=[N+]=[N-])N1CCN(C(c2c(CC)nccn2)=O)CC1C C(=O)(CCCCCF)NCC(C(=O)NCc1c(C)csc1)CC1CC1 C12(C(=O)NC(Cn3cc(-c4cc(NC)c(C)cc4)nn3)C)CCC(O)(CC1)CC2 C1(OC)CN(C(C2CCCN(C(C)C)C2)=O)C2(CCCC2)C1 CC(C)CC(O)CNC(=O)C(CCF)NC(c1ncccc1N)=O C(CC(=O)NC(C(O)CO)C1CC1)(C(C)C)NC(C(n1ccc(C)n1)C)=O Cc1cnc(C(=O)NC(C)(CNC(=O)C(N2CCCCCC2)C)C2CCC2)cn1 C(=O)(CC1=CCCCC1)CC(N1CCCCCC1C1CCCC1)=O N#Cc1ccc(F)c(C(N2CC3CC2CN3C(=O)CCCN2CCCC2)=O)c1F C1(NC(c2ccc(C#C)cc2)=O)CC2CC(NC(C3OCCO3)=O)CC2C1 c1(C(=O)NC2CCN(C(Cc3c(C)scc3)=O)C2C(C)C)cc2n(n1)CCO2 CN1CC=C(CC(=O)N2CCCN(C(=O)CN3CC(C)(C)C3)CC2CO)CC1 c1(C(=O)NCCCC(C)(C)NC(CC2C(C)CCCC2)=O)nc2ncccn2n1 C(=O)(C1CCc2c[nH]nc21)NC1C(NC(=O)Cc2ccccc2Cl)CCC1 C1(CN(C(C2CCC(CC)O2)=O)C)CN(C(c2conc2C)=O)CC12CC2 N1(C(C(C(C)C)SCC)=O)CCC2(CCCN(C(=O)CC3CCC(=O)NC3)C2)C1 CN1CC(C(N2CC3CC3(C(=O)NC3C4CCCOC34)C2)=O)CC1=O N1(C(CC=C)=O)CCC2(CNC(=O)CCSCCCC)CCCCC12 Cc1cccc2c1OC(C(=O)NC1CC(C)CN(C(C3CC(C)N(C)C3)=O)C1)C2 N1(C(c2c(C)nco2)=O)CCC(C(=O)NCC2CC(O)C23CCC3)C(O)C1 c1(C(N2C(CNC(c3ncsc3C3CC3)=O)CCC2)=O)cc2c(cc1Cl)NCC2 N(C1c2ccccc2OCC1F)C(c1c(C)ccc([N+](=O)[O-])c1C)=O c1(CN2CC3C(C(N4C(C(C)C)COCC4)=O)C3C2)ncccc1[N+](=O)[O-] C1(C(NOC(C(=O)OC)C)=O)CN(C(=O)CCP(C)(C)=O)CC1(F)F c1(SCC)ccc([N+](=O)[O-])cc1C(=O)N(C(=O)Cc1sccc1S(N)(=O)=O)CC CC(C)C(C)(O)C(=O)NCC12CC(CN1C(c1[nH][nH]c(=N)c1Br)=O)C2 C1(OC)CC(O)CN(C(=O)C(C)NC(=O)CN2CCCCC2=O)C1 N1(c2ncnc(C)c2C#N)CC2CCCC(NC(=O)CN(C)C(N)=O)C2C1 C=CCCCC(C(=O)NCCCNC(C)=O)NC(c1cccn1C)=O N1(C(C2CN(C)C2)=O)CCCC1CCC(=O)N(C1CC1)Cc1ccoc1 S(=O)(=O)(c1cccc(Cl)c1)NC1CCC(CC(=O)NC(c2ccccn2)C)CC1 N1(C(CCOCC)=O)CC(C)CN(C(C2(C)CCC(=O)NC2)=O)CC1C C1(NC(=O)C(C2CCCCC2)F)CN(C(=O)Cn2nccn2)CC1C1CC1 Cc1ccccc1CC(N1CC2(NC(=O)CSc3ccccn3)CC1C2)=O Cn1ccc2c(C(=O)NC3CCCCC3NC(C34CC(F)C3C4)=O)ncnc12 N1(C(C(=O)NCc2ccc(OC(C)C)cc2)=O)CCCC2NC(=O)CCC12 CCCC(C)=CC(=O)N(CC(=O)N(CC(C)C)C(C)C)CC(C)C c1(CN2CC3CN(S(CC=C)(=O)=O)C3C2)ccc([N+](=O)[O-])cc1Br CC1CC(C(=O)NC(CNC(c2cc(-c3ccccc3F)no2)=O)CO)CN1C N1(C(c2c(CC)cccn2)=O)CCC(F)(F)C(O)C1.c12ccsc1C(=O)NC2 Cc1c(C(N)=O)cccc1C(=O)NC1CC2(C1)CN(C(c1cncc(O)c1)=O)C2 C1(C(=O)NC2(CNC(C(COCC)C)=O)CC(F)(F)C2)CCCS(=O)(=O)C1 C1(C(N2C(CC)CN(C(=O)Cc3cc(OC)no3)CC2)=O)CC(C)(C)OC1(C)C c1(C(N2CC(NC(CC(=O)NCC#C)=O)C(F)CC2)=O)ccc2nn[nH]c2n1 C=C=CC(C)C(=O)NC1CC(OCC(=O)NC(C)(CO)C2CCC2)C1 Cc1noc(N)c1C(=O)NC(c1nocc1C(=O)NCC1CC(=O)N(C)C1)C N1(C(C(CC2CC2)NC(C=Cc2ccc(C)o2)=O)=O)CCc2nncn2CC1 CC1CN(C(=O)C(C#N)CC2CC2)CC1NC(=O)C(C)Sc1cccc(F)c1 Cc1cncc(CC(=O)N(C2C3CN(c4cc(C(F)(F)F)ncn4)CC23)C2CC2)c1 C(CCC(=O)NCC(CNC(=O)C(O)C1CC1)CO)OCC=C CC1C(N(C(=O)C2=CCN(C(c3ccc(=O)n(C)c3)=O)C2)C)CCCC1C Cc1ccc(C(N2CCCC2C(C)NC(C23CCN(CC2)C3)=O)=O)nc1C C(=O)(C(C)C(F)F)N(C(C)CNC(=O)Cn1ccnc1)CC N1(C(C2C(CNC(C(C)C(F)F)=O)CCO2)=O)CCC2C(O)C(C)(C)C12 c1(CC)nc(Cl)[nH]c(=NCC2(C)CCCN(C(=O)C(n3cc(Cl)cn3)C)C2)c1Cl O=C(CN=c1cc[nH]cc1)NC(C(=O)NC1CCCOC1)c1cccs1 C(=O)(C(F)(F)CF)NC(C)C(c1ccc(O)cc1)NC(=O)COc1ccccc1 CCCCCC(CC)C(=O)NC1CCCC12CN(C(c1nccc(Cl)c1F)=O)C2 C1(CC(N2CCC(N(C(c3cnc(CSC)s3)=O)C)C2)=O)CCNC(=O)C1 Cc1ccn(C)c1C1CN(C(C(CO)CO)=O)C(=O)C1CC N1(C(c2nc(C)sc2C)=O)CCN(C(=O)CCc2cn[nH]c2)C(c2cn[nH]c2)C1 c1(SC)nscc1NC(=O)C(c1cnn(C)c1)NC(c1ccc[nH]1)=O C#CC(C)(C)C(=O)NCC=CCC(=O)NCC1(CSC)CC1 c1(C(=O)Nc2ncc(-c3cc(OC)cc(C)c3)cc2C)cc(OC)c(O)c(Cl)c1 N1(C(C2C(OC(C)=O)C2)=O)CC2(COC(CNC(C3(C(C)C)CCC3)=O)C2)C1 c1(N(C2C(C)CCNC2)C(=O)CCCn2cccn2)cc(C#N)ncn1 c1(NC(C(=O)NC)=O)cccc(C(N2CCC(NC(C)=O)C2)=O)c1 C1(CCC)CN(C(c2ccccc2Cl)=O)CCN1C(=O)CCC1(C)CCC(=O)N1 N1(C(c2cnc(C(=O)OC)s2)=O)CC2(CCCC(CNC(=O)C(C)O)O2)C1 C1(C)(CNC(C2C=CC(NC(C(CC=C)N(C)C)=O)C2)=O)CCC(=O)N1C C1(NC(c2c(OCC(C)C)n[nH]c2)=O)CC2CN(C(=O)CSC3CC3)CC2C1 C1(NC(c2c(C)noc2C)=O)CC2CCC1CC2NC(=O)CSCCC(F)(F)F C(CC(CC)C(=O)NCC(C)N(C(c1cc(C(F)F)no1)=O)CC)=CC C1(C(N(CC(CN(C)C)O)C)=O)CSCN1C(C1(CF)CC1)=O Cc1ccc(C(=O)OC(c2cccc(C(F)(F)F)c2)C)c(C)c1.C1(=O)CCCO1 N1(C(CNC(=O)OC)=O)C2CCC1C(C(=O)NCCc1cnc[nH]1)C2 C1(C(=O)NCC#CC(=O)NCc2ccc(CC)o2)CC(N=[N+]=[N-])C1 C1(c2cn(CC(=O)N(C)C)nn2)COCCN1C(c1ccc(Br)o1)=O C#CC12CCCC1CN(c1nnc(C3=CC(Br)=S3C)n1CC)C2 N1(C(C(C)=C2CC2)=O)CCC(C)(CCNC(c2nsnc2O)=O)C1 C1(C(N2C(C(N)=O)CC2)=O)(NC(C23CCC(C2)C3)=O)CC=CC1 C1(N(C(CCOCC(C)C)=O)C)CCN(C(=O)C(COC(C)(C)C)C2CCC2)C1 c1(OCC(=O)NCC2CC2NC(c2nnc(O)cc2O)=O)cc(F)cc(Cl)c1 CC1CC(CNC(=O)CCNc2ncccn2)CN1C(c1sc(F)cc1Cl)=O c12cccc(c1)CO2.c1(-c2cn(C(C(C)O)C)nn2)cnc(C(=O)O)nc1 c1(C(=O)NC2C(NC(c3cc(COC)oc3C)=O)C2)ccc2c(n1)CCC(C)C2 c1(CC)cc(C(N2CCC(CC(=O)NC(C)C3CC3)C2)=O)on1 C12(CNC(C(CCC)(C)C)=O)CCCC1CN(C(c1cnc3n1CCOC3)=O)C2 C1(C(N(CCCCCC)CCO)=O)CC2CC2N1C(C1C2C=CSC12)=O N1(C(c2c(C)cccc2C)=O)CC2CCCC(N(C(=O)CC3CCCC3)C)C2C1 C(C(CNC(c1nnc(S)n1C)=O)S(C)(=O)=O)NC(c1cncc(OC)c1)=O O(NC(=O)C(c1cccnc1)NC(c1ccc(Cl)cc1)=O)CCCC N1(C(C2(OC)CCN(C(c3coc(C(F)F)c3)=O)C2)=O)CCC(F)(F)C(O)C1 CC1CN(C(=O)CCC(C)(C)C)CC(C)CN1C(=O)CC#N C1(NC(C2(OC)CCSC2)=O)CN(C(=O)Cc2c[nH]nc2C)CCC1CO C1(CC)CN(c2cc(NCC(C)(C)C3CC3)ncn2)CC(CC)O1 C1(C(=O)NC23CC(NC(CCc4c(C)noc4Cl)=O)(C2)C3)CCC2(CCC2)CO1 N1(C(C2CCCC(=O)N2)=O)CCC12CN(C(=O)C(O)CC1CCOCC1)C2 C(=O)(C1CSc2ccccc21)N1CC2(CC(CNC(CCNC(=O)CO)=O)C2)C1 c1(C(N2C3C(NC(CC=CCC)=O)CC(C3)C2)=O)c(C)sc2ccc(F)cc12 C1(C(N2CCC(NC(c3c(C)cns3)=O)CC2C)=O)CCc2ccccc2O1 C1(CN(C(Cc2c(C)csc2)=O)C)CCCCN1C(c1sc(C2CC2)nc1C)=O CCC(C(=O)NCC(=C1CN(C(c2c[nH]nc2-c2cccs2)=O)C1)F)C(F)(F)F N1(C(C2C(CC)CCO2)=O)CCC(C(=O)Nc2cc(C)cnc2OC)C(O)C1 c1(C(N2CCC(NC(=O)CO)C(F)C2)=O)cnc2c[nH]nc2c1 c1(C(CCC)OC)nc(-c2ccc(Cl)cc2)nn1-c1ccc(F)cc1 C(=O)(C1=NN(C)C(=O)CC1)NC1C(NC(c2c(OC)cccc2C)=O)C1 C1(c2ccc(C)o2)(C(=O)N(CC(N2CCC(N(C)C)C2)=O)C)CCOCC1 C1(C(=O)NC2(C)CCC(NC(=O)COC(F)F)CC2)CCc2n[nH]cc2C1 C1(N(C)C)COCC1NC(=O)C(c1cccnc1)NC(=O)C=CC1CCC1 c1(C(=O)OC)ccc(CC(=O)NC2CCCC2NC(=O)CSC(F)F)s1 N1(C(C(c2n(C)ncc2)(F)F)=O)CC2(CCN(C(C3CCC(=O)NC3)=O)CC2)C1 c1(C(CCC)C)nc(CCC(=O)NCC(F)(F)F)n(-c2nccn2C)n1 C=C1COCC1C(=O)NCC1(CC2CCC2)CC1 c1(NC(C2C(NC(C=CC(C)C)=O)CCCC2)=O)nc(Cl)ccc1Br N1(C(CN(C)CC)=O)CC2(CCN(C(=O)C(C)(C)n3cncn3)CC2)C1 C1(N(CC)CC)CCCN(C(=O)Nc2coc(C(N)=O)c2)C1 c1(C(=O)NCc2c(C)c[nH]n2)c(CNC(C23CC(C#N)(C2)C3)=O)cnn1C C12(C(N3CC(O)CC(C)(O)C3)=O)CC(CCO1)N(C(C1CC1C1CCC1)=O)C2 c1(C(N(C(CNC(CC(=O)OCCC(C)C)=O)C)C)=O)ccc2ncn(C)c2c1 N1(C(CCC(=C)C)=O)CCCC(NC(=O)C(c2ccncc2)C)C1C CCCC(C(=O)NCC1(C)CN(C(=O)COC(C)=O)CCO1)C(C)C c1(C(N(C)CC2CCCN(C(c3cnc(OCC)s3)=O)C2)=O)c(C)cccc1Cl O=C(CC(O)CSc1ccccc1)NC1CCCC1NC(C1CCCC1CF)=O c1(C(N2CCCC(NC(C(C)NC(=O)NC)=O)C2)=O)cc(F)cc(Cl)c1N Cc1ccc(OCC(=O)N(C)C(C)C2CC2)c(Cl)c1 N1(CC(=O)Nc2cccc([N+](=O)[O-])c2F)C(=O)C2CC=CCC2C1=O c1(C(=O)NC(CNC(C2(Cl)CC23CCC3)=O)CO)cc2c(O)cccc2[nH]1 C12(NC(C3CN(C(c4c(C)snc4)=O)CC3(F)F)=O)CCC(CC1)C2(C)C Cc1ccnn1C(C)C(=O)NCC1CC(O)(CNC(c2cc(Br)no2)=O)C1 C1(O)(CN(C(=O)CSC(F)F)C)CCN(C(c2cc(F)ccc2O)=O)CC1 C(N=c1[nH]c(=NC2CCCCCCC2)c2cc(Cl)ccc2[nH]1)C1CN(C(=O)OC)C1 C(=O)(CC(C(C)(C)C)NC(C1CCCSC1)=O)N(C1(CO)CCC1)C C12(NC(c3cnc(C(C)(C)C)[nH]3)=O)CC1CN(C(C1CCCOC1)=O)C2 C(CN=C(NCC1CCCN(C(=O)C(C)(C)C)C1)NC1CSC1OC)=CCCC C#CCCCCC(C(=O)Nc1ccc(C(=O)OC)cc1)N1CC(=O)N(C)CC1C C(=O)(C(O)CC1CCOCC1)NCC(C)(C1CC1)NC(c1cc(C(N)=O)c[nH]1)=O Cc1[nH]nc(C(N2CCC(CCC(=O)NCC3CC3(F)F)CC2)=O)c1Cl c1(NC(=O)Nc2c(C(=O)NC3CC(=O)NC3)cc(F)nc2)ccc([N+](=O)[O-])cc1 c1(C(=O)NC(C2C3CC4C(C3)C24)C)ccc(-n2cc(Br)cn2)nn1 c1(CNCCN(C(c2ccc(Cl)cc2)C)C)nn(C)c2c1CCC2 N1(C(=O)Nc2ncc(COC)s2)CCC2(C1)OCCO2 CCCC(CC(=O)NC1CC2CCC1(CO)C2)NC(c1ccnc(C)c1C)=O C(=O)(CCC(C)S(C)(=O)=O)N(C1CCN(C(=O)CCCCC(=O)OC)CC1)CC c1(CNC(C#C)Cc2ccccc2)ccc2c(n1)OCCO2 C1(CC)(CNC(C2CN(C(=O)C(C)CC3CC3)CCO2)=O)CCOCC1 C1(CN(C(=O)C(C)c2cncs2)C)CCN(C(C2CC2Cl)=O)CC1 CC1(C)CC(CC(N2CC(=C(F)CC(=O)NC(=O)CSCC3CCCC3)C2)=O)C1 C1(OCC)CC(N)(C(=O)Nc2ccc(Oc3cccc(CC)c3)cc2)C1(C)C N1(C(=O)Nc2c(CCOCCOC)ocn2)CCCC(c2cn(C)cn2)C1 C(=O)(C1CCCc2c[nH]nc21)NCC(CNC(c1cc(CC2CCC2)c[nH]1)=O)F C1(C(=O)NCc2ccc(C#N)o2)CC2C=CC1N(C(C1(Cl)CC1)=O)C2 CCCCC(CNC(C1CCC(N(C)C)CC1)=O)NC(=O)CCC(N)=O C1(C(=O)OC)NC2CC1CC2NCc1ccc(CSN(C)C)cc1.c1(C)ccccc1 N1(C(C=CC(CC)=CC)=O)CCN(C(=O)CCCC2CC2)C(c2nccn2C)C1 C1(C2CN(C(=O)CC(C)NC(N)=O)C2)(NC(c2nc(C(C)OC)oc2)=O)CC1 N1(C(CCCCC)=O)CCC2(CCC2)C(CNC(c2c(CO)noc2C)=O)C1 CCC(CN(C(=O)C(F)C1CCCC1)CC)NC(=O)Cn1ccnn1 C1(CNC(C(C)CN(C)C)=O)CCN(C(c2cccc(C(F)(F)F)c2)=O)CC1C C(N=c1[nH]c(=NCN(C)C)[nH]c2c1COC2)C1CCCN(S(C)(=O)=O)C1 C(=O)(CC(F)(F)C(F)(F)F)N1C2CC(NC(c3cn(CC)nc3)=O)(C2)C1 C1(C(=O)NC2C=CCN(C(c3cnc(SC)nc3O)=O)C2)CCc2nc[nH]c2C1 N1(C(c2ccc(C(N)=O)cc2)=O)CCN(Cc2cn3ncccc3n2)CC(O)C1 N1(C(CCc2cc(C)no2)=O)CCN(C(=O)C#CC2(C)CC2)CC2CCCCC12 C1(NC(CCN(CCC)C)=O)(COC)CCN(C(c2cc(C(F)F)cs2)=O)CC1 c1(CC)c[nH]nc1C(=O)NCC1CC(O)(CNC(C23CSCC2C3)=O)C1 C(C(C(=O)NCC1CNC(=O)CO1)C(C)(C)C)NC(c1ccc(CC)cn1)=O CC(C)CCC(O)C(=O)NCC1CN(C(c2c[nH]cc2C2CC2)=O)C1 C1(CC(=O)N(CC(C)NC(=O)CCC(C)(C)C)C)Oc2ccccc2NC1=O c1(NC(COC2CCN(C(C(CC)N(C)C)=O)C2)=O)ccc(C)c(C)c1F C1(CN(C)C(C2CCC(=O)N2)=O)CCCN(C(c2ncc[nH]c2=O)=O)C1 Cc1nc(-c2cccc(Cl)c2)sc1C(N1CCC1CN(C)C)=O CCC(C(=O)NCCCCC(C)NC(c1cc(C)n(C(C)C)c1)=O)C(C)C CCC(C)C(CN(C)C)NC(N1CC(C)C12CC2)=O C1(CNC(CCOCCCNC(=O)C#CC2CC2)=O)CC12CCOCC2 C1(C(N2CC(C(C)NC(=O)C#CC(=O)N(C)C)OCC2)=O)CCCN2CCCC12 C(=O)(C#CC1CCCC1)N1CCC(CNC(c2cnc(C#N)s2)=O)C1 C(=O)(C1CCOc2ccccc21)NCCCN(C(c1c(C)ccc(OC)n1)=O)C C1(OC)CC(C(=O)N(C)CC2CCSC2)N(C(=O)C(C)c2ccsc2)C1 CCC(CC)CCCC(=O)N1CC(NC(C2(OC)CCOC2)=O)CC(C)C1 Cc1cc(S(N)(=O)=O)ccc1OC(c1ccnc(C)c1C)=O c1(C(=O)NCC2CN(C(c3ccc(Cl)c(Br)c3)=O)CCO2)cccc2c[nH]nc12 N1(C(c2nccc(N(C)C)c2)=O)CC(C2CN(C(=O)C=CCF)C2)C1 C1(NC(COCCC(C)C)=O)CN(C(=O)Cc2n[nH]c(=N)s2)C(C)(C)C1 c1(C(=O)NCC2N(C(C3C(OC)CCC3)=O)CC2)c(C)ccc(N)c1C C1(NC(C2CCC=CCCC2)=O)CCN(C(C2(Cl)C3CCC(=O)C23)=O)CC(O)C1 C=CCC(CNC(=O)CCC1CCCO1)NC(=O)Cc1coc(C(F)F)n1 C1(SC)CN(C(c2cscc2C(N)=O)=O)CC1NC(=O)C(C)N1CCC1 C1(C(=O)NCc2c(C)ccc(C)n2)CC(C)(C)CCN1C(C1CC(O)CN1C)=O C(=O)(C(C)C(=O)N1CCC(NC(=O)CSc2nc[nH]n2)CC1)OC C1(NC(C)=O)CN(N(C)C2CCc3ccccc3C2C)C1 c1(OC)cc(C(=O)Nc2cccc(NC(=O)C3CC3)c2)ccc1C(F)(F)F c1(C(N2CC3C(NC(C4=C(C)CCC4)=O)C3C2)=O)cccc2c1COC2 c1(CC(N2CC(CNC(C(C)=C3CC3)=O)C(C)(C)C2)=O)ccc2nn[nH]c2c1 C1(C(=O)NCC(CC=C)NC(c2nnc(O)nc2O)=O)CCCC12CCOCC2 Cc1nc(NC(C2CC3(CC3)CN2Cc2ccc3c(c2)CCO3)=O)c(Br)cc1Br C1(C(N(CCNC(=O)CCc2cc[nH]n2)CC2CC2)=O)CC2(C1)CC(O)C2 C1(C(N(CCCNC(c2coc(O)n2)=O)CC)=O)C2CCC1(C(N)=O)C2 C(c1cncnc1O)=CC(=O)N(C1CCC(Nc2ccnc(CO)n2)CC1)C O=C(C#CC1CCOCC1)NC1CCOCC1NC(=O)CC1COCC1O c1(C2(CC(=O)N(C3CCCC3)CCNC(=O)C(F)C3CC3)COC2)ccccc1 CC1CCN(C(=O)CCCN2CCCCC2)C1CNC(=O)C1=CCCC1 N1(C(c2cncc(N(C)C)n2)=O)CC2(CNC(C3(N(C)C)CCC3)=O)CCC1C2 N1(C(COC(Cc2ccc(C)o2)=O)=O)CC(C)CC(C)C1 C1(NC(c2n(CCCC)ncc2)=O)CC(C)CN(C(c2ccnc(Cl)c2O)=O)C1 C1(C(N(CCC)CC2CCN(C(c3sccc3C)=O)CC2)=O)NC(=O)OC1C C1(CNC(C2CCC(=C)CC2)=O)CC2(C1)CN(C(c1csc(Cl)c1Cl)=O)C2 N1(C(CCNC(CCCSC)=O)=O)CC(C)CC1(C)C C1(CC(=O)NC2CCC(CNC(CCC3(C)CC3)=O)C2)CCCC(F)(F)C1 c1(C(=O)NCCC(C)N(C(CCOCCOCC)=O)C)ccc(F)c(C#N)c1 C1(CC(C)C)(C(=O)NC2CCCC2NC(C2CSCC(=O)N2)=O)CCNC1=O N1(c2ncc(S(=O)(=O)NCCC(C)F)cc2Cl)CCc2cc(Cl)cc(F)c2C1 C(C(C(=O)NCC(C)N(C(c1ccnc(O)c1)=O)CC)C(C)(C)C)OCC=C c1(CC)ccc(NC(c2n[nH]cc2NC(=O)CO)=O)cc1 C1(C(N(CCS(C)(=O)=O)CC)=O)CCCN(C(=O)OCCl)CC1.C(C)(C)(C)O c1(CC)ccnc(C)n1.n12cc(nn1)CCOCC(O)CN(C)C(=O)CCC2 c1(C(=O)NC(C(C)C)CO)cnc2ccc(C3=CC(C)(C)C3)cn12 C1(OCC)CC2CN(C(C3CCN(C(C4CNC(=O)C4)=O)C3(C)C)=O)CC12 C1(NC(CCC(=C)C)=O)CC(C)CN(C(=O)C(C(C)(C)C)C2CCC2)C1 c1(C(=O)NCC(C)NC(C(C#C)(C)C)=O)cc2[nH]nnc2cc1OC N1(C(C(C)OCC)=O)CCCC(CN(C(c2cnc(C3CC3)[nH]2)=O)CC)C1 N(S(=O)(=O)N1CC(C)OC(C)C1)(CC)Cc1ccc(F)cc1 C12(C(=O)NCc3c(CC)nn[nH]3)CC(CO)(CN1C(C1CC3CCCC3C1)=O)C2 C(C)(C)(C(=O)N(CC(C)NC(=O)CNC(=O)OC(c1ccccc1)CO)C)OC N=c1[nH]c(=NCc2ccoc2)[nH]c(=NC2C3C4CCC(C4)C23)[nH]1 c1(CC)cc(C(=O)NCC2CC3CCC2N3C(=O)CN2CCC(C)C2)ccc1O c1(NC)ccc(-c2ncc(C(F)(F)F)cc2Cn2cc(COC(C)C)nn2)cc1F C12(CCNC(CNC(CN(C)C)=O)=O)CCC1CN(C(c1nnn(C)c1N)=O)C2 CCCCC(C(=O)NCCCCCNC(=O)Cc1cccc(CC)c1)N(C)C c1(NC(=O)NC(C)C(=O)N(C)C)n[nH]c2cccc(-c3cccc4nonc34)c12 c1(OC)ccc(C(C)OC)cc1OC.C(C)(C(C)NC(=O)NC1CC1)NC=O c1(C(N2CC(NC(C(CC)NC(C)=O)=O)C(F)C2)=O)cccc(F)c1O c1(OC)c(Cl)ccc(C(=O)NCC(C2(O)CCN(C(=O)Cn3nccn3)C2)C)c1F C1(C(N(C(C)C(=O)NC2CC(CSC)C2)CC#C)=O)CC2CCCC2C1 c1(OC)ccncc1C(N1CC(NC(C2CC(OC)C2)=O)C2CC12)=O N1(C(C(c2cccc(C)c2)=O)=O)C2CCC1C(F)C(NC(c1cccs1)=O)C2 C=C(Cl)C(C)(C)C(=O)NCCOC1CN(C(c2ccc(NC)cc2)=O)C1 C(=O)(CS(=O)(=O)C1CC1)N1C(C)CC(CNC(c2cn(CCC=C)nn2)=O)C1 c1(C(=O)NC(c2cc(F)ccc2F)C)ccc2c(c1)S(=O)(=O)CCC2 N1(C(c2c(C)con2)=O)CC(C(=O)NCC(C)(O)C(F)F)C(F)(F)C1 C(=O)(C(Cn1cccn1)NC(=O)COC(F)(F)F)NCC(C)(C)C1CC1 CCC(C)CC(C)C(=O)NC1CCC(CNC(=O)CC2CCOCC2)C1 C1(C(=O)Nc2cccc(NC(c3c(CC)onc3C)=O)c2)CC2(C1)CC(F)C2 C1(Cl)(C(=O)NCCC2OCCCN(C(C3(OC)CCC3)=O)C2)CC12CCOCC2 C1(CC)CN(C(=O)OC(C)(C)C)CCC1NC(=O)Nc1nccs1.C1CSC1 Cc1c(C(=O)N(CC(=O)Nc2cnc(O)c(F)c2)C)[nH]ccc1=O N(C1c2ccccc2CC1O)C(=O)Nc1nccs1 CCC(CC)C(C(=O)N1CC(NC(C23CC(CO)(C2)C3)=O)C(F)C1)OC C1(CNC(CCCC)(CC)c2nnnn2C2CCOC2)CC2C3CCC(C3)C2C1 Cc1nn2c(c1C(=O)NC1CC(NC(=O)C(C)OCCC(C)C)C1)CCCC2 c1(CNC(c2cccc(CC(F)(F)F)c2)C2CC2)ccnc(Cl)c1F C1(CC(=O)OC)CN(Cc2ccc(-n3cccc3)c(F)c2)C2COCC2O1 N#CC1CCCCN1C(C1CC(O)CN1C(=O)CCC(F)(F)F)=O C=CC(CC)CC(=O)N1CCN(C)CC1C(=O)NCCC(C)(C)C#CC c1(C(N(C2CCC(NC(c3nccn3C)=O)C2)C)=O)cn2c(n1)CCCC2 N1(C(c2c(C)snn2)=O)CCC(O)(C(C)CNC(c2cc(C(N)=O)c[nH]2)=O)C1 Cn1cccc1CCC(=O)N(CCCNC(C1CC(O)C1)=O)CCO Cc1cnc(O)n1-c1cccc(C(N2CCC(C(C)NC(=O)C=CCF)C2)=O)c1 C1(C(=O)NC(CC=C)CNC(=O)C(F)(F)C2CCCCC2)(CC)CCCSC1 N1(C(Cn2cc(-c3cc(C)no3)nn2)=O)CCCC1P(C)(C)=O C(Cc1ccccc1)(C(=O)NC1(C)COC1)NC(=O)OC c1(C(=O)NCC(CNC(C(C=C)O)=O)(C)C)c(C)[nH]c(-c2ccncc2)nc1=O n1(CC)nc(C(=O)NCC=CC(=O)NC(C2(C(=O)OC)CC2)C)ccc1=O c1(C(c2ccn(C3CCC3)n2)NC(c2cc(CO)[nH]n2)=O)ccccc1 c1(CNC(=O)NC2CC2CN2CC3CC(CO)C(C3)C2)ccc(F)c2occc12 c1(OCC(N2CC(OCCNC(c3occ(C)c3C)=O)C2)=O)cc(F)cc(F)c1 C1(NC(CC=C(C)C)=O)CCOCC1C(N1CCC1CN=[N+]=[N-])=O C(=O)(C1=CC2CCC(C1)C2)N(CC(N1CC(C#CC)C1)=O)C c1(C(=O)NCC2(C(C)(C)O)CN(C(CC=CC)=O)C2)cc2c(s1)CCCNC2=O C(=O)(CCCC(=O)NC1CC(O)(CNC(C2(C)CCCO2)=O)C1)N(CC)CC C1(NC(c2scc(C)c2C)=O)CN(C(c2ncsc2C(C)C)=O)CCC1CO C1(CNC(CC=C)=O)CN(C(c2cccnc2C(F)F)=O)CC1c1ccccc1 Cc1cc(O)cc(=O)n1CC(N1CCCC1(C)CNC(c1nccnc1Cl)=O)=O C1(C(N2CC(CCNC(C(C)NC(C)=O)=O)C(C)C2)=O)CCC(F)(F)CC1 C1(NC(C(CC=C)(F)F)=O)CN(C(=O)Cn2cnnc2)C2(CCOCC2)C1 c1(C(C)C(=O)NCC(C)(O)CNC(=O)CC#N)cccc2ccccc12 Cc1cc(Cl)ccc1CNCCCCCCn1cc(C(C)(C)O)nn1 N1(C(C2C(NC(c3ccnc(C)n3)=O)C=CCC2)=O)CCC2CN(C)CCC12 CC(C)(CF)C(=O)NC1CCC(C(=O)NCCCC(=O)Nc2scnc2C)CC1 C(=O)(N=c1ccn(CCCO)[nH]1)C1C(CNC(C(C)SC(C)C)=O)OCC1 N1(C(C2N(CC)C(=O)CC2)=O)CCCCC(CNC(=O)CN2CC(=O)NC2=O)C1 C(=O)(CC(C)C(C)(C)C)N(C(C(=O)NCc1c(CC)onc1C)C)C Cc1cc(C(=O)NCC2(NC(c3cnc(O)o3)=O)CCCCCC2)c(F)cc1F C1(C(=O)NC(C(C)C)CCNC(c2cc(Br)co2)=O)CCn2ccnc2C1 N1(c2nnc(C#N)s2)CCN(CC(=O)NCC2CCN2C(=O)CC2CCCC2)C(=O)C1 n1(CC(N2C3CN(C(CC(CCC)O)=O)C(C3)C2)=O)c([N+](=O)[O-])cnc1C N1(C(CC(OCC)OCC)=O)CCCC(F)(C(=O)NCc2cnns2)C1 C(=O)(CS(=O)(=O)c1ccccc1Cl)N1CCN(C(=O)CC2CCC(F)(F)C2)CC1 N(C1CCCc2sc(Br)cc21)CCC=CCN c1(C(N2CCC(NC(C(CC)NC(N)=O)=O)C2)=O)cc(C)c(N)cn1 C=Cn1ncc(C(=O)N(CCC(=O)NCC=CCCOC)C2CC2)c1N c1(C(=O)NCC(C)Cc2cn[nH]c2)cc2c(ccn2C)s1.C12CCCCN1CC2 c1(C(N2CC(NC(C(C)CC(C)(F)F)=O)C2)=O)cc2c(s1)CCCCCC2 c1(C2N(C(c3c(F)cccc3Br)C(=O)NC)CCNC2)nc2ccc(C)cc2[nH]1 C1(OC)CN(C(=O)CN2CCOCC2=O)CCC1NC(=O)CCC1CCCOC1 C1(N(C)C(c2cc(Br)c[nH]2)=O)CN(CC(=O)NCc2ccccc2)CCC1O CC1CC(NC(C2CC2C(F)(F)F)=O)CN(C(=O)C=Cc2cncc(Br)c2)C1 Cc1ccc2c(c1)CC(C(=O)NCC1(F)CN(C(=O)C(C)OCC(C)C)C1)S2 C(CC(C(=O)Nc1cnn(CC(C)C)c1)NC(c1nc(C)oc1C)=O)OCC C(C(C)(O)CC(=O)NCC#CC(=O)NCc1ccc(OC)cc1C)OC N1(C(CN(C(=O)CC2CCOC2(C)C)C)=O)CCCC(O)(C#C)C1 c1(OC)ccc(CCC(N2CCN(C(c3ncsc3C3CC3)=O)CC2)=O)cn1 N1(C(C2CC(C)OCC2)=O)CCCCC12CN(C(=O)CN1CCOCC1)C2 c1(C(C(=O)NC(CCSC)CO)NC(=O)C(C)N=[N+]=[N-])c(C)cccc1Br N1(CC=C)C(=O)c2ccc(C(=O)NCCN(C(=O)CC3(O)CCC3)C)cc2C1=O c1(OC)ccccc1C(C)C(=O)NCCC(O)CNC(=O)CC1CCC1 C(=O)(C(C)(C)CCO)NC.C12(CCC(OC(C)(C)C)CC1)C(=O)OC2.OC C=CC(CCC)CC(=O)NCC(CNC(=O)COc1cn[nH]c1)S(C)(=O)=O N1(C(c2cc(C)oc2)=O)CCCC(NC(=O)C(N2CCOCC2)C)CC1 c1(OC)nc(C(N2CC(NC(C3(O)CCOCC3)=O)C(O)C2)=O)sc1C C=CCCCCCC(=O)NCC1(C)CCCN1C(c1ccc(C#N)c(Cl)c1)=O N1(C(CCCCC=C)=O)CCC2(C1)CN(C(=O)C=C1CCCC1)CC(C)O2 C1(OC)CN(C(=O)OC(C)(C)C)C(C)(CNCC(C2CCCCC2)O)C1 c1(NC(C=NOC)=O)cccc(NC(=O)CC2CCN(C(C)=O)CC2)c1 c1(C(N2CC(C(C)NC(c3c(C)cc[nH]3)=O)OCC2)=O)nnc2ccccc2c1 C1(N(C(=O)NCc2nccc(OC)c2)Cc2ccccc2)CC2(CCC2)C1O CC(C)C(C)(C)C(=O)NCCCC(O)C(=O)NCCNC(=O)CO C1(CN(C(C(C)=C(C)C)=O)C)CCCN(C(c2cnc(C(C)C)[nH]2)=O)C1 C1(C(=O)NC(c2cccnc2)C(C)C)CCc2nc(C3=COCCC3)sc2C1 c1(CC)nc(N2CC3CC2CN3C(C2CCCN2N=O)=O)cc(C#N)n1 CCC(C)(C(F)(F)F)NC(=O)CCN(C(c1cccnc1S)=O)C1CC1 c12ccc(cc1)CN(C(C(=O)NCC(=O)OC)C(C)C1CC1)C2.C1(C2CC2)CC1 C(c1cnn(C)c1)=CC(=O)NCC(CN(C(C(Cc1c(C)nc[nH]1)O)=O)C)C CCCCC(C(=O)NCC1CC(NC(=O)C(C2CCCOC2)OC)C1)C(C)C Nc1ccc(C(=O)NC2CC(O)(CNC(c3coc(CO)c3)=O)C2)nc1N N1(C(c2ccc(OC)s2)=O)CC(NC(c2c(Cl)cnn2C)=O)CC1C N1(C(CC(CC)CC)=O)CCCN(C(=O)CN2CC(=O)NC2=O)CC1CO N(C(=NCC(C)c1cccc(F)c1)NC1CCCCC1)Cc1c(CC)noc1CC C=CCCCC(=O)NC1CCN(CCCSC)C1.C12CC1NC2=O c1(C(=O)NC(CNC(COCC=C)=O)CCCC)oc2ccccc2c1COC N(C1CCSc2ccc(F)cc21)C(N(CC(c1ccccc1)C)C)=O C1(NC(C(C)n2cncn2)=O)CC(O)CN(C(=O)CCc2c(Cl)cccc2Cl)C1 CCC(CC)C(=O)N1CCOC(Cn2cc(Cn3ccsc3=O)nn2)C1 c1(CC(N2CCC(C)(NC(C(C3CCOC3)OCC)=O)C2)=O)ccc(O)c(Cl)c1 N1(C(c2cn(CCCOC)nc2)=O)CCCC2CN(C(C3CC(C)C3)=O)CCC12 C(=O)(Nn1cnnc1CC)C1CCC(C(N2CC(C(=O)OC)(CC)C2)=O)O1 C1(NC(C2CCCNS2(=O)=O)=O)CCC2(CC1)CCN(C(c1ccon1)=O)CC2 C(=O)(C1=NN(C)C(=O)CC1)N1CCC(CC#C)C1.C12CCCCN(C1)C2=O CCC(CCC(=O)NCC1CC1Cl)NC(C1Cc2nccn2C1)=O C1(C(=O)NC(CNC(N)=O)C(C)C)(NC(Cc2ncc(C)o2)=O)CCOCC1 c1(C(=O)NCC2(F)CN(C(C(C(CC)O)(C)C)=O)C2)cc(F)c2cn[nH]c2c1 C(=O)(CCC1=CCCCC1)N1CC(C(=O)NCC(C(C)(C)C)CO)(CCO)C1 O=C(C(O)C1=CCCCC1)NCC1CCN(C(C2(C3(O)CCC3)CC2)=O)C1 C(CNC(=O)CNC(c1ccsc1)=O)(CC(C)C)NC(CC(C)OC)=O N1(Cc2n(C)cnc2)CC2CC(NC(=O)OC(C)(C)C)CC(C2)C1 CCC(CCCC(=O)NC1CC2CC1C(O)C2O)NC(c1csnn1)=O CC1C(NC(C2(CCN(C)C)CCCC2)=O)CC2CCC1N2C(=O)CN(C)C1CC1 N1(C(=O)NCCc2ncc(C)cc2Cl)CCCC2(CCCO2)C1 C(=O)(CCOC(=O)C=C(C)C1CC1)N1CCCC1.CCC(C)N(C)C c1(C(=O)OC)cc(NC(=O)C2=COCCC2)cc(CO)c1.c12cc(on1)NC2=O Cc1nc(CC(=O)NC2CC(C(C)NC(C3CCCC(O)C3)=O)C2)[nH]c1C N1(C(C(CCCC)CC)=O)CCCC2CN(C(=O)Cc3sc(C)nc3C)CCC12 c1(OC)ccsc1C(=O)NC1(C(=O)OC)CCC1.C12CC1C(=O)NC2 CCC(O)CC(=O)N1CCCC(CCNC(=O)CN2CCN(C)CC2)C1 C1(CCCC)CCCN(C(=O)CONC(c2conc2C)=O)C1 N1(C(COC(CC)(C)C)=O)CC=CC1(C)C(=O)NC(C1CCCCC1)C(N)=O N1(C(CCCC)CN(c2ccccc2C)C(=O)CCC)CCCC(C2CC2(F)F)C1 C(=O)(C(CNC(c1c[nH]nc1OC)=O)C(C)(C)C)NCC(C(CC)(C)C)O CC(CCC(C)(C)C)C(=O)NCCC(C)(C)CNC(C1C=CCCC1)=O CC(C(=O)NCC1CN(C(C2C3CC4C(C3)C24)=O)C1)C(F)(F)F C1(CC)CN(C(=O)C(c2ccccc2)C)CCN1CC(=O)Nc1cc(Cl)cs1 N1(C(C(C2CCC(C)CC2)CC)=O)CC(C)(C)CC1CNC1OCCC1(C)C N1(C(C(=O)NC2CCOC2)c2ccoc2)CCN(C(C2CC=CCC2)C2CC2)CC1 c1(-c2cn(CC(C)(C)O)nc2)nc(CCCO)nn1CC1CC2CCC1C2 C1(CC(=O)NCCCN2CCCC2)CCN(C(c2cncn2C(F)F)=O)C1 c1(C(N2CC3CC(NC(C4(F)CC4)=O)CC2C3)=O)nc[nH]c2ncc(Br)c1-2 c1(C(N2C3C(NC(c4c(C)nc(C5CC5)[nH]4)=O)C(C3)C2)=O)cnc2[nH]nnc2c1 N1(C(CC2(NC(C)=O)CC2)=O)CCC2CC2(C(=O)N(c2ccccc2)CC)CC1 N1(C(c2ccc(C)cn2)=O)CC2CCC(C1)N(C(c1ccsc1C)=O)C2 C(C1=NOC2CN(C(C3(O)CC3)=O)CC12)NC(Cc1ccc(S(N)(=O)=O)s1)=O C12CCN(N3CC=CC3CO1)C2.c1ccc(CCn2ccnc2)nc1 N1(C(C(CCC)c2ccccc2)=O)CC(C(N2CC(O)C2)=O)C(F)(F)C1 C#CC1(F)CCN(C(C2(CCC)CCN(C(C3CC(SC)C3)=O)C2)=O)CC1 c1(C(N(CC(C)NC(C2(C(=O)NC)CC2)=O)C)=O)cn(C2CCCCC2)nn1 C1(CNC(C2C(OCC)C2)=O)CN(C(c2cn(C3CC3)nn2)=O)CC1(F)F Cc1ncc(C(=O)NC(C)CC(C)NC(c2cccc(F)c2)=O)n1C N1(C(C(C)CF)=O)CCC2(CC1)CCN(C(C1CC(F)CN1)=O)C2 C(=O)(CC(F)(F)C(F)F)NCC1OCCN(C(C2CC(C(C)C)OCC2)=O)C1 Cc1cc2nc(NC3(CNc4cc5ncnn5cn4)CCC3)cc(=O)n2o1 C1(C(=O)OC)OC(C(=O)NCC2COCCN2C(=O)Cn2cnnc2O)CC1C C1(NC(C2CCC(NC(C3C(=C)C3C(=O)OC)=O)C2)=O)CNC(=O)C1(C)C Cc1ccc(C(=O)NC2(CNC(c3cccc(F)n3)=O)CC2)c(F)c1F CCCCC(CNC(=O)CC1CC(C(F)F)C1)NC(C1(C)CC1C)=O Cc1ccc(C)c(C(=O)NC(C)C(=O)N(C)CC2COC(=O)N2)n1 Cc1c(F)ccc(Cl)c1C(=O)N(C)CC1CCCN1C(=O)CC1COCCO1 C1(CC(=O)NCC(C)CN(C(=O)C(F)(F)c2cccnc2)C)CC=CCC1 c1(C(N(C2CCN(C(C3(CC)CCOC3)=O)CC2)C)=O)cc(F)c(F)cc1O CC1CCCCC1(CNC(C1CCCSC1)=O)NC(C1CC2(CCCO2)C1)=O C(=O)(C(C(F)(F)F)C(F)(F)F)N1C(C)CC(NC(=O)CNc2nccs2)C1 N1(C(C(CCCC)F)=O)CC2CC(NC(=O)C=C(C)c3ccco3)CC1C2 c1(OC)cc(Cl)c(Cl)cc1C(=O)NCC1COC(C)(C)CN1C(C1CCCO1)=O C=CCC(C)C(=O)N1CCC(C)C1CNC(=O)COc1cccc(Cl)c1 N1(C(C2N(c3cc(OC)ncn3)CC2)=O)CCc2c(Cl)cc(Cl)cc2C1 c1(C(C(=O)NCC(=C)CCNC(C23CCC2C3)=O)O)ccc(F)cc1 c1(OC)cc(I)c(C(N2CC(C(=O)Nc3cc(Cl)sc3Cl)C2)=O)cc1OC C1(C(N(CCCC(C)C)CCO)=O)COC2(C1)CN(C(=O)C=C(C)C)C2 c1(CCC)ccc(OCCCCC(=O)NC(CC)CO)cc1 N1(C(CN(C2COC2)CCC)=O)CCN(C(=O)C2CC2)CC1c1ccncc1 C1(C(=O)NC2CCN(OC)CC2)CC2CCCC2N1C(C1CC2CCC(C1)C2)=O C1(C(=O)NCC2(C)CCOC2)CC12CCN(C(C1CNC(=O)O1)=O)CC2 C1(C(NCP(C)(C)=O)C)CCCCCC1NC(=O)CCCC1CCCO1 N1(C(c2cnc(OCC)nc2)=O)CCN(C(c2ncc(Br)cc2Cl)=O)C(CO)C1 c1(NC(C(C2SC(=N)NC2=O)C)=O)ccc(C(F)(F)F)nc1N(C)C Oc1cnc(CNCc2cccc(OC(F)F)c2)c(O)c1 c1(SCC)cncc(C(=O)NCC(C2CCCCC2)(C)NC(c2cnc[nH]2)=O)n1 c1(C(=O)NCC(CCOC)NC(C(C)SCCCC)=O)cn2cccnc2n1 C1(CCN(C(C=C(C)Cl)=O)C2CC2)CCCCN1C(=O)CC1CCCOC1 N1(C(CCCCCC#N)=O)CCn2nc(CNC(c3cnsn3)=O)cc2C1 C1(C)(C(=O)NCC(C(C)C)(C)NC(=O)COC2CC=CC2)CCC12CCC2 N12CCN(C3CCCCC13)C(=O)c1ncc(s1)C2=O.c1(OC)ccccc1C#N N1(C(c2c(C)ccn2C)=O)CCC2CC2(NC(=O)C(=Cc2c[nH]cn2)F)CC1 c1(C(=O)NC(c2nnn(-c3cccc(C)c3)c2C)C)ccnc(F)c1C c1(C(N(CCNC(C(C=CC)O)=O)CC)=O)nnn2c1C(=O)NCC2 c1(CC(=O)NCC(=O)OCc2ccccc2)cccnc1Br C12(CNC(C(C)C3CCOC3)=O)CCC(CC1)CN2C(c1coc(C#N)c1)=O N1(CCC)CCCC(C(=O)NC2CCC(NC(C34CCC(C3)OC4)=O)CC2)C1 CC1CCc2c(NC(C3CN(c4nc(Cl)nc5c4COCC5)C3)=O)csc2C1 C1(CN=[N+]=[N-])CCN(C(=O)CCNC(=O)CN2CSCC2=O)CC1 N1(C(C2C(C(C)C)CCO2)=O)CCC(C(=O)NC2(C)CC(CO)C2)C(C)C1 N1(C(c2cc(CC)on2)=O)CC2OCCN(C(c3cc4ccsc4n3C)=O)C2C1 c1(C(=O)NC(C2CN(C(c3cc(OC)n[nH]3)=O)C2)C)ccc2[nH]c(C)c(C)c2c1 Cc1ccccc1C=CC(=O)NC1CC(C)N(C(c2cn(C)c(=O)cn2)=O)C1 C1(C(=O)NC(c2cnsc2)C)CCN(C(C2CCCN2C2CC2)=O)CC1C c1(C(C)=O)cc(C(=O)N(CC(C)NC(C2CCC(=O)N2C2CC2)=O)C)c(C)o1 C=CC1CN(C(=O)CNC(=O)C2CC2)CC1NC(=O)Nc1cccnc1Cl C(=O)(CCCCC(=O)NCC1CC(C(=O)N(CC(C)(C)CO)C)=NO1)OC N1(C(c2nc(OCC)oc2)=O)CCC(C(=O)NC2CC2c2ccsc2)C1C(C)C c1(SCC(c2ccc(Br)cc2)C)ccccc1NCC(C)S(C)(=O)=O Cc1c(C=CC(=O)N(CCNC(c2conc2C(C)C)=O)C2CC2)cnn1C C(=O)(C(C)(C)CS(C)(=O)=O)N1CC(C)C(NC(=O)CNC=O)C(C)C1 c1(SCC(=O)NC2CC(C)(NC(c3ccc(NC)nc3)=O)C2)ccc(F)cc1F Cc1cn2c(C(N3CC4CC3C4NC(c3cc(C4CCC4)[nH]n3)=O)=O)cnc2s1 c12cc(nc(C)n1)NC(C)CN2.c1(CCC(C)SCC)ccccc1 c1(C(=O)NCC(C2CC2)OC)c(CNC(C2CCS2(=O)=O)=O)cnn1C Cc1ccc(C(=O)NC(C2CCN(C(=O)C=Cc3cocn3)C2)C)c(N)c1F c1(CCCOC(C2(CCC)CC2)=O)ccc(I)cc1 Cc1cc(C(=O)NC(C)CCNC(c2cc(C3CCC3)[nH]n2)=O)ncc1C(F)F c1(OCC)ccc2cc1-2.c1(C(N(C)CC)=O)ccc(F)c(Nc2occc2Br)c1 CCC(CNC(C1(NC(=O)CC(CC)c2ccc(Br)cc2)CC1)=O)CC(F)(F)F c1(C(=O)NC2CCC(CNC(C(CC(C)C)O)=O)CC2)cn(C)c2ccccc12 C1(C2CCN(C(=O)COCC3CCCO3)C2)(NC(C(C)CF)=O)CC1 CC1=C(C(=O)N(CC(C)NC(c2ccc(Br)c(C)c2)=O)C)CCCC1 C1(NC(Cn2ncc(CC)c2)=O)CC(NC(=O)Cc2cnc[nH]2)C12CCC2 C1(C(=O)NCC(CC)(C)NC(=O)CC2CCC2)CCCC(=O)N1 c1(C(=O)NCC(CN(C(=O)CCF)C)O)c(S(N)(=O)=O)ncn1C C12(C(N3CCC(F)(CNC(=O)CCCCc4cnc[nH]4)C3)=O)CCCC1C2(F)F C(=O)(C1=CC2(CCOCC2)C1)N1C(C)C(NC(=O)C=CC2CCCO2)C(C)CC1 N1(C(c2cncc(F)n2)=O)CCC(C2CCN(C(C3CC3F)=O)CC2)C1 C(CCCC(=O)NC1CC(C)N(C(c2cnn(C3CC3)c2)=O)C1)OCC C(=O)(C(C(C)CC)N(C(=O)CCOCCOC)C)NCC(C#C)(C)C CC1(C)C(NC(=O)C(F)n2ccnc2)C(C)(C)C1NC(=O)CCC1CCCO1 C(CCC(=O)N1CCCC1CCNC(=O)COC1CC1(F)F)SC C(=O)(C(C(C)(C)O)NC(=O)C(C)C1(O)CCC1)NC(CCC)CCO c1(NCc2c(C)cccc2)cc(N(C)Cc2nnc(CO)s2)nc(C(F)(F)F)n1 C12(C(N(C)CCC3CCN(C(CCC(=C)C)=O)CC3)=O)CC(CO)(C1)OC2C N1(C(c2ccc(C)c(C)c2)C(=O)OC)CC2CCN(C(C3C4COCC34)=O)C2C1 C(C(CC(C)C)C(=O)NCCC(=O)NC(N)=O)NC(C(CC=CCC)C)=O N1(C(C2(C)CC2(F)F)=O)CC2CCN(C(=O)CCc3cccc(Cl)c3)C(C2)C1 C1(C(C)C)C(=O)NCCN1C(c1cc(CCNC(=O)CC2CC2)on1)=O C1(NC(c2cn(CCC)nc2C)=O)CC2(CCN(C(=O)C(O)C(C)(C)CC)C2)C1 N1(C(CC(C)CF)=O)CC2(CNC(c3cnn(Cc4cccs4)c3)=O)CC1CO2 c1(C(N2CCC(F)(C(=O)Nc3cc(Cl)c(Cl)cc3I)C2)=O)c(Cl)ccnc1Cl C(=O)(C(F)C(C)CC(C)(C)C)NCCN(C(=O)C(CC)N(C)C)CCC C(=O)(CN=c1[nH]c(N2CCNC(=O)C(F)(F)C2)nc2c1CCCC2)N1CCC(C)C1 C1(C(=O)NCC(CNC(c2cnsc2C)=O)OC)(CC)CCCCO1 N1(C(C2C(C)(C)C2(C)C)=O)CC2CC(C(=O)NCCCO)(C2)C1 c1(C2(OCCO)COC2)cccc(Cl)c1.N12CC3CC3(C1)Nc1ccnc(n1)C2=O Cc1ccc(C(=O)NC(CNC(=O)Cn2cc(C3CC3)cn2)C2CCC2)nc1C C12(CNC(c3c(SC)ccs3)=O)CC1CN(C(=O)C(C)(C)O)C2 C1(C)(NC(C)=O)CCN(C(c2ccc(OCC3CC(F)(F)CO3)cc2)=O)CC1 c1(N(C)Cc2scc(C)c2)[nH]c(=NCCCn2cnnc2)nc2sccc12 c1(OC)ccc(S(=O)(=O)NN(C(=O)CCCC(N)=O)S(N)(=O)=O)c(CC)c1 N1(C(C(C(=O)OCC)(C)F)=O)CC2OCC(NC(C3CCS(=O)(=O)CC3)=O)C2C1 C12(NC(=O)C(F)(F)F)CCCN(C1)C2.C1(CCCF)CC2CCCC12 c1(C(=O)NC2C(CNC(c3c(CCC)n[nH]c3)=O)C2)cc2c(C)cccn2n1 CC1(C)CC(C(=O)NOCC(N)=O)CN(C(=O)C(F)C(C)(C)O)C1 Cc1n[nH]c(C)c1CNC(C1CCN(C(=O)C(C)C2(O)CCC2)C1C(C)C)=O C1(CNC(C(C)(C)OC)=O)CC(C(=O)OC)C12CCC2.C12CC(C1)NC(=O)C2 N1(C(C(CC#C)C)=O)C(C)C2CC1C2NC(c1ccc(Cl)c(F)c1)=O N#Cc1cnc(NCC2CCCN(C(=O)CC34CCC(CC3)OC4)C2)c(Cl)c1 Cc1ccc(CC(=O)N(CC(O)CN(C)C(C2CCCCC2(F)F)=O)C)c(Cl)n1 C1(NC(c2cccc(OC(F)F)c2)=O)CN(C(=O)CCC2CC2)CCC1CO c1(C(=O)NCCCN2CCN(C(CC(CC)O)=O)CC2)cnc(C)nc1C(C)C C(=O)(C(O)C(F)(F)F)Nc1cccc(-n2cc(-c3scc(C#N)n3)nn2)c1 c1(CNC(c2cncc(CC)n2)=O)cc2n(n1)CCN(C(C1CC3(CC3)CO1)=O)C2 C1(CNC(CC2CCC(SC)O2)=O)CCN(C(C2(OC)CCCCC2)=O)CC1O Cc1[nH]nc2c1CCC(C(N1CCC(C)N(C(=O)CCCCC(N)=O)CC1)=O)C2 c1(C(N(C2CN(C(=O)CCCCCC(C)(C)C)C2)C)=O)c[nH]c(=O)c2ccncc12 c1(OC)ccc2c(c1)CCCC2c1noc(Cc2cccc(OCF)c2)n1 CS(=O)(=O)c1ccc(C(=O)NC2CC(CNC(C3(F)CC=CC3)=O)C2)cc1 C1(C(N(CCOCCN(C(C(C)=C(C)C)=O)C)C)=O)CCc2cnc(C)n2C1 c12ccc([nH]1)C(=O)N(CC)C2.c1(NC(CCO)C2(C(=O)OC)CC2)ccccc1 c1(C(=O)NC(C(C)NC(C(COC)(F)F)=O)CO)c(F)cc(C(F)(F)F)cc1F C1(NC(=O)C=CC2CC2)CCCC(NC(c2ccc(-c3ccccc3)cc2)=O)C1 N1(C(C2CN(OC)C(=O)C2)=O)CC(C(N2CC3(CC(F)C3)C2)=O)C2(CC2)C1 Cc1cc2c(cc1C)C(C(=O)N1CCOC(CNC(=O)C3=CCCS3)C1)CO2 C=Cc1ccc(C(N2C(C(=O)NCCOCC3CCCC3)CC2C)=O)cc1 CC(C)C(C)(O)C(=O)NC1CN(c2nnc(-c3ccccc3)o2)CCC1C CC(C)(C)C(C#N)C(=O)N1CCC(CNC(C2CCC23CCOCC3)=O)CC1 CC1c2ccccc2CCN1C(=O)C(c1cccc(Cl)c1F)(F)F c1(C(C)(C)C)nc(CNC(=O)CC2(O)CN(CC(O)C=Cc3cnc[nH]3)C2)n[nH]1 C(=O)(C1=NOC(C)C1)NCCN1CCC(NC(C(CCC)=CC)=O)CC1 C1(F)(C(=O)NCCCN(C(C)C)C(c2ccc(C(C)F)cc2)=O)CCOCC1 n1(CCC)nccc1C(=O)N(CC(N1CCC1C(=O)NCC(C)C)=O)C c1(NCOC2C(C(=O)O)CCC(N(C)C)C2)ccc(CC#N)c2c1OC(F)(F)O2 C1(C)(C(=O)NCC2(O)CCN(C(C3C(C)OCC3)=O)CC2)CC2CCC(C1)S2 C12(CC(=O)NC3(CO)CN(C(=O)CN(C4CCC4)C)C3)CCCC1C2 C1(C(N2CCC(CC(=O)NC3C(C)(C)C3(C)C)C2)=O)CC2C(C1)C2(C)C Cc1ccc(SCC(=O)NCC2CCC2NC(C2CCN(C3CC3)CC2)=O)cc1 CC1CN(C(=O)C(=Cc2c[nH]cn2)F)CCCN1C(=O)C=CCN1CCCC1 C1(NC(=O)OC(C)(C)C)CC(O)CN(C(C2(C#N)CC2C(F)(F)F)=O)C1 c1(C(N2CC(CC(=O)NC(c3nn(C)cc3O)C)OCC2)=O)ccc(Cl)c(Cl)c1 N1(C(c2c(C)nccn2)=O)CC(NC(=O)Cc2cccc(F)c2O)CC12CCC2 C1(CNC(=O)C(=O)Nc2cccc(Br)c2)CCCN(C(c2ccns2)=O)C1 C(=O)(C#CC1CCOC1)NCCCCN(C)C(C1CCCCCC1(F)F)=O c1(NC(C2CN(C(C(=C)F)=O)CC(C(F)(F)F)C2)=O)cc(O)c(OC)c(O)c1 CN1C(=O)C(=O)N(CC(N2CCN(C(C3CSCCS3)=O)CC(CO)C2)=O)C1=O CC1(C)C(C)(C(=O)NC2CCCCN(C(c3cn(C4CC4)nn3)=O)C2)C1(C)C c1(CNS(C)(=O)=O)ccc(C(=O)NC2CC(NC(C34CCCC3C4)=O)C2)o1 C(=O)(CC(F)(F)CC(=O)N(C1CCCN(C(C2CCCN(C(C)=O)C2)=O)C1)C)OC N1(C(C2N(C(c3cc(COC)on3)=O)C(C)CC2)=O)CCCC(F)(F)C1 c1(-c2nc(-c3c(Cl)ccc(CC)c3)n(CCCC(F)F)n2)cc2ccccc2[nH]1 N1(C(CCC=CC)=O)CCC(C(=O)NCCC(CCC)C2CC2)C12CC2 N1(C(c2nc(CCC)sc2)=O)CC2CC1CCC2NC(=O)C=C1CC(CC)C1 CCC(CN(C)C)CC(=O)NCC1(O)CC(C(=O)N(C2CCN(C)C2)C)C1 C1(N(C)C(C23CCC(CO2)C3)=O)CCCCN(C(=O)C=Cc2cncs2)C1 C(=O)(C(F)(F)C(F)F)N1CCCC(C(C)NC(c2cc(C)nnc2)=O)C1 Cc1nc(C(N2CC3CC3(CNC(=O)C(F)C(C)(F)F)C2)=O)ccc1C#N c1(CC)cccc(C(=O)NC2(CCCCNC(C3CCCCCC3)=O)CC2)n1 c1(NCCO)ncnc2sccc12.C12COCCN(C1)Cc1c(cccc1)C2=O C1(CNC(C=C(CCC)C)=O)CCCC12CCN(C(C1OCCCO1)=O)CC2 C(C(CC(C)C)C(=O)N1CCC(C(N2CC(C)CCC2CO)=O)C12CC2)OC C1(C(=O)NC2(CC=C)CCN(c3cc(=O)n(C)cn3)C2)CCCC2(C1)CC2(F)F C(=O)(CC(O)C(Cl)(Cl)Cl)NC1CCCCCN(C(C2(COCCOC)CC2)=O)C1 C1(CNC(COCCC)=O)CC2CN(C(c3cccc(-n4cccn4)c3)=O)CC12 Nc1ccc(OC(=O)CCc2ccccc2Br)cc1.C1CO1 CCCCCS(=O)(=O)CC(=O)NC(C)CCNC(=O)C(n1ccc(C2CC2)n1)C S(=O)(=O)(C1CN(C(=O)OC(C)(C)C)C1)CCNC(=O)NC(C(C)O)(C)C C1(C)(CC)C=C(C(=O)NC2CN(C(=O)Cn3cnc(C(N)=O)n3)CC2C)C1 N#Cc1csc(C(=O)NCCCN(C)C(c2ccc(C(N)=O)s2)=O)n1 C1(C(N2CCC(NC(=O)C#CC3CC3)C(F)C2)=O)CCC2C(CC1)C2(F)F N1(c2nc(OC)c(C)cn2)CCC(C2CCN(C(=O)CC(=O)NC3CC3)CC2)C1 c1(C(N2CCC(CN(C)C(C3CC4C(C3)C4(C)C)=O)C2)=O)cc2n(n1)CCCC2 C(=O)(CCCCCNC(c1scnc1C)c1nnnn1CC(F)F)OC Cc1ccc(NC(=O)CCC(=O)O)nc1 CC1CCCN(C(=O)CC2COCC2(C)C)C1CNC(C1CN2CCN1CC2)=O C(=O)(C(c1ccccc1)=C(C)C)OC(=O)C(C)Nn1nc(C)oc1=O C1(=CCN)CCN(C(c2cc(N3CCCC3)ncn2)=O)CC1.CC(C)(C)C=CC=O N1(C(CC(CC)OC)=O)CCCC(C)(NC(=O)CC(C)(C)c2ccc(C)cc2)C1 C1(NC(=O)C=CC(F)F)CC2(C1)CC(NC(c1cc(O)ncn1)=O)C2 c1(C(N2C(CN(C(=O)C=Cc3cn[nH]c3)CC)CCC2)=O)ccc(C)cc1N c1(CC(=O)NC23CC2CN(C(=O)C=Cc2ccco2)C3)cn2cc(F)ccc2n1 C1(NC(CC2(OC)CC2)=O)CCCN(C(c2ccnn2-c2ccncc2)=O)C1 C(=O)(CC(C)C(C)C(C)C)N1CCC(CNc2nc(OC)cc(OC)n2)C1 c1(C(=O)NC(CCCNC(c2n(C(C)C)ccn2)=O)C)ccc(O)cn1 C(=O)(C(F)(F)C(O)CC)N1CCCC(CC)(NC(=O)CCC(=O)NCC)C1 N1(C(c2cc(CC)c(C)s2)=O)CCCCC(NC(c2sccc2Cl)=O)C1 CC1CCC(CN2CC(C)(NS(C)(=O)=O)C2)CC1C.C12(CCC1)C(=O)N2 c1(C(N2CCC3(C(N4CCC(=C)CC4)=O)C(C2)C3)=O)ccc(Br)c2cccnc12 Cn1nc(COC(C2CCNC2=O)=O)cc1C(C)(C)C C1(NC(CCN(CCCCC)C)=O)CN(C(c2cncc(C)c2)=O)CC1(C)C C(=O)(CS(=O)(=O)NC1CC1)NCC1(F)CC(NC(=O)CCN2CCC2)C1 C1(C(=O)OC)C(F)(F)C12CC(C(N1CC(CN(C(=O)C(F)=C3CCC3)C)C1)=O)C2 N1(CCC(=O)NCCNC(C2CN(C(C=C(C)Cl)=O)C2)=O)CCCCC1C Cc1cc(C#N)nc(NC(C2CC(O)CN2c2nc(C)cc(C#N)n2)=O)n1 c1(C(=O)NC(CC)CNC(c2sc(C(C)(C)C)nc2C)=O)cc[nH]c(=N)c1N CN1CC2CC1C(=O)O2.c1(SC)ccc(F)cc1.c1(C2CN2)ccccc1 C(CCN(C)C)(C(=O)N(C)CC1CCSC1)NC(c1c(C)cc[nH]1)=O c1(NC(C2(C)N(C(Cc3cc(C)n(C)n3)=O)CCC2)=O)ncc(CO)cc1Br C=C1CCC(C(=O)NC2(C)CCN(C(=O)CC3CC4(CC4)CO3)C2)CC1 c1(CCC(=O)NC2CC(NC(=O)Cc3ccsc3)C2)cnc(SC2CCCC2)o1 C=CCCCCC(=O)N1CCC(C(C)C)CC1CNC(c1c(OC)noc1C)=O N1(C(C2CN(C(C(N)=O)=O)CC(F)C2)=O)CC2CNC(=O)C2C1 N1(C(c2occ(C)c2C)=O)CCCC(C)C1CNC(c1sccc1CN(C)C)=O n1(CC(=O)NC2C3CCN(C(Cc4cc(OC)no4)=O)C32)cc2ccccc2n1 N1(C(C(C(C)C)OC)=O)Cc2n[nH]cc2C1C(=O)N1CC(C2=NOCC2)C1 C1(COC)CN(C(=O)CCCCC2CC2)CCN1C(=O)C=CC(C)(C)SC C(=O)(C1=CC2CCCCCC12)NCCCCCNC(c1c(C#N)scc1)=O CCC(C)C(C)(O)CNC(C1CN(C(=O)CSC2CC2)CCO1)=O c1(CC(N2CCC(NC(c3c(C)ccnn3)=O)C2C2CC2)=O)nc(F)c(F)cc1F n1(CCC)ncc(CN2CCCCC2CNC(C2CC2C2CC2)=O)c1C N1(C(C=CC=CC)=O)CCCC(C)(C)C1CNC(c1cc(C2CC2)[nH]n1)=O O=C(C1=NOC(C2(O)COC2)C1)NC1CCCCN(C(c2ccc(F)cn2)=O)C1 c1(CNC(C(CC2CN(C(C(C=C)C)=O)C2)F)=O)ccc(F)cc1F C1(CC(=O)NCC2(F)CN(C(c3c(C)ncs3)=O)C2)CCCCC12CC2 N1(CC)CCC(NC(=O)N(C)CCOCC2(C)CC(OC)(OC)C2)CC1 CCC(CC)(CO)C(=O)N1CCCC(N(C(=O)Cc2cnc[nH]2)C)C1 C=CC1CN(C(=O)CCC(=O)OC(C)(C)C)CC1N(C(C1CCCO1)=O)C(C)C N1(C(c2ccoc2Br)=O)CCC(CNC(C2COC2)=O)CC1 c1(N(CCCNC(Cc2c(CC)n[nH]c2CC)=O)C(C)C)cnc(C#N)cn1 C1(C(=O)NC(c2noc(C)n2)CC)CCCN1NC(=O)c1ccnn1CC N1(C(C2C(C)CCN2C(C2(C)CCN(C)C2=O)=O)=O)CC2(CNC(=O)N2)C1.CCO N1(C(c2csnn2)=O)CCC(F)(c2cn(CC3C4CCCC34)nn2)C1 c1(CC(=O)NC(CCN(C(C2CC(OC)C2)=O)C)C)sc(C2CCC2)nc1C Cc1nnc(Nc2cc(CNC(C3C(NC(=O)OC(C)(C)C)C3)=O)on2)s1 C(=O)(C1COc2ccccc21)NCC(CNC(c1c(C)noc1C)=O)S(C)(=O)=O Cc1ccc2cc(C(N3C4CCC3C(NC(c3cccnc3S)=O)C4)=O)oc2c1 C(=O)(CS(=O)c1ccc(Cl)cc1)NCC(CC)NC(=O)CC1CC(C)(C)C1 c1(C(N(CCCN(C(C=C(C)C2CC2)=O)C)C)=O)cc(C2CCCC2)nn1C C1(OC)CN(C)C(C)(C(=O)NC2CC(NC(c3cnc(N)c(Br)c3)=O)C2)C1 c1(CC(=O)NC2(C(=O)NCC3N(C(C)=O)CCC3)CCSC2)ccc(C)cc1 N1(C(=O)CCN2CCCS2(=O)=O)CCN(C(=O)Cc2ccc(F)cc2)C2(CC2)C1 C(=O)(CC(C)P(C)(C)=O)NC1(CO)CCN(C(c2c(C)csc2)=O)C1 O=Cc1sc(CN2CC(O)CC2C(=O)Nc2ccc(O)cc2O)c(Br)c1Br c1(C(=O)OC)cc(Cl)c2[nH]c(-c3ccc(F)cc3)nc2c1.C1(=O)CCCCO1 C(CN=C(NCC(C)(C)C)NC1CCS(=O)(=O)C1)c1cnc(OC)c(Cl)c1 N1(C(C=C(CCN(C)C)Cl)=O)CCC(NC(C2C3CC4C(C3)C24)=O)C12CC2 O=C(CN=C(NC1CC1)NC1CC(c2ccc(F)cc2)C1)N1CCCC1 c1(CCC)cc(C(=O)N(C2CCCCC2N(C(=O)CC(C)(F)F)C)C)c(C)o1 c1(COCC(=O)NCCC(C)(C)NC(=O)CS(N)(=O)=O)ccc(F)cc1Cl C1(CN(C(c2cc(OC)ns2)=O)C)CN(C(C23CC(CO2)C3)=O)CCO1 c1(CC)cc(C(=O)NC(Cn2ccnc2)CC(=O)N2CCC(NCCO)C2)ncn1 N1(C(c2cc(F)cc(Cl)c2)C(=O)NCCCC)CCCC(F)(F)CC1 C1(CNC(c2coc3c2COC3)=O)CCCCN(C(C2C=CCC2)=O)C1 c1(C(=O)NCC2CC(O)CN2C(c2cc(=O)cc[nH]2)=O)cccc(Br)c1Cl N1(C(C(C)n2cnnn2)=O)CCC(C(=O)NCc2ccncn2)C(O)C1 c1(C(C)C)noc(CCC(=O)N(CCCCNC(=O)C(=O)NCC(F)(F)F)C)n1 c1(CN(c2ccc(Cl)cc2)C(C(C)C)(C)c2nnnn2C2CC2)cc(Br)ccc1Cl CC1COc2ccc(C(N3CCC(CNC(C4CC4C(N)=O)=O)CC3)=O)cc21 C1(F)(C(=O)NC(CSCC)(C)C)CCCN(C(c2sccc2OC)=O)C1 N1(C(C(C)C2(O)CCC2)=O)CCOCC1CC(=O)NC1CC1CC(C)(C)C C1(NC(c2ncn(C(C)(C)C)c2)=O)CC(C2CCN(C(c3cnsc3)=O)C2)C1 c1(C(C)(C)C#N)ccc(NC(C2CC(F)CN2C(=O)CCCC#N)=O)cc1 C(=O)(C(C)CC(F)F)NCCc1c(CNC(Cc2cncc(C)c2)=O)nco1 c1(C(=O)OC)cn(CNc2ccc3c(c2)c(C)nn3C)c(C)c(Br)c1=O C1(C(N2CCN(C(C3C4NC(=O)C(CC4)C3)=O)CC2)=O)CCc2nnc(O)n2C1 CC(C)CC(CNC(C1COCCN1CC(F)F)=O)NC(C1(C2CC2)CC1)=O c1(OC)cc(O)cc(OC)c1CN1CC2CC2(C(=O)Nc2ccc(Cl)c(Br)c2)C1 c1(C(=O)NCCOCCN(C(C2(C=C)CCC2)=O)C)ccc(F)c(N)c1 C(=O)(C(O)C)N.N1(CC(NOCC(C)(C)C)=O)CCOC1=O N1(C(C(F)OC)=O)CCCC2(C1)CN(C(C1(c3ncc(C)o3)CC1)=O)C2 N1(C(CC(=C)Br)=O)CC(OC)C(NC(C2CCCCC2)=O)C1 CC(C)(C)[Si](C)(C)OCCN(C(c1ccnc(O)c1)CC(=O)OC(C)(C)C)C(N)=O C=C(Cl)C(C)(C)C(=O)N1CCN(C(=O)CNC(=O)CN(C)C)CC1 CCS(=O)CC(=O)NC1CC1NC(=O)CC1(CO)CCCC1 Cn1nc(CNC2CC(NC(=O)OC(C)(C)C)C23CCC3)c2cc(F)ccc12 N1(C(C2C(CC)CCO2)=O)CCC(C(C)(C)C)(CNC(=O)C(C)n2ccnc2)C1 C(=O)(C(C)(C)C(F)F)NCCCN1CCC(N2CCN(C)CC2)CC1 c1(NC(C(c2cncnc2)C)=O)cn(C2CN(C(=O)NN3CC4CC4C3)C2)nn1 N1(C(C2C(C)C2(F)F)=O)CCC2CN(C(c3cn4cccnc4n3)=O)CC12 C12(NC(C3CN(S(C)(=O)=O)C3)=O)CCCC1CN(C(c1cncn1C)=O)C2 c1(-c2n(C(C3CCCO3)C)nc(C3CCCC3)n2)cnc(C2CC2)nc1O Cc1c(C(=O)NCCCC2(NC(=O)CSc3n[nH]c(=N)s3)CC2)cns1 C(C)(CC(C)NC(=O)CC1CC2CC2C1)NC(CN(c1ccccc1)CC)=O c1(OC)cccc(OC)c1C(N1CC(O)CC1C(=O)NCc1cc(Br)no1)=O C(=O)(CC(C(C)(C)C)NC(C1CC(C)CC(C)C1)=O)NCC1CC(OCC)C1 CCCC(CCC)C(=O)N1CCC(NC(c2ccc(C(C)C)o2)=O)C1C(C)C C1(C(N(CCCCNC(c2c(C)cns2)=O)C)=O)CC2(CCCC2)CO1 N1(C(c2c(CC)c(C)sc2)=O)CCc2nc(=N)[nH]cc2C1 C(CC(=O)NC(C(=O)N(C)CCC1CN(C)C1)c1ccco1)SCCC N1(C(C(CC=C)N(C)C)=O)CC2(CNC(=O)C=Cc3ccccn3)CCC1CC2 N1(C(CCC(C)CN(C)C)=O)CC2CCC(C1)N2C(=O)COc1cccc(O)c1 CC1(C(N2CC=CC(NC(=O)COCC3CCCO3)C2)=O)CCCCO1 N1(C(C2C(C)C2C)=O)C(C(=O)NC2CCS(=O)(=O)C2)CC2CC12 C=CC(C)(C)CCCNC(C1(NC(c2ncc(C)cc2F)=O)CCCC1)=O Cc1cnsc1C(N1CCC(C(=O)NCCc2c[nH]nc2O)C1)=O C1(CC(C)NC(C2N(CC)CC2)=O)CC2CCC(C1)N2C(c1cccc(Cl)c1)=O C1(C(C)NC(=O)CCc2cnco2)CN(C(c2cnn(C(C)C)n2)=O)CCO1 C(=O)(C(C(C)C)NC(C1CC1c1cnc(C)s1)=O)OC N1(C(c2nnn(C)n2)=O)C(CNC(=O)C(c2ccccc2Cl)O)CC2COCC12 C(=O)(C(C)(C)C(O)C(C)C)N(CCNC(c1csc(C)c1C)=O)C(C)C c1(C(N(C(C)C(=O)NCC)CCC)=O)c(NC(c2cnc(Cl)s2)=O)cnn1C Cc1ccc(C(=O)NC2CC(NC(c3c(C)coc3CC(N)=O)=O)C2)cc1Cl c1(OCC)ccc(CCNC(=O)CN2CCCC2Cc2nn[nH]n2)cc1 N1(C(c2ccc(SC)s2)=O)CC2CC2(CNC(c2cc(Br)ccn2)=O)C1 Cc1sc(=O)n(CC(N2CC(N)CC(N)C2)=O)c1C Cc1cncc(C)c1C(N1CC2CC2(CNC(=O)CCc2cnccn2)C1)=O c1(C(=O)OC)c(C(=O)NCC2(C)CCCN2C(C2CCC(=O)N2)=O)n[nH]c1C c1(CC(=O)NC2CCCC(NC(C3(C)CCCC3)=O)C2)c[nH]c2c(F)cccc12 c1(CNC(C(C2CN(C(c3occc3C)=O)C2)OC)=O)cn(C)nc1C CCC(C)C(C(=O)N1CCN(C(c2cc(OC)ns2)=O)C(C)C1)N(C)C c1(NC(C)CSC(F)F)nc(N2CC3C(C2)C3(C)C)nc2sccc12 Cn1nc2c(c1C(=O)NCC1(C)CCCN1C(C1C3COCC13)=O)COCC2 c1(CC)cc(C(=O)NCC(c2ccccc2)(C)NC(=O)C(C)OC)cc(F)c1 C1(CCNC(C2C(C(C)(C)C)CC2)=O)CN(C(c2ccccc2O)=O)CCO1 C1(OC)CN(C(=O)Nc2ccc(C(F)(F)F)cc2)CC1CC(C)(C)C C1(C(N(C)CC2(O)CN(C(c3nc(CCC)oc3)=O)C2)=O)(CCF)CCOCC1 C(CC(C)C)(C(=O)NC(C)CNC(=O)C(c1ncccc1F)(F)F)NC(C)=O C1(CNC(C2CCC(F)(F)C2)=O)C2CCC(C2)N1C(c1ccc(C(F)F)cc1)=O C1(NC(c2[nH]n(C)c(=O)n2)=O)CN(C(C2(C)CCCOC2)=O)CCC12CCC2 N1(C(C(CNC(C2(O)CCC(C)CC2)=O)O)=O)CCCC2CC1C2(C)C c1(NC(C=C)C)nc(N(C)CC)nc2sccc12 CC(COc1ccccc1)C(=O)NCC1CCN(C(=O)COC23CC(C)(C2)C3)C1 C=CCC(C)(C)C(=O)NCC1CN(C(C2CC(C)(O)C2)=O)CCO1 CN1CCCC1(C)c1cn(CCCNC(C2CC3CC3C2)=O)nn1 C1(C(=O)OC)CC(C)N1C(c1cc(CCNC(=O)C(C2CCC2)OC)on1)=O Cc1c(C)c(C)c(CN(C)CCN2CCC(F)(F)CC2)c(C)c1C c1(OC)ccc(Cl)cc1CC(=O)NCC1C(C)CCN1C(=O)CC1CSCCS1 C1(NC(=O)CC(F)F)CC2CN(C(c3cc(C(F)F)no3)=O)CC2C1 C(=O)(C(C(C)C)SC)NCCC1CN(C2(CNC(c3cc(CC)no3)=O)CC2)C1 CC(C)C(C)NC(=O)NC(C)CCN1CCCC1 C12(C(=O)OC)CCOCC1CN(C(c1cccc(CC(=O)OC)c1Br)=O)C2 CC1(C)C(NC(c2c[nH]ccc2=O)=O)CC1C(=O)NC1CCC(F)(F)C1 N1(C(C2CCN(C(C)C)CC2)=O)CC(C(=O)N=c2cco[nH]2)C2(CC2)C1 c1(CNC(=O)Nc2c(F)ccnc2Cl)cnc(N2CCCC2)c(Br)c1 CCCCCC(O)C(=O)N1CC(F)CC1CNC(=O)CCc1cccc(O)c1 N1(C(C2OCC(C)C2)=O)CCC(F)(CNC(c2cc(CO)n(C)n2)=O)CC1 c1(OC)ccccc1CC(=O)C(=O)NCC(CO)NC(c1nc(O)sc1C)=O c1(CN2CCOCC(C(=O)NC(C(CC)C)C)C2)cc2ccncc2[nH]1 N1(C(C(CC=C)C)=O)CC2CCC(CNC(=O)CC(CC)C3CCC3)C2C1 c1(OC)ccc(CCC(=O)N(C(C)CN(C(=O)CCC(C)O)C)C)cc1[N+](=O)[O-] c1(CC)ccc(C(=O)NCC2(CNC(c3ncccc3C)=O)CCC2)cc1 C1(C)(NC(C2C(C)CCC2)=O)CCN(C(=O)COc2ccc(CO)cc2)C1 C(=O)(C(C)(C)C(=O)NC1CN(C(C2CCCCC2)=O)CC1n1ccnn1)OCC C1(C(N2C(C)(C)C(CO)C2)=O)CCN(C(c2ccsc2)=O)C1(C)C C1(NC(C(CC(C)C)OC)=O)CC2CCC1CN2C(=O)CNC(=O)CSC C1(S(C)(=O)=O)(C(N2CCC(=CCNC(C(C3CCCO3)OC)=O)CC2)=O)CCC1 Cc1c(C(=O)N(CCCCC(=O)NCC2CCCCCCC2)C)cncc1F c1(C(N2CCC(F)(F)C(Nc3ncc4[nH]ccc4n3)C2)=O)c(F)cc(Cl)cc1Br C(N1CCOCC2(COCC3CCCN23)C1)N1c2ccc(S(C)(=O)=O)cc2CC1 c1(C(=O)NCC2CC(OC)CN2C(=O)C=Cc2cnc[nH]2)n[nH]c2c1CCSC2 CCCS(=O)(=O)C(C)C(=O)N1CCC(NC(c2cc(C)c(CC)s2)=O)C(O)C1 c1(CC(C)NC(C2CCC(CNC(c3ccc(CC)o3)=O)C2)=O)ccc(C)cc1 C1(C)(C(N(CC(C)NC(C2(C(=O)NCCO)CCC2)=O)CC)=O)CC(O)CN1C Cc1ncc(C(N2CCCC(CNC(c3ccc(O)cc3)=O)C2)=O)n1C c1(C(=O)NC2CCCN(C(CCCSC)=O)CC2)cc2c(nc1O)CCCCC2 C1(NC(C=CC(=O)OCC)=O)(COC)CCCN(C(c2ccc(F)cc2F)=O)C1 CCC(CC)C(C)C(=O)N1CC(O)CC1C(=O)N(C(C)C(C)(C)C)C C1(NC(Cc2cccc(OCC=CC)c2)=O)CCNc2ccccc2C1 C12(C(N3CC(OCC)C3)=O)CCCC1CN(C(=O)CC1CC3C=CC1C3)C2 Cc1cccc(C(C)CNC(N2CCN(c3ncc(F)cn3)CC2)=O)c1 c1(C(N2CCCC(CNC(=O)C=Cc3cnc[nH]3)C2)=O)cnn2c1OCC(O)C2 N1(C(CC(CC)(F)F)=O)CC(NC(c2ccc(Cl)cc2C(F)F)=O)C(C2CC2)C1 C#Cc1ccc(C(N2CC(OC)C(NC(c3c[nH]nc3C(F)F)=O)C2)=O)cc1Cl S(=O)(=O)(c1cc(CNC(C2CCC(C(N)=O)O2)=O)co1)NC(C)(C)C C(=O)(C(Cc1ccc2c(c1)OCO2)CN=c1[nH]c2cc(Br)cnc2s1)OC N1(C(C(C2CCOC2)OC)=O)CC2CCC1C(CNC(=O)CC1C=CCC1)C2 c1(C(=O)NC(C(=O)NC2C(OC)CC2O)Cc2cnc[nH]2)c[nH]c(=O)cn1 c1(CCC(=O)OCCCC)c(C)nc(S)nc1C.c12ccc(c(C(F)(F)F)c1)o2 CC(C)CCC(O)C(=O)NC1COCCC1NC(c1n[nH]c2c1CCSC2)=O c1(C(=O)NC(C)CNC(c2cc3ccc(F)cc3o2)=O)cc2c(nn1)CCCO2 CC1CC(NC(c2cnccn2)=O)CN1C(c1ccc(C(F)(F)F)[nH]1)=O C1(C(=O)NC(CC=C)CNC(=O)CCN2CCCC2)COCCC1(F)F c1(C(C)=O)cc(C(=O)NC(C)CC(C)NC(=O)Cc2cccc(CO)c2)c(C)s1 C1(C(=O)NC2(CC(=O)OC)CN(C(=O)CCC3CC3)C2)CC=C1N=[N+]=[N-] c1(C2(C(=O)NCC(N(C)C(C3CNC(=O)C3)=O)C3CC3)CC2)ccc(F)cc1 CC1CCN(C(c2cc(C(N)=O)c[nH]2)=O)CC1NC(=O)CN(C)S(N)(=O)=O N1(C(C(C(C)(C)O)F)=O)CC(C2CN(C(=O)C=CSc3ccccc3)C2)C1 c1(CS(C)=O)cccc(C(=O)NC2CCCC2CNC(=O)CN2CC3CC3C2)c1 C1(CNC(Cc2nc(C)sc2)=O)CC2(CCN(C(=O)CC3CS(=O)(=O)C3)C2)CO1 CCC(C)CC(C)C(=O)NC1CC2(C1)CC(NC(C1CN(C(=O)NC)C1)=O)C2 c1(C(C(=O)N(CC(C)C)C)NC(=O)C(C)NC(N)=O)ccccc1 N1(C(CC(=O)OCC)=O)CCCC(CO)(NC(c2cc(C)c(F)cn2)=O)C1 Cc1ccc(C=CC(=O)NCC2CCN(C(C3CC4CC4C3)=O)C2)cc1F c1(C(=O)NC(CNC(CCCCC)=O)C(C)(C)C)cccc2oncc12 c1(N2CC(COC)OCC2)cc(Nc2c(OCC)cncc2Br)nc(C)n1 C(=O)(CS(=O)CCC(F)(F)F)N1CCC(C(C)NC(c2ncnn2C)=O)CC1 C1(N(C)C(c2cc(C3(C)CC3)n[nH]2)=O)CCC(NC(c2c[nH]c(CO)c2)=O)CC1 c1(NCC)cc(Cl)ccc1C(N1CCOCC1CN(C(=O)C(O)C(C)C)C)=O C(C(CC(C)C)C(=O)N1CCC(CF)(NC(C2CC3C=CC2CC3)=O)C1)OC c1(C(N2CCN(Cc3c(C)ncs3)CC2)=O)c(F)cccc1Cl C#Cc1ccc(Br)c(C(=O)NCCn2cc(CC(C)(O)CC)nn2)c1 N1(C(C2C(C)CN(C(c3cn(C)c(=O)n3C)=O)C2)=O)CCC2(CC1)CC2C#N C(C)(CO)(CC(C)C)NC(CC1OCCN(C(C2CCC(CC)O2)=O)C1)=O C1(NC(C(C#N)C2CC2)=O)CCCC(NC(c2cccc(-c3ccoc3)c2)=O)C1 C12CN(C(=O)O1)C(C)C(=O)NCCNC2=O.c1(N(CC(=O)NC)C)ccccc1.NCC c1(C(=O)NC(C)(CNC(C2CC=CCC2)=O)CO)ccc(CC#N)cc1 C=C(C)C(C)(C)C(=O)NCCOCCN(C(=O)Cc1ncn(C)c1C)C N1(C(C=CCOCC)=O)CCC(C2(O)CN(C(=O)Cc3sccc3C)C2)CC1 N1(C(C(C(=O)OC)OC)=O)CCC(O)CC1C(=O)Nc1ccc(Cl)cc1C(C)C C1(NC(C(CC)NC(C)=O)=O)CC(C)CN(C(c2snc(O)c2Cl)=O)C1 c1(N(C(=O)C(C)N(C)CC2CC2C)CC=C)ccccc1 N1(C(C)=O)CC(C(N2CCCC2(C)c2ccccc2)=O)Oc2ccccc21 c1(OC)c(C(N2CC(NC(C3CCCCC3C(N)=O)=O)C2)=O)cnn1C N1(C(CN2CCC(C)CC2)=O)CC2CC(NC(c3cncc(Cl)c3)=O)C2C1 Cc1cncc(C=CC(=O)NCC2CCN2C(=O)C(C)CCCO)c1 CN1N=C(C(=O)NC2CN(C(c3ccccc3F)=O)C3(CCOC3)C2)CCC1=O N1(C(C(CC)=CC)=O)CCC(C(=O)NOC2CCC2)(CO)C1 C1(C(=O)NCCC2CCN(C(=O)Cc3csc(Cl)c3)C2)CC2(CCOCC2)CO1 c1(C(=O)NC2CCC(CNC(CC(CCSC)O)=O)C2)cc2c(ccn2C)s1 C#Cc1cccc(CC(=O)N(C2CC(NC(=O)CN3CCCCS3(=O)=O)C2)C)c1 CC1(C(N2CC(c3cc[nH]n3)C2)=O)CCCN1C(C1(F)CCCCC1)=O CC1COCC(CC(=O)NCC2CCC2C(=O)Nc2cccc(CC3CC3)c2)O1 C1(CNC(C2CC(C)(C)OCC2)=O)CC2CCCCC2N1C(=O)C=CCO C1(CC)CCCCN1CCc1cccc(Cl)n1 c1(CN(C)C)ccc(C(=O)NCC(CN(CCCn2ncc(C)c2)C)C)cc1 C1(NC(c2on(C)c(=O)c2)=O)CC2CC1CN2C(=O)C=CC1CCC1 C1(C(=O)NC2(NC(C(C)N(S(C)(=O)=O)C)=O)CC2)CCCN1C(=O)OC(C)(C)C Cc1c(C(=O)NC2CCCC2CNC(C2CC(N(C)C)C2)=O)cccc1Cl.C(C)(C)(C)O C1(C(=O)NCC(C2CCN(C(CN(C)CC)=O)CC2)O)COCCC1(F)F C1(C(N2CCC(C)(N(C)C)C2)=O)CCCCC1(F)F.C12CC(F)CN1C2=O CN(C)NC(=O)CCC(=O)NC1CC1C(=O)N=c1cc[nH]cc1F N1(C(C(CC=CC)C)=O)CCCN(C(=O)COCC(=O)NC)C(CO)C1 CC(CCC(=O)NCC1CCCC1NC(C1(C(F)(F)F)CCN(C)C1)=O)N(C)C N1(C(c2ccncc2O)=O)CCC(O)C2(CCN(Cc3sccc3Cl)CC2)C1 C(C)(C)(CCC(=O)NCC1(NC(c2cc(=O)cc[nH]2)=O)CCOC1)OC CC(C)CCCC(=O)N1CCC(C)(C)C1CNC(=O)COCC1(F)CC1 C1(NC(c2cnn(CCC)c2Cl)=O)CN(C(=O)OC(C)(C)C)C(C)(CC)C1 c1(C(=O)NC(C(C)C)C(C)NC(C2CC(F)(CO)C2)=O)cc(Cl)ccc1[N+](=O)[O-] c1(CCN(CCCOC)Cc2noc(C(C)(C)C)n2)n[nH]c(=NC)s1 Cc1cc(C(N2CC3CC2CN3Cc2ncccc2Br)=O)c(F)cc1F C1(NC(c2cc(CC)n(CCO)n2)=O)CCCCN(C(=O)C(C)OC)C1 C1(CC(=O)NCC(=O)OCC#C)CC(C)N(C(=O)CCc2cncnc2)C1 Cc1nc(C)c(C(N2CC(F)CC2C(=O)NCCF)=O)o1 N1(C(c2cncc(C#C)c2)=O)CC2CCC(N(C(=O)CCCOCC)C)C2C1 CC(Cn1ccnc1)C(=O)N1CCC(C(C)(C)NC(=O)C=Cc2cccs2)C1 C1(CCCNC(c2c(OCC)n[nH]c2)=O)CCN(C(c2cnns2)=O)CC1 c12cc(no1)CN2.C1(C(=O)OCC)CCN1C(=O)CN(C)C(N)=O C(=O)(CC(C)CC)N1CCC(NC(c2c(C(=O)OC)scc2)=O)C1 C1(C(C)NCc2c(C)ccc(Br)c2)Cc2cc(F)ccc2O1 C(=O)(C(Cc1cn[nH]c1)NC(=O)CSC1CC1)N(C1CC(SC)C1)C CC1C(=O)CCN1Cc1cn(-c2cccc(C(F)(F)F)c2)nn1.N1CCCCC1 Nc1nccnc1C(N1CCC1C1CCN(C(=O)CN2CC3CC3C2)CC1)=O Cc1ccc(CCC(=O)NCCCNC(c2cnc(CC3CC3)s2)=O)cc1C N1(C(c2ccc(Cl)nc2)C(=O)NC(C)C2CC2)CC(N(C)C)C(C)(C)C1 c1(CN(CC(=O)NCCC(=C)CNC(c2ccccc2)=O)C)c(C)ncnc1C C1(NC(C2(COC)CN(C(c3ccc(CC)[nH]3)=O)C2)=O)C=CCCCC1 CCCCC(C(=O)N1CCOCC1C(=O)NC(C)C(=O)N(CC)CC)C(C)C C(=O)(C(CNC(c1cc[nH]n1)=O)CC(C)C)N(C(CC)CC)C1CC1 c1(C(=O)NCC(CC)NC(=O)Cn2cccn2)ccc(=O)n(CCO)c1 N1(C(C(C(CC)C)O)=O)CC(NC(=O)CCCOC(C)C)CC(C)(C)C1 N1(C(c2cnc(CC)s2)=O)CCCCC1CCNC(c1ccc(SC)s1)=O N1(C(C(CCNC(CCCOC)=O)OC)=O)CC2(CNC(=O)N2)C1 CCC(C)CC(C)C(=O)NC1CC(CO)N(C(=O)CN2CC=CC2)C1 c1(OC)ccc(Cl)c(C(N2CC3C(NC(c4ccncc4O)=O)C3C2)=O)c1Cl c1(N2C(CNc3cccc(C)n3)CCC2)ccc(-c2cncc(C#N)c2)nc1C N1(C(c2cc(Br)c(Cl)s2)C(=O)NCCCC)CCCC(O)(c2ccccc2)CC1 c1(C(N(CCNC(CC=CC(C)(C)C)=O)CC2CC2)=O)n[nH]c(C2CC2)c1Cl N1(C(c2cnn(CCC)c2C)=O)CCC(NC(C2CC(CC(F)F)C2)=O)C(F)C1 C(=O)(CC(C)CCCCC)NC1(CC=C)CCN(C(c2cnn(C(C)C)n2)=O)C1 CN1CCCCCC1C(=O)N(CCCCCC(=O)NC1CCC(=O)NC1)C C1(CN(C(=O)Cc2cncc(O)c2)C)CC(F)CN1C(=O)CCC(F)F n1(CC(=O)OC(c2ccc(C)cc2Cl)C)c(C)nc2ccccc2c1=O C1(NC(C(C)n2cccc2)=O)(CO)CCN(C(C2(Cl)CC2(F)F)=O)CC1 N1(C(C(C)OCCCC)=O)CC2CC(N(C)C(c3sc(CCC)nc3C)=O)C1C2 c1(OC)ccc2c(C(=O)NC3CC4CC(C3)N(C(=O)C(C)O)C4)cc(=O)oc2c1 n1(CCCNC(=O)Cn2cc(C3(C(=O)O)CC3)cn2)nc2n(c(=O)c1=O)CCC2 C1(NC(c2c(SC)ccs2)=O)CC2CC(NC(=O)Cc3csc(=N)[nH]3)C1C2 c1(C(N2CC3(C(C(=O)NC45CC(C(=O)OC)(C4)C5)C3)C2)=O)ccc2c(c1)CCO2 Cc1cc(C(N2CCCC2C2(O)CN(C(=O)C(c3cncnc3)C)C2)=O)[nH]c1C c1(C(C)C)nccn1CC(=O)NCCCC1(NC(=O)CC2CCCC2)CC1 c1(CNCc2c(OC)nccc2)[nH]c(=NC2CCC(F)CC2)nc2c1ncn2C CC(C)(C)C(CO)C(=O)NC1C2CN(C(c3cc(C(F)F)ccn3)=O)CC12 c1(C(CNC(C2CC(=C)C2)=O)NC(=O)Cn2ccc(CC)n2)cccc(Cl)c1Cl c1(C(=O)OCC)ccnc(NC(c2nccn2C(C)C)=O)c1.C12CC1CNC2=O c1(C(=O)NC2C(C(=O)NC(c3ccc(Br)cc3)C)C2)ccc(Cl)nc1 C12=CNC(=NCCNC1=O)C=C2.C1(CC(=O)N(CCOC)C)CCCS(=O)(=O)C1 CC(C)S(=O)(=O)C(C)C(=O)NCC(CNC(=O)C(c1ccccc1F)(C)C)CO C1(NC(C(N2CCC(N(C)C)CC2)C)=O)CN(C(=O)CC23CC(C2)C3)CC1(C)C C1(NC(=O)CC2CCOC2=O)CCC(O)CN(C(c2cccc(F)c2F)=O)C1 N1(C(c2ncc(OC(C)C)nc2)=O)CC2CC(CF)(CO2)C1 C1(O)(C(C)NC(=O)C(=O)NCC(F)F)CCN(C(=O)C(F)(F)C2CCCC2)C1 N1(C(C2CC(=C)C2)=O)CCN(C(c2cnoc2C)=O)CC1CO C1(CNC(C(c2cccc(C)c2)C)=O)CCN(C(=O)Cn2cc(C)cn2)C(C)C1 CCC(CC)(CO)C(=O)NC1CC(NC(=O)Cc2c(C)noc2Cl)C(O)C1 C(C)(C)(CC(=O)NC(C)CN1CCCC1=O)N(C(c1ccn(C(C)C)n1)=O)C C1(C(N(CCCCO)CC)=O)CC(O)CN1C(c1n[nH]cc1OCC)=O c1(N)cc(C)ccc1C.c1(CC)ccc(C(=O)OC)cn1.N12CCCCC1C2=O C1(C(=O)NC(COCC)C)CN(C(c2cc(Cl)cc(Br)c2O)=O)CC(F)(F)C1 C1(C(N(C(C)CNC(c2cc(N)ccc2O)=O)C)=O)CC(F)(F)CCC1(C)C c1(OCC)oc(C)nc1C(N1CC(NC(C23CCC(CC2)C3)=O)C(C)C1)=O c1(OC)ccc(F)c(C(N2CC(NC(=O)CCS(C)(=O)=O)C(F)C2)=O)n1 CON(CCC(=O)NCC(=O)NC1CC1)C(=O)C1CCC(F)CC1 C(=O)(CC(O)C(Cl)(Cl)Cl)NCC(C)(C(C)C)NC(C=C(COC)C)=O C(=O)(C1CNC(=O)c2ccnn21)N1CC(O)(CNC(c2cnc(CC)[nH]2)=O)C1 c1(C(=O)NC2CCN(C(CC(C(=C)C)OCC)=O)C2)cnc2cc(C)ccc2c1 C(=O)(CC(C)C(=O)OC)Nc1cc(O)no1.C(C(=O)NC)NC(C1CC1COCC)=O c1(CNC(C2(C#N)CC2)=O)nnc2n1CCN(C(=O)CN1CCC(CO)CC1)C2 N1(C(C(C)NC(C)=O)=O)CC2(CCNC(=O)CC3CC3(Cl)Cl)CCC1CC2 C1(NC(C2CCCN(CC)C2)=O)CCN(C(=O)C=Cc2cccc(F)c2)C1(C)C C12(C(N3CC(C(C)C)NC(=O)C3)=O)CCN(C(C3(C)CCC(=O)C3)=O)CCC1C2 C(=O)(CC(F)(F)c1ccccc1)NC1CC(N(C(C(c2cn(C)cn2)C)=O)C)C1 N1(C(CCC(C)N(C)C)=O)CC2OCCN(C(c3ncoc3C3CC3)=O)C2C1 Cc1cc(C(N2CCC(NC(C3CCOC3)=O)C2(C)C)=O)c(N)c(Cl)c1 c1(C(=O)NC2CC(CNC(c3cc(C)oc3C)=O)OCC2)ccc(F)c(Cl)c1 C1(NC(c2ccc(CCCC)cc2)=O)C2CCC1N(C(=O)C(C(C)CC)OC)C2 CC1=NOC(C(=O)N(CC(n2cc(-c3cnc[nH]3)nn2)C)C2CC2)C1 C1(NC(c2ccn(CC)c2C)=O)CCCC12CCN(C(C1CCNC1=O)=O)CC2 c1(C(N2C(CN(C(c3ccc(C)s3)=O)C)CCC2)=O)cnc(Cl)cc1N C1(C2CC2)CC(OC)C(=O)N1C.c1(CN)ccccc1F.C12CC(C(F)F)(CO1)C2 N1(C(Cc2ccc(-c3nc(C)sc3)s2)=O)CC2CCC2(NC(c2cn[nH]c2)=O)C1 C(CN=c1[nH]c2ccccc2o1)C1C(C)CCCN1C(=O)C(C)C1CCOC1 C(c1cc(F)cc(F)c1)=CC(N1CCN(C(=O)NCC(=O)OCC)CC1C)=O c1(C(=O)NC(CC)CNC(C2(C(C)C)COC2)=O)cnn(C(C)(C)C)c1Cl N#Cc1ccc(NCC(=O)NCC2CCCN(C(=O)C=C(Cl)Cl)C2)cc1 C(=O)(C(C)(C)C(C)(C)O)NC(CC(=O)NC(c1n(CC)ncn1)C)C1CC1 C(C(C)(C(C)C)NC(c1cccc(SCC#N)c1)=O)NC(C=NOC)=O c1(Cc2n(CCC)nc(-c3occc3C)n2)c(Br)c(C(C)C)nn1C C1(CN(C)C(C2(C(F)F)CC2)=O)CN(C(C2C=CCS2)=O)C1 C1(NC(C2CCCCC2)Cc2n(C)cnc2)CCCOCC1 O=C(CS(=O)(=O)C1CC1)NC1CN(C(c2cc3ccccn3c2)=O)CC(F)(F)C1 C1(CNC(=O)C(F)C2CCC2)CC(O)C(O)CC1C(=O)NCC1CC2(CC2)CO1 C1(CNC(C2CN(C(C)=O)C2)=O)CC2(CCN(C(c3cccc(N)c3)=O)C2)CO1 c1(N2CC(NC(c3n(C)nc(CC)c3Cl)=O)C(C#N)C2)ncc2ccccc2n1 c1(CC)cc(CC)[nH]c(=NC(CNC(C2CCCN2C)=O)C(C)C)n1 C=CCCCCCN(C(=O)CC1CC(C)N(C(c2nccs2)=O)C1)C N1(C(c2c(-c3c(C)cccn3)c(C)[nH]n2)=O)CC2(CCCC2)C1C(=O)N(C)C CCC(CC)N=c1nc(N2CCC(c3n[nH]c(C)n3)C2)c2c([nH]1)CSC2 CC1=NNC(=O)C1CC(=O)NC(c1ccccc1)C(=O)NCCC(F)(F)F N#Cc1ccc(CN2CC3C(C2)N3C(c2cccc(Br)c2)=O)cc1Cl C1(NC(C(C)C2CCCC2)=O)C2CC1CN(C(=O)C(F)=CCCF)C2 C12(NC(C(CC)SC)=O)CCCC1CN(C(c1ccccc1C(C)=O)=O)C2 C=CC(C)(C)CCCNC(C1CN(C(=O)COc2cnn(C)c2)CC(C)O1)=O C1(C(N2CC(C(C(=O)N(C(C#C)C3CCC3)C)OC)C2)=O)CC2(CCC2)C1 N1(C(=O)OCC(C)C)CCN(C(c2sc(Br)cc2Cl)C(=O)NC(C)C)CC1 C1(C(N2CC(CC)N(C(=O)COC(C)(C)C)CC2)=O)OCC2CCCC1C2 N1(C(C2(CCc3ccccc3)CCC2)=O)CCN(c2ncc(F)cn2)C(CO)C1 c1(C(=O)NCC(C)(C2CCC2)NC(C2ON=C(C)C2)=O)cn2ccsc2n1 c1(C(C)(F)F)ccccc1C(=O)NCC(F)CNC(c1ccc(C#N)s1)=O C(C(=O)NCc1ncoc1CCNC(C1CCC(=O)C1)=O)(C(C)C)NC(C)=O N1(C(C2CC(C)(OC)C2)=O)CC2CCC(C1)N2C(=O)CCCF CCCC(C)CCCC(=O)N1CC2CCCC(C1)N2C(C1CN(C(C)C)C1)=O C1(NC(c2c(C)cccc2)=O)CCCC12CCN(C(c1ncoc1C)=O)C2 O=C(C1Cc2ccc(F)cc21)N1CC2(CCCC2NC(C2(C3CCC3)CC2)=O)C1 Cc1nc(C(C)NC(c2c[nH]nc2CNC(=O)CCCn2ccnn2)=O)c(C)o1 C(CC(=O)NCCCn1ccnc1)(C(F)F)NC(c1cc(C(C)C)on1)=O c1(C(=O)NCCCNC(CSc2n(C)ccn2)=O)ccc(F)c2c1CCC2 N1(C(C(C=C)O)=O)CC(NC(=O)Cc2nocc2C)CC(C)(C)C1 C(CCC(C)CC(=O)N1CCCC(C(=O)NCc2cccc(C)c2)C1)=C(C)C C1(C(=O)NCC2(NC(c3cccs3)=O)CCC2)CC(=O)c2cc(F)ccc2O1 c1(C(=O)NCC=CC(=O)NCC(C)(O)C2CCC2)cccc(CO)n1 N1(C(C2(COCC)CC2)=O)CC2CCC1C(NC(C1CSCCS1)=O)C2 C1(NC(C=C(CCC)C)=O)CN(C(=O)C(C)(C2CC2)OC)CC1(C)C Cc1noc(C(=O)NCC23CC(NC(=O)CCC4CCCCC4)(C2)C3)c1C Cc1nn(C)c(C)c1OCC(N1CC=CC1CNC(C1COC(=O)N1C)=O)=O CC1CC=C(C(=O)NCC2(Nc3ncn(C)c(=O)c3Br)CC2)CC1 c1(CNC(C2(COC)COC2)=O)cc(C(=O)Nc2cnn(C)c2)n(C)n1 N1(C(C(C)C(F)F)=O)CCC(C2CCN(C(=O)C(C)C(F)(F)F)CC2)CC1 c1(C(=O)NCC2C(NC(C3CCN(CC)C3)=O)C2)cc2nc(C)sc2[nH]1 c1(C(N2CCN(C(c3c(=O)ccn(C)c3)=O)C(CF)C2)=O)occ2c1CCCC2 CCC(CC)C(F)C(=O)NCCN(CC(C)O)C(=O)CNC(=O)C1CC1 N1(C(C2N(C(C)C)CCC2)=O)CCN(C(c2sc(C#N)cc2Cl)=O)CC12CCC2 c1(COCC(=O)NCc2ccc(C(=O)NC(C3CCCC3)C)o2)ccnc(O)c1 C1(OCC)CN(C(N)=O)C(C)(CNC(C2CN(C(=O)C3=CCCS3)C2)=O)C1 C1(NC(C(CCSC)O)=O)C(C)CCN(C(=O)C(C2CCCCC2)C)C1C N1(C(CN(c2ccncc2)C)=O)CC2C(NC(C3(C#N)CC3(C)C)=O)C2C1 N1(C(C2C(C)(C(F)(F)F)C2)=O)CCCC(C)(CNC(=O)C2=CCCOC2)C1 N1(C(C(C=C)(C)O)=O)CCC(N=c2cccn[nH]2)CC1C C(=O)(CC(c1ccccc1)SC)NCCN(C(C1(C)CC1(F)F)=O)CC C1(NC(Cc2cc(C)c(CO)cc2)=O)CCN(C(=O)Cc2cc[nH]n2)CC1(C)C c1(CN2CC(CNC(C3CCN(C)C3)=O)C2)c[nH]c2cc([N+](=O)[O-])ccc12 c1(C(=O)NCCN(C(=O)CC2CC2C)CC)cc(CO)oc1C C12(C(=O)NC(C)CC3CN(C(c4c(N)cnn4C)=O)C3)CC(C)(C1)OC21CCC1 C#Cc1nccnc1NC(C1CCN(Cc2cccc(O)c2Br)C1)=O c12ccc(cc1)C(C)NC(=O)C2C.c1(CN(C(=O)C(=O)NC)CC)ccccc1 n1(CC(=O)NCC(CNC(c2nccnc2SC)=O)OC)cccc(C)c1=O c1(C(N2C(CC(N3C(C)CN(C)CC3)=O)CCC2)=O)cnc2ncccn12 Cc1cncc(C(=O)NC(C)CCCCNC(c2nc[nH]c2C(C)(C)C)=O)n1 C=C(F)C1(CC(N2CCC2CC(=O)NCC2(COCC)CCC2)=O)CCC1 Cc1sc(C(=O)N(C2CN(C(=O)COCC3CCOC3)C2)C)c(C)c1C C1(NC(c2cc(C)on2)=O)CC2(CCN(C(C3CC(C)CC(C)C3)=O)C2)C1 C(c1cccc(F)c1Cl)=CC(N1CCC(NC(c2c(CCC)nco2)=O)C1C)=O N1(C(c2cc(CC)nn2C)=O)CCC2CN(C(c3cnc4[nH]ccnc3-4)=O)CC12 C(=O)(N=c1nc(C2CC2)[nH]s1)NC1=CN=C(OC)C(Br)=C(F)C1 c1(C(N2CCN(C(=O)C(F)C(F)(F)F)C(CC3CC3)C2)=O)ccc2oncc2c1 Cn1ncc2cc(C(N3CCC(O)(C(=O)Nc4cnnc(Cl)c4)C3)=O)ccc12 CCCC(CCC)CC(=O)N1CC(F)CC1C(=O)NCCC1CC1 CC1(C)CC(n2cc(C3CCCN3Cc3c(F)cc(Cl)cc3F)nn2)C(C)(C)O1 N1(C(c2n(C)ncc2)=O)CCOCC1C1C(CC(=O)NC(CN(C)C)CO)OCC1.C(=O)C C=C(C)CC(C(=O)NCCN(C(C)C)CC)NC(=O)CC1CC(CC)C1 c1(CNC(C(CC)NC(c2ccc(CSC)o2)=O)=O)ccc(O)cc1F N1(C(CCCOCC)=O)CCC2(C1)CN(C(=O)CSCCOC)CCO2 C1(Nc2nc(N3CCCCC(CC)C3)c3c(n2)ccs3)CC2(C1)C(F)(F)C21CC1 N1(C(c2nccs2)=O)CC2(C1)CN(C(C1(CF)CC1)=O)CC2CO C(=O)(C(C)S(C)(=O)=O)N1CCCC(CCNC(C(n2ncc(C)c2)C)=O)C1 C(=O)(C(C)C(O)CC)N1C(CNC(c2cc(CCC)n(C)n2)=O)CC(O)C1 c1(OC)cccc2c(Nc3sc(OC4CCCC4)nc3C)cc(C)nc12 N1(C(C=Cc2c(C)nccc2)=O)CCCC(C2CC2NC(=O)C(O)C2CC2)C1 C(=O)(C(C)C(C)(C)C)NCC1(C)CCN(c2snc(C(=O)OC)n2)C1 CCC1=C(C(=O)NC2C=CCC(C(=O)Nc3cnn(C(F)F)c3)C2)CCCO1 Cc1ccc(C(=O)N(C)CC2(NC(=O)Cc3c(C)n[nH]c3C)CC2)cc1Cl c1(C(N2CCC(F)C(NCc3c(F)ccc(Cl)c3F)C2)=O)cc(F)c(F)c(Cl)c1 C1(C(=O)NC(C(=O)OC)C)(CO)CN(C(c2ccc(Sc3nncs3)o2)=O)C1 CC1CC(C(=O)N2CC3CC2(C(=O)NCC2(CC4CC4)CC2)C3)=NO1 c1(N2CCC(C3(NC(C4CCCN(CC)C4)=O)CC3)C2)ncc([N+](=O)[O-])c(=N)[nH]1 Cc1nc(C2CCC2)oc1C(N1CCC(O)(CNC(C2CC(C)(C)CO2)=O)C1)=O N1(C(C(CC)N(CC)CC)=O)CC2CC(NC(c3cc(OC)no3)=O)C(C2)C1 C1(C)(CNc2ccc(C(C)(C)C)s2)CC2(CC2)C1 C12CN(CCC1O)C2=O.c1(C(C)=O)cccc(Nc2csc(C)n2)c1 CC1(C)C(CNC(C2(P(C)(C)=O)CC2)=O)CCN1C(=O)CCSc1ccccc1 N1(C(CCC(=C)Br)=O)CCN(C(c2ccc(Cl)nc2N)=O)C(C)C1 c1(OC)cc(CCC(C)NC2C(F)(F)C23CC3)ccc1O N1(C(C(C)SCC)=O)CC(N(C)C(c2ccc(CO)cn2)=O)C2(CC2)C1 c1(C(=O)NCC23CN(C(c4cncc(N)n4)=O)C(C2)CO3)ccnc2ncnn12 Cc1ccc(OCCCC(=O)NC2CCC2NC(=O)C(F)(F)F)c(C)c1 Cc1nc2ccc(C(=O)NCC3(NC(c4cc[nH]n4)=O)CC3)cc2s1 c1(C(N(C2(CC(=O)NCC(C)CO)CCC2)CC)C)ccncc1 C(=O)(C1CCCc2n[nH]cc21)NCC=CCNC(c1cnc(CC)s1)=O C1(CN(C(=O)CC2CC3CCC2C3)CC)CCN(C(c2oc(C)cc2C)=O)CC1 c1(C(=O)NCC(CCOC)NC(c2cc(C)c(C)nn2)=O)cc(Cl)cnc1C CCCC(CCC)CC(=O)N1CCC(C(=O)N(CC(C)C)C)(C(C)C)C1 C1(NC(N)=O)CCCCN(C(c2c(-n3cccn3)cccc2F)=O)C1 c1(OC)cc(C)c(S(=O)(=O)NC(=O)C(=O)Nc2cc(Br)cc3c2OCC3)cc1Cl N1(C(C2CCC(=O)O2)=O)CC(C(=O)NC2(CC3CC3)CCC2)C2(CC2)C1 CCC(C)C(C(=O)C(=O)C=CC(=O)NC1CC1)N(C)C.n1(CC=C)cncn1 C(=O)(CC(O)CC(C)(C)C)NCCC(C)NC(C(c1ccccc1)OC(C)C)=O N1(C(c2cc(CC)no2)=O)CC2CCCC(NC(c3coc(C4CC4)n3)=O)(C2)C1 c1(C(N2C(CNC(CCC(C)=O)=O)CC2)=O)cc(Cl)cc(Cl)c1[N+](=O)[O-] Nc1c(C(N2CC=CC(NC(=O)C=CCF)C2)=O)nnc2ccccc12 C(=O)(C1CCCc2c1ncn2C)N1CCOCC(NC(c2nccc(C)c2)=O)C1 c1(NCc2c(C)cncc2)[nH]c(=NCC2CCCC(CO)O2)nc2sccc12 c1(C(=O)NC2C(NC(C(CCOC)(C)C)=O)CC2)cc(C)c(Cl)c(N)c1 Cc1ccc(C(=O)NCCn2cc(C(=O)NC3CCN(C(C)C)C3)nn2)c(C)n1 c1(C(=O)NC2C(NC(c3n(C)ccn3)=O)CC2)cccc2ncnc(O)c12 c1(C(=O)NC(CN(C(C(C)Cc2cccnc2)=O)C)C)ccc2c(c1)OCCN2 c1(NC(C2C(C(=O)Nc3c(OC)cccc3Cl)C2)=O)ccc2nc(CO)[nH]c2c1 c1(C(=O)NCCNC(=O)CC2CCCCO2)ccc(F)c(F)c1Cl C1(C)(NC(C2C(CC)CCN2C(C2CC3(C2)CC(O)C3)=O)=O)CCCC(C)(C)C1 C1(NC(CC(=O)NC2CC2)=O)CN(C(=O)CSC(F)(F)F)CC1C1CC1 CC(C#N)CN=C(NCc1nn(C)cc1S(C)(=O)=O)NCc1cccs1 c1(OCCNC(c2cccc(C#N)c2)CCOC)ccc2ncn(C)c(=O)c2c1 CC1CN(C(c2nccc(Cl)c2F)=O)CCC1CNC(C1(CO)CCCC1)=O N1(C(C(CC#C)C)=O)CCC(C(F)(F)F)CC1CNC(C1C2CCOCC12)=O c1(C(=O)NCC(C2CC2)NC(C(C)(C)F)=O)ncc2ccccn12 CC1=C(C(=O)NC2CCCN(C(=O)CCc3nccn3C)C2C)CCO1 c1(OCC)ncc(C(=O)NC2CN(C(c3c(F)cccc3F)=O)C2)cc1Cl C1(CC(=O)NCCOCCN(C(=O)CC(=O)N(C)C)C)CCC(C)(C)O1 C1(NC(C2CC(O)(CNC(C3CCCC3)=O)C2)=O)CC2(CC2)C1 c1(NC(c2scc(C(N3CCC(OC(C)=O)C3)=O)n2)=O)ccc(C2CC2)c(Cl)c1 c1(OC)cc(Br)c(C(=O)NCC23CCCCCC2NCC3)cc1OC c1(C(=O)NC(CNC(C(c2c(OC)cccc2)C)=O)C2CC2)ccc(=N)[nH]c1Cl CCCCC(F)C(=O)N(C)CCOCCCNC(c1cn(CCO)nn1)=O c12cnn3c1CN(CC3)CC(=O)NC2.c1(CC)cc(N2CCCC2)ccn1 Cc1ccnc(C(N2CC(C(C)(C)O)(CNC(c3onc(C)c3C)=O)C2)=O)n1 c1(C(N2CC(C(C)(C)O)(CNC(CCC=C)=O)C2)=O)cccc2c1OCC2 c1(C(C)=O)ccc(NC(c2cc(Cl)c(C)cn2)=O)c(F)c1F N1(C(=O)OC(C)(C)C)CC(NC(C2CCN(C3CCOC3)C2=O)=O)CC(F)C1 C(=O)(C(O)C(C)CC)N1CCC(N(C(c2c(CC(=O)OCC)nccc2)=O)C)C1 c1(C(N(CCOC)CCNC(=O)CCC2CC(OC)C2)=O)scnc1Cl c1(NC(CC2CCN(C(C(CNC)C)=O)C2)=O)cccc(OC)c1 N1(C(c2ccn(C)n2)C(=O)NC(C)C2CC2)CCN(C)CC1C1CC1 c1(C(=O)NCC2CC2CNC(c2ccc(CF)cc2)=O)ccc2nccn2c1 N1(C(c2n(C)nc(C3CCCC3)c2)=O)C2CCC1C(CNC(=O)CCS(C)=O)C2 CC1=C(C(=O)NC2CCN(C(C3CCC(=O)N3)=O)C2C)Cc2ccccc2O1 N1(C(C2CNC(=O)C2)=O)CCOC(CCNC(C2CC(N3CCCC3)C2)=O)C1 c1(C(=O)NCCCNC(=O)Cc2ccsc2)coc2c1C(=O)NCCC2 c1(C(=O)NCCNC(c2c(Cl)ncc(OC)c2)=O)ccc2nnnn2c1 c1(C(N2C(C(C)C)CN(C(=O)CC(C)C3CC3)CC2)=O)ccc2ccnn2c1 c1(C(=O)NC2(C(=O)NC(C3CCOC3)CO)CSC2)cc2occc2[nH]1 CC1(CNC(c2cnc(N(C)C)o2)=O)CCN(C(C2CSCN2C(N)=O)=O)C1 C12(NC(c3ccc(OC(C)C)cc3)=O)CCC(CN(C(=O)CC3CC(F)C3)C1)C2 N1(C(c2c(COC)noc2)=O)CCC(NC(C2CCC3CC3CC2)=O)C12CCCC2 C(C)(CCC(=O)NCCNC(C1CN(C(=O)C(N2CCSCC2)C)C1)=O)SC C(CC(F)(F)Cn1cc(CCCC)nn1)NC(CCC=C)=O CCCCCC(C)(C)C(=O)NCCCC(O)C(N1CC2(COC(C)(C)C2)C1)=O O=C1CCC(C(=O)NCCN2CCN(C(=O)C#CC3CCOC3)CC2)=NN1 c1(NC(CN(C(C2(C)CCCNC2=O)=O)C2CC2)=O)ccc2ncnn2c1 CC(C)CC(C(=O)NC(C)(C)CCNc1ncc(O)cn1)C(C)C c1(C(C2CCN(C(C3CCN(C(C)=O)CC3)=O)CC2)O)ccc2c(c1)OCCO2 O=C1CS(=O)(=O)c2cc(NC(=O)CC(C(F)F)N3CCOCC3)ccc2N1 c1(CNC(CN(C)C)CCO)ccc2c(c1F)CCC2 N1(C(C(Cc2cc[nH]n2)NC(c2ccc(C#N)o2)=O)=O)CC2CCCC2(CO)C1 CC1=C(C(=O)NC2C3CN(N(C)C)CC23)CCCO1.C1(C=O)CCn2cncc2C1 c1(OC)ccc(C(=O)NC2CCC(N(C)C(c3coc(C)c3)=O)CC2)cc1N Cc1cc(=NC2CCC(NC(=O)CN3C(=O)CC(C)(C)C3=O)CC2)[nH]c(CO)n1 N1(C(CC=C)=O)CCC(CNC(=O)CCSC)C12CC2 CC(O)C(C)(C)C(=O)N1CC2C(C(=O)N(C)CCc3cnc[nH]3)C2C1 c1(C(=O)OC(C)(C)C)ccc2c(c1)CCCCN2C1CCCCC1=O C(=O)(C1=NN(CCO)C(=O)CC1)NCC(CC)NC(=O)C(C)(F)C(=O)OC C1(NC(C(CC=C)OC)=O)CCOC12CCN(C(c1nn(C)c(C)c1Cl)=O)CC2 CCC(O)C(C)C(=O)NCC=C1CCN(C(C2(N(C)C)CCC2)=O)CC1 C1(NC(CN2CCC(OC)C2)=O)CC(F)CN(C(=O)C(C)(F)c2ccon2)C1 C1(NC(=O)CC2CCC(F)C2)(CO)CCN(C(=O)COc2ccccc2)CC1 C1(C(N2CC(NC(C(c3c(C)cccc3)C)=O)C(O)C2)=O)CC12CC(C)(C)C2 c1(CC)nc(C(=O)N(C2CCOC(C(CC)CC)C2)CC2CC2)cc(=N)[nH]1 C1(CNC(C2(CC=C)CCC2)=O)CC2CCCCC2N1C(c1cncc(F)c1)=O Cc1cc(C(N2CCSCC2)=O)c2cc(-c3cc(F)c(O)cc3F)ccc2n1 C1(C(=O)NCC2CCC(C(=O)NC3(CC)CCCCC3)C2)CC2CC(=O)C1O2 CC1=NN(C)C(=O)C1CC(=O)N(C1CCN(C(c2ccc(=N)[nH]n2)=O)C1)CCO Cn1c(O)nc2c(C(=O)NC3CC(NC(C45CCOC4CCOC5)=O)C3)cccc12 N1(C(CCC(C)N(C)C)=O)CC2(CNC(C3CC(C4CCC4)C3)=O)CCC1CC2 C1(NC(C2C(C)(CC)C2)=O)C2CCN(C(c3ccnn3-c3ccncc3)=O)CC12 c1(CN(C)C(c2ccccc2C(=O)NC(C)(C)C)=O)cc(Cl)ncc1Cl N1(C(CC2CCC(C(C)C)CC2)=O)C2CCC1C(CNC(C)=O)C2 c1(OC)ncc(C(=O)NC2CN(C(C3CC(=O)NC3(C)C)=O)C2)cc1Cl O=C(CCCCCc1ccccc1)NCCC1CCCN1C(C1CCCC1O)=O c1(C(C(=O)NC2(CC)CN(C(=O)CN3CCCC3)C2)C)sc(CN(C)C)nc1C c1(C(C(=O)NCC(CNC(c2c(NC)nccc2)=O)CO)O)ccc(Cl)cc1F C1(C(N(CCCNC(c2cn(C3CC3)nn2)=O)C(C)C)=O)CCC(=O)CC1 c1(NC(C2C(CC)N(C(=O)CCc3nnnn3C)CC2)=O)cccn2nccc12 Cc1ccc(C(C)CC(=O)N2CCC(N(C(=O)CN(C)C3CC3)C)C2)cc1 c1(C(=O)NCCNC(c2cc(C(C)C)cc(C(C)C)c2O)=O)ccc2cnnn2c1 c1(C(c2c(C(N3CC(C(=O)OC)NCC3)=O)nccn2)=O)cccc(C)c1Cl C1(NC(c2ccc(CC)cc2)=O)CCN(C(C2(C)CC2C)=O)CC1C(N)=O C(=O)(CC(P(C)(C)=O)P(C)(C)=O)NC1(CC=C)CN(C(=O)CC(CC)CCC)C1 C1(CN(C(=O)CC2(CO)CC2)C)CCCN1C(=O)C(=O)NC(C)(C)CNC1CC1 C1(CNC(C2N(C(=O)NC)CCC2)=O)CC2(CCOCC2)CN1C(C1CCSC1)=O Cc1conc1CC(=O)NCC1CC(F)(CNC(=O)CC2CC2(C)C)C1 C#CC1(C(=O)OC)CCN(C(C2CC(F)C2)=O)CC1.C12CC(C1)N(C)C2=O C(=O)(C(C)CCCC(C)C)NC1C(C=C)CN(C(=O)Cc2c(C)ncnc2C)C1 C(C(O)C(=O)NCC(C(C)C)NC(=O)CCNC(=O)Oc1ccccc1)OC CC(C)C(C)(O)C(=O)NC1CCC(c2cn(-c3cc(O)nc(O)c3)nn2)CC1 c1(C(Cc2nc(C)c(C)o2)=O)ccc(F)c(-c2cn(C(C)C)nn2)c1 CS(=O)c1cccc(NC(c2ccnn2CCF)=O)c1 c1(C(=O)NC(c2ccc(Cl)cc2)C)cc2cc(S(N)(=O)=O)sc2s1 c1(C(=O)NC(CCCC)CNC(=O)CCF)cc(Br)cc2cccnc12 c1(C(N2CCCC(N(C(C(C)(C)F)=O)CCO)C2)=O)ccc2c(c1)C=CS2(=O)=O C1(C(=O)NCCN(C(c2c(CC)nn(C)c2)=O)C(C)C)CCC2C(C1)C2(F)F C1(N(C(C2CC(C)(F)C2)C(=O)NS(C)(=O)=O)C)CCC(C(N)=O)C1 C(=O)(C(C)(CC)CC=C)NCC(CC(=O)NC(CC=C)CC)O C1(c2ncc(-c3n(C(C(NOCCCOC)=O)C)ccn3)s2)C2CCC(C2)C1C C(=O)(C1CCCc2sccc21)NCC1C(C)(C)CCN(C(CC2(OC)CC2)=O)C1 C1(C(=O)NCCN(CCC)C(C2CCCC(F)C2)=O)CCCC1S(C)(=O)=O c1(C(=O)NCC(CNC(C2N(C)CCOC2)=O)O)cc2c(F)c(F)ccc2s1 C1(C(=O)NC(C(C)NC(CSCCOC)=O)CO)CCCC(C)(C)CC1 C(=O)(C(CNC(c1cnc(C2CC2)o1)=O)CC1CC1)NCC1C(OC)CCC1 C=CC1(C(N2CC(OC(F)F)C2)=O)CCN(C(=O)Cc2cnn(C)c2)C1 Nc1ccc(C(N2CC3(NC(=O)CC45CCCC4C5)CC2C3)=O)c(F)c1 Cc1nn(C)cc1C(C)NC(C1OCCC1NC(C1CC2CCC2C1)=O)=O c1(C(=O)NC2(C3CCN(C(=O)C(O)Cn4cncn4)C3)CC2)cccc(O)n1 Cc1c(N2CCSC(C)CC2)ncnc1NC(C1CCCC1)CN(C)C CC1OC2CCC1(C(=O)NCC(=O)NCc1cccc(CC3CC3)c1)C2 C1(F)(CNC(C(C)(C)OCC)=O)CCN(C(c2ccccc2-c2cn[nH]c2)=O)C1 C1(CC=C)(C(=O)NCCC2CC(NC(C3CC3C(N)=O)=O)C2)CCOCC1 N1(C(CCC2CCC(C)O2)=O)CCCC12CCN(C(c1cnoc1)=O)CC2 N1(C(C)=O)Cc2nccn2CC(NCC2(Oc3ccccc3)CC2)C1.C(=O)C(C)(C)C N1(c2c(Cl)cnc(OC)n2)CCN(C(c2ccc(C(C)C)c(Cl)c2)=O)CCC1C c1(C(C)NC(=O)C(F)OC(F)(F)F)nocc1C(=O)NCC(C)N=[N+]=[N-] C1(C(N(CCCCNC(C2CC2c2cnn(C)c2)=O)C)=O)CC2C=CC1O2 c1(C(N(Nc2ncc(C(=O)OCC)cn2)CC2CC2)=O)ccc(CC)cc1Cl C1(NC(C(c2ccccc2)OC)=O)CC2CC1CN(C(C1(C(N)=O)CC1)=O)C2 CC1=C(C(=O)N2CCC3CCC23CNC(c2ccncc2N)=O)SCCO1 N1(Cc2c(C)nccc2)CCCC2C1CCN2C(c1cc(Cl)c(O)cc1F)=O CC(CC(N)=O)C(=O)N1CCC2CC12C(=O)NC(C)(C)CCN(C)C c1(CC)c(C(=O)NC2CCC(NC(=O)C(C)C(F)F)C2)cccc1C c1(C(N(C(C)CCNC(C2CCN2C2CCCC2)=O)CCC)=O)c[nH]c(=N)o1 c1(-c2ccc(C(=O)N(c3ncc(Br)c(I)n3)CCO)nn2)ccc(F)cc1[N+](=O)[O-] c1(C(N2CC3C(CNC(c4ccnnc4O)=O)C3C2)=O)cc2c(Cl)ccnc2s1 C=CCCCCCCC(=O)N1CCCCCC1C(=O)NCCn1nncc1C Cc1cc(C(N2CCCCC2C2CCN(C(c3ncccn3)=O)CC2)=O)ncn1 C(CCC(C)C)(C(=O)N1CCC(O)(CNC(=O)CCS(C)=O)C1)NC(C)=O N1(C(c2c(C)cco2)=O)CC2CCN(C(c3nc(Br)c[nH]3)=O)CC12 c1(CCC(=O)N(CCOC2CCC(C)CC2)C2CC2)c[nH]c2ccccc12 c1(C(=O)NCC2C(NC(C3(C)ON=C(C)C3)=O)C2)cc2c(cc1N)CCC2 c1(C(=O)NCC(CN(C(c2nc(CCC)oc2)=O)C)C)sc(C)nc1C CC(C)C(CC1CCCCC1)C(=O)NCC(F)CNC(=O)C1=NOCC1 c1(OC)cc(NC(=O)C(CC(C)C)N(C)C(c2cnsc2)=O)ccc1O c1(C(=O)NC(C)CC(=O)NC2(CO)CC2)ccc(O)c(F)c1 C1(CC(N2CC(OCCNC(c3cccnn3)=O)C2)=O)CCCC2(CC2)C1 C(CCC(O)C(=O)NCCN1CC2CC2C1)OCC(=O)NCCO.C1(N)CC1 CC1(C)CCN(C(C2Cc3cccnc3C2)=O)CC1CNC(c1coc(Cl)c1)=O N1(C(c2n(CC)ncc2)=O)CCC(C)C(N(C)C(c2sccc2C(C)(C)C)=O)C1 N1(C(CC(C)n2ccnc2)=O)CC=CC(C(=O)NC2CC(O)CC2O)C1 c1(C(=O)NC2CCCCN(C(C(C)SC(C)C)=O)C2)n[nH]c2ccc(Cl)cc12 N1(C(C(N)CCN2CCOCC2)=O)CC(F)(F)C(F)(F)C1 c1(C(=O)NC(CNC(C(Cc2c(OC)cccc2)=O)=O)C)c(C)nc(C)n1O N1(C(CC2(OC)CCC2)=O)CCC2CC(C1)CN(C(c1cc(C)nnc1O)=O)C2 c1(CCC(N2CCC(N(C(=O)C(CC)CCOC)CC)C2)=O)c(C)ncnc1O c1(NC(C2CC3(CCN(C(c4c(C)cc(F)cc4)=O)C3)C2)=O)cc(F)cnc1C#N N1(CCC#C)CCC(C(=O)NCC(C)(C2CC2)NC(=O)CCC2CCCO2)CC1 c1(C(=O)NCC(C)(O)CNC(C2CCn3cnnc3C2)=O)cnn2c1OCCC2 N1(C(=O)N(C2CCCCC2)C2CC2)CCOC2(CCCOC2)C1 C#Cc1cncc(NC(C2CN(C)CCN2C(c2ccc(CC)cc2)=O)=O)c1 c1(NC(C2CCN(C(C(C=CC)O)=O)C2)=O)ccc(O)c(F)c1 c1(OC)nc(C)sc1C(=O)NCC1(CO)CCN(C(=O)C(C)(C)NC(C)=O)C1 c1(C(N2C(C(=O)NCC(C(=O)OC)(C)C)CC(C)(C)C2)=O)cc2cccnn2c1 c1(CC)ncc2c(n1)CCC(C(=O)Nc1ncccc1Cl)C2 c1(C(=O)NCC(=C)CCNC(C2CCCN(CC)C2)=O)cc(C)c(C)cc1C C1(COC)CC(CNC(c2nocc2Br)=O)N(C(=O)C2=CCSC2)C1 Cc1nocc1N(C)C(=O)NC(Cc1ccccc1)C(=O)N1CCNCC1 N1(C(C(CC)=O)=O)CC2CN(C(C3CCC(C)O3)=O)CC12 C(CC(C(=O)NCCCCC(=O)N(C1CC2C=CC1C2)C)OC)OC c1(C(=O)NC2CCC(CNC(C(C)n3cncn3)=O)CC2)cccc(Br)c1O C(F)(F)(C(=O)N1CC(N(C(=O)CN(C)Cc2ccccc2)C)C1)C1(OC)CCC1 C1(N(C(c2c(CCC)occ2)=O)C)CCC(NC(=O)CSc2nncn2C)CC1 C1(CC(=O)NCc2nccc(=NCC3(CN)CC3)[nH]2)CCC2(CCOCC2)CO1 Cc1ccccc1CNc1ccc(N(c2cccc(C(=O)NC(N)=O)c2)C)cc1 CCC(C)C(CC(=O)N(CCCO)C)NC(C1C2CCC(F)C12)=O CC1N(CCCC2CNC2)CC12CCC2 C1(CNC(CC(C=C)C)=O)CC2(CCC2)CN1C(c1c(Cl)ccc(O)c1N)=O N1(C(C2(C)CCCC2O)=O)CCOCC(CNC(c2cc(CC3CC3)on2)=O)C1 c1(CC(N2CC(OC)(CNC(C3(C)CC3(F)Cl)=O)C2)=O)cc(F)cc(Cl)c1 c1(CNC(CSC)=O)ccccc1CNC(c1cc(C2(O)COC2)on1)=O Cc1cc(C(=O)NC(C2CCN(C(C3(C)CCCC3)=O)C2)C)cc(N)c1 C(CC(C(C)C)NC(C1CC(C)N(C)C1)=O)NC(C(c1cc(C)sc1)(C)C)=O C1(NC(C=COCC)=O)(CNC(=O)Cn2ccnn2)CC2CCC1C2 C(=O)(C1CCCc2cccnc21)NC1C(O)CCN(C(C(C)(C)C(F)(F)F)=O)C1 C1(C2CC2)(C(=O)NCC2CC(NC(CC(C)n3ccnc3)=O)C2)CCC1 C(=O)(C1CCOc2ccc(Cl)cc21)N(CCC(F)(F)F)CCOC O=S(=O)(c1ccc(Br)cc1CO)NC1CCCCC1.C12=C(F)C=C(C=C1F)C2 n1(CC(=O)NC(C2CCCN2C(=O)C2=CCC2)C)cc(Br)ccc1=O c1(C(=O)NCC(CNC(CC(CCCC)O)=O)O)ccc2c(c1)OCC(=O)N2 N1(CCCNC(C2CC(CC)C2)=O)CCC(NC(C2CCCC2C)=O)C1 CC(C)C(CNC(=O)CCC1CCCN1C)NC(=O)CSc1n[nH]c(O)n1 CCCCCCC(=O)N1CCC(CO)C(NC(c2cc(Br)c(C)nc2)=O)C1 N1(C(C2(CC)CCCN2C(=O)COc2cccnc2)=O)CCC2(CCCOC2)C1 Cc1cc(CC(N2CC(CNC(=O)CNc3nc(C)cs3)C2)=O)cc(C)c1 c1(C(=O)NC2CN(C(c3coc(Cl)n3)=O)C3CC23)ccc2nc(S)oc2c1 n1(CC(=O)NC(C)(CNC(C2CC2(Cl)Cl)=O)CO)nc(Cl)ccc1=O C12CCC3(CC1)CC3NC(=O)N2.c1(C)cccc(C(C)(C)C)c1.CO CCCC(CC1CCCC1)C(=O)NCCCCCNC(=O)CN(S(=O)(=O)CC)C N1(CC)CN(c2nnc(C(c3cc(C)on3)C)n2C)C(C)CO1 N1(C(C(C)OCC#C)=O)CCC(C(C)NC(=O)CCc2nncs2)C1 c1(OC)cc(C(C)NC(C2OCCC2F)=O)ccc1OC(F)F C1C(CC(=O)O)c2cn1nn2.Cc1nc(C(=O)NCC(C)(C)CO)cs1 N1(C(=O)C(O)Cc2ccco2)CCOC(CNC(C2(CF)CCC2)=O)C1 c1(-c2nc(-c3ccc(OCC)cc3)nn2C2CCC=CCCC2)nnc(O)cc1O N1(C(c2nc(C)oc2)=O)CC2CN(Cc3ccc(I)cc3O)C2C1 N12CCC3(CCCCC3O1)CC(CCCO)C(C)N(C)C(=O)C2=O c1(C(N(C(C)CNC(C2(c3cc[nH]n3)CC2)=O)C)=O)cc2c[nH]cnc-2n1 C1(C(=O)NC(C(C)(C)NC(CCCN(C(C)=O)C)=O)C)CC2OC1C1CC21 C(=O)(C(O)CC(C)(C)C)NC1(CCNC(C(CSC)O)=O)CC1 Cn1c(=O)ccn(CC(N2CCCC(CCNC(=O)CC3CC34CC4)C2)=O)c1=O C1(C(=O)NCC(=C2CN(C(c3[nH]c(=NC)sc3)=O)C2)F)CC(C(C)(C)C)=NO1 N1(C(C)=O)CC(C)N(N(C(=O)NCc2ncc(OC)cn2)C)C(C)C1 C(c1ccco1)=C(C)C(=O)NC1COCC1CNC(=O)CN(C1CCCC1)C c1(C(N2C(CNC(c3ccc(CC)[nH]3)=O)CCCCC2)=O)ccc(CC)nc1C Clc1ccnc(N2CCC(NC3CC(CC4CC4)CN3)C2)c1 C1(CNC(NC(CC)CC)=NCCNC(C)=O)CCc2cc(OC)ccc2C1 N1(Cc2scc(C)n2)CC(Cc2ccccc2)OC(C)C1.c12nccc(n1)N2 c1(CC)ccc(CCC(=O)NCC=CCNC(=O)C(C2CCCCC2)O)cc1 N1(C(C(C(C)C)O)=O)Cc2ccccc2CC1CC(=O)NC1CCCOC1 C1(NC(CC(=O)OCC)=O)CCN(C(=O)CC(C)N2CCCC2=O)C(C)C1 C1(C(N(CCOC)CCNC(=O)C(=O)NC2CC2)=O)CC12CCOCC2 C(=O)(C1OC(=O)c2ccccc21)NCC(C)(O)CNC(=O)C(F)(F)C1(O)CCC1 c1(-c2cc(C(=O)NCC3(NC(C4CCCC4F)=O)CC3)on2)ccc(F)cc1 C1(C(=O)NC2(C(=O)Nc3cnn(CC4CC4)c3)C(C)CCC2)CCOCC1(C)C c1(NC(=O)C(C)CF)ccccc1.CC1C(=O)NCC2(CC2)NC(=O)O1 C12(C(=O)NC3C=CC(C(=O)N(C(C)CN(C)C)C)C3)CCC(CO)(CC1)C2 C1(NC(c2csc(C(C)=O)c2)=O)CC1C1CCN(C(=O)CC2=CCN(C)CC2)CC1 c1(CNC(C(C(C)C)SC)=O)nnc2n1CCN(C(C1CC13CCC3)=O)C2 c1(C(=O)NCC2CCN(Cc3ccc(C)nc3Cl)CC2)cc2cc(Br)ccc2[nH]1 C1(NC(CC(C)OC)=O)CC2CCC(C1)N2C(C1(c2ccn(C)n2)CC1)=O N1(C(c2c(C(=O)OCC)con2)=O)CCC(CNC(=O)CC2COCCO2)CC1 C(CCC(=O)N1CC(=O)N(C)C(C)C1)(C(C)C)NC(C1(OCC)CC1)=O CC1CCCc2nc(C(=O)NCC3CCCN3C(=O)C=Cc3ccccc3)cn21 C1(C)(C(=O)NCCCOCCN(C(C(CC)F)=O)C)CNC(=O)N1 C(=O)(C1CCCc2nn[nH]c21)NCC(CNC(C(C(C)(C)C)=O)=O)(C)O C1(C(=O)NCc2c(C)ncs2)CC(C)(C)CCN1C(=O)CCn1cccc1 C(=O)(C(C)CCCC(C)C)N1C(CC)CN(C(=O)CCCCOC)CC1 C1(NC(c2ccc(C)[nH]2)=O)CN(C(c2cc(C(C)(C)C)n[nH]2)=O)CC2(CC2)C1 C1(CNC(CNC(=O)OC)=O)COCCN(C(=O)C(CN(C)C)N(C)C)C1 C(=O)(C(O)C(F)(F)F)NCCC1(NC(c2nccc(N)c2)=O)CC1 C1(N(C(C(C)(C2CCC2)NC(c2cccnc2O)=O)=O)C)CCCCCC1O c1(C(N(CC(CNC(C(CC)(C)C)=O)C)C)=O)nnn2c1C(=O)NCC2 CC12CC(C(N3CC(NC(c4cccs4)=O)CC3(C)C)=O)(C1)C(C)(C)O2 Cc1oc(C(C)C)nc1C(=O)NCC=CCNC(c1csc(-c2cccs2)n1)=O C(=O)(C(O)CNC(=O)C(C1CC1)NC(c1cc(C(N)=O)[nH]n1)=O)NC C=CCC(CC=C)C(=O)NCCN(c1nc(C(C)=O)c(C)s1)C1CC1 C1(CN(C(=O)C=Cc2ccco2)C)CCN(C(C2CC(N3CCCC3)C2)=O)CC1 c1(NC2CC(C(=O)NC(C(CC)O)C)C2)cc(O)nc(O)n1 CC1(C)CC1(C)CNC(=O)C(O)C1CN(C(=O)COC2CC2)C1 C1(COC)(CNC(=O)Cc2cc[nH]c2)CN(C(=O)CCCN2CCCCC2)C1 c1(C(=O)NC2CC(NC(=O)CCn3cnnn3)C2)ccc(-c2cn[nH]c2)cn1 Cc1cc(=NCC(CNC(C2CCCN2C=O)=O)C(F)(F)F)[nH]c(Cl)n1 N1(C(C(=Cc2cccs2)C)=O)CC(NC(=O)COC2CCOC2)CC(C)(C)C1 C(=O)(C(C)C(O)C(C)C)NCC(C(=O)N(C)CC1CC1(F)F)OC N1(C(C(C)NC=O)=O)CC(NC(c2cc(F)ccc2Br)=O)CC(F)(F)C1 N1(CCCC)CCN(CCCNc2ccc(Cl)cc2)CC1 Cc1ccc(O)c(CC(N2CCN(C(=O)CCS(C)=O)CC2CCO)=O)c1 C1(C(=O)NCCN(C(CC)C)CC)CN(C)CCN1C(=O)CSc1nc[nH]n1 N1(C(C(CCC)O)=O)C2CCC(C2)C1C(=O)Nc1ccc(N(C)C)cc1C CCCCC(O)CC(=O)NC1CC(CNC(c2sc(OCC)nc2C)=O)C1 N1(C(c2cc(CNC(C3(OC)CCC(C)C3)=O)sc2)=O)Cc2nc(C)sc2C1 CC1CCN(C2CCN(C(c3cc(Cl)c(I)s3)=O)CC2)CC1 c1(CN(C(=O)N=C(C)CCN2CCCC2)Cc2ccccc2)cccc(C#N)c1 Cc1ccc(O)c(CNC(c2ccc(CNC(=O)C(C)c3ccco3)cc2)=O)c1 Cc1noc(C(=O)NCCCCNC(C2CCC(C)C2)=O)c1C c1(CNC(C2(CC)CCCN2C(=O)C=Cc2ccncn2)=O)ccc(F)c(O)c1 c1(C(N(C2CCNCC2)C)=O)cccc(C(=O)O)n1 c1(OCCC(=O)OCC)cccc(F)c1.CC(CC(C)NC(=O)Cc1cn(C)nn1)N c1(CC)csc(CCC(N2CC(C)(NC(=O)C(C)Cc3ccco3)C2)=O)n1 C1(O)(C(N2CC(OCCNC(C3(CCN(C)C)CC3)=O)C2)=O)CC2CCC1C2 c1(CN(C(=O)CC2(O)CCC2)CC)ccc(CNC(C2CC(=O)N(O)C2)=O)cc1 Cn1nc(C(=O)NCCOCCn2cc(CCO)nn2)c(Br)c1Cl C(C(C)N=c1nc(N(C)Cc2cnc[nH]2)c2c(F)cccc2[nH]1)OC(C)C C(=O)(C1=CCCN(C(=O)C(C)(C)N2CCCC2)C1)N1C(C)CC(C)(C)C1 c1(OC)cc(C(C)Nc2ccc(OC(=O)N(CC(C)O)CCO)cc2)ccc1O N1(C(C2(CCOC)CCCC2)=O)CCCC(NC(C2(CCO)CC2)=O)C1C C1(NC(CCN(C(C)=O)C)=O)C2CCN(C(=O)CC3CC(C)(C)CO3)CC12 Nc1cc(F)c([N+](=O)[O-])cc1C(N1CCOCC(O)C1)=O C(=O)(C(=O)N=S(C)(C)=O)NCC1C(C)CN(C(=O)CC2CN3CCN2CC3)CC1 C=CCC(CC(C)C)C(=O)Nc1ccc(NC(C2CN(C3COC3)C2)=O)cc1C CC(C(=O)NCC12CC(NC(=O)CCCCCc3ccccc3)(C1)C2)C(F)(F)F c1(NC(N(C)CC2CCCSC2)=O)cnc(C#N)c(Br)c1 c1(C(=O)OC)cc(C(=O)OC(c2ccn(CCSCC)n2)=O)cc(C#N)c1 c1(C(N2C(CCNC(c3ccc(C)cn3)=O)CC(OC)C2)=O)c(C)ccnc1C N1(C(C2(C(N(C(C)C)C)=O)CC2)=O)CCN(C(=O)C(O)C(F)(F)F)C(CF)C1 C(=O)(C#CC(C)(C)O)N1CC(C(C)NC(c2cnc(Cl)s2)=O)OCC1 C12CCN(CC1)C(=O)C(OC)C(=O)N2.c12ccc(cc1)[nH]c2=O.C(C)(=O)OCC C12(NC(C3CCCC(NC(C4(C)CC4)=O)C3)=O)CC1COC21CCC1 C(C(O)C(=O)NC1CCC1)NC(CCNC(COC)=O)=O C(c1ccc(F)c(F)c1)=C1CN(C(C2C(C)CN(C(=O)CC(F)(F)F)C2)=O)C1 C1(CNC(C=CC(CC)C)=O)CN(C(=O)C(C)CS(C)(=O)=O)CC(C)(C)C1 C1(NC2(c3n(C(C)C)nnn3)COC(CC3CC3)C2)CCc2nnnn2CC1 N1(C(CCC(C)C)=O)CCC(NC(C2CCC(C)(C)CO2)=O)C(O)C1 c1(NCC(CCC)C)cc(N2CC(OC)CC(OC)C2)nc(COC)n1 c1(C(N2CC(O)(CNC(C3(C)C(C)(C)C3)=O)C2)=O)ccc(Cl)c2ccccc12 CC(C)P(=O)(OC)C(=O)CCn1cc(CN)nn1 C(=O)(C1=NNC(=O)C1)NC(C(C)NC(c1ccncc1C(F)(F)F)=O)C C12(C(=O)NC3CCN(CCOC)C3)CCC(CC1NC(C1CCC1OC)=O)C2 c1(C(CNC(c2ccccc2-c2ccncc2)C)O)ccc(-n2cnnc2)cc1 N1(C(c2cc(C(C)C)on2)=O)CC2CCC1C(NC(=O)CCc1cn[nH]c1)C2 c1(CC)cccc(C(N2CC3(CC(NC(C4CCC(O)CC4)=O)C3)C2)=O)c1C CCC(C)(C)C(C)CC(=O)NC1(CNc2ncc3ncnc-3[nH]2)CC1 Cc1cc(CNC(C2COC(CNC(=O)C(C)(C)c3ccsc3)C2)=O)ccn1 N1(C(c2cccn(C3CCC3)c2=O)=O)CCCN(C(C2CCC2)=O)CCC1 Cc1ccc(Cl)c(O)c1C(N1CCC(CNC(C2CC3(C2)CC3F)=O)C1)=O C1(NC(CCN(CCC)C)=O)CC1C1CCCN(C(c2cc(C)nc(O)n2)=O)C1 N1(C(c2c(C)cncc2)=O)CCCOC(CNC(=O)Cc2nncn2C(C)C)C1 Cc1ccc(C(=O)NC2C3CCN(C(C4CSCCS4)=O)C23)cc1-n1cccc1 c1(C(CNC(CC=C(C)C)=O)NC(C2OCC2(C)C)=O)ccccc1F CN=c1nc(NC(C)(C)CCOc2ncccc2Br)cc(C)[nH]1 CCC(CC(=O)NCCC(F)(F)F)N(C(=O)C(CC1CCC1)OC)C C1(NC(c2ccc(C#C)cc2)=O)CC2CCCC(C1)N2C(C1(C(C)C)CC1)=O c1(C(N2CC(C(C)NC(=O)C=CC(F)(F)F)OCC2)=O)nccn2ccnc12 C12(CS(N3CCC(Br)=C(C)C3)(=O)=O)CC3CC(CC(C3)O1)C2 c1(C(N2CC(CCC)C(NC(C34CCC(C3)C4)=O)C2)=O)ccc(F)c(O)c1F N1(C(c2nc(C)oc2C)=O)CC(C(N2CCC(N3CCC3)C2)=O)CCC1C c1(C(=O)NC(CNC(c2c(O)ccc(C)c2)=O)C)cn2cc(Cl)cnc2n1 CC1(C)CC1(c1cccs1)C(=O)NC1CC(CNC(=O)CCc2cnco2)C1 CCC(C)CN=c1cc(C)c(C(=O)N)n[nH]1.C(C)=O O(NC(=O)C1=NOC(CN(C(c2sncc2C)=O)C2CC2)C1)CCOC c1(C(CNC(=O)NC(c2ncc(Cl)s2)C)(C)C)ccccc1[N+](=O)[O-] c1(N(C2CNCCC2(F)F)C(c2cc(CC)on2)=O)cc(C)nc(SC)n1 C1(N(C(=O)C(C)CO)CCC)CCN(C(c2ncoc2COC)=O)CC1 N1(C(c2ncn(C)c2)=O)CC(NC(c2cccc3ccsc23)=O)C(N=[N+]=[N-])C1 c1(COC)ccc(C(=O)NC23CC(CNC(=O)CC4CC5CCC4O5)(C2)C3)cc1 c1(C(C)C)cccc(NC(=O)NC(C23CC(NC(C4CCSC4)=O)(C2)C3)=O)c1 c1(C(=O)NCCN(C(C(C(=O)OC)C)=O)C)c[nH]nc1S(N)(=O)=O C1(C(N2CC(C)(C(=O)NCCC(C)N(CCC)C)C2)=O)CCC(C)CC1 Cc1cnc(C(=O)NC2C=CC(CNC(C3(C(=O)NC4CC4)CCC3)=O)C2)cn1 C(=O)(CCCCSC)NCC(CC=C)NC(=O)CNC(=O)C1CC1 Cc1ccccc1C(C)(C)C(=O)OCC1CCN(C(C2CCC(O)C2)=O)CC1 C(=O)(CC(C)(C)CC(=O)N1C2CCCC1CN(C(=O)COC1CC1)C2)OCC c1(N(C(c2cc(-n3ccnc3)cs2)C(=O)NCCOC)C)ccc2sccc2c1 c1(C(N2CC(CNC(CCOCCC)=O)C3C2C3)=O)ccc2nnnn2c1 CC(C)C(=O)NNC(=O)c1ccc(-n2cc(CN(CCO)C3CC3)nn2)cc1 c1(C(=O)Nc2cc(C)n(C)c(=O)c2)ncn2cc(Cl)ccc12 Cc1ccc(C(N2CCCC2C(N2CCC3(CC2)CC(=O)N3)=O)=O)c([N+](=O)[O-])c1 C1(NC(CC(C)N2CCCC2=O)=O)CN(C(c2cc(Cl)c[nH]2)=O)CC2CC12 N1(CC(N2CCCC2Cn2cc(C3CC3)nn2)=O)CCOCC1CC1CCC1 N#Cc1ccc(-c2cncc(NC(c3cc(F)c[nH]3)=O)c2)nc1 c1(CN2CC(O)(CNC(c3cc(Cl)cnc3O)=O)C2)cccc2ccoc12 C1(C(=O)NCC(C)CNC(=O)Cc2ccsc2)CC2CCC2C1 C(CCSC)(C(=O)NC(CCNC(c1c[nH]nc1C1CC1)=O)C(C)C)OC C1(NC(=O)NCCC(=O)NC(CC)C)CC(OCC)C12CCCC2 C(=O)(CCCC(=O)NCC(C)(O)CNC(c1c[nH]nc1[N+](=O)[O-])=O)NC(C)C c1(NC(C2N(C(c3n(C)ncc3)=O)C3C(C2)C3)=O)c2c(nn1C)CCC2 c1(C(=O)NC2(CCCNC(C3CCCS3)=O)CC2)ccnc(CO)c1 C1(NC(C2(NC(c3ccc(C)s3)=O)CCSC2)=O)CCN(C)C(C)C1 N(C1CCOc2c(Br)cccc21)C(CN1C(=O)C(c2ccc(Cl)cc2Cl)CCC1)=O CC1CC(NC(c2ccc([N+](=O)[O-])[nH]2)=O)CN(C(c2ccccc2)=O)C1 C1(C(N(CCNC(c2cc(COC)on2)=O)C)=O)CCN2CCC1C2 C(=O)(CCC(C)(F)F)NCC(CCOC)NC(c1cc(Br)cnc1O)=O C1(CNC(CSSC)=O)CCCC12CCN(C(C1CC3CCCC13)=O)CC2 N1(C(C(C(C)(C)O)F)=O)CCC2(CCCN2C(=O)C(F)C2CCC2)CC1 C(C(C)(C(=O)NC1CCCN(C(=O)CO)C1)OC)OC N1(CC(=O)NCC(CN(C)C(c2cnccn2)=O)O)CCCCC1 C1(OC)CN(C(=O)C=C(C)I)C2(CCCC2)C1 Cc1cccc(S(=O)(=O)NCc2ccccc2C2(C)NC(=O)NC2=O)n1 c1(OC)c(F)cc(N(C)CCOc2cccc([N+](=O)[O-])c2)cc1F C=CCC(C(=O)N(C1CCN(C(c2c[nH]ccc2=O)=O)C1)C)OC Cc1c(Cl)cc(C(N2C3COCC2CC(NC(=O)OC(C)(C)C)C3)=O)cc1I c1(C(=O)NCC(CC=C)NC(=O)CC(C)COC)cc(C(F)F)ccc1F N1(C(c2ccc(SC)cc2)=O)CCCC2C1CCN2C(c1cnc(S)n1C)=O C=CC1(C(=O)NCC(C2CC2)NC(=O)CCc2c(C)noc2Cl)CCCCC1 C1(NC(CC23CC(C)(OC2)C3)=O)CC12CCN(C(C1(C3CC3)CC1)=O)CC2 C1(C(=O)Nc2cc(Br)cc(F)c2F)CC(c2c(F)cccc2F)=NO1 c1(C(N(C2CC(SC)C2)C)=O)coc2c1CN(C(c1cncc(C)c1)=O)C2 Cc1ccc(OCC(=O)NCC2CCN2C(=O)C(C)NC(C2CCC2)=O)c(C)c1 C(=O)(C(CO)C(C)(C)C)N1CCCC(CCNC(COCCCOC)=O)C1 N1(CC(=O)OC)CCN(C(c2ccc(NC(C3CCCC3C)=O)s2)=O)CC1(C)C c1(NC(C(C(C)O)NC(C2C(C(=O)OC)CC2)=O)=O)cccc(C#N)c1 c1(C(=O)NC2CCC(NC(c3nc(C)c(Br)cc3)=O)C2)cc(Cl)c(Cl)cc1F N1(C(C2(O)CC2)=O)CC2CN(C(C3(N(C)C)CCCC3)=O)CC(C1)O2.CCS N1(C(Cc2c(C(=O)OC)c[nH]c2)=O)CCN(C(=O)Cn2cncc2C)C(C2CC2)C1 CCC(O)C(C)C(=O)N(CCN(C)C(c1nn(C)c(N)c1C)=O)C(C)C Cc1[nH]nc2cc(C(=O)NCC3CC3CNC(=O)C#CC3CCOC3)ccc12 C=CC(C)(C)CC(=O)NCC(C1CCCC1)NC(C1CCC(F)(F)CO1)=O c1(-n2cc(C(C)OC(c3c(CC)scn3)=O)nn2)cc(Cl)cc(Cl)c1 c1(CC(=O)NCC(N(C)C(C2CC2(C)C)=O)C2CC2)nc(-c2ccccc2)no1 N1(C(c2cn(CC)nc2)=O)C(CNC(=O)CC2CCCCC2C)CC2COCC12 Cc1cc(C(=O)N(C2CCN(C(=O)C=Cc3cccc(Cl)c3)C2)C)cc(C)n1 C12(C(N3CCC(NC(Cc4ccc(OC)cn4)=O)CC3)=O)CCC(CC1)C(C)O2 c1(C(CCC2(C)CC2)NC(c2n(C)nnn2)C2CCOCC2)ccc(CC#N)cc1 N#CC1(NS(=O)(=O)C(F)(F)F)CCN(Cc2cncc(O)c2)C1 c1(C(=O)NC2CCN(C(c3c(C)cn(C)n3)=O)C(C)C2)cc(O)c2ccoc2c1 C1(NC(c2cncnc2)=O)CC(O)CN(C(c2ccc(-c3ccccc3)o2)=O)C1 c1(C(C)NC(=O)NC(CCC)C2CC2)c(Cl)cccc1Cl CC(C)CC(=O)NC1CC1NC(=O)Cc1cnoc1 N1(C(C(CCC)CCC)=O)CCCCC2(CCN(C(=O)C(C)C3CCCO3)C2)C1 Cc1cc(C)c(NC(=O)C(N2CC3CN(C)CC3C2)COC(C)(C)C)c(C)c1 N1(C(C2CCC(N(C)C)C2)=O)CCN(C(c2csc3nccn23)=O)C(C2CC2)C1 CC1CNc2c(C(N3CC4CCN(C(c5cnns5)=O)CC4C3)=O)cnn2C1 C1(NC(c2ccc(Br)s2)=O)CCC12CCCN(C(c1ccco1)=O)C2 CC1CC(NC(C23CCCN2CCC3)=O)CCN1C(c1ncccc1Cl)=O CC1CC=C(C(=O)NC2CCCCCN(C(=O)C(C3CCCCCC3)O)C2)CC1 Cc1cc(CCC(=O)NCCCC(C)NC(C2CN(C(N)=O)C2)=O)on1 N1(C(COCCCOC)=O)CC2(C1)SCCC2NC(c1cccc2nnnn12)=O c1(N2CCC(NC(C(CCCC)CC)=O)CC2)ncnc2ccc(F)cc12 c1(SC)cn(C)nc1C(N1CCC(N(C(C2CC(OC)C(OC)C2)=O)CC)C1)=O C1(C(=O)NC(CNC(C2(CC)CC(F)(F)C2)=O)C)CC2(CCC(F)(F)CC2)C1 C(C(C)C)(C(O)C(=O)N1CC(C(C(=O)N(C)Cc2occc2C)OC)C1)OC CC(O)C(C)(C)C(=O)NCC=C1CCN(C(c2ccnc(C(=O)OC)c2)=O)CC1 C1(NC(Cc2c(C)n[nH]c2)=O)C2CN(C(=O)C(C(C)C)OCC(C)C)CC12 Cc1cccc(C)c1OCCC(=O)N1CCC1CNC(=O)C=CS(C)=O C12=NC(=NCCSCCN1)Nc1cccnc12.N=c1nc(Cl)cc(CCCO)[nH]1 c1(C2C(CC)CC2)nc(-c2ccc(C(F)(F)F)cc2)nn1CCOC C(=O)(C(CC)(CC)CCCCCC)N1CCCC(CN(C(C(CC)=CC)=O)C)C1 c1(OCCC)cccc(C(=O)NC(C)C(C(C)C)NC(=O)C=C2CCCC2)c1 c1(C(=O)NCc2ccc(CN(C(C(C)OCC=C)=O)C)cc2)nn(C)cc1Cl NCCC(F)(F)CNC(=O)COC(=O)C(c1ccccc1C(N)=O)N C(=O)(C(F)(F)F)COC1(CC(=O)NCCC(C)NC(=O)Cc2ccccc2)CC1 n1(CC(N2CC(c3c(CNC(C=CC(C)(C)C)=O)nco3)C2)=O)ccccc1=O N1(C(c2cc(CC)n(C)n2)=O)CCC(NC(=O)C(O)C(F)F)C12CC2 CCC(Cc1cccc(C)c1)C(=O)NCC1(CNC(=O)C(C)N(C)C)CCCC1 c1(OC)ccc(C(C)C(=O)NCC2CCCN2C(C2SCCS2)=O)cc1F c1(C(=O)NC(C2CCCC2)CNC(c2cn[nH]c2)=O)ccnn1CCF Cc1cc(CNC(C2CC3CCC2N3C(=O)CC2CSC2)=O)cc(C)c1 c1(C(=O)NC(c2ccccc2F)CNC(CCC=C)=O)ccc(OC)c(Cl)n1 c1(C(N2CC(NC(C3CC(OC)C3)=O)C(C)CC2)=O)c(Cl)ccc(O)c1Cl c1(OCC(=O)NCC2C(C)CCNC2=O)ccc2nc(O)[nH]c2c1 C1(NC(CN(C)C)=O)CCN(C(c2ccc(N)c(Cl)c2O)=O)CC1(C)C c1(C(N(CCCCNC(=O)CN(C)S(N)(=O)=O)C)=O)cc2occc2s1 Cc1nc(F)ccc1-c1nc(NC(c2c[nH]nc2-c2cccc(C#N)c2)=O)cs1 c1(N(C(=O)C(C2CC2)NC(=O)CN2CSCC2=O)C)ccc(Cl)cc1F Cc1cccc(C)c1NC(=O)CN1CC2CC1CN2Cc1c(Br)ccnc1Br C(=O)(CCCCCc1cccs1)N(C1CC(NC(C2C(CC)OCC2)=O)C1)C Cc1cnn(C)c1CC(=O)NCCCC(C)NC(c1cn(C)cn1)=O C1(C(N2CCCC(CNC(C3CC(OC)C3)=O)CC2)=O)CC2CCC1NC2=O C1(N(C(CCC#C)=O)CC)CCC2(CC1)CN(C(=O)C=C(CC)CC)CCO2.CC C(CCCCCC(=O)NCC(C)(C)CNC(=O)CC(c1ccc(C)cc1)C)SC C1(C(=O)OC)CC(N=c2cc(C#N)cn[nH]2)C12CCC2 C1(NC(=O)CSc2ccncc2)CCCC12CCN(C(=O)C1=CCCCO1)C2 C1(=CCNC(c2cn(CC)nc2)=O)CCN(C(=O)C(C)C2CCCC2)CC1 c1(CNC(=O)C(=O)N(C2CC2)Cc2cccc(OC)c2)cc(F)ccc1Cl c1(OC)cc(CCC(=O)NC2CC2Sc2cccs2)ccc1O.C1(=O)CN1 C1(C(N(C2(C)CCC2)C)=O)CN(C(=O)CCc2ccn(C)n2)CC1(F)F c1(CC(=O)NCC(CN(C)C(C2CC3CCC2C3)=O)O)ccc2sccc2c1 c1(CC)cccc(S(=O)(=O)N2CC3CN(C(c4cccnn4)=O)CC3C2)c1 c1(C(=O)NC2(CC=C)CCOC2)cn(CCF)nc1C.c12cc(n[nH]1)C(=O)NC2 c1(C(=O)NCC(C(=O)NCc2ccccc2CC#N)N(C)C)ccnnc1O C1(NC(CC(C)N(C)C)=O)Cc2nccnc2CN1C(=O)CCc1ccccc1 N1(C(C2CCN(CC)C2)=O)CC(F)(F)CC1C(N1CCC(C)(O)C1)=O c1(N2C(CNC(c3cccc(OC)c3)=O)CCCC2)nc2ncc(Cl)cc2o1 C1(OC)CN(C(C2CCCCC2NC(c2cc(C3CC3)[nH]n2)=O)=O)CC12CC2 N1(C(C2(C(C)C)CCC2)=O)CCC(C(C)(O)CNC(=O)C=CCO)CC1 C(=O)(C1=CN(CCC2CCN(C(C3N(C)CCOC3)=O)C2)CC1)OC(C)(C)C C12(CC(N3CCC(N(C(CS(=O)(=O)NCC)=O)C)C3)=O)CCCCC1C2(F)F Cc1cc(NC(=O)C(CO)NC(C2(C)CCOCC2)=O)cnc1O c1(C(=O)NC2C(SC)CN(C(=O)C(C)(F)F)C2)c[nH]c2cccc(Cl)c12 CC1CC(C(=O)NCCN(C)C2CC2)CN(C(=O)Cn2cnnc2O)C1 c1(CC(N2CCC(CN(C(c3[nH]cc(CC)c3)=O)C)C2)=O)cccc(CC)c1 c1(C(C(=O)NCC2(CNC(CCSC)=O)CC2)C)cc(C)cc(F)c1 Cc1[nH]nc(Cl)c1C(=O)NCC1(C(N)=O)CN(C(C2CCO2)=O)C1 C(CC(C)C(C)(C)C)NC(C1C(CNC(C(c2ccn(C)c2)C)=O)CCO1)=O C1(C(=O)NCCOCCOCCCNC(CC(=O)NC)=O)C(Cl)(Cl)C1(C)C Cc1nc2cc(C(=O)NC3CCCCN(C(=O)CCCCC(C)C)C3)cnc2s1 c1(C(C(=O)N(CCNC=O)CC2CC2)(F)F)nc2ccccc2s1.C(=O)(C(F)F)N c1(SC)nc(O)nc(C)c1C(N1CCCC(NC(C2CC(Cl)(Cl)C2)=O)C1)=O C1(CNC(CCN(C)CC)=O)C2CN(C(C3CCC(=O)N3)=O)CC12 C1(N(C(CCc2c(C)n(C)nc2)=O)C)CCC2CN(C(=O)CCOC3CC3)CC12 N1(C(C(C(C)C)SC)=O)CCN(C(c2ccc3c[nH]nc3c2)=O)CC(C)C1 C(=O)(N=c1cc(CC(C)C)[nH][nH]1)OC(CCc1c(Cl)ccc(OC)c1)=O C(CS(=O)(=O)CC(=O)NC1CCOCCC1C(N1CCOCC(C)(F)C1)=O)OC c1(C(C(=O)NCC(C)C)N(C)CCn2cc(Br)cn2)cc(F)c(Cl)cc1Cl C(C)(C(=O)NCC1(NC(c2cnoc2C)=O)CC1)(C1(C)CC1)OC CCC(C)CCC(=O)NCC(C)(C)CNC(c1cc(C(=O)OC)ccc1N)=O C1(C(N2C(CN(C(C(C)N(C)C)=O)C)COCC2)=O)CC12CCCCC2 C12(C(N3CCC(N(C(CC=C(C)C)=O)C)C3)=O)CC1COC2(C)C c1(C(C(=O)NC(C)C)N(CCN(C)C)CC)ccn(C2CC2)n1 CS(=O)(=O)CCCC(=O)NCNC(C1CCC1NC(=O)C(C)C)=O.C1(=O)C(CO)N1 C1(CC(=O)N(CCCC)C)CN(C(C2CC2OC(C)=O)=O)C(C)(C)C1 C1(NC(=O)CC2CCC2(F)F)CCC(CNC(=O)CN2CCCC2=O)CC1 N1(C(c2cc(NCc3cc(OCC)ncc3)cn2C)=O)CCOC(C#N)C1 N1(C(CCNC(=O)OCC)=O)CCC(C2CC2)(NC(=O)CCCN(C)C)C1 N1(C(CC(=C)C)=O)C2CCC1C(C)C(NC(c1ccn(CCC)n1)=O)C2 N1(CC)CCC(NC(=O)CCC2CCN(C(C3CC3C(F)F)=O)CC2)C(C)C1 CC1CCCCN1CCOC(C1(NC2CCC2C(C)(C)C)CCOCC1)=O C1(C(=O)NCCn2ncc(C(=O)NCCc3onc(C)n3)c2)CCCC(=O)C1 C(=O)(C1CCCc2nc[nH]c21)NC1CCN(C(CC2=C(C)CCC2)=O)CC(O)C1 c1(OC)ncc(C=CC(N2CCN(C(C3CCCC4CC34)=O)C(C)C2)=O)cn1 c1(CNC(=S)NCC2CCC2)cc2c(s1)CCC2 CC(C)C(O)(C(=O)N1CCC(C)(C)C(NC(C2CCCCCC2)=O)C1)C(F)(F)F c1(CN(C(c2cn(C)nn2)C(=O)NCC=C)C2CC2)ccc(Br)cc1 C=CCC(CNC(=O)C(C)(C(C)C)OC)C(=O)NCC(C)(F)C(C)(C)F c1(OC)ncc(C(=O)N(CC(C)NC(c2cncc(C(C)(C)C)c2)=O)C)cc1F c1(CC)cccc(C(N2CCC(NC(c3cc(C)cc(O)n3)=O)C2)=O)c1F N1(C(C=Cc2cnc(C)s2)=O)CCCC(NC(c2c(CO)noc2C)=O)C1C c1(CCCC)ccc(C(=O)NC(C)C(C(C)C)NC(=O)Cc2cncn2C)cc1 C(=O)(C(O)c1ccco1)NCCOCCCNC(CNC(=O)OC)=O CCCCC(CC)CC(=O)NCC(CCCC)NC(C1(CC)CCOC1)=O C#Cc1cc(C(=O)NC(C)(C)CC(=O)N2CCCC(C(C)O)C2)ccc1C N1(C(c2c(C)n[nH]c2C)=O)CCN(C(=O)Cc2ccc3nn[nH]c3c2)C2CCC12 c1(CNC(C2(OCC)CCOC2)=O)cncc(C(=O)N(CCC(C)(C)O)C)c1 c1(CNC2C(CNC(=O)C(C)OC)CC(OC)O2)ccc(C(F)(F)F)nc1 CCN=C(NCCC1COCCO1)NC1CCN(c2cnn(C)c2)C1 c1(C(N(CC(C)CNC(=O)C(C)CC(N)=O)C)=O)cc(F)cc(Cl)c1N N1(C(C2(OC)CCC2)=O)CC2CCCC(C1)N2C(C1CCOC(C)C1)=O C1(C(=O)NC2C3CN(C(C4(CC=C)CCOC4)=O)C2C3)CCc2nnc(O)n2C1 c1(OC)ccccc1C(=O)NCCOCCNC(=O)C=Cc1sccc1Br Cc1cn(C)nc1C(=O)NC(C)CC1CN(C(C2(O)CC(F)(F)C2)=O)C1 C1(C(=O)NCC2(CNC(C(C)=C(C)C)=O)CCC2)CCC(F)C1 C1(CC=C)(NC(c2nccn2C)=O)CN(C(=O)Cn2nccc2C)C1 Cc1ncc(C(=O)NCC2CCCN2C(C2C3CCN2CC3)=O)c(O)n1 c1(C(=O)NC2CCN(CCNC(c3coc(Cl)n3)=O)CC2)cnc2[nH]cnc2c1 Cc1c(NC(C2CC2NC(c2cc(O)cc(F)c2)=O)=O)cccc1Cl Cn1ccc2cc(C(N3CC4CN(Cc5cc(Cl)ccn5)C4C3)=O)ccc12 C(=O)(CN=c1cc[nH]cc1)N1CC(C(=O)NC2(C3CC3)CC2)CC(C)C1 C(=O)(C1=CC2CCCCCC12)NCCCNC(c1c(Br)cn(C)n1)=O c1(NCC=C=C)nc(C)cc(=NC2CCCN(c3nc(C)cc(C)n3)C2)[nH]1 N1(C(Cn2ncc(C(=O)O)c2)=O)CCCC(CN2CCC(CO)CC2)C1 C(=O)(CC(C(=O)N1CCC(CCNC(c2ccsn2)=O)C1)NC(C)=O)OC c1(OC)ccccc1C(=O)NC1CCOC1C(N1CCSCC1C)=O C1(c2cn(CC(COC)O)nn2)CCN(C(c2sccc2C2CC2)=O)C12CC2 O=C(C1=CCCCCC1)N1CC(CC(F)C(=O)NCC=Cc2nccs2)C1 c1(C(=O)NCCC2(O)CN(C(C(C)NC(CC)=O)=O)C2)cncc(Cl)c1 c1(C(N2CC(OCCNC(CCc3n(C)ccn3)=O)C2)=O)ccccc1Cl C1(Nc2cc(CC)ncn2)CCCCN(C(=O)C=Cc2ccco2)C1 c1(OC)ccc(CNCC2CC(OC)C2)c(Br)c1OC S(=O)(=O)(c1ccc(NCCC(F)F)nc1)NC(c1nc(C)oc1C)C c1(CC)ccc(F)c(C(=O)NC2CCC(CNC(C3(O)CCCCC3)=O)C2)c1F N1(C(c2c(C)cc(Br)c(F)c2)C(=O)NC(C)C)CCN2CCCC2C12CCC2 C(=O)(C1CCCc2ncnn21)N1C2C(NC(CCCCCC=C)=O)CC(C2)C1 c1(C(CNC(=O)COCCCF)NC(C2(F)CCOC2)=O)ccccc1Cl Cn1[nH]c(=NC(c2ccccc2)C=O)c([N+](=O)[O-])c1C(F)(F)F.c1cscc1Cl c1(CN(C(=O)CSCC)CC)ccc(F)cc1.C12(CCCNC1=O)C(=O)NC2 c1(OC)cccc(OC)c1CN1CCCC1CO.N1(C(=O)CN)CCS(=O)(=O)CC1 CC(C)CCCC(C)C(=O)NC(C(=O)NCCOC1CC1(F)F)C1(C)CC1 N1(C(c2c(C)noc2C)=O)CC2CN(C(C3CCN3C3CCCC3)=O)CC2(C)C1 CC(C)C(N)C(c1ccccc1)NCC(=O)Nc1n[nH]cc1-c1ccncc1 CC1=C(C(=O)NCC(C)CNC(C2(F)CCOC2C)=O)Cn2nnnc2N1C Cc1nc(C(C)C)[nH]c(=NC(C)C2CCCCN(C(c3cn(C)cn3)=O)C2)c1Br C1(CC)CN(C(=O)C(c2cccnc2)C)CCN1C(c1ccc(CO)cc1)=O CC1(C)CCCN(C(c2csc(CC3CC3)n2)=O)C1CNC(=O)CNC=O c1(CNC(C(CSC)(C)NC(=O)CCCOC(C)C)=O)ccc(C)c(C#N)c1 N1(CC(N2CC(CCCNC(C3C(C)C3)=O)OCC2)=O)C(=O)NC(C)(C)C1=O CC1=C(C)CC(C)(NC(C2C=CC(NC(C3CCCCC3)=O)C2)=O)CC1 C1(CC(=O)NCC(C)NC(=O)C(C)OCC2CCCCO2)CCCCC1(F)F c1(NC(C2(NC(c3ccc(N(C)C)nc3)=O)CC2)=O)cc2cc(F)ccc2[nH]1 C1(C(=O)NC2(C(N(C)OCC(F)(F)F)=O)CCC2)CCC=CCC1 C1(NC(=O)OC(C)(C)C)CC2CC(NC3(C)CCC(=O)NC3)CC12 C(=O)(CCC(C)CN(C)C)N1C(CC)C(NC(=O)CCOC)CC1 C1(C(=O)NCC(CNC(CC2N(C(C)C)CCC2)=O)(C)F)CC2(CCCC2)CO1 C1(C(N(CC(CC)O)CC)=O)COC(CNC(c2cnn(C)n2)=O)C1 n1(CC(=O)N(C)CC2CCN(C(C(COC)(C)O)=O)CC2)cnc([N+](=O)[O-])c1 C1(CNC(c2cnns2)=O)CN(C(=O)Cc2ccno2)CCC1(F)F C(=O)(C#CC1(CC)COC1)N1CCN(C(CC(COC)C)=O)C(CC(F)F)C1 c1(OC)c(C(N2CCCC(OC(c3ccn(C)n3)=O)C2)=O)sc(C)c1Br C1(C)(C(N(CCCCCCNC(C2C(C)CC2)=O)C)=O)CC2(CCC2)C1 CC(C)(C)C(CNC(=O)CCCC1CCCC(=O)N1)NC(=O)Cn1nccn1 N12CCC(C3CC3)(C1)CNc1ncc(s1)C2=O.C(=O)(C(C(C)C)SCC)O.CCO C=CCC(C(=O)N1CCN(C(C)CNC(c2ncccc2O)=O)CC1)OC c1(OC)cc(C(=O)NC(C(=O)NCC(c2ccccn2)C)C2CCC2)on1 N1(CC(N2CC(OCC(=O)NC(C3(n4cncn4)CC3)C)C2)=O)CCOCC1=O C(=O)(CCC(C)(F)F)NCC(Cc1csc(CSc2ccccc2)n1)OCC c1(C(=O)NCC(CC)NC(=O)COCC(F)(F)F)cc(=O)c(C)c[nH]1 N1(C(c2c(C)n(C)nc2)=O)CC2CN(C(c3cnn(C4CCOC4)n3)=O)CC2C1 c1(N2CCCCC(NC(=O)Cc3cccnc3)C2)ncnc2cc(C3CC3)nn12 Cc1ccncc1C=CC(=O)NCC1C2CCC(C2)N1C(c1csc(C)c1C)=O C(C(=O)NCc1cc(C(=O)N(C)CC2CCC(=O)N2)n(C)n1)(C(C)C)SC N1(C(C2CCN(C(c3nc(CCC)oc3)=O)C2C(C)C)=O)CCCNC(=O)C1 C#Cc1cn(C)nc1C(N1CCSCC1CCNC(=O)Cc1cncn1C)=O C(CC(F)F)(C(=O)NC1CCCC1OC)OC.c12nocc1C(=O)NC2 c1(C(=O)NCC(O)CNC(C2C(F)(F)C23CC3)=O)c(F)ccc(F)c1F C(C)(C(CO)NC(c1cc(-c2ccccc2)[nH]n1)=O)NC(C1(CSC)CC1)=O c1(C(=O)NC(C)CCNC(=O)CCC2CCN(C)C2)nc2ccccc2cc1Cl C1(O)(CNC(C(c2cccc(OC)c2)O)=O)CCCN(C(=O)CCSC)CC1 N1(C(C(C2CCC2)OC)=O)CCCN(C(c2c(F)cc(Cl)cc2F)=O)CC1CO c1(C(N2CCNCC2)=O)cc(N(C(=O)C2=NNC(=O)C2)C2CCC2)ccc1O CC(CC(F)F)C(=O)N(C)CC1(NC(=O)CSCC2CCCO2)CC1 N1(C(CC2CCC(=O)O2)=O)CCN(C(c2ccc(F)o2)=O)CC1CF N1(C(C)=O)CC2CC1CC2Nc1cc(C(F)(F)F)n(C)n1.C12(CC1)C(=O)N2 N1(C(C(C(=C)Cl)(C)C)=O)CC2(CCCC(CNC(=O)CC3CC34CC4)O2)C1 CCC(COC)(CC)C(=O)NCC(C)CN(C)C(c1cccc(C2CC2)c1)=O C=CC1(CC(=O)N(C)CC2(O)CN(C)C2)CN(C(C2(C(=O)NC)CC2)=O)C1 N1(CC)CC(NC(=O)CNC(c2c(C)nn(C)c2N)=O)CCC1=O c1(N2CCC(CC=C)(NC(=O)Cc3occc3C)C2)c([N+](=O)[O-])cnn1C c1(C(=O)NC2CN(C(CN(C)CC)=O)CC(O)C2)ccc2c(c1)COC(C)(C)O2 c1(C(N2C(CNC(c3cncc(C#C)c3)=O)CC(F)C2)=O)cc(F)c(F)cc1Cl C(C(N=c1[nH]cnc(C2CC2)c1Br)c1ccc(OC(C)(C)C)cc1)CO c1(C(=O)NCC(CN(C(c2cnsc2C)=O)CC)(C)C)cncc(C)c1 C#Cc1ccc(C(=O)NC(CC=C)CC(=O)N2CCCC2(C)CO)cc1 CCC(C)(COC)C(=O)NCCOC1CCN(C(C2CCCC(=O)N2)=O)CC1 C1(NC(c2nc(CC)oc2)=O)CCCCCC1C(=O)NC1CC1c1ccnn1C c1(C(N2C3C(C(N(CC(C)C)C)=O)C(C3)C2)=O)cc(O)ncc1F NC(=O)CC(O)C(=O)NCC(N1CCN(C(=O)CNC(C2CCC2)=O)CC1)=O C(C(C)(COC)C(=O)NCC(C(=O)N(C(CC1CC1)CO)C)C(C)C)OC C(=O)(C1=CCCCC1)N1CCC(C(N2C(C)(CCC)CC2)=O)(OC)C1 CN1CCN(C(=O)C(O)C(C)(C)C)CC1CNC(c1ccnn1C1CCC1)=O c1(CC)cc(C(=O)N(CCCNC(C2CCNC2=O)=O)CC)cc(C)c1 CN1CC(C(=O)OCc2nnsc2C(F)F)C(c2ccccc2)C1 N1(C(Cc2c(C)c(Br)ccc2)C)CCC2CC2(C(=O)N(CC)CC2CCC2)CC1 n1(CC=C)nc(-c2ccnc(-n3nc(C)cc3C)c2)nc1C[SH]=O.c1cncnc1 c1(C(N(C2CN(C(C3CCCC(O)C3)=O)C2)C)=O)cc(C(F)F)ncn1 C(c1cc(C)cc(C)c1)=CC(=O)NC1CN(C(CC(CC)(F)F)=O)C(C)CC1 N1(C(C(CC)n2ccnc2)=O)CC2CCC(CNC(=O)C(C(C)C)OC)C2C1 Cc1c(C(N2CC3(CC(NC(=O)CCC(=O)N(C)C)CO3)C2)=O)nc2sccn12 CC1CC(C(=O)NC2CC23CCN(C(=O)C2=CCCCCC2)C3)CC(C)(C)C1 C1(C(N2CCC(NC(C3CCSC3)=O)CC2)=O)CC2(C1)CC(C)(C)C2.C(CCO)SC N1(C(c2nc(OC)oc2)=O)CCN(C(c2cncc(C)n2)=O)CC1CF N(C1CCc2ccccc21)C(N1CCCCC(F)(F)C1)=O c1(C(=O)NC2C(NC(C=C(COC)C)=O)CS(=O)(=O)C2)cnc2c(cnn2C)c1 CCCC(C)(C)CC(=O)NC1CC(C)N(C(c2cncnc2)=O)C1 N1(C(C(=O)NC(CC)CNC(=O)C=CSC)C)CCCCCC1 C(=O)(CC(C)C(C)C)N1CC(CNC(C(C=C)(C)C)=O)C1 C1(C(=O)NC(C2CCC(NC(=O)Cc3cncnc3O)C2)C)CCC(C)(F)CC1 CC(C(C)(C)NC(c1csc(-c2ccsc2)n1)=O)NC(C1CCCN1C)=O C1(NC(=O)Cc2cc(Br)ccc2F)CC(C2CCNCC2)C1 c1(C(N(CC=CCNC(CCOC)=O)C2CC2)=O)ccc2c(c1)CC2 C1(NC(c2cc(CNC(c3c(CC)nco3)=O)oc2)=O)CC12CCCCCC2 C(=O)(C1=C(C)OCCS1)N(C1CC(C(N2CCC(CCC#C)C2)=O)C1)C N1(C(c2nc(CC)oc2)=O)CC2CS(=O)(=O)CC2(NC(c2cnncc2O)=O)C1 CON=CC(=O)NCC(C)(C)CNC(=O)C(F)c1ccsc1 c1(C(=O)Nc2ccc(C(=O)Nc3cccc(Cl)c3O)nc2)cc(Cl)c(Cl)cc1F C1(O)(CNC(C2(OC)CCSC2)=O)CCN(C(C2(Sc3ccccc3)CC2)=O)C1 c1(CNCCCCN(C)C)c[nH]c2c(F)cccc12 N1(C(CC2(C)CC2)=O)CCC(CCC(=O)NC2CCCN2C)C1 C(CN=C(NCC1(c2ccccc2)CCC1)N1CCC(CS(C)(=O)=O)C1)OCC Cc1noc(COCC(=O)N(CCCCCNC(c2cscc2Cl)=O)C)n1 N1(C(CCC(C)OC)=O)CCC2(CC1)CN(C(C1(F)CCCN(C)C1)=O)C2 Cc1ccnc2nc(C(=O)NC3CC(NC(C4CC4(F)F)=O)C3)nn12 C1(C)(C(=O)NC2CC(NC(c3nc(C(C)(C)C)[nH]n3)=O)C2)CCNC1=O C(=O)(C1=C(Cl)CCC1)NC(C1(C(N2CCC(C(N)=O)C2)=O)CC1)C O(NC(=O)C(O)C1CN(C(c2cccc[n+]2[O-])=O)C1)Cc1cn(C)nc1 c1(NC(C2CN(C(C(C)(C)O)=O)CC(F)C2)=O)cc(F)c([N+](=O)[O-])cc1Br CC(C)CC(C)CC(=O)NC(C)(C)CCNc1ccc(C#N)nc1 c1(OC)cccc(NC(=O)C(O)CCNC(c2cccc(C3CC3)c2)=O)c1 CN=c1[nH]cc(C(=O)NCCC2CCCN(C(C3CC3C(F)(F)F)=O)C2)s1 N1(C(C2CCCN2Cc2cc(Br)c[nH]2)=O)C2CCC1CC2 C1(NC(CC(CC)NC(C(CCC)NC(N)=O)=O)=O)COCC(C)(C)C1 C1(C(=O)NC(COCC)C(C)C)C=CCCN1C(=O)CCOC c1(C(N2CC(C)C(NC(c3cncn(C)c3=O)=O)C2)=O)ccc2ccncc2c1 N1(C(c2cc(CC(=O)OC)on2)=O)CCN(C)C(C(=O)NCC2C=CCCC2)C1 c1(OC)ccccc1C(N1CCN(CC(C)NC(c2n[nH]c(C)n2)=O)CC1)=O c1(-n2c(C)ncc2)ccc(C(C(=O)NC(C)C)N(CC(C)(C)C)C(C)C)cc1 C1(C(=O)NCC(C2CC2)NC(NOCC(=O)OC(C)(C)C)=O)COC2(CCC2)C1 Cc1cc(C#N)c[nH]c1=NC(=O)C1CCCN1C(=O)Nc1ccccn1 S(=O)(=O)(c1ccc(Cl)cc1)N1CCN(c2ccc(N(C)C)cc2)CC1 c1(C(N2CC3C(CNC(C=CC(CC)C)=O)(C3)C2)=O)nccn2cc(C)nc12 c1(C(=O)NCC(CC)(CC)NC(=O)CC#N)ccc(C)c(F)c1F C1(C(N2C(CN(C)C)CCC2)=O)CC(C)(C)CCN1C(c1c[nH]c(=O)cn1)=O O=C(N=c1ccn(-c2ccccn2)[nH]1)C(=O)N(C1COC1)C1CC1 c1(OC)cc(CN2CCC2C(N2CC3C(C2)C3(F)F)=O)cc(OC)c1O N1(C(CCC)=O)CC=CC1(C)C(=O)N(C)C(c1nccs1)C c1(C(N2CCCC(N(C(=O)C(C)C#N)CC)C2)=O)ccc2c(Cl)nccc2c1 c1(C(N(C2C3CN(C(C(CC)C)=O)CC32)C)=O)cc(C)c2ncccc2c1 c1(-c2c(OC(COC)C)ccc(C(C)=O)c2)ccc(N(C)C)c(C(=O)OC)c1 c1(COC)ccc(NC(C2CC2c2nc(Br)cs2)=O)cc1OCC(F)F CCC(C)CC(=O)C(=O)NC1(C)CCC(NC(c2cc(C)[nH]n2)=O)CC1 C#CCC(C)(C(=O)NC(C)CC1CC1)NC(c1cc(OC)no1)=O C12(NC(c3ccc4cncn4c3)=O)CCCC1(F)CN(C(=O)C(Cl)=CCl)C2 N12CC(OC(C)C1)CCNC(=O)C1(CC1)C2=O.c1(NC)cc(C2(C)CC2)on1 N1(C(C2CC(=C)C2)=O)CCCC(NC(c2ccccc2CN(S(C)(=O)=O)C)=O)C1 C(=O)(CCC(C)CN(C)C)NCCCCC1CN(C(c2cnn(CC)c2C)=O)C1 Cc1cc(C(=O)NC2CCN(C(=O)CC3CC4CC4C3)CC2O)cc(Cl)c1 CCC(CC(=O)NC1CC(N(C(=O)CCc2ncc[nH]2)C)C1)SC C12(CNC(CCOC(C)C)=O)CC(NC(C3CN4CCC3CC4)=O)(C1)C(C)(C)O2 C1(C(=O)NCCCCCNC(Cc2c(C)ccs2)=O)CC=CCC1C(F)(F)F c1(C(=O)NC2CCC(CNC(c3cc(CC)n(C)n3)=O)CC2)cnc(Cl)c(Cl)c1 C(=O)(N1OC2CCC1CC2)C1CCN(C(c2c(C)n(C)nn2)=O)CC1(C)C CS(=O)(=O)C1CCCC(NC(C23CC(F)C2C3)=O)C1 C1(C(=O)NCC2C(NC(COCCCCC)=O)C2)(CC=C(C)C)CCCCC1 c1(NC(C23CC(C(=O)NC(COC)C)(C2)C3)=O)cccc(-c2cn[nH]c2)c1 O=C(C1=CC(O)CCC1)NCC1CC1NC(c1c(O)cccc1F)=O C(C(C)(C)C(=O)NCc1cnn(CCO)c1)N(C(Cn1ccc(C)c1)=O)C c1(C(=O)NC2CCCN(C(=O)COC3CCC3)C2)cnc(O)c2cccnc12 N1(C(C=Cc2ccn(C)c2)=O)CC(NC(=O)C2=CC(C)(C)C2)CC(F)C1 CC(C)CC(O)C(=O)N1CCC(NC(c2cc(-c3ccc(C)o3)[nH]n2)=O)C(O)C1 n1(C(C(=O)NCCCCCN(C(=O)COC(C)(C)C)CCC)C)nccc1C c1(C(N2CCN(C(c3ccc(C)cc3N)=O)CC2)=O)cnn2cc[nH]c(=O)c12 N1(C(c2c(C)nccc2)=O)CCC(NC(C2(F)C(F)(F)C2(F)F)=O)C(C)(C)C1 c1(CCC(=O)NC(C=CC(=O)N(CCCC)C2CC2)C)nnc(C)n1C C(=O)(C1=NN(C)C(=O)CC1)NCC1(NC(C(C(C)O)C)=O)CC2CCC1CC2 CC(CC(=O)N1CC2(NC(=O)C(c3ccc(Br)s3)=O)CC1C2)C(F)(F)F N1(C(C(C)SC(C)C)=O)CC(C)(C(=O)NCc2cc(F)cc(F)c2)CC1(C)C Cc1cc(F)c(C(N2CCOC(C(C)NC(=O)C=CI)C2)=O)cc1F Cc1cc(C)cc(C=CC(=O)NC23CC(C)(C2)OC32CCC2)c1 C(CC1CC1)(CN=c1[nH]c(N2CCC(n3cncn3)CC2)nc2c1COC2)OC c1(C(=O)NCCC(C)NC(COCc2nnc(C)s2)=O)cnc2c(c1)CNC2=O c1(COCC(N2CCN(CC(=Cc3ccccc3)F)CC2)=O)ccccc1Cl c1(C(=O)NC2C(CO)CCN(C(C3(C)CCN(C)C3)=O)C2)cnc2n1CCOC2 CCCC(C)(CC)C(=O)N1CC2CCCC2(CNC(=O)CCc2cn(C)nn2)C1 c1(C(=O)Nc2scc(CC(=O)Nc3nc(C)sc3)n2)cccc2ccoc12 Cc1cc(CNc2ccccc2-n2cncn2)ncc1Cl CC1CCCCN1CC(N1CC(F)(C(=O)NCCC2CC(O)C2)C1)=O c1(C(N(C2CCC(CNC(=O)CN(C(C)(C)C)C)C2)C)=O)cccnc1SCCC CC1CN(C(=O)CCC(=O)N(C)C)CCN1C(=O)Cc1c(F)cncc1Cl Cc1ccc(Br)c(C(N2CCCCC(NC(c3ccon3)=O)C2)=O)c1N O=C1Cc2cc(C(=O)Nc3cccc(C4CCOC4)n3)ccc2N1 c1(C(=O)NC23CCCN(C(CC(C=C)(C)C)=O)CC2C3)cnc2ccccc2n1 C1(C(=O)NCC2N(C(COC)=O)CCOC2)CCc2ccccc2C1 c1(-c2cn(C3C(NC(CN(C)CC)=O)CCC3)nn2)cc[nH]c(=N)c1 C1(C(=O)NC2CC(C(N(C)C)=O)C2)CCCCC1C(N)=O C(C(F)(F)F)OC(C(=O)NCC(=O)N(CCN(C)CCN1CCC1)C)C1CC1 CN1C(C(N2CC(F)(c3cn(C)cn3)C2)=O)CCS1(=O)=O C(=O)(C(CC(F)F)C1CCC1)N(CCN(C(=O)C1CC1)C1CC1)C1CC1 C1(c2cn(CCCCC=C)nn2)CC2(CC(NC(=O)C(F)CC)C2)C1 c1(C(N2CC(CCCCNC(C(C(C)C)C)=O)C2)=O)cc2c(F)c(Br)ccc2[nH]1 C(=O)(C(C)C(C)(F)F)N1CC=CC(NC(CCc2ccc(OC)cc2)=O)C1 c1(CC(N2CCC3(NC(C45CC(F)(C4)C5)=O)CC3C2)=O)ccc([N+](=O)[O-])cc1 c1(C(=O)NC2C3CC2N(C(c2coc(Cl)c2)=O)C3)ccc([N+](=O)[O-])cc1F C1(NC(c2cc(OC)ncc2)=O)CC2(CCN(C(=O)C(O)C(F)F)CC2)C1 N1(C(c2c(C)ncs2)=O)CCC(F)(C(=O)Nc2ccnc(C#N)c2)CC1 CCC(C(=O)OC(F)F)NCc1ccc(OCC(F)(F)F)o1.C(C)(C)O c1(C(N(C2CN(C(c3nnc(O)cc3O)=O)C2)C)=O)ccnc(F)c1N N1(C(Cn2ncn(C)c2=O)=O)CC2CCCC2(CNC(=O)CC2CCNC2=O)C1 CC1(C)CCOC1CC(=O)NC(C)(CO)C(=O)N1CC(N(C)C2CC2)C1 C1(C(=O)NC(C=C)C)CCN(C(=O)C=Cc2ccccc2C)CC1CO c1(CC)noc(C)c1C(=O)NCC1CCCCC1NC(C1CC=C(C)CC1)=O C(=O)(CCCCC(=O)N1CCCC(NC(C2CCCCC2O)=O)C1)OCC C(c1nc2ccccc2o1)=CC(=O)NC1CCN(C(c2nnc(C)s2)=O)C1 C1(NC(N2CCN(c3cccc(OCC)c3)CC2)=O)CNC2(CCC2)C1 N1(C(c2c(C)c[nH]n2)=O)CCCC2C(CCCN2C(=O)Cc2ccno2)C1 CCC(C)CCN(C(=O)CCOC(C)=O)C1CC1.C12(C)CCN1C(=O)C2 CN1CCCC(CNC(C2(CNC(C3CCCN3C=O)=O)CCCO2)=O)C1 c1(OC)cc(OC)nc(C(=O)NCC2(O)CC(NC(=O)CC3C4COCC34)C2)n1 N1(C(C(CCC)NC(c2ccc(OC)cc2)=O)=O)CCOC(C)(C)C1 c1(C(N(C(C)CNC(C2Cc3nccn3C2)=O)C)=O)cc(Cl)c(F)cc1N C1(C(=O)NC(C)C(CO)NC(c2cc(O)cc(=O)o2)=O)CCc2nncn2C1 C1(C(C)C)CCN(C(=O)C(CNC(C2CCC(=O)N2)=O)CC2CCCC2)C1(C)C c1(C(=O)NCC2C(n3cc(C(COC)(C)O)nn3)CCC2)nccc(C)c1Br S(=O)(=O)(c1cnc(NCc2cc(O)ncn2)c(Cl)c1)NCCC(COC)(C)C c1(CC)cccc(NC(=O)C(C)(CNC(=O)CN(C)C(C)=O)CC)c1O n1(CC)cc(C(=O)NCCN(CC(C)O)C(C2CCSC2)=O)c(C2CC2)n1 C1(C(N(CCC(=O)NC(C(C)C)C2CC2)CC)=O)CCC=CCCC1 N1(CC)CC2CC(N=c3ccc(C(c4c(CC)cno4)=O)c(OC)[nH]3)CC1C2 Cc1c(C(=O)NC2CN(C(c3cnn[nH]3)=O)C(C)(C)C2)cccc1C#N O=C(CCCn1cccn1)NCC=CC(N1CC(OC(F)F)C1)=O N1(C(c2nccc(CC)c2)=O)CCOCC(NC(c2c[nH]nc2C(F)(F)F)=O)C1 C1(C(=O)NC(C(=O)NC2(C#C)CC2)CCOC)CCCC(C)(C)C1 c1(C(=O)NC2CN(C(CCSCCCC)=O)C2)n[nH]c(C)c1[N+](=O)[O-] c1(C(=O)NCC(CC=C)NC(=O)CCc2cnc[nH]2)ccc(CC)cc1F c1(NC(C2N(C(CCC)=O)CC2)=O)c(F)cc(Cl)cc1I.C1C(=O)N1 CCC(CCCC(=O)NC1(C)CC2CCC1C2)NC(=O)C1=C(Cl)CCCC1 C(=O)(C(C)C(C)CC)N1CCN(c2nccc(CNC(C(F)=CCC)=O)c2)CC1 c1(C(=O)NC2C(NC(C(C(F)(F)F)OC(C)=O)=O)CC2)cc(F)c(F)c(Cl)c1F C(=O)(C(CO)C(C)(C)C)N1C(C(=O)NCCc2ccc(C)cn2)CC1C C(C(COC)CC(=O)Nc1ccc(Cl)nn1)OC CC(C)CC(CNC(=O)Cc1ccsn1)NC(c1ccc(C(N)=O)cn1)=O c1(NS(=O)(=O)CCC2COCCO2)ccc(CC(O)CF)cc1 c1(C(=O)OC)ccc(CC(=O)NC(C)CN(C)C(C2CCC(C)O2)=O)cc1F C1(OC)C(OC)CN(C(=O)C(c2c(C)noc2C)C)C1CNC(c1ccc[nH]1)=O C(=O)(C(C)S(N)(=O)=O)NC(CN1CCN(C(CC2(OC)CC2)=O)CC1)(C)C c1(CCC(=O)N(CCC)CCNC(C2(F)CCOC2C)=O)cccc2c1OCO2 C1(N(C(=O)CC2CC=CC2)C)CCCN(C(c2cccnc2C(F)F)=O)CC1 N1(C(CCCC=C)=O)CCN(C(c2cn(C(F)F)cn2)=O)C(c2ccncc2)C1 CC1CC2(CC(C(N3CC(CCNC(C4(c5ncccn5)CC4)=O)C3)=O)C2)C1 C(CC(N)C(=O)N(CCC(=O)O)Cc1ccccc1)N(C)C Cc1nn(CC(N2CCN(C3CN(C(C4COCC(C)O4)=O)C3)CC2)=O)c(=O)o1 C1(CNC(CCNC(N)=O)=O)C2CN(C(c3n[nH]c(-c4cccnc4)n3)=O)CC12 C12CC(O)CN1C(=O)C1CC1c1cn(nn1)C2.c1(C=O)cccc[n+]1[O-].CO CN1Cc2cc(S(=O)(=O)NC(N3CCOCC(O)C3)=O)ccc2OC1=O c1(OC)ccc(C(=O)C(=O)NCC2CCCCN2C(=O)CSC2CC2)cc1 C1(CNC(c2ccc(OC)s2)=O)COCCN(C(C23CC=CC(C2)OC3)=O)C1 Cc1ccc(C(N2CCOC(C(C)NC(=O)C=C3CCN(C)C3)C2)=O)c(Cl)c1 C(=O)(CCCCCC#N)NC(C1CCN(C(=O)Cc2ccc(Cl)nc2)CC1)C C1(CN(C(=O)C(Cn2cncn2)NC(c2cnn(CO)c2)=O)C)C(C)(C)C1(C)C Cc1cc(N)c(C(=O)NCC2CN(C(=O)C3=NOC(C)C3)CC23CCC3)cc1C C1(C(N(CCC(C)NC(c2c(C)cc(C)o2)=O)C)=O)CC12CC(F)(F)C2 c1(C(=O)NC2(C)C(NC(Cc3ccc(C)o3)=O)CCC2)cc2ccc(F)cc2o1 Cc1cccc2c1NCCC2C(=O)NCC1CN(C(=O)CC2CCC(C)C2)C1 Cc1ccccc1CC(=O)NC1CCCC(NC(C2(C)CC2(Cl)Cl)=O)C1 C(=O)(CCC(=O)N(C)C(C)C)NCC(CC)(C)NC(c1ccncc1Cl)=O c1(Nc2c(C(=O)Nc3c(Cl)ncc(OC)c3)nccc2)ncnc2n[nH]cc12 C(=O)(CC(O)C(C)C)N1CCC(CC=C)(NC(=O)C=CC2CCCC2)C1 C1(C(=O)NC23CC(C2)N(CC#C)C3)CC2CCC(C1)C2(F)F.C1C(=O)NCCS1 Nc1ccc(C(=O)NCC(CO)NC(c2ccc(CO)nc2)=O)nc1Cl c1(C(N(C)CC2(NC(C(C)C3CCOC3)=O)CC2)=O)ccc(CN(C)C)nc1 Cc1cc(NC(C2CCCCC2O)=O)ccc1NC(=O)CN1CCC(C)(O)C1 C1(C(=O)NC(CNC(COCCC(C)C)=O)(C)C)CC(=O)C1C N1(C(C(C(C)C)C#N)=O)CC2CN(C(c3ccc(OCCF)cn3)=O)CC2(C)C1 C12(CC)CC(C(=O)NC(C)(CNC(=O)C(C(C)C)n3cnnn3)CO)(CO1)C2 C1(C(N(CC(C)N(C(COCC=C)=O)C)C)=O)CCn2nccc2C1 c1(C(=O)NC(C2CCCN2C(=O)C(O)CC2CC2)C)cnnn1C N1(C(COC(C)C)=O)CC2CCN(C(c3cccc(OCCF)c3)=O)C2C1 C(=O)(C1CCCc2ncnn21)NC1CCC(CNC(CC(=O)OC)=O)C1 N1(C(CC(C(C)C)OCC)=O)CC2CCCC2(NC(=O)CCCSC)C1 C1(C(=O)NCc2ccc(Br)cc2)CC(F)CN(C(=O)COc2cccnc2)C1 c1(OC)cccc(C(=O)NC2COCC2NC(c2n[nH]c3c2CCC3)=O)c1C CCC(C)(C)C(c1nnnn1C1CCCC1)NCc1cc(-c2ccccc2)cs1 CCC(C)(CNC(=O)C#CC1CC1)C(=O)Nc1ccc(O)cc1C N1(C(CSCCC)=O)CCC(O)C1(C)C N1(C(c2cc(C3CC3)cnc2Cl)=O)CCC2(CCOC2=O)C1 C=C1CCC1C(=O)NCC1CCC1NC(C1(NC(=O)NC)CC1)=O c1(C(=O)NC(CCN(C(C2(C#C)CC2)=O)C)C(C)C)ccc2ccccc2n1 C(C(C)(C)CC(=O)N1CCCC1CNC(C1CC1CN(C)C)=O)OC(C)=O c1(C(=O)NC(C)CCNC(=O)C(C)OC2CCOC2)ccn2cncc2c1 Cc1cc(C(=O)N(C(C)CNC(c2cnn(CCO)c2C)=O)C)c2nccn2c1 c1(C(N2CC(CNC(c3n(CCCC)ncc3)=O)C(O)C2)=O)cccc(O)c1F c1(CCC(c2nnnn2CC2CCOC2)OC)cccc(OC)c1.c1(CC)noc(CC)n1 C1(NC(C(=O)NC(C)C)=O)CC(O)C1(C)C.c12ccoc1C(=O)N(C)C2 c1(C(=O)NCCC(Cn2cc(SC)nn2)(F)F)ccc2c(c1)NC(=O)CNC2=O c1(CNC(=O)NCc2cnc(C3CCOCC3)[nH]2)ccc(Cl)c(F)n1 N1(C(c2c(CC)ccs2)C(=O)NCCNC(C)=O)CCS(=O)CC(C)C1 c1(C(N2CCCC(NC(C3CC4CC3CC4O)=O)CC2)=O)ccc(F)c(F)c1F n1(CCCN2CC(C(=O)OC)(Cc3ccccc3)C2)ncc(Cl)c1C N1(C(C(CCCCC)O)=O)CC(C2CCCN(C(=O)CC3CC4(CCC4)C3)C2)C1 C(=O)(C(C(C(C)C)OC)N1CCCOC(C(=O)NCC)C1)NCCC(=O)NCC C1(C(N(CC)Cc2ccoc2)=O)CC2(CCN(C(C3CCC(=O)NC3)=O)C2)C1 C1(NC(c2sccc2F)=O)(CF)CCN(Cc2ccn(CCF)n2)C1 N1(C(C(C(C)C)SC)=O)CC(NC(c2cn(C)nc2C(F)F)=O)CC2(CCC2)C1 C1(N(CCC)C(C2CCCC2O)=O)CCN(C(=O)CCc2c(C)n[nH]c2C)CC1 C(=O)(C(C)OC)N(CCCNCCCC)C c1(OCCCC(=O)NCCCNC(C2C(C)C2)=O)ccccc1F c1(C(C)(C)C)ncc(C(=O)NCC2CC2CNC(=O)CCc2ncc[nH]2)o1 C1(CN(C(C2(CCOC)CCC2)=O)C)CCN(C(=O)C(c2ccnn2C)C)CC1 CC1(NC(C2CC2(C)Br)=O)CCN(C(c2scnc2C2CC2)=O)C1 C(c1ccc2[nH]ccc2c1)=CC(=O)NCC1(O)CN(C(CC(CCC)O)=O)C1 c1(C(N(CCC(C)NC(C23CC(F)(C2)C3)=O)C)=O)cc(C(F)(F)F)ns1 c1(C(N2CC3(CC2CO)CCS3(=O)=O)=O)nc2cncnc2nc1O c1(C(N(CC(C)NC(C2CC3CCCC(C2)C3)=O)C)=O)nn(C)c2ccccc12 N1(C(c2nc(C)sc2C)C(=O)NC2CCCC2)CCCC2CCCC12 C1(NC(C(C)NS(CC)(=O)=O)=O)CC(O)CN(C(C23CCCCC2C3)=O)C1 C(C(C(C)(C)C)NC(=O)C(O)CCC)NC(C(C)(C)NC(CC(=C)I)=O)=O CCCCCCC(=O)NC(C)C(C)(C)C(=O)NCCC1CCOC1(C)C c1(C(=O)NC23CCCN(C(CCCC=C)=O)CC2C3)cc2c(O)cccc2n1C C1(C(C)C)CN(C(=O)C(C)(C)n2cc(-c3ccns3)nn2)CCS1 C1(NC(c2c(CCC)n[nH]c2)=O)CN(C(=O)Cc2csnn2)C(C)(C)C1 C1(CNC(CNC(=O)OC)=O)CC(F)(CNC(=O)C(Br)=C(C)C)C1 N1(C(C2(C(=O)OCC)CC2)=O)C2CCC1C(NC(=O)C(=O)N(C)C)C2 C1(C)(C(=O)NCc2c(C(N(C)CCO)=O)n[nH]c2)CC=CCC1 C(=O)(C(Cc1ccccc1)NC(=O)COCCc1cn(C(C)C(=O)O)nn1)OC C(CCCCC(=O)NCC1COCC1NC(c1cc2n(n1)CCC2)=O)OC N1(C(CC2CNC(=O)O2)=O)CCC2C(NC(c3ccc(Cl)cc3)=O)C12 C1(NC(CC(=C)Br)=O)CN(C(=O)CSCC(F)F)CC1C C(C)(CC(=O)NCC(C)(F)CNC(=O)CCCn1cc(C)cn1)OC Cc1nccc(C(=O)NC2(C(N3CC(OCF)C3)=O)CCCC2)n1 Cc1cccc(COCCOCCC(=O)N(C2CN(C(=O)CNC(N)=O)C2)C)c1 C(=O)(C1CCCc2nn(C)cc21)N1CC(NC(CC(CC)C(F)F)=O)C1 C=CC(C)(CC)C(=O)NCC(C1CCN(CC(O)Cn2cccn2)CC1)OC C(CO)(CCCCNC(c1cccc(C)c1)=O)NC(CC(C)SC)=O n1(CC(N2CCCC(NC(c3cn(CCSC)nn3)=O)C2)=O)ccc(O)nc1=O c1(C(N(C(C)CN(C(=O)CC(F)(F)Cl)C)C)=O)nnc(O)nc1O c1(CNC(C2CCN(C(c3cncs3)=O)CC2F)=O)ccc(Cl)cc1C(F)(F)F N1(C(C(=O)OC)C)CCN(C(c2cccc(F)c2)=O)CC1 CC1COCCC1N(C(=O)C(C1CC1)NC(=O)CCn1cncn1)C c1(CNC(=O)C(=O)Nc2ccccc2OC2CCCCC2)nc2ccccc2s1 C1(NC(=O)OC(C)(C)C)CC2(CCC(C(=O)NS(=O)(=O)CCCC3CCC3)CC2)C1 O(S(=O)(=O)c1ccsc1C#N)Cc1c(C)ccc([N+](=O)[O-])c1 C12(CNC(=O)C(F)OC(F)(F)F)CC(CCO1)N(C(=O)C1=COCCC1)C2 N1(C(C2(CC=C)CC2)=O)CC=C(CCNC(c2cn(CC(F)F)cn2)=O)CC1 C1(NC(C(CC)Cc2cccc(C)c2)=O)CN(C(=O)CN2CC=CC2)CCC1O c1(C(=O)NCCC(C)(C)NC(c2cnc(C(C)O)s2)=O)coc2c1CCCC2 C(=O)(CCC(F)(F)C(F)(F)F)N1C(CNC(C2CC2c2cccnc2)=O)CC1 N1(C(c2ccc(COC)o2)=O)CC2(CC1CNC(C1(C(=O)NC)CC1)=O)CC2(F)F N1(C(C2(C)CC2(F)F)=O)CCC(C)(CNC(C2(F)CCCC2)=O)C1 NC1CC2CCC1CN(Cc1cc(F)c(F)cc1Br)C2 N1(C(CN(C)CC)=O)CCC2CN(C(c3cnn(C4CCC4)n3)=O)C2C1 CCC(C(=O)NCC1(F)CC(NC(c2ccc(O)c(F)c2)=O)C1)C(C)O N1(C(C(CC(=O)OC)C)=O)CCC2CCCC12C(=O)NCC(C)(O)C(F)(F)F C=CC(C)(CC)C(=O)N(CCC(c1cccs1)NC(=O)CS(=O)(=O)CC)C C(=O)(CC(C(F)(F)F)NC(C1CCCC(=O)C1)=O)NC1CCN(OC)CC1 c1(NC(CC2(C)CCN2C(C2Cc3ccccc3C2)=O)=O)ccc2ncnn2c1 C1(CCNC(CCCOCCC)=O)CSCCN1C(=O)C=CC1CCCO1 C1(C(N(CC#C)Cc2ccccc2)=O)CN(C(=O)CCC2CC(C)C2)CC1(F)F c1(SC)ccc(C(N2CC(NC(=O)C(O)CCn3cncn3)C(SC)C2)=O)cc1 C1(CC(=O)NC(N(C)CCC2CC2)=O)CCCCCN1C(C1CCO1)=O c1(C(=O)NCCC2N(C(CC3C(CC)C3)=O)CCC2)c(Cl)ccc2ccncc12 c1(C(N2C(CNC(=O)C(=O)NCC(F)(F)F)CCCC2)=O)ccc(F)c(F)c1F C=CC(CC(=O)NCC1CC(O)CN1C(=O)COC(F)(F)F)c1ccco1 N#CC1(C(=O)NC2CCC(NC(=O)CC3CCCCO3)CC2)CCCCC1 C(=O)(C(C)C(C)(C)C)N1CC(CCC=C)(C(=O)NCc2cn(C)nn2)C1 CCCCCC(C)CC(=O)NCC(C)(C)CC(=O)N1CCCC(C)CC1 c1(C(C(=O)NCCCC2CC2)N(C2CCCCC2)CC)ccn(CC)c1.C1(C)CC1 Cc1cc(C(=O)NC2CCCN(C(=O)CCc3ccccc3C)C2C)nc(C)n1 c1(C(=O)NC2CC(C(=O)OC)CN(CC)C2)[nH]c2cccc(Br)c2c1COC C1(C(=O)NC2CCCC2SC)(CC)CCN(C(=O)CC2CCN(C)C2=O)CC1 N1(C(CSC)=O)CC(F)CC1C(=O)NCC1COCC1O C1(C(=O)NC(C2CCOC2)C#C)CN(C(=O)C(C)NC(=O)COC)C(C)(C)C1 c1(OC)cc(C(N2CCC(NC(=O)C(F)n3cccn3)C2)=O)c(C)cc1Br c1(-c2c(CN3CCCC(c4nc(C)on4)C3)c[nH]n2)ccc2c(c1)CCCN2 N1(C(c2cccc(C(C)C)c2F)=O)CCN(C(=O)C(C)CN(C)C)CC(O)C1 N1(CC(C2CC2)OC)CCC(=O)N(CCc2cc3ccccc3o2)C1=O C1(C(N(C2CCN(C(=O)CCc3cnoc3)CC2)C)=O)CCCC(F)C1 C(=O)(CCCCCS(N)(=O)=O)NC1C(NC(c2c(OC)cccc2Cl)=O)COC1 Cc1cc(S(N)(=O)=O)sc1C(=O)NCCN(C)C(C1CC(OC(F)F)C1)=O C=CC1(C(=O)NCC2CN(C)CCN2C(c2ccc(O)cc2F)=O)CCCCC1 C1(CNC(C(C)CC2CCC2)=O)CC2(CC2)CN1C(c1ccnc(Cl)c1N)=O c1(COC)cccc2c1CN(C(=O)NCC1(F)CCN(C(=O)OC(C)(C)C)C1)CC2 C(=O)(C#CC1CCCO1)NCCCCNC(CC(CC(=O)OC)C)=O N1(C(CCCOC)=O)CC2CC1C2CNC(=O)Cc1ccc(O)nc1 C1(CNC(C(CC)(C)C)=O)C(C)CCCN1C(c1cc2ccsc2s1)=O C1(NC(c2ncn(CC)n2)=O)C2CC1N(C(c1ccc(N(C)C)cn1)=O)C2C Cn1ccc(C(=O)NC2C=CCN(C(c3cc(=O)c(Br)c[nH]3)=O)C2)cc1=O CC(CCCCNC(C1CCCCC1O)=O)NC(=O)Cc1cocn1 C1(C(C)(C)C)C(=O)N1.C1(C(=O)NCCN(CCC)CCC)CCCC(CF)C1 Cc1ccc(C(=O)NCC23CCC(CC2NC(c2coc(Cl)n2)=O)C3)cc1F N1(C(c2cc(SC)oc2)=O)CCC(O)(CNC(C2CC(C(C)C)=NO2)=O)CC1 N1(C(Cc2c(C)cnn2C)=O)CC2(C1)CN(C(c1cc[nH]c(=N)c1)=O)C2 c1(C(=O)NCC(C)N(C(c2cn(CC(N)=O)nn2)=O)CC)cc(Br)n(C)n1 c1(C(=O)NC2C(C)(CNC(c3c(C)cns3)=O)CCC2)cccn2cnnc12 C1(NC(C=C(COC)C)=O)CC(O)(C2CCN(C(=O)C3=NOC(C)C3)CC2)C1 CC12COCC1(C)CN(C(C13CC(CN1C(C1C4CCCC14)=O)C3)=O)C2 C1=CCCN(N2CCC(OC(F)(F)F)CC2)C1 N1(C(CCN(C)C(C2C3CCC(F)(F)C23)=O)=O)CC2CC=CCC2C1 C(C(CC(C)C)NC(c1ccc(CNC(=O)CNS(C)(=O)=O)s1)=O)OC N1(C(C(c2cccc(OC)c2)O)=O)CC(NC(c2ccc(F)o2)=O)CC2(CC2)C1 C=CCCCC(C(=O)N1CCCC(C)(OC)CC1)NC(=O)C(O)CCC(C)C N1(C(c2c(C)nc(CO)o2)=O)CCCC2C1CCN2C(=O)C1=CCCOCC1 CC(C)(C)C(C#N)C(=O)NC(C)(C)C=CC(N1CCOCCC1C1CC1)=O N1(C(c2c(C)ncn2O)=O)CCC(C2CC(NC(c3cnc4sccn34)=O)C2)C1 C1(CC(=O)NC(CNC(C2(OC)CCOC2)=O)C(C)C)CC2CCC(C1)N2C N(C(=NCCC(C)=O)NCC1CCC(c2ccc(Cl)cc2)O1)CCC(C)OC c1(CC(=O)N(C2(O)CN(C(=O)CC3C(OC)CC3O)C2)CC)cc(Cl)n(C)n1 N1(C(c2ccc(CC)[nH]2)=O)CCC(CO)(NC(=O)C=Cc2cn(C)cn2)C1 C1(C(=O)NC(C)CNC(c2cscc2Br)=O)CCOC2(CCC2)C1 CCN=c1cc(C(=O)Nc2cccc(Cn3ccnc3)c2)[nH]c(=N)[nH]1 C1(C)(NC(C2N(CCC)CCC2)=O)CCC(NC(=O)C(C#N)CCC)CC1 c1(N(CCc2ccccc2)CC2ON=C(C)C2)cccc(C)c1.O(N)C c1(CC)cc(CC)[nH]c(=NC(CCNC(=O)COc2cccc(Cl)c2)C(C)C)n1 CN1CCC(O)(CC(N2CC(CO)(NC(C3CC4CCC(C3)O4)=O)C2)=O)CC1 C1(CC(=O)NC2CN(C(C(C)=CC)=O)CC2c2cncn2C)CCCCC1(F)F c1(C(C)C)cccc(C(=O)NC(C2CN(C(c3cnn(C(C)C)c3N)=O)C2)C)n1 c1(C(=O)OC)ccccc1C(N1CCC(F)CC1)=O.C12C=CC(C1)C(=O)N2 c1(OC)cc(Br)c(NC(C2CSCCN2C(=O)CCCCBr)=O)c(Br)c1 C(=O)(C(C(O)C(F)(F)F)C(C)(C)C)NCCCN(C(=O)Cc1ccc(O)cc1)C C(=O)(CCCCC(C)(C)C)N1C(C(=O)NCC(=C)C)CC2(CC1)CC2 C(=O)(C(F)(F)CO)N(C(C)CCNC(=O)CCN(C1CCOCC1)C)C C(=O)(CCN=C(NCCc1ncc(C(=O)O)s1)N1CCC(OC(C)C)CC1)NC C(C(C(=O)N1CCCC1C(C)NC(c1cc(-c2ccoc2)[nH]n1)=O)N(C)C)OC c1(SCCC(=O)NCC(CCCC)NC(=O)C(C)C(C)C)ccc(Cl)c(Cl)c1 c1(CC(=O)NCC(C)CNC(c2cn(C)[nH]c2=N)=O)cc(F)c(F)cc1F CN1CCc2cc(C(=O)NC3CCC3NC(=O)C(O)C3CCCC3)ccc21 N1(C(C(c2ccccc2)C)=O)CCN(C(c2ccn(CO)n2)=O)CC1C(C)(C)C C#Cc1cccc(CNC(=O)CC2CNC(=O)O2)c1 C(=O)(CC(C)C(C)(C)C)NC(C(C)C)C(C)NC(=O)CCc1ccccn1 C1(NC(c2cc(CC)on2)=O)CCC(O)CN(C(C2CCC(C)(C)C2)=O)C1 c1(C(=O)NC2(CNC(c3cnn(C)c3)=O)C(C)CCCC2)nc[nH]c2nccc1-2 N1(C(C2CC(=C)C2)=O)CC(CNC(C2(c3cc[nH]n3)CC2)=O)C(C)C1 c1(C(N2CCN(C(C3(F)CC3)=O)CC23CCC3)=O)ccc2c(c1)OC(F)(F)O2 C1(NC(C=CC)=O)CCC2(CCN(C(c3nnn(CC4CCCO4)c3C)=O)C2)C1 C1(NC(C2CC2C(F)(F)F)=O)CCN(CC(F)(F)F)C1=O C=C(C(=O)NCC1CCCN(Cc2cnc[nH]2)C1)C(F)(F)F C1(NC(C(C)CNC(C2CC=CC2)=O)=O)CC2CCCC2C1 C1(C(C)(C)C)CCN(C2=CCc3ccccc32)C1 N1(C(CSC(C)C)=O)CCC2CN(C(c3c[nH]nc3Cl)=O)C(C)C12 CC1CCN(C(C23CCCC2C3(F)F)=O)C(c2nnc(S)n2C)C1 C(=O)(CC(C)(C)CC(F)(F)F)NC1(CN(C)C(C2C(C3CC3)C2(F)F)=O)CC1 c1(C(=O)NC)ccc(C)c(NC(=O)NC(c2ccccc2)CC2CCCCC2)c1 N1(C(c2c(C)[nH]cc2)=O)CC2CC(C(=O)NC(C)Cc3nccn3C)(C2)C1 N1(CCc2ccc(C)cc2)CCN(c2nnc(-c3cn[nH]c3)n2C)CC1=O CC(CC(F)(F)F)C(=O)NC(C1CC1C(=O)NC1(CO)CC2(CCC2)C1)C CS(=O)C=CC(=O)N1CCC(C)(CNC(c2nc(Br)c[nH]2)=O)C1 N1(C(Cc2c(C)nc(O)[nH]2)=O)CCC(NC(C2CCCC(C)(C)C2)=O)C(O)C1 C(CCN(C(=O)CC(C)c1ccccc1)C)(C(C)C)NC(c1cc(CC)no1)=O C(=O)(CCC(C)(F)F)NCC1CCCC(NC(c2c(OC)oc(C)n2)=O)C1 Cc1ccc(-c2ccc(C(=O)Nc3nnccc3C)nc2)c(C#N)c1 CC(N=c1[nH]c(Cl)nc2c1S(=O)(=O)CC2)C1CCCN(C(C2CCCCS2)=O)C1 c1(-n2cc(N(CC(=O)OC)Cc3ccc(C)cc3)nn2)cc(C(F)(F)F)ncc1F c1(N2CCC(CC=C)(NC(=O)CCN(C)CC)C2)nc(C)nc(C)c1C Cc1cc2[nH]c(C(N3CC4CN(C(=O)CCC5CCC5)C4C3)=O)cc2s1 C1(C(N)=O)CCN(C(C2C=CCN(C(c3ccc(O)nn3)=O)C2)=O)CC1 C(=O)(CC(F)(F)c1ccccc1)N(C(CNC(C(CC)OC)=O)C1CC1)C Cc1ccncc1C(N1CCOC(CCCNC(=O)CCc2ccon2)C1)=O c1(OCC)cc(CNC(=O)Nc2cc(Cl)c(Br)[nH]2)nn1-c1ccccc1 c1(OCC)cccc2c1CCCC2N=c1ccnc(N(CCC(C)C)C)[nH]1 C#CCC(C(=O)N1CCCC(CNC(=O)CC2CC2CC)C1)C1CC1 c1(C(=O)OC)ccc(C(=O)NC2CCN(C(C3CCCO3)=O)C2C(C)C)cc1Cl N1(C(C(Cc2cc[nH]n2)NC(C2CC3CCC3C2)=O)=O)CCC12CCCOCC2 C(CN=c1nc2c(cnn2C)c(NCCSCC)[nH]1)OCCC.C(COC)O N1(C(C(CC=C)C)=O)CCC(NC(=O)CC(C)(C)C)CC(O)C1 c1(NC(C)=O)ccc(OC)c(OC(c2cccc(NC(CC)=O)c2)C)c1 C1(C(N2C(C3CCN(C(c4c(C(C)C)onc4)=O)C3)CCC2)=O)CC(F)C(=O)N1 C=CC(CC)CC(=O)N1CCN(C(=O)CC2COCCOC2)C(CC)C1 c1(CC)ccccc1C(=O)NCC1CCCC1NC(=O)Cc1cnns1 N#CC1CCN(C(C2(CO)CCN(C(c3cc(C(N)=O)[nH]n3)=O)C2)=O)CC1 CN1CC2(COCCN2C(c2ccccc2CC#N)=O)C1=O c1(CNC(N2CCC3CCOCC3C2)=O)ccc2ccncc2c1 CCC(CCC(=O)NCC1(C(C)C)CCCC1)NC(c1n[nH]cc1Cl)=O C(CC(C)C)(C(=O)NC(C)C(CO)NC(=O)COC(C)(C)C(F)(F)F)NC(=O)OC C1(C(=O)NC2CN(C(C(c3ccncc3)C)=O)C(C)C2)CCCC2CCCCC12 C(C(CCO)CC(C)C)NC(c1c(C)scn1)c1nnnn1C1CC1 C1(CNC(C(C(C)C)F)=O)CN(C(=O)Cc2cc(C3CC3)on2)CCC1(C)C c1(C(=O)NCC2(C)N(C(C=C3CCC(C)C3)=O)CCC2)coc2c(Cl)cccc12 C1(CC(=O)NC(CC#CC)C)COCCN1C(c1ccc(C#N)o1)=O C(CCN=c1cccc(S(=O)(=O)N2CCSCC2C(C)(C)C)[nH]1)SCC C1(C(F)(F)F)(CC)CN(C(=O)NCC(C)Cc2ccncc2)CCO1 N12CCCC(C1)C2C(=O)NC(C)CC.N1(CC#C)CCC(OCC(F)(F)F)C1 C1(NCCCCO)CC2(C1)CC(CNC(C13C(NC4CCCO4)C4CC1C3C4)=O)C2 C12(COC)CC(NC(C3CC34CCC4)=O)(CN1C(=O)C(c1ccc(Cl)cc1)O)C2 c1(C(=O)NC(c2onc(C)n2)C)coc2c1CN(C(c1conc1C)=O)C2 C1(C(=O)NCC(CNC(C2CC(CCC)C2)=O)O)(CC)CCC(=O)N1 N1(C(c2n(C)cnc2)=O)CC2CC(C(N3CCn4cncc4C3)=O)C(C2)C1 c1(C(N(CC=C)C2CC2)=O)cncc(CC=CC=CC(=O)N)c1.c1(SCC)ccccc1 CC(CF)CC(=O)N(C1(O)CCN(C(=O)CNC(=O)OC(C)(C)C)C1)C.C(C)(C)(C)S c1(C(N(C(CN(C(c2nc(C(C)C)oc2)=O)C)C)C)=O)cnn(C)c1C(N)=O N1(C(CC(CCC=C(C)C)C)=O)C2CCCC1CN(C(=O)CC(O)C1CCCC1)C2 N1(C(CC(CCC)NC(C2CCCCNC2=O)=O)=O)CCC2(CCOC2)CC1 C#Cc1ccc(F)c(C(N2CCCN(C(=O)C(C)Cc3cnn(C)c3)CC2)=O)c1 c1(C(=O)NC(CNC(Cc2c(C)cc(C)s2)=O)(C)C)cnn2c1S(=O)(=O)NCC2 C(C(=O)N1CCC(CCCO)C1)(C(C)C)OC c1(NC(C(=O)NC(C)CC2CCCO2)=O)cn(C)nc1-c1ccc(F)cc1 N1(CC)CCC2(CCOC2)C(C)C1.c1(CCCOC)cn(CCC(=O)OC)nn1 C(=O)(C1=NOC(C(C)(C)C)C1)NCC1N(C(c2oc(C)c(C(N)=O)c2)=O)CC=C1 CC1CC(=O)NCCN1C(C1(C)CN(C(C2SCCS2)=O)C(C)(C)C1)=O CCCCC(C(=O)Nc1cnc(C(C)C)nc1)NC(C1COCC1(C)C)=O Nc1cnc(Cl)c(C(=O)NCCC2CCCN(C(=O)Cn3ccccc3=O)C2)c1 C1(C(=O)NCCSCC(=O)NCC2(C3CC3)CCOC2)CCCOCC1 C(=O)(CCC(F)(F)F)N1CC(NC(C2C(C)NC(=O)N2)=O)C1 N1(C(c2csc(-c3ccco3)n2)=O)CCC2(CCN(C(C3CCCCS3)=O)C2)C1 c1(NC(c2ncc(-c3c(NC(COC)=O)cccc3)cn2)=O)c(C)ccnc1Cl C1(C(=O)NC(c2ccncc2)(C)C)CCCN(C(=O)CC2CCC(=O)C2)CC1 C1(C(N(CC=CC(=O)N(C(C)C)CCN(C)C)C)=O)CCCC(F)C1 C(=O)(CCCC(C)NC(C1CCSCC1)=O)N(C(C)C)CC1CCCO1 CCC(CC)(CO)C(=O)N1CC(NC(C2(C3CCCO3)CCC2)=O)C(C(F)F)C1 c1(C(N(C(CC(=O)N(CCC(C)O)C)C)C)=O)ccnc(OCC2CC2)c1 C1(C(N2CC(C(C(N3CCCC3CC)=O)OCC)C2)=O)CCC2(CC1)CC2(F)F c1(-c2ccc(-n3cncc3)cc2)ncn2c1CN(c1ncnc3sccc13)CC2 C1(NC(CCSCC)=O)CCC(N(CCO)Cc2ccc(OC)nc2)CC1 N1(C(CN(CCOC)C)=O)CCCCC1CN(C(=O)Cc1nc[nH]n1)C.CO C1(CNC(C2C(=C)CC2)=O)(SC)CCOCC1.c12nc(cs1)CNC(=O)C2 C12(C(=O)NCC3N(C(=O)C(c4ccccc4)F)CC(O)C3)CCN(CC1)CC2 c1(C(N2CCN(C(C3CCCCC3)=O)C3CC23)=O)cc2c(F)cccc2s1 N1(C(C(C)(O)c2ccccc2)=O)CCC2(CC1)CCN(C(=O)CCCC1CC1)C2 Cn1nc(C(N2CC(NC(c3nncs3)=O)C(C3CC3)C2)=O)c2c1CCSC2 CCC(C)(C#N)C(=O)N1CCC(OCCNC(=O)C(CO)N(C)C)C1 CN1CC(F)CC1C(=O)NCC12CC1CN(C(=O)CN1CC(C)(C)C1)C2 c1(NC(CC2(NC(c3ccc(C(=O)OC)s3)=O)CC2)=O)cncnc1S c1(NC(=O)NCCN2CC(C3CCCC3)C2)ccc2c(n1)OCCO2 c1(NC(C=CC=CC(=O)Nc2ccccc2-c2ccccc2)=O)cccnc1F c1(C(=O)NC2(C)CCN(C(c3nc(C)oc3)=O)C2)ccc(F)c(C)c1Cl Nc1c(C(N2CCC(NC(=O)CS(=O)(=O)C3CC3)C2)=O)ccc(Cl)c1Cl N1(C(C(C=CC)O)=O)CC(CNC(c2nc(Br)c(C)s2)=O)C(F)(F)C1 c1(OCC)ccc(C(=O)NCC2(NC3(c4ncccc4Br)CC3)CC2)c(F)c1 C(=O)(C#CC(C)(C)CNC(C1(OC)CCC1)=O)N(CC(C(C)C)OC)C C(=O)(CCC1=NNC(=O)CC1)NC1(C)CCN(C(CCC2OCC(C)(C)C2)=O)CC1 C=CCC(C)(C)CC(=O)NC(Cc1cnc[nH]1)C(=O)Nc1conc1OCC C(=O)(CS(=O)(=O)CC(=O)N(C)CC1CCCN(C(=O)Cc2ccccc2)C1)OC N1(C(CC2(C)CCCO2)=O)CCC(c2ccccc2)(NC(C2CC23CC3)=O)CC1 CC1CC2(CCN(C(C3CC(F)(F)C3(C)C)=O)CC2)CN1C(=O)CC(C)(F)F N1(C(C2ON=C(C(C)(C)C)C2)=O)CCC2(CC1)CC(CNC(C1CCCC1)=O)C2 CCCCC(O)CC(=O)NC12CCN(C(C3(COC)CCC3)=O)CC1C2 CN1C(=O)NCC1C(=O)NCC12CC1CN(C(c1coc(N(C)C)n1)=O)C2 C1(O)(CC(=O)N)CCN(N(C(C)CO)CC)CC1.c1(C)ccc(C(N)=O)nc1 Cc1cc(C(N2CCCC(CC(=O)Nc3ccc(Cl)c(C)c3)C2)=O)cc(O)n1 CC(C)(C)CCCC(=O)N1CC2CC1CCC2NC(c1cc(Cl)ncc1Cl)=O N1(C(c2ccc(CC)[nH]2)=O)CCC(C)(CNC(=O)C(c2cnccc2C)(C)C)C1 CC1CC(C(=O)NCCCC(C)(C)NC(=O)CC2(O)CCC2)CCS1(=O)=O C1(C(N2C(C(N)=O)CC2)=O)(C(=O)NCCC2CC3CCC2O3)CCCCC1 C(=O)(CC(C)(C)CCNC)N1CCCC(CNC(C(C(C)C)NC(C)=O)=O)CC1 C1(C)(C(N(C(CNC(C(C)CC2CC2)=O)C)C)=O)CC=CCC1 Cc1c(C(=O)O)ccn1Cc1nc(C(C2CCN(Cc3ccccc3)CC2)C)on1 C(=O)(C1=CCCN(C(=O)C(CO)C(C)(C)C)C1)N(C(C)C(C)(C)O)C C(C(CCC)C(=O)NCCC(=O)OC)NC(C(C)OCCC=C)=O c1(C(=O)NCCOC(C2N(C(C)=O)C(=O)CC2)=O)ccnc2ncsc12 c1(N(C)Cc2ccns2)nc(N(C)Cc2nc(O)n[nH]2)c2c(n1)CCS2 c1(CC)cn2c(C(N3CCC(C(=O)O)C3C)=O)cccc2n1 c1(Nc2c(C(=O)OCCNC(C)=O)cccc2)ccccc1C#N C1(C(=O)OCC)CN(C(=O)Nc2ccccc2Oc2cccc(F)c2)C2CC12 C1(C(=O)NCc2cc(C)[nH]c2)CC2C=CC1N(C(c1nnc(S)n1C)=O)C2 CCC(CC)(CCNC(c1ccc(=O)oc1)=O)NC(C1CCC(C)(C)C1)=O [N-]=[N+]=NC1CCCN(S(=O)(=O)C2CCOC2)CC1 N1(C(c2cc(C)c(C3CC3)cc2)C(=O)NC(C)(C)C)CCCC2CCNC(=O)C12 C1(C(N2C(CNC(c3cnc(C)[nH]3)=O)CCC2)=O)CC1C1CC(F)(F)C1 N1(CC=C)CCC(NC(=O)CN(C)C(c2cccc(F)c2)=O)CC1 C=C(C)CC(C)C(=O)N1CC2CC1C2NC(=O)C(O)CC c1(C(=O)NC2C(NC(c3cc(C(=O)OC)sc3C)=O)CCC2)cc(O)nc(C)n1 C(C(=O)N(C)CC1CN(C(c2cc(-c3cccs3)[nH]n2)=O)CCO1)(C(C)C)OC N1(C(c2cc(SC)nn2C)=O)C2CCC1C(NC(c1cnc(CC(C)C)[nH]1)=O)C2 c1(C(=O)NCC2(CN(C(Cn3c(C)nnn3)=O)C)CC2)cccc(F)c1Cl C1(C)(C(N2CC(O)(CCNC(C3OCCN(C)C3=O)=O)C2)=O)CCCCCCC1 C1(C(N2CCN(c3cncc(F)c3)CC2)=O)(ON)CCCCC1 C1(CNC(C(CC)CC)=O)CCCCCN1C(c1cc(Br)n(C)c1)=O C1(C(N(CCC(C(C)C)NC(C2(C#C)CCC2)=O)C)=O)(CF)CCC(F)(F)CC1 Cc1c(NC(=O)CCN(C)C(C2(C#N)CCCO2)=O)cccc1F N1(C(CS(CC)=O)=O)CCC(C2(NC(=O)CC3(O)COC(C)(C)C3)CC2)C1 c1(CCC)cccc(C(N2CC3C(NC(C4(CC)CCCCC4)=O)C3C2)=O)c1 c1(CC)ccc(F)c(C(N2CC(F)(CNC(C3CCC(C(N)=O)C3)=O)C2)=O)c1 N1(C(=O)OC)CC2(C)CC1(CNC(=O)NCCCc1ccncc1Br)C2 N1(C(C2N(C)CC2)=O)CCN(C(C2CCC(=O)N2)=O)CC(C)(F)C1 c1(C2C(N)C2)ccc(OC)cc1.C(F)(F)(C(F)(F)F)OC.O=S1(=O)CCN1 Cc1cc(C2CCC2)ccc1C(=O)NCC(O)CCNC(=O)C(C)(C)C#N N1(CC2(NC(CC=C=C)=O)CC2)CCN(C(c2cnccc2C(N)=O)=O)CC1 c1(CC)ccc(C(N2CC(O)(CCC(=O)NCC3CCCCS3)C2)=O)[nH]1 c1(CCOC)n[nH]c(=NCC2(CNC(c3ccsc3Cl)=O)CC2)s1 N1(C(CCC=CCC=C)=O)CC(NC(c2ccc(SC)cc2)=O)CC12CCCC2 C1(CN(C)C(=O)NCC(C)(C)C(=O)NCc2ccccc2)CCN2CCCC2C1 N1(C(=O)CCCc2cccnc2)CC2CC(C1)N(C(=O)CCc1ccoc1)C2 CCCCCCC(=O)N1CC2CC1(CNC(C1COC(C)C1)=O)C2 C(=O)(C1CCCc2nc[nH]c21)NCC(C)(C)NC(Cc1ccc(OC)cc1)=O Cc1ccc(CN=C(NCc2nc(C3CC3)n[nH]2)NC2CCCC(C(N)=O)C2)cc1 C1(C2(O)CN(C(=O)OC(C)(C)C)C2)(NCc2c(OC)cc(C)c(C)c2)CC1 C1(C(=O)NCC2CCC3(CN(c4nc(Cl)ncc4Br)C3)O2)CCCCC1C1CC1 C1(C)(C(N(C2CC(OC)C2)C)=O)CC(O)CN1C(=O)CCc1ccc(C)o1 C=CCC(C)(C)CC(=O)NCCCNC(=O)Cc1ccn(C(C)C)n1 c12cn(nn1)CC(=O)N1CCCC1C1(C)N(CC1)C(=O)C21CC1.C1(SC)CCC1 Cc1nc(C(N2CCCC(NC(C3CC(OCCN(C)C)C3)=O)C2)=O)sc1C N1(C(C2(SC)CC(=O)C2)=O)CCC=C(C(=O)NCCOCP(C)(C)=O)C1 C1(NC(C2(OC)CCC2)=O)CC2CCC1(CNC(c1oc(C)cc1C)=O)C2 c1(C(N(C2CN(C(C3(C=C)CC3)=O)CC2F)C)=O)cc2c(o1)CCCC2 c1(OC)cc(CC(=O)NC(C)C(C)NC(c2cccc(F)c2OC)=O)ccc1C N1(C(c2cc(Cl)ccc2F)=O)CCC2(CCC2N2CCC(CO)CC2)CC1 N1(C(C(C(C)C)C#N)=O)CCc2sccc2C1CNC(c1cc(F)cc(F)c1)=O c1(OC(C(=O)OC)C)ccc(-c2ccccc2)cc1S(=O)(=O)N(C)C c1(OC(C(=O)NCC(CC=C)NC(c2ccncc2)=O)C)cccc(SC)c1 C1(CC)CCN(C(c2cn(C)nn2)=O)C1C(=O)N(C1CCN(CC)C1)C C(C)(CCCC(C)C)NC(C)=O.C12CCCN1C(=O)NC2COC C#CCC(C)(C)N(C(=O)CN(C(=O)C(O)C1CCC1)C)CCOC c1(N2CC(C)C(NC(c3ccc4nsnc4c3)=O)CC2)ncccc1[N+](=O)[O-] c1(C(N2C(C(C)NC(CSCCOC)=O)CCC2)=O)nc(Cl)ccc1OC(C)C c1(CC)cc(C(=O)NC2CCC(NC(C3CSCN3C(C)=O)=O)C2)ccc1O N1(C(CC2CC(=C)C2)=O)C2CCC1C(C)C(NC(=O)CCC1C(=O)ON=C1C)C2 c1(C(=O)NC(C)C(C)NC(=O)C(C)C(F)F)cc(Cl)ncc1N c1(C(N(C2CCN(CC(=O)NC(C)C)C2)C)=O)ccnc(-n2cccn2)c1 N1(C(C2C(C)N(C)CC2)=O)CCC(C=CC(=O)N(CC(F)F)C(C)C)CC1 c1(C(C)(C)C(=O)NCCC2CC(NC(=O)CNC3CCCC3)C2)cccc(Cl)c1 c1(C(N(CCCCN(C(C(C(C)O)C)=O)C)C)=O)ccc2c(c1)COC2 C(=O)(C1=C(Cl)CCOC1)N1C(C(N2CCCC(C)(O)C2)=O)CSC1 N1(C(c2occ(C)c2)=O)CCC(C)C1CNC(c1ccc(CCO)cc1)=O C12(C(N(CCOC)CCOC)=O)CC(CN(C(=O)CC3CC(O)C3(C)C)C1)C2 C(=O)(CS(=O)(=O)Nc1c[nH]nc1F)NC(C)(CNC(=O)C1CC1)Cn1cccn1 c1(C(Cc2cn(CCN3CCC(CC(=O)OC)C3)nn2)(C)C)ccc(F)cc1Cl C(CCCCN=c1cc(C)nc(NCc2nnc(O)n2C2CC2)[nH]1)N(C)CC c1(OC)c(NC2CC(C)N(C(c3nn(C)cc3C)=O)C2)ncnc1C N1(C(CC2(C=C)CC2)=O)CCC(CC(C)NC(c2ccccc2C(N)=O)=O)CC1 c1(CNC(C(n2cc(-c3nn[nH]n3)cn2)C)=O)ccc2c(c1)COCC2 C1(C(=O)NCC2CCC(C(=O)NCC3(C(=O)OCC)CC3)C2)CS(=O)(=O)CCO1 C1(NC(C=Cc2n(CC)ncc2)=O)CN(C(=O)CS(=O)(=O)NC)C(C)(COC)C1 Cc1ccc(C(=O)NCC(C)CNC(=O)CC2=CCOCC2)c(N)c1Br c1(NC(N2CC(C)C(n3cc(CC(O)C(F)(F)F)nn3)C2)=O)cccc([N+](=O)[O-])c1F Cc1ccc(C2CC2C(=O)NCC2(NC(C3CCN(C)CC3)=O)CCOC2)cc1 c1(NC(=O)NC2CCC(C(=O)NC3CC3)CC2)ccc2ccc(Br)c(Cl)c2n1 C1(NC(C2C(c3onc(C)n3)C2(C)C)=O)CN(C(=O)C=CC(=O)N(C)C)CCC1O N1(C(CCOCCOC)=O)CCN(C(c2cncs2)=O)CC1C1CCC1 Cc1cc(N)cnc1C(=O)NCC(CO)NC(c1ccc(CN(C)C)nc1)=O C1(NC(=O)C2=CCCOC2)CN(C(=O)C=CSc2ccccc2)CC2(CC2)C1 C1(C(=O)NC(C2CCN(c3ccnc(C(=O)OC)n3)C2)C)CCC2(CCC2)CC1 C1(C(=O)NCC(CNC(Cc2n(C(C)C)cnn2)=O)C)CC(C2CC2)=NO1 C1(CC(=O)CCO)CC2(CCC2)C1.C1CCC(=O)N1CCCO.C(C(F)(F)F)O c1(C(N2CC(C)(C(N(C3CCC3(C)C)C)=O)C2)=O)ccsc1C#N Cc1cnc(C(=O)NCC(C)NC(c2cc3occc3n2C)=O)cc1C#N CCC1C(=O)Nc2ccc(C(=O)NCC(F)CNC(=O)CC3OCCO3)cc21 C(=O)(C(CCC(N)=O)N=[N+]=[N-])NCCOCC1(NC(c2[nH]n(C)c(=O)n2)=O)CCCC1 C1(C(=O)NCC(C)N(C(c2ccnc(OC)n2)=O)C)CCc2nn[nH]c2C1 C1(C(=O)NC2CCN(C(C3(S(N)(=O)=O)CC3)=O)C2)Cc2c[nH]cc2S1(=O)=O C1(CCC)C(=O)NCCN1C(C1CN(C(c2cc(Cl)n[nH]2)=O)CC1C(C)C)=O Nc1c(C(=O)NC2C3CN(C(C4CC4C(F)(F)F)=O)CC23)ccc(Cl)c1O C1(CC(N2CCC(CN(C(=O)C(c3nc(=N)[nH][nH]3)=O)C)C2)=O)CCC(F)(F)CC1 c1(C(=O)Cn2cc(C(=O)NCCN(CCOC)C)nn2)c(CN)noc1C.OC N1(C(c2nn(CC)c(C3CC3)c2)=O)CCC(NC(C2CCC(=O)N2C)=O)CC1C C(N=c1ncc(I)c[nH]1)C1C(C)CN(C(c2cnn3c2CCC3)=O)C1 c1(C(=O)NCC2(O)CN(C(C(C(CC)C)OC)=O)C2)c(C)sc2ccc(F)cc12 N1(C(CS(CC)=O)=O)CCC(C2(NC(=O)Cn3cc[n+](C)c3)CC2)CC1 c1(CC)nn(C)c(Cl)c1C(=O)N(CCC(C(C)C)NCc1cc(Cl)ccc1F)C N(C(=NCCOCC(F)(F)F)NCc1cc(C)cs1)C(C=C)C CCC(O)C(C)C(=O)NCc1ccc(CNC(=O)C(C)OCC2CC2)cc1 C1(C(N(C)OC2CCCC2)=O)COCCN(C(=O)CC2CCCCC2O)C1 c1(C(N2C3CN(C(C(CC=C)C(C)C)=O)C(C3)C2)=O)cccc2c1nc(O)n2C N1(Cc2cc(C)n(C)n2)CCC(C(=O)Nc2ccc(F)c(C(N)=O)c2)C(O)C1 N1(C(COCC(=C)C)=O)CC(C(=O)NCC2(NC(N)=O)CCCCC2)C2(CC2)C1 C1(NC(CC(=O)OC)=O)CS(=O)(=O)C2CN(C(c3cc(C(F)F)ncn3)=O)CC12 CC(C)CN=C(NCC1CCOC1C)NCCC(F)F N1(C(C(C)(C)n2cc(CCN3CC3)nn2)=O)CCC2NCCC2C1 C1(CCOC)CCCCC1N(C(C1CCN(C(=O)COc2cn[nH]c2)C1)=O)C C1(C)(CNC(C(COC)C)=O)CCCN(C(=O)CN2CCC2)C1 c1(C(=O)NC2C(CNC(CCSc3nc(C)[nH]n3)=O)C2)cnc2ncccn12 C#Cc1ccc(NC(N2CCC(O)(CC(=O)OC)CC2)=O)cc1 N1(N2CCOCC(C)(F)C2)Cc2ccccc2C1=O.C C#CCC(C)C(=O)N1CCC(CNC(=O)CN2CCCCC2=O)C1 c1(C2(NC(C)C(=O)Nc3ccccc3)CNC2)ccccc1 c1(C(N2CCOC(C)(C(=O)OC)C2)C(=O)NC)cc(F)c(F)cc1OC C1(c2nnnn2CC(F)F)(NCc2c(OCC#C)cccc2)CC(C)N(C)C1 N1(C(C(CC=C)CC)=O)CCC=C(C(=O)N2CCC(n3cccn3)C2)C1 N1(C(C=C(C)c2ccsc2)=O)CCC2(C1)CN(C(c1nnn(C)n1)=O)CC(C)O2 c1(CC)cc(C(=O)NC2(CNC(=O)CC3(C)CCCCC3)CC2)ccn1 c1(C(N2CC3CC2CN3C(c2ncccc2Br)=O)=O)c(F)cccc1F C(CC(C)(C)C)(C(=O)NC1CC1CC(C)C)NC(c1cc(C)nc(C)n1)=O CN1CCN(C(=O)CC2CCCN(C)C2)C(CNC(c2cc(Cl)c(Cl)n2C)=O)C1 c1(OCC(=O)NCC(C)(C)NC(c2coc(Cl)c2)=O)ccccc1Cl c1(C(=O)NC(C)CNC(C2CCC3CCC(=O)N23)=O)cc2cc(O)ccc2[nH]1 CC(C)(CCC(=O)NCCn1cc(CNC(=O)CN2CCCCC2=O)nn1)CO c1(C(=O)NCC(Cn2cc(Cc3ccn(C)n3)nn2)OC)conc1C(C)OC CCCC(CNC(C1(CC)CCCO1)=O)OCC c1(CNC(c2c(OCCCC)cc(OC)cc2)=O)ccc(S(=O)(=O)NC)o1 Cc1nn2cc(C(N3CCOCC3CNC(=O)C(c3cncnc3)C)=O)nc2s1 C1(C(=O)NC)CCCCN1CC(=O)N(C1CCCCC1)Cc1ccc(F)cc1 CC(F)(F)C(C)(C)C(=O)N1CCC2(CC1)CC2C(=O)N1CC(O)CO1 CC1CCC(O)(CNC(C2CCC(NC(=O)CCCN3CCCC3)C2)=O)CC1 N1(C(CCC(C)NC(=O)CN2CCCC2)=O)CC2CC1CC2CF C1(N(C(CCCOCCC)=O)CC)CCN(C(=O)C(N2CCCCC2)C)C1C C(=O)(CC(C)(C)CC(F)F)N(C)CCNC(C12CCC(CC1O)C2)=O Cc1ccc(C(=O)NCC2CCCN2C(c2cnc[nH]2)=O)[nH]1 CC1CCCC(C)N(C(=O)CC2CC(NC(=O)C(C3CCCCC3)O)C2)C1 c1(CC)conc1CC(N1CC(C(O)C(=O)NCc2occc2C)C1)=O n1(CC#C)cnnc1C(=O)NC1(CC(=O)NCCCC2(O)CC2)CCC1 N1(C(C(C)OCCOC)=O)CCCC12CCN(C(=O)CC(C)N(C)C)C2 C(=O)(C(CNC(C1(NC)CCSC1)=O)C(C)C)OCC c1(C(N2CC(NC(C3N(S(C)(=O)=O)CCC3)=O)(CO)C2)=O)c(F)ccc(Cl)c1N N12CCCC1(c1ccccc1)NC(=O)C2C1C(C)C1.C1(CC2CC2)COCCO1 C1(C(=O)NCC2(NC(CC3CCCC(C)C3)=O)CCOCC2)CC(=O)NC(=O)C1 C1(C)(NC(C(C)=C(CC)C)=O)CCCN(C(c2cn(CC3CCCO3)nn2)=O)C1 N1(C(C=C(C)c2ccco2)=O)CCN(C(C2CCC(O)CC2)=O)CC(CO)C1 c1(C(N(C(C(=O)OCC)C)C)=O)cn(CCNC(C2CCC2C#N)=O)nn1 c1(C(=O)NC2C(CNC(CCCNC(=O)OC)=O)CC2)nccnc1N c1(C(N2CC(O)(C(C(=O)NCC3CC34CC4)F)C2)=O)ncccc1O CC1OC2(C(=O)NCC3CCC3NC(=O)CSc3ccccc3F)CC1C2 C(C(C)(O)CC(=O)N1CC(=O)CC1C(N1CC(CO)CC(C)C1)=O)OC CC(C)CC(C(=O)NC1COC2(CCC2)C1)NC(=O)CN1CCCCC1=O C12(CNC(C(c3ccc(F)cc3)(C)C)=O)CCC1CCN2C(c1ccncc1)=O c1(OC)ccc(I)cc1NC(C1CC(F)CN1C(c1[nH]ccc1C)=O)=O C=CC1(C(=O)NC2CCCCC2CNC(c2ccnnc2Cl)=O)CCOCC1 CCCC(C)(O)C(=O)NCC1CC(O)(CNC(c2cc(C)c(Cl)cn2)=O)C1 S(=O)(=O)(c1cc(Cl)c(Br)cc1F)NC1CCN(Cc2c(C)c(Cl)ncc2)C1 c1(C(C)C)ccc2c(c1)C(NC(c1c(F)ccc(N)c1F)=O)CCO2 Cn1cc(N)c(C(=O)NC2CC(F)(CNC(c3cncc(-n4ccnn4)c3)=O)C2)n1 n1(CCOCC)nnnc1C(CCC1CCCO1)N(CCCCO)CC C(=O)(C1=CCCOC1)NCC1(F)CC(N(C)C(c2ccc(C(=O)CF)cn2)=O)C1 C1(CNC(C2(CC)CCNC2=O)=O)COCCN(C(=O)CCCc2cccs2)C1 N1(C(CN(CCOC)C)=O)CCN(C(=O)Cc2cc(C3CC3)on2)CC1C C1(C(N2C(CN(C)C)CC2)=O)CCc2nnc(-c3ccc(F)cc3)n2C1 N1(C(c2c(O)ccc(CC)c2)=O)CCC2CCN(C(C3(OC)CC3)=O)CC2C1 C1(CCNC(C23OCC(CC)(C2)C3)=O)CN(C(=O)C(C)C(=O)OC)CCS1(=O)=O c1(C(=O)NC2(CC)CN(C(C3CCC4(CC4)C3)=O)C2)cnc2ccnn2c1C C(CCCCCN(C(=O)C(C)C1(O)CCC1)C)NC(c1c(C)ccs1)=O c1(C(=O)NCC2(COC)CN(C(C3(OC)CC3)=O)C2)cccc2nc(O)n(C)c12 CC1CN(C(c2ncn(C)n2)=O)CC1CNC(=O)CCC(=O)c1cccc(N)c1 CCC(C)C(C(=O)NC1CCCC(CNC(=O)CNS(C)(=O)=O)C1)NC=O C(CO)(CCCCNC(c1cncc(OC)c1)=O)NC(CCC)=O CC1(C)C[Si]2(CCCC2)CN1C(=O)CCC1CCCC1 N1(C(c2c(C)[nH]cc2)=O)CC2ON=C(CNC(c3ccc4sccc4c3)=O)C2C1 C(=O)(C1=C(C)C(C)(C)OC1=O)N1CCCC(CNC(CC(CC)OC)=O)C1 c1(C(=O)NCCC2CC(NC(C3CCN(OC)CC3)=O)C2)cc2c(s1)CCC(C)C2 c1(C(N(C2(CC(=O)NCC(C)N3CCC3)CC2)C)=O)cc(C(C)(C)C)on1 Cc1ccccc1C(C)CC(=O)N(C)CCNC(c1cncc(N)c1)=O C(c1csc(Br)c1)=CC(=O)NCC1C(NC(c2c(C)cc[nH]2)=O)C1 CC12CCN(C1)CCC2.c1(CNC(=O)C(C2CCOCC2)O)ccc(F)cc1 Cc1ccc(F)c(CN2CCC2C(=O)Nc2ccc(-n3nc(C)cc3C)cc2)c1 N1(C(C2CC(OC)C(OC)C2)=O)CCC2(CC1)CN(C(=O)CC1CC1)CCO2 C(=O)(C(C)(C)C(F)(F)F)NCC1C(NC(c2c(C)n(-c3ccccc3)nc2)=O)C1 c1(OC)cccc(C)c1NC(c1cn(CCSc2ncccc2F)nn1)=O c1(N(CCN2CCNCC2)CC2CCC(C)S2)ncnc2c1c(Br)cn2C CCC(C#N)(CC)C(=O)NC(CNC(C1CC1c1ccn(C)n1)=O)CO Cc1ccc(-c2cc(C(=O)NC3CCC(NC(=O)C(O)C4CC4)C3)no2)c(C)c1 C1(C(N(CCNC(C2CN(CC)C(=O)CC2)=O)C)=O)CC2(C1)CC21CCC1 C(CN=C(NCCOC(F)F)NC1CCCN(c2ncccn2)C1)OC(C)=O C=CC(CC)C(=O)NC1CC=CCC1C(N1CCC(C(C)O)CC1)=O N1(C(C(CC(C)C)C(N)=O)=O)CC2(C)CN(C(c3ncccc3F)=O)CC2(C)C1 N1(C(C(COC)OC)=O)CCC(C(=O)N(CC(C)(C)COC)C)(CO)C1 c1(C(=O)NCC(C2CCCC2)NC(c2cc(Cl)sc2Cl)=O)ccc(F)cn1 CC(C)(C)CCC(CO)NC(=O)OC(C)(C)C.C12CC(C1)C(=O)NCCC2 C#CCCC(O)C(=O)N1CCN(CCNC(=O)CNS(C)(=O)=O)CC1 CC(C)(CCS(C)(=O)=O)C(=O)N1CCN(C(C2CCCC(F)(F)C2)=O)C2(CC2)C1 C1(C(=O)Nc2ccc(Cl)nc2)CC2CN(C(=O)COc3ccc(F)cc3)CC12 N1(C(C2(OC)CCC2)=O)CC2CCC1CC2NC(C1CCCN(C(C)C)C1)=O CCCCCC(O)C(=O)NCC1CCN(C(=O)Cc2ccc(Cl)c(OC)c2)C1 N1(C(Cn2c(C)c(Cl)cn2)=O)CC2CCCC(NC(=O)Cc3ccns3)C2C1 Cc1cn2c(n1)CC(C(N1CC3CC(NC(C4CCCSC4)=O)CC3C1)=O)CC2 N1(C(CC(CC)(F)F)=O)CC2OCCN(C(c3c[nH]cc(C)c3=O)=O)C2C1 C1(C2CCN(C(C3CC3N)=O)C2)(OC(C(=O)OC)C(C)C)CC1.CCOC(=O)C1CC1 N1(C(C=CS(CC)(=O)=O)=O)CCCCC(C2CN(C(=O)CCC[N+](=O)[O-])C2)C1 C1(NC(CNC(=O)OC)=O)CN(C(=O)Cc2ccccn2)C(C)(C)C1 c1(C(N2CC(CNC(c3cnn(C)c3F)=O)CC2(C)C)=O)cc(S(N)(=O)=O)cs1 C1(CNC(c2cc(CO)[nH]n2)=O)CN(C(=O)CCc2nc(O)n[nH]2)CCO1 Cc1ccc(CN(C2CC(NC(=O)C(c3cncn3C)O)C2)C)cc1C CCCCCCC(CC)C(=O)NC(C)CCCNC(C1(COC)CCCCC1)=O C(=O)(C(F)CC1CN(C(=O)C(C)c2ccsc2)C1)N(CC(C)OC)C N1(C(c2cnc(C(C)=O)s2)=O)CCC(NC(C2C3CC4C(C3)C24)=O)C(F)C1 C(=O)(CCC(C)C)NC(C(=O)NCCc1ncc(C)o1)Cn1cccn1 N1(C(c2c(C)nc(CCCC)s2)=O)CCCCCC(NC(=O)C(C)COC)C1 c1(C(N(C2C(O)CCN(C(c3c[nH]c(=NC)s3)=O)C2)C)=O)ccc2cncn2c1 N1(C(C(N2CCCCC2)C)=O)CC(C)(C(N2CC(CO)CC2CO)=O)CC1(C)C c1(OCC)cc2ccccc2cc1C(=O)Oc1ccc(C2(CO)CC2)nc1 C1(NC(C(C=C)(C)C)=O)CCN(C(=O)CCCc2cc(C)ccc2C)CC(C)(C)C1 N1(C(CCOCCOC)=O)CCCCC(NC(c2cn(C)c(=O)n2C)=O)C1 CCC(CCCC(=O)NC(CC1CC1)CO)NC(=O)CN(C)C(C)=O c1(OC)ccccc1NC(c1cc(C2CCCCC2)[nH]n1)C N1(C(c2c(CNC(Cc3c(C)n[nH]c3)=O)cco2)=O)CCCCC(C)(C)C1 N1(C(C2(CCCC)CCCC2)=O)CCCN(C(c2cccc(F)c2C)=O)CC1 Cc1cc(N)cnc1C(N1CC(C)(CCC(=O)NCC2COCC2(C)C)C1)=O C(=O)(CC(CNC(C)=O)CC(C)C)NCCCN(C(=O)CCCCC)CC CCCC(CNC(=O)C(=O)N(CC(F)F)C)C(=O)N(CCCC(C)C)C N1(CC(=O)Nc2csc(Cc3cccc(Br)c3)n2)CCCC12CC1CCC2C1 c1(C(N2C3CC(CC(NC(C4C(C)C4)=O)C3)C2)=O)c[nH]c2ccccc2c1=N CC1CCC(C(=O)Nc2ccc(F)cc2CO)CN1C(=O)C1=CCCC1 C(=O)(C1=CCS(=O)(=O)C1)N1CC(O)CC(NC(c2cccc(OCC)c2)=O)C1 N1(C(C(CC)C)=O)CC2(CO)CC1(C(=O)NCC(n1ccnn1)C)C2 c1(C(=O)NCC2N(C(CC=C)=O)CCC2C)c(C(F)(F)F)cccc1Cl N1(C(C=C(C)Cl)=O)CCC2(CC1)CN(C(=O)Nc1ccccn1)CCO2 C1(NC(CCC=CCC=C)=O)CCN(C(C2CCCCC2(C)C)=O)CC1CO C1(NC(=O)CCNC(c2n[nH]cc2[N+](=O)[O-])=O)C2CCCCCC12 C1(NC(CCOCCOC)=O)CC2(C1)CC2CO.C12CCN(CC1)C(=O)C2 c1(C(=O)NC(C)CCCNC(C2(c3cncnc3)CCCC2)=O)c[nH]c(=O)cn1 C1(N(C)C(C2CN(C(=O)NCC3(OC)CCCSC3)C2)=O)CCN(C(N)=O)CC1 C(CC(C(=O)NC1CC(C)(OC)C1)NC(c1cn[nH]c1)=O)OC c1(C(=O)NCC(C)N(C(c2ccsc2C(F)F)=O)CC)ccc2nc(S)oc2c1 C1(NC(=O)CCCCn2cc(CNS(=O)(=O)C3CC3)nn2)CCCCNC1 C1(CC(C)NC(=O)C(C)(C)O)CCN(C(C2(C(F)(F)F)CC=CCO2)=O)CC1 N1(C(c2cc(CC(C)C)ncc2)=O)CC2CCN(C(C3(CC(C)C)CC3)=O)C2C1 C12(NC(C(CC)(C)O)=O)CCCC1N(C(=O)C=CCOc1ccccc1)CC2 C1(C(=O)NCC2(C(N)=O)CN(C(c3c(C)scn3)=O)C2)CCSC(C)C1 C(=O)(CCCCC(C)(C)C)NCC(CCC)NC(=O)C(F)(F)C(F)(F)F Cc1cc(C)c(C#N)c(NCC(C2CCCC2)NC(=O)CCC(N)=O)n1 c1(C(=O)NCC(=O)N(C2CCN(C(C(CCC)C)=O)C2)CC)cc(F)cc(F)c1 C1(C(CNC(COCCOC)=O)CNC(=O)CCF)CCCCC1 C1(NC(C(C=CCCC)O)=O)COCCC1NC(=O)Cc1ccsc1C CC(CN=c1[nH]c2cccnc2s1)NC(C1CC(N=[N+]=[N-])C1)=O C1(SCC)CCCN1C(=O)C(OC)OC.C1(c2cn(CCC(=O)NC)nn2)CC(SC)C1 C1(CNC(=O)C(F)CC2CCCC2)CN(C(=O)C2=CCOCC2)CCCO1 c1(C(=O)NCC(C)N(C(=O)C(C)(C)CO)C)nc(C(F)(F)F)n2c1CCCC2 Cc1nn(-c2ccc(F)cc2)c(C)c1NC(C1CC(F)CN(S(=O)(=O)C2CC2)C1)=O C1(CC(=O)NCCCN(C(=O)Cc2ccc(F)cc2)CC)CC2(CCC2)C1 C1(NC(C(c2ccc(C)o2)C)=O)CN(C(C2(CO)COC2)=O)CC(C)(C)C1 CC1CC(C)(C(=O)NCCCN2CCC(NC(C3CC(F)(F)C3)=O)C2)C1 C1(NC(C2CN(C(C(C)OCC)=O)CC2(F)F)=O)CCCCCC1(C)C C(=O)(C#CC1CCCCO1)N(C1CCCN(C(c2c(N)ncc(OC)c2)=O)C1)C c1(-c2cnc(C)nc2)ncn2c1CN(C(c1cnc(F)c(F)c1)=O)CC2 C1(NC(C2(C#C)CCC2)=O)CCCC(NC(=O)CCNS(=O)(=O)C(F)(F)F)C1 c1(C(N2CC(F)CC(NC(C3CC(=C)C3)=O)C2)=O)ccc2nc(Cl)nn2c1 Cc1cn(C)nc1C(N1CCC(OCC(=O)N(CCO)C(C)C)C1)=O c1(NC2C(C(N)=O)COC2)nc2c(c(=NC3CCn4ccnc4C3)[nH]1)CCC2 CC1CN(C(C2CCCSC2)=O)CCN1C(c1ccc(C2CCCO2)[nH]1)=O c1(SC(C2CCCN2C(=O)C(C)(C)C(=O)N(C)C)C)nc2ccccc2s1 CC1CN(Cc2ccc(OC(F)(F)C(F)(F)F)cc2)CC(C)S1=O c1(C(=O)NCC2(F)CCN(C(C(C)n3cccn3)=O)CC2)cc2c([nH]1)CCOC2 C1(F)(C(=O)Nc2ccc(OC)cc2F)CC(N=c2nc[nH]c3[nH]c(Br)cc23)C1 Cn1c(O)ncc(C(N2CC(NC(=O)Cn3cc([N+](=O)[O-])cn3)C3CC23)=O)c1=O C(=O)(C1=C(C)CCCC1)NCC1N(C(C(C(C)C)NS(CCCC)(=O)=O)=O)CC1 CC(CCN=C(NCCc1cccs1)NC1CC1C1CCCCO1)C(F)F CCC(CCC(=O)NOCCO)NC(=O)Cc1ccco1 Cc1cc(C)cc(S(=O)(=O)N2CC(NC(c3cc(Br)ccc3I)=O)C(F)C2)c1 O=C(CC(C(F)(F)F)NC(=O)C(C1CCCCC1)F)NCC(F)F N1(c2cc(C(C)=O)ncn2)CC2(CC(C)CCCC2)C1 C(=O)(C1=CS(=O)CCC1)N1CCCC(CNC(c2ccccc2C(F)F)=O)C1 CCCC(CCCNC(=O)C(C)(O)Cc1ccccc1)OC C(CCC(C(=O)NCCOC)NC(C1C2CCC(C2)C1C)=O)OCCN=[N+]=[N-] C(=O)(CC(F)(F)C(F)(F)F)NCC(C1CCN(C(CSCCC)=O)CC1)(C)O CC1(C)CC(NC(c2cnc3nccn3c2)=O)CCN(c2ncc(Br)c(O)n2)C1 C1(NC(c2cncc(Cl)n2)=O)CN(C(c2cc(Cl)nc(Cl)c2)=O)C2CCCCC12 n1(CC(=O)NCCCC2(NC(c3c(SC)snn3)=O)CC2)ncc(C)cc1=O Cc1c(C(=O)NCC2CCCC2NC(c2cn(C)nc2C(C)(C)C)=O)cnn1C N1(C(=O)C(N2CC3CC2CC3O)=O)CCC(O)C(C2CCCC2)C1 n1(CC(=O)NC2CCC2NC(C2CCC=CCC2)=O)c(=O)n(CO)c2ccccc12 c1(C(N2C3(CN(C(c4scc(C(N)=O)c4)=O)C3)CC2)=O)nc2ncccn2n1 C1(NC(Cn2cc(CNC(CC(C)(C)SC)=O)nn2)=O)Cc2ccccc2C1 c1(C(=O)NCC(=O)NC(c2nncs2)C)cc(CO)n(C)n1 C1(CC)CN(C(=O)CNC(=O)CCC(C)C)CCN1C(c1cocc1C)=O C1(NC(c2cnc(C)cn2)CC)CCCC1(C)C c1(C(=O)NC2C(NC(c3cnc(C)[nH]3)=O)CC2)ccc(Cl)cc1Cl CC(CC(F)F)C(=O)NC.C(=O)(NOC(C)C)C1(CC2CCC2)CC1 C(=O)(CS(=O)c1ccc(Cl)cc1)N(CCC)CCNC(=O)C(F)CC C(=O)(CCCCC(=O)NC1CN(C(C2(C)CCC(F)(F)C2)=O)CC1C)OC N1(C(c2cc(CSC)c(F)cc2)=O)CCOCC(C)(CNC(C2CC2CF)=O)C1 C1(C(=O)NC2CC(NC(Cc3nn(C)c(Cl)c3)=O)C2)C2CCN(CC2)S1(=O)=O C1(NC(CNC(=O)OC)=O)CC2CCC1N(C(C1CC3CCC1C3)=O)C2 C1(CC(=O)NCCC(C)N2CCC2)CCCCC1NC(c1ccsn1)=O C1(C2CCCOC2)(NC(=O)CCNC(C2CCN2C2CCCCCC2)=O)CC1 CCC(CC)(C(=O)N1CCOC(C)(CNC(=O)COCC2CCC2)C1)OC Cc1c(C(N2CCC(CO)(NC(C3CC3C(N)=O)=O)C2)=O)csc1Br CCC1=NOC(C(=O)NC2CC(NC(c3ccc(COC)[nH]3)=O)CC2O)C1 n1(CC(=O)NC2CC(C)(C)CN(C(C3(O)COC3)=O)C2)[nH]cc2c(=O)ncnc1-2 N1(C(CCC(C)N(C)C)=O)CCCC12CCN(C(=O)C1=CCCCO1)CC2 c1(C(N2C(CNC(c3c(OC)ccs3)=O)CCC(C)C2)=O)cnn2c1NCCC2 C1(C(=O)NCC2N(C(C)=O)CCC2)CCN(C(=O)CN(C)C)C1C(C)C C1(C(=O)NC2CC2C(=O)NCC2CCCCC2)CCCN(Cc2ccccc2)C1 c1(OC)cc(C)sc1C(=O)NCC#CCNC(c1cccnc1O)=O c1(OC)c(CN2CCC(F)(CO)CC2)cccc1Cl.C1(C(C)C)C(=O)NC(=O)N1C O=C(C1CCc2ccccc21)NCC1CC(NC(C2CC3(CCCCO3)C2)=O)C1 N1(C(=O)NCCc2c(C)cccc2C)CC2COCCC2(C(=O)O)C1 Cc1cc(=NCC2(O)CC(NC(C3CCCN3N=O)=O)C2)[nH]c(S(C)(=O)=O)n1 S(=O)(=O)(c1ccc(C#N)c(NCC(O)C2(C)CC2)c1)N(C(C1CCCO1)C)C Cc1ccc2c(c1)SC(C(=O)Nc1ccc(F)cc1CO)C2 Cc1cc(C(N2CC(CNC(C3CC3F)=O)C3CC23)=O)sc1Cl c1(N2CCC(C(CN3CCC(C)C3C)=O)CC2)cccc(Cl)c1F C1(CNC(CCc2ncc(C)[nH]2)=O)COC(C)(C)CN1C(=O)C(C)C(C)(C)C CC(C)C(O)C(=O)NCC(C1CCCCC1)NC(=O)CC(C)c1ccccc1 N1(C(C(C(C)C)CO)=O)CC=C(CCNC(=O)CCOc2ccc(F)cc2)CC1 c1(OC)cccc(C(=O)NCC2CC(C)N(C(C3(CO)CCCO3)=O)C2)n1 N1(CC(=O)OCC)CCN(C)CC1NS(CC1N(CC(=O)OC)CC(F)C1)(=O)=O C#CCCCC(=O)N1CC(NC(C23CC(C(F)F)(C2)C3)=O)C(C)C1 c1(C(=O)NCC(C(C)C)NC(C2C(OC)CCCC2)=O)cnc2sc(C)cn12 C1(CC(=O)NCC23C(CN(C(CCN(S(C)(=O)=O)C)=O)C2)C3)CC(C)(C)OC1=O C1(COC)(NC(=O)C(C)n2ccnn2)CCCN(C(c2csc(=N)[nH]2)=O)C1 C=C=CC(C)C(=O)NC1(CNC(c2coc(C(=O)OC)n2)=O)CCOCC1 c1(OCC)ccccc1C(N1CCNC(C(=O)NCCc2ccccc2)C1)=O c1(C(N(CC(=O)NC(c2ccccc2)CC2CCC2)CC)=O)cc[nH]c1C(=O)O N1(C(C(CC=CC)NC(=O)C(=O)Nc2ncc[nH]2)=O)CCCCC(C)C1 c1(C(N(CCC(=O)NCc2ccc(C)o2)C(C)C)=O)cnn(C)c(=O)c1 c1(CC(=O)NCC(CCOC)NC(C2(C)CC2C)=O)ccc(F)cn1 N1(C(CSCC)=O)CC2CC(NC(C3(C(C)C)COC3)=O)CC1C2 C(=O)(C(C(C)CC(C)C)N(C)CCN1CCN(C)CC1)NCC(C)C C(=O)(C1CNC(=O)c2ccnn21)N1CCC2(CCN(C(C3(C)CCC3)=O)C2)C1 c1(CN(C(=O)C(=O)NC(c2ccc(OC)cc2)C)CCOC)cc(F)cc(F)c1 C1(C(N2CC(NC(C3(COC)CC3)=O)CC2(C)C)=O)CCc2nc(=N)[nH]cc2C1 CCC(C#N)(CC)C(=O)NCc1ccc(CNC(c2ccc(C(N)=O)[nH]2)=O)cc1 c1(C(=O)NCC2(O)CCN(C(C3(C)CCCN3)=O)C2)ccc(F)c(F)c1 c1(C(=O)NC2C(CO)CCN(C(C(C=C)O)=O)C2)cc2cc(F)ccc2o1 C12(CNC(CCC)=O)CCC(CN(C(c3cnncc3O)=O)C1)C2 C1(NC(c2cc3sccc3[nH]2)=O)CN(C(C2(O)CCOC2)=O)Cc2nccn2C1 C1(CCCNC(=O)CC2COC(=O)C2)CN(C(c2cccc(F)c2)=O)CCO1 C1(C(=O)NC(C)CC2CN(C(C3CC3(C)C(F)(F)F)=O)C2)CC(F)C(=O)N1 c1(C(C)=O)cc(OCCOC)c(F)cc1N C1(CC)CN(C(=O)CCc2cn(C)nn2)CCC1NC(C1(O)CCC(C)CC1)=O C(C(C)C(=O)OC)NC(C)Cn1cc(C(c2ccccc2)OC)nn1 CCC(O)C(F)(F)C(=O)NCC(C)NC(c1ncoc1C1CC1)=O N1(C(c2c(CC)nc[nH]2)=O)CC23CCCC2(C1)CN(C(C1(C)CCCO1)=O)C3 N1(C(c2cc(CNC(C(C)=CCC)=O)[nH]n2)=O)CCOC(C)C1C N1(C(C2C=CCN(C(C(OC)OC)=O)C2)=O)CCC(=C(F)F)CC1 C(=O)(C1CCc2ccc(OC)cc21)N1CC(NC(C2C(OCC)C2)=O)C(CC)C1 CCCS(=O)(=O)CC(=O)N1CC2CCCC2(CNC(C2CCS2(=O)=O)=O)C1 c1(SCC)ccccc1C(=O)NCC(C)(C)CN(C)C(C1CCC1(OC)OC)=O N1(C(c2cc(C)nc(C)c2)=O)CCCC2(C1)CN(C(=O)CN1CCCCC1=O)C2 N1(C(c2cc(C)cc(Cl)c2)=O)CC(NC(=O)CC2CCSCC2)CC12CCOC2 N1(C(c2c(C)nccn2)=O)CCC(CNC(=O)C(c2ccc(Cl)s2)=O)C1(C)C CC(CCN(C)C)C(=O)NC1C2CN(C(=O)CC3CCCC3O)CC12 C1(C(=O)NCc2ncc(C(=O)OC)nc2)CN2CC3CC2(CO1)C3 CCC(CC(=O)N1CCCN(C(C2(O)CCC2)=O)CCC1)C(C)C c1(NC(C(c2cnn[nH]2)N(C2CCC(C)C2)CC#N)=O)cccc(OC(F)F)c1 C1(C(N2CC(OC(COC)C)C2)=O)CCC(C)(C)N(C(=O)C(C(C)C)OC)C1 c1(CC)cccnc1S(=O)(=O)NCc1cc(Cl)cnc1-c1ccn(C)n1 c1(CCC)cc(C(=O)NCCOCCCN(C)C(c2csc(O)n2)=O)n[nH]1 Cc1cc(F)c(C(=O)NCCC(C)NC(=O)C(N)Cc2cnc[nH]2)cc1F Cc1nn(C)c(C)c1CCCNC(=O)COC(=O)CNc1ccncn1 CC(CC(=O)N1CCN(C(c2csc(S)n2)=O)C(C(C)(C)C)C1)C(F)F c1(NCC(COC)(F)F)nc(N2CC(=O)N3CCCC3C2)nc2ncn(C)c12 C1(CNC(C2CCCC2)CC)CCN(CC#N)C1 CC1=C(C(=O)N(C)CC2(O)CN(C(C3CCC(F)C3)=O)C2)COCC1 C1(C(C(=O)N(CC(C)O)CCNC(=O)CCF)OC)CCOCC1 C12(NC(=O)CCOC3CCCC3)CCN(C(c3ccnc(Cl)c3O)=O)CC1C2 N1(C(c2c(OC)cc(O)nc2)=O)CCC2CCC(NC(c3ccncc3)=O)C1C2 C=CCC(C(=O)N1CC(C(C)NC(c2ccc(C3CC3)s2)=O)C1)C(C)C C1(C(N2CCC(N(C(=O)CCOC3CCC3)C)CC2)=O)CCC2CC2CC1 c1(C(N2CCC(c3cn(C4CC4)nn3)C2)=O)ccc(CC2CCC2)c(Cl)c1 C(=O)(CCS(=O)(=O)NC)N(CC(CO)(CO)NC(C(CCC)N(C)C)=O)C c1(C(N2C(C(=O)NC(CCCC(C)C)C)CC(O)C2)=O)c[nH]c2ccccc12 N1(C(c2ccc(C)cc2)=O)CCCC2C(NC(c3cn(C)nn3)=O)C(C)(C)C12 C1(C(=O)NC(C)CCNC(C2CCC(C(N)=O)CC2)=O)CCCC2C1C2(F)F C1(O)(C(=O)NC(C2CCN(C(CCNC(C)=O)=O)CC2)C)CC2(CCOCC2)C1 N1(C(COCCOCC)=O)CCC2(CC2)CC1C(=O)NC(C(O)CO)C1CC1 N1(C(C(F)OC)=O)CCC(CNC(=O)COc2cccc(C#N)c2)CC1C C1(CC(=O)NCCSCC(=O)NCC2CCCS2)COCCO1 C(=O)(C1CCCc2ncccc21)NCCN(CCc1c(C)nn(CC#N)c1C)C C=C(C)CCC(=O)NC(C)CCCCNC(=O)C(N1CCSCC1)C C1(OC(CCC(=O)NCCCCCCC)=O)CC(c2ccc(OC)cc2)=NO1 C1(CNC(C(C)(C)NS(C)(=O)=O)=O)CCC2(CN(C(=O)CC#N)C2)O1 CCCCC(C)(F)C(=O)N1CC2(CNC(=O)C(C(C)C)NC(N)=O)CC1CO2 n1(CC)cc(Cl)cc1C(N1CCC(NC(C23CC(CO)(C2)C3)=O)CC1)=O C#Cc1ccc(C(=O)NCc2cc(C(N3CC(O)CC3C)=O)on2)cc1C c1(OC)c(CC(=O)NCC2CCC(NC(=O)CN(C)C3CC3)CC2)cccc1Cl C12(C(=O)NCCC(C)NC(=O)CCCF)CCC(C1)C2 N1(C(C2(CSC)CC2)=O)CCC(CCN(C(=O)CCc2cc(C)sc2C)C)CC1 C1(N(C(=O)CC2(N(C)C)CC2)C)CCCN(NC(C2(C3CCCCO3)CC2)=O)C1 C1(NC(C(CC)(C)O)=O)CCC(C)N(C(C2CCC(C(=O)OC)C2)=O)C1 C1(CNC(CCS(C)=O)=O)CC2(CCN(C(c3cccn4cnnc34)=O)C2)CO1 Cc1nc2ccc(C(=O)N(CCCCCNC(=O)CCCC(F)(F)F)C)cn2n1 c1(C(N2CC(CC)N(C(C3CC(OC)C3)=O)CC2)=O)ccc(C)c(Cl)c1F CC1=C(C(=O)NCC2CN(C(C3CC34CCc3ccccc34)=O)C2)CCCO1 C1(CC=C)CCCN(C(=O)CC2(C)CN(C(=O)CC3CC=CCC3)C2)C1 c1(C(=O)OC)cccc2ccc(N3CCC(Oc4ccc(Cl)cn4)CC3)nc12 c1(C(N(C)CC2OCCN(C(C(CC)C#N)=O)C2)=O)cccc(=O)n1C N1(C(C(COC)NC(c2csc(C)n2)=O)=O)CCC(F)(F)C(CO)C1 C1(NC(COCCOC)=O)CCN(C(c2ncc(OC)cn2)=O)C2CC12 CCC(C)C(C(=O)N1CC2CC2(CNC(c2ccco2)=O)C1)c1ccccc1 C1(CC(=O)NC2CCN(C(=O)N(C3CCCC3)CCO)C2)CCc2ccccc2O1 CCCCCC(C)CC(=O)N1CCN(C(c2ccc(C(N)=O)[nH]2)=O)C(CF)C1 C1(NC(c2cn[nH]c2)=O)CN(C(C2CC3CCC2O3)=O)CCC12CCC2 CC1CN(C(=O)CC(O)CNC(C2(O)CCCCCC2)=O)C(C)CO1 CCC(C)C(O)C(=O)NCc1csc(CNC(C2(Cc3ccccc3)COC2)=O)n1 C(CC1CC1)(C(=O)NC1(C2CCCO2)CCC1)NC(C1C(C)CC1)=O C1(CC(=O)NCC2(F)CCN(C(CCSC)=O)C2)CCOCC1(C)C CCCC(C)C(=O)N1CC(C)C1C(=N)c1ccc(OCC(=O)O)cc1 N1(C(c2cnccc2C(F)F)=O)CCC2(CCCN(C(C3C=CCCC3)=O)C2)C1 CC1C(N(C)C(C2COCCN2C(=O)CCc2cscn2)=O)CCCC1C N1(C(CCCNC(C2CC(C)(COC)C2)=O)=O)CC(OCC#C)C(OC2CC2)C1 CCCC(C(O)C(=O)Nc1ccc(OCC)nc1)NC(=O)CC(C)C Cn1cc(C(N2CCN(CC(=O)NCC3CC4CCC4C3)CC2)=O)ccc1=O C1(NC(C2C(C)OC(C)C2)=O)CC2CCC1N(C(c1c[nH][nH]c1=N)=O)C2 Cn1ccc2ccc(-c3nc(C(=O)N(C(C)(C)C)C)cs3)cc12.C12CN(CCO1)C2 C12(C(=O)NC3CCN(C(=O)CC4CCCCO4)C3)CCC(C(F)(F)F)(CC1)CC2 CS(=O)(=O)c1cc(C(=O)NC2CCC(CNC(c3cnc(O)o3)=O)C2)co1 C1(CC)CC(O)CN1C(=O)CC1CN(C(c2occc2COC)=O)CCO1 C1(NC(C(C)N(C)C)=O)C2CC(NC(c3cccc(N4CCCC4)c3)=O)CC12 c1(C(=O)NC(CCCC)CNC(c2ccn(C3CCC3)n2)=O)cc2cn[nH]c2cn1 Cc1cccc(Cl)c1C(=O)NC1CCCCC1CNC(C1CC1(F)F)=O c1(C(=O)NCC2CC(OC)CN2C(=O)CC2CCC(=O)NC2)cnc(O)c(C)c1 N1(C(C(CCC)NC(C23CCC(C2)C3)=O)=O)CC(N(C)OC)C1 CCC(CNC(c1ccnnc1C)=O)(CC)C(=O)NCc1ccnn1CC c1(CNC(CCCC#C)=O)ccc2c(c1)CN(C(=O)CCCCc1cnc[nH]1)C2 c1(C(=O)NC2C(NC(c3c(C)cns3)=O)C2)occ2c1CCC2 C1(C(N(CCCC=C)C)=O)C=CCCN1C(=O)CCc1ccncn1 Cc1cn2nnc(C(=O)NCCC(O)CNC(C3C4COCC34)=O)c2c(O)n1 N1(C(C(C=C)(C)C)=O)CCC2CN(C(c3cc(Cl)ccc3OCC)=O)CCC2C1 c1(OC)c(C(=O)NC2CCCN(C(=O)CCC3C(=O)ON=C3C)C2)cccc1F C1(C(=O)NC(c2coc(CNC(=O)CC3CCC(C#N)C3)c2)C)CC2COCC2C1 c1(C(N2CCC(N(C(CC(C)N3CCCC3=O)=O)C)C2)=O)cncc(C#N)c1 c1(C(=O)NC(CN(C(c2cccc(C)c2O)=O)C)C)cc2c(nc1N)CCC2 c1(C(C(F)(F)F)OC(C(c2ccc(OC)cc2)C)=O)cc(Cl)ccc1Cl C1(NC(c2cnc3ncccn23)=O)CCC2CN(C(=O)CC3(CO)CC3)CC2C1 O(NC(=O)C(C(C)N(C)C)C(C)C)C(C(=O)N1C(CC)CC(O)C1)CC(C)C C12(C(=O)NC(c3nc[nH]n3)C)CC(c3ccccc3)(C1)CS(=O)(=O)C2 c1(C(=O)NCCCN(C(=O)C(C)(C)O)CC)nn(CC)cc1Cl Cc1nn(C)c(C)c1C(=O)NCC(O)CNC(C1(C(C)C)CCCO1)=O C1(NC(c2cscc2Cl)=O)CCN(C(=O)Cn2cc(C3CC3)nn2)CC1 C1(S(=O)(=O)c2ccccc2)(C(=O)NC(c2ccc(OC)c(Br)c2)C)CC1 C1(NC(c2cnncc2NC)=O)CCN(C(C2(CC)CC(C)(C)C2)=O)CC1C C1(CC(=O)NCC(C)CN(C)C(C2CNC(=O)N2)=O)COC(=O)C1 CC(C)C(C(=O)N1CC(C(C(=O)N(CC(C)(F)F)C)N(C)C)C1)n1cnnc1 C12(NC(c3cn(CC=C)nc3)=O)CCN(C(c3coc(Cl)n3)=O)CC1C2 C(=O)(CCCF)NCC(C1CCCCC1)NC(C1(C(N(C(C)C)C)=O)CC1)=O N1(CC(=O)N(CC(C)NC(=O)C(C)c2ccco2)C2CC2)CCP(C)(=O)CC1 c1(C(N2C3C(N(C(c4cnc(C)[nH]4)=O)C)CC(C3)C2)=O)ccc2ncn(C)c2n1 O=C1CC2COC(CN3CCC(c4ncccn4)C3)CN12 CCC(C)(CO)C(=O)N1C2CCC(C2)C1CNC(C1CCCS1(=O)=O)=O N1(C(CCN(C(=O)C)CC#C)=O)CCN(C)C(C)(C)C1.C(CC)=CC C1(C(=O)NC2CC(CCNC(c3nn(C)c(O)c3)=O)C2)CC12CCC(C)(C)CC2 C(C)(CCCC(=O)NCc1sccc1C)NC(C1(CC#C)CCC1)=O C1(CNC(C(c2ccc(F)cc2F)C)=O)CN(C(=O)CCC(F)(F)F)CCN1C N#Cc1cncc(C(=O)NC2CCN(C(C3CC3c3ccncc3Cl)=O)C2)n1 C(CC(C)CC)(C(=O)Nc1ccc(O)c(Cl)c1)NC(CC(CC)CC)=O C(C(O)CC(=O)NCC1CC1NC(=O)Cc1cnccc1OC)N(C)C C=CC1(CC(=O)NCC(CC)NC(c2cc(CCC)ccc2N)=O)CCCCC1 C(C(C)C(C)C(=O)N1CC(OCCC(=O)NCc2csnc2C)C1)OC C1(NC(C(C)NS(CC)(=O)=O)=O)CCC2CC1CN2C(=O)CC1CCCCC1 c1(CN(CCOC)Cc2ccc(OC)cc2F)cc(C)nnc1C CCCC(C)CC(=O)NC1CN(C(C2CCC23CCC3)=O)C1 N1(C(C(CC)O)=O)CCCC(NC(=O)C(c2ccccc2C(F)(F)F)(F)F)CC1 C(=O)(C(F)C(=O)NC(C)(C)CC(=O)NC(COC)C(C)C)OCC C(=O)(C(C)(O)CC(F)(F)F)NCC1N(C(CNC(C)=O)=O)CCC1 N1(C(C2N(C(c3cc(C)no3)=O)C3C(C2)CCC3)=O)CCCC(C2CC2)CC1 C1(c2n(CC)nnn2)(NCCS(=O)(=O)N(C)C)CCOCC1CC1CC1 C#CC1CCCN(C(=O)C(c2cn(C)nn2)NC(c2ccccc2F)=O)C1 C1(OCC(=O)N(CCNC(C(C)C)=O)C)CCN(C(C2CCC(O)CC2)=O)CC1 c1(C(=O)NCC(C2CCCN2C(C2CCS(=O)CC2)=O)(C)C)cncc(F)c1 C(=O)(CC(F)(F)CC(=O)OC)NCC(CNC(C(CC)c1cccnc1)=O)C C1(NC(CCOCCCOC)=O)CCC(CNC(c2ccn(C(F)F)n2)=O)CC1 N1(C(c2cc(OC)c(F)c(F)c2)=O)CCC2(CCC2NC(=O)C(C)OC)CC1 c1(C(=O)NC2C3CN(C(COCCC=C)=O)CC2C3)ccc2c(c1)CC(C)O2 n1(CC)nc(C(=O)NCC2CCN(Cc3ncccn3)C2)c2ccccc2c1=O C1(CC(=O)NCCC(CNC(CSCC)=O)OC)CCn2cncc2C1 N1(C(CC2C(C)(C)OCC2)=O)C2CC=C(C(=O)C3CCCC3)C1CC2 Cc1c(C(=O)NCC(O)CNC(=O)C(C)(F)F)sc2[nH]cnc(=S)c12 C1(CCNC(c2[nH]cc(CC)n2)=O)CN(C(=O)CCc2cncc(F)c2)CC1C C1(CC(=O)NC)CC2CCC1O2.C(C(C)(C)C)N(C(=O)CCC1OCCO1)C N1(CC(=O)N(CCC(=O)NCCC2(CO)CCC2)C)CCCC1C Brc1nc(CNC(c2nnnn2CCC2CC2)C2CC3CC3C2)co1 N1(C(CCCOC)=O)CCC2C(C1)NC(=O)CN2C(c1cc(C)ncn1)=O Cc1cccc2[nH]c(C(=O)N(C)CC3CCCN3C(=O)COCCN(C)C)cc12 C1(CC(=O)OCCc2ccc(F)cn2)CCCC(F)(F)C1 C1(CNC(CN2CC(C)C2)=O)C2CCN(C(=O)C(C)c3ccsc3)CC12 C(C(CC(C)C)C(=O)N1CCC(C(=O)NCc2n[nH]cc2C)CC1(C)C)OC C1(O)(CC(=O)NC2CN(C(C3C(C#C)C3(C)C)=O)C2)CCCN(C)C1 c1(C(N(C)CC2CCCN(C(CCCC#C)=O)C2)=O)cc2cccnn2c1 CC1CN(C(=O)CCCC#N)CC(C)N1C(C1(C)CCC(=O)CC1)=O CC(CN(C)C)CC(=O)NC1CCC(NC(C2(COC)CC(F)(F)C2)=O)C1 N1(C(C(CCC)OCC)=O)CCC(C2CCN(C(c3cncnc3)=O)CC2)C1 C1(NC(N2CCC(c3scc(C(C)=O)n3)CC2)=O)Cc2nnc(C)n2C1 c1(C(N(C)CC2(NC(COCCOCC)=O)CC2)=O)nccc2ncccc12 c1(C(=O)NCC2C3CN(C(c4cc[nH]n4)=O)CC23)ccc2c(O)nc(S)nc2c1 c1(C(=O)NCC2CCN(C(=O)CSCC3CCCO3)CC2)cc2ccccn2c1 C(CN=c1[nH]c(=NCC2CCCC23CC3)[nH]c2c1CSC2)N1CCC(C)(F)C1 Cc1nsc(N)c1C(=O)NC1CC(C)(NC(c2sc(C(C)C)nc2C)=O)C1 N1(C(C(F)=C(C)C)=O)CC(O)CC1(C)C(N1CC(c2cc(O)n[nH]2)C1)=O c1(CNC(CSC)=O)ccc2c(c1)CCN(C(=O)C(C)(C)F)CC2 C(CCC)(C(=O)NC(C)CCCNC(CC(C)(C)C)=O)=CCC.C(=O)(CNC)N c1(C(=O)NC2(C)CCN(C(c3cnc(CC(C)C)s3)=O)C2)ccc(F)c(F)c1 N1(C(=O)CS(=O)(=O)C2CC2)CCOC2(C1)CN(C(C1CCCOC1)=O)C2 Cn1cc(SCC(=O)NC2CCCC2NC(C2CC23CC3)=O)cn1 N1(C(C2(C)CCCCC2)=O)CC(NC(C2CC(C(F)F)C2)=O)CC(O)C1 C1(NC(C(C(C)C)OCC)=O)CN(C(=O)CCCCCOC)CC12CCOCC2 C(=O)(C#CC1CCCC1)NCCC(=C)CNC(=O)CC1CCc2ccccc2C1 CC(C)C(C(=O)NC1(C(=O)NCC(c2ccco2)O)CCCC1C)C(C)C N1(C(CCc2cc(C)sc2C)=O)CCN(C(C2CCC(C)(O)CC2)=O)C(C)C1C C1(OC(C)C(=O)NC2(C)CN(C(c3cc(Br)co3)=O)C2)CCCCCC1 Cc1ccc(C(=O)N(C)CC2(NC(c3cc[nH]c(=N)c3)=O)CC2)cc1Br C1(C(=O)N(CC(C)NC(c2cc(C3CCC3)no2)=O)C)(OC)CCSC1 CC1CCN(C(C23COCC2CN(C(=O)CC2OCCO2)C3)=O)CC1(F)F C1(NC(C)=O)CCC(NC(=O)C(N2CCC(Cc3ccccc3)CC2)=O)CC1 C1(NC(C(C)C)=O)CC2(CCC(NC(=O)C(C)C3CCCO3)CC2)C1 C1(NC(C2CCCN(C)C2)=O)C2CCC1CN(C(=O)CCc1ccsc1)C2 c1(CN2C(C(=O)Nc3cccc(I)c3)CC2)cc(Br)ccc1[N+](=O)[O-] C(=O)(C1(C)Cc2cccc(Cl)c21)N1CC(NC(C2CC=C(C)CC2)=O)C1 Cn1[nH]c(C(N2CCCC2C2(NC(c3cccnc3N)=O)CC2)=O)nc1=O C1(C(=O)NC23CC(NC(c4nn(CC)nc4Br)=O)(C2)C3)CCc2nccn2C1 n1(CC(=O)N(CCNC(C2(C(=O)OC)COC2)=O)CC)nccc1C N1(C(c2ccc(C#C)c(C)c2)=O)CCC2CCN(C(=O)CCSC)CC2C1 c1(-c2ccc(OC)cc2)nc(N2CCCC(C(C)(C)O)C2)ncc1C C1(CN(C(CCc2nc(C)sc2)=O)C)CCCN(C(c2coc(C)n2)=O)C1 c1(C(=O)NC2CN(C(CCCOC)=O)C2)ccc(OC)nc1Cl N1(C(=O)COCc2ccccc2)CCN(C(=O)Cc2ccno2)CC1C1CC1 c1(NC(=O)OC)cc(C(=O)NCC=CCNC(=O)C(C(C)C)SC)ccc1F c1(C(N2CC3C(CNC(c4cc5sccc5[nH]4)=O)(C3)C2)=O)nnn2c1CCCC2 C1(CNC(C(N(C)C)C2CC2)=O)CCN(C(c2ccnc(CO)c2)=O)C1(C)C N(C1CNCCc2ccccc21)CC1NC(=O)C2=C1NC(=O)NC2c1ccccc1 C(C)(CCN=C(NCCc1ccc(O)c(C)c1)NC1CCC1)SC c1(C(=O)NC(C)C(=N)NOCc2ccccc2)ccc(O)cc1 C(CCCCC(=O)NC(C)C(C)F)NC(C#CC(C)C)=O C1(NC(C=CCN(C)C)=O)CN(C(=O)C(c2cccc(Cl)c2F)(F)F)CCC1F CC(C)(C)C#CC(=O)N1CCCCC(C(=O)NCC2COC(C)(C)C2)C1 N1(C(C2CCN(C(c3c(C)cns3)=O)CC2O)=O)CCCCCCC1C CS(=O)(=O)c1ccc2c(c1)CCN2C(N1C2CCC1CC(=C)C2)=O CC(F)(C(=O)NC1CC(NC(C2CCCN2c2nccs2)=O)C1)C(F)(F)F c1(OCC(=O)Nc2scc(-c3ccc(CC)o3)n2)ccc(F)c(Cl)c1 C12(NC(CC3(OC)CC3)=O)COC(C1)C(NC(C1CC(C(C)C)C1)=O)C2 CCCCCCN(CC(=O)NCC(C)N(C(=O)CSc1cscn1)C)C c1(C(=O)NCC2C(NC(CC3(C)CC3)=O)CC2)ccc(OCC2CC2)nc1 C(C(=O)NCCC1(NC(c2ccsc2-n2cnnn2)=O)CC1)(C(C)C)SC N1(Cc2cn(CC)nc2)CCC2C1CCCN2C(c1ccc2ncccc2c1)=O c1(C(=O)NCC2(F)CCN(C(c3[nH]cc(C)c3)=O)C2)ccc2cc[nH]c2c1F C12(Cc3cccc(F)c3)CCN(CC1)C2=O.N1(NC(C(C)SC)=O)CC2CC2C1 c1(C(=O)NCC2N(C(=O)Nc3cc(C)c(Cl)cc3)CCC2)nc2ccccc2[nH]1 c1(C(=O)NC2(C)CC(NC(C(C)NC(COC(C)C)=O)=O)C2)cccc(F)c1 Cc1cc(C(CC#N)NC(NOCC2CCCC2C)=O)ccc1F N1(C(c2nccc(N)c2Cl)=O)CCC(NC(=O)COC(F)F)C(CO)CC1 C(=O)(C(C(C)O)NC(N)=O)NC(C)C(CO)NC(=O)C1=CCCC1 Cc1cc(O)ncc1C(=O)N(C1CCCN(c2ncccc2C(N)=O)CC1)C c1(CCC)cc(C(N2CCCC2C(=O)Nc2cnn(C(F)F)c2)=O)n[nH]1 C1(N(C)C(c2cn(C3CCOCC3)nn2)=O)CN(C(=O)CC(C)(F)F)CC1F C#CCCC(O)C(=O)N1CCN(C(c2ccsc2Cl)=O)C(c2ccccc2Cl)C1 Cc1cccc(NC(C2CSCN2C(C2CCOC2)=O)=O)n1 CCCCC(C(=O)NCC(C)Cn1cccn1)NC(=O)CCn1ccnn1 C(=O)(CN=S(C)(C)=O)NCCN(C(=O)CCCn1ccnn1)CC N1(C(C2CN(C)C2)=O)C(CNC(C2CC3CCCCC(C2)C3)=O)CC2COCC12 C1(CC(=O)NC2CC(NC(c3cnc(OCC)s3)=O)C(O)C2)CCC(F)(F)CC1 c1(-c2cn(CC(N3CCOC(Cn4cncn4)C3)=O)nn2)cc(Cl)c(Cl)cc1Cl c1(C(=O)NC2C(NC(c3ccc(OC)nc3)=O)C2)nncc2c1CCCC2 CC1(CNC(=O)CCc2cc(Cl)no2)CCCN(C(C2(C3CCC3)CCC2)=O)C1 C(=O)(C1=CC2C=CC(C1)C2)NCC1CCC(C(=O)NCCCOCC)C1 C1(N=[N+]=[N-])(C(N(C(C#C)C)C)=O)CCN(C(c2cc(C(N)=O)co2)=O)C1 C(=O)(C(C(C)C)SC)NCC(CC=C)NC(=O)C=CCOCc1ccccc1 C1(NC(c2cnoc2)=O)CN(C(=O)C(O)CN2CCCC2)CC12CC2 C1(CNC(c2oc(CC)c(C)c2)=O)CCC(C)(C)CN1C(C1CCCO1)=O CC1CN(C(=O)CNC(=O)NC2(c3ccccc3)CCC2)CC(C)S1 N1(C(c2c(CC)n(C)nc2)=O)C2CCC(C(=O)NC(C)C(=O)N(C)CC)C1CC2 c1(C(N2CC(C)C(NC(=O)CC3CCCOC3)CC2)=O)ccc([N+](=O)[O-])c(O)c1 Cc1ccc(CN2CC(CC(N3CCCC3Cc3ccc(Cl)s3)=O)C2)c(F)c1 N1(C(C(C)C(F)F)=O)CCC2(CC1)CC2C(N1CCC(C)(O)CC1)=O C#CCCCCCCC(=O)N1CCCC1C(N1CCCC1C(F)(F)F)=O C1(CNC(C=CC(=O)NC2CC2)=O)(CO)CCN(C(C2CCCCC2O)=O)C1 CCCC(O)(CCC)CC(=O)NC1(CNC(C2OCC2(C)C)=O)CCC1 N1(C(Cc2n(C)cnn2)=O)CC2CCC(C1)N2C(c1ccns1)=O Cn1cc(C(=O)NCC2CN(C(c3cc(F)cs3)=O)CC2(C)C)c(O)nc1=O CC(CCCCNC(=O)C(C)(C)C1CCCC1)NC(C1CC(N(C)C)C1)=O CN1CC(C)(C)CC1C(N1CCCC1C(C)(C)CNC(C1(C)CCCCO1)=O)=O N1(C(CCSCCC)=O)CC(C(=O)NCCN(CC(C)O)C)CCC1(C)C C(c1c(Cl)cccc1Cl)=C(C)C(=O)NC1CCCN(C(=O)C=C2CC2)CC1 N1(C(C2(C(=O)NC)CC2)=O)CC(C)(C)CC1C(=O)NCC(C)N=[N+]=[N-] c1(CCNC(C2CN(C)NC2=O)=O)cccc2nccnc12 N1(C(c2c(CC)cncc2)=O)CC2CC(C(=O)NC3CC(C)(OC)C3(C)C)(C2)C1 C1(CNC(C(COC)OC)=O)COCCN(C(=O)CCC2CCC(=O)C2)C1 c1(C(N2CC3CC(CNC(COCCCC)=O)C3C2)=O)nn(C)c2c1CSCC2 C1(C(C)NC(COC(CC)CC)=O)CCCN1C(=O)CCc1cnn(C)c1 C1(CCC(=O)N(C2CC3CC3C2)C)CCCN(C(=O)Cn2nccn2)C1 N1(C(COC2(C)CCCC2)=O)CCCC(CNC(=O)CCC2(C)CCC(=O)N2)C1 c1(OC)cc(Cl)c(C(=O)NC2CC2NC(=O)COCCF)cc1Cl Nc1ccc(C(N2CCN(C(C3CC3C(N)=O)=O)C3CCC23)=O)c(F)c1F CON(CCC(=O)N(C)C)C(=O)c1c[nH][nH]c1=N.C123CCC(CC1O2)C3 c1(CC)cc(C(=O)N(CCCNC(=O)COCCF)C2CC2)n[nH]1 c1(C(=O)NC(C(C)C)(C)CNC(=O)CC2CCC(=O)N2C)n[nH]c2c1CCC2 C(c1ccc(=N)[nH]c1C)=CC(N1CCC(N(C(CS(CC)(=O)=O)=O)C)C1)=O Cc1c(NCCc2ccc(Br)o2)ncnc1N1CCOCC(C)C1 CC1(C)CCCC(C(N2CCC2C(=O)NCc2cc(Cl)ccn2)=O)C1 C(=O)(CS(=O)(=O)CC1CCCO1)NC1C(NC(C2C(C)OC(=O)N2)=O)C1 Cc1nonc1CC(=O)NCCN(C(c1cscc1Cl)=O)CC1CC1 C=CCC(CC(C)C)C(=O)N1CCOCC(CO)C1.C12C3CC4C(C3)C14NC2=O c1(C(=O)NCC2CCN(C(C3CN(C)C(=O)C3)=O)C2)ccnc2c1cnn2C C(=O)(C1=NNC(=O)C1)NCC1C(NC(CC(C)N(C)C)=O)C1 CC(CN(C)C)CCC(=O)N1CCC(CCNC(c2csc(C(F)(F)F)c2)=O)C1 c1(OC)cc(C)c(Cl)cc1C(=O)NC1CCCC1NC(=O)Cn1cc(C#N)cn1 Cc1csc(=NCC(=O)NCCC2CCN(C(=O)C=C3CCC(C)C3)C2)[nH]1 C1(NC(=O)COc2ccc(Cl)cc2)CN(C(c2ccc([N+](=O)[O-])o2)=O)CCC1O C(=O)(C(CC1CC1)N(c1nccn1CC(F)(F)F)C)NC C1(CNC(C2CC3(CCO2)CC3)=O)CC(C(=O)N2CCCC(CCO)CC2)=NO1 c1(C(C(=O)NCC(C)(C)NC(c2nccc(C(F)F)n2)=O)(F)F)cccc(Cl)c1 CC(C)(CNC(C1CCCCO1)=O)CNC(=O)Cn1ccc(C(F)(F)F)n1 CON(C)C(=O)CN=C(NCC1CCCC(C)(C)C1)NC1CC1 c1(CC(N2CCCC(CN(C(CC(C)N(C)C)=O)C)C2)=O)nc([N+](=O)[O-])n[nH]1 C(C(C(=O)N1CCN(C(C)=O)C2CC12)C(C)(C)C)NC(C(CC)(C)C)=O C=CCC(CC=C)C(=O)N(C)CC1(O)CN(C(=O)Cn2cc(C#N)cn2)C1 c1(CCC(=O)NC2CCN(C(=O)Cc3cnsc3)CC2)c(F)cccc1Cl c1(C(N2CCCCC(C(=O)NC3(C)CC3)C2)=O)ccc2c(c1)CCN2C(C)(C)C C1(C(N(C2OCC(C)C2)C(=O)CN2CCOCC2C)=O)CCCCC1C c1(C(N2COC3CS(=O)(=O)CC23)=O)ccc2c(n1)CNCC2 N1(C(C)=O)CS(=O)(=O)CC1C(=O)NC(C)CCNC(C1SC2C=CC1CC2)=O C1(C(N2CCC(C(C)NC(c3[nH]cc(C(C)=O)c3)=O)C2)=O)Cc2ccccc2O1 C1(NC(C(C)=C(C)C)=O)CCSC12CN(C(=O)Cc1csc(Br)n1)C2 CC(C)CS(=O)(=O)CCC(=O)N(C)CC1(NC(=O)CC2CCOCC2)CC1 c1(CC)cc(C(=O)NCC2COC(CNC(=O)CSc3nnnn3C)C2)sc1C C1(C(N(C(C(=O)N(CC)Cc2cnn[nH]2)C)CC)=O)CC(F)CN1C C(=O)(C1=NOC(C)C1)N1C(C2(NC(c3c(CC)sc(=N)[nH]3)=O)CC2)CCCC1 Cc1c(C(=O)NC(C)CCNC(=O)CSC(C)C)csc1Br C=C1CCN(C(c2cccc(C)c2)=O)C(C(=O)N(C2CCCCC2)C)C1 C1(C(=O)Nc2cnc(C)s2)CC2(C1)CN(C(c1ccc(Cl)cc1I)=O)C2 C1(C(N(C)Cc2nnc(C)o2)=O)CCC(C)N1C(c1cn(CCO)nn1)=O CCC(C)C(O)C(=O)NCCCNC(c1ccnc(-n2cc(F)cn2)c1)=O C(CN=c1ccc(-c2nccs2)c[nH]1)=CCNC(=O)OC(C)(C)C c1(C(=O)NCC2(NC(C3(C#N)CC3)=O)CCOC2)ccc2n[nH]cc2c1 C(=O)(C(CCC)CCCS(C)(=O)=O)NC1C(NC(C2(C)CC(=C)C2)=O)CC1 C1(N(C(=O)Cn2ncn(C)c2=O)C)CCCN(C(=O)C(C)(C)O)CC1 c1(C(=O)NCC2CN(C(C=COCC)=O)CC23CCC3)cc2nc(C)ccc2o1 CC1CCCCC1C(N1CC(CCNC(c2nccnc2N)=O)C1)=O C(=O)(C(O)CC(F)F)NCC(CO)(CO)N(C(=O)COc1ccc(O)cc1)C c1(C(=O)NCC2CCN(C(c3c(C)nn[nH]3)=O)C2)cc2c(nn1)CCCO2 CC1(C)CC(C(=O)NCCC2(O)CCN(c3nnc(CO)s3)CC2)CCO1 Cc1c(C(N2CCCC(C(=O)NCc3ccco3)C2)=O)cccc1Cl c1(C(N2CCC(N(C(c3cc(-c4cccs4)[nH]n3)=O)CC)C2)=O)ccc(F)cc1 Nc1cc(C(F)(F)F)ccc1C(=O)NCC(O)CNC(C1CC1(F)F)=O Cc1cc2sc(C(=O)NCC3CC(F)CN3C(=O)CN3CC4CCC3C4)cc2s1 C1(O)(C(C)NC(=O)CCNC(=O)CO)CCN(C(=O)C(c2nc(C)cs2)C)C1 C12(NC(c3cnn(CC)n3)=O)CC1CN(C(=O)Cc1ccsc1Cl)C2 CC1CN(CC2(C)CCN(CC(c3cnn(C)c3)=O)CC2)C(C)CO1 N1(C(C(CC)Cc2ccc(N)cc2)=O)CC(NC(C2CC(=O)N2)=O)CC(F)C1 CC1(C#N)CCN(Cc2cnc(-c3ccccn3)nc2)C1.Cc1ccc(C)s1 C(CCN(C(=O)C(COC)OC)C)(C(C)(C)C)NC(C1(C(=O)NC)CC1)=O N1(C(CC(c2c(C)cccc2)C)=O)CCCC(NC(=O)Cc2ccns2)CC1 c1(NC(C2CCN(C(C(C)CCBr)=O)CC2)=O)cccc2sccc12 C1(C(=O)O)CC2C1CCN2CCc1cccc(F)c1.c1(C(C(C)C)N)cc(C)no1 CCC#CCN=c1[nH]c(=NCC(C(C)C)OCC)[nH]c2cc(C)ccc12 n1(CC)cc(Cl)c(C(=O)NC2CCN(C(C3CCC4CC34)=O)CC2)n1 N1(S(c2c(OC)cccn2)(=O)=O)CC2CCC1CN2C(=O)C(c1ccccc1)O C=CC1OCCC1C(=O)NCC1COC(CNC(c2csc(COC)c2)=O)C1 N1(C(c2cnc(C(C)O)s2)=O)CCC(NC(c2ccncc2)=O)C(O)C1 c1(N(C)C)ccc(CN=c2[nH]c(-c3ccc(Br)cc3F)cs2)cc1F C1(NC(=O)C#CC2CC2)CCCC12CN(C(c1ccnc(C3CCCC3)n1)=O)C2 c1(OC)ccc(C(=O)NC(C)CN2CCN(C(C3C4CCCC34)=O)CC2)c(F)n1 c1(C(=O)NC(C)CNC(=O)C=Cc2ccco2)nn(C)cc1C(=O)O c1(OC)cncc(C(=O)NCCC2CN(C(C3CC3C(F)F)=O)CCO2)n1 C(=O)(C1CCCc2nc[nH]c21)NC1CN(C(c2ccc(OC)cc2)=O)CC1OC Cc1cc(=NC2CCc3c(Br)cc(Cl)cc3C2)[nH]c(=NCCCOCC(C)C)[nH]1 c1(C(c2ccc(Cn3cc(Br)cn3)o2)=O)cc(Cl)cc([N+](=O)[O-])c1O CCCCCCC(=O)NCC(CC(F)(F)F)NC(=O)C(C)OC1CCCC1 c1(OCC(=O)NCC(CC)NC(c2coc(Cl)c2)=O)ccc(F)cc1Br c1(N(C)C)cccc(CN2CC(NC(C3(N4CCCC4)CCOCC3)=O)C2)c1 Cc1cccc(CN2CCC(C(N3CCCC3CC3CCNCC3)=O)C2)c1 C1(NC(C2C3(CC(NC(c4c(C(C)C)ocn4)=O)C3)C2)=O)CC2(C1)CC(C#N)C2 N#Cc1cc(S(=O)(=O)N2CCC3(CCSC3)C2)ccc1N1CC=CC(O)C1 C1(CNC(C2CCC(=C)CC2)=O)CCN(C(=O)CCC(=O)N(C)C)CC1O N#Cc1c(NC(c2csc(=NCc3cnc(O)nc3O)[nH]2)=O)cc(F)cc1F C1(C(N2C(C3(NC(COC)=O)CC3)CCC2)=O)CCN(C)C1=O N1(C(CCOC(C)C)=O)C2CCCC1CC(n1cc(-c3cnn(C)c3)nn1)C2 c1(CC(N2C(CN(C(C(C)C3CCCO3)=O)C3CC3)CCC2)=O)cc(O)nnc1O C1(C(=O)OC)CS(=O)(=O)CC1C1CC1.C(=O)(CS)NCCOCCOC.C1(=O)NCCN1 N1(CC(=C)C)CCN(S(=O)(=O)N2CCC3(CC2)OCCO3)CC1 c1(C(=O)NC(CNC(c2c(C(=O)OC)coc2)=O)(C)C(C)C)ccc(Cl)cc1C N(C(=NCCN1CCCCC1)NCC1CCSC1(C)C)C(C)CC(F)F C(=O)(C1=NNC(=O)C1)N1CC(NC(C(C)Oc2ccccc2Cl)=O)C1 c1(C(=O)NC23C(CN(C(C(C(C)C)(C)O)=O)C2)C3)ccc2nnc(S)n2c1 C1(CC(=O)N(C(CC)CNC(=O)CCc2nc(C)no2)CC)CCC(=O)O1 CC(C(=O)NC(C)(C)CCCCNC(c1cnc(Cl)[nH]1)=O)C(C)(C)C c1(CC(N2C(CNC(C3C(C)CCC3)=O)C3CCC2C3)=O)cn2c(n1)CCCC2 S(=O)(=O)(CC(=O)NCC1CCN1C(=O)C(C)OCCN(C)C)NC c1(C(N(C(C(=O)NCC(CC#C)(C)CO)(C)C2CC2)C)=O)ccc2c(c1)CCC2 CC1=C(C(=O)NC2CC3CCC2(NC(C2C=CCCC2)=O)C3)CCO1 C1(c2n(-c3c(C)cccc3)nc(-c3ccc(F)cc3)n2)CCCC2(CC2)C1 c1(C(=O)NCCCC(C)NC(C(C)(C)OCC)=O)cccnc1C(F)F N1(C(C2(C#N)CCOC2)=O)CC2(C1)CN(C(c1ccc(Br)s1)=O)C2 C1(NC(C(C)(C)NC(C=COC)=O)=O)CC2(CCN(C(=O)NC3CCCC3)C2)C1 N1(C(C2C3C(NC(c4[nH]c(=N)sc4)=O)C4C(C3)C42)=O)CCc2ccccc21 c1(Cn2c(C(C(CCCC)OCC)NCC3CC3)nnn2)cc(Cl)c(Cl)cc1Cl CCC(C)CCC(O)CC(=O)NC1CC2CN(C(=O)CC(C)CN(C)C)CC2C1 C1(NC(C(=O)NC(C)C)=O)CN(C(c2cc(F)c[nH]2)=O)CC1C N1(C(COCCCC#C)=O)CCCC(N2CCN(C(C3CCS3(=O)=O)=O)CC2)C1 C1(C(=O)NCC(CNC(C(n2c(C)ccn2)C)=O)(C)C)CCc2ccccc2O1 C=C1CC(C)(NC(c2coc(CNC(=O)C(C3CCC3)OC)n2)=O)C1 Cc1cccc(NC(c2ccc(CN3CCOCC3)c(F)c2)=O)c1[N+](=O)[O-] C1(C(=O)NC(COC(C)C)C(=O)NC2CCC(CO)C2)COCCO1 C1(C(=O)NCc2n(CC)nnc2C)CCC(C)(C)N(C(C2CCCC(=O)N2)=O)C1 N1(C(c2ccc(C(N)=O)cc2)C(=O)NCC=C)CCC2(C1)NC(=O)N(C)C2=O N1(C(C(CCSC)O)=O)CCC2C(CCN2C(=O)CSc2ccc(C#N)cc2)C1 C1(NC(CCC(=O)NCCC)=O)CCCCN(C(C2(C#N)CC(C)C2)=O)C1 C(C(C)(C)CC(=O)N1CC(O)(CO)C1)NC(c1cn(CC)nc1)=O O=C(C(O)CC(O)CO)NCC(c1ccco1)O N1(C(C2CCCN(C(Cc3ccn(CC)n3)=O)CC2)=O)CCC(O)C(C)(C)C1 c1(C(N2CCC(NC(CC(CC)C)=O)(CF)C2)=O)c(N)cc(Cl)cc1F C1(NC(=O)C(O)CCC(F)(F)F)CCCC(NC(c2csc(Br)n2)=O)C1 N1(C(c2cccc(C)c2C)=O)CCN(C(c2nccn2C)=O)C2CCCC12 N1(C(C2OCCN(C(C)=O)C2)=O)CCCCCC(NC(=O)Cc2n[nH]c(=N)s2)C1 N1(C(C(CSC)OC)=O)CCC(C(C)(C)C)(NC(=O)C(C)(CO)OC)C1 c1(C(N(C2CCN(C(=O)COCC(F)(F)F)C2)C)=O)cccc2nn(C)nc12 CCC(C)C(CC(=O)N1CC(CO)CC1(C)C)NC(c1cc(Cl)ns1)=O C1(C(N2CC3CCN(C(CCOC)=O)C3CC2)=O)Cc2ccccc2NC1=O c12cccc(c1)CNC(=O)C(C)NC(=O)NC2.c1(NC(N)=O)cc(Cl)ccn1 c1(CCC(=O)NC2CC(NC(=O)C(Cl)=CCl)C23CCC3)cc2ccccc2o1 C12(CNC(C(CC)F)=O)CC(NC(c3ccc(COC)cn3)=O)(CO1)C2 N1(C(CC(C)O)=O)CCC(O)(C(=O)NC(C)(C)C)C1.C(=O)(CCOCCF)N(C)C C#CCCC(C(=O)NC(CC(C)C)C(N)=O)NC(=O)CC12CCC(CC1)C2 C(=O)(CCCCCCNC(=O)CC1CCCCCC1)NC(C)Cc1cnc[nH]1 N1(C(c2[nH]cc(C(=O)OC)c2)=O)CCCC(C)(CNC(c2cnnn2C)=O)C1 C(=O)(C(c1ccoc1)NC(C1CCO1)=O)NCCOCCC N1(C(=O)NCc2ccn(CCF)n2)CC2CC1CS2=O C1(O)(c2cn(CCOC3CCN(C(c4cc(OCC)no4)=O)C3)nn2)CCOCC1 CCC(C)CCCCC(=O)N1CC2CCC(C1)N2C(C1OCCC1(C)C)=O CC(CC(C)NC(c1ncsc1C(F)(F)F)=O)NC(=O)CC(C)F C1(CC(=O)NCC2(O)CCN(C(c3cnc(O)c(Cl)c3)=O)C2)CCS(=O)(=O)CC1 N1(C(CC2CC(CC)C2)=O)CCn2ncc(CNC(C3CC(O)C(F)C3)=O)c2C1 C1(CNC(C2CN(CC)C2)=O)CCCC2(CN(C(c3cccc(Cl)c3)=O)C2)O1 C1(C(C)O)CCN(C(=O)C(=O)NCCCC2CCCN2)C1 c1(SC(C(=O)N(CCNC(=O)Cn2cnnc2)CC)C)nncn1C N1(Cc2nc(C)sc2)CCOC(CNC(=O)CCc2cnccn2)C1 N1(C(C=C(C)C(C)(C)C)=O)CCC(C2CC2)C1CNC(=O)CCCF.N1CSC1 c1(SCC(N2C(C(C)NC(=O)CNC=O)CCC2)=O)c(Cl)cccc1Cl c1(OC)cc(C(c2nnnn2C2CC2)Nc2ccc(O)c(Cl)c2)ccc1C#N C1(C(N(C2CCCC(C)(C)C2)C)=O)CNC(=O)CN1C(=O)CCc1nccs1 C1(CNC(Cc2cn(C)nc2Cl)=O)CCCCN(C(=O)C=CSc2nc[nH]n2)C1 O=C1CC(C(=O)NC(C(=O)NCC2CCCC(=O)N2)C2CCC2)=NN1 CN1CCc2nc(C(N3CCC4CN(C(c5cncc(F)c5)=O)CC34)=O)sc2C1 N1(C(C2CC(=C)C2)=O)CCOC2(CCCN(C(=O)C(c3cnn(C)c3)C)C2)C1 Cc1nc(C(N2CCC(NC(c3c[nH]c(Br)c3)=O)C(C)C2)=O)c(C)n1C1CC1 C(=O)(C(C)(C)CC(C)(C)C)N1CCC(CC(=O)NCc2cc(C)ns2)CC1 CC1N(C(C2(C(=O)NCC3CCCC4(CC4)C3)CCCO2)=O)CC(C)OC1(C)C c1(C(N2CC(OC3CN(Cc4c(SC)cccc4)C3)C2)=O)cc(F)ccc1C C1(C)(CNC(C(c2ccncc2)C)=O)CCCN1C(c1cc(C(F)F)no1)=O N1(Cc2ccc3c(c2)O3)CCS(=O)(=O)CC1CO.CCCCOC C1(CC#C)(C(=O)NC2CC2NC(=O)Cc2cc(C(F)(F)F)n[nH]2)CCCO1 c1(N(C(c2ccc(OC)c(CC)c2)C(=O)NCCC)C)c(Cl)cccc1[N+](=O)[O-] CCC1=C(C(=O)N2CCCC(NC(C3CN(N4CCCC4C)C3)=O)C2)CCCO1 c1(C(N2CCCC(CNC(CC3C=NN(C)C3=O)=O)C2)=O)nccc2[nH]ccc12 N1(C(CNC=O)=O)CCOC2(CCCN(C(c3cn(C4COC4)nn3)=O)C2)C1 C(=O)(N=c1cc(C)n(C)[nH]1)c1c(F)ncc(-c2ccc(OC)c(F)c2OC)c1 C1(C(=O)NCCCn2cc(-c3c(C)ocn3)nn2)CSCC(=O)N1 N#Cc1cccc(CNC(C2CCN(C(C3CC3c3nc[nH]n3)=O)CC2)=O)c1 c1(C(N2C(C(=O)Nc3cnc4ccccn34)CSCC2)=O)ccc2ocnc2c1 C1(C2(CN(C)CC3CCN(C(c4cnco4)=O)CC3)CC2)CCCNC(=O)C1 C1(Cn2ncc(C)c2)CCN(C(=O)Nc2cc(C)n(C)c2)CC1C Cc1cncc(C(=O)NC(C)CN(C)C(C2CCN(C)C2)=O)c1Cl C1(CC(=O)NCC(F)(F)F)CCCN1C(=O)CCC.C1(OC(=O)C2CC2)CCOC1 Cc1n[nH]c(C)c1S(=O)(=O)N1CCC1C(=O)NC1CCC12CNC2 C=CCC(CC=C)C(=O)NCC1(CNC(c2cnnc(C3CC3)c2)=O)CC12CCC2 Cc1c[nH]c(C(=O)NCC(F)CNC(c2ncncc2F)=O)c1C C(=O)(CS(=O)(=O)CCOC)NC(CC)CCC(=O)NCC(C)(O)COC c1(SC)cnn(C)c1C(=O)NCC(C)(C)CN(C(=O)CCOC1CCOC1)C CC#CCC1C(=O)N2CCN(C(C)C2)C(=O)C2CCCC(C2)C(=O)N1.OC.NC N1(C(C=CC)=O)CCN(C(c2ccc(C(C)=O)cc2)=O)C(c2ccncc2)C1 C12(C(N3C(C(=O)NC4CC(N5CCCC5)C4)COCC3)=O)CCCC1C2(F)F C1(C(=O)OCC)COCCN1C(=O)C(=O)N(C1CCOCC1C)C N1(C(CSC(C)C)=O)CCCC(C2CN(C(=O)CN3CCC(C)C3)C2)C1 C1(CCC)(NC(c2nnsc2C)=O)CCCN(C(c2[nH]c(C3CC3)nc2C)=O)C1 Cc1cc(C(=O)NC(C(=O)Nc2cc(CO)cc(C)c2)C(C)C)nc(C)c1 N1(C(Cc2cc(C)n(C)n2)=O)CCOCCC1C(N1CCC(N(C)C)C(C)C1)=O N1(C(C(CC#C)C)=O)CC2(C1)CN(C(=O)C(C)OCC(C)C)C2 c1(C(C)=O)cc(C(N2CCC(C)(CNC(=O)Cn3nccn3)CC2)=O)cc(C)c1 CC(C)CC(C)CC(=O)N1CC(CNC(c2cc3cnccc3o2)=O)C(O)C1 CCCCC(=O)NC(CNC(C1(CNC(=O)OC(C)(C)C)CCCC1)=O)CC CCC(CC)C(C(=O)N1CC(O)(C(C)NC(C2CC(CF)C2)=O)C1)OC C1(C(=O)NCCCOC)CC(OC)CN1C(c1cn(-c2ccccc2Cl)nn1)=O CC1OCCC1(F)C(=O)NCC1(NC(=O)CC2(C)CCCC2)CC1 C1(n2cc(C3(NC(Cc4nc(CC)sc4)=O)CCC3)nn2)CC2CCC1(C(=O)O)C2 N1(C(C2C(OCC)C2C)=O)CCC2(COC(CNC(C3CCCOC3C)=O)C2)C1 N1(C(CCOC(C)C)=O)CCN(C(C2(n3cncn3)CC2)=O)C2CCCC2(C)C1 c1(-c2nc(-c3ncc(SC)cc3C)on2)cccc2c1CN(c1ccccc1)C2 N1(C(CC(CC)CC)=O)CCN(C(c2scc(C)c2C)=O)C2CCCC12 N1(C(c2cc(CCC)on2)=O)CCN(C(c2cc3occc3s2)=O)CC1CF C1(CC)CC(CC(=O)NC(C2CCN(C(=O)C(Br)=C(C)C)CC2)C)CCO1 c1(OC)ccc(CN=C(NCc2ccc[nH]2)NCC2CCCCC2)cc1F C(=O)(C(O)CC(F)(F)F)N1CC(NC(c2ncc(F)cn2)=O)C(C(F)F)C1 C(CCC(=O)N1CCC1C(=O)NCC(=O)NCCOC)OCC C1(NC(C(C)OCOC)=O)CN(C(=O)CSc2cccc(C)c2)C(C)(C)C1 C(=O)(C(C)(C)c1ccccn1)NCC(CNC(C1(CC#C)CCC1)=O)OC c1(N(c2ncnc(CC)c2F)CC2CCC(N)C2)ncc(Cl)cc1[N+](=O)[O-] C1(C(=O)N2CC(n3cc(-c4csnn4)nn3)CO2)CCc2ccccc2O1 C#CCC(CC#C)C(=O)N(CCC)CCNC(c1nc2ncccn2n1)=O c1(C(N2CCC(NC(c3c(OC)cccc3I)=O)C2)=O)ccc(C#N)cc1F CC1(C)CN(C(C2(C)CCC2)=O)CC1C(=O)NCCC1CCOCC1 Cc1ccc(Cl)c(N)c1C(=O)NC1CCCC1CNC(C1CC(n2cccn2)C1)=O c1(C(=O)NCC2N(C(CC(C)c3cnn(C)c3)=O)CC=C2)ncccc1O C(=O)(C1=C(Cl)CCCC1)NC1C(NC(c2ncc(C)c(C)c2)=O)CCCC1 C1(NC(C(CC)(C)CC)=O)CCN(C(C2(OC)CCC2)=O)CCC1CO C1(CCNC(C(C)C2CCC2)=O)CN(C(=O)Cc2cc(C3CC3)no2)CC1C N12CC(CCC13CC3)NC(=O)C2.c1(CC)cccc(F)c1C(=O)OCC N1(C(c2ccc(CC)cc2)=O)CCCC2(CCN2C(=O)CN2CCSCC2)C1 N1(C(CC2(C=C)CCC2)=O)CCCN(C(=O)C(C)c2ccco2)CC1C(C)C N1(C(CCCCC)=O)CCC2(COC(CNC(c3snc4ccccc34)=O)C2)C1 N1(C(C2CC(C)(NC(c3nc(CC)sc3)=O)C2)=O)CC(C2=NOC(C)C2)C1 Cc1ccn(C)c1C(=O)NCCCN(C(=O)C(N1CCCC(O)C1)C)CCO C1(CC(=O)NCCC2N(C(CCC(=O)N(C)C)=O)CCOC2)CCCC(C)(C)O1 c1(NC(c2c(Cl)n[nH]c2C)c2n(CCCCCC)nnn2)cc(NC)cc(F)c1 Cn1cc(C(N2CC(CSC3CC(=O)NC3=O)CCC2=O)=O)c2cccnc12 c1(C(N(CC#C)C)=O)coc(CNC(=O)C(C)C#N)n1 N1(C(=O)CCF)CCCC1C#CC(=O)OC(c1ccc2c(c1)COCO2)CC(N)=O N1(C(C2CC(C)C2)=O)CC(CCNC(=O)CN2CC(=O)NC2=O)C(C)C1 c1(C(N2CC(C(=O)NC3CC(C)CC(C)C3)C(C)(C)C2)=O)cnn2cccc2c1 c1(C(=O)NCC2(NC(C3CC(CCC)C3)=O)CCCC2)cncc(Br)c1 CC1CN(C(=O)Cn2cc(C3CC3)cn2)CCC1C(N1CCC(O)(CO)C1)=O C1(NC(=O)CCn2cncn2)CN(C(C23CC2C3)=O)C2(CCOCC2)C1 CC(CCCN=c1[nH]c(=NCc2ccsc2)[nH]c2ccsc12)c1ccccc1 [N-]=[N+]=NC1CN(C(C2COCCO2)=O)CC1NC(c1cccc2c1NCC2)=O C1(n2c(-c3ccoc3Cl)nc(C(C)C)n2)CCCS(=O)(=O)C1 C(=O)(C(C(C)C)N(C)C)NC(C1CCN(C(c2c(CC)scc2)=O)C1)(C)C C(=O)(C1CCC(=O)c2cccn21)N1CC(NC(c2c(SC)cccc2)=O)(CO)C1 Cc1ccc(C(=O)NCCC(C)NC(C2CCN(C)S2(=O)=O)=O)c2c1CCC2 C1(CC(N2CCCC(C(=O)NC(C)CN3CCCC3=O)C2)=O)CCC=CCCC1 C1(NC(c2cn(CC)nc2C)=O)CN(C(=O)CSC(F)(F)F)C2(CCOCC2)C1 c1(C(N2CC(C3CC3)(C(N3CCC34CC(CO)C4)=O)C2)=O)cccc2c1CCC2 Cn1nc(C(N2CC3C(NC(c4cccnc4O)=O)C3C2)=O)c2c1CCSC2 c1(C(N2CCC(N(C)C(c3coc(C4CCOCC4)n3)=O)C2)=O)ncc(F)cn1 C1(NC(C2C3(CC(C)(C)C3)C2)=O)CN(C(=O)CCCC#N)CC2(CC2)C1 N1(C(C2C(C)(C)C2(F)F)=O)CCN(C(C2COCCC2(F)F)=O)CC12CCC2 N1(C(c2c(CC)cncc2)=O)CC2CC(C)N(C(=O)C(C)N(C)C)C2C1 n1(C(C)C)cnnc1CC(=O)NC1CC(CNC(c2ccccn2)=O)C1 N1(C(C(OC)OC)=O)CC(O)(CNC(C2CCC2(C)C)=O)C1 c1(NCc2c(C)ccs2)cc(NC(c2nnc(O)o2)C)ncn1 C1(NC(c2cnc(CC)s2)=O)CN(C(=O)C(N2CCCC(C)C2)=O)CC1C c1(CC(C(N2C(C)CC2CO)=O)C)ccc(O)cc1 C(=O)(C1CCCc2ccnn21)N1C(CN(C(C(=O)NC(C)C)=O)C2CC2)CCC1 CCC(C)(CC)C(=O)NCCCCCNC(=O)C(c1cc(F)cc(F)c1)O C123COCC1CN(C2)C3=O.c1(CC)nc(CNC(c2ccccc2)=O)cs1 C1(C(C(=O)NC(CNC(C2(OC)CC2)=O)(C)C)C)CCCCCC1 CCC(CC(F)F)C(=O)N(C1CCN(C(=O)CC2CCS(=O)(=O)CC2)C1)C c1(C(=O)NC2C(C)COCC2)cc(F)ncc1NC(c1cc(=O)ccn1C)=O c1(N(C)CC2N(C(CN3CC(=O)N(C)C3=O)=O)CCCC2)cc(O)nc(=O)n1C S(=O)(=O)(c1ccc(NCCOc2ccc(F)cc2)c(C#N)c1)NC(CCC)CO C(=O)(CCCC(=O)N(C)C)N(CCCC(=O)Nc1ccc(OC)cc1)C1CC1 CCC(C(=O)NOCC(=O)NC1(CF)CCC1)n1cccn1 C1(CC)Oc2cc(Sc3ccc(CN4CCC4(C)C(C)C)cc3)ccc2NC1=O CCC1=C(C(=O)N2CCCCC(C(=O)NCc3cnn(C)c3C)C2)CCCO1 Cc1cccc(C(F)(F)C(N2CCC(CCNC(C3CCOC3C)=O)CC2)=O)n1 CC1(C)CCC1(O)C(=O)NC(CCO)C(F)F C(=O)(C1=NNC(=O)C1)N(CCNC(CCc1nc(C)c(C)o1)=O)C(C)C N1(C(CC2(C)CC2)=O)CCN(C(=O)C#CC2CCOC2)C2(CCC2)C1 C12(NC(C3CCC3)=O)CCC1CN(C(c1ccc(Cl)s1)=O)C2 c1(C(=O)NCC(C)(C)NC(C2CC23CCOCC3)=O)cc2c(o1)CCCC2 C12(CNC(C(C)SC)=O)CCC(CC1NC(c1ccc(Br)cn1)=O)C2 CC1CCC(C(N2CC3CC(C)C3C2)=O)CN1C(=O)C=C1CCC(C)CC1 C(=O)(CCC(=O)C(C)(C)C)N1CC(CC(=O)NC2CC(C)(C)OC2=O)(OC)C1 C1(CC(=O)N(CCN(C(CCC(C)c2ccccc2)=O)C)C)CCC(=O)NC1=O c1(C2ON=C(C)C2)cccc(-c2ccc(OCc3cccc(C)c3)cc2)c1 C(=O)(C(F)(F)CCn1cccn1)NC(C1CCN(C(C=NOC)=O)CC1)C c1(C(N(CC(C)CNC(c2cnn(C)c2Br)=O)C)=O)nnc(O)cc1O c1(CNC(C)CCc2ccc(Cl)cc2)c[nH]c2cccc(Br)c12 CC1CC(NC(c2cn(C(F)F)cn2)=O)CN1C(=O)CN(c1ccccc1)C N1(C(c2cc(=O)cc[nH]2)=O)CCOCC2(COCCN2C(=O)CCC2CCC2)C1 C(=O)(C#CC1CCOCC1)N(C1CCOC(C)C1)CC(NOC(C)C)=O C1(C(C(=O)NC2(C)CC2)N(C)CCn2ccccc2=O)C2CC=CCC12 C=CCN(OC)C(=O)CC1C(C)CCCN1C(=O)C1=C(CC)OCCC1 CCCCCCCCC(F)C(=O)NCC(C)(CO)NC(=O)Cc1cccc(C)c1 c1(-c2cn(CCCCNC(C3(C)CS(=O)(=O)C3)=O)nn2)ccc(Cl)c(F)c1 C1(C)(NC(c2ccc(CC)s2)=O)CCN(C(C2CCN(C(=O)OC)CC2)=O)C1 N1(C(c2c(OC)scc2)=O)CCCC(NC(c2cc(NC(C)=O)ccc2C)=O)CC1 n1(CCC)cc(C(=O)NCC(C)(O)CNC(=O)C(C)n2cnnn2)c(C)n1 C(=O)(CC#CC)N(CC(=O)NC(CC=C)C1CC1)CC CCCCC(C)C(=O)NCc1cc(O)nc(CNC(C2CCC2(F)F)=O)n1 c1(C(=O)NC2CC(CCNC(C(C(=O)OC)C)=O)C2)ccc(C)c2ccccc12 c1(CC)cccc(C(=O)NCC2CC(O)CN2C(=O)COCCCF)c1 Cc1ccsc1CNC(=O)CC1(CNC(=O)CC2(O)CCC2)CC1 C(=O)(CC1=CCCC1)N1C(C2(NC(C3CC4CCC3C4)=O)CC2)CCC1 C12(C(=O)NC3CCN(C(C(CC)N(C)C)=O)CC3F)CCC(CC1)C(C)O2 C(C1c2ccccc2CCN1C(=O)CN(C)C)NC(c1c(CCC)nns1)=O n1(CC)nccc1C=CC(=O)NCCC(C)(C)NC(c1cnn(C2CC2)c1Cl)=O C1(CC)(CC)CC(NC(=O)C(O)C2CCC2)CN1C(=O)CCc1cnn(C)c1 c1(C(=O)NCC(=O)NCCNC(C2CC2(Cl)Cl)=O)ccc2cc[nH]c2n1 C1(NC(c2coc(C3CCCCC3)n2)=O)CCN(C(=O)C(F)=C2CCC2)CC1F c1(OCC(=O)NC(C2CN(C(=O)CN3CCC3)C2)C)cccc(C(F)(F)F)c1 c1(C(N(C2CCCC(NC(CCCOC)=O)C2)C)=O)ccn2ccsc12 N1(C(c2nc(CC)sc2)=O)CCN(C(=O)CCOc2ccc(Cl)c(F)c2)C2CC12 c1(OCC=C)cccc(S(=O)(=O)NC2CCC(NC(=O)OC(C)(C)C)C2)c1 c1(C(=O)NCC(CC)NC(c2nc(C)nn2C)=O)cc(C(N)=O)cc([N+](=O)[O-])c1 C1(NC(c2nn(CC)nc2C)=O)CCN(C(C2CC2C)=O)CC1C Cc1ccc(OCCCNC(=O)C(C)n2cccn2)cc1C C1(N(C(C(C2CCN(C(Cc3cc(C)on3)=O)C2)F)=O)C)CCCC(C)(C)C1 N1(C(c2scc(CNC(CCSCCC)=O)c2)=O)CCOCCC1C C#CCCCC(C)C(=O)N1CCC(C(N2CCC(OC(C)C)C2)=O)CC1 C1(CNC(C2(C)CCC(C)C2)=O)CC2(C1)CN(C(C13CCC(CC1)O3)=O)C2 c1(C2(C)C(C(N3CC(N4CCN(C(CC#N)=O)CC4)C3)=O)C2)cc(F)ccc1F N1(C(c2n(C)cc(Cl)c2)=O)CC(C)(C)OCC1CNC(=O)C(F)(F)c1nccs1 C12(CC(N3CC(C)C(NC(C4CCCCC(=O)N4)=O)C3)=O)CCCN1CCC2 c1(C(CNC(c2n(CC)nnc2C)=O)NC(=O)C(C)C)ccc(F)cc1F C1(NC(C(=Cc2ccccn2)C)=O)CCCCN(C(=O)CN2CCOCC2C)C1 c1(C(N2CC3C(C(=O)Nc4onc(C)c4C#N)(C3)C2)=O)ccc2ncncc2c1 CCC(CC(=O)N1CCCCC1CC(N1CC(CF)(CO)C1)=O)C(C)C N(C(=NCCCCC(F)(F)F)NCC(=O)N(C)C)Cc1ccc(SCC)cc1 c1(C(=O)NCC2N(C(C(CC)OC)=O)CC(CO)C2)cc(C(N)=O)ccc1OC C=C(C)CCCC(=O)NCCC1CCC(NC(=O)C=Cc2cscn2)C1 O=C(C1=CCCCCC1)NCC1CCN1C(C12C=CC(CC1)C2)=O CC(F)CN=c1[nH]c(N2CCCc3cnn(C)c3C2)nc2cccc(F)c12 c1(CCN2CC(C(N3CCCC(O)C3)=O)C2)nccc(F)c1Cl C#CCC(CC(F)F)C(=O)N1CCCC(C(C)C(N2CCN(C3CC3)CC2)=O)C1 CC(C(=O)NCC(CNC(c1ccnc(-n2cccc2)c1)=O)CO)C(C)(F)F Cc1ccc2[nH]c(C)c(C(N3CCC(C4CCCN(C(=O)CCF)C4)C3)=O)c2c1 c1(SC)cc(C(=O)NCCc2n[nH]cc2C(=O)N(C)CC2(CC(C)C)CC2)co1 C1(CCC(=O)N(C2(C(=O)NCC(C)N(C)C)CCC2)C2CC2)CCCCO1 C(=O)(CC(C)CC(=O)N1Cc2occ(C(=O)N(C3CCNC3=O)C)c2C1)OC c1(C(=O)NC(C)CC(C)NC(=O)C(C)C#N)ncc([N+](=O)[O-])n1C C1(CNC(c2n(C)ncc2C2CCC2)=O)CCN(C(c2cnc[nH]2)=O)C12CCC2 c1(NC(c2nnnn2C(C)CC)CCOCC=C)ccnc(C)c1 c1(CC)[nH]c(C(=O)NC2CN(C(C3CCCS3)=O)C(C)(C)C2)c(C)c1C(=O)NC c1(OC)ccc(C(=O)NCC2CN(C(=O)CCC(C)(F)F)CC2O)cc1N c1(C(=O)NCCN2CCN(C(CCCCC=C)=O)CC2)cccc2ncc(Br)cc12 N1(C(c2c(CC)nco2)=O)CCC(C)C1CNC(=O)CC(c1ccc(F)cc1)C C1(OC)CC2CC(NC(=O)CC(CNC(c3cc(C)cc(C)n3)=O)OC)CC12 S(=O)(=O)(c1cc2c(cc1F)NC(=O)CO2)NCCC1(C)CCOCC1 C1(=O)C2=NOC3(CCN(C3)CN1)C2.c1(C(C)C)c[nH]c2cc(F)ccc12 C1(C(=O)NCC(CC(=O)N2CCOCC2C(C)C)OC)CCOC(=O)CC1 C(c1c[nH]c(=N)c(C)c1)=CC(N1C2C(NC(CCCC)=O)CC(C2)C1)=O N1(N2CCC3(CC3)C2)CC(CO)C(C2CC2)C1.CC(C)(C)OC=O c1(C(N(CCOC)CCNC(C23CC(C)C2C3)=O)=O)cnc2[nH]cncc1-2 c1(OC)ccc(C(=O)NCC#CCOC2CCC2)nc1N.OC Cc1cc(Br)c(C(=O)NC2CC(C)CN(C(=O)CC3CC3)C2)cc1F c1(C(=O)NC2CC(C)(COC)N(C(=O)C(C)=C3CC3)C2)cc(C)[nH]c(=NC)n1 C1(NC(c2nnnn2C)(CSCC)C)C=CCCCC1 C(C(C)(C)CNC(c1cc(C2CC2)sn1)=O)N(C)C(C1CCS1(=O)=O)=O c1(NC(CNC(=O)NC2CCCO2)CO)cn(CCF)nn1 c1(CNC(N2CC(OC)C2)=O)ncc(OC2CC2c2ccco2)c(=N)[nH]1 CS(=O)(=O)c1ccccc1C(N1CCC1C(=O)Nc1cccc(C2CC2)n1)=O C1(C(=O)NCC(N2CCN(C(c3cnc(C)nc3)=O)CC2)=O)CC(C)CC(C)C1 N1(C(=O)NCc2nc(CCC)on2)CCC2(CCC2O)CC1 c1(CNC(C2C(C(C)C)CCC2)=O)ccc(CNC(C2(C)CCCS2)=O)cc1 C1(C(N(C2CCN(C(C3(CF)COC3)=O)CC2)CC)=O)CCC(=O)N(C(C)C)C1 c1(C(=O)NCC2(F)CC(NC(CN(C)CC)=O)C2)cccc(Cl)c1C(C)=O.C CN1CCN(C(=NCc2ccc(CO)s2)NC2COCc3ccccc3C2)CC1=O C1(C(=O)NCC2CCC(CNC(=O)C3=CCCC3)CC2)CCc2nccn2C1 N1(C(C(=O)N(C)C)=O)C2CCC1CC(F)(CNC(C1CCn3nnnc3C1)=O)C2 c1(CC(C)NC(=O)CC2CCCN2C(=O)CCCF)ccn(C)n1 N1(C(C2C(C)CC2)=O)CC2CC(NC(c3nc(C(F)(F)F)cn3C)=O)C1C2 N12CCC(C(=O)O)(C1)NCC2=O.c1(CC)nc(C(C)(C)C)no1 CC(CC(=O)NCC1CCCC1NC(c1ccc(CN(C)C)s1)=O)n1cccc1 CCC(C)C(O)CC(=O)N1CCC(C)CC1C(=O)NCCCC1CCC1 c1(-c2nc(CNC(CC=C)C)on2)c(N)cc(CC)cc1F C12(NC(C#CC(C)(C)C)=O)CN(C(c3cc(F)ccc3F)=O)CC1CS(=O)(=O)C2 N1(CC(=O)Nc2ccc(C(N)=O)cc2)CCC2(CC1)CC2c1nn[nH]n1 C(c1ccccc1)=CC(C)C(=O)NCC1(CNC(c2cc(Cl)c(Cl)s2)=O)CC1 C(CC(C(=O)NCCS(N)(=O)=O)NC(=O)C(C)CC)SC C1(N(C(C(CNC(c2c(CC)c[nH]c2)=O)N(C)C)=O)C)CC2CCC1CC2 C1(CC)(NC(c2cccc(C)c2Cl)=O)CCN(C(C2CSC(C)=N2)=O)CC1 c1(C(=O)NCC(N2C(C(C)(C)CNC(=O)C(O)CF)CCC2)=O)ncc(Cl)cn1 CCC(C(=O)NCCN(C)Cc1cc(C(=O)NC2CCC2)n[nH]1)OC C(=O)(C1CCc2c[nH]nc21)NC1CCC(NC(C=C(CC)C)=O)C1 Cn1ncc([N+](=O)[O-])c1C(=O)NCC(O)CCNC(=O)CCOCC(C)(C)C c1(C(=O)NCC(C)N(C(=O)C(C)O)C)cc(C2CC2)ccn1 c1(C(=O)NCC2CC(O)CN2C(=O)C=CBr)cccnc1Cl N1(C(C(C)(C)C(N)=O)=O)CCC2(CCC2)C(NC(C23CCOC2CCOC3)=O)C1 C(=O)(CC(CCCC)NC(=O)CCC(C)SC)N(C1CCCCCC1)CC#C CC1(C)CN(C(c2ccnc(CNC(C3CCC3(F)F)=O)c2)=O)C2CCCC12 C(C(COC)CC(=O)NC1CCCCC1CNC(=O)C(c1cnn(C)c1)=O)OC C1(NC(CC2CCCN(C)C2)=O)CN(C(=O)CC2CC3(CC3)C2)CC2(CCC2)C1 Cc1ncc(C(N2CCC(CCNC(=O)C(n3ccc(C4CC4)n3)C)C2)=O)o1 N1(C(C2(C)CC=C(C)CC2)=O)CC=C(CCNC(C2CCC23CCC3)=O)CC1 C1(NC(C(C)(C)NC(=O)NCCC)=O)CN(C(C2CC2(Cl)Cl)=O)CC1O.C1CO1.OC C1(CNC(C2CC23CC3)=O)CN(C(=O)Cc2ccc(Cl)s2)CC12CC2 Cc1oc(C(F)(F)F)nc1C(=O)N(C1CCCN(C(=O)C(F)CC2CCC2)C1)C N1(C(c2ccc(CC)nc2)=O)CC2CC(NC(C3(C(N)=O)CC3)=O)C2C1 Cc1nn(C)c(=O)c(C(=O)NC2CN(C(=O)C=CCF)CC3(CCC3)C2)c1C N1(C(C(=O)N(C(C(N)=O)C2CCC2)CCC2CCCC2O)=O)CC2(C1)CC2(F)F C1CS(=O)(=O)C2CN(C(CCCCN)=O)CC12.c1nccc(C(F)F)n1 C(=O)(CCCC(=O)N1CC(n2cc(CS(=O)(=O)CC)nn2)CO1)C1C(CC)C1 C1(CNC(C(CC)C)=O)C(C2CC2)CCN1C(c1ccc(Br)cc1)=O c1(C(N2CC(O)(CCNC(C(C)OCCN(C)C)=O)C2)=O)ccc2ccsc2c1 C1(NC(c2sc(C)c(O)n2)=O)CC2(C1)CC(CNC(=O)C(C)OCCC(C)C)C2 N1(C(c2nc(N(C)C)oc2)=O)CCCC(C2CN(C(C3(F)CCC3)=O)C2)C1 N1(C(CCOC)=O)CCN(C2CCCN(C(c3cc(C(F)F)[nH]n3)=O)C2)CC1 C(CCCCC(=O)NC1CC(NC(N)=O)C1)N(C(C(CCOC)C)=O)C c1(C(=O)NC2CCC(CNC(CC3(OC)CC3)=O)C2)ccc2c(c1)CCCO2 N1(C(C2CN(C(C(CCCC)O)=O)CC2CC)=O)C(CO)CCC12CCC2 CC1CN(C(C2(CC(C)(C)C)CC2)=O)CC1N=c1ccnc(C(C)(C)C)[nH]1 C1(C(=O)NCc2n(C(C)C)ccn2)CC=CCN1C(=O)CCN(C)C C1(NC(c2c(C)scc2)=O)COC2(CCCN(C(c3cnnc(O)c3)=O)C2)C1 c1(OCC)cc(CN2CC(C)(CNC(=O)NC(C)C)C2)c(Br)cc1O N1(C(=O)NCc2ccc(OC)cc2Br)CC2CN(c3ccc(C)c(C)c3)CC2C1 Cc1ccn2cc(C(=O)NC3(CNC(C4CC45CCCC5)=O)CCCC3)nc2c1 c1(C(=O)NCCC2(OC)CCC2)cc(CNC(=O)CC2CCCCC2)[nH]n1 CC1=NOC(C)(C(=O)NC2CCC(F)(CNC(C3CN(S(=O)(=O)CC)C3)=O)C2)C1 C12(C(=O)NC3CCN(C(C45CC(CC(C)C)(C4)C5)=O)C3C)CCCCC1C2(F)F c1(C(=O)NCC2C(NC(C=C(COC)C)=O)COC2)cc2sc(Cl)cc2[nH]1 C1(NC(C2(OC)CCCOC2)=O)CN(C(=O)CCCCC(N)=O)CC2(CC2)C1 C1(NC(=O)CC(F)(F)Cl)CN(C(=O)Cc2ccc(F)c(Cl)c2)CCC1CO CCC(CC)C(C)C(=O)NC1CCCC1Cc1cn(CCOC2CCOC2)nn1 c1(C(=O)NCC2C3CN(C(C(C)OCCC=C)=O)C(C3)C2)ccc(F)c(O)c1F CC#CCC(CO)NC(=O)CCC1(C)CN(C(C2CCNC(=O)C2)=O)C1 c1(-c2cn(C3C(c4ccc(C)cc4)CCC3)nn2)c[nH]c(C)cc1=O C1(N(C(c2ccc(OCC(F)F)cc2)C(=O)NC)C)CCCC(C)C1C O=C(CCCS)NC1(CNC(C2(CCC3CC3)CC2)=O)CC1.C1(S)CCCCC1 Cc1n[nH]c(C)c1CC(C)C(=O)N(CC(O)CN(C(=O)Cc1cn[nH]c1)C)C c1(C(=O)NC2CC(F)(CNC(CS(=O)(=O)NC)=O)C2)ccc(O)c2ccccc12 C12(CNC(C3(C)CCN(C(CCOCCOC)=O)C3)=O)CC1CCC2(F)F c1(NC(=O)NC(Cc2nccc(C(F)(F)F)n2)C(F)(F)F)ccc([N+](=O)[O-])nc1 Cc1c(NC(C2(C)CCN2Cc2cccnc2O)=O)cnc(Cl)c1Br CC1=C(C(=O)N2CC(CNC(C3CCCC(C)CC3)=O)C(C)C2)CCC1 c1(C2(C)C(N(C)C(c3cn(C4CCOC4)nn3)=O)C2)ccccc1F C1(C(N2CC(CNC(c3c(C)ncs3)=O)OCCC2)=O)CCn2c(O)nnc2C1 C1(NC(CSc2ccc(NC(CC)=O)cc2)=O)COCCN(C(=O)C=CBr)C1 C1(C(=O)N)CC2CC(C1)N(C(=O)COC1CCCC1)C2.O=C(CCCC(F)F)N Cc1ccc(C(=O)CNC(=O)CNc2cccs2)nc1 S(=O)(=O)(c1ccccc1Cl)NC(C(C)O)C(=O)OC(c1ccccc1)CF c1(C(N2CCCC(C)(NC(=O)C(F)CC3CCCC3)C2)=O)ccc2occc2c1 CC1CCC(CCNC(=O)NC2(C)CS(=O)C2)O1 C(=O)(CC1=NN(C)C(=O)C1)N1CCC(C)(CC(=O)N(CCC)CCN(C)C)C1 N1(C(c2c(C)ocn2)=O)CC2C(NC(C3CCCN3c3ncccn3)=O)C2C1 CC(C)(C(=O)NCC1C=CCN1C(=O)CCCNS(C)(=O)=O)C1CCCCO1 Cc1c(C(=O)NCCN(C(=O)C(F)=CC2CC2)C)cnn1CC(C)C N1(C(C2(C=C)CCOCC2)=O)CC2CCC(NC(C3CCN3CC)=O)(C2)C1 C(=O)(C1=CC2CCCC12)N1CCCCC(NC(c2ccc(C(C)C)nc2)=O)C1 C1(NC(C2C(OCC)C2)=O)CCC(NC(c2cnccc2C(C)(C)C)=O)CC1 C(=O)(C1=NOC2(CCC2)C1)NCCCCCCN(C(CC(C=C)CCC)=O)C N1(C(c2c(C)snn2)=O)CC2CC2C1CNC(=O)CC1CCCCC1 C1(NC(c2c(C(CC)(F)F)cccc2)=O)CCc2cnn(C)c2C1 C12(CNC(C=CC(=O)OCC)=O)CCCC1CN(C(=O)CC1CCCS1(=O)=O)C2 C(C)(C)(CCCNC(c1ccccc1N(C)C)=O)NC(c1ccc(C(C)=O)o1)=O CC1(C)CC(NC(c2ccoc2C2CC2)=O)CN(C(C2CC2(C)Br)=O)C1 C1(CCC(=O)NCC2(C(N)=O)CN(C(=O)Cn3ccsc3=N)C2)CCCCO1 C1(CC(=O)NCCCC2(C)CC2)CCC2(CCN(C(=O)OC(C)(C)C)C2)C1 N1(C(c2occ(C)c2C)=O)CC(NC(=O)C(c2cc(F)cc(F)c2)C)C(C)(C)C1 N1(C(C#CC(C)C)=O)CC(NC(c2cccc(-c3nn[nH]n3)c2N)=O)C2(CC2)C1 C1(CNC(C2CCC=CCCC2)=O)CCCN(C(=O)Cc2cnoc2)CC1 C(CCCC(=O)NC(C1(C(=O)NC(CC2CC2)C(=O)OC)CC1)C)OC C1(CC(N2CCC(n3cc(CN(C(C)C)CCO)nn3)C2)=O)CC2(CCC2)C1 c1(N2CCC(C=C)CC2)nc(=NCc2cc(C)ccn2)[nH]c2c1CCC2 C1(CC(=O)NC2CC23CCC3)CN(C(c2cccc(C3CC3)c2)=O)CCO1 N1(CC(=O)NCC2(CNC(c3ccn(C)c3)=O)CC2)CCCC(C(N)=O)C1 c1(C(N2CCCCC(NC(C(C)C(C)(C)C)=O)C2)=O)cccc2cnccc12 Cc1cc(=NC(C)c2ncc(C)cn2)[nH]c(=NCCC(Cl)=C(Cl)Cl)[nH]1 c12ccc(O)c(c1)OCC(=O)N(CCC)CC(=O)N2.C1(COC)CCOC1 N1(C(c2ccc(CS(C)=O)cc2)=O)CCC2(COC(CNC(=O)CNC=O)C2)C1 N1(C(CCN(CC)CC)=O)CCCC(N(C(=O)C=Cc2nc(C)co2)C)CC1 CCCCC(CC(=O)NC1(c2ccccc2C)CC1)NC(=O)CNS(N)(=O)=O N1(C(c2ccnnc2)=O)CCC2C1CCN2C(c1occc1Br)=O c1(C(=O)NCCCOCCNC(C2(C)CC(=C)C2)=O)ccnc(C(C)C)n1 C1(NC(c2ccn(CCCC)n2)=O)CCC12CN(C(=O)Cc1ccn(CC)n1)C2 C1(C(=O)NCCCCCCNC(c2cncnc2)=O)CCc2nnc(O)n2C1 C1(C(=O)NC(C2(O)CN(C(c3cn(CC)nn3)=O)C2)C)CC2CCCC12 C1(CC(=O)NCC(=O)NC2CC2)CCN(C(=O)CNC2CCSC2)C1 N1(C(C2CN(C(c3c(C)csc3)=O)CC2C)=O)CC2(C1)OC(=O)NC2C N#CC1CCCCC1NC(C1C2CC2CN1C(c1cccc(F)c1F)=O)=O C1(NC(Cc2nc(C)[nH]n2)=O)CC(CNC(=O)CCSc2nnnn2C)C(O)C1 CC(C)C(O)C(C)(C)C(=O)NCC(C)(C)OCCNC(=O)C(CO)N(C)C N1(C(C(CC)OC)=O)CCCC(F)(CNC(c2ccc(OC)nc2Cl)=O)C1 c1(CC)ccc(C(=O)NCCOCCNC(C2CC2(C)Br)=O)cc1Cl Cc1nn(C)c(C)c1C(=O)NCC1CCCN(C(c2ccc(N(C)C)cn2)=O)C1 C1(CC)C(C(=O)NC(C)(CNC(=O)CCC2CC2)C(C)C)CCN1C C1(CNC(CCc2cc(C)cc(C)c2)=O)CCN(C(=O)C=CBr)CC1(F)F c1(C(N(C)CC2OCCN(C(C(CN(CC)CC)F)=O)C2)=O)cc(C)cc(C)c1 C(=O)(CC1CCCc2ccccc21)N1C2C(CNC(CCOCC)=O)C(C2)C1 CN1CCN(c2ccccc2CC2CCCCN2Cc2ccccc2)CC1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CC=CC(N1CCC(CCCC)CC1)=O)(C)C c1(CCN(C)CCOC)ccccc1.C(C1CC1)=CC(=O)N c1(OC)ccc(Cl)c(F)c1C(=O)NCCNC(=O)NC1CC1c1ccoc1 N1(C(C2N(C(Cc3c(C)cnn3C)=O)CCC2O)=O)CCCSC(C)C1 C12CCN(C1C(=O)NCc1nn(C)cc1C)C(=O)C2.C1(CC)CC(N(C)C)C1 CC(C(C)C(=O)NCCN1CCC(O)C1)NC(=O)CCn1ccnc1 C=CCC(CNC(c1cncnc1)=O)C(=O)NC1(CO)CC(C)(C)C1 C#CCC(C)(C(=O)NC(CC)C(=O)OC)NC(c1cnco1)=O C1(CNC(C(CC(C)C)N(C)C)=O)CCCC2CN(C(=O)C(C)CC(C)(C)C)CC12 c1(NC(CC)CNC(=O)C=Cc2ccccc2)nc(Cl)nc2c(C)nn(C)c12 N1(C(CC(=C)Br)=O)CCC2(CC1)COCC(CNC(c1cnc[nH]1)=O)O2 Nc1ccc(C(=O)NCCC2CCC(NC(=O)C(F)(F)c3cscn3)C2)nc1Cl C1(Oc2ccc(C(=O)NC(C(=O)NCC(CC)SC)OC)cc2)CCC(C)CC1 O=C(C#CC1CCCO1)N(C1CCCN(C(c2cnc3sccn23)=O)C1)CCO C1(CN(C(C(C)Nc2scc(C)n2)=O)C)C2CN(C(c3c[nH]nc3C)=O)CC12 C(=O)(CC(C(F)F)NC(C12CCN(CC1)C2)=O)N(C(C)C(C)C)CC C=CC(C)(CCOC)C(=O)N(CCNC(=O)C(C)(C)CC(F)F)C(C)C C1(CNC(CNS(c2c(C)cco2)(=O)=O)=O)CCc2nccn2CC1 C1(NC(c2cnn(CC)c2C2CC2)=O)CC2CN(C(=O)CCCC(=O)OC)CC12 N1(C(=O)C=C2CCCC2)CCC(C2CCCN2C(=O)CN2CCC2)CC1 C(=O)(CCCCNS(C)(=O)=O)NCC(C(C)C)NC(c1cn(CC(N)=O)nn1)=O N1(C(c2nn(CC)c(C)c2)=O)CCCC(F)(CNC(=O)C(C)(C)S(C)(=O)=O)CC1 CC1(C)C(CNC(=O)CSc2ccccn2)CCN1C(=O)Cn1ncccc1=O N1(C(c2ccc(C)c(N)c2)=O)CCCC2C(NC(=O)C(N)=O)C(C)(C)C12 C1(NC(C2C(C(=O)OC)C2)=O)CC2CCC1N2C(C1CCCN1C(C)=O)=O C(=O)(C1=C(C)OCCS1)N1CCCN(C(C(C2CCOCC2)OCC)=O)CC1 S(=O)(=O)(c1ccc(Br)s1)CN(CC(N1CCCC1)Sc1ccc(N)cn1)CC1CC1 C1(C(=O)NCC(C2CCC2)NC(C2(C)CSC2)=O)CCC2(CC1)CC2(F)F Cc1nc(CN(C)CCN(C(=O)Nc2ccco2)CC2CC2)ccc1Br.C1CC1 C1(NC(c2c(COC)ncs2)=O)CN(C(=O)C(C2(O)CCCC2)F)C(C)(C)C1 C=CC(C)(C)C(=O)NCc1nc(C)c(C(N2CC(C)(C)C2)=O)o1 CC(C)CCC(F)C(=O)N1CCC2CC12C(N1CC2(CCCC2)C1)=O C1(C(=O)NCCCc2cn(CCCn3cccn3)nn2)CCC2(CCC2)C1 CCC(CC)(CO)C(=O)NCC1CN(C(=O)CCc2ccncn2)C2CC12 C1(CNC(c2c(C)csc2)=O)CN(C(=O)COc2ncccn2)CCC1(F)F C1(C(N)=O)CCCC(C(=O)N(CCCNC(C2(c3ccccc3F)CC2)=O)CC)C1 Cc1cccc(N(C(C)C)CCc2ccc(Br)cc2)c1NC(=O)C1CC1 C1(C(=O)OC)CCN(C(=O)C(C)(C)N(S(C)(=O)=O)C(C)C)C1 c1(C(N(CCN(C(C2ON=C(C)C2)=O)C)C(C)C)=O)n[nH]c2cc(Cl)ccc12 N1(C(C(C)OC)=O)CC2(C1)CN(C(C1(C)CC3CCC(C1)S3)=O)CC2CO C1(NC(C(C)n2ccnc2)=O)CC(C)(NC(=O)C(O)Cc2cn(C)cn2)C1 C1(C(=O)NCC(CC(C)C)NC(COCc2onc(C)n2)=O)CN2CCC1CC2 c1(-c2ccc(CCSC)s2)nc2c(s1)CN(Cc1ccc(Cl)s1)CC2 c1(C(=O)NCCC(C)NC(C2C(C=C)CC2)=O)ccc(C(C)C)nc1O C1(C(=O)NCC(C)N(C(=O)C(O)Cc2cnc[nH]2)CC)Cc2cc(Cl)ccc2O1 N1(C(C(CC)SC)=O)CCC2(CC1)OCCCC2NC(c1cc(F)cc(F)c1)=O C1(C(=O)NCC(C)CN(C(=O)Cc2cn(C)cn2)C)OCCC1(C)C Cc1cc(C)c(-n2nc(CCN(C)C)nc2C2CCCCC2F)c(C)c1 N1(C(c2ccc(C(=O)OCC)[nH]2)=O)CCC2CN(C(=O)CC(C)CF)CCC12 C12(NC(c3ncn(CC)n3)=O)CC3CCC(C1C2)N3C(C1COCCC1(F)F)=O N1(C(C2CCN(C(CC=C)=O)CC2O)=O)CC(=O)N(C)CC1C(=O)OC C(C(=O)NC1(CCNC(C2CC(O)C(F)C2)=O)CCCC1)(C(C)C)OC C#Cc1ccc(C(=O)NC2CN(C(=O)CC3=CCCC3)C3CC23)cc1F c1(-n2c(-c3nn(CC)c(CO)c3)nc(-c3ccoc3)n2)ccc(N(C)C)nc1C c1(C(=O)NC2C(CC(=O)NC3CC3F)C(O)C2)occ2c1CCC2 C(=O)(C(C)C(O)C(C)C)N(CCC)CCNC(c1cc(OC)nc(C)c1)=O C12=NNC(=NCC(O)COCC1)S2.c1(CC)cc(OC)c(OC)c(Cl)c1 O=C(O)CC(O)C(=O)ONC(=O)NC(C1CC1)C1CC1 C1(CN(C(c2c(CC)cno2)=O)C)COCCN1C(=O)C=Cc1cnc[nH]1 CC(=O)C(C)CC(C)C(=O)NCC1C(n2cc(-c3ccc(F)c(Cl)c3)nn2)C1(C)C C1(C(=O)NCC(CNC(C2(n3cccn3)CCOCC2)=O)O)CCCS(=O)(=O)C1 C1(=CC(=O)NC(CNC(=O)C(F)CC2CC2)C2CC2)CCOc2ccccc21 C1(F)(C(N2CCC(C(C)(C)O)C2)=O)CCN(C(c2cn(C3CC3)cn2)=O)C1 C1(C(=O)NCC(C)CNC(=O)COC2CCCC2)COC(=O)O1 Cc1ncnc(C(=O)NCC2(O)CN(C(=O)C(=O)N(C)C)C=C2)c1C N1(C(c2cc(C)cs2)C(=O)NC(c2ccccc2Br)C)CCOC(C)(C)C1 n1(COC)ccc(C(=O)NC2CC(C(F)C(N3CC=CC3C(C)O)=O)C2)n1 N1(C(C(CC(=O)OC)C)=O)CCN(C(C2(CC3CC3)CCCO2)=O)CC(C)C1 C1(C(=O)NC(CC#CC)CO)N(C(c2ccc3c[nH]nc3c2)=O)CC12CCCC2 N1(C(c2cc(SC)nn2C)=O)CCN(C(C2CCCN2N=O)=O)CC(O)C1 C(C(CN(C)C)CC(=O)N1CCC(F)(F)C1)NC(C)=O.N1CCCC1CC=O Cc1ccc(F)c(C(=O)NC2CC(N(C(=O)C(C)NC(c3ccoc3)=O)C)C2)n1 C1(CC)CN(c2nncs2)CCC1N=c1[nH]nc(C(=O)OC)cc1C(=O)O C1(C(=O)NC(CNC(c2nc(OCC)oc2)=O)C)CCc2cnc(C)n2C1 c1(OC(C2CSCN2Cc2nnc(-c3ccc(Cl)s3)o2)=O)ccccc1F c1(N(C2C=CC(NC(=O)CCC(C)C)C2)C(C)=O)nc(C(F)(F)F)c(Br)s1 C(CC(C)(C)CC(=O)NC(c1ccccc1)CNC(C1CC1(C)C(F)F)=O)OC C1(C(=O)NCC(CC)O)CC(O)C(O)CC1CNC(c1csc(C#N)c1)=O C1(NC(Cc2nc(C)[nH]n2)=O)CC(CNC(c2coc(C3CC3)n2)=O)C1(C)C N1(C(CC=C)=O)CCC(C2(O)CCN(C(c3cnc[nH]3)=O)C2)CC1 c1(C(=O)NCC2C(C)CCCN2C(=O)CC2CCC(O)C2)cccn2nncc12 CN(S(=O)(=O)NCCOC(F)F)CCC1CCCC12CC2 C(=O)(C1=NN2CCCN=C2N1)N(CCN(C(C)C)C(c1cncnc1)=O)C N1(C(C(C)CC2CCC2)=O)CC(CO)C2(C1)CN(C(=O)CSc1n[nH]c(=N)s1)C2 c1(N2CCC(COC)C2)nc2c(c(=NC3CC3C(C)C)[nH]1)CCCCCC2 c1(OC)ccc(CC(=O)NCC2CC2NC(=O)CC(C)C2CCCO2)c(OC)c1 c1(C(=O)NC2(C(N(C)C)=O)CC2)ccc(CNC(=O)CC2(C)CCCO2)nc1 CN1CC(CCNC(C2(CCNC(=O)Cc3cnns3)CCC2)=O)C1 CC1(C)C(C)(C)C1(Br)C(=O)NC1COCC1NC(=O)CCC1CCOC1 C1(C(=O)NCc2ccccc2CNC(C2CCC(C)(C)C2)=O)(CC)CCCOC1 N1(C(c2c(OC)cnnc2)=O)CCC(NC(C2OCCC2(C)C)=O)C(C)(C)C1 O=C(C(CNC(=O)OC(C)(C)C)CC1(C(=O)O)CC1)NCC(O)CF C(C(C(=O)NCCC(C)COC)NC(=O)COC)OC.C1(O)CC=CC1 C(=O)(C1=CCCS1)NC1C(C(N(CCC#N)C2CC2)=O)C1 c1(C(=O)NC(C)(C)CCNC(=O)COC2CCOC2)ccc(OC(F)(F)F)cn1 Cc1nn2c(C)cccc2c1C(=O)N(C)CCN(C(=O)CS(=O)(=O)C(C)(C)C)C C1(CNC(c2c(COC)cc[nH]2)=O)CCC(C)CN1C(c1cc(Cl)cnc1O)=O Cn1cnc(C#N)c1C(=O)NC1CN(C(C2(c3cnn(C)c3)CC2)=O)C1 CC(C(=O)N(CC(O)CN(C(=O)C=Cc1ccc(Cl)nc1)C)C)S(N)(=O)=O c1(C(=O)NCC2CCN(C(=O)CN3CCCC3=O)C2)cc2c(O)ncnc2cn1 C1(C(N(C)CC2CCN(C(C3CC(C#N)C3)=O)C2)=O)CCN(CCO)C(=O)C1 C1(C(N(C2CCN(C(C3(CF)CC3)=O)CC2)C)=O)CC(=O)N(C2CCCC2)C1 C1(C(N(C(C(C)SC)C)C)=O)C2CN(C(c3ncccc3N)=O)CC12 c1(C(=O)OC)cc(C(=O)NC2CC(C)N(C(c3cc(C)no3)=O)C2)ccc1Cl CCC(c1ccc(OC)cc1)=CC(N1CC2CC2(NC(=O)C=C(C)C2CC2)C1)=O Cc1cnc(CC(=O)N(C(C)CN(C)C(C2CCN(C3COC3)C2)=O)C)s1 C12CCCN1C2.c1(C2CN(C(=O)OC(=O)CCSC(F)(F)F)C2)cccnc1 CCC(C(=O)OC)C(=O)NCC(C)N(C)C(C1CCOCC1(C)C)=O C1(CCC=C)(C(=O)OC)CN(N2CCCC(OC(=O)NC)CC2)C1 C1(C2CC2)(NC(C(CC)NC(C)=O)=O)CCN(C(=O)Cn2cc(CO)nn2)C1 N1(C(C2CC(F)CN(C(=O)CCN3CCOCC3)C2)=O)CCN2CCOCC2C1 C(CC(C)(C)C(=O)NOCc1ccccc1)NC(CC1CCN(C)C1=O)=O c1(NC(=O)CC2COCCN2C(c2ccc[n+]([O-])c2)=O)c(O)cccc1Br C12(CC(=O)NCC3(C(N)=O)CCC3)CCCC1C2.n12ccc(n1)C(=O)NCCC2 C1(F)(CNC(c2cc(C)n(C(C)(C)C)n2)=O)CCCN(C(=O)CC2CCOC2)C1 O=C(C1=NOC2COCC12)NC1CC(C(=O)NCC2Cc3nccn3C2)CC1O C(=O)(C1=C(C)OCC1)NC(CNC(C(CC)OCC)=O)C(C)(C)C C(=O)(CC1=CCCCC1)NC1(CCNC(C(C)Oc2ccccc2)=O)CC1 N1(C(CSCCC#N)=O)CCC2CCN(C(=O)CCCC(F)F)C2C1 C(C(C)(C(=O)N(CCCCCCNC(c1ccc(CC#N)cc1)=O)C)OC)OC C1(NC(C(F)=CC)=O)CCC(NC(=O)Cc2cncn2C2CC2)CC1 C(=O)(C(C(C)(C)C)NC(C1CCCSC1)=O)N1CC(C)(C)C1C1CC1 c1(C(=O)NC2C(CC)N(C(=O)C3CC3)CC2)cc2c(C)cc(Cl)cc2[nH]1 N1(C(C(COC)NC(=O)CC(C)(C)C(F)F)=O)CCc2c(cnn2C)C1 C1(CC)COCCN(C(=O)CNC(C2CC(N(C)CC)C2)=O)C1 C1(CC(NOCC(=C)C)=O)CCCN(C(c2cc(Cl)cs2)=O)C1 N1(C(CNC(c2ccc(F)cc2)=O)=O)CCCC12CCN(c1cn[nH]c1)C2=O C(=O)(C1=NOC2COCC12)N1C(C(=O)NCC(CSC)(C)O)CCOCC1 C12CCCN(C1)C2=O.c1(C(C)Nc2csc(-c3ccco3)n2)ccccc1O c1(SC)nc(N2CC3(CCC(NC(c4cc(O)no4)=O)C3)C2)c2ccccc2n1 c1(C(CNC(=O)NCCN(CCC)C(C)C)CC)cccc(Br)c1 CC1(C)CC(C(N2CCCC(NC(=O)Cc3ccccc3F)CC2)=O)CNC1=O C12CN(CC1C)C2=O.c1(C2(NC(CC=CC=C)=O)CC2)ccc(OC)cc1 c1(CCC(=O)NC2(CC(=O)NC(c3cccc(F)n3)C)CCC2)ccccc1Br CCC(O)C(C)C(=O)N(CCCNC(c1cccc(N)n1)=O)CCO C(C)(C)(CCOC)NC1(CC(=O)OC)CN(C(=O)CCCF)C1 c1(OC)cc(C(N2CC3C(C2)N3C(c2ccccc2N(C)C)=O)=O)cc(Br)c1 N1(C(c2c(Cl)cc(C)c(F)c2)=O)CCOC2CN(C(=O)CC3CCCCO3)CC12 C=C(Cl)C(C)(C)C(=O)N1CCC(CCOC)(NC(=O)C(C2CCCCC2)F)C1 N1(C(C2C(C)(C)C2NC(=O)COC2CC2)=O)CCC2OCCC2C1 CC1(C(=O)NCC2(C(=O)NCC3CNC(=O)C3)CC2)CCCO1 c1(OC)ccc(N)c(C(=O)NCC2CC(NC(c3cnc(C)nc3SC)=O)C2)c1 c1(NC(C(=O)NCCCN(CCN)C(C2CCCO2)=O)=O)cccc(Cl)c1.CO C(=O)(N(CCC(=O)NC1CCSCC1)OC)c1n(CCC)cnc1 C12(NC(Cc3cncc(C)c3)=O)CCC(C1)N(C(C1(Cl)CC1(C)C)=O)C2 C(C(CC)CC(C)C)NC(c1c(Cl)noc1C)c1n(C(CC)C)nnn1 c1(CC)cc(C(=O)NCC2CCCN2CCOC)sc1C N1(C(CC(C(F)F)NC(=O)CCc2cccnc2)=O)CCC2(CNC(=O)N2)C1 N1(CCC)C(=S)NC(c2ccc(C3CC3C)o2)C(C(=O)OCC)=C1CF CCCCC(C(=O)NC(CN=[N+]=[N-])C(=O)NCCc1cccnc1F)C(C)C CCC(CNC(c1csc(O)n1)=O)(CC)C(=O)NC1CCC2(CCC2)C1 c1(OC)cc(Cl)c(Br)cc1C(N1CC2(CNCCO2)C1)=O CCCC(C(C)C)(c1nnnn1C(C)C)NC(c1cn(C2CC2)cn1)C C(c1cccc(Cl)c1)=CC(=O)NC1C(NC(C2C(C)CCO2)=O)CCC1 Cn1cnc2ccc(C(N3CC4CN(C(c5cc(O)nc(Cl)c5)=O)C4C3)=O)cc12 C(C)(C(=O)N(CC=C)OC)C1CN(C(CC(=C=C)C)=O)C1 CC(CNC(=O)CC1CCCSC1)CC(=O)NCCCCC1CC1 C1(NC(c2c(C)c(C(C)C)[nH]n2)=O)CC2(C1)CC(NC(=O)C(F)C1CCCC1)C2 C(=O)(C(C)CCCC(C)C)N1CCC(C(=O)NC2CC(Cl)(Cl)C2)(OC)C1 c1(CC(=O)NC2CC(F)(CNC(CC(C)O)=O)C2)cccc2ccsc12 N1(C(c2ncn(C)c2)=O)CCC2(NC(C3CCC3)=O)CCCC12 C1(C(=O)NCC2N(c3nnc(C)s3)C3C(C2)COC3)CCn2c(C)cnc2C1 C(=O)(C(C(C)(C)C)N(C)C)NC(CNC(C1(SC)CCSC1)=O)C(C)C C1(NC(C2CCCC(F)C2)=O)(CO)CCCN(C(=O)COc2ccsc2)C1 c1(NC(C2C(C(=O)NCCOCCN(C)C)C2)=O)ccc(C2CC2)nn1 N1(C(=O)C=Cc2ccsc2)CC2CN(C(c3ccc(C4CC4)nc3)=O)C2C1 C(CCC(C(=O)NCC(F)(F)F)NC(=O)CC1CCCSC1)OC c1(C(C(=O)N(CCCNC(CC2CC(SC)C2)=O)C2CC2)(C)O)ccc(F)cc1 C1(C2CCN(C(=O)CCCc3cnn[nH]3)C2)(NC(=O)CC2CCCC23CC3)CC1 Cc1c(C(=O)NCCOCCN(C)C(c2cc3c([nH]2)CCC3)=O)cc(N)cc1O C(=O)(C(=O)C(C)(C)C)NC1C(OC)CN(C(c2nc(C(C)(F)F)cs2)=O)C1 c1(NC(CCN(C)C(c2cccc(-n3ccnc3)c2)=O)=O)cccnc1CO c1(CNC(N2C(C(=O)Nc3cccc(Cl)c3)CCC2)=O)ccc([N+](=O)[O-])c(Br)c1 c1(C(=O)OC)cc(=NC(=O)CN2CCC(O)(C(F)(F)F)C2)cc(C)[nH]1 N1(C(C(C)N(C)C2CC2)=O)CCC=CC1C(=O)NC(CC1CC1)C1CC1 C1(NC(CSCC(=O)OC)=O)CCC2(CC1)CN(C(=O)C(C)CC(C)C)CCO2 N1(C(C(C)NC(C)=O)=O)CC(F)(F)CC1C(=O)Nc1ccc(C)c(C(F)(F)F)c1 c1(CC)ccccc1C(=O)NCC(O)CC(=O)NC(c1ccc(C)s1)C C(=O)(CCC(C)N(C)C)NCCc1cnc(C)s1.C12(CCC1)C(=O)OC2=O C=CC(C)CC(=O)NCc1nnn(C)c1C(=O)NCC1CC1Cl N1(C(c2[nH]n(C)c(=O)n2)=O)CCC2CN(C(=O)CC3COC(=O)C3)C2C1 C1(OC)(CNC(C2CC2Br)=O)CN(C(c2cc(C(F)(F)F)n[nH]2)=O)C1 c1(OC(C)C(=O)NC2CC(CNC(C3(C(N)=O)CC3)=O)C2(C)C)ccc(F)cc1 N1(C(C2OCCC(NC(c3c(OC)cncc3)=O)C2)=O)CCN(C)CC1C C1(NC(c2ccc(C)nc2)=O)CCN(c2nccc(Br)n2)CCC1CO N1(C(COC)=O)CCCC2(CNC(c3cnn(CCC(F)(F)F)c3C3CC3)=O)CC12 Cc1cnc(N(C)Cc2cc(Br)cs2)c(S(=O)(=O)NC2CCC2C)c1 c1(C(N2CC(CC)C(NC(=O)C3=CCC3)CC2)=O)c(C)nc2ccccn12 c1(-n2cc(CC3CCN(C(c4c(C)n(C)nc4)=O)C3)nn2)ccc(F)c(Cl)c1 Cc1ccc(C(=O)NCc2nc(C(=O)NC3CC34CCCC4)c(C)o2)c(C)n1 n1(C2C(C)C2)nc(-c2ccco2)nc1-c1cc(Br)cs1.c12ccc(cc1)OCC2 C1(CC(C)NC(c2ccnnc2)=O)CCN(C(c2cscc2C2CC2)=O)CC1 N1(C(C2COCC(C)O2)=O)CC2(C(N3CC(F)(C#N)C3)=O)CCC1CC2 c1(-n2ncc(C(CC)NC(=O)NCCC3CC(C)C3)c2)ccc(Cl)cc1 Cc1ccc(C)c(C(=O)NCC2CC(CNC(c3cncc(Cl)c3Cl)=O)CO2)n1 C(=O)(C1=CCCC1(C)C)NCC(C)(C)OCCNC=O.C1(N)COC(=O)C1 C1(NC(Cn2nnc(C)n2)=O)C2CC3CN(C(=O)C(C)CC(C)(C)C)C1C3C2 C#CCC(C(=O)N1CCCC1CN(C(c1cc(CC)no1)=O)C1CC1)C1CC1 Cc1nc(C)c(C(=O)N(C2CC(NC(=O)Cn3cnc(=N)[nH]3)C2)C)[nH]1 Cc1ccc(CC(=O)NCCC(=O)NCCc2csnn2)s1 N1(C(CC(CC)SC)=O)CCN(C(c2ccco2)=O)C(c2cccc(F)c2)C1 c1(C(N(CCC(=O)N2CCC2N2CCCC2=O)C)=O)cccc([N+](=O)[O-])c1 C(CCN(C)C(c1sccc1F)=O)(C(C)(C)C)NC(C(C)CO)=O C1(C(=O)NCCC(C)(C)N(C)C)CC(NC(c2cc(Cl)ns2)=O)C1(C)C N1(C(C=C(C)Cl)=O)CC2CCC1C(NC(=O)Cc1cn(C)nc1C)C2 N1(C(c2c(CC)noc2)=O)CC(F)(F)CC1NC(=O)CC(C)OC C1(C(C)(C)NC(Cc2n(C)nnc2)=O)CCN(C(C2(C)CC2F)=O)CC1 c1(C(=O)NCC(=C2CN(C(C3C(C)C3)=O)C2)F)cc2ccccn2c1 CCC(C)CC(=O)NCC1CCCC1C(=O)NCc1csnn1 c1(SC)ncc(CN2CCOC(C(=O)Nc3cc(I)ncn3)C2)c(Cl)n1 Cc1cc(C(=O)NC2CCN(C(=O)C(O)C(C)C)C2C(C)C)nn1C(C)C C1(NC(=O)CSc2ccc(F)cc2)COCCC1NC(=O)CC1CC1(Cl)Cl C1(NC(C2CN(S(=O)(=O)C(F)(F)F)C2)=O)CN(C(=O)CC(Cl)Cl)CC12CCC2 C1(=CC(N2C(CCCC)CCC2)=O)CCN(C(c2cnc(Cl)cn2)N(C)C)CC1 c1(CNC(C2(CNC(C3C(CCC)C3)=O)CCCO2)=O)cnc(C)cn1 C(C)(C(=O)N1CCC(C(C)(C)NC(=O)Cc2ccc(C)c(Cl)c2)C1)(C(C)C)OC c1(CC(CN2CC(=O)N(C3CCCC3)CC2)O)ccc2c(c1F)CCC2 c1(C(=O)NC(C#C)CCC)ccc(CC(C)(C)C(N)=O)cc1 C1(NC(C2(OC)CCC2)=O)CCCC(CNC(=O)CSc2nccn2C)C1 CCC(C)(C)CN=c1[nH]c2c(c(=NC3CCC4(CCC4)CC3)[nH]1)COC2 CCC(C)(O)C(=O)N1CC2(NC(=O)CCN3CCOCC3=O)CC1C2.C1CCS1 C1(C(=O)NCC2(OCC)CC2)CC12CCN(C(c1cc(F)c[nH]1)=O)C2 CCC1=C(C(=O)NC2CCC2NC(=O)Cn2cc(C)cn2)SCCO1 N1(C(c2n(CCC)ncc2)=O)CC2(CC2)CC1CC(=O)NCC1CC=CC1 N1(C(C2=CC=NCC(OC)=N2)=O)CCCC2(C1)CN(C(=O)CC(C)(C)C(F)F)C2 C=CCC(C)(CC)C(=O)N1CCC(C(C)NC(c2ncncc2N)=O)C1 Cc1ccn2c(C(=O)NCC3CCC(NC(C4CC(C)CO4)=O)CC3)cnc2c1 N1(C(C2(C(CC)=O)CC2)=O)CC2CCC1C1CN(C(c3ccc(C)o3)=O)CC21 n1(C(C)C)cnc2c(N(C)Cc3ncco3)[nH]c(=NCCN3CCC(C)C3)nc12 C1(CCNC(c2c(C)[nH]nc2Br)=O)CCN(C(C2CCC2)=O)CC1(F)F c1(C(N2CCC(NC(c3ccc(C)o3)=O)(CF)C2)=O)cc(C)c(F)c(C)c1 c1(C(N2CCC(C3N(C(c4ncc(C)cn4)=O)CCC3)C2)=O)nccc(Cl)c1C c1(C(C)NCC2CCC(O)CC2)cc(F)c(O)c(F)c1 CC(C)C(C(=O)N1CC(NS(=O)(=O)CC(C)C)C(F)C1)c1ccc(F)cc1 N1(C(C(CC(CC)C)C)=O)CCC2(CC1)CN(C(=O)CC=C(Cl)Cl)C2C(C)C CN=c1[nH]c(SC)ncc1CN1CC(C)(C(N2CCCC(F)(F)CC2)=O)C1 c1(C(N2CC(NC(c3cnn4c3CCC4)=O)C(O)C2)=O)cc(F)cc2cc[nH]c12 c1(C(=O)NC(CN(CCC)C)(C)C)conc1CNC(c1ncoc1C(C)C)=O C1(C(N2CCC(NC(C3(C)C(C)C3)=O)C2)=O)CC2(CSC2)C1 c1(CC)cccc(C)c1C.C12CCC(CC1)C(c1nnnn1C1CC1)OC(=O)CN2 C12(C(N3CC(NC(C4(C)CCN(C)C4=O)=O)C3)=O)CCC(N=[N+]=[N-])C1C2 C1(F)(C(C2CC2)OCC(C2SCC(C)C2)=O)CC2CC1(c1ccccc1)C2 N1(C(C(C(C)C)=O)=O)CCCCC(C(=O)NCc2cnc3n2CCC3)C1 C=CC(C)(O)CC(=O)NCc1ccc(CNC(=O)CCP(C)(C)=O)cc1F N1(C(c2cn(CCF)nn2)=O)CC(CO)C2(C1)CN(C(=O)C1CC1)C2 c1(C(N2CC(CNC(C3CC(=O)NC3)=O)C(F)(F)C2)=O)c(F)ccc(F)c1Cl C#CCCCC(C)C(=O)N1CCN(C(=O)Cc2c(C)cc(C)cc2C)C(C)C1 n1(CC)cnc2c(NCC(C)C(F)(F)F)[nH]c(=NCc3ccc(Cl)o3)nc12 c1(CCCC(=O)NCC2C(NC(COCC(=O)NC)=O)CCC2)nnc(C)n1C N1(C(C2C(C)(CC)C2)=O)CC(O)(CCNC(C2(CC(=O)N)CCCC2)=O)C1.C1CC1 c1(CC)cccc(C(N2CC(CC(C)NC(c3cc(O)nc(Cl)c3)=O)C2)=O)c1N c1(C(=O)NC2C3CC2N(C(=O)COCCF)C3)cccc2c1OCCO2 c1(C(=O)OC)cc(F)cc2c1CCN(C(c1ccc3nnn(C)c3c1)=O)C2 C1(CNC(C2CC(CC)(CC)C2)=O)CCC(CNc2ccnc(Cl)n2)CC1 N1(C(C(=COCC)C#N)=O)CC2(COC(CNC(C3CCC(F)CC3)=O)C2)C1 C1(C(N(CCC)CC)=O)CC(NC(c2cccc(OC)c2C)=O)C12CCC2 CCCC(C)C(=O)N1CC2CC1C2C(=O)Nc1cccnc1Cl c1(C(N(C(CN(C(C(C)OC)=O)C)C)C)=O)ccc(Br)cc1NC(C)=O N1(C(CN(CCOC)C)=O)CCCC(C2CCN(C(c3c[nH]c(=N)s3)=O)C2)C1 c1(C(N(C)CCOCCCNC(=O)CS(C)(=O)=O)=O)ccc2c(c1)NC(=O)C2=O c1(C(=O)N)ccccc1.C1(C(=O)N)CN(CC2CC2F)C1.C(CCOC)=CCSCC C1(C(=O)NCC2CCN(C(C3CCCCC3(F)F)=O)C2)Cc2ccccc2C1 c1(NC(CC)CSC)ncc(C)cc1S(=O)(=O)N1CCOC(OCCCO)C1 Cc1ccc(C)c(OCCC(=O)NCC2(NC(c3n[nH]cc3F)=O)CCOC2)c1 n1(CC(=O)NC2CCN(C(=O)C(F)=CC3CC3)CC2F)ccc2ccccc12 Cc1ccc(=O)n(CC(=O)NC2CCN(C(c3cccc(Br)c3C)=O)C2)n1 C1(F)(CNC(CCC=C)=O)CCCN(C(C2CC3CCCC3C2)=O)C1 C(=O)(C1=CCCOC1)NCC1N(C(CCSC)=O)CC(O)C1 C(C(C)(C)C(=O)NCc1coc(C)n1)N(C(C1CCC(CC)C1)=O)C Cc1cn2c(n1)CC(C(N1CC(CNC(c3ccc[n+]([O-])c3)=O)CC1(C)C)=O)C2 c1(OC)cc(C)c(C(=O)NC2CC(=O)N(OCC3(C)CCCN3)C2)cn1 C(=O)(C(F)C1=CCCCC1)N1CC2CC(C1)NC2=O.N1(CC(=O)OC)CC2CC2C1 C1(CNC(=O)CC2CCCC2CNC(N2CCCC2)=O)CCCC2(C1)OCCO2 N1(C(C(CC=C)C)=O)CCCC2(CCCN2C(C2CC(C(F)(F)F)C2)=O)C1 c1(OCC)ccnc(NC2CCCN2C(C2CCCN2S(C)(=O)=O)=O)n1 c1(C(C(=O)NCC2CC2)N(C(CC)CC)C)cnc(C(C)C)s1 N1(C(=O)NC(CCOC)C)CCc2ccccc2C1CC c1(C(=O)NCC(C)(F)CNC(C2C3COCC23)=O)cccc2c1CCC2 N1(C(C(C2CC2)OCC)=O)CC(NC(c2cnoc2C2CCC2)=O)CC(C)(C)C1 c1(C(CC)NC2CC(CNC(=O)Oc3ccccc3)C2)nnn(C)c1C(F)(F)F c1(C(=O)NC(C2CCCC2)CNC(C2CC2(F)F)=O)cncc(Cl)n1 N1(C(c2cnc(CC)[nH]2)=O)CCC(C)(CCNC(=O)Cc2ncccc2C)C1 C(COC)(CC(=O)N(CCCCC(=O)N(CC(=O)OC)C)C)NC c1(C(=O)NC(C2CCN(C(CSCC=C)=O)C2)(C)C)ccc(CCO)cc1 c1(CNC(C2CC3CC3N2CCN2CCNC2=O)=O)cccc([N+](=O)[O-])c1F C1(NC(C2(CC)CCCN2C(c2cc(C3CC3)n(C)n2)=O)=O)CCCCCCC1 C1(NC(C2CCN(C(C3CNC(=O)N3)=O)C2)=O)CCCN(O)C1=O CC1(C)C(C(=O)NCCc2nn[nH]n2)CCN1C(c1cccc(CO)c1)=O CCCCC(CC)CC(=O)NC1CCC(CCC(N2CC(CO)C(C)C2)=O)C1 C1(NC(=O)NC(c2ccc(C(=O)OC)o2)C)CCOC(C(C)C)C1 c1(C2C(C(N3CCCC(NC(N)=O)C3)=O)C2)cc(C(F)(F)F)ccc1Cl C(=O)(CCC(=O)N1CC(NC(=O)CCN(C)C)C(O)C1)Nc1nnc(C(C)C)s1 N1(C(c2ccc(C(N)=O)[nH]2)=O)CCC(O)(C2CCCN2c2nnc(C3CC3)s2)C1 N1(CC2(C)CCCO2)CCC(N)CC1.n12cc(nn1)NC(=O)COCCOCC2 c1(C(CC)NC(=O)NCCC2CC(O)C2)nocc1C C(=O)(CCCCCC(C)C)N1CCCC(N(C(c2cccnc2)=O)CC)C1 c1(C(N(CC(C)O)CCNC(c2cnn(CC)n2)=O)=O)c(SC)nc(O)nc1C C1(NC(C=NOC)=O)CCC2(CCCN(C(c3scnc3Cl)=O)C2)C1 C12(C(N)=O)CCCC1(C(=O)NC1CCCN(c3ccccc3)C1)C2 N1(C(c2cn(C)nc2)=O)CCC(N(CCO)C(C2CCSC2)=O)CC1 N1(C(CCC2N(C)CCC2)=O)CCN(C(C2CC3(CC3)C2)=O)C2CCCC12 C#CC(C)(C)C(=O)NC1CCCC(N(C)C(c2ncsc2NC)=O)C1 C(=O)(CC(C)(C)CNC(c1cccc(CO)c1)=O)N1CCN(CCOC)CC1 C1(C(N2CCN(C(C3C(=C)C3)=O)C(C)C2)=O)C2CCC1(C)C2(C)C C1(CNC(C(C)N(CCC)C(C2CC(n3ccnc3)C2)=O)=O)CCCC1 C(=O)(C1COc2ccccc21)NCCn1cc(C(NOCCCCC)=O)nn1 Cc1cncc(C(=O)NCC2CC2NC(=O)CCc2cccc(O)n2)n1 N1(C(c2cnc(OCC)c(Cl)c2)=O)CC(NC(c2csc(Cl)n2)=O)CC2(CC2)C1 CCCS(=O)(=O)CC(=O)N1CC2C(CNC(C3CCC(NC(N)=O)CC3)=O)C2C1 C1(COC)(NC(=O)CCC2(C)N=N2)CCN(C(c2ccc(OCCF)cc2)=O)C1 c1(C(=O)NC(C)C(=O)C2CCOC2)ccc(Oc2ccccc2Cl)nc1 C1(C2CCN(C(C3SC4C=CC3CC4)=O)C2)(NC(C(C)=C(C)C)=O)CC1 N1(C(CCN(CC)CC)=O)CCCC(N(C)C(C2COCCN2C=O)=O)CC1 C1(C(N)=O)CCCN(S(=O)(=O)NCC(c2ccc(Cl)o2)O)C1 CCCCCCCCN(C(=O)CC1CCN(C(C)=O)CC1)Cc1cc(C)on1 c1(C(N2CC(C)OC(CNC(C3(C4CC4)CC3)=O)C2)=O)cnn2cccc2c1 C1(NC(CCN(CCC)C)=O)CCC(C)(C)CC1CNC(c1ccsc1CC)=O C(C(C)C(C)C(=O)N1CCC(C2CCCN2C(c2csc([N+](=O)[O-])c2)=O)C1)OC C1(C)(CNC(C2C3CN(C(c4cncc(C)c4)=O)CC32)=O)CCOC2(CCC2)C1 CC(C)(CC(=O)N1CCC(NC(=O)C(c2ncccc2F)(F)F)C1)CC(F)(F)F N1(C(C(C)S)=O)CCCC2(CCN2C(=O)CC2(Sn3ccnc3)CC2)C1 S(=O)(=O)(c1ccc(F)cc1)NCC(=O)NC1CC(NC(=O)C=CCO)CC1O C1(CNC(c2cc3ccncc3s2)=O)CN(C(C2CCCO2)=O)CC2(CCC2)O1 C1(C(=O)NC(C)CCCCNC(=O)CCn2cnnn2)CCC2(CCC2)C1 CC(C)CCC(=O)N1CC2CC2(c2nc(CCc3ccc(C(C)C)cc3)no2)C1 c1(N(C)CC2C3COCC23)ccc(S(=O)(=O)NC2CC3(C2)CC32CCC2)cc1C#N C1(N(c2ccc(C#N)s2)C(=O)OC)CCCNC1C.CC1CC2N1C2=O c1(OC)ncc(Cl)cc1C(N1CCCOC(CCNC(=O)C(C)NC=O)C1)=O c1(OC)cc(C(=O)NC2CCN(C(=O)CCC(C)SC)CC(O)C2)cc(F)c1F N1(C(C2(C#N)CC2)=O)CC2CCCC2(NC(C2COCCN2C=O)=O)C1 C(CCC(C)C(=O)NC1(CC(=O)NCC2Cc3nccn3C2)CCC1)OC C1(NC(c2c(C)nco2)=O)CC12CC(NC(=O)Cn1ncc(Br)n1)C2 c1(C(=O)NCc2onc(-c3ccc(C(=O)OCC)cc3)n2)ccc(F)c(Cl)c1F c1(C(=O)NC(C2CN(C(c3n(CC=C)ccc3)=O)C2)C)ccc(OC)cn1 c1(OCC(=O)NCC2C(NC(CCC(=C)Cl)=O)C2)ccc2ccccc2c1 S(=O)(=O)(c1cccc(=NCC2CCCC(C)(C)CC2)[nH]1)NC(CCCC=C)C CCC(CC)CCCC(=O)N1CCC(CC(=O)NCC(C)(O)CO)C1 C12(C(=O)NC(CNC(c3cccc(CC)c3)=O)C)CCCC(C(=O)OC)(CC1)C2 C1(NC(c2c(CCC)occ2)=O)CC2(C1)CN(C(=O)CCC1CC1(C)C)C2 C#CCC(C)(CNC(=O)COCCNC(c1cnc(C)n1C)=O)CO C1(COC)CN(C)CCN1C(c1nc(C)co1)C(=O)NCCN1CCOCC1 c1(C(=O)NCC(CNC(C(C)NC(C)=O)=O)(C)O)ccc(F)cc1Br N1(C(C(=O)NC2Cn3c(COC)nnc3CC2)=O)CC(C)(C)C(O)C(C)(C)C1 Cc1ccccc1-c1nsc(NCc2ncn(Cc3ccccc3)n2)n1 Cc1cnc(C(=O)NC2CCOCC2C(=O)NCC2CCC(=O)NC2)cn1 N1(C(c2ccccc2Cl)C(=O)NCC(=C)C)CCC(C#N)CC12CC2 n1(CC(N2CC(O)CC(NC(c3nn(C)c(F)c3)=O)C2)=O)cc(S(C)(=O)=O)cn1 C1(C)(CNC(C2C(C(C)C)C2)=O)CC(NC(=O)CCN2CCOCC2)C1 C(=O)(C(CO)C(C)(C)C)NCC1(CC(=O)NCC(C)CC(F)(F)F)CC1 c1(C(N(C(CN(C(C(CC(C)C)F)=O)C)C)C)=O)ccc2ccccc2c1F C1(=O)CCC(F)(F)Cn2cc(nn2)C(C)(C)N1C.S(=O)(=O)(C1CC1)COC(=N)O CN1CCCCC(C(=O)NCC2C3CCC(C3)N2C(c2cc(CO)[nH]n2)=O)C1=O C(=O)(C1=Cc2ccccc2OC1)NCCCCCNC(C1CCC(C)(O)CC1)=O N1(C(c2cncc(C)c2)=O)CCC2(CCCN2C(=O)C(CO)C(C)C)CC1 c1(OC)csc(C2CC2)c1OC.c12cnc(nc1)NC(=O)C(C)n1cc-2nn1 C1(NC(CC2(CC)CCC2)=O)COCCN(C(c2c[nH]nc2C(F)(F)F)=O)C1 N1(C(c2scc(CC)n2)=O)CC2CCC(C1)C2NC(c1ccc(Br)c(C)c1)=O c1(SCC(=O)N(CCNC(C2CCCOC2)=O)CC)nc2ccccc2[nH]1.C1(S)CC1 CCCCC(O)CCC(=O)N1CCCC1CNC(c1cc(C2CCC2)nn1C)=O c1(NC=O)ccc(C(=O)NCC(CNC(C2(c3ccccc3)CC2)=O)CO)cc1 C1(NC(C=CCCC)=O)C(C)CN(C(c2ccnn2C2CCOCC2)=O)CC1C CC1NC(=O)CCC1NC(C1(CNC(=O)CC2CC3(CC3)CO2)CCC1)=O NC1(C(=O)NC(c2ccccc2)CO)CCC2CCC12 c1(CCC(=O)NCC2CC(NC(c3ccn(COC)n3)=O)C2)cc(C)nn1C c1(CNC(c2cc(C)c(-c3ccccc3OC(C)C)s2)=O)cccc2nn[nH]c12 N1(C(c2c(CC)nccn2)=O)CCN(C(C2CCCC23CC3)=O)CCC1C Cc1c(Br)ccc(C(N2CC(O)(CNC(C3CCC(F)(F)C3)=O)C2)=O)c1F C1(NC(C2C(C(=O)OC)C2)=O)CCCCC1CNC(=O)CSc1n[nH]c(C)n1 c1(OCC)cncc(C(=O)NC2CC(CNC(c3cnn[nH]3)=O)C2)c1 N1(C(COCC)=O)CCN(C(C2(c3ccccc3)CC2(F)F)=O)CCC1C C(C1C(=O)N1)N(C)C.C1(CNC(=O)OC(C)(C)C)CCCS1 c1(C(=O)OCCC(C)C)cc(C(=O)C(C)N(CC(C)C(C)C)C)c[nH]1 C1(CNC(c2c(C)n[nH]c2)=O)CCN(C(C2CCSC2)=O)C12CC2 N1(C(CSC)=O)CCOC(CC(=O)NC2CN(C)CC2C)C1 n1(CC(=O)NC2CC(C(F)F)C2)cc(Br)cn1.c12cc(no1)CNC2=O N1(C(C(CC(C)C)F)=O)CC(O)(C2(CNC(C3CC4(C3)CC(O)C4)=O)CC2)C1 N1(C(C2C(C)C2C)=O)C2CCC1CN(C(=O)COc1ccccc1)CC2 CCCCC(C(=O)N(C(C)CNC(c1[nH]ccc1C)=O)C)N1CCCS1(=O)=O C1(NC(CCC(=O)NC)=O)COCCN(C(C2(C)CCC(=O)N2)=O)C1.C(C)(C)N CC(C)C(C(=O)N1C2CCC1CC(N(C(=O)CCC1CC1(C)C)C)C2)C(C)C c1(C(N2CCCC2CS(C)(=O)=O)C(=O)N(C)C2CC2)ccc(C)cc1C C1(NC(c2ccc(Cl)nc2O)=O)COCCN(C(C2(C3CCCO3)CC2)=O)C1 c1(CC)ccc(S(C)(=O)=O)cc1C(=O)N(C1CCN(C(=O)CN(C)C)CC1C)C C(C(C(=O)N=c1ccn(C(C)C)[nH]1)NC(c1cnc(CC2CC2)o1)=O)OCC CCC(C#N)C(=O)NCC1CC(NC(C2CCS2(=O)=O)=O)C1 c1(C(=O)NCCN(CC(C)O)C(C2CCOCC2(C)C)=O)ccnc(Cl)c1F N1(C(C(N)c2ccoc2)=O)CCC(C(=O)NCC2COCCN2)CC1 c1(CNC(=O)NC2(C)CCSC2)cc(Cl)ccn1 Cc1c[nH]c(C(=O)NC(C(=O)NCC(F)(F)C(C)C)C2CCCO2)c1C C1(CC(=O)NCCOCCNC(c2n(C=C)ncc2)=O)CCC2(CCOCC2)CO1 c1(OC)ccccc1N1CC(C(=O)NCc2cccc(CN)c2)CC1=O C1(C(=O)NCCOC2CN(C(C(C(CC)O)C)=O)C2)CC12CCOC(C)C2 CCC(C)(C)C(C)CC(=O)N(C1CCCN(C(c2cc(Cl)n(C)n2)=O)C1)C C1(NC(C2COCCOC2)=O)CCOCC1NC(C1(c2cccnc2)CC1)=O C(=O)(CC(C)C1CC1)NC(C1(c2ccon2)CCC1)CNC(C1CC(SC)C1)=O c1(NC2CC(NC(CCC(C)SC)=O)C2(C)C)ncnc2cc(C3CC3)nn12 N1(C(C=CCC)=O)CCOC(CCCNC(=O)Cc2csc(-c3ccoc3)n2)C1 C1(N(C)C(c2ccc(C(F)F)cc2)=O)CN(C(C2(CC#N)COC2)=O)CC1(C)C c1(CN2CCC(NC(CC(CC)O)=O)C(O)C2)cc([N+](=O)[O-])cc(O)c1O C(=O)(C(O)CC(C)(C)C)NCCCC1CCN(C(C(C)NC=O)=O)CC1 C1(N(C(=O)CC2(O)CCOC2)C)CCC(NC(=O)C(C)(C)c2cccnc2)CC1 N1(C(CC(C)CNC(c2cnc(O)o2)=O)=O)CCC2CCC(C1)S2 c1(NC(c2c(C)cc(SCC)o2)=O)cc(Cl)ccc1C.C12CCN(C1)C(=O)CO2 c1(C(=O)NCC2(CN(C(C(CC)OC)=O)C)CC2)csc2c1CCCC2 C(CCC(C)C(=O)NCCCC(=O)NC1CCN(C(C)=O)C1)OC c1(NC2CCCC(CN(C)C)C2)nccc(=NCCS(=O)(=O)C(F)(F)F)[nH]1 C(C(=O)NC(C1CN(C(c2csc(CO)n2)=O)CCO1)C)(C(C)C)NC(C)=O N1(C(c2cc(C)on2)=O)CC2CC(C1)CN(C(c1cn3c(C)cccc3n1)=O)C2 CCC(C(=O)N(C)CCOC)N(C)C(c1ccnn1C1CCCC1)=O.C1(=O)CO1 c1(C(=O)NCC2(C)CCN(C(=O)CC3CCOC3)C2)cc2n(n1)CCCNC2=O c1(C(C(=O)NCC2CC(NC(c3c(S)ncs3)=O)C2)C)ccncc1C.CC CCC(C(=O)NC(c1nocc1C(=O)NCc1c[nH]nc1C1CC1)C)C(C)(C)CC C1(NC(C(C)CF)=O)CN(C(=O)C(C)(C)c2ccno2)CC1CC1CC1 CC1(C)CC(NC(c2cc(Br)c[nH]2)=O)CN(C(c2coc3c2COC3)=O)C1 N1(C(C2COC3CN(C(C(C)N(C)C)=O)CC32)=O)CCCC2(CCc3c[nH]nc32)C1 c12ccccc1C(c1nnnn1C)NC2CCO.c1(NCC)cccc(C(C)C)c1 N1(C(c2cc(C)c(Cl)cc2C)=O)CCC2(CCC2)C(CNC(=O)C(C)C2CC2)C1 C1(NC(C)=O)CCN(CCn2ccc(C)n2)C1C c1(C(=O)OCC)c[nH]cc1C(=O)NC1CCC(NC(=O)C=CC(C)C)C1 C(=O)(C(C)CC(C)C)NCCOCCOCCNC(c1cc(COC)[nH]n1)=O C1(C(C(N2CCC(CNc3ncc(Br)cn3)CC2)=O)O)CCCCCC1 c1(CCC(=O)NCC2(CNC(C(C)=O)=O)CCCC2)c(C)nc(S)nc1C c1(C(N2CCC(NC(c3coc(C4CC4)n3)=O)C2)=O)ccccc1C1CC1 C1(C(=O)NC(C(=O)OCC)CO)C(O)CCN1C(c1ccccc1OC(C)=O)=O N1(C(CCC(C)O)=O)CC(O)CC1CNC(c1ccnc(F)c1)=O N1(C(CN(C(CN(C(C(C)C)=O)C)=O)CCO)=O)CC(C2CCCCC2)C1 C1(SC(N2CC(CCCCNC(c3cc(C4CC4)on3)=O)C2)=O)CC2CCCC2C1 N1(C(C(C(CC)O)(C)C)=O)CCc2ccccc2C(NC(=O)CSC(F)F)C1 Cc1snc2sc(C(N3CCCC(C(=O)Nc4cnc(Cl)nc4)C3)=O)cc12 Cn1c(C(=O)Nc2ncc(Cl)nc2Br)cc2cc(Cl)ccc12 N1(C(=O)OC(C)(C)C)C(C(=O)N=c2nc(C(F)F)[nH]s2)CCC12CCC2 c1(CC(=O)NCC(CO)NC(=O)C(F)CC2CCC2)csc(Cl)c1 C1(C(=O)OCc2nsc(N3CC(C(O)C(=O)OC)C3)n2)CCCC12CN(CC)C2 c1(CN(C(=O)CCC=CC(C)C)CCOC)ccccc1.C12CC1OC2=O C1(C)(C(=O)NCC2N(C(c3c(CC)nco3)=O)CC2)C=CCCC1 C1(C(=O)NCCCCN(C(CC(CC)C)=O)C)Cc2nnsc2S1 C1(NC(C=CCNC(CC2C(C)CCO2)=O)=O)CC2CC1OC(=O)N2 C1(NC(COCCCC(C)C)=O)CC(O)CN(C(=O)CC(F)(F)F)C1 CCC(O)C(C)C(=O)N1CCCC(NC(c2ccc(=N)[nH]c2Cl)=O)C1 CS(=O)(=O)CCCC(=O)N1CC2C(CNC(=O)CCOc3ccc(Cl)cc3)C2C1 c1(C(=O)NCCC(C)NC(C2(C3CC3)CCCO2)=O)ccc2c(c1)SCCN2 N1(C(CC(C)n2ccnc2)=O)CCCCCC1C(=O)NC1CCCN(O)C1=O C1(C(=O)NCC2C(NC(c3ccc(C(C)(C)C)cc3)=O)C2)C2CC(=O)CC(=O)C12 Cc1cc(O)c(C(=O)N(CC(C)NC(C2CC3CC3C2)=O)C)cc1Br C(C(=O)N1CCN(Cn2cc(-c3ccc(F)nc3)nn2)CC1)(C(C)C)NC(C)=O c1(CC(=O)N(CC)CC2CCN(C(c3ccsn3)=O)CC2)nc(F)c(F)cc1F N(C(=NCc1ccccc1)NC(c1nnc(C2CCC2)s1)C1CC1)CC(=O)NC CN1CCC(C)(C(=O)NC(CC2CC2)CC(=O)NCCn2cnnc2)C1 N1(C(CCCC(C)NC(=O)OC(C)(C)C)=O)C2CCC1CC(O)C2 N1(C(C2OCC(C)(C)C2)=O)CCCN(C(=O)C2=C(Cl)CCCC2)CC1CO c1(C(N2CCC(C#C)(C(=O)NC(C)C(C3CC3)OC)C2)=O)c[nH]c2cnccc12 N1(C(C(C)SCCCC)=O)CCOCC1C(=O)Nc1ccc(O)cc1 c1(OCC(C)C)ccc(C(N2CCC(Sc3ccc(Cl)cc3)CC2)=O)cn1 Cc1cc(CNC(=O)Cc2c(C)noc2C)oc1C(=O)NC(C)C(C)O N1(C(C2N(C(CC3CNC(=O)O3)=O)CCC2)=O)CC2(CC2)CC1CO c1(C(=O)NC(C2CCN(C(C3C(OC)C3)=O)CC2)C)cc2n(c1)CCOC2 c1(C(=O)NCCCCNC(C2CCC3CC23)=O)c[nH]nc1OCC(F)F C(=O)(C1=C2CCCN=C2NN1)N(C(CNC(c1c(CC)sc(=N)[nH]1)=O)C)C C1(C(=O)NCC2CCN(C(Cc3c(C)scc3)=O)CC2O)CCCCN(C)C1=O C(=O)(C1CCc2cc(F)ccc21)NCC1CN(C(CCC(C)SC)=O)CC1C C12(CC(=O)NC(c3cccnc3)C(=O)NCCN3CCCOC3=O)CCC(CC1)C2 c1(OCCC)ccc(CNC2COC(C)(C)OC2)c(C)c1 C1(NC(c2cc3n(n2)CCCC3)=O)CCN(C(C2CCC2)=O)CCC1CO c1(OC)cc(C)c(NCCOCC(C)C)cc1Br Cn1ccnc1S(=O)(=O)NC1CN(Cc2ccc(-c3ccc(Cl)cc3)o2)CC1F C1(OC)CN(C(=O)Cc2nnc(C)o2)CC1NC(=O)C(c1ccc(Cl)cc1)O Cc1cc(C(=O)NCC2(O)CC(NC(=O)CCC3CCCN3C)C2)cc(F)c1 c1(NCc2c(NC(c3c(Cl)cc(OC)nc3)=O)cccn2)c(Cl)c(F)nc(F)c1Cl C=Cc1ccc(C(=O)NCCC2CC(NC(c3cc(C)cc(O)n3)=O)C2)cc1 C12C3CCN(C13)C(=O)CCNC(=O)C=CC(=O)N2.CNC.C(N)(=O)N c1(C(=O)NCC2(C)CCN(C(c3ncc[nH]c3=O)=O)C2)cc2c([nH]1)CCOC2 N1(C(c2c(OC)csc2)=O)C2CCC1CN(C(=O)C(=Cc1ccncc1)C)C2 c1(CNC(C2CNCCCO2)=O)sc2ccccc2c1Cl C1(C(N(CC(=C)C)C)=O)CC12CCN(C(c1nccc(C)c1N)=O)CC2 c1(CC2CCN(C(c3nn[nH]n3)C)C2)c(F)cccc1Cl Cc1cc2cc(SC(C)CN(C)C(C3CC(O)CN3C(N)=O)=O)c(Cl)cc2[nH]1 C=CCC(CNC(c1ccc(C)n1C)=O)C(=O)NC(C)(COC(C)=O)CO C1(C(=O)NC(C(C)(C)O)CO)CCN(C(C2CC23CCOCC3)=O)C(C)(C)C1 Cc1ccc(-n2ncc(C(=O)NC3CN(C(=O)C(C(C)C)N(C)C)C3)c2C)cc1 c1(C(N(C2CCN(C(=O)COCC3CC3)CC2)CC#C)=O)ncc(F)cc1N C#CCC(CC(F)F)C(=O)N1CC(NC(=O)C(CCCC)NC(N)=O)C(C)C1 c1(N)ccc(N)cc1C.c1(C(c2nnnn2C(C)(C)C)SC)nc(Br)cn1C c1(CC)conc1CC(=O)NCC(C1CC1)NC(c1ncsc1C)=O CS(=O)(=O)CC(=O)N1CCCCC1C1CCCN(C(=O)CCc2ccccn2)C1 C(=O)(CCCCCC(=O)NCC1(NC(=O)CCC(C)(C)C#N)CC1)OCC c1(C(=O)NC2CC(C)(NC(CCNC(C)=O)=O)C2)sc2ncnc(N)c2c1C N1(C(C(COC)(C)O)=O)CC=C(CC(=O)Nc2ccc(C(C)C)nc2)CC1 c1(C(=O)NCC(=O)NCCCN(C(C2(C)CC2Br)=O)CC)ccncc1 c1(C(N2CCOCC2CNC(C2C(C)C2C)=O)=O)cnc(NOC)c(Cl)c1 Cn1ncc(C(=O)NCCC2CCCN2C(=O)C(C#N)C2CC2)n1 C1(C(=O)NC(CN(C(c2c(C)n(C)c(C(C)C)c2)=O)C)C)CCCC(C)(C)CC1 Cc1cncnc1C(C1CCC1)NCCCCc1cn(-c2ncccc2C)nn1 N1(CC(=O)NC2(C)CN(C(CCn3ccc(C)n3)=O)C2)CCC(N(C)C)CC1 c1(C(N2C(CNC(c3c(C)nsc3)=O)CC(O)C2)=O)ccc2ncccc2c1 N1(C(C2N(C(CC3CCC(C)C3)=O)CC3CC32)=O)CC(O)(C2CC2)C1 C1(NC(C(c2ccnn2C)C)=O)CCC12CN(C(c1ccc(Cl)cc1F)=O)C2 CC1CN(C(=O)CCF)CC(C)C1NC(=O)C=Cc1cnc[nH]1 c1(C(=O)NC(C(=O)N(CCC)CCC)c2ccco2)ccn(C)c1C N1(C(C(C(C)O)N(C)C)=O)CCOCC(C)(CNC(=O)CCN2CCCC2)C1 c1(C(N2CCC(O)(C(=O)Nc3c(C#N)cno3)C2)=O)cc2ncsc2[nH]1 n1(CCCC)ccc(C(=O)NC(C)CCNC(=O)C(O)(C2CC2)C2CC2)n1 O=C(CCCN=c1nc(N2CCC3CC3C2)c2ccccc2[nH]1)NCC(F)F CC1(C(=O)NCC2(C)CCCN2C(c2cc3occc3s2)=O)CCCC1(F)F C(N=c1[nH]c2ncc(Br)cc2s1)C1CC(=O)NCC1 C=CCC(CC(C)C)C(=O)N1CCC(C)C(CNC(C2CC2C2CC2C)=O)C1 Nc1nccnc1C(N1CCOC(CNC(=O)Cn2nnc(C3CC3)n2)C1)=O c1(CC)cncc(C(=O)N(C2CCCC2)CCNC(=O)CCN2CCOCC2)c1 C(=O)(CC(C)C(C)(C)NC(c1cccnn1)=O)NCC(CC)CC C1(NC(CCNS(C)(=O)=O)=O)CCN(C(c2ccc(=N)[nH]c2Cl)=O)CCC1(F)F CCC(C)(O)C(=O)N1CSCC1C(N1CCC1CNC(=O)OC(C)(C)C)=O C1(C(=O)NC2(C)CN(C(=O)C(F)C(C)(C)O)C2)CCc2ncnn2C1 c1(C(C)=O)ccc(S(=O)(=O)C(=O)NC2(CSc3ccc4ccsc4c3)COC2)cc1 C1(C)(C(=O)NC2CC(NC(CCc3c(C(=O)OC)nco3)=O)C2)CCCC1(F)F N1(C(=O)N)CCCCC1.C(=O)(NCCNC(=O)OCC)OC c1(NC)cc(C(=O)NC2(C)CN(C(c3cnc(C(C)(C)C)o3)=O)C2)cc(Cl)n1 c1(C2C(C(N(C(c3ccccc3)C(C)C)C)=O)C2)csc(C(F)(F)F)n1 CC(C1CCCCC1)=CC(=O)NCC1C2CN(C(=O)C(=O)NC3CC3)CC12 Cc1cc(C(N2CC(CNC(=O)C(F)(F)C3CC3)C2)=O)cc(S(C)(=O)=O)c1F N1(C(C2(OCC)CCCC2)=O)CCC(N(C)C(C2(C)CC2(F)Cl)=O)CC1 O=C1c2cccnc2N(C2C3C(CCCC2)NC(=O)N3)CCCCN1 CC1CC(C(=O)NCCCc2cnc[nH]2)CCN1C(=O)COCc1nc[nH]n1 C1(NC(c2[nH]cc3c2CCCC3)=O)CC2CCCC(C1)N2C(C1(F)CC1)=O C(=O)(C(CCF)NC(=O)C(C)CC1CCC1)NCc1cc(CC)no1 CC1CN(C(=O)COC2CC(NC(C3CC(C)(C)C3)=O)C2)CC(C)(C)C1 c1(C2CCC(=O)N2)ccc(NC(C23CC2CN(C(c2coc(CO)c2)=O)C3)=O)cc1 C1(NC(C(CC)=CC)=O)CC2CN(C(c3ccncc3Cl)=O)CC2C1 c1(SCCC(=O)Nc2nc(NC(=O)OC(C)(C)C)sc2)coc2cc(Cl)ccc12 Cc1ccc(Cl)cc1CN1CCCC1CNC(c1cn(C2CCOCC2)nn1)=O C1(C(=O)NCc2c(CC)nn(C)c2)CC(C23CC(C2)C3)CN1 C1(C(N(CC(C)(C)C(=O)N2CCC(CO)C2)C)=O)C2CCC(F)(F)C12 C(=O)(C1CCCc2cncn21)N1CC=C(CNC(C2(COC)CCCC2)=O)CC1 N1(C(C2(C)CCCN(C(C(C)S(C)(=O)=O)=O)C2)=O)CCCCC(C)(C)C1 c1(C(N2C(C(=O)Nc3c(COC)nn[nH]3)C(CC)CC2)=O)cc(OC)ccc1N c1(OC)cc([N+](=O)[O-])c(C(=O)Nc2ccc3occc3n2)cc1OC C1(C(C)(C)C)CN(C(=O)C=Cc2cn[nH]c2)CCN1C(=O)COCC(F)(F)F N1(C(C2(C)CCCCCC2)C(=O)NC(C(=O)OC)C)CCCC(C)(C#N)C1 c1(C(=O)NC2CC(NC(CC(CC)O)=O)C2)cc2cccnc2s1 C=CCC(CC)C(=O)NCCOCCC(=O)NC(CO)CC(F)(F)F C1(CC(=O)NCC2(CC(=O)OC)CC2)CCCN(C(C2CCCN(C)C2)=O)C1 N1(C(C2C(CNC(c3c(CC)c[nH]c3)=O)CCC2)=O)CC2(C1)CN(C)CCO2 CC(C)(C)C(O)CONC(C1C=CCN1C(c1ocnc1C1CC1)=O)=O N1(C(C2(C)CN(C(C3(OC)CCCC3)=O)C2)=O)CC2CCC(C1)C2CN(C)C N1(C(C=C(CC)C)=O)CCOCC(COC)C1 c1(CSC)cnc(CNCCC(F)(F)CO)nc1 c1(Cn2c(C3(C)CCC(=O)O3)nc(-c3ccco3)n2)ccc2ccccc2c1 c1(OC)ccc(NC(C23CC(CO2)N(C(c2ccccn2)=O)C3)=O)cc1C N1(C(C(C)OCCCC)=O)CCCCC1CN(C)C(c1cccnc1)=O C12(C(=O)NC(C(C)O)CO)CCC(NC(C3COCCC3C)=O)(CC1)C2 C1(C(=O)NC2(CO)CN(C(c3cscn3)=O)C2)CCCCC1F c1(C(=O)NCC2(CCNC(c3cc(C(C)C)no3)=O)CC2)cn2c(n1)CCCC2 C1(CNC(C(C(=C)C)(C)C)=O)CN(C(c2c(C)nn(C)c2N)=O)CC(C)(C)C1 CC(C)C(CO)C(=O)N1CCC(N(C)C(c2ccc(F)nc2F)=O)CC1 C12(C(N(C3CC(OCC)C3)C)=O)CC(CO)(CN1C(c1n[nH]c(C)c1C)=O)C2 c1(OC)cc(C(N2CCN(C(=O)CCN(C)C)CC2C(C)C)=O)c(OC)cn1 Cc1nc(C(N2CCC(O)C(NC(c3cc(F)ccc3F)=O)C2)=O)c(=O)[nH]c1C n1(CC)c(C)cc(C(N2CC(NC(C3C(C)(C)C3(C)C)=O)C(SC)C2)=O)c1C c1(C(=O)NCC(=O)N(CCCCN(C(c2cc(C)sn2)=O)C)C)ccc(O)cc1 c1(OCCOC)ccc(F)cc1C(=O)NC12CC(C1)N(C(=O)CN(C)C(C)=O)C2 c1(OC)ccc(F)c(CN2CCC2C(=O)NC(c2cccc(Cl)c2)C)c1 C=CCC(C)(O)C(=O)NCc1ncccc1C(=O)NCC(=C)F C1(C(=O)NCC(C)(CO)NC(=O)CC2CC2)CC2CCC1CC2 c1(CC)ccc(S(=O)(=O)N2CCC(F)(NC(=O)Nc3cc(Br)ncc3Br)C2)cc1 C1(NC(=O)NCC2CC=CC2)(CO)CC2CCC1C2 c1(NC2C(CC)CN(C(=O)C3=CCCO3)CC2)ccc(C)cc1[N+](=O)[O-] C(C(C)(C)C(=O)NCC1CN(C(=O)CC(=O)N(C)C)CC1C)NC(C)=O Nc1c(F)cc(C(N2CC3CCC(CNC(c4sccc4Cl)=O)C3C2)=O)cc1F c1(C(=O)NC2CN(C(C(C=C)(C)C)=O)CC2(C)C)ccc2[nH]ccc(=O)c2c1 C1(CN(C(c2cnn(CC)n2)=O)C)CN(C(C2CCCCO2)=O)CC12CC2 Cc1ccc(CCC(=O)N2CC(OCCNC(C3(C)COC(=O)C3)=O)C2)cn1 c1(CC)ccc(C(=O)NC(C)CCCCNC(C2CC2CF)=O)c(C)n1 C1(CNC(C23CCC(C2)C3)=O)CC2CN(C(C3(C(=O)OC)CC3)=O)CC12 C12(CNC(COCC)=O)COC(CN)(C1)C2.C1(CCC(=O)C2C(CC)C2)CCOCC1 C1(OC)CN2CCCC2(C(=O)NCCCn2cc(CCC3CCCCC3)nn2)C1 C1(CNC(C=CC)=O)C(C)CCN1C(c1cc(C(N)=O)c[nH]1)=O N1(C(c2c(C)n(C)nc2)=O)CC2CCC(C1)N(C(c1ccn3cncc3c1)=O)C2 C1(C(=O)NCCN(C(=O)CC2CC=CCC2)CCOC)CCc2nnc(O)n2C1 C(CNC(c1cc(C2CC2)[nH]n1)=O)(C(C)(C)C)NC(C1C(C)C1C)=O C1(C(N2CCC(C(=O)NCCC(C)CO)C2)=O)CC2CCC(C1)C2 N1(C(CCCCCOC)=O)CCC2(CCN(C(=O)CCn3cc(C)cn3)CC2)C1 C12(C(N(C(CCNC(C3(CC=C)CC3)=O)C)C)=O)CCC(N=[N+]=[N-])C1C2 C1(NC(CCOCCC)=O)CN(C(=O)CSCC2CCCO2)CC1(C)C CCC(CCCC(=O)N1CCC(C)C1(C)C)NC(=O)CCCCNC(C)=O C=CC(C)CC(=O)N1CC(C(=O)NOCCC(C)O)C(C)C1 c1(OC)ccc(OC)c(C(=O)NCC(O)CN(C(=O)CCCCCF)C)c1 N1(C(C(C(C)C)OC)=O)C2CCC1CC(NC(C1C=CC=CC=C1)=O)C2 c1(C(=O)Nc2ccc(C(=O)NCC3CCC3)nc2)cccc(F)c1I c1(C(=O)NCC(CC(C)C)NC(C(CC#C)C)=O)cnn2cc(OC)ccc12 CC12CC(C(N3CCC(NC(C4CC5(CC5)CO4)=O)C(F)C3)=O)(CCO1)C2 CC1(C)C(NC(=O)Cc2cnsc2)CC1CNC(c1cnc(O)s1)=O N1(C(c2cc(COC)sc2)=O)CCN(C(C2CCCCC2F)=O)CC(O)C1 CCC(Cc1ccccc1)C(=O)NCC1CC(O)CN1C(=O)CN(C)C1CC1 C1(CN(c2ccc(Cl)cc2)CC)CCCN1NC(=O)C1CC1 c1(C(=O)NC(CC)CNC(C2CCN(C(C)=O)C2)=O)c(O)noc1C N1(C(CCC(=O)NC)=O)CC(C)CN(C(c2[nH]nc(OC)c2Cl)=O)C(C)C1 C=C1CCC(C(=O)NC(C(=O)N2CC(C)(C)C2C(=O)OC)C(C)C)CC1 N1(C(CCC2CCN(C(CC3N(C)CCC3)=O)C2)=O)CCC(C)(CCO)C1 N1(C(COCc2c(C#C)cccc2)=O)CCCC1C1CCCCN1C(C)=O c1(C(N(C2CN(C(C(C)OC)=O)C2)C)=O)ocnc1C C1(C(N(CCOCCN(C(C#CC(C)C)=O)C)C)=O)CCC(C)(C)OC1 c1(OCCC(N2CC(O)(CN(C(c3cc(C)sn3)=O)C)C2)=O)ccc(F)c(F)c1 N1(C(C2=C(C)OCC2)=O)CC2(NC(c3cc4ccncc4[nH]3)=O)CCCC2(F)C1 c1(NC(C2C(CNC(CC3(NC(N)=O)CC3)=O)C2)=O)cccc(CO)n1 c1(CCNC(c2c(C)cnn2C)c2nnnn2C(C)(C)C)ccc(Cl)c(F)c1 CCC(CCC(=O)NC1CCSC1)NC(=O)Cc1ccco1 CC1(C)CC(CNC(c2ccc(C(F)F)s2)=O)N(C(c2cc(O)cc(O)n2)=O)C1 C1(C(=O)NCc2cc(-c3cccc(OC)c3)no2)CCn2ccnc2C1 Cc1nc(C(C2CC2)NC2CC2C)sc1-c1ccccc1 C(C#N)(N(CC)CC)OC.C(C)(C)O c1(C(=O)OCC)cc(-c2ccnn2C)sc1NC.c12cc(cn1C)NC2=O C(=O)(C(C)(C)CCCNC(c1cccc(CO)n1)=O)NCC=C c1(CCC(C)NC(=O)CC2CN(C(=O)C(CN(C)C)N(C)C)C2)cccnc1 N1(C(C(C)(C)OC(C)C)=O)CCC(CO)C(NC(C2CC(C)CC(=O)N2)=O)C1 C(N1CCCC(O)(CO)C1)n1c(-c2ccc(CC(C)C)cc2)nc(C2CC2C)n1 Cc1c(C(N2CCC(NC(=O)C(C)n3cccn3)C2C)=O)csc1Br N1(C(Cc2cc(C)on2)=O)CCCCC1CN(C)C(C1(CO)CCCC1)=O C=CC1(C(=O)NC2CCC(NC(C3CCCN3C(C)=O)=O)C2)CCCCC1 C(CNC(=O)CC1(NC(=O)C(C)N(C)C)CCC1)(CNC(=O)COC)OC CC(C)CC(C(=O)NC1CC12CC(NC(=O)CC(C)(C)O)C2)n1ccnc1 c1(CC)ccccc1C(=O)NC(C(=O)N1CC=CC1CF)C(C)C C1(O)(CC(=O)NC2CCSCC2)CCN(Cc2csc(Br)c2)CC1 CCC(C)(C)CC(=O)NC1C2CCN(C(=O)Cc3c[nH]nc3O)C12 C(=O)(CC(F)(F)C(F)(F)Br)NCc1c(Cn2cc(C(CC)N(C)C)nn2)nco1 c1(CN2CC(C(=O)Nc3ccnc(Cl)c3Cl)C(F)(F)CC2)cc(Cl)cc(Cl)c1O CC(C)CC(C(=O)NCC1(N2CCCC2)CC1)N(C(=O)CC1C=CCCC1)C c1(C(=O)NC(C(C)NC(c2ccc(COC)o2)=O)C)c(Br)ccc(F)c1C C(CCC(=O)NC1(C)CC(C)(C)C1)(C(C)C)NC(c1c(C)ccc(O)c1)=O C1(CC(=O)NC(c2ncc(C)s2)C)CCCCN1C(=O)Cc1nonc1C c1(C(N(C2CC(C(=O)NCc3cn(CC)nc3)C2)C)=O)ccc(CO)c(Cl)c1.C(C)=O c1(OC)cc([N+](=O)[O-])ccc1CNC1CCC(C(N2CC3CC3C2C#N)=O)CC1 C1(O)(CNC(C(C)C(F)F)=O)CCCN(C(=O)CN2C(=O)CN(C)C2=O)C1 C(=O)(C(F)(F)c1cccnc1)NC1CC(CNC(C2CC(n3cnnc3)C2)=O)C1 C=CC(CC)CC(=O)NC(CO)C(=O)N1CCC(CC(C)(C)C)C1 Cc1cc(CN2CCC(C(N3CC(CC(=O)NC(C)(C)C)C3)=O)C2)cc(C)c1 C1(C(=O)NCC(NOC)=O)CCCCN(C(=O)C(C)CC(F)F)C1 N1(C(=O)CCCCC2CC2)CC(C(=O)NCCC2CCOCC2)C(F)(F)C1 C1(C(=O)OCC)CC(F)(C(N2CC(N(C(=O)CC3CC4CC4C3)C)C2)=O)C1 Cc1ncn(C)c1NC(C1CCC(NCc2ccncc2O)CC1)=O C1(C(N2CCCC(NC(CCCOCCC)=O)C2)=O)CCCC(C)(C)O1 c1(C(=O)NC(c2nc(C)cs2)CC)ccccc1-n1cc(C2CCCSC2)nn1 C12(CCCC1)CNC(=O)C(=O)N2.C12CN(C1)C(=O)C2.C1(SCC)CC1 c1(C(=O)NCC(CC)NC(C2CCCCN2C)=O)c[nH]c(=N)c(C)c1 N1(C(c2cc(C(C)C)no2)=O)CCC2(CC1)CC2NC(=O)COC1CCCOC1 CC1(C)CN(Cc2c(Br)cccc2Br)CCC1NC(c1ccc(C(F)F)cn1)=O c1(COC)nc(=N)[nH]cc1C(N1CCOCC1CCNC(c1cnsn1)=O)=O C(=O)(C(C)(O)C(C)C)N(CC(Cc1ccccc1)NC(CSCCOC)=O)C C1(C(=O)NCC2(Nc3ccnc(F)n3)CCC2)CCCC12OCCO2 C1(C(=O)NC(c2c(CC)cccc2)CC(=O)O)CC(C2CC2)=NO1 c1(C(=O)NC2CCC(CNC(=O)COc3ccon3)C2)c(F)cncc1Cl c1(C(N(CC(C)NC(=O)CC(O)C2CC2)CC)=O)cccc(C)c1O CC1C(NC(c2ccc(Cl)cc2F)=O)CCCN1C(=O)CN1C(=O)CN(C)C1=O N1(C(C(C)NC(C)=O)=O)CCC(C)C(NC(c2csc(Cl)c2)=O)C1C C(=O)(CC(=O)N(c1ccccc1)C)OCC=C.C1C(=O)NC(=O)O1 N1(C(C(CSC)OC)=O)CCC(CCNC(=O)CC2CCNC(=O)C2)CC1 C1(C(N(CC(CC)NC(c2coc(Br)n2)=O)C)=O)CCCCNC1=O CC#CCCC(=O)N1CCCC1C(N(C)CC1(OC)CC(C)(C)C1)=O C1(C#N)(C(=O)NC2(C)CCN(C(COCCOCC#C)=O)C2)CCOCC1 CC(C(=O)N1CC(C(C)(C)O)C1)N(N1CC(CF)C1)C.C(CF)C=O c1(C(=O)NC2C(CC(=O)NCCN(CCO)CC)CCC2)cc2n(n1)CCC2 C1(COC)CC(CNC(=O)Cn2cc(Cl)cn2)N(C(C2CNC(=O)O2)=O)C1 C1(CC)CN(C(=O)CC(=O)NCC(F)(F)F)CCN1C(c1cc(CSC)on1)=O C1(NC(C=C(C)C(C)C)=O)CN(C(=O)CCc2ccc(C)cc2C)CC12CCC2 C(CCCC(=O)NC(C(=O)N(C)Cc1ccoc1)C1CCOC1)OCC N1(C(CC2(C)CCOC2)=O)CC2(CO)CC1(C(N1CCC(CO)CC1)=O)C2 N1(C(C(=O)Cc2ccccc2F)=O)CCCC2(NC(c3ccncn3)=O)CC2C1 c1(C2(C(=O)NC3CC(n4ccnc4CO)C(O)C3)CCCC2)c(F)cccc1F c1(CC(=O)N(CC(=O)NCCCF)C)ccccc1 c1(C(=O)NC2CCCN(c3nccc(C)n3)C2)cc2cc(F)ccc2s1 C(=O)(C1Cc2c(Cl)cccc21)NC1(CC=C)CCN(C(c2c[nH]cc2CC)=O)C1 Cc1nc(C(=O)NCC(C)NC(=O)C2=CCCO2)c(C)s1 c1(N(C)Cc2ncc(Br)s2)nc2c(c(=NCC3CC(C)(C)CCC3O)[nH]1)CSC2 CC(C)CCC(C(=O)N1CC(O)C(C2CC2)C1)N(C(=O)C=CC(C)(C)C)C1CC1 C=CCCCCC(C(=O)NCCO)N1CCN(C2CCC2)CC1.C1(C)CCCO1 C(=O)(C1=C(Cl)CCC1)N1C(CN(C(C(c2cc(C)oc2C)C)=O)C)CCC1 c1(OCC(=O)N(C)CCN(C)C(C2C3CCN2CC3)=O)ccc(F)cc1F C#CCC(C(=O)OC)NC(=O)C(C)(C1CC1)N(C)C(c1ocnc1CC)=O CC1CC2(CC(N(C(=O)C(C)C(C)N3CCCCOCC3)C(=O)OC(C)(C)C)C2)C1 C1(CNC(C2C(c3cn(C)nc3)C2)=O)CC2CCCCC2N1c1nnco1 c1(C(N2CCC3(CC2)CN(c2nnc(C4CC4)s2)C3)=O)nccc2ncncc12 C(CCC(C)C)(C(=O)NC1(C)CCCCC1(C)C)NC(c1n(C=C)ncc1)=O c1(C(N2CCC(CCC(N3CCC=C(Cl)C3)=O)C2)=O)cnn2ccccc12 C1(c2c(C(=O)OCC)non2)C2CC3C(C2NC(=O)CSCC(C)C)C13 CC1=C(C)CC(C(N2CCCC(C)(NC(c3ccc(C4CC4)cc3)=O)C2)=O)CC1 C1(CN(C(C2CCCC(F)C2)=O)CC)CCCN(C(c2cc(CC)no2)=O)C1 C1(NC(c2cc(C)ncc2)=O)CN(C(c2cnc(O)n2C)=O)CC2CCCC12 N1(C(c2c(CC)c[nH]c2)=O)CC(C)C(Nc2ncnc3ccccc23)C(C)C1 C12(CNC(C(C)NC(=O)Cn3cnnn3)=O)CCC1CN(C(c1ccc[nH]1)=O)C2 N1(C(c2nc(NC(C)=O)sc2)=O)CCC(NC(=O)CCC2CC(F)(F)C2)C1C N1CC2OCC(NC(Cc3cc(CC)on3)=O)C(C2)C1.C1(C)(C(=O)N)CCCC1O Cc1nc2cc(C(=O)NC3CC(CNC(=O)C(O)CC(C)C)C3)cnc2s1 CC(C)(CNC(C1(C2CCCCO2)CC1)=O)CC(=O)NC1CCC2CC12 N1(C(C(C=C)CC)=O)CCC2(CCN(C(=O)C(C)n3cccn3)CC2)C1 OC1(c2ccccc2)CCN(N2CCC(O)(c3ccc(F)cc3)CC2)CC1 c1(C(=O)NC2(CCNC(c3c(C)ccnc3)=O)CC2)cccc(C)c1Cl C1(CCNC(=O)CNC(C2CCC2)=O)CSCCN1C(=O)CCc1cnc[nH]1 C(C)(N=c1[nH]c(=NCC(C)Oc2ccccc2)[nH]c2ccsc12)c1c(C)cccn1 C(CC(O)C(=O)NC(Cn1ccnn1)C(=O)NCC1C2CCCC12)SC N1(C(c2ccc(C(F)F)cc2)=O)CC2CC(NC(c3c(C)nns3)=O)C1C2 N1(C(c2c(O)ccc(C)n2)=O)CC2CCCC2(NC(=O)C=C2CCCCC2)C1 c1ccc(C(C2CCCC2)Cc2csc(CCN3CCOCC3)n2)cc1 N1(C(c2cccc(NC(C)=O)c2)=O)CCCN(C(C2CC2C(N)=O)=O)C(CO)C1 N1(C(C2CC(CNC(CC3CCC(C)C3)=O)OC2)=O)CCOC2COCC2C1 C1(CNC(C2(SC)CCC2)=O)CN(C(C2CC=CC2)=O)CC(C(F)(F)F)O1 C1(NC(C2CCCC23CC3)=O)CN(C(=O)CCc2ccc[nH]2)CC(F)(F)C1 N1(C(Cc2ccc(C)o2)=O)CCC(C)(CCNC(c2c(C)nn(C)c2C)=O)CC1 c1(C(=O)OC)cnc(C)[nH]c1=NC(CCN(C)C(C1CCCCC1)=O)C(C)C Cc1cc(C=CC(=O)NCC2CCC(NC(=O)C(O)C3CCC3)CC2)c[nH]c1=N O=C1NC2(CCN(C(C3CC(F)(F)CN3Cc3nc(Br)cs3)=O)CC2)CO1 C1(OC)CN(C)C(C)(C(=O)NCC2CC(NC(=O)CCc3ccc(C)cc3)C2)C1 C1(CN(C(c2ccn(C)n2)C(=O)NC)C)CCc2nccn2C1 c1(C(=O)NC2CCCC(N(C)C(c3coc(O)n3)=O)C2)c(F)c(N)cc(Cl)c1F N1(C(C(C)(C)c2sccc2Cl)=O)CC(O)CC2CCCCC12 CCC(C)CCCC(=O)NC1(C(=O)NC2CC2(C)C(F)F)CCCCC1 C(c1cnc[nH]1)=CC(=O)NC1CC(NC(=O)CCC2CC(F)(F)C2)C1 c1(C(=O)NC2C(NC(Cn3c(C)ccc3C)=O)CC2)cc(F)c(CO)c(F)c1 C1(CNC(C2CCCCO2)=O)CN(C(c2cc(C3CC3)cs2)=O)CC1O C1(CNC(C(CC)CC)=O)Cc2ccccc2CN1C(=O)Cc1cccc(Cl)c1 c1(OC)cc(C(=O)NCC(C)(C)CN(C)C(C2CC2C(C)(F)F)=O)ccc1Cl C1(C2CCCN(C(=O)C(F)C3CCC3)C2)(NC(c2n(C)c(C#N)cc2)=O)CC1 C12=CNNC1=NC(=O)C1(C)CCN1C2=O.c1(OC)cc(Nc2ccccc2)ncn1 CN1CCC(N(C(=O)CCN(C)Cc2ccc(F)cc2)C)CC1 N1(C(c2cc(CCC)on2)=O)CC2C(C(N3CCC(C(C)C)CC3)=O)C2C1 CCCC(C(=O)N1CCOC(CC(=O)NCCc2cscn2)C1)NC(C)=O c1(NC(C2C=CCN2C(c2cc(O)ccn2)=O)=O)cccc(-n2cc(Cl)cn2)c1 C1(CN(C(C(C)OCC)=O)C)CCCCN1C(c1cncc(O)c1)=O C1(O)(CNC(C(CC(=C)C)C)=O)CCCN(C(=O)CN2CC(C)(C)C2)CC1 C(=O)(C(O)CC(C)C)NC1(C(=O)NCCc2cc(C)n[nH]2)CCN(C)C1 c1(C(N(C2CCCCN(C(=O)CCCC#N)C2)C)=O)cc(C2CC2)nc2ccnn12 C12(C(N3C(C)CC(NC(COCCOC)=O)C3)=O)CCCC1C2(F)F c1(C(=O)NCC(c2ccccn2)N(C(CC)C)C2CC2)cnc2c(c1)COC2 Cc1cccc(Cl)c1C(c1nnnn1C1COC1)NC1(c2ccccc2)CC1 C1(C(=O)NCCOCCNC(CCOCC)=O)CN2CCN1CC2 C=C(C)C(C)(O)C(=O)N1CCN(C(c2sc(C)nc2C)=O)C(C)C1 C1(CC)CC2(CCC2)CN1C(c1cscc1-c1cccc(OC)c1)=O C1(C(=O)Nc2cccc(NC(C(C)O)=O)c2)CCc2nccn2C1 CCC(CC)(C(=O)NC12CC(C1)N(C(=O)NN1CCCC1=O)C2)c1ccccc1 C1(CNC(C(COC)(F)F)=O)CN(C(c2coc(C)n2)=O)CC12CC2 c1(C(=O)NCCN(CC(C)O)C(c2sc(CC)c(C)c2)=O)c(C)[nH]c(C)c1C c1(C(N(C(C)CCNC(c2cc(O)ncn2)=O)C)=O)ccc(O)cc1Cl c1(C(N(C)CC=CC(N2CC(O)(CCO)C2)=O)=O)cc(O)n(C)n1 c1(C(CC)(C)C)n[nH]c(=NC(C)(COC)CNC(=O)Cc2c(F)cccc2Cl)s1 C1(C(N)=O)(CNC(C2(C(C)(F)F)CCC2)=O)CN(C(C2CCCC2O)=O)C1 C1(C(=O)NCCC=C=C)CCCC(NC(C2(C)COC(=O)N2)=O)CC1 C1(CCCC)CN(C(=O)CCOC2CC2)CCN1C(c1cnn(C)c1F)=O C1(NC(C(C)Sc2nnnn2C)=O)CCCC(CO)CC1.c12ccc(cc1)[nH]2 C(=O)(C(=O)C(C)(C)C)N(C1CC(C(=O)NCCOC(C)C)C1)C Cc1ccc(S(=O)(=O)N2CCN(C(=O)CCS(C)(=O)=O)C3CC23)cc1C C1(NC(CNC(C)=O)=O)C=CCC(C(=O)NCCC2CC=CCC2)C1 N1(C(c2cnc3snc(C)c3c2)=O)CC2CC(C1)CN(C(=O)CC(C)C(F)F)C2 C1(C2CCC2)(C(N2CCN(C(CCCC)=O)CC2)=O)CC1(F)F C(CC(F)F)(C(=O)NCCCN(C1CC1)CC)OC.c1(C(=O)N)cn(C(C)C)nc1C CCC(C)(C)C(C)CC(=O)N1CCCC(n2cc(-c3cnc(O)c(C)c3)nn2)C1 C1(C(C)NC(=O)CCN(C)C)CCN(C(=O)C(C)c2cc[nH]n2)CC1 C1(N(C(CN2CCN(C)CC2)=O)C)CN(C(c2ccccc2CO)=O)CC12CC2 C1(NC(C(C)=C(C)C)=O)CN(C(C2CCOC2(C)C)=O)CC12CC2 c1(C(=O)NCC2(NC(c3c(CCC)n[nH]c3)=O)CCCC2)cc(Cl)c(Cl)cc1N N1(C(CN(S(C)(=O)=O)C)=O)C(CNC(C2(C)CC=CCC2)=O)CC2CCCC12 c1(OC)cc(CN2CCC(C(C)NC(=O)Cn3cccn3)CC2)cc(Br)c1 C1(NC(c2nnn(-c3ccc(F)cc3)c2C2CC2)=O)CC2CCC1C(O)C2O C1(NC(=O)CC2CC2C2CC2)CC2CC(NC(c3ccccc3O)=O)CC12 c1(C(N2CC(C(=O)NC(C3CCCC3)C)(CC)C2)=O)ccnc(C)c1 c1(CC)c(F)c(-c2nc(-c3cc(C)n(CCOC)c3C)no2)cc(F)c1F C1(CSCC)CCN(C(=O)NCc2ccc(C(C)C)cc2)CC1 c1(C(N(CCC(C)NC(c2c(C(C)C)noc2)=O)C)=O)nccnc1C(F)(F)F c1(CCC(N2CCC(CNC(C(CCOC)C)=O)C2)=O)ccc(O)c(F)c1 N1(C(CCC(=O)NC)=O)CC(CNC(=O)C2=CCCO2)CC(C)(C)C1 N1(C(Cc2c(OC)cccc2)=O)CCC2(CCCC2C(N2CCC(C)C2)=O)C1 N1(C(C(CSC)(C)C)=O)CCC2(CCCCN(C(C3(F)CCCN(C)C3)=O)C2)C1 C(C(CC(C)C)C(=O)NCC1CN(C(=O)Cc2cnoc2)CCCO1)OC C1(O)(CN(C(c2[nH]cc(CC(C)C)c2)=O)C)CCN(C(C2(F)CC(CF)C2)=O)C1 Cc1cc(C(=O)N(C)CCOCCCN(C)C(C2CC3CCC23)=O)oc1C C12(C(N3C(CN(C)C(c4cnc(Cl)c(F)c4)=O)CC(F)C3)=O)CC=CC(C1)OC2 N=c1[nH]c(C(=O)NC2CC(NC(=O)C(O)C3CC3)C2)c(-c2ccccc2)s1 Cc1cccc2[nH]c(C(=O)NC3CCCN(C(=O)C(C)C4CCC4)CC3)cc12 c1(CCC)onc(C)c1C(=O)N(CC(C)NC(=O)CN1CCCC(C)C1)CC CC1CCOC1CC(=O)NCC1CCCC1CNC(=O)Cc1cnn(C(F)F)c1 c1(NC(C2C(CCC)CCC2)=O)ncnc(Cl)c1C(N1CCCC1(C)C(C)C)=O C(C)(C(CC(=O)NC(C12CCC(CO1)C2)C)NC(=O)CNC(=O)CN(C)C)OC N1(C(c2cc(C#N)no2)=O)CC2CCN(C(C3CCCC(F)(F)C3)=O)CC12 C1(CN(C)C(=O)NCC(C)(C)CN2CCCC2)CC(CN)CC1O CC(C(=O)N(CCCCNC(=O)C(C)C(=O)NC(C)(C)C)C)c1cc[nH]n1 c1(OC)ncc(Cl)cc1C(=O)NC1CC(NC(C2CC=CCC2)=O)C1 C(=O)(CCCCCCC(=O)OC)N1C(CNC(c2n(CC)ncc2)=O)CCC1 Cn1c([N+](=O)[O-])cnc1C(N1CCCN(c2ccc(C(F)(F)F)nn2)CC1C)=O c1(OCC)ncc(C(=O)NC(C(=O)NCC2COC(C)(C)C2)C2CCCO2)cn1 N1(C(CC(=O)NCC#C)=O)CCC2CN(C(=O)C(C)(COC)CC)CC2C1 c1(OC)ccc(NC(=O)C(=O)NC2CC(CC(=O)OC(C)(C)C)C2)c(C)c1 N1(C(CCCCCC)=O)CCC(C)(C)C1CC(N1CCSC2(CCC2)C1)=O c1(C(=O)NCC2CC(NC(CC3CC(=C)C3)=O)C2(C)C)nc(C(C)C)ccc1N Cc1c(C(=O)NC(C(N2CCC(O)CC2)=O)C2CCCC2)cccc1Cl c1(CC)noc(COCC(=O)N(C2CN(C(=O)C(O)c3ccco3)C2)C)n1 c1(C(N2C(CNC(C(C)(C)OC)=O)CC2)=O)ccc(=O)n(-c2cnn(C)c2)c1 Cc1cc2ccc(C(=O)NCC(CO)NC(=O)C(C)S(N)(=O)=O)cc2o1 C1(C(=O)NCC2CCCN(C(COCC=C)=O)C2)Cc2ccc(C)cc2S1 C1(N(C)C(c2cncc(C(F)F)c2)=O)CCCN(C(c2cscc2CO)=O)CC1 Cc1cc(C(N2CC(NC(=O)CCS(C)(=O)=O)C2)=O)cc2nn[nH]c12 C1(NC(c2c(SC)n(C)nc2)=O)CCCN(C(C2CC(N(C)C)C2)=O)C1C c1(NC)ccccc1C(=O)NC(C1CCCN1C(C1CCCC12CC2)=O)C c1(C(=O)NCC(C)(C)Cn2cc(-c3ccc(Br)cc3)nn2)ccn2ncccc12 C(CCC)(C(=O)NCCCC1(NC(=O)CC2CCN2C(C)=O)CC1)=CCC c1(C(N2CC(OC)C(NC(=O)CC3C=CCC3)C2)=O)cc(C2CC2)ccc1Cl C#Cc1ccc(C(=O)NC(c2n[nH]c(C)n2)C(=O)N(CC(C)C(F)(F)F)C)cc1 C1(C(N2C(C(=O)NCC3(O)CCCC3)CSCC2)=O)CC12CCOCC2 c1(C(C(=O)OC)N(C)C(c2cc(NC(C)=O)cs2)=O)cccc(OC)c1 C1(C)(CC)C=C(C(=O)N2CCN(C(=O)CCOCCCOC)CC2CC(F)F)C1 Cc1cnnc(O)c1C(=O)NCCCCC(C)NC(=O)C(O)CN(C)C c1(CC(N2CCN(C(CN(CCOC)C)=O)C(CO)C2)=O)nc2cccnc2[nH]1 C1(F)(CNC(C2(C)CC=CCC2)=O)COCCN(C(c2cccnc2O)=O)C1 c1(C(N2CC(F)CC(NC(C(C)CO)=O)C2)=O)ccc2c(c1)CCCS2(=O)=O C1(CCNS(C)(=O)=O)CCCN1N1CCC(C2CCCC2)C1 O=C(CC(=O)NC1COCC1NC(=O)CC1CC2CC2C1)NCC1CC1 CC1(C)CC(C(N2CCOCC2C2CC2)=O)CCN1C(c1cc(Cl)c[nH]1)=O c1(C(=O)NCC(C)(CO)NC(c2nc(C(C)OC)oc2)=O)c(C)cnn1C CC1CCC(CC(=O)NC2CC(NC(c3cc(C4CCOC4)[nH]n3)=O)C2)OC1 C1(CC(=O)NCC(C(=O)OC)(F)F)CCCN(C(=O)CC2COCC(C)O2)CC1 C(C(COC)C(=O)NC1CN(C(=O)CCC=Cc2ccccc2)CC1SC)OC C1(NC(c2cccn2C2CC2)=O)CCCN(C(=O)C(O)C2CCCC2)C1 c1(Nc2cccc(CCOC(N(C)C)=O)c2)nccn2c(CO)nnc12 Cc1cc(CCNC(=O)CC2C=CC(NC(C3CNC(=O)O3)=O)C2)n[nH]1 C1(C(=O)NCC(C2CCN(C(=O)CC#N)CC2)F)(CC)CCCCO1 C1(CCC)CN(C(C2(CC)CN(C(=O)C=Cc3cn(C)cn3)C2)=O)CCO1 Cc1cc(OCC(=O)NCCCCCNC(C2(O)CC2)=O)cc(C)c1 N1(C(C(COC)NC(C)=O)=O)CCCC2C1CCCN2C(=O)CCCCCOC N1(C(C2N(C(C(=O)NCC)=O)CC(O)CC2)=O)CC2CCCC(O)C2C1 c1(C(N(C)C)=O)ccccc1C(=O)NC1CC(C(=O)NC2(CC(F)(F)F)CC2)C1 C1(CC(=O)NC(C2(O)CCN(C(C(C(C)C)F)=O)C2)C)CCCNC(=O)C1 CCCC(C)(CC)C(=O)NC(C)CNC(c1cnn(-c2ccc(Cl)cc2)c1C)=O C1(CC)COC(CC)CN1C(=O)CN(C(=O)CC(=O)OCC)C1CCCC1 N1(C(C)=O)CCN(C(=O)N(c2ccccc2)C(=O)CSc2cnc(C)s2)CC1 c1(C(N(CCCNC(=O)C=Cc2ccccc2)C)=O)cc(=O)n2ccsc2n1 CC1CC(NC(=O)C=Cc2ccc(Br)s2)CC(C)N1 C1(C(CNC(=O)CC2CCC2)NC(C2(C#C)CC2)=O)CCCCC1 C1(NC(CCSC)=O)CCCN(c2ncncc2C#N)CC1 C1(CNC(C#CC(C)(C)C)=O)CC2(CN1C(c1ccc(C#N)[nH]1)=O)CC2(F)F c1(C(=O)NCCN(C(C(F)=CCC)=O)C)cc(C(F)(F)F)ccc1N C(=O)(C(F)(CC)C(=O)OC)N(C1CCN(C(COCC)=O)CC1)C c1(OC)nn(C)cc1NC(=O)COc1ccc(OCC2CCCCC2)cc1 C12(NC(C(C)(F)F)=O)CC(CO)(C1)OC21CCN(C(c2nc[nH]n2)=O)CC1 c1(C(N2CC(CNC(C(CC)(CC)CO)=O)C2)=O)cccc2[nH]cc(C#N)c12 N1(C(c2cc(CC)c(C)s2)=O)CCN(C)C(CNC(C2CCN(C)C2)=O)C1 C1(NC(Cc2ccc(C(C)=O)s2)=O)COC2(CCN(C(c3nocc3Cl)=O)C2)C1 N1(C(C(N2C(C(=O)OC)C(O)CCC2)=O)=O)CC(O)CC2(CC2)C1 CC1CN(C(C2CC(=O)C2)=O)CC(C)N(C(c2cc(Cl)ccn2)=O)C1 C(=O)(C(CCC1CCC1)NC(c1ccc(O)cc1)=O)N(CCC=C)CC C=CCC(CCCCC)C(=O)NC1CCC(CNC(=O)CN2CC(C)(C)C2)CC1 C(=O)(CS(=O)(=O)CCC(F)(F)F)NC1CCCC(CNC(C(CCC)(C)C)=O)C1 C1(NC(CC2(CC)CCC2)=O)CS(=O)(=O)CC1NC(c1cnccn1)=O Cc1cc(=O)c(C(N2CCSCC2C(=O)NC2CCC=CCC2)=O)c[nH]1 C1(C)(NC(c2cncc(NCC)c2)=O)CCCN(C(=O)CC2CC2C2CC2)C1 C(=O)(C(C(C)C)C(C)C)N(CC(C)(C)C)C(C1CCCN(C(CC)=O)C1)=O CCC(CNC(c1cc(Br)cn1C(C)C)=O)(CC)NC(C1C=CCC1)=O C(=O)(C1=NNC(=O)CC1)NC1CN(C(c2cnc(OCC)nc2)=O)CC(O)C1 CC1(C(N2CC(CNC(=O)Cn3ncccc3=O)C(O)C2)=O)CCCS1(=O)=O C#Cc1cccc(C(=O)NC(C2CCN(C(C3CCCN3C)=O)C2)C)c1 C(=O)(C1=CC(O)C(NC(=O)CCC2CCCN2C)C1)N1C(C)(C(C)C)CC1 C1(C(=O)O)(C(=O)NCC2CN(CC(F)(F)F)C2)CC2(CCC2)C1 C(=O)(C(C(C)C)NC(=O)C=Cc1ccncc1)NC(C(=O)OCC=C)(C)C N1(C(CCOC2C(NC(C(=Cc3ccco3)C)=O)C2)=O)CCC(F)(F)C(O)C1 C(CN=c1nc(N2CCC=C(Cl)C2)c2[nH]ccc2[nH]1)(C1CCC1)OC C1(C(N(C2CCN(C(C3CCCC3O)=O)CC2)CC#C)=O)CC12CCCCC2 N1(C(c2nccc(C)c2N)=O)CCC2CN(C(C3C4CCCOC34)=O)CCC12 Cc1nc2ccc(C(=O)NC(C)CN(C)C(c3c(O)ccc(F)c3C)=O)cc2o1 C1(CC)CCCN(C(C2C=CCN2C(=O)CCCOCCOC)=O)C1 C=C(C)CCC(=O)N1CC2CC2(CNC(c2oc(C3CC3)nc2C(F)F)=O)C1 C1(CNC(C(C)OCCOCC)=O)(CO)CCN(C(c2cnn(C)c2N)=O)C1 CCC(CC(C)C)C(=O)NCC(c1ccc(F)cc1)NC(c1cc(OC)ns1)=O N1(C(C(C(CC)C)NC(=O)N)=O)CCC(F)(F)CC1C.C(C)(C)(C)OC C1(C)(CNC(C(CC2CN(C(CCC3(C)N=N3)=O)C2)F)=O)COC(=O)N1 Cc1cc(C(=O)NCC2CCCCC2C(=O)NCCS(N)(=O)=O)nc(O)c1 c1(C(N2CCOCC2CC2CCOC2)C(=O)NCC)cc(C(F)(F)F)cc(F)c1 N1(C(=O)OC(C)(C)C)CCC(S(=O)(=O)OCC2CC2c2ccccc2)C1 C1(CNC(C(C2CC2)OC)=O)CC(C(F)(F)F)CN1C(C1(c2ccncc2)CC1)=O c1(NC2CC(OC)C(OC)C2)ccc(S(=O)(=O)NCc2nncs2)cc1Cl C=CC(C(=O)NCC(C)=CC(=O)N(C)Cc1ccco1)OC c1(C(=O)NCCOC)ccccc1NS(=O)(=O)CC1CCS(=O)(=O)C1 N1(C(c2c(C(C)C)cn(C)n2)=O)CCCOC(CNC(c2ccccn2)=O)C1 C=Cc1cc(C(=O)N(CCN(C)C)Cc2ccc(C#N)cc2)cc(F)c1 c1(C(=O)NC(CN(C(C2N(C(CCC)=O)CSC2)=O)C)C)onc2ccccc12 C(=O)(CCCCCNC(C)=O)NCC1C(NC(c2cnn(CC)n2)=O)C1 c1(C(=O)NC2CCN(C(C(C)c3ccsc3)=O)C2)cc(N)cc(O)c1F C1(NC(C2(C#N)CCOC2)=O)CN(C(=O)C2=C(Cl)CC2)C2(CCCCC2)C1 c1(C(N(CC(C)NC(c2c(Cl)cc(C)s2)=O)C)=O)cc(N(C)C)cc(C#N)c1 c1(SC)cc(=NC(=O)C(=O)N=c2cc3n([nH]2)CCCC3)cc[nH]1 C1(C2CC2)(C(=O)NCC(CNC(c2c(C)ccnn2)=O)CO)CCOCC1 CC1(C)CC(O)CN1C(C1CC(F)CN1C(C1CC1c1ccccc1)=O)=O c1(OCC(=O)NCC(C)N(C(=O)C(O)CC(N)=O)CC)cccc([N+](=O)[O-])c1 n1(CC)nc(C(N2CCC(NC(c3cn(CC(F)(F)F)cn3)=O)C2)=O)ccc1=O C1(C(=O)NCC2C(C)CCN2C(c2csc(Cl)n2)=O)CCC2(CCCC2)CC1 N1(C(c2cnn(C)c2Br)=O)CCC(NC(c2ccnc(S)c2)=O)C1(C)C N1(C(CN2C(C)CCC2C)=O)CCN(C(=O)CN(c2ccc(Cl)cc2)C)CC1C c1(CNc2cccc(-c3c(SC)cc(F)cc3)n2)c(F)cc(F)cc1F c1(C(N2CC3CC2CO3)=O)c(C)cc(Cl)cc1Br.C1(C(C)=O)CC1C=O N1(C(CCS(=O)(=O)NC)=O)CC2(CCN(C(C3CC(OC)(OC)C3)=O)C2)C1 c1(C(N)=O)cccc(CC(N2CC(O)(CNC(C3(C(F)F)CCCO3)=O)C2)=O)n1 N1(C(C(=O)NC2CCN(C(CCC(CC)C)=O)CC2)C)CCCc2ccccc21 C1(OC)CCC(C)(C(=O)NCC(C)(C)OCCNC(=O)OC(C)(C)C)CC1 CC(C)C(C(=O)N(C1CC1)Cc1ncc(C(N2CCC(C)(O)C2)=O)cn1)NC=O CCCC(CC(=O)NCC(F)Cl)NC(c1c[nH]c(C)cc1=O)=O c1(C(=O)NCC2C(F)(C(=O)OCC)C2)[nH]c2ccc(C(F)(F)F)cc2c1C C1(CNC(CN(C2CC2)CC)=O)CN(C(C2CCCC2CF)=O)CCO1 c1(OC)nc(Cl)ccc1C(=O)NCC1CC1CNC(c1cc(C)ncc1Cl)=O C(=O)(C1CCOc2ccccc21)NCC1C(Nc2nc(C(C)(C)C)nc(=N)[nH]2)C1 CC(C)C(CCNC(=O)C(C1CCCCC1)F)NC(=O)C(C)CN(C)C C(=O)(C(CC(F)F)NC(C1CCOC1)=O)NCCc1cnc(C)o1 C(CCC(C)CC(=O)N1CC(NC(c2csc(CO)n2)=O)C(CC2CC2)C1)=C(C)C C(C)(CN=c1[nH]c2c(c(=NCC3CC4(CC4)CO3)[nH]1)CCC2)c1ncc(C)s1 C#CCCCCC(=O)N(CCC(C)NC(=O)CC(c1ccccc1C)C)C C1(C(=O)NCCCOCCNC(C=CSC)=O)CCC(=O)N1C(C)=O c1(OCC)ncc(S(=O)(=O)N2CCC(Cc3nccs3)C2)cn1 C(=O)(C(CCN(C)C)NC(=O)CCCF)N(CCN(C)C)C.C(C)(=O)O n1(CC)nnnc1C(C)(CCCl)NCC(C)C(=O)NCCC(F)(F)F C1(NC(C(C)OC)=O)(COC)CCN(C(C2C3(CC3)C23CC3)=O)C1 c1(NC(C(C)N(CCC)CCc2ccccc2)=O)ccc(CCOC)cc1 c1(N2CCC(CC=C)(NC(c3cc(F)cnc3Cl)=O)C2)ncnc2c1cnn2C O=C(C(CC(F)F)C1CCC1)N1C(CC(=O)NCCOc2cn[nH]c2)CC1 c1(C(=O)NC2CCC(C(=O)NCCOCCCC)C2)ccc(C)c(Cl)c1 CCCCCCCCC(=O)NC(C)(C)CCC(N1CCC2(CCC(CO)C2)C1)=O C1(NC(C2C(C)CC2)=O)(CNC(=O)CS(=O)(=O)N2CCN(C)CC2)CCCCC1 c1(C(=O)NC(C)CN(C(=O)CNC(C2CCCC2)=O)C)coc2ccc(O)cc12 C1(C(=O)NCCC(C)N(C)C(C2CCCS(=O)(=O)C2)=O)(OC)CCCCCC1 C(=O)(CCCC(C)(C)NC(c1ccc(F)s1)=O)NC(C)CS(C)=O c1(C(=O)NC2(C)CCCC2NC(C2CC(F)(F)C2)=O)noc2c1CCCCC2 N1(C(C=Cc2cccc(C)n2)=O)CC2CCC(C1)N(C(c1c[nH]c(Br)c1)=O)C2 c1(C(N2C(CNC(c3nc(CCC)sc3)=O)CC2)=O)nccc2cccnc12 CC1CN(C(=O)CSCC(F)(F)F)CCC1NC(=O)CCc1cnc[nH]1 C(=O)(C(O)CCN(C(c1sncc1C)=O)CC)NC(c1ccccc1)C#C CCC(C)CCC(=O)NCCCCCCNC(c1[nH]c(O)nc1C)=O N1(C(C(CC2CN(C(C3(SC)CC3)=O)C2)F)=O)CCC(=C(F)F)CC1 c1(SCC)cccc(C(N2CCC(N(C(=O)C(C)Cc3ccccc3)C)C2)=O)c1 c1(CC(=O)NC(C(C(C)C)NC(c2c(C)n[nH]c2C)=O)C)cc2ccccc2o1 Cc1cnc(C=CC(=O)NC(C)(C)CNC(=O)C(C)SC(F)(F)F)[nH]1 CC1(NC(=O)CCCNC(N)=O)CCCN(C(C2CC3CCC2CC3)=O)C1 c1(CN(C(=O)COc2ccccc2)Cc2ccccc2F)noc2c1CCCC2 C(C1=NOC2CCCC12)NC(C=CC(C)(C)NC(C1C(C)(C)COC1)=O)=O C(=O)(CC(C)(C)C(C)(F)F)NC1CC(N(C(C=Cc2cncc(C)c2)=O)C)C1 CC1CCCC(CC(=O)NCCCCNC(=O)C(=Cc2cccnc2)F)O1 C1(=O)CCCC(=O)N1.n1(CCOC)nccc1CCCCCN(C(C)C)C1CC1 C1(C(C)C)CN(C(=O)CC(C)(C)C#N)CCCN1C(c1cnc(C(F)F)o1)=O C1(CNC(CC=C=C)=O)CCCC2CN(C(c3cc(C#N)cs3)=O)CC12 N1(C(c2c(C)cccn2)=O)CCN(C(=O)Cn2nccn2)C2CCCCC2C1 C(C(C)(C)CNC(C1CC1c1ccn(C)n1)=O)N(C(=O)C=Cc1cncs1)CC C1(CC(=O)N(CC(F)F)C(C)C)CCCN1C(=O)CCn1cccn1 c1(OC)nc(C)ccc1C(=O)NCc1ccc(CCNC(C2CC(F)C2)=O)cc1 C1(C(=O)NCc2nc(C(C)OC)[nH]n2)(CNC(=O)C(C)OC(C)C)CC12CCC2 c1(OC)ccc(C(=O)NCC2CCN(C(C3CCC34CCC4)=O)C2)nn1 c1(C(=O)NCCC2CN(C(C3CC3Cl)=O)C2)cccnc1SCc1ccccc1 c1(C(=O)NCC2N(C(c3cn(CCC)nc3)=O)CC(F)C2)cccc2c1CCN2 O=C(CC1=CSC2=NCCN12)NCC1(F)CCCN(C(=O)CSc2ncccn2)C1 C1(C(C(=O)OC)O)CCN(CCCc2ccc(Cl)cc2)CC1 C1(CNC(=O)COC2CC(F)(F)C2)CC2(CO1)CN(C(=O)C=Cc1cc[nH]n1)C2 Cc1cc(O)ccc1C(N1CCCC(NC(c2ccoc2C2CC2)=O)CC1)=O CC1(C)CC2(CC2C(=O)NC(C2CCCN2C(=O)CCc2ccoc2)(C)C)C1 Cn1cc(NC(=O)COC23CCCN(CCC2)C3)c2ccccc12 C1(O)(CNC(=O)COCCO)CCCN(C(c2ccc(-c3ccc(Br)s3)s2)=O)C1 Cc1ccc(NC(=O)C(CNC(C2(C)CCCNC2=O)=O)CC2CC2)cc1C#N N1(C(C(CC)OCC)=O)CC(C(=O)N(CCCN2CCCC2)C)C(C)(C)C1 C(=O)(CCCCC#N)NC(c1cncc(F)c1)CNC(CCCCC=CCC=C)=O c1(CCC(=O)NCCCn2cc(CS(=O)(=O)C3CC3)nn2)cccnc1Br Cc1ccc2c(CCNS(=O)(=O)CC3OCCO3)cn(C)c2c1 C=CCCC(CC(C)C)C(=O)NC1CC(CNC(C2(C#N)CCOC2)=O)C1 c1(CC(N2CC(C)(NC(c3ccc(C)cc3Br)=O)C2)=O)ccn2cncc2c1 N1(C(CCc2c[nH]c(=N)[nH]2)=O)CC(NC(c2cn(C3CCCC3)nn2)=O)C2CC12 CC(C)(CC(=O)N1CC(C(F)(F)F)C1COC(F)F)C(F)F.n1(CCS)cc(C)nn1 CC(=O)CCCCC(=O)N1CC(C(=O)NCCNC(C2CC(C)N(C)C2)=O)C1 C(C(C(=O)NCC1(F)CC(NC(=O)C(C)CN2CCOCC2)C1)OC)OC CCCC(C(=O)NC(C)(C)C(C)NC(=O)CCc1ccc(F)c(F)c1)C(C)C c1(C(N2CCC(CSC)C2)C(=O)NCCC2(C)CC2)ccc(C2CC2)c(F)c1 C1(C(=O)NCCn2c(CC)ncc2)CCC(O)CN1C(=O)C1=C(C)CC1 N1(C(CCCOCCC)=O)CCCCC12CC(NC(=O)C(C)CSC)C2 C1(NC(CC(C)C(F)F)=O)CCCC12CN(C(c1ccnn1CC(F)(F)F)=O)C2 C1(CNC(C(C)OCC#C)=O)CCC(C(N2CC3CC2C3)=O)C1 c1(C(c2nnnn2CCCO)NCC2(OCC)CC2)c(Br)cnn1C.C1(CO)CC1 N1(CC)CC(NC(C2(CNC(=O)CC(C)CN(C)C)CCCC2)=O)CCC1=O C1(CC)CCCC1(C)C(=O)NC(C1CN(C(=O)CCC2CC(F)(F)C2)C1)C N1(C(=O)C2=CCC2)CCN(C(C2CCCC2C(F)(F)F)=O)C(CS(N)(=O)=O)C1 N1(C(C(C)CNC(=O)C(F)C(C)(F)F)=O)CC(O)CC12CCCC2 c1(C(=O)NCCOCCCC#C)coc(CNC(C)=O)c1 c1(C(N(C2CC(CNC(COC)=O)C2)C)=O)ccc(=O)n(C)c1 Cn1cc(S(N)(=O)=O)cc1C(=O)NCC1CCCC(NC(C2CCSCC2)=O)C1 O=C(C(F)(F)CO)NCCC1(O)CN(C(c2ccns2)=O)C1 CCC(C)(CNC(=O)CC(C)CNC(=O)CC1(O)CCOCC1)C(N)=O c1(CN2CCCC(NC(CCC(=O)NCC)=O)CC2)cn(C)c2ccccc12 C1(F)(CNC(C(C)SCC)=O)CCCN(C(=O)C(C)(O)CC)CC1 c1(CC(=O)NCC(C2CCCN2C(C(C)C#N)=O)(C)C)ccc(F)cc1Cl c1(C(N(CCNC(c2ccc(CO)s2)=O)C2CC2)=O)cnc(-c2ccoc2)s1 C12(C(=O)NCC=CCNC(C(c3ccccc3F)(C)F)=O)COCC1C2(F)F C1(C(=O)NCC(C)OCCF)CCCCCN1C(c1ccncc1)=O CCCC(C(=O)NC1C2CCN(C(=O)CSc3nnc(S)n3C3CC3)C12)SC CCC(C(=O)N1CC(O)(CCNC(C2(C(N)=O)CCC2)=O)C1)Sc1ccccc1 CC1(CNC(=O)C(N)=O)CCCC1NC(C1CCCN1C=O)=O C(CC(O)C(=O)N(C1CN(C(C)C)C1)C)NC(C(C)C1(O)CCC1)=O CCC(CC(F)F)C(=O)NCCCCC(C)NC(C1(CO)CCCC1)=O N1(C(CC(C)CF)=O)CCN(C(c2ccc3nccn3n2)=O)C2CCCC12 C(CCCCC(=O)N(CCCN=[N+]=[N-])C)NC(CC(CC)C)=O C1CCCN(C(C23CCC2CC3)=O)C1.C(=O)(C(C)C#N)OC C12(CNC(c3cccc(C)c3C)=O)CCCC1CCN2C(C1CCSCC1)=O N1(C(C(CC(C)C)ONC(C2(C)COC(=O)N2)=O)=O)CC(=O)N(C)C(C)C1 C12(C(=O)NCC3CC(CNC(COCCC)=O)OC3)CCC(F)(CC1)C2 N1(C(C2(CCCC)CCC2)=O)CC2CC2(CNC(=O)Cc2ccsn2)C1 C(=O)(CCCCC(C)(C)C)NC(CSCC)C(=O)N(CCC1CC1)CC C(=O)(C(C)(O)CCc1ccccc1)NC(C)CNC(=O)Cc1cnn(C)c1 N1(C(c2c(CC)n(C)nn2)=O)CC(C(N2CCC(C)CC2)=O)CCC1C N1(CC2=CCCC2(C)C)CCOC(C)(CNC(=O)CNC=O)C1 C1(C(C)C)CCN(C(=O)CCC2CCCN2C(C2CC2C2CCC2)=O)CC1 c1(C(=O)OCC)ccc(F)cc1C(=O)Nc1cccc(NC(C2CC(C)(F)C2)=O)c1 C1(N(C(=O)CSc2cnn(C)c2)C)CCCCN(C(c2cc(C(N)=O)[nH]n2)=O)C1 N#Cc1nn(CC(F)F)cc1C(N1CCN(CCC(F)(F)F)CC1)=O c12ccncc1S(=O)(=O)N2.C1(CS)CCCC12CC2.C1(C(=O)NCC)CCN(CC)C1 CC12CC(C(=O)NC3CCN(C(C4CC4C(N)=O)=O)C3)(C1)C2 N1(C(C2CNC2)=O)COC2CCCCC2C1.c1ccc([N+](=O)[O-])cc1Cl C1(C(=O)NC(C(CO)NC(C(COC)C(=O)OC)=O)C)CCCC(C2CC2)C1 N1(C(c2ccn(C)n2)=O)CC2CC(NC(=O)Cc3cn(C)nc3Cl)C1C2 CCCC(C(=O)N1CCCC1(C)CNC(=O)CN(C)S(N)(=O)=O)N(C)C C(=O)(C1CCOc2c(F)cccc21)N1CCCC(NC(=O)CCc2cncs2)C1 N1(C(C2OCC(C)C2)=O)CCN(C(c2csc(Cl)c2Cl)=O)CC1CO C(=O)(C(F)CC(C)(C)NC(c1ccc(C(F)F)o1)=O)NCc1n(CC)c(C)nc1 c1(C(N2CCC(Cn3cc(C(C)(C)C)nn3)C2)=O)nccn2ccnc12 C1(CN(C(=O)CS(=O)(=O)NC2CC2)C)CCCN(C(c2cncc(CO)c2)=O)C1 N1(C(C(CC(=O)Nc2cc3sccc3[nH]2)C)=O)CCN(C(=O)NCC)C2CC12 C(C(CNC(=O)Cc1ccns1)C(F)(F)F)NC(c1ccc(COCC)cc1)=O N1(C(C=CCC)=O)CCN(C(c2sccc2C)=O)CC1CC1CC1 c1(CN2C(C(N3CCOC(O)C3)=O)CC2)n[nH]c2ccc(Br)cc12 O=C(C#CC1CCOC1)N1CC(CC(N2C(CO)CC2CO)=O)C2(CC2)C1 c1(SCC(=O)NCC(CNC(C2C(C)C2C)=O)CO)ccccc1[N+](=O)[O-] N1(C(C)=O)CC(O)CC1C(=O)NCCCCNC(c1nn[nH]c1Cl)=O c1(NC(NS(CC)(=N)=O)=O)c(Br)ccc2c1OC(F)(F)O2 c1(OCC(=O)NC2C(CNC(C3(C)CCCO3)=O)CCC2)cc(Cl)cc(Cl)c1 CCCCC(C)C(=O)N(CCCNC(=O)COc1ccc(Br)nc1)CC c1(C(=O)NC23CCN(C(C4C(C)CCCC4)=O)CC2C3)ccc(F)cc1[N+](=O)[O-] N1(C(C(C)(C)C(F)(F)F)=O)CC2CCCN(C(=O)C(O)CC3CCCCC3)C2C1 c1(OCC=C)cc(Cl)ccc1C(N1CCC(NC(=O)C#CC(C)C)C(C)C1)=O C1(NC(C(F)=CCC)=O)CCCC(CC(=O)NCC(c2ccccc2)C)C1 C1(CNC(CCS(C)=O)=O)(CO)CC12CCN(C(=O)CC1CCCCC1)CC2 CC1(C(=O)Nc2cccc(NC(c3ccncc3)=O)c2)CC(C#N)C1 O=C1CC2(CCC2)C(C(=O)NC2CCCN(C(=O)C(F)CC3CC3)CC2)CN1 CN1CCC(C(N2CCN(C(=O)CCCCC3CCC3)CC2C2CC2)=O)CC1=O c1(CNC(C(C2(C)CC2)NC(=O)COCCN(C)C)=O)ccncc1Cl CN1CC(CC(=O)NC2(CNC(C3CCCCC(=O)N3)=O)CC2)c2ccccc21 Cc1ccc(CC(=O)OCC2OCC3CCC2C3)c(F)c1F C(=O)(C1=CN2CCS(=O)(=O)N=C2C=C1)N1CCC(NC(C(C(C)C)SC)=O)C1C c1(SCC)ccc(C(=O)NCC2CN(C(=O)Cc3cn[nH]c3)CCO2)cn1 N1(C(c2c(C)oc(C3CC3)n2)=O)CCN(C(=O)CCC(C)CN(C)C)CC1CO c1(C(=O)NCC(CNC(C(C)CCC(C)(C)C)=O)F)cc(C#N)c2n1CCCC2 CCCCCCC(C)C(=O)NC1CN(C(=O)CCN2CCOCC2)C1 CC(C(O)C(=O)NC(C)(C)CCNC(=O)C1=C(Cl)CC1)c1ccccc1 c1(C(N2CC(C)C(NC(=O)CCc3cc(Cl)no3)CC2)=O)n[nH]c2cccnc12 C123CC(CCO1)C2CC(=O)N1C=COCC1C(=O)N3.CC(C)(C)O N1(C(CC(=O)OC)=O)CC2(NC(=O)C(F)n3ccnc3)CCC1C2 N1(C(C(CC)OC)=O)CCC(NC(c2cncc(C(C)C)c2)=O)C(O)C1 C=CCC(CC)C(=O)N1CCN(C(c2ccc(CC)cc2)=O)CC1 Cn1cnc(C(=O)NCC(C2CCCN2C(C2CCCOCC2)=O)(C)C)cc1=O C1(C(=O)NCC2(NC(=O)CCOCC3CCCO3)CC2)CC2CCC2C1 N1(C(c2c(C)n(C3CCC3)nc2)=O)C2CCC1CN(C(c1ccncc1)=O)C2 NS(=O)(=O)c1ccc(CC2C(NC(=O)COCCn3cc(CO)nn3)COC2)s1 CCCCCCCCC(=O)NC(CC)CCC(=O)NC1CCCC1C#N c1(C(N2CC(C)N(C(C3CCS(=O)(=O)C3)=O)CC2C)=O)cc2ccoc2cc1F c1(C(=O)NCC(CC)(F)F)c[nH]c2cc(-c3cccc4ccccc34)cnc12 c1(OC)nc(C)cnc1C(N1CC(CNC(c2cc(C)ncn2)=O)C(C)C1)=O C#CCC(C)(CNC(=O)CC(C)(C)CNC(=O)C=CCOCCOC)CO CC(C)(C)CC(O)CC(=O)NCC1CC(F)(F)CN1C(=O)CC1=CCOCC1 CC(C(=O)N1CCC(CC(=O)NCCOC2CCC2)CC1)C(F)(F)F C(C(=O)NC1COCC1NC(c1nn(C)cc1Cl)=O)(C(C)C)OC CN1CC(C(N2CCC(O)(CN(C)C(c3cc(O)nn3C)=O)C2)=O)NC1=O c1(C(C)=O)cccc(OC(C)C(=O)NCC2CN(C(C3C=CCC3)=O)CC2C)c1 c1(-c2c(OC)c(C)ccc2)ccn2cc(C(=O)NC3CCCCC3O)nc2c1 N1(C(c2n(CC)cc(Cl)c2)=O)CC2CCOC2(CNC(=O)CN2CCOCC2)C1 c1(OC)cc(C(N2CCCC2CNS(=O)(=O)C2CC2c2ccccc2)=O)ccc1Br CCC(C)C(C(=O)N1CCN(C(=O)NC)CC1)NC(=O)C(C)C(F)F C1(C(=O)NCC2CCCCCN2C(=O)C2=CCCCC2)CC2CCC(C1)C2 c1(CN2CC(C3OCCN(C(Cc4ncn(C)n4)=O)C3)C2)cc(F)c(F)cc1Br N1(CCN(C(C2(n3cncn3)CC2)=O)CCC2CC2)CC(C(=O)CC)CC1=O.OC C1(C(=O)NCC(CC)NC(=O)CCc2cc(C)nn2C)CCN(C)C1=O C1(CC)(CC)CC(NC(=O)C(C)OC)CN1C(c1cc(CF)on1)=O C=CC(C)(C)C(=O)N1CCC(CCN(C)C(C2CC2(C)C(F)(F)F)=O)CC1 C(CCCCNC(c1cc(C(F)F)[nH]n1)=O)N(C(CO)C(=O)OC)C C12(CNC(C=CC=CC)=O)CCCC1N(C(c1cn3c(n1)COCC3)=O)CC2 C1(NC(Cc2cc(C)on2)=O)CCCC(C(=O)NC(C)(C)CCO)CC1 C1(NC(C2CC3COCC3C2)=O)CC2(CCN(C(c3cc(CCO)on3)=O)C2)C1 N1(C(CNC(CCC)=O)=O)CC(F)(CNC(C2CCS2(=O)=O)=O)C1 C(=O)(C(CC(C)c1ccccc1)N(C)C)NCCOC C1(NC(CC2(CC=C)CCCC2)=O)CN(C(=O)COCC)C2(CCOCC2)C1 C(=O)(C1=NOC(C)C1C)NC(CNC(c1c(C)ncnc1C)=O)C C1(NC(c2nccc(C)n2)=O)CN(C(=O)Cc2cnccc2C)CC1S(C)(=O)=O C1(NC(c2cc(C)ns2)=O)CC(C2CCN(C(C3CC(C)CC(=O)N3)=O)CC2)C1 CCC(C(=O)NCCn1cc(CNC(c2ccc3nnnn3c2)=O)nn1)C(F)(F)F c1(C(N(CCCNC(C(C)n2ccnn2)=O)C)=O)cncc2ccccc12 Cc1ccc2cccnc2c1C(=O)N(CC(C)CNC(=O)C(O)c1cnc[nH]1)C C(=O)(C(C)(O)C(C)(C)C)N1CC2C(CNC(c3c(C)ccc(C)n3)=O)C2C1 C1(C(N2CC(CNC(c3cc(CC)nn3C)=O)OCC2)=O)C2(CCC2)C12CCC2 N1(C(C(CCC)F)=O)CCCC2(C1)CN(C(=O)C(C)C1CCCO1)C2 C1(C(=O)NC2C(NC(CNC(N)=O)=O)C2)CCC=CCC1 C1(CNC(c2cnc(O)o2)=O)CCCCN1C(=O)CC1CS(=O)(=O)C1 C1(NC(c2ccc(CC(C)C)cc2)=O)CC2CN(C(=O)C(C)C)CC2C1 N1(C(=O)C=CC(F)(F)F)CCC2CCCN(C(c3nccc4[nH]ccc34)=O)C2C1 N1(C(CC2(C(=O)OC)CC2)=O)CC2CC1CC2NC(C1CC2(C1)CC(O)C2)=O C1(C(=O)NCC(=O)NCC)COCCN1CC.C12CCC1CNC2=O C(=O)(CC(C)(C)C(F)F)N1CCC(NC(c2c(OCC)noc2C(F)(F)F)=O)C1 N1(C(C2CCC(OCC)CC2)=O)CC2COCC2(C(=O)OCc2ccccn2)C1 C1(C)(C(=O)NCCC(CCNC(C2(CC=C)CC2)=O)C)CCNC(=O)C1 c1(N(C)C)ccc(C(N2CC3CC3(CNC(=O)C(C)(C)O)C2)=O)c(F)c1 c1(NC(C2(N(C)C)CC2)=O)cc(OC2CC2)cc(=O)o1.C1(C(=O)O)CC(=C2CCC2)C1.CO C(=O)(CC(CC(C)C)NC(c1sncc1C)=O)N1CC(OC)C(OC)C1 c1(CC(=O)NC(c2nccn2C)C)cc(O)ccc1Br C=C(C)C(CC(=O)NC1CN(C(c2cc(Cl)ncc2N)=O)CC1(C)C)OCC CC1C(NC(c2ccc(N)cn2)=O)CCCN1C(c1ccc(C2CC2)cc1)=O N1(C(COCCCC)=O)CCCCC1C(=O)NCc1nc(C)c(C)o1 C1(CNC(c2ccc(CSC)o2)=O)CN(C(=O)C(=Cc2cnc[nH]2)C)CCO1 c1(CC)cccc(C)c1NC(C1CCC(C)N(C(=O)CS(=O)CC)C1)=O C1(NC(C2(C#N)CCC2)=O)CN(C(=O)CCc2ncc[nH]2)CCC1C(F)(F)F CCCC(C(=O)NCC1CCN(c2nc(Cl)nc(C)c2F)CCC1(F)F)C(C)C c1(C(=O)NC(CNC(C(C)O)=O)CO)ccc(S(N)(=O)=O)cc1 C(C)(CO)(C(=O)NC(C1CCN(C(C2(O)CCCC2)=O)C1)C)OC C1(C)(NC(C(C)N(S(CC)(=O)=O)C(C)=O)=O)CN(C(=O)Cc2c[nH]nc2C)C1 c1(CC(=O)OC(CC(CC)C)C)nnc2n1CCCC2 N1(C(C(C(C)C)CC2CCCC2)=O)CC2CCC1CN2c1nc(C(F)(F)F)ns1 N1(C(C(=O)NC(c2ccccc2)C)C2CCCC2)CCC2COC(=O)NC2C1 c1(C(C2N(CC(=O)NCc3scc(C)n3)CCC2)O)cc(Cl)ccc1Cl C(=O)(CCC(CC)CC)NCC(C(=O)NCCOCC#C)(C)CC Cc1cc(C(=O)NC(C(N2CCSCCC2)=O)C2CCCC2)n(C)n1 c1(CC)ccc(Br)cc1C(=O)NC1CC(F)CN(C(=O)COC(C)=O)C1 CCC(C)N(OC)C(=O)C1CCN(C(c2ccn(C)c2)=O)C1 C1(CNC(CCCOC)=O)CN(C(=O)CC2CC3CCC(C2)C3)CC1(F)F N1(N2CC(c3c(C)coc3)C2)CCOCC1(C)c1cn(CCC)nn1.C(=O)O C1(C(N(CCC(=O)OC)CC#C)=O)CCCC(C)(C)C1.C(=O)(C(C)C(=O)OC)NC Cn1cc(-c2cc(C(=O)NC3CCC(NC(c4ccoc4)=O)C3)n[nH]2)cn1 c1(CCNC(CCN(C)C)=O)c[nH]c(=NCc2ccc(F)nc2F)[nH]1 CC(O)CCCN(C)C(c1n[nH]cc1CNC(C1(CO)CCOC1)=O)=O c1(CC(=O)NCC(C2CC2)NC(c2c(C)cc(C)s2)=O)csc2sc(C)cc12 c1(NC(C(CNC(=O)CCc2cccnc2)O)=O)ccc(C2CC2)c(F)c1 c1(C(N2CCC(CNC(C3CCCS(=O)(=O)C3)=O)CC2)=O)cccc2c1OCC2 c1(N2CCCC(CCCC)C2)ccc(S(=O)(=O)NCCCS(=O)(=O)CC)cc1F N1(C(C(CN)C2CC2)=O)CCN(C(c2cc(O)nn2-c2ccccc2)=O)CC12CC2 CC1=CCC(C(F)(F)F)(C(=O)NCC2CCN(C(=O)CNC=O)C2)CC1 Cc1cnccc1-c1cc(CNC(=NCc2ccccc2)NC2CCCC2)[nH]n1 c1(C(N(C(C)CNC(=O)C=Cc2cccc(Cl)c2)CC)=O)cc(C)ccc1Cl C1(c2nnnn2CC2CC2)(Nc2cccc(CC)c2)CC2C=C(C)CC(C2)C1 n1(-c2n(C)ccn2)nc2c(cc1=O)C1(CCOCC1)CN2C1CNCC1 c1(C(N2CCC(NC(C3(CC)CC3(F)F)=O)C2)=O)cnn(C(C)(C)C)c1Cl C1(CCC)(NC(c2c(C)coc2C)=O)CCCN(C(c2cccnc2O)=O)C1 C1(CNC(CCOCC)=O)CCCC2CN(C(=O)C(C)(C)CO)CC12 C(C)(CCC(=O)N1C2COCC1C2)OC.C12CCCC1CC(=O)N2 C12(NC(C(C(CC)C)OC)=O)CCCCCC1N(C(c1oc(C)nc1C)=O)CC2 CS(=O)(=O)C1CCC(C(=O)OCC(c2ccc(C(F)(F)F)c(Cl)c2)=O)C1 C1(C(N2CCCN(CC)CC2)=O)CN(C(c2n[nH]cc2[N+](=O)[O-])=O)CCC1(F)F Cc1ccccc1-n1ccc(NC(=O)C(N2CCCC2c2ccc(Cl)s2)=O)n1 c1(C(N2C3C(NC(CS(CC)(=O)=O)=O)C(C3)C2)=O)c(F)cc(C)cc1F C1(NC(CCC)=O)CCCCCN(C(c2cc(OC)ccc2C2CC2)=O)C1 C1(NC(c2n(CC)cnn2)=O)CS(=O)(=O)CC1NC(C1CC(SC)C1)=O N#CC12C3C4C1C1C2C3C41C(=O)NCC1CCC(NC(C2CCCCCC2)=O)C1 N1(Cc2c(OC)ccc(O)c2)CCC2(CCCN(C(c3ncoc3C)=O)C2)C1 c1(C(N(CC(C)NC(C2CC2C(=O)OC)=O)CC)=O)nnn(CC)c1C1CC1 N1(C(c2n(CCC)ncc2)C(=O)NC(C)C(=O)OCC)CC(CO)CC(F)(F)C1 c1(C(=O)OC(C)(C)C)nc(-c2cn(CCC3CCN(C(=O)OC)C3)nn2)c(C)o1 CCCC(C(=O)NC1CN(C(=O)CCSC2CCCC2)CCC1O)C(C)C C(=O)(CCCCCC(C)(C)C)N1CCC(N(C(=O)C(O)CC(C)(C)C)CC)CC1 C12(C(N(CCCNC(c3c(CC)[nH]nc3Cl)=O)C)=O)CCN(C1)S(=O)(=O)C2 C=CC(C)(CC)C(=O)N(C)CC1CCCCN1C(c1cc(Cl)nn1C)=O Cc1nc(Cl)cc(Cl)c1C(=O)NCC1CCNC(=O)C1.C12CCN(CC1O)C2=O C#Cc1cncc(C(N2CCCC(CNC(=O)CC3CCN(C)C3)C2)=O)c1 C1(C(N2CCC(C(C)NC(C(F)=C(C)C)=O)C2)=O)CN(C)CCO1 C1(NC(c2cnn(C)n2)=O)CCCOC12CCN(C(=O)C(C)(C)CF)CC2 C12(CNC(CS(=O)(=O)NC)=O)CCC(NC(C3CNC(=O)N3)=O)(CC1)CO2 c1(C(N2CCCC(CNC(C3CC4C(C3)C4(F)F)=O)C2)=O)ccc([N+](=O)[O-])nc1 C1(NC(C2(C#C)CC2)=O)CCCC(CNC(c2cc(C(N)=O)cn2C)=O)C1 N1(C(CCC2CCN(C(C3(C#N)C(C)(C)C3)=O)C2)=O)Cc2cccnc2C1 N1(C(C(C)NC(CC(C)N(C)C)=O)=O)CC(O)(C2CC2)C1 c1(SCC(=O)OC)scnc1NCC1(NC(Cc2ccnn2C2CC2)=O)CC1 CC(C)(C)CC(O)C(=O)NCC1(CNC(=O)CC2CCC2(C)C)CCC1 C1(C(=O)OCC)(CN(C)Cc2cn(C(C)C)nn2)CC(F)(F)C1 C12(NC(C(C)CN(C)C)=O)CCC(CN(C(C3CCC(C)(O)CC3)=O)C1)C2 C1(C(=O)NC2(CCCNC(C3C4COCC34)=O)CC2)(OC)CCC(F)(F)CC1 C1(CC(C)C)CCCCN1C(=O)C(C)(C1CC1)N(C(=O)CCc1ccc[nH]1)C c1(C(=O)NCC2(CNC(C(C)OC(C)C)=O)CCCCC2)[nH]cc2c1CCCC2 N(C1CCc2cc(C)ccc21)C(C(=O)Nc1ccc(OCC)c(OC2CCC2)c1)=O C(N=c1ccc2ncc[nH]c-2n1)C1OCC(CNC(C2CC23CCSCC3)=O)C1 N1(C(C(c2cnn(C)c2)C)=O)CC2CC2(CNC(C2SCCS2)=O)C1 N1(C(c2ccc(CC)cn2)=O)CCN(C(=O)CCc2cnc(O)[nH]2)CC1CF C(=O)(CS(=O)(=O)CCOC)NC(CC)CNC(=O)C(=O)Cc1ccccc1 CC1C(NC(=O)C(F)=C2CCC2)CCCN1C(=O)CC(c1cccc(F)c1)O N1(C(CC(=O)NC(CC)=O)=O)CCc2cc(-c3ncc[nH]3)ccc21 Cc1cc(C(N2CCC(NC(=O)C(C(C)O)N(C)C)C(O)C2)=O)cc2nc[nH]c12 N1(C(c2on(C)c(=O)c2)=O)CCC(NC(C2CCC(=O)NC2)=O)C(F)(F)CC1 Cc1nc2cccnc2n1N(C(=O)Cn1cncn1)C c1(C(=O)NC2C(CNC(CNC(CC)=O)=O)CCCC2)cc(C)c2[nH]cnc2c1 c1(C(=O)NCC(CCCC)NC(CSCC=C)=O)cccn2cc(C)nc12 N(C(=NCC(C)C1CCCCC1)NCC(c1cnn(C)c1)OC(C)(C)C)C(C)C C1(COC)CN(C(c2c(O)cccc2O)=O)CCN1C(c1cnc(Cl)nc1)=O c1(OC)cc(CN2CCC(CCN(C)C)CC2)cc(Br)c1 c1(CN(C)Cc2ccc(Br)cc2)cc(F)ccc1O N1(C(C=COCC)=O)CCOCC(NC(=O)C(C)(C)C(C)O)C1 C1(N(C2CCN(C(COC)=O)C2)C(=O)CC2CCCC(C)O2)CCCCC(=O)N1 CCC(C(C)(F)F)NC(C1CN(C(C2(C#N)CCC2)=O)CC1F)=O C1(N(C)C)CCC(C(N2CC(CO)C(NC(C3CCN3S(C)(=O)=O)=O)C2)=O)CC1 c1(NC(C(CCC(C)(C)N)O)=O)ccc(S(=O)(=O)NC2=NCCS2)cc1 C(=O)(C(C)S(C)(=O)=O)N1CCC(COC)(CNC(=O)C2=NOCC2)C1 N1(C(C(c2cccc(C)c2)O)=O)CC2CC(CNC(=O)COC(C)C)C2C1 C(=O)(CCC(C)(C)F)NCC1(NC(CNC(C(CC)C)=O)=O)CCCC1 N1(c2c(C(C)=O)cccn2)CCC2(CC1)CC2(C)C(=O)NCc1sc(C)nc1C CCCC(CC1CCCC1)C(=O)N1CCC(CNC(=O)CCC(C)(C)F)C(O)C1 c1(C(=O)NC2CN(C(CC(C(C)C)O)=O)CC2C)cc2ncccc2[nH]1 C(=O)(CC(C)(C)C(F)(F)F)N1CC(Cn2cc(C(CC)N(C)C)nn2)C1 N1(C(C2CC(C)OCC2)=O)CC2CCC(N=c3[nH]c(C(C)(C)C)nc(=N)[nH]3)C2C1 c1(C(=O)NCC(C)(C)NC(C2(C)CC2(Cl)Cl)=O)ccc(Cl)cc1 C1(NC(C(N2CCSCC2)C)=O)CC2CN(C(C3CN(C)CCO3)=O)CC12 c1(OCC)ccccc1C.c1(C(C)(C)NCCOC(C)=O)nnnn1CC(F)F C1(NC(C(C)OC)=O)CN(C(C23CCC(C2)OC3)=O)CC(C)(C)C1 C(=O)(C(C)CC(C)C)NC1CC(NC(=O)OCC)C1.C1CC(OCOC)C(OC)C1 CC(C)(C)CCCC(=O)NCC(CC1CC1)C(=O)NC12CCC(CC1)CC2 C1(CC(C)C)CN(C(C2CC=CCC2)=O)CCN1C(=O)CNC=O c1(CC(N2C(C)C(NC(c3ccn(C)c3)=O)CC2)=O)ccc(S(N)(=O)=O)s1 C1(c2cn(CC(C)N(C)C)nn2)C2CN(C(=O)CCCC3CCC3)CC12 C1(NC(C(COCC)C)=O)CN(C(c2cccc(OCCF)c2)=O)C2(CCC2)C1 C(=O)(CC(C)(C)COC(C)=O)NCCCCC(=O)N1CC(CCC#C)C1 N1(C(C2C(CC)CC2)=O)CCCC2(CC1)CC2.C12CCCC1C(=O)NC2 Cc1ccc(C(N2CCC(n3ccnc3C)C2)C(=O)NC(C)C)nc1 C=C(Cl)CC(C(=O)NCC1CC(=O)N(C)C1)NC(C1CCCCN1C)=O n1(C(CC)C)nc(C(=O)NCC2CCN(C(=O)CCC3CCN(C)C3)C2)cc1C CC(C)C(C(=O)N1CC2CC1C2CNC(=O)C(C(C)C)N(C)C)n1ncc(N)n1 Cc1nc(C(C)C)oc1C(=O)NC(C)(CNC(C1CC(N(C)C)C1)=O)C(C)C CC(C)CCC(F)C(=O)N1CC2(CC2)CC1C(N1CCC(OC(C)C)C1)=O C(CC(=O)N(CCCNC(=O)C(F)C1CC1)C)N(C(COC)=O)C.C(C)(C)(C)O N1(C(C(c2cccc(CO)c2)C)=O)CC(NC(=O)Cc2csc(Cl)c2)C2(CC2)C1 N1(C(c2n(CCC)ncc2)=O)CC(O)CC1CNC(=O)C(O)CSC c1(CNC(C(C2CN(C(C(C)SC(C)C)=O)C2)O)=O)ccc(F)cc1O C#CC1COCCN1C(c1c[nH]nc1CNC(c1c[nH]c(C#N)c1)=O)=O N1(C(c2n(CC=C)ccc2)=O)CC2CCC(N(C)C(c3csc(C)c3C)=O)C2C1 c1(CC)noc(CCC(=O)N(C(C(=O)NCCOC)C2CCOC2)CC)n1 Cc1c(C(=O)NC2(CNC(C3C=CCS3)=O)CC(F)(F)C2)ccc(F)c1F Cc1c(C(=O)N(CCCN(C)C(c2cc(C3CC3)[nH]n2)=O)C)nc2sccn12 O=C1NCC2C(C(N3CCC(N(C(=O)CC4CCCC4)CCO)C3)=O)C12 C(CCC(=O)N1CC(CNC(c2ncsc2C2CC2)=O)C1)NC(N)=O CC1(CNC(CCc2n(C)cnn2)=O)CCCCC1NC(c1cnc(O)n1C)=O N1(CC(N2CC(C)C(NC(C3(CC(F)F)CC3)=O)CC2)=O)CCc2sccc2C1 c1(C(=O)NC2C(C)CN(C(=O)C=CC3CCOCC3)C2)c(N)cc(Cl)cc1F n1(C(C)C)nccc1C(=O)N(C)CCOCCC(=O)NCC1(O)CCOC1 C1(C(=O)NC2(COC)CC2)CN(C(c2ccncn2)=O)CC1C(F)(F)F C(C(=O)N1CC(NC(c2ccoc2)=O)C1)(C(C)C)N(CC)CC N1(C(c2nc(C)oc2)=O)CC2CCC1CN(C(c1cnc(C)nc1)=O)C2 C1(CNC(C(CC)F)=O)CN(C(=O)CSc2ccncc2)CC12CCOCC2 C1(C(=O)NCCC2CCCCC2O)CC=CCN1C(=O)CCc1ccccc1O Cc1cnc(C(=O)NC2CCC2NC(C2CCC(C(F)F)CC2)=O)cn1 c1(C(N2C(CNC(c3nc(COC)oc3)=O)CCCC2)=O)ccc(F)cc1N C123CC(CO1)N(C2)C3=O.CCC(C)C(=O)NCC(=O)NCc1cc(C2CC2)on1 C1(C(N(CCNC(C=C(CCN(C)C)Cl)=O)C)=O)CCC2CC1CO2 C1(NC(CC2(OC)CC2)=O)CCN(C(=O)Cc2cc[nH]n2)C1C c1(SC)ncc(CN(c2cc(C#N)ncn2)C2CNCC2(F)F)c(C(F)(F)F)n1 C(=O)(C#CC1CCCO1)NCCCC1N(C(CCC(=O)NCCC)=O)CCCC1 C1(NC(=O)CCSC2CCCC2)CCCC(NC(c2ccccc2F)=O)C1 C(CCC(=O)N(CC(C)NC(=O)CCCN1CCC1)C)OC(C)=O c1(C(N2C3CN(C(CCc4cccc(C)n4)=O)CC2C3)=O)c(F)cc(F)cc1Cl c1(C(N2CC(C)C(NC(=O)Cc3ccn(C(F)F)n3)C2)=O)ccc(F)c(Cl)n1 C1(C(=O)NC2(CNC(c3ccc(CO)s3)=O)CC2)CC(C2CCC2)C1 Cn1nc(C(=O)NC(CC2CCCC2)C(=O)NC2CCC(N(C)C)C2)cc1O O=C1CCC(C(N2CC=C(CNC(C3CCCCC3(F)F)=O)CC2)=O)CCO1 C1(CC=C)(NC(=O)COC)CCCN(C(C2CC3CCCC23)=O)C1 c1(CC(N2CC(CC)C(NC(c3oncc3C)=O)CC2)=O)ccc(S(N)(=O)=O)s1 C(=O)(C(C)(O)C(C)C)N1CC2(C(C(=O)NCc3onc(C)n3)C2)C1 C1(CNC(=O)CC2CC(O)C2)CCCC(NC(C2(c3cccnc3)CCC2)=O)C1 CCC(C)(COC)C(=O)N1CCC(c2nnc(CNC(=O)CC(C)SC)s2)CC1 c1(CNC(C=CSC)=O)ccc(CN(C)C(C2(c3cccc(C)c3)CC2)=O)cc1 N1(C(CC2(C=C)CCC2)=O)CC2=C(C1)CN(C(c1ncc(C(C)=O)cc1C)=O)C2 O=C(CCCCC1CC1)NCCC1CCC(NC(c2ccn(CCF)n2)=O)C1 C1(C(c2n(CC(=C)C)nnn2)(CC)NC(C)CCSCC)CCCCCC1 c1(C(=O)NC(C2CN(C(=O)CC(C)(C)C)CCO2)C)ccc2cc[nH]c2c1 c1(C(N(C)CC2CCN(C(=O)CC3(C)CCCO3)C2)=O)cnc[nH]c1=N c1(N(C(C)CC(=O)OCC2CC2)C)cc(=O)n(-c2ccccc2)n1C C1(C(=O)NCC(C)(C)NC(=O)CSCc2ccccn2)Cc2c[nH]cc2S1(=O)=O Cc1n[nH]c(C)c1CCC(N1CC(NC(C2C3COCC23)=O)CC1C)=O C(C(C(=O)NOCC(C)O)NC(C1CC(C)=NO1)=O)OC(C)C c1(C(=O)OC)ncc(C(N2CC(C)(Nc3ncoc3C3CC3)C2)=O)s1 N1(C(CC(C)SC)=O)CCCC(F)(CNC(c2occc2-c2ccccc2)=O)C1 c1(C(=O)NCC(C)N(C(c2ccccc2OC(C)C)=O)CC)c(C)cccc1Cl C(CO)(C(O)CCC)NC(CCCNC(C1(CC=C)CCOC1)=O)=O c1(NC)cc(F)ccc1C(=O)NC(=O)C(c1cccc(OC)n1)(F)F C(=O)(CCCCC(C)C)N(C(C(N1CCC(OCCOC)C1)=O)CC)C Cc1nc(C(N2CCCCC2CCN(C)C(C2C3CC4C(C3)C24)=O)=O)[nH]c1C C1(C(=O)NCC2CCC(CNC(c3ccns3)=O)CC2)CN2CCC1CC2 N1(C(C(CC)(C)O)=O)CCC2(CC1)CN(C(=O)CC1CC1C(F)(F)F)CCO2 C1(C(=O)NCCc2ncn(CC)c2)C2CC3C(C2NC(=O)CCC2CC2)C13 N1(C(c2cc(C)[nH]c2)=O)CCC2CCCC12C(=O)NC1CCC2(CC2)C1 c1(NC(CCC(=O)OC)=O)cc2cc(Br)[nH]c2nc1C c1(CC)onc(C)c1C(=O)NCc1ccc(C(=O)NCC2CCOCC2C)o1 c1(C(N2CCC(F)(CO)C2)=O)ccc(CNS(=O)(=O)CN2CCCCC2=O)cc1 C12(CNC(=O)COC(F)(F)F)CCC(CN(C(=O)CC3CCC34CCC4)C1)C2 c1(NCc2cc(CC)on2)ccc(S(=O)(=O)NCCN2CCOCC2)cc1Br c1(OC)cc(C(=O)NCCC(C)NC(C2CCC(C)(C)CO2)=O)c(F)cn1 N1(C(C2C(CC)N(C)CC2)=O)CCC2CCN(C(=O)COC)C2C1 C(=O)(CC(CC)CC(F)(F)F)NC1(CO)CN(C(c2cc(OCC)no2)=O)C1 C1(NC(=O)COCCc2ccsc2)CC2CCC(C1)N2C(=O)CCCSC1CC1 C(=O)(C1=NNC(=O)CC1)NC(C(CCc1ccccc1)NC(COC)=O)C N1(C(C(COC)O)=O)CCCN(C(c2sc(CO)nc2C)=O)C(C(C)C)C1 c1(C(N2CCC(C)C2C(=O)NCC2OCCC2(C)C)=O)cccc(F)c1F C1(OC)CN(C(=O)CC2NC(=O)NC2=O)CC1NC(c1nnc(C)s1)=O c1(CNCc2c(C(C)(C)C)con2)ccc(S(N)(=O)=O)s1 CC1=NOC(C)(CNC(=O)C(C)(C)CN(C(=O)C(C)OCC2CC2)C)C1 C1(CC)CN(C(=O)CNC(C)=O)CCN1C(=O)CC1CC1.C(=O)(CCC1CCCC1)N CC(C)C(CNC(C1(CN(C)C)CC1)=O)C(=O)NOC1CCCC1 N1(C(C(C)OCCC(C)C)=O)CCC2CC1CN2C(c1cnc(C(F)(F)F)s1)=O N1(C(c2ncn(C)c2)=O)CC(NC(=O)CS(C)(=O)=O)CC12CCCOC2 c1(N(c2n(C)ccn2)C2CCCCC2)ccc(S(=O)(=O)NC2CC2)cc1N C(=O)(C(O)CC(F)F)N(CC(C)(C)CNC(=O)Cc1ccc(C(C)=O)s1)CC N1(C(c2nc(C)n(C)n2)=O)CCC2CCC12CNC(c1ccncc1Cl)=O C=C(C)C(CC(=O)N(CCCNC(c1c(Br)n[nH]c1C)=O)CC)OCC CC1CCC(C)N1CC(=O)NCCc1cc(C(=O)NC2CC(Cl)(Cl)C2)no1 c1(OC)ccc(C(=O)NC2(C)CC(NC(C3COC(=O)N3)=O)C2)c(Br)c1F c1(N(CC(=O)N(C2CCN(C(C(C)S(N)(=O)=O)=O)C2)C)C)ncnc2[nH]cnc12 C1(OCC)CCC(C)(NC(=O)C(N2CCC(C(=O)NC3CC3)CC2)=O)CC1 N1(C(C2C(=C)C2)=O)CCCCCCC1C(=O)NCCN(C(C)C)CC c1(C(=O)NC2CCCCN(C(CCC(=O)NC)=O)C2)c[nH]c2cc(C)ccc12 c1(C(N2CCC(N(C(=O)CSc3nncn3C)CC)CC2)=O)c(O)cccc1F Cc1cc(CCC(=O)NCCc2cc(C(N3CCCC3C(C)(C)O)=O)no2)on1 c1(CN2C(C(=O)NCCN(C)C)CC3(CC3)C2)cc(Cl)c(F)c(Cl)c1 N1(C(c2occ(C(=O)OC)c2)=O)CCCN(C(=O)C2=CCCC2)CC1 N1(C(C(CC)OC)=O)CCCC2(CCN(C(c3c(Cl)cnn3C(C)C)=O)CC2)C1 Cc1cccc(CC(N2CCN(C)CC2CNC(=O)C=Cc2ccc(Cl)s2)=O)c1C C1(C2CCN(C(C=C(CCC)C)=O)C2)CCCCN1C(C1CCCC(O)C1)=O Cc1nc(C2CC2)ncc1C(=O)NCC1CC(NC(c2cnc(N)c(F)c2)=O)C1 NS(=O)(=O)CC(O)CNC(=O)NCc1ccc(N2CCCCC2=O)cc1 c1(OC)c(C(=O)N(C2CN(C(c3coc(O)n3)=O)C2)C)cc(Br)cc1F C1(C)(CNC(C(C)N(C)C)=O)CCN(C(=O)CC2(CO)CC2)CC1 c1(C(N2CC3(OCC(NC(CCSCCC)=O)C3)C2)=O)cc2c(cc1O)OCO2 c1(NC(N(CC(C)NC(c2ccccc2)=O)Cc2nc(C)on2)=O)ccc(Br)cc1 Cc1nscc1CN(C)C(C1(C)CN(C(=O)CCC2CCC(C)C2)C1)=O N1(C(c2ccc(C#C)o2)=O)CC2CN(C(c3cc4cn[nH]c4cn3)=O)CC2C1 c1(C(=O)NC2CN(C(c3cc(C)oc3)=O)CC2C)cc2cccc(C)n2n1 C1(O)(CNC(c2cnc(CCCC)s2)=O)CCN(C(c2[nH]c(C)nc2CC)=O)C1 c1(CC)nc(C)c(C(=O)N(C2CCN(C(=O)C(C)(CO)OC)C2)C)s1 Cc1cn2cccc(C(=O)NCC(C)(O)CNC(=O)Cc3cnn(C)n3)c2n1 C1(C)(CC)CCCN(C(C2CCC(O)CN2C(=O)CS(C)(=O)=O)=O)C1 c1(C(=O)NC2CN(C(CCC=C(C)C)=O)C2)ccc(-n2ccnc2)c(Cl)c1 c1(CC)ccc(C(N2CCC(NC(=O)CN3CC4CC4C3)CC2C)=O)c(N)c1 N1(C(Cc2c(C)occ2)=O)CCC2CN(C(=O)Cn3ccccc3=O)CC12 C1(c2cccs2)(C(N2CCCC(NC(c3c(C)snn3)=O)C2)=O)CC2(CCC2)C1 CCC(C(C)C)C(C(=O)NCC(=O)OCC)N(C)CCC1CCOC1.C(C)(C)(C)O CCC1Cc2c(cccc2)CNC1=O.c1(CC)nc(C(C)C2CC2)no1 c1(C(=O)OC)cc(C(N2CC(O)(CNC(C3(C)CC(C)C3)=O)C2)=O)c(C)s1 c1(OC)ccc(Cl)cc1C(N1CC2CC1CC2C(=O)NCc1ccc(F)cc1)=O C(=O)(CCCC(=O)N(C)C)N1CC(N(C(C(C)C2CCCC2)=O)C)C1 c1(C(=O)NCC(C)CN(c2ncccn2)C)cc(N)c(N)cc1F C1(C)(CNC(C2(C(N)=O)CCC2)=O)CN(C(c2cc(N)c(F)cn2)=O)CCO1 N1(C(C2CC(OC)CN2C(c2ccc(Br)cc2Br)=O)=O)CC2OCCOC2C1 N#Cc1ccc(Br)cc1CN1CC(NC(c2cc(Br)cc3cn[nH]c23)=O)C(F)C1 C(C(CNC(c1cccnn1)=O)CO)NC(C1(CC(C)C)CCC1)=O C1(C(N2CCCC3(CN(C(=O)CC4CC4)C3)C2)=O)CC(c2ccccn2)=NO1 c1(OCC)nccc(C)c1C(=O)NC(CNC(=O)C(F)CC)CO C1(C)(C(=O)NCCn2ncc(C)c2)CCN(C(=O)C(O)CC2CCCC2)C1 C1(C(=O)NCCCCC)CC(O)CN1C(=O)CS(=O)CC N1(C(CCCNS(C)(=O)=O)=O)CCCC12CCCN(C(c1ccc(=O)oc1)=O)C2 c1(COCC)cc(C(=O)NC(C)CC(C)NC(=O)CC2(C(=O)OC)CCC2)no1 N1(C(c2n(CC)ncn2)=O)CCCC(C)(C)C1CNC(C1CC(C#N)C1)=O N1(C(C2CC(=C)C2)=O)CCOC(CC)CC1.c12c[nH]cc1CNC2=O N1(C(c2c(COC)nns2)=O)CC(CNC(=O)CCCCCSC)OC(C)(C)C1 N1(C(COCCN(C)C)=O)CCCCC1C(=O)NC1(CO)CCCCC1 Cc1nc2c(s1)CN(C(=O)CC1(C)CCN(C(C3CC(=O)CCO3)=O)C1)C2 N1(C(C(CCC)C)=O)CCN(C(c2cnc(C3CCC3)[nH]2)=O)CC1C1CCC1 C1(C(=O)NCCN(C(=O)C(Cc2ccccc2)C2CC2)CC)CCN(C)C1=O c1(C(=O)NCC(C)N(C(C(C)N(C)C)=O)CCO)ccnc(C2CC2)c1 CC1(C(N2CC(=C(F)CNC(c3coc(-n4ccnc4)c3)=O)C2)=O)CC2CC2C1 c1(CNC(C(C2CCN(C(=O)C(c3ccccc3)=O)CC2)C)=O)cnc(Cl)cn1 Cc1cc(C)c(NC(N2CCC3(CC3)C2)=O)cc1C Cc1cccc2c1OCC2C(=O)N1CC2CCC1CN2C(=O)C(F)CC1CC1 C1(CNC(C2(CC(C)C)CC2)=O)CCN(C(=O)CC2CCSCC2)C12CC2 CC1(C)C(CC(=O)Nc2cccc(F)c2)CCN1C(c1ccncc1)=O C(=O)(CCS(=O)(=O)NCCl)N1CC(COC)C1(C)C c1(OC)cccc(C(O)C(N2CC3C(CNC(C4CS(=O)(=O)C4)=O)C3C2)=O)c1 c1(CNC(=O)CC2CCC(NC(C3CC=CCO3)=O)C2)ncccc1F N1(C(C2C(C)(C)CCCC2)=O)CC2CC(NC(=O)C3=CC4(CCOC4)C3)CC2C1 c1(CNC2CC(NC(c3cccnc3S)=O)C2)c(F)ccc(F)c1Cl C#Cc1cc(F)c(C(=O)NCC(C)NC(C23C=CC(CC2)C3)=O)cc1F c1(C(N(CC(C)NC(=O)C(C2CCCCCC2)O)C)=O)cccc(C2CC2)c1 N1(C(=O)CCc2cnn[nH]2)CC2CCOC2C1.C1(=O)CCCN1 CON(CC1CCCO1)C(=O)CCN=[N+]=[N-] N1(C(C(=O)Nc2c(N(C)C)cnc(Cl)c2)=O)CC2CN(c3ccccc3)CC2C1 Cc1nc(Cl)ccc1C(N1CC(N(C)Cc2cc(C(F)(F)F)ccc2O)C1)=O C(=O)(C(CNC(C1CCN1C)=O)CC1CC1)NC(CN(CCCC)C)C C=CC(C)C(C)C(=O)NCC1CC(NC(=O)Cc2c(C)n[nH]c2C)C1 c1(OC)cc(CC(N2C(C)C3CC2C3NC(C2(CC(C)C)CC2)=O)=O)ccc1C C1(F)(C(=O)NCCC(C)NC(c2cccc(NC(C)=O)c2)=O)CCC(C)CC1 Cc1nc(NCC(N2CCN(C(C3C(C)CC3C)=O)CC2)C)c(C)c(O)n1 c1(CN(C(C2CC2c2ccccc2)=O)CC)cnn(CC2CCCCC2)c1Cl N1(C(C2N(C(CCC#C)=O)CCSC2)=O)CC(C)(C)OC(C)(C)C1 C1(NC(=O)CCN(C)C)CCCN(CC(=O)Nc2c(NC(C)=O)cncc2)C1C C(=O)(CC(C(F)(F)F)c1nccn1C)NCCCN(C)C(c1nc(Cl)cs1)=O CC1OC2(CN3CCCC3C3CN(C(=O)CSc4ccccc4)C3)CC1C2 N1(C(CSCC(N)=O)=O)CCN(c2ccccc2CNC(C2CCC(O)C2)=O)CC1 C1(C(=O)OCc2nn(C)c(=O)n2C)CCC2(CC1)C(C(=O)OC)C2(F)F N1(C(=O)NC2C(C(=O)OC(C)(C)C)C2(C)C)CC2C3C=CC(C2)C1C3 Cc1ncccc1-c1cn(CC2CCN2C(C2(C(C)C)CCC2)=O)nn1 C(=O)(CCCCCC(C)C)N1CC2C(CNC(c3c(CC)cc(C)cc3)=O)C2C1 C1(C(=O)NC(CC(=O)NC)C2CC2)CC12CCN(C(=O)CC(C)(C)C(C)=O)CC2 N#CC12CCC(C(N3CCC4CN(C(=O)CC5CC5)CCC34)=O)(CC1)CC2 C1(NC(CC(CC)SC)=O)C2CCC1N(C(=O)C(c1cccnc1)OC)C2 C1(CNC(c2n(CC)ncc2)=O)C(C)CCN1C(c1nc(C)cs1)=O Cc1cc(F)cc2[nH]c(C(=O)N(CC(C)NC(=O)CC3(C)CCCC3)C)cc12 N1(C(c2coc(O)n2)=O)CCC(CNC(C2(C(F)F)CC(O)C2)=O)C(F)(F)CC1 N1(C(C(CC)Cc2ccccc2)=O)CCCC(C)(Cc2cn(CCC(C)C)nn2)C1 N1(C(C2(C(C)C)CC2)=O)CC2(C1)CN(C(C13CCC(N=[N+]=[N-])C1C3)=O)CCO2 c1(C(=O)NC2(Cc3ccccc3)CC2)ccc2c(c1Cl)OC(F)(F)O2 C1(CO)CCCN(C(C2CCC(NC(=O)COC3CC4CCC3C4)C2)=O)CC1 C1(CCNC(C(C)N(C(C)=O)C)=O)CCN(C(=O)CCOCCN(C)C)C(C)C1 O=C(N=c1ncn(C2CCCC(O)C2)[nH]1)C1CC(O)c2ccccc2C1 C(C(C(=O)NOCC1CCOC1)C(C)(C)C)NC(c1ccc(C)cn1)=O CCC(CNC(=O)Cc1cc[nH]n1)(CC)C(=O)N1CCCC(C(C)(C)O)C1 Cc1cc(C#N)ccc1NC(N1CC(CNS(=O)(=O)c2cn[nH]c2)C1)=O CC1CN(C(c2cn[nH]c2)=O)CCC1NC(c1cccc(-n2ccnc2O)c1)=O c1(OC)cc(Cl)c(Cl)cc1C(=O)NCCN(C(=O)Cc1ccccc1SC)C C#Cc1ccc(NC(C2CCOCCN2C(=O)C(Cl)Cl)=O)c(C)c1 CC(C(C)(C)C(=O)NC(c1nc[nH]n1)C1CC1)NC(C1CC=CC(O)C1)=O C1(CNC(c2cnco2)=O)CN(C(c2cccc(OCC(F)(F)F)c2)=O)CC1O C1(C(=O)NCC(C)NC(=O)CC2CCCN2C)CCCC(F)(F)CC1 C1(C(N2CC(CNC(C3CC(=O)NC3)=O)C2)=O)Cc2cc(Br)ccc2O1 c1(C(=O)NC2C(n3cc(C(CC)O)nn3)CCCC2)c2c(nn1C)CCOC2 CC1CCCN1CC(=O)NC1CN(C(C2CCCN2S(C)(=O)=O)=O)C1 c1(N2CC3C(CNC(C4CCCCO4)=O)(C3)C2)ncc2c(n1)CCC2 c1(NC(C(C)NCc2ccc(F)nc2)=O)ccc(C(F)(F)F)c(N)c1 CCCC(C)CC(C(=O)NCC(C)(C)C)N1CCOC(CC(=O)NC(C)C)C1 N1(C(c2cc(C)on2)=O)CC(C)OC2(CCN(C(=O)CSc3nccs3)C2)C1 c1(CC)nn(C)c(C(=O)N(CCC(C)NC(C2CCOCC2)=O)C)c1Cl C(CCNC(=O)C(O)CCc1ccccc1)(C(C)C)NC(C1N=C(C)SC1)=O C1(NC(C(CC)=CC)=O)CCC2CN(C(c3ccc(F)c(O)c3)=O)CCC2C1 Cc1cc(C(N2CC(NC(=O)CO)C(F)C2)=O)nc(Cl)c1 N1(C(Cn2cc(C(C)O)nn2)=O)CCCN(C(=O)C2=NOCC2)CCC1 C1(NC(c2ncn(CC)c2)=O)CC2(C1)CC2C(=O)NC1CCCC(C)C1 c1(N2CC(C)N(C)C(C)C2)ncc(S(=O)(=O)NCCCSC(F)(F)F)cc1Cl c1(OC)cc(C(C)(C)NC(C2CCCC2n2cc(COCCC#N)nn2)=O)sn1 N1(C(CC=C=C)=O)CC(NC(=O)Cc2ccc(I)cc2)CC1(C)C C(=O)(C#CC1CCCCC1)N1CCN(C(C2C(C)(C)CO2)=O)CC1CO C(=O)(C#CC1(C)CCCO1)Nc1c(C)n[nH]c1C.C1(=O)C(C)NC2(CC2)N1 C1(C(N2CCCC(NC(CCOC)=O)(CO)C2)=O)CC2C=CC1CCC2 N1(C(c2ccc(SC)o2)=O)CCCN(C(=O)C(C)c2ccsc2)CC1CO CC1OC(C)CC1C(N1CCC(NC(C23CCCCC2C3)=O)C1)=O c1(-c2ccc(NC(C)=O)nc2)ccc2cc(O)c(C(=O)Nc3ccno3)cc2c1 N1(C(C2C(=C)C2)=O)CCC(NC(=O)C(C)NC(=O)Nc2ccoc2)C(C)C1 c1(C(N2CCC(C(=O)O)(COC)C2)=O)cc2ccccc2n1C C12(NC(C(CCSC)OC)=O)CCCC1N(C(c1cc(F)cc(F)c1)=O)CCC2 Cc1nc2cncc(C(=O)NCC3(CNC(=O)C(C)C(C)C)CCCC3)c2[nH]1 c1(C(=O)NC23CCCC2CN(C(C24CC5CC2C4C5)=O)C3)c[nH]c2cccnc12 c1(C(N2CCC(NC(C(C)Oc3c(OC)cccc3)=O)C2)=O)ccc(I)cc1O N1(C(C(C(C)C)=O)=O)CCC2(C1)CN(C(=O)CCc1cccs1)CCO2 N1(C(CC(=C=C)C)=O)CCCC(O)(CN(C(=O)CCc2cnccn2)C)C1 C1(CC(=O)NC2CCN(C(C(C)(F)F)=O)C2)CCC2(CCC2)CO1 Cc1ccc(OCC(=O)NC2CCC2CNC(=O)CC2CC2)cc1 c1(C(N(CCOCCN(C(C(C=C=C)C)=O)C)C)=O)cccc(N)c1O C1(C(=O)NCc2occ(C(=O)Nc3ccc(O)nc3)c2)CC12CCCCC2 N=c1c(C(=O)NCC2CC(O)CN2C(C2CNC(=O)C2)=O)c[nH]cc1Br N1(C(c2c(CCC)n[nH]c2)=O)CCC(C(=O)N2CCCC(C)(C#N)C2)=C(F)C1 CC1(C)CCOC1CC(=O)NC1CC(NC(=O)CC2CCCCCC2)C(O)C1 c1(C(N2CCC(NC(c3cncc(F)c3)=O)(CO)C2)=O)cncc2ccsc12 Cc1ccc(Cl)cc1N1CCN(Cc2cn(CCc3cncnc3)nn2)CC1 C(=O)(CCC(F)(F)Cn1cc(CN2CCOCC2C)nn1)NC1C(CCC=C)C1 N1(C(c2c(C)nc(O)[nH]2)=O)CCCN(C(C2CCCO2)=O)CC1C(C)C CC(C)CC(C(=O)NC12CCN(CC1)C2)N(C(=O)C(C)NC(N)=O)C C1#CCCC(O)CC(NC2CC2C2CCCC2)C1 c1(NS(C)(=O)=O)cccc(C(N2CCCCC2CN2CCC(CC#N)CC2)=O)c1 C1(C(=O)NCC(NOC)=O)CCN(CCC(C)=O)CC1 C12CCC(CC1)NC(Cc1ccccc1)C(=O)N2.c1(OCC)ccccn1.O(N)C Cc1nc(C(=O)NC(C)(C)CNC(=O)C(C2CCOCC2)F)c(C)n1C C(CCC(C)C(=O)NC1CN(C(=O)C(F)CC2CCOC2)CC1(C)C)OC N1(Cc2cc(C)[nH]c2C)CCc2ccsc2C1C N(C1CN(C(=O)C=CC=C(Cl)Cl)Cc2ccccc21)C(C(c1n(C)ncc1)O)=O N1(C(CCCNC(C)=O)=O)CCCN(C(C2OCCC2C(C)C)=O)C(C)C1 S(=O)(=O)(c1cnn(C)c1)N(CC(=O)NCCS(=O)C(C)(C)C)C C(=O)(N1CCC(C(=O)NCC23CCCC(CO2)C3)O1)c1cc(COC)on1 c1(CNC(=O)CN2CCCCCC2CC(F)(F)F)nc2cccnc2s1 c1(C(=O)NC2C(C)CCN(c3nnc(C(N)=O)s3)C2)cn(C)c(=O)nc1O n1(CCC(=O)NC(C)CN(C)C(c2nc(Cl)cs2)=O)cnc2sccc2c1=O N1(C(=O)Cc2cnoc2)CCN(C(C2(C(F)F)CCCO2)=O)C2(CCC2)C1 c1(C(=O)NCC(C2CCC2)NC(C2(C=C)CC2)=O)cc2nccn2c(O)n1 CCC(CC)CC(F)C(=O)NC(c1ccccc1)C(=O)NC1CCC(N(C)C)C1 N1(C(C(C)=C(C)C)=O)CC(C)(CNC(=O)Cn2cc(C(F)F)cn2)CC1(C)C c1(C(N2CCC(F)(CNC(C(C=C)(C)O)=O)CC2)=O)ccc2c(c1)ncn2C C(=O)(C(F)C(C)(C)O)N1CC(C)(OCC(=O)NC(C=C)C2CCC2)C1 C1(NC(CC2COCC(C)O2)=O)CCN(C(c2ccnc(SC3CC3)c2)=O)C1(C)C C1(N(c2snc(C)n2)C)CCC2CN(C(c3ns[nH]c3=O)=O)CC12 C(=O)(C1=CCC(N)C1)N(CCCF)CC1CCC1.C#CCO c1(OC)c(I)cc(NC(c2csc(CSc3ccc(O)cc3)n2)=O)cc1I n1(CC)cnc2[nH]c(=NCC3CC4(CCCC4)C3)nc(N(C)Cc3ccco3)c12 CCCC(C(O)C(=O)NCc1nc(C)sc1C)NC(c1ccccc1F)=O S(=O)(=O)(c1cccnc1NCCc1ccco1)NC(c1nc2c(s1)CCC2)C c1(C2(C(N3CCC(C(C)NC(CCC(=C)C)=O)C3)=O)CCC2)cccc(C#N)c1 c1(C(N(C)CC2CCCN(C(C3(COCC)CC3)=O)C2)=O)ccc(Cl)c(Cl)c1O CN1CCCC12CCN(C(C1CCCCCN1C(c1nnc(S)n1C)=O)=O)C2 C1(O)(CNC(CN2C(C)CCC2)=O)CCN(C(=O)C=CCF)C1 C(CC(C)C(=O)NC(C)C(=O)NCc1n[nH]c(C)n1)=CC c1(C(N2CCN(C(COC)C)CC2)=O)ccc([N+](=O)[O-])cc1C C1(C(=O)NC2C(CC(=O)N(C3CCCCCC3)CC)CCC2)CC(C)(C)CCO1 N1(C(c2ccn(CC)c2C)=O)CCC(NC(=O)CCc2ccncc2)C(C)C1 c1(C(N2C(CC)CN(C(=O)C=Cc3cccs3)CC2)=O)cc2c(o1)CCCC2 c1(C(=O)NCCC2N(C(c3c(N)nccc3)=O)CCOC2)cc(F)cc(F)c1 c1(OC)c(F)cc(C(=O)NCCC(O)CNC(c2sccc2C)=O)c(N)c1F c1(CC)cc(C(=O)NC(CNC(=O)C=CBr)CC)c(C)nn1 N1(C(CCN(C(C2C(C#N)CC2)=O)C2CC2)=O)CCC12CCCSC2 c1(SC)ccc(N)cc1C(N1CC(CCNC(=O)C=Cc2ccco2)C(C)C1)=O c1(C(N2CCC(CN3CCOCC3)CC2)=O)occc1C1=CCNCC1 c1(C(N2CCC(CNC(c3c(F)ccc(C)n3)=O)C2)=O)cc2c(nn1)CCCO2 C(CC(C(C)(C)C)NC(C1C(C2CC2)C1(F)F)=O)N(C(CCC(=C)C)=O)C N1(Cc2cccc(OCC)c2O)CC2(CCC(C(=O)NC(CC)CO)O2)C1 c1(C(=O)OC)cc(NCCNC(=O)C(C)CN2CCOCC2)cn1C C1(CCNC(C(CC)n2nccc2C)=O)CCCCN1C(c1nnsc1C)=O N1(C(C2C(C)C2)=O)CCOC2(CCC(NC(c3ccc(S(C)(=O)=O)o3)=O)CC2)C1 Cc1noc(Cl)c1CC(=O)NC1CN(C(=O)Cn2cnc(C(F)(F)F)c2)C1 c1(C(=O)NCCCCNC(C(C2CC(OC)C2)F)=O)cc(SC)n(C)n1 c1(C(=O)NCCn2cc(-c3ccncc3Cl)nn2)cccc2sccc12 C(N=c1cc[nH]cc1S(=O)(=O)NCCCOC1CC1)C1(OCCO)CCOC1 c1(CC(=O)N(CC(C)C)CCSc2cn[nH]c2)ccc(-c2cncc(N)c2)cn1 c1(C(NC(CCC=C(C)C)C)=O)noc2c1CC(C)CC2 C1(C(=O)NCc2c(CN(C)C(c3cnc[nH]3)=O)cccc2)CCn2ncnc2C1 C1(NC(Cc2nnc(C)o2)=O)CCOCC1NC(C1(C)COCCO1)=O C(=O)(C(C)(C)S(=O)(=O)C1CC1)N1CCCC(NC(C(CCC)NC(C)=O)=O)C1 N1(C(C(C)(C)OCC)=O)C2CC1CN(C(C1CC13CCOC3)=O)C2 c1(NC(=O)Nc2cc(CC)no2)[nH]c2ccccc2c1COC c1(-c2n(CCC(C)(C)C)nc(-c3cc[nH]n3)n2)noc2nc(C(F)(F)F)ccc12 c1(CNC2(c3n(C4(C)CC4)nnn3)CCSC2)cccn2cncc12 S(=O)(=O)(CC(=O)NC1CCCC1C(N1CCC(CO)CC1)=O)NC C1(OCC(=O)NCC(c2ccccc2)CC)CCNC1=O C12(NC(Cc3ccn(C)n3)=O)CC1CN(C(c1csc(Cl)n1)=O)C2 c1(C(N(CCN(C(=O)C(O)c2cnc[nH]2)C)C)=O)nncc2c1CCCC2 C1(NC(C)=O)CC2(CCC(CNC(c3cscc3C)=O)OC2)C1 N1(C(C(CC(C)C)OC)=O)CCC2(CC1)CC(NC(c1n[nH]cc1C)=O)CCO2 C1(C(=O)NC(C)CC(C)(C)C)CN(C(=O)CCc2cnn[nH]2)CC(C)(C)C1 c1(CC)ccccc1C(N1CC2CC2(C(=O)NCC(CC)CC)C1)=O C1(NC(=O)Cn2cnc(Br)c2)CCCN(C(=O)C(F)(F)C(F)F)CC1 C#CCCCCCCCC(=O)NC(C)(CNC(C1(O)COC1)=O)C(C)C Cc1nc(N2CCC(N(C(c3cc(CC(C)C)on3)=O)CC3CC3)C2)n[nH]1 c1(-c2cn(C(C(=O)OC)C)nn2)ccccc1CNC(c1cc(Br)c[nH]1)=O C1(C(C(=O)OC)C)CCCN(C(c2c[nH]cc2C)=O)C1.C(C(C)C)N(CCO)CC CN1CCC(CC(=O)NC2(C(=O)N(C3CC4CC4C3)C)CC2(C)C)CC1 C1(NC(C=CCSC)=O)COC2(C1)CN(C(=O)COCC(c1ccccc1)C)C2 c1(C(=O)NC2C(C(N3CCC(NC(C)=O)C3)=O)C2)cc(O)cc(F)c1 C1(n2cc(C(=O)NO)nn2)(NC(C)=O)CCN(C(c2ccc(Cl)nc2)=O)C1 CC1(C)CC(CNC(C23CCC(F)(CO2)C3)=O)CN1C(c1ccncn1)=O C1(C(F)(F)F)(NC(=O)NC(c2occc2Br)C)CCCN(C(=O)NC2CC2)C1 O=C1C=C2CN(C(c3csc4ccccc34)=O)CCC2S1 N1(C(C(C(C)C)n2ccc(Br)c2)=O)CCCCCC(NC(=O)C2=CCCS2)C1 C12(C(=O)NC3C(NC(C(CC(C)C)O)=O)CCC3)CC3CC(C1)CC(F)(C3)C2 c1(C(N2CCN(C(=O)Nc3ccc(F)cc3)CC2)=O)cc(F)cc2cc[nH]c12 N1(C(CCC2C(C)C2)=O)CCC2(CC(NC(c3ncc[nH]c3=O)=O)C2)C1 c1(C(=O)NCC2C3N(C(CC(CC)SC)=O)C(CC3)C2)c(N)cc(F)cc1Cl c1(N(CCCC)C(c2cscc2-c2cccc([N+](=O)[O-])c2)=O)cccn2nccc12 C#Cc1cccc(C(=O)N(C(CNC(=O)Cc2cnn(CC)c2)C2CC2)C)c1F c1(NC(C2N(C(c3cc(CC)nc(C)c3)=O)CCC2)=O)cc2n[nH]cc2cc1C C1(C(=O)NCC(C(=O)NC)(C)C)CCN(C(c2n[nH]c(=N)[nH]2)=O)C12CCC2 C1(CC(=O)NC(CC)Cn2cncn2)CCN(C(=O)CC(C)(C)C)CC1(C)C N1(C(CC2(CC)CCC2)=O)CCN(C(c2cccc(C(=O)NC)n2)=O)C(CO)C1 c1(C(=O)NCCOCC(=O)Nc2ccc(C)nc2)cc2ccccn2n1 CC1CN(C(C2CCSC(C)C2)=O)CCN1C(=O)Cc1cccc(C(N)=O)c1 CC1CC(F)(F)CCN1C(C1N(C(c2ccc(F)c(F)c2)=O)CCC1(C)C)=O N1(C(C2C(C(=O)OC)CC2)=O)CCCCC(NC(=O)CC2CC(OC)C2)C1 N1(c2nc(C)nc(C#N)c2)CCCC(C2CC2NC(c2ncncc2Cl)=O)C1 c1(NCCOCC)ccc2c(F)cnc(Cl)c2c1 C(CN=c1[nH]c(=NC2CCS(=O)C2)[nH]c2c1CCCC2)N1CC(OC)C1 C1(CC(=O)NCC2(NC(C3CC3F)=O)CC(F)(F)C2)CC2(CCC2)C1 C(=O)(C1COc2cc(F)ccc21)OCC[Si](C)(C)C N1(C(c2cc(COC)no2)=O)CCC(CCN(C(=O)CCC=CBr)C)CC1 c1(C(N(CC(CC)NC(CC=C)=O)C)=O)sc(-c2cnccn2)nc1C N1(C(C2C(CCOC)C2)=O)CC(CNC(c2ccc(F)cc2C)=O)CC1(C)C N1(C(C2CC2(F)F)=O)CCC(C2CCCCN2C(c2cnn(C(C)C)n2)=O)CC1 N1(C(=O)NCCCSCCN(C(=O)OC(C)(C)C)CC)CCOCC1C1CCC1 C(=O)(C(C)CC(F)(F)F)N1C(C(NOCC(=O)OC)=O)CC(F)CC1 C(=O)(C=CSc1nc[nH]n1)NCC(CC)NC(=O)COCCCC(C)C CC1SCCCC1C(=O)NC(Cc1ccco1)C(N1CCC(C(C)C)(CO)C1)=O N1(C(c2c[nH]c(=NC)s2)=O)CCC2(CC2C(N2CCCC(C)(CC)C2)=O)C1 C(=O)(C(CC)C(=O)N1CCC1C(=O)NC1C(O)CC1O)OCC N1(C(C2(CC)CCC2)=O)CCC2CN(C(C3(CSC)CC3)=O)CCC2C1 C(CNC(=O)Cc1ncc(C)s1)(CC(C)C)NC(C(C)NC(CC)=O)=O C(CCC(=O)NCCC(C)NC1(O)CCC1)OCCOC.C(C)(C)(C)OCCNC(=O)N C1(C(=O)NC2(CO)CCN(C(C(CCOC)OC)=O)C2)CC2(C1)NC(=O)NC2=O N(C(=NCCN1CCOC1=O)NCCF)C(C)COc1cccc(F)c1 CN1CCN(CC)CC1.C1(C(C(=O)O)(F)F)CCN(CC(O)CN(C)C)CC1 Cc1cc2ccc(C(=O)NC(C)C(CO)NC(C3(C)C(C)(C)C3(C)C)=O)cc2o1 C1(N(CC#C)C(C2(n3cc(Cl)cn3)CC2)=O)CCN(C(C2(CC)CCCO2)=O)CC1 Cc1cc(C(=O)NCC(CO)NC(=O)CC2CC=CCN2C)c(C)n1C C1(NC(C(COC)OC)=O)CC2(CCCCN2C(=O)CC2CCCNC(=O)C2)C1 CC(C)CC(C(=O)NC1CC(NC(C23CC(C)(CCO2)C3)=O)C1)C(N)=O C1(C#C)(C(=O)NCC2(OC)CCCCC2)CCN(C(=O)C=CC(F)F)C1 C1(CNC(CN(CC)CC)=O)CC2CCCC2N1C(=O)CN1CCCCCC1 c1(C(=O)NC2C(NC(C(C)NC(N)=O)=O)CC2)sccc1-n1cnnn1 c1(CC(=O)NCC(O)CNC(C2CC2C2CCOCC2)=O)ccc2c(c1)CCO2 CCC(C(=O)NC1CCCN(C(=O)CCn2ccnc2)CC1)C(F)(F)F N1(C(C2CCC(C(C)=O)O2)=O)CC2CC(C1)CN(C(C1(C)CCC(C)C1)=O)C2 CC1CCN(C(=O)Cn2ccc(O)nc2=O)CC1CNC(c1cnoc1)=O c1(C(=O)NCCN(OC)C)cnc(CNC(=O)CC(C)C2CCCO2)nc1 N(C(=NCC1CCOC1)N1CCCC(O)CC1)Cc1cc(C)ns1 N1(C(C(C)O)=O)CC(NC(=O)Cc2ccn(-c3ccc(Br)cc3)n2)C2CC2C1 C=C(Cl)CC(C(=O)Nc1ccc(Cl)c(O)c1)NC(C1CCCCC1OC)=O N1(C(CCN(C)CC)=O)CCN(C(=O)CS(C)(=O)=O)CC(CO)C1 N1(C(c2ccc(OC)c(Br)c2)=O)CC(C(=O)O)C2(C1)CN(C(=O)CC(C)O)C2 C1(C(=O)NCC=CCC(=O)NC(COC(C)C)CO)CCN(C)C1 c1(C(N(C2CCN(C(CCC(C)CN(C)C)=O)C2)C)=O)cccc2nc[nH]c12 CC1(C)C(C(N2CCC(NC(C3CC4CC4C3)=O)C2)=O)CCS1(=O)=O C#Cc1ccc(C(N2CCC(NC(=O)CC3CCCC3)C2C(C)C)=O)o1 C(CN=C(NCC1=CCOCC1)N1CCC(F)(F)C1)OCc1n(C)c(O)nn1 C(C)(C)(C(=O)NCC1CC(F)(CNC(=O)CNC(=O)OC)C1)OCC CC1(C(N2CCOC(C(=O)NC3(CCF)CC3)C2)=O)CC2CC2C1 CC1CC1(C#N)C(N1CC(CCNC(c2nc(C(F)(F)F)cs2)=O)C1)=O c1(CNc2nccc(CC(C)C)c2F)cc2c(cn1)COCC2 Cc1cccc2c1CN(C(=O)CC1(C)CCN(C(c3ccnnc3O)=O)C1)C2 C1(NC(C2CC3CCC3C2)=O)CCCCN(C(=O)COc2ccc(Cl)cc2F)C1 c1(C(=O)NCCCC(C)NC(C2(C3CC3)CCOCC2)=O)cncc2nc[nH]c12 c1(C(=O)NCC(CN(C(CCc2cnc(C)s2)=O)C)O)c(Cl)nn(C)c1Cl N1(C(c2c(C(=O)OC)cn(C)n2)=O)CCCCC(NC(c2ccc(F)o2)=O)C1 C12(C(=O)NC(C)CC(C)NC(=O)Cn3nnc(C4CC4)n3)CCCC(C)(C1)OC2 C(C(CC(C)C)C(=O)N1CC(CC(F)F)C1)NC(CCSCCC)=O CC(C)(O)C(C(=O)Nc1cncc(F)c1)NC(=O)CCn1ccnc1 CCCCC(C)C(=O)NCc1ccc(C(=O)NCC2CC(C3CC3)=NO2)s1 c1(C(=O)NCC2(OC)CN(C(c3c[nH]c(=NC)s3)=O)C2)cccc2c1nnn2C n1(CC(N2CCC(CCNC(c3cc[nH]n3)=O)C2)=O)nnc(-c2ccsc2)n1 NS(=O)(=O)C1(C(N2CC(NC(=O)CCc3ccncn3)C(F)C2)=O)CC1 c1(C(=O)NCC2C(C)(C)C(NC(=O)OC(C)(C)C)C2)n[nH]c2c(Br)cccc12 c1(C(N2C(CNC(C3(CC=C)CC3)=O)CCC2)=O)cc(Br)ccc1OC C1(c2cc(C)[nH]n2)CN(C(=O)C(=O)Nc2ccc(N3CCCCC3)cn2)CCO1 CC1(CNC(=O)Cn2[nH]cnc2=N)CCCN(C(C2(C(F)F)CCCO2)=O)C1 C1(CNC(C2C3CC(=O)CC23)C)CCC(CC(=O)NC2CC2)CC1 C(C)(C(C)(C)C(=O)NC1CC(=O)N(c2ccc(OC)cc2)C1)NC(CCC)=O NS(=O)(=O)c1n[nH]cc1C(N1CC2CCC1CN2C(=O)CCc1cc[nH]n1)=O CC1OC2(C(N3CCC(CN(C(=O)C(C)OC(C)(C)C)C)CC3)=O)CC1C2 C1(C(N2C(CNC(C(COC)C)=O)COCC2)=O)CCOC(C)(C)C1 Cc1csc(=O)n1CCC(=O)N(CCCN(C(=O)CC1CCOC1)C)C N1(C(CCOCCSC)=O)CCN(C(=O)Nc2cnn(C)c2)CC1C1CCCC1 C12(C(=O)NCC3CCCN(C(c4nc(C(C)C)sc4)=O)C3)CCOC1CCOC2 CC(C(=O)N1CCC(CNC(c2sccc2C(F)F)=O)C1)P(C)(C)=O c1(CC(C)OC(CCCC)=O)ncc(Cl)cn1 C(CC(C(=O)NC(COC(C)C)C(=O)NCC(O)CCC1CC1)OC)OC c1(C(N(C(C)C(=O)NCC(O)C(F)F)CC)=O)ccc(C)c(F)c1F C=C(CNC(=O)C(C)SCC)CCNC(=O)C(O)CC1CC1 C(=O)(C(CNC(=O)C=Cc1ccncc1)C(C)(C)C)NC1C(CC(C)(C)C)C1 C1(C(N2CC(=C(CNC(C3N(C)C(=O)NC3)=O)F)C2)=O)COC2COCC12 C1(C(=O)NCCC(C)NC(C2N(C(C)C)CCC2)=O)CCCOCC1 C1(C(=O)OC(C)(C)C)C(C(=O)NCc2cn(C3CCOC3)nn2)C1(C)C c1(OC)cncc(C=CC(=O)NC(CNC(=O)CN(C)C(C)=O)CC(C)C)c1 c1(C(=O)NCC=CCNC(c2cn(C)nc2Cl)=O)c[nH]c2cccnc2c1=O C#CCC(C)(C(=O)N(CC)Cc1cccnc1)NC(=O)C(CN(C)C)CC N1(C(C(C)N(C(=O)CCc2nc(=N)[nH][nH]2)C2CC2)=O)CCC(O)(CO)CC1 C(C(CC(=O)NCCc1cccc(O)n1)C1CCC1)NC(Cc1cc(C)sc1)=O c1(C(C)NC(=O)NCCO)ccc(OCC(=O)OC)c(C(F)(F)F)c1.CC C(CC(C)C)(C(=O)Nc1cnn(CCN(C)C)c1)N(C(c1c(C)csc1)=O)C N1(C(C(C)(C)C2CCCC2)=O)CCC(O)(CCNC(c2ccc(C(=O)O)s2)=O)C1 c1(C(=O)NCCCOCCNC(c2cc(C(C)C)[nH]n2)=O)cncc2c1CCC2 C1(C(C)C)C(C(=O)NCCSC(F)(F)F)CCN1C(C12CCC(CC1)C2)=O C1(NC(CCCOCC)=O)CC2CC1CN2C(=O)CCCC1CCOCC1 C12(C(N(C)CCNC(=O)CCc3nccs3)=O)CC(CN1C1CC1)C2.C1(C)CC1 c1(OC)ccc(CNC(c2ccc(CNC(C3CCCN3C)=O)cc2)=O)cc1 N#Cc1ncc(C(=O)NCC(O)CNC(C23CC(Cc4ccccc4)(C2)C3)=O)s1 C1(S(C)(=O)=O)(C(=O)NCC2(CCNC(C(CN(C)C)(C)C)=O)CC2)CC(O)C1 C1(C(=O)NCCC=CCC)CCC(NC2CCN(C(=O)NC)C2)CC1 C=CCCC(C)(C)C(=O)N1CCCC(C(C)C(=O)N2CCC2c2ccccc2F)C1 C1(NC(C2(COC)CCCO2)=O)CN(C(=O)COCc2scnc2C)CCC1C C1(NC(c2scc(OC)c2)=O)CCN(C(C2CC2F)=O)CC1 N1(c2c(C)cccc2)CCCC(NC(c2cccc(C(=O)O)n2)=O)C1=O CCCC(C(=O)N(c1ncc(COCC)s1)CC)OCCO.c12ccc(cc1)NC2.SC C1(C(=O)NCC(CC)(C)OC)(NC(C2CC2C2CCC2)=O)CCN(C)C1 C(=O)(CC(C)P(C)(C)=O)N(C(C)C)CCN(C(=O)C(C)CC(N)=O)C C(=O)(C1=CCCCO1)NC1CN(C(C(C(C)C)c2ccncc2)=O)C1 Cc1ccn2c(C(=O)NC(CNC(c3ccc(Cl)s3)=O)C(C)C)cnc2c1 c1(CNC(C2(OCC)CN(C(=O)C(C(C)C)C3CC3)C2)=O)nnn(C)c1C Cc1csc(C)c1C(N1CCC1(C)CC(=O)NCC1(O)CC1)=O c1(C(N2C(C(N3C(C)(C)C(CO)C3)=O)C3CC3C2)=O)ccc([N+](=O)[O-])o1 N1(CC(=O)NC(COCOCC)C)CCCC(CN(C)C)CC1 C1(C)(CC=C)CCCN(C(=O)Cc2ccnc(OC)c2)C1 c1(CC(=O)NC2CCN(C(c3cnn4ccsc34)=O)C2)cc(F)ccc1F CCC(C(=O)N1CCC1CC(=O)NC(c1cc(C)on1)C)C(F)(F)F C(CC(F)(F)F)N(C(CCN(C(=O)Cc1cscn1)C)=O)C1CC1 N1(C(c2ncc(OC)nc2)=O)CCCC(NC(=O)Cc2cn(C)nc2C)C(F)C1 Cc1cc(C)c(C(=O)NCCN2CCN(C(C3CCCN3C)=O)CC2)o1 S(=O)(=O)(c1ccc(C)cc1)C(C(=O)NCCCCC(C)NC(C(C)=C(C)C)=O)C Cc1ccc(CC(C)C(=O)N2CC(N(C)C(c3cnco3)=O)C2)cc1 C(=O)(C1=Cc2cc(F)ccc2OC1)NC(CNC(C(c1ccc(CC)s1)=O)=O)C Cc1cccc(CCC(N2CC3CC3(NC(c3ccn(C4CCC4)n3)=O)C2)=O)c1 C1(CNC(C2(CC)CC2(F)F)=O)COCCN(C(=O)C(C)(C)c2nccs2)C1 C1(C(N2CCC(CO)C(O)C2)=O)(OC)CCN(c2ncc(OC)cn2)CC1 N1(C(c2cn(C)c(=O)cn2)=O)CCC(NC(=O)C2=CCS(=O)(=O)C2)C2(CCC2)C1 C(C(C)(C(C)C)C(C)C)NC(C1(OC)CCN(C(=O)CCCCC(N)=O)C1)=O c1(C(N(CCCN(C(C(CC=C)C)=O)C)C)=O)ccc(F)cc1C(F)(F)F N12CCC(C1)OCC2=O.C(=O)(CCC1CC1CC1CC1)OCOC.C1CO1 c1(NC(CCC2CCN(C(CN(CCCO)C)=O)C2)=O)ccccc1Cl c1(C(=O)NC(CNC(c2c(C)csc2)=O)C2CCC2)cnc2c(c1)NCC2 C#CCC(C)(C(=O)NCC1CCS(=O)(=O)C1)NC(=O)COC1CCC1 C1(OC)CCN(C(=NCCSC)NCc2cccc3c2NC(=O)CO3)C1 Cc1cc(C(=O)NCC(C)NC(=O)CCCC2CC2)c(C)cc1Cl N1(c2c(C)c(NCC3(C4CC4)CCC3)ncn2)Cc2ccccc2C(CO)C1 c1(SCC)cnccc1C(=O)NC(CNC(=O)C(F)CC1CCOC1)C(C)C N1(c2nc(SC)c(C)cn2)CC(C)(C)CCC1CNC(=O)CC1(C)CCCO1 N1CCC(C)N(C(=O)C(C)C(C)CC)CC1.c1(CCCC)nc(NC2CCCC2)cs1 N1(C(CCOC(C)=O)=O)CCC2(CCC(NC(=O)CC3CCC(=O)N3)C2)CC1 C(CCCC(=O)NCCN(C(=O)Cc1cc(C)on1)C)NC(C)=O c1(CSCC(N2CCCC2)C)cccc(NC(=O)NC2CC2(Cl)Cl)c1 c1(OCC(N)=O)cccc(C(=O)Oc2ccc(C(F)(F)F)cn2)c1 c1(NCCOC(c2ccc(C)cc2)C2(C)CCC2)ccc(F)cc1Cl N1(C(c2c(OC)n[nH]c2)=O)CCC2(CC1)CC2(CO)CNC(=O)CCCC(F)F C12(C(C)C)CC(C(=O)NCc3ccc(C4CCCO4)[nH]3)(CO1)C2 Cc1ccc(C(=O)NC2(C)CCC(NC(C3CCC(N(C)C)C3)=O)CC2)c(N)n1 C(C1=NOC2(CCC2)C1)NC(C(C1CN(C(C(C)SC(C)C)=O)C1)O)=O C12CCC(CC1)OCC(=O)N1CCC(CC#C)(C1)C(=O)N2.C(CC(C)C)OCF C1(CNC(C2(C)CS(=O)(=O)C2)=O)CC2(CCN(C(=O)Cc3cc[nH]n3)C2)CO1 C1(N(C(C2N(C(Cc3c(C)ccs3)=O)CSC2)=O)CCO)CCC(C2CC2)C1 c1(C(N(CCNC(c2cnc(CCC)s2)=O)C)=O)c(C)oc2ncnc(O)c12 N1(C(=O)C(=O)NCC2CN3CCCCC3CO2)CCC2(CCOC2)CC1 C(=O)(C(C#N)C(C)C)NC1(C)CCN(C(c2cnc(C(C)C)s2)=O)C1 C1(Cl)(C(=O)OC)CC12CCN(C(C1CCCS1)C(=O)NCC(C)C)CC2 C12(NC(C(c3cccc(Cl)c3)CC)=O)CCC(CC1)N(C(C1CC1C(F)F)=O)C2 c1(C(N(C2CCCC2O)CC)=O)n[nH]c2cccc(F)c12 c1(C(=O)NCC(C)N(C(COCCOC)=O)C)ccc2oc(N(C)C)nc2c1 c1(CC)cc(C(=O)NCC=CCNC(=O)C(F)(F)C(C)O)cc(O)n1 C1(N(c2ccccc2)C)CCN(C(C(=O)NC)C(C2CC2)OC)CC1.C1CCOC1 C1(C(NOC(COC)COC)=O)CCC(NC(=O)CC2(CSC)CC2)CC1 c1(C(=O)NCC2C(NC(c3nc(COC)sc3)=O)CCC2)c(C(F)F)n[nH]c1C c1(C(=O)NCCC(CNC(c2c(CC)noc2)=O)O)cccc2c(C)[nH]nc12 C12(CNC(CC3C(NC(c4ccc(OC)o4)=O)CCC3)=O)CC(CO)(CO1)C2 Cc1c(F)cc(C(=O)NCC2CC3(CCC3)CN2C(=O)CC(C)CF)c(F)c1N Cc1[nH]nc2c1CC(C(N1CCCC(C)C1CNC(c1csc(S)n1)=O)=O)CC2 n1(CCS)nnnc1N(CCCC)C.c1(N)ccc(-c2cccs2)o1 N1(C(CCC)=O)CCCCC1CCNC(C1CC=CC(O)C1)=O c1(C(=O)NCC2C(NC(=O)C=CCO)CCC2)cc2ccc(Br)cc2nn1 Cc1nccc2c(=O)c(C(N3CCN(C)CC3C(C)C)=O)c[nH]c12 c1(NCC(CC=C)(C)C)nccc(=NC(C)COC(F)F)[nH]1 CC(Cc1ccccn1)C(=O)NCC(C1CC1)N(C(=O)C(c1ccccc1)=O)C c1(C(N(C(CN(C(Cn2nc(C)c(Cl)c2C)=O)C)C)C)=O)c([N+](=O)[O-])cnn1C c1(CN2CCC(CC(=O)NC(c3ccc(Br)cn3)C)C2)ccc(Br)c(F)c1O C(=O)(C(O)CC(O)CO)N1CCC(C=C)(C(N2CCCCC2)=O)C1 c1(C(N2CC(NC(c3c(C(C)C)[nH]cc3)=O)C2)=O)ccn2ncccc12 CCCC(CCCNC(=O)Cc1csc(C)c1)NC(=O)CCC(=O)N(C)C CCCCCC(C)CC(=O)N(CCCNC(c1cc(S(N)(=O)=O)c[nH]1)=O)CC N1(C(N=c2ncc(C#N)c[nH]2)=O)CC2(CCCCC2)CC1CO CCCC(O)CC(=O)OC(c1cc(C)cc(Br)c1)C C(=O)(C(O)CCCNC(c1snnc1C)=O)N(C1CC1)CC c1(SC)cc(C(=O)NC2CCC2NC(c2nccn2C)=O)c(C)o1 N1(C(C2(C)CC2)=O)CC2CC(NC(=O)CCc3ncco3)CC2C1 c1(C(N2CCN(C(C3C(C)CCO3)=O)CC2CCO)=O)cnc2ccnn2c1 C(CCCCCC(=O)NCc1csnc1C)NC(C(CCCC)C)=O c1(C(C(=O)NCc2ccc(C)cc2O)C)cn(C)c2ccccc12 CC(CO)(CCF)NC(c1coc(CNC(C2CC(F)(F)C2)=O)n1)=O C12(C(=O)NC(C)CNC(C3CC(=O)N(C4CC4)C3)=O)CCCCN1CCC2 C1(CNC(CC(C)SC)=O)CN(C(c2ccc(OC(C)C)nn2)=O)CCN1C c1(C(C)=O)c(Cl)nc[nH]c1=NCC1CC1CNC(=O)C=CCO C1(C2CN(C(=O)CC3CCC(C)C3)C2)(NC(c2cc(OC)n[nH]2)=O)CC1 c1(C(N2CCC(C(N3CCC(C=C)C3)=O)C2)=O)cccn(C)c1=O c1(CC)cnccc1C(=O)NCC(CNC(=O)C(c1cccc(C)n1)(F)F)CO C1(CNC(C2CCCC2(F)F)=O)CC2(CCN(C(=O)Cc3nncs3)C2)CO1 c1(OCC)ccc2c(c1)CCC(c1nc(C3CC=CC3)nn1CCS(C)(=O)=O)C2 C(=O)(C(Cc1cccc(F)c1)CC(F)(F)F)OC(F)F.Cc1c2cnn1C(CC(=O)O)C2 c1(-c2cn(Cc3ccc(C)c(C)c3)nc2)cnc2cc(C(=O)NCC#N)ccn12 CCCCC(O)C(C)C(=O)N1CC(C2CCCN(C(C3(CC)CCCO3)=O)C2)C1 c1(C2C(C(=O)NCCC(C)N(C(=O)CN(C)CCO)C)C2)cccc(C#N)c1 Cc1cc(Br)nc(Cl)c1NCC1CC2(CC2)C1 C(CC(CNC(=O)C(CC(c1ccc(CSC)s1)=O)N(C)C)OC)OC(C)C.C(C)(C)OC C(C(CC1CCCC1)C(=O)NCCCC(F)(F)F)NC(C(C)OCCOC)=O C1(C(=O)NC2CN(C(c3cn(C)c(O)n3)=O)CC2(C)C)CN(CP(C)(C)=O)C1 Cc1ccc(C#N)c(N2CCOCC(CNC(C3(C)CC=CCC3)=O)C2)n1 C1(C(N(CCNC(C2CCN(C(=O)OC)CC2)=O)C)=O)CCc2n[nH]cc2C1 C1(NC(C(CCSC)O)=O)CN(C(=O)Cc2ccc(Cl)nc2C)C2(CCC2)C1 C1(CNC(C(CC#C)C)=O)(NC(=O)CCc2ccc(C)nc2)CC2CCC1CC2 c1(NC(=O)NCC2CCCC2c2ccccc2C(F)(F)F)ccc(O)c(Cl)c1 c1(C(C(=O)NC(CC)C)N(C(C(=O)OCC)C(C)C)C)cc(F)cc(N)c1N C1(NC(c2csc(C3CC3)n2)=O)(CO)CCN(C(=O)C=Cc2cscn2)C1 N1(C2CCN(C(CN(C(c3cn(CC=C)nn3)=O)C3CC3)=O)C2)CC(C)CC1=O CC1CN(C(c2nccn2C)=O)CC1NC(c1nccnc1N)=O Cn1c(Cl)nc2nc(Cl)nc(NCC34CC(NC(=O)CSC(F)(F)F)(CO3)C4)c12 c1(C(N2CC3CC(NC(c4c(C)onc4CO)=O)C3C2)=O)ncc([N+](=O)[O-])n1C C(C)(CC(C)(C)C)(c1n(CC=C)nnn1)NC(c1ccn(C)c1)C C(C1=CCN(C(C)C(=O)Nc2ccccc2)CC1)NC(C1CCC(CC)CC1)=O C1(C)(C(N2CC(COC)C2)=O)CN(C(=O)Cc2c[nH]nc2C)C(C)(C)C1 CCC(C)CCC(O)CC(=O)N1CC(C)(NC(c2cc3c(cn2)CCCC3)=O)C1 C(C(C)C(C)C(=O)N(C)CC=CC(=O)N(C(CCO)C(F)F)C)OC CCC(CCCC(=O)N1C(C(=O)OC)CC1C)NC(c1c(C)cnn1C)=O C(=O)(C1CCOc2ccccc21)NC1CC(NC(c2c(C)csc2)=O)C1 c1(C(N2CCC(N(C(c3cc(C4CCCNC4)no3)=O)CC)C2)=O)ccccn1 c1(OC)ccc(C(=O)NCC2COCC2NC(C2(F)CC2C)=O)cc1N N1(c2nc(C)c(Br)cn2)CC2CCC1CN2Cc1cc(Cl)cc(C)c1O C1(C(N(CC(=O)NCCCC(=C)Cl)C2CCC2)=O)CCCCCC1 N1(C(C(CC)SC)=O)CC(CNC(c2cocn2)=O)C(O)C1 Cc1nccc(C(N2CCC23CN(C(C2(n4cccn4)CC2)=O)C3)=O)c1C c1(CN2CCC(NC(C3N(C)CCOC3)=O)C(C)(C)C2)ccc2ccn(C)c2c1 N1(C(c2cc(C(CC)CC)no2)=O)CC2(CC(NC(c3ncc(Cl)s3)=O)CO2)C1 Cc1ccc(C)c(C(=O)NC2CN(C(=O)COCc3nnc(S)n3C)CC2O)n1 C1(C(=O)NCCN(C(c2ncncc2N)=O)CC)CCN(C(=O)OC)CC1 C#Cc1ccc(C(N2CC=CC(NC(C3(C)CCN(C)C3=O)=O)C2)=O)c(C)c1 CC1(NC(c2nc(Br)cnc2N)=O)CCCN(C(C2(F)CCCCC2)=O)C1 C(C(C)CN=c1ccn2c(Br)cnc2[nH]1)NC(c1cnc(CC)[nH]1)=O c1(OC)ccc(CC(O)C(=O)NCC2CC(NC(=O)Cc3cocn3)C2)cc1 c1(C(C)C)cc(C(=O)NCCNC(c2cc(C(F)(F)F)ccn2)=O)ccc1F C1(C(N(CCCN(C(CC(C(=C)C)OCC)=O)C)C)=O)CCCN(S(N)(=O)=O)C1 CCCCCCC(=O)NCCOC1CCN(C(=O)C(F)(F)c2ncccn2)C1 CCC(CCCC(=O)N=c1ccn(C2CC2)[nH]1)NC(=O)C(C)=CC(C)(C)C C(=O)(NNC(=O)COc1ccc(C)cc1)Nc1nc(CN(C)CC)on1 C1(C(=O)NCC(C2OCCCO2)(C)C)CN(C(=O)OC(C)(C)C)CC2(CCC2)O1 N1(C(c2[nH]nc(CC)n2)C(=O)NCC(C)C)CCCCC1COC(F)F CC(C)CC(O)C(C)C(=O)N1CCC(OCC(N2CCC(NC(N)=O)CC2)=O)C1 C1(CC(N2C(CC)CC(O)C2)=O)CCCN(C(C2(C)CCSCC2)=O)CC1 C1(F)(CNC(=O)CSC2CC2)CC(NC(=O)C(F)F)C1 C1(NC(C2C(=C)C2)=O)CCN(C(=O)Cc2csc(=N)[nH]2)C(C)C1 C(N=c1[nH]c(N2CCOC3CC23)nc2ccccc12)C1(OC)CCOCC1 C(CC(C(C)C)NC(c1ccc(OC(F)F)cn1)=O)NC(C1C(C)=C1)=O N1(C(c2c(=N)[nH][nH]c2)=O)CCC(NC(=O)CC2CC3CCC2O3)C(F)C1 c1(C(N(C)CCOCCNC(C2CC2F)=O)=O)cc(Cl)c(Cl)cn1 C(=O)(C1CCCn2cnnc21)N(C1CCCN1C(=O)C1=C(C)OCCS1)CC c1(C(=O)NC(C)CCNC(C2(CS(N)(=O)=O)COC2)=O)csc(C(F)(F)F)c1 C1(O)(C(=O)NC2CCN(CCC)CC2)CCN(C(C2CC3CCC2O3)=O)CC1 N1(C(CS(CC)(=O)=O)=O)CCC(C(=O)N(CC(O)C2CCC2)C)C(C)(C)C1 c1(CC)ccc(OC)cc1C(=O)NCC1CCCN(C(C2CC2F)=O)C1 N1(C(CC#N)=O)CCCCC1C1CCCN(C(C2(N3CCCCC3)CC2)=O)C1 c1(CCC)ccc(NC(C2CCOCC2)c2nnnn2C2CC2)cc1 c1(C(N2CCCC(N(C(c3cc(CC)no3)=O)C)C2)=O)cncc(P(C)(C)=O)c1 CC1(F)COCCN(C(=O)CCCCCNC(=O)C=CC2CCC2)C1 c1(C(=O)NC2C(NC(c3cc(C)ns3)=O)C2)ccnc(-n2cccn2)c1 C(CCCC)(C(=O)N1CCS(=O)C(C)C1)NC(CC=CC)=O c1(CC)oc(C(N2CCC2CNC(c2cc(C)c(C)o2)=O)=O)cc1C c1(C(=O)NCC2C(NC(c3n(C=C)ncc3)=O)C2)cn2nc(C)cc2[nH]c1=O C1(CNC(C(CC=CC)C)=O)CN(C(=O)CC2(O)CCOCC2)C2(CCC2)C1 C12(C(NOC(=O)Cc3ccns3)=O)COC(C1)C(NCCC(C)C)C2 Cc1nc(NCC(C)(C)OC(F)F)cc(NC(C)C(N2CCCCCC2)C)n1 S(=O)(=O)(c1ccc(Cl)cc1)NCCC(N1CC(C)CC(CC2(CC)CC2)C1)=O C1(CNC(C2(CC)COC2)=O)CN(C)CCN1C(c1ccc(Cl)c(C)c1)=O N1(C(CSCCCC)=O)CC2(CCOCC2C(N2CCSCC2)=O)C1 C12(C(=O)NCCCN(C(c3c(C)nn(C)n3)=O)C)CCCCN1CCC2 c1(CC2N(C(=O)NCC3C(C)C3C)CCC2)cccc2ccccc12 c1(C(N2CC(C)(NC(=O)CCCc3nccs3)C2)=O)cccc(C2CC2)n1 c1(C(N2CCC(n3cc(CNC4CCC4)nn3)C2)=O)cc2cccn2c(O)n1 CC1CCC=C1C(=O)NCC1C(C(=O)NCC2CCN(C)C2)C1(C)C c1(C(=O)NC(CC2CN(C(C(C(=O)OCC)CC)=O)C2)C)cc(Br)cnc1O C1(N(C(C(C)Cc2ccccc2)=O)C)CCCN(C(=O)CS(=O)(=O)N(C)C)CC1 CC(C(C)(C)NC(=O)COCC(F)F)NC(=O)COC1CCCOC1 C(=O)(C(=O)NC1(C(=O)NCCOCCN(C)C)CC1)NCC c1(CN2C(C(=O)Nc3nc(Cl)cs3)CCC2)cc(F)c(F)cc1Cl c1(CNC(CCCC)=O)cccc(C(=O)NCCCN2CC=CC2)n1 Cc1cccc(C(N2CC(CNC(=O)Cc3cn(C4CC4)cn3)CC2C)=O)c1Cl CCCCC(O)C(C)C(=O)NCC(C)CN(C)C(c1cc(OC)n[nH]1)=O CC(C)CC(C)CC(=O)NCC1(F)CC(NC(c2cc(F)c(Cl)cc2Cl)=O)C1 C1(C#N)(C(=O)NC2C(CNC(C3C(=C)CC3)=O)CCC2)CCc2ccccc2C1 C1(NC(C=NOC)=O)CC2(CCN(C(=O)C(C)NC=O)CC2)C1 c1(C(N2CC(CCNC(Cc3c(C)ocn3)=O)OCC2)=O)c(N)ccc(F)c1F C(=O)(CC(CNC(C)(C)C)C1CCC1)NCC(C)NC(=O)CC1CCCO1 c1ccc2c(c1)CCC(CSC1CCC3(CC1)COC3)C2 N1(C(C=C(C)Cl)=O)CCCCC1C1CCCN1CC.C(CO)NC(C)=O N1(C(C2CCC(C)C2)=O)CC2CC(C1)CN(C(=O)CSCCN(C)C)C2 n1(CC)cc2ccc(C(=O)NC3CN(C(=O)CC(C)NC(N)=O)CC3C)cc2n1 C1(CN(C)C(C2(N3CCOCC3)CC2)=O)CCN(C(=O)CC#N)C12CC2 C12(NC(C3N(S(CC)(=O)=O)CC3)=O)CCCC1(F)CN(C(=O)C(F)(F)C1CC1)C2 c1(NC(=O)NC)n[nH]c2c1C(C(F)(F)F)CC2.C(=O)(C(=O)NC1(NC(C)=O)CC1)NC C1(C(=O)NCCN(C(c2ccc(Br)o2)=O)CC2CC2)CCC2CCC(=O)N12 c1(CC(=O)NC23CC(C2)N(C(=O)CN2CSCCSC2)C3)ccc(Br)cc1F C=CCC(C(=O)NC(CCOCCO)C(=O)NC1CCC1C(=O)NC)OC C1(CNC(c2ccc(-c3cn[nH]c3)cc2)=O)COCCN1C(c1csc(Cl)n1)=O C1(C(C)NC(c2cc(CNC(C=CC=CC)=O)on2)=O)CC2(CCC2)C1 c1(CCC)onc(C)c1C(N1CSCC1C(=O)NCCc1ncc(C)o1)=O C1(N(C2CC(n3cc(COC(=N)O)nn3)C2)C)CCCC(=O)C1 C1(NC(CC=CCC)=O)CCN(C(C2CCOC2CC)=O)C1C1CC1 Cc1nn(-c2ccccc2)nc1C(=O)NC(C1CCCN1C(=O)C(C)O)(C)C c1(C(=O)NC2C=CCN(C(c3ccc(C(C)=O)[nH]3)=O)C2)cc2c([nH]1)CCCC2 C1(NC(C2(F)CCN(C(=O)C(F)F)CC2)=O)CCS(=O)(=O)CC1 C1(C(N2CC(N(C)C(C3C4C5CCC(C5)C34)=O)C2)=O)CCc2ccc(F)cc2O1 C1(C(N(CCCNC(c2[nH]cc(C(C)=O)c2)=O)C)=O)CC2(C1)CC21CCC1 N1(C(C2(C)ON=C(C)C2)=O)C2CCC1CC(NC(C1(N(C)C)CCCCC1)=O)C2 C(N=c1nc(O)c2cnn(C(C)(C)C)c2[nH]1)C1CCN(C(CCP(C)(C)=O)=O)C1 N1(C(C(c2cncc(F)c2)C)=O)CCCC(C)(NC(C2CC(C(C)C)=NO2)=O)C1 C(=O)(CC1CC(=O)c2ccccc21)NCC1(F)CC(NC(CCC=C(C)C)=O)C1 c1(NC(CCN(C(CC2ON=C(CC)C2)=O)C(C)C)=O)cc(C)c(O)c(C)c1 Cc1cc(C(=O)NCC2CN(C(=O)CC3CCOC(C)(C)C3)CCN2C)cc(O)c1 C12(NC(CN(C)S(N)(=O)=O)=O)CCOC(CNC(c3cccc(F)c3)=O)(C1)C2 c1(C(=O)NCC(CCNC(C2C(OC)CC2)=O)O)cc2c(s1)CCS(=O)(=O)C2 N1(C(CC2C(NC(C3N(CC)CC3)=O)CCCC2)=O)CCc2nocc2C1 Cc1ccc(F)c(C(N2CC3CC3(NC(=O)CCCn3c(C)csc3=O)C2)=O)c1 N1(C(=O)CC2CCN(Cc3cscn3)C2)CCN(CCCO)CC1 N1(C(C(c2ccc(CC)s2)=O)=O)CC2CCC1C2NC(=O)C=CC=C(C)C C1(O)(CN(C(C(C)OCc2ccccc2)=O)C)CCCN(C(=O)CSC2CC2)C1 N1(C(CC(=O)OCC)=O)CC2C(C(=O)N(C)CC3(CO)CC3)C2C1 C1(NCc2ccc(NC(C3CC(=C4CC4)C3)=O)o2)CC(C(=O)O)C12CCOCC2.[SH2](C)CC1CC1 c1(C(N(C2CCN(C(c3n(CC)ncn3)=O)C2)C)=O)cc(F)c(F)c(F)c1N Cc1ccc(Br)c(C(N2CCN(Cc3cccc(O)c3O)CC2CO)=O)c1F c1(C(N2CCCCC(CNC(C3C(C)(C)OCC3)=O)C2)=O)cnn2ncccc12 c1(NC)nc(C(=O)OC2CC(C(=O)OC(C)(C)C)C2)ccc1[N+](=O)[O-] CCCC(C)(C)C(=O)NC1C2CC(NC(C3CCCN3C(C)C)=O)CC12 c1(-c2ccc(COC)s2)nccnc1N(CCC(C)C)CCN(C)C CC1CN(C(=O)CN2C(=O)CN(C)C2=O)CCC1NC(c1cc(F)ccc1Cl)=O C(=O)(C(F)C(F)(F)F)NCC(CNC(C1C2CCC12)=O)O C(=O)(C1=C(C)CCCC1(C)C)N1CCC(N(C)Cc2ccc(C#C)s2)CC1 CC(CNC(=O)C(N1CCOCC1)=O)CN=c1[nH]n(Cc2ccccc2)cc1Br CCC(=O)CCC(=O)N(C(C(=O)NC1CCC2CCC12)C1CC1)C O=C1CC(C2CCCN(C(=O)NCCC3COC3)C2)C(=O)N1c1cccc(Cl)c1 C#Cc1cn(C)nc1C(=O)NCC1CN(C)CCN1C(=O)C(C)CC=CC c1(N(C(c2nc(C(F)(F)F)no2)C(=O)NCCCCCC)C)c(I)cnn1C N1(C(C(CCCOC)C)=O)CC2CC(O)C1C2NC(=O)CCc1ccc(C)nc1 c1(CC)c[nH]c(C(=O)NC2CC(NC(=O)Cn3cc(C4CC4)cn3)C2)c1 C#CCC(C)(C(=O)NC(C)(CC)CCC)NC(=O)C(N1CCNC1=O)C Cc1cc(C(=O)NC2CN(C(=O)Cn3nccn3)CCC2F)nc2ccccc12 C1(N(C(C(C2CCCCC2)C)=O)C)CCC(NC(C2CC2F)=O)CC1 c1(NC(C2COCCN2C(=O)CCC(O)C(F)(F)F)=O)cccc(CF)c1 C1(CC2CCC2)C(=O)N1.C1(CC(=O)OCC)(CC=CC=C)CCC1 C(=O)(CC(O)CNC(C1(CCF)CCC1)=O)N1CC(CCOC)C1 C(=O)(CCC(=O)C(C)(C)C)N(CCC(=O)N1CCCC1)CC1C(C)(CC)C1 N1(C(C2C=CCC2)=O)CCCCC(CNC(C2(Cc3ccccc3)CC2)=O)C1 C(=O)(N=c1[nH][nH]c(C)c1C)C1CCN(C(c2cc(OC)c(Br)cn2)=O)C1 C12(NC(c3n(CC)ncc3Cl)=O)CCC(CC1NC(c1cn(C3CC3)cn1)=O)C2 c1(NC(=O)CC2(NCc3cccc(Cl)c3Br)CCC2)ncc(Cl)cc1I C1(C2CC2)(CNC(C(CC=C)N(C)C)=O)CCN(C(=O)CCC2CCCCC2)C1 n1(CC)ncc(Cl)c1C(=O)NC(CN(C(=O)C(F)CC1CCOC1)C)CC C#Cc1cnc(C(N2CC(C(O)C(=O)N(C)Cc3sccc3C)C2)=O)c(C)c1 C=CCC(CC(=O)NC(C)CNC(C)(C)C)NC(=O)C(CCCC)N(C)C CC1OCCN(C(=O)C(C)Cn2ccnc2)C1C(=O)NCCCC(C)(F)F N1(C(CCSCC(=O)OC)=O)CCCC(CO)(CNC(=O)Cc2cccs2)C1 CS(=O)c1ccc(CC(N2CCCC(CCNC(=O)Cn3ccnn3)C2)=O)cc1 C1(C(N2CCC(C)(NC(c3ccc(COC)o3)=O)C2)=O)CC2CCC1CC2(F)F N1(C(C(c2cncnc2)C)=O)CCC2CN(C(=O)CCOC3CC3)CC2C1 C1(N(C(C2C(CNC(C3C(C(C)C)OCC3)=O)CCC2)=O)C)CC2CCC1CC2 C12CCCCN1S(=O)(=O)CCc1c[nH]nc12.c1(C(C)C)ccccc1C(F)(F)F N1(c2c(F)cnc(OC)n2)CCC2(CC(C(=O)NC(c3ccsc3)C)=NO2)C1 c1(C(=O)NCCC(C)NC(c2c(C)cno2)=O)cnc2c(C)cccn12 c1(C(N2C(CNC(C3CCCN(C)C3)=O)CCC2)=O)cccc2c1C(C#N)C2 CC(C)(C)CC(O)CC(=O)NC1CC2(C1)CC2C(=O)NC1C2CCCC12 C(C(=O)NC1CSC1)(C(C)C)NC(c1c(COC)noc1)=O CN(C)S(=O)(=O)N1CCN(c2nc(N3CCCC(F)C3)c3ncccc3n2)CC1 CCC(C)(CCNC(c1ccc(C(F)F)cc1)=O)NC(=O)CC1COCC(C)O1 C1(C(C)C)CCCN(C(=O)C(CCC2CCC2)NC(=O)CC2CC(F)(F)C2)C1 c1(NC(C(CC(=C)Cl)NC(C2CCCN(CC)C2)=O)=O)cc(C)c(F)cc1O C1(=CC(=O)NCCO)CCN(C(=O)Cc2cnns2)CC1.O=C(CNC(=O)C1CC1)N c1(C(N(CC(=O)NC(CC#C)C(N)=O)CCOC)=O)[nH]ccc(=O)c1C c1(C(=O)NCC2CN(C(CCS(C)=O)=O)CC23CC3)cc2c(nc1O)CCOC2 CCCCCCOC(C)C(=O)NCC1(F)CC(NC(=O)CC(C)SC)C1 c1(CC)cc(S(N)(=O)=O)co1.c12ccc(cc1)N(C)CC1N(C(=O)C2CC)CC1 C1(NC(C(CC)CC)=O)C2CC3CN(C(=O)Cn4ncc(Cl)c4C)C1C3C2 Cc1cn2c(n1)CCC(C(=O)NCCNC(=O)Cn1c(O)nc3ccccc13)C2 c1(C(=O)NCC2CN(C(c3cn(C)nc3O)=O)C2)ccc(Cl)c2cccnc12 c1(C(N2CC(O)(CCNC(C3CCCCC3O)=O)C2)=O)ccc2ncncc2c1 C1(CNC(=O)CCc2cnc[nH]2)CC(F)CCN1C(=O)CC1CCCOCC1 CCCC(C)(C)C(=O)NCCC1CC(NC(=O)CCC2CCC(C)O2)C1 C1(CNC(C2CC(C)N2C(=O)CN2CCOCC2)=O)CC2C=CC1O2 CC(C)C(C(=O)NCc1nc(=O)o[nH]1)C(C)NC(c1ncc(F)cn1)=O C1(O)(CNC(CC(C)N(C)C)=O)CC2CCC(C1)N2C(C1(c2cccs2)CC1)=O N1(C(C(C)=C(C)C)=O)CCC(C)C1c1cn(Cc2occc2C)nn1 Cc1ccc([N+](=O)[O-])c(C(N2CCCC(NC(=O)CCC=CBr)C2)=O)c1 N1(C(C(n2nnnc2C2CC2)C)=O)CCN(C(c2coc(Cl)c2)=O)C2CCCC12 C=CCN=C(NCC(O)CF)NCC(C)(C1CCC1)N(CCO)C(=O)OC(C)(C)C c1(CC(N2CC3CN(c4ncnc5[nH]ccc45)CC3C2)C)cc(Cl)cc(C#N)c1 C=CCCCC(=O)N1CC(O)(C(F)C(=O)NC(CCC)C(=O)N(C)C)C1 S(=O)(=O)(c1cnc(N2CCCC(CS(N)(=O)=O)C2)c(Cl)c1)N(CC(CCC)C)C N#Cc1ccc(OC(c2cnc(NC3CCCC3)c(Cl)c2)=O)cc1 N1(C(C2CN(C)C(=O)C2)=O)CCCC(CO)(NC(=O)CCc2ccc(F)cc2)C1 C12(C(CNC(=O)CCSC)NC(c3cnn(CC)n3)=O)CCC(CC1)C2 C1(C(=O)NCC2(CNC(=O)COCC3CC3)CC2(F)F)COCC2(CCC2)O1 Cc1cccc(C(=O)NCC2(CNC(C3CCCCC3C(=O)N(C)C)=O)CC2)c1 Cc1c(C(=O)NC2CCc3cn(C)nc3C2)cc(Br)cc1[N+](=O)[O-] C1(CNC(C(C)C(F)F)=O)CC12CCN(C(C1(c3ncco3)CCC1)=O)CC2 c1(C(=O)NC(CC)CNC(c2[nH]c(O)nc2C)=O)c(O)cc(=O)n2c1COCC2 c1(N2CC=CC2)nc2c(c(=NCCN3CCCCC3)[nH]1)COC2 C(C(C)(C)C(=O)NC1CN(C(c2cc(Br)oc2C)=O)CC1C)OC N1(C(COC2C(C)CCCC2)=O)CC2(CC2)CC1CNC(=O)CCNS(C)(=O)=O CCC(CNC(c1cc(C2CCOC2)[nH]n1)=O)(CC)NC(C1CC(F)C1)=O C1(C(=O)NCCN(C(C)C)C(c2ccc3nn[nH]c3c2)=O)OCCOC12CCC2 c1(C(=O)NCC(CN(C(=O)C=CC2CCOC2)C)O)cc(-c2ccncc2)no1 N1(C(C(CC)(C)O)=O)CC(NC(c2cc(C(F)(F)F)nc(C)c2)=O)C(C2CC2)C1 C1(NC(=O)CNC(N2CCCC2)=O)CN(C(C2CC3COCC3C2)=O)CC1(C)C.C C1(NC(C2CCC(C)(C)C2)=O)CCC12CCN(C(=O)C(C)(C)c1cc[nH]n1)CC2 c1(C(C)C(=O)NCC2CCC2NC(=O)C(C)SC(F)(F)F)ccc(Cl)s1 CC1CCN(C(C2CCOC(C)C2)=O)C(C)C1NC(c1nccc2occc12)=O c1(C(=O)NCC(CCNC(c2c(C(C)C)cnn2C)=O)O)cc(F)c(F)cc1Cl c1(CC)nc(C(=O)NC(C)CC(C)NC(=O)Cn2cc(Br)cn2)c(C)o1 C(=O)(C1=NN(C2CC2)C(=O)CC1)N1C2C(NC(C3(C)C(C)CCC3)=O)C(C2)C1 N1(OC(=O)CN=[N+]=[N-])CCCC(C(=O)Oc2c(C)nn(-c3ccc(Br)cc3)c2)C1=O N1(C(CCc2cc(C)no2)=O)CCC2(CC(C(N3Cc4cncnc4C3)=O)C2)C1 CN1CC2(CC2)CC1C(=O)NCC(C)(C)CC1CN(C(C2CCCO2)=O)C1 C(=O)(C#CC1CCCOC1)NCC12N(C(c3c(N(C)C)ccnc3)=O)CC(C1)C2 C1(C(N(C)CC=CC(=O)N(C2CC2(C)C)C)=O)OCCCC1(C)C C12(C(=O)NCCc3c(C)ocn3)CCCC1CCN2C(C1CCNC1=O)=O C1(O)(C(C)NC(=O)COCCCF)CCN(C(=O)CC(C)(C)c2cccs2)C1 C1(NC(CC2C(OCC)CC2)=O)CCOC(CC)C1.C(CCSCC)NC=O C=Cc1cc(C(=O)NCC2CC2CNC(c2c(C#N)cnn2C)=O)cc(F)c1 N1(CC)CCC(S(N)(=O)=O)C1.c1(C2c3n(nnn3)CCCN2)cccc(OC)c1 CC(C)(C)C(CO)C(=O)NC1CCC(NC(C2OCCCO2)=O)CC1 N1(C(C2N(CC#C)CCC2)=O)CCCOC(CNC(C2(O)COC2)=O)C1 N#Cc1cccc(NC(C2CCCCC2(C)NC(C2CC(=O)CC(=O)N2)=O)=O)c1 C1(NC(c2c(N)nc(Cl)cc2)=O)CCN(C(c2ns[nH]c2=O)=O)CCC1CO Cc1ccc2ncc(C(=O)NC3C4CCN(C(=O)CC(C)C(C)C)C34)cc2c1 c1(NC(CCCOC)=O)cc(=O)c(O)c[nH]1.C1(=O)NCCN1 CCCCCCC(=O)N1CC(CC(C)C2(NC(=O)C(C)Cn3ccc(C)n3)CC2)C1 Cc1cnccc1C=CC(N1CCC(C(C)NC(=O)CC(C)C2CC2)C1)=O Cc1nnc(CCNC(C2(NC(=O)C(F)C3CCC3)CC(F)C2)=O)n1C c1(C(=O)NCC(C(=O)NCC(C(=O)OC)OC)C)ccc(O)nc1 c1(OCC)cc(-c2nc(NCc3ccccn3)cs2)cc(F)c1F C1(O)(CNC(CC2CN(C)C2)=O)CCCN(C(=O)Cc2cccc(F)c2F)CC1 c1(CNC(=O)CCCc2cnn[nH]2)cccc(NC(=O)CCc2ccon2)c1 N1(C(c2nccc(N(CCCC)C)c2)=O)CCC12CCNCC2 N1(C(C=Cc2cccc(N)c2)=O)CC(C2CN(C(C3CC34CCCOC4)=O)C2)C1 C1(OC)CCCN(C(=O)C(c2ccnn2C)NC(C2C3CCC(F)C23)=O)C1 C1(CNC(CCSCC)=O)COCCN(C(C2CC2C(C)O)=O)C1 C1(CNC(C)=O)CC2(CCN(C(=O)C(O)C3CCCC3)CC2)C1 N1(C(c2c(COC)nn(C)c2Cl)=O)CCC2CN(C(=O)C=CSC)C2C1 CP(C)(=O)CN1CC(C(N2CCOC(CCNC(=O)CCF)C2)=O)C1 c1(NC(C2CCCCN2Cc2ccncc2Cl)=O)ncc(Br)c(O)n1 c1(C(=O)NCC(C)(C2CC2)NC(C(F)=C(C)C)=O)ccc2nn[nH]c2c1O N1(C(C)=O)CCC(C(=O)N(C)CCNC(C2(C(C)(C)C)CCC2)=O)C1 C1(C(=O)NC2C(NC(C3CCC3)=O)CC2)CN2CCCC1C2 C12(CNC(Cc3c(SCC)cccc3)=O)CCCC(CN1C(=O)C(N)=O)C2 C(=O)(C1CCc2ccccc21)N1C(C(=O)NCC(C(=O)OC)C)CNC(=O)C1 C1(O)(CCNC(c2c(C)ncs2)=O)CCN(C(c2cccc(C)n2)=O)C1 C1(COC(C2C(C)(c3cccs3)C2)=O)CC(c2cccc(Cl)c2)CCC1=O C1(C)(C(N(CCN(C(COCCCC#C)=O)C(C)C)C)=O)CCCNS1(=O)=O C1(C(N2CCC(CCNC(C3(OC)CCC3)=O)CC2)=O)CCc2ccccc2O1 c1(C(=O)NC2C(C)N(C(=O)CC(C)(C)C)CC2)ccc(S(=O)(=O)CF)cc1 N1(C(C2N(C(CCC(C)SC)=O)CC2)=O)CCOCC2(CCC2)C1 C1(C)(CC)CCCN(C(=O)CC2CC3(C2)CN(C(C2CC2(C)C)=O)C3)C1 C(CNC(C1CC2C=CC1C2)=O)(CC(F)(F)F)NC(c1ccc(Cl)cc1F)=O Cc1ccc(C(=O)NCCCC(C)NC(c2n[nH]cc2[N+](=O)[O-])=O)c(F)c1 c1(CCNC2CCN(C(=O)NC(c3ccccc3)C)C2)cccc(Br)c1Cl c1(CC(=O)NCC2(NC(C3CNCC3(F)F)=O)CCOCC2)cc(F)ccc1Br CC1(O)CCC(C(=O)NCCCCCCNC(c2ncoc2C2CC2)=O)CC1 N1(C(Cn2nc(C)oc2=O)=O)CCOCC(NC(C2(CS(C)(=O)=O)COC2)=O)C1 c1(CC2(C)CCN2C(=O)CCNc2cncc(C(C)C)c2)ccc(F)cc1F C(=O)(CS(=O)(=O)CC1CCCO1)NCCCN(C(C)C)C(C1COCCN1C)=O Cc1c(C(=O)N(C)CC2CCCN2C(c2cnc(C3CCC3)o2)=O)cccc1F c1(CC(=O)NC2CN(Cc3c(F)cccc3I)C2)cc(Br)ccc1F N1(C(C2C(CC)CCC2)=O)CCCN(C(c2ccc(=O)n(CCO)c2)=O)C(C)C1 c1(OC)ccc(C(=O)NCC(C(C)C)NC(=O)C(C)C(C)O)c(Br)c1 C(CC(=O)NCc1csnc1C)(C(C)C)NC(C1(CCOC)CCC1)=O c1(C(c2nnnn2C)NC(CCC)C2CCCC2)cc(I)n(C)n1 c1(C(=O)NCC(CC(C)C)NC(C2CC2C)=O)cccc2nonc12 n1(CC(=O)NCC(C)(C)CNC(=O)C(F)CC2CCOC2)ccc([N+](=O)[O-])n1 N1(C(C2(C#N)CC2C(F)(F)F)=O)CCN(C(=O)C=Cc2ccco2)CC(CO)C1 c1(CNC(C(=O)N(CC(C)CO)C)=O)ccc(-c2ccnn2C)cc1 CC(C)C(C(c1nnnn1C1CCC1)NC(c1ccn(C)n1)(C)C)C(C)C Cc1ccc(O)c(CC(=O)NC2CC(CCNC(C3(C)COC(C)CO3)=O)C2)c1 C(=O)(CC(=O)N(C)C)N1CC(CC(F)C(=O)N2CC(O)(C(F)(F)F)C2)C1.CNC Cc1sc(C)c(C(=O)NC2CCCCC2NC(c2c[nH]c(C(N)=O)c2)=O)c1C c1(NC(c2ccc(Cn3cc(COCC(N)=O)nn3)cc2)=O)cc(O)nc(O)n1 C1(CCNC(C2CN(C)C2)=O)(OC)CN(C(C2CCC(C(C)C)O2)=O)C1 Cc1ccc(SCC(=O)NCC(C2CC2)NC(=O)CN(C)C2CC2)cc1 C(=O)(C(CC(C)C)C(N)=O)N1CC(CC(C(=O)NC(CCC(C)C)C)F)C1 c1(CC(=O)NC2C(NC(Cc3ccc(CC)cc3)=O)COC2)ccc(Cl)c(C)c1 C1(C(CNC(c2nc(C(C)OC)oc2)=O)F)CCN(C(C2CS(=O)C2)=O)CC1 N1(C(CN(C)CC)=O)CC(N(C)C(c2nc(C)[nH]c2C(F)(F)F)=O)C(C)(C)C1 C(=O)(C(C)CC(F)(F)F)NC(CN(C(c1cnn(C(C)C)c1N)=O)CC)C c1(CC(=O)NCC(CC(=O)NCc2cnc[nH]2)C2CCC2)coc2ccccc12 C1(C(N(CCN(C(c2c(OC)ccnc2)=O)C)C)=O)CCCC2CCCCC12 N1(C(C2(C)CCCS2)=O)CC2(C(=O)NC3(CO)CCC3)CCC1CC2 C=C(C)CCC(=O)NCC(F)CNC(=O)C(C)NC(=O)C(C)(C)C c1(C(C)C)cncc(C(=O)NCC2CN(C(=O)C(N3CCSCC3)C)CC2C)c1 C(C)(C(O)C(=O)NCC1(CNC(c2cccc(-c3nccs3)c2)=O)CC1)OC c1(C(=O)NCC(CC=C)NC(C2(C(C)(F)F)CC2)=O)cnc2[nH]cc(C)c2c1 C(c1ccc(Br)cc1Cl)=CC(C(=O)NC)N1CCNCC1 c1(C(N2C3CN(C(=O)CC(F)F)C(CC3)C2)=O)nc2c(F)cc(Cl)cc2s1 CC1(C)C(NC(=O)CNC(N)=O)C(C)(C)C1NC(=O)CCN1CCCCC1=O C(=O)(C1=CC2CCCC12)N(CC)CC1CCN(C(c2cncnc2)=O)CC1 c1(C(=O)NC(CCCNC(C(C)=C2CCCC2)=O)C)c(Cl)ccc(F)c1F CC1(C)CCC(C)(NC(C2CCC2NC(c2cnnc(O)c2)=O)=O)C1 Cc1ccc(C(C(=O)NCC2(F)CCN(C(c3ccncc3Cl)=O)C2)C2CC2)cc1 C1(C(=O)NCCNC(N(C)C)=O)C2CC3C(C2NC(C2CC4C=CC2O4)=O)C13 Cc1ccc(C(N2CCCC(NC(=O)COC3CC3(F)F)CC2)=O)cc1[N+](=O)[O-] C1(C(=O)NC2C(CNC(c3sncc3Br)=O)C2)CCNC1=O C1(C)(COC)CC(NC(=O)C=C(C)C(F)F)CN1C(c1ccnc(C2CC2)n1)=O c1(C(=O)NC(CN(C)C(c2ccc[nH]2)=O)(C)C)ccn2nccc2c1 c1(C(N2CC(C#N)OCC2)=O)cc2cccc(-c3cncc(OCF)n3)c2s1 c1(Cn2cc(CCCSCC)nn2)ccc(C(=O)NCc2cccnc2)cn1 N1(CC(=O)Nc2c(NC(=O)NCC)coc2)CCn2ncc(C(=O)N(C)C)c2C1 C(=O)(C1COc2ccccc21)N1CC(NC(Cc2n(C)cnc2)=O)C(O)C1 C12(C(=O)NC3CCN(C(C4CCC(C)C4)=O)C3)CC(C1)S(=O)(=O)C2 C1(C(=O)NC(C)CNC(=O)COC2CCC2)COC(C)(C)CO1 CC1OCCC1(C)C(N1CC(NC(c2ccncc2F)=O)C(O)C1)=O N1(C(C=C(C)C(F)F)=O)CCC2(C=C(C(=O)NC3(C)CS(=O)(=O)C3)C2)C1 C1(C(N2CC(C(C)NC(c3ncoc3C3CC3)=O)OCC2)=O)CC(=O)NC1(C)C N1(C(C2CC(N(C)CC)C2)=O)CCCN(C(c2ccc(C)c(Cl)c2)=O)CC1 CC1(C)CC2(CC2C(=O)NCC2CC2CNC(=O)COCCF)C1 c1(CN(c2ccccc2)C(=O)NCC(CC)C#N)cccc(C)c1C C(=O)(C1=C2CCCN=C2NN1)N1CC(CNC(CCCCC)=O)C2(C1)CCC2 c1(CC)nnc(N2CC(CNC(=O)CCc3ccc(Cl)s3)CC2C)nc1CC CC1(C)COC2(CC3(CC2)COO3)C1.c1(CCNCc2ccn(C(F)F)n2)ccccc1 Cc1cccc(CC(N2CC(C)CC2C(=O)NC2CC2(F)F)=O)n1 C(=O)(C(O)CCCNC(C1COCCO1)=O)N1C(C)(CCO)CC1 C(CCCCCC(=O)NC(C)(CNC(c1c(O)cccc1F)=O)C(C)C)SC N1(C(c2ccc(CNC(=O)CCc3ccc(Cl)cc3)cc2)=O)CCn2nccc21 C1(C)(C(=O)NCC(N2CCCC2)C)CN(C(C23CSCC2C3)=O)C(C)(C)C1 Cc1cc(C(=O)NCCC(C)NC(C2CCC(=O)NC2)=O)cc(C)c1C#N N1(C(C2C(C=C)C2)=O)CC(CO)(NC(C2CC(N3CCCC3)C2)=O)C1 C(c1cc(C)cc(C)c1)=CC(N1CCC(C)(NC(C=C(COC)C)=O)C1)=O C(C1=CCCCC1)(n1c(-c2ccc(O)cc2)ccn1)Nc1cccc(C(N)=O)c1 N1(C(CSC(C)(C)C)=O)CC2(CCC(C(=O)NCc3ncc[nH]3)O2)C1 C12(NC(c3cc(C(F)(F)F)n[nH]3)=O)CCCC1N(C(=O)C=Cc1ccsc1)CC2 C1(CNC(c2cccnc2C2CC2)=O)C2CN(C(=O)Cc3csc(Br)c3)CC12 N1(NC(C(C)CN)=O)CCC(O)(CCn2cc(C3(O)CCOC3)nn2)CC1 C1(NC(C2CCC(CC)O2)=O)CN(C(C2(CC)CC2)=O)CC2(CCC2)C1 c1(N(C)C)ccc2[nH]c(C(=O)NCC3(O)CCN(C(C4CC4F)=O)CC3)cc2n1 N1(C(COC(C)C)=O)CC(NC(=O)CC(O)CN(C)C)C2CCCC2C1 c1(C(N2C(CC)CN(C(=O)C(C)(F)CC)CC2)=O)ccc(P(C)(C)=O)nc1 N1(C(C2(C)C(CC)CCC2)=O)CCCN(C(c2ccn(C)c2C)=O)CCC1 N1(C(C)C)CCCC(CC(=O)NC(C)CCNC(c2c[nH]cc2C(C)(C)C)=O)C1 C(=O)(CCC(C)(C)C)N1CC(CC(C(=O)NC(C)CC2CC2)F)C1 c1(C(=O)Nc2ccc(Cl)cc2OC)c(N2CCN(C)C(CC)C2)nc(=N)[nH]c1C C#CC1CC2CCC1N(C(=O)CC1CC(C)N(C(=O)C3=NOCC3)C1)C2 S(=O)(=O)(c1ccc(OC(F)F)cc1)N(C(C1CNCCO1)C(=O)NCCC)C Cc1csc(C(=O)N(CC(O)CN(C)C(C2CC2(F)F)=O)C)c1Cl N1(C(C=C)=O)CC(C)CN(C(=O)C=CCCC)C(C)C1.CCCCCC=CC(=O)N C1(C2CCOCC2)(CNC(CC=CC)=O)CCN(C(c2cc(OC)n[nH]2)=O)C1 N1(C(CNC(CCC)=O)=O)CC(NC(=O)Cc2nncn2C)CC2(CC2)C1 c1(C(=O)NC(C(C)NC(CCC=C)=O)C(C)C)ccc(F)c(Cl)c1F C(=O)(CS(=O)(=O)CCC(F)(F)F)NC1C(CNC(c2cc(C)n(C)n2)=O)CCC1 CC1(C)CN(C(C2CCC(=O)NC2)=O)CC1C(=O)NC1CCCC1N=[N+]=[N-] n1(CC)ccc(CC(=O)NC(C2CCCC2CNc2cc(C3CC3)on2)=O)n1 C(C)(CNC(C12CCC(CC1)CO2)=O)(CC(C)C)NC(c1cn(CC)nc1)=O c1(C(N2CCC(NC(C3(OC)CCOCC3)=O)CC2)=O)sc2cccnc2c1Cl C1(CNC(c2cnc3sccn23)=O)CCCN(C(=O)CN2CC=CC2)CC1 CN1CC=C(CC(=O)NCC2CCN(C(c3ccc(O)nc3)=O)C23CCC3)CC1 c1(C(=O)NCC(C)NC(c2nc(OCC)sn2)=O)cnc2ccc(F)cc2c1 C#CC1(C(=O)NOCc2ccccc2F)CCN(C(c2cccc(C)c2)=O)C1 c1(OC)cc(Cl)c(C)cc1C(=O)NC1CC12CCN(C(c1nonc1N)=O)CC2 C1(N(C(=O)COCC2(C)CCCC2)C)NCCC1(C)C c1(C(=O)NC2CCCC(CNC(CCCC=C)=O)C2)cc2c(=O)[nH]ccn2n1 Cc1ccn(C)c1C(=O)NCCCOCCCNC(=O)C(C)n1cccn1 CC(C)S(=O)(=O)CC(=O)N(C)CC1CN(C(c2cnnn2C)=O)CC12CC2 Cc1cccc(OC(C)C(=O)N(C2CC(NC(=O)C(F)(F)CC3CC3)C2)C)c1 N1(c2snc(C)n2)CCCC(CO)(NC(C2CN3CCC2CC3)=O)C1 c1(C(=O)NCCCC2CCCCN2C(=O)CC2CC(F)C2)ccc2occc2n1 N1(C(C(c2cncnc2)C)=O)CC=CC1C(=O)N(C)Cc1cn(C)nn1 c1(CNC(c2nc[nH]c2C(=O)O)=O)csc(=NCc2cc(Br)co2)[nH]1 C1(CCN(C)C)C(=O)NCCC(=O)N1.C(=O)CCCCC1CC1 C1(C(N2CCC(CC)(CC)C2)=O)CC2CC1CC2NC(=O)Cc1cccnc1F C1(C(N2CC(O)(CN(C)C(C3(CC4CCC4)CC3)=O)C2)=O)(CC)CNC(=O)C1 c1(CC(=O)N(CC(=O)NCC(c2ccnn2C)C)CC)ccc(C)c(F)c1 c1(CCC(=O)N(C(CN(C(CSC)=O)C)C)C)ccc2cccnc2c1 C1(C(N2CC(CNC(C3CCN(CC)C3)=O)(COC)C2)=O)CCC(C)(C)CC1 c1(C(=O)NCCC2N(C(Cc3cc(C)sc3)=O)CCSC2)c(Br)c(C)nn1C c1(OC)cc(C(N2CC(NC(C3CSCCS3)=O)CC2(C)C)=O)cc(N)c1OC N1(C(C=Cc2ccc(OC)cc2)=O)CCC(NC(=O)C=C2CC2)C(C)(C)C1 Cc1ncsc1C=CC(=O)NC1CC(CCNC(=O)COc2cccc(O)c2)C1 Cc1ccc(=O)n(CC(N2CCN(C(C3CCSC3)=O)C(CCO)C2)=O)n1 C(C)(C)(CCCC(=O)NOCCCCO)NC(Cc1c(C)ccnc1)=O N1(C(c2c(C)cco2)=O)CCN(C(=O)C(C)C2CCC2)CC1C(C)C c1(OC)ccc2cc(C(=O)NCC(O)CNC(=O)Cn3ncnn3)[nH]c2c1 C1(CCNC(c2csc(C3CC3)n2)=O)COCCN1C(=O)CCCn1ccnn1 C(c1ccc(Cl)cc1F)=CC(N1CCC(NC(=O)CC2CCOC2=O)(CF)C1)=O C1(NC(=O)C=Cc2ccc(Cl)s2)CCC2CN(C(c3csnn3)=O)CCC2C1 c1(CC)ncoc1C(=O)N(C(C)CCNC(c1cc(C(C)C)[nH]n1)=O)C c1(C(C)NC(C2CN(S(C)(=O)=O)C2)=O)ccc2c(c1)CN(C(C1(CF)CC1)=O)C2 N1(C(CCc2cnc(C)[nH]2)=O)CC2COCCC2(C(=O)OC(C)(C)C)C1 C(c1ccnc(Cl)c1)=CC(=O)NC1CC(NC(N)=O)C1 C12(C(=O)NCC(CC)N(C)C(c3csc(C)c3)=O)CCC(N=[N+]=[N-])C1C2 C1(CCOC)(NC2CCCO2)CCN(Cc2noc(CCCC(=O)OC)n2)CC1 c1(NC(C2C3CN(C(CNC)=O)CC32)=O)ccc(Cl)c(I)c1 C(=O)(C(C(=O)OC)C(C)NC(=NCCNS(C)(=O)=O)NC1CCC1)OC N1(C(CC=CC)=O)CC2CCCCC2(CNC(=O)CCCOCC)C1 Cc1cc(C(=O)NCC2CC2NC(=O)CCc2cncnc2)c(Br)c(C)c1 C1(F)(CN(C(CNC(=O)NC)=O)C)CC(CNC(C2CCN(C(C)=O)C2)=O)C1 Cc1cn(C)nc1C(=O)NCC1CCCCC1NC(C1(c2cc[nH]n2)CCC1)=O N1(C(c2c(C)non2)=O)Cc2n[nH]cc2C1C(=O)N(C1CC2(CC2)C1)C N1(C(C)C)CC(C(=O)NCC(O)CNC(=O)COCc2nc[nH]n2)CC1=O Cc1ccc(F)c(C(=O)NCC2CC2NC(c2nc(Cl)c(Cl)s2)=O)c1 c1(CC)ccc(C(=O)NC2CCC(F)(CNC(=O)C(F)C3CCC3)C2)c(C)n1 c1(C(C)C)cc(C(=O)N(CC(C)NC(=O)Cn2cnc(Br)c2)C)on1 C1(C(=O)NC2CC(n3cc(C4(O)CCOC4)nn3)C2)CCOCC1F c1(C(=O)NCC2CC(F)(CNC(COCCC)=O)C2)ccc(C)cc1[N+](=O)[O-] N1(C(Cc2cccc(C#C)c2)=O)CCC(CNC(=O)CCCC)C(F)(F)C1 C1(N(C)C(C2CC=CCC2)=O)C2CN(C(=O)CCc3ccc(O)cc3)CC12 C1(C(N2CCC(C)C2CNC(C2CC(n3cnnc3)C2)=O)=O)C2CCC1(C)C2(C)C C=CC1OCCC1C(=O)NCCC1(NC(c2cc(CC)c[nH]2)=O)CCC1 c1(CN2CCN(C(CC(C)C)=O)C3C2C3)cc([N+](=O)[O-])ccc1O c1(C(=O)NC2CCC(NC(C3(C#C)CC3)=O)CC2)nnc2c(F)cccc2c1O c1(C(N2CC(C)N(C(=O)CSC3CC3)CC2)=O)cc(P(C)(C)=O)ccn1 C1(C)(NC(CCOCCC(=O)OCC)=O)CCC(C)C1.C1(CC(=O)NCC)(O)CC1 C1(CC(=O)NCC(C)(C)NC(c2cn(C3CCOC3)cn2)=O)CCCNC(=O)C1 C1(S(C)(=O)=O)(C(=O)OC)CC(NC(c2ccc(C(C)C)c(C)c2)=O)CCC1 c1(C(=O)OC)ccc(C=CCN(CC)Cc2nc(C)cc(C)n2)cc1.c1(=O)cn1 c1(C(=O)Nc2ccc(I)nc2)ccc(-c2cncc(C3CCCC3)c2)c(F)c1 n12nc(C)c(c1C)COC2.c1(SCC)ccc(-n2cc(CCCN)nn2)cc1 c1(CNC(C2CCCC(Br)CC2)=O)cc(Br)cc2c1OCC2 c1(OC)cc(CC(=O)NC(C)Cn2nc(C)c(C(=O)O)c2C)cc(Cl)c1 N1(C(C2OCC(C)(C)C2)=O)CCC2(CC1)CN(C(=O)CC(F)F)C2 C=C(C)CC(C(=O)N1CCC(=CCNC(=O)C(N2CCSCC2)C)CC1)OC C1(CNC(CN(C2CCCC2)C)=O)COCCN1C(c1occc1F)=O C(=O)(C1=C(c2ccccc2)SCCO1)NCC1(CNC(CCCCC=C)=O)CC1 N1(C(CCc2onc(C)n2)=O)CCCN(C(c2cc3c[nH]cnc-3n2)=O)CC1C C1(NC(COCC)=O)CCC(C)N(C(=O)CCc2nc(C3CC3)n[nH]2)C1 C1(NC(Cc2ccn(CC)n2)=O)CS(=O)(=O)CC1NC(=O)C(=O)C(C)(C)C c1(C(N(CCNC(=O)CC2COCCO2)C2CC2)=O)cc(C(F)(F)F)ccc1O c1(CC(=O)NCC2N(C(c3c(COC)noc3)=O)CCC2)c(OC)cccc1F O=C1CN(C2CC3CCC2CN3)CCN1 C1(NC(C(CSC)(C)NC(c2ncc(F)cc2C)=O)=O)CC2CC1C(O)C2O c1(C(=O)NCC(N(C(C(CC)SC)=O)C)C2CC2)c(F)ccc(O)c1O C1(CC(=O)NC)CN(C(=O)C(C)OC)CCN1C(c1cc(O)ncn1)=O C1(C(=O)N(CCCNC(c2cc(C)nn2C)=O)CCO)(OC)CCCC(C)(C)C1 CS(=O)(=O)C1(C)CC1.C1(N(C(=O)NCC2CC2)CO)CCN(C2CC2)C1 Cn1ccc2c(C(N3CC4CC(NC(c5ccc[nH]5)=O)C(C4)C3)=O)ncnc12 CC1(NC(C2COCCO2)=O)CCN(C(C2CC3(CC3)C2)=O)C1 C1(CC)(NC(=O)CCF)CCN(C(C2CCC3CC3CC2)=O)CC1 CON=Cc1ccc(C(=O)NC2CCC2NC(=O)C2=CCc3ccccc32)cc1 C1(CN(c2ccnn2C)C)CC(O)CCN1S(=O)(=O)CC1CCC1 N1(C(CCC#C)=O)CCCCC1CC(=O)NCC(=O)N(C)CC c1(C(=O)NCCC2N(C(c3c(CC)nco3)=O)CCCC2)cccc(S(C)=O)c1 C1(CNC(c2c(C)nc(O)[nH]2)=O)CC2CCC(C1)N2C(=O)CCCn1cccc1 Cc1c(C(=O)NC23CCN(C(=O)CSc4cccs4)CC2C3)[nH]c2c1CCCC2 C1(CC)CN(C(=O)COc2cn[nH]c2)CCN1C(=O)CCc1cccnc1Cl c1(C(C)(C)NC(=O)NC2CC(C3CC3)C2)cc(Br)ccc1F CC1(C)CC(C(=O)NC2CCCC(O)C2)(CNC(=O)Cc2ccco2)C1 O=C1NCCCCC1CC(N1CCSCC1CCNC(C1CC12CC2)=O)=O CCC(C)C(C(=O)N1CC=CC(NC(=O)Cc2ccc(Cl)c(F)c2)C1)OC Cc1ccc(C(=O)NCC(C(C)C)NC(=O)CCc2ccnc(C)n2)nc1 N1(C(C(c2scc(C(=O)OC)c2)=O)=O)CCN(C(C)=O)C2(CCCC2)C1 C1(C#N)(C(=O)NC(CCCC)CNC(=O)CCNC(=O)C(C)(C)C)CC12CCC2 N#Cc1ccc2[nH]cc(CN3CCC(NC(c4cccc(Br)c4)=O)C(F)C3)c2c1 c1(OC(C)C(N2CC(C(=O)NCc3nncs3)CC2(C)C)=O)ccc(F)cc1F CN1CC(C)(C(=O)N(CCC(=O)NCC2CCN(C(N)=O)CC2)C2CC2)CC1=O N(C(=NCc1nc(C(C)(C)C)co1)NC1CC1)C(C1CCCC1)C CC(C)C(CCNc1cccc(OCC(=O)N(C)C)c1)NC(=O)C1=CCCO1 C1(C(=O)NC2CCC(NC(C3CCCN(C)C3)=O)C2)C2CC3C(C2=O)C13 C1(C(=O)NC2CCC(CNC(C3C(C)C3)=O)C2)CCCC(C)C1 N1(C(COCC)=O)CCOC(C)C1C(=O)Nc1cncc(SC)c1 N1(C(CC=CC=C)=O)CC2CCC1C1CN(C(c3c[nH]cc(Cl)c3=O)=O)CC21 c1(C(=O)NC2CCCCN(C(C(C)OCC)=O)C2)ccc2c(c1)CN(C)C(=O)N2 C=CC(C)(CCOC)C(=O)N1CCC2CN(C(C3CC(n4cccn4)C3)=O)C2C1 C1(C(=O)NCCC2N(C(c3cnc(C(C)C)s3)=O)CCC2)CCOC(C)C1 c1(C(=O)NC2(C(=O)NC(CCCCC)C3CC3)CC2)ccccc1C#N c1(C(=O)NCC(C)(C2CC2)NC(C2OCC(C)C2)=O)ccc(N)c(N)c1 N1(C(C=CC)=O)CCC(NC(=O)COc2ccc(Cl)cc2N)CC1C1CC1 c1(CC(=O)Nc2nccc(Br)c2Br)cnc2ncccn12 O=C1NC(=O)C(CC(N2CCCCC2CC(N2CC(OC(=O)N3CC3)C2)=O)=O)N1 CCCC(CC)CCC(=O)N(C1CCC(NC(c2scnc2Cl)=O)CC1)C C(c1cnccn1)=CC(=O)NCC1C2CN(C(C3CCCS3(=O)=O)=O)CC12 N1(CCO)CCN(c2ccc(Br)cc2)CC1.Cn1cc(C(C(F)(F)F)NC(=O)N)cn1 c1(C(N(CCOCCN(C(C2(COC)CCOC2)=O)C)C)=O)cc(Cl)cnc1O C1(CN(C(CCn2c(C(C)C)ncc2)=O)C)CN(C(C2COCCO2)=O)CCO1 C=C1CCN(C(=O)C#CC2CCOC2)C(C(N2CCOC(C3CC3)C2)=O)C1 C(CS(=O)(=O)CC(=O)N1CCC(O)(CCNC(c2ccc(COC)[nH]2)=O)C1)OC C(=O)(C(C)(C)CC(C)C)NCC(CC(=O)NC(CCCC)CCC)O c1(C(=O)NC2CN(C(C(C)CN(C)C)=O)CC2(C)C)cc2c(nn1)CCOC2 N1(C(CC2N(C(c3c(C#C)c[nH]n3)=O)CCC2)=O)CCOC2CCCCC12 N1(C(c2cn(CC=C)nn2)=O)CCC(CN(C(=O)CN2CCCCC2)C)CC1 C1(CNC(c2cncc(C)c2)=O)CCCCN(C(=O)C(C)C(C)(F)F)CC1 C1(NC(c2c(C)c(C3CC3)on2)=O)CCN(C(c2cnc(O)n2C)=O)CC1F C1(C(=O)Nc2scc(C#N)n2)C2C(CN1C(c1cscn1)=O)C2(C)C c1(N(C)C(=O)OCC(c2ccc(Cl)s2)=O)noc2c1CN(C(C(C)(C)C)=O)CC2 C=CC1(C(N2CC(c3nncs3)C2)=O)CCN(C(c2ccnnc2)=O)C1 CN1CCCCC1CC(N1CC(N(C)C)C(CNC(c2cnsc2)=O)C1)=O C(=O)(C(O)C(C)SC)NCC1(CNC(c2cnn(CC)n2)=O)CC1 N1(C(C(COC)NC(=O)COc2cccnc2)=O)CC2CC(CO)C(C2)C1 C#CC1(NC(C2CC(C)CN(C(C3CCCOCC3)=O)C2)=O)CCCOC1 C1(CCNC(c2ccn(CCF)n2)=O)CN(C(=O)CC2CCC(=O)N2)CCO1 C(N=c1[nH]c2cc(C)ccc2o1)C1CCC(NC(c2cc(C)cc(C)n2)=O)C1 CN=c1ccc(C(=O)NCC2(C)CN(C(C3(C)CCC(=O)NC3)=O)CC2C)c[nH]1 c1(C(=O)NC2(CNC(c3cn(CC(C)C)nc3)=O)CCC2)sccc1C#N C(c1ccn(C)c1)=CC(=O)N(CCC(N1CCC1(CC)CC)=O)CC#C Cc1cc(=NCCC(F)(F)Cl)[nH]c(NC(c2ccccc2)CCC2CC2)n1 C1(n2cc(CCC(C)O)nn2)CN(C(=O)Cc2c(I)cnn2C)CC1C N1(C(C2CCCC(CNC(C3(CC)CC3)=O)C2)=O)CCCC(F)(F)C1 Cc1ccc2c(C(=O)NC(C3CCN(C(c4c(C)coc4C)=O)C3)C)coc2c1 CCC(CC)CC(=O)N(CCC(=O)NCC1CCN(C)C1=O)CCO C1(N(C(CC(C)OC)=O)C)CCC2CN(C(c3n[nH]c(CO)n3)=O)CC12 N1(C(CC2(C=C)CC2)=O)CCC(C(F)F)(CNC(=O)Cn2cnccc2=O)C1 C12(CCOC)CCN(CC1)C2=O.c1(NC(c2cc(OC)n[nH]2)=O)ccc(Cl)cc1 Cc1cc(C(F)(F)F)ccc1S(=O)(=O)NCC1CC(C)N(C)C(C)C1 C(C)(CCC(=O)NC12CC(C(=O)Nc3ncccc3F)(C1)C2)OC c1(C(C(=O)N(CCCNC(C2CC2[N+](=O)[O-])=O)C)O)cccc(Br)c1 CC1(C)CN(C(c2cc(N)nc(Cl)c2)=O)CCN(C(C2(C)CCCOC2)=O)C1 C(=O)(C(O)CC[S+](C)C)NC1(c2ccccc2)N(C(=O)OC(C)(C)C)CCC1 N(C1CCC(N)c2ccccc21)C(C1(O)CC(C(=O)OC)C1)=O C1(CC(N2CCC(OC)C2C)=O)C2CCCC2N1C(=O)COC1CCOC1 N1(C(CN(C(=O)C2CC2)CCO)=O)CCN(C(C23CCN(CC2)CC3)=O)C2CC12 C12(C(=O)NC(CC(C)NC(c3coc(C#N)c3)=O)C)C3CCC(CC13)C2(F)F C#Cc1ccc(Cl)c(C(=O)NCC(O)CNC(=O)C(C23CCC(CC2)C3)CC)c1 c1(N2C(CNC(c3scc(C)c3)=O)CC2)nc2ccc(F)cc2s1 c1(OC)ccc(F)c(NC(C2CN(C(=O)CCCCCl)CCC2O)=O)n1 c1(NCC2C(C(=C)C)OCC2)nccc(=NCc2nc(CC)nn2C)[nH]1 c1(C2C(C(=O)N(c3ccccc3)c3ccccc3)C2)cccc(Cl)c1 N1(C(C2(CC)CCN(C(c3cccc(F)c3F)=O)C2)=O)CCC(F)(F)CC1C Cc1coc2c(C(N3CC(O)(C(C)NC(c4cscn4)=O)C3)=O)cccc12 C1(NC(c2cnn(CCO)c2)=O)CCC(NC(=O)C(F)OC(F)(F)F)C1 c1(CNC(N2CC(C)C2C(C)C)=O)ccccc1Br C1(C(=O)NC(CNC(c2nccc(OC)c2)=O)C(C)(C)C)CCOC(=O)CC1 CC(C)C(O)C(C)C(=O)NCC1CCC1NC(=O)C(C)(C)C c1(NC(C2CCN(C(CNC(CCC)=O)=O)CC2)=O)ccc2occc2c1 C1(C(=O)NCC(C)N(CC)CC)CCCCCN1C(c1coc2c1COC2)=O CCC(C)CC(=O)C(=O)NCc1nc(C(=O)OC)co1 C1(C(=O)NC(CCCNC(C(=O)NCC)=O)C)CCC(F)(F)CO1 CCCCC(CC)CC(=O)NCC(C)(CC(C)C)NC(=O)CN(C(=O)C(C)C)C C(N=c1cccc(S(=O)(=O)NCC(C)CC2CC2)[nH]1)c1cc(OC)c(Cl)cc1 C12(CNC(C(C)NC(N)=O)=O)CN(C(=O)CC3CCCCC3O)CC(F)(C1)C2 C1(=CC(=O)NC2CCN(C(CC(C)(C)O)=O)C(C3CC3)C2)CCCCCC1(F)F Cn1nc(C(F)(F)F)cc1C(=O)N(CC(N)=O)C1CC1.N12CCCC(C1)C2 C1(NC(c2ccc(C)c(C)n2)=O)CCCC12CCN(C(=O)CCNS(C)(=O)=O)C2 N1(C(c2cc(CCC)[nH]n2)=O)CC(OC)CC1(C)CNC(c1cnn[nH]1)=O c1(NC(C(c2nnnn2C)C)=O)cccc(C(=O)NCC2(C3CC3)CCCO2)c1 C(=O)(CC(C)C(C)C(C)C)NC1CC(NC(C=Cc2c(C)ncs2)=O)C1 c1(C(=O)NC(C)CCCNC(=O)C(C)(C)c2cccs2)ccnn(C)c1=O c1(C(N(CCCCOC)C)=O)csc(CNC(C2(O)CCSC2)=O)c1 N1(C(c2nn(CC)c(C)c2)=O)CCC2CCN(C(=O)CCS(C)=O)CC12 CCC(C)(CNC(c1n[nH]cc1C)=O)C(=O)NC1COCC(C)(C)C1 c1(N(C(=O)CO)C(C2CC2)NCC(N2C(C)C3CC2C3)=O)ccc(C#N)c(Br)c1 C1(C(=O)NC(C#C)C2CC2)(NC(c2ccc(C)s2)=O)CCc2cc(Br)ccc2C1 C(C(C)C(=O)NCCC(=O)NCc1cncn1C1CC1)N(C)C1CC1 C1(C(=O)NC2C(C(=O)NOC3CCCC3)CC2)CC12CCCCC2 c1(CCNC(=O)NCC(n2cc(Br)cn2)C)ccc(C(C)(C)C)nc1 C(C(C(=O)N1CCCC1CCC)C(C)C)NC(C=CC)=O c1(C(=O)OC)cc([N+](=O)[O-])cnc1C.C1N=C2NC(=NC(=N)N2)N2CCC1C2 c1(OC)ccc(-c2nc(C3CCCOC3)n(-c3ccc(F)cc3)n2)cc1 c1(CC(=O)NCC(CNC(=O)C2=C(Cl)CCCC2)CO)c[nH]c2cnccc12 CCC(CC(=O)NC1CC1C(=O)OC(C)(C)C)C1CC1.c12cccc(c1)NC2=O C12(C(N3CCC(C)(NC(C4=C(C)CCCC4)=O)C3)=O)CCC(C1)c1ccccc12 C1(NC(C(CC(CC)C)C)=O)CN(C(=O)CC(C)n2cccn2)C2CCCCC12 c1(CC(=O)NCC(CC=C)NC(c2ccc(C)cc2F)=O)cc(F)cc(F)c1 c1(OC)nccc(Br)c1C(N1CCCC1CNC(=O)C(C)C1CC1)=O c1(CCNC(C(C2CC=CCC2)NC(c2ccc(CC)o2)=O)=O)ccc(C)cc1 Cn1c(-c2ccc(-c3c(F)cc(Br)cc3F)cc2)nnc1NOCC(=O)O N1(C(C(COCC=C)c2ccccc2)=O)CCC(C)(NC(=O)C=C(C)C)CC1 N1(C(c2cnc(C)[nH]2)=O)CCC2C(CCCN2C(c2cccc(F)c2C#N)=O)C1 C1(NC(c2c(C)nc(C)s2)=O)C2CC3CN(C(=O)C#CC4CC4)C1C3C2 N1(C(c2cc(CC)c(C)s2)=O)CCC(C)C(CNC(=O)C(C)=C2CCC2)C1 c1(C(=O)NCCC(C)NC(c2cncc(F)c2)=O)cnc2c(c1)COCC2 N1(CC)CCOCC1C(=O)NCCC(C)(C)NC(c1cscn1)=O c1(C(=O)NCC2(F)CC(NC(c3cncc(F)c3)=O)C2)cnc2ccc(F)cn12 c1(NCCNC(=NCCC)NCC(C)(C)OC)ccc2nnn(C)c2n1 N1(C(C2CCCN(C(COC)C)CC2)=O)CCC(C2CCN(C)C2)C1 CC(CN(C)C)C(=O)NCCC1CCN(C(=O)C(=O)NCC#N)C1 N1(C(c2cnn(CCOC)c2C)=O)CCC(CNC(=O)CCS(C)(=O)=O)CC1C C1(N(C(c2cncc(C(C)C)c2)=O)C)CCN(C(=O)COC(C)(C)C)CC1C c1(CC(=O)N(CC(CN(C(=O)CSC2CCCC2)C)O)C)ccc(Cl)s1 C1(CCNC(C2C(C)=CCS2)=O)CCCN(C(c2cc(CO)ccn2)=O)C1 c1(OC)cnnc(C(=O)NC(C)(C)CC(=O)N2C(CO)CC2CO)c1 C#Cc1cccc(C(=O)NC(c2cccnc2)C(=O)NCCCc2ccco2)c1 N1(C(C(C2CCOC2)OC)=O)CCC(CF)(NC(=O)C2=CCCS2)C1 N1(C(C=Cc2c(C)nsc2)=O)CCN(C(=O)Cc2cnccn2)C2CC12 C1(NC(CC2(C=C)CC2)=O)CCN(C(c2ccc(C)n2C)=O)CC1O c1(CC(=O)NC2(CN(C(=O)Cc3cnnn3C)C)CC2)c(F)cccc1Cl CC(C)C(F)C(=O)N(CC(=O)NC1CC(C)(C)C1)C(C)C c1(NC(C2(C)CCN(Cc3ccsc3)CC2)=O)cc(F)cc(C#N)c1 C1(NC(c2cnn(CC)c2C)=O)CS(=O)(=O)CC1N=c1cc(C)c(C#N)c(C)[nH]1 C(C)(C)(CC(F)C(=O)N1CC(C(F)(F)F)C1)n1cc(CCC[Si](C)(C)C)nn1 c1(CC)ccc(C(C)=CC(=O)NC2(CO)CN(C(=O)CC(CSC)CC)C2)cc1 N1(C(C2N(C(C3(NC(C)=O)CC3)=O)C3C(C2)C3)=O)CCC2(CO)CCCC12 c1(OCC)cc(CN2CCC(O)C(C(N3CCOC(CO)C3)=O)C2)ccc1Cl N1(C(C(C(C)C)NC(N)=O)=O)CC2CC1CC2NC(C1CCC(F)(F)CC1)=O CC(C)CCCCC(=O)NC1CN(C=O)CC1C1CC1.c1(N)cccn1C CCCC(O)C(=O)NC1CCN(C2CCN(C(=O)NC3CC4C=CC3C4)C2)CC1 CC1CC(CO)CN(C(c2conc2CNC(=O)CN2CC=CC2)=O)C1 N1(C(C2N(C)CCCC2)=O)CCN(C(=O)CSc2ccc(F)cc2Cl)CC(O)C1 C1(C(N(CC#C)CC)=O)CCN(C(=O)C=CC=CCC)CC1 c1(N(C)CC2(n3cc(N)cn3)CC2)cc(F)c(C(=O)O)c(F)c1 C12(NC(C(C3CCC3)OC)=O)CC(CNC(C3CCC=CCCC3)=O)(C1)OC2C Cc1cc(CO)oc1C(=O)NCC1(CNC(=O)Cn2cncn2)CCCC1 N1(C(Cc2ccn(C)n2)=O)CCC12CCN(C(=O)C(c1ccccc1Cl)O)CC2 C1(NC(c2ncccc2C2CC2)=O)CC2(CCN(C(c3ccc(O)nc3)=O)C2)C1 c1(-n2cc(C(=O)NC3(C)CC(NC(=O)C(F)F)C3)nn2)ccc(Cl)cc1 C=CCC(CC=C)C(=O)NCC1(C(N2CC(c3cc[nH]n3)C2)=O)CC=CC1 C(C(=O)N=c1ccn(C(F)F)[nH]1)NC(C(C(CC)C)c1ccccc1)=O c1(C(=O)NC(C(C)NC(c2c(C)occ2)=O)C)cc(Br)cc2cccnc12 C(CS(=O)(=O)CC(=O)N1CCCN(C(c2cnc[nH]2)=O)C(CO)C1)OC c1(C(N(C(C)CNC(c2ncoc2C2CCCO2)=O)C)C)cc2ccccc2o1 C#CCCCCC(c1nnnn1C1CCC1)NCC(C)(C)S(C)(=O)=O c1(CC)cccc(F)c1NC(C1C2CN(C(c3cncc(C#N)c3)=O)CC12)=O CS(=O)c1ccc(CC(=O)NC2CCC2NC(c2ccccc2O)=O)cc1 N1(C(C(C)OCCCCCC)=O)CC=CC(NC(C2CS(=O)C2)=O)C1 N1(C(=O)Nc2nc(CC3CCCO3)cs2)CCN(c2ccc(F)cc2)CC1 C(=O)(C(C)CCN(C)C)N1CC(COC)(NC(c2oncc2C)=O)C1 C(CNC(=O)Cc1ccsn1)(CC(=O)NCc1cncn1C)OC Cc1cnc(NC(=O)CN2CCN(C(=O)CC3CC3)CC2)c([N+](=O)[O-])c1 C1(C(=O)OC(C)C)CC12CC(C(=O)NCCCCNC(=O)C(C)N1CCCC1)C2 C1(C(=O)NC(C2CN(C(C(CC)(C)C)=O)C2)C)CCOCC12CCCC2 N1(C(C(C)c2ccco2)=O)CC2=C(C1)CN(C(=O)C#CC1CCOC1)C2 c1(CC)cc(C(N2CCC(C3CCCN3Cc3cn(C)nc3Cl)C2)=O)ccc1Cl C(=O)(C(C)S(N)(=O)=O)N(C)CC1N(C(C(CC)OC)=O)CCCC1 C(=O)(CCC(C)(C)F)N(C)C.C1(=O)CCS(=O)(=O)NC2CC(C2(C)C)N1 C1(C(N2CCC(CC=C)(NC(c3scnc3CC)=O)C2)=O)CC2CCC(C1)C2 Cc1nc2c(C(=O)NC(C3CCN(C(C4CCOC4C)=O)C3)C)cccc2o1 C1(F)(C(=O)NCC2(C)CN(C(c3cccc(Br)c3)=O)C2)CCOCC1 N1(C(c2cc(C)[nH]n2)=O)CCC2(CC1)CC2C(=O)NCCS(C)(=N)=O c1(C(=O)NCC(CNC(C(C)OCOC)=O)C)ccccc1N1CCN(C)CC1 C1(CC(=O)N(CCCNC(=O)CN2CC3C=CC2C3)CC)CCOCC1(C)C c1(C(C)(C)C)nocc1C(=O)NC1CCN(C(c2cccnc2)=O)C1 N1(C(CNC(C2C(=C)C2)=O)=O)CC(C(=O)NC(COC)CC)CC(C)C1 c1(SC(C)C(=O)NC2CCC(NC(=O)Cc3csc(=N)[nH]3)C2)ccc(F)cc1 C(=O)(C1=CNC2=NCCC2=C1)N1C(CN(C(C2C(CC)CCO2)=O)C)COCC1 O=C(CCCN(CCc1cccnc1)C1CC1)NCC(=C1CN(C(=O)C=CBr)C1)F c1(C(=O)OC2C=CCCCC2)cnc(Cl)c(Cl)c1 c1(CC(N2C(CN(C)C(C3CC4CC3C4)=O)COCC2)=O)cccc(F)c1F Cc1nn(C)c(Cl)c1NCc1c(CNC(C2(C(=O)N(C)C)CC2)=O)cnn1C c1(C(=O)NCC2CCCC(NC(C(CC)(C)CC)=O)C2)ccc(F)c2occc12 C1(C(=O)NCC(N(C(=O)C=Cc2ccccc2Cl)C)C2CC2)CCCCCC(=O)C1 C1(CC(N2CC(CC(C)NC(CCCCC#C)=O)C2)=O)CCC2(CC1)OCCO2 CN1CC(=O)N(Cc2ccc(O)nn2)C1=O.N1(CCO)C(=O)NCC=CC1 C1(NC(c2c(CC)noc2)=O)CCC2CCN(C(=O)CCn3cncn3)C1C2 C12(NC(c3cc(CC)on3)=O)CCCCC1N(C(=O)Cc1ccc(C)s1)CC2 C=CCC(CC(=O)NCC12CC=CC(C1)OC2)NC(C12CCC(C1)C2)=O C12(C(=O)NCC(C)N(C(=O)CSCCC#N)C)CC(C)(C1)OC21CCC1 c1(CC)cc(C(=O)NC(C(C)NC(C2CC3C=CC2CC3)=O)C(C)C)cc(N)c1 c1(CC(=O)NCC2CCN(c3c(OC)cncn3)C2(C)C)ccc2c(c1)OCO2 c1(OC)ccc2cc(C(=O)OC3CC34CC4(F)F)[nH]c2c1 c1(NC(c2ccc(Cl)c(Cl)c2F)C)cccc(S(=O)(=O)NCC(CO)N(C)C)c1 CC(C(=O)NCC1CC2CN(C(=O)CC3OCCCO3)CC12)C(C)(C)C Cc1ccsc1C=CC(=O)NC(C1CCN(C(=O)CSCC(N)=O)CC1)CO CC1CC(NC(c2n[nH]c(=N)[nH]2)=O)CCN1C(=O)CSc1ccccc1Cl c1(NC)cncc(C(N2CCC(C(C)(C)NC(C3CC(C)C3(C)C)=O)C2)=O)c1 c1(CCC(N2C(C(=O)Nc3ccc(F)cc3O)CCC2)=O)ccccc1[N+](=O)[O-] N1(C(CCOC)=O)CCC(NC(=O)C(C(C)C)n2cnc(C)c2)C(C)(C)C1 O=C(C1=NN(C2CC2)C(=O)CC1)NC1(CO)CCN(C(c2cnco2)=O)CC1 C12(CC(=O)NC3C(NC(=O)COCC4CCOC4)CCC3)CCCN1CCC2 C1(OC)CC2CCC1CC2C(N1CCC(N(C)C(=O)OC(C)(C)C)C12CC2)=O C(=O)(CCC(C)(C)C)NCC1(OCC)CN(C(C2N(CCC)C(=O)CC2)=O)C1 N1(C(=O)C=Cc2ccc(Cl)s2)CC2(CC(NC(=O)C(F)(F)CO)CO2)C1 Cc1cc(C(=O)NCC(C(C)C)NC(=O)C(C)Sc2ccccc2)ncc1Cl Cc1cc(=NCCCCS(N)(=O)=O)[nH]cc1S(=O)(=O)NCCCC(C)(C)C(=O)O N1(C(CC2(OC)CCC2)=O)C2CCC1CN(C(=O)Cc1n[nH]c(C)n1)C2 n1(CC=C)ncc2ccc(NC(=O)C(=O)NCC(c3ccco3)OC)cc12 CCCC(C)(CC)C(=O)NC1CCC(C(N2CC(=O)NC(C)(C)C2)=O)C1 C1(CC#C)(C(=O)N(CCCn2ccnc2)C)CCN(C(=O)C(C)OC)C1 C12(CNC(c3n(C=C)nnc3)=O)CCC1CCN2C(=O)CC1CN2CCC1CC2 CC(C)C(C)(CNC(=O)CN1CCC(N(C)C)C1)NC(C1CCC1)=O c1(OCC)ccc(C(=O)NC(CO)CCc2ccccc2)c(C)c1 c1(C(N(C2CCN(C(c3csc(C)c3C)=O)CC2)CC)=O)c(OC)ccnc1O C(CCCC(=O)NC1CC(n2cccn2)C1)NC(C(CC)SC)=O C1(C(N(C(CNC(c2cn(CC)nc2C)=O)C)C)=O)CC2(C1)CC(F)(F)C2 C1(O)(CC=C)CCN(C(=O)CC(C(C)OC)NC(=O)C(O)CCSC)CC1 c1(CN2CC(C(=O)Nc3ncco3)SCC2)c(Cl)cccc1I N1(C(Cc2cccc(COC)c2)=O)CCN(C(=O)Cc2n[nH]c(C)n2)C(C)C1C c1(C(=O)NCC(CNC(=O)C(C)=CC(C)(C)C)OC)cc2c(s1)CN(C)CC2 N1(C(c2cc(S(C)(=O)=O)ncc2)C(=O)NCCC#N)CC2C3CCC(CC3)C2C1 C1(OC)CC(NC(=O)CC(C2CC2)NC(C2CNC(=O)O2)=O)C12CCC2 c1(C(N2CCCC2Cc2ccc(Cl)cc2)=O)ccnc(OC2CCCC2)c1 c1(SC)cc(F)ccc1C(=O)N(C)CC1CN(C(c2[nH]ccc2C)=O)CCO1 C1(CC(=O)NCC(CNC(c2c(C(C)C)con2)=O)(C)F)CC=CCN1C C(C1c2ccccc2CN1C(=O)CCC(N)=O)NC(c1c(C)n2c(s1)cnc2)=O C12(C(N3C(C(CC)C)CCC3)=O)COCC1CN(C(=O)CCC1(Cl)CC1)C2 N1(C(c2c(CC)cco2)=O)CCN(C(c2coc(Cl)n2)=O)C(C)CC1C C1(C(=O)NC2C(C)(CN(C(CC(CCC)O)=O)C)CCC2)CC2(CCCC2)CO1 C(CN=C(NCc1n[nH]c(CO)n1)NCc1ccccc1)SC.C1(S)COC(C)(C)C1 c1(C(=O)NCCCNC(C(C)N(C)CC)=O)cc(OC(F)F)ccc1F C1(C(N2CC(C(C(=O)NCCC(O)C(F)F)OC)C2)=O)C2CN(C)CC12 N1(C(c2nn(CC)c(C)c2)=O)CC2(CNC(=O)C(O)C(C)OC)CCC1CC2 c1(CCC(=O)N(CC(CC)NC(C2C=CCC2)=O)C)nc(CSC)no1 CCCCC(COC)N=c1nc2scnc2c(N2C3CCC(C3)C2CO)[nH]1 C1(CNC(C(C)OCC=C)=O)CN(C(c2cnc(N(C)C)s2)=O)CC1O c1(C(N(C)CC2CCN(C(=O)C3CC3)C2)=O)noc2c1COCC2 C(CCN=c1[nH]cnc2c1CCCC2)N(C)C(c1cnc(C2CCOC2)s1)=O c1(C(N(C)CCC2CCN(C(CSC)=O)C2)=O)n[nH]c2c(C)cccc12 N1(C(CC2N(C(=O)C=CCO)CC2)=O)CCN2CC(O)CC2C1 c1(NC(C2(C(N)=O)CN(C(=O)COCCCF)C2)=O)ccc(C(O)CF)cc1 N1(C(COC2CN(C(C(C#C)(C)C)=O)C2)=O)CC2(CCN2C)C1 S1(=O)(=O)C2CCN(N3CCN(CC3)CCN1)C2.N1(C(C)=O)CCCC1 C(=O)(CC(C)CCCCC)N(C1CCC(NC(CCCCC#C)=O)CC1)C N1(C(CN(S(C)(=O)=O)C)=O)CCCC(CN2CC(C(=O)OC)C2)C1 n1(CC(=O)NC2(CNC(C(C)(C)C(F)F)=O)CCOC2)cc2ncccc2n1 N1(C(C2(CNC(C(COC)C)=O)CCCO2)=O)CCC(C)(C(C)C)C1 C1(C(=O)NCCC2(C=C)CCC2)CCCN(C(c2cc(CCC)cnn2)=O)CC1 C1(C(N(CC(N2CC(O)(COC)C2)=O)C2CCC2)=O)C2CN(C)CC12 c1(-c2n(CC)c(N(C)Cc3cccs3)nn2)nn(C)c(=O)c2ccccc12 Cc1cn2c(n1)C(C)N(S(=O)(=O)c1scc(Cl)c1Cl)CC2 c1(CCNC(N2CCC(c3cncs3)CC2)=O)ccc2cc[nH]c2c1 N1(C(C2(CCOC)CC2)=O)CCOC(C(=O)NCC(CC)CO)C1 c1(C(=O)NCC(CC)NC(c2nncs2)=O)ccccc1SC(F)F O=C1Cc2cc(C(N3C4CN(C(=O)Nc5ccc(F)c(Br)c5)CC34)=O)ccc2N1 CN(CCc1ccccc1)ONCCSc1ccccc1.CC O=S1(=O)CCC2(CC1)CN(c1nc(=NCC3CCCO3)[nH]c3c1COCC3)CCO2 CC1=CCN(C(C2CC(C)N2C(=O)Cc2ccc(F)cc2)=O)CC1 CC(C(=O)N1CCCc2ccnn21)NC(=O)C(=O)N(CC1CC1)CC1CC1 c1(OC)ccc(C(N2CCOCC2C(=O)NC2CCC(=O)NC2=O)=O)c(I)c1 c1(C(=O)NC(CCC=C)CO)cc(-c2cc[nH]n2)c2[nH]ccc2c1 C1(C(N(C(CN(C(C2(OC)CCSCC2)=O)C)C)C)=O)CC=C(C(C)C)CC1 n1(C(C)C(=O)NC2CCC(N(C(=O)CO)C)C2)cnc(C#N)n1 C1(C)(NC(c2nnc(C(C)C)s2)=O)CCCN(C(c2cc(CO)[nH]n2)=O)C1 C1(CNC(C=C(COC)C)=O)COCCN1C(c1ncc[nH]1)=O C1(C(=O)NC(c2ccccn2)C(=O)NCCOCC(C)C)OCCCC1(C)C C1(NC(C(C=CC)O)=O)CCN(C(=O)CCC(=O)Nc2nnc(C)s2)C1CC C1(C(=O)NC(CCCC=C)C2CC2)CCC2CCC1N2C(=O)Cn1ccc(C)n1 C(=O)(CC(O)CC(C)(C)C)NC1(C(N2CCSCC(C)C2)=O)CC(O)C1 Cc1cc(F)ccc1C(O)C(=O)NCC1CCCCN(C(=O)C(O)C(C)(C)C)C1 c1(C(N2CCC(CC=C)(NC(c3cc(OC)n[nH]3)=O)C2)=O)ccc2scnc2c1 c1(NC(C(C(C)C)OCC=C)=O)cc(CC)ccc1O Cc1noc(Cl)c1CCC(=O)NC(C)CC(C)NC(c1nncn1C1CC1)=O C1(NC(c2ccc(SCC)nc2)=O)CCCC12CN(C(C1CCC(OC)C1)=O)C2 c1(C(N2CCC(C)C2CNC(=O)Cc2cnc[nH]2)=O)ccc(Br)cc1C#N C(=O)(CC(C)C(F)(F)F)NC1C(CC)CN(C(C23CC(CO)(C2)OC3C)=O)CC1 C1(CC=C)(NC(C2CCCOCC2)=O)CC2CCC(C1)N2C(C1CC1OC)=O C12(CN(C)C(c3cnc(=N)[nH]c3)=O)CCC(CC1)CC2 c1(NC(C)(C)C)ccc(S(=O)(=O)NCC2(N(C)C)COC2)cn1 C1(C(N2CCCC(O)(CCNC(C3(OC)CCC3)=O)C2)=O)CN2CCCC2CO1 c1(N2CC3C(CNC(=O)NC(COC)=O)(CCCC3)C2)c(C)c(C)nc2ncnn12 N1(C(C(CC=CC)C)=O)C2CCCC1CN(C(=O)C1=C(C)OCCC1)CC2 NC(=O)CCC(=O)N1CC(F)CC1CNC(C1CCNC(=O)C1)=O C1(NC(C(CC2CCC2)N(C)C)=O)CCCCC1NC(C1(CO)COC1)=O C(=O)(C(COC)CC(C)C)N(CCCNC(c1c(C)nc(CCC)s1)=O)CC c1(C(=O)NC2C(CC)CN(C(C3(C)CC=CC3)=O)C2)cccc(Br)c1Cl C(=O)(C1=C(Cl)CCC1)C(=O)CCCC1CCOCC1.C1(CC(=O)N)CCCC1N C1(C(=O)NCCC2CCN(C(C3CC4CC4C3)=O)CC2)CC2COCC(C1)C2 CC1NC(=O)CCC1NC(C1CN(C(=O)C(C)N2CCCC2)CC1(C)C)=O C1(C(=O)NCC(CC(C)C)NC(C2(C)C(C)(C)C2(C)C)=O)CCCC(C)(C)C1 Cc1cc(C(=O)NC2CC(F)CN(C(=O)C(C)NC(N)=O)C2)c(C)cc1C c1(-c2cn(-c3ncc(Cl)cc3C(F)(F)F)nn2)cc2ccccc2nn1 C1(C(=O)NCC(C#C)OC)CC(O)CN1C(=O)C(C(C)C)OC.SCC c1(C(=O)NC2CC(CCNC(C3C(C)(CC)C3)=O)C2)cncc2ccccc12 N1(C(C=CCN(C)CC)=O)CCOC(C)(CNC(C2CCC(C)(C)CC2)=O)C1 c1(C(=O)NCC(N(C)C(C2CCS(=O)(=O)C2)=O)C2CC2)ccnc2c1cnn2C Cc1nn(C)c(C)c1C(=O)C(N1CCN(C(C2CC(=O)NC=CC2)=O)C(C)C1)=O c1(C(N2CC(CCO)(OC)C2)=O)cc(C)c(C)nn1.C(=O)(CO)NCCSC C12(NC(c3c(C)nn[nH]3)=O)CCC(CC1n1cc(-c3cccnn3)nn1)C2 C1(NC(=O)CSc2nnc(S)s2)CN(C(c2cnn[nH]2)=O)C2(CCCOC2)C1 c1(CC)cc(Cl)ccc1C(N1CC(N(C(=O)COC(C)CC)C)C(O)C1)=O Cc1cc(F)c(F)cc1C(=O)NC1CN(C(c2cc(Br)cs2)=O)CCC1F c1(C(N(C2CCCN(C(c3nnc(C)s3)=O)C2)CC)=O)cnn2c1CCCC2C c1(NC(CC2CCC(NS(CC(C)C)(=O)=O)CC2)=O)cnc(Cl)cc1Cl C(=O)(C1=CCN(C)C1)N1CC(C(C(=O)NC(C2CSC2)C)F)C1 c1(C(N2C(C(C)C)CN(C(C3(C)CC3(Cl)Cl)=O)CC2)=O)cnn2ccn(C)c12 c1(C(C)C(=O)NC2(CN(C)C(c3cc(C(F)F)[nH]n3)=O)CC2)ccc(F)cc1F Cc1c(NCc2ccc(C(N)=O)c(F)c2)nc[nH]c1=NCC1CNC(=O)C1 N12CCC3(CC1)CC3C2=O.N1(C2(c3cc[nH]n3)CC2)CC2CCC=CC12 C1(n2cc(C(C)O)nn2)CCN(C(C2CN3CCN2CC3)=O)CC1O N1(C(C(CCN(C)C)O)=O)CCCCC(NC(=O)CCc2ncnn2C)C1 C(=O)(CC(C(C)(C)C)NC(c1cc(C)c(O)nn1)=O)N1C(C)(CCC)CC1 C12(NC(C(C(C)O)C)=O)CCOC(CNC(C3(C#N)CC4CC4C3)=O)(C1)C2 C(CCCC(=O)N1CCCCC1C(N1CCN(CC2CC2)CC1)=O)(OC)OC C1(NC(CN(CCOC)C)=O)CC(C)(CO)C1.C12(CC1)C(=O)N2C N1(C(c2c(C(=O)O)[nH]cc2)=O)CCC(=O)CC1C1CCCC1 C1(CNC(C=CCCC)=O)CN(C(=O)CC2COC(=O)C2)CCN1C C1(C(=O)NCC2(NC(c3ccc(N)c(Cl)c3)=O)CC2)Cc2cc(Cl)ccc2O1 Cc1ccc2c(=NCC(C)(F)F)[nH]c(N3CCOC(c4cccnc4)C3)nc2c1 N1(C(CCC(C)N(C)C)=O)CCC2(CCCN(C(c3ccnc(Cl)c3N)=O)C2)C1 c1(C(N2CCCC(NC(CCC=CC(C)C)=O)(CO)C2)=O)cnc2[nH]cnc2c1 c1(C(=O)NCC2CCCN(C(=O)C=Cc3ccccc3F)C2)cc(O)nc(O)c1 N1(C(c2n(C=C)nnc2)=O)CCC(O)(CNC(c2nc(OC)c(C)s2)=O)CC1 C1(C(N(C(CF)CF)C)=O)C(NCC=C)C2CCCC12.C(C)(C)(C)S c1(C(=O)NC(CN(CCOC)C(c2cccc(CO)n2)=O)C)cccc(Cl)c1N N1(C(C2CC(OC)C2)=O)CCC(C)(CCNC(c2cc[nH]c(=N)c2)=O)C1 CC1=NS(=O)(=O)NC(C)=C1CC(=O)N1CCN(C(C2CCC(C)(C)C2)=O)CC1C c1(NC(CC(C)(C)CNC(c2coc(C(N)=O)c2)=O)=O)ccc2nn[nH]c2c1 Cc1ncc2c(C(=O)NC3CC(NC(C45CCCCC4OCC5)=O)C3)nccn12 N1(C(=O)CC2CCCC2)CCC2CCN(C(C34CC=CCN3CCC4)=O)CC2C1 CC(C)CS(=O)(=O)CCC(=O)N1CC(C)CN(C(C2CCCC(C)C2)=O)C(C)C1 N12CCCCCCC1C2=O.N1(C(Cc2c(C)nsc2)=O)CCN(C)C(C(C)C)C1 c1(C(n2cccc2)CC)nc(-c2ccc(Br)cn2)nn1Cc1ccccc1 c1(C(N2C(CNC(c3c(COC)n(CCO)nc3)=O)CC2)=O)ccn2ccsc12 c1(C(=O)NCC2(O)CN(C(C(n3cc(Cl)cn3)C)=O)C2)cnc(N)c(Br)c1 c1(N(C)Cc2c(C)sc(Br)n2)ccc(S(=O)(=O)N(C(C)C(C)C)C)cn1 c1(N2CCC(OC(C)C)CC2)ccc(S(=O)(=O)NC(CO)C2CCC2)cc1F C=C1CC(C)(C(N2CCC(NC(C34CC(c5ccccc5)(C3)C4)=O)C2)=O)C1 O=C1CSc2ncc(C(=O)NC3CS(=O)(=O)CC3NC(c3ccoc3)=O)cc2N1 CC(O)C(C(=O)NC1CCCC(NC(=O)OC(C)(C)C)CC1)Nc1ncccn1 c1(C(=O)NCC2C=CCN2C(=O)CC2CS(=O)(=O)C2)cnn2c1OCC2 N1(C(C(C(C(C)C)OC)O)=O)CC2OCCN(C(c3cc(F)cc(F)c3)=O)C2C1 C(N=c1cc(N2CC(CN3C(C)CCC3C)C2)nc(C)[nH]1)c1c(OC)scc1 C1(NC(Cc2nc(C)sc2)=O)CCC2(C1)OCCO2 N1(C(Cc2cccc(C)c2F)=O)C2CCC1C(F)C(NC(c1sccc1F)=O)C2 Cc1cc(Cl)c(C(N2CC3CN(C(=O)CCc4nncs4)CC3C2)=O)cc1C Cc1ccc(C)c(C(N2CCN(C)CC2CNC(c2nc(C)sc2C)=O)=O)c1 c1(CC(N2CC(C)(NC(=O)C(F)C3CCOC3)C2)=O)ccc2c(c1)NC(=O)C2 CCC(C)C(CO)CN=c1nc2sccc2c(NCC23CC(C)(CO2)C3)[nH]1 C=CCC(CNC(c1cscc1CC)=O)C(=O)NCC(O)C(N)=O C(=O)(C(CNC(=O)C(C)CC(F)(F)F)CC(C)C)N1CC(C(=O)NC)OCC1 c1(OC)ccc(CC(=O)NC2(CO)CCCN(C(c3cccn3C)=O)C2)c(Cl)c1 N1(C(C(c2ccncc2)C)=O)CCSCC1CCNC(=O)COC(F)(F)F C(C(C)N=c1[nH]c(=NCC2(CO)CN(C)C2)[nH]c2ccccc12)NC(=O)OC N1(C(c2c(CCC)nco2)=O)CCC(C(N2CCC(C)(CO)CC2)=O)C1(C)C C(=O)(CCC(C)(C)C)N1C(C(=O)NC(CC#C)CC#C)CC(OC)C1 CC1CN(C(=O)OC(C)(C)C)CC(C)N(C(C23CC2CCC3(F)F)=O)C1 C1(NC(c2cncc3ccsc23)=O)CC2CCC(C1)N2C(C1C2CCCC12)=O CCC(C)C(O)C(=O)NCC(O)CNC(=O)CC(C)N1CCCC1=O c1(OC)ccc(S(=O)(=O)N2CCOCC(CNC(=O)CCCCC3CC3)C2)cn1 c1(C(=O)NCCC2=CCCCC2)ccc(=O)n(C)n1.CC1CCCC12C(=O)N2C CC1Cc2cc(S(=O)(=O)N3CCCC4COCC34)cc(Cl)c2O1 CC(C)C(C)(O)C(=O)N1CCC(CO)(CNC(c2nccc(N)n2)=O)C1 N1(C(CCN(C2CCCCC2)C)=O)C(CNC(C2CCC2(F)F)=O)CC2CCCC12 C1(C(=O)NC(C(C)NC(c2csc(C(F)(F)F)n2)=O)CO)CCOC(C)(C)C1 C1(C(=O)Nc2c(C(=O)OC)ccs2)CC(F)CN(Cc2cccc(Br)c2O)C1 C1(O)(CC(=O)NC2CC(CNC(C(c3cnn(C)c3)C)=O)C2)COC(C)(C)C1 Cc1ccc(C(=O)NCCC2CC(NC(c3ccc(N)c(Cl)n3)=O)C2)c(=O)n1C Cc1cnc2nc(C(N3CC(O)(CN(C)C(C4(C)CC(C)(C)C4)=O)C3)=O)nn2c1 C1(CNC(C2CC(N(C)CC)C2)=O)CCC2CN(C(=O)Cc3scnc3C)CC12 CC(C(=O)N1CC2CC2(CNC(=O)CC2(Oc3ccccc3)CC2)C1)C(F)F C1(NC(CC2(C=C)CCC2)=O)CCN(C(C2(CCC)CCC2)=O)CCC1CO N1(C(CNC(C(C2CN(C(c3nccs3)=O)C2)OC)=O)C)CCOC1=O Cc1ccc(C(=O)NC2CC2CNC(c2ccc(Br)s2)=O)cc1CO c1(C(=O)NC(C(C)C)CNC(C23CCCC(C2)OC3)=O)ccc2c(c1)OCO2 c1(C(=O)NC2C(C)CCN(C(C3(CCF)CC3)=O)C2)cccc2nc(CO)[nH]c12 Cc1cc(C(=O)NC(C2CN(C(c3cc(Cl)no3)=O)C2)C)cc(O)n1 N1(C(C(=O)NC2COC(C(F)F)C2)=O)C2CCC1c1cc(F)ccc12 c1(C(N2CC(O)CC(NC(c3ncc(F)cc3F)=O)C2)=O)ccn2cnnc2c1 Cn1ncc(C(=O)N=c2cc(OC(F)F)n(C)[nH]2)c1S(N)(=O)=O Cc1c(CC(=O)NC(C)CN(C)C(C2C3CC4C(C3)C24)=O)cnn1C Cc1nc(CO)ncc1C(=O)NCC1(O)CCN(C(C2(C)C=CCC2)=O)C1 CC1CC(NC(=O)C=Cc2ccoc2)CN(C(=O)COCCc2ccccc2)C1 C1(NC(C(C)SC(C)C)=O)CN(C(c2ccnn2CCF)=O)Cc2nccn2C1 CCC(C)C(O)C(=O)NC(C)CN(C(=O)C(=O)NC1CC1)C CCC(F)(F)CC(=O)NCC1CC2(CC2)CN1C(=O)CC1CCCN(C)C1 c12cccc(c1)CNC2=O.N1(C(C(=O)NCC=C(C)C)=O)CCCCCC1 CC1CN(C(C2COC(=O)C2)=O)CC2(CCN(C(C3CCC3)=O)CC2)O1 N1(C(C(Cc2ccccc2)NC(C)=O)=O)C2CCCC1CC(N=[N+]=[N-])C2 C(=O)(CCCCc1cnc[nH]1)NC1C(CNC(c2c(C)occ2)=O)COC1 C1(NC(=O)NCCC(C(=O)OC)C)CCCN(c2ccccc2Cl)C1=O C1(C(=O)NC(C2N(C(CC3(C=C)CC3)=O)CCC2)C)CCC(N(C)C)CC1 C1(CNC(C(CCC)OCC)=O)CCC(C)(C)CN1C(=O)CCC(C)(C)C c1(C(N2CCC(CNC(COCCC)=O)C2(C)C)=O)cnc(O)c2cnccc12 N1(C(CS(CC)(=O)=O)=O)CCC2C(NC(C3(CC4CCC4)CC3)=O)C2CC1 C#CCC(CC(=O)N1CC=CCO1)NC(c1cnc(Cl)s1)=O n1(C(=O)N(CC2CC2)CC(=O)C(Cl)(Cl)Cl)ccnn1.c1(C)cccnc1.N12CCC(C1)C2 C1(NC(C2CCC(C)O2)=O)CCC2(C1)CN(C(C1CNC(=O)O1)=O)C2 c1(C(=O)NC(CNC(C(COC)NC(C)=O)=O)CC(C)C)cccc2ncnn12 N1(C(CC(C)Oc2ccccc2)=O)CCC(NC(=O)C(O)c2ccsc2)CC1 c1(C(C)NCCC)cncc(Br)c1C.n12nnnc1C2(C)CCOCC(=O)OC.C c1(C(N2CC(C)(C(=O)NCC)C(OC)C2)=O)cn(CCO)c(C)cc1=O S(=O)(=O)(c1cccnc1)N1CC(NC(c2sccc2Cl)=O)C2(C1)CC2 C1(CNC(CCC)=O)CC2(CCN(C(c3ccc(N)c(F)c3)=O)C2)CO1 C1(OC)CN(C(=O)C(c2cccnc2F)(C)C)CC1NC(c1nc(Cl)oc1C)=O C1(NC(CCOC(C)C)=O)CC(NC(=O)Cc2nc(C3CC3)n[nH]2)C(O)C1 C(C)(C)(C(=O)NCCN1CC2CC2C1)NC(C(C)c1ccco1)=O CC(c1ccccc1C)=CC(=O)N(C1CCCC(NC(C2CCC2)=O)C1)C C1(N(C(C(C2CC2)SC)=O)C)CCCCN(C(c2cncc(Cl)c2)=O)C1 N1(C(C(C=C)O)=O)CC2CCC(C1)C(NC(=O)C(c1ccc(Cl)cc1)C)C2 C1(NC(C(C)Oc2ccccc2)=O)C2CN(C(C3CC(C(F)F)C3)=O)CC12 c1(-c2ccc(-n3cc(CCC(C)(C)C#N)nn3)s2)c(F)cccc1F CC1CCCC(CCNC(=O)C=CCN(C)C(c2cc(CO)n(C)n2)=O)O1 CN=c1nc(NC(CN(C)C)C(C)C)[nH]c(=NCCc2cccnc2C)[nH]1 c1(C(N2CC(C)C(NC(C3CCCO3)=O)C2)=O)nc(S(N)(=O)=O)c2ccccn12 CC1(C)CCCC(CCNC(=O)CONC(c2cc[nH]c2C2CC2)=O)C1 c1(CC(N2CC(C)C(CNC(=O)CCS(C)(=O)=O)CC2)=O)cc(F)c(F)c(F)c1 C1(NC(=O)CCSc2ccccn2)CCCCC1NC(C1CC1C(F)(F)F)=O c1(OC)ccc(O)cc1C(=O)NC1(CCNC(=O)C(C)N=[N+]=[N-])CC1 c1(CNC2CCN(C(c3ccc(C)s3)=O)CC2O)c[nH]c2cccc(C)c12 c1(C(=O)NC(c2cn(C3CCCCC3O)nn2)(C)C)ccc(N)cc1Br N1(C(CCCSC)=O)CCC2(NC(=O)Cn3cccn3)CCCCC12 C12(C(=O)NCC=CCCC)CCC(CC1NC(=O)CC(C)F)C2 Cc1cc(C(=O)NCCCN(C(=O)CCC2CCC(=O)N2)C)c(C)n1C C(=O)(C#CC1CCC1)NCC1C(CNC(c2c(-c3n(C)ccn3)nn[nH]2)=O)C1 C(C(C)(O)C(C)C)NC(CC(C1CC1)NC(c1c(C)nco1)=O)=O c1(OC(=O)NCC2CC(OC(C)(C)C)C(O)C2)ccc(F)cc1O C1(F)(CNC(C(C)(F)F)=O)CCCN(C(=O)CCc2cnc(C3CC3)o2)C1 Cc1[nH]nc(C(N2CCCC(N(c3ccnc(N(C)C)c3)C)C2)=O)c1Cl CC1(C)CCC(O)(CNC(=O)C(C2CCC2)NC(C2CCCC2C2CC2)=O)C1 N1(C(C2CCC(=O)C2)=O)CCN(CC(=O)NC2CCC3(CC3)C2)CC1 c1(C(=O)NCCC(C)NC(c2cc(CCC)n(C)n2)=O)c(N)cc(OC)cc1F Cc1sc(N)c(C(=O)NC(C)C(C)NC(c2cccc(OCCOC)c2)=O)c1C N1(C(C(C(C)C)CNC(c2cccc(=O)o2)=O)=O)CCC(F)(F)C(O)C1 c1(C(N2C(C)C(NC(c3ccc(C(N)=O)o3)=O)CC2)=O)ccc(N)c(Cl)c1 C1(CCC(N2C(C(C)(C)OC)CCC2)=O)CCN(C(C2COCCO2)=O)CC1 c1(-c2cncc(CCC(=O)NCCO)c2)ccc(SCCCn2ccnc2)cc1 C(=O)(CC1=CCN(C(=O)CC(C)n2cccn2)CC1)N(CCC#C)C N1(C(c2ccc(OC)c(I)c2)=O)CCCC(C2CCCN(c3nnco3)C2)C1 c1(NCCN(C)C(c2coc(C3CCC3)n2)=O)cnc(C#N)cn1 N1(C(CC(=O)NC2CC2)=O)CCC(NC(=O)CC2CCCC2)C(F)C1 C12(C(N(C(C)C3CC3)C)=O)CCC(CN(C(c3cc[nH]c3C3CC3)=O)C1)C2 C(=O)(CCCCC(=O)OC)N1CC(C(NOCCC(C(CC)CC)O)=O)C2(C1)CC2 C12(CNC(c3cnc(C(F)F)s3)=O)CCC(NC(C34CCCCC3C4)=O)(CO1)C2 c1(C(=O)NCc2ncc(CC)s2)cccc(S(=O)(=O)NCCc2nc(O)n[nH]2)c1 Cc1cc(NC(C)CO)ncc1S(=O)(=O)N(C12CCC(CC1)CC2)C C1(CCC)CC(C(=O)NC2CCN(C(C3(C(C)C)CC3)=O)CC2)CCO1 c1(OC)cc(C(C)NC(=O)CC2CC2C(F)(F)F)ccc1OCC#N N1(C(c2sc3cc(C)sc3c2)=O)CCC(NC(=O)CN(C)C)C12CCCC2 N12CCC(O)(CC1)SCC2=O.C1(OC)CCC(CNC(=O)CCN2CCC2)CC1 C1(CCNC(CCNC(=O)NC)=O)C(C)CCCN1C(c1ccc([N+](=O)[O-])s1)=O C(C(CC)(CC)C(=O)N=c1ccn(C(F)F)[nH]1)NC(C=CCC)=O c1(C(=O)OC)c(NC(C2CN(Cc3ncccc3C)CCS2)=O)n[nH]c1C C1(CNC(COCCOCC#C)=O)(NC(c2cocn2)=O)CCC1 c1(C(=O)NC2CCC(N(C(c3cc(C)oc3)=O)C)C2)cc(Br)cnc1N c1(CNC(=O)CCc2ccccc2F)cc(Br)c(O)cc1O.C12CCCN1CC2 C(CCN(C(=O)CCc1ccccc1O)C)(C(C)C)NC(c1cnc(CC)s1)=O c1(C(=O)NCC2(C)CN(C(=O)CC3CCCOC3)CCO2)ccc2c(c1)OCC2 C(=O)(CCCCC#N)N(CC(C)NC(c1cn(C(C)(C)C)cn1)=O)C c1(C(=O)NC(CNC(c2cn(CC=C)nc2)=O)CO)c(C)[nH]c2ncccc12 c1(C(N2CCC(CC=C)(C(=O)NCC3(C(C)C)CC3)C2)=O)cc(C)ncc1C C#Cc1ccc(C(=O)NCC2OCCC2C(=O)NCCNC(=O)NC)o1 CC1(C)CN(C(c2ccc(Cl)c(O)c2)=O)C(CNC(C2CCNC2=O)=O)CO1 C1(c2n(CCCC)nc(-c3cccc(OC)c3F)n2)CC2CCCCC12 N1(C(c2ccc(C)s2)=O)CCC2C(CCN2Cc2cc(Br)cc(C)c2O)C1 c1(C(=O)NC2C(CCC)CN(C(=O)C(O)CN(C)C)C2)c(C)nn(CCC)c1C N1(C(=O)NCC(Cc2ccccc2)N(C)C)CCC(O)C(C)(CNS(C)(=O)=O)C1 C1(NC(c2cc(CS(C)(=O)=O)on2)=O)CCN(C(c2coc(O)n2)=O)C1C1CC1 c1(C(=O)NC(C2CN(C(=O)CN3CCCOC3=O)CCO2)C)cccc(Cl)c1F C(C)(C)(CCNC(c1ocnc1C)=O)NC(COCCOC)=O.C(C)(C)(C)OC(=O)C C#CC1(NC(=O)CC(C(C)NC(=O)CC2(O)CCOC2)SC)CCCCC1 N1(C(C)CC2CCCC2)CC(NC(=O)CCc2cccs2)CC2(CCOCC2)C1 Cc1ccc(CC(=O)N(CCCCCCCCF)C)cc1[N+](=O)[O-].C(C(=O)O)N Cc1nc(-c2cc[nH]n2)sc1NC(C1CCOC1CN)=O c1(OC)ccc(CC(C)C(=O)OCC2CC2c2cnn(C)c2)cc1 c1(-c2cc(C(=O)NC(C3CCCC3)(C)C)on2)ccc(Cl)cc1 C1(C(=O)OC)(C(=O)OC)CCOCC1.n12ccc(n1)CNC(=O)N(C)C1CC2C1 C(=O)(CC1=CCCC1)NC(C(C)NC(C(C1CCOCC1)OCC)=O)CO N1(C(C=C(C)CNC(c2c[nH]c(=N)o2)=O)=O)CCCC12CCNC2 CCC(C)C(C)C(=O)NC1C2CN(c3cc(O)nc(C)n3)CC12 C(=O)(C(C1=CCCSC1)N1CCNS(=O)(=O)CC1)NC(C)C Cc1cc(C(=O)NC(C2CCCN2C(=O)C2=CCCS2)C)c(C)cc1Cl Nc1cc(F)cc(C(=O)NC2CCCN(C(=O)CC=C(Cl)Cl)CC2)c1F N1(Cc2cccc(-n3ccc(C)n3)c2)CC(O)(C2(CN(C)C)CC2)C1 N1(C(c2sc3ncn(C)c3c2)=O)CCOC2(CCN(C(C3CCCS3)=O)CC2)C1 c1(C(=O)NC(C(C)C)C(C)NC(c2csnc2Cl)=O)cc(S(N)(=O)=O)co1 C#CCC(C)(C)C(=O)N1CCCC1CNC(C1CCC2(CCC2)C1)=O C1(C(=O)OCC)CC2(CC2)CN1C(=O)C(=O)Nc1cnc(Oc2ccccc2)s1 C=CC(C)(CC)C(=O)NCC(F)CNC(=O)CCCOc1ccccc1F c1(SCCC)ccc(C(=O)NC(CN(C(=O)Cc2cnccc2C)C)CC)cc1 C1(C(N2CC3(C2)CN(C(C24CCCC2CCC4)=O)C3)=O)CCCNS1(=O)=O C(=O)(C(C)S(N)(=O)=O)NC(CN(C(=O)CCc1ccc(OC)c(Cl)c1)CC)C N1(C(C(C2CC2)OCC)=O)CCCC1(C(=O)N(C(CC)C1CC1)C)CC c1(C(CC)=O)ccc(OCC(=O)NC2CC(NC(=O)C=C3CCC3)C2)cc1 C1(C(=O)NCc2cc(C)on2)CN(C(C2CNC(=O)CN2)=O)C(C)(C)CO1.C(C)(C)(C)O c1(C(N2CCN(C(CC3CC(C)C3)=O)CC(O)C2)=O)cc2c(nn1)CCCC2 C(=O)(CCCCCNC(C1CCN(C)C1)=O)NC(c1nncs1)C C(=O)(CCCCCCCC1CC1)N1CCC(NC(CC2CCN(C)C2)=O)C1 c1(C(=O)NCC(C(=O)N2CCC2C2CCCC2)N(C)C)ncncc1N C1(NC(C2CCCN(CCC)C2)=O)CC2(CCC(NC(=O)CC(C)(C)C)CC2)C1 C(C(CC(C)C)C(=O)NC1CCN(C(c2coc3c2COC3)=O)C(C)C1)OC c1(C2c3nnnn32)ccc(C)c(Br)c1.C1(N(CCC)CC2CC2)COC1.C1CS1 c1(NC(C2CC(C)C2)=O)cn(C)c(CN2CCOCC2)n1.c12ccc(cc1)SC2 C1(NC(c2ncn(C(C)C)c2)=O)CCN(C(=O)CCCC#N)C(C2CC2)C1 C1(C)(CC)C=C(C(=O)NCCCCC(C)NC(c2nnc(C3CC3)s2)=O)C1 c12ccncc1OC2.c1(OC)cc(C(=O)NC2CCC2)[nH]n1.C(=O)NCC1CC1.C(C)O Cn1cc2cc(C(=O)NC3CCC(NC(C4(c5ccon5)CC4)=O)C3)ccc2n1 c1(OCC)nc(Br)cnc1NC(C1CCC(CNC(c2nc(Cl)sc2Cl)=O)CC1)=O c1(C(=O)NCCN(C(C2CCC(C)CC2)=O)C)cnn2cc[nH]c(=O)c12 c1(C(N2CC(CNC(C3N(C)C(=O)NC3)=O)C2)=O)cn2ccccc2n1 C1(C(N2CC(C)(NC(Cn3cc(C)c(C(F)(F)F)n3)=O)C2)=O)CCCCC(=O)N1 c1(CC(=O)NCC(CNC(C2CC(CCC)C2)=O)OC)ccccc1 C#Cc1cc(F)c(C(=O)NC(C)CN(C(=O)CCC(C)(C)F)C)c(F)c1 C1(C(=O)NC2(CN(C)C(c3ncccc3OCF)=O)CC2)C2CCC(=O)C12 C(CCC(C)C(=O)NCC1CCCN(C(c2nncs2)=O)CC1)OC N1(C(c2ccc(C(=O)NC)o2)C(=O)NCC)CCN(CC2CCCCC2)C(C)C1 C(=O)(C(C)(C)CC(C)(C)C)N1CC(NC(CCC#C)=O)C(O)C1 Cc1ccc(-n2cc(-c3ccccc3I)nn2)cc1.O(CO)CC(=O)O c1(C(=O)NCC(CNC(C2CCC(=C)CC2)=O)C)ccc(N)c(C)c1F CC(C)(C)CC(O)CC(=O)N1CCCC1CN(C(C1(C2CC2)CC=CC1)=O)C1CC1 CCC(CC)(CC(=O)OC)C(=O)N1CC(C2(NC(c3nc(Cl)sc3C)=O)CC2)C1 CC1CCCCC1(C)C(=O)NCCCCC(=O)N(C)CCc1ccccc1 C12(NC(c3ccn(CCOC)n3)=O)CC3CC(C1)CC(NC(=O)CSC)(C3)C2 C12(O)CCN(C1)C(=O)CC2.c1(C(CC)(C)NC(N2CCCCC2)=O)noc(C)n1 c1(C(=O)NCC2CC3(CN(C(c4c(C)con4)=O)C3)C2)coc2c(C)cccc12 c1(OC)cc2c(cc1CN(C)C(c1ccc3c(n1)CCC3)=O)OC(C)C2 c1(CN2CC(C)SCC2)c(F)cc(Br)cc1Cl C(CC(CC)C(=O)NC12CC(C(=O)NCC3OC(=O)CC3(C)C)(C1)C2)=CC C1(O)(CC)CCN(C(c2cc(CNC(C3CC3c3ccco3)=O)on2)=O)C1 C1(CNC(c2ccc(C#C)cc2)=O)CN(C(C2(O)CCOC2)=O)CC2(CCC2)O1 S(=O)(=O)(c1cc([N+](=O)[O-])ccc1C#N)NC1CCC(c2n(C)ccn2)C1 N1(C(C2(C(C)(F)F)CCC2)=O)CCCC(CNC(=O)CCCc2ncco2)C1 c1(OC)cc(OC)c(C(C(=O)NCC(=O)C2CC2)SC)c(OC)c1 Cc1nc(C(=O)N(CC(O)CN(C)C(C2CC=CCO2)=O)C)[nH]c1C CC1ON=C(C(=O)NCC2CC(F)(CNC(c3cc(Cl)c(Cl)n3C)=O)C2)C1C C(C)(C(C)(C)C(=O)NC(C1CCCO1)CO)NC(C(C)n1cnnn1)=O c1(C(=O)NCC(C)NC(=O)CCc2ccsc2)cc(F)cc([N+](=O)[O-])c1 c1(C(=O)NCC2C(NC(CCCCC)=O)C2)coc(S(=O)(=O)N2CCOCC2)c1 c1(NC(c2c(CNC(c3ccncn3)=O)cc[nH]2)=O)ncccc1C(F)F Cc1nc(C(N2CCC(N(C(=O)CCCc3n[nH]c(=N)s3)C)C2)=O)nn1C c1(OC)ccc(C(=O)NC2CC2C(=O)OC)cn1.C1(CNC(=O)COC)CCC1 N1(C(c2cnc(OC)c(Cl)c2)C(=O)NC2CC2)CCC2(CCC(OC)CC2)CC1 C(=O)(CCP(C)(C)=O)N(CCCCN(C(C(CC)OC1CCCC1)=O)C)C C#Cc1ccnc(C(=O)NC2CCN(C(C3CN4CCC3CC4)=O)C23CC3)c1 Cc1noc(C)c1C=CC(=O)NC1CC2(C1)CN(C(=O)CCc1cnco1)C2 CCCCC(CC)C(=O)NCCCN(C(=O)C(C)NS(=O)(=O)c1cccs1)C1CC1 C12(NC(C=CC)=O)COCCC1CN(C(=O)Cc1ccc(F)c(CSC)c1)C2 N1(C(c2c(F)ccnc2Cl)=O)CC2CC(C1)CN(C(c1ccc(O)cc1F)=O)C2 CN1CCN(C(=O)CCNC(C2CCC2)=O)C(CNC(=O)C=C(C2CC2)C2CC2)C1 CC(O)C(C(=O)NC(CN(C(=O)CC(=O)OC(C)(C)C)C)(CO)CO)N(C)C C1(CNC(C(C)OC)=O)CN(CCc2ccc(Cl)cc2Cl)CCC1(C)C C#Cc1cccc(CC(=O)N(CC(=O)NCCN2CCC3CC23)C(C)C)c1 n1(CC(C)C)ccc(C(=O)NC2(CNC(=O)CCc3ccccn3)CCOC2)n1 N1(C(CC2(C=C)CC2)=O)CC2CCC(NC(c3ccccc3SC)=O)CC2C1 N1(C(C(C=C)OC)=O)CCC2(CC1)CN(C(=O)C(C)CCCC(C)C)C2 c1(C(=O)NC2CCC(NC(=O)C=CC3CCCC3)C2)nc(C2CC2)ncc1Cl c1(C(N2CC(F)(CNC(C(C)NC(C)=O)=O)C2)=O)cc(-c2ccccc2)ccn1 C1(NC(C(CC)OC)=O)CCCCC1NC(C1(F)CCCCC1)=O CN1C(=O)N(CCC2(CN)CC2)C(=O)C1c1ccc(N2CCCS2(=O)=O)cc1 C12COCCN(C1)C(=O)COC(Oc1c(C)c[nH]n1)OC2.C1(OCC)CCCS1(=O)=O N=c1nc(N2CCOC(SCC3CSC3)C2)[nH]c(CO)n1 C1(CNC(c2ccon2)=O)CC2CC1CN2C(C1CN2CCC1CC2)=O c1(C(=O)NC2CC2C(=O)Nc2ccc(F)c(Br)c2)cc(O)nc(Cl)c1 N1(CC)CCCCC1C(=O)N(C(C)CCNC(=O)CSCc1cccs1)C C1(C(=O)NCCNC(c2n[nH]c(C)c2F)=O)CCc2c(n[nH]c2C)C1 C1(C(N2CCCCC(N(C)C(C3CC(C#N)C3)=O)C2)=O)CCCN(S(N)(=O)=O)C1 c1(C(=O)NCC2CCCN(C(CC3C(C)=NOC3=O)=O)C2)cn2cccnc2n1 c1(C(=O)NCc2scc(CNC(CS(N)(=O)=O)=O)n2)cc2n(n1)CCNC2=O C1(C(N(CCN(CC)CC)C)=O)CCN(C(=O)CC2CC=CCC2)CC1(C)C CN1CCOC(C(=O)NCCC(O)CNC(=O)CCc2cncs2)C1 c1(CNC(CCC(OC)OC)C)ccc2c(c1)CCOC2 N1(C(C2(F)CCN(C(C(C)OC(C)C)=O)CC2)=O)CCCN(C)C(=O)C1 N1(C(C=CCC)=O)CCC2CC12C(N1CCCCC1CC(N)=O)=O C1(NC(Cc2ccc(OC(C)C)cc2)=O)CN(C(=O)C(=O)N2CCC2)CCC1C C(=O)(n1ccc(CNC(=O)Nc2ccc(OC3CC3)nc2)n1)OC(C)(C)C S(=O)(=O)(c1cccc2nccnc12)N1CC(C(=O)Nc2cncnc2)SCC1 N1(C(C(C)(C)OCC)=O)CCC2(CC1)COCC(CNC(=O)C(C)(C)N(C)C)O2 N1(c2ncc(C(=O)NC3CC3c3cc(C)c(Cl)cc3)cn2)CCc2ccccc21 C12(CC=CCC1)C(=O)C2.c1(N)cccc(CC2CC2(C)C)c1.N1(CC(=O)OC)CCOCC1.C C1(NC(=O)COc2ccc(Cl)cc2)CC1C1CCN(C(c2cnn[nH]2)=O)CC1 C(=O)(C(C)(C)CCCNC(c1coc(CC)c1)=O)NC1CCCC(C#C)C1 c1(C(N(C)Cc2ccc(CO)o2)=O)cccc(CNC=O)c1.C1(=O)CN1 c1(CC)cc(C(=O)NCCOCCCNC(C2(COC)CCCO2)=O)on1 c1(C(N2CCC(C(=O)NCC(C)C)CC2)=O)cc(C(F)(F)F)ccc1F c1(C(N2C(NCC=C)CCC2)C(=O)NCCCC)ccc2c(c1)C(C)C(C)O2 c1(C(=O)NC(C)CC2CN(C(C3CCCO3)=O)C2)c(O)nnc2c1CCCC2 N(C1CCc2c(Cl)cccc21)C(=O)NC1(C(F)(F)F)CCOC1 c1(C(c2n(CC)nnn2)NCCc2ccsc2)nc(C)ccc1F N1(C(CC(C)C)=O)CC2CCC(C1)C(NC(c1cc(OC(F)F)ccc1F)=O)C2 c1(NC(N2CC(CCCCNC(=O)CCc3cnoc3)C2)=O)cccnc1 C1(C(=O)NC(COCC)C(=O)NCc2[nH]nnc2C)CCCCN1CC c1(OCC(CNC(=O)Cc2ccc(N3CCOCC3)cc2)O)ccc(Cl)c(Cl)c1 c1(C(=O)NCC2CC(NC(=O)CCCn3cccn3)C2)cccc2cnsc12 C(CCCC(C)(C)C(=O)NNC(=O)CSC)NC(c1cncc(C(=O)OC)c1)=O c1(C(=O)NCCN(CCOC)Cc2ccc(Cl)cc2)ccc2c(c1)NCC2 C(=O)(C1=C(Cl)CCCC1)NC1(COC)CCN(C(=O)CC2COCCO2)CC1 C12(C(N3CCC(CCNC(c4ccc(CO)nc4)=O)C3)=O)CCOCC1C2 C1(NC(c2cc3ccoc3cc2F)=O)COC2(CCCN(C(=O)C3CC3)C2)C1 C1(C(=O)NCC(C)(C2CC2)NC(c2nncn2C2CC2)=O)CCCC12OCCO2 N1(C(c2ccc(OCC)c(C)c2)=O)CCCC2CCN(C(=O)C=C(Cl)Cl)CC12 N1(C(CCC=CC)=O)C(CNC(=O)CC(C(F)(F)F)OC)CC2CCCCC12 c1(CN2C(CNC(c3ccc(C)cc3)=O)C=CC2)c[nH]c2nccc(Cl)c12 CCC(C)CC(=O)C(=O)N1C(C(=O)NC2CCCC(C(=O)OC)C2)CC1C N1(C(CN(C)CC)=O)CC(C(=O)Nc2cncc(C)c2)CCC1C c1(C(=O)NC(CNC(C(C)SC)=O)C2CCC2)ccc(F)cc1OC(F)F c1(C(=O)NCC(CC)NC(C2(C3CC3)CCCO2)=O)cncc(Br)c1 C1(C)(C(N2CCC(OCCNC(c3c(CC)scc3)=O)C2)=O)CC(C)=NO1 N1(C(C(C)C2CCC2)=O)CCC(C)(C(=O)NCc2cc(C3CC3)n[nH]2)CC1 Cc1cccc(C2CCCCC2C(=O)N(CC(N2CCN(C(N)=O)CC2)=O)C)c1 C1(CCOC(F)F)(O)CCC12CCC2.c1(CN)ccc(-n2cncn2)cc1 N1(C(C(C)(CO)NC(c2nncs2)=O)=O)CCCC(C)(O)C1 C1(O)(C(C)NC(C2(C)CC=CC2)=O)CN(C(C2CC3CC3C2)=O)C1 N1(C(CCNC(=O)NC)=O)CCC2(NC(C3OCCCO3)=O)CCCC12 c1(C(=O)NCCC2CC(NC(C3C(C)(COC)C3)=O)C2)sc2sccc2c1Cl C12(NC(c3nn(C)c(Cl)c3)=O)CCCC1N(C(c1cocn1)=O)CC2 N1(C(CC2N(C(c3ccc(C(C)C)o3)=O)CC2)=O)CCc2ccccc2C1 C(CNC(=O)C(C)n1cncn1)(CC(=O)Nc1cnc(C(C)C)nc1)OC c1(C(=O)NCC2N(C(Cc3c(C)non3)=O)CC2)ccc(=O)n(CC(C)O)c1 CCC(C)(C(=O)NCC(CNC(c1cc(C)c(C(F)F)c(C)c1)=O)CO)C(N)=O C1(C(N2CCCC(C)(CNC(C3(C)CC=CCO3)=O)C2)=O)CCc2nnnn2C1 C#Cc1ccnc(C(=O)N(C)CCN(C)C(C2(c3ccncc3)CC2)=O)c1 N1(CC(=O)NC2C3CN(C(C(=O)NCCOC)=O)CC32)CCc2c(O)n[nH]c2C1 CCCC(C#N)C(=O)N1CCC(c2ccccc2)(NC(=O)Cc2ccon2)CC1 c1(SCc2cn(C3C(C(=O)OC(C)(C)C)CCCC3)nn2)cc(Cl)ncc1N c1(N(C2(COCC)CCC2)C)nc2ncn(C)c2c(=NCC2(F)CCOC2)[nH]1 C(=O)(C(C(C)(C)C)C1CCC1)C1C(c2cnc(C)s2)C1.N12CCC(C1)C2=O N1(C(=O)NC2CCN(C(c3ccccc3)=O)CC2)CCc2c[nH]nc2C1 C1(C(N2CC(NC(C(C)NC(CC)=O)=O)C2)=O)CCC(C)CC1 c1(C(=O)NCC2C(NC(c3c(C)scn3)=O)CC2)sc(C)c(Br)c1C c1(CN(C(=O)CN(C2CC2)C)C)cccnc1.c1(C(=O)N)cccs1 c1(N2CC3CC(NC(C(C)CO)=O)CC3C2)nc(Cl)nc2sccc12 Cc1c(F)ccc(C(=O)N(C2CN(C(=O)Cc3cnc[nH]3)CC23CC3)C)c1F c1(C(=O)NC(CCCC)CNC(=O)C(C(C)C)NC(C)=O)cn2cccnc2n1 c1(NCC)c(NC2(CC(=O)Nc3cn(CCC)nc3)CCC2)cccc1C N1(C(COCc2onc(COC)n2)=O)CC2CC1C2NC(C1CCC(=O)N1)=O C(=O)(C(C(C)O)NC1CCN1C(C1CCN1C(C)(C)C)=O)OC C(c1ccccc1Cl)=CC(=O)NC1(C)CCN(C(C2CN(S(N)(=O)=O)C2)=O)C1 C1(CNC(C(c2cccnc2)C)=O)CCC(C)(C)CN1C(c1ccncc1F)=O c1(CC)cccc(CC)c1Cc1nc(C2(C(C)C)CCCC2)on1 N1(C(CC2COCC(C)O2)=O)CCC(NC(=O)CNC(c2ccsc2)=O)C(O)C1 n1(CCC#N)cccc(NCC2C3CCCC23)c1=O c1(N2CCCC(C(=O)NC)C2)nc2c(c(=NC(C)c3cc(C)oc3C)[nH]1)COC2 c1(N(C)Cc2c(C)ccs2)nc(N(C)CCC2CCCO2)nc2c1CC(C)CC2 c1(C(N(C(C)C(=O)NOCCOC)CC)=O)cc2ncccc2[nH]1 N1(C(=O)NC(C2(O)CC2)C)CCOC(C)(C(C)(C)C)C1 Cc1coc(C(=O)NCC2COC(CNC(c3cnc(NC4CC4)s3)=O)C2)c1 c1(CC(=O)NC2CC(CNC(C(c3c(C)nn(C)c3)C)=O)C2)ccc(C#N)nc1 Cc1c(CC(=O)NCCCCC(=O)N2CCC(N(C)C)CC2)ncn1C C(C(C)(C)C(=O)NCC1CCN(C(=O)C=Cc2cocn2)C1)N(C)C C1(N(C(CC=CC=C)=O)C)CCCN(C(=O)CCNC(=O)NC)CC1 c1(C(N2C(C)C3CC2C3NC(C2CCC2)=O)=O)ccnc(P(C)(C)=O)c1 C1(C(N2C(CNC(c3[nH]cc(C(N)=O)c3)=O)CCC2)=O)NC(=O)C2CC12 C1(CNC(N2C(c3ccc(C)s3)CCC2)=O)CC12CCSCC2 c1(CN2C(C)CCC(NC(C3CCS(=O)(=O)C3)=O)C2)ccc(C#N)c(Cl)c1 c1(C(=O)NCC2(NC(c3ncc[nH]3)=O)C(C)CCCC2)cc(F)cc2ccoc12 C(CCC(=O)N1CCCC1C(C)(C)NC(=O)Cc1cccs1)=CCC=C C1(C(N2CC(OC)C(NC(c3cc(CC4CC4)on3)=O)C2)=O)CCCC1C1CC1 Cc1nn(-c2ccccc2)c(Cl)c1C(=O)N(c1cc(C#N)cs1)C C1(NC(CCc2cc(C)no2)=O)CCCC(N(C(=O)C(=O)N(C)C)C)C1 CN=c1ccc(C(N2CCC=C(C(=O)N(CC(CC)OC)C)C2)=O)c[nH]1 N1(C(c2sc(C)c(O)n2)=O)CC2CCC(NC(c3ccsc3)=O)CC2C1 C(=O)(C1COc2ccc(Cl)cc21)NCC1CCN(C(CCC=C(C)C)=O)CC1C C1(O)(CN(CCC(C)C)C(=O)NC)CN(N2CC(C)C2)C1.c1(C=O)cn(C)cn1 Cc1ccc(Cl)c(C(=O)N(C(C)CNC(c2nc3sccn3c2C)=O)C)c1N C(=O)(CC(C(F)F)NC(C1C2CCCC12)=O)N1C(C(C)C)C(C)(C)C1 C(=O)(C1=NOC(CNC(=O)CC2CSCCO2)C1)N(CC)Cc1ccc(O)cc1 c1(CCn2cc(CNC(c3cccc(C)n3)COC)nn2)nc2ccccc2s1 c1(C(=O)NCC(C)(C2CC2)NC(C2CC(OC)C2)=O)c(C2CC2)nc2sccn12 CN1CCCC12CCN(C(=O)C(=O)Nc1ccc(N(C)C(N)=O)cc1)CC2 N1(CC(=O)NC(CNC(C(c2ccccc2)SC)=O)C)CCN(C)C(=O)C1 CC(C)(CC(=O)N1CCCCC1CF)NC(=O)Cc1cccc(F)c1 N1(C(c2c(C)c[nH]n2)=O)CCCC(O)(CN=c2[nH]nc(C(F)F)s2)C1 c1(C(N2C(CN(C(c3cnccn3)=O)C3CC3)CCC2)=O)cnnc(O)c1 Cc1cc(C(=O)NC2CC(F)(CNC(c3csc(O)n3)=O)C2)cs1 C1(C(N(C2CCCCN(C(c3cn[nH]c3)=O)C2)C)=O)Cc2cc(F)ccc2O1 C1(CC(=O)NCCN(C(=O)CNC(C2CCCCC2)=O)CCC)CC2(CC2)CO1 Cc1cc(Cl)c(NC(=O)N(C)Cc2cn(C)nc2C)cc1Cl c1(C(=O)NC(C)CCN(C)C(C2(CC(F)(F)F)CC2)=O)cc(F)c(F)c(F)c1F C(c1ccncc1)=C(C)C(=O)NC1CCCN(C(=O)CN2CCSCC2)C1 N1(C(N2CCCN(CCc3cccs3)CC2)=O)CCCC1C1CCCO1 Cc1nc2c(N3CCC(C(C)NC(C4CC(C)CC(C)C4)=O)C3)ncnc2s1 C1(CCN(C)C)CCN(C(=O)C(=O)N(n2cccn2)C)C1 c1(OC)cccc(-n2cc(-c3cccc(Oc4cc(Br)cn4C)c3)nn2)c1F Cc1cc(C(=O)NCC(C)CNC(=O)CC2CCC3CC23)cc(N)c1O Cc1nn(C)c(C)c1CC(C)C(=O)NC1CC1CNC(C12CCCC1C2)=O C1(C(=O)NC(CCCC)CNC(=O)CC2(C)CC2)CCCCCCC1 C(CCN=c1nc(N2CCCC(F)C2)c2c([nH]1)COC2)OCCC(C)C Cc1c(C(N2CC3CC3(NC(=O)C(F)CC3CCOC3)C2)=O)cnn1CCC#N C1(CCNC(C(CCC)OC)=O)CN(C(c2ncccc2N)=O)CCS1(=O)=O N1(C(CCCNC(C(C)n2cccn2)=O)=O)CCOCCC1C1CC1 N1(C(c2c(C)nn[nH]2)=O)CCN(C(c2ccn3cccc3c2)=O)CCC1C N1(C(C=CCCC)=O)CC(C)(C)CC1CNC(c1ccc[nH]1)=O C1(O)(CNC(C(C)(C)c2cscc2Cl)=O)CCCN(C(c2ccc(F)cc2)=O)C1 c1(C(N2C3CN(C(=O)Cc4cccc(Cl)c4)CC32)=O)c(O)ccc(Br)c1O c1(C(=O)NC(COCC)C(=O)N2CC=CC2CF)ncc(F)cc1N CC1CN(C(=O)CCCn2cccc2)CC1(C)CNC(c1nc(C2CC2)cs1)=O c1(C(=O)NCC(C)N(C(=O)Cc2cn3ccsc3n2)C)ccn2ccccc12 C1(CC)C(NC(c2cnc(C)s2)=O)CCN1C(=O)Cc1cncn1C c1(C(N2CCC(C)(NC(c3conc3C3CC3)=O)CC2)=O)cccc2c1CCO2 C1(C(=O)NC(CO)CCOC)(NC(C2CCN(C(=O)NC)CC2)=O)CCCCC1 C1(O)(C(C)NC(=O)CNC=O)CCN(C(=O)CCc2cncc(O)c2)CC1 c1(CNC(c2cc(C)[nH]n2)=O)cccc(CNC(=O)COC(=O)CO)c1 N1(C(c2ccc(CCC)[nH]2)=O)CCC(N(C(=O)C(C(C)C)n2cncn2)C)CC1 C1(C(N2CCCC(NC(c3c(C)csc3)=O)CC2)=O)CCC2(C1)CC2(F)F C1(NC(CCOCCC)=O)CC(CNC(c2ccnn2C(C)C)=O)CC1O c1(N2CCC(N(C(=O)C=CC=C(Cl)Cl)C)C2)ncncc1I Cc1nc(CC(=O)NC(C)(C)C(C)N(C(=O)CN(C2CCC2)C)CCO)cs1 C1(CNC(C(C2CCCC2)N(C)C)=O)CC2CC2N1C(=O)COc1ccsn1 N1(C(COCCSC)=O)CCC(F)CC1C(=O)NC(c1cccc(O)c1)C CC1C(N(C(C2CC(NC(=O)CCNC(=O)CO)CCO2)=O)C(N)=O)CCCC1C c1(OC)cc(CCC(N2CC3CC3(CNC(=O)C(C)OC)C2)=O)ccc1Cl CCCCCCCCC(=O)N1CCCC1C(N1CC(C)N(C)C(C)C1)=O C(C)(C)(CCCO)NC(c1cc(CNC(CC=CCC)=O)[nH]n1)=O CS(=O)c1ccc(CC(=O)NCC2CC2NC(c2cccc3nncn23)=O)cc1 C1(C)(C(=O)NC(C(C)C)CNC(C2(Cl)CC23CCC3)=O)CCC(C)(C)CC1 c1(C(N(C2CCN(C(=O)CC3(CC)CC3)C2)CC)=O)cn(CCC(C)C)nn1 N(C1CCCc2c1cnn2C1CC1)C(Cn1c(C)cc(C(=O)O)n1)=O c1(C(=O)NC2CC(CNC(COC3(C)CCOCC3)=O)C2)c(N)cc(F)cc1F C1(NC(C2CCN(C(C)(C)CCCl)C2)=O)CCOCC1n1cc(CCO)nn1 C1(C(=O)NC2CCCCC2C(F)(F)F)C2Cc3cc(Br)ccc3C12 c1(C(N2C(CC)CN(C(c3cc[nH]n3)=O)CC2)=O)cc(Br)cn(C2CC2)c1=O C1(C(N(c2cccc(O)c2)CC)=O)COCCN(C(=O)CCC2CCCO2)C1 CC1CCN(C(C2CCCCS2)=O)C(C)C1NC(c1nonc1N)=O N1(C(C=C(C)C)=O)CCCCC(NC(c2cc(C3CC(F)(F)C3)[nH]n2)=O)C1 CCC(F)(F)CC(=O)N1CCC(NC(c2cccc(C(F)(F)F)n2)=O)CC1C c1(CNC(C(C)OC(C(c2cnn(C)c2)C)=O)=O)cc2c(s1)CCC2 C12(C(=O)NCCCN(C(c3n(C)nc(C4CC4)c3)=O)C3CC3)OCCCC1C2(F)F C1(O)(C(C)NC(CC=C)=O)CCN(C(=O)CS(N)(=O)=O)CC1 N1(C(C2(C)CCN(C)C2=O)=O)CCC2(CC1)CC2CNC(c1n[nH]cc1Cl)=O c1(OC)cccc(F)c1CN1CCC(NC(=O)C2=C(C)OCC2)CC1 Cc1cc(C(=O)NCC2CN(C(=O)CC3CN(C)C3)CC2O)oc1C c1(CC(=O)NC(C)CCCNC(C2CC(=C3CC3)C2)=O)cccc(SC2CC2)c1 Cn1nc(C(=O)NCC(C)(O)CNC(C2CC3CC3C2)=O)cc1[N+](=O)[O-] C(CN=c1ccc(C(C)(C)C)c[nH]1)NC(=O)NCC(Cc1cccc(C)c1)OC c1(C(N2CC(CNC(=O)C=CC3CC3)C(O)C2)=O)ccc(Br)c(F)c1F c1(C(N2CC(CNC(CC(=C)C)=O)C(C)C2)=O)cc(Cl)cc2c1OCC2 c1(CNC(CN(C(C2CC(n3ccnc3)C2)=O)CC)=O)ccnn1C c1(C(=O)NCC(C)NC(CCN(CC(F)(F)F)CC)=O)nsc2ccccc12 c12nnnn1C2.c1(CNC(c2nccn2-c2ccccc2)C)ccccc1 c1(CC)nc(C)ncc1C(=O)NCC(C)CN(C(=O)Cc1ccc(F)cc1Cl)C N(C1CCN(CC)c2ccccc21)C(C(CCC)C)c1nnnn1C1CC1 C1(C(=O)OC)(CNC(c2ccon2)=O)CN(C(=O)OC(C)(C)C)C1 CC1CN(C(=O)Cn2ccnn2)CC(C)N1C(=O)Cc1ccc2c(c1)CC2 N1(C(C2CCCC(OCC)C2)=O)CCC2C(C(=O)OC(C)(C)C)CC12 CC1CCCC(C(N2CC(OCCC(=O)NC3CCCCC3C#N)C2)=O)CC1 c1(C(C)C(F)(F)F)ccccc1C(=O)NC(CO)C(C)NC(C1CC1C(F)F)=O N1(C(c2nn(C)c(Br)c2)=O)CCC2CN(C(=O)Cc3cccc(F)c3)CC12 c1(C(=O)OCC(=O)NC(C(=O)OC(C)(C)C)C2CC2C(=O)O)ccc2c(n1)CCC2 N1(C(C2N(C)C(=O)CC2)=O)CCCC(NC(c2csc([N+](=O)[O-])c2)=O)CCC1 C1(CC)(NC(=O)NC2CN(C(=O)CC3CCCCC3)CC2O)CCOCC1 N1(C(C2CCN(C(C)=O)C2)=O)CCC2(NC(=O)C3=COCCC3)CCCCCC12 Cc1c(C2CC(Cc3ccccc3)N(Cc3cccs3)C2)cnn1C c1(C(=O)NC2(C)CC(NC(c3ccsc3C(F)F)=O)C2)ccc(O)nn1 c1(C(=O)NCCCC2(NC(=O)CC3CC3)CC2)cccc(F)c1 c1(C(=O)NC2(CC=C)CN(C(c3cn(CCOC)nc3C)=O)C2)nccnc1C Cc1nc(SCC(=O)N(CCCNC(=O)CSC(C)C)CCO)n[nH]1 C1(C)(C(=O)NC2(C)CN(C(CC3CC(C)(C(=O)OC)C3)=O)C2)CCCC1(F)F C1(C(=O)OC)(CNC(=O)CC2CCN2C(=O)C=C(C)C(C)C)CCC1 C1(C2CCN(C(c3cnn4cc[nH]c34)=O)CC2)(NC(c2ccc(C)nn2)=O)CC1 C1(C(CC)C)CCN(C(=O)COCCNC(c2ncccc2O)=O)CC1 c1(C(=O)OC)cccc(C(N2CC(NC(C3CCS(=O)CC3)=O)C(C)C2)=O)c1 Cc1ccc(CCC(=O)NC2CC(F)(CNC(C3CCCC(C)C3)=O)C2)cc1C c1(C(=O)NC(C(C)C)(C)CNC(C2(c3ccnn3C)CC2)=O)cc(F)cc(Cl)c1 CC(C)C(C(=O)NCc1ccc(F)nc1F)C(C)NC(c1ncccn1)=O C1(NC(CN(C)CC)=O)CCC(C)(CNC(c2ccc(SCC(N)=O)cc2)=O)C1 C(=O)(CN=S(C)(C)=O)N(C(CCNC(C1(NC(C)=O)CCCC1)=O)C)C c1(C(N2CC(C(C)NC(CC(C)OC)=O)C2)=O)csc2cncn12 c1(C(=O)NCC(CNC(c2cc(Cl)c[nH]2)=O)F)c(F)ccc2ccncc12 c1(C(=O)NC2C(NC(CNC(CC)=O)=O)CCC2)c(O)cc(=O)n2c1COCC2 n1(CC)c(NC(C2CCCCN2C(C2CCC(C)O2)=O)=O)nc2cc(Cl)ccc12 CP(C)(=O)c1ccc(C(=O)NC2COCCN(C(=O)COc3cn[nH]c3)C2)o1 c1(C(=O)NC2CCCC(NC(c3cc(C#N)[nH]c3)=O)C2)ccc(F)c2occc12 c1(CNCc2c(C)ccc(OCC(F)(F)F)n2)nc2cc(Br)ccc2o1 c1(CCC=C)cn(C)nc1C(=O)OCC.N12CC(C1)NC(=O)C2=O N1(C(c2cnc(OC)c(C)n2)=O)CCCC12CCCN(C(c1cc(C)ns1)=O)C2 CCC(C)C(O)CNC(c1cc(CNC(C2(C(C)=O)CC2)=O)ccn1)=O c1(C(N(CCN(C)Cc2c(C)ccnc2Cl)C)=O)cc2ccccc2o1 c1(C(=O)NCC2(CCNC(CC3(C(=C)F)CCC3)=O)CC2)cc(N)c(Cl)cn1 CC1CC(C(N2CCCC2CN(C(=O)CCCCc2ccccc2)C)=O)C1(C)C C(=O)(CCCCN(C)C)NCc1scc(C(N(CC(CC)C)C)=O)n1 CCCC(C(=O)N1CCC(OCCN)CC1)NC(C)=O.N1(C=O)CSCCSC1 c1(NC(c2c(NC(C)=O)cccc2F)=O)c(-c2ccc(I)cc2)ccc2c1OCO2 Cn1cc(Cl)c(CC(=O)Nc2nc(C3CCCNC3)cs2)n1 c1(C(=O)NC2(C)CC(NC(c3c(CC)csc3)=O)C2)cc2ccsc2s1 C1(O)(CN=[N+]=[N-])CCN(C(c2cccc(C(O)C(OC)=O)c2)=O)C1 c1(C(N2C(C(=O)NC(CC)C)CN(C)C2=O)=O)ccc([N+](=O)[O-])cc1OC C(=O)(C(C)(CO)NC(c1csc(C#N)c1)=O)N(CCC)CCN(C)C CC(C)(CNC(c1ccc(N)cn1)=O)CCNC(c1ccccc1OCC1CC1)=O C(=O)(CCC(C)(C)C#N)NCC(N1CCCC(C)C1)c1ccccc1 C1(C(=O)NC(C2(O)CN(C(c3cc(C4CCC4)no3)=O)C2)C)CC2(CC2)CO1 c1(NC(=O)N(C(C)CNc2ncncc2Cl)C2CC2)cc(N2CCCCC2)ccn1.NCC N1(C(CCC(=O)N(C)C)=O)CC(C2CCCN(C(c3sccc3C#N)=O)C2)C1 c1(OC(CC)CN(C(=O)C(N)=O)CC(=O)C2CC2)ccc(F)cc1F C(=O)(C(F)C(C)CNC(c1cnn(C)c1C#N)=O)N(CC)CC1CCCC1 N1(C(c2ccccc2F)=O)CCN(NCC=CC(=O)NCCCOCC)CC1C N1(C(CC(CC)C)=O)CC(=O)NC2CN(C(c3cccc4c[nH]nc34)=O)CCC12 c1(C(=O)NCC2N(C(C(C=C)O)=O)CCC2)ccc(NCC(N)=O)c(Cl)n1 c1(C(N2CCC(N(C)C(c3cc(F)n(C)n3)=O)C2)=O)ccc2c(c1)nnn2C C(CC(=O)NCC(C)C(F)(F)F)(C(F)(F)F)NC(CCOC(C)=O)=O C1(C(N(C)Cc2ccsc2)=O)C2CN(C(=O)CCN3CCC(F)C3)CC12.C(=O)CN N1(S(c2c(NCc3ncn(CC)n3)nccc2)(=O)=O)CC(CO)OC2(CCC2)C1 c1(-c2nc(C(c3cncc(F)c3)C)nn2C2CC2)nccc2ncccc12 c1(C(N2CCOCC(CNC(C3CC3C3CC3)=O)C2)=O)nnc2ccccc2n1 c1(NCC2(C)ON=C(C)C2)ncnc(NC(c2ccccn2)C)c1C c1(CN(CC(CC)OC)C)cc(C)cc(C)c1 C(=O)(C(CCOCCO)NC(C1CC=CC1)=O)N1CC(C(CC)CC)C1 C(CCC(C)(C)NC(C1CN(C)C(=O)N1)=O)NC(C(C)Cc1ccncc1)=O N1(CCc2nc(C)c(C)o2)CC(=O)N(Cc2ccccc2OC(F)F)C1=O N1(C(C(c2ccccc2)C)=O)CCC(F)(F)C(CNC(=O)C2=COCCO2)C1 c1(CC(=O)Nc2cccc(CF)c2)ccc(Cl)cc1F.C12CCN(CC1)C2=O c1(CC=C)ccccc1C(=O)NCC(C1CC1)N(C(=O)C(C)(C)n1cncn1)C N1(C(CN(C(c2ncn(CC)c2)=O)C)=O)CC(F)(F)CC1CO CC1(C)COc2cc(CNc3cc(F)cc(F)c3)nn2C1 CC(C)CC(CNC(c1ncc2ccccn12)=O)C(=O)N1CC(O)C1 Cc1cccc(C2CC2C(N2CCC(CNC(C3CCO3)=O)CC2)=O)c1 N1(C(CSCCC)=O)CCCOC(CNC(=O)CN2C(=O)CCC2=O)C1 c1(CCC(=O)N(C2CCN(C(C3CC34CCC4)=O)C2)C)c(C)noc1C.CN Cc1ccc(-c2nc(C(=O)NC3CN(C(=O)C(=O)NCC4CC4)C3)co2)c(C)c1 C1(n2cc(CCCCC)nn2)CC2CCC1(C(=O)N(c1cccc(OC)c1)CC)C2 CC1CCC(CC(=O)NCCCN2CCN(C(=O)Cc3csc(S)n3)CC2)CC1 C12(CC(C)(C)C1)C(C)C(=O)NCc1cccc(n1)NC2=O.C1(CO)CNC(=O)O1 c1(C(N2CC3OC(C)(C)OC3C2)=O)cccc2ccc(Cl)nc12 Cc1ccc(C)c(OCC(=O)NCC(C)NC(C2CCCCC2)=O)c1 N1(C(c2c(CC)n(C)nc2)=O)CCC2(CC2C(=O)NC2(C)CCCC2C)C1 C1(NC(C(C2CCOCC2)C)=O)CN(C(c2nn(C)cc2Cl)=O)CCC12CCC2 C=CCC(CC=C)C(=O)N1CC(NC(c2cn(C)c(C(F)F)n2)=O)CCC1C N1(C(C2CCCN(C(=O)CNS(=O)(=O)C(F)(F)F)C2)C)CCc2ccccc2C1 c1(C(N2C(C)CCC2)=O)cc2c(s1)C1(CCN(Cc3ncccc3F)CC1)OCC2 C1(C)(C(=O)NCC(C)NC(=O)CCCNC(=O)C(C)(C)C)CC(O)CN1C CC1=C(C(=O)NCC2C=CCN2C(c2cn(C(C)C)nn2)=O)C(=O)OC1(C)C c1(OC)cncc(C=CC(N2CCC(NC(=O)C(C3(O)CCCC3)F)C2C)=O)c1 C1(NC(c2cnc3ccsc3c2)=O)COC2(C1)CN(C(c1cnco1)=O)C2 c1(C(N(C(C)CN2CCCCC2)C)=O)c(O)cccc1F C1(CNC(CSCC#C)=O)CN(C(c2ccn(CCC)n2)=O)CC12CC2 c1(C(=O)NCCOCCN(C(C(F)OC)=O)C)cnn2c1OCC(O)C2 c1(C(=O)NCC(CNC(c2[nH]c(CC)c(Cl)n2)=O)O)c(O)ccc(Cl)c1F c1(CN2CCC(C(N3CCC(O)C(F)C3)=O)C2)cnc2cc[nH]c2c1 C12(C(C)C)CC(NC(=O)Nc3nc(CN(C)C)cs3)(C1)C2 c1(C(N2CC(C(C)(C)O)(CNC(c3c(C)ncs3)=O)C2)=O)scc2c1CCCC2 C1(NC(c2ccn(CC)c2C)=O)CN(C(C2C=CCS2)=O)C(C)(COC)C1 N1(C(c2c(C)cccc2)=O)CCC2(CNC(C3CSC3)=O)CCCCC12 C1(C#N)(C(=O)NCC(CNC(=O)Cc2csc(C(C)(C)C)n2)OC)CC(C)C1 N1(C(c2c(CNC(C3CCSC3)=O)cco2)=O)CC2COC(=O)C2C1 C1(c2nnc(CNC(c3cn(C(C)C)nc3Br)=O)s2)CCCCN1CC C(C(=O)NNC(=O)NC1CCCC1)C(CC(=O)OC)c1ccsc1 CC1CCC(=O)N(CC(C)(C)NCCCC2N(C(=O)OC(C)(C)C)CCCC2)C1 CCC(C)(CNC(c1ccn(CCNC(=O)Cc2ccsc2C)c1)=O)OC C12(CNC(C(C)(C)OC)=O)CCCCC1CN(C(c1cc(CO)n(C)n1)=O)C2 c1(C(=O)NC(C(C(C)C)NC(=O)CSc2cn[nH]c2)C)csc2ccccc12 N1(c2nccc(C(=O)OC)n2)CCC(NC(C2C3COCC23)=O)C1(C)C c1(C(=O)NC(C)CNC(=O)CC2CCCOC2)ccc(OC(F)(F)F)c(Cl)c1 CCCC(C)(C)C(=O)N1CCCC1CSc1cncc(-c2cccs2)c1 Cc1cccc(-c2noc(NCC(c3ccccc3C)C)n2)n1 N1(CCC(N2CCC(CCNC(c3ncn(C)n3)=O)C2)=O)C(=O)NC(C)(C)C1=O N1(C(=O)CC2(O)CCCCC2)CC2=C(C1)CN(C(c1ccn(C3CCC3)n1)=O)C2 Cc1cccc([N+](=O)[O-])c1N1CC(O)(C(C)NC(c2cc3n(n2)CCO3)=O)C1 C1(CNC(CN(C)C)=O)C(CNC(c2cnn(C(C)(C)C)c2)=O)C1(F)F C(=O)(CCCCC(C)(C)C)NC(C)C(CO)NC(C1CC12CCOCC2)=O C1(CNC(c2c(OC)ccc(O)c2)=O)CN(C(=O)C(F)=CCCF)C2(CCC2)C1 c1(C(=O)NC2C(NC(=O)CC3CCCCC(=O)N3)C2)ccc2c(c1)C(=O)CCC2 c1(C(=O)NCC2CN(C(c3n(CC)ncc3)=O)C2)nc[nH]c2nccc1-2 C1(NC(C(C)(N(C(c2c(C)csn2)=O)C)C2CC2)=O)CCCCCC1O CCCC(CCC)CC(=O)NCC(C)(C)CNC(c1cc(F)ccc1F)=O C1(NC(C2(COCCOC)CC2)=O)C2CN(C(=O)Cc3cncnc3O)CC12 CC1CCc2onc(C(=O)N(C3CN(C(=O)C#CC4CCCOC4)C3)C)c2C1 CCC(C(=O)OC)C(=O)Nc1ccccc1N1CCN(c2cc(SC)no2)CC1 C1(C(=O)NCCNC(=O)NCC#N)(NS(C(C)C)(=O)=O)CCOCC1.C(C)(C)(C)O CC(C)C(C(=O)OC(C)(C)C)NC(c1ncccc1N(C)C)=O.C1(C)CC1C#N N1(C(C2CCN(CC(C)C)C2)=O)CCC(CNC(=O)C(C)CSC(F)(F)F)CC1 c1(NCC2N(C(C3(CC)CCNC3=O)=O)CC2)nc(Cl)nc2sccc12 N1(C(C2CN(C)C(C)(C)C2)C(=O)NC(C(=O)OC)C)Cc2ccccc2C1 C1(NC(c2cnn(CC)n2)=O)CC(NC(=O)Cc2cc(F)cc(F)c2)C12CCC2 C1(CNC(CCCc2c(C)ccs2)=O)CCN(C(c2cnsn2)=O)CC1C N1(C(C(C)NC(N)=O)=O)CC2CC3CC2C1C3NC(c1ncc(F)cc1F)=O N1(C(C(C)NC(COC)=O)=O)CC(C2CN(C(C3(C)CCC(F)(F)C3)=O)C2)C1 Nc1cc2ccccc2c(C(=O)NCC2CCN2C(=O)CC2CCOC2)n1 c1(C(N2CCCN(C(CC(CC)C(=O)OC)=O)CC2)=O)c(OC)ccc(C)c1OC c1(OC)ccc(CC(N2CC(N(C)C(C3CC(C)(F)C3)=O)C3(CC3)C2)=O)c(C)c1 NS(=O)(=O)C1(C(=O)NCC2(CNC(=O)CC(F)(F)C(F)F)CC2)CCCC1 C1(C(N(C2CCN(C(C3COC3)=O)CC2)CCOC)=O)CCCCN1C CC1CC(C(N2CCC(O)(CN=c3[nH]nc(C(N)=O)s3)CC2)=O)CCS1(=O)=O C(=O)(C(F)(F)C(F)(F)C(F)(F)F)N1CCC(N(C)C(c2cc[n+]([O-])cc2)=O)C1 C(CCC(C(=O)N(C)C)NC(=O)NC1(C)CN(C(c2ccc(Cl)cn2)=O)C1)OC c1(C(=O)OC)c(F)cc(Nc2nc(SC)ncc2OCC)cc1F C1(CC)CCC(C(N2CCOC(CN(C)C(C3CCCN3C3CC3)=O)C2)=O)CC1 Cn1cncc1CC(=O)NCC1OCCC1C(N1CC(c2ccon2)C1)=O Cc1nc(CNC(=O)Cn2cc(Cl)cn2)oc1C(N1CCCCC1SC1CC1)=O c1(CNCCN2CCN(C(c3n(C)cc(Br)n3)C(=O)O)CC2)cc(F)cnc1O CC1CN(C(=O)C(F)(F)c2csc(Cl)n2)CCN1C(=O)OC(C)(C)C c1(C(N2CCC(NC(Cc3cn(C)nn3)=O)(CO)C2)=O)cccc2cnsc12 c1(CC(=O)NC2(CCNC(CCCSC)=O)CC2)ccc(O)c(F)c1 C1(CC)(CC)CC(NC(=O)C(C)S(N)(=O)=O)CN1C(C1CCC(C#N)CC1)=O c1(C(=O)NC2(COC)CN(C(=O)CC(C)OC)C2)cc(C(F)F)cc(Cl)c1 n1(CC)nc(C)cc1C(=O)NC(CCOC)C(=O)Nc1cnn(C)c1C(N)=O C1(C)(CC(=O)N(CCOC)CCNC(=O)CCN2CCCC2=O)CCS(=O)(=O)N1 N1(C(c2n(CCC)ccc2)=O)CC(F)(F)CC1CNC(C1CC1C(C)(F)F)=O c1(C(N2CC(CC(N3CC(C)C(O)C3)=O)C2)=O)ccc(F)c(Br)c1F c1(C(=O)NC(CC)CNC(=O)CC2COCCO2)[nH]c2cc(Cl)ccc2c1C O=S(=O)(c1ccc(Cl)cn1)NC1CN(Cc2coc3ccccc23)CC(F)(F)C1 C1(CNC(CSC2C(=O)OCC2)=O)CCCN(C(c2ccc(O)nn2)=O)C1 CC(C(=O)NC1C=CCN(C(=O)Cc2c(F)cccc2Cl)C1)C(C)(F)F C=CCC(CC)C(=O)N1CC2(CO)CC1(C(=O)NC1CCCC3CC13)C2 c1(C(C)NCC(CO)N(C)C)cccc2ccccc12 C1(C(C)OC(C2(S(C)(=O)=O)CC2)=O)CCC2(CCCCCC2)O1 C1(CC(=O)N(CCCCCNC(C2C(c3n(C)ncc3)C2)=O)CC)CC2(COC2)C1 N1(C(C2(CCNC(C3(F)C(C)(C)C3(C)C)=O)CC2)=O)CC(C)(C2CCC2)C1 C1(CN(C)C)COCC1NC(C1COCC1NC(=O)CN1CCOC1=O)=O C1(CNC(CC2CC(C)(C)OC2)=O)CCN(C(c2cccc(O)c2F)=O)C1(C)C N1(C(CCSCCC)=O)CC2C(CNC(=O)CCCCc3ccc(F)cc3)C2C1 N1(Cc2ncc(-c3cn(C(C)C(=O)O)nn3)cn2)CCc2ccc(Cl)c(Cl)c2C1 C1(NC(Cc2cn(CC)nc2)=O)CCN(C(c2cc(OC)cnc2F)=O)CC1O N1(C(C2C(C)C2)=O)CC(CNC(c2cc(Br)n(C)c2)=O)CC(C)(C)C1 O=C(C(O)C(F)(F)F)NC12CC(C(=O)NCCc3nccs3)(C1)C2 c1(C(=O)NCCN(C(CC(C)CN(C)C)=O)CC2CC2)ccnc(Cl)c1O c1(C(=O)N(CCSC)C(C)C)ccc([Si](C)(C)C)cc1 C=C1c2ccccc2C(=O)N1CCC(=O)NC1CCCN(C(=O)CC(C)CF)C1 N1(C(Cc2c(Cl)cn(C)n2)=O)CC2CC(C1)CN(C(=O)C#CC1(C)CCCO1)C2 CCC(C)C(C(=O)NCC1CCN1C(=O)Cc1cccc(Cl)c1F)N(C)C C1(C(=O)NCc2c(C)csc2)CN(C(=O)CCc2cn(C)cn2)CCO1 C1(c2c(C)cccc2)CN(C(=O)C(=O)NC(C2CC2)C2CC2)C(C)CO1 C#CC1CCN(C(=O)C(=O)NC2CCN(CCC(F)(F)F)C2)CC1 C(CC(C)C(=O)NC1(C(=O)NCc2cc(C3CC3)on2)CSC1)=CC C1(CNC(C(N2CCC(C)SCC2)c2cccnn2)=O)C2CCCCCCC12 C1(C)(CNC(C2(CNC(CCOCC(C)C)=O)CCCO2)=O)NC(=O)NC1=O C1(C(C)NC(C2CCC(C(F)F)CC2)=O)CCN(C(C2(CO)COC2)=O)CC1 Cc1cc(C(N2CCOCC(CNC(=O)C(F)C(C)C)C2)=O)cc(C)c1C#N c1(C(N2C(CN(CCOC)C)CCC2)=O)ccc(SC)c(Br)c1 c1(C(N2C(CC)CC(F)C2)C(=O)NCC2CC2)cc(OC(F)F)cc(F)c1 c1(NC2CC(C)CN(C(=O)OC(C)(C)C)C2)nc2c(Br)cccc2s1 C#CCCCC(N)C(=O)Nc1ccccc1CN C(=O)(C(C)S(=O)(=O)C(C)C)N(C(C)C)CCN(c1nc(C(F)(F)F)n[nH]1)C N1(C(=O)Nc2ccc(C)cc2C)CC2CCCCC2(NC(=O)C(C)(C)O)C1 c1(-n2c(C3C(SCCOC)C3)nnn2)c(C)cccc1C C1(C(C)C)(C(=O)NC2CCN(CCF)C2)CCCN1C(C1CC2(CCC2)C1)=O N1(C(C(C2CCOC2)NC(Cn2c(=N)nc[nH]2)=O)=O)CCCC(C2CC2)CC1 N1(C(c2ncc(C(=O)NCC)nc2)=O)CCN(C)CC1CNC(=O)CCCOC C(=O)(C(C(C)C1CCOCC1)N(C1CCCCCC1)C)NCC(C)C C1(C(=O)NCC2(C)CN(c3cc(O)nc(O)n3)CCO2)CCc2c[nH]nc2C1 CCCCC(C)C(=O)NCCCCN(C)C(c1cnn(-c2ccc(F)cc2)n1)=O N1(C(C(CC2CC2)NC(c2ccc(CC)s2)=O)=O)CCC2CCC12 S(=O)(=O)(c1ccc2nc(O)oc2c1)N1C(C(=O)NC(c2cccc(Cl)c2)C)CC1 CCS(=O)CC(=O)NCC(C(=O)C(F)(F)c1ccccc1)=O.c1(NCC2CC2)cncn1C c1(CC)nc(Cl)cc(NNC(=O)NC2CCN(c3cc(C)cc(C)c3)CC2)n1 N1(C(C(C=C)O)=O)C(CC(N2CCCCC2C(F)F)=O)C2CCCC12 CC1(C)CCCC(C(=O)NCC2CCC(NC(=O)Cc3cnoc3)CC2)CC1 C1(C(N(CCCN(C)C)CC)=O)CC(=O)CN1C(=O)Cc1cnnn1C C12CCC3(CCC3)CN1C2=O.C1(CC)CC2(C1)CC2N(C(=O)COCC(F)F)CC C1(C)(C(=O)NCC2C(NC(C3C(C)(C(F)F)C3)=O)C2)C2CC3CC(C2)CC1C3 C(=O)(CCC(=O)NC(C1CN(C(=O)C(c2ccccc2)O)C1)C)NCC c1(NC(C2C(NC(c3ccsn3)=O)C3CCC2C3)=O)cc([N+](=O)[O-])c(F)cc1Cl c1cc2nc(N3CCC4(CC3)CC4CN3C4CCC3CC4)[nH]c(=NC3COC3)c2[nH]1 C12(C(N(C3(C#C)CN(C(c4cc(C5CC5)on4)=O)C3)C)=O)CCC(C1)C2(C)C N1(C(C(CC)(F)F)=O)CCN(C)C(C(=O)N(C)CC2CC(F)(F)C2)C1 c1(OC(C)=O)cc(C)c(Br)cc1C(N1CCOCC(NC(=O)C(C)O)C1)=O N1(C(C2OCCN(C)C2)=O)CCOCC(F)(CNC(c2cc(CCO)on2)=O)C1 C1(CC)CN(C(C2CCCCS2)=O)CCC1NC(c1c(CC)cccc1F)=O Cc1c(-n2cc(C3CC3C(=O)NN3CCCC(CCO)C3)nn2)cccc1F N1(C(CCC=C)=O)CCOC2(C1)CN(C(c1ccoc1CC(N)=O)=O)C2 c1(C(=O)NCC2(F)CCN(C(CC(C)C(F)F)=O)C2)n[nH]c2c1CCOC2 CC1(C)CCCC(CC(=O)NC2CCCN(C(c3cocn3)=O)C2)O1 C1(C(N2C3C(CNC(C(CC)NC(N)=O)=O)C(C3)C2)=O)CC2(CCC2)CO1 CC1COC2(C1)CN(C(C1CC(NC(=O)C=Cc3ccco3)CCO1)=O)C2 C1(CC(N2CCC(CCNC(c3n(C=C)ncc3)=O)C2)=O)CCCS(=O)(=O)C1 N1(C(CN(C(C)=O)C)=O)CCC(C2CCCN(C(C3CC(CF)C3)=O)C2)CC1 N(C1c2ccccc2CC1O)C(C1CC12CCN(Cc1ccccc1I)CC2)=O S(=O)(=O)(c1cccc(=NCC(CC(C)C)c2ccc(F)cc2F)[nH]1)NCC#CC CN=S(C)(=O)c1cccc(C(=O)NC2CN(C(=O)CC3NC(=O)NC3=O)C2)c1 C1(CNC(=O)CC2COC(CNC(COCCC)=O)C2)COC2(CCC2)CO1 C(=O)(C(O)C(C)CC)NCc1cccc(NC(CCCCOCC)=O)c1 c1(N(CC)CC)ccc(C(N2CC3CC3(CNC(=O)C(C)(Cl)Cl)C2)=O)cn1 C(N=c1[nH]c(=NCC2CC2C2CC2)[nH]c2c1COCC2)c1nnn(C)n1 CCC(C(C)C)C(C(=O)N(C1(C)CC1)C1CC1)N1CCOC(C2CCC2)C1 c1(N2CCC3(CCCC(C)(C)C3)C2)nc(=N)[nH]c(=NC2C3CCC(F)(F)C23)[nH]1 C1(c2c(F)cnc(OC)n2)CN(S(=O)(=O)c2ccccn2)CC12CCOCC2 c1(C(=O)N)ccc(C(C)C)nc1.C(C(=O)NCC1(CO)CCC1)(C1CCOC1)OCC c1(C(=O)NC2C(F)CCN(C(C(C#N)C3CC3)=O)C2)csc(S(N)(=O)=O)c1 C1(C(=O)NCC2CC3CCC(C2)N3C(=O)CO)CCC2(CCCCC2)C1 c1(NCC2(CNC(c3c(COC)noc3)=O)CC2)cccc(F)c1[N+](=O)[O-] C(=O)(CCC(C)(C)[N+](=O)[O-])N1CC=C(CCNC(CCN(C)CCO)=O)CC1 c1(C(N2C(C3(O)CN(C(c4c(Cl)cn(C)n4)=O)C3)CCC2)=O)nnc(Cl)cc1N c1(SCC)cccc(C(=O)NCC2CN(C(=O)C(C)(C)C3CCCO3)CCO2)c1 C1(C)(NC(=O)NC2CC(CNc3nccc(C(C)(C)C)n3)C2)CCC(C)=C(C)C1 N1(C(C2(CC)CCNC2=O)=O)Cc2ccccc2CC1CNC(=O)CO C12(Cn3c(N4CC(C)CN(C)CC4)nnn3)CC3(C)CC(C)(C1)CC(F)(C2)C3 C1(NC(CCCC2C(C)C2)=O)COC2(C1)CN(C(=O)C1=CCCCC1)C2 Cc1c(NC(C2(C)CCCCN2)=O)cccc1F Cn1nc([N+](=O)[O-])c(Cl)c1C(N1CCCC(NC(c2cc3scnc3[nH]2)=O)C1)=O CON(CCC(=O)NC1(C)CCCC1C)C(=O)CC(C)(C)C(C)=O Cn1cnc2nc(-c3ccccc3)[nH]c(=NC3CC(F)(F)C3)c12 c1(C(=O)NCC2CCCN(C(=O)CN3CCCC3=O)CC2)[nH]nc2ncccc12 Cc1c(C(N2CC3CC(C2)N(C(c2csnc2Cl)=O)C3)=O)oc2ccccc12 C1(C(=O)NC2C(O)CCN(C(CN3CC(C)(C)C3)=O)C2)CCc2ccccc2C1 C1(NC(C2C(OCC)CC2)=O)CC2CC1CC2C(N1CCC(OC(C)=O)CC1)=O c1(OC)ccnc(Cl)c1CN1CCOCC(C(=O)NCCc2ccncn2)C1 CCCC(C)C(=O)NC(Cc1ccccc1Br)C(=O)NCC12CCC(C1)C2 CC(C(=O)N1CCC(N(CCO)C(C2CCC2(C)C)=O)CC1)C(F)F N1(C(C2(Cl)C(C)(C)C2)=O)CC(CO)C2(CCN(C(=O)C=C3CCCC3)CC2)C1 N1(C(c2cc(CC)n(C)n2)=O)CCC(NC(C2C=CCCC2)=O)C(O)C1 N1(C(C2CC(C(C)C)C2)=O)CCCC1CNC(C1(C(C)(C)C)CCC1)=O C(C)(CN=c1nc2scnc2c(N(CCC(=O)N(C)C)C)[nH]1)Nc1ncc(C)nc1 c1(CNC(N2CCN(OCC(=O)O)CC2)=O)cc2n[nH]cc2cc1Cl c1(C(N(CCCCC)CCO)=O)ccc(CN2CCCCC2)o1.n12cc(nn1)C2 C1(NC(=O)CCc2cncc(F)c2)CCN(C(C2C=CCC2)=O)C12CCC2 c1(C(=O)NC2CN(C(CC(CCC)O)=O)CC3(C2)CC3)cccc2ncccc12 c1(C(=O)NCC(C)(C)OCC(=O)N(C(CC)C)C)cnn2c1CCC2 c1(CC)cccc(C(=O)N(CC(C)NC(c2ccc(C)n2C)=O)C)c1 C(=O)(C1CCc2ccc(C)cc21)NCC(CCOC)NC(=O)C(C)CC(F)F N1(C(CCc2cc(C)[nH]n2)=O)CC(=O)CC1C(=O)OCC1CCCCC1C O=C(CC1=NNC(=O)C1)NC1CCCC(CNC(=O)Cc2csc(NC=O)n2)C1 c1(C(=O)NCCCC(C)NC(C(CC)C(F)(F)F)=O)[nH]c2ccccc2c1C C1(C(=O)NC2C3N(C(CN(C(C)C)C)=O)C(CC3)C2)CC2CCCN2C(=O)N1 C1(C)(COC(c2n(C)ccc2-c2c(Cl)cccc2Cl)=O)CCCCN1S(C)(=O)=O Cc1ccn(CC(N2CCC(O)(C(C)NC(C34CC(CO)(C3)C4)=O)C2)=O)c(=O)c1 c1(OC)ccc(CC(O)C(=O)NCCCCCN(C)C(c2ccns2)=O)cc1 Cc1cc(Cl)nc2cc(C(N3CCC(CNC(C4CC4F)=O)C3)=O)ccc12 N1(C(C(C)S(C)(=O)=O)=O)CCC(F)(F)C(CNC(=O)CC2CCCC(=O)N2)C1 c1(CCC)nsc(N)c1C(=O)NCC(O)CNC(=O)Cn1cc[n+](C)c1 c1(C(=O)NCCCN(C(=O)CCSC)CC)cc(C)c(OC(F)F)c(C)c1 C1(CNC(=O)CCc2ccoc2)CC2CCCC2N1C(C1CS(=O)(=O)C1)=O C=CCCCCCNC(C1CC(C)N1C(=O)COc1ccccc1)=O c1(CCC(=O)N(CCCCN(c2nnc(CC)o2)C)C)ccc(S(C)(=O)=O)cc1 O=C(C1=CSCS1)NC(CNC(C1CCCS1)=O)C1CC1 N1(C(c2cscc2Br)=O)CCC(N2CCC(F)(CO)C2)C2(CC2)C1 C(C)(C(C)NC(=O)CC1(N(C)C(C2(CCF)CCC2)=O)CC1)SC CCCS(=O)(=O)C(C)C(=O)N1CCC(n2cc(-c3ccc(SC)c(Br)c3)nn2)C1 C1(C(=O)NC(C2CC2C(=O)NCCC(O)C2CCCC2)C)CC2(C1)CC21CC1 c12cccc(c1OC)C(=O)OC2.C1(C(C=C)C)CN(C(=O)OC(C)(C)C)CCO1 N1(C(CSCC)=O)CCC(C2CCN(C(c3cccc(C4CCCC4)c3)=O)C2)C1 Cc1cc(Cl)c(C(=O)NCCCCNC(C2(Cl)CC23CCC3)=O)cc1C C(=O)(C(C)(C)CCCF)NCCCCCN(C(=O)CC1CC(=O)NC1=O)C c1(C(=O)NCC2C(NC(C3(COC)CCC3)=O)C2)c(Br)ccc(C)c1F Cc1nc(C(N2CC(O)CC2CNC(C2CC2C(C)(C)O)=O)=O)c(=O)[nH]c1C C1(C(N2CCC(NC(c3c(CC)ncs3)=O)(CF)C2)=O)COC2COCC2O1 C12CN(C3(CCC3)C1)C(CCC1CC1)C(=O)NC2.c1(CC)nocc1C1CC1 CC1(C(N2CCC(O)C(NC(C3(F)CC=CC3)=O)C2)=O)CCC(O)CC1 C1(CO)CCCN(CC(c2nnc(-c3ccccc3)n2C2CC2)O)C1 C(=O)(C1=C(C#N)CCC1)NCCN(C(C1(OCCOC)CC1)=O)C c1(OC)ccc(CN2CCCC(COC(C)C)C2)c(OC)c1 N1(C(C(C2(O)CN(C(CCCC#N)=O)C2)F)=O)CC2COCC2C1 c1(C(N(C2CN(C(C(C(C)O)C)=O)C2)C)=O)cc2nc(F)ccc2o1 C(N=c1[nH]c2ccccc2[nH]1)c1cccc(NC(N(C)C)=O)n1 C1(C(=O)NC(C(=O)Nc2c(C)ccnc2)CCF)CN(C)CC(C)O1 c1(C(=O)NC2C(NC(C3(CC#C)CCC3)=O)CCCCC2)cc(C)n(C)c(=O)c1 Nc1cc(CC(=O)NCCC2CCN(C(c3cscn3)=O)C2)ccc1[N+](=O)[O-] C1(CNC(c2cc(C)c(C)nn2)=O)CC2(CCC2)CN1C(c1ncc[nH]c1=O)=O c1(C(=O)NC2C(C(N3CCC(=C)CC3)=O)CCC2)ccc(F)c(F)c1F C1(C(=O)NCC2CC(NC(c3nc(C)oc3)=O)C2)(CO)CC(C)(C)C1 c1(OCC)cccnc1C(=O)NC1(CF)CCN(C(c2cc(C)oc2C)=O)C1 Cc1cc(C2CCC2)ncc1C(=O)NC1CCC(NC(=O)CNC(=O)C2CC2)CC1 N1(C(c2ccc(C#C)o2)=O)CCOC(C(=O)NC(C2CCCCO2)(C)C)CC1 CCC(C)CCC(=O)NCC1(C(N2CC(C(C)(C)C)C2)=O)CC12CCC2 N1(C(CNC(=O)OC)=O)CC2(C=C(C(=O)NC(C3CCC3)C)CO2)C1 c1(C(=O)NCCC2(NC(c3nc(CCC)oc3)=O)CC2)cnc(C(C)C)n1C C(CCCC(=O)NCCN(C(=O)C=C1CN2CCC1C2)C)OC c1(OC)cc(F)cc2[nH]c(C(=O)NCCC(C)N(C(=O)CCC(C)SC)C)cc12 CC1CCN(C(C2CCO2)=O)CCN1C(c1csc(-c2ncc[nH]2)n1)=O c1(OC)ccc(C(=O)NCC2CCN(C(=O)Cc3ccoc3)CC2O)cc1C C1(C(=O)NCCC(CC)CO)CCCCN(C(C2COCCO2)=O)C1 C1(Cn2c(-c3ccc(C)o3)nc(-c3c(C)occ3)n2)CCC2(CCOCC2)CO1 c1(CNC(C(CC)OC)=O)ccc2c(c1)CN(C(=O)Cc1ncc(Cl)s1)C2 C1(CCNC(CCC(=O)NC)=O)CC(F)(F)CN1C(c1ccc(C(N)=O)cc1)=O C#CC1(O)CCN(C(=O)CC2CCC(NC(=O)Cc3cncn3C)C2)C1 c1(OC)cccc(C(C)N(C(c2ncccc2C)C(=O)NCCCF)C)c1 C1(Cn2c(N3CCC(N(C)CC4CCCO4)C3)nnn2)CCOC2(CCC2)C1 C(=O)(C(CCC)NC(=O)COCCN(C)C)NCC(CCC)C.C(C)(C)(C)O CC1=CCCN(C(=O)C(C2CCN(C(=O)Cn3cc(CN(C)C)nn3)C2)F)C1 C(=O)(C1=CCCSC1)NC(CNC(Cc1c(OC(C)C)cccc1)=O)C c1(C(C(N2CC(OCCNC(C(C)NC(C)=O)=O)C2)=O)C)c(Cl)cccc1Cl C(CNC(c1cccc(Cl)c1Cl)=O)(CC(F)(F)F)NC(c1cn[nH]c1)=O c1(NC(C(CSC)=O)=O)ccccc1-c1ccno1 C=C(C)C(C)(C)C(=O)Nc1ccc(N2CCOCC2)c(C)c1 n1(CC2N(CC(CN(C)CC)O)C(C3CC3)CC2)ncc2ccccc12 C12(COC)CN(C(c3cn(C)nc3C)=O)C(CNC(c3n[nH]c(C)c3O)=O)(C1)C2 C1(C(=O)NCC(CCC)O)(CCOC)CCN(C(=O)C=CC2CC2)CC1 C1(C(N)=O)CCCCC1C(=O)NC1CCN(c2ccccc2)C1 N1(C(=O)CC2CCCSC2)CCC(N2CCN(CCO)CC2)CC1 c1(C(N2C(CNC(C(CSC)(C)O)=O)CCC2)=O)cc2ccc(O)cc2[nH]1 c1(NC(=O)Oc2cccnc2F)ccc(CCCC2(C(F)(F)F)N=N2)c(F)c1 c1(CC)cc(C(N2CCC(CO)(NC(=O)Cc3nnc(C)s3)CC2)=O)ccc1O CCCC(CC)N=c1nc2c(ncn2C(C)C)c(N2CCC(NC(N)=O)C2)[nH]1 C(C(=O)NOCC(=C)C)N(C(C(CC=C)C1CC1)=O)CC1CC1 N1(C(c2cn(CN(C)C)nc2C2CC2)=O)CCC2(NC(=O)C3=COCC3)CC2C1 c1(C(N2CC(NC(C(C)(C)OC)=O)C3C2C3)=O)ccc(C)c(F)c1F C1(NC(c2c(C)nsc2)=O)CCN(C(C2CCCC(C)CC2)=O)CC(O)C1 N1(C(c2c(C)cc(F)nc2)=O)CCC2CCC(C1)N2C(=O)CSCc1cccs1 Cc1cnc(C(=O)NC2(CCNC(=O)CC3(C)CC3)CC2)cc1Br c1(C(=O)NCC2N(C(C3(C)CC4CC4C3)=O)CCC2)cnc(C2CCC2)nc1O c1(C(=O)NCC2CCC(NC(C3CC(=O)OC3)=O)C2)ccc(Cl)nc1Cl c1(C(N2CC(NC(C3CCC(C)(C)O3)=O)C3(C2)CC3)=O)ccnc2ccsc12 C(C(=O)N=c1ccn(C2CN(c3ccc(C#N)cc3)C2)[nH]1)=CC(=O)OC(C)(C)C N1(CC(=O)NC2CC(NC(=O)C(n3cc(Cl)cn3)F)C2)CCC(F)(F)C1 C1(CN(C(c2scc(OC)c2)=O)C)CCCN(C(c2cnc(SC)n2C)=O)C1 C1(CNC(C(F)OC)=O)C2CN(C(c3cc(C(F)(F)F)ncn3)=O)CC12 c1(C(N2C(CC)CN(C(c3cc(O)ccc3Br)=O)CC2)=O)nc(O)nc(O)c1F c1(OC)ccc(N)c(C(=O)NC2CCN(C(c3ccnn3C)=O)C2C)c1 Cc1cc(N2CCC(COC(=O)Cn3cc(Cl)cn3)C2=O)ccc1Br c1(CN2CC(COC)C2(C)C)cnc2ncccn12 N1(C(c2nc(C(C)NC(C(COC)C)=O)oc2)=O)CCC(N(C)C)C(C)C1 N1(C(C(C)OCC=C)=O)CC2OCCN(C(c3n[nH]cc3CC)=O)C2C1 CC1(C)C(NC(c2coc(Cl)n2)=O)CC1CNC(c1cccc(C(F)(F)F)n1)=O N1(C(c2nc(COC)[nH]n2)=O)CC2CC(NC(=O)C(C)(O)COC)C2C1 N1(C(C=Cc2cnc(C)s2)=O)CCC(CNC(=O)CC2CC2(Cl)Cl)CC1C C=CCCC(CC(C)C)C(=O)NC(C1CCN(C(=O)C(F)=CC2CC2)C1)C C1(C(N2C3CC(CNC(c4n[nH]c(C)c4Cl)=O)C2CC3)=O)CCn2cncc2C1 N1(C(CC(CN(C)C)O)=O)CC2(C)CN(C(c3nc(=O)n(C)[nH]3)=O)CC2(C)C1 C12(NC(c3[nH]cc(C)c3)=O)CC(CNC(c3ccc(O)nc3C)=O)(C1)OC2C c1(C(N(CCCCNC(c2scc(C)n2)=O)C)=O)c(C)coc1C1CC1 O=C1C(c2ccc(Br)cc2)CCN1C1CCN(C(C2(C(F)(F)F)CCCC2)=O)C1 CC(C(=O)NCC(O)CN(C)C(c1ccc(-c2nnco2)cc1)=O)S(N)(=O)=O N1(C(c2cc(OC)no2)=O)CCN(C)C(C(N2CC(O)(C(F)F)C2)=O)C1 C(c1ccccc1C#N)=CC(=O)N(C)CC1(c2ccon2)CC1 C1(NC(c2nc(CC)oc2)=O)CCN(C(c2csnc2C2CC2)=O)C1C(C)(C)C C1(NC(C)=O)CCN(C(=O)CCC2(NC(=O)C(C)(Cl)Cl)CCC2)C1 Cc1ccc(Cl)c(O)c1C(=O)NCC(C(C)(C)C)NC(=O)CSC(C)C c1(NS(C)(=O)=O)ccc(C(F)(F)F)cn1.CC1C(=O)N2CC(C2)C(=O)N1C1CC1 n1(CC)ccnc1C=CC(=O)NC1CC2(C1)CC2NC(C1CCS(=O)(=O)N1)=O N1(C(=O)NCC(CC)N(CC(C)(C)C)C)CCOC(CC(=O)OC)C1 C1(CN(C)C(c2ncc(F)cn2)=O)CCCCN(C(=O)C=CS(C)=O)C1 C=CC1(C(=O)NC2CC23CCOCC3)CCN(C(=O)CCC(=C)Cl)CC1 N1(C(C2CCC(CC)O2)=O)CCN(C(c2cnc(C)cc2Cl)=O)C(C(C)C)C1 CC1(CNC(C2C3CCCC23)=O)COCCN(C(c2ccc(N)cc2Cl)=O)C1 N1(N(C(C(=O)NC(c2c(C)ncs2)C)=O)C)CCC(C(=O)C(F)(F)F)CC1 N1(C(c2ccc(C(N)=O)o2)=O)CCC2(CC1)CN(C(C1CCCS1)=O)CC2CO CC(C(C)NC(C1CC1(C(N)=O)C(=O)OC(C)(C)C)=O)NC(=O)C(C1CC1)N(C)C N1(C(c2ccc(OC)cc2)=O)CCCN(C(C2CN(C)C(=O)CN2C)=O)C(C)C1 C(c1ccccc1C)=CC(=O)N(CC(CNC(C1CCCC(OC)C1)=O)C)C C(=O)(C(C)Cc1cnc[nH]1)N(CCN(C(COC)=O)C)C C1(C)(C(N2CC(CNC(CCOCCCOC)=O)OCC2)=O)CCS(=O)(=O)CC1 C(C)(N=c1[nH]c(Cl)ncc1OC)C1N(C(c2c(COC)nn[nH]2)=O)CCCC1 c1(C2C(NC(=O)NC(C)(CO)C3CCCO3)C2)nc(-c2ccccc2)cc(O)n1 C1(NC(=O)CC2CCC(F)(F)C2)CC2(C1)CC(C(=O)NC1CC13CCOCC3)C2 c1(C(=O)NC(C)C(C)NC(C2CCC=CCC2)=O)cncc2nc(O)[nH]c12 CC(CN1CCC(O)CC1)CN=C(NCC1CCOC1)NC1CCCC1 N1(C(C2CN(C(C)=O)C2)=O)CC2CC1CC2NC(c1ccc(F)cc1Br)=O c1(C(=O)NCCCCCCCn2cc(C3CCC3)nn2)cnn2c1OCC(F)C2 c1(NC(C2CCC(NCc3sccc3Cl)C2)=O)cc(F)c(Cl)cc1F CC1CN(C(=O)CC(C2CCC2)C2CCC2)CC1NC(c1cc(C2CC2)on1)=O c1(C(N2CCCC(CCC)(NC(=O)C(CC)CC)C2)=O)ccnc2[nH]ncc12 c1(C(=O)NCC(CNC(c2nc(C)nc(O)c2)=O)F)cc(Cl)cc(Cl)c1O N1(C(c2cc(OCC)n[nH]2)=O)CC(NC(c2cc(O)n(C)n2)=O)CC(F)(F)C1 C(=O)(C1=NOC(C)C1C)NC(CN(C(c1coc(C)c1)=O)CC)C C(=O)(C(O)C(C)(C)C)N(Cc1c(CCNC(C(C)SCCCC)=O)ocn1)CC N1(C(=O)OC(C)(C)C)C2CC=C(C(=O)CC(O)C3CC3)C1CCC2 c1(C(N(C2CCN(C(c3c(CCC)occ3)=O)C2)CC)=O)n[nH]c(C)c1C c1(OCCOC)cncc(CN(C=O)CC2CCCC(c3cccc(Cl)c3)C2)c1 C1(C(=O)NC(C2CCN(C(c3c(CC)n(C)nn3)=O)C2)(C)C)CC12CCOCC2 Cc1cnc(C(=O)NC(c2ccccc2)CNC(c2cnn(C)c2Cl)=O)cn1 c1(CNS(N(C)CC(c2ccccc2)O)(=O)=O)cc(O)cc(F)c1 N1(C(C(c2ccccc2F)OC)=O)CCC12CN(C(=O)CN1CC3CCC1C3)C2 N1(C(c2c(C)ccs2)=O)CCCC12CCCN(C(=O)C1=CCC(C)CC1)C2 c1(C(=O)NC(c2cn(C(CC=C)CC)nn2)C)cccc2c1CNC2=O N1(C(C=C=C(C)C)=O)CC2(CC(CC(N3CC4(CC4)CC3C)=O)C2)C1 C(=O)(CC(C)(C)O)N(C(CNC(C1NC(=O)CC1c1ccccc1)=O)C1CC1)C c1(OC)cc(C(=O)NC2CC(NC(C3(O)CCCC3)=O)C2)c(OC)cc1Cl c1(-n2cc(CSCCNC(C3C(CN(C)C)C3)=O)nn2)c(F)cc(F)cc1F CC12CCC(C(=O)NCC3(CNC(c4nnn5c4CSCC5)=O)CC3)(CC1)CO2 c1(NCCN(C(CCCOCC)=O)C)cncc(Cl)n1 Cc1ccc(NC(c2ncoc2CNC(C2(C)CC(=O)N(C)C2)=O)=O)c(C)c1 C1(C#N)(N(C(=O)C(c2ccccc2F)NC(=O)OC(C)(C)C)C)CCOC1 N1(CC(CCC)C)CCC(C(=O)NC2CCS(=O)(=O)CC2)C(O)C1 c1(C(=O)NCC(CCCC)NC(=O)CC(C)COC)cc(C(N)=O)ccc1OC c1(NC2C(C)CN(C(=O)CCC3CCCC3)CC2C)ncccc1S(C)(=O)=O C1(C(=O)O)C=CCN(C(=O)Nc2ccnc(N3CCCC3)c2)C1 Cc1cncc(C(=O)NCc2cn(C3CCCN(C(=O)CO)C3)nn2)c1C Cc1cc(C(=O)NC(C)CCCNC(c2cnc(-c3ccoc3)s2)=O)nc(C)c1 C1(c2ccccc2)(NC(C=COCC)=O)CCN(C(=O)CC2(O)CC2)CC1 c1(C(=O)NC2CC(CNC(C(C)(C)N(C)C)=O)C2)cccc(Br)c1F C(CC1C(=O)Nc2ccccc21)NC(c1c(Cl)nc(C(=O)O)c(Br)c1)=O CC1(C)CC(O)(CC(N2CC3(CC(NC(C4CC4(F)F)=O)C3)C2)=O)CO1 CCCC(C(=O)NCCNC(c1cn(CCC2CC2)nn1)=O)NC(C)=O C1(C(N(C(c2ccc(F)cc2)C)C2CC2)=O)CN(C(C2(O)CC2)=O)CC1F C1(C2CCN(C(C3CC4CC4C3)=O)C2)(NC(C(C)OCCOC)=O)CC1 c1(OC)ncc(C(=O)NCC2(CNC(c3cccnc3)=O)CCCC2)s1 N1(C(C(C)OC2CCCC2)=O)CC(C(=O)NC2CCCCCC2)C(C2CC2)C1 c1(C(=O)NC2CCCN(C(=O)C(F)(F)CO)C2)nc2n(c1Cl)CCCC2 C1(CC)CN(C(=O)Cc2ccc(OC)cc2)CCC1NC(=O)COCCF c1(NC(CCCCNC(c2c(COC)noc2)=O)C)[nH]c(=O)n(C)c(=O)c1C#N C(C(C(=O)N(C)CC1CCCO1)C(C)(C)C)NC(c1n[nH]c(C)c1C)=O C1(NC(=O)CNC(=O)CCCc2cccs2)CCCN(C(=O)Cn2ccnc2)C1 N1(C(c2cc(C)oc2)=O)CCC(O)(C(C)NC(=O)C=CSc2nc[nH]n2)C1 c1(OCC=C)ccc(COC2CCN(C(=O)CC3(CC)CCOC3)C2)cc1 C1(C(C#C)C)CCN(C(=O)C(CC2CC2)NC(c2nnsc2N)=O)CC1 Cc1ccnc(C)c1C(N1CC(O)(c2cn(Cc3ccno3)nn2)C1)=O N1(C(C(C(C)C)NC(=O)CC2(N(C)C)CCC2)=O)CCC2C(CCN2C)C1 C(=O)(C(CC(C)C)C(C)C)NC1(C(=O)NCCc2cc(C)[nH]n2)CSC1 C1(NC(C2(CCC=C)CCCC2)=O)CN(C(=O)Cc2nnc(O)s2)C2(CCC2)C1 c1(C(=O)NC2CCN(C(C(CCC)O)=O)C2)ccc(F)c(O)c1 c1(-c2c(C)nn(C)c2C)ccc2nccc(C(=O)NCCc3ccccc3)c2c1 c1(CC2(OCC)CCC2)ccc(S(=O)(=O)N(C)CCOC2CCCOC2)cc1Cl Cc1cc2[nH]cc(C(N3CC4CCC4(C(N4CC(C)C4)=O)C3)=O)c(=O)n2n1 c1(C(=O)NCCCN(C(=O)CCC2CCCCCC2)C)cn2cccnc2n1 C1(NC(C=CC(=O)OC)=O)CN(C(c2cc(-c3ccc(F)cc3)on2)=O)CC1O n1(CC)ncc(C(=O)NC2C(C(=O)N(C3CCOC3)C)C2(C)C)c1C c1(OC)ccc(Br)cc1NC(C1CN(CC(N2CC(C)OC(C)C2)=O)C1)=O C1(C(=O)NC2CCN(C(CC(CC)O)=O)C2)CCC(C)(C)CC1 C1(C(=O)NCC2C=CC(NC(=O)CCC3(C)CC3)C2)(OC)CCSCC1 N1(C(C2C(C(=O)OCC=C)C2)=O)CCCC2(C1)CN(C(=O)CC1C=CCCC1)C2 N1(C(C2(OCC)CCC2)=O)CC2CCC1C2.c1(C(=O)NC(=O)C2CC2)[nH]cnc1C C(=O)(CCC(F)(F)F)NCC1(O)CCN(C(C(CO)NC(=O)OC(C)(C)C)=O)C1 C1(C)(NC(C=C(COC)C)=O)CCN(C(=O)CC2CC3C=CC2C3)CC1 C(=O)(C(C)(F)C(F)(F)F)NCC1N(C(c2c(Cl)cn(C(C)(C)C)n2)=O)CC1 C(=O)(C1CCCc2cncn21)NC1(C)CC(NC(CCCn2c(C)ncc2)=O)C1 C1(NC(CCCCCC)c2nnnn2C2COC2)COc2c(F)cc(F)cc2C1 C(=O)(C1=CC2CCC(C1)C2)NCCSCC(=O)NCC1CCCC2(CC2)C1.NCO N1(C(=O)OC(C)(C)C)CCCN2C(=O)N(Cc3ccc(C(C)(C)C)o3)C(=O)C2C1 Cc1nn2cc(CC(=O)NCCN3CCC(CNC4(C)CCC(C)C4)C3)nc2s1 Cc1csc(=O)n1CCC(=O)NC(C)(C)CNC(C1CC1(C)C(C)C)=O C(=O)(C(=O)C(C)(C)C)NC(C1CCCN(C(C(COCC)(C)C)=O)C1)C C1(CC)CN(C(=O)C(c2cc(F)ccc2F)=O)CCN1C(c1cccn1C)=O c1(OC)cc(C(=O)NC2(CC(=O)NC(CO)C3CC3)CCC2)c(Br)cn1 N1(CCC)CCCC(C(N2CCC(CF)(NC(=O)COCP(C)(C)=O)C2)=O)C1 C(C)(C)(C(=O)NC(C1CCCO1)CNC(=O)Cn1cc(COC)nn1)SC c1(C(N2C(C)(C)CC(CNC(C3CNC(=O)O3)=O)C2)=O)cnn2c1NCCC2 N1(C(=O)C=CC2CC2)CCCN(C(c2cc3cccn3cn2)=O)CCC1 N1(C(C(COCC)C)=O)CCN(C(c2cnncc2NC)=O)CC2(C)CCCC12 Cc1cc(S(=O)(=O)N(C2CCNCC2)Cc2cc(C#N)ccc2Cl)c(C)cc1Cl c1(C(=O)NCCC2(NC(Cn3c(C)c(Cl)cn3)=O)CC2)ccc(C(N)=O)c(Cl)c1 N1(C(C2CC3CC3C2)=O)CCCC(C2CCN(C(c3cnoc3)=O)CC2)C1 c1(C(=O)NC2C3(CC(NC(Cc4c(C)noc4)=O)C3)C2)nn(C)c2c1CCC2 C(=O)(C1=CN=C2N=CNN2C1)NCC1CC(NC(c2n(CCC)nc(C)c2)=O)C1 N1(C(CC=C=C)=O)CCCC2(CCN(C(=O)CN3C(=O)C(C)C(C)C3=O)CC2)C1 C#CC(C)(C)C(=O)NCC(C(C)(C)C)NC(=O)CCC1CCCCO1 c1(C(N(CCCCN(C(C2C(C(=O)OC)C2)=O)C)C)=O)nnc(C)cc1O N(C1COc2ccc(Br)cc21)CC(N1CC(C)OCC1)=O C12(C(N3CCCC(CN(C)C(C4(C(N)=O)CCC4)=O)C3)=O)CCC(CC1)C(C)O2 c1(-c2cc(CNC(CCCn3cc(COC)nn3)=O)no2)ccc(C)cc1 c1(C(=O)OCC)c[nH]c(=NC2CC(CNC(=O)C3=CC(C)(C)C3)C2)cn1 c1(CC(=O)NC23CC(C2)N(C(C2CC4C=CC2C4)=O)C3)ccc2c(c1)CCC2 N(C(=NCC1(C)CC1Br)NC1CN(C(=O)CCC2CCCCO2)C1)CC(C)(F)F C(CC(CC)C(=O)N(CCCC(=O)NCCSCCO)C)=CC Cn1cc(NC(=O)CO)cc1C(=O)NCc1cc(-c2ccccc2)n[nH]1 Cn1cc(F)cc1C(=O)NCCC1CCCN(C(c2ncccc2Cl)=O)C1 c1(OC)cc(Br)cc(F)c1C(N1CCC(CC(=O)NCc2ccc(Cl)c(F)c2)C1)=O Cc1cc(-c2noc(CNC(=O)C(=O)NCCc3cncc(C)n3)n2)cc(C)n1 c1(C(=O)NC(CNC(C(C=C=C)C)=O)CC=C)cccc(F)c1OCC c1(SCNC(C(c2c(C)nn(C)c2)N2CCOC(C3CC3)C2)=O)ccc(F)cc1F C1(N(C(c2c(CC)cns2)=O)C)CCCN(C(c2oncc2C)=O)CC1 Cc1ccc(CC(C(=O)NCC(C)NC(=O)C(c2cccn2C)=O)N(C)C)cc1 C(=O)(C(O)CC(C)C)NSc1nc(C)c(C(N2CCCC(NC(=O)C3CC3)C2)=O)s1 C1(NC(COC(CC)C)=O)C(C)(C)CN(C(=O)C(CC)(CC)CC)CC1(C)C N1(C(c2c(F)ccc(C#C)c2)=O)CCC2(CCC(C(=O)N(C)CCOC)O2)CC1 C(=O)(C1Cc2ccccc21)NC1C2CN(C(C(CC=C)(C)C)=O)CC1C2 c1(C2C(C(=O)NCc3ccccc3-n3ccnc3)CCC2)ccc(Cl)cc1 c1(C(N2CC(CN(C(C3(C)CCC(C)C3)=O)C)C2)=O)c(O)cccc1F N(C1COc2cc(C#N)ccc21)C(C1CC2(CCN(C(=O)OC(C)(C)C)C2)OC1)=O CCC(CC)(C(=O)OC(C)C)C(=O)NCC(C1CC1)NC(=O)C(CO)NC(C)=O CC12CCN(CC1)C2=O.C1(CC(=O)NCC2CCCSC2)CC2C=CC1CC2 c1(C(=O)NCCC(=C)CNC(=O)CCOC2CCC(C)CC2)ccc(=O)n(C)c1 N1(C(C2(C)C(CC)CCC2)=O)CC(CNC(C2SCCS2)=O)CC12CCC2 C1(C(N2CCN(CC)C(=O)C2)=O)CC12CCN(C(c1c(Cl)cccc1Br)=O)CC2 Cc1cc(C(=O)NC2CCCC2CN(C(=O)Cc2conc2C)C2CC2)c(C)o1 c1(CN2CCC(=CC(=O)Nc3ccncn3)CC2)c(O)cccc1F CC(C(=O)N1CCCC(CNn2cc(C(N3CCCC3)=O)nn2)C1)C(F)(F)F Cc1nc(C(=O)NCC2CCC(NC(=O)CC3CCCC3C)CC2)nn1C c1(N2CCC3NC(=O)C2C3)nccc(=NC2CCN(C3CCC3)C2)[nH]1 N1(C(C2CCCCN(C(CCC(C)CN(C)C)=O)C2)=O)CC2CCC(CO)(C2)C1 c1(C(=O)NC23CC(C(=O)OCC)(C2)C3)cn(C)nc1-c1ccco1 c1(C(=O)NC2CN(C(C3C4COCC34)=O)CC2CC2CC2)ccn2nncc2c1 CC(C#N)CCC(=O)N1CCN(CCNC(C2CC3C(C2)C3(F)F)=O)CC1 C1(CNC(C(C2CCC2)OC)=O)(Cn2cc(C3CCCC3O)nn2)CC12CCC2 N1(C(COCCCC#C)=O)C2CCC(C2)C1C(=O)NCc1ccns1 C(=O)(C1=Cc2ccccc2C1)N1CCC(CNC(C2CS(=O)(=O)C2)=O)C1 N1(C(c2c(CC)c[nH]c2)=O)CCCC(CO)(CC)C1 C(=O)(C(O)C(C)(C)C)N(CC(=O)N(C(CC#C)C)CC)CC C1(NCc2cc(CC)no2)CCN(CCNC)CC1 C1(NC(C=C(C)C(F)F)=O)CC2CCC1N2C(c1ccnn1-c1ccncc1)=O N1(C(c2ncn(CC)n2)=O)CC(NC(=O)CCc2n[nH]c(=N)s2)CC12CCOC2 N1(C(Cc2c(C)n[nH]c2C)=O)CC2(C1)CN(C(=O)C(F)C(F)(F)F)C2 C1(CC=C)(NC(=O)C(COC)N(C)C)CCN(C(C2CC(C#N)(OC)C2)=O)C1 CC12CC(C(=O)NCC3CC4(CC(NC(=O)Cc5cscn5)C4)C3)C(CO1)C2 c1(OC)cccc2c1C(C(=O)N1CC(F)CC1CNC(C13CCC1CC3)=O)CC2 CC1=C(c2cc(C(=O)NCCc3cccn3C)c3ccccc3c2)CCCC1 c1(C(=O)NCC2(O)CN(C(c3cnoc3C3CCOCC3)=O)C2)cncc(F)c1 C#CCCC(C(=O)OC1CCN(C(=O)OCC)CC1)C(F)(F)C(F)(F)F C1(CC(=O)NC(CC)CN2CCCC2)CN(C(C2(C(F)F)CCCC2)=O)CCO1 CC(C)(O)C#CC(=O)NCC1COC(CNC(c2ccc(C3CCC3)nc2)=O)C1 c1(NC2CC(CC)C2)cc(NCC2CCC(C)(C)O2)nc(C)n1 Cc1nc(NC(c2snnc2C)C)cc(=NCc2ccc(C(F)(F)F)c(C)n2)[nH]1 C(=O)(CCCCC(C)(C)C)N1CCCC(C(N(C2CCN(CC)C2)C)=O)C1 C1(Cl)(C(N2C(CNC(C3NC(=O)C(F)C3)=O)CC2)=O)CC2CCC1O2 Cn1cc(S(N)(=O)=O)c(C(N2CC(CNC(C34CCCCC3OCC4)=O)C2)=O)n1 C1(C)(C(=O)NCc2c(C(=O)NC(c3ccccn3)CC)n[nH]c2)CCC(C)C1 c1(C(N2CC(NC(C3ON=C(C)C3C)=O)C(C)C2)=O)cc(Br)cnc1O N1(C(=O)OC(C)(C)C)CCCC2CN(C(=O)Cc3ncsc3)CCC12.C(F)F C(=O)(CC1=NN(C)C(=O)C1)N1CC(CC(C)NC(c2cnc3sccn23)=O)C1 N1(C(C2N(C)CC2)=O)CC2CC(C1)CN(C(=O)Cc1c[nH]c3cnccc13)C2 c1(C(N2CC3C(C(=O)Nc4c(OC)cccc4)(C3)C2)=O)cc(C#N)ccc1F C1(C(=O)NCC(C)NC(=O)CCc2cn[nH]c2)CC12CCc1ccccc12 C1(C(=O)NCc2c(C(N(CC(C)C#N)CC)=O)con2)CCN(C)C(=O)C1 c1(CN(CCCN(C(=O)Cc2cc(C3CC3)sn2)C)C)cc(F)ccc1F n1(CCC)ccc(C(=O)NCC(C)(CO)NC(c2ccsc2C)=O)n1 c1(CC(N2CC(O)(CNC(c3cc(O)nc(Cl)c3)=O)C2)=O)ccccc1[N+](=O)[O-] c1(CN(C)C(C2CC(N(C)C(C3CCN3C(C)(C)C)=O)C2)=O)ccoc1 C1(CCOC)CN(C(C2CNC(=O)O2)=O)CCN1C(c1ccsc1OC)=O c1(C(C(=O)N(CCNC(c2c(C)occ2)=O)C(C)C)C2CC2)ccc(F)cc1 C1(c2nnnn2C)(c2ccccc2)CC2(CCNC2)C1.CCCCC(CC)N N1(C(=O)COC2CCOC2)CCC2(CC1)CCN(C(C1CCCC(CF)C1)=O)C2 C1(C(=O)NC)CCN(C(=O)CC(C)CNC(=O)CC23CCCC2C3)C1C c1(C(=O)NCC(C)NC(CNS(CCCC)(=O)=O)=O)nc(C)ccc1C c1(OC)ccccc1C(C)CC(=O)NC(C)CCNC(c1ccc(C(N)=O)o1)=O N1(C(C2CN(C(N)=O)C2)=O)CC(CNC(c2ccnc(O)c2)=O)C(C(F)(F)F)C1 C1(CC=C)(C(=O)Nc2cncc(C)c2)CCN(C(=O)CC(C)(C)OC)C1 C1(CN(C(=O)CN(C)C(=O)C2CC2)C)CN(C(C2(C)CCOCC2)=O)CCO1 c1(C(N2CCCC(NC(c3cc(C(C)C)n(C)n3)=O)C2)=O)ccc(S(C)=O)cc1 Cc1cc(C)n2nc(C(N3CCC(CNC(C4(C)CC=CC4)=O)CC3)=O)cc2n1 CCCCCCCCNC(c1ncc(COC)s1)c1nnnn1C1CCC1 c1(C(N2CC(C=C)(CC(N3CCC(C)(C)C3C)=O)C2)=O)cnn2ccc(Cl)c(F)c12 c1(C(=O)NCC2N(C(C(C)N(C)C)=O)CC(O)C2)cccc2c1C(=O)CC2 CC(C(F)(F)C(F)(F)F)=CC(=O)N(CC(C)(C)NC(C1CC(C(C)C)C1)=O)C N1(C(c2c(OC)scc2)=O)CCN(C(=O)COc2cc(F)ccc2F)C(CF)C1 CCCCC(C(=O)NCCCCN=[N+]=[N-])NC(=O)Cn1ccc(C)c1.O(N)CC N1(C(CC)=O)CCCC(C(=O)NCC(O)CNC(c2cnn(C3CC3)c2)=O)C1 C=C1CCN(C(C2CC3(CCC3)C2)=O)C(C(=O)NC2CN(C)CC2(F)F)C1 C#CCC(CC(F)F)C(=O)NCC1CCC2(CN(C(C3COCOC3)=O)C2)O1 C12(NC(CN3C(C)CC3)=O)CCOC(CNC(c3cc[n+]([O-])cc3)=O)(C1)C2 Cc1cc2[nH]c(C(N3CC(CO)(NC(=O)Cn4nc(C)c(C)c4C)C3)=O)cc2o1 C1(CC(=O)N(C(CC#C)C)C)CC(C)N(C(=O)Cc2cnn(C)c2C)C1 C=CCC(CC=C)C(=O)NC(CN(C(c1cnc(C(F)F)s1)=O)CC)CC CCCCCCC(C)C(=O)N1CCC12CN(C(C1CCCS1(=O)=O)=O)C2 c1(C(N2C3CN(Cc4ccc(C)c(C)c4)C(C3)C2)=O)c(F)cc(F)c(F)c1F C1(NC(C(=C)F)=O)CCCC(CNCc2ccc(F)nc2)C1 CC(F)(F)CCC(=O)Nc1cccc(NC(C23CC(C(=O)N(C)C)(CO2)C3)=O)c1 C(=O)(C(F)(F)C1=CCOCC1)N1CC(CNC(C2(N(C)C)CC2)=O)C(F)(F)CC1 C1(C(=O)NCC(n2cccn2)C)(N(C)C)CSC1.C12CC(C1)C(=O)N2 C1(NC(C2(C(=O)NC)CCC2)=O)CN(C(=O)COCCOC)C2(CCCCC2)C1 O=C(CC1CSCCO1)NOCC=CCl.N1(C=O)CCC1 C1(N(C(CC2(NC(C(CN(C)C)O)=O)CCC2)=O)C)CCCC1(F)F C(=O)(CN=c1cc[nH]cc1)NC(CNC(c1c(OC)n(C)nc1)=O)C(C)C(C)C Cn1cnc(C(=O)NCc2ncoc2CNC(=O)Cn2cc(C#N)cn2)cc1=O c1(C(N2CCN(C(c3cccc(Cl)c3F)=O)C3C2C3)=O)cnc2c(F)cccn12 N1(C(C2CCN(C(C3CN(OC)C(=O)C3)=O)C2)=O)CCC2(CC1)CC2C#N CC(CC(=O)NC1CN(C)C1)NC(=O)CN(C1CCCC1)C C(=O)(C(C)(C)CN=c1[nH]c2c(c(=NCc3cnc(Cl)cc3C)[nH]1)COC2)NC C1(CNC(c2n(C)ncc2)=O)CN(C(c2ccc(O)c(F)c2)=O)CCC12CCC2 C1(O)(C(CNC(C(C)SC)=O)(C)C)CN(C(c2ccc(C)[nH]2)=O)C1 C1(C(=O)NCC(C)C(=O)N(C)CCn2cnnc2)CCC(=O)N1C N1(C(C=C(CCC)C)=O)C2CCC1C(C(=O)NC13CC(C)(C1)C3)C2 c1(CNC(C(C)(F)F)CCO)cc2cc(Br)ccc2s1 C1(CC=C)(NC(c2ccnn2COC)=O)CCN(C(=O)C(COC)N(C)C)C1 C(N=c1[nH]c(=N)[nH]c(=NC(C)C2CCOCC2)[nH]1)c1c(C)coc1C N1(C(c2c(F)cc(OC)cc2F)=O)CCOC2CN(S(=O)(=O)CCN(C)C)CC12 C(=O)(C1CCc2ccccc21)NC(c1cn(Cc2c(C)cc(Br)s2)nn1)(C)C Cc1cccnc1CNC1CCC(C(=O)Nc2ccnn2Cc2ccccc2)C1 C(=O)(CCCCN1CCCC1)NC1CC(NC(COC)=O)C1 C1(C(=O)NCC(CN(C(C2CC(=C)C2)=O)C)O)Cc2cc(OC)ccc2O1 C1(NC(C(Cn2cncn2)NC(c2n(CC)ncc2)=O)=O)CCCC12CC2 c1(C(=O)NCCNC(C2(c3cncnc3)CCCC2)=O)cc2n(n1)CCCC2O N1(C(c2c(C)snc2)=O)CCC(C)(CNC(c2cscn2)=O)CC1 C1(C(N2C(C(=O)NC3(CCOC)CCCC3)C(C)C2)=O)CN(C)CCN1C N1(CC(N2C(C(C)NC(COCCCOC)=O)CCCC2)=O)CCCCS1(=O)=O c1(CC(C(N2CC(c3cn(-c4c(C)occ4)nn3)(O)C2)=O)C)ccc(F)c(F)c1 c1(CC)ccc(C=CC(=O)NCC2C(C)CCN2C(C2CC(C)OC2C)=O)o1 C(=O)(CCCC(C)(C)C)N(CC(CNC(CNC(CCC(C)C)=O)=O)C)C C#CCCCCCC(=O)N1CC2CCC1CC2NC(C1CCC(CC)CC1)=O CCCC(CC)CCC(=O)NCC(C)N(C(=O)CN1CCCC(N(C)C)C1)C N1(C(C(C)NCCCCCO)=O)CC2C(C1C(=O)NCc1ccccc1)C2(C)C C1(C(=O)NC(CCN(C)C(C2(N(C)C)CCC2)=O)c2cccs2)CC(Cl)(Cl)C1 N1(C(COc2c(C)ccc(C)c2)=O)CC2CCC1C(NC(=O)C=CC1CCCO1)C2 N12CC(C)CC1C2=O.Cc1nocc1C(N1CCC(N(C)C)C1)=O C1(NC(=O)C2CC2)CC(O)CN(C(=O)C(c2ccc(Cl)cc2)(F)F)C1 CN1CCc2cc(CC(=O)NC3CCOC(CNC(C4CC=CC4)=O)C3)ccc21 c1(CNC(=O)CONC(=O)C2(CC=C)CCC2)nccc(C)n1 C1(NC(CC2(C)N(C(c3c(C)noc3N)=O)CC2)=O)CC2(CCOC2)C1 N1(C(CN(C(C(CC)O)=O)C2CCC2)=O)CC(O)CC12CCCC2 N1(C(C(C)OCCOCCOC)=O)CC(CNC(=O)CCOC)CC(C)C1 O=C(C1CCCn2ccnc21)NC1C2CCN(C(C3(CF)CC3)=O)CC12 CC1OCCC1N=c1[nH]c(=NCCn2ccnn2)c2cc(Cl)ccc2[nH]1 N1(C(C(C(C)C)OC)=O)CC2CCCC1C2CNC(c1csc(O)n1)=O c1(OC)cnc2[nH]c(C(=O)N(C(C)CNC(=O)C=C3CCC3)C)cc2c1 c1(C(=O)NCC2CCCC2O)ccc(C(=O)NC2CC(OC)C2)cn1 C(=O)(C1=CCCCCC1)NC(C(C)C)C(=O)N1CC(F)(F)C1C1CC1 N1(C(C2(C)CC(C)(C)C2)=O)CCC(CO)C(NC(=O)Cc2cncc(C#N)c2)C1 N1(C(C2C(CC(C)C)C2)=O)CCOCCC1C(=O)NCCCC1CCOC1=O C(=O)(CC(C)CC(C)(C)C)NCC(c1ccccc1)NC(c1c(CC)onc1)=O Cc1onc(C2CC2)c1C(N1CC(F)(CNC(c2snc(O)c2Cl)=O)C1)=O C1(COC)(CNC(C2C=CCC2)=O)CCCN1C(c1n[nH]cc1Br)=O C(C(C(=O)NCC1(NC(C2COC(=O)N2)=O)CC1)n1cc(CC2CC2)nn1)OC Cc1cccc(C(N2CCC(C(F)C(=O)NCCCSCCO)C2)=O)n1 C1(C)(C(=O)NCc2c(CN(C)C(C3OCCCO3)=O)cccc2)CCCS1(=O)=O C1(NC(c2ccc(CO)o2)=O)CCCC1C(=O)N(C1CCOC1=O)CCF C1(C(=O)NCC(Cc2ccccc2)N(C(CCOC)=O)C)CCN(C)C1 C(=O)(C(CC(C)C)NC(=O)CC1CC2CCC1O2)NCC1CN(CC)C(=O)C1 N1(C(C(CC)NC(N)=O)=O)C2CCC1CC(C(=O)N(C(C)C(=O)NCC)CC)C2 C1(C(=O)NCc2c(C(=O)NCC(C3CCCC3)C)n[nH]c2)CCC(F)(F)C1 C1(NC(C(c2nc(C)sc2)=O)=O)CS(=O)(=O)C2CN(C(=O)C(C)(C)C)CC12 N1(CC(C)C)CC(C(=O)NC(CNC(c2c[nH]c(Br)c2)=O)C(C)C)CC1=O c1(C(N(C2CCCC2)CCNC(COCCC#C)=O)=O)cc(C)ccc1F C(c1ccccc1)=CC(N1CCC(COCCCCCn2cc(C3CC3)nn2)C1)=O CC(C(C)C(=O)NCC(C)(C)CN(C)C)NC(=O)CC1CCCCCC1 c1(C(=O)NC(CCN(C(c2ccc(SC)o2)=O)C)C)ccncc1F c1(C(N2CCN(C(C3C(CC)C3)=O)C(CO)C2)=O)cc2ncc(Br)cc2o1 C1(C(=O)NCC2(C)CC(CN)C2)CCCC(C(F)F)C1 C(=O)(CC(CN(C)C)C(F)F)NC(C(C)C)CCNC(=O)CCCc1nccs1 C1(C(=O)NC(C)Cc2nncn2C)CC(C)CN1C(C1CCCCC1O)=O c1(C(N2C(CNC(C3OCCN(C(C)C)C3)=O)CCC2)=O)cc(S(C)(=O)=O)cs1 N#Cc1ccc(C(=O)NCCC2CCN(C(C3C=CCC3)=O)C2)nc1 N1(C(c2c(C)oc(C(C)C)n2)=O)CCN(C(=O)CC2CCC3CC23)CC12CC2 CC1(NC(=O)C2=CCCC2)CCCCC1C(=O)NCC(C1CCCC1)O N1(C(C2(NCC=CC)CCC(C)C2)=O)CC2C3COCC3C2C1 Cc1cc(Br)c(NC(=O)CCC2CCCN2Cc2c(F)ccc(C)c2Br)c(Br)c1 C(CC(C(=O)OC)NC(C1CCCN1C(=O)C(C)NC(=O)NC)=O)=CC N1(C(c2c(C)cco2)=O)CC(NC(C2CN(CCOC)CCO2)=O)CC1COCC C1(O)(CN(C(COC(C)C)=O)C)CCN(C(=O)CSC2CCOC2=O)CC1 c1(C(=O)NC2(CF)CCN(C(C3(C(F)(F)F)CC3)=O)C2)cccc2nsnc12 Cn1c(=O)n(CC(=O)NC2CC(CNC(C3SCCS3)=O)C2)c2ccccc12 Cc1occc(=O)c1OCCOC1CCN(C(=O)CC(F)(F)F)CC1 CC1CN(C(=O)CCCC(F)F)C(C)CN1C(=O)Cn1cc(F)ccc1=O C1(NC(CC(=C)C)=O)CCCN(Cc2cc(C(=O)OC)ccc2Br)C1C c1(C(=O)NC23C(CN(C(c4scc(C)c4)=O)C2)C3)cc2ccccn2c1 c1(NCC(C)C2CCC2)cc(=NC2COc3ccc(Cl)cc32)[nH]c(C(F)(F)F)n1 c1(C(N2C3C(NC(=O)C=Cc4ccc(F)cc4)C(C3)C2)=O)ccc2n[nH]cc2c1 C1(CNC(C2(N(C(CC=CC)=O)C)CC2)=O)CCC(=O)N1 c1(C(N2CCC(CNC(C(CC=C)CC)=O)(OC)C2)=O)c(C)cc(O)nc1C CC(=O)CCCC(C)C(=O)NCC1(C(=O)NCC(O)CNC(N)=O)CC2(CC2)C1 N1(C(C(N)=O)=O)CCC(NC(C2CCC(=O)N2)=O)C12CCCC2 C1(C)(C(N2CC(NC(C(c3ccc(N)cc3)C)=O)C2)=O)CCC(=O)CC1 C1(NC(CCC#CC)=O)CC2CN(C(c3cscc3C(F)(F)F)=O)CCN2C1=O N1(C(C2CCCC(NCc3ccc(OC)cc3OC)C2)=O)CCCC(C)(O)CC1 c1(OC)ccc(Br)cc1-c1cn(CC2CC(CCNC(=O)C(C)(C)OC)C2)nn1 C1(NC(c2ccc(OC)nn2)=O)CN(C(=O)Cc2cc(F)ccc2F)CCC1C C1(NC(c2ccc(C(C)C)nc2)=O)CCC(C)N(C(c2ccc(Cl)s2)=O)C1 CCC(C)(C#N)C(=O)NCC1(C(N)=O)CN(C(=O)CC2(C)CCOCC2)C1 c1(C(N(C)CC2(C)CCC2)=O)c(NC(CC2(CSC)CC2)=O)noc1C N1(C(c2ccc(CC)nc2)=O)CC(C)C(C)(C(=O)NC2CCC(F)CC2)C1 N(C1CCc2cccc3cccc1c23)C1C2CN(C(C(=O)N(C)C)=O)C1C(O)C2 N1(CCCC)CCOCC1C(=O)NC(CNC(c1oc(C)nc1C)=O)CO c1(OC)cc(C(N2CCC(N3CCCC3)C2)C(=O)NCC2CCC2)cc(Cl)n1 c1(C(=O)NC2C(C(N(CC(C)CO)C)=O)CC=CC2)cc2ccccc2[nH]1 C1(C(=O)NCC2(c3c(C)cccc3)CC(OC)C2)CC(c2cccc(F)c2)=NO1 N1(C(C(c2ccoc2)NC(c2c(C)nc(C)nc2)=O)=O)CCN(C)CC(C)C1 Cc1noc(C(N2CCCC(CNC(C3(C)CCCC3)=O)C2)=O)c1C N1(c2nnc(C)o2)CCCC(C)(CNC(=O)Cc2c(C)noc2C)C1 C1(NC(c2c(CC)nns2)=O)CCN(C(=O)CC2CCCCC2C)C12CCC2 Cc1cccc(-n2cc(C3CCN(C(=O)CCc4ccccc4)C3)nn2)n1 N1(C(C=Cc2cc(C)no2)=O)CC2(CC(CNC(=O)CSc3nc[nH]n3)C2)C1 c1(N2CCC(O)(C(C)NC(=O)Cc3ccoc3)CC2)ncc(S(C)(=O)=O)cc1Cl N1(C(C=Cc2ncn(C)c2)=O)CC2CC(NC(C3CC34CC4)=O)C2C1 Cc1ccc2nc(C(=O)N(C)CCN(C(=O)C=CC3CCCO3)C)ccc2c1 N1(C(C(C)c2ccco2)=O)CCC2C(CCN2C(N(C)C)=O)C1 c1(OC)cnc(Cl)c(CN(C2CCN(Cc3ccc(C(=O)OC)cc3Cl)C2)C)c1 C12(C(=O)Nc3cnc(COC)nc3)CCC(C(=O)Nc3ccncn3)(CC1)CC2 Cc1cc(C(=O)NC2CCC(CNC(=O)Cc3cnn(C)c3)C2)sc1Cl c1(-c2n(CCCOC)nc(-c3ccccn3)n2)cnc2n1CCC2 Cc1sc2ncnc(N(C(C)CNC(c3cc4ccc(F)cc4s3)=O)C)c2c1C C(=O)(CC(F)(F)Cl)N(C1CCN(C(=O)C(C(C)C)SC)C1)CC N1(C(C2N(C)CCC2)=O)CCC2C(CCN2C(=O)Cc2ccco2)C1 Cc1ccc(C=CC(N2CCN(C(=O)CCS(C)=O)C(C)C2)=O)c(C)c1 N1(C(CC(C=C)C)=O)CCC(O)(CN(C)C(C2CCCS(=O)(=O)C2)=O)CC1 N1(C(C2C(C)(C)C2)=O)CCC2(CC1)CC2CNC(c1ccoc1)=O N1(C(C(CC2CC2)OC)=O)CCC(CNC(C2(C)CNC(=O)C2)=O)C12CC2 c1(C(N2CC(NC(=O)CCN3CCCC3)C3(C2)CC3)=O)cc2cccnc2s1 N=c1[nH]c(C(F)(F)F)ccc1C(N1CC2CC2(CNC(=O)C=C2CCC2)C1)=O CC1C(C)N(C(c2ccc(CO)cc2)=O)CCN1C(c1ccncc1Cl)=O c1(C(N2CC(CNC(C3CC(F)C(=O)N3)=O)C2)=O)ccc(F)c2ccncc12 Cc1ccc2c(CC(=O)NCC(C)(CO)NC(C3CCCOC3)=O)coc2c1C CCC(CC(C)C)C(=O)N1CC(CF)(NC(=O)CN2CC=CC2)C1 C1(CC(=O)NC2(C(=O)NC3CCN(CCOC)C3)CCC2)CCC(C)(C)C1 c1(C(=O)NCc2cn(CC(C)NC(=O)CC3CC3)nn2)ccc2nnn(O)c2c1 C1(C(=O)NCCCCC2C(C)C2)CCCCCCN1C(=O)CC1CCCC12CC2 C1(CC)CN(C(c2cc(Cl)ccc2F)=O)CCN1c1nc(C2CC2)ncc1F N1(C(c2onc(CC)c2C)=O)CCC2(C1)CN(C(c1ccnc(OC)c1)=O)C2 C1(C(=O)NCC(CNC(c2ccc(CC)cc2O)=O)OC)CCc2c[nH]nc2C1 c1(CC(N2CC(C(N)=O)(CNC(C(CC)C)=O)C2)=O)coc2cc(OC)ccc12 Cc1cc(=NCCCCC(C)NC(c2cc(C)n(C)n2)=O)[nH]cn1 C1(COC)CCN(C(=NCCCCl)NCc2cc(CO)ccn2)C1.C(N)(=O)N c1(C(=O)NC2CC(C)N(C(=O)Cc3ccns3)CC2)ccc2cnccc2n1 C12(NC(C(N3CCC(C)CC3)=O)=O)CCC1CN(C(c1cc3n(n1)CCC3)=O)C2 CCCCCC(O)C(=O)NCCCC1(NC(=O)Cc2ccc(C)nc2O)CC1 n1(CC(=O)NCC2CC(CNC(=O)CC3CC=CC3)C2)ccc(C2CC2)n1 c1(CC(=O)NCC(CNC(C(N2CCC(O)CC2)C)=O)OC)ccnc(O)c1 CN1CCCC1CCC(=O)NCC(C)(C)NC(c1cc(-c2ccccn2)no1)=O c1(CC(N2CCN(C(c3nc(C)c(C)s3)=O)CC2CO)=O)ccc2c(c1)CCO2 C1(NC(c2cc(C(=O)OCC)on2)=O)CCOCC1NC(=O)C(C)=C(C)C N1(C(C(CCCC)O)=O)CC2CCN(C(c3ccc(S(C)(=O)=O)[nH]3)=O)CC2C1 N1(C(c2cnc(C)o2)=O)CC2(CCCC2NC(c2c(C)n[nH]c2C)=O)C1 CCC(C)C(C)CNC(=O)C(C)(CO)NC(=O)CN1CCNC(=O)C1 CS(=O)(=O)c1ccc(C(=O)NCC2CC(NC(=O)CC3(CO)CC3)C2(C)C)o1 c1(C(=O)NC(C(=O)OC)(C)C2CCCO2)ccc(C(C)(C)C)nc1 CC(C)C(CNC(=O)COC(F)(F)F)NC(=O)CCOC1CCCOC1 C1(C(=O)NC(CCOC)CNC(=O)Cc2cc(C3CC3)no2)CCC(=O)N(C)C1 C1(CN(C(c2c[nH]c(=NC)s2)=O)C)CCCN(C(=O)C(C)(C2CC2)OC)C1 c1(C(C)C)nc(NCC(Cl)(Cl)Cl)cc(=NC(C(C)(F)F)c2ccccc2)[nH]1 c1(NC(CNC2(c3nnnn3C)C(C(C)C)CC2)=O)cc(F)c(F)cc1F Cc1ccc(C)c(CNC(=O)C=CC(C)NC(C2CC3CCC3C2)=O)n1 C1(C(N2C(C(N3CCC(O)(COC)C3)=O)CC(O)C2)=O)CC2(C1)CC(C)C2 C(=O)(C(C)(C)C1CCCC1)NC1C(CNC(CCOC)=O)C1 c1(CCNC(C(n2cc(CC(C)(C)CO)nn2)C)=O)ccc2ocnc2c1 Cc1ccnc(C(N2CC(CF)(NC(=O)CCn3cccc3)C2)=O)c1 C(c1ccc(=N)[nH]c1)=CC(N1C(CNC(C2CCN(C(=O)NC)CC2)=O)CC1)=O C(C(=O)NCCC1(CO)CCC1)(C(C)CC)NC(c1c(CC)oc(C)c1)=O N1(C(C(CCC2CC2)NC(c2cc(C3CC3)on2)=O)=O)CCCCCCCC1 N1(C(c2c(C)cccc2O)=O)CCC2(CO)CN(C(=O)Cc3cnns3)CC2C1 c1(NC(=O)NCc2cn(CC)nn2)ccc(C(OCP(C)(C)=O)C)nc1 N(C1CC(F)(F)c2ccccc21)S(c1cccc(N(C)CCC2CCC2)n1)(=O)=O S(=O)(=O)(C=Cc1ccccc1)N1CCC(CC(=O)Nc2ccc(Br)nc2Cl)CC1 c1(CC(N2CC(C(C)NC(=O)CCCC3CC3)C2)=O)ccc2cnccc2c1 C(=O)(C(O)CCCC)NC(CC#C)C(=O)NCC1(C)CC2(CC2)C1 C1(=O)C2=NN(C(=O)CC2)C(C)C1=O.c1(CCC)nsc(CO)n1 N1(C(C2C(C)CC(=O)N2)=O)CC2C3CCC(C2C1)N(C(C1CCCSC1)=O)C3 C1(NC(c2nccc(C)n2)=O)CC2CC1N(C(=O)CC1C(C)(C)C1(C)C)C2 C1(NC(Cc2c(C#C)cccc2)=O)CCCC2CN(C(=O)C(O)C3CCC3)CC12 CCC(CNC(=O)C(c1cccc(OC)c1)C)(CC)NC(C1CC1C1CCC1)=O c1(CC(N2C(CC)C(NC(=O)Cc3c[nH]nc3O)CC2)=O)ccc(F)c(Cl)c1 C(=O)(C1=CS(=O)CCC1)NCC1CCC(NC(C(CC)N(C)C)=O)CC1 O=C(C1CCCc2nc[nH]c21)NCC1CC(NC(C23CCC(CC2)C3)=O)C1 Cc1cc(S(=O)(=O)NCC2CCCC2C(=O)O)sc1Cl C(=O)(C1c2ccc(Br)cc2CCN1C(=O)C(O)C1CCCC1)OC C1(C(=O)NC(C2CCN(C(COCc3cnc(C)s3)=O)C2)C)CCOC(=O)N1 C1(N(C(COCCCCCC)=O)C)CCC2CN(C(=O)C(C)OCC(C)C)CC12 N1(C(c2ccn(C(C)C)n2)=O)CC(NC(C2(c3cc[nH]n3)CCC2)=O)CC(O)C1 c1(CC)nn(C)cc1C(=O)NCCN(C(C1CCCSC1)=O)CC c1(N(CCOCC)C)nc(=NC)nc(NC(C)COC(F)(F)F)[nH]1 C1(CCNC(C2(F)C(C)C2)=O)CSCCN1C(c1cncc(OC(F)F)c1)=O N1(C(c2cccc(-c3cn(C)nc3)n2)=O)CCC2(CCN(C(=O)CNC=O)CC2)C1 C1(C(=O)NC2(CC=C)CN(C(c3cc(CO)oc3C)=O)C2)NC(=O)OC1C C1(NC(C2(c3cc(C)no3)CC2)=O)CN(C(=O)CC2CCCCC2C)CC1(C)C C(=O)(C(C)(C1CC1)NC(c1ccn(C(F)F)n1)=O)NC(C1(C(=O)OC)CC1)C N1(C(C=Cc2ncn(C)c2)=O)CCN(C(=O)CC(C)(C)C)C2CCCCC12 N1(c2n(C)c(Cc3nc(Br)c(Br)n3C)nn2)CCC(F)C(O)C1 CCCCC(C)C(=O)N1CCCC(NC(=O)Cc2coc(C(F)F)n2)C1 C(=O)(C(C(C)(C)C)N(C)C)NC1(C2N(C(c3cccc(SC)n3)=O)CCC2)CC1 c1(C(N(C2CCC(NC(C=C3CCC(C)C3)=O)CC2)C)=O)cnc2[nH]cncc1-2 C#CCCCCC(=O)N1CC2(CC(NC(C3(CF)CCC3)=O)C2)C1 c1(C(=O)NCC2C(NC(C(CC)OC)=O)CCC2)[nH]c(C)c(C(=O)O)c1CC C#CC(CNC(=O)CCC1CCN(C(c2cnn(C)c2C)=O)C1)CC(C)(C)C c1(CN2C(C(=O)Nc3cc(O)nc(CO)n3)CC2)ccc([N+](=O)[O-])cc1 C=C=CC(C)C(=O)N(C1CN(C(=O)C(C)Nc2nc(C)cs2)C1)C C(=O)(C(C#N)C(C)(C)C)NCC(C)NC(C1(O)CCSCC1)=O N1(C(C(C(C)NC(C2CCCCO2)=O)(C)C)=O)CC2(C)CC1CCO2 N1(C(C(C=C)OC)=O)CCC(O)(CNC(=O)C(C)(C)C=C)CC1 C(=O)(C(C)(O)C(F)(F)F)NCCC1CCCN(C(C(C)=C(CC)C)=O)CC1 c1(NC(C)C=CC(=O)OC(C)(C)C)ccc2nnc(O)n2c1 c1(CC)cnc(C(=O)NCC2CCCC2C(=O)N(CC(C)(C)COC)C)nc1 c1(C(=O)NCC(C)N(C(c2cn(C)nc2C)=O)CC)ccc(S(N)(=O)=O)o1 c1(NC(C2C3CN(C(C(CCC)C)=O)CC32)=O)c(Br)cc(Br)cc1[N+](=O)[O-] CCCCC(O)C(C)C(=O)N1CC(C(C(N2CCC(OC)CC2)=O)OC)C1 C1(O)(CNC(C=C(C)C)=O)CCN(C(=O)CSCC(c2ccccc2)C)C1 c1(C(N(C2CCCCN(C(C3(CC=C)CC3)=O)C2)C)=O)ccc2c(c1)ncn2C C1(CNC(c2c(OC)ccc(C)c2)=O)CC2(CCN(C(=O)CC3C=CCC3)CC2)C1 c1(CC(=O)NCC(C)CN(C(=O)C(F)(F)CO)C)ccc2nc(O)[nH]c2c1 c1(C(N(C2CCCN(C(C3CC4CC4C3)=O)C2)C)=O)c[nH]c2cc(O)ccc12 CN1NC2=NC(c3ccc(Br)c(Cl)c3)C1=C2.N1CCCC(N)C1 c1(C(N(C(C(=O)OC)C)C)=O)cnc2ccc(C#N)cn12 c1(OC)cscc1C(=O)NC1(CC(=O)N(C(C)CC2CC2)C)CC1 c1(NS(C)(=O)=O)ccc(C(=O)NC2CC(NC(=O)CSc3ccccn3)C2)nn1 CC(C)CC(C(=O)NC1CCN(C2CC2)C1)ONC(=O)CCc1ccccc1 c1(CC)c(C(=O)NCC2(C)CCCN2C(=O)CC2C=CS(=O)(=O)C2)cnn1C O=C(C1=CC2(CCN(C(=O)Cn3cnnn3)C2)C1)NC1CC(F)(F)C1 n1(C(C)C)ccc(C(=O)NC2CN(C(C3(C(C)C)CC3)=O)CC2C)cc1=O Cc1cccc(CC(=O)NC(CCNC(=O)C(C)Cc2ccnn2C)C(C)C)c1 C1(CNC(C(C)=CC)=O)CCN(C(=O)C(COC)N(C)C)CC1 C1(NC(c2ccsc2)=O)CC2CC1CN2C(c1cnc(C2CCOCC2)s1)=O C12(NC(C3CC(C#C)(O)C3)=O)CN(C(=O)CNC=O)C(COC)(C1)C2 C=CC1CN(C(=O)CC2CN(C(c3nc(Cl)cs3)=O)CCC2C)CCO1 c1(C(C)NC2CCC2)ccc(CN(c2ccnc(N3CCCCC3)n2)C)cc1 c1(C(N2C(CN(C)C(c3ccc(Cl)s3)=O)COCC2)=O)nncc2c1CCCC2 C12(C(=O)NCCCP(C)(C)=O)CCCC1CCN2C(c1cc(C2CC2)[nH]n1)=O c1(C(=O)NC2CC(NC(c3n(CC)ccc3)=O)C2)ccc(Br)cc1 CC1=C(C)CC(C)(C(N2CCC(CNC(=O)C=CS(C)=O)CC2)=O)CC1 c1(C(=O)NCC2(NC(C3C(C)(C)CC3)=O)CCC2)ccc2sc(=N)[nH]c2c1 C(=O)(CC(C)CC(C)(C)C)N1CC(NC(c2c(C)nns2)=O)C2(C1)CCC2 C(=O)(C(F)C(=O)NCC1(NC(C2CCN2CC)=O)CC(F)(F)C1)OCC CC1C(NC(=O)CC2CCCS2(=O)=O)CCN1C(C12CCC(C1)C2)=O CCC(C)C(C(=O)NCCC(O)CCC)NC(C1CCN(C)C1=O)=O c1(C(=O)NC2(COC)CN(C(C(C=C=C)C)=O)C2)cc2c(F)cc(F)cc2o1 C1(NC(=O)Cn2nccn2)CC(CO)N(C(c2c[nH]nc2Br)=O)C1 S(=O)(=O)(c1ccc(F)cc1)NCC(N1C(C)CCCC1C)=O c1(C(=O)NC(C2CCOC2)CNC(c2c(OC)c[nH]n2)=O)cc(Cl)cc(Cl)c1 CN=c1[nH]nc(CC(=O)NC(C)(CNC(c2ncncc2Cl)=O)C2CC2)s1 c1(-c2nnc(CN(C(=O)NCCCl)Cc3cccnc3O)o2)ccc(Cl)cc1 c1(C(=O)NC(C(=O)NC2(C=C)CCCC2)CC2CCCC2)c[nH]c2nccc-2c1 CC(C(F)C(=O)N1CC(CNC(=O)C2=NOCC2)OC(C)(C)C1)C(F)(F)F c1(C(N2CCN(C(c3c(C#C)c[nH]n3)=O)CC2C(C)C)=O)cc2c(ccn2C)s1 c1(C2CCCN(c3cc(NCCN(CCC)CC)ncn3)C2)cccc(C)n1 CC1(C)OCCC1(C)NCc1ccccc1Cn1cccn1 c1(C(C)C)nccn1CC(=O)NCCNC(C1CCCC1c1nncn1C)=O c1(CCC)nnsc1C(=O)NCCCN(CCCNC(=O)C(F)(F)C1CC1)C C1(C(N(c2ccc(F)cc2)C)=O)CC2CCC(C1)C2N c1(CCN=C(NC2CC(C)(F)C2)NC2CCCCC2)cccc2cc[nH]c12 N1(C(CCC2C(C)(C)C2)=O)CCCCC2(C1)CN(C(C1CC=CCC1)=O)C2 c1(C(N(C2CCN(C(C3C=CCC3)=O)CC2)CC)=O)cc(Cl)sc1Cl C(C(CCNC(=O)C(C)(C1CCC1)NC(=O)C(C)CSC)OC)OC C1(NC(=O)C=Cc2cnc[nH]2)CCCCC12CCN(C(C1(CO)CCCO1)=O)C2 N1(C(C(C)N(C(=O)C(C)n2cnnn2)C2CC2)=O)CCC(NC(COC)=O)C1 N1(C(N2CCCCC(CC)C2=O)=O)C2CCC1CC(=O)NC2 C1(CC(=O)NCCN(C(c2cnn(C)c2N)=O)CC)CCCC(F)(F)C1 C(=O)(C(C(C)C)NC(N)=O)NC(C1CCOC1)CNC(C1(CC=C)CCC1)=O N1(C(c2cc(C)[nH]n2)=O)CCN(C(c2c(F)ccc(C)c2N)=O)CC(CO)C1 N1(Cc2c(OC)ccc(O)c2)CC2CCN(C(c3ccc(I)cc3O)=O)C2C1 N12CCC3CC(C3C1)C2=O.N1(CCN)CCC(C(C2CCS(=O)(=O)C2)=O)CC1 c1(C(N2CC3C(NC(Cc4n[nH]c(=NC)s4)=O)C(C3)C2)=O)cc2c([nH]1)CCOC2 Cc1cc2c[nH]nc2cc1C(=O)NCC(C)N(C(=O)CCC1CCC1)C C12(C(=O)NC(C)CC(=O)NCC3C4CCCCC34)CCC(C1)OC2C C1(NC(CC(C(C)C)O)=O)CC(O)(C2CCN(C(=O)CCn3ccnc3)CC2)C1 N1(C(C(N2CCNC2=O)C)=O)CC(C(=O)N(C2COCC2(C)C)C)CC1(C)C C1(NC(=O)NCc2cn(CCCCO)nn2)CC12CCOc1ccccc12 N1(C(C=CC2(C)COC2)=O)CC2COCCC2(NC(=O)CCC(F)(F)F)C1 C1(NC(=O)CCOC2CCOC2)CCC(C=O)CC1.CCC(CC)C1CC1 N1(N2CCC(Oc3ccc(OCCC)cc3)C2)CCc2nc(C=O)sc2C1.CC Cc1ccc(F)cc1C(F)(F)C(=O)OCCCOc1ccccc1C(F)(F)F Cc1cc(C(=O)N(C2CCC(NC(=O)C(F)(F)C3CCCCC3)C2)C)ns1 c1(CC)ccc2cc1NC(=O)N1C(CC1)C(=O)N2.C(C(F)(F)F)OC(C)=O C=CCC(CC)C(=O)N1CC2CC2(NC(C2C3CCC2(c2ccccn2)C3)=O)C1 c12ccc(cn1)[nH]c2=O.c1(CC(=O)NCCN(CCC)C(=O)NC)[nH]ccc1C n1(-c2c(F)ccc(C)c2)nc(C2COc3ccccc32)nc1C(C1CC1)C1CC1 c1(C(N(CC(CC)NC(c2cn(C)nc2OC)=O)C)=O)cccc(C(C)C)c1 CN1CC(NC(=O)CCC2CCN(C(C3C4CCCOC34)=O)C2)C(F)(F)C1 N1(C(c2c(OC)cc(C)cc2)=O)CCCC12CCCN(C(C1(CCF)CC1)=O)C2 N1(C(Cc2c(C)noc2C)=O)CC(C)CN(C(=O)CCOC2CCC2)C(C)C1 Cc1sccc1NC(=O)COC(=O)CCCN1CCCCC1 C1(NC(c2cc(CC)c(CC)o2)=O)CCN(C(=O)COCC2CCC2)CC1F c1(CC)cc(C(N2CC(NC(=O)C(c3cccc(O)c3)(C)C)C(C)C2)=O)n(C)n1 c1(CC)cnc(O)c(C(=O)NCC(C)(F)CNC(=O)CCc2cnn[nH]2)c1 C1(CNC(CCC2CCN(C(COCC(=C)C)=O)C2)=O)CCOCC1(C)C Cc1c(C(=O)NC23CC(NC(=O)COCC(F)F)(C2)C3)nn(C)c1N C(=O)(C1=CC2C=CC(C1)C2)N1CCC(O)(CNC(c2cscc2F)=O)C1 C(=O)(CCCC(C)NC(c1c[nH]c(=NC)s1)=O)NCc1c(C(C)C)ocn1 Cc1noc2cc(C(=O)NC3(CNC(=O)Cn4cccnc4=O)CC3)ccc12 C(=O)(C(F)(F)CCc1ccccc1)N1CCC(C)(NC(CC2C(C)C2)=O)C1 C1(NC(C2CCC(C)(C)C2)=O)CCCCCN(C(c2cncs2)=O)C1 CC1CCN(c2cc(C(F)F)ncn2)C1CNC(=O)CCC(C)N(C)C C(=O)(CCCCCC(C)C)NC1(C)CC(NC(c2cc(OCC)no2)=O)C1 c1(NC(=O)NC2(C)C=CCC2)c(C#N)sc2ncccc12 C12(C=O)CC3CC(C(=O)N1)C2C3.C1(OCC(=O)N(CCCN)C)CCCCCC1 S(=O)(=O)(c1cc(C(F)(F)F)ccc1F)NC1CCC(NC(C(C)O)=O)C1 CCC(CCCC(=O)N1CC2CC1CN2CC)NC(=O)CC1CCOC1 C1(NC(C(C2CCCCC2)OC)=O)C2CCC1N(C(c1cc(C)cc(C)c1)=O)C2 C1(CN2CC(CNC(Cc3c(C)ccc(C)c3)=O)C2)COc2ccccc2O1.C(C)C N1(C(c2ccc(C(Cl)Cl)cc2)C(=O)NCC(F)F)CCCC(C2CC2(F)F)C1 CCC(C)CCCC(=O)NC1CC(C)(NC(=O)CC2COCCN2C)C1 N1(C(C(=O)Nc2c(C)c(Cl)ccc2)C2CC=CC2)CCCC2(CNC(=O)C2)C1 c1(C(=O)NC23CCN(C(CCCCC)=O)CC2C3)ccc2nc(C)nn2c1 C1(C(N2CCCC(CN)C2)=O)CC2CCN(C(c3cccc(O)n3)=O)CC12 C1(CN(C(C2(C(C)C)CCC2)=O)C)CCCCN1C(=O)C=C1CCN(C)CC1 Cc1ccnc(C(=O)NCc2cccc(CNC(=O)Cc3ccn(C)n3)c2)c1 c1(OC)ccc(CN2C(C(=O)Nc3cc(O)ccn3)CC3CC23)c(OC)c1Cl C12(NC(C(CC)n3cncn3)=O)COC(C1)C(NC(c1ccc(=N)[nH]c1Cl)=O)C2 c1(CC(CNC(CCOCCOC)=O)NC(=O)C(C)OC)ccccc1C(F)(F)F c1(OC)ccc(COCC(N2CCC(CN(C(=O)CCCSC)C)CC2)=O)cn1 C1(NC(CC2(C=C)CCC2)=O)COC2CN(C(=O)CNS(C)(=O)=O)CC12 C1(C(=O)NCC(C(=O)NCCN2CCC3CC23)N(C)C)C2CC3C(C2=O)C13 c1(C(=O)OC(c2ccon2)C)cc(-c2ccncc2)no1 C1(CNC(c2c(C)n(C3CCC3)nc2)=O)CCN(C(=O)CCC2(C)CC2)C1(C)C c1(C(C(=O)NCC2N(C(CCC#CC)=O)CC2)(F)F)cc(F)cc(F)c1 N1(C(COC(CC)C)=O)CCC(C(C)C(=O)NCCN(C)C(C)C2CC2)C1 C1(O)(CC#C)CCN(C(=O)C=CC2CCCN2C(=O)CCc2cncn2C)CC1 C(CCCC(=O)N(C1CCCC1)CCCNC(=O)C(F)=CC1CC1)(OC)OC c1(CC(N2CCC(N(C(=O)Cc3cccc(O)c3)C)C2)=O)ccc2c(c1)CCC2 C1(NC(C2N(C)CC2)=O)CN(C(C2(C)CC(F)C2)=O)CC1c1cccc(F)c1 c1(C(C)=O)c[nH]c(C(=O)NCC(F)CNC(c2cnc(C(C)C)[nH]2)=O)c1 c1(SCC)cc(Br)ccc1C(N1CCSC(C(=O)Nc2ccc(F)c(F)c2)C1)=O Cc1nc(CC(C)C)oc1C(N1CC(NC(=O)N(C(C)C(C)C)C2CC2)C(C)C1)=O N1(C(Cc2n[nH]c(=NC)s2)=O)CCCC(NC(c2nc(C)oc2C)=O)C1C C1(NC(C2CN(CC)C2)=O)(CNC(=O)C2=C(C)CCC2)CCCCC1C C1(CC(=O)NCC2(O)CCN(C(C(=O)NCC)=O)C2)CSc2ccccc2NC1=O C(=O)(C1=CCCOC1)NCC1(C)N(C(C2C=C(C)CS2)=O)CCC1 N1(C(CC2(OC)CCCCC2)=O)CCC(NC(C2CCCS2)=O)CCC2(CC2)C1 O=C(CN=C(NCc1nccc(C(F)F)n1)NC1CC1)NC(=O)CCC(F)(F)F n1(CCC)cc(-c2cscc2CC(=O)NCC(C)F)cn1 Cn1cc2c(n1)CC(C(=O)NCCC1CC(NC(=O)CCc3cn[nH]c3)C1)CC2 C12C3CCCC1CN(C3)C2=O.N1(C(C)=O)CCC(C(=O)NC2CNC(=O)O2)CC1 CCC(CC(=O)NCCCN1CCC(CO)C1)NC(C1CN(C)C1)=O c1(C(N2C(C(N3C(C)(C)C(CO)C3)=O)CC=CC2)=O)cc2cccn2cn1 c1(C(=O)NC(CCCCNC(c2ccc(COC)o2)=O)C)cccc2nccn12 c1(OC)cccnc1C(N1CCCC1CCC(=O)NCc1cncn1C)=O C1(CNC(c2cn(CC)nc2)=O)CN(C)CCN1C(c1cnc(C(C)OC)s1)=O CCCCCCCCOCC(N1CCC(C)C1CNC(C1C2CCCC12)=O)=O CCC(C(C)(C)O)NC(c1cccc(CNC(c2cccc(O)n2)=O)n1)=O C1(C(C)NC(C=CCOC)=O)CN(C(c2cc(CSC)ccn2)=O)CCO1 C(=O)(C(C)CC(C)(C)O)NCCN(C(=O)CC(C(C)C)OC)CC CC(C)CCCCCC(=O)NCC1CC(C)N(C(c2cnc(O)n(C)c2=O)=O)C1 c1(OC)ccn2ccnc2c1C(N1CC2CC1C2NC(=O)CC1C=CCC1)=O C1(NC(C2CC(=C)CN2C(=O)CCSCC)=O)CCC(=O)N(CCOC)C1 C1(NC(=O)NC2CC(C(C)C)OC2)COCCC1O N1(C(CC(C(=O)OC)(C)C)=O)CCCC1C1CCCN1C(c1cn(C)nc1C)=O C(CCC(=O)NC)C1N(C(=O)NC(CC#C)C)CC1 Cn1ccc(=O)c(C(=O)NCCC2(C)CCN(C(=O)CCC3CC(F)(F)C3)C2)c1 c1(C(N2CC(N(C(=O)Cc3cn(C)nn3)C)C(O)C2)=O)n[nH]c2c1COC2 CCC(CNC(=O)CCN(C(C1OC2CCC1C2)=O)C1CC1)C(C)(F)F N1(c2ccc(OC)cc2)CCCC2(CCN(N3CC=CCC3OC)CC2)C1 c1(NC(N2CC(C)S(=O)C(C)C2)=O)ccc2c(c1)CCC2(C)O C1(CC)(NC(C2CCCN(C)C2)=O)CCCN(C(=O)C(C)S(N)(=O)=O)C1 Cc1nsc(N)c1C(N1CC(N2CCN(C(=O)CCC3CCC(C)O3)CC2)C1)=O CC(C)C(O)C(=O)NC(C1CCN(C(c2cnn(CC3CCCC3)c2)=O)CC1)C Cc1cc(-c2cn(CC3CCN3C(c3sccc3NC3CC3)=O)nn2)cc(Cl)c1 Cc1cc(C(=O)N(C2CCCCC2NC(C2CC2F)=O)C)c(Cl)cc1Cl C1(CCNC(c2c(CC)ocn2)=O)CN(C(=O)Cn2cnc(C(N)=O)n2)CCO1 Cc1cc(N)ccc1C(N1CCOC(C)(CNC(=O)C(C(C)C)n2cnnc2)C1)=O Cc1cc(=O)c(C(N2CCN(C3CN(C(=O)CCOC4CC4)C3)CC2)=O)cn1C C1(C(C)(C)CNC(=O)CSCC(F)F)CCCN(C(C2CC3CCC3C2)=O)C1 N1(C(C2CCN(CC)C2)=O)CCCC2(C1)CN(C(C1(O)CC(C)(C)C1)=O)C2 c1(CN2CCC(O)(CCNC(Cn3c(=N)scc3)=O)CC2)ccc2c(c1)COC2 c1(C(=O)NCCNC(c2cc(C(=O)OC)oc2C)=O)cc2ccc(F)cc2[nH]1 C1(C(=O)NCC(C2CC2)NC(CC=CCCCCC)=O)CC(=O)NC1(C)C CCC(Cc1ccccc1)C(=O)N1CCC(N(C(c2cscc2CC)=O)CC)C1 CC1CN(C(c2cc(O)cc(Cl)c2Cl)=O)CCCN1C(c1coc(C(N)=O)c1)=O c1(C(=O)NCC(CNC(CN(C2CCCC2)C)=O)F)ccc(Cl)cc1C(F)(F)F c1(C(=O)NCC2CC(O)(CNC(=O)CC34CC(C3)C4)C2)ccc([N+](=O)[O-])c(O)c1 N1(C(C23CCC(COC)(OC2)C3)=O)CCCN(C(=O)CC2OCCCO2)C(C)C1 c1(C(N2C(C)CCC(NC(=O)C3CC3)C2)=O)c(O)nc2ccccc2c1Cl c1(C(=O)NCC2(F)CCCN(C(C(CC)F)=O)C2)ccnc2c1nnn2C c1(N(CCC)C)cc(S(=O)(=O)NCc2c(F)cc(F)c(F)c2F)ccc1C#N CC(C)CC(C(=O)N1CCC(NC(=O)N(C)C)C1)NC(=O)CC1CC=CCC1 c1(N(C2CCC2)C)nnc(-c2nc(C3CC3)[nH]c2Br)n1C.S(=O)(=O)(CCOC)NC c1(-c2cnc(C(=O)Nc3ccc(-c4nn[nH]n4)cn3)nc2)cccc(Cl)c1O c12ccc(c(F)c1)-c1c[nH]nc1C(=O)N2.C1(C(N(C)C)=O)CCCN(C)C1 N1(C(C#C)=O)CC(NC(c2cccnc2N2CCCC2)=O)CC1CO Cc1cnccc1CCNC(=O)C(C1CCC1)NC(=O)Cc1ncccn1 CC(C)C(C(=O)NC1CCC(CNC(C2(C)COCCO2)=O)C1)n1ncc(N)n1 CCC(CN(C)C)C(=O)N1CCCCC1CCCO.C1(C)(CNC=O)CC(C)=NO1 C(=O)(C(F)(F)CCCNC(=O)OC(C)(C)C)NC(c1cn(C)nc1)C1CC1 Cc1cc(NC(c2c(-c3ccoc3)cncc2F)=O)ccc1N c1(C(N(CCC(COC)OC(F)(F)F)CCCC)C)ccc(Br)cc1 C1(N(C(C2(F)C(C)C2)=O)C)CN(C(c2cc(Br)cs2)=O)CC1(C)C C=CCN(OC)C(=O)C(CC(C)(C)C)NC(c1nc(C)c(C)nc1C)=O C1(F)(CNC(=O)CCc2nccs2)CC(NC(c2c[nH]nc2Br)=O)C1 N1(C(c2ccc(N)c(Cl)n2)=O)CC2CCCCN2CC1CNC(=O)C=C(Cl)Cl CC1CN(C(c2ccc(Cl)nc2N)=O)CC1(C)CNC(C1CCC12CCC2)=O O=C(C(F)C(F)(F)F)N1CC(C2CN(C(C3(n4cncn4)CC3)=O)CCO2)C1 N1(C(c2c(OCC)cccn2)=O)CC(NC(C2CN(C)C2)=O)CC(C)C1 C1(N(C(CC(C)n2cccn2)=O)C)CN(C(=O)Cc2cccnc2)CC1(C)C CC1COCC(C(=O)NC2CC(CCC(=O)NOCC(C)(C)C)C2)O1 N#Cc1cc(C(=O)NCC2CCC(NC(c3csc(Cl)c3)=O)C2)c[nH]1 C(CCC(=O)N(O)Cc1cn(Cc2conc2C2CCCCC2)nn1)OC C1(NC(CCc2ccn(C)c2)=O)CN(C(=O)CC2CCCO2)CC1O CC(C)C(C(=O)N1CC(CNC(C2CCSC2)=O)C1)NC(c1ccccc1)=O C1(C(N2CCC(C)(CNC(=O)C(c3ccccn3)O)C2)=O)CC1C1CCCCC1 C1(NC(c2nc(C(F)F)cs2)=O)CC2(C1)CC(NC(C13CC4CC1C3C4O)=O)C2 n1(CC)c(CNC(=O)CC(C)CNC(=O)CCC2CC2(F)F)cnc1C c1(C(N(CCCNC(C2CC2CC(C)C)=O)CC)=O)sc(OC)nc1C CCC(C)C(C(=O)N(C)Cc1nnnn1C)N(C)C(c1cncn1C(C)C)=O C1(c2cn(CC(COC)O)nn2)CCCCN1C(c1cccc(C(F)(F)F)c1)=O c1(CC(=O)NC2C3CN(C(C(C)NC(=O)NC)=O)CC32)ccc(O)c(F)c1 C1(C(=O)OC)CCOC1COC(=O)COCc1nccn1C c1(C(N(CC(CC)NC(c2ccc(CO)cc2)=O)CC)=O)nccc(OC)c1C C1(CC)CCC(C)CN1C(=O)C(CC(N)=O)NC(=O)CC1CCCOCC1 C(CCC1CCC1)(C(=O)NC1CN(CC(F)F)C1)NC(CSCC(=O)NC)=O N1(C(C2N(C(=O)NC)CCC2)=O)CC(C)CCC1CNC(c1nocc1Cl)=O c1(C(N(C2CCCOC2)C)=O)cccnc1CNC(=O)CCCC#N Cc1ccn2cc(C(=O)NC3CCCN(C(C4(CO)COC4)=O)C3)nc2c1 N1(C(C(C)SC)=O)CCC(OCCNC(c2cncn2-c2ccccc2)=O)C1 C1(C(=O)NC(c2ccc(F)cc2)C)C2CCN(C(=O)CC3OCCO3)CC12 Cc1ccc(CN2CCC(C)(C(=O)Nc3cc(C(C)(C)C)ccc3O)C2)c(C)c1 C(=O)(C(O)CC(C)(C)C)N1C(C(N2CCC(C)CC2)=O)CCCC1 CC#CCCCC(=O)NCC(CCC)NC(C1CN(C(C)=O)CCO1)=O Cc1nn2ncccc2c1C(=O)OCC(c1ccc2[nH]ccc2c1)=O c1(C(=O)NCC(=O)NC2CC(O)(CNC(C3CSC3)=O)C2)cccc(F)c1F c12cccc(c1)CCNC2=O.N1(C(C)C)CCC(C(=O)NCC(C2CC2)N(C)C)C1 CC1CC(CNC(c2cn(C(F)F)cn2)=O)CN1C(=O)CCSc1ccccc1 C(CS(=O)(=O)C1(Cc2c(C)n[nH]c2C)CC1)OC C(CCCC(C)NC(C1(C(F)F)CCOCC1)=O)NC(C1C(C)C1(F)F)=O C1(C(=O)NCCC(C=C)C)CC(NC(c2cc(CO)[nH]n2)=O)C1(C)C C1(NC(c2c(OC)ccs2)=O)CCCC12CN(C(=O)CC1OCCOC1(C)C)C2 C12(NC(=O)CCc3ccc(F)cc3)CCCC1N(C(C1C3CCCC13)=O)CC2 c1(C(N2CC(N(C(CC3C=NN(C)C3=O)=O)C)C2)=O)nn(C)cc1S(N)(=O)=O N1(C(C(CC)C#N)=O)CCC(C2CC2)(CNC(c2cnc(C)[nH]2)=O)C1 C=CC(CCC)CC(=O)NC(C)CNC(c1nnc(C)s1)=O C1(NC(c2cc(C)cc(F)c2)=O)CN(C(C2CC(N=[N+]=[N-])C2)=O)CCC12CCC2 c1(C(N2CCCC23CCN(C(C2(CC4CC4)CC2)=O)C3)=O)nccc2ncncc12 C=CCC(CC=C)C(=O)NCCC1CCCC(NC(c2ccc(F)c(Cl)c2)=O)C1 N1(C(COc2cc(C)on2)=O)CC2(CCC2)CC1C(N1CC2(CCCC2)C1)=O N1(C(C(C)(C)c2cscn2)=O)CCN(C(C2CC(F)(F)C2(C)C)=O)CC(CO)C1 C1(C(C)C)(C(=O)NCC(C2CCCC2)NC(c2nccnc2N)=O)CNC(=O)C1 c1(CC)c(C(N2CC(NC(=O)Cn3cnc(C#N)n3)C(C)C2)=O)csc1C C1(CC=C)CCCN(C(=O)C(CC)N(C(=O)CCNC(C)=O)C)C1 CS(=O)(=O)C1CC(NC(=O)CC2CCCN2Cc2cc(C(F)(F)F)ccc2O)C1 Cc1cc(N)ccc1C(N1CCC2(CC2NC(C2CCCN(C)C2)=O)C1)=O CC1(CNC(c2ccc(-c3cccs3)o2)=O)CN(C(=O)CCOC2CC2)CCO1 N1(C(CCC(C)NC(C2CC(CF)C2)=O)=O)CC2COCC2C1 c1(CO)cccc(S(=O)(=O)N2CC3CCC2CN3S(=O)(=O)CC2CC2)c1 C1(C(=O)NC2CN(C(CS(CC)(=O)=O)=O)CC(C)(C)C2)CCC2(CCOCC2)O1 c1(OC)nc(C(N2CC(CNC(C3CSCCS3)=O)C(C)C2)=O)cc(O)n1 C1(C(N2C(CNC(COCP(C)(C)=O)=O)CC2)=O)CC(c2cccc(F)c2)=NO1 c1(C(=O)OC(C)(C)C)cncc(NC(C2COCCN2Cc2ccccc2)=O)c1 N1(c2n(CCC#C)c(CCC(F)(F)CO)nn2)CCn2cnnc2C1C CN1CCCC(C)(CNCc2c(C(F)(F)F)n[nH]c2C(=O)O)C1 C=C=C(C)CC(=O)NCC1CC(C)N(C(c2cnn(CC(F)(F)F)c2)=O)C1 C1(c2n(CCC)nnn2)(NC2(C(=O)OCCOC)CCCC2)CCCC2CC12 C#CCC(CC#C)C(=O)NC1CN(C(=O)COc2cc(Cl)ccc2C)CC1O C=C(C)C(C)(C)C(=O)N1CCC(CO)(NC(=O)C(CO)c2ccccc2)C1 C1(CN(C)C(c2ccn(CCF)n2)=O)C2CN(C(=O)C=C(Cl)Cl)CC12 C(=O)(C1=Cc2ccccc2C1)C(=O)CC1CN(c2ncc3scc(Br)c3n2)CC1C N1(C(c2n(SCC)ncc2)=O)CCCC(NC(c2ccoc2Cl)=O)C1 C(=O)(CC1CCC(C)(C)c2ccccc21)NCCC(C)NC(CCCC)=O c1(NCC2CCN(C(=O)CC(c3ccc(F)cc3)O)C2)nc2ccc(Cl)cc2s1 C(=O)(CC(C)C(F)(F)F)NC1C(CC)N(NC(=O)OC(C)(C)C)CCC1 C(=O)(C1CCCc2sc(C)nc21)NCCC(C)(C)NC(CCC(CCCC)C)=O Cc1cc(OCCNC(=O)NCc2cnc(N(C)C)o2)cc(C)c1 C(=O)(C(C)(C)CCNC(c1cnc(O)c(F)c1)=O)NC1C(SCC)CCC1 CCN=c1[nH]c(C)c(C(N2CC(NC(=O)Cc3ccn(C(F)F)n3)C(C)C2)=O)s1 C(=O)(C=CS(F)(F)(F)(F)F)NC1C(NC(C2C(C)(C)C2C(F)F)=O)CCCC1 N1(C(COc2cn(C)nc2)=O)CCN(C(c2nc(=N)cc[nH]2)=O)CC(O)C1 C1(CC)C(NC(=O)CCc2nncs2)CCCN1C(=O)Cc1ncoc1C c1(NCCS(=O)(=O)NCC)[nH]c(=NC(C)CN(C)C)nc2sccc12 Cc1nc(=N)[nH]cc1C(N1CCN(Cc2nccs2)CC1)=O C(=O)(CCN1C(=O)CCc2cc(F)ccc21)C(NOC(CC)CC)=O.OCC C(=O)(CC(O)CCCC)N1CC(CCNC(CCCC#C)=O)OCC1 c1(OC)nc(Cl)c(C(=O)NC2CC(CNC(=O)CCc3ccc[nH]3)C2(C)C)s1 c1(SC)cc(C(=O)NC(CCNC(c2ccoc2C)=O)C(C)C)ccc1N CC(C)C(F)(CNC(C1(C)CC1)=O)C(=O)NCCN1CC=CC1 C1(C(N2CC=CC2CF)=O)CCC(C(F)(F)C(F)(F)F)CC1 c1(C(=O)NCCCNC(C2CCC(C(N)=O)CC2)=O)ccc2c(n1)CCC2=O Cc1ccc2c(c1)C(NC(=O)N(c1cn(Cc3ccc(Br)c(Cl)c3)nn1)C)CC2 N1(C(C(C)OCC)=O)CC2CCN(C(C3CCSC3)=O)C2C1 C1(CNC(CCCOCCOCC)=O)CN(C(C2(C#N)CC2)=O)CC1C N1(CC(=O)NCC#CC#CCO)CCN(C(C2CCC(=O)O2)=O)CC1 c1(CNc2ccc(CCCNC(C)=O)cc2)ccc(S(=O)C(F)(F)C(F)(F)F)cc1 Cc1c(CC(=O)NC2CC(C)(NC(c3cc(CN(C)C)n[nH]3)=O)C2)ncn1C N1(C(C(CCC)CC)=O)CC2(C=C(C(=O)NCCC(O)C3CC3)CO2)C1 N1(C(C=CCC)=O)CCC2(CCC(NC(C3CC4CCC3O4)=O)C2)C1 Cc1nc(C(C)(C)C)c(C(=O)NCCC(C)CCNC(=O)Cc2cccs2)s1 c1(-c2cn(C(C)C(=O)N3CC(NC(=O)C(F)(F)F)C3)nn2)c(Cl)cc(Cl)cc1Cl C1(CC(C)C)COCCN1C(=O)C(=O)NC(C)CCCl.n1(CC)cc(-n2cccc2)nn1 c1(CC)cc(Br)c(CN2CCC(C(c3ccc(F)cc3)c3cccs3)C2)s1 C1(N(C(=O)CC2CCC23CCC3)C)CC2CCC(C1)N2C(c1ccccc1)=O C1(NC(=O)Cc2ccon2)CC1C1CCN(c2ncc(Cl)cn2)CC1 O=C(C1=CC2C=CC1C2)N1CC2CC1CN2C(c1ccncc1Cl)=O CCC(CC(=O)NCCCC(C)NC(c1c[nH]ccc1=O)=O)C(C)(C)C N1(C(CCSc2cccc(OC)c2)=O)CC(C)CN(C(=O)COC(C)=O)C(C)C1 C(=O)(CCC(=O)NCC1CC1CC(N1CC(O)CC1CO)=O)NCCC N1(C(c2c(C)c(O)cc(N)c2)=O)CCC2(CCC2CNC(C2C(C)C2C)=O)CC1 CC1=C(C)CC(C(=O)NCC2CCC2C(=O)NCc2ccc(C)cc2C)CC1 c1(C(=O)NC(C(C)NC(C2CCN(C(C)(C)C)C2=O)=O)CO)c(F)cccc1Cl C(=O)(CC(C)(C)N(C)C(c1cn(C2CC2)cn1)=O)OC.C1(C)(C(=O)N)CC(C)=NO1 c1(C(=O)NC2C(NC(c3cc(C)cc(Cl)c3)=O)CCOC2)cnc(Cl)c(F)c1N c1(C(N2C(CNC(c3ncccc3Cl)=O)CC(OC)C2)=O)c(C)cc(F)cc1C c1(C(C)(C)C)ccc(NC(C2CCC(NS(=O)(=O)CC#N)CC2)=O)c(I)c1 Cc1ccc(O)c(C(=O)N(C(c2ccccc2)CNC(C2CC=CCC2)=O)C)n1 C1(CNC(C(C)(C)NC(C(C2CCC(=O)N2)C)=O)=O)CC2(CCC2)C1 C(C(=O)NC(C1CCN(c2cc(C(F)F)ncn2)C1)C)(C(C)C)NC(=O)OCC CC1(CNC(c2ccc(CF)cc2)=O)CC(F)(F)CN1C(=O)C=Cc1ncc[nH]1 C(=O)(N1CCC(C(=O)NCC(=O)OC(C)(C)C)O1)c1c(C)oc(Cl)n1 c1(CN(C)C(C2CCCC(=O)CC2)=O)cc(Cl)c(Br)cc1F C1(C(=O)NCC2(O)CC(NC(=O)CC3C=CCCC3)C2)CCC2(CCCC2)CC1 N1(C(C2C(CC)CCO2)=O)CC2C(C(=O)NCCOCCOC)C2C1 C1(C(N2CC(NC(c3cncc(C)c3)=O)CC2(C)C)=O)CC2(COCCO2)C1 c1(CC)cc(C(N2CCN(C(=O)CN3CCCC3CO)CC2C)=O)cc(O)n1 C(CC(=O)N1CCOCC1)(CC(C)C)NC(c1c(C)cc(O)nn1)=O C12(NC(CC3CC(OC)C3)=O)CCC(CN(C(=O)Cc3ccc(F)cc3Cl)C1)C2 c1(C(N2CCC(C)(C)C2CNC(=O)CC2CCCCO2)=O)ccc(S(N)(=O)=O)o1 C1(NC(c2n(C)cc(Br)c2)=O)CC2CC1N(C(C1(C)CC3CC3C1)=O)C2 c1(C(N2C(C(C)NC(c3cc(CCOC)on3)=O)CCC2)=O)ccc(O)nc1Cl C(=O)(C1=CCC2CCC1N2C(C1(SC)CCC1)=O)NCC(CCC)C C1(CCNC(c2n(CC)ncn2)=O)CCN(C(=O)CCC(C)OC)CC1 c1(CNC(C(CNC(C2CC2Cl)=O)OC)=O)ccncc1Cl C12(CNC(CSCCC)=O)CCC1CCN2C(c1cc(C(C)(C)C)nn1C)=O N1(C(C(=O)Nc2c(CC)cccc2C)c2ccsc2)CC(C)(C)OC2(CCC2)C1 C1(C2CC2)(CNC(c2nc(C(C)C)oc2)=O)CCN(C(=O)CC(C)(O)C2CC2)C1 C1(NC(Cc2ccn(C)n2)=O)CCCC(NC(c2ncc[nH]c2=O)=O)C1 c1(CC(=O)NC2CC3CCC(C2)N3C(=O)C=CBr)ccc2ncccc2c1 c1(CNC(c2c[nH]c(=N)s2)=O)ccc(CNC(C2CCCCS2(=O)=O)=O)c(F)c1 N1(C(C=Cc2c(C)n[nH]c2)=O)CCC2C(CCCN2C(C2(C(C)C)CC2)=O)C1 c1(C(=O)NCC2CCCN(c3c(C(=O)OC)nccn3)C2)cc2ncccc2s1 C1(NC(C(C)(C)C2CCCC2)=O)CCCN(C(=O)CNC=O)CC1 c1(C(C(N2CC(CNC(C3(C)CCCC3)=O)C2)=O)O)ccc(F)c(Br)c1 C1(C(=O)NCCN(C(c2c(C)oc(C(C)C)c2)=O)C)CCc2ccc(F)cc2O1 C(C(C)(O)C(=O)NCC1(NC(c2nccc(C(F)(F)F)n2)=O)CCC1)OC CC1CN(c2ccccc2)CCN1C(c1cnc(-n2cccn2)cn1)=O CC1CCCC(CC(=O)NC2(CCNC(c3ncccn3)=O)CCC2)C1 C1(C(=O)NCC2CC(O)(CNC(c3nn(C)c(O)c3)=O)C2)CC2OC(=O)OC2C1 N1(C(c2cncc(NC)c2)=O)CCC(C)C(CNC(=O)C(C)(C)c2ccns2)C1 N1(C(C(C)S)=O)CCC2C1CCCN2C(c1c(C(F)(F)F)cc(Cl)cc1Br)=O C1(N(C)C(=O)OC(C)(C)C)CCCN(C(=O)NCc2cc(Cl)n(C)n2)C1 N1(C(c2c(C)ccs2)=O)CC(F)(F)CC1CNC(=O)CCc1ccc(Br)cc1 C(N=c1[nH]c(=NC2CCCC(O)C2)[nH]c2c1CSC2)C1CCCN(CC)C1 N1(C(CC(C)(C)C)=O)CC2CCC1CN2C(c1cnc(N)c(Br)c1)=O c1(OC)cccc(Br)c1NC(C1CC2CC2N1Cc1ccc(OC)c(Cl)c1)=O CC(C)C(C(=O)N1CCCC(C)C1)NC(=O)CSCC(N)=O C(=O)(C1=CC2(CCOC2)C1)N1CC2(CN(C(C3(C)CC3(F)F)=O)C2)C1 c1(C(N2CCC(c3ccc(F)cc3)C2)C(=O)NCCOC)ccc(C)cn1 C#CCC(CC(=O)N1CCC(OC(C)C)CC1)NC(=O)CCCCn1ccnn1 CCCCC(C)C(=O)NCC1CCN(C(=O)C(O)CCc2ccccc2)C1 c1(OC)ccc(CCCC(=O)NC2CCCC2NC(C2CC2(C)C)=O)cc1 c1(C(=O)NC2CCN(C(C(C)CC(N)=O)=O)CC2C(N)=O)scc2c1OCCO2 CN1Cc2ccc(C(=O)NC3CCN(C(=O)CSC(F)(F)F)CC3F)cc2C1 C(=O)(C1=CC(C)(C)C1)NC(C(C)NC(C1(OC)CCOC1)=O)CO CN1CCCC1C=CC(=O)NCC1CCC1NC(=O)Cc1ccc(C(F)F)cc1 C1(N(C(=O)CCSC)CCCC)CC(C(=O)OCC)C12CCNCC2 N1(CCOCCCNC(C2(C)CSC2)=O)CC2CCN2C1 c1(C(N2CCCC(NC(C(C)C#N)=O)CC2)=O)cc(Br)cc2cccnc12 n1(CC)ncc(S(=O)(=O)NC(C)=O)c1NCc1csc2ccc(Br)cc12 C(=O)(C(C)C(F)(F)C(F)F)NCC1(OC)CN(C(=O)CSC(F)(F)F)C1 C1(CC(N2CCCC(NC(c3ccoc3)=O)C2)=O)CCC2(CCOCC2)CO1 c1(C(=O)NCC2CCN(C(C(C)OCC)=O)C2)cnc2ccoc2c1 c1(C(N2C3CN(C(C4N(CC)CC4)=O)C(C3)C2)=O)c(Br)ccc(F)c1C c1(CN2CCCC(N(C(c3cnc(NC(C)=O)o3)=O)C)C2)ccncc1C#N C=CCC(CC)C(=O)Nc1ccc(OCCC)c(N)c1.C12CC(F)CN(C1)C2=O Cc1ccc(C)n1CC(=O)NC(C1(O)CN(C(=O)COC2COC2)C1)C C1(NC(C2CC(CSC)C2)=O)CC2CCC1(NC(CCC(=O)C(C)=O)C1CC1)C2 S(=O)(=O)(c1ccc(=NCC2CSCCO2)[nH]c1)CCN1C(C(N)=O)=NCC1 CN1CCC2CCN(C(C3C4CCCC4CN3C(c3cc(O)n(C)n3)=O)=O)C2C1 C(c1cccnc1C)=CC(=O)NCC(c1cccc(C)c1)NC(CC(=C)C)=O C#Cc1ccc(C(=O)NC(CNC(c2coc(C#N)c2)=O)CC=C)c(F)c1Cl N1(C(Cc2cc(C)on2)=O)CC(NC(c2sccc2C(C)C)=O)C2(CCCC2)C1 N1(C(Cn2cc[n+](C)c2)=O)CCC(NC(=O)C=C(C2CC2)C2CC2)C(CO)CC1 C(c1ccc(Cl)nc1)=CC(N1C(C)CC(CNC(c2cc(O)nn2C)=O)C1)=O N1(C(C(c2nncn2C)C)=O)CC2(CCN(C(=O)CC3CC4CCC3C4)CC2)C1 c1(C(CNCC(c2ccccc2C)OC)O)ccc(F)c(Cl)c1 C1(OC)CN(C(=O)C(F)CC2CCOC2)CC1C(=O)N(C1CC(SC)C1)C c1(C(C)CC(=O)NCC2CCN(C(C3(F)CCC3)=O)C2)ccc(F)cc1F C(=O)(C#CC1(C)CCCO1)NCC1(OC)CCN(C(C2CCCC(O)C2)=O)C1 C1(F)(C(=O)NCCN(CCC)C(C)C)CCN(C(C2CC(C)OC(C)C2)=O)CC1 c1(C(C)=O)cc(C(N2CC(N(C(=O)CC3(C)CC3(Cl)Cl)C)C(O)C2)=O)oc1C NC(=O)CC(C(=O)NCCSC(F)F)NC(c1cc(CO)[nH]n1)=O C=Cn1nncc1C(=O)NC12CC(NC(C3CC4CC4C3)=O)(C1)C2 C1(O)(C(C)NC(c2c(C)cnnc2)=O)CCN(C(C2CCO2)=O)CC1 C1(OC)Cc2ccccc2C1N(C)C(c1ccc2ncccc2c1)=O O=C(CC(C(F)F)n1cccn1)N(CCC1(O)CN(C(=O)C=C(Cl)Cl)C1)CCO C=CC(C)(C)CC(=O)N1CCC(CF)(NC(c2ncc(Br)cc2F)=O)C1 C(=O)(CCCC(=O)N(C)C)N1CC(N(C)C(C2CCOC2=O)=O)C1 C(=O)(C(F)(F)C1=CCOCC1)N1CC(CNC(c2c(OC)nn(C)c2)=O)C1 C1(C(N(C2CN(C(=O)CCc3ccn(C)n3)C2)C)=O)CC12CCSCC2 c1(C(C#N)NC(C2C(C)(C)C2)=O)ccccc1F N1(CCNCc2c(NC(C)=O)cccc2)CCCN(C2CCOC2)CC1 c1(OC)noc(C(=O)NCC2(C)CCN(C(C3(C#N)CC3)=O)C2)c1Br C(=O)(C(C)C(O)CCCC)NC1C(CNC(C2(CCC=C)CC2)=O)CCCC1 C(=O)(C1=NNC(=O)C1)N(C)CCC1CCN(C(c2cnccn2)=O)CC1 N1(S(c2c(NC(CC)=O)nccc2)(=O)=O)CCc2cccc(Br)c2C1 N1(C(C(CSC)(C)NC(=O)C=Cc2cccnc2)=O)CC(=O)N2CCCC2C1 CC1(C)COCC(C(N2CCOC(CNC(=O)Cc3ccsc3)C2)=O)O1 C1(C(C)CNCC(O)CO)CCCCN1C(=O)NC1CCCC(C(F)(F)F)C1 CC(CCCCNC(=O)CC1(C)CCCO1)NC(c1nc(C(C)(C)C)no1)=O c1(CNC(C2N(C(c3cnc(CC)nc3)=O)CC(OC)C2)=O)cc(C)cc(F)c1 N1(C(C2CC(C)(CC)C2)=O)CCCC(CCNC(=O)C(C)CN2CCCCC2)C1 C(C)(C)(CC(=O)NC12COC(C)(C1)C2)N(C(=O)CCCN(C)C)C c1(C(=O)NCCC2CCCN(C(C(C)CCO)=O)C2)cnc2ncnn2c1N c1(C(=O)NC(=O)CN)ncccc1O.C1(CC)CCCN1C(=O)C(=O)N(CC)C C1(NC(c2c(CC)ocn2)=O)CC2CC(C1)N(C(=O)Cc1cc(C)no1)C2 N1(C(c2c(CC)[nH]cc2)=O)CCC(C)C(NC(C23CC(CN2C2CC2)C3)=O)C1 Cc1cc(C(=O)N(C(C)CNC(C2CC2F)=O)C)c2[nH]cnc2c1 c1(OC)ccc(C(N2CCC(C(C)NC(c3cc(C)nn3C)=O)CC2)=O)c(Cl)c1 c1(N(CCCNC(C)=O)C(=O)CN(C2CC2F)C)ncnc2[nH]cnc12 N1(C(c2cc(C)cc(C)n2)=O)CCC(C)N(C(C2CCCN2N=O)=O)CC1 C(CCCC(=O)N1CCC(CN(C)C)C1)N(C(CC=CC)=O)C c1(OC)ccc(O)c(C(=O)N(CCCCNC(=O)CC2CC(O)C23CCC3)C)c1 N1(C(Cc2c(C)nn(C)c2)=O)CCC(NCc2ccc(C(C)(C)C)cc2)C(C)C1 C(=O)(C(C(C)(C)O)NC(=O)CCS(C)(=O)=O)N(CCCOCC)CC C1(F)(CNC(c2c(C)nsc2)=O)CCCN(C(C2CC(=O)N(C(C)(C)C)C2)=O)C1 c1(C(=O)NC(CC)CNC(C2OCCC2CC)=O)cccc(OC)c1 c1(NC(=O)CCSc2cn(-c3ccccc3)cn2)cc(F)ccc1F C1(NC(c2c(C)cno2)=O)(CO)CCCN(C(C2CC=CCO2)=O)C1 c12cc(Br)c(s1)[nH]2.n1(CC2CN(C(COC)=O)C2)cc(C2CCCOC2)nn1 N1(C(C(COC)COC)=O)CCCCCCC1C(N1CCC(C#N)C1)=O CC(C(=O)N(C)CC1(NC(c2cnc(O)cc2C(F)(F)F)=O)CC1)S(N)(=O)=O N1(C(CN(S(CC)(=O)=O)C)=O)CC(O)C(O)C1CNC(c1cccnc1O)=O C#CC1CN(C(C2CCCN(C(=O)CS(=O)CC)C2C)=O)CCN1C C1(CC)COCCC1N=c1[nH]c2c(c(=NCc3ncoc3C)[nH]1)COC2 N1(C(COCCC#C)=O)CC(COC)CC1CNC(C1CC(=O)N(C(C)C)C1)=O Cc1ccccc1C1(C(=O)NCC2(O)CCN(C(=O)C3=NOCC3)C2)CC1 N1(CCOC)CC(C(=O)NC(C)CC(C)NC(C2CCOC(C)C2)=O)CC1=O C1(CN(CCCNC(=O)CCN(S(C)(=O)=O)C)C)COCC1(C)C CC(C)C(C#N)C(=O)N(CCCN(C)C(C12CCCN(CC1)C2)=O)C c1(CN(C)C)cccc(C(N2CCSCC2CCNC(c2ccoc2Cl)=O)=O)c1 C1(NC(c2c[nH]nc2-n2cnnn2)=O)COC2(CCCN(C(=O)C3CC3)C2)C1 CC1(CNC(c2cc(C3CC3)[nH]n2)=O)CCN(C(C2CCC(=O)N2)=O)C1 c1(C(N(C2CCCN(C(C3N(CC)CCC3)=O)C2)C)=O)cn(C)c(=O)nc1O CCC(C)CCC(=O)NCC1CN(C(C2(CO)COC2)=O)CC1O N1(C(c2cc(C)on2)=O)CCC(C(N2CCC(c3ccccc3O)CC2)=O)CC1 C1(CN(CC)Cc2ccccc2)(OC(=O)CCC2CCCO2)CC1(C)C N1(C(C)=O)CC(C)CCC1CNC(C1CC(=O)N(C2CCCCCC2)C1)=O N1(C(c2[nH]cc(CC)c2)=O)CC2(CCC(NC(=O)C(CC)N(C)CC)CC2)C1 C1(C)(C(=O)NCC2N(C(Cc3n(C(C)C)cnn3)=O)CCCC2)CCN(C)CC1 C(CC(=O)NCC1CCOC1)(C(F)F)NC(C(C)N(C)C)=O C1(NC(C(C)CO)=O)CCCCN(C(c2sc(F)cc2Cl)=O)C1 N1(c2nc(CC)nc(=N)[nH]2)CCCC2C(NC(=O)C(C)CC)C(C)(C)C12 Cn1ncc2c(NC3CCc4ccccc43)nc(N3CCCC(C(F)F)C3)nc12 N1(C(C2C(=C)C2C(=O)OC)=O)CCCC1CC(=O)NCCN=[N+]=[N-] C1(CC(=O)NCC2OCCN(C(C=CC=CCC)=O)C2)CCCC2(CCC2)O1 C(=O)(C(C)CCCC(=O)N(C(C)CNC(=O)CC1CCC1)C)OC c1(CC(C)N(C(=O)C(=O)NC2CCCC2)C)ccc(C(C)(C)C)cc1 c1(NC(C2(C)N(C(c3c(N(C)C)cccn3)=O)CC2)=O)ccc(F)c(F)c1 c1(NCC(c2ccc(F)cc2)(C)F)ncnc(-c2cccs2)n1 C12CCCCC1C(=O)NCCS2.C(C(=O)NCC=C)=CC=C.OC C(=O)(CCCCCCCS(C)(=O)=O)NCc1c(CNC(C(CC)F)=O)cccc1 C#Cc1ccc(C(=O)NC(CC2CC2)C(=O)NCCC#CCC)nc1 c1(C(N2C(C(C)NC(=O)C(=Cc3c[nH]cn3)F)CCC2)=O)cnc2cc[nH]c2c1 C=C(C)CCCC(=O)N1CCCC(C(C)NC(=O)CC2(C(F)(F)F)CC2)C1 N1(C(Cc2c(C)ccnc2)=O)CCN(C(c2cc[nH]c2C)=O)C(C)CC1C c1(C(C(=O)NC(CC(C)C)CNC(C2(CCO)CC2)=O)C)nc(F)ccc1Cl N1(c2nc(C)nc(C)c2C)CCC(C2(NC(c3cccn(C)c3=O)=O)CC2)CC1 C(CN=c1[nH]c(=NCCc2ccc(C)nc2)[nH]c2c1CC(C)CC2)N1CCC(C)C1 O=C1CN(CC(=O)NCCO)CCN1.C1(O)(N)CCN(C(=O)COc2cn[nH]c2)C1 c1(NC(=O)C(C)Cc2ccccc2Cl)ccc(CNSC(C)C(=O)NCC)cc1 C(c1cncnc1O)=CC(=O)NCCN(CCC)C(c1ccsn1)=O N1(C(C(C)CO)=O)CC(O)CC1C(=O)NOC1CC1 C=CC1COCCN1C(C12CC(CO1)N(C(=O)C=Cc1ccccc1C)C2)=O Cc1cnc(C(N2CCC(CNC(C3(C)CC(C)(C)C3)=O)C23CC3)=O)c(O)c1 CC(CCNC(C12CC(NC(c3cccc4[nH]ncc34)=O)(C1)C2)=O)CC(C)(C)C c1(C(=O)NC23CC(NC(CCc4cc(C)[nH]n4)=O)(C2)C3)c(F)ccc2c1OCO2 c1(C(N2CC(NC(=O)Cc3ccccn3)C(F)C2)=O)ccc(Cl)c(I)c1 N1(C(CCC(C)OC)=O)CCN(C(c2ncoc2-c2ccccc2)=O)C(CF)C1 C1(N(C2CS(=O)(=O)C2)C(Cc2cc(C)n(C)n2)=O)CCC2(CCNCC2)CC1 Cc1ccncc1CC(=O)NC1CC(C)(NC(=O)CCC2CCCN2C)C1 Cc1sc(-c2nc[nH]n2)nc1C(=O)NCC1CC(NC(=O)C=CS(C)=O)C1 c1(C(N(C)CC2CCN(C(=O)CCc3ccc[nH]3)C2)=O)nc(O)nc(O)c1F CCC(CC)C(C)NC(=O)C(C)(C)CNC(=O)CC1CCCOCC1 N1(C(C(C#C)(C)C)=O)CCCC2(CCN(C(c3cc4ncccn4n3)=O)CC2)C1 N1(C(C(c2ccc(Cl)s2)C)=O)C2CCC1CC(n1cc(C3(C)CCCO3)nn1)C2 C(C(=O)N1CCC(C(C)(C)CN(C(=O)C(O)CN(C)C)CC)CC1)(C(C)C)SC N1(C(c2cn(CC=C)nn2)=O)CCN(C(c2cn(C)c(=O)n2C)=O)C(CCO)C1 C1(F)(C(=O)NCC(C)N(C)C(c2cnc(-c3ccccc3)[nH]2)=O)C(C)(C)C1(C)C C12(CNC(C(CO)N(C)C)=O)CCC(C1)N(C(=O)C1=CCOC1)C2 Cc1snnc1C(=O)NCC(c1ccccc1)N(C(=O)CCOCC(C)C)C C(=O)(C(F)(F)C(O)CCCCCC)NC(CNC(C(C)SC)=O)(C)C C1(C)(OC)CC(NC(=O)CC2CCN(C(c3cnn4c3CCC4)=O)C2CO)C1(C)C C1(C(=O)NCC2C(NC(CN(C)CC)=O)C2)(C(F)F)CCCCC1 O=C(C1=NNC(C(F)(F)F)C1)NCC1(CNC(c2cc(O)cc(O)n2)=O)CCC1 N1(C(CCCOCCC)=O)CCOCC(NC(=O)C(N2CCC(CC)CC2)=O)C1 c1(OC)ccc(CCC(=O)NCC(C)NC(C2Cc3nnsc3S2)=O)cc1C c1(NC(C2CCC(NC(C3(F)CCCC=C3F)=O)C2)=O)ccc(CO)c(F)c1 c1(OC)ccc(C2(C(=O)NC(CC)C(=O)NCCOC(C)(C)C)CC2(Cl)Cl)cc1 FC1CC(N=c2[nH]c3c(c(=NCCn4ncc(Br)n4)[nH]2)CCCCC3)C1 c1(C(C)C(=O)NC2CC(NC(=O)CC3CC4(CC4)CO3)C2)cccc(O)c1 C(=O)(CCCC(C)(C)C)N1CCCN(C(C(C(C)C)C)=O)CC1 N1(C(c2nnn(CC)c2C)=O)CCC2(CC2NC(=O)CCC2CC2(F)F)C1 C1(O)(CNC(C=C(C)Cl)=O)CCN(C(=O)C(C)Oc2ccccc2C(N)=O)CC1 c1(CCC)n[nH]cc1C(=O)NC(C(=O)NC1C(C)C1C)C1(C)CC1 CC(O)(C(=O)N1CC2CCC2(C(N2CCCC2C(N)=O)=O)C1)C(F)(F)F C(CC(C)C)(C(=O)N1CCN(C(c2cnc(Cl)[nH]2)=O)CC1C)NC(C)=O Cc1ccc(C(=O)NC2(CO)CCCN(C(c3cccnn3)=O)C2)c(C)c1 N1(C(CCC=C)=O)CCOC2(CCCN(C(C3(S(N)(=O)=O)CCCC3)=O)C2)C1 N1(C(=O)NC)CCCC(O)(CNC(c2ncsc2NC(=O)OC(C)(C)C)=O)C1 c1(C(=O)NCC2CCC(F)(CNC(CCN(C)CC)=O)C2)scc2c1CCCC2 C(CCC(C)C(=O)N1CCCC(F)(CNC(C2(F)CC=CC2)=O)C1)OC CCC(CC)CCC(=O)NC(C1CCCN1C(=O)C(F)CC1CCOCC1)C C#CCCCC(=O)N1CC(C=C)(CC(N2CCC(N(C)C)C2)=O)C1 c1(OC)ccnc2c(NCC3CC(C)CN3C)cccc12 C12(CNC(C(N3CCOCC3)C)=O)CCC(CC1)N(C(=O)C(O)C1CCCC1)C2 C=C(C)C(C)(C)C(=O)N1CC(CNC(c2cc(C)cc(C)c2)=O)C(C(F)(F)F)C1 c1(OC(C(=O)NC(C)CNC(C2(O)CCSCC2)=O)F)ccc(Cl)c(F)c1 c1(C(=O)NC(C2CCN(C(c3nccnc3O)=O)C2)C)cc(Cl)c2n[nH]cc2c1 N1(C(C(=O)NC(C(=O)OC)CCC2CC2)C)C(=O)c2cccc([N+](=O)[O-])c2C1=O N1(C(CC(C)SC)=O)CCCC12CCCN(C(c1ccc(F)cc1Br)=O)C2 CC1C(C)S(=O)(=O)CCN1C(=O)Nc1[nH]nc2ccc(C(C)(C)C)cc12 N1(C(C(C(C)O)NC(C)=O)=O)CCC2CN(C(=O)CC=C(Cl)Cl)CC2C1 C1(NC(c2cnc(C3CC3)[nH]2)=O)CC(O)CN(C(=O)CCn2cncn2)C1 c1(CNC(C2CC(NC(c3cc(CN(C)C)on3)=O)C2)=O)ccc(Cl)nc1 Cc1csnc1C(=O)N(C1CCCC1)CCNC(=O)C(n1ccnc1C)C c1(CC(=O)NC2CCC(C(F)(F)F)O2)cc(F)ccc1C(F)(F)F Cc1cc(=NCCN(C)C)[nH]cc1S(=O)(=O)Nc1cccc(C)c1C C1(CNC(C(CC)=CC)=O)CN(C(c2ccccc2O)=O)CCN1C c1(C(N2C(C(C)NC(C3C=CCC3)=O)CCCC2)=O)cc(O)nc(O)n1 Cc1cc(N2CCC(Cn3cc(Br)cn3)C2)nc(N2CCOC(CC(C)C)C2)n1 c1(C(N2CC3(CN(C(COCCC)=O)C3)C2)=O)cc2cncc(C)c2s1 C(CCCC(=O)NC1(C(C)O)CC1)NC(c1c(C(C)C)noc1)=O c1(NC(C)=O)ccc(C(N2CCC(C)CC2)=O)cc1.C12(C)CC(C1)C(=O)N2 c1(CN(C(=O)CC2CCN2C(C2CC(F)CN2C)=O)C)ccc(O)cc1 C1(CCOC)CC(F)(F)CN1CC(c1cn(C)nc1C)=O C1(CNC(C2(CC(C)C)CC2)=O)CCC(C)CN1C(C1CC(C(F)(F)F)C1)=O c1(C(N(C)CC2COCCN2S(C)(=O)=O)=O)ccc(C2CCC2)cc1 c1(-c2ccc(NC(=O)NC3C(CC)N(CC4CC4)C(=O)C3)cc2)ccc(F)c(C)n1 C(=O)(C#CC1(C)COC1)NC(CNC(C1NC(=O)CC(C)C1)=O)C N1(C(C2CCC(=O)O2)=O)CCOC(CCNC(c2cn(CC(F)(F)F)nn2)=O)C1 C1(O)(C(C)NC(C2C(C=C)C2)=O)CCN(C(c2cc(C)n(C(C)C)c2)=O)CC1 N1(C(CCCNC(c2ccc(OC)cc2)=O)=O)CC2CCCC(CO)(C2)C1 CCC(C)C(C(=O)NCc1cc(C(=O)N(CC(C(C)C)OC)C)cs1)OC N1(C(Cc2nnc(C)s2)=O)CCN(C(c2ccc(OC(F)F)cc2F)=O)CC1C CC1c2c(Br)cccc2CN1Cc1c(Cl)cc(Br)c2scnc12 N1(C(c2cc(C)[nH]n2)=O)CCN(C)CC1CNC(C1(Oc2cnn(C)c2)CC1)=O C1(NC(c2c(CC)cccn2)=O)CC2(C1)CC(NC(C1CN(C(=O)O)C1)=O)C2 c1(SC)cc(C)c(C(N2CCC(C)(NC(C3CCC4(CC4)C3)=O)C2)=O)o1 C1(N(C2CN(C(c3cnc(CC)s3)=O)C2)C)CCN(C(=O)COC(C)C)CC1 c1(C(C)C)ccc(C(N2CC(N(C(=O)C(C)CO)C)C3(CC3)C2)=O)cc1F c12sc(nc1C)[nH]2.CCC(CNC(=O)CC1CC1(C)C)NC(=O)C1CC1 Cc1ncnc(NCCC2CCC(C(=O)NC(=O)C3CC3)CC2)c1Br c1(C(=O)NCC2CN(C(c3c(C#C)c[nH]n3)=O)C3C2C3)cc2cccnc2[nH]1 C1(C(=O)NCCCC(C)NC(c2c(CC)n(CC)nn2)=O)CCC2(CC1)CC2 N1(CCNC(C(C)OCC=C)=O)CCN(C(C2CC2c2cccc(C)c2)=O)CC1 c1(C(=O)NCC(C)N(C(=O)C2=C(C#N)CCC2)C)nn2cccnc2c1Br c1(C(=O)NC(CC)CNC(=O)C=C(C)c2ccco2)ccc(C)c(F)c1F c1(CC)cccc(NC(=O)C(n2cc(CCOCc3nc(C)cs3)nn2)C)c1 C1(CNC(C(CC)c2ccccc2)=O)CN(C(c2cc(C#N)n(C)n2)=O)CCN1C c1(C(=O)NCC(CCC)NC(C2(C)CCOC2)=O)cc2cnccc2[nH]1 C1(C(=O)NCc2ncc(C)o2)CC2CC1CC2NC(=O)Cn1cccn1 c1(-n2cc(C3CN(C(c4c(CC)occ4C)=O)C3)nn2)cc(F)cc(F)c1 c1(C(=O)NCCOCCN(C(C2CC(OC)C2)=O)C)csc2c1CCC(C)C2 CCC(CC)(CC(=O)O)N(C=O)C(c1ccccc1)C.c12cn(nn1)CC2 N1(C(CCCCOCC)=O)CC(NC(=O)C(F)n2cccn2)C(C2CC2)C1 CC1Oc2ccccc2OC1C(=O)NCC1CCCN1c1ccn2nccc2n1 N12CC(CC1=O)NC(=O)C2.c1(NC(=O)OC)nccc(C)n1 c1(CCC(=O)NCCCOCCNC(c2nncs2)=O)cccnc1Cl N1(C(=O)C(c2ccccc2)Oc2ccccc2F)CCC2(CCCNC2)C1 C(C(C)CC(=O)N1CCC(SCC)CC1)NC(C1(C(=O)OCC)CC1)=O N1(C(C(=O)NCC)=O)CC(C(=O)NC2CCCN(CCO)C2)C2(CCC2)C1 c1(CCC)c(C(=O)NC2CCC(NC(c3csc(C)n3)=O)C2)cnn1CCO N1(C(c2cc(C)n(CC)c2C)=O)CCCN(C(c2cc(C#N)c[nH]2)=O)CC1C C(=O)(C1=NNC(=O)C1)NCC(CC)NC(=O)C(C)(C)c1ccncc1 C(=O)(CCCCC(N)=O)NC(C(C)NC(c1n(CC)ccn1)=O)C C1(O)(CNC(c2c(C)nc(CC)s2)=O)CCN(C(=O)C(F)=CCCF)CC1 C1(C(=O)NCC(CNC(c2cccc3nsnc23)=O)O)CC12CCC(F)(F)CC2 c1(CC(=O)N(C(CC(=O)NCCCCCC)CC)C)csc2nc(C)cn12 N1(C(CC(COC)C)=O)CC2CCCC(NC(C3CCCSC3)=O)C2C1 N1(C(C2CC3C(C)(C)C3C2)=O)C(CNC(c2nncs2)=O)CC2COCC12 c1(C(=O)NC(CNC(c2[nH]n(C)c(=O)n2)=O)CC(F)(F)F)ccc2nnnn2c1 c1(C(N2C(C)(CNC(=O)CC3COCCO3)CCC2)=O)cc2cc(Cl)ccc2o1 c1(C(N(CC(C)NC(=O)COC(F)F)C)=O)ccc2c(c1)OCC2 c1(OCC)cc(C(N2CC(NC(c3cncnc3C)=O)CC(C)C2)=O)cc(F)c1 C(=O)(C(C(C)(C)C)NC(=O)C(CN(C)C)C(C)C)NCC1(CSC)CC1 C(C)(C)(CCCNC(c1nn(CC)cc1Br)=O)NC(COCC#C)=O c1(C(=O)NCCN(C(C2CC3C(C2)C3(F)F)=O)CC)ccc2c(n1)OCC(=O)N2 CCCC(C(O)C(=O)NC1CC2CC1C(O)C2O)NC(=O)C=CC1CCOCC1 CC1OCCN(C(c2cccn(C)c2=O)=O)C1C(=O)NCC(C)C(C)(F)F N1(Cc2cc(C)ns2)CC2(C)CN(C(c3coc(Cl)n3)=O)CC2(C)C1 N1(CCCNC(C(Cn2ccc(C)n2)C)=O)CCN(C(C23CC(CO2)C3)=O)CC1 C1(C(=O)OC(CNC(C(CCC)Cl)=O)=O)CCC2(CCCN(C(C)(C)C)C2)C1 O=C(CC=C1CC(CCC(=O)NC2(CCO)CC2)C1)NCC(CNC1CC1)O Cc1cn2cc(C(=O)NC3COCC3NC(C3CC4(CCCO4)C3)=O)nc2s1 Cc1ccc(CCC(=O)NC(c2c(C)noc2C)C)cc1C C1(CN(C(C=CCCC=C(C)C)=O)C)CN(C(=O)CC(=O)OC)CC12CC2 C(=O)(CCCCC(C)C)N1CCC(CNC(CCC(CC)C)=O)C(C)C1 CCCC(CC)C(C(=O)NC(C)C(=O)OCC)N1CCC(CN=[N+]=[N-])C1 C1(CCc2cnc[nH]2)C(=O)NN(CC)CC(=O)N1.C=C1CC(C(=O)OC)C1 C1(CNC(=O)Cn2cc(C3CC3)cn2)(Nc2nnc(O)s2)CCOCC1 C1(NC(c2ccc(CC)[nH]2)=O)CN(C(=O)C(c2ccccc2F)OC)CC1OC N1(C(C(CC=CC)NC(c2ccc(=O)oc2)=O)=O)CCCCCCC1C C1(C(=O)OC(C)C)CN(N2CC(n3cncn3)C2)C1 CC1C(NC(=O)C2=NNC(C(F)(F)F)C2)CCCN1C(C1CCC(=O)N1)=O Cc1cc(-c2cn(C3(C)CCCCC3O)nn2)ccc1N C1(NC(C(C)SCc2ccccc2)=O)CN2CCC1C2 C(=O)(C(C)(C)C1=CCSCC1)NC1C(NC(c2c(C)csc2)=O)COC1 C=CC(C(=O)NCC1(C(C)(C)O)CN(C(=O)CC(C)OC)C1)OC c1(CN(C)CC2CN(C(=O)Cc3cccc(Cl)c3)C2)cc(F)cc(Br)c1 C#CC1CCCN(C(C23CC(CO2)N(C(C2CC2CC(C)C)=O)C3)=O)CC1 CCCC(C)C(=O)N(CC(C)C(=O)NCCOC(=N)O)C C#Cc1ccc(C(=O)NCCC(=O)NCc2ccc(OC)cc2)cc1C c1(CNC(=O)NC2C(CC)(CC)CC2)ccc(-c2nn[nH]n2)c(F)c1 N#Cc1c[nH]c2ncnc(N3CCCC3C(=O)NCCCc3cccnc3)c12 C(CCC1CCC1)(C(=O)NCCC(C)(C)C)NC(c1cc(CC)[nH]n1)=O c1(C(=O)OC)ccnc(NC(C2CCCC2)CNC(=O)C2CC2)c1.C(=O)(C(C)SC)N CCC(CC)CCCC(=O)NC1CN(C(c2ccc(OC(F)F)cn2)=O)CC1C C1(C(=O)ONC(CC)=O)CCN(C(=O)CCNC(=O)Cn2cnnn2)C1C(C)(C)C C1(CNC(C2C(C=C)C2)=O)CCC2(CN(C(c3cnn(C(C)(C)C)c3C)=O)C2)O1 C1(CNC(=O)C(O)Cc2cccc(Cl)c2)CN(C(=O)Cc2cnc[nH]2)CCCO1 C(CC)(CCC(=O)N1CCSC2CCC12)NC(CC1(C(=C)F)CCC1)=O C1(NC(C2(F)CCCC2)=O)CCCC(c2ccccc2)CC1 C(=O)(C1=CNS(=O)(=O)N=C1C)N1CCC(NC(c2c(CC)occ2)=O)C2C1C2 C1(NC(=O)C(F)C2CCCC2)CC2(C1)CC2C(N1CCCCC1CCO)=O c1(C(=O)NC2CC(NC(CCC(=C)C)=O)CC2O)ccc(C)c(C)c1 CCCCC(F)C(=O)NCC1CC(CC(N2CCC(CC)C2)=O)C1 CCC(C#N)N(C(C(=O)NCCC#N)C1CC1Cl)C CCCCCCC(C)C(=O)NC(CCF)C(=O)NCc1ncsc1C CCC(CNC(C1CC12CC2(F)F)=O)(CC)NC(=O)C=C(C)C1CC1 c1(C(N2CC3CC(NC(C4CCCC(=O)N4)=O)C3C2)=O)cc2n(n1)CC1(CC1)C2 C1(OC)CCC(CCC(N2CCN(CC3(NC(=O)CCCF)CC3)CC2)=O)CC1 C(CCC(=O)NCCCOCC1CC1CNC(=O)Cc1ccon1)N(C(C)C)C c1(C(=O)NCC2(F)CC(NC(C(C)OC)=O)C2)cccc2c(C)ccnc12 CP(C)(=O)C(c1ccccc1)NC(=O)COC(c1csnc1Cl)=O CCC(CC)(C(=O)NCC1(CNC(c2nc(=N)cc[nH]2)=O)CCOCC1)C(C)C Cc1cn2ccnc(C(N3CCC(C)C(NC(=O)CCCC4CC4)C3)=O)c2n1 c1(C(=O)NCC(C2CC2)NC(C(C(=C)Cl)(C)C)=O)ccc(F)c(C)c1Cl CCCCCCCC(=O)NCCC1(NC(=O)Cc2c(OC)cccc2F)CC1 C1(NC(CCN(C)CCO)=O)CCN(C(c2ccc(Cl)c(C#N)c2)=O)CC1(C)C CC1(C)CCCOC1C(=O)NC1C(C(=O)NC2CC(=O)NC(=O)C2)C1(C)C O=C(CC1CS(=O)(=O)c2ccccc21)Nc1cc(F)cc(Br)c1F C1(NC(C(C)=CC)=O)CCC2(CC1)CC2NC(=O)CCc1cnn(C)c1C c1(C(=O)NC(CNC(c2c(C)nc(CO)o2)=O)C)cc(N(C)C)ccc1F C(C)(CCC(=O)NC1CCOC1)NC(c1c(C)occ1)=O CC(C)C(C)(O)C(=O)NCCC1(C(=O)NCCC2CCCCCC2)CC1 c1(C(C(=O)Nn2cnnc2SCCC2CC2)OCC=C)ccc(N(C)C)cc1 Cc1c(N(C(c2ccc(Br)cc2)=O)CC2CCCO2)cccc1[N+](=O)[O-] Cc1c[nH]cc1C=CC(=O)NC(c1cccnc1O)C(=O)NC1CC(C)OC1=O C(F)(F)(C(F)C(F)(F)F)OCCC(=O)O.c12ccccc1C(=O)NCC1CCCN21 c1(N(C)C)ccnc(C(=O)NC2CC2NCc2csc(-c3ccsc3)n2)c1 C(=O)(CCCCCNC(C)=O)NCC(C)(CC)NC(CN(CCC)C)=O c1(OCC)ccccc1N1CCOCC1.N12CC(C1)N(C)C2=O CC(CC(C)NC(C1CN(C(=O)CCc2ncccn2)CCN1C)=O)C(F)F C1(C2CCN(C(=O)C(F)(F)C(O)C3CC3)CC2)(NC(Cn2c(C)nnn2)=O)CC1 n1(CC)cc(C2OCCC2NC(=O)C2CC2)cn1.C12CN(C1)C(=O)CSC2 Cc1cc(C(=O)N(CC(C)CNC(C2CC2c2ccccc2)=O)C)ccc1O c1(N(C)C)ccc(Br)c(C(=O)NC2CC(N(C(=O)Cc3cncn3C)C)C2)c1 CC1CCCCC1NC(=NCC1CC1[N+](=O)[O-])NCc1ncccc1F C1(C(N2CCC(CN(C(c3c(C)cn(C)n3)=O)C)C2)=O)COCC(=O)N1C(C)C c1(C(=O)NC2(CN(C(=O)CC3COC4CC3C4)C)CC2)cc2cc[nH]c(=O)c2s1 C1(C(N2CC(OCCC(=O)NC3CCN(C(=O)NC)C3)C2)=O)CSCC(=O)N1 S(=O)(=O)(c1c[nH]c(C(N2CC(NC(C3(O)CCOC3)=O)CC2(C)C)=O)c1)N(C)C C=CC1(C(=O)NC2CCCC2(C)C)CCN(C(=O)C(C)CCOC)CC1 c1(N2CCC3(C(C(N4CC5CC5C4)=O)C3)CC2)ncnc2cccnc12 c1(C(C(=O)N(CC(=O)N(CC)CC)CC2CC2)O)cncn1C C1(CN(C)C(c2ncccc2Cl)=O)CC(F)CN1C(C12CC(C1)C2)=O Cc1cc(CNC(C2(CN)CCCO2)=O)oc1C.C1(C)CCN(C2CC2)C1 C1(CN(C(C2(F)CC2C)=O)CC)CCCN(C(=O)C=C(C)C(C)(C)C)C1 C#Cc1ccc(C(=O)NCC(N2CCCOC(C)C2)=O)cc1 C1(NC(CC(C)(C)O)=O)COCCN(C(C2CCCN(C(=O)C3CC3)C2)=O)C1 N1(C(C(CCC)N(C)C)=O)CCN(C(c2nncn2C2CC2)=O)CC1CO C1(NC(c2n(CC)nnc2)=O)CC2CN(C(c3cocn3)=O)CC2C1 c1(CCNC(C2(C)N(C(C(C=C)O)=O)CC=C2)=O)nnc2n1CCS2 Cc1ccc(N)cc1C(=O)NCC(C)(C1CC1)NC(c1cc(F)cs1)=O CC(CS(C)=O)C(=O)NCCCN(CCCCNC(=O)CC1(O)CCCCC1)C c1(CC)ncccc1C(=O)NCC1CC1CNC(c1cc(C(N)=O)c[nH]1)=O Cc1cc(C(=O)N(CCC(=O)Nc2ccc(F)cc2)C(C)C)nc(C)c1 C12(CNC(=O)Cc3cnsc3)CC1CN(C(c1c[nH]nc1F)=O)C2 N1(CC)CCC(C(=O)NCC(O)CN(C(=O)CSCCC(C)C)C(C)C)C1 Cc1nc(C(C(=O)NC2CCC2)N(C2CC3CCC2O3)C)nn1C C1(CO)CC(=O)NC1=O.C(C1(C)CONC(=O)O1)OC.OC N1(C(C(=O)NCCOCC(F)(F)F)=O)CCCCCC1n1cccn1 c1(-c2cn(C)nc2)nc(C2CC2(C)C)n(-c2cnnn2C)n1 c1(C(N(C)Cc2c(OC)cc(OC)nc2)=O)cc2nc(C)sc2[nH]1 N1(C(C(CC)CCOC)=O)CCN2CCN(C(=O)Cc3csc(C)c3)CC2C1 C1(NC(C(C)NC(N)=O)=O)CCCN(C(c2ccnc(F)c2Cl)=O)C1C C(=O)(CCCN1CCCC1)NCC1(C(C)NC(c2cc(Cl)cs2)=O)CC1 N1(C(C(C)OCC)=O)CCOC2(CCC(NC(c3cscn3)=O)CC2)C1 c1(N2CCC(NC(=O)CCC3COC3)C(F)C2)ncnc2cc(Br)ccc12 S(=O)(=O)(c1cnn2ccc(=NCc3cc4cnccc4o3)[nH]c12)NCC(CC)O N1(C(Cc2nc(C)oc2)=O)CC2(CCN(C(C3CCN(C)S3(=O)=O)=O)C2)C1 C(=O)(C1=C(c2nccn2C)N(CC)C(=S)NC1c1cc2sccc2s1)OCC N#Cc1ccccc1CN1CC(OC(C(F)(F)F)C2CCOC2)CC1=O C1(CC(=O)NCC(C)OC=C)CCCCN1C(=O)CNC(=O)CC c1(C(=O)NC2C(CNC(c3c(CC)occ3)=O)COC2)cn(C2CC2)nc1C c1(C(=O)NC(CCCCNC(c2c(CC)[nH]c(=N)s2)=O)C)ccc2nonc2c1 N1(C(C(C)=C(CC)C)=O)CC(O)CC1(C)C(N1CCOC(C)C1CO)=O C(=O)(C(F)C(F)(F)F)N(C1CCN(C(=O)CC2CCCCC2N)CC1)CC(C)C N1(CC)CCCC1C(N1CC(C)(NC(C2CCN(C(=O)NC)C2)=O)C1)=O C1(NC(N2CC(C(N(C)C)=O)CC2(C)C)=O)Cc2ccccc2C1O Cc1c(C(=O)Oc2cccc(F)c2)cccc1I.C12CCN(CC1)C2=O O=C(C#CC1CCCO1)N1CCCCC(CNC(c2ccc3[nH]ccc3n2)=O)C1 N1(C(C23OCC(CC)(C2)C3)=O)CCCCC(CNC(=O)C=Cc2nc(C)cs2)C1 C(=O)(CCCS(C)(=O)=O)N(c1ccc(N(C(=O)SCCC#N)CC)cc1)CC c1(CNC(C2CCCC(CC(F)(F)F)C2)=O)nc2c(s1)CCN(C(=O)CO)C2 N1(C(C(C)CNC(=O)Cn2cc(Cl)cn2)=O)CC2CC2C2CC12 n1(CC)cnc2nc(=NC3C=CCC3)[nH]c(NCCC3(CCCO)CCCC3)c12 C1(OC(=N)O)(COC)CC(C(F)F)C1.c1cn(CCNC(=O)C2CC2)nn1 c1(CC)oc(C)cc1C(N1CCCC1(C(=O)NC12CC(C1)C2)C(C)C)=O N(C1CSCc2ccc(Br)cc21)C(c1sc(CC)c(C)c1)=O c1(C(=O)NC2CC(NC(C3CCC(=C)CC3)=O)C2)cc2ccc(F)cc2o1 c1(CCC(=O)N(C(C)C)CCNC(=O)CC2CN(C)C2)n[nH]c2ccccc12 c1(OC)ccc(C(C)CC(=O)NCC23CC(NC(C4OCC4(C)C)=O)(C2)C3)cc1 c1(C(N(C2CC(NC(C3(OC)CC3)=O)C2)C)=O)cccc(Br)c1N N1(C(c2c(C(C)C)scn2)=O)CC(C)N(C(c2csnc2Cl)=O)CC1C N1(C(C2C(C(=O)NCC(C)(C)C)C2)=O)CC(C#N)C2(CCC2)C1 CC1(C)CC(C(=O)N2CC3CC2CN(C(c2cscc2F)=O)C3)=NO1 N1(C(c2c(Cl)cnc(CC)n2)=O)C2CCC1CN(C(=O)CC1COCC1(C)C)C2 C1(CCNC(CN(CCOC)C)=O)CN(C(=O)COC2CCCC2)CCS1(=O)=O c1(C(=O)NC(CC)CNC(=O)CC2CCC(C(F)(F)F)O2)c(C)cccc1C c1(CCNC(CN(C(=O)Cc2cncs2)CC#C)=O)cn[nH]c1 c1(CCC(N2CCC(N(C(C(C=C)O)=O)CCC)C2)=O)cc(F)cc(F)c1 C1(NC(c2cc(C(F)(F)F)ncn2)=O)CCN(C(=O)C(F)(F)C2CC2)CC1F c1(C(C(N2CCC(CNC(CC(C)F)=O)C2)=O)(C)C)ccc(C(C)(C)C)cc1 c1(C(=O)NCCNC(C2C3CC4C(C3=O)C24)=O)cc2cccn2cn1 Cc1cc(C(F)(F)F)nc(-c2nc(CC3CCCC3)nn2-c2ccnnc2)n1 N1(CCNC(C(=O)NC(CC)CCc2ccccc2)=O)CCC(N(C)CC)CC1 c1(NC(c2cccc(Br)n2)c2n(CC(=C)C)nnn2)ccnc(P(C)(C)=O)c1 C=C(Cl)CCC(=O)NCC1(F)CC(CNC(c2cnc(CC)[nH]2)=O)C1 N1(C(C(C)OCC2CC2)=O)CC2CC2(NC(C2CCOC2(C)C)=O)C1 Cn1ncc(C(N2CCC3(CC(NC(=O)OC(C)(C)C)CO3)C2)=O)c1S(C)(=O)=O C1(CNC(CCOCC(C)C)=O)COCCN(C(C2CCC2(C)C)=O)C1 N1(C(C2(C)CC=CCO2)=O)CCCC2(C1)CN(C(=O)C(c1ccc(O)cc1)=O)C2 c1(CC)nc(C(=O)NCCCN(c2ccccc2)C)c2ccccn12 c1(OC)nc(C)sc1C(=O)NCC1CC1CNC(=O)CC1CCCC1 C1(NC(C(C)=CC)=O)CCC2(CC1)CN(C(=O)Cc1ccc(O)c(Cl)c1)CCO2 CC1C(C(=O)NC(c2ccccc2Br)C(=O)O)C(O)C(=O)N1C c1(C(N(CC(C)NC(CC2(COC)CC2)=O)C)=O)ccc2c(c1)S(=O)(=O)NC2 c1(C(N2CCCC(F)(CNC(C3CC3C3CC3)=O)C2)=O)ccnc2ccnn12 CS(=O)(=O)C1(C(N2CC=CC(NC(c3c[nH]nc3-n3cnnn3)=O)C2)=O)CC1 c1(C(=O)NCc2c(C(=O)Nc3c(C(=O)OC)csc3)scc2)c[nH]c(C)cc1=O C1(CNC(CNC(=O)OC)=O)CC(C(=O)N(C2CCOC2=O)C)CCO1 C1(NC(COCCCOC)=O)CN(C(C2CC(=O)CCO2)=O)CC12CC2 C1(C(N(C)CCNC(=O)Nc2c(C)nc(C)o2)=O)CC12CCOc1ccccc12 c1(C(N2C(CNC(c3ncc(C)cc3C)=O)CC(F)C2)=O)cnc2c[nH]nc2c1 c1(C(=O)NCCC2CC(NC(C(C(C=C)C)C)=O)C2)cn2cnnc2cn1 C#CCC(C(=O)NCc1ccc(CC)cc1)C1CC1.C(=O)(CCC1CC1(C)C)NCC C1(NC(CCN(CC)CC)=O)CC(C)(C(=O)NCC)C1.C(=O)C(F)(F)F c1(C(N2C3(CN(C(c4cncc(O)c4)=O)C3)CC2)=O)cc2nccnc2cc1F C(=O)(C1=NN(C)C(=O)CC1)N1CCC(C)(C(N2CC(C)S(=O)CC2)=O)C1 c1(C2(C(=O)NCC(C3CCCCN3C(=O)CCF)O)CCC2)cccc(O)c1 c1(C(=O)NC2CC(O)(CNC(c3cnc(C4CC4)o3)=O)C2)cnc2c(c1)CCC2 C1(C(N(CCC(=O)Nc2ccccc2)C)=O)CNCC2(CCC2)C1 C(=O)(C1=CCCCC1)NCc1occ(C(=O)NC2CC(C)(C)OC2)n1 C=C(F)C1(CC(N2CCOC(C(C)NC(=O)Cc3nnc(O)s3)C2)=O)CCC1 N1(C(CNS(NC)(=O)=O)=O)CC=C(CCNC(=O)C(C)C2CCC2)CC1 CCC(CO)C(=O)N1CCCC1Cn1cc(CN2CCCCC2=O)nn1 C(CCCCCNC(=O)CCF)NC(c1cc(COC(C)(C)C)on1)=O c1(C(N2CCC(OCCNC(C3CC(F)C3)=O)C2)=O)ccc2c(c1)OCCO2 C1(C(=O)NC2CCN(C(c3ccnc(C)n3)=O)C2C)CC1C1CCCCC1 C(CN=C(NC1CC1)N(C)C(=O)NCC)(c1cccs1)NC(=O)NC(C)(C)C C1(CNC(=NCC)NCC2(C3CC3)CC2)C2CC3CC(C2)CC1C3 c1(-n2cc(CN(C(CN(C)Cc3ccccc3)=O)C3CC3)nn2)cc(F)cc(F)c1 C12(C(N3CC(CCCCNC(c4c(C)occ4)=O)C3)=O)CCN(CC1)CC2 c1(CNC(CCC(C)C2CCCCC2)=O)cc(N)c([N+](=O)[O-])cc1Br c1(OCC)ccc(NC(C2CCOC2CNC(=O)CC2CCN(C)C2=O)=O)cn1 Cc1c(F)cc(CN2CC(NC(c3cnn(C4CCCC4)c3)=O)C(F)C2)cc1Br CC1CN(C(=O)CC2CCCCO2)CC1CNC(c1cncn1C)=O CCC(CC(=O)NC(C)C(C)NC(c1cc(C)no1)=O)c1ccc(OC)cc1 Cc1cc(C(=O)NCC(C)(C(C)C)NC(=O)CN(C)C(=O)C2CC2)cc(N)c1Cl C1(C(=O)NCCCCNC(C2CCN(CC)C2)=O)Cc2cc(Cl)ccc2C(=O)O1 N1(C(CCCC#C)=O)CCC(NC(C2CC(CC)C2)=O)CC(O)C1 c1(CC(C)N(C(C2C(CC)OCC2)C(=O)NC(C)C)CC)ccc(F)cc1 C1(NC(C2(C#N)CCCOC2)=O)CCCCCCC1NC(=O)C(Cl)=CCl N1(C(C=C(C)C(C)C)=O)CCN(C(=O)Cc2nc(C(F)(F)F)nn2C)C(C)C1C C1(CNC(C=CCN(C)CC)=O)CC2(CC2)CN1C(c1cc(C)n(C(F)F)n1)=O c1(C(N2CCC(N(C(=O)COC3CC=CC3)CC)C2)=O)cc([N+](=O)[O-])c[nH]1 C1(NC(CCCOCCOC)=O)CN(C(c2cnn(C)c2C(C)C)=O)CC12CC2 S(=O)(=O)(c1ccc(=NCC2(C)CCCO2)[nH]c1)NC(C)(C)CN1CCCC1 CC1CC=C(C(=O)NCC2CCC2NC(c2nc(Br)sc2Cl)=O)CC1 C1(C(N2CC(C)N(C(c3ccn(CC#N)n3)=O)CC2)=O)CCc2cn(C)nc2C1 Cc1nc(-c2cnn(CC(N)=O)c2)sc1CC(N1CCOCC1)=O.C(C=O)NC=O C(=O)(C1CCCn2ccnc21)NC1C2(CCN(C(COC3(C)CCC3)=O)C2)C1 C12CCN(CCC1(F)F)C2=O.C12(CCCC(=O)OC)CCOC1CC(=O)NC2 CC1CCN(C(c2nc(C(F)(F)F)cs2)=O)CC1N(C)C(C12CCCC1C2)=O CC(C)(O)C#CC(=O)NCC1(C)CCN(C(C2CCN2C(=O)OC(C)(C)C)=O)C1 CCCN=C(NCc1cccc(C)c1C)NCC(C(F)(F)F)n1cccn1 N1(C(C(c2ccncc2)C)=O)CCC(C(=O)NC(CO)C2(O)CC2)C(C)C1 C1(CC=C)(NC(c2cc(=N)[nH]c(Cl)n2)=O)CCCN(C(=O)C(CC2CC2)OC)C1 C(C1CCCN1C)=CC(=O)NC(CCOC)CNC(=O)CCOCCCOC C(C)(CC(=O)NC(C)(C)CNC(=O)Cc1cc2ccccc2o1)(C(F)F)N(C)C c1(NC(CCSCCCC)=O)cccc(C(=O)NCCN(C(=O)CC)C)c1 CC(C)C(CC1CCCCC1)C(=O)NC1CCCC(NC(=O)C2=CCCOC2)C1 C1(NC(C(C)OCCCC)=O)CN(C(=O)CC(C)(C)O)CC1S(C)(=O)=O c1(OC)nccc(C(=O)NC2CCC2CNC(=O)Cc2ccc(C)o2)n1 C1(CC(=O)NCCC(C)NC(=O)CCc2ncc[nH]2)CC=CCC1 CC(O)CCN=c1[nH]c(=NCc2nc(CC3CC3)n[nH]2)c2cccc(F)c2[nH]1 c1(CC)ccc(C(=O)NCCN(C(c2cc(-c3ccco3)[nH]n2)=O)C2CC2)o1 C1(C)(CC)C=C(C(=O)NCc2ccc(C(C)NC(c3ccccn3)=O)cc2)C1 N1(Cc2cn(CCC)nc2)CCN(C(=O)NC2CC(CNC(C)C)C2)CC1=O CC(C)C(CC(=O)NCCN(C(=O)C1=CCCSC1)C12CCC(CC1)C2)c1ccon1 N1(C(C(c2cn(C)nn2)NC(CC2ON=C(C)C2)=O)=O)CCC(F)(CF)C1 S(=O)(=O)(c1ccc(NCCC2CCCC2)c(C#N)c1)NC(CCC)C1CC1(C)C CC1CCC(=CC(=O)N(C)CCOCCNC(=O)CC2CCC2)CC1 C(C(=O)NCCCC1CCC1)(C1CCCO1)NC(=O)OC(C)(C)C Cc1cccc(CC(=O)NCC2CC(C(=O)NCC3CC(C)OC3C)CO2)c1 CNS(=O)(=O)N1CCC(C(=O)NC2C=CCN(C(=O)C=CSC)C2)CC1 C1(NC(C(N2CCCCCC2)C)=O)CC2(C1)CC2Nc1ncncc1I C1(C2CCC2)(NC(COC(C)(C)CNC(=O)C(F)=CC2CC2)=O)CCC1 C12CCN(CC1c1ccccc1)C2=O.Cc1nn(C)cc1-c1ncc(C(C)C)s1 c1(OC)nc(C)c(Br)cc1C(N1CCC(NC(C2(O)CCC2)=O)C1)=O N1(C(C(CC=C)c2ccccc2)=O)CC2CCCC2(N)C1 C1(C(=O)NC(C2N(C(COCCC=C)=O)CCC2)C)CCCOC1CC N1(C(=O)C=Cc2cn[nH]c2)CC2(CCN(C(C3CCC4CCC34)=O)C2)C1 N#Cc1sccc1C(=O)N.O=C(COC1CCC1)NC1CC1C(F)(F)F N1(C(C(C)OC(C)=O)=O)CCCC(F)(CNC(=O)CC2COCC2(C)C)C1 CCCC(C)CC(=O)N1CC(CNC(C2CCCCN2C)=O)CC1C N1(C(CC2N(C(C(CC#C)C3CC3)=O)CCCC2)=O)Cc2n[nH]cc2C1CO C(=O)(C(C)P(C)(C)=O)NC1(C)CN(c2c(C(=O)OC)nccn2)C1 c1(OCC)sccc1C(=O)N(C(C)CNC(c1cnc(C2CCC2)o1)=O)CC c1(CCC)nc(=NC(C)(C)CNC(=O)CN2CC3CC3C2)s[nH]1 C1(CC(=O)N(CC(CN(c2nnc(C3CC3)s2)C)O)C)CCCC(F)(F)C1 N1(C(CCNC(COC)=O)=O)CCCN(C(=O)CC(C)(C)C)C(CO)C1 C1(CC(=O)NC2CC(CNC(C3(COC)CCCCO3)=O)C2)CCCCCCC1 c1(OC(C(=O)NC(CCOC)CNC(c2cnoc2C)=O)C)cc(F)cc(F)c1 N1(C(C(CC(C)C)OC)=O)CC(N=[N+]=[N-])CC1C(=O)NCCCOC(F)(F)F c1(C(=O)NCC(CC)NC(c2snnc2C)=O)cc2c(OC)ccc(F)c2[nH]1 c1(-c2cn(C(C(=O)NC3C(C(=O)OC)C3)C)nn2)cc(F)c(F)c(F)c1 C12(CNC(COCC(C)(C)C)=O)CCCC1CCN2C(=O)Cc1nncs1 c1(C(=O)NCC2CCC(NC(C(CC)C(C)C)=O)C2)cc2c(Cl)cccc2s1 c1(CC(=O)NON2CC3(CCCC3)C2)cc2ccccc2[nH]1 N1(C(C)=O)CCCCC1C(=O)NCCCCNC(=O)C(C)c1cccs1 C(=O)(C(C)CC(C)(C)C)NCc1cc(C)c(C(=O)NCCC(O)C(C)C)o1 c1(C(N2CC(OC)C(NC(=O)Cc3ccccc3)C2)=O)ccc([N+](=O)[O-])cc1F CCCC(C)(C)CC(=O)NCCCCCCC(=O)NCC1CCCCC1(CC)CC C(=O)(C1Cc2ccc(F)cc21)N1CCN(CC(=O)OC)C(C)C1 c1(N(N2CCC(c3cn[nH]c3)CC2)C(C)=O)ccc(F)c(Cl)c1 CCCCCC(F)C(=O)N1CCN(C(=O)C(c2ccc(C)cc2)=O)C2CC12 Cc1nnc(CCC(N2CCCCC2CNC(N2CCOCC2)=O)=O)n1C c1(C(N2CCC(N(C(C)=O)C)C2)=O)ccc(NC(=O)Cn2cncn2)cc1 CC(c1ccccc1Cl)=CC(=O)N(C(C)CNC(=O)Cn1ccc(=N)[nH]1)C C(=O)(C1CCC(=O)c2cccn21)NC1CC(C)N(C(C2CCC(C)(C)C2)=O)CC1 C1(C(N(CCNC(=O)CC2CC3CC3C2)CC)=O)CCN(C)S1(=O)=O N#Cc1cncc(NC(C2CCC(CNCc3ccc(C(=O)O)cc3Cl)CC2)=O)n1 c1(C(N2CC(C(C)NC(c3c(C)cns3)=O)OCC2)=O)nn(C)c2c1CCCC2 C1(C)(CNC(c2n(CC)nc(C)c2)=O)CC(F)(F)CN1C(C1CCNC(=O)C1)=O CCC(CCOC)NC(C1(NC(=O)CC2CCC(=O)C2)CSC1)=O CC1CC(CC(=O)NC(C)CS(N)(=O)=O)CN1C(=O)C(c1cccn1C)=O CN1N=C(C(=O)NCC2CCN(C(=O)CC3CCC(C)(C)O3)C2)CCC1=O CC(C)CC(CNC(=O)C(C)C#N)C(=O)N(C)Cc1cocn1 c1(C(=O)NCC(CN(C(=O)CCC2CCCC2)C)(C)C)cccc(C(F)F)c1F C(C(CC(=O)NCC1OCCC1(C)C)NC(=O)CCc1csnn1)OC N1(C(=O)NCC2CC(OCC)C2)CC(C)(C)C1c1nccn1C N1(C(=O)OC(C)(C)C)CCOCC1CCNC1CCCN1c1ccc(C(N)=O)o1 C1(C(N2CC3C(NC(C(C4CCC(C)CC4)CC)=O)(C3)C2)=O)CC(C)(C)OC1(C)C N1(C(CC2C(C)OCC2)=O)CC(C2CC2C(N2CCCC2C(N)=O)=O)C1 c1(C(N2CCC(CC=C)(NC(=O)CNC(N)=O)C2)=O)[nH]nc2cc(F)c(Br)cc12 CCC(C)C(C(=O)NC(C1CN(C(C2CC(CF)C2)=O)C1)C)OC C(C(C)(C)CNC(=O)CC1CCCCC1)N(C(C12CC(C)C1C2)=O)CC C(=O)(CC(C)(C)c1ccc(F)cc1)N1C(C(C)NC(=O)CC2CC=CCC2)CCC1 c1(CC)ccc(C(=O)NCC(C)(F)CNC(C2(C(C)(F)F)CCC2)=O)c(O)c1 C(=O)(CCC1CCc2ccccc21)NCC(CC)NC(c1nnc(O)nc1O)=O C(c1ccco1)=CC(=O)NCC(=O)NCCCNC(CCN(C)C1CC1)=O c1(NCCc2n(C)cnn2)nccc(=NCCc2ccc(-c3cccs3)cc2)[nH]1 N1(CC(C)(C)F)CCN(C(=O)CC2CCCO2)CC1 C1(C(C)(C)NC(=O)CNc2cn[nH]c2)CCCN1C(=O)CC1CCC1 c1(NC(=O)CCC2CCN(C(C3CC4(CC4)C3)=O)C2)csc(Cl)c1 c1(NC2CC3(CN(C(CC=C)=O)C3)OC2)ncnc2[nH]nc(C)c12 c1(C(N2C(C(N3CCC(C(F)(F)F)C3)=O)CCCC2)=O)ccc2c(c1)CCC2 C(=O)(C(F)(F)C(F)(F)C(F)F)N1CCCC(CNC(=O)C2=CCOC2)C1 N1(C(c2nc(=N)[nH][nH]2)=O)CCN(C2CN(C(c3cc(O)no3)=O)C2)CC1 c1(CNC(c2c(CC)noc2)=O)ccc(C(=O)NC(CC)(CC)CO)cc1 C=C(C)CCC(=O)NCC1C(C)CCCN1C(=O)CCSCc1ccccc1 N1(C(C(C)c2cccs2)=O)CCCN(CCO)CC1.C(CCC1(NC=O)CC1)S C(=O)(C1Cc2ccccc21)N1CC(C)(NC(c2c(C)coc2C)=O)C1 C(C)(CCC(=O)NCc1nc(SC)ns1)NC(C(CC)SC)=O C1(N(c2cccc(OC)c2Cl)S(=O)(=O)CC2CCC2)CCCC12CCNCC2 C(=O)(C(C)(C)CCC#N)N1CCC(C)(CC(=O)NC(C(=O)N(CC)CC)C)C1 C(CNC(C)=O)(CC(=O)NC1CC1C(=O)NC(c1ccco1)CO)OC N1(C(CN(C)S(N)(=O)=O)=O)CCC(C)(NCCCN2CCC2)CC1 N1(C(c2ncnc(C)c2C)=O)CC2CC(NC(=O)CCOCCN(C)C)C(C2)C1 c1(C(C(=O)N(C(CNC(CCC#CC)=O)C)CC)C)ccc(Br)cc1C N1(C(CCC=C)=O)CCC(N(C(=O)C(C)COC)CC)CC1 CN(C)S(=O)(=O)N1CCC(C(=O)NCC2CCCN2C(=O)C2=CCS(=O)(=O)C2)C1 C1(NC(CC=CC)=O)CN(C(=O)CC(CC)CCCC)CC2(CCC2)C1 CC1(C)CCCOC1C(=O)NC1CC(NC(=O)CC2CCC=CCC2)C1 Cc1c(C(=O)NCC2CC(NC(=O)CC3CCCO3)C2)cnn1CC(F)(F)F C1(NC(C2CC2F)=O)CN(C(=O)CN2CCCC2)CCC1c1ccc(F)c(F)c1 c1(CNC2CCCC2)ccc(CNCCOC(C2CCN(CC)CC2)=O)cc1 N1(C(C2CC3C=CC2C3)=O)CCCN(C(C2COC3(CCC3)C2)=O)CC1 Cn1cccc(C(N2CCC(C)(CC(=O)NC3CCOCC3F)C2)=O)c1=O N1(C(C(C)CNC(=O)C(=O)C(C)(C)C)=O)CCCC2(CCCC2)C1 c1(CN(C2CCC(C)C2C)C(COc2c(C)cccc2)=O)cccc(C#N)c1 C1(OCC#C)CCN(C(C2CCCC2NC(=O)CC(C)n2ccnc2)=O)CC1 c1(CN=C(NCC2C(C)C2)NCCCOCC2CC2)cc2ccccc2cc1Cl N1(C(Cc2cc(C)on2)=O)C2CCC1C(F)C(NC(C1(F)CC1)=O)C2 C=CCC(F)(F)C(=O)NCCC(C)(C)NC(=O)CC1CCC(C)C1 O=C(C1=NNC(=O)C1)N1CC(C2CC2)(C(=O)NC2CC(CO)C3CC23)C1 Cc1ccc(O)cc1C(=O)NC1(C)CC(NC(=O)CSc2ccc(F)cc2F)C1 Cn1c(COCC(N2CCOCC2CNC(C2CNC(=O)N2)=O)=O)nnc1S C1(NC(Cc2c(C)cccn2)=O)CC(F)CN(C(=O)CC(C)(C)CN(C)C)C1 C(=O)(C(C)(C)CCS(C)(=O)=O)N1CC2C(NC(c3cnc(OC)c(C)c3)=O)C2C1 Cc1cnn2cc(C(N3CCC(CCNC(=O)C(C)CC(C)(C)C)C3)=O)cnc12 c1(C(=O)NCC2CCCC(NC(c3scc(OC)c3)=O)C2)cccc(Cl)c1C Cc1nc(C(=O)NCCC2CN(C(c3nncn3C3CC3)=O)C2)c(C)o1 c1(C(N2CC(C#C)(C(=O)NC(c3cscn3)CO)C2)=O)cc[nH]c2nccc1-2 c1(OC)ccc(C=C(CCC(=O)OCC)C(=O)N2CC(C3CCCO3)C2)c(C)c1 Cc1ccc(Cl)c(C(N2CCN(C(=O)CC3(N4CCCC4)CC3)CC2CF)=O)c1 C1(N(C(C2CN(C)C(=O)N2)=O)C)CCCCN(C(=O)C=Cc2nccs2)C1 C(CNC(c1cnoc1C)=O)(CCNC(C1C=CCS1)=O)OC c1(C(N(CCNC(C2(C)CCCCC2C)=O)CC)=O)cccc2ncsc12 N1(C(c2cnc(CC(C)C)s2)=O)CCC(C(C)NC(C2CC3(CC3)C2)=O)CC1 CCC(O)C(C)C(=O)N1CCC(C)(CNC(c2cc(=O)n(C)o2)=O)CC1 CCCC(CCC)C(=O)N(C(C)C(=O)N(CCC(=O)OC(C)(C)C)C)CC c1(CC)c(C(=O)NC(C23OCC(C(N4CCC(CC)C4)=O)(C2)C3)C)cnn1CC C(CS(=O)(=O)CC(=O)NCC(C1CCN(C(C2CCOC(C)C2)=O)CC1)C)OC N1(C(C(=O)NC2C(CNC(c3cn(CC=C)nc3)=O)COC2)C)CCN(C)CC1 C(N=c1[nH]c(=NCCC(C)C(C)C)[nH]c2c1CCC2)c1cc(C)nc(Cl)c1 c1(CCC(N2CC(CNC(C=CC=CCC)=O)(COC)C2)=O)ccc(OC)nc1 Cc1ccc(C(N2CCOC(C(=O)Nc3cnc(F)c(C)c3)C2)=O)cc1C N1(C(Cc2c(CC)cccc2)=O)CC2CC1CN(C(c1c(C)csc1C)=O)C2 C1(CCC(C=CC(C)NC(CCc2nc(C)sc2)=O)=O)CCCC2CC12 N1(C(C(CN(C)C(c2ccc(O)nc2)=O)(C)C)=O)CCC2(CCC2)CC1 C(C(C(=O)NOC1CCCC1)C(C)C)NC(CC1ON=C(C)C1)=O N1(C(CCCC#CC)=O)CC(C)(CNC(=O)C(C)OCCOCC)CC1(C)C C=C(Cl)CC(C(=O)NC(C(O)CO)C1CC1)NC(=O)Cn1ncccc1=O C1(NC(CC(=O)NCC#C)=O)CC2CN(C(=O)CC3(CS(C)(=O)=O)CC3)CC2C1 c1(C(C2CCCCC2)NC(=O)NCC2CN(CC(F)(F)F)C2)cccc(O)c1 C1(C(=O)NC2CC23CCN(C(c2cncs2)=O)CC3)COc2ccc(F)cc2C1 c1(C(=O)NC2C(C(=O)NC(C=C)C)CCC2)ccc(F)c(C)c1Cl N1(S(CC)(=O)=O)CCCCC1C(=O)NC1CN(C(c2cn(C)c(C(F)F)n2)=O)C1 C1(C(=O)NCCCCC2CCC2)CCC(C2CC2)N1C(=O)C1=NOCC1 C1(CNC(Cn2ccc(C)n2)=O)CN(C(c2nn(C)cc2Cl)=O)CCC1C C1(CC(=O)NCC(C)NC(CNC(=O)NC)=O)CCC(=O)N1C C(=O)(N=c1ccn(C(F)F)[nH]1)c1ccc(CNC(=O)CCCF)nc1 N1(C(C(CCC)NC(=O)Cc2ccc(C)cc2)=O)CCC2(CC1)CC2C#N c1(C(=O)NCC(CO)NC(=O)C(F)n2ccnc2)cc(F)cc(Br)c1F C1(NC(C(CC)OC2CCCC2)=O)CCCN(C(=O)CCCc2sccc2C)C1C O=C(N=c1cnc(Cl)c[nH]1)C1CCC2(CN(Cc3ccncc3[N+](=O)[O-])C2)O1 C1(CNC(C2C(C)(C(F)(F)F)C2)=O)C2CN(C(C3(C)CCOC3)=O)CC12 Cn1c(=O)[nH]c(NCC2COC(NC(=O)CNC(=O)CCCCO)C2)c(C#N)c1=O N1(C(Cn2c(CCC)nnc2S)=O)CCC2CN(C(c3cnn(C)n3)=O)CC2C1 C1(C)(N(C(c2cccc(C(C)C)c2)C(=O)NCCC(=O)OCC)C)CCN(C)C1 CCC(CC(F)(F)F)C(=O)N1CCN(C(c2c(C)nn(C)c2OC)=O)CC1 C(N=c1[nH]c(=NCC2(CSC)CCC2)[nH]c2c1SCC2)C1(CCOC)CC1 CC(C)C#CC(=O)NCC1(F)CC(CNC(=O)CCC(=O)NC2CCCC2)C1 c1(CNC(c2cncc(Cl)c2Cl)=O)nnc2n1CCN(C(c1csc(O)n1)=O)C2 c1(C(=O)NC(C(CO)NC(C2(OC)CCCC2)=O)C)cnc(O)c(Cl)c1 c1(SCCC(=O)NCC2C(NC(c3ncn(CC)n3)=O)C2)nc2ccccc2s1 c1(C(N2CCCCC(N(C)C(C3COC(=O)C3)=O)C2)=O)cccc2oc(O)nc12 N1(Cc2c(C)c(Br)cc(F)c2)C(=O)C2CC=CCC2C1=O C12(C(N(CC(C)O)CCNC(C(C(C)C)n3ccnc3)=O)=O)CCCC1C2(F)F C1(NC(C2CC(Cl)(Cl)C2)=O)CC2CCC1C(NC(c1ccc(C3CC3)s1)=O)C2 C1(C(=O)NCC(CC)O)CC(NC(=O)CCOC2CCC2)CCO1 c1(C(N2CCCC(N(C(CCNC(C)=O)=O)C)C2)=O)cccc2ncccc12 C(=O)(C1CCn2cc(-c3ccccc3)nc21)NCC(CCOC)O CCCC(C(=O)N1CCC(NC(C23CC=CC(C2)OC3)=O)C(C)C1)S(N)(=O)=O C(C1=Nc2ccccc2S(=O)(=O)N1)N.C(C(O)CNC)OCC C(=O)(C1=NOC2(CCOC2)C1)NC1CCN(C(c2c(NC(C)=O)c[nH]c2C)=O)C1 c1(NC(c2nnnn2C(c2ccccc2)C)C2(CC)COC2)cccc(C)c1 C(=O)(CS(=O)(=O)C1CCCC1)N1CC(NC(C(CN(C)C)(C)C)=O)C2C1C2 C1(CCNC(C2(SC)CCC2)=O)CN(C(=O)C(C)OC)CCO1 C=CCC(F)(F)C(=O)NCC1N(C(c2ccncc2Br)=O)CCC1(C)C C#Cc1cccc(NC(C2CCCC2CC)(c2nnnn2CCOC)C)c1 C(=O)(C(CCF)NC(=O)C(CC)=CCCC)N(CCCC=C)CC C1(C(=O)NCC(C)(C)OCC(=O)NC(C(=O)NCCC)C)C=C(C)CS1 c1(C(=O)NCC(C(C)C)(C)NC(=O)Cc2ccoc2)cc(F)c(F)c(C#N)c1 C(=O)(C1=CCN(C)C1)N1CCC(C(C)C(=O)NCCOCC2CC2)CC1 c1(C(=O)NC(C)(CNC(c2ccc(F)c(Cl)c2)=O)CO)cc(F)c(N)c(F)c1 c1(OCC)cc(OCCOC)c2c(c1)COC(C(=O)NC1CCCC(CC)C1)CC2 C1(NC(CNS(NC)(=O)=O)=O)CN(C(C2CC3(CC(OC)C3)C2)=O)CC12CCC2 c1(C(=O)NCC2C(NC(c3c(CC)ocn3)=O)C2)sccc1S(C)(=O)=O N1(C(Cc2ncc(C)s2)=O)CCC2CN(C(=O)CC3CCC(C)(C)CC3)CC12 N#Cc1cn(CC(N2CCC2CNC(=O)CC2CCCCCC2)=O)c(=O)nc1O C(=O)(C(C)CS(C)=O)NCc1cccc(CNC(c2n(C=C)nnc2)=O)c1 C(CCC(C)C)(C(=O)N1CCCC(CC)(NC)C1)NC(c1cncc(CC)c1)=O c1(C(=O)NC2(CCNC(C3C(C)(C)C3(C)C)=O)CCC2)cc2c(cn1)CCCC2 C(=O)(C(F)(F)C(F)(F)C(F)F)NC1CCCC(NC(c2ccncc2)=O)C1 c1(NC(C2N(Cc3scc(C)n3)CCC2)=O)cnc(Cl)c(Br)c1C c1(C(=O)NC(CC=C)CNC(=O)C=C(C)C(F)F)cnnc(C2CC2)c1 c1(C(N(CC(CC)NC(=O)CC2(C)CCCO2)C)=O)c2c(nn1C)CCOC2 C1(C(=O)NC2CC(C(C)NC(=O)Cn3cc(CO)nn3)C2)(OC)CCCOC1 C(CCCCC(=O)N1CC(NC(N2CCCCC2)=O)CC(O)C1)NC(N)=O CC(C)CCC(C(=O)N(C12CC(C1)C2)C)NC(C1CC2CC1CC2=O)=O C1(NC(C(C)(F)F)=O)CC(NC(=O)CCOC2CCOCC2)C12CCC2 C1(C)(NC(C(COCC)C)=O)CCN(C(C2CCCC2O)=O)CC1 C1(O)(CC)CCCN(C(=O)C(C)C2CCC2)C1.C1(=O)CCN1C(C)C C1(CC)CCCC1(C)C(=O)NCC(C)N(C)C(c1nccs1)=O N1(C(CC2(NC(=O)Nc3ccnnc3)CC2)=O)Cc2ccccc2CC1CCO C1(CCN(C)C(C2CCC2(F)F)=O)CCN(C(=O)C=CC2CCC2)CC1 Cc1ccc2[nH]cc(C(=O)NC(C3(O)CN(C(=O)CC4CCCC4)C3)C)c2c1 C=CC1OCCC1C(=O)NCC=C1CCN(C(=O)C=Cc2ccco2)CC1 c1(OC)ccncc1C(N1CCC(C(C)C(=O)NCC(COC)CO)C1)=O c1(C(N2C(CN(C(CC(=C=C)C)=O)CC)CCC2)=O)cc(Cl)cnc1C C1(NC(C(CC)NC(N)=O)=O)CC2CCC1N2C(c1cn(C)cn1)=O C1(CCCC)CN(C(=O)CN(CC(C)C)C(C2CC(C)C2)=O)C(CC)CO1 c1(C(=O)NCC2N(C(c3scc(OC)c3)=O)CCC2)ccc2nccnc2c1 C(=O)(C(C)(C)C)OCCOCC(c1nc(C(C)(C)C)on1)O N1(C(Cc2ccc(OC)c(O)c2)=O)CCN(C(c2sc(O)nc2C)=O)C(C#N)C1 c1(C(CN2CCC(NC(=O)C(=O)NC(C)C)CC2C)OC)cc(Cl)nc(Cl)c1F C1(C(=O)Nc2ccc(Br)nc2C(F)(F)F)CC12CCC1(CC1)CC2 N1(C(Cc2c(C)noc2)=O)CCCC2C1CCN2C(=O)CC(O)C(C)C C(=O)(C(C)(CNC(C1CCN1C(C)(C)C)=O)CC)N(C1CC(CC)C1)C O=S(=O)(c1cccnc1)N1CCC2(CCN(Cc3nccnc3Cl)C2)C1 c1(COCC)ncc(C(N2CCC(C(=O)NC3CCC3)C2)C(=O)N(C)C)[nH]1 N1(C(CCS(C)(=O)=O)=O)CC2CC1CN(C(c1coc(C(F)F)n1)=O)C2 Cc1cc(F)c(C(=O)NC2C3CC2N(C(c2ccc(F)s2)=O)C3)cc1F N1(C(C(C2CCCC2)NC(C2(C(CC)=O)CC2)=O)=O)CCC(C(=O)NC)C1 c1(OC)cc(C(=O)NC(c2ccccc2)C(C)NC(=O)CSC(C)C)cc(F)c1 N1(C(CNC(C(C)(C)SC)=O)C)CCN(C(=O)CN(C)C)CC1 CS(C)(=O)=NCC(=O)N1CCC(CNC(c2csnc2Br)=O)C1 c1(N2CC(CC)SCC2)nc(N(C)Cc2ncn(C)n2)nc2c1CCCC2 CCC(CC(=O)NCC(C)(C)CN(C(=O)CN1CCCC1CO)C)C(F)F CC(C(=O)N1CC2CC1C2NC(C1(c2c(F)cccc2F)CCC1)=O)C(C)(F)F C1(=CC(N2CCC(C)(CNC(COCC#C)=O)C2)=O)CCC(C)(C)CC1 C=CCC1C(=O)N1C.C1(C)CCCCN1C(=O)C=Cc1nccs1.OC C(=O)(C(C)(O)C1CCOC1)NCCOCC(=O)NCCN(C(=O)CC=CC)CC c1(C(N2CC3C(C(=O)NC4(CC5CC5)CCC4)C3C2)=O)ccc2cc[nH]c2c1 N(C1CCc2ccccc21)N1CC(C(N(CCC(=O)O)C)=O)C1 CC1(C)CCOC1C(=O)NCC#CC1CC1.C12(CCCCC1)CC(=O)N2 c1(OC)cc(F)c(F)cc1NC(C1CCN(Cc2cn(C)nc2C)CC1)=O N1(C(CN(C(C(CC=CC)C)=O)C2CC2)=O)CCC(C)(C#N)C1 C1(CNC(c2ccc(CC)o2)=O)CC2(CCN(C(=O)Cn3nnc(C)n3)C2)CO1 Cc1ccc(C(N2CCCC2CNC(C2(C)CC3CCC2O3)=O)=O)cc1F C=C=C(C)CC(=O)NC(C)CC1CCN(C(c2cccc(C3COC3)c2)=O)CC1 Cc1cc(C)c(C(=O)NC2C=CC(CNC(C3(C(F)(F)F)CCC3)=O)C2)c(O)n1 c1(CC(C)C)ccccc1C(=O)NCCCNC(=O)Cc1ccc(C(N)=O)cc1 C12(C(N3CC(CNC(C4N(C(C)=O)CSC4)=O)C(C)CC3)=O)CCCC1OCC2 c1(C(=O)NCC2N(C(C(C(C)C)n3ncc(C)c3)=O)CCC2)cc(C)nc(C)c1 C1(NC(c2c(CCC)n(C)nc2)=O)CC2CC(C1)N(C(=O)CC(CC)CC)C2 C1(C)CCCCC1(C)C.C1(N2C(=O)C(C)N2C(=O)CCC=CC)CCOC(C)(C)C1.CC N1(C(C(C)(C)CO)=O)CC=C(CCNC(=O)CN2CCC(C)(O)C2)CC1 C(=O)(CC(C)(C)c1ccccc1)NCC(C)NC(C1OCCOC1C)=O C(=O)(C1=NN2CC(C)CN=C2N1)NC(CCN(C(C1(CC)COC1)=O)C)C1CC1 c1(NCC)ccc(C)nc1C(N1CCCC(CNC(C2CC2OC)=O)C1)=O N1(C(C2CC(CNC(C(F)=CCC)=O)C2)=O)CCC(C)C2(CCC2)C1 C1(C(N(CC(CC)NC(=O)CCC23CCC(CC2)C3)C)=O)CNC(=O)C(C)(C)C1 C(=O)(C(C)S(=O)(=O)C(C)C)NCCCC(C(=O)CO)C.c1(N)ccc(Cl)cc1 C1(C)(C(=O)OC)CCN1C(=O)C(C1(C)CC1)NC(=O)CC1CSC1 N1(C(c2n(CC)ncc2Br)=O)CCOCC(F)(CNC(=O)CC(C)SC)C1 C1(OC)CCC2(CC(=O)NCC3(O)CN(C(=O)CC4CC5(COC5)C4)C3)CCC12 C1(NC(CCNC(C)=O)=O)C2CC1N(C(C1(CF)CCC1)=O)C2C C1(C)(C(=O)NCC(C)(C)C)C=CCN1C1CC1.C1(C(=O)NCCO)CC1C(=O)N.O C(=O)(C(F)(F)C(F)F)NCC(CNC(c1c(OC)cc(C)s1)=O)F C1(NC(C=COCC)=O)CN(C(=O)C(c2csc(C)n2)=O)CCC1C C1(NC(C(C2CC2)OC)=O)CCCN(C(c2cc(-n3cccc3)ccn2)=O)C1 CCC(C)(CNC(=O)COC(CCSC)C(=O)NC1CCC1)C(N)=O.OC c1(N2CCCC(NC(Cn3c(C)ncc3)=O)C2)ncnc2c1CCO2 C12(C(N3CCCC(NC(C4(C#C)CCCC4)=O)C3C)=O)CCCC(C)(C1)OC2 c1(C(N2CCCC(NC(C3(C(C)(C)C)CCC3)=O)CC2)=O)cc2ccncc2s1 C1(CC(=O)N(C(C(=O)NC(CC=CC)CO)C)CC)CCC(C)(C)O1 C(=O)(CS(=O)c1ccc(Cl)cc1)NCCNC(c1cncc(OC)c1)=O N1(Cc2ncccc2F)CC2(C)CC1(C(N)=O)C2.C12(CC1)C(C)NC2=O c1(C(N(CC(CC)NC(c2occc2C)=O)C)=O)csc2nnsc12 CC(C)CCC(C(=O)NCC1=CCCOC1)NC(=O)CN1CC2CC2C1 Cc1cnc(C=CC(=O)NCCC(C2CN(C(=O)CC(C)C)CCO2)O)[nH]1 CC(C)(O)C(F)(F)C(=O)NCC(CO)NC(C1COC(=O)C1)=O C(=O)(C(C(C)CC(C)C)N1CC(C(=O)OC)C2(CC2)C1)NCC=C N1(C(C2(C)CC=CCC2)=O)CCCC(CNC(c2ncsc2C2CC2)=O)CC1 Cc1cc(-c2cn(C3CC3)nn2)cnc1C(=O)NC12CCCC1C2 C(C(COC)CC(=O)NCCn1cc(C(=O)NC(c2cnn[nH]2)(C)C)nn1)OC c1(OC)cc(CC#N)cc(NCC2(c3ccc(Br)cc3)CCOC2)c1Br Cc1ccc(C(=O)NCC2CCOC2C(=O)NC(CCO)C(F)(F)F)cc1C CCCC(CC)CC(=O)N1CCC(CC(=O)NCCCc2ccccc2)C1 N1(C(CC(C)OC)=O)CCC2CN(C(c3c(Cl)nc4ccccn34)=O)CC2C1 Cc1c(C(=O)NCC(C2CCC2)NC(=O)CO)c(C(F)(F)F)nn1C C=C1CON(C(=O)C2CCCC(NC(=O)COCC3CC3)CC2)C1 c1(C(=O)NCCCCN(C)C(C2(C)CCCC2O)=O)noc2c1CC(F)(F)CC2 Cc1[nH]nc(Cc2nc(-c3ccccn3)nn2CC2CCOC2)c1Br Cc1ccc2c(c1)ncn2CC(N1CCCN(C(C2CCCC2C)=O)CCC1)=O Cc1nn(C(C)C)cc1C(N1CCOC(CCNC(=O)CCCN(C)C)C1)=O C(C(=O)NNc1cccc2ncccc12)c1c(-c2c(C)nn(C)c2C)cccc1 c1(C(C(C)C)NC2CC(OC)C2)cccnc1.C1C(=O)N1C c1(OC)ccc2[nH]c(C(=O)NCCN(C(C3(C)CCCS3)=O)C3CC3)cc2n1 c1(C(N2C3CN(C(c4c(C)ccc(C)c4)=O)CC32)=O)cc2cc(Br)ccc2s1 C1(CNC(CCc2ncn(C)c2)=O)(CNC(c2[nH]cnc2C#N)=O)CC12CCC2 c1(N(Cc2cc(C)no2)CC2CNCCO2)ncnc2sc(C(C)C)cc12 C=C(Cl)C(C)(C)C(=O)OCC(=O)Nc1ncc(Cl)c(OC(=O)NC)n1 c1(C(=O)NCC2(OCC)CN(C(=O)CCSCC(N)=O)C2)cccc(Cl)c1F C1(C(N(C(CNC(C2(OCC)CCC2)=O)C)C)=O)CCC2CC12 C(=O)(C(C(=O)N1C2CCC1CC(CNC(=O)CCCC(C)C)C2)C(C)C)OCC C1(C(=O)OC)(C(=O)N(CCCNC(C2CC2Cc2ccccc2)=O)C)C=CCC1 CCCC(N=c1[nH]c(N(C)Cc2cc(CC3CC3)on2)nc2c1CCCC2)C(C)C c1(C(=O)NC(CC)CN(C)C(c2cc(OC)cs2)=O)ccc(SC)c([N+](=O)[O-])c1 N1(C(C(CCC)NC(N)=O)=O)CC(NC(c2ccc(OC)nc2F)=O)C2(CC2)C1 c1(C(C)C)ccc(CNc2ccc(NC)cc2)cc1 C1(CNC(C=CC(C)(C)C)=O)CN(C(=O)C2=C(Cl)CCOC2)C2(CCC2)C1 C1(C(=O)NCCN2CCC3CCCCC3C2)CC2CCC(C1)S2(=O)=O CCCCC(CC)C(=O)NC1(CCC(N2CC(C)(O)C2)=O)CCCC1 N1(C2(CC(=O)NC(C)CNC(=O)Cn3cncn3)CC2)CCS(=O)(=O)CC1 C1(CC(=O)OC)CCN(C(=O)Cn2cc(S(=O)(=O)NC)cn2)CC1C1CC1 N1(C(c2c(C)nco2)=O)CCC2CN(C(C3CC3c3ccccc3Cl)=O)CC12 N1(C(Cn2nc(C)c(Cl)c2C)=O)CC(NC(=O)C(O)CN(C)C)CC(C)(C)C1 N1(C(C(C(CC)C)O)=O)CC2CCC1C(CNC(c1cnco1)=O)C2 C1(CNC(CCSc2nc(C)[nH]n2)=O)C2CN(C(c3cncnc3)=O)CC12.C1(CO)CC1 N1(C(C(=Cc2ccco2)C)=O)CCCN(C(=O)CS(=O)(=O)N2CCCC2)C(C)C1 C#CC1CN2CCN1CC1N2CCCC1C.c1(C=O)scc(C)c1C.OC N1(C(C2CC(=C)C2)=O)CC(C2CCCN(C(c3cnc(C4OCCO4)s3)=O)C2)C1 C1(CNC(CC2(C=C)CCC2)=O)CN(C(c2cnn(C)c2CCC)=O)CC1C C(=O)(CC(C)C(C)C)NC1(C)CN(C(C2C(c3cn(C(C)C)nn3)C2)=O)C1 N1(C(C(C)CC(N)=O)=O)CCN(C(C2CCC3CC3CC2)=O)CCC1C Nc1cc(C(=O)NC2CCCC(NC(=O)C=CCN3CCC3)C2)cc(O)c1Cl C1(C(=O)NCC(C)N(C)C(c2ccc(OC(C)(C)C)cn2)=O)CN2CCN1CC2 N1(C(C2C(O)CCN(C(CCSCCCC)=O)C2)=O)CCn2nccc2C1 c1(C(=O)NC(CNC(C(CC)(C)C)=O)CCOC)c[nH]c2cc(F)ccc12 C(C(C)CN=c1cc(NC(=O)OC)nc(C)[nH]1)NC(C(C(C)C)OCC)=O CC1CC(NC(=O)C(N(C)C)N(C)C)CN(C(C2CS(=O)(=O)C2)=O)C1 C1(C(N2C3CC(CN(C(CSC)=O)C3)C2)=O)Cc2cc(C)c(C)cc2O1 c1(OC)c(CC(=O)NCC(C(C)(C)C)NC(=O)CC2C(C)C2(F)F)cccc1F C1(F)(C(=O)Nc2cc(OC)n[nH]2)CCN(C(c2cncc(C(F)(F)F)c2)=O)C1 Cc1csc(CNC(N2CC(N3CCCC3)C2)=O)c1Cl CCCC(C(=O)N1CCN(C(=O)CCCn2cncn2)CC1)N1CCN(C)CC1 Cc1nn(C)c(C)c1CC(C)C(=O)NC1(C)CN(C(c2nn(C)c(CN)c2Cl)=O)C1 N1(C(CN(C)C2CC2)=O)CC(C)(C(N2CC(N3CCNC3=O)C2)=O)CC1(C)C C1(N(C(C(CNC(c2n(CC)ncc2)=O)C)=O)C)COC(C)(C)C1 Cc1nc(NCc2cc(C(C)(C)C)on2)cc(=NC(C)c2cc(Br)n(C)n2)[nH]1 CCC(CC(=O)OC(C)C(=O)C1CCCC1)C(=O)O c1(CCOCC(N2CC(NC(C(COC)(C)C)=O)(CO)C2)=O)cccc(C#N)c1 c1(SCC(N2CC(CNC(CSCCC)=O)OCC2)=O)ccsc1[N+](=O)[O-] c1(COCC(=O)NCCOC2CN(C(c3ccc(CC)[nH]3)=O)C2)ccccc1C N1(C(C(=O)NC2CC2)=O)CC2(C1)CN(C(c1n[nH]cc1Cl)=O)CC2CO C1(NC(C2CC(C)(O)C2)=O)CN(C(c2cccc(N)n2)=O)CCC1CO C(N=c1[nH]c2c(c(=NCCC3(CO)CC3)[nH]1)CCCC2)C1CCC(C(O)=O)O1 C1(NC(Cc2c(C)scc2)=O)CC2(CCC(NC(C3CC3Cl)=O)CC2)C1 Cc1cc(F)ccc1C1CCC(C(N2CCC(n3cnnc3N)CC2)=O)N1 N1(C(C2(C#C)CCC2)=O)CCCC(O)(CC23CC(C(=O)NOCC4CC4)(C2)C3)C1 C1(C(C#C)C)CCN(C(C2CC2C(C)NC(=O)CN(C)CC)=O)CC1 c1(C(N2CCN(C)CC2CNC(C2CCCO2)=O)=O)cc2cncn2c(O)n1 C1(NC(C(CCCC)O)=O)C2CC3CN(C(=O)CN4CC(=O)NC4=O)C1C3C2 C1(CNC(c2c(C)[nH]c(C(C)(C)C)c2)=O)CCC2(CN(C(C3C(C)C3C)=O)C2)O1 C(=O)(C1CCCc2sccc21)NCC1(C)COCCN(C(=O)C#CC2CCC2)C1 N1(C(c2cc(OCC)ncc2)=O)CCN(C(C2CC(C)C2)=O)C(CN(C)C)C1 N1(C(CNC2CC(NC(=O)CC3C=CCC3)C2)=O)CCOCC(O)C1 c1(C(N2CCC(O)C2)C(=O)NCCCC2CC2)cnc(C(F)(F)F)cc1Cl C12(C(N3CCC(NC(c4ccc(OC)nc4)=O)C3)=O)CC3CC(C(=O)N1)C2C3 c1(C(=O)NC(CCNC(C(C=C)O)=O)C)ccncc1C(F)F N1(C(CCCC=C)=O)CCC(C(F)(F)F)C(NC(c2cncc(O)c2)=O)C1 C1(C(=O)NS(CCOC(C)C)(=O)=O)CCC2(CCN(C(c3ccno3)=O)CC2)C1 c1(CNC(C(C2CCCO2)NC(C=CCN(CC)CC)=O)=O)cc(C)cc(C)c1 c1(CCCNC(=O)C(N2CCCC2CC2CCOC2)=O)ncc(Br)cn1 c1(NC(=O)CCc2cncs2)ccc2c(c1)Cc1ccccc1-2 N1(CC(N2CCC3CN(C(c4cncc(Cl)c4)=O)C3C2)=O)Cc2ccccc2C1 N1(C(C2N(C(C(C)SC(C)C)=O)CC3(CC3)C2)=O)CC2CSCC(C2)C1 C(=O)(C(C)C(CC)CC)NC1CC(C(N(CC)Cc2cnn(C)c2)=O)C12CCC2 C1(NC(COCCCC)=O)CC12CCC(NC(c1n[nH]c(C3CC3)c1C)=O)CC2 c1(COC)ccc(C(=O)NC2CCC2NC(c2cc(C3(C)CC3)n[nH]2)=O)[nH]1 c1(C(N2CC(NC(CC(C)F)=O)C(S(C)(=O)=O)C2)=O)ccc2c(c1)NC(=O)C2 N1(C(C(CC)Cc2ccccc2C)=O)CC(NC(=O)C(C)C2CC2)CC(C)(C)C1 C12(NC(c3c(OC)cccc3)=O)CCCC1N(C(C1CC3CC3C1)=O)CCC2 N1(CCNC(C(CCC)OCC)=O)CCC(N=c2[nH]c3cc(C)ccc3o2)CC1 c1(C(N2CCC(N(C(C3CC3c3cncs3)=O)CC)C2)=O)ccc2c(c1)CCC=C2 c1(N(C(C)C)C)c(Cn2cc(C3(C4CC4)CC3)nn2)nn2c1CCC2 N1(C(C)C)CC(CNC(=O)CC2CCCCN2C(=O)C=Cc2cscn2)C(C)C1 Cc1cc(F)c(C(=O)NC2CC2C(=O)Nc2cc3c[nH]nc3cc2F)cc1Br c1(N2CCC(O)(CNC(c3cc(C)[nH]c3)=O)CC2)nc2c(cc1C#N)CCCC2 CC(CC(=O)NCC(O)CNC(C1(O)COC1)=O)C(F)(F)F c1(C2(CC)CCC2)cn(C2CN(C(c3cc(C(=O)O)no3)=O)C2)nn1 C(C(=O)N1CCC(CCCNC(C2CCN2C2CCCC2)=O)CC1)(C(C)C)OC CCCC(C#N)C(=O)N1CCN(C(C)C(=O)NCC(C2CCCCC2)O)CC1 C1(C(=O)NCCN(CCOC)C(c2ccc(C(=O)CSC)s2)=O)CCCCS1.C(C)C Cn1cc(C(N2CCC(F)(C(=O)NC3CC(N4CCCC4)C3)C2)=O)c(C(F)F)n1 c1(OC)ccccc1CN(C1CCCN(C(C2(C)CC2C)=O)C1)C(c1ccco1)=O N1(C(CC(C)c2ccco2)=O)CCCC(C2CN(C(C3OCCCO3)=O)C2)C1 N1(C(CC(CC(C)C)C)=O)CCOC2(CCN(C(=O)C(C)(C)CO)C2)C1 c1(C(=O)NC2C(CC)CN(C(c3cscc3F)=O)CC2)cc(F)cc2nc[nH]c12 C1(C(N2CC(COC)OCC2)=O)CC2(CCC2)CN1C(=O)C1=C(C)OCCC1 C1(NC(c2ccc(CNC(COCCOCC)=O)o2)=O)CCCC2(CCC2)C1 c1(CSCCNC(=O)CC2CCCC2)c[nH]c2ccccc12 N1(C(C(CC=C)(C)C)=O)CC2CCCC(C1)N2C(c1c(C)cc(C)nc1C)=O C1(COC)CN(C(C2CCC2c2nc[nH]n2)=O)CCN1C(c1cccc(O)n1)=O C12(NC(C(C)N(CC)CC)=O)CCC(CC1)N(C(C1C(C)C1C)=O)C2 C1(C(=O)N(CC2CCN(C(=O)COC3CC3)C2)CC2CC2)C2CCN1CC2 S(=O)(=O)(c1ccc(Cl)s1)N1CCN(c2nc(SC)nc(C(F)(F)F)c2)CC1 c1(C(=O)NCCN(C(COC(CC)C)=O)C)ccnc2c1nnn2C N(C(=NCCC(C)C)N1CCCC2(C1)CC2(F)F)C(N(C)Cc1ccc(C)cc1)=O N1(C(N2CCCCC(CNC(=O)CC3CCCOC3)C2)=O)Cc2ccccc2C1 C1(C(=O)NC(COC)C(=O)Nc2cnc(O)c(F)c2)CNC(=O)CC1C C1(CC)CCCC1CNC(c1ccn(CCNC(C2CC(OC)C2)=O)c1)=O C1(CNC(C2CCO2)=O)COCCN(C(c2cc[n+]([O-])cc2)=O)C1 c1(CNC(C2(CCNC(C(n3cc(Cl)cn3)C)=O)CC2)=O)ccc(O)c(F)c1 c1(CNC2CC(F)CN(Cc3c(OC)ccc(O)c3)C2)cc(C#N)ccc1F C1(=CC(=O)NCC2CC(NC(C3(SCC)CC3)=O)C2)CC2CCC(C1)N2C C1(NC(CC(CCC)(C)C)=O)CCC2(CCN(C(c3csnc3C)=O)C2)C1 c1(C(=O)NCCC2CCCN(C(C(C(C)C)O)=O)C2)ccc2nc(O)sc2c1 CC1(C)C(C(N2CCCC2CCNC(C2CC23CC3)=O)=O)CCS1(=O)=O Cc1cc(Cl)ccc1OC(C)C(=O)NC1CC(C)(NC(=O)CC2COC(=O)C2)C1 C12Cn3c(C)nnc3CN1C2=O.C1(SCC#C)COCCN1C(=O)OC(C)(C)C C1(CNC(C2CN(C(CCC(=O)NCCC)=O)C2)=O)CC12CCCCC2 N1(C(C(C)OCCCC)=O)CC(C)CN(C(c2cc(N)c(F)cc2F)=O)C(C)C1 C1(NC(CCOC)=O)CC2CN(C(c3cnc4cc(C)ccn34)=O)CCN2C1=O c1(C(=O)NC2C(CNC(C(C)NC(CC)=O)=O)CC2)cc2cc(F)ccc2[nH]1 c1(C(=O)NC2CCN(C(c3ccco3)=O)CC2O)nc2ncccn2n1 CC1CN(C(=O)CN(CC(C)N(C)C)C)CC1(C)CNC(=O)C1CC1 C12(C(N3CCC(C(C)NC(=O)CSc4ccccc4)C3)=O)CCC(CF)(C1)OC2 N1(C(CC2C(C)=NNC2=O)=O)Cc2[nH]nc(C(=O)N(c3ccc(F)cc3)C)c2C1 c1(C(=O)NCC(C(=O)NCc2cc(C)nc(O)c2)N(C)C)cccc(C#N)c1C C1(C(N2CCC(CNC(c3cnc(CC)s3)=O)CC2)=O)CCC2(CC1)OCCO2 Cc1noc2ncc(C(N3CC4=C(C3)CN(C(C3(C#N)CC3C)=O)C4)=O)cc12 C#Cc1cccc(C(=O)NC2CN(C(c3ccoc3CCC)=O)CC2C)c1F Cn1nc(C(N2CCC3(NC(=O)Cc4cnc[nH]4)CCCC23)=O)c2c1CCSC2 c1(NC(C2CCCC(NC(c3c(F)cncc3F)=O)C2)=O)cncc(F)c1I C(=O)(C1=CNC2=NCCC2=C1)N1C(CNC(CC2CC(C)C2)=O)CC2COCC21 O=S(=O)(Cc1cscn1)N(CCC1CC1)CC1CCOC1 C1(C(N2CCC(NC(=O)CN3CCS(=O)CC3)C2)=O)CN2CCCC2CO1 n1(CC)ccc(C(N2CCCCC(NC(C3CCOC(=O)N3)=O)C2)=O)cc1=O Cc1cc(C(=O)NC2CC(CC(=O)NC(C)Cc3ccc(C)o3)C2)ncn1 CC1(CNC(=O)CNC(c2cscn2)=O)CCN(C(C23CCCCC2C3)=O)C1 C1(CC(=O)NCCC(C)CO)C2CCC1CN(C(c1onc3ccccc13)=O)C2 c1(CC(C(=O)NC2CN(C(C(C)(C)OC)=O)CC2O)O)ccc(OC)cc1 N1(C(Cn2c(C)nnc2C2CC2)=O)CC2CC(C1)C2O c1(OC)ccc(CNC(=O)NC(C)C(O)C(=O)OC(C)(C)C)c(F)c1 c1(CC(=O)N(C)CC2CN(C(=O)CNC=O)CCO2)ccc(S(=O)C2CC2)cc1 CCC(C)CCC(=O)NC(C)CCCCNC(c1cccc(CC#N)c1)=O C1(O)(C(C)(C)C(=O)NCC2CCN2C(c2ccc(F)o2)=O)CCCCC1 N1(c2snc(C)n2)CC2(CC2)CC1CNC(=O)CCc1cccnc1 C1(NC(C2CC=CC(NC(C(CC)(C)COC)=O)C2)=O)CCc2nncn2C1 CCCCCC(C)(C)C(=O)NC1CCCC1NC(c1oc(C(F)(F)F)nc1C)=O Cc1nc(-c2ccco2)cc(C(=O)N(C2CC(NC(C3CCCS3)=O)C2)C)n1 C1(NC(c2c(N)nccc2)=O)CC(NC(C23CC(CO)(C2)C3)=O)C12CCC2 C(=O)(CS(=O)CCC(F)(F)F)N1C2C(CNC(CN(C)C)=O)C(C2)C1 C1(Cl)(C(=O)OC(c2ccc(C)c(Br)c2)C)C2CCCC(=O)C12 c1(C(N2CC(CN(C)C(C3CC(C)(C)C3)=O)C2)=O)c[nH]c(=O)c(C(N)=O)c1 c1(CC(=O)N(CCCN(C)C(C2CC3CC3C2)=O)C)ccc(C#N)cc1F C1(CC(=O)N(CC(C)(C)NC(c2cnccn2)=O)C)CC2CCC1O2 CC(C)CCCCC(=O)NCCC1CN(C(c2scnc2C(C)C)=O)CCO1 c1(C(c2nnnn2C2CC2)NCCF)cc2ccccc2o1 Cc1occc1C1CC1C(=O)NCC(CCC1CC1)n1cccn1 N1(C(C2OCCN(C(CC(C)C3CC3)=O)C2)=O)CC2(CCC2O)C1 N1(C(Cc2c(SC)cccc2)=O)CCCC2(NC(=O)CC(C)(C)C)CC2C1 C1(C(=O)NC2CN(C(CCCOC(C)=O)=O)C(C)(C)C2)CCn2c(O)nnc2C1 c1(OC)ccc(C(N2CCCC2CN(C)C(c2conc2C(C)C)=O)=O)cc1O N1(C(c2ccc(C(F)(F)F)cc2)C(=O)NC(C(=O)OC)C)CCC(O)CC(C)C1 C12(NC(c3cc(OC)ncc3Cl)=O)CCOCC1CN(C(=O)C1=CCCC1)C2 CC1C(NC(=O)CCCCN2CCCC2)CCCN1C(=O)CSC(=N)N C1(C(N(C)Cc2cc(C)n(C)n2)=O)CCCN(C(c2csc(F)c2)=O)C1C Cc1ccccc1C1(C(=O)N(C)CC2CN(C(c3ccc(=O)oc3)=O)C2)CC1 c1(CC)conc1C(N1CCC(C(=O)N(C(C)C(N)=O)C)C1)=O C(=O)(CCCS(C)(=O)=O)NCC(CNC(C1CCN(C)S1(=O)=O)=O)O c1(C(N2CCC(N(C(c3n(OC)cnc3C)=O)C)C2)=O)cc(C)sc1S(N)(=O)=O C12(NC(CSCC)=O)CC(CO)(C1)OC21CN(C(=O)C2=CCSC2)C1 c12ccc3c(c1)N(CC(C)(C)O3)N(CCN(CC)CC(C)F)C2C(=O)NCCC C1(C(N2CCC(N(C(c3cnc[nH]3)=O)CC)C2)=O)CCCCC12CCC2 O=C1CC(N2CCCC2)CN1.c1(-c2scc(C)n2)ccccc1Br c12cc(c[nH]1)S(=O)(=O)NC2=O.c1(OC)ccc(I)c(CN=c2[nH]nc(CO)o2)c1 S(=O)(=O)(c1ccc(Cl)c(Cl)c1)N1CC(CNC(c2cc(Cl)nc3n[nH]cc23)=O)C1 C1(CNC(C2(CC(=O)OC)CC2)=O)CCC(NC(=O)CCCc2cnn[nH]2)CC1 N1(C(=O)NC2CC(OC(C)(C)C)C2)CC(CNC(C2(O)CC(F)(F)C2)=O)C(O)C1 CC(C)(C#N)CCC(=O)N1CCC(C)(NC(c2csc3c2CCCC3)=O)C1 c1(C(=O)NC(CCNC(C=Cc2cnc(C)s2)=O)C)c(C)ncn(C)c1=O c1(CCC(=O)NCC2CCN(C(C(CC#C)(C)C)=O)CC2)n[nH]c2c1CCCC2 c1(C(=O)NC2C(C)CCN(C(=O)CC3CC4(CC4)CO3)C2)ncc([N+](=O)[O-])n1C N1(C(c2n(C)c(S)nc2)=O)CCC2CC1CN2C(=O)Cc1ccc(C#N)cc1F C(N=c1[nH]c(C)nc(Cl)c1Br)c1cc(OC)nc(C)c1 CCC(CC)C(F)C(=O)N(CCCOCCN(C)C(C1(COC)CCCO1)=O)C C12NC(=S)N(c3ccccc3)C(C(C)(C)C)=C1C2=O.C#Cc1ccc(OC)c(CC)c1 c1(OC)c(CC(=O)NCCCCNC(=O)CCS(C)(=O)=O)cccc1C#N c1(C(C(=O)NCc2ccc(F)cc2)N(C)Cc2cn(C)nn2)cc(Cl)cc(Br)c1 c1(C(N2CCC(F)(C(=O)Nc3c(OC)nccn3)C2)=O)cc2c(cn1)OCCC2 c1(C(N2C3C(NC(CC(=O)NCC)=O)CC(C3)C2)=O)ccc(S(=O)C(C)C)cc1 C1(CC(=O)NCCNC(c2cc(-n3ccnc3)cs2)=O)CC2CCC1O2 N1(N(c2cc([N+](=O)[O-])ccc2Oc2ccccc2)C)CCC2(CCCCC2)CC1 n1(CC(=O)N(C23CCCC2CN(C(=O)C(C)(C)C)C3)C)ccc2c(N)cccc12 c1(OC)cc(C(C)C(=O)NC23CC(NC(=O)CC4(C)CCOC4)(C2)C3)ccc1O c1(NC(=O)NCCOCCOCC#C)ccc(Br)cc1Br c1(C(C(F)(F)F)OC(Cc2cc(C)n(C3CC3)c2C)=O)cn(C)c2ccccc12 C1(C(C)C)N(C(C2CC(C3CC3)=NO2)=O)CC12CCN(C(=O)CO)CC2 CC1C2CCC(C2)C1C(=O)O.C1CCCCC(=O)N2CCC(C2)C(=O)N1C C(=O)(C(C)(C)C(C)(C)O)N1CCCC(NC(C(C)(C)CC2CC2)=O)CC1 Cc1cc(O)ncc1C(=O)NCC1(O)CCCN(C(=O)CN2CC=CC2)C1 CC1CCN(CC(N2CC3CC3(NC(c3cc(Br)cn3C(C)C)=O)C2)=O)CC1 c1(C(C)C)ncc(Br)c(=NC2CC(C(N3CCCCC3C#N)=O)C2)[nH]1 c1(C(=O)NCC(c2ccccc2)NC(CC2C(C)(C)C2)=O)nncn1C1CC1 c1(COCC)nnc(-c2nc(C3CN(CC(C)C)CCO3)n[nH]2)n1CCN(C)C C1(NC(C2C(C)(C)C2(F)F)=O)CC(CNC(=O)Cn2cc(C(F)F)cn2)C1(C)C Cc1c(C(=O)Nc2ncc(-c3ccncc3)cc2C(F)(F)F)cccc1I Cc1nnc(CC(C)C(N2CCC(F)(CF)C2)=O)n1C S(=O)(=O)(c1ccc(CC(=O)NCCCN(C(=O)CC2CCC(=O)N2)C)s1)NC CC#CCC(C(=O)N1CCC(N2CC(O)C2)C1)NC(C1CCN(C(C)C)CC1)=O c1(OC(CCC2C(N(C(=O)Cn3cccn3)CC)C2)=O)cc(F)cs1 c1(C(N2CCC(NC(c3c(C)cc(F)cc3)=O)(CF)C2)=O)n[nH]c2c1COCC2 N(S(=O)(=O)N(C)C)CC(=O)NCC(C)N(C)C(c1c(C(F)(F)F)cnn1C)=O C1(C(=O)NCC2CCC(NC(C(C)(C)F)=O)CC2)CCn2c(O)nnc2C1 C1(C(=O)NC2(CC=C)CCN(C(=O)CC(F)F)CC2)CCc2nn(C)cc2C1 N1(C(C)=O)CCC(C)(C(=O)NCC#CCNC(c2cc[nH]n2)=O)C1 CC(C)C(CC(=O)NCCC(C)N(C)C(c1cnc(S(C)(=O)=O)s1)=O)C(C)C Cc1[nH]c(C#N)cc1C(N1CCC1CNC(=O)CCc1ccc(N(C)C)cc1)=O c1(C(=O)OC)cocc1C(N)=O.C(C(C)(O)CN)NC(=O)C=CC(C)(C)C N1(C(C2CCCCN(C(C(C)(C)SC)=O)C2)=O)CC2(C)CC1CCO2 N1(C(C2(C)CCOC2)=O)CCCCC(C(=O)NCc2nccs2)C1 C1(NC(C(COC)C)=O)CC2CCC1N2C(c1ccc(N(C)C)cc1)=O C(CC(=O)NCC1CC12CC2)(C(F)(F)F)NC(c1ccc(C#C)cc1)=O N1(C(CC(C)c2ccco2)=O)CCC=C(C(=O)NCC2CC2C2CCC2)C1 C(CCCCC(=O)NCC(C)C(F)C(=O)Nc1ccc(F)cc1)=CC Cc1ccnc(C(=O)NC(CO)C(C)NC(C2CC23CCOCC3)=O)c1F C1(C2CCN(C(c3c(CC)ccs3)=O)CC2)N(Cc2nncs2)CC12CCC2 C1(CCOC)(NC(C(C)OCC=C)=O)CCCN(C(=O)CNC(=O)CN(C)C)C1 N1(C(CC(C)N(C(=O)C(c2ccnn2C)O)C)=O)CCOCC(O)C1 C#Cc1ccc(C(=O)NC(C)C(C)NC(c2c[nH]c3ccncc23)=O)c(F)c1Cl Cc1cc(S(=O)(=O)N2CCS(=O)(=O)CC2C(=O)N(C)C)ccc1Cl Cc1ccc(CC(N2CCOC(C(=O)NCc3sc(C)nc3C)C2)=O)cc1 C=CCC(CC=C)n1cc(C2CCCCN2)nn1 C(CCCCCNC(C1C(C#N)C1(C)C)=O)N(C(=O)CCSc1ccccc1Cl)C Cc1csc(CC(=O)NC2CCC(CNC(c3n[nH]cc3F)=O)C2)c1 n1(CC)cnnc1-c1cn(CC(F)CCNC(c2ccn(CCF)n2)=O)nn1 Cc1cnc(C(=O)NCC(CNC(C2(C)CNC(=O)C2)=O)CO)cn1 Cc1ccc(-c2cn(CC3CN(C(C4CC4(Br)Br)=O)C3)nn2)s1 C1(CNC(=O)CC2CSCCS2)C2CCCC1N(C(C1CC13CC3)=O)C2 C=C(C)C1OCCC1CNC(=O)CC1(C)CCN(C(C2(O)CCCCC2)=O)C1 c1(C(N2C(CNC(COC)=O)C(C)(C)CCC2)=O)ccnc2cc(OC)ccc12 c1(C2(NC(N3CCCC3)=O)CCC2)ccc(NCc2ncccn2)cc1 c1(NC(C(CC(F)F)NC(C(CCC)OCC)=O)=O)cc(C#N)ccc1C c1(C(NOC(CC(=O)OC)CNC(=O)Cc2ccccc2)=O)cccc(C)c1C N1(C(=O)NCc2cnn(C=C)c2C)CCc2cc(F)cc(Cl)c2C1 C1(C(=O)NC2(CSC)CC(O)C2)CCC(NC(C2C3CC4C(C3)C24)=O)CC1.CCF C1(NCC(CC)C(=O)O)CCC2CCCCC2C1 c1(C(=O)NC23C(CN(C(C4(CCOC)CC4)=O)C2)C3)cccc2c(C)[nH]nc12 c1(NC(C(=O)N(C)CC2CC2)=O)ccc(NC2CCNC2=O)nc1 N1(C(c2ncccc2CC)=O)CCC2(CC1)CN(C(=O)CC1(N(C)C)COC1)C2 FC1(F)C2CC(N=c3[nH]c(=NCCc4ccccc4)[nH]c4c3CCC4)CCC12 n1(C(CC)C)nc(C2CC2)nc1-c1cc(Cl)n(C)n1 O=NN1CCCCC1C(=O)NCCC(O)CNC(C1CC(F)(F)C1)=O CCC(C(=O)NCC(C)NC(c1cn(-c2cccnc2)nn1)=O)N1CCCC1=O N1(C(C2(CC)CCOC2)=O)CCCC(CCNC(c2ccc(COC)o2)=O)CC1 CCCCC(O)C(C)C(=O)N1CCC2(C)NCC2C1.c1nncn1C c1(CC)ncccc1C(=O)NC1CCC(NC(c2cc(C)n(CC)n2)=O)C1 CC1(CC(=O)NCC(CO)NC(c2ccccc2)=O)CC1(F)F c1(CNC(C2C3CC3CN2C(c2ccsc2Cl)=O)=O)ccnc(F)c1 C(=O)(C(F)(F)CCn1cc(CCO)nn1)NC(C)CCN(C)C S(=O)(=O)(c1ccc(C#N)c(NC(c2n[nH]c(=N)s2)CO)c1)N1CCC(C)(C)C1 C(=O)(C1=NN(C)C(=O)CC1)NC(C(C)NC(c1ccc2nc(O)oc2c1)=O)(C)C CC(C)(CC(F)C(=O)Nc1ncccc1Br)c1nn[nH]n1 c1(C(=O)OC)ccnc(N2CC3(CN(C(C4(O)CCOC4)=O)C3)C2)c1[N+](=O)[O-] C1(CNC(c2ccnc(OC)n2)=O)CC12CCN(C(=O)Cc1ncc(Cl)s1)CC2 C=CCCCC(C(=O)NCc1ccc(Cl)nc1)NC(C1CCOC1C=C)=O c1(C(=O)NC(C2CCCN2C(=O)C(F)F)C)ccc(F)c(C(F)F)n1 c1(C(=O)NCCN(C(C(C=C=C)C)=O)CC(C)O)n[nH]c(CCC)c1[N+](=O)[O-] C1(CNC(Cc2cc(C)sc2)=O)CCC(C)(C)CN1C(C1CCC(C)(C)CC1)=O CC(CCC(=O)N1CC2(CC2)C1)NC(=O)CC1CCCN(C)C1 C(C(C(=O)N1CC2CCC(C1)C2O)C(C)(C)C)NC(Cc1c(C)occ1)=O C1(O)(CCNC(C(C)c2ccco2)=O)CCN(C(c2cnc(C(F)F)nc2)=O)C1 C1(NC(C2CCN(C(C)=O)C2)=O)CCN(C(c2sccc2Cl)=O)C1(C)C C1(C(N(CC(C)NC(c2ccc(C#C)o2)=O)C)=O)CN(C)C(=O)CCO1 C1(CC(=O)NCC(CNC(c2c(C)n(C)cc2)=O)(C)C)CC(F)(F)C1(F)F c1(C(=O)NCc2ccc(-c3cc(C)c(F)cc3Cl)cn2)c(Cl)cc(Br)c(Cl)c1Br C1(C(=O)NC(CNC(C2CN(C(C)C)C(=O)CC2)=O)C)CCCCC1P(C)(C)=O N1(C(C(C)Oc2cccc(C)c2)=O)CC2(C)CN(C(C3CC3(F)Cl)=O)CC2(C)C1 N1(CCNC(C(C2CCCCC2)OC)=O)CCN(C(=O)Cn2ccc(C)n2)CC1 Cc1cc(=O)n(CC2CCC(=O)N2C)c(O)c1CN1CCOCC1C#N C(N=c1nc2ncn(C)c2c(NCC(C2CCS(=O)(=O)C2)=O)[nH]1)c1nnn(C)n1 Cc1ccc(O)c(CC(=O)NCC2CCC2NC(=O)C2CC2)c1 N1(C(C)=O)CCC(C(=O)NCC(CO)NC(c2ccc(CN(C)C)o2)=O)C1 C(=O)(C1=NOC(C2(O)COC2)C1)NC1CC(NC(Cn2c(C)cnc2)=O)CC1O C#Cc1cnn(CC(=O)NC(C)CN(C)C(C2(C)CCCCC2)=O)c1 c1(OC)ccc(C(N2CCC(F)(C(=O)Nc3cc(C#N)nn3C)C2)=O)c(F)c1 CC(C)CCC(C)NC(C1CCCC(NC(=O)C=CC2CCCN2C)C1)=O c1(C(C(=O)NC2CCOC2)N(CCN=[N+]=[N-])C)cn(C)nn1 C12(CNC(Cc3scc(C)c3)=O)CCC(CN(C(c3c(C)cnn3C)=O)C1)C2 CC(CC(F)(F)F)N(C)C(C1COCCC1NC(c1cc(Cl)cn1C)=O)=O Cc1ccc(C(C)C(=O)N(C)CC2(NC(c3ccncc3)=O)CC2)o1 C(=O)(C(Cc1ccco1)NC(C1CC=CC1)=O)NCC(C)CF N1(C(C(C(CC)C)N)=O)CCC(C2CN(C(C3CC4C=CC3C4)=O)C2)CC1 c1(N(C)Cc2cn(C)nn2)nc(=NCC2(C)CCCS2)[nH]c2c1SCC2 C(=O)(CC(F)(F)C(F)(F)F)N1CC2CC(CNC(C(C(CC)(C)C)OC)=O)C2C1 N#CC1CC12CCN(CC1CCC(c3nc(C(N)=O)no3)O1)CC2 C=CCC(CC=C)C(=O)NC(C)(C)C(C)NC(=O)C(=O)Nc1cccc(C)c1 C(CCCC(=O)NC(C)CNC(c1cccc(CCN(C)CCN)c1)=O)OCC Cc1nc(F)ccc1-c1cn(CCN(C(=O)CC2CC(N(C)C)C2)C)nn1 C(C)(C)(C(C)CC(=O)NC(c1ccnn1CC)C)NC(C1C(OCC)C1)=O.C(C)(=O)O CCCC(C(=O)NC1(CF)CCN(C(=O)CCCc2ncc(C)o2)C1)C(C)C C1(O)(CNC(C2C(=C)C2)=O)CC(CNC(=O)C(F)=CC2CC2)C1 CCC(F)(F)CC(=O)N1CCC(C)C(NC(c2cnc(C(C)OC)s2)=O)C1 CC(CCCCNC(=O)Cc1cnsc1)NC(=O)Cc1nn(C)cc1Br C(C(C(=O)NCC1(O)CCCC1)C(C)(C)C)NC(C1(C(C)=O)CC1)=O Cc1c(NC(c2ccc(C(=O)C(F)(F)F)s2)=O)cc(C(F)(F)F)cc1F c1(N(C(C2CCCN(C(C3CCCOC3)CC)C2)=O)C)nccc(C)c1[N+](=O)[O-] c1(NCCC(=O)NC)cc(NC2CC3CC3C2)nc(C)n1 c1(SC)nn(C)cc1C(=O)NCC(C(C)C)NC(c1occc1C)=O c1(C2C(=O)N2)nnnn1C1CCOCC1.n12ccnc1C2(CC)N(C)C.SC.OC CC1(C)CCCC(N2CC(OCC(=O)NCCO)C2)C1 c1(CC(=O)NC2CC(C)(NC(C3CC=CC3)=O)C2)noc2ccccc12 C1(NC(COC2(C#C)CCC2)=O)C2CC3COC1C3C2 C1(C(=O)NCCC(C(C)C)NC(C2(CO)CCCO2)=O)CCCN2CCCCC12 N1(C(c2[nH]cc(CC)c2)=O)CC(NC(C2=CN=C(O)CC2)=O)C(C)C1 C=CC(C)CC(=O)N1CCCC(CC(N2CCN(C(=O)C=CBr)CC2)=O)C1 C(=O)(CCCC(F)F)NCC(CC=C)NC(c1cncc(OCC(F)F)c1)=O N1(C(C2CN(C(C)C)C2)=O)CC=C(C(=O)N2CC3(CCCO3)C2)C1 N1(CC(COC(COC)C)O)CC(NC(c2c(Cl)n[nH]c2C)=O)CCC1C C(=O)(C(C)(C)C(F)(F)F)N1C2CC(CNC(C=Cc3ccc(C)o3)=O)C1CC2 C(=O)(C1CCCc2n[nH]cc21)NC1C=CCN(C(c2n(CC)ccn2)=O)C1 N1(C(CC(C(C)OC)NC(=O)C#CC(C)(C)C)=O)CCc2ncn(C)c2C1 N1(C(CCC(=O)NCC)=O)CCN(C(C2COCC2C(=O)OC)=O)C(C(C)C)C1 C=CCC(C)(C)CC(=O)N1CCC(C(=O)NC(C)CCCC(C)C)C12CC2 N1(C(c2cnc(NC(C)=O)s2)=O)CCCC(O)(CN(C(=O)CC(C)(F)F)C)C1 N1(Cc2cnc(OC)nc2)CCC(=O)N(CC2COC3(CCC3)C2)C1=O c1(C(=O)NC2C(C)(C)N(C(C3CC3C3CC3)=O)CC2)nccc2ccncc12 c1(C(=O)NCC2C(NC(COCCOCC)=O)COC2)ccc(C)c(OC)c1 C1(C(=O)NC(CCCCNC(C(CC)(F)F)=O)C)CCN(C)C(=O)C1 N1(C(C(CSC)(C)C)=O)CCC2CN(C(=O)CCCC(C)C)C2C1 C1(NC(=NCC)NCCc2ccc(C(F)F)cc2)CCc2nnc(OCC)n2C1 c1(COC(C)C)ccccc1NC(=O)NCCC1CCOC(C)C1 C1(NC(C=CCN(C(Cc2ncc(CC)[nH]2)=O)C)=O)CC2CCC1O2 n1(CC(=O)NCC2N(C(CC(C(C)C)C)=O)CC2)c(O)nc2ccccc2c1=O C(CS(=O)(=O)c1cccc(Br)c1)NC(c1ccc2cnn(C)c2c1)=O c1(C(N2CC3C(CNC(Cc4c(C)noc4Cl)=O)C3C2)=O)ccc(O)c(F)c1 c1(C(=O)NC2CC(C)(NC(CSc3ccc(OC)cc3)=O)C2)ccc(N)c(N)n1 c1(NC(=O)C(N2CC3(CCCC3)C2)=O)ccc2ccnn2c1 C1(C(=O)NCC2CC(NC(CC(C)N(C)C)=O)C(O)C2)CC2(CCO1)CC2 Cc1cc(-n2cc(CSCCNC(C3CCC(C#N)CC3)=O)nn2)cc(C)n1 N1(C(C)C)CC(C(N2CCC(NC(=O)Cc3cnnn3C)C2)=O)CC1=O Cc1cc(S(N)(=O)=O)sc1C(=O)NC(CC(=O)O)C(=O)O C(N=C(NC1CCC1)N1CCCC(S(C)(=O)=O)C1)c1cc(C)oc1C N1(C(C(c2cccc(C)n2)(F)F)=O)C2CCC1C(CNC(C1CC3CC3C1)=O)C2 C1(C(=O)NC(COC)C(=O)NC(c2n[nH]c(C)n2)C)CC12CCOCC2 C1(NC(c2cc(CCCCC)[nH]n2)=O)CC2CN(C(c3cscc3Cl)=O)CC2C1 c1(CCC)onc(C)c1C(=O)NC1CC1CNC(C1(C)CC2CC2C1)=O C1(C(=O)OC)(C(F)F)CCC(NC(=NCc2conc2C(C)C)NC2CC2)CC1 O=C(CS(=O)(=O)C1CC1)NCC12CC1CN(C(=O)CCOC1CCOCC1)C2 N1(C(CC2(C)CCCO2)=O)CCC2CCN(C(=O)C=CI)CC2C1 N1(CCCl)CCCC1C(=O)O.C1(SCC(=O)NC)COCC1n1cc(C(=O)OC)nn1 c1(-c2cc(C(=O)NCCCN(C(C3(CC)CCC3)=O)C)on2)cccc(F)c1 C1(C(=O)NC(C(C)C)C)(NC(=O)CCN(C)C)CCOCC1 C(=O)(C1CCCc2n[nH]cc21)NC1(CCOC)CCN(c2nccnc2F)C1 c1(N(C)C)ncc(NC(C2(C)CCCN2C(C2CNC(=O)C2)=O)=O)cc1Br c1(NC(C2CC3CC3N2C(=O)CN2CCOC2=O)=O)ccc(F)cc1Br CC(CC(=O)NCCNC(C1CCC(n2ccnn2)CC1)=O)C(C)(C)C N1(C(C)C)CC(C(N2CCN(CC(C)O)C(CC3CC3)C2)=O)CCC1=O c1(C(=O)NCC2N(C(C(C3CC3)OC)=O)CC2)ccc(N)c(CC(C)C)c1 c1(C(C)=O)c(C)[nH]c(CC(=O)N(CCCNC(=O)CSc2n[nH]c(O)n2)CC)c1C CCCS(=O)(=O)C(C)C(=O)NCCCNC(=O)Cc1noc2ccc(O)cc12 C(CC(C)(C)CC(=O)NCC1(NC(c2nc(Cl)c(Cl)s2)=O)CCOC1)OC C(CC(=O)N1C2CCCC1COC2)(C(F)(F)F)N(C1CCOCC1)C C(CC)(C(=O)N1CC(O)(CO)C1)=CC.C(=O)(CC(C)C)N(C(=O)CN)C C1(C(N(C(C=C)C)C)=O)CCN(C(C2(CF)CC(=O)C2)=O)CC1(C)C C(=O)(C1=C(Cl)CCC1)N(CCCNC(c1cnc2n1CCS2)=O)CCO c1(C(=O)NCC(=O)NCC(=O)N(CC(F)Cl)C)ccccn1 C(C)(CO)(C(=O)NCC12CC(NC(=O)CC3SC(=N)NC3=O)(C1)C2)OC C1(C(=O)NC(c2ncc[nH]2)(C)C)CCN(C(=O)C2C3CC(=O)CC23)O1 C=C(C)CC(C(=O)N1CCNC(=O)C1C)NC(=O)CCC(C)OC N1(C(C2CC2c2ccccc2F)=O)CCC(=C(F)F)CC1 Cc1cc(C)c(C(N2CCCC2C2CCN(C(=O)CC3CC3(C)C)C2)=O)o1 N1(C(C2=CCCC(C)(C)C2)=O)CCCC2CCN(C(=O)COC(F)F)CC12 O=C(CCC(CF)CF)NCCn1cc(C(=O)Nc2ccc(O)cc2F)cn1 C(C(=O)NC(C)C(C)C(=O)Nc1cc(O)ccc1C)(C(C)(C)C)OC C12(NC(CCC)=O)CC(C)(C1)OC21CCN(C(c2nc(O)sc2C)=O)CC1 C1(NC(C(CC2C(C)C2)C)=O)CCC2(CCN(C(=O)CN3CCCCC3)C2)C1 O=C(C1=CCCN(C(c2ccc3occc3c2)=O)C1)NC1=COC=CC(Cl)=C1 C1(CNC(=O)CC2CC2(Cl)Cl)CN(C(=O)COC2CCOC2)CCCO1 CCCC(C(=O)N(CC(c1ccc(F)cc1)C)C(C)C)NC(N)=O c1(NC2CCCN(C(=O)CCCCc3ccccc3)C2)ncnc2[nH]cc(I)c12 CC(CC(N)=O)C(=O)NCC1(F)CCC(CNC(=O)CC2CCC(=O)N2)CC1 C(=O)(CC1=CSC2=NCCN12)N(CCCCN(C(C1CN(C(C)=O)C1)=O)C)C(CC)OC c1(C(=O)NCC(C)CNC(C2CC2F)=O)ccc(CN2CCOCC2)o1 C1(C(=O)NCCNC(c2c(C#C)ccc(F)c2)=O)Cc2nn[nH]c2C(C)C1 N1(C(C(C)NC=O)=O)CCC2(CCCN(C(=O)CS(=O)(=O)N3CCOCC3)C2)C1 C1(C)(C(=O)Nc2cn(CC)nc2)CCCN(Cc2ccc(OC)nc2Cl)C1 N1(C(C2C(C)C2)=O)CCCCC1CN(C(=O)C(O)COCc1ccccc1)C C1(S(C)(=O)=O)(C(N2CC(C(C)NC(=O)CC3CCCCC3F)C2)=O)CCCC1 CC1(C)C(C(=O)NC2CCN(C(=O)Cc3cncnc3)C23CC3)CCS1(=O)=O C12(O)CC(C1)CNC2=O.O=C(CCSC1CCC1)NCC1CN(C2CC2)C1 n1(CC(=O)NC2CN(C(CC(CC=C)(C)C)=O)CC2F)c(=O)oc2ccccc12 C12(NC(C(C)C)=O)CCCCC1N(C(=O)CCc1nc3ccccc3o1)CC2 c1(NC(C2CCN(C(c3cc(CN4CC4)[nH]n3)=O)C2)=O)cc(C2CC2)cnc1Cl c1(C(=O)NC(C(=O)NC(CCCC)CO)C)ccn2ccnc2c1 c1(OC)cc(OC)c(C(N2CCC(C(=O)Nc3ccc(I)c(F)c3)C2)=O)cc1Br C=CCCCCC(=O)NCCCC(C)(c1ccccc1)NC(=O)COCC(=O)OC C=C1CC2(C1)CC(C(=O)NC1(C)CCN(C(c3ccsc3C#N)=O)C1)C2 N1(C(c2cc(C(C)C)no2)=O)CC2(CC2)CC1CNC(C1CCCO1)=O N1(C(C23C(CN(C(C(CCN(C)C)O)=O)C2)C3)=O)CCC(F)(C#N)C1 c1(C(C)C(=O)NC2CC2CNC(=O)CCN(CC(F)(F)F)C)ccccc1 C1(NC(CC(=O)NCC#C)=O)CCCN(C(c2ncc[nH]2)=O)CC1 C(=O)(CS(=O)(=O)C(C)(C)C)NCC1CN(C(CCSCCCC)=O)C(C)(C)C1 c1(SC)cccc(NC2(CO)CN(C(=O)C(F)CC3CCCCC3)C2)c1[N+](=O)[O-] C1(NC(c2cc(C)oc2C(F)(F)F)=O)CC2CC1N(C(=O)CCCN(C)C)C2 N1(C(CCCSc2ccc(OCC(=O)NCC)cc2)=O)CCC2(CC1)OCCO2 CC1C(NC(c2c[nH]c(=N)o2)=O)CCCN1C(C1CCOC(C)(C)C1)=O Cc1ccc2c(=NCCc3c[nH]c(=N)s3)[nH]c(NC(CC(N)=O)C3CC3)nc2c1 Cc1cn(C(C)C)cc1C(N1CCCCC1CNC(c1ccccc1CO)=O)=O C1(CC(=O)NC2CC3(C(N)C3)C2)Cc2ccccc2C1 Cc1cc(C(=O)NC(C)CCCNC(=O)CN2CC(F)(F)C2)on1 c1(CC)ccc([N+](=O)[O-])c(C(=O)NC2CC(NC(=O)C(C)(C)C3CCC3)C2)c1 C(C(C)C(=O)NOCc1cnccn1)N(C(c1c(C(C)C)cccc1)=O)C CC(C)CC(C(=O)C(=O)CCOC1CCC1)c1ccccc1.C1(CN)CC1N N1(C(c2cc(C)[nH]n2)=O)CCCCC(NC(=O)COCCc2ccccc2)C1 C(CC(C)(C)C(=O)N1CCOC(CCNC(C2COCCO2)=O)C1)OC C1(C(N2CC(NC(Cc3c(OC)nccc3)=O)C(C)C2)=O)CC(C)(C)OC1(C)C CS(=O)CCC(=O)NCCC1(NC(C2SCCS2)=O)CCCC1 CCCC(Cc1ccccc1)C(=O)N1CCN(c2ccccc2)CC1C Cc1c(C(N2CCCC(NC(=O)CCC3CCOC3)C2C)=O)cccc1C1CC1 C1(C(=O)NC2CC(CCC(=O)N(C3CCC(C)C3)C)C2)C2CCCC(=O)C12 C1(C)(CC)C=C(C(=O)N2CCC(C(=O)N(C3CCC3)CCO)(CC)CC2)C1 n1(CC)ncc(NC(c2cn(CCNC(C3CC3(C)C)=O)nn2)=O)c1C N1(C(C(N2CCCCCC2)C)=O)CCN(C(=O)CC2(C)CCC2)C(C)C1 C1(F)(CNC(CC2CCN(CCCC)C2)=O)COCCN(C(=O)C(=O)N(C)C)C1 N1(C(c2c(C)cno2)=O)CC2(CCC(CNC(C3CCC(F)C3)=O)O2)C1 N1(C(c2ccn(C)n2)=O)CC2CC(C1)N2C(c1ccccn1)=O c1(C(=O)NC(CC=C)CNC(C2CC2c2ccccn2)=O)cn(C(C)C)nc1C C(C1c2ccccc2CN1C(C1C2CC3C(C2)C13)=O)NC(c1ncccc1CO)=O C=C1CC2(C1)CC(C(=O)N(CCC)CCNC(=O)CC(C)COC)C2 c1(C(=O)NC2CN(C(C(C(C)C)NS(C)(=O)=O)=O)CC2O)cc2nc[nH]c2cn1 CC1Oc2ccccc2C1NC(=O)NC1CCCN(S(=O)(=O)c2ccccc2)C1 c1(OC(C(=O)NCC(C)(CC)NC(CCC)=O)C)cccc(C(C)=O)c1 CC1(C)CCC(CNC(C2CC3CCC(C2)C3)=O)N(c2ncnc3[nH]cnc23)C1 c1(C(=O)NCC=CCNC(Cc2ccc(C#N)cc2)=O)nccc2c1CNC2=O C(=O)(C(CCNC(c1cnncc1O)=O)OC)N(CCCOC)CCO c1(C(=O)NCC2(F)CCN(C(c3nn(C)c(O)c3)=O)C2)ccc2cccnc2n1 C1(CC)CCCC1.CCC(=O)NCCN(C(=O)CN(C)CC)N1CC1=O C(CCNC(c1cccnc1C1CC1)=O)(C(C)C)NC(C1N(CC)CC1)=O n1(CC)cc(C(=O)N(C2CC(NC(=O)CC3CC(O)C3(C)C)C2)C)c(C)n1 CN1CCCc2cc(CC(=O)NCC(CO)NC(=O)C=C3CC3)ccc21 C(=O)(CC(F)(F)C(F)F)NC(CCNC(c1c(C)oc(C(C)C)n1)=O)C(C)(C)C C1(NC(C(=O)NCC)=O)CC2(C(=O)Nc3cccc(OC)c3OC)COC1C2 CC(N=c1[nH]c2c(c(=NC(C)C3CC3)[nH]1)CSC2)c1cn[nH]c1 C1(COC)(CNC(c2c[nH]nc2C(F)F)=O)CN(C(=O)C(C2CCCC2)O)C1 C(=O)(CC1=NNC(=O)C1)N(CC(CC)NC(=O)CC1CCCOCC1)C c1(OC)nc(C)ccc1C(N1CCCC(N(C(=O)C(c2ccccc2)C)C)C1)=O N1(C(CCC=C(C)C)=O)CC(NC(c2cn3ccnc3s2)=O)CC12CCCOC2 C1(CC(=O)NCc2cccc(F)n2)CCN(C(c2cc(F)c[nH]2)=O)CC1 c1(C(=O)NCC(C2CC2)NC(c2ccoc2Br)=O)noc2c1CCCC2 Cc1nn(C)c(C)c1CC(=O)NC1CN(C(=O)CC(C)(C)C)C2CC12 C(=O)(C(C)CCCC(C)C)NC(CCN(C(C(C=C)O)=O)C)C c1(NCC2CCN(CC(=O)Nc3ncc(Br)cn3)C2)ccc(F)c(CO)c1 N1(C(Cc2cncc(C)c2)=O)CC2CCCC2C1C(=O)N(C(C)CN(C)C)C C1(C(C)C)CN(C(c2ccc(CF)cc2)=O)CCCN1C(=O)C(C)OCC(C)C Cc1cc(C(c2cn(CCc3[nH]nnc3C)nn2)(C)N(C)C)no1 c1(CC(=O)NCC2N(C(=O)OC)CCC2C)ccc(OC)c(O)c1 c1(CC(N2CC(CNC(CC(C)C)=O)C3C2C3)=O)ccc2c(c1)CCCC2 N1(C(C(N2CCCC(C)C2)=O)=O)CCN(C(C2C(F)(F)C23CCC3)=O)C2(CCC2)C1 c1(C(N2CCC(NC(CC=C)=O)(CF)C2)=O)cc(C)c(C)nn1 c1(C(N2C3CN(Cc4nc(C)sc4)C(C3)C2)=O)nc2c(s1)CN(C)CC2 c1(C(N2C3C(NC(CC=C)=O)CC(C3)C2)=O)oc2ccc(C)cc2c1C CC1CN(C(=O)C(C2CC2)N(c2ccccc2)C)CCN1C(c1ccncn1)=O c1(OC)nc(Nc2ccsc2NC(=O)CCn2ccccc2=O)nc2[nH]cnc12 c1(OC)c(C)cc(C(N2CCC(O)(CNC(C34CCC(CC3)C4)=O)C2)=O)cc1Cl c1(NCC2CCCC(=O)N2)ccc(S(=O)(=O)N2CCC=C(Cl)C2)cc1F CCCC(CC(=O)NCC)NC(C1(C)CCC(NC(=O)OC(C)(C)C)CC1)=O c1(CCN2CCC(O)(C(=O)OC(C)(C)C)CC2)nc2ccccc2o1 c1(C(C(=O)NC2CC(NC(c3c(C(C)C)cco3)=O)C2)C)cccc(O)c1 C(=O)(CCCC(=O)NC1(CCNC(=O)CCc2ccc(C)s2)CCC1)OCC C1(C(N2CC(C)C(NC(=O)Cn3nnc(C(C)(C)C)n3)C2)=O)CC2CCC1CC2 c1(C(=O)NC(CNC(C(CC=CC)CC)=O)(CO)CO)csc2c1CCC(C)C2 N1(C(CCc2cccc(C)c2)=O)CCN(C(c2cc(C)cs2)=O)CC1CO C(C1=CCN(C(c2ccnc(OC(F)F)c2)=O)CC1)NC(c1ccncc1O)=O C1(N(C)C)CCN(C(C2CC2NC(c2cccc(CCO)c2)=O)=O)CC1 CC(CCNC(=O)OCc1cnn(C)c1)C(=O)OC(C)(C)C.C CCCCC(CC)NC(c1ccnc(CSC)c1)=O.C12(CC1)C(=O)N2 n1(CC)nc(C(=O)NC2CN(C(=O)CC(F)F)CC2SC)c2c1CCOC2 Cc1ccc(F)cc1C(=O)N(C)CCN(C(=O)Cc1cncc(Br)c1)C CN(C)S(C)(=O)=Nc1nc(-c2nc(CO)nn2C2CCOC3(CCCC3)C2)cs1 c1(OC)cc(C(=O)NC2CC(C(=O)NCC3CCN(C)C3C)C2(C)C)n(C)n1 N1(C(c2ocnc2C(F)F)=O)CCN(CC(F)F)C(c2ccccc2)C1 C1(CNC(C=CSC)=O)CC(C)CCN1C(=O)COc1cccc(F)c1 c1(OC)ccc(F)c(-c2cn(CC(N3CC(C(=O)O)C(C)(C)C3)=O)nn2)c1 c1(OCCC(N2CCN(C(C3(O)CCSCC3)=O)C3CC23)=O)cccc(Cl)c1Cl N1(C(C2C(OC)(OCc3ccccc3)CC2)=O)CCc2c(C(=O)O)cccc21 N1(CC(=O)NC(CCNC(C(CCC#C)O)=O)C)C(=O)NC2(CCCC2)C1=O C(=O)(C(=O)CC(C)C)NC(CC(=O)N1CC(C)(OC)C1)(C)C C(CC(C(=O)N1CC2CC2(C(=O)NCC2(CC(C)C)CCC2)C1)OC)OC C1(NC(c2ccc(C)cc2)=O)CCCC2CCC1N2C(C1C2CC3C(C2)C13)=O c1(OC)ccnc(C(=O)NCCCCCCNCc2ccc(C(=O)O)cc2)c1 c1(NC2CC(NC(CC)=O)C23CCC3)nc(C)c(C#N)cc1Cl c1(C(=O)NCC2CCC(C)N(C(C3CC(C)(C)C3)=O)C2)c(O)cc(Cl)cc1Cl c1(CNC(C(=O)N(C(C)C)C)=O)cccc(Cl)c1OC(F)F CC1CN(C(c2cc(CNC(=O)CC(C)C3CC3)[nH]n2)=O)CCN1C1CC1 c1(CC2CC2NC(c2scc(C(=O)NC3(C)CCC3)n2)=O)ccccc1F CCCS(=O)(=O)CC(=O)NCCC1CCN(C(=O)CCCOC)C(C)C1 C(=O)(CC(C)C(F)F)N1CCC(CCN(C(C(c2c(C)noc2C)C)=O)C)CC1 N1(C(C(CC)OC)=O)CCC(NC(=O)C=C(C)c2ccccc2)C(OC)C1 c1(C(C(CS)COC)CC)cc(S(=O)(=O)N)ccc1Br C1(C(CC)(O)CNC(c2csc(=N)[nH]2)=O)CCC(C)CC1 N1(C(C(c2cccs2)OC)=O)CC2CCC(C1)N2Cc1cnsn1 c1(NC(C2N(Cc3ccc(CC)s3)CCOC2)=O)ccc(Br)c2cc[nH]c12 c1(C(N2CC3C(NC(C(C)OCCOC)=O)(C3)C2)=O)cc(C)nc2ccnn12 Cc1noc(Cl)c1CCC(=O)NCC(C)CN(C)C(c1nn(C)cc1Cl)=O N1(CCC(=O)NC2CC(CNC(CN(C(C)=O)C)=O)C2)CCCC1=O CCCCCC(F)C(=O)N1CC2(CNC(C3(C)CCOC(C)C3)=O)CC(F)(C1)C2 c1(CNc2ccc(C(=O)NCCC)cn2)nccc2ccccc12 C(=O)(CC(C)C(F)F)NC1C=CC(CNC(c2c(C)onc2C(C)C)=O)C1 C1(NC(C=CCOC)=O)CC2CC(C1)N(C(=O)CSc1ccc(F)c(F)c1)C2 C#CCC(CC#C)C(=O)NC1CN(C(C2(CC=C)CCCC2)=O)CC1(C)C c1(C(=O)NCCN(C(CN2CCCC(CC)C2)=O)C)nn(C)c2c1CCC2 c1(C(=O)NC(CCCC)CNC(=O)C=Cc2cnc[nH]2)cccc2cccnc12 C12(C(N3CCN(C(CCSC)=O)C(CCO)C3)=O)CCC(O)(CC1)CC2 CC1CN(C(=O)Cc2ccns2)CC1(C)C(=O)NC1CN2CCC1CC2 Cn1nc(C(=O)NC2CCCCN(C(C3C=CCC3)=O)C2)c2cc(F)ccc12 C#CC1(C(=O)NCc2ncn(C(C)C)n2)CN(C(c2cc(Cl)c[nH]2)=O)C1 N1(C(C=C(C)C)=O)CCCN(C(c2cc(C)n(C)n2)=O)CC1C N1(C(C)=O)CCCCC1C(=O)NCCC1CC1.c1(C(C2CC2)S)conc1C(F)F C1(C(N(C2CCC(NC(=O)CC3(CO)CC3)CC2)C)=O)CC2(C1)C(F)(F)C21CC1 C1(CC(N2CCC(C(CC)CC)C2)=O)CC2(CC(NC(=O)OC(C)(C)C)C2)C1 Cc1cc(C(=O)NC(C)CNC(=O)CCc2cccc(C#N)c2)cc(C)c1 N1(C(=O)CN2CSCCSC2)CCCC12CCN(C(C1C3CC4C(C3)C14)=O)C2 N1(NC(=O)C(F)(F)Cc2cn(CC(C(C)C)CC(=O)O)nn2)CCCCC1C C#CCC(CC(=O)N(C(C)C(C)C)CCC(C)C)NC(=O)C1CC1 c1(C(N2CCCC(O)(CN(C(c3nc(C)sc3)=O)C)C2)=O)c[nH]c2cccnc12 c1(-n2cc(NCC(C3CN(C(CCC=C)=O)C3)=O)nn2)cccc(C(C)(C)C)c1 C1(NC(C(CCC)Cl)=O)COC2(CCN(C(=O)C(C(C)C)NC(C)=O)CC2)C1 c1(OC)ccc(C(=O)N(C(C)CCNC(=O)C(C)(F)F)C)c(Br)n1 N1(C(CSC(C)C)=O)CCC(C)(C)C1C(N1CCCC(C(F)F)C1)=O CC1CCCN(C(=O)CCOCC(F)F)C1CCNC(c1c(F)cncc1Cl)=O C(CCCC(=O)NC(C)Cc1cncn1C)N(C(c1cnc(OC)s1)=O)C C12(C(N(CCCN(C(C3CCN(C(=O)OCC)C3)=O)C)C)=O)CCCC(CO1)C2 c1(-c2cn(CC3CCN(C(C(CC)(C)O)=O)CC3)nn2)ccc(Cl)cc1F n1(CC)ncc2c1CC(C(=O)NCC(C)O)CC2.C(CC(C)C)O.C1(=O)CO1.C1CO1 CC1CC(NC(c2cccs2)=O)CN(C(C2CC2C(c2ccccc2)=O)=O)C1 N#Cc1cc(N2CCC3CCN(C(=O)CC4=CCCCC4)C3C2)ccc1[N+](=O)[O-] CC1CC(CCNC(c2csnc2Cl)=O)CCN1C(c1cc([N+](=O)[O-])c[nH]1)=O CC(=O)CCCCS(=O)(=O)N1CCC(Cc2nccn2C)C1 C=CCCCCCCC(=O)NCC1CC1C1CCCN(C(=O)COc2ccsn2)C1 CC1(CCNC(=O)C(=O)NC2CCN(c3ncco3)CC2)CCOCC1 N1(C(c2c(C)onc2)=O)CC2CC(NC(c3n[nH]c4c3COCC4)=O)CC2C1 c1(C(C(=O)NCC2COCC2NC(=O)C(C2CC2)OC)OC)c(F)cccc1F c1(C(=O)NC2(CO)CN(C(CCCC3C(C)C3)=O)C2)cccc(N=[N+]=[N-])c1 C(C(=O)NCC1CCCO1)(C1=NOC2COCC12)N1C(C#N)COCC1 CC1(C(=O)Nc2cccc(C3CNC(=O)C3)c2)CNCC1(F)F c1(C(=O)NCC(CC)NC(=O)C(F)CC2CCCCC2)c(N)cc(C)cc1F C1(CNC(c2c(C)scn2)=O)C2CC2CN1C(=O)CC=C(Cl)Cl C1(CNC(C(C=C)(C)O)=O)CC(C(=O)N2CC(CC)(OC)C2)=NO1 C1(C)(CNC(C(C)Sc2ccccc2)=O)COCCN(C(c2cncs2)=O)C1 N1(C(CC2(O)CC(C)(C)OC2)=O)CC2(CCC2)CC1CNC(c1cc(F)c[nH]1)=O CC#CCC(C(=O)NCC(F)C1CCC1)NC(=O)CC(C)CN(C)C N1(C(c2c(C)cn(C)n2)=O)CCC2(C1)CN(C(C1(c3ccnc(Cl)c3)CC1)=O)C2 c1(CC(=O)NCCC(C)NC(=O)C(c2cccc(Cl)c2)O)nsc2ccccc12 CC1CN(C(C2(C)CC3CC3C2)=O)CCC1N(C)C(C1CN(C2CCC2)C1)=O N1(C(=O)OC(C)(C)C)CCC2CC2(CNc2occc2F)CC1 c1(C(N2CC(C(C)NC(C(C3CCC(=O)N3)C)=O)C2)=O)ccc(O)cc1Cl C1(CNC(c2c(CC)cc[nH]2)=O)CC(C(=O)NC2CCSCC2)=NO1 C1(OC)CN(C(=O)CC2CCCC2)CC1NC(c1cnn(CC(F)(F)F)c1)=O c1(C(N(C(CN(C(C2CC(OC)C2)=O)C)C)C)=O)ccc(N2CCNC2=O)cc1 C1(C)(C(N2C(CNC(Cc3cnc(C)[nH]3)=O)COCC2)=O)CCCC1(F)F CC1CCCN(c2ccc(-c3cn(-c4n(CCC)ccn4)nc3)cc2)C1 C1(=O)C(Cc2cnco2)N1.C(CC(C)N(C)Cc1cccs1)OC Cc1ccc(O)nc1CNC(c1c(CNC(=O)C(C)CO)nnn1C)=O N1(C(CSCC)=O)CCC(O)(CN(C)C(c2sc(-c3nc[nH]n3)nc2C)=O)C1 c1(N(CCCCCC=C)C)nc(NC2CCCCCC2F)c2sccc2n1 C(=O)(CC(C)CSC)N(CCC(=O)NCC(C)(C)CO)CC#C CCC(C(C)(F)F)NC(C1OCCC1CNC(c1cnc(C)nc1)=O)=O C(=O)(C(O)C(C(C)C)OC)NCC1C(O)CCN(C(Cc2cn(CC)nc2)=O)C1 C1(NC(C2CC(N(C)C)C2)=O)CC(F)CN(C(c2ccnc(C(N)=O)c2)=O)C1 c1(C(=O)NC)ccc(C(=O)NCC(C)CNC(c2cc(C#N)c[nH]2)=O)cn1 N1(C(C=CC=CC)=O)CC(CNC(c2cn(C3CC3)nc2C)=O)OC(C)(C)C1 Cc1ccc(C(=O)N(C(C)C(N2CCCC(C)(F)C2)=O)C2CC2)cc1F N1(C(c2ncnc(OC)c2F)=O)C2CCC1C(F)C(NC(=O)C(C)(C)CF)C2 N1(C(C2(c3c(OC)cccc3)CCC2)=O)CCC(NC(C2CC2C)=O)C(F)C1 Cc1cc(C(N2CCC(CC(C)NC(c3ccc(C#N)s3)=O)CC2)=O)nc(O)c1 N1(C(c2cc(C)cc(F)c2)=O)CC2CCCC2(NC(=O)CC23CCC(CC2)C3)C1 CC1(C)CCCC1(O)NC(=O)Cn1cc(C2CCC2(C)C)nn1 C12(NC(C(CSC)O)=O)CCCC1(F)CN(C(c1c(Cl)cccc1Cl)=O)C2 Cc1ccc(CC(=O)NCCCC2(NC(=O)C=CC(F)(F)F)CC2)cn1 c1(C(=O)NC(CNC(c2ccc(OC)c(Cl)n2)=O)CO)c[nH]c2c(Cl)cccc12 c1(NC(C)=O)cc(Cl)ccc1C(=O)NCCCNC(c1c[nH]cc1C(C)(C)C)=O Cc1ccc(-c2cn(CC3C(CNC(C4(C)CSC4)=O)C3(F)F)nn2)cc1 Cc1noc(C)c1CC(N1CCCC(CN(C2CCS(=O)(=O)C2)C)C1)=O C(CCCC(N)=O)(C(=O)NCc1cc(O)nc(Cl)c1)N1CC(O)(CN(C)C)C1 C1(CC(=O)NCC(CN(C(COCCC(C)C)=O)C)(C)C)CCCCC12CC2 Cc1cc(NC(=O)C(C)(C)CC2CCC2)ccc1NC(=O)CCc1ccon1 N1(C(C23CCCCC2C3)=O)CCCCC(C2CN(c3ncc4ncnc-4[nH]3)C2)C1 C1(N(C(CNC(CNC(C(C)(C)NC(C)=O)=O)=O)=O)CCCO)CCCCCC1 C(=O)(CCC(=O)NN(C)C)NC(C)CCCNC(C1CCCCC1)=O N1(C(C2(CCC=C)CC2)=O)CCCCC(CCC(=O)NC2CCC(O)C(O)C2)C1 N1(C(C2(C#C)CC2)=O)CCCC2(C1)CN(C(=O)CC(C)P(C)(C)=O)C2 C1(F)(CNC(c2cc(C)c(C)s2)=O)CCCN(C(=O)COC(C)(C)C)CC1 CN=c1ccc(C(=O)NCC2CC2CNC(c2cnn(C3CCCCC3)c2)=O)c[nH]1 C1(C(N(CCNC(C)=O)C)=O)CC12CCN(C(C1CC(=O)C1(C)C)=O)CC2 c1(OCC)ccc(Cl)cc1CC(N1CCC(CCNC(C2CC2C(C)C)=O)C1)=O C1(NC(C=Cc2cnc(C)s2)=O)CCN(C(=O)C(C)N(C)C)C(C)C1 c1(C(=O)NC2CN(C(CCNC(COC)=O)=O)CC2F)ccc(O)nc1Cl C(=O)(CC(F)(F)C(F)(F)F)NC1(C)CCN(C(CC2CCCC(C)(C)O2)=O)C1 CCC(CCC(=O)N1CC(c2ocnc2CNC(c2cc(C#N)[nH]c2C)=O)C1)OC c1(-n2cc(CC3(F)CN(C(c4nc(C(C)=O)sc4)=O)C3)nn2)c(F)cccc1F Cc1nn(C(C)C)cc1C(=O)NC(C)CCNC(c1ccc(CC(C)C)o1)=O CCCC#CC(C)(C)NC(=O)C(c1ccco1)Oc1ccccc1 N1(CC)CCCC(C(=O)N(C(C)CNC(c2[nH]ccc2-c2cccs2)=O)C)C1 Cc1cn2cc(C(=O)NC3CCCCN(C(C4(C)CC5CCC4O5)=O)C3)nc2s1 c1(CN2CCN(CCN=[N+]=[N-])CC2)ccc(C(F)(F)F)c2c1CCCC2 CC12CN(C(=O)C=Cc3cnc[nH]3)CC1CN(C(=O)CC1CCCCC1(F)F)C2 c1(C(N(CC(CNC(C(C)OCOC)=O)O)C)=O)cnc(C(F)F)c(C)c1 CCC(CC)(CCOC)C(=O)N1CCC(NC(=O)Cc2ncccc2C)C1 c1(NC(C(c2ccnn2C)C)=O)cc(Cl)cnc1O.c12ccc(nc1)CNC2=O O=C1Cc2c(N3CCOC(C(=O)Nc4ccc(I)cc4Cl)C3)ncnc2N1 n1(C2CCN(c3ccc(OC)cc3)C2)ncc2c(O)nc(=NNC(=O)OC)[nH]c12 CN1CCC(C(=O)NC2(C(=O)N(C3CC4(CCC4)C3)C)CCC2)C1=O CCCCCCC(C)C(=O)OCC(C)CSC1CCC1 c1(C(=O)NCC=CCNC(c2[nH]c(CC)c(Cl)n2)=O)csc2nccn12 c1(C(N(CCNC(=O)CC(c2cccs2)NC(=O)NC)CC)=O)ncncc1C C1(NC(C(C)SCC)=O)CCCN(CC2CC2(C)C)C1 c1(C(C)(C)C)cccc(C(=O)NCC(O)CNC(=O)C(F)=C2CCC2)c1N N1(C(C=CC(=O)OCC)=O)CCCC(C(=O)NCc2cncc(N(C)C)c2)C1 Cc1ccc(CC(=O)NCC(C)(C)NC(=O)C=CC=C(Cl)Cl)o1 C(=O)(C1=CCCC1(C)C)NC1CCN(C(C2C(OC)CCC2)=O)CC1C C(=O)(C1=C(Cl)CC1)NCCOCCN(C(=O)C(c1ccc(Cl)s1)=O)C Cc1cc(C(=O)NCCC2CC(NC(c3snc(C)c3N)=O)C2)cc(O)n1 c1(C(=O)NCCCN(CCCNC(c2c(CC)cc[nH]2)=O)C)cnc(C)c(C)c1 c1(C(N(C)CCN(C(=O)C(F)C2CCC2)C)=O)cccnc1SC(F)F CC1CCC(NC(=O)Cc2cccc(O)c2F)CN1C(c1cc(C#N)c[nH]1)=O c1(SCC)ccc(C(=O)N(CC(O)CNC(=O)C(C)NC(=O)NC)C)o1 C1(CNC(=O)CSc2cn[nH]c2)C2CCN(C(=O)CCC3CCOC3)CC12 c1(C(=O)NCCCN(C(C2CCC(F)C2)=O)C2CC2)cc(F)c(Cl)cc1Cl c1(NC(C2N(C(c3c(C)ccnc3)=O)CCC2O)=O)ccc(Br)c(C)c1C C(F)(F)(C(=O)NC(C)CNC(C1(c2nc[nH]n2)CC1)=O)C1(OC)CC1 c1(C(N2C(C)CN(Cc3ccc(Cl)nc3Cl)CC2)=O)cc([N+](=O)[O-])cc(Br)c1O CCCCC(O)C(C)C(=O)N(CC(=O)NCc1cccc(C)c1)C1CC1 N#Cc1ccc2ncc(C(=O)OCC)n2c1.C12CCCN(C1)C2.c12ncn(n1)C2 Cc1cc(Cl)cc2[nH]c(C(=O)NC3CS(=O)(=O)CC34COC4)cc12 C1(CN(C(c2c(CC)nco2)=O)C)CCC(CNC(C2C(C)(C)C2(C)C)=O)CC1 N1(C(C(N2CCC(C)CC2)=O)=O)CC2(CNC(C3COC4(CCC4)C3)=O)CC1CO2 N1(C(=O)CC2CCCC2)CC2CCCC1C2c1cn(CC2CCCCC2)nn1 C12(NC(C3(C)CCC(F)(F)CC3)=O)CCCN(C(C3(C#N)CC3)=O)CC1C2 C(c1ccc(N)c(N)c1)=CCNC(C(=O)NCCC1(OCC)CCOCC1)=O C1(C(N2CC3(CN(C(c4ccc(F)c(F)c4)=O)C3)C2)=O)CCc2nn[nH]c2C1 C12(CNC(C(C)N3CCC3)=O)CCCC1N(C(c1cncc(Cl)c1Cl)=O)CC2 c1(C(N2CCN(C(c3c(C)c[nH]n3)=O)C(C(F)(F)F)C2)=O)ccc2[nH]ccc2c1 Cc1cc(F)c(C(N2CCCC(N(C)C(c3cnnn3C)=O)C2)=O)c(F)c1 C1(C(N2C(C(=O)NC)CCC2)=O)CN(C(c2cc(C)cc(O)c2)=O)CC12CCC2 N1(C(=O)Cn2cncn2)CC2(CCC(CNC(=O)C(F)(F)C(O)C3CC3)O2)C1 N1(C(c2cc(C(=O)OCC)c(C)o2)=O)CCC(NC(=O)C(O)C2CC2)C(F)C1 C1(c2cn(C(C)CC3OCCOC3(C)C)nn2)CCN(C(=O)CO)C12CC2 C1(CNC(c2n(C(C)C)cnc2)=O)CC(C)CN(C(=O)C(c2ccnn2C)O)C1 C1(NC(Cc2c(C)n(C)cn2)=O)CCN(C(c2c(C3CC3)cnn2C)=O)CC1C N1(C(C(CCNC(C(CC)=CCCC)=O)O)=O)CC(C)C(C)C1C C(=O)(C1COc2ccccc21)N1CCC(NC(c2ccc(Cl)[nH]2)=O)(CO)C1 C1(CC(N2CCC(NC(C34CC(C)(OCC3)C4)=O)C2)=O)COCC2(CCC2)O1 O(C1CCc2ccc(Br)cc21)C(c1c(C)cc(C(N)=O)cc1C)=O C1(CNC(Cn2c(CCC)ncc2)=O)CC(F)(F)CN1C(=O)CCCC(N)=O C1(NC(C2(OCC)CC2)=O)CN(C(c2c[nH]c(=S)cn2)=O)CC12CC2 Cc1ccc(C(=O)NC2CCC2NC(=O)CCCn2cccc2)c(C)n1 O=C1NCc2c(C(N3CC4(CCN(C(=O)C5=NOCC5)CC4)C3)=O)cccc21 CC1CN(C(=O)OC(C)(C)C)CCCN1C(=O)CS(C)(=O)=O N1(C(CC(C)OC)=O)CCC2CCC(NC(=O)C(C)(C)c3ccno3)C12 N1(C(C(CC(=C)C)OC)=O)CCC2CCN(C(=O)C(C3CCCC3)OC)CC2C1 C12(C(=O)NCC3(O)CN(C(c4cc(N)c(F)cn4)=O)C3)CCOC1CC(=O)NC2 N1(C(CCC(C)OC)=O)CCCC2(NC(=O)C(=Cc3ccccc3)C)CCCC12 c1(CC(=O)NCCN(C(C2(C(C)C)CCCO2)=O)CC2CC2)nc([N+](=O)[O-])n[nH]1 C(=O)(C1Cc2ccccc21)NCC1C=CC(NC(CC2CCN(C)CC2)=O)C1 N1(C(C2C(OC)CCC2)=O)CCN(C(c2ccnc(C)c2)=O)CC1C c1(C(N(C2CC(C(NOC3CC(CC)C3)=O)C2)C)=O)cc(C)sn1 C(CN=c1cc[nH]cc1S(=O)(=O)NC(C1CCCC1O)C)SC(C)C c1(OC)cccc2c(C(=O)NC3CN(C(C4CCC(=O)N4)=O)CC3(C)C)n[nH]c12 c1(C(=O)NC2C(C)N(C(c3ccc([N+](=O)[O-])[nH]3)=O)CC2)ccn2nccc2c1 c1(CC)c(C(N2CC(CNC(c3cnc(C)o3)=O)(OC)C2)=O)cccc1F Cc1nc(C)c(C(=O)NC2CC3CC2N(C(c2cnc(Cl)cc2N)=O)C3)nc1C c1(C(=O)NC2CC(C(N(CCC#N)CCC)=O)C2)cc(C)no1 CC(C)C(CCN(C(=O)C1=CCCC1)C)NC(=O)CCc1ncc(F)cn1 C1(C(=O)NCC2(OC)CN(C(=O)COCc3ccncc3)C2)CC(C)OC1C C#Cc1ccc(F)cc1C(=O)NC1CC(N(C(=O)C(C)CC=C)C)C1 CS(C)(=O)=Nc1ccc(C(N2CCC(NC(C3CCC3)=O)C(O)C2)=O)cc1 CC1CN(C(C2CN3CCC2CC3)=O)CCC1NC(C1(S(N)(=O)=O)CCC1)=O c1(C(=O)NC(C2CCN(C(=O)C(C)(C)n3cc(Br)cn3)C2)C)csc(=N)[nH]1 N1(C(Cn2nnc(=N)[nH]2)=O)CCC2(CCCN(C(c3ccon3)=O)C2)C1 C1(N(N2CC(CC)C2)C(C2(C)CC=CC2)=O)CCN(C(c2csc(C)c2)=O)CC1 CC1CN(C(C23CC2C3)=O)CC2(CCN(c3ccc(C#N)cn3)CC2)O1 C(N=c1nc2c(ncn2C)c[nH]1)C1CCCCN(C(CC(C(C)C)C)=O)C1 c1(C(N2CCCC(C)(CNC(C(C)CF)=O)C2)=O)snc2ccccc12 CN1CCC(C)(C(N2CCC2CNC(=O)Cc2c[nH]nc2O)=O)C1=O c1(NC(C(N2CCN(CC)CC2)=O)C)ccc(Br)cc1[N+](=O)[O-] CCCC(C(=O)NCC1CCCN1C(C1C=CC=CC=C1)=O)NC(C)=O c1(CN2CCC(F)(C(=O)Nc3ccccc3Cl)C2)cccc(O)c1Br CCCCC(O)C(=O)N(C)CC1CCCN(C(=O)C(CC)CO)C1 C1(N(C)C(=O)NCC2COC(=O)O2)CC2CCC(C1)N2C C12(CNC(=O)CCN3CCOCC3)CCC1CCN2C(c1cscc1Cl)=O C1(C)(C(=O)OC)C2CCC(C2)C1NC(=O)NCc1nc(C)c(C)[nH]1 Cc1cc(C(=O)NCC2(NC(=O)CC(F)(F)c3nccs3)CCCC2)cc(N)c1 N1(C(C(=O)Nc2cccc(OC)c2)c2cn[nH]c2)CC(CO)CC(C(C)(C)C)C1 CCCC(C)CC(=O)NC1(c2ccccc2)CN(C(C2CC(=O)NC(C)C2)=O)C1 c1(C(N(C2C(N(C(=O)C=CC3CC3)C)CCCC2)C)=O)cccc2[nH]nc(O)c12 C#Cc1cc(F)c(C(=O)NCC2CN(C(C3(F)CC=CC3)=O)CC2(C)C)c(F)c1 CC(C)CC(C)(CO)NC(C1CCC1NC(=O)CCC(C)(F)F)=O Cc1n[nH]c(C)c1CC(=O)N(C1CCN(C(=O)Cc2cscn2)C1)CCO C1(OC)CCC(CONC(c2ccoc2CNC(=O)CCC2CCC(=O)C2)=O)CC1 C1(C)(C(=O)NC2CCC(CNC(c3ccc(CC)o3)=O)C2)CC2(CC2)C1 C(C(=O)N1CCC1CC(=O)N(C(C)CCSC)C)(C1CC1)OCC Cc1ccc(N)c(C(=O)NC2CC(F)(CNC(C3CC4(CCC4O)C3)=O)C2)c1 N1(C(c2snc(C)c2N)=O)C(C)C2CC1C2NC(C1CCCN1S(C)(=O)=O)=O C12(CNC(c3ccc(C)c(CO)c3)=O)CC(CCO1)N(C(c1cnnn1C)=O)C2 C(=O)(CC(C(=O)NC1CC(CNC(C2CC(C)(C)C2)=O)C1)N1CCCCCC1)OC C1(NC(CCNC(C)=O)=O)CC2CC(NC(c3ccc(OCCF)cc3)=O)C2C1 CC1CN(C(c2cnn(C)c2C2CC2)=O)CCCN1C(=O)C(F)c1ccco1 c1(C(=O)NCCC2CN(C(C3(C)CC4CCC3C4)=O)C2)cc2ccccc2cn1 c1(OC)ccc(OC)c(OC)c1C(N1CC2(CC2)CC1C(=O)OC)=O.C(=O)(N(C)C)O N1(C(C2=CCC(NC(c3cnc(CC)s3)=O)C2)=O)CCC(C)(C)C(O)C1 c1(OCC)ccc(C)cc1NC(C1(C2CCCO2)CCC1)=O N1(C(c2conc2C)C(=O)NCCOC)CC(CC(F)(F)F)OC(C)C1 C1(C(=O)NCCCOC(F)(F)F)CN(C(c2coc(C(F)F)c2)=O)C2(CCC2)C1 C(=O)(C1=C(Cl)CCC1)NCC1N(C(c2cccc(C(N)=O)c2)=O)C2C(C1)C2 c1(C(=O)NCC(CCOC)NC(=O)C(C)NS(C)(=O)=O)cccc(C(C)(F)F)c1 Cc1ccc(F)cc1C(N1CC(CNC(=O)COC2CCCC2)C(C(F)F)C1)=O c1(C(=O)Nc2cccc(C(=O)NC(CC)CO)c2)c(C)cccc1F N1(C(C2C(C(=O)OCC)C2)=O)CCN(CCNC(=O)C=Cc2cnc(C)s2)CC1 c1(NCCNS(C)(=O)=O)ccc(C(c2nnnn2CCc2cccs2)N(C)C)s1 Cc1cc([N+](=O)[O-])cc(C(=O)NC(C)(C)CNC(c2n[nH]c3c2COC3)=O)c1Cl C1(N(C)C(C2C3CCCC23)=O)CN(C(c2nnc(C(C)(C)C)s2)=O)CC1(C)C c1(C(=O)NCC2(O)CC(NC(C(CCC)N(C)C)=O)C2)c[nH]c2cc(Cl)ccc12 C#Cc1cccc(N(C)C(C2CC(=O)CN2C(=O)CN2C(=O)CNC2=O)=O)c1 c1(C(=O)NC2CN(C(=O)C=Cc3ccc[nH]3)CC2C(F)F)ccc2occc2c1 N1(C(C(C)OC(=O)OCC)=O)CCC(C(=O)NCc2nc[nH]n2)C1 N1(C(CC(CC)NC(C2CCCC(=O)N2C)=O)=O)CCn2nc(C)nc2C1 N1(C(CC2CC(NC(CC3(N(C)C)CC3)=O)C2(C)C)=O)CCCN(C)CCC1 CCC(C)(CC)C(=O)NC1CC1CNC(c1ncsc1C(C)C)=O c1(CC(=O)NC2CN(C(c3cc(CC(C)C)[nH]n3)=O)C2)ncnc2sccc12 Cc1cc2c(C(=O)NCC(CO)NC(=O)C(C)CC3CC3)nccn2n1 N1(C(C2CCC(C)(F)CC2)=O)CC2CC(NC(C3CCN(C4CC4)CC3)=O)CC2C1 c1(C(N2CC(N3CCN(Cc4ncccc4F)CC3)C2)=O)c[nH]c2cc(Cl)ccc12 N1(C(CCC)=O)CCC2CCN(C(c3cn(C4CCOCC4)nn3)=O)C2C1 N1(C(C=CC(C)(C)NC(c2ccc(=N)[nH]n2)=O)=O)CC2C1CCCC2 N1(C(COCC)=O)CCCC(N(C)C(C2CC3CC3C2)=O)CC1 Cc1cncc(CCC(=O)NCC2CCCCC2NC(=O)Cn2cnnc2O)c1 c1(NC(=O)CC2CN(S(=O)(=O)c3ccccc3Cl)C2)nc2cccc(Br)c2s1 C=C(C)C(O)CC(=O)NC1CCCN(C(=O)CSc2nccn2C)C1 C(CCCCC(=O)N1CC=CCC1)NC(C1C(C)CCC1C)=O c1(-c2nnc(N(CC)CC)n2CC23CCC(C2)C(=O)N3)ccnc2[nH]cnc12 c1(C(=O)NCC(CCOC)NC(c2cnc(COC)s2)=O)cc(F)ccc1F C1(NC(c2c(CC)ncs2)=O)CC(C)CN(C(=O)C(C)n2cccc2)C1 N1(C(c2ncn(CC)n2)=O)CCCC2CCN(C(c3cnn4c3CCC4)=O)CC12 N1(C(c2cc(OC)ncc2OC)=O)CCC2(CC1)CCN2C(c1ccoc1Cl)=O c1(C(N2CCC(C)(NC(COC(CC)C)=O)CC2)=O)n[nH]c2c1CCC(C)(C)C2 C1(C(=O)NCC=CCNC(=O)CCC2CCCOC2)CC2(CCOC2)C1 CC(CC(=O)N1CCN(C(c2cc(Cl)n(C)n2)=O)C2CCC12)CC(C)(C)C C1(CC(=O)NCCN(C(c2c(C(C)C)ncs2)=O)C(C)C)CCCC(=O)C1 C(=O)(CC(O)C(C)CC)NCc1c(C(=O)NC(C#CCC)(C)C)n[nH]c1 Cc1[nH]c(=N)ccc1C=CC(N1CCCC(NC(=O)C(F)CC(C)C)C1)=O Cc1cccnc1C(=O)NCC1CN(C(c2cc(Br)sn2)=O)CCO1 C=C(C)CCC(=O)NC1CN(C(=O)C(CC)CC)CC1c1nccn1C CC1(C)CCOC(CCNC(c2csc(C(F)F)c2)c2nnnn2CCCF)C1 O=S(=O)(c1c[nH]ccc1=NC1CCC(CCO)CC1)N1CCCC1CCCO c1(C(N2CCC(C(C)NC(CC=CCC)=O)C2)=O)ncc(C)cc1F N1(CC(C)C)CC(C(=O)NC2CCCC(CNC(C3CS(=O)(=O)C3)=O)C2)CC1=O N1(CC(N2CCC(CCNC(c3c(C)n(C)nc3)=O)C2)=O)C(=O)CCCC1=O N1(C(CCCOC(C)=O)=O)CC23CCCC2(C1)CN(C(c1c(Cl)cnn1C)=O)C3 c1(C(N(C2CC(C#N)C2)CC(N2C(C(=O)OC)CC2)=O)=O)ccc(=NC)[nH]c1 C(=O)(C1=C2CCCN=C2NN1)N1C(C)CCC(NC(C(C)=O)=O)C1 N1(C(c2cc(OC(CC)C)ncc2)=O)CC2CN(C(=O)C(C)(F)F)CC2(C)C1 CC(CC(N)=O)C(=O)NC1CC(CCNC(c2cc(C3CC3)nn2C)=O)C1 CCC(C(=O)NCC1(CNC(c2ccc(Cl)c(N)c2)=O)CCC1)C(C)C C(C(=O)NCC(F)(F)CO)(C(C)(C)C)NC(CCC(C)OC)=O CN1N=CC(CC(N2CCC2CC(N2CCC(O)(CC3CC3)C2)=O)=O)C1=O N1(C(C(N(C(=O)C(CO)NC(N)=O)C)C2CC2)=O)Cc2ccncc2C1 Cc1nc(C(C)C)oc1C(N1CCC(OCCNC(C2CC23CCC3)=O)CC1)=O CC1OC2CCC1(C(=O)NC(c1nc(C(=O)NC3CC(C)OC(C)C3)co1)C)C2 N1(C(CC=CCC)=O)CCOCC1CC(=O)NCC1(F)CC(O)C1 c1(OC)cc(C(N2CC(NC(=O)CC(F)F)C(F)C2)=O)cc(N)c1O c1(CC)cc(C(=O)NCC(C)N(C(C2(c3oncc3C)CC2)=O)CC)ccc1O n1(CC(=O)NCC(CNC(CC(CC)SC)=O)O)cccc(O)c1=O Cc1ccccc1C(=O)NC1CN(C(C2(N(C)C)CSC2)=O)CC1C c1(C(=O)NCCN(CC(C)O)C(c2nncc(OC)c2)=O)cc2c(s1)CCOC2 c1(C(=O)NC2CN(C(c3cccc(OC)c3)=O)C3C2C3)cnc2ncccn12 C1(C(=O)OC(C)(C)C)CCCCC1N=c1ccnc(C2CC2)[nH]1 Cc1cc(Cl)c(Cl)cc1C(N1CCCC1C(C)NC(C1(F)CCC1)=O)=O c1(C(=O)NCC(C)CNC(=O)CNC(c2ccncc2)=O)cccn2ccnc12 C(=O)(C(F)CC1CCC1)C(C=CC(=O)OC(C)(C)C)=O.C(COCCNC(N)=O)N c1(CCC(=O)NCC23C(CN(C(CCN(C(C)=O)C)=O)C2)C3)ccc(F)c(F)c1 N1(C(C)=O)CCCC1(C)C(=O)NCC1CCCN1C(=O)C(CO)NC(=O)COC C1(NC(CCCC=C)=O)CCCN(C(=O)C2=CCCC2)C1CC c1(C(N2CC(CNC(C3=CCCC3C)=O)OCC2)=O)ccc2cccnc2c1 c1(C(N(C(C)CNC(=O)CN2CCC(C)(C)C2)C)=O)cccc2c1NCCC2 C1(NC(C(c2ccccc2)N(C)CC)=O)CN(C(c2cnsn2)=O)CCC1C CCC(CC(=O)NC1C2CCCCC12C(N1CCC(N=[N+]=[N-])CC1)=O)C(F)F Cc1ccc([N+](=O)[O-])c(CNC(=O)C(=O)Nc2ccc3nnn(C)c3c2)c1 NC1CC2C(C(=O)N(C3CC3)Cc3ccc(Br)s3)C2C1 C1(CC)CN(c2cc(C#N)ncn2)CCN1C(c1ncc(Cl)cc1C)=O CN1N=CC(CC(N2CCCCC2CNC(=O)Cn2nnc(=O)[nH]2)=O)C1=O Cc1cc(C)cc(C=CC(=O)NC(C2CCN(C(c3ccc[n+]([O-])c3)=O)C2)C)c1 c1(CN(C2CC2)NCC)ccc(CN)cc1.c12ccc(cn1)c(=O)[nH]2 C1(C2(C(N3C(C(N4CC(n5ncc(C)c5)C4)=O)CCC3)=O)CC2)CC2C=CC1C2 c1(C(=O)NCCCCC(C)NC(CCC)=O)cncc(OCC(F)F)n1 Cc1cc(CN(CCC2(CC(C)(C)C)CC2)CC2CN3CCN2CC3)cc(C)c1 N1(C(CCSC)=O)CC2CCN(C(c3ccc(N(C)C)cc3F)=O)CC2C1 CC(C)(C)CCC(F)C(=O)NC(c1cccnc1)C(=O)NC1(C)CC1 N1(C(c2ccnc(OCC)n2)=O)CCC(C)C(CNC(=O)CCCC(N)=O)C1 c1(OC)cccc(NCC(=O)NCc2cccc(NC(=O)C(C)(C)SC)c2)c1 C=CCCN=C(NCC1COC(=O)O1)NC1CCC(OC)CC1 Cn1cnc2nc(=NCC#CC3CC3)[nH]c(NCc3nc(C4CCOC4)n[nH]3)c12 C(=O)(CC(F)(F)F)NCCOC(CNC(CCC1CC(OC)C1)=O)(C)CO C1(NC(COCCC=C)=O)CN(C(C2CCC2C(C)(C)C)=O)CC1N=[N+]=[N-] N1(C(C(C(=O)OCC)C)=O)CC(=O)NCC1C(N1CCC(C)(CO)CC1)=O c1(CC(N2C(C)C(NC(=O)COCCF)CCC2)=O)ccc2c(c1)CCC(=O)N2 c1(C(N2CCOCC(NC(C(C)OC)=O)C2)=O)ccc(P(C)(C)=O)cc1 C=CCC(C)(CC=C)NC(=O)NCCC1CCC(C)(C)CO1 C12(NC(=O)CC3CCCO3)CCC(C(=O)NC3CCCC3)(CC1)C2.C(CSC)O c1(CC(CNC(C2CC(OC3CC3)C2)=O)NC(C(C)SCC)=O)ccccc1 c1(OC)ccc(Br)c(C(=O)NC2CC3(C2)CN(Cc2cc(F)cc(Br)c2)C3)c1F C1(NC(C2C(CC)OCC2)=O)CCCC12CN(c1cc(C)nc(C(C)C)n1)C2 Cc1ccc(C#N)cc1C(=O)NC(CNC(c1ccoc1Br)=O)C1CC1 O=C1CNc2ccc(S(=O)(=O)Nc3cccc(-c4ccccn4)c3)cc2N1 C1(NC(C2(C)CC2(Cl)Cl)=O)CC2CC(C1)N(C(c1cncs1)=O)C2 c1(C(=O)NCc2cn(-c3c(F)cc(Br)cc3F)nn2)ccc2c(c1)OC(F)(F)O2 C(C)(CC(=O)NC(C)(CNC(=O)CCCOCCOCCOC)CO)OC C(=O)(CCC(=O)NC(C)CC(C)NC(C1CCCC1C(=O)OC)=O)NCC N1(C(C(=O)N(C2CCN(C(CCC=C)=O)C2)C)=O)CCC(CC)C1C(C)(C)C c1(C(N2CCCC(CC(N3CC(C)C(O)CC3)=O)C2)=O)cc(F)c(F)cc1Br c1(C(=O)NC2C(C(=O)NC(CC#C)C(=O)OC)C2)c(O)ccc2ncccc12 n1(CC(=O)NC2(CNC(C(C)SC)=O)CCC2)nc(C)c2cccnc12 C(=O)(C1=CC2(CN(C(C3(C(=O)OC4CC4)CC3)=O)C2)OC1)NC1(O)C(C)OCC1 Cc1onc(-c2ccsc2)c1C(=O)NCC(C)CNC(c1ccsc1C)=O C(CCCCCNC(=O)CC1CCOCC1OCC)NC(C(F)=CCC)=O C1(C)(CC)CCN(c2nnc(-c3ccc(-c4cccs4)cc3)n2C)C1 c1(OC)ccc(C)cc1C(=O)N(CCNC(=O)CCc1cnoc1)C1CC1 C1(NC(C2(C)CCOCC2)=O)CC2(C1)CN(Cc1ccc(Br)c(Br)c1)C2 C1(C(=O)NCC2CC(C)(C)N(C(c3cc[nH]c(=N)c3)=O)C2)CC2CCC1C21CC1 c1(C(=O)NC2C(OC)CN(C(c3c(CC)cc[nH]3)=O)C2)cc2c(O)ncnc2cn1 C(=O)(C(C)(C)C(F)(F)CC)NCC1N(C(c2cc(CC)no2)=O)CCCCC1 C1(C(=O)NCc2cc(C(=O)NC3C=CCCC3)sc2)CC12CCOCC2 c1(C(=O)NC(C)C(C)NC(c2c(C(N)=O)cnn2C)=O)csc2nnsc12 c1(CN(C(=O)CCCn2cc(CCO)nn2)Cc2cccnc2F)ccncc1F C(C)(C)(CCCF)NC(CCCN(C)C(C1CCS1(=O)=O)=O)=O c1(C(N2CCN(C(c3ccc(C)nn3)=O)CC2)=O)cnc(C(C)C)nc1O c1(C(N2CCN(CC(C)(C)NC(C(CSC)O)=O)CC2)=O)cc(C)[nH]c(=NC)n1 Cc1onc(C2CC2)c1C(=O)NCC1CC(NC(=O)CCC(=O)N(C)C)C1(C)C C1(C(=O)NCC(C2CCC2)NC(=O)Cc2cnco2)CC2(CC2)C1 C1(NC(C(C)c2cc[nH]n2)=O)CCC2(CCN(C(C3COC(=O)N3)=O)CC2)C1 c1(CCC(N2C(CNC(Cc3onc(C)n3)=O)COCC2)=O)cc(F)ccc1F C1(NC(c2cc(C(C)(F)F)n[nH]2)=O)CC2CCC1CN2C(=O)CC1CCCO1 c1(NCC(c2ccccc2)OC)ncnc(N2CCCC(C)CC2)c1C C1(C)(CNC(c2c(CC)occ2)=O)CCCN1C(C1CC(C)(C)C1)=O C1(CC#C)CCN(C(C2(CNC(=O)CCC3(C)CC3)CCCO2)=O)CC1 c1(C(=O)NC2CCN(C(C(C=CC)O)=O)C2C)cncc([N+](=O)[O-])c1 c1(C(=O)NC2(CNC(CCCC=C)=O)CCCCC2)cnc2cccnc2c1 C1(C(=O)NCC(CC)NC(c2cc(OCC)ccc2N)=O)CCOC(C)(CC)C1 S(=O)(=O)(c1c(F)cc(C#N)cc1F)N1C(Cc2ccccc2)CC(C)C1 N1C2CCC1CC(CCO)C2.C(C(=O)N1CC(C=O)C1)(C(C)C)SC c1(C(=O)NCC(CNC(=O)COC(F)(F)F)OC)cnc(C)s1 N1(C(c2c(NC)c(F)ccc2)=O)CC2=C(C1)CN(C(c1cc(COC)on1)=O)C2 N1(C(C)=O)CC2CC1CN(N1CCC(O)(Cc3ccc(F)cc3)C1)C2 CN1CCCCCC1C(=O)NC1CC2(C1)CC2C(=O)NCC1CCCC1 c1(C(=O)NCCC(C(C)C)NC2CCCCC2)ccc([N+](=O)[O-])c(N(C)C)c1 C(C)(C)(CCC(=O)NCc1ccc(O)cc1F)NC(C1C(c2n(C)ncc2)C1)=O C(=O)(C1=CCC(F)(F)CC1)NC1CCC(C)N(C(=O)Cc2ccccc2CO)C1 C1(C)(C(=O)NCC(CCOC)NC(=O)COCCCF)CCC(=O)NC1 N1(C(C(C=C)O)=O)CCC(C)N(C(c2cc(SC(F)(F)F)c[nH]2)=O)CC1 c1(NC(C2CN(c3ncc(I)cn3)CCC2O)=O)ccc2nn[nH]c2c1 CCC(C(=O)NC1CCC(CNC(=O)COc2ccccc2)C1)C(F)(F)F CCCC(C)(O)C(=O)NC(CNC(c1nccnc1C)=O)CC c1(CC)noc(C)c1C(=O)N(C1CC(NC(=O)CC2CCC23CCC3)C1)C c1(CC(=O)NCCC(C)NC(=O)C(C)NC(C2CCC2)=O)ccc2ccoc2c1 c1(OCC)ccc(F)c(C(=O)NCC(CC)NC(c2nnc(O)nc2O)=O)c1N c1(CC(C(=O)OC)NCC2CC(O)C2O)cccc(C)c1 C1(O)(C(=O)Nc2ccc(OC)nc2)CCN(Cc2ccnc(Br)c2F)CC1 n1(CC)ccc(C(N2CCCC(NC(=O)CN3C(C)CCCC3C)C2C)=O)cc1=O c1(CCC(=O)N(C)CC2N(C(C(C)c3ccco3)=O)CCC2)ccccc1Cl CC(O)C(F)(F)C(=O)NCC1(NC(c2coc(C(C)(C)C)n2)=O)CCCC1 C(=O)(C(C)N=[N+]=[N-])N(CCNC(CCCS)=O)C.C(COC)SCC c1(C(=O)NCC23C(CN(C(C(C4CC4)OCC)=O)C2)C3)ccc(Cl)cc1Cl c1(CCCC(=O)NCC2CCCCN2C(=O)CCC(F)F)ccc(CO)cc1 CN1CC(NC(C2(C)CCN(C(C3CC(C)(O)C3)=O)C2)=O)CCC1=O C1(CN(C(c2cc(C)nn2C)C(=O)NCCOCC)C)CCOCC1(C)C CS(=O)(=O)c1ccsc1C(N1CC2(C1)SCCC2NC(c1ccnnc1)=O)=O c1(OCCOC(C)(C)C)nc2c(c(=NCC34CCC3CCN4CC)[nH]1)COC2 CC1(C(=O)NCCC2CN(C(c3cnc(-c4cccs4)s3)=O)C2)CC1(Cl)Cl C(=O)(NNc1nc2cccnc2s1)c1oc2ccc(C)cc2c1 C1(C(N(CCN(C)C(C2COCCN2C2CC2)=O)C)=O)CCn2nnnc2C1 N1(C(C(C=C)C)=O)CCOCC(C(=O)NC(C2CCCCC2)CO)C1 c1(C(=O)NCCOC2CN(C(c3c(C)snn3)=O)C2)cc2cc(Cl)ccc2[nH]1 C(C)(C)(CCCC(=O)N1CCC(O)C(F)CC1)NC(C1(CC(=O)OC)CC1)=O C1(C)(C(N(CC(=O)N(C)CCC2CCCO2)C2CCC2)=O)CC=CC1 c1(C(=O)N)ccnc(C(=O)O)c1.CC1(Cc2cn(CC3C4CCCC34)nn2)CCCO1 C1(C)(CC)CC(NC(c2cccn(C)c2=O)=O)CN1C(c1ccnc(O)c1F)=O C(N=c1[nH]cnc2ccc(OC)cc12)C1(O)CN(C(C(COCC)N=[N+]=[N-])=O)C1 C(=O)(CC(O)CN(CC(C)O)CC)NCC(C(=O)NCC)NC(=O)OC(C)(C)C CCC(C(=O)NCC(C)CN(C)C(c1cnc(O)n(C2CC2)c1=O)=O)C(F)(F)F c1(NC(c2cc(CNC(C3C(OC)CCCC3)=O)oc2)=O)c(C)nn(C)c1C S(=O)(=O)(c1cccc(Cl)c1)N1CCCC(C(=O)Nc2ccc(F)nc2)C1 Cn1ncc(S(C)(=O)=O)c1C(=O)NCCCOCCCNC(=O)CCCF c1(C(C)NC(CN(C(CCC)C)Cc2ccccc2)=O)ccc(F)c([N+](=O)[O-])c1 C(=O)(C#CC(C)C)N(C)CC1N(c2snc(C(=O)OC)n2)CCC1 Cc1ccc(F)c(C(N2CCCCC2CNC(c2ncn3c2CCC3)=O)=O)c1O c1(OC)ccc2[nH]ccc2c1C(=O)NCc1cn(CC(O)COC)nn1 Cc1cc(C)c(NCCCc2ccc(OC(F)F)cc2)cn1 CC(CCC(=O)NCC(=O)N(C)C)NC(c1cc(F)n(C)n1)=O N1(C(c2ccc(Br)cc2)C(=O)NC(C(=O)OC)C)CCC(O)(CC(C)C)CC1 c1(OC)cccc(C(C(=O)NC23CC2CN(C(C2CC(C)=NO2)=O)C3)C(C)C)c1 c1(C(=O)NC23C(CN(C(CCOCC(C)C)=O)C2)C3)cc2c(Cl)nccc2s1 N1(C(C(C)NC(CN(C)C(C23CC(F)(C2)C3)=O)=O)=O)CC2CC(NC)CC2C1.CO C1(CNC(C(CCC)C)=O)CCN(C(=O)C(O)CN(C)C)CC1(F)F C(=O)(C(C)CC(N)=O)NCCCCCCNC(C(c1cc(C)oc1C)C)=O C(C(C)C(=O)NC(Cc1ccccc1)CCNC(C1(Cl)CC1)=O)OC CCC(C(=O)N1CCCC(N(C)C(c2c[nH]c(=NC)s2)=O)CC1)C(C)(F)F c1(C(N(CC(=O)NC2CC(CC)OCC2)C(C)C#N)=O)cc(F)ccc1F C(CCCN=c1[nH]c(=NC2CN(S(=O)(=O)CC)C2)c2c(F)cccc2[nH]1)=CC N1(C(c2c(C)cnnc2)=O)Cc2occ(C(=O)NC3(C)CC4CCC3C4)c2C1 N1(C(c2ccc(CNC(c3ncc(OC)nc3)=O)nc2)=O)CCN(CCO)C(C)C1 c1(C(N2C(CNC(C(CC)COC)=O)CC(F)C2)=O)ccc(N)c(F)n1 c1(C(N2C(C)CC(NC(CCn3c(C)cc(C)n3)=O)C2)=O)ccc(N)c(F)n1 N1(C(CC(=O)NCC2(F)CC(NC(=O)CC3CCOCC3)C2)=O)CCCCC1 C1(SCC(=O)NC2(CCO)CN(C(=O)C(F)CC3CCC3)C2)CCS(=O)(=O)C1 C12CC(C1(C)C)OC2=O.c1(C(=O)COC(CC)=O)cn(C2CCC2)nn1 C1(C(=O)NCCCC2(NC(C(F)=C(C)C)=O)CC2)CC2(C1)CC1(CC1)C2 C1(CC#C)(C(=O)N(C)CCSC)CCN(C(C2C3CCCCC23)=O)C1 Cc1nn(-c2ccc(F)cc2)c2ncc(C(=O)N(C(C(=O)O)C(C)C)C(C)C)cc12 CC(C1CCCCC1)=CC(N1CC2(CC(NC(=O)C(C)N3CCC3)C2)C1)=O C1(C(N2C(CCCNC(CCCC=C)=O)CCCC2)=O)CCC2(CC1)CC2 C12(C(N3CCC(COC)(NC(c4cnn(C)n4)=O)C3)=O)CCC(CO)(CC1)CC2 C=C1COCCN(C(C2COCC2NC(C2CCCN(C)C2)=O)=O)C1 Cc1nn(CC(N2CC(C3(NC(C4CC(N(C)C)C4)=O)CC3)C2)=O)c(C)c1C c1(CC=C)ccccc1C(=O)NC(C(=O)NCc1ccnc(F)c1)C1CCCC1 Cn1cccc(C2CCN(C(=O)OC(C)(C)C)C2)c1=O.c12cc(=O)n([nH]1)C2 Cc1nc([N+](=O)[O-])cn1CCC(N1CCCC(C)(NC(=O)CCC2CC2C)C1)=O N1(C(C(=O)NCCn2c(C)cc(C)n2)C)CCC(C)C(Cc2ccccc2)C1 C(=O)(NN=c1cc[nH]c2ccccc12)NC1C(c2n(C)ncc2)OCCC1 c1(C(=O)NC2C(CNC(=O)CC3CCOCC3)CCCC2)cc2n(n1)CCO2 C1(CC)(CC)CC(NC(C2CC(C)CC(=O)N2)=O)CN1C(=O)CC1CC=CC1 N1(C(C2C(C(N)=O)CC2)=O)CCCN(S(N)(=O)=O)CC1 c1(CCCNC(=O)CO)ccccc1.CN1CC(C(=O)NCCCNC(C=CC#N)=O)C1 C1(C(=O)NCCN(CC(C)O)C(c2ocnc2C2CC2)=O)CC2(CCC2=O)C1 C1(NC(c2ccc(OCC#C)cc2)=O)CN(C(=O)Cc2cccnc2)CCC1F N1(C(c2c(CNC(C(CSC)O)=O)ocn2)=O)CC(O)(C2CC2)C1 C12(COC(C(c3ccccc3F)(C)F)=O)C(=O)C3CC1C2C3 c1(CC)cc(C(=O)NCc2nocc2C(=O)N(C2CCCCC2)C(C)CO)n[nH]1 N1(C(C(C)CS(C)=O)=O)CCC2(CC1)CN(C(=O)CSCc1ncc[nH]1)CCO2 C1(N(C2CCCC3CC23)C(C2CCC(OCCO)CC2)=O)CCC2(CC1)CNC2 c1(-c2cn(C3CC(C(N4CCCC(CC)C4)=O)C3)nn2)cc(O)ccc1Cl N1(C(C2N(C(CCC)=O)CCC2)=O)CCC(C)(C)C1CNC(=O)C(CC)C(C)C N1(C(c2cc(C(C)C)on2)=O)CCN(C(C)=O)C(c2ccncc2)C1 N1(C(C(C=C)(C)O)=O)CC=C(CCNC(C2CCCCC2C2CC2)=O)CC1 C1(C)(C(=O)NC(C)C(C)NC(c2ccsc2)=O)CCCN(C(=O)CN(C)C)C1 N1(C(C(CSC)OC)=O)CCCCC1C(=O)NC(C)C N#Cc1ccc(O)c(NC(C2CCC(n3cc(CN4CCCC4)nn3)C2)=O)c1 N1(C(CCc2n(C)ncn2)=O)CCC(F)C(NC(C2CCC3(CC2)CC3)=O)C1 C1(CN(C)C)C(=O)N1.C1CC(=O)N1.C(C(C)SC)NC(=O)NC Cc1cc(C(=O)NCCNC(=O)CCN(CC(F)(F)F)C)n2ncc(C#N)c2n1 c1(C(=O)NCC(CN(C(=O)COC2CCC2)C)(C)C)cc2cc[nH]c(=O)c2s1 c1(OC(C)C(N2CCC(NC(c3c[nH]c(Br)c3)=O)C2)=O)ccccc1F C1(C(=O)NC(C)CCN(C)C)(NC(c2n[nH]cc2Cl)=O)CC(F)(F)C1 N1(CCC(C)(C)C(=O)N2CCC(NC(=O)C(F)(F)F)CC2)Cc2ccccc2C1 c1(C(C(=O)NCCC(C)N(C(C(F)=CCC)=O)C)N(C)CC)ccccc1 CN(C1CCc2c(F)cccc21)C(C1(c2ccc(N(C)C)cc2)CCCO1)=O Cc1onc(CC(N2CCN(C(=O)C=C3CCCCC3)C(C)C2)=O)c1C#N N1(C(CC(C(C)OC)NC(C2CC=CC2)=O)=O)CC2(CCOC2=O)C1 c1(OCC)ncc(C(=O)N(C2CCN(C(=O)CC3(OC)CCC3)CC2)CC)cn1 CCCC(C)CC(=O)NCc1cn(CC2CN(C(C3CN(C)C(=O)N3)=O)C2)nn1 c1(OCc2cn(C(C)C)nn2)cccc(C(N)=O)c1.c12cc(ncn1)CNC2=O c1(C(=O)NCC2(COC)CN(C(C(CCC)C)=O)C2)ccc2cnccc2c1 C1(OC(=O)NCCC2(C(C)OC)CC2)CC(C)N(C(=O)C(C)C2CCCC2)C1.N c1(C(N2CCCN(C(COCCOC)=O)CC2C)=O)ccc2c(c1)OCC(=O)N2 c1(C(=O)NC2CC3(C(NC(=O)CN4CCCC4=O)C3)C2)ccc(Cl)cc1F N1(C(CCCC2C(C)C2)=O)CC2CC(C1)CN(C(=O)CC(C)(C)O)C2 c1(CC)cccc(C(N2CC(Cc3cnn(-c4ccccc4)c3)C2)=O)c1F C1(CC#C)(C(=O)NC(c2cnccc2C)C)CCN(C(=O)C(C)C2(O)CCC2)C1 N1(C(C23CN(C(=O)CC4(O)CCOCC4)C(C2)CO3)=O)CCn2c(O)nnc2C1 C=C=CCCC(=O)NCc1nc(C(=O)NC(C2(O)CCCC2)(C)C)co1 c1(C(=O)NC2C(C(N3CCC(C)(C)C3)=O)CCC2)ccc2occc2c1 C1(C(N(C)CC2(O)CCOC2)=O)CC(NC(C2CCCSC2)=O)C(O)C1 N12CCC(CC1)N(CCO)C(=O)C2.CC1CC(CO)N1C(=O)C(=O)NC(C)C N1(C(CC2CC(NC(CC3C(C)CCC3)=O)C2)=O)CCOC2CCCC12 C1(C(N(CC#C)CC=C)=O)CCC2(CC2)N1C(=O)CC1C(=O)NN=C1C CC(C(C)C(=O)NCCCCN(C)C(c1nn(C)c2c1CCC2)=O)C(C)(C)C N#Cc1ccc(C(N2CCC(CNC(=O)C(F)(F)CC3CC3)C2)=O)cc1O c1(C(=O)NCCCC2(NC(c3cc(C(N)=O)oc3)=O)CC2)cccc2sncc12 Cc1ccc(CNC(=O)C(Cn2cccn2)NC(c2ccc(CO)s2)=O)cc1 c1(NC(C23CC2CN(C(c2ccc(O)cn2)=O)C3)=O)cnc(O)nc1O C1(NC(Cc2cc(C)sc2)=O)CN(C(C2(C(C)(F)F)CCOCC2)=O)CCC1F N1(C(c2c(C)cno2)=O)CC2CC1CC2NC(c1cc(Br)ccc1C)=O C=CCCCC(C(=O)N(C)CC)NC(c1cc(CC)no1)=O.C1(CC)(OC)CCCC1 S(=O)(=O)(c1ccc(I)cc1)N1C(C(=O)N(c2c(Cl)cc(Cl)cc2I)C2CC2)CCC1 c1(OC)cccc(CCC#N)c1.C1(C2CC2)C(=O)OC2CC(C2)C(=O)N1 N1(C(C)=O)CCC(C)(c2cn(CC(=O)NOC3CCN(CCO)CC3)nn2)C1 N1(C(C(C)CN(C)C(N2CCOCC2)=O)=O)CCC(CF)(CO)C1 C1(c2n(C)ccn2)CN(C(c2ccc(Cl)o2)=O)CCN1C(=O)C1=C(Cl)CCC1 C(=O)(C1Cc2ccccc21)N1CC2C(CNC(c3c(C)nn(CC)c3Cl)=O)C2C1 C1(CC(N2CC(N(C(CCc3n(CC)ccn3)=O)C)C2)=O)CCCCN1C C=CC1CN(C(=O)CCc2cn(C)nn2)CC1NC(=O)CN(C(=O)COC)C CC1(C)CCCCC1C(=O)NCC1CN(C(c2cnsn2)=O)CC(C(F)(F)F)O1 C1(CCNC(c2ncn(CC)n2)=O)CCN(C(c2c[nH]nc2C(C)(C)C)=O)CC1 C1(C(=O)NC2(CNC(CC3C(CC)C3)=O)CCC2)CCC(C)CC1 Cc1ccc2ncccc2c1NC(C1(CNC(C2CC2(C)C)=O)CC1)=O CC1(C(=O)NCC(F)CNC(C2(C(F)F)CCCCC2)=O)CCCCC1 C12(C(N3C4CCC3CC4)=O)CCCN(CC1)C2.C123CC(C1)(C2)C(=O)N3 N1(C(CC2(CC)CC2)=O)CC2(CO)CC1(C(N1CCC(OC(C)=O)C1)=O)C2 N1(Cc2ncc(OCCOC)[nH]2)CC(NC(=O)Nc2ccccc2)CCC1=O c1(CCNC(C(C)N(C(C(C)C)=O)C)=O)cn(C)cn1 C(=O)(C(C)(C)C(O)C(C)C)N1CCCC(N(C(=O)C(=O)C(C)C)CC)C1 CC1=C(C)CC(C(=O)N(C)CC2CCCN2c2nc(C(F)F)nc(=N)[nH]2)CC1 C1(CC)CN(Cc2ccc(OCCNC)cc2Br)CCN1C(C1(C)CCCN1)=O C12(CN)COC(C1)C(NC(=O)Cc1cn(C3CC3)nn1)C2 C1(OC)(CNCC2CCCCC2c2cccc(Br)c2)CCCCCCC1 c1(NC(C2C3(CCN(C(c4cc(C(C)C)on4)=O)C3)C2)=O)ccc(Br)cc1C#N O=C(C(CC=CCl)c1ccccc1)NC1CCN(C(c2cnc[nH]2)=O)CC1O C1(N(C(C(F)=CCC)=O)CC)CCCN(C(=O)CCc2nc(C)cs2)C1 CC1(C)CN(C(c2c[nH]nc2Cc2ccccc2)=O)CCC1CC(N)=O c1(C(N(C(C)C(N2CCC(CO)C2)=O)C2CC2)=O)cccc(O)c1F c1(C(N2C3CN(C(C(CCCOC)C)=O)C(CC3)C2)=O)coc2c1C(=O)CCC2 C(=O)(C1CCCc2ncnn21)N1CCC(NC(c2onc(C)c2C)=O)C(C)(C)C1 C1(C(N(CC=C)CC2CC2)=O)CCC(C)CN1C(=O)C=CC(=O)OCC c1(OC(C)C)ccc(C(=O)NCCCC(C)(C)NC(C2CC2(C)C)=O)cc1N C1(CNC(CCN(C(c2ccc(C)cc2)=O)C)=O)COc2ccccc2O1 C(CCCCC(=O)NCC1CC2(C1)CN(C(=O)C(C(C)C)SCC)C2)OCC c1(C(N(C)CC2(NC(c3c(CC)nn(C)c3)=O)CC2)=O)ccc(C)c(C)c1 C1(CNC(C2C(c3ccc(N)cc3)OCCC2)=O)(CO)COCC2COCCN12 N1(C(c2cnc(CNC(C(C=C)(C)CC)=O)nc2)=O)CC2OC(=O)N(C)C2C1 c1(C(C(=O)NC(C)CCNC(=O)CCN2CCOC2=O)(C)C)cccc(F)c1Cl c1(CC)cscc1C(=O)NCC(O)CNC(C1CC(C(F)F)(OC)C1)=O c1(OC)cc(O)ncc1C(=O)N(C(CCNC1CCC1)C(C)C)CC(C)C c1(CC)cc(C(=O)NCC2(COC)CCN(C(C3CC(C)CO3)=O)C2)n(C)n1 c1(C(N2CC(C(N(CCCF)CC)=O)C(C)(C)C2)=O)cccn2nccc12 N1(C(C(C)Sc2ccccn2)=O)CCCC2C1CCN2C(C1(C)COC1)=O CC1(CNC(C2CCS(=O)(=O)C2)=O)CCCN(C(C2CC3CC2C3)=O)C1 C1(C(=O)NCCOCC(=O)NCCCOCC#C)CCCC1CC C(C)(CCC(=O)N1CC(CO)(NC(=O)C(CC)Nc2cccnc2Cl)C1)OCC c1(C(N2C(C)CC(CNC(c3cscn3)=O)C2)=O)ncnc2c1CCCC2 c1(C(=O)NC2CC3(CC(CNC(C(C)=C(CC)C)=O)C3)C2)ccc(S(N)(=O)=O)o1 c1(C(=O)NCC2(O)CCN(C(CSC)=O)C2)ccc(Br)cc1F c1(N2CCCC(CCNC(C(CO)NC(N)=O)=O)C2)ncc(Br)cc1C#N c1(C(=O)NC2CC(CCNC(C(CSC)(C)C)=O)C2)ccc(F)cc1Cl C1(C(=O)NCC(C)CNC(=O)CCC(=O)c2cccs2)CNC(=O)CC1C c1(OCC)nc2ccc(C(=O)NCCNC(c3sc(Cl)cc3Cl)=O)cc2[nH]1 Cc1sccc1CC(N1CCC(CC(C)(C)C)C1)=O.C1CCCN1c1ncns1 c1(C(C(=O)NC2CCC2)N(C2CC3CCC2O3)C)cncc(Br)c1 c1(CC(=O)NC2(C)CCN(CCc3ccc(OC)cc3)C2)cc(C)cc(F)c1 C(=O)(C1=CCCCCC1)NC1(CN2CCN(C(C3(C)CCC(C)C3)=O)CC2)CC1 c1(C(=O)NC2(CC=C)CN(C(=O)C(C)(O)C=C)C2)cc(Cl)c2ccccc2n1 c1(COCC(=O)NCC2C=CC(NC(=O)COC3CC3)C2)ccccc1Br C1(CNC(c2c(COC)noc2)=O)CN(C(C2CC(C)(C)C2)=O)CCCO1 c1(C(=O)NCC2CCC(NC(c3cnc(SC)[nH]3)=O)CC2)c[nH]cc(F)c1=O c1(COC)c(C(N2CCCC2C)=O)oc2ccccc12 CC1(NC(c2cccc(Cl)c2)=O)CCCN(C(c2cnsc2)=O)C1 C1(CC)CCN(C(c2cnc(O)o2)=O)C1C(=O)N(C)Cc1cnc(C)s1 c1(CC)cccc(C(N2CC(OCCNC(=O)CSc3cccc(C)c3)C2)=O)c1 C(=O)(C1=C2CCCN=C2NN1)N(CCNC(c1c(C)nc(C2CC2)o1)=O)C(C)C C1(C(=O)NCCc2ccc(C)s2)(NC(c2cnn(C3CC3)c2)=O)CCCC1C N1(CCNC(=O)C(N2CCN(Cc3ccc(Cl)cc3)CC2)=O)CSCCSC1 C(=O)(CC1=CCOCC1)NCC(CC)NC(=O)C(CO)c1ccccc1 N1(C(C(C(CC)C)O)=O)CCC2(CC1)CCN(C(=O)C(C)NC(N)=O)CC2 N#CC1(C(=O)NCC2CCC2NC(C2CC(n3cnnc3)C2)=O)CC=CC1 C1(NC(c2c(CC)nn(C)c2)=O)COC2(C1)CN(C(=O)CS(=O)CC)C2 CC#CC1CN(C(=O)C(C)(C)CN(C(=O)CCOCC2CC2)C)C1 C1(C(F)(F)F)(OCC)CC(C(=O)NCC(C)NC(=O)C(O)Cc2ccccc2)C1 c1(C(N2CC(C(C)NC(=O)CSC(F)F)C2)=O)cnn(-c2ccccn2)c1 c1(C2(C)COC2)nocc1C(N1CCCC1CNC(c1sccc1C1CC1)=O)=O N1(C(C2CN(CC)C(=O)C2)=O)CCOC2(CCN(C(=O)CCC3CCCO3)C2)C1 C1(O)(CNC(c2ccnc(O)c2)=O)CCCN(C(c2[nH]nnc2C2CC2)=O)C1 C1(C(N(C)CCn2ccnc2)=O)CCC(NC(=O)C(=O)C2CC2)C1 c1(C(=O)NCC2CC(SC)C2)ccc(F)c(OC)c1.C1(C)(OC(=O)N)CCCC1 C1(NC(c2cnc(C)n2C)=O)CCN(C(C2CC2C2CC2)=O)CC(C)(C)C1 C(=O)(C(O)C(C)(C)C)NCc1ccc(N2CCN(C(C(CC)O)=O)CC2)nc1 CC1CCN(C(=O)CCCCN(CC(N)=O)C)CC1NC(=O)Cc1cnsc1 N1(C(c2ccn(C(C)C)n2)=O)CCC2(CCCN(C(=O)CCCF)C2)C1 C1(CNC(c2cnsn2)=O)CCC2(CCC2)CN1C(=O)C=C(C1CC1)C1CC1 N1(C(CC2N(C(c3cc(CC)ncc3)=O)CCOC2)=O)CCS(=O)CC1C C#Cc1cccc(C(=O)NCCCC(c2ccccc2)NC(=O)C(C)S(N)(=O)=O)c1 C1(C(=O)NC2CCC(Nc3c(C)c(Cl)ncn3)CC2)CC2CCCCCCC12 C(C(C(C)C(C)C)NC(=O)C=CCN1CCCC1)NC(CCSCCCC)=O c1(-c2ccn(C(C)C)n2)nc(-c2ccc(C(F)(F)F)cn2)nn1CCCC(F)F CC1CCCC(c2cn(CC3CN(C(=O)CN4CCCNC4=O)C(C)C3)nn2)CC1 CCCCN=C(NCc1coc2ccccc12)NCC1(CO)COCCN1C C1(O)(CNC(c2cnco2)=O)CCN(C(=O)COCCc2cccs2)C1 c1(OC)cc(C(N2CCN(C(=O)C(C)O)CC2CO)=O)c(N)cc1F N1(C(=O)CC2CCNC3(CC3)C2)CCc2ccc(Br)cc2C1 c1(SCC(=O)NC(C(CO)NC(C2(C#C)CCC2)=O)C)ccc(C)c(C)c1 C1(NC(C(CC)C)=O)CC2(CCCN(C(c3nc(Cl)c(Cl)s3)=O)C2)C1 c1(OC)cc(CN(C)Cc2cc(-c3ccccc3C)cn(C)c2=O)ccc1OC n1(CC(=O)N(C2CCC(Oc3ccc(F)cc3)CC2)C2CC2)ncc2ccccc12 c1(C(N2CCC(OCCNC(=O)CCCC(F)F)C2)=O)scc2c1OCCO2 c1(C(N2CC3CC(C2)N(C(C2CNC(=O)C2)=O)C3)=O)ccc2snnc2c1 c1(C(N(C)CCC2CCCCN2C(c2ccsc2)=O)=O)cccc(C#N)c1 N1(C(C2(COCC)CC2)=O)CCC2(CC1)CC(C(N1CC3CC3C1C#N)=O)CO2 N1(C(c2csc(Cl)c2)=O)CCCC2(NC(C3(c4cccs4)CC3)=O)CCCC12 N1(C(c2nc(CC)oc2)=O)CCCCCC1CNC(C1CC=CCC1C)=O C1(CC)CN(C(C2(C)CCC(=O)N2)=O)CC1C(=O)NCc1cncn1CC C1(c2ccccc2)(CNC(N(C2CC2)CC)=O)CCOC1 c1(C(N(C2CCN(C(CC(CC)CN(C)C)=O)CC2)C)=O)nsc2ccccc12 C1(CNC(C(C)NS(C)(=O)=O)=O)CCN(C(=O)CC2CC2CC(C)(C)C)C1C c1(C(N2CCCC(CNC(C3C(C)C3)=O)CC2)=O)c(Br)ccc(N)c1F N1(c2snc(C)n2)CCC2(CCCN(C(c3ccc4c(c3)C(C)(C)C4)=O)C2)C1 n1(CC)nc(C(N2CCOC(C(=O)Oc3snc(C(N)=O)c3C#N)C2)=O)cc1C C(=O)(C1=CC2(CCN(C(=O)C3=CCCOC3)C2)C1)N(CC(C)N(C(C)=O)C)C N#Cc1ccc(OCc2sccc2C(=O)O)cc1.C12CC(C1)NC(=O)C2 N1(C(c2c(CC)ocn2)=O)CCC(OCC2CCN(C(=O)C(F)(F)CO)C2)CC1 C1(COC)CN(C(c2ncc(OC)cn2)=O)CCN1C(c1cc(F)cs1)=O C(=O)(C(F)(COC)C(=O)NCC1(CNC(c2cnc(OC)s2)=O)CC1)OC.C1CC1 CC1(CCO)CCN(c2cc(NCC3CC3Cl)ncn2)C1 C#Cc1c[nH]nc1C(N1CC(NC(C2CCC23CCC3)=O)CC1CO)=O CCC(C)C1CCC1.N(COC1CCC1)CCC CC(C)S(=O)(=O)C(C)C(=O)NC1CCC1NC(C1([SH]=CCN2CCCCC2)CC1)=O N1(C(CCCCC=C)=O)CC2CCCCC2(NC(C23CCC(C)(C2)OC3)=O)C1 N1(C(C=CC)=O)CCC(NC(c2cccc(Cl)c2)=O)C(CC)C1 N1(C(COCc2ccc(OC)cc2)=O)CC(NC(C2(O)COC2)=O)CC(O)C1 c1(C(=O)NCC2CCN(C(C3C(C)C(=O)C3)=O)CC2)cc(F)ccc1O C123CCC(CC1)(CC2)C(=O)N3.c1(C(COC(C)(C)C)=O)cc(F)c(O)cc1Br c1(C(=O)NCCC(C)N(C(=O)Cn2cnc(Br)n2)C)cc(N)nc(Cl)c1 C1(NC(CCCC=C)=O)CC2(CCCN(C(c3cc(C)ncc3C)=O)C2)C1 N1(C(C2(NC(=O)Cc3ccc(F)cc3)CCN(C)C2)=O)CC(C2(C)CC2)C1 C1(C(=O)NCC2C(NC(CC3(C)CCC3)=O)CCC2)CCC2(CCC2)CC1 c1(CC)nc(Cl)c(F)c(=NC(C)CNC(=O)C(C)C(C)C)[nH]1 C(=O)(C(F)(CNC(=O)CC(C1CC1)C1CC1)C(C)C)N1CC(OC)C(OC)C1 C1(C(CC)NC(=O)NC(c2cccc(OC(F)(F)F)c2)C)CCC(F)(F)CC1 C(=O)(C(C(F)(F)F)OC1CCN(S(=O)(=O)CCc2sccc2Br)C1)OCC N1(C(C)=O)CC(C)CN(C(=O)C(F)=CC2CC2)C(C)C1 C12(C(=O)NC3CN(C(c4ccn(C)c4)=O)CC(F)C3)C3C4C1C1C2C3C41C(N)=O c1(C(N2CCC(COC)C2)=O)ccc(-n2cc(CCC(C)(C)O)nn2)cc1 S(=O)(=O)(c1cccc2c1OCO2)NC1NC(=O)CSC1 C1(OC)CC(C(=O)NOCC(F)(F)F)CCN1C(=O)CSCCN(CC)CC C1(N)CN(C)CCO1.C(CCC(=O)C)OC.C12(CCCO1)C(=O)OC2=O.C12CC1NC2 N1(C(CCSCCC)=O)CCCC(C(C)NC(C2CC(=O)N(C(C)(C)C)C2)=O)C1 C(=O)(C1=CCS(=O)(=O)C1)N1CC(CCC)N(C(c2cc(C(F)F)nn2C)=O)CC1 c1(C(N(C2CCCN(C(c3cc(C)n(C)n3)=O)C2)CC)=O)cc(Cl)c(F)cc1C c1(C(=O)NC2C(C)CCN(C(c3cncn(C)c3=O)=O)C2)c(F)ccc(Cl)c1F C1(NC(C2(C)CCOC2)=O)CCC12CN(C(=O)CNC(c1ccccn1)=O)C2 c1(C(=O)NCCN(C(c2cccnc2OC(F)F)=O)CC)ccc(F)c(F)c1 C(=O)(C(O)CC(C)C)NC(CCSC)C(=O)N(C1CCN(C)C1=O)C c1(OC)ncc(C(=O)NC2CC(C)N(C(=O)CNc3cccc(C)c3)C2)c(C)n1 c1(OCCNC(c2ccnc(F)c2I)=O)ccc(Cl)c(Cl)c1 C(CCC1CC1)(C(=O)NCc1cccnn1)NC(C(C)OC1CCCC1)=O c1(CC(=O)NC(c2ccccc2)CC=C)ccc(N2CCCCC2)cc1 CC(C)CCCC(C)C(=O)NC(C(=O)NCC(C)CO)C1CC1 c1(CNC(C(C2(O)CN(C(c3ncn(CC)c3)=O)C2)F)=O)ccc(C)c(O)c1 O(NC(=O)C1=NOC(CNC(C2(CC3CC3)CCC2)=O)C1)CCCN(C)C C(=O)(C1CCCc2scnc21)N1CC(O)(C(C)NC(C2CC(OC)C2)=O)C1 N12CCn3ncc(c3C1)C2.CC1CCCCCC1NC(=O)OC(C)(C)C N1(C(C2(N(C)C)CCC2)=O)CC2CCN(C(c3ccn4ccnc4n3)=O)CC2C1 C1(C)(CC)CCC(C(N2CC(O)(c3cn(Cc4ccc(OCC)s4)nn3)C2)=O)O1 Cc1ccc(F)c(CC(=O)NC2CN(c3ncnc(Cl)c3C)CCC2C)c1 CCC(O)C(C)C(=O)N1CCC(N(CCOC)C(c2cccnc2O)=O)CC1 C1(SC)CCN(C(c2ccc(CNC(c3cccnc3CN)=O)[nH]2)=O)CC1 C(=O)(C1CCc2cc(F)ccc21)NC(C(C(=O)OC)(C)C)C C=CCC(CNC(=O)CC(C)CN(C)C)C(=O)Nc1ccc(OC)nc1C c1(C(=O)NC2CC(NC(c3cccc(OCC)c3)=O)C2)cnc2ncccn12 C(F)(c1ccccc1)=CC(=O)NC1CC(C(C)NC(C2CCC(C(F)(F)F)C2)=O)C1 c1(C(N(CCNC(=O)NC(C)C2CC2)CC2CC2)=O)cc(C(F)(F)F)cc(Cl)c1 C(=O)(C(C)(F)C(C)(C)F)NCC1(NC(Cc2n[nH]c(=NC)s2)=O)CCC1 C1(OCC)COCCC1NC(=O)NCc1ncc(-c2ccccc2C(F)(F)F)cn1 c1(C(N2CCN(C(C(C)CF)=O)C(C3CCC3)C2)=O)ccc(N)c2cnccc12 C1(N(C)C(c2cnc(C3CC3)s2)=O)CN(C(=O)C=CC2CC2)CC1(C)C C1(NC(C2(COC)CC2)=O)CN(C(=O)CCc2ccc(N)cn2)C2(CCC2)C1 C1(C(N(C2CN(C(=O)C(C#N)C3CC3)C2)C)=O)CCS(=O)(=O)N1 O=C(N1CC(n2cc(C3(c4ccccc4F)CC3)nn2)CO1)C1(C2CCC2)CCC1 C1(C(=O)NCC(C)N(C)C)C2CC3C(C2NC(=O)C=CCN2CCC2)C13 C(N=c1cc(F)nc[nH]1)c1c(SC)n(C)nc1 CC(C)CC(=O)NC1(C(=O)NCCCCN(C(=O)CC2CCC2C)C)CC1 c1(-c2cn(C(C)C(=O)N(C)CCN3CCOCC3C)nn2)ccc(O)cc1F CC1CN(C(=O)C(F)OC(F)(F)F)CC1(C)CN(CCc1cnc[nH]1)C(C)=O c1(C(=O)NC(CNC(c2c(C)[nH]nc2Br)=O)(C)C)ccc(Cl)cc1N N1(S(c2cnc(C)n2C)(=O)=O)CC(C(=O)O)CC12CCOCC2 N1(C(CCN(C)C)=O)CC(C2CC2)(C(=O)NCC2CCCC(C)(C)O2)C1 C1(NC(c2cn(-c3ncccn3)cn2)=O)CCN(C(=O)CN2CCSCC2)C1 C1(NC(c2c(C)nsc2)=O)CCCN(C(=O)C(C)(C)C(F)(F)F)CC1F C(CCCCC(=O)N1CC(NC(c2ccc(F)cc2OCC)=O)CC(C)C1)OC c1(C(N2CCC(CNC(CCC=CC)=O)C(C)C2)=O)cc2ccccc2cc1F C1(C(CC)C)CCN(C(=O)CCN(CCO)C(C2CC(=O)CCO2)=O)CC1 Cc1ccc2c(c1)C=C(C(=O)N1CCCC(NC(C3CCCSC3)=O)CC1)CO2 CC(C)CCCCC(=O)NCC1CCCCC1NC(=O)CN1C(=O)CCC1=O C(C)(CCCNCc1cnn(C(C)C)c1C(C)C)(c1nnnn1C)OC C12(C(=O)NC(C(CO)NC(Cc3nc(C)oc3)=O)C)CCC(CC1)C2(C)C N1(S(CC2(C)COC2)(=O)=O)CCCC2C(=O)NCC12 N1(C(C(C)CN(C(=O)Cn2cnc(C#N)n2)C)=O)CC2CC1C1CC21 c1(C(N2CCC(C(=O)NC(C(C)C)CCO)C(O)C2)=O)cc(Br)ccc1[N+](=O)[O-] C(=O)(C(F)(F)C(F)(F)F)N1CCCC(CNC(=O)Cc2cc(F)ccc2Cl)C1 C1(NC(C2CCN(CC(C)C)C2)=O)CN(C(=O)C(C)(C)CF)CCC1(C)C N1(C(C(C)(C)N(C)C)=O)CC(Nc2ccc(N3CC(O)C3)nc2)C(C)(C)C1 C=CC(C)(C)C(=O)N1CCC(CNC(=O)C(C2CCOCC2)F)CC1 C(CCCCC(=O)NCc1nc(CNC(C23CCCCC2C3)=O)cs1)OC N1(C(C2C(C)N(C(=O)CCC(F)(F)F)CC2)=O)C2CCCC1COC2 c1(COC)cccc(C(=O)NCC(C)CN(C)C(c2ccc(C(F)(F)F)s2)=O)c1 C1(NC(C2CCC(C(N3CCC(CN(C)CCO)C3)=O)CC2)=O)NC(=O)OC1C CCCC(CNC(C1CC1C(=O)OC)=O)C(=O)N1CC2(CC(N(C)C)C2)C1 c1(C(=O)NCCN(C2CCCC2)C(c2c(C)con2)=O)c[nH]cc(Br)c1=N C#Cc1ccc(C(=O)N(CCCNC(C2CCC(F)C2)=O)C2CC2)c(C)c1 C1(C(=O)NC2CCN(C3CC3)C2)CN(C(c2ccccc2Cl)=O)CCO1 C1(C(N(C2CCN(C(C3CCC=CCCC3)=O)CC2)C)=O)CCc2ccnn2C1 C1(C(=O)NCC2N(C(=O)CN3CCCCC3)CCN(C)C2)CN2CCCN1CC2 N1(C(c2c(C)c(I)ccc2)=O)CCC2CN(C(C34C5C6C7C5C3C7C46)=O)CCC12 CN1N=C(C(=O)NCC=CCNC(C2CC3CC2CC3O)=O)CCC1=O N1(C(c2nc(C(C)=O)sc2)=O)CCC(C2(NC(c3ccc(C)c(C)n3)=O)CC2)C1 C(C)(C(O)C(=O)NC1CC(F)(CNC(c2cc(C(C)C)nn2C)=O)C1)OC C1(NC(CCc2c(C)n[nH]c2C)=O)CC12CCN(C(c1ccc(F)s1)=O)CC2 N1(C(C2CN(C(c3ccc(C#N)n3C)=O)CC(C)O2)=O)CCn2nccc2C1 C(c1c[nH]c(=N)c(C)c1)=CC(=O)NCC1(F)CC(CNC(C(CC)(C)OC)=O)C1 C1(NC(CSCC(C)C)=O)CC(NC(c2ccncc2N(C)C)=O)C(O)C1 N12CCOC3(C1)CN(C3)C(=O)C=Cc1cc(co1)C2=O.S(=O)(=O)(CC)NCC C1(CNC(C2(CC)CCCCC2)=O)CCN(C(=O)C(F)(F)CO)CC1CC c1(C(N(CCOCCCNC(C2C(C=C)OCC2)=O)C)=O)cnc([N+](=O)[O-])n1C Cc1cc(N)n2ncc(C(=O)NC3CCN(C(=O)CC4CCOC4)C(C)C3)c2n1 C=C1CCC1(C(=O)OC)C(=O)NC(CNC(c1cc(CC)no1)=O)CO c1(C(=O)NC)c(NC(C2CC(C(=O)OC)C2)=O)cnn1-c1ccccc1 CC(C)CC(C)CC(=O)N1CCCCC1CCCNC(=O)CCc1nncn1C C(C(O)CC(=O)NCCCc1ncc[nH]1)NC(c1nc(C)sc1)=O c1(NCC23CCC(NC(C=CC)=O)(CC2)CC3)[nH]c(=O)n(C)c(=O)c1C#N c1(CNC(=O)NC(C(=O)OC)C(C)C)cc2cc(C)c(C)cc2o1 c1(C(=O)NCCC2(C)CCN(C(C3C(CC)C3)=O)C2)c(F)c(F)cc(F)c1F c1(C(N2C(CNC(CC=C)=O)COCC2)=O)[nH]c2ccccc2c1C#N C1(CNC(C2C(CC)C2)=O)COCCN(C(=O)C=Cc2cccs2)C1 c1(-c2cn(CC(CCNC(C3N(N=O)CCC3)=O)F)nn2)ccc(F)c(Cl)c1 n1(CC)nc(C)c(C(=O)NCCC2CCCN(C(c3cnns3)=O)C2)c1Cl N1(C(CCCNC(C)=O)=O)CC2(COC(CNC(=O)CSc3ccc(F)cc3)C2)C1 C=CC(C)(C)CC(=O)NC1CCN(C(=O)CCC23CC(C(=O)OCC)(CO2)C3)C1C C1(CNC(C(C)C2CCC2)=O)CC2(CCN(C(c3c[nH]c(=N)nc3O)=O)C2)CO1 c1(C(=O)NC2C(CC)CN(C(c3c(Cl)cnn3C)=O)CC2)cnn2c1OCCC2 C1(CCC(C)C)CCCN(C(=O)CC2CNCCO2)C1 c1(C(c2n(CCC)nnn2)Nc2cnn(CCO)c2)cc(I)cn1C C12(C(N3C(COC)CCC3)=O)COC(C1)C(NC(=O)C(C)C1CC1)C2 c1(C(N(CC(C)N(C(c2cn(CC)nc2)=O)C)C)=O)c(O)cccc1Cl c1(OC(CC)C(=O)NCC(F)CNC(C2(CCO)CC2)=O)cccc(C)c1 c1(NC(C2CCC(F)C2)=O)ccc2cc(C3CCCCC3)[nH]c2c1 c1(N(C)CC)ccc(C(=O)NC2CCCC2CNC(C2(n3cccn3)CC2)=O)cc1 c1(C(=O)Nc2cncc(C(=O)Nc3ccc(C)cc3)c2)cc2cccc(F)c2s1 C12(CN(C(=O)C(O)Cn3cncn3)C3CCOC3C3CNC3)CCC(CC1)CC2 c1(C(c2nnnn2C(C)C)NCCc2ccnc(OC)n2)c(F)cc(Br)cc1F C1(NC(C2(C)CC=CCO2)=O)CCCCN(C(=O)Cn2cnc(C(F)(F)F)n2)C1 C1(S(C)(=N)=O)(CN(CC(=O)NCc2cccc(O)c2)C)CC1 CCC(CC)C(C(=O)NC1CC=C(C(=O)NCC(C)C(=O)NC)C1)N1CCOCC1 N1(C(CSCC)=O)CCC(NC(=O)C(SC)SC)CC1C c1(C(=O)NC2CC(O)(CNC(C3(C)CC=CC3)=O)C2)ccc(S(C)(=O)=O)s1 CC1OCCOC1C(N1CCC(C)(CC(=O)NCCCCNC(N)=O)C1)=O CC(C)CC(CNC(=O)C(C)C1CCC1)C(=O)N1CCOC(CCO)C1 C1(C(=O)NCCCOCCNC(=O)COc2ccsc2)CCN(C2CCC2)C1 N1(C(C23OCC(C(C)C)(C2)C3)=O)CC(N(C(=O)CCC(F)F)C)C(C)(C)C1 N1(C(Cn2c(C)nnn2)=O)CCCCC1CN(C)C(C12CCC(C1)C2)=O C=CCC(CC(C)C)C(=O)NC(CCC1CC1)C(=O)NCCCN1CCC1 N1(C(CC2CN(C)C2)=O)CC2CC3CC2C1C3NC(c1cn2ncccc2n1)=O c1(C(N2C(C)CCC(CNC(COCCCC)=O)C2)=O)ccc(Cl)c2cccnc12 C#Cc1cc(F)c(C(=O)NC2CC2NC(=O)C(CCSC)OC)c(F)c1 C(=O)(C(C)(C)CC#N)NCC(C(=O)NCC(C)(C)CCO)CC1CC1 CCC(CC)CCCC(=O)NC(CC)CC(=O)NC(c1cnccc1C)C C1(CC(N2C(C(N(C)C)=O)CC2)=O)CCCCC1NC(=O)CC1CCCOCC1 N1(C(C(N2CC(C)C2)C)=O)CC(NC(=O)CSc2nncs2)CC1C CCC(C(=O)NC1CCN(C(=O)CSC2CCOC2=O)CC1)C(C)(C)CC c1(C(=O)N(C(C2CCCSC2)=O)C2CC2)csc(CN(C(C)=O)C)c1 N1(C(c2n(C)ncn2)=O)CC2CC(NC(=O)CC3CCCCCC3(F)F)CC1C2 C1(CC)C(NC(C2CNC(=O)N2)=O)CCN1C(c1c[nH]c(C(=O)NC)c1)=O n1(CC(=O)NCC23CCC(CN2C(=O)C(F)F)C3)ccc2ccccc2c1=O Cc1ccc(CC(=O)NC2CCCC2C(=O)N(C)Cc2cncn2C)o1 C(CCCNC(C)=O)(C(=O)O)NC(=O)Nc1cccc(COC)c1 C1(CNC(=O)C(O)Cc2cnc[nH]2)CC(F)CN1C(=O)CCc1cccc(F)c1 C#CC(CNC(=O)CC1CCN1C(c1c[nH]c(=N)o1)=O)CC Cc1nc(C2CC2)nc(O)c1C(=O)NCC(CC(C)C)NC(=O)CC1CCCO1 c1(CNC(C)Cc2ccc(C#N)cc2)cc(C#N)c(Cl)cn1 C1(NC(c2cc(CNC(Cc3n(C)nnc3)=O)nn2C)=O)CCOC(C)(C)C1 C(CC(=O)NCC(F)CNC(=O)CCOCCNC(=O)OC(C)(C)C)=C(C)C.CCO CC(CNC(c1cccc[n+]1[O-])=O)CC(=O)NCCC(C)(C)CO c1(CNC(c2ncc(OC)nc2)=O)ccc(O)c(OC(C2(C(F)(F)F)CC2)=O)c1 C1(NC(C2CC(=O)OC2)=O)CC2CN(C(=O)CC3(O)CCCOC3)CC12 c1(C(N2CC(c3ccccc3)(NC(C3C(=C)C3)=O)C2)=O)cccc(C)c1 C1(CC(=O)NCC23COC(C(=O)NC4CC(O)C4)(C2)C3)CN2CCC1CC2 C(=O)(C1CNc2ccccc21)NCC1(CCNC(C(c2ccnn2C)C)=O)CC1 C1(NC(=O)CC23CCCC2CCO3)CCN(c2c(OC)cccc2)CC12CCC2 c1(C(N2CCN(C(c3cnc(C(C)=O)s3)=O)C3C2C3)=O)ccc2c(c1C)CCC2 c1(C(N(C2CCC(NC(c3cc(CCC)on3)=O)C2)C)=O)c(C)csc1Cl C1(NC(Cc2ccc(C)s2)=O)COCCC1NC(=O)C1=C(Cl)CC1 C1(c2n(CC(C)CO)nc(C3CSC3)n2)CC12CCCc1ccccc12 CC(C)C(F)(F)CC(=O)NCC1(F)CC(NC(=O)Cc2cn3ccsc3n2)C1 c1(CC)c(C(=O)NCC2CCC(C)N(C(=O)C(C)=C(C)C)C2)cccc1C Cn1nc(C(C(=O)NCC(F)F)N(C2CC2)C(C)C2CC2)c(Br)c1Cl c1(C(=O)NC(C)CC(C)NC(C2CCC(=O)O2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 C(=O)(C1=CN=C2N=CNN2C1)NC1(CO)CN(C(C2CCC(C)O2)=O)C1 c1(C(C)C(N2CCC(NC(=O)CNC(C3CCC3)=O)CC2)=O)ccc(Cl)c(Cl)c1 C1(C(=O)NCCN(C(c2cnc(C(=O)OC)s2)=O)C)Cc2cc(F)cc(F)c2O1 c1(C(=O)NC(C(=O)NC(C=C)C(F)(F)F)CCF)cc(O)cc(F)c1 N1(C(C(C)C)=O)CCC(C(F)(F)F)C(NC(c2ccccc2-n2ccnc2)=O)C1 C12CC(C(O)C1)NC2=O.C1(C)(CC=C)CN(C(=O)C(O)Cn2cncn2)C1 c1(C(N(CCN(C(C2(CC=C)COC2)=O)C)C)=O)cnc2sc(C)cn12 C(=O)(C(C(C)C)C(C)C)NC(C(CC)C)C(=O)N1CC=CC(O)C1 C1(N(C(C)=O)C)CCCC(N(C(=O)C2=CCC2)C)C1 C=CC1CCCN(C(=O)CC2(C)CCN(C(C3CCOC3(C)C)=O)C2)C1 c1(OC)cc(CN(CCCCCCc2ccc(C)cc2)C=O)ccc1Br N1(C(Cc2cc(C)no2)=O)CCC2(NC(=O)C(O)CC(F)(F)F)CCCC12 N1(c2nc(C)cc(CC)n2)CCN(C(C2C(C)(C)C2(C)C)=O)CCC1C CCCCC(C)(F)C(=O)NCC1COCCN(C(c2cc(C)c(C#N)[nH]2)=O)C1 N1(c2ncc(C(=O)OCC)cn2)CCN(C(=O)C(C)=C(C)CC)C(CC)C1 C12CC(C(O)C1O)CN2.n1(CC(C)(C)C)c(C(c2nnnn2C)OCC)cnc1O C#CCCC(O)C(=O)NCC1(NC(=O)C(CSC)c2ccccc2)CC1 C1(NC(CN(C(C(C(C)C)OC)=O)C(C)C)=O)COC2(CCC2)C1 C12(C(N3CC(C)C(NC(c4cc[n+]([O-])cc4)=O)C3)=O)CC(C)(CCO1)C2 N1(C(C2C(CC(C)C)C2)=O)CC(F)(CNC(C2(Cc3cccnc3)CC2)=O)C1 C1(CNC(=O)CC2CC(O)C23CCC3)CCCC2CN(C(=O)C3=COCC3)CC12 Cc1c(C(N2CC(NC(c3cccc(CO)c3)=O)C(O)C2)=O)cncc1N C1(NC(c2cccc(-n3cnnn3)c2)=O)CC2CCC(C1)N2 N1(c2n(CC=C)c(C(C3CCS(=O)(=O)C3)(C)C)nn2)CC2CC(F)(C2)C1 C12(C(N(C(C(=O)NNC(=O)C(C)(C)C)C3CCCO3)C)=O)CCN(CC1)C2 c1(C(N2CC(N(C(C3CN(C(C)=O)C3)=O)C)C(C)(C)C2)=O)cccc(C)c1C#N N1(C(C2(C(N)=O)CC2)=O)CCC(C2CC2)(CNC(c2ccc(C3CC3)o2)=O)C1 C12(CCCCC1)c1nnc(n1CCO)N1CCC(CC1)N2.CC(C)(C)OC(N)=O c1(C(=O)NCC(C(C)(C)C)NC(c2cnn[nH]2)=O)cc(F)ccc1C1CC1 c1(C(=O)NCC(CO)NC(c2cc(CC)ncn2)=O)n[nH]c2ccc(OC)nc12 c1(OC)cc(C(=O)NC(C)CNC(=O)C(C)N(C)C(C)=O)ccc1S(N)(=O)=O c1(C(N2CCCC(F)(CNC(C3C(C)C3)=O)C2)=O)cc2c(OC)cc(Cl)cc2[nH]1 c1(C2CCCN(C(CN(C)Cc3cc(C(F)(F)F)no3)=O)C2)nnc2n1CCCC2 N1(C(c2ccc(F)c(F)c2)C(=O)NC)CCCOCC12CCCC2 C12(NC(CCC(N)=O)=O)CN(C(c3occ4c3CCCC4)=O)CC1CS(=O)(=O)C2 c1(C(C(=O)NC2C(CNC(c3nc(Cl)cs3)=O)CCC2)(F)F)ccc(F)cc1 C1(C#N)(NC(CC#C)=O)CCN(C(=O)CCc2ccc(F)cc2)C1 C#CCC(C)(CC)C(=O)N1CC(CNC(=O)COCC(F)F)C1 c1(C(N2C(CNC(C=CC(CC)=CC)=O)CC2)=O)cnc(CC)s1 c1(C(=O)NCC(F)(F)F)ccc(CNC(CCNC(C2C(C)C2)=O)=O)o1 c1(CC(=O)NC2CCCC(N(C(C(C)=CC)=O)C)C2)coc2c(OC)cccc12 C=CC1(C(=O)NC2CCCCC2CNC(C2CC23CCC3)=O)CCOCC1 c1(C(=O)NCCOCCCN(C(=O)C2=CCOCC2)C)c(N)cc(Cl)nc1Cl c1(OC)sccc1C(=O)N(CCCNC(=O)Cc1csc(C)c1)CC1CCCC1 C1(NC(CC(=C)C)=O)CN(C(=O)C(C)Cn2ccnc2)CC1C C(=O)(C(CNC(=O)C(C#N)CCC)CCC)NCC1CCN(CCC)C1 CC(CCCCNC(c1nn(C)cc1Cl)=O)NC(C1CCC(F)(F)C1)=O CCCCC(=O)N1CSCC1C(=O)N(C)CCNC(C1CC1F)=O c1(C(CCCCNC(C(=O)NCCN(C(CC)C)C)=O)=O)c[nH]c2ccccc12 CCC(CC)C(F)C(=O)N(CCC(C)(C)NC(c1cnncc1C)=O)C C1(C(C)NC(c2cn(CC3CC3)nn2)=O)CCCCN1C(c1cc[nH]n1)=O N1(C(C(C)SCC)=O)CCC(O)(C(C)NC(=O)Cc2cccc(C)c2Cl)CC1 N=c1[nH]cc(CC(N2CCC(NC(c3cnc(C4CCCO4)s3)=O)C2)=O)[nH]1 N1(C(C(CCCOC)C)=O)CCC2CC2(NC(c2cc(C3CC3)on2)=O)CC1 c1(N(C2CCCN2)C(CCC2CCCN(C)C2)=O)ncnc2c1cnn2C C(=O)(CC(C)C(=O)N1CCCCC1C(=O)NCC1CC1C1CCC1)OC c1(C(=O)NCC2CCN(C(C3CC(C#N)C3)=O)C2)cc2cc(F)c(F)cc2[nH]1 C1(C(=O)NCC(CC)N(C)C(c2ccc(CO)cc2)=O)CCC=CCC1 C1(NC(CCc2cc(C)n(C)n2)=O)CN(C(C2CCC(C)(C)C2)=O)CCC1CO C1(NC(C(CN(C)C)O)=O)CCN(C(=O)CCC(=O)N(C)C)CC1O C1(N(C(C(C)SC)=O)CC2CC2)CCCN(C(c2cc(C)c(C)[nH]2)=O)C1 N1(C(c2n(CCC)ncc2)=O)CC2CN(C(=O)CC3CSCCS3)CC2C1 c1(C(=O)NCCC2N(C(C3CC(=C)C3)=O)CCC2)cc(C2CC2)nc(Cl)c1 c1(COC)ccc(-c2cn(CCCNC(c3cc(O)n(C)n3)=O)nn2)cc1 Cc1c(Br)ccc(NC(=O)CC2CN(C(c3cccc(Br)n3)=O)CCO2)c1C N1(C(c2ccc(C(N)=O)[nH]2)=O)CC2CC2(CNC(=O)CCNC(C2CCC2)=O)C1 C1(NC(=O)C(=O)N(C2CC2)Cc2ccccc2F)CCCC(C2CC2)O1 c1(CNC(c2ccccc2N2CCOCC2)C)ccc(N2CCCC2=O)cc1 c1(C2N(C(C3C(C)C(=O)NC3)=O)CCC2)ccc(Cl)c(Cl)c1 c1(CCNC(c2csc(CNC(=O)C(F)OC(F)(F)F)n2)=O)ccncc1F CCCCC(CC(=O)NCC=CBr)NC(C1CCC(=O)NC1)=O c1(SCc2nnc(-c3cc(C(=O)OC)c(C)o3)o2)cc2c([nH]1)CCCC2 N1(C(c2c(NC)cccc2)=O)CC(CNC(=O)CC(C)n2cccc2)C(C)(C)C1 CC1(C)CC(NC(c2sccc2S(N)(=O)=O)=O)CN(C(=O)CCc2ncco2)C1 C1(CNC(CN2CC(C)C2)=O)CC2CCC1N(C(=O)CCc1ccc(O)nc1)C2 CC(C)(C)CC(O)CNC(=O)C(CCC1CC1)NC(=O)CCc1cncs1 c1(OC)cc(C(N2CCC(N(C)C(c3ccccn3)=O)CC2)=O)ccc1Br c1(N2CCCC(C)(F)C2)ccc(S(=O)(=O)N2CCCC2c2ccco2)cc1F N1(C(c2cc(C)[nH]c2)=O)CCCCC1CCC(N1CCC(OCCO)C1)=O N1(C(C=CCCC)=O)CCC(c2cn(CCCC=O)nn2)C1.n1(CC=CCl)cccc1 C1(NC(=O)CCn2cncn2)CN(C(c2sccc2Cl)=O)CCC1O N#Cc1cc(CNCC2CCCN2C2CCCC2)ccc1Cl C1(=CC(=O)NCC2C(C)CCN2C(C2(C)COC2)=O)CCC(C)(C)CC1 c1(C(N2CCC(CC=C)(NC(C3CC34CCOC4)=O)C2)=O)cccn2ccnc12 c1(C(N2CCC(NC(C3(C#C)CC3)=O)(CO)C2)=O)cc(Br)cnc1C N1(C(C2(OC(C)=O)CC2)=O)CC(CCNC(c2ccc(CF)cc2)=O)OC(C)C1 c1(C(=O)NCC2C(CNC(c3c(C)nsc3C)=O)CCC2)ccc(O)c(CO)c1 C1(CC(N2CCCC(N(C)C)C2)=O)CC2(C1)CN(C(C1CCOC(=O)CC1)=O)C2 N1(C(C(n2ccc(C)n2)C)=O)C2CCC1(CNC(c1c(CO)noc1C)=O)CC2 CN(C)S(C)(=O)=NCc1cccc(NC(=O)C(=O)NC2COCC(C)N2)c1 N1(C(C(C2C(CC)C2)OC)=O)CCCC(OCCN(C)C)C1 C(CC(CC)C(=O)NCC1(F)CC(NC(=O)C(C(=O)OC(C)C)OC)C1)=CC.OCC C1(CC)CN(C(=O)C=C(C)C(F)F)CCN1C(=O)COc1cccc(F)c1 N1(C(c2n(CC)ncc2Cl)=O)CC(CO)C2(C1)CN(C(=O)C(C)(O)COC)C2 C(CS(=O)(=O)NC1CC2(CC2)C1)OC(C)(C)C CC1CCCc2ccccc2C1NCCc1ccc(OCc2ccccc2)cc1 Cc1nc2c(F)cccc2c(C(=O)NCC=CCO)c1O C1(N(C(=O)CNc2ccsn2)CC)CCCN(C(=O)C(F)CC2CC2)C1 CC1=CCCN(C(=NCC2CCc3cc(Cl)ccc32)NC2CCS(=O)(=O)C2)C1 c1(C(N2CC3C(NC(C(CC)O)=O)CC(C3)C2)=O)coc2c(C)cccc12 Cc1noc(N)c1C(N1CC(CNC(=O)C(C)CC2CCC2)C(O)C1)=O N1(C(c2c(C)[nH]c(=N)s2)=O)CCC(C)(C)C1CNC(c1ccc(CO)o1)=O CC1CCN(CC(C(=O)NCC2C3CCN2CC3)NC=O)CC1 c1(OC)cccc(C(N2CCC(NC(=O)C(C)CN(C)C)C2C(C)C)=O)c1 C1(F)(CNC(c2ccnnc2)=O)CCC(CNC(C2CCN(C3CC3)C2=O)=O)C1 N=c1[nH]c2ccc(C(=O)NCC3CCCC(NC(C4CC(O)C4)=O)C3)cc2s1 c1(-c2cn(C(C(=O)NC(c3ccc(Br)s3)C)(C)C)nn2)ccc(C#N)cc1F CCC(O)C(C)(C)C(=O)NCC1COCC1NC(c1cnc(OC)cc1C)=O c1(C(C)NC(=O)NCCC(c2nn[nH]n2)C2CC2)cnc(SC2CC2)o1 C#Cc1ccc(F)c(C(=O)NC2CC(F)CN(C(C3CCOC(=O)CC3)=O)C2)c1 c1(OC(C)(C)C(=O)NCCC(N2C3COCC2C3)=O)cccc(C(F)(F)F)c1 C1(C(N2C(CC)CN(C(=O)CCCCC3CC3)CC2)=O)CCC(=C(F)F)CC1 c1(NC(C2C(CC)N(C(=O)Cn3nnnc3C)CC2)=O)ccc(C)c(F)c1 C(C)(CCCCNC(c1n[nH]c(C)c1Br)=O)NC(C(C1CC(F)(F)C1)OC)=O C1(C#N)(C(N2CCC(C)(CCNC(C3CC4(CC4)C3)=O)C2)=O)CC2C=CC1C2 N(C(=NCCC1CCN(C)C1)N1CCC(C)(COC)C1)CCC(=O)OCC c1(-n2cc(-c3c(=N)[nH]cnc3)nn2)nc2cc(F)c(F)cc2[nH]1 n1(C(C)C)cc2c(n1)C(C(=O)NCCCCNC(C1CCS(=O)(=O)CC1)=O)CCC2 Cc1cccn2nc(C(N3CCC3CNC(c3n[nH]cc3[N+](=O)[O-])=O)=O)cc12 c1(OC)ccc(C(=O)NCCCNC(=O)C(C)C2CCC2)c(Cl)c1 CCC(C)C(O)CC(=O)NC1(CCCNC(=O)Cn2ccnc2C)CC1 O=C(C1CCCn2cnnc21)NC1CC2CCC(C1)N2C(=O)C1=CS(=O)CCC1 C(=O)(C#CC1(C)CCCO1)NC(C1N(C(Cc2cccc(OC)n2)=O)CCC1)C CC1N(C(=O)COC2(C)CN(C(=O)C(N3CCCCC3)C)C2)CCCC12CCC2 c1(C(=O)NC(CC)(C)CNC(=O)COC(C)C)ccc(OC)c(F)c1N CCCC(C)CC(=O)N1CC(C(=O)Nc2ccsc2)C2(CC2)C1 c12cc(O)nc(n1)N1CCC(C1)N(CCc1ccccc1)C2.n1(CCC)ccnc1 N1(C(c2c(C)n(C)nc2)=O)CCC(CNC(C2CC2c2cccnc2)=O)C(O)C1 C1(OC)CCC12CC(NC(=O)C(=O)NCC(CSCC(F)F)OC)C2 c1(C(=O)Nc2n[nH]c(C)c2C(N)=O)cn2c(n1)C(=O)CCN2 C1(C(N(C(C2CCOCC2)C)C)=O)CN(C(C2OCCC2(C)C)=O)CC1C1CC1 C1(=CC(=O)NCC2(CNC(=O)Cc3cnns3)CC2)CCSCC1 CC1CN(C(=NCCC2(OC)CCCCC2)NCCS(C)(=O)=O)c2ccccc21.N(C)C C(N=c1cc(C2CC2)nc(Cl)[nH]1)C12CC(NC(CC3C(CC)C3)=O)(C1)C(C)O2 N1(C(CN(CC)CC)=O)CCC(NC(=O)Cn2ccnc2C)CC1 CC(C(=O)N1CC(CN(C(=O)CCc2cn[nH]c2)C2CC2)C1)n1cncn1 C1(OC)CC(S(=O)(=O)NCCCCN(C)C)C1.C1(CO)(OC)CCC1 C(=O)(C(C)(C)CCOC1CCCC1)NC1CC(NC(C=CC(C)NC(N)=O)=O)C1 N12CCCC(C1C)NC1CCN(C1)CC2=O.C(c1ccoc1)=CC(=O)OCC C(=O)(C1CCc2ccccc21)NC1(C(=O)NCCC2(C)CCC2)CCC1 c1(CC)c(N2CC3CC(NC(c4sccc4F)=O)C3C2)ncnc1Cl Cc1cc(C(=O)NC(C2(O)CN(C(c3cn(C4CC4)nn3)=O)C2)C)cc(N)c1 C1(C)(NC(C(C)Oc2ccc(C)cc2)=O)CCCN(C(=O)Cc2ccco2)C1 CCCS(=O)(=O)CC(=O)N1CCC(C)(NC(c2cc(CSC)oc2C)=O)C1 C#CCCCCCC(=O)N1CC2CC(NC(c3cc4ncccc4[nH]3)=O)C(C2)C1 C1(C(=O)NCc2c(C)n(C)nn2)CCN(C(c2ncncc2Cl)=O)CCO1 Cn1c([N+](=O)[O-])cnc1C(=O)NCC1CC(NC(=O)Cc2csc(C(F)F)n2)C1 C(=O)(C1=COCCO1)NCC(CC)(C)NC(C1CCN(C)C(=O)C1)=O c1(C(N2C(CNC(C3CC4C=CC3C4)=O)C(O)C(O)C2)=O)cccc2scnc12 c1(C(=O)NC(CNC(CN(C)C2CC2)=O)C2CC2)cccc2[nH]nc(O)c12 N1(C(CCCc2ccc(C)s2)=O)CCC(C)C1CNC(=O)CN(C)C c1(COC)nc2n(n1)CCCC2NC(=O)Nc1ccc(-c2ccc(O)nn2)cc1 C1(C(=O)NCC(=O)N(C)C)CCCC12CCN(Cc1cc(Br)cc(F)c1O)C2 C1(C(=O)NCC(N2CCC(CN)C2)=O)CCCCN1CCO.c1(C)ncccc1Cl c1(C(N2CCN(C(=O)CC3CCC3)C3C2C3)=O)cc2cc(F)ccc2[nH]1 c1(NC(CC2OCCN(C(C(n3ccc(C)n3)C)=O)C2)=O)cnc(O)cc1C CS(=O)(=O)c1ccc(-c2ncsc2C(=O)Nc2cccc3ccnn23)cn1 C1(NC(Cc2ccc(C)cc2)=O)CC12CCN(C(=O)C(O)C1CCC1)CC2 Cc1cc(C(=O)NC(C)(C)C(C)NC(=O)C(c2cc(F)cc(F)c2)C)cc(C)n1 N1(C(C(COC)(C)O)=O)CCN(C(c2ccoc2Br)=O)C(CC(F)(F)F)C1 C1(NC(CCCOC(C)=O)=O)CCC2(CC1)CN(C(C1CCCCC1C)=O)C2 C(c1ccc2ncccc2c1)=CC(N1C2CCC(NC(C3CC(O)C3)=O)(C2)C1)=O CCC(CC)C(=O)NCC(=O)NCC1(NC(C2C(C#N)C2(C)C)=O)CCOC1 N1(CC(=O)Nc2c3ncn(CC)c3nc(Cl)n2)CCC(S(=O)(=O)C(C)C)CC1 c1(NCCc2ncc(C)c(CC)c2C)cc(=NC(C)c2cnsc2)[nH]c(C)n1 C(CC(CC)C(=O)N1CCCC1(C(N1CC(S(C)(=O)=O)C1)=O)CC)=CC C1(CNC(C(C)OCC#C)=O)CC2COCC2N1C(C1CCC(=O)C1)=O C(=O)(CC(C)C1CC1)N(CCC(=O)NC(C#C)C1CC1)CC1CC1 Oc1[nH]c(=NCC2CCC=CO2)nc(N2CCC(C3CC3)C2)c1Cl C12(C(N(C)CC3N(C(CC4C(C)C4(F)F)=O)CCCC3)=O)CCC(O)(CC1)CC2 S(=O)(=O)(c1c(O)cc(Cl)cc1Cl)NCC(=O)Nc1ccc(OCC2CC2)cc1 CCCC(CC)C(=O)N1CCN(C(c2coc(Cn3cccn3)c2)=O)C(CC)C1 c1(NC(C2(C)CC23CC3)=O)cccc(Cl)c1 N1(C(C2C3CN(C(c4c(C)oc(CO)c4)=O)C2C3)=O)CCCC(N=[N+]=[N-])C1 N1(C(c2ccc(CC)c(C#N)c2)=O)CCC2(CC1)CC(C)N(C(C1CC1C)=O)C2 c1(N(C)Cc2cccc(F)c2)cc(S(=O)(=O)N(C2(CO)CC2)C)ccc1C#N CN1CCC(C2(C(=O)NC3C4CC3N(C(C3CCC(=O)O3)=O)C4)CC2)CC1 N1(C(COC(C)C)=O)CCN(C(C23CC(F)C2C3)=O)C(c2cc(F)ccc2F)C1 c1(C(N2CCC(NC(CCC#C)=O)C2(C)C)=O)ccc2c(c1)OCCO2 N1(C(C2ON=C(CC)C2)=O)CC2(CCC2)CC1C(N1CC2(CCC(=O)O2)C1)=O C#CCCC(O)C(=O)NC(C)CN(C)C(C1CN2CCC1CC2)=O CC1CN(C(c2cccnn2)C(=O)NC2CCCC2)CCCO1 CC1CCC(NC(=O)CN2C(=O)CNC2=O)CN1C(c1cccc(C2CC2)c1)=O CCC(CC)CC(F)C(=O)NCC1CC(C)N(C(=O)C(C2CCOCC2)=O)C1 c1(C(N(C)CC2CN(C(=O)Cc3ccon3)C2)=O)cc2ccc(Br)cc2s1 C1(N(C)C(c2cc(C(N)=O)co2)=O)CCCC(NC(C2(C)CC2(F)F)=O)C1 CC1CCCC=C1C(=O)N1CCC(C)(NC(c2cc(CO)[nH]n2)=O)C1 c1(OC(C)=O)ccc(C(n2cc(-c3cnn(CCCOC4CC4)c3)nn2)C)cc1 C1(NC(=O)Cc2cc(Br)cs2)CCN(Cc2cncnc2)CC1F c1(NCc2c(CC)noc2CC)nccc(=NCCC2COCCO2)[nH]1 c1(C(N2CC(SC)C(O)C2)C(=O)NC(C(=O)OC)C)ccc(I)cc1 CC1CC2CN(C(C3CCCS3)=O)CC2N1C(=O)CCc1ccc[nH]1 c1(OC)ccc(C(F)(F)CNC(=O)N(C)Cc2nnc(-c3cccs3)o2)nc1 C1(OC)(CNC(C2CC(n3cnnc3)C2)=O)CN(C(=O)CC2CCCC2O)C1 C1(CC(=O)NCCCOCCN(C)C(c2ccc(C(F)(F)F)o2)=O)CCC(O)C1 N#CC1(C(=O)NCc2nc(CNC(=O)CC3CC=CCC3)cs2)CCCOC1 c1(C(=O)NC(C)CNC(=O)C=CC2(C)COC2)cc([N+](=O)[O-])c(N(C)C)cc1F N1(C(c2c(C)cncc2)=O)C2CCC1CC(NC(C1(C)CSC1)=O)C2 O=C(CN=c1ccnc(N2CC3CCOC3C2)[nH]1)N=S1(=O)CCCCC1 N1(C(C(C)n2cccn2)=O)CCCCC2(C1)CN(C(=O)C(F)F)C2 CCCC(C(=O)NC1CC(CNC(=O)Cc2cc(CC)nn2C)C1)NC(C)=O C1(C(=O)NC(C2CCCC2)CNC(c2cc(OC)n[nH]2)=O)CC(C)(C)OC1(C)C N1(C(C(=O)NC(C)C)c2ncco2)CCC2(CCN(C)C2=O)C1 CC1CCCC(n2cc(CNC(=O)CNC(=O)CN3CC=CC3)nn2)C1 C1(CNC(CCC(=C)C)=O)CC2(CCN(C(=O)Cc3cc(Cl)sc3Cl)C2)CO1 N1(C(C#C)C)CCN(C(C2(CC=C)CN(C(=O)CC3C(=O)NN=C3C)C2)=O)CC1 C#CC1(O)CCN(C(C2(CC=C)CN(C(=O)CSC(F)(F)F)C2)=O)CC1 c1(CCC)cc(C(=O)N(C2CCN(C(=O)C(C)CF)C2)CCO)nn1C C(=O)(CCP(C)(C)=O)NCC1C(C(=O)NC(c2c(C)cccc2)C)OCC1 Cc1ccc(F)c(CC(=O)NCC2(C(N3CCOC(CC4CC4)C3)=O)CC2)c1 CCC(C)C(C(=O)NCc1cc(COC)no1)N(C)C(c1ccccc1C)=O N1(C(C2(F)CCN(C(C=CCOC)=O)CC2)=O)CCCCC(C)(C)C1 N1(C(c2ccc(Br)nc2)C(=O)NCc2cccc(OC)c2)CCCC1C1OCCO1 CC1ON=C(c2nc3c(s2)CCN(C(c2ccc(Cl)o2)=O)C3)CC1=O C1(CNC(=O)CCN2CCC(F)C2)CCCC2(CN(C(=O)CCC3CC3)C2)O1 c1(CC)nc(C)c(I)c(=NCC=Cc2ccc3ccccc3c2)[nH]1 N1(C(CCSCCC)=O)CC2(COC(CNC(=O)C(C)n3cccn3)C2)C1 c1(C(=O)NCC2(O)CC(C(=O)NCC3CCCN3C(N)=O)C2)n[nH]c2c1COC2 C(C(CNC(C1CCCC1)=O)C(F)(F)F)NC(=O)Cc1ccns1 c1(C(N2CCN(C(c3nnc(O)cc3O)=O)C(CO)C2)=O)n[nH]c2c1CCSC2 C1(CCC)CC(=O)N2CCCC2CC(=O)N1.c1(CC)ccsc1C(=O)OC N1(C(Cc2n(C)cnn2)=O)CCC2(NC(C3CC4(C3)CC4F)=O)CCCC12 c1(OC)ccc(CN2CCC(C)(C(=O)Nc3nnc(Br)s3)C2)c(Br)c1O c1(C(=O)NCC2CCC(NC(C3(C)C(C)CCC3)=O)CC2)nc(Cl)ccc1F n1(CCC(=O)NCC2CC(C(=O)OC(C)(C)C)C2)ccccc1=O c1(C(N(C2CCN(C(c3cc4ccncc4[nH]3)=O)C2)C)=O)cc(F)c(O)c(Cl)c1 C(=O)(C(CC(C)C)C(C)C)N1CC(C=CC)C(C(=O)NCCSCCCO)C1 N1(C(CCN(C(C(CC2CCCC2)OC)=O)C(C)C)=O)CC(C)(C)OCC1C N1(C(C(C)N2CCCC2)=O)CCC(C(C)(C)C(=O)N2CC(O)(CCO)C2)C1 CC1CCN(CC(N2CCCC(CNC(C3CC3Br)=O)C2)=O)CC1 C(CC(=O)NC1CCN(C(C2CCC(C(N)=O)CC2)=O)C1C)(C(N)=O)NC(C)=O C1(C(=O)NC2C(CNC(C3C(C(=O)OC)C3)=O)CCCC2)CCc2c[nH]nc2C1 n1(C(C)C)cc(CN(C(C(=O)NCCCOC(C)(C)C)c2csnn2)C)cn1 CCC(CN(C)C)CC(=O)NCC1CCCC1C(=O)OC.C12(CC1)C(=O)NC2 C(=O)(CCC1=CCCCC1)N1CCN(C)CC1C(N1CCC(CO)C(O)C1)=O N1(C(COC2CN(C(c3ccc(C)cn3)=O)C2)=O)CC(C)C(F)(F)C1 N1(C(=O)Cn2nnnc2C)CCC(C)(Nc2c(OC)cccc2)CC1 C1(NC(C=Cc2scc(C)n2)=O)CCN(C(c2ccnc(C(N)=O)c2)=O)C1(C)C N1(C(c2c(C)n3c(s2)ncc3)=O)CC2CCN(C(C3CC3C(F)(F)F)=O)CC2C1 C12(CC(N3CCC(NC(C4CCN(C)C4=O)=O)(CF)C3)=O)CNC(=O)C(C1)C2 C12(C(=O)NC(CC=C)C(=O)OCC)CCCCC(NC(=O)OC(C)(C)C)(C1)C2 C1(CCOC)CN(C(c2ccc(N)cc2O)=O)CCN1C(=O)C(C)n1ccnn1 CCCS(=O)(=O)C(C)C(=O)NCC1CC2CCC1N2C(=O)C(C)(F)F c1(CC(=O)NCCN(C(=O)Cc2cc[nH]n2)C)ccc(N2CCN(C)CC2)cc1 c1(C(=O)NC2CCC(NC(CC3CC(C)C3)=O)C2)ccccc1-n1ccnn1 C(CC(=O)NC(C)(C)CCNC(c1csc(O)n1)=O)(C(N)=O)NC(C)=O Cc1cc(C2(C(=O)NCC3CC(CNC(=O)C=CCF)C3)CC2)cc(Br)c1 N1(C(C(CC(C)C)O)=O)CCN(C(=O)Cc2cccc(Cl)c2Cl)CCC1C C1(CN(C(C2C(C)(CC)C2)=O)C)CCN(C(=O)CCOC(C)=O)CC1 CCC(CC(F)(F)F)NC(=O)CC1CCC(NC(C2CCC(O)C2)=O)C1 C1(CCC)CN(C(=O)C=CC(=O)NC2CC2)CCN1C(=O)CC1CCCCO1 CC1CN(C(c2cnco2)=O)CCC1NC(=O)C(c1ccc(F)cc1)CO N1(C(c2cncc(C#N)c2)=O)C2CCC1CC(NC(C1CCC(C3CC3)C1)=O)C2 C1(C(N)=O)CC2CCCC(C1)N2C(=O)NNC(=O)c1ccccc1OC(F)(F)F N1(C(c2cc(C)ns2)=O)CCC(C2CCCN(c3ccc(C#N)nc3)C2)CC1 N1(CC(=O)NCC(C)(F)CNC(=O)CCCN2CCOC2=O)CCC(O)CC1 Cn1ccc(CCC(=O)NC2CCCC2CC(=O)NC2(CCC(F)(F)F)CCC2)n1 Cc1cccc2c1OC(C(=O)NCCN(C(c1nccnc1N)=O)CC1CC1)C2 N1(C(Cc2c(C)nc(C)s2)=O)CCOC2(CCN(c3ccc(C#N)nc3)CC2)C1 C(CN(C)C)(C(C)(C)C)NC(CC(C)NC(=O)C=Cc1cn[nH]c1)=O N1(C(C(C)C2CCCC2)=O)CCCC(C(=O)N(C2CCCC2)Cc2ccccc2)C1 N1(C(c2cc(C)oc2)=O)CC2CC1CN2C(=O)CCC1CCCCC1 C1(CC(=O)NCC2CCC(C(N(C3CC(C)C3)C)=O)C2)COCC(C)O1 Cc1ccc(CNC(=O)CCCNC(=O)CC2(NC(N)=O)CC2)cc1F C(C(C)(C(=O)NCCC1CCN(C(C2C(C(=O)OC)C2(C)C)=O)CC1)OC)OC n1(CC(=O)NC2CCC2NC(=O)CCC2CC(F)(F)C2)cc(C#N)cn1 CN1CCN(CCNC(=O)NCc2cnn(CCF)c2)CC1 N1(C(C2(CC)CC2)=O)CCN(C2CCCN(C(C3OCCC3C)=O)C2)C(=O)C1 c1(C(=O)NCC(F)CNC(c2cccc[n+]2[O-])=O)ccc(C2CC2)c(Cl)c1 CCCC(CCCO)C(=O)N(C(CNC(c1cc(OC)no1)=O)C1CC1)C n1(CC)cc(CN(c2noc(C3CC3)c2C)C)c2ccccc12 C1(NC(C2(C)CC(=C)C2)=O)CC(F)CN(C(c2ccc(N(C)C)cn2)=O)C1 N1(C(CC(=O)OCC)=O)CC2CCC(C1)N2C(=O)CC1CCC(O)C1 c1(CC(CCC)NCCC(C)Br)cccc(I)c1 c1(CNC2CN(C(C(CCC)C)=O)CC2C)ccc2ccncc2c1 c1(C(N2CCC3C(C(=O)NC(CC)(C)CO)C3C2)=O)cc2ncccc2[nH]1 CC1=NOC(CC(=O)NC2CC(C)(NC(c3sccc3C(F)F)=O)C2)C1 C1([Si](C)(C)C)(CNC(CCN(C(=O)CCn2ccnn2)CC)=O)CC1 c1(N)ccc(F)cc1.c1(N(CC(=O)OCC)C(CO)C2CC2)ccccc1 Cc1cccn2c(CC(N3CC4CC3CC4NC(C3(C(N)=O)CC3)=O)=O)cnc12 c1(C(N2CCC(NC(c3c(C)nns3)=O)C23CCC3)=O)cc2ccc(F)cc2o1 c1(OC)nc(C(=O)NC(C2CCCN(C(=O)C=Cc3cc[nH]c3)C2)C)ncc1F O(N=C1CCCCCC1)CC(=O)NCCCNC(C1CC1C(=O)OC)=O C=CCC(CC(=O)N(CC(C)C(C)C)C)NC(=O)CCN1CCOCC1 N1(CC2C(NC(C(=O)OC)=O)CCC(C)(C)C2)Cc2ccccc2C1=O C1(NC(=O)C=CCO)CN(C(c2ccc(F)cc2)=O)CC2CC12 N1(CC2(OC)CCOC2)CCCC2(CC=CCO2)C1 CN1CCCC(N(C(=O)C(c2cnn(C)c2)NC(C2CN(C(N)=O)C2)=O)C)C1 c1(C(=O)NCCOCCN(C(C2CC(CF)C2)=O)C)cc(CCO)on1.C1CO1.CC c1(C(=O)Nc2n(CCOC)ncc2)cc2n[nH]cc2cc1-c1cccc2ncnn12 C1(C(=O)NC2CCN(C(c3cc(OC)n[nH]3)=O)C2)CCn2c(Br)cnc2C1 Cc1cc(C)c(C(=O)NCCN2CCCN(C(C3CNC(=O)N3)=O)CC2)c(C)c1 c1(C(N2CC(NC(c3cnc(C)[nH]3)=O)C(O)C2)=O)cc2n(n1)CCNS2(=O)=O C1(NC(c2nccc(C)n2)=O)CCC2(CC1)CN(C(c1cnns1)=O)CCO2 C1(CNC(c2ccn(-c3ccccc3)n2)=O)CCCC1NC(C1CCCC1)=O C12(CNC(N3CCC(c4cscc4Br)C3)=O)OCCCC1C2(F)F N1(C(CC#N)=O)C2CCC(C2)C1CC1(C(F)(F)F)N=N1.c12ccc(cc1)CNC2=O c1(NC(C2CC(=C)CN2Cc2ccc(I)c(O)c2)=O)nc(C)ccc1C#N C(=O)(C(O)CC(F)(F)F)NCC1(C)CCCN(C(COCCSC)=O)C1 C(CCCC(=O)NCCCC1(NC(=O)CCCF)CC1)OCC COn1cnc(C)c1C(=O)NC(C)C=CC(=O)Nc1cn(C)nc1OC C(C(F)(F)Cl)N(C(=O)C(=O)Nc1cnsc1)C C(C(C(=O)N(CCC(=O)NC(C)COC(F)(F)F)C)N(C)C)OC C1(C(=O)NCC2C(C(=O)NCCC(=O)N(CC)CC)CCO2)NC(=O)OC1C c12ccc3cc(nnc3c1)N2.c1(-c2c(C)onc2)nc(C(C)O)nn1C(C)C C#CCC(O)C(=O)NC(Cn1cncn1)C(=O)NCC1CC(F)(F)C1 C1(CNC(c2csc(NC=O)n2)=O)CN(C(c2ccn(C(F)(F)F)n2)=O)CC1O c1(C(=O)NC2(CNC(C3(C)CCCNC3=O)=O)CC2)cc(Br)n2ccccc12 CCC(CC(=O)N1CC(CNC(c2cccc(N)c2F)=O)CC1C)C(C)C N1(C(C(C)NC(c2ccc(C(F)(F)F)[nH]2)=O)=O)CCC2(C1)CN(C)C2 CC(=O)C(C)(C)CC(=O)NC1CN(C(c2nn[nH]c2Cl)=O)CC12CC2 C(=O)(C(CC)C(C)(C)CC)N(CC(C)NC(c1ccc(C#N)[nH]1)=O)CC N1(C(C(CC=C)NC(C)=O)=O)CC2(CCC(CNC(c3n[nH]cc3CC)=O)O2)C1 CCC(CC(C)O)N=c1cccc(S(=O)(=O)N2CCC(N(CC)CC)C2)[nH]1 C1(NC(C2C(C)(C)C2)=O)C2CC(CN(C(=O)CN3CCC(CO)CC3)C2)C1CO S(=O)(=O)(c1ccc2nc(NCCn3cc(Br)cn3)sc2c1)NC1CCC(C)CC1 c1(OCC)oc(C)nc1C(=O)OC(C)C(N)=O N1(C(C2(COC)CC2)=O)CCCN(C(c2cc3sc(C)cc3[nH]2)=O)C(C(C)C)C1 Cc1ncc(S(=O)(=O)N2CCC3(CC3C(=O)Nc3ccc(O)cc3Br)C2)n1C C1(C(=O)OC)C(C(=O)NC(CNC(c2ccc(F)o2)=O)C(C)C)C1(C)C CC1CCC(C(N2CC3(CC3)CC2C)=O)N(C(C2C3CCCOC23)=O)C1 CC(C)(C)C(CC(=O)NC1CCCCN(c2ncnn3c(Br)ccc23)C1)C(F)F c1(C(CCNC(c2nnnn2C2CCCCC2)CCF)OC)ccccc1Cl c1(CNC(C(C)SCCCC)=O)cnn2c1CN(C(=O)CCCCCO)CC2 C(=O)(CCN=c1[nH]ccs1)NCC1(C)CCN(C(c2sc(C)c(O)n2)=O)C1 CCC(F)(F)CC(=O)NCC1CCN(C(C2CC2c2ccc(Br)s2)=O)C1 c1(N2CCCCC(N(C)C)C2)nc(=NCC2CC2)[nH]c2c1CSC2 N1(C(c2scc(C)c2)=O)CCC(C(C)CNC(c2cnc(C(C)C)s2)=O)CC1 C(=O)(C(O)CCS(C)=O)NCCC(C)(C)NC(c1[nH]cc(CC)c1)=O Cc1cccc2c1OC(C(N1CCCC(C)(NC(C3CC(F)(F)C3)=O)C1)=O)C2 CN1CCN(C(C2CC(NC(c3csc(Cl)c3)=O)CCO2)=O)CC1 c1(C(C)=O)cc(C(N2CC(N(C(=O)C(=O)C3CC3)C)C3(CC3)C2)=O)ccc1O C1(CNC(c2occ(C)c2)=O)CCC(NC(=O)C(C)Cn2ccc(C)n2)CC1 C1(C(=O)NC(CCCC=C)C)CCC(O)CN1C(C1(OCC)CC1)=O c1(OC(C)C)ncccc1C(=O)NCC1(C)CCN(C(=O)CN2CC(C)(C)C2)C1 c1(CNC(C2N(C(c3ccc(OC)nn3)=O)CC2)=O)nc(Cl)ccc1Cl C1(C(F)F)(CNC(c2cnc(CC)o2)=O)CCN(C(=O)CCF)C1 C(=O)(CCN(C(=O)COCC(C)C)C(c1csnn1)C1CC1)NC(CC)C CC1CN(C(=O)Cc2cc(C3CC3)on2)CCC1N(C)C(C1CC(Cl)(Cl)C1)=O c1(CC)[nH]nc(C(N2CCC(CCNC(=O)COc3ccn(C)n3)C2)=O)c1C CCCCC(C)(F)C(=O)N1CC(CC(=O)N(CC(F)Cl)C)C2(CC2)C1 c1(C(N2C3CN(C(CC(CC(C)C)O)=O)CC2C3)=O)ccc(O)c2ccccc12 C#CCC(O)C(=O)N1CSCC1C(N1CCCC1C(N)=O)=O c1(NC(C2CCN(S(=O)(=O)CCCCl)C2)=O)nc2ccc(C(F)(F)F)cc2s1 C=C=CCC(=O)N(CCCNC(=O)C(C)CN1CCCCC1)CC1CCCC1 c1(C(=O)NCC2(OC)CN(C(c3[nH]ccc3C3CC3)=O)C2)cc(C)cc(F)c1 CC1CN(C(C2(C)CCCOC2)=O)CC1CNC(C1CCC(C(C)(C)O)CC1)=O N1(C(c2c(C)ncs2)=O)CCc2c(C(N3CCC4(CNC(=O)O4)C3)=O)csc2C1 N1(C(C(C)(CO)NC(C)=O)=O)CCC(C2CN(C(C3(C)CCSCC3)=O)C2)CC1 C1(NC(COCCC)=O)CC(=O)N(C2CN(C(=O)CP(C)(C)=O)C2)C1 C1(NC(C(C2CC2)NC(=O)CCc2ccccc2)=O)CCn2cncc2C1 N1(C(C2CC(C)OCC2)=O)CCC(CO)(CNC(c2ccc(O)nn2)=O)CC1 N1(C(=O)OC(C)(C)C)CCc2ccccc2C1CCC(=O)NC1CC1 C(=O)(CC(C)P(C)(C)=O)NCC1CCCN(C(c2cc(C(C)C)nn2C)=O)C1 C1(CNC(Cn2c(C(C)C)nnn2)=O)CN(C(=O)CCC(C)(C)F)CCC1C CCCC(CCC)C(=O)Nc1cccc(CNC(c2cccc(CC)n2)=O)c1 c1(-c2c(C(c3n(CC)nnn3)NCc3n[nH]c(CC)n3)c[nH]n2)cccc(C)c1 C(C)(C)(CCC(=O)NC1CS(=O)(=O)CC1NC(c1ccc(Br)cc1)=O)OC C(=O)(CC(C)C(F)(F)F)NCC1N(C(c2c(C)nc[nH]2)=O)CCCC1 CC(F)(F)C(C)(C)C(c1nnnn1C1CCCC1)NCC1(CF)CC1 N1(Cc2ccc(OC)c(OC)n2)CCC2(CCC(OC)C2)C1 c1(CCC(=O)NCC2(F)CC(NC(c3ccc(CC)s3)=O)C2)ccc(OC)cc1 C1(C(N2CC(N(CC)CC)C2)=O)CCC(CNC(C2CCOC2C)=O)CC1 N1(C(C(C)C)=O)CCCC(O)(CCNC(c2conc2C2CC2)=O)C1 C1(C(N(C(CC(=O)N(CCCOC)CCO)C)C)=O)CCCC(=O)C1 c1(C(C(=O)NC2C(CNC(c3ccn(CCCC)n3)=O)CC2)O)cccc(F)c1 CCCCC(O)C(C)C(=O)N1CCC2CC2(C(=O)NCc2cncnc2)CC1 Cc1cc(Cl)ncc1NC(=O)C(CC(C)C)N(C)C(c1ccc(O)c(F)c1)=O C1(C(=O)NCCCNC(C(CN2CCN(C)CC2)(C)C)=O)CCCCCS1(=O)=O CCC(C)C(C(=O)NCC(C)C(C)(C)C)NC(=O)Cc1ccc(C)s1 C12(C(N3C(CC)CN(C(C4CC=CCC4)=O)CC3)=O)CC3CC(C1)CC(C)(C3)C2 c1(OC)cc(OC)nc(C(=O)NC(C)CC(C)NC(c2cnc(Cl)n2C)=O)n1 N1(C(CCc2cnc(C)s2)=O)C(C)CN(C(c2ccc(CO)c(Cl)c2)=O)CC1C C(C(=O)N1CC(N(C)C(c2cn(C3CC3)cn2)=O)C1)(C(C)C)c1cnc(C)s1 C(=O)(CC(C)(C)CC(F)(F)F)NCC1CCCN(C(c2cnn(CC)c2C)=O)C1 N1(C(Cc2cc(C)cc(C)c2)=O)CCC2(CCC(NC(=O)CN(C)C3CC3)C2)C1 c1(C(N2CC(NC(C(C)OC)=O)C(F)(F)C2)=O)cccc(S(=O)(=O)N(C)C)c1 CC1CCCN(C(=O)Cc2ccco2)C1CNC(=O)Cc1conc1C1CCC1 C=C(C)CC(C)C(=O)N(C1CCN(C(=O)C=Cc2cncn2C)CC1)CCO c1(C(N2CCC(N(C(=O)CN3CC4CC4C3)CCC)CC2)=O)ccc(C#N)n1C C1(c2cccc(Cl)c2)(C(=O)NC(C(C)NC(C=C(COC)C)=O)CO)CC(F)(F)C1 C1(C(N(CCCOCCN(C(COCC=C)=O)C)C)=O)CCC2CC12 C(C(CNC(=O)C(c1ccccc1)C)C(F)(F)F)Nc1c(C(=O)OC)cn(C)n1 C(=O)(CC1CCCc2oc(C)nc21)N1CCC(C(=O)OCC)CC1C C(CC(=O)N(CCNC(=O)CC(=O)OC)C(C)C)(C1=CCCC1)OCC CC(C(=O)NCC1CCC(NC(c2scnc2C2CC2)=O)C1)C1=CCCC1 c1(CNc2cc(N3CCC(C=C)C3)ncn2)c(C)nc2ccccn12 C1(C(=O)NC2CC(O)(CNC(C(C)NC(N)=O)=O)C2)CCC(C)CC1 C1(C(=O)NC(CNC(C=CC=CC)=O)C)(CC)CCOC1 C12(NC(CNC(C)=O)=O)CCN(C(c3cc(N)ccc3C)=O)CCC1C2 N1(C(c2n(CC)ncc2)=O)CCC2(CC1)CC(NC(=O)C(C)C1(O)CCC1)CO2 N1(C(CCc2ccc(C)s2)=O)CC2CC(NC(=O)CCC=CBr)C(C2)C1 N1(C(c2ccc(C)o2)=O)CCC2(CCC2)C(CNC(C2(C)CCOC2)=O)C1 Cc1c(C(=O)NC2CCCN(C(=O)C=CS(C)=O)CC2)cccc1C1CC1 C#CCC(C(=O)NCc1n[nH]c(C)n1)NC(=O)CC1CC(O)C1(C)C CCS(=O)(=O)CC(=O)N(C)CCN(C)C(c1cnc(Cl)s1)=O C1(NC(C#CC(C)(C)C)=O)CN(C(=O)Cn2cnnc2)CC1C1CC1 Cc1[nH]nc2ncc(C(=O)N(CC(Cc3ccccc3)NC(=O)CC#N)C)cc12 c1(C(=O)NCCN(CCC)C(C2(F)CCCC2)=O)n[nH]cc1F c1(C(N2CC(NC(C3CC(CC(F)F)C3)=O)C2)=O)ccc2nccnc2c1 c1(NC(C2CCCCN2Cc2ncccc2Br)=O)cccc(Br)c1O c1(CNC(C(CC=C)NC(C23CCC(OC)C2C3)=O)=O)nc(O)ccc1C C(=O)(C(C)(C)CC(F)(F)F)N1CCC(N(C(C2CCN(C)C(=O)C2)=O)CC)CC1 C1(C2CCOCC2)(CC2N(C(C#CC(C=C)(C)O)=O)CC2)CCN(C(=O)CC)C1 c1(C(=O)NCCC2CC(NC(c3c[nH]nc3-c3cccs3)=O)C2)cc(=O)cc[nH]1 Cn1nccc1C=CC(N1CCOC(C(N2CC(N3CCCC3=O)C2)=O)C1)=O N1(C(c2cc(Br)n[nH]2)=O)CCCC2(CCN(C(c3cnc4sccc4c3)=O)C2)C1 c1(COC)nc(=N)[nH]cc1C(=O)NCC1CCCC1OC(c1cncc(C)n1)=O c1(C(=O)NCC2C3CN(C(C(CSC)(C)C)=O)CC32)c(F)cc(C)cc1F C(=O)(C(C)S(N)(=O)=O)N(C1CCCCC1)CCNC(C(C)(C)OC)=O C1(NC(C(C(C)C)(C)O)=O)CC2CCC1CN(C(=O)CCC1CCC(=O)N1)C2 c1(N2C(C(N3CCCC(CCOC)C3)=O)CC2)ncc(C)c(SC)n1 N1(C(c2ccc(NC)cc2)=O)CCCC(N(C(=O)C(C)Cn2cccn2)C)CC1 c1(COC)ccncc1CNC(=O)C(N1CCC(C(C)(C)C)CC1)=O C1(CNC(C(C)OC)=O)CN(C(c2ccccc2C)=O)C2CCN1C2 C1(C(N(CC(=O)NCCc2cnc(C)s2)CC)=O)OCCOC1C c1(C(N2CCC(CN(C)C(c3ccc(N)c(Cl)c3)=O)C2)=O)n[nH]c2c1COCC2 C12CCOCC1NC2=O.c1(CC)c(C)noc1-c1ccncc1 N1(C(=O)CC2CC2)CC2CC1CN2C(c1ccc(Cl)[nH]1)=O CCCC(O)CC(=O)N1CC(NC(C2CCCC3(CC3)C2)=O)C(C)(C)C1 CC1CN(C)C(=O)CN1C(=O)C(CNC(=O)CCC(C)(C)C)CC1CCCC1 N1(C(c2cnc(C)[nH]2)=O)CCCC2(CCN(C(c3cnc(Cl)nc3)=O)C2)C1 C1(NC(CSc2nc(C)[nH]n2)=O)CCN(C(c2ccnn2C(C)C)=O)CC(O)C1 Cc1[nH]nc(C(=O)NC2CCC2CNC(C2(C(N)=O)CC2)=O)c1Br C(c1ccc2ncsc2c1)=CC(N1CCCC1c1nnc2n1CCCC2)=O C1(COC)(NC(C2CC(C)CO2)=O)CCN(C(c2nocc2Cl)=O)CC1 N1(C(C(C(=O)OC)OC)=O)CCC(CNC(c2cc(C)co2)=O)C(F)(F)C1 N1(C(CCC(c2ncc[nH]2)C2CC2)=O)CCC(C2=NOCC2)C1.C=CCNCC=C c1(C(=O)NCC(COC)NC(=O)C=CC(C)(C)SC)csc(C(F)F)c1 c1(C(N2CC(NC(c3c(OC)nn(C)c3)=O)C(OC)C2)=O)coc(S(C)(=O)=O)c1 Cc1c(S(=O)(=O)NCC2CC3(CCOCC3)CO2)oc2ccccc12 C1(C(C)(C)NC(CCN(C)CC)=O)CCN(C(C2CS(=O)(=O)C2)=O)C1 N1(Cc2c(C)nc(C)s2)CCC(NC(c2ccoc2C)=O)CC1C C12(C(N(C3CC(F)(F)C3)C)=O)CCCC1CN(C(c1nocc1Cl)=O)C2 c1(C(=O)NC2CC3CN(C(CCC=CC(C)C)=O)C2C3)nc[nH]c2nccc1-2 c1(CC(=O)NC2(CC(=O)NCC3CCCCO3)CCC2)cccc(F)c1[N+](=O)[O-] N1(C(c2cn(C)nn2)=O)CCC2(CC1)CCN(C(c1ccnn1CC(F)F)=O)C2 Cc1ccc(CC(=O)NCC2(CNC(=O)CO)CCCC2)c(Cl)n1 c1(CC)cccc(CC(N2CC(NC(=O)COC3(C)CC3)CC2COC)=O)c1 c1(C(N(C2CCCC2)CCCNC(CCOCCC#C)=O)=O)cnc(O)c(C)c1 CC1(CNC(=O)CO)CCCN1C(=O)CNC(c1ccccc1)=O N12CCOC(C1)C2=O.C(C(C)(C(C)C)NC(=O)CCC=C(C)C)NC(C)=O C1(n2c(C(N(C)C)=O)nc3ccccc32)CCc2ccccc2C1 C(C)(C(=O)NC(C1CN(C(=O)C(=C2CCCCC2)F)C1)C)(C1(C)CC1)OC Cc1nn2c(C)cccc2c1C(N1CC2CC2(NC(C2CNC(=O)N2)=O)C1)=O c1(C(N(CC(O)CN(C)C(C2(C)CCC(=O)O2)=O)C)=O)cc(F)c(F)cc1F C1(NC(C)=O)CN(C(C2(c3cc[nH]n3)CCC2)=O)CC1C(c1cccc(N)c1)=O CCCCCC(C)CC(=O)N(CCC(=O)NC1CCN(C2CC2)C1=O)C(C)C CCCCC(O)C(=O)NC1CN(C(C2CC(S(C)(=O)=O)C2)=O)CC1O C12(CNC(CNC(C3CC(C#N)C3)=O)=O)CCC1CN(C(=O)Cn1cncn1)C2 c1(N(CC(CN(C)C)(F)F)C)nccc(N2CCC(N(C)C)CC2)n1 CN1CCC2(CC1)CN(c1ncccc1S(=O)(=O)N1CCC(CO)C(F)(F)C1)C2 N1(C(C2CCN(CC)CC2)=O)CCCN(C(=O)CC2CCCC2O)CC1 C1(CNC(CC2ON=C(CC)C2)=O)CCN(C(c2cc(C)oc2C)=O)C(C)C1 C(CCC(C)(C)C)(c1ccn(C)n1)NC(=O)NC(c1onc(C)n1)(C)C O=S(=O)(c1ccc(N2CC=C(CO)CC2)c(Cl)c1)NCCCc1ncccc1F C(=O)(CC(C)C(F)(F)F)N1CCC(N(C(c2nc3ccccc3s2)=O)CC)C1 C(CCCCCN(C)C(c1ccc(CCC)cc1)=O)NC(CN(CCC#C)C)=O Cc1cccc(C(=O)NCCC2(O)CCCN(C(=O)C=CC3CCOC3)C2)c1F N1(C(C(C2CCCC2)OC)=O)CCOCC(NC(c2ccc(O)nc2Cl)=O)C1 N1(C(C2(CCNC(CCCC#C)=O)CCC2)=O)CCOC(C)C1C N1(C(C(F)OC)=O)CC(NC(=O)C2=CCCC2(C)C)CC12CCCCCC2 N1(C(CC(C(F)F)NC(c2c(CC)cno2)=O)=O)CCN(CC)C(C)(C)C1 C(=O)(C(C)CC(F)(F)F)NC(CC(=O)N(C(CC)CO)C)C(F)F C(C1CCC(C)CC1)=C(C)C(N1CCC(CN(C)C(C2CCC(C)O2)=O)CC1)=O C1(CNC(CCCC)=O)CC2CCC(C1)N2C(c1conc1C1CCC1)=O N1(C(C=C(C)Cl)=O)CC2CS(=O)(=O)CC2(NC(C23CCC(F)(CC2)CC3)=O)C1 c1(OCC)ccc(C(N2CCCC2C(C)NC(C23CCC(C2)C3)=O)=O)cc1Cl C(=O)(C(C(C)(C)C)N(C)C)NC(C)C.C(=O)(C(O)CCSC)N(CCCCCNCC)C c1(C(=O)NCC2(F)CCC(NC(CC=CC=C)=O)C2)cc(Cl)c2n[nH]cc2c1 CC(C)C(N=[N+]=[N-])C(=O)NC1CC(C(N2CCC(F)(F)C(O)C2)=O)C1(C)C CC1C(C(N2CCC(N(C)C(C3CCC(C(N)=O)CC3)=O)C2)=O)C(O)C(=O)N1C c1(NCC)cc(F)ccc1CNC(=O)NC(C)Cc1ccccc1F C1(NC(c2ccc(CC)o2)=O)CN(C(c2scnc2C2CCCC2)=O)CCC1F C1(C(=O)NC2CN(C(=O)C3CC3)C2)CCC(C)N1N(C(C1CS(=O)(=O)C1)=O)CC CC(C)C(C(=O)N1CC(NC(c2ccc(C(F)(F)F)[nH]2)=O)C(C)C1)n1cncn1 c1(C(N2CCC(O)(c3cn(CC4CC4)nn3)CC2)=O)ccc(F)c(C2CC2)c1 N1(C(c2cccc(C(N3CCC4(CC4)C3)=O)c2)=O)CCC(O)C(NS(C)(=O)=O)C1 C(c1ccccc1)=C(C)C(=O)NCC1(C(=O)NC(C)(C)CCCF)CCCCC1 c1(C(C)=O)cc(C)c(C(=O)NCCCn2cc(-c3cccc(F)n3)nn2)o1 C1(CNC(CN(C2CCCC2N)CC)=O)CNCCC1C N1(C(C2CCN(C(C)=O)CC2)=O)CCCC(NC(=O)C(N2CCSCC2)C)CC1 C1(CC=C)(NC(C2CC(C)CC(C)C2)=O)CCCN(C(=O)C(C2CCC2)OC)C1 S(=O)(=O)(c1cccc(C#N)c1)NCC(=O)NC1C2N(C(CC(C)C)=O)C(CC2)C1 C(=O)(C(F)(F)C(F)(F)F)NCCCN(C(C(C1CCC1)OC)=O)C c1(C(=O)NCC(CCOC)NC(c2ccc(C(F)F)s2)=O)ccc2nn[nH]c2n1 Cc1cc(CCCC(=O)NCC2CCCCN2C(=O)CC(C)(C)C2CC2)c(C)s1 c1(OC)ncc(-c2cc(CNC(c3cccc(C)c3)=O)ccn2)cn1 C1(OC)CCC2(C(=O)NC3(CN(C)C(C4C=CCS4)=O)CC3)CCC12 C12(NC(c3cncc(Cl)c3)=O)CCCC1CN(C(C1CCC=CCCC1)=O)C2 c1(C(C(=O)NCCC(C)NC(C2CC23CC3)=O)N2CCCC2)cccnc1 c1(C(N2CCC(N(C(=O)C(F)CC)CCC)C2)=O)c[nH]c2ccc(F)cc12 Cc1cc(NC(=O)CC2(C)COCCO2)n(C2CS(=O)(=O)C2)n1 Cc1ccc(S(=O)(=O)CC(C)NC(=O)NC2CCC(CN)CC2)s1 N1(C(C(C)NC(CC)=O)=O)C(CC(N2CC(N(C)C)C(C)C2)=O)C2CCCC12 c1(CNC(c2cc(Br)ncc2Br)C)cc2ncccc2[nH]1 c1(C(=O)NCC(C2CC2)NC(CC2ON=C(CC)C2)=O)onc2c1CCCC2 C1(CC(=O)N(CCCCN(C)C(c2cnnn2C)=O)C)CCCC(C)(C)CC1 C1(C(C)NC(c2cc(CCO)on2)=O)CCCN(C(=O)CCc2cnoc2)C1 C(=O)(C1=C(Cl)CCOC1)N1CC(F)=C(C)CC1 C(c1ccc(Cl)cc1)=CC(=O)NCC1N(C(C2(C)CCCO2)=O)CCCC1 N1(CCCNC(C2CC(CNC(C(C)N3CCCC3)=O)C2)=O)CCOC1=O Cc1cc(C(N2CCCC(C)(C(=O)NCCC(=O)N(C)C(C)C)C2)=O)nc(C)n1 C1(NC(c2c(CC)csc2)=O)CCN(C(c2ccc(N)c(SC)c2)=O)CC(O)C1 c1(C(N(C(CNC(CC(=C)I)=O)C)C)=O)cccc(Cl)c1 N1(C(c2ccn(CC)c2C)=O)CC(CNC(=O)CSc2nc[nH]n2)CC1(C)C C1(C(=O)NC2CN(C(C3C(C)OCO3)=O)C2)CCCC(=O)N1C C(=O)(C1CCC(O)c2ccccc21)NC1CC(CNC(c2c(CC)nns2)=O)C1 C(=O)(CCCCCNC(C)=O)NC(CCNC(C1(CCC=C)CC1)=O)C(C)C c1(C(N(C2CCCN(C(C(=C(C)C3CC3)F)=O)CC2)C)=O)nccc2occc12 C#CC1(C(=O)NCc2nnn(CC)n2)CCN(C(=O)C2=CC(C)(CC)C2)C1 CCCC(O)CC(=O)NC1(C)CCN(C(C2CC2(F)F)=O)C1 c1(-c2ccc(CBr)cc2)ccc(-n2ccnc2)c(Br)c1 C1(NC(C(CC)C2CCC2)=O)CN(C(c2oc(CO)nc2C)=O)CC1C(F)F c1(-c2nccc(C(=O)Nc3cc(C(C)=O)c(C)cn3)c2)cc2c(cc1O)OCO2 C(c1cccnc1)=CC(=O)NC(C1CC(NC(CN(C2CC2)CC)=O)C1)C Cc1c(C(N2CCCC(n3cc(C4(C)CCCO4)nn3)C2)=O)cccc1[N+](=O)[O-] c1(CN(c2nccc(C)n2)CC2CCNCC2)ncc(Cl)cc1F c1(C(N(C2CCN(C(c3csc(O)n3)=O)C2)CCC)=O)c[nH]nc1Br C1(C(=O)NCC2(CNC(c3ccc(C(F)F)s3)=O)CCC2)CC(F)C(=O)N1 c1(CC)ncccc1C(N1CCC(C)C1CNC(=O)Cn1ncn(C)c1=O)=O C1(NC(C2COCCO2)=O)CCCCCCC1.CC1(C)C2C1CNC2=O C(=O)(CCC(CC)OC)NC1CCC(C(=O)NC(C=C)C(F)(F)F)C1 c1(C(=O)NCC(C)CNC(c2cncc(F)n2)=O)c(F)cccc1F c1(OC)cc[n+]([O-])c(C(=O)NCC2CCCCN2C(c2cnc[nH]2)=O)c1 c1(CNC(=O)C(=O)N(CC(O)CO)CCF)cccc(C(=O)O)n1 N1(C(C(C)O)=O)CC2CCC1C1CN(C(=O)COc3c(Cl)cccc3Cl)CC21 c1(C(N(C)CC2CC2)=O)ccc(O)nc1.C1(Nc2ccccc2)CC(=O)N(C2CC2)C1 N1(C(CN(C(=O)OC)C)=O)CCN(C(c2cnc(O)n2C)=O)CC1CC1CC1 c1(C(=O)NCC(CC=C)NC(=O)Cc2cccnc2C)cn(C)nc1Br C1(CNC(C2C(CC)C2)=O)CC2CCC(C1)N2C(=O)C(COC)COC C12(CC)CC1CN(C(=O)C(C1CN(C(c3nonc3N)=O)C1)OC)C2 C12(C(N3C(CNC)CCC3)=O)CC3CC1C2C3.C1(C(=O)N)C(C=C(C)C)C1(C)C Cc1cncc(CNC(=O)C(C)=CCNC(=O)CC2CC3CCC2O3)c1 C12(CNC(CCc3cn(C)nc3)=O)CCCCC1N(C(C1CCS1(=O)=O)=O)CC2 Cc1ccc(C(=O)NCC2CCCC2NC(C2CCCN(C)C2)=O)c(O)c1 C1(C(=O)NCCN(CCOC)C(c2cc(C)ccc2F)=O)CC2(CCC2)CO1 c1(OC(C)C)cnc(=NCC2C(C)CCCN2C(C2COCCO2)=O)[nH]c1 C=CC(C)C(=O)NCC(C1CCC1)NC(=O)CCCc1n[nH]c(=N)s1 C(=O)(CC(C)(O)C(F)(F)F)NCCCN(C(C(C(=O)OCC)F)=O)C C1(NC(c2ccc(OC)c(Cl)n2)=O)CCC2(CC1)CC2NC(c1cscc1Cl)=O N1(C(=O)NCc2cc(N3CCCCCC3)ncn2)CCC2COCC12 c1(CNC2C=CC(C(=O)Nc3cc(OC)nnc3)C2)ccc(F)c([N+](=O)[O-])c1 N1(C(C2CC(OC)C2)=O)CC(CNC(c2cnc(Br)c(N)n2)=O)CC12CCC2 c1(CC(C)C(=O)N(C)CC2(NC(C3CCS(=O)CC3)=O)CC2)ccc(Cl)cc1 C(=O)(C(CC(C)C)C(C)C)N1C(C)=NOC(CC(=O)NC2CCC(N=[N+]=[N-])CC2)C1 c1(OC)cc(C(N2CCCC(C)C2CNC(=O)COC2CCC2)=O)c(Cl)cc1Cl N1(C(c2c(C)nc(O)cc2)=O)CCC2(CC1)CC2C(N1CCC(C(C)C)C1)=O N1(CC2N(CC(C)(C)O)CC(CC)OC2)CCOCCC(O)C1 C1(C(N2C(CCC)C(=O)NCC2)=O)CCC(C)(C)N(C(=O)C2=C(Cl)CCC2)C1 c1(OC)cc(C(=O)NCC2CCC(NC(c3nocc3Cl)=O)CC2)ccc1C#N CCC(C)CC(C(=O)Nc1cccnc1C)NC(=O)CCc1ccnn1C C12(C(N(C3C(C)CCC3)C)=O)CCCC1CCN2C(C1CN(C)C1)=O C1(NC(C(C)Oc2cccc(C)c2)=O)C(C)CN(C(c2ccsc2C)=O)CC1C C(=O)(CC(CN(C)C)C(F)(F)F)NC1C2(CN(C(COCC(=O)NC)=O)C2)CC1 C1(NC(C(C(CC)CC)C)=O)CCN(C(=O)COC2CCCOC2)CC12CCC2 N1(C(C2CCC(CCC)CC2)=O)CCCC(C)C1CNC(=O)C(C)SC N1(C(C2N(C)CC(C)(C)C2)=O)C2CCC1CN(C(c1cc(N)ccc1F)=O)C2 Cc1cc(F)cc(C)c1NC(C1CCC(C)(C)N(C(=O)NC2CCCC2)C1)=O C(N=c1cc(C(C)C)nc(Cl)[nH]1)C1(CNC(c2ccc(COC)s2)=O)CCCC1 C(=O)(CCC(C)N(CC(C)(C)CO)C(C)=O)N(CC(CC)CC)C1CC1 C1(NC(c2c(C)nn(C)c2)=O)CC(F)CN(C(=O)CC2CCCC2)C1 c1(CC)ccc(Br)cc1C(=O)NC1CC2CC1N(C(C1CCOC1)=O)C2 C(CCN(C)C)(C(=O)N(C)Cc1ncccn1)NC(COCCC#C)=O C1(C(N2C(CCCNC(c3ccc(CO)cc3)=O)CCC2)=O)CC2(C1)CC2F CCCC(C(=O)NC1CC2(C1)CC(NC(C1(C#N)CC3CC3C1)=O)C2)C(C)C c1(C(=O)NC2CN(C(CC(=C)Br)=O)C(C)CC2)cc2ccccc2nc1O c1(C(N2CCCC(NCc3cccc(CC(=O)OC)c3)C2)=O)cn2c(n1)SCC2 c1(CNCc2ccc(C(=O)OC)[nH]2)cnn2c1CCCC2 C(=O)(CCC(C)CC)NCC(CCCC)NC(=O)C(C)NC(N)=O c1(N(C2CCC3(CC2)CNC3)C(CCCC#C)=O)ncnc2cccc(F)c12 C(=O)(C(C(C(C)C)C(C)C)NC(=O)CN1CCC2(CCC2)CC1)OC N1(C(CC(C(C)C)C)=O)CCC2(C1)CN(CC(N)=O)CC(C)O2 c1(-n2cc(CN(CCC)C)nn2)ccc(N=[N+]=[N-])cc1F C1(S(C)(=O)=O)(C(N(C(C)CNC(=O)CC(C)C(F)F)CC)=O)CCC1 c1(C(N2C(CNC(C(C)O)=O)CC3(CC3)C2)=O)cc(F)c(O)c(Br)c1 C1(NC(=O)CNC(C2CCOC2)=O)C=CCC(C(=O)NCc2cnn(CCF)c2)C1 c1(C(=O)NCC2C3CN(C(C(C(C)C)(C)O)=O)CC32)cc2ccoc2cc1F C1(O)(CNC(CN(C)Cc2ccncc2)=O)CCCN(C(C2(C)CC=CC2)=O)C1 C(=O)(C(CNC(C1(CC=C)CC1)=O)OC)NCC(=O)NCC=C N1(C(c2c(C)nsc2)=O)CCN(C(=O)CC2CCC3(CCC3)O2)C(CC2CC2)C1 C1(CNC(C(C)SC(C)C)=O)CCN(C(=O)Cc2ccccc2O)C12CCC2 N1(C(C(CC=C)C)=O)CC(N(C(=O)C(C)(C)CSC)C)CC1(C)C c1(OCC)cc(OC)cc(Nc2cn(-c3cccc(Br)c3)nn2)c1 CC1CN(C(C2(CO)CCCO2)=O)CC1(C)CNC(=O)CC(C)(C)O C(=O)(C(O)CCCNC(c1cn(C)cn1)=O)NCc1cccc(CC)c1 n1(CC(=O)NCC(CNC(CC(=O)OCC)=O)O)nc(C)c2cccnc12 c1(C(=O)NCCC2(O)CCN(C(C3C(C=C)C3)=O)C2)c(C)nc(C2CC2)nc1S CCC(C)C(=O)NC(C1CCCN1C(=O)Cn1cc(C(=O)OC)cn1)C c1(C(=O)NCC2(CNC(C3(C)CC4(CC4)C3)=O)CCCC2)cc2cccnn2c1 C1(NC(C(C)N(C)C)=O)CCCOC12CCN(C(c1csc(F)c1)=O)CC2 c1(NC(=O)NC(c2ccncc2)C)cnn(C2CC2)c1 C(=O)(C1c2ccccc2CN1Cc1nc(Br)ccc1F)NC(C)CN(C)C c1(C(=O)NCCN(C(C(C(C)C)SC)=O)C)cc(C)nc(C(C)CC)n1 C1(CNC(C(N2CCOCC2)C)=O)CN(C(=O)CN2CCCNC2=O)CC1(C)C c1(C(=O)NCCC2CCC(NC(C(C)OCC)=O)C2)cc(C)cc(C)c1O C=CCC(CC(=O)NC1CC(O)C1O)NC(=O)CC1CC1(C)C C1(C(=O)NCC2(NC(C(C)c3ccsc3)=O)CC2)C(F)(F)C12CCC2 N1(Cc2ccc(CNC(C(n3cc(CN)nn3)C)=O)cn2)CCOCCC1=O N1(C(C2(C#C)CCCC2)=O)CC2CC(C1)CN(C(=O)C(C)(C)CC(=O)OC)C2 CCCC(C)(CCC)C(=O)N1CCCN(C(C23COCC2C3)=O)CC1 c1(C(N2CC(C(C)NC(c3c(C)cnnc3)=O)OCC2)=O)ccc(O)c(F)c1F N1(C(=O)NCCN(C(=O)C(C)SC(C)C)CC)CC=CCC1 Cc1ccc(F)c(OCC(N2CC(F)(F)CC2CCNC(=O)C(C)(C)CF)=O)c1 c1(CNC(=O)C=CCNC(c2[nH]ccc2C2CC2)=O)cc(C(F)F)[nH]n1 c1(NCCC(CC)C)cc(NCC2CC3(CC3)CO2)ncn1 CCC(C)(C#N)C(=O)NC(CNC(C1CC2CCOC12)=O)C(=O)OC(C)(C)C C1(CN)(NC(=O)NCC=Cc2ccco2)CCN(Cc2ccccc2)CC1 c1(CC)ccc(C(=O)NC2(C(=O)N(CC)Cc3cnco3)CCC2)cn1 C1(NC(CC=CC)=O)CCS(=O)(=O)C12CN(C(c1cc(C)[nH]n1)=O)C2 CC1CCCN(C(=O)C=Cc2cnc[nH]2)C1CCNC(=O)CC1(CO)CC1 C1(C)(C(=O)OC)CCCN(C(C2CCN(C(c3ccncc3)=O)C2)=O)C1 C1(=CC(=O)NCC(=O)NC2COCC2NC(C2CC3CC3C2)=O)CCOCC1 c1(C(=O)NC2C(C(=O)Nc3c(C(N)=O)cc(Br)cc3)C2)cnn2cccnc12 c1(C(=O)NCC2N(C(CCC=CC)=O)CC(OC)C2)cnn2ccsc12 C1(NC(CC(=O)N(CC#C)CC)=O)CC2CC(C1)CN(C(=O)C(C)(CC)OC)C2 C1(C(C)CO)CCN(C(C2CCN(C(=O)CC(C)CN(C)C)C2C)=O)CC1 C1(NC(C(C=CC)O)=O)C(C)(C)CN(C(=O)CCc2cnc(C)s2)CC1(C)C N1(C(CCn2c(C)cc(C)n2)=O)CCC2(CC1)CC2NC(c1ccc(F)cn1)=O C1(C(N2CC(F)(CNC(c3ccn(C(C)(C)C)n3)=O)C2)=O)CCC12CCOCC2 c1(C(=O)NC2CCCC(NC(=O)CCOC3CC3)C2)ccc2cnccc2c1 N1(C(C2(OC)CCN(C(=O)CN3CCCC3)C2)=O)CC(C2=NOC(C)C2)C1 c1(N2CC3(CN(C(c4cc(C)c(F)nc4)=O)C3)C2)ncnc2cc(F)ccc12 N1(C(c2c(C)cc(CC)o2)=O)CCC2(CC1)CC2C(=O)N(C)Cc1cnc[nH]1 N1(C(CSCCCC)=O)CCC(C(=O)NC2CC(OC)C(OC)C2)C1(C)C Cc1ccc(C(N2CCCC(CCNC(c3nonc3N)=O)CC2)=O)c(C)n1 c1(C(C(C)NC(c2cccc(C)c2)C(=O)OC)=O)ccc2c(c1)CCC2 C(=O)(C(C)CC(=O)OC)N(CC(CN(C(c1cc(COC)[nH]n1)=O)C)O)C c1(C(C)C(N2CCC(NC(C3(C#N)CC3)=O)C2)=O)cccc(C2(C)CC2)c1 C1(NC(C2C(C(N)=O)COC2)=O)CN(C(c2cc(C3CC3)on2)=O)CC(F)(F)C1 C(=O)(CCCCCCC(=O)NC(C)(CNC(=O)CC(=O)OC)CO)OC Cc1csc(C(C(F)(F)F)NC(=O)C(C)NC2CC2)n1 CC1CCN(C(c2cc(CN(C)C)c[nH]2)=O)CC1NC(=O)C(F)n1cccn1 Cc1c(C(=O)NCC2=CCN(C(=O)CC(O)CN(C)C)CC2)nc2sccn12 c1(C(N2CCC(C)C(NC(=O)CCF)C2C)=O)ccc2c(c1)CCCCC2=O c1(CC(=O)NC2C(C)CN(C(=O)CCCN3CCCC3)C2)cccc(Cl)c1Cl c1(CC)cc(C(=O)NCC(CNC(=O)CSCC)NC(c2cscn2)=O)no1 C1(COC)(CNC(C2CCCOC2C)=O)CCCN1C(c1nonc1N)=O c1(OC)nccc(C(=O)NCCC2CCCN(C(c3csnn3)=O)C2)c1Cl N1(C(c2ccc(C(N)=O)s2)=O)CCCC(NC(=O)CC2CCCNC(=O)C2)CC1 c1(C(N2CCC(N3CCC(O)C3)C2)C(=O)NCCOC)c(C2CC2)cnn1C C=CCC(C(=O)NCc1occc1C(=O)NCC(CCC)CCO)C(C)C C(CO)(CCF)OCC(=O)NC1C(CCC(=O)Nc2nc[nH]n2)C1 N1(C(C(COC)C)=O)CCCC(C)(NC(=O)Cc2cnn(C3CC3)c2)C1 c1(C(=O)NC2CCN(C(CCC(C)SC)=O)CC2O)cc2c(F)cc(C)cc2[nH]1 N1(C(c2ccn(C)c2)=O)CCC2CN(C(c3ccnc(Cl)c3F)=O)CC12 N1(C(COCC=C)=O)CCN(C(c2cc(N(C)C)c(C3CC3)nn2)=O)C2CC12 C1(=CC(=O)NCCNCCC2(NC(=O)C=CCO)CC2)C2CC3CC(C2)CC1C3 CC1CN(C(c2nc(=O)cc(N)[nH]2)=O)CCC1CNC(c1cnc(C2CC2)[nH]1)=O C(C(N=c1[nH]ccn2nnnc12)c1ccncc1)N1CC(=CC(F)(F)F)C1C(=O)O N1(C(c2cc(C(C)C)n(C)c2)=O)CCCC(N(C(=O)C(O)C(F)(F)F)C)CC1 C1(C(=O)NC2CC(NC(CCC(=C)C)=O)CC2O)CC2COCC2C1 Cc1nc(C(N2CC(=O)NCC2C(=O)NCCN(CCCF)C)=O)ccc1C#N C1(C(=O)NCCNC(COC)=O)CCN(C(c2ncc(F)cn2)=O)C(C)(C)C1 CC(C)S(=O)(=O)CC(=O)NC1(c2ccccc2)CCN(C(C2(C)CC=CCC2)=O)C1 C1(OC)(CO)CCCN(C(C(=O)NCC2CCCO2)c2ccoc2)C1 C12(NC(CCNC(=O)CO)=O)CCOCC1CN(C(C1CC3(CCC3O)C1)=O)C2 c1(C(N2C(C(=O)NC3(CC(C)(C)C)CC3)CC=CC2)=O)ncn2ccccc12 N1(C(C2(OCC)CC2)=O)CCCCC1.c1(C(N(CC)C)=O)csc(CC)n1 c1(C(=O)NC(CCNC(c2ccc(CC)cc2F)=O)C)c(C)nc2sc(C)nn12 c1(NC2C(C(=O)OC)CCC2)ncnc2ccc(O)cc12 c1(C(C)NC2CNC2(C)C)nc(Cl)ccc1Cl Cc1nc(-c2ccccn2)nc(S)c1Sc1ccc(N2CC(C)OC(C)C2)o1 c1(CC(=O)NC2CC(CCNC(=O)C(Cl)=CCl)C2)cccc2nsnc12 c1(C(=O)NC2(CO)CCCN(C(C3CC3C(F)F)=O)C2)sc2cccnc2c1Cl C=CCC(C)(C)CC(=O)NCCOCCCN(C(=O)C(C#N)C1CC1)C N1(C(=O)CCOC2CCCCC2)CCC2(NC(C34COCC3C4)=O)CCCC12 N1(C(N(C)CCNC(=O)CN2CCCCCC2=O)=O)CC(=O)N(C)C1=O.C1CC1 c1(C(N(C2CCCCN(C(c3c[nH]c(=N)s3)=O)C2)C)=O)cn2cccc(Cl)c2n1 C1(C(=O)NC(C(C2CCCCC2)NC(CSCC(=O)OC)=O)C)CCC(=O)NC1 CCCS(=O)(=O)CC(=O)NC1(C2CCCN2C(C23CCC(CC)(C2)OC3)=O)CC1 CN1CC(CC(=O)NC2CC(NC(C3(c4cccs4)CCCC3)=O)C2)C(O)C1 O=S(=O)(c1ccc(NCCOC2CC2)cc1Br)NC1CCOCC1CO.C1(N)CC1 CN=C(NCc1cc(F)ccc1F)N1CCC2(CCOCC2)CC1 CCCCCC(F)C(=O)NC(CCN(C)C(c1ocnc1C)=O)C(C)C C(=O)(CC1=CCN(C(=O)C2=C(C)CC2)CC1)NC(CC)CO C1(NC(C2(NC(C(c3cncnc3)C)=O)CSC2)=O)CCOC2(CCC2)C1 CC(O)C(C)(C)C(=O)NCC(O)CNC(=O)Cc1nncn1C c1(C(N(CC(O)CNC(=O)C=CC2CCCO2)C)=O)ccc(Br)c(F)c1F C1(C(=O)NC2C3CN(C(c4c(C)cccc4C)=O)C2C3)CCn2nnnc2C1 C12N(CC1(C)C)C(=O)CN(C)C2.c1(C(C(C)C)O)cn(Cc2ccccn2)nn1 CC1CC(C(N2CCCNC(=O)C2)=O)CCN1C(c1cccc(C(F)(F)F)c1)=O N1(C(c2ccc(C)s2)=O)CCOC(CCNC(c2ccccc2C(C)O)=O)C1 C1(C(=O)NCC2(NC(C(C)C(F)F)=O)CC2)CCC2(CCC2)OC1 C1(C(=O)NCCCCNC(c2c(C(C)C)cccc2)=O)CCC(=O)N(C(C)C)C1 c1(C(=O)N(CCCn2cncn2)C2CCC2)ccc(-c2cnsc2)cc1 c1(C(=O)NCC2CCC(NC(c3nc(C)n(C)n3)=O)C2)c(C(C)C)nn(C)c1Cl C(=O)(CC(C)C(C)(C)C)N1C2C(CNC(COc3ccc(CC)cc3)=O)C(C2)C1 c1(NC(C2CNCCN2C(c2ccnc(O)c2)=O)=O)ccnc(Br)c1 C(C1COC(C)(C)O1)=CC(=O)NCCC(C)NC(c1cc(C2CC2)on1)=O C1(CCNC(=O)C(=CC2CCCCC2)F)CCCCN1C(=O)C=C.C(CC(F)(F)F)SCO c1(C(=O)NCCCN(C(c2cc(Br)c[nH]2)=O)CC)c[nH]nc1F N1(C(C(C)(C)N(C)C)=O)CCCN(C(=O)CC2OCCC2(C)C)CCC1 CC1CCCN(CCN(C(=O)CSC2CCCCO2)C2CCC2)C1 C(C1c2ccccc2CCN1C(c1nccc2ccsc12)=O)NC(C(C)C)=O c1(C(=O)NC(CNC(C2C(C=C)CC2)=O)(CC)CC)cc([N+](=O)[O-])ccc1SC C(=O)(CCS(=O)(=O)Cc1ccccc1)NCC(=O)Nc1c(C)cccc1C N1(C(C2CCC(C)O2)=O)CC2(CC(NC(=O)CC3(C)CCCCC3)C2)C1 CC1(C)CCN(C(=O)Cc2ccc(F)cc2)CC1NC(=O)C=Cc1ccncn1 c12cccc(c1)CNC(=O)C1(CC1)N(C)C2=O.C1(CCF)(NC(C)=O)CC1.CC(=O)O c1(C(=O)NC2(C3CN(C(C4=C(C)CC4)=O)C3)CC2)cnc2c(C)nsc2c1 c1(C(N2CCN(C)C(CNC(c3sccc3Cl)=O)C2)=O)csc2cnccc12 C1(OC)CC(CNC(c2c(F)cnn2C(C)C)=O)N(C(C2CCCN2C)=O)C1 C1(NC(CCc2ccn(C)n2)=O)CC2CC1N(C(C1CC=CCO1)=O)C2 C(CCC)(C(=O)N1CC(=O)CC1C(=O)NCC(C)(CC)CC)=CCC CCCC(CCC)=CC(=O)NC(C)(CNC(=O)C(C)CCOC)CO Cc1cc2c(C(=O)NCCCCNC(C3CCC(F)(CO)C3)=O)cccc2o1 C1(CNC(c2[nH]c(=NC)sc2)=O)CCN(C(c2cn(C)nn2)=O)CC1C C1(C(=O)NC2CCC(C#N)CC2)(CC)CCN(C(c2scnc2Cl)=O)CC1 N1(C(c2cn(CCC)nn2)=O)CCC(NC(c2c(C)coc2C(C)C)=O)C(O)C1 C(CC(C)C)(CS(C)(=O)=O)N(C(=O)OCC1CCN(CCNC(C)=O)CC1)C c1(N2CCC(NC(c3ccc(Br)cc3Cl)=O)C2)ncnc2cc(Br)ccc12 N1(C(C=Cc2nc(C)sc2)=O)CC(N(C)C(C2CC23CCCCC3)=O)C2(CC2)C1 C(CCC(=O)N(CC(C)N(C(=O)CSCC(C)C)C)C)N(CC=C)CCO C(=O)(C1=CCS(=O)(=O)C1)NCCN(C(C1C(C#C)C1)=O)Cc1cccc(Cl)c1 Cc1c(F)ccc(C(=O)NCC(C2(O)CCN(C(=O)CCCC#N)C2)C)c1Cl c1(C(c2nnnn2CCOC)NC(C=C)COC)ccc2cc(F)c(F)cc2n1 C=C(Cl)CC(C(=O)N(CCOCCOCC)CC)NC(=O)C(=O)NC c1(OCCC(=O)NCC(CNC(C=CC(=O)OCC)=O)O)ccccc1F C#CC1(C(N2CC(F)(CF)C2)=O)CCN(C(c2ccc(C(N)=O)o2)=O)C1 N1(C(=O)Nc2n[nH]cc2-c2ccc(N3CCCC3)nc2)CCC(F)(F)CC1 C(=O)(CC(O)CCCCC)N1CCC(C#C)(C(=O)NC(c2nncn2C)CO)C1 c1(N2CCC(C(C)NC(CNC(C)=O)=O)CC2)nccc(C#N)n1 c1(N2CCC(NC(C)=O)C(F)C2)ncnc2c1cnn2C(C)(C)C C12(CNC(c3ncn(C(C)C)c3)=O)CCC1CCN2C(c1ccc(F)c(Cl)c1)=O C1(C(=O)NC(C)CC2CCCC2)C2CC3C(C2NC(c2cncs2)=O)C13 C1(C(N2CCN(C(C3(SCC)CC(=O)C3)=O)CC2)=O)CCc2ncc(C)n2C1 C1(C(=O)NCCCC#C)CCC(O)CN1C(=O)CCc1nncs1 C(=O)(CCCCCCN=[N+]=[N-])NC(CNC(C1N(C)CCOC1)=O)C(C)(C)C N1(C(C2(C)N(C(c3n(CC)ccc3)=O)CC=C2)=O)CCn2c(C)nnc2C1 c1(NC(CNC(c2c(CC)noc2)=O)C(C)C(C)C)ncnc2sc(C)c(C)c12 c1(C(N2CCNC(CO)C2)C(N2CCSCC2)=O)ccc(C(=O)OC)c(C)c1 c1(OC)c(Cl)ccc(Cl)c1C(=O)NCC(F)CNC(=O)CCS(C)=O N1(C(C(CC2CC2)OC)=O)CC(N=[N+]=[N-])CC1C(=O)N(C(CCO)C(F)F)C c1(NC(C)=O)ncc(C(=O)N(CC(C)CNC(=O)CC(C)c2ccncc2)C)o1 C1(CCCNC(=O)CC2CCSCC2)CCCCN1C(c1cccc(CF)c1)=O c1(C(C)N(C(=O)CC2C3CNC2C3)C)nc2ccccc2[nH]1 C(N=C(NC(C)C)N1CCCC2(CC2)C1)c1ccc(OC(C)=O)cc1 c1(C(=O)NCC2C(C)CN(C(=O)CN3CCC3)C2)cnc2c(c1)CCCO2 c1(CNC23CC(C(N(CC=C)C(C)C)=O)(C2)C3)ccc(C)c([N+](=O)[O-])c1 C1(NC(CC(=O)NCC)=O)CC(C)CN(C(=O)CCc2ccc(F)nc2)C1 CC1C(=O)N(SC2CC(c3ccccc3)C2)CCN1CC1CCCCO1 C(CC(C(=O)N1CC(C)=C(C)C1)NC(=O)Cc1cc(C)cs1)OC C12(CNC(c3cnc(OC)c(Cl)c3)=O)CN(C(c3cnoc3C)=O)CC1CCO2 C(C(=O)NC1(CN2CCN(C(c3cc(C)n(C)n3)=O)CC2)CC1)(C(C)C)SC N1(C(C=Cc2n(CC)ncc2)=O)CCN(C(c2ccc(CO)s2)=O)CC(CO)C1 S(=O)(=O)(c1cccc(F)c1)NCC(=O)NCC#CCNC(CCC(=C)Cl)=O C12(CNC(c3ccc(Cl)cc3Cl)=O)CN(C(=O)CC3CCCO3)CC1CCO2 C1(C)(C(=O)NCC(C)NC(c2cc(C(=O)OC)c(C)o2)=O)CCCCCC1 N1(C(C(CC)C(C)O)=O)CC2(CCCN(C(c3c[nH]nc3-c3ccco3)=O)C2)C1 C1(NC(C2(CC=C)CC2)=O)CCCC1(C)CNC(=O)Cc1cnco1 CN1CC(C(N2CCN(Cc3cn(CC4CCOC4)nn3)CC2)=O)NC1=O CC(CC(=O)NCCC1(NC(c2cc(N)ccc2Cl)=O)CCCC1)C(F)F c1(CNC(C(=O)NCC2N(C(CCC=C)=O)CCC2)CCC)ccc(Cl)cc1F CC1C(NC(=O)CCCN2CCCCC2)CCN1C(c1coc(Br)n1)=O N1(C=O)CC(O)(N(C(=O)OC(C)(C)C)C)C1.C(=O)(C(C)SC)N.C(C)(C)C.C(COC)OC.C C(=O)(CC(CNC(=O)Cc1ccc(C)nc1)OC)Nc1cn(CC)nc1 COn1cnc(C)c1C(=O)NCCC1CC(NC(c2c(C)noc2N)=O)C1 C(=O)(C1CSc2ccccc21)NC1C(NC(CC(C)(C)C#N)=O)CCC1 C1(NC(C(C)(C)c2cc[nH]n2)=O)CC2(CCN(C(C3(CO)CC3(F)F)=O)C2)C1 N1(C(c2cc(N)c(Cl)nc2)=O)CCC(C2(NC(c3occc3Cl)=O)CC2)C1 c1(C(N2CCN(C(c3cnc(C)o3)=O)CC2CCO)=O)cn2ccccc2n1 Cc1ccc(C=CC(=O)NC(CNC(C2CC2c2cccc(F)c2)=O)C(C)C)s1 C12(CNC(CCC(C)C)=O)CCC(C1)N(C(C1CCC(=O)O1)=O)C2 C1(COC)CN(CC(=O)NC(=O)Nc2ccccc2)CCO1 C1(CNC(=O)CC2(N(C)C(C3CC(C)(O)C3)=O)CC2)CCCCC1n1ccnc1 C(=O)(CC(C)P(C)(C)=O)NC1C2CN(C(C(C(C)C)N(C)C)=O)C1C2 n1(CC)ncc2cc(C(N3CC(C(=O)O)C(C(C)C)C3)=O)cnc12 C1(F)(CNC(C(C)NC(CC)=O)=O)CCC(CNC(=O)COC2CCCC2)C1 Cc1cc(CC(=O)NC23CC(CNC(=O)CCC4CC4(C)C)(C2)C3)sn1 CCC(C)C(O)C(=O)N(CC1CCC1)CC.c1(NCC)nnn(-c2ccccc2)c1C O=C(C1=CCSC1)N1CCOC(C2(NC(=O)C(c3ccccc3)=O)CC2)C1 C=C(Br)CCC(=O)N1CCCC1CN(C(=O)C(N1CCSCC1)C)C1CC1 N1(C(CCCCCC=C)=O)CCCC(C2CCN(C(C3SCCCS3)=O)CC2)C1 c1(NCC(C)CCCO)nccc(=NC(C)(C)Cc2cccc(Cl)c2)[nH]1 C1(OC(C(c2c(Cl)cccc2Cl)(C)C)=O)CCN(CP(C)(C)=O)CC1 N1(C(Cc2c(C)scc2)=O)CCOC(CC(N2CCCCC2C(N)=O)=O)C1 Cn1cnc2cc(C(=O)NCCC3CCN(C(=O)CCC(C)(C)F)C3)ccc12 c1(C(=O)OC(CC)C(=O)Nc2cccc(C)c2)ccc2nc(C3CC3)[nH]c2c1 N1(C(C(C)(F)F)=O)CCCCC(NC(c2cccc(OC(F)F)c2)=O)C1 N1(CCC(c2cnccc2Cl)=O)C2CCC(C2)C1Cc1ccccc1 c1(C(=O)NC(C)Cn2cncn2)cn(CCNC(=O)CCN2CCC2)nn1 N1(C(C(=O)NCCC)C2CCC2CC)CCCC1COCc1cnn(C)c1.C1CC1 C1(C(N2CCC(C(=O)NCC(C3CCC3)OCC)(CF)C2)=O)CC2(C1)CC(O)C2 C(=O)(C(CC(C)C)N1CCCC1CC)OCc1cncc(OCC)c1 c1(C(c2nnnn2CC)NC(C(=O)NCC)C)cc(-c2cccnc2)n(C)n1 C1(O)(COC)CCN(C(=O)C(c2cn(C)nn2)NC(=O)C(F)C2CCCC2)CC1 O=C1CCCCC1OC(c1ccc(Br)cn1)=O C1(NC(c2c(C)cc(C)nc2)=O)CCC2(CC1)CC2C(=O)O.C12CCC1NC(=O)C2 C#CC12CCC(C(=O)NC3CCN(C(c4cn(C)nn4)=O)C3)(CC1)CC2 Cc1cnn2c1CN(C(=O)CCCCN(C)C(C1(C#N)CC(=O)C1)=O)CC2 c1(CCNC)nnc(N2CCCC(CC3CC(C)C3)C2)n1C.C(C(F)(F)F)OCC c1(CC(=O)NCC(C(=O)NCC2(C(C)(C)OC)CC2)O)ncn(C)c1C CC(C)(O)C#CC(=O)N1CCCC1C1CCN(C(=O)CCOCC(F)(F)F)CC1 C1(C(=O)NCC(CN(C(c2cncc(NC)c2)=O)C)C)C2(CCC2)C12CCC2 c1(CC)ccc(C(N2CC(C(C)NC(c3cnoc3CC)=O)C2)=O)[nH]1 c1(CNC(C2CCC3CC3CC2)=O)ccc(F)c(Cl)c1.C12=CC(=O)N(CC1)CC2 C(=O)(CC(C)CF)NCC(CCOC)NC(c1oc(CC(C)C)nc1C)=O N1(C(C(CN(C)C)c2ccccc2)=O)CCCN(C(=O)OC(C)(C)C)C(CO)C1 c1(S)cccnc1.C12(C(=O)NCCN(C(C3CC3CCOC)=O)C3CC3)CCC1C2 N1(C(C(CC=C)NC(C)=O)=O)CCN(C)CC1CNC(c1ccnn1CC#N)=O CCCN=C(NCC1CCC(=O)NC1)N1CCC(Cc2ccc(OCF)cc2)C1 N1(CC2CC(CNC(c3cc(C(F)(F)F)ccn3)=O)C(O)C2)CCS(=O)(=O)CC1 c1(C(=O)OC)ccc(C(=O)NCc2sccc2C(=O)NC2CCCO2)o1 c1(OCC(C)C)ncccc1C(=O)NCC(C(C)C)NC(C1C=CCC1)=O C1(OCC)(CNC(=O)N(C(c2ccccc2)CO)C)CCCS(=O)(=O)C1 c1(C(C)C)cc(N2CCC(C)C(NC(=O)Cc3c(O)ncnc3O)C2)nc(Cl)n1 c1(NCCS(CC)(=O)=O)ccc(S(=O)(=O)NC(CO)CCF)cc1Cl C1(F)(C(N(C2C(=O)NCC2)CCO)=O)CCN(C(=O)C=Cc2ccccc2)C1 CCCCC(C)(C)NC(C12CC1CCN2C(=O)Cc1csc(C)c1)=O c1(OC)cc(C(=O)NC(C)CNC(=O)CCC(C)(C)F)cc2cccnc12 C(CN=c1nc2c(cnn2C)c(NCC23CC(C)(CCO2)C3)[nH]1)c1cnc(C)[nH]1 c1(C(C)C)ncc(C(=O)NCC(C2(O)CN(C(=O)C(F)=CCCF)C2)(C)C)s1 C1(NC(C=CC=CC)=O)CCN(Cc2nc(-c3cc(C)oc3C)no2)CC1C N1(C(C(C)=CC)=O)CCC2(CC1)CN(C(c1cncc3nc(O)[nH]c13)=O)C2 c1(OC)ccccc1C=CC(N1CCCC(NC(c2ccc(Cl)cc2)=O)C1C)=O N1(C(CC2CC(C)(C)C2)=O)C2CCC1(C)C2(C)C C1(C(N(CCCOCCNC(C(C)=C2CCCC2)=O)C)=O)CCC(C)(C)O1 Cc1cc(O)ncc1NC(C1(C(C)NC(C2CC2C2CCCC2)=O)CC1)=O N1(C(c2cncc(C3CC3)c2)=O)CC=C(CNC(c2ccc(CO)o2)=O)CC1 CCC(COC)C(=O)N1CCC(NC(C2CCN(C(=O)OCF)CC2)=O)CC1 C1(CNc2c(C)n(C3CCCCC3)nc2)CC(c2ccc(F)cc2)=NO1 CC(C)C(C)N=c1[nH]c(=NCCn2cc(Br)nn2)[nH]c2c1COCC2 c1(NCC2(C)OCC(C)(C)OC2)nc2ncc(Cl)cc2o1 N1(C(CC=CCC)=O)CC2(C(=O)NC)CC1CCO2.N12CCC1C2=O N1(C(=O)CCn2ccccc2=O)CCN(C(C2CCCS2)=O)C2COCC12 C1(O)(CNC(CCCOCCOCC)=O)CCCN(C(c2cc[n+]([O-])cc2)=O)C1 c1(-c2n(C)ncc2)ncc(Cl)n1C.c1(N)cccc(Cl)c1 C1(C)(C(N(CCCNC(c2cnn(C)c2)=O)CC)=O)CCN(C)C1=O N1(C(c2c(C)cc(O)cc2)=O)CC2CC1CCC2NC(=O)CC1CN(C)CC1O N1(C(CCCc2nc(C)sc2)=O)CC2CCC2(NC(=O)Cn2nnc(=O)[nH]2)C1 C1(C(=O)NCC(CCOC)NC(=O)Cn2ccc(C)cc2=O)COCC(C)(C)O1 CC(C)(C)CCC(F)C(=O)N1CCC(C)(CC(=O)NCCCS(C)(=O)=O)C1 N1(C(COCC=C)=O)CCC2CCCC(C1)N2C(=O)Cc1cc(F)c(F)cc1F c1(C(=O)OCC)cncc(CNc2nc(C3CCCC3)ns2)c1 CCCCCCC(=O)NC1CC(O)(CNC(c2ccc(CN(C)C)nc2)=O)C1 C12(NC(CCC(=O)NCC)=O)CCCC1N(C(=O)CCc1cnco1)CC2 N1(C(C2(CCCC)CC2)=O)CCC2(C1)CN(C(c1cn(CCCC)nn1)=O)C2 C1(CNC(=O)CNC(c2cccs2)=O)CN(C(=O)CN2CC=CC2)CCC1CO CN1CCN(C(=O)CC2CCN(C(C3CCO3)=O)CC2)CC1C1CC1 C1(CNC(CC2CN(C)C2)=O)CC2(CCN(C(=O)CC3COC(=O)C3)CC2)C1 c1(OC)ccc(C(C)(C)NC(=O)N(C)CC2(F)CC2)cn1 c1(C(=O)OCC)cccc(N2CCC(NC(=O)CCC3C(=O)ON=C3C)C2)n1 C1(C(=O)NCCC(=O)NC(C2CCCCO2)(C)C)CC2CC1CC2O CCC(CC)CCC(=O)N1CC2(CCCC2)C1C(N1CC(F)C1)=O C1(COC)CC(CNC(c2nocc2SC)=O)N(C(=O)CCC2CCC(C)O2)C1 c1(C(=O)NCCOC2CCN(C(c3cc(Cl)ccc3O)=O)CC2)n[nH]c2c1CCC2 N1(C(c2c(C)ocn2)=O)CCC(O)(CNC(=O)CNc2ccccn2)C1 O=C(N=c1[nH]c(Cl)ncc1O)C1CC(F)CN(C(c2cc(F)c[nH]2)=O)C1 N1(C(=O)CCc2ccccn2)CCN(C(C23CCC(CO)(CC2)C3)=O)CC1CO C1(CC)CN(C(=O)C(c2ccccn2)C)CCN1C(c1ccc(C(C)C)cn1)=O c1(C(N(CCC(C)NC(Cc2cnc(C)s2)=O)C)=O)ccc(C(C)C)nc1 C(=O)(C1=CC2CCC(C1)C2)N1CCC(NC(Cc2ccc(C)cc2C)=O)C12CC2 N1(C(c2cccc(C#N)n2)=O)CC2OCCOC2C1.C12CC(C1)C(=O)N2 C(=O)(C(CNC(c1nsnc1O)=O)(CC)CC)N1CCC(CCOC)C1 c1(C(N2CCC(C)C2CNC(C2CC23CCC3)=O)=O)ccc2ccnc(O)c2n1 c1(CC(=O)NCC(C)N(C(C=Cc2c(C)cccc2)=O)C)nsc2ccccc12 N1(c2cc(C)nc(C)n2)CCC2C(CCCN2C(C2CCCN2C=O)=O)C1 N1(C(CC)=O)CC2(OC(C3CCC(NC(c4scnc4C)=O)C3)=O)CC1(COC)C2 CC(C)(C(=O)NC1CCN(C(C2CC2C(C)(F)F)=O)CC1)C(F)(F)F C12(C(=O)NC3CC4(CCCO4)C3)CCCC1N(C(c1cccc(F)c1O)=O)CC2 c1(-n2cc(C3N(C(c4cc(COC)on4)=O)CCC3C)nn2)ccc(C)nc1C C1(NC(C(COC)COC)=O)CCN(C(c2nn(C)cc2N)=O)C12CCC2 Nc1cccc(C(N2CCC(NC(=O)CN3CCCNC3=O)C23CC3)=O)c1F N1(C(CC2CC(CC)C2)=O)CCC2(CC2)CC1C(=O)N(C)CCOCCCF C1(NC(c2n(-c3c(C)cccc3)nnn2)C(C)C2CCC2)CCC(CC)CC1 N1(C(CC(COC)COC)=O)CCN(C(C2CCS(=O)CC2)=O)CC(O)C1 N1(C(C(C2CCOC2)NC(=O)CC2CCOCC2)=O)CC2(COC(=O)C2)C1 C(=O)(CCS(C)(=O)=O)OC(C(C)C(c1nnc(-c2ccccc2)o1)C)=O c1(C(=O)NCC(CC)NC(c2ccc(C)cn2)=O)cccc2nc(C(F)F)[nH]c12 N1(C(COc2ccc(C)cc2)=O)CC2CCCC(NC(=O)C=Cc3cc[nH]n3)C2C1 Cc1cn2nnc(C(=O)NCCC(C)NC(C3(C)CC3C)=O)c2c(O)n1 Cc1nc(NCC23CC(C2)N(Cc2ccccc2)C3)cc(O)n1 N1(C(CN(C2CC2)CC)=O)CCOC2(CCCN(C(c3cnc(Cl)cn3)=O)C2)C1 N1(C(c2oc(C)c(C(F)(F)F)n2)C(=O)NCCC#N)CCCC(N=[N+]=[N-])C1 CCCC(C)(O)C(=O)NC1C2CCN(C(c3cc(CCCO)on3)=O)CC12 c1(CNC(C(c2cn(C)nc2)O)=O)nnn(C)c1C(=O)NCCOC(=O)C1CC1 C1(C(N2CCN(C(C3CCCCC3)=O)CC2CF)=O)CC2(CO1)CC(F)(F)C2 Cc1ccn(CC(C)C(=O)N(C)CCN(C)C(C2CCCC2c2nc[nH]n2)=O)n1 CC1CCN(C(c2cc3c([nH]2)CCC3)=O)C(C)C1NC(=O)COC1(C)CCC1 Cc1cc(C(=O)NCC(C)NC(C2CCN(c3nncs3)CC2)=O)cc(N)c1O C(=O)(C(F)(F)C(O)C(C)C)N1CC(N(C(c2c(CCC)n(C)nn2)=O)C)C(O)C1 C1(C(=O)NC2C(NC(C3C=C(C)CS3)=O)CC2)C2C3CCC(C3)C12 c1(C(=O)NC(CN(C(=O)COC2CCOC2)CC)C)cc(C2CC2)cc(F)c1 c1(C(=O)NC2CN(C(c3cc(CC)n(CCO)n3)=O)C2)cc(Cl)c(O)c(Cl)c1 C1(CCCC)CN(C(c2cscc2C)=O)CCN1C(c1cnn(CCF)c1)=O C(=O)(C(O)Cn1cncn1)NCC1C(NC(C(C)OC2CCCC2)=O)CC1 N1(C(C(N)=O)=O)CCN(C(c2ccn(CCF)n2)=O)C2CCCCC2C1 CC1(C)COCC(C(=O)NC2CCCN(C(c3nocc3C3CC3)=O)C2)O1 C1(OC)CCC12CN(C(=O)CC1CCCCC1)C2.C12CCCC1NC2=O N1(C(C2(C#C)CC2)=O)CCN(C(=O)COCCF)C(c2cccc(CC)c2)C1 c1(OCc2c3cccc(C(C)C)c3[nH]c2)cccc2c(O)ncnc12 c1(OC)cc(CC(N2CCN(C)C(=O)C2C(C)C)=O)cc(F)c1F c1(SCc2scc(CNC(=O)CC3CCOC3)n2)ccc(-c2nn[nH]n2)c(F)c1 C(CC(C)C(=O)NCCCC(C)NC(=O)CC12CC(C1)C2)=CC C12(CNC(=O)CONC(C3CNC(=O)O3)=O)CCCC1OCC2 C1(C2CCC2)(NC(=O)NCc2ccc(OCC3ON=C(CC)C3)cc2)CCC1 c1(C(=O)NC(C(C)NC(c2c(C)cc(OC)nc2)=O)(C)C)cccc2c1CCN2 C1(C(=O)N(CC(=O)NCCO)CCO)CCN(CCCc2c[nH]c(Br)c2)C1 C1(C)(N(C2C3COCC23)C)CN(CC(=O)N(C(C)C(=O)N(CC(F)(F)F)C)C)C1 Cc1ccccc1C=CC(=O)NC(CNC(c1cnn(C(F)F)c1)=O)C1CCC1 C1(C)(NC(C)=O)CCCN(C(=O)C(C(C)C)NC(=O)CNSC(F)F)C1 C12(NC(CCCOCC)=O)COC(C1)C(NC(=O)C(c1ccc(C)o1)C)C2 C1(S(=O)(=O)N(C)C)(C(=O)OC)CCC1.c12ccnc(n1)NCC2 c1(C(C(=O)NCCCC)N(C)Cc2nn(C)nc2C)cccc(S(C)(=O)=O)c1 C(=O)(CCCCCNC(c1cc(C)n(CC)n1)=O)N(CC=C)CCC C1(NC(c2cn[nH]c2)=O)C2CC3CN(C(=O)Cc4ccc(C5CC5)cc4)C1C3C2 C(C(C)(C)CNCc1cc(CO)on1)OCC c1(C(=O)OC)cc(C(=O)OCCCCCC(N)=O)ccc1Br c1(C(N(C2CC2)CC2N(C(CC#N)=O)CCC2)=O)cc(S(N)(=O)=O)c(Cl)o1 Cc1cc(N2CCC(OCc3nccc(N4CCCC(CO)C4)n3)CC2)nc(C)n1 C12(NC(c3ccc(C#C)o3)=O)CCCC1CN(C(c1ccc(N)cc1C)=O)C2 N1(C(C#CC(C)C)=O)CCC(C2CC2)(CNC(C2CCC(F)CC2)=O)C1 C1(C)(NC(CCCOCCOC)=O)CCCN(C(C2CC3CC2C2CC32)=O)C1 c1(OC)ccc(CC(=O)NCC2C=CCN2C(c2sccc2C#N)=O)c(Cl)c1 CC(C)(CCCNC(c1ccc(O)c(F)c1)=O)C(=O)N1CCC(CCO)C1 C1(C(=O)NOC(C)C=C)(CC=C)CCN(C(=O)C(O)CCSC)C1 c1(C(C(=O)NC(C(=O)OC(C)C)C)C)ccc(SCc2ccns2)cc1 N1(C(c2c(CC)nco2)=O)CCC2CN(C(=O)C(C)Oc3ccc(F)cc3)CC12 C1(NC(C=CCC)=O)CCCC12CCN(C(=O)C(N1C(=O)CCC1=O)C)CC2 C(=O)(C(COC)C(F)(F)F)NCC(CC=C)NC(=O)Cc1ccc2nc[nH]c2c1 Cc1ncnc(O)c1CCC(=O)NC(C)CN(C)C(C1CCC2(CC2)C1)=O c1(C(=O)NCC(C(C)C)NC(c2ccccc2-n2cnnn2)=O)ccc(O)nn1 C=CC(C)CC(=O)N1CC2CC2(CNC(=O)CCc2nnc(C3CC3)o2)C1 C1(CC(N2CCN(CCc3cn(C4COCC4O)nn3)CC2)=O)CC2(CC2)CO1 c1(CNc2cn(C)c(C(N3CCOC(C#N)C3)=O)n2)cc(Br)ccc1Cl Cc1nccc(C(N2CC(O)(C(F)C(=O)NC(c3cscn3)C)C2)=O)n1 c1(C(N2CCC(NC(CN(C)CC)=O)C2)=O)cnn(C(C)(C)C)c1Cl n1(CCC=C)cc(C(N2CC(CNC(c3coc(N(C)C)n3)=O)(OC)C2)=O)nn1 CC(N=[N+]=[N-])C(=O)N1CCCCC1CCC(=O)NCC(C1CC1)C1CC1 C1(NC(CC2(C)CC2(F)F)=O)CCN(C(C2(CF)CC2(F)F)=O)CC1 N1(C(C2(COC)CC=CC2)=O)CCN(C(c2cc(C)c(N)cn2)=O)C(CF)C1 C1(F)(CNC(c2c(CC)ncnc2)=O)CCN(C(c2csc(Cl)n2)=O)CC1 c1(NC(C2CC(NCc3ccsc3)C2)=O)cnn(CC(F)(F)F)c1 c1(C(N2C(C(=O)NCC3CCCCC3)C=CC2)=O)ccc(F)c(OCC(F)(F)F)c1 CC(C)(O)CC(=O)N1C(C(=O)NCC2CC(F)(F)C2)CCC1C1CC1 CON=Cc1ccc(C(=O)NCC2(C(N)=O)CN(C(=O)C(C)=C3CCC3)C2)cc1 N1(C(CC2C(OC)COCC2)=O)CCCN(C(C2CC3(C2)CC(O)C3)=O)C(C)C1 c1(OC)ccc([N+](=O)[O-])c(C(C(=O)OC(C)(C)C)N(c2ccc(I)cc2Cl)C)c1 c1(OC)ncc(Cl)cc1C(=O)NCCCNC(=O)CN1CCC(F)(F)C1 n1(CC(=O)NCC(c2ccc(I)cc2)=O)ccc2nc[nH]c(=O)c12 C1(NC(c2c(CNC(C3C(C(C)C)OCC3)=O)c[nH]n2)=O)CC2C(C1)C2(F)F c1(COC)ccc(CC(N2CC=CC(NC(C3CN(C)CCO3)=O)C2)=O)cc1 C1(C(N2CCC(N(CC(C)C)C(c3c(C)nco3)=O)CC2)=O)CCC(C)(C)CO1 Cc1cc(C(N2CC(CNC(=O)C=CCN3CCCCC3)C(C)C2)=O)c(C)o1 C1(C(N2CCN(CCC)CC2)=O)N(C(=O)CC)CCC1(C)C.OCC CC(C)(C(=O)NCC1CC1CNC(c1cc(CC2CC2)on1)=O)C1CCC1 N1(C(c2cc(C)sc2)=O)CCN(C(=O)C(C)Oc2ccccc2F)C(C)C1C Cc1cccc(CNC(C2(CNC(c3cccs3)=O)CCCO2)=O)c1O N1(C(C2CN(C3CN(C(C4CC(F)(F)C4)=O)C3)C2)=O)CCN(CCO)CC1 c1(-c2cccc(COC)c2)cnc(F)c(C(N2CCCC(C)(O)C2)=O)c1 c1(OCC)c(C(N2CCC(Cc3cn(CCC(C)(C)C)nn3)C2)=O)c(C)nn1C C1(CCN(C(CC=C=C)=O)C2CC2)CC(F)(F)CN1C(C1CC(OC2CC2)C1)=O C1(C(N2CCCC(CNC(c3cnc(C(C)C)nc3)=O)C2)=O)CCC(O)C(=O)N1 C12(C(N3CC(C(C)NC(=O)CCc4cccnc4)C3)=O)CC(CN1C1CC1)C2 C(C1(C)CCCc2ccccc21)NC(C(N1CC(C)c2c(c(Cl)ccc2)C1)C)=O C12(CCNC(COCCC=C)=O)CCC1CN(C(C1(Cl)CCCCC1)=O)C2 c1(CNC(Cc2cnc(C)s2)=O)cncc(C(=O)NCC2CCN(C)C2)c1 c1(Nc2cn(C(C)C)nn2)nccc(N2CCC(N3CCCCC3)CC2)n1 C(CCC(C)C(=O)NC1CC(C)(CNC(=O)CC2CCOCC2(C)C)C1)OC c1(C(=O)Nc2scc(CC)n2)n[nH]c2cc(N3CCC(C(=O)O)C3)ccc12 c1(C(=O)NCCOc2cccc(Br)c2)ccc(C2=CCCC2)cc1 c1(C(C(=O)NCC#CCNC(C2(C)ON=C(C)C2)=O)(F)F)nc2ccccc2s1 c1(C(=O)NC2C=CCN(C(C3CC(C#C)(O)C3)=O)C2)cccc(S(N)(=O)=O)c1 N1(C(C2(CC=C)CCCN2C(c2cc(C)c(C)o2)=O)=O)CCCCCCC1C c1(C(=O)NC(C2C(C(=O)NC(c3ccn(C)n3)CC)C2)C)cc[nH]c(=N)n1 C(=O)(CC(CC)SC)NCC(CC=C)NC(=O)Cc1csc(S)n1 N1(CC)CC(NC(N(CCCCC(=O)N2CC(CF)C2)C)=O)CCC1=O C1(NC(c2cnn(-c3ccccc3Cl)c2)=O)CCOCC1C(=O)NCC1CCCC1 N1(C(c2c(CC)non2)=O)CCCN(C(c2ccc(C)cc2OC)=O)CC1CO CCC(O)C(C)(C)C(=O)NC1CN(C(C2CCC(=O)C2)=O)CC1F C(CN=c1cc(C#N)nc(C)[nH]1)(N(C(c1cc(C)cc(F)c1)=O)C)C1CC1 c1(C(N2C(C)CC(NC(c3c(C)ocn3)=O)C2)=O)ccn2nccc2n1 C=CCC(C(=O)NC1COCC1CNC(C1COCC1C(F)F)=O)NC(C)=O N1(C(CCc2cnc(C)o2)=O)C2CCC1CN(C(=O)C(C)Oc1ccccn1)C2 Cc1ccccc1C(=O)Nc1cn(C2CC2c2ccccc2)nn1 CC1CC(NC(=O)CCc2cncnc2)CCN1C(C1CC2CCC1C2)=O Cc1cc(F)sc1C(=O)N(C)CCN(C)C(C1(O)CCCC1)=O c1(C(=O)NCc2ccc(CNC(c3ccc(C)nc3)=O)cc2)nn(C)c(C)c1Cl N1(C(COCCCCC)=O)CCC(F)(C(=O)NC(C)(COC)C2CC2)C1 C(=O)(C(C)(F)C(=O)NCC1CCN(C(C2COCCO2)=O)C1(C)C)OC C1(F)(CNC(=NC)NCC2CC(=O)N(CC3CN(C(C)=O)C3)C2)COCCOC1 C1(C(N(C2CCNC2)CC)=O)CCC(C)(C)N(C(=O)C(C2CCCCC2)=O)C1 C(C1CCCN1C(c1cc(C2CC2)on1)=O)=CC(=O)NC1CC(C(C)C)OC1 CCCCC(O)C(C)C(=O)NC(C)CCC(=O)NC(CC)CC(F)(F)F C(C1CCCN1C(=O)Cc1cc(C)n(C)n1)=CC(=O)NCC(CC)N(C)C C1(OC)C(NC(=O)C#CCNC(=O)C(=Cc2cn[nH]c2)C)CC1(C)C N1(C(C=C(CCC)C)=O)CC(CO)C2(C1)CN(C(C1(CC)CCCCC1)=O)C2 c1(C(=O)NCCN(CCC)C(c2cc(C)[nH]c2C)=O)c(CC)noc1C O(N(C(=O)c1cc(COC(c2cnc(O)c(F)c2)=O)cs1)C(C)C)CC Cc1cc(CC(=O)OCC2COCC2C(F)(F)F)cc(C(F)(F)F)c1 N1(C(C(C)N(CC)CC)=O)CCCC(CNC(C2CC(O)C2)=O)C1 N1(C(c2cnc(C(C)(F)F)s2)=O)CCC2C(CCCN2C(C2(C)CC2(F)F)=O)C1 C1(NC(=O)CC2CC2(Cl)Cl)CN(C(=O)COc2cccc(F)c2)CC12CCCC2 C1(NC(=O)CCc2cscn2)CCC12CN(C(=O)C(c1ccccc1F)O)C2 c1(C(N2CC(NC(CCC(=C)C)=O)C(C)C2)=O)cc(F)cc(F)c1F c1(C(C(=O)NC(c2cn(CCC3CCCC3=O)nn2)CCC)F)ccccc1 C1(NC(C2(N(C)C)CCC2)=O)CCCCC1CNC(c1cncc(Cl)n1)=O N1(C(C2CC(=C)CN2Cc2ccc(N(C)C)cc2O)=O)CCC2(C1)CC2(F)F c1(N(C2CCN(CC)C2=O)C)nc(N(C)CP(C)(C)=O)c2c(n1)CCS2 N1(C(c2c(N)cc(Cl)nc2)=O)CCCC2(NC(c3cccc(F)c3F)=O)CC2C1 Cc1cc(N2CCCCC(CNC(C3CCCNC(=O)C3)=O)C2)n2ncnc2n1 C1(CC(C)(C)C)CCCCN1CC(=O)Nc1cccnc1C(F)(F)F C1(CC)CC(C(=O)NCCC2(NC(c3nnn(C(C)C)c3C)=O)CCC2)CCO1 C12(C(=O)NC(CCCNC(Cc3nc(C(C)C)sc3)=O)C)CCC(C)(C1)OC2 c1(C(N2CC3CCC2CC3)C(=O)NCCOCC)cc(C)c(Br)c(Cl)n1 C(=O)(C(C(C)C)NC(c1conc1NC(=O)CN(C(=O)C(C)C)C)=O)OC C1(c2ccccc2)(CNC(c2nnnn2C2(C)CC2)CCOCC)CCOCC1 N1(C(C(C(=O)OC)OC)=O)CC(C(=O)NC2C3CCCC2COC3)CC12CCC2 c1(CC)ccccc1C=C(C)CNC(N1CCC(C)(N(C)C)C1)=O O=C1OCCC2CN(C(C3CCN(Cc4cc5cc(Cl)ccc5[nH]4)C3)=O)CCN12 Cc1c(Cl)ccc(C(N2CCC(O)C(NC(c3cscc3F)=O)C2)=O)c1N c1(CNC(C2CCC(C(F)(F)F)CC2)c2n(C3(C)CC3)nnn2)nccc(Cl)c1F CCCC(C)CC(=O)NCC1C(O)C(O)CN1C(=O)Cc1ccc2c(c1)CC2 C1(C(=O)NC2C(C=C)COC2)N(C(=O)COCC2CC2)CCCC1(C)C Cc1cc(CN(C)CC2CCC(C(N3C(C(=O)C4CC4)CCC3)=O)CC2)ccn1 c1(CCC(=O)N(C(c2cnn(C)c2)CC)C(=O)CO)cccc(C)c1.C1(=O)CO1 N1(C(c2c(CC)nc[nH]2)=O)CCC2(CC1)CC(C)N(C(=O)CC1CCOCC1)C2 N1(C(CC(=O)NCC)=O)CCC(CCCCNC(=O)C(C)CF)CC1 c1(CCNC(CCC(C)=O)=O)cc(F)ccc1Br.C1CCCCC1 c1(CC)nc(N2CCC(C)(N3CCCC3)C2)sc1C.CCCC(C)N(C=O)C C1(C(=O)NCC2CC2Cl)CN(C(c2ccsn2)=O)CC12CCC2 C1(C(=O)OC2CN(C(=O)OC)C2)CC(C)(C)OC(C)(C)C1 C(=O)(C(C)CC(N)=O)N1C(C(=O)NCc2ccn(C)n2)(CC)CCC1 Cc1ccc(C2SCCN2C(C2(C)CCN(C(=O)C(C)S(N)(=O)=O)C2)=O)cc1C N1(C(C(C)(C)C)=O)CCOC(CNC(c2cccc(NC(=O)C3CC3)c2)=O)C1 C(C(C(C)C(C)C)NC(C1C2CC3C(C2)C13)=O)NC(C1C(C)=C1)=O c1(C(=O)NC(CNC(C2CCC(C(C)C)CC2)=O)C)nc2ccccn2n1 c1(CN2CCC(C(=O)NC(c3ccno3)C)C(O)C2)cc(Cl)c(Cl)cc1F C(CN=C(NC1CCOC1)NC1CCOC1)c1c(C)cncc1.C1CC1 C1(CC)C(C(=O)N(C2CN(C(=O)OC)C2)C)CCN1C(C1CC2CC2C1)=O C1(NC(C(C)=C2CCCC2)=O)CC2(CCCCN2C(C2CCS(=O)(=O)C2)=O)C1 c1(NC(C2C(C)N(C(=O)C(=O)C3CCCC3)CC2)=O)ccc2ccoc2c1 C(C)(CN=c1[nH]cncc1Cl)N(C(c1c(C)oc(C(C)C)n1)=O)CC(C)(O)CC(C)C CC1CN(C(=O)CCCF)CCCN1C(c1cn[nH]c1)=O c1(C(C(=O)NC2CCOC2)N(C2CC2)CC)sc(C(=O)OC)cc1OC C1(C(N2CCC(CC(=O)NOC3CC4CCC3C4)C2)=O)C2CCCC(=O)C12 c1(C(=O)NCC(N(C)C(C2(CO)CCCO2)=O)C2CC2)cnc(S)nc1 C1(C(=O)NCC(C(C)C)(C)O)CC12CCN(C(=O)C(C)(C)C1(O)CCC1)CC2 CCCCC(O)CC(=O)N1CCCC(NC(c2ccc(SC)o2)=O)C1 C1(NC(C(C2CCOCC2)C)=O)CCCN(C(C2(c3ccnn3C)CC2)=O)CC1 C(=O)(CCC(=O)C(C)(C)C)NC(CC#C)CC(=O)NC(C)CCNC(N)=O c1(NC(C23CC2CN(Cc2ccn(CCF)n2)C3)=O)nc2c(s1)COCC2 c1(C(=O)NC23CCC(CN(C(CN(C)CC)=O)C2)C3)c(C)c2cnccn2c1C Cc1cc(Br)ncc1S(=O)(=O)Nc1nc(-c2nccn2C)cs1 c1(CC)cccc(C(N2CC3(CC3C(=O)NCCn3cc(CC)cn3)C2)=O)n1 CCC(CC)CC(F)C(=O)NCCOC1CN(C(=O)C2=CCCSC2)C1 C1(C(CNC(c2n(C(C)C)ncn2)=O)(C)C)CCN(C(C2CC2C(C)O)=O)CC1 C1(CCC(=O)NCCC(CC)C)CCN(C(c2cc(C)c(C)[nH]2)=O)CC1 N1(C(CC(C)OC)=O)CCCC2(CCN(C(C3C=CC=CC=C3)=O)C2)C1 c1(C(N2C(CNC(CC(C(C)C)O)=O)CCCC2)=O)ccc2c(c1)N(C)C(=O)C2 N1(CCc2ccccc2)CC(N=c2cc(COCC(F)F)nc(C(F)(F)F)[nH]2)C1 CC(C(=O)NCCCC1CCN(C(c2c[nH]nc2Br)=O)CC1)C(F)F CC1CCc2sc(C(=O)NCC3CC3CNC(c3cc(O)cc(O)n3)=O)cc2C1 c1(NC(=O)NCCSc2ccc(C)cc2)ccc2c(c1)nc(C)c(=O)n2C C1(CNC(C2C(C=C)C2)=O)(NC(=O)C=CC(=O)OCCCC)CCOC1 CCC(C)(C)CCCC(=O)NC1(C)CCN(C(c2cccc(F)c2F)=O)CC1 c1(C(=O)NC2C(CC)N(C(C3CCCCC3(C)C)=O)CC2)ccc(OC)nc1Cl N1(C(CCc2c(C)cccn2)=O)CC2(CCN(C(C3(C(=O)C4CC4)CC3)=O)C2)C1 N1(C(C=CC2N(C)CCC2)=O)CCCC(O)(CNC(c2cnn(C)c2N)=O)C1 c1(OCCC(=O)NCC2C(NC(c3ccn(CC)n3)=O)COC2)cccc(C)c1 C(=O)(C(CO)C(F)(F)F)NC(C(CC)C)C(=O)NCCCn1ccnc1C CN1CCOC(C(=O)NCc2ccc(C(=O)NC3CCC3)cn2)C1 c1(C(=O)NC2CCCN(C(C(CCCC)N)=O)C2)ccc2c(c1)CCCC2=O c1(NC2n3nnnc32)ccc2occc2c1.N1(CC(C)SC)CCCC1=O CN1CCNCC1CNC(=O)C(N1CCN(C2(c3ccccc3)CC2)CC1)=O c12ccccc1N2.CCC(C1CC1)(C1CC1)NC(=O)NC1CCCC1 CC1c2nncn2CCN1C(=O)C(O)CCNC(=O)CS(C)(=O)=O C(=O)(CS(=O)(=O)CC(=O)NC(C)CCNC(c1c(C)cc(F)cc1C)=O)OC N12CCCC1CN(C)CC2=O.C1(CC(=O)NC)C=CCCC1.c1(C(=O)O)ccco1 c1(N(C)C)ccc(-c2cn(CC(=O)N(CC(O)C(F)(F)F)C)nn2)cc1 N1(C(COCCC#C)=O)CC(NC(C2Cc3nccn3C2)=O)C(C)(C)C1 c1(C(=O)NC2CC(C(=O)NC3(C)CC3)C2(C)C)ccc(O)c(F)c1 N1(C(C(=O)NCCCCNC(Cc2nc(C)oc2)=O)C)CCCC(O)C1 c1(C(=O)NCC)ncoc1C(=O)NCC1CC(NC(=O)C(C)(C)OC)C1 c1(C(=O)NC2CCC(CCNC(C3C(=C)CC3)=O)C2)cc(CC)nn1C C1(C(N2C(COC)(CNC(=O)CN3CCCC3=O)CCC2)=O)CCC(=O)CC1C c1(CC(=O)N(CCNC(C2(CCC)CCC2)=O)CCC)cn(CC)nc1C C1(CCO)(NC(C(=O)NCc2ccccc2)=O)CCCOC1.C12CC1NC2=O C(C(C(=O)N1CCSC(C)C1)C(C)C)NC(c1c(C)scc1)=O c1(C(=O)NC(CN(C(=O)CN2CCC(C)C2)CC)C)nccc(OC)c1OC c1(C(N2CC(CC)C(NC(=O)COCC3CC3)CC2)=O)sc2cccnc2c1Cl c1(NC)ccccc1C(N1CCC(F)(C(=O)N(CC(C)COC)C)C1)=O CC1CN(C(=O)C(C)(C)CCCNC(=O)CCCn2cccc2)CC(C)N1C Cc1sccc1C(=O)N(C1CCCC1)CCNC(=O)C(n1cc(Cl)cn1)C C1(NC(=O)Nc2ncc[nH]2)CCN(Cc2ncc(C3CC3)o2)CC1O N1(C(c2c(C)n(C)cn2)=O)CCN(C)C(CNC(=O)CCc2ccncn2)C1 C=Cc1ccc(C(=O)NC(C)(C)C(C)NC(=O)CSC(F)(F)F)cc1 c1(OC)ccnc(C(=O)N(C2CCC(NC(=O)C(c3ccc(O)cc3)=O)C2)C)c1 C1(CNC(C(C2CC2)OC)=O)CN(C(C2CC3(CCC3)C2)=O)CCO1 O=C1NCC2(CCN(C(C3(F)CCN(C(=O)Cn4cccc4)C3)=O)C2)O1 c1(NC(=O)C(c2ccnc(F)c2)N2CCCC(O)C2)ccc2c(c1)OCCO2 C1(NC(c2c(CC)cncc2)=O)CC=C(C(=O)NCC(CO)C(C)(C)C)C1 C1(C(=O)NCC(c2ccccc2)O)(CNC(=O)C=CC(F)F)CC=CC1 N1(C(c2cn(C(C)(C)C)nn2)C(=O)NCC=C)CCC(C)C1C1CC1 N1(C(c2c(OC)csc2)=O)CC(CNC(C23CC(F)C2C3)=O)CC1(C)C C1(OCC(=O)NC(CC)CNC(c2nnn(C(C)(C)C)n2)=O)CCCOC1 C1(C(=O)NC2CCC(NC(COCCCC)=O)C2)CC12CCOCC2 Cc1cccc(C(O)C(N2CCCC2CNC(c2nnn(C)c2C)=O)=O)c1 c1(CC)cc(C)c(C(=O)NC(CNC(=O)C(c2cccnc2)OC)CCOC)o1 C1(CCNC(=O)CCn2cnnn2)CN(C(c2cccc(CSC)c2)=O)CCO1 CN1CC(O)CC1C(=O)N(C(C1CN(C(C2(C)CC2)=O)C1)C)Cc1cccnc1 N1(C(CCC(C)=O)=O)CCC2(CC1)CC2NC(c1ccsc1)=O CC1(CNC(C2CC3CC3C2)=O)CCN(C(=O)Cn2nnnc2-c2ccsc2)C1 C1(C(=O)NC(CC)CN(C)C)C2CC(O)C(C2)N1C(c1cccc2occc12)=O Cc1ccc(Cl)c(NC(=O)C(=O)N2CC(NC(=O)CN3CCCCC3)C2)n1 CC(N=c1[nH]c(=NCc2nc3ccccc3o2)[nH]c2c1SCC2)c1ccccn1 C(=O)(C1Cc2cccc(Cl)c21)N(C1(c2ncon2)CC1)C c1(SC)cc(C(=O)NC(C2CCOC2)CNC(=O)C=Cc2ncc[nH]2)co1 N1(C(C#CC)=O)CCOCC(C(=O)Nc2cc(C(=O)OC)c(C(C)C)o2)C1 CC1CC(C(=O)OC2CCCN(c3ccccc3)C2=O)CCS1(=O)=O c1(C(N(C(CCNC(CSC)=O)C)C)=O)cnn(CC(F)F)c1C C(CN=c1[nH]c(=NCCCN(C)C)c2sccc2[nH]1)c1nccc(C)n1 c1(C(=O)NC2CC(CC)(CC)N(C(C3CCCSC3)=O)C2)ccc(C#N)c(C)n1 C1(O)(CNC(=O)CCc2ccncn2)CCCN(C(C2CCN(C3CC3)CC2)=O)C1 N1(C(c2cc(CO)on2)=O)CCN(C(C2(C(=O)NC3CC3)CCC2)=O)CC1 c1(CNCCCOCC(=O)NCC2N(C)S(=O)(=O)CC2)cc2c(cc1Br)OCO2 C(=O)(CCCCN(C(=O)CC1(CSC)CC1)C)NCC(C1CCCC1)OC CCCC(O)C(=O)NCCCC(C)NC(=O)C(C)(C)C1CCCCC1 S(=O)(=O)(c1ccc(I)cc1)N1CCC(CC(=O)Nc2cnccc2Cl)C1 c1(C(=O)NCCC2CCN(C(c3c(CC)onc3C)=O)CC2)ccnc(Br)c1Cl c1(CNC(C(N2C(C)COC(CO)C2)=O)=O)ccc2c(n1)NCCC2 N1(C(c2c(C)cc(C)s2)C(=O)NCCCOCC2CC2)CCC(C)(C)C1C CC1(C)COC(CCC(N2CCC(CNC(C3CNC(=O)C3)=O)CC2)=O)C1 C1(C(=O)NCCC#CCC)CCC(C)(C)N(C(c2n[nH]c3c2COC3)=O)C1 CC(C)CCC(C(=O)NC1CCC(CO)CC1)NC(=O)CC#N C(C)(C)(CC(=O)NCC1CC(F)(CNC(=O)CCCC#N)C1)SC N1(C(=O)Nc2c(OC(C)=O)cccc2)CCCC2(CCCOC2)C1 C1(NC(CCC)=O)CN(C(C2CCC(=O)N2CCC)=O)CC2(CCC2)C1 CCCC(CC)CC(=O)NCC(C)(C)CNC(C1CC1c1nccn1C)=O N1(C(COC)=O)CCCC1C1(C(=O)NC(C)(C)CCF)CC1 c1(C(N2CCC(NC(C3(OC)CC3)=O)C(F)C2)=O)cc(F)c(N)c(F)c1 N1(C(C(C)=O)=O)CCSC(C(=O)Nc2ccc(-n3nc(C)cc3C)cc2)C1 C1(CCC)CN(C(c2cnc(O)n2C)=O)CCN1C(c1cc(C(F)F)nn1C)=O C=CCCCCCC(=O)NCCOCCCNC(C1CC1c1ccccc1Cl)=O C(C(=O)NC(C)CC(C)NC(c1c(C)ncn1C)=O)(C(C)(C)C)NC(C)=O c1(CC)nc(-c2ccnc(-n3cncn3)c2)n(CC(C)CO)n1 CN=c1ccc(C(N2CCC(C(=O)N(C)CC3CC3C)C2C)=O)c[nH]1 N12CC(F)(C1)N(CCO)C(CN(C)C)C(=O)NC1C(C1C)C2=O.CCOCC c1(C(CNC(c2ccn(CC)n2)=O)NC(C2CCS2(=O)=O)=O)ccc(NC)cc1 O=C1CCC(NC(=O)CCC2CCCN2C(C2CCCO2)=O)C(=O)N1 c1(COC)ccc(C(=O)N(CC(C)N(C(=O)C(O)C(F)F)C)C)cc1F C1(C2(NC(CC=CCC)=O)CC2)CCCN1C(=O)CCc1cnn[nH]1 c1(C(=O)NC2(CCCNC(c3ccc(C#C)cn3)=O)CC2)ccc(S(N)(=O)=O)s1 C(C)(CNC(=O)C(=O)NCC(F)F)(CC)NC(CCN(CCCCC)C)=O N1(C(c2cnc(C)nc2)=O)CC2(CCN(C(=O)CC3CCCCN3C)C2)C1 N1(C(c2onc(-c3c(OC)cccc3)n2)=O)CC(C2CCN(C(=O)CO)CC2)C1 C1(C(=O)NC(CC=C)C)CC2(CCC2)CN1C(C1CCOC1(C)C)=O c1(CC)nc(C)c(C(=O)NCCCC2(NC(=O)CC3(O)CCCC3)CC2)s1 Cc1cc(=N)[nH]cc1C(N1CCCC(CNC(C2(Br)C(C)C2C)=O)C1)=O C12(C(=O)NCC(CC)NC(C3(O)CCC(C)CC3)=O)CCC(C)(C1)OC2 C1(C(=O)NCCC(C)OC)CCCN1C(=O)CSCCC(C)C C(=O)(CCCC(C)=O)N(C1CC(NC(C2(COC)CC=CCC2)=O)C1)C n1(CC(=O)N(C2CCN(C(=O)CN(S(C)(=O)=O)C)C2)C)nc(O)ccc1=O c1(CC)noc(CNC(=O)C(c2cccs2)NC(=O)C(C)c2ccco2)n1 C#CC(C(C)(C)OC)NC1(CO)CCC1.OC c1(C(N2CCC(CNC(CCCC=C)=O)CC2C)=O)cc2c(CC)cccc2[nH]1 c1(OC)cnncc1C(=O)NC1(CCC(=O)NC(C2CCCCC2)CO)CCC1 C=CC(C)(CC)C(=O)NC1CC(CCNC(c2occc(=O)c2OC)=O)C1 CCN(OC)C(=O)CNC(=O)C(n1cc(COc2cccc(N)c2)nn1)C CC(CC(=O)N1Cc2occ(C(N3CC(F)CC(F)C3)=O)c2C1)C(C)(C)C N1(C(CCSC)=O)CCC2CN(C(=O)CC3CCCCC3(C)C)CC2C1 C1(C(=O)NCC23CC(NC(C4Cc5cscc5C4)=O)(C2)C3)CCn2cncc2C1 C(CCC(=O)NCC1CC2(CCCO2)C1)(C(C)C)NC(c1nc(C)sc1)=O NS(=O)(=O)c1ccc(-c2cc(CN3CC(O)C(F)C3)ccc2F)nc1 C12(COC)CCOC1CN(C(C(=O)NC1CCOC1)C1CC1(C)Br)C2 C12(C(=O)NC3CCC(C)(CNC(CCCOCC)=O)CC3)CC1COC21CCC1 C1(NC(CCCCCC#C)=O)C2CCCN(C(=O)C(=O)NCC3CC3)C2C1(C)C c1(OC)cccc(CC(=O)NCCC2(CNC(=O)CCSC3CC3)CC2)c1 Cc1nccnc1C(=O)NC1CC(C(F)F)(NC(C2CC3C=CC2C3)=O)C1 c1(CS(=O)(=O)NC2CCN(c3nnn(C)n3)C2)ccc(Cl)c2ccccc12 c1(C(=O)NC2CC(CC)(CC)N(C(=O)CS(C)(=O)=O)C2)c(Cl)ccc(Cl)c1O c1(CCC)cc(C(=O)NC2(CC)CN(C(=O)C=C(Cl)Cl)C2)n(C)n1 Cc1cc(Cl)nc(Cl)c1CNc1cn(C)c(C(=O)NCC#CC(=O)O)n1 C(=O)(C1=CCC(C)CC1)N(C1CCCN(C(C(C)SC)=O)CC1)C C#Cc1ccnc(C(=O)NC(C2CCCC2)CNC(C2(C)CCNC(=O)C2)=O)c1 CCC(CC(F)(F)F)C(=O)N1CCC(C(C)NC(=O)CC2C=CCCC2)CC1 c1(C(N2CC(C(C)(C)C)N(C(=O)CC(F)(F)F)CC2)=O)cc2cccnc2[nH]1 C(=O)(C1=NOC2(CCN(C(=O)C(C)(C)C3CC3)C2)C1)NCc1cccc(C=C)c1 C1(C(N(CCC)CCO)=O)(NC(c2cc(COC)on2)=O)CCN(C)C1 N1(C(CC(CC)OC)=O)CC(NC(=O)C(F)=CC2CC2)C2(CCC2)C1 CCC(C)C(C(=O)N1CCC(CCN(C(=O)CN2CCOCC2=O)C)CC1)OC N1(C(COCCC=C)=O)CCC(OCCNC(=O)CC(F)(F)Cl)CC1 CN1CC=C(CC(=O)N2CC3CC2(C(=O)NCCCc2ncc[nH]2)C3)CC1 c1(C(=O)NCCC(C)NC(C2(C)COC(=O)OC2)=O)cc2n(n1)CC(F)C2 c1(OCC)ccccc1C(C)NC(=O)Cn1cc(CC(=O)OCC)nn1 c1(N2C(C3(OC)CC3)CCC2)nc(NC(c2n[nH]c(CC)c2Cl)=O)cc(C)n1 Cc1cccc(C(=O)NC2COCCC2C(N2CCC2(C)C(C)C)=O)n1 C(=O)(CC1=NNC(=O)C1)NC(C1CCN(C(C=Cc2ccc(CC)o2)=O)C1)C c1(NC(C2N(C(c3c(CC)nn(C)c3)=O)C(C)CC2)=O)cn(C)c(=O)nc1O N1(C(=O)OC(C)(C)C)CCC(C)(NC(=O)CCF)CC1.c12ccc(cc1)CO2 c1(OC)ccc(C(N2CC=CC2(C)CNC(c2cc(C(N)=O)c[nH]2)=O)=O)cc1 c1(C(=O)NCCC(C)NC(C2=C(C)CCCC2)=O)cn(C)c2ccccc12 Cc1coc(C(N2CC(NC(=O)CCCSc3ccccc3)C(O)C2)=O)c1C c1(C(=O)NC(c2ccnc(O)c2)C)ccc2c(c1)CC2 c1(NCC2OCCN(C)C2)ccc(C(F)(F)F)cc1S(=O)(=O)NCCCF C1(O)(CN(C(CCc2scc(C)n2)=O)C)CCN(C(c2cncc(N)n2)=O)C1 c1(N(C)Cc2ccsn2)ccnc(NCC2CCN(CC(F)F)C2)n1 C1(F)(C(N2CCC(c3ccc(C)cc3)(C)C2)=O)CNCC1C1CC1 C1(NC(=O)NC(C(=O)OC)C(C)C)CCCC12CN(C(C)Cc1ccccc1)C2 C12(C)CN(CCC1(C)OC)C2=O.C1(CCCOC)CC1(F)F C1(O)(C(=O)Nc2cn(CC)nc2)CCN(C(=O)Cc2cccc(Br)c2)C1 C(=O)(C1Cc2ccccc21)N(CCCCCCNC(C(C)(C)SC)=O)C C1(NC(N2CCN(SC)CC2)=O)CC2(CCC2NC(C)C)C1 N1(C(CCN(C(c2n(CC#C)cnn2)=O)C)=O)CCC2(CCOC2=O)C1 C12(NC(C(C)=C(C)C)=O)CCCCC1CN(C(C1CC(=O)NC1(C)C)=O)C2 C1(C(=O)OCC)CN(C(=O)Nc2ccc(OC(C)CCC)c(C)c2)CC12CC2 C(=O)(C(C)(C)CC(C)C)NC(CC)CCC(=O)NC1CCCC1N C1(NC(C=COCC)=O)CCC2CN(C(C3(C)C=CCCC3)=O)CC2C1 c1(OC)nc(NC(C2CCN2S(=O)(=O)CCCCl)=O)cc(O)n1 c1(CC(=O)NCC2(O)CC(C(=O)Nc3ccccn3)C2)ccc(F)cc1 c1(C(=O)NCC2(NC(CN(C3CCCC3O)C)=O)CC2)ncccc1N C1(OC)CCC12CC(C(=O)NCC1(C(C)(C)O)CN(C(c3sccc3C)=O)C1)C2 C(=O)(CC(F)(F)Br)N1C(CNC(C(n2c(C)ncc2)C)=O)C=CC1 C(CNC(C1CCCN1CC(F)(F)F)=O)(CC(C)C)NC(CCCOC)=O C12CC13CCC(CC3)NC(=O)CC(=O)N2.c1ncc(F)cn1.C1(OCC)CCNC1 C1(NC(c2ncc(C)nc2)=O)CCN(C(=O)C(CO)NC(=O)C(C)C)C1(C)C C1(CNC(c2c(CC)cco2)=O)CCCN(C(=O)CC(C)C)C1.N(C)C C1(C(N2CC(C#C)(N(C)C)C2)=O)CC(C)CN(C(c2cc(O)ncn2)=O)C1 N1(C(c2cnc(C(C)(C)C)[nH]2)=O)CC2CC1CC2CNC(=O)C=CCO S(=O)(=O)(c1ccccc1)NCC(N1CCN(c2ccc(OC)nn2)CC1)(C)C c1(CNC(c2nc(CC)oc2)=O)nc(C(=O)NC2CCC(F)CC2)c(C)o1 Cn1cnc(C(=O)NCCC2(O)CCCN(C(C3CC(C)(C)CO3)=O)C2)cc1=O N1(C(C2CCCN(Cc3ccc(OC)cn3)C2)=O)CCCC2(CCOC2)C1 N1(CC)CCN(c2ncnc(Cl)c2F)C(C)C1.C1(C(C)C)C(=O)N1 Cc1sc(Cl)cc1S(=O)(=O)N(C)CC1OCCCC1(C)C N1(C(C=C(CCC)C)=O)CCN(C(C2(C)CCCOC2)=O)C2CCCC12 C(=O)(C(CC)C(C)(F)F)NCC1(NC(Cc2ccc(OC)cc2)=O)CCOC1 N1(C(C=C(C)C2CC2)=O)CC2CCC(CNC(=O)CN3CCOCC3)C2C1 N1(C(CC(=O)OCC)=O)CCC2(CC1)CCN(C(=O)C(C)(C)c1sccc1C)C2 CCC(CC(=O)N1CC(C2CCC2)C(O)C1)N(C(=O)CC#N)C CCC(CC(=O)N1CCCC(NC(c2ccnc(OC)n2)=O)C1)SC c1(N(C(=O)CC2CCC2)C2CC2)ccc(C(=O)NC(C(C)NC(C)=O)C(C)C)cc1 C1(CC)CN(C(c2occc2Cl)=O)CCN1C(c1nc(C(F)(F)F)oc1C)=O C1(C(N2C(C)CC(NC(c3cc(C#N)oc3Cl)=O)CC2)=O)CCC2(CCCC2)C1 N#Cc1cc(C(=O)NCC2CCCC2NC(=O)C(c2ccccc2)O)co1 C(=O)(C(O)CC(C)(C)C)N1CC(C(=O)Nc2ccc(C)nc2Cl)SCC1 Cc1snnc1C(=O)NC(C1CCCC1)CNC(C1CC1F)=O C1(NC(C2CCCCC2O)=O)CCC2CN(C(=O)Cn3cccn3)CCC2C1 N1(C(c2c(OCC)scc2)=O)CCCN(C(c2cccc(OC)c2)=O)CC1C c1(C(C(=O)NC)N(CC(C)C)C)ccc(C(F)F)cn1 c1(N2CC(CCC)C(CO)C2)nc(=NCC2(C)CCCO2)[nH]c2c1COCC2 C1(NC(C2(NC(CC(C)SC)=O)CC(COC)C2)=O)C2(CC2)C12CC2 CCCC(C)CC(=O)NC1C2CC3C1C3C2C(=O)NCC1CN2CCC1CC2 CC(C)CC(CN(C)C)N=c1[nH]c(=NCC2CNC(=O)C(C)(C)C2)c2sccc2[nH]1 c1(SCC)ccc(C(N2CCCC2C=CC(=O)NCC2(CO)CC(C)C2)=O)cc1 C1(n2cc(NC(CC3N(C(COCC(C)(C)C)=O)CCC3)=O)nn2)CCCCC1O O=C(C1=Cc2ccccc2C1)OCC(F)(C(=O)NC1CCCCC1)C(F)(F)F C(=O)(C1SCCc2ccccc21)NCC12OCCC(NC(C(=O)N(C)C)=O)(C1)C2 Cc1cnc(CNC(C2CCN(C)CC2)C)c(C(=O)O)c1 C1(NC(=O)C(c2cccc(Br)c2)O)CN(Cc2ccc(Br)s2)CCC1(F)F c1(SCC)ccc(CNC(c2sc(Br)cc2F)=O)nc1 C1(C(C)C)N(C(C2CCNC(=O)C2)=O)CC12CCN(C(=O)CC1CN(C)C1)CC2 c1(C(=O)OC)ccccc1C(N1CCC(O)(C(C)NC(=O)C=C(C)C)C1)=O CCC(CC)CC(=O)N1CCCCC(C(=O)NCCc2cncs2)C1 c1(C(=O)NC(C)C(C)NC(c2cnc(C(F)(F)F)c(F)c2)=O)cc(=N)[nH]c(Cl)n1 C(=O)(CC(C1CC1)NC(C12CSCC1C2)=O)NC1(CSC)CC1 C(=O)(C(C)(CC)CC)N1CC(CC=C)(NC(C2CC2(C)Br)=O)C1 c1(OC)c(CC(N2CC(NC(=O)COC3CCOC3)CC2C)=O)cccc1F CC(C)C(C)C(=O)N1CCCC1CCCNC(=O)C=Cc1ccccc1 C1(C(C(=O)NC(C(=O)NC(C)C)C)(C)C)CCCN(C(C2CC2(Cl)Cl)=O)C1 c1(NC(N2C(C)(CCO)CCC2)=O)nc2ccccc2n1-c1ccccc1 N1(C(c2cncc(C)c2)=O)CCC(NC(=O)C(C)OCC(C)C)CC(C)(C)C1 CC1CC2CC2CC1C(=O)NC1CC(CNC(c2csc(C(F)F)c2)=O)C1 C1(C2CCOCC2)(C(N(CCN(C(c2cccc(C)c2Cl)=O)C(C)C)C)=O)CC1 c1(C(C)CC(=O)NC2C=CCN(C(C3COC3)=O)C2)ccc(F)c(Br)c1 C1(C(NOCC=CC)=O)CCC(C)(C)N(C(c2[nH]ccc(=O)c2C)=O)C1 N1(C(=O)NCc2ccc(CCCCCC)s2)CC2CC(C1)c1cccc(=O)n1C2 Cc1cccc2nc(C(C)OC(C(C3CC3)NC(N)=O)=O)cn12 C(=O)(CC1=CCN(C(=O)CC2CCC=CCC2)CC1)N1C(C(=O)NC)CCC1 c1(C(N2CC(NC(c3c[nH]ccc3=O)=O)C2)=O)ccc2sc3ccccc3c2c1 C1(CC(=O)N(CCNC(c2c(C)sc(Br)n2)=O)C2CC2)CC(O)C12CCC2 C(=O)(CC1=CCOCC1)N1C(C)(C(N2CCCSCC2)=O)CC(O)C1 c1(CC)nnc2n1CCCC2C(=O)N(c1cc(C)ccc1Br)C C=CCC(CC(C)C)C(=O)NC1(C(=O)NCC(C)O)CCN(C)C1 C1(C(=O)NC2(C)CC2)CN(C(c2c(F)ccc(Cl)c2F)=O)CC(F)(F)C1 CCC(C)CCC(=O)N1CCC(C)(CNC(c2csc(C#N)c2)=O)C1 C(CC(=O)NCC(C1CCCCC1)O)(C(C)(C)C)NC(Cc1c(C)n(C)cn1)=O C1(NC(c2c(C)ccc(C)n2)=O)CCC2(CC1)CN(C(=O)CC(Cl)Cl)C2 c1(C(=O)NC2CC3(CC(NC(C(C4CC4)OC)=O)C3)C2)ccc2ncc(C)n2c1 N1(C(C2(NC(=O)NCC)CCCC2)=O)CCC(C(C)NC(=O)C(C)(C)F)CC1 c1(OC)ccc(NC(C)=O)cc1C1CCN(C(=O)CCCn2cc(C)cn2)CC1 Cc1cc(C(N2CC(NC(=O)C(C)CF)C(C)(C)C2)=O)cc2ccsc12 C(C)(CC(=O)N(CC(O)CNC(=O)Cc1ncoc1C)C)OC CC(CN=c1nc2ncn(C)c2c(NCC2(C)CCC(F)(F)C2)[nH]1)n1ccnc1 N1(C(c2c(SC)cccc2)=O)CC(NC(c2ccccc2Cl)=O)CC2(CC2)C1 CN=C(NCCOC(N1CCc2ccccc21)=O)N1CCC(N(C)C)C1 C1(NC(COCCCC)=O)CCC2(CC1)CC2NC(=O)COCCCN=[N+]=[N-] C(CC(C)C(=O)NC(Cn1ccnn1)C(=O)NCc1coc(C)n1)OC C1(CNC(CC2CC(NC(C(CO)N(C)C)=O)C2)=O)CCCCC1CO C1(CNC(c2scc(C(C)(F)F)n2)=O)(CNC(=O)CNS(N)(=O)=O)CCCCC1 C1(N(CC(C)C)C(C2N(C(C(C)=CC=C)=O)CC2)=O)CC2C=CC1C2 c1(C(=O)NC(c2ccc(F)cc2)C(C)S)cccc2c1OCCO2 C(=O)(CCCCCCCCCO)N1CCN(C(c2c(Cl)ccc(SC)c2)=O)CC1 N1(c2ccc(-c3ccc(-c4cccc(O)n4)cc3)o2)CCc2[nH]nc(O)c2CC1 c1(OCC)cc2cc(c1O)C(=O)N2.C(C(C)CCOC)OC C(c1ccn(C)c1)=CC(=O)NCC=CCC(=O)NC(C1(OC)CCC1)C c1(C(=O)NC2(C(=O)OC)C(C)(C)C2)coc(S(N)(=O)=O)c1 C1(CN(C(=O)C(F)(F)C23CC(C2)C3)C)CN(C(C2CCC23CCC3)=O)CCO1 c1(C(=O)NC(CC(C)NC(c2coc(C(F)F)c2)=O)C)cncc2[nH]ccc12 C(=O)(C(C)(C)CC(=O)NC1(C(=O)NCC(CSC)OC)CCN(C)C1)OC CCC(C)(C(=O)NCC(C1CCCN1C(=O)Cc1nocc1C)(C)C)C(N)=O c1(C(=O)NCC2(NC(=O)C3=CCCCC3)C(C)CCCC2)ccc2[nH]ccc2n1 N1(C(C2NC(=O)OC2)=O)CCCC(C2CCN(C(c3cnc(O)s3)=O)CC2)CC1 N1(C(C(C)OC(C)(C)C)=O)CCC2(CCC(CNC(C3CC4CC4C3)=O)O2)CC1 C1(C(N(CC(C)(C)CNC(=O)C(C)C2CCC2)CC)=O)CN(C)CCO1 C(=O)(C1COc2ccc(Cl)cc21)NCC1N(C(COCC=C)=O)CCC(C)C1 c1(NCc2ccc(NC(=O)OC)cc2)ncc([N+](=O)[O-])cc1C C(=O)(CC(C(F)F)NC(c1ccc(C2CC2)o1)=O)NCC#CC O=C(CC(CNC(c1cn(C2CC2)nn1)=O)C1CCC1)NCCN1CCC1 C12(N(C(CC3(CSC)CC3)=O)COC)CCN(C(=O)CCc3ccc(F)nc3)CC1C2 C1(C(=O)NC(C)(C(=O)O)c2ccccc2)CC1C1CCNCC1 C1(C(=O)Nc2nc(C)c(I)s2)CC(F)CN(Cc2ncccc2Br)C1 Cc1nc2ccccn2c1CC(=O)N(CCCNC(=O)CC(C)(C)O)CCO c1(C(=O)NC(C)C(CO)NC(c2ccc(=N)[nH]c2)=O)cc2c(s1)C(C)(C)CCC2 c1(NC(CCC)CCCNC(C2(CO)CCC2)=O)nccc(C(N)=O)c1[N+](=O)[O-] c1(C(=O)NC(C)C(CO)NC(=O)C2OC(C)(C)C2C)cc2c(s1)C(C)(C)CCC2 C1(C(=O)NCCC(C)CCNC(C23CCC(CC2O)C3)=O)CCCCCCC1 C=CCC(C(=O)N1CCC(NCC2CC(OC)C2)CC1)NC(C)=O N1(C(C(C(C)C)CO)=O)CC2CC1CN(C(c1ncccc1CO)=O)C2 c1(C(N2CCCC(C3CC(N)CCO3)C2)C(=O)NC(CC)C)nccnc1Cl c1(C(=O)NCCCN(C(=O)C(C)C(C)O)CC)ccc2c(c1)CCN2C1CC1 C1(CC)CN(C(=O)Cc2ccon2)CCC1N=c1[nH]c(Cl)nc(C)c1Cl N1(CCC(C)C)CCOC(C(=O)NC(C)C(c2ccccc2)N(C)C)C1 CCCC(CC(=O)NCc1ccc(=O)n(C)c1)NC(c1cc(C(=O)OC)oc1C)=O N1(C(C2ON=C(C)C2)=O)CCN(C)CC1CNC(=O)C(C)(F)CC1CCCC1 Cc1nn(-c2cccnc2)cc1C(=O)NC(c1nccn1C)C(C)C N(C(=NCCCCC1OCCO1)NCc1ccnn1C)CCOC C(=O)(C(CO)C(F)(F)F)N1CCCC(CCNC(C(C)(C)OC)=O)C1 C1(OC)CN(C(=O)C=CC2CCCN2C)CC1CNC(=O)Cc1ccccc1 C12(OC)CCC(C(N3CCOC(C)(CNC(=O)C(=O)NCC4CC4)C3)=O)(CC1)C2 C1(CNC(Cc2c(C)ccs2)=O)(CNC(=O)C(N2CCNC2=O)C)CCOCC1 C(=O)(C1=CCCC1(C)C)NC1CCN(C(CCC)=O)CC1C Cc1cc(C2CC2)ncc1C(N1CCN(C(C2SCCS2)=O)C2CC12)=O c1(C(N(CC(C)O)CCNC(c2ccc(O)c(Cl)n2)=O)=O)cc2cnccc2[nH]1 c1(CC(C(=O)NCC=CCNC(Cn2ncc(C)c2)=O)C)ccc(F)cc1F Cc1cccc2nc(CNc3cc(C4CCCO4)n(C)n3)[nH]c12 CC1CCN(C(c2n[nH]c(O)n2)=O)C1C(=O)NCCP(C)(C)=O C#CC(C)(C)C(=O)N1CCCC(C2CCCCN2C(C2CC23CC(O)C3)=O)C1 c1(OC)ccc(-c2csc(CC(=O)NC(c3ncc(C)s3)C)n2)cc1 C1(C(=O)NC(C2CN(C(=O)CCCS(N)(=O)=O)C2)C)CCc2ccc(F)cc2O1 c1(N2CC3C(CNC(=O)CCc4nc[nH]n4)C3C2)nc2ccc([N+](=O)[O-])cc2s1 Cc1c(C(=O)NCC(F)CNC(c2ccc(OC3CC3)cc2)=O)noc1C1CC1 c1(CC(=O)NCC(C2CC2)NC(C2CS(=O)(=O)C2)=O)ccc(F)cc1Br C1(N(CC(CC)CC)C(CC)=O)CCC(NC(=O)CCc2nc(O)n[nH]2)C1 C1(C(N(C(c2ccccc2)CNC(=O)C2CC2)C)=O)CSCCS1 N1(C(c2c(Cl)cc(C)nc2)=O)C2CCC1CC(OC1CNC1)C2 C1(N(C(CCN2C(C)CCCC2)=O)C)CCCN(C(c2c[nH]c(=O)cn2)=O)CC1 C1(C(=O)N(C2CN(CCOC)C(=O)C2)CC(C)C)CCC2(CN(CC(C)C)C2)O1 c1(C(=O)NC2C(NC(CSCC(=O)OC)=O)COC2)cnc2scc(C)n12 C12(CC(=O)NC3C(NC(C=CC(=O)NC4CC4)=O)COC3)CCCN1CCC2 C12(CC)CN(C(=O)CC3CCCC(C)O3)C(CNC(c3nc(O)sc3C)=O)(C1)C2 C1(CC(=O)NC(CC=C)C2CC2)N(C(=O)CCCCCC)CCC1(C)C c1(CCNC(CN(CC(C)C(=O)O)C2CC2)=O)ccc2c(c1)OCCO2 Cc1cc(F)ccc1C1(C(=O)NCC2CCCC2NC(C2(O)CCC2)=O)CC1 CCC(CC(=O)NC(CN(C(=O)Cc1csc(S)n1)C)CC)C(C)C CC1(C)CC(CNC(=O)CCc2ccccc2F)N(C(=O)CCCCO)C1 CC(C)CC(C)CNC(C1COCCC1NC(=O)CCn1ccnc1)=O c1(NC(C23C(CN(C(c4ccc(O)c(I)c4)=O)C2)C3)=O)ccc2ncnc(O)c2c1 C1(C(N2CC(CNC(c3ccsn3)=O)OCC2)=O)CCn2c(O)nnc2C1 CC(C)CC(O)C(C)C(=O)N1CC(NC(c2c[nH]c3cnccc23)=O)C1 C1(O)(CNC(C(C)CC2CCCC2)=O)CCN(C(=O)CC2CCNC2=O)CC1 C#CC1(C)CCN(C(C2COCCC2NC(C2CCCN2CCC)=O)=O)CC1 C1(C2CCC2)(C(=O)NCC2CC(C)(C)N(C(=O)COC3COC3)C2)CC1(F)F N1(C(c2cc(Br)ncc2OC)C(=O)NC)CCC2CCC(C1)N2C c1(C(N(C)CC2CCN(C(C3(F)CCC(C)CC3)=O)C2)=O)ccc2ncccn12 CC1(C)CC(C(F)(F)F)(C(=O)NC2CC2NC(c2coc(C3CC3)n2)=O)C1 C=C1CN2C(=O)CCC2(C(=O)NCC2CN(C(c3nccc(OC)c3N)=O)C2)C1 C1(C(=O)NCc2cccc(C#C)c2)CC12CCN(C(C1(F)CC=CCC1)=O)CC2 C1(C(=O)NC(C2CCC2)C)CCC2(CCC2)CN1C(=O)OC(C)(C)C Cc1nc2cc(C(N3CCC4(CC(NC(C5(F)CCC5)=O)CO4)C3)=O)cnc2s1 CC1CC(C2CN(C(C34COC(C3)C(NC(=O)C(F)OC(F)(F)F)C4)=O)C2)=NO1 c1(C(C(=O)NCCOCCCN(C(C(=O)NC(C)C)=O)C)(F)F)cccc(Cl)c1 CC1(C)CC1CCC(=O)NC1(CNC(=O)Cc2cccs2)CCC1 c1(C(=O)NCCC(C)N(C(=O)CCOCCN(C)C)C)ccc([N+](=O)[O-])c(O)c1 c1(C(=O)NC(C2CCN(C(c3cc(Br)n[nH]3)=O)CC2)C)cc[nH]c(=N)c1N C1(C)(C(N2CC(C)C(NC(=O)C(C)(C)C(N)=O)C2)=O)CCCC(F)(F)C1 C1(NC(CC2C(C)(C)OCC2)=O)CCN(C(=O)CC2CC3CCC2C3)CC1F c1(N2CCOCC(c3[nH]ccn3)C2)nc2c(c(=NC3CCSC3)[nH]1)COCC2 C1(C(=O)NCC(C)(CO)NC(c2cc(F)c[nH]2)=O)CCCCC12CCC2 c1(N(C)CC2CCCS2)nccc(=NCc2c(C(F)(F)F)cccc2Cl)[nH]1 C1(C(=O)NCC2(F)COC2)C2CCCC1CN(S(=O)(=O)Cn1cccc1)C2 Cn1cnc(C=CC(=O)NC2CCCCC2NC(c2ccnn2C2CC2)=O)c1 C1(CC)CN(C(c2cc(C(C)C)n(C)n2)=O)CCN1C(=O)CSCc1cccs1 c1(NC(C2CCC(NC(C)=O)CC2)=O)cnc(C2=COCC2)cn1 C12(C(=O)NCC(C)N(C(C(CC)CC3CCCCC3)=O)C)CCC(CC1)C(C)O2 c1(CC(N2CCC(NC(COC(C)C)=O)C(F)C2)=O)ccc2c(c1)COCC2 C1(NC(C(C(C)O)(C)C)=O)CN(C(c2ccccc2Br)=O)C2(CCCC2)C1 C1(C(N(CC=C)CC)=O)CCCCCCN1C(=O)CCCC(OC)OC C1(C(=O)NCC2(N(C)C)CC2)CN(C(=O)C(C2CCCCC2)F)C2(CCC2)C1 Cc1ccc(C)c(C(=O)NCC(O)CC(=O)NCCOc2ccccn2)n1 c1(CC)ccc(O)c(NC(=O)C(C2CCOC2)NC(=O)C(O)C(F)(F)F)c1 N1(C(c2cncc(SCC)n2)=O)CCCN(C(=O)CC2COCCO2)C(C)C1 c1(CC)cc(F)c(C(=O)NC2CC3CC2N(C(C2CC(C(F)F)C2)=O)C3)cc1F C1(CC)(NC(=O)CNC(=O)CN(C(=O)COC)C)CCCN(C(=O)CC#N)C1 C1(CC(=O)NCCCCCCn2cc(CC3(O)CCC3)nn2)CCCCCO1 C1(C(CNC(CC#N)=O)F)CCN(C(=O)CC2CC3CC3C2)CC1 c1(OC)nccc(CNC(=O)NC2CCCOC2c2nccn2C)c1Br C1(C(=O)NC2CN(C(c3c(CC#N)ccs3)=O)CC2O)CC12CCS(=O)(=O)CC2 CC1CCC(N(C(=O)CC2CCC(NC(C34CC3CNC4=O)=O)C2)C)CC1 c1(CN(c2c(C(=O)O)cccc2F)C)cccc([N+](=O)[O-])c1 C1(CNC(C2(C(=O)OCC)CC2)=O)CCC(C)(C)CN1C(C1CCN(C)C1=O)=O CCCCC(C)C(=O)NCCCC1CCCCN1C(c1scc2c1CCCC2)=O C(N=c1[nH]c(=NCCSC2CCCC2)[nH]c2cccnc12)c1c(CC)noc1C c1(N2CCC(C)OC(C)C2)nc2ccccc2nc1N1CCSC(C(F)(F)F)C1 C(C(=O)NCC12CC(CNC(c3cnccc3C)=O)(CO1)C2)(C(C)(C)C)OC C12(CNC(C3ON=C(CC)C3)=O)CCCC1N(C(=O)Cc1cnn(C)c1)CCC2 Cc1ccc(-c2nc(Nc3ccccc3CO)cs2)cc1-c1ccccc1C#N C1(C(C(=O)NC2(CCOC)CCCC2)C)CCCN(C(=O)C=Cc2ccsc2)C1 C1(C(=O)NC2C(C)CCN(CC(=O)NC3CCCCC3)C2)CC2CCCCN2C1 Cc1cc(C)c(C(N2CCCC2C(C)NC(=O)C(C)Oc2ccccc2F)=O)[nH]1 c1(NC(=O)NCCS(=O)(=O)NCC)nccc2ccc(F)cc12 C1(S(C)(=O)=O)(CNC2CC(C(=O)Nc3c(C(=O)OCC)nccn3)C2)CCC1 c1(C(N(C)CC2CCCN(C(CSCC=C)=O)C2)=O)ccnc(C)c1O C1(NC(C2(CC)CCC2)=O)CN(C(=O)CC(C)CC(=O)OC)CC1N=[N+]=[N-] N1(C(C(N2CC(C)C=C(C)C2)=O)=O)CC(C)c2ccccc21 c1(COCC)nc(C(=O)NCCCNC(c2nnn(C(C)(C)C)n2)=O)cs1 N1(C(c2c(CC)occ2)=O)CCC(C(=O)NCC2=NOC(C)C2)CC1(C)C N1(C(C(CC=C)C)=O)CC2(C1)C(NC(=O)CCCCF)CCS2(=O)=O CC1C(C(=O)N2CCC3CC2CN(C(C2(C)CC2)=O)C3)=Cc2ccccc21 C1(C(=O)OC)CN(C(=NCCCCl)NCCC(N2CCN(C)CC2)C)CC12CCC2 O=C(C1=Cc2cccc(Br)c2OC1)NC1CN(C(C2CC23CC(O)C3)=O)C1 c1(OC)cc(C(=O)NCC2CN(Cc3c(Br)ccc(F)c3F)C2)ccc1C#N c1(OC)ccc(C=CC(=O)NC2(CNC(C3CNC(=O)N3)=O)CC2)cc1O C1(C(=O)Nc2c(C)n(C(C)C)nc2)N(C(=O)C(C)CC#N)CCCC1(C)C C1(NC(=O)Cc2cn(CC3CCOC3)nn2)CCOC(c2ccc(F)cc2)C1 S(=O)(=O)(c1c[nH]c(C(=O)NCCC(C)N(C)C(C2(OC)CCSC2)=O)c1)NCC C1(NC(C(CC)OC)=O)C2CC1N(c1ccnc(-c3ccccc3)n1)C2 C1(NC(c2ccc(CCC)[nH]2)=O)CC(CO)N(C(=O)Cn2nc(C)nc2C)C1 C(=O)(CC1=NNC(=O)C1)N1C(C)CC(NC(=O)C(c2ccc(O)cc2)=O)C1 C(=O)(C1CCCc2scnc21)NCC1(O)CCN(C(C2CC(C#C)(O)C2)=O)CC1 N1(C(C2(C(C)C)CC2)=O)C2CCC(C2)C1CC(=O)NCCC[Si](C)(C)C C1(C(=O)NC(=O)C(=O)N(c2ccc(NC3CC3C)cc2)CC)CCC(C)(C)CO1 O=C(NNc1ccc(F)c(F)c1)C1(n2cc(CN3CCCC3)nn2)CCOCC1 CN1Cc2ccc(C(=O)NCC(CNC(=O)CC(F)(F)C(F)F)CO)cc2C1=O c1(OC)ccc(C(N)=O)cc1C(=O)NC1(CCNC(=O)C(C)(O)C2CC2)CC1 Cc1ccc(C(N)=O)cc1NC(=O)NCC1CCCC1c1nncn1C c1(C(C(=O)NC(C(=O)OC)C)N(C)CCc2cccs2)ccc(C(C)C)cc1 c1(C(N2CC(CO)(NC(=O)C=Cc3cnc[nH]3)C2)=O)ncc(Cc2cnn[nH]2)s1 c1(CC(N2CCCC(CN(C)C(c3cnn(C)c3)=O)C2)=O)cc(F)ccc1Cl CC1CN(C(=O)CC2(N(C)C(N)=O)CC2)CC1C(=O)Nc1cnncc1O N1(OC(CCl)OC(N2C(C)C(OC(C)(C)C)CCC2)=O)CCc2scc(Br)c2C1 c1(C(N2CCC(O)(C(=O)NCc3cnn(CCF)c3)C2)=O)ccncc1Cl N1(C(c2c(F)ccc(C)c2N)=O)CCC2(CC1)CC(C)N(C(C1CCC1C)=O)C2 c1(SCC2(CC(=O)NCCOC)CNC2)ccc(C)cc1 N1(C(Cc2c(C)ccs2)=O)CC(CNC(C23CC(C(C)(C)C)(C2)C3)=O)CC1C C1(C(=O)NCC(O)C2CCC2)(COC)C=CCN1C(C1CCOCC1)=O CCCCCC(CC)C(=O)N1CC2CC1(C(=O)NCCC1CC1)C2 C#CCC(C)(C(=O)NC(CCC)C(=O)N(C)C)NC(=O)C(CC)OC(C)C c1(C(=O)NCC2CC(OC)CN2C(=O)C(N)=O)nnc(O)cc1C c1(C(N2CC3CN(C(C4CC=CCO4)=O)CC3C2)=O)ccc2ncc(=O)[nH]c2c1 C1(C(=O)NC(C(=O)N(CC(=O)NC)CCC)C2CCCC2)CC(OC)(OC)C1 c1(C(=O)NC2C=CC(C(=O)NC(c3scc(C)n3)C)C2)c[nH]c2nccc-2c1 C1(F)(CNC(CCOCC(C)C)=O)CCC(NC(C2C3COCC23)=O)C1 Cc1cc([N+](=O)[O-])cc(C(=O)NC2CCCC2CNC(C2(N(C)C)CCC2)=O)n1 C(=O)(C(=O)C(C)(C)C)NCC(C(=O)NC(C)CC1CC1)OC C1(C(N2C(C#C)CCCC2)=O)CCN(C(=O)Cc2cnn(CC)c2)O1 N1(C(C(=CC2CCC(C)CC2)C)=O)CC2CCN(C(=O)C3=CCOCC3)C(C2)C1 CC(C)(CC(F)C(=O)N1CC(O)(CO)C1)NC(=O)C(O)CN1CCCC1 CCCCC(C)C(=O)NC1(C)CCN(C(=O)CCc2nc(-c3ccoc3)no2)C1 C1(CC(=O)NC2CCN(CCNC(CC(=C=C)C)=O)CC2)CC(O)C12CCC2 C1(C(=O)Nc2nnc(C)o2)CN(Cc2cccc(Cl)c2)CCS1 N1(C(CCSc2n(C)nnn2)=O)CCCN(C(C23COCC(C2)OC3)=O)CC1 c1(C(=O)NCc2c(C(=O)NC(C3CCCO3)CC)c[nH]n2)ccc(O)nn1 c1(C(=O)NCC2CN(C(C3(C)CC=CC3)=O)C2)ccc(Cc2ccccc2)cc1 c1(SC(C2(C(=O)OC)CCOCC2)=O)ccc(C2=CCCCO2)c(OC)c1 N1(C(C2(C)COC2)=O)CC(F)CC1CNC(C1COC(=O)N1)=O c1(CCC(=O)N2CC(CF)C2)cccc(O)c1.n12ccc(n1)-c1cn(nn1)CC2 Cc1nc(NC2CCN(C(C3CC(C)(F)C3)=O)C2C)ncc1[N+](=O)[O-] Cc1ccc(C(N2CCC(C)C(NC(C3(C)CCCCO3)=O)C2)=O)c(O)c1C N1(C(N2CCC(Cc3ccco3)C2)=O)CCCCC1C(O)C(F)F CCC(C#N)C(=O)NCCC1COCCN1C(=O)CCN(CCC(C)(C)C)C c1(OC)cnc(Cl)c(C(N2CCC(CC(=O)Nc3nc(Cl)cnc3Cl)C2)=O)c1 CC(CO)(C(=O)NCC1CCCOCC1)NC(C1CCSCC1)=O C1(C(=O)NC(C)(CNC(C2CC(n3cnnc3)C2)=O)C2CC2)OCCOC1(C)C c1(C(N(C(C(=O)NCC2CC(F)(CO)C2)SC)CC)=O)ccc2ccoc2c1 CC(C)(C#N)CC(C)(c1nnnn1C1CCOCC1)NCC1=CCCOC1 c1(C(N2CCCC2CC(C2CCCC2)O)C(=O)NC(C)C)ccnn1CCF.SCC c1(C(=O)NCC(CC)NC(c2ccoc2)=O)ccc(N(C)C)c(F)c1 C1(C(=O)NCCC(C)c2cn[nH]c2)(NC(C=C(COC)C)=O)CCN(C)C1 N1(C(C2(CCC)CCC2)=O)CC2(CCN(C(C3(CO)CC3)=O)C2)C1 c1(C(C(=O)NC2(CO)CN(C(C(CC)N(C)C)=O)C2)OC)cccnc1Cl CCCC(C)C(C)NC(=O)NC12CC(C1)C2 C1(CN(C)C(C2(C)COC2)=O)COCCN1C(c1cc(-c2ccccc2)co1)=O CC1CCCCC1NC1(C(=O)Nc2ccccc2)CCOCC1 O=S(=O)(c1ccc2[nH]c(=NC3CCC(F)(F)C3)sc2c1)NCCc1cnc[nH]1 N1(C(CCC(CC)C)=O)CCC(C)(C)C(CNC(c2ccc(CO)o2)=O)C1 CCN=C(NCC1C(C)(C)C1(C)C)N1CCN(C(C)=O)CC1 C1(CC(=O)NCC(CCOC)NC(=O)C(C)(C)c2ccsc2)CCCNC1=O C1(CN(C(C(C2CCCC2)OC)=O)C)CC(F)CN1C(c1coc(C(C)C)n1)=O N1(CC=C)CC(C)N(NC(=O)C(O)C(C)(C)SC)CC1C C=CC1CCCCN1C(c1cc2occc2s1)C(=O)NCCOC N#Cc1ccccc1-c1cnc(C(=O)NCCCn2ccnc2)cn1 C1(CNC(CCOCCN(C)C)=O)(NC(=O)CC2CC2)CCC(F)(F)CC1 N1(C(C(CC)COC)=O)CCN(C(c2c(-c3ccco3)noc2CC)=O)CC1C c1(CC)ccnc(C(=O)NCC2CC(F)CN2C(=O)CC2CC3CC3C2)c1 N1(C(C(CC#C)O)=O)CCC(O)(C2(NC(=O)C(C)Cc3ccccc3)CC2)CC1 c1(CC(=O)NCC(C)NC(C2C(C#C)C2)=O)ccccc1CC N1(C(C2N(C(C)=O)CSC2)=O)CCCC(C2CC2NC(c2conc2C)=O)C1 Cc1cnc(C(N2CCCC(N(C(=O)C(C)n3ccnc3)CCO)C2)=O)nc1 C1(CCNC(C2CCC2(C)C)=O)(OC)CN(C(=O)CCN2CCOC2=O)C1 CCN=C(NCCc1ccccc1OC)N1CCN(CC)C(C)C1 C1(OC)CN(C(c2snc(O)c2Cl)=O)CC1NC(=O)CCc1ccnc(C)n1 c1(C(=O)NC(CC)CNC(c2c[nH]nc2C)=O)cc(Cl)c(O)cc1C N1(C(C(Cc2ccc(OC)cc2)C)=O)CCC(NC(=O)C(C)(C2CC2)OC)C(C)C1 C1(C(N(C2CN(C(C(CCCC#C)C)=O)C2)C)=O)CC2CCCC(C1)C2(F)F C1(C(=O)NCC2CCC(NC(Cn3cnc(C#N)n3)=O)C2)CC2(CCCC2)CO1 CC1(C)CC(O)CCN(C(c2ccsc2Cl)C(=O)NCC(F)F)C1 CC(C(=O)NCCC1(NC(=O)COc2ccc(Cl)cc2)CCC1)C(C)(C)C c1(CNC(c2c(C)snc2)=O)ccccc1C1CCN(C(=O)C(C)C(F)F)CC1 C1(CC=C)(NC(=O)C=Cc2ccncc2C)CCN(C(=O)CCCC(=C)C)CC1 c1(CC(N2CCCC(CNC(C=C(CCN(C)C)Cl)=O)C2)=O)ccc2c(c1)CCC2 n1(C(CC(N2CCC(NC(CCCCC)=O)C(O)C2)=O)C)cnc2ccccc12 c1(OC)cc(C)c(NC(=O)CC2(NCCc3cccc(Cl)c3O)CCC2)c(O)c1 Cc1nn(C)c(C)c1C(=O)NCC12CCC(CC1NC(=O)Cc1nccn1C)C2 C1(CNC(CC(C=C)C)=O)CN(C(c2ccc(N)c(F)n2)=O)CC(C)(C)C1 C1(CC(=O)N(C2CCN(Cc3ccccc3Cl)C2)CCCl)CC2CCC1C2 CCCC(C)CC(C)(c1nnnn1CC)NNc1ccc2c(c1)CCC2.CC C1(C(=O)NCCOCCOCCNC(C2C(C=C)OCC2)=O)CC2(CCC2O)C1 N1(C(C2(Cl)C(C(C)=O)C2)=O)CCC(O)(C(C)NC(=O)C(C2CCCO2)C2CC2)C1 C1(N(C(C2CC(OCC)C2)=O)C)CCN(Cc2cn(C(C)C)cn2)C1 N(C(=NCC1CC1)NCc1cc(Cl)cn1C)C(CC)CCC c1(OCC)ccc(C(C(=O)NC(C)(C)C)N(C)CCc2cc[nH]n2)cc1SC.C(C)C N1(C(c2nc(COC)oc2)=O)CCC2CCN(C(c3cc(COC)cs3)=O)CC12 C1(C(=O)NC(c2nn[nH]n2)CC)CC12CCN(C(c1c(Cl)ccnc1Cl)=O)CC2 C1(NC(=O)C=C2CCCCC2)CN(C(C2(Br)CC2)=O)Cc2nccn2C1 c1(CC)ccc2c(c1)C(CC(=O)OCC(=O)N(C)OC)C(=O)N2 C(=O)(CCCC(=O)NCC(C)CC(=O)NC(C)CN1CCCC1=O)OC C12(C(=O)OC)CCCCC1(C(N1CCC(CNC(=O)CC3CSC3)C1)=O)CC2.OC Cc1cnc(NCCc2cc3cnccc3o2)c(S(=O)(=O)NCC2CCCO2)c1 N1(C(CNC(=O)NCCl)=O)CCCC1CC.C=CC(=O)OCC c1(C(N2C(CN(C)C(c3cc[nH]n3)=O)CC(F)C2)=O)cccc(N)c1Br Cc1ccc(CN2CCC3(CC3C(N3CCC(CC#N)CC3)=O)C2)cc1Br c1(C(=O)NC2CC(C)(NC(CCC(C)OC)=O)C2)cc(C2(C)CC2)ccc1F C12(C(N3C(C(=O)OC)C=CC3)=O)COC(C1)C(NC(C1CC(O)CN1C)=O)C2 C(=O)(C(C(C)CC=C(C)C)NCC(=O)Nc1ccc(NC(=O)NC)cc1)OCC c1(NC(C)=O)cccc(C(=O)NC(C2CCCN2C(=O)C=Cc2cscn2)C)n1 C(=O)(CC(C)(C)NC(C1CCCCN1C)=O)N(C(C(N)=O)C1CC1)C Nc1cc(Cl)nc(Cl)c1C(N1CC2CC1CN2C(c1ccnnc1)=O)=O S(=O)(=O)(c1ccc(Br)c(C)c1)NC(Cc1cc(C)cc(C)c1)C(=O)O N1(C(c2cn(CC(F)F)nc2C)C(=O)NCC=C)CCC(C)=C(C(=O)OC)C1 c1(OC(C)(C)C)cccc(CNC2CCNCC2CO)c1 n1(CCOC)nnnc1C(c1nscc1Br)NCCCSC N#Cc1ccc(C(N2CCC(CC(=O)Nc3nccn4ccnc34)C2)=O)cc1F C1(C(=O)NC(CC(=O)OC)C2CC(F)(F)C2)CCCCCCC1=O c1(C(=O)NC(C(C)C)CNC(C2CCN(C3COC3)C2)=O)[nH]nc2ncnc(O)c12 C1(NC(COCC#C)=O)CN(C(c2ccccc2CCC)=O)Cc2ccnn2C1 Cc1c(C(=O)NC2CCCN(C(C3CCS(=O)(=O)N3)=O)C2)nn2ccccc12 c1(CN(C(COCC#C)=O)C)ccc(CNC(C2(F)CCCCC2)=O)cc1 Cc1ccc(C(=O)NC2CCC2C(=O)NCC2CCCN2C)o1 c12ccc(cc1)Cn1ncc(c1-c1ccccn1)CS2.NC1(C(=O)O)CCOC1 c1(C(C(=O)OC)N(C)C(c2cnc(-c3cnn(C)c3)s2)=O)ccccc1Cl Cc1oc(C(=O)NCC(O)Cn2cccn2)cc1Br N1(C(c2[nH]cc(C(C)=O)c2)=O)CCC(C(N2CC(COC)C2)=O)C1CC C(=O)(C(F)CCC(C)C)NC(COC)CNC(c1nn(C)cc1Cl)=O c1(C(N2CCN(C(C=CC(CC)=CC)=O)C(C)CC2)=O)cc2n[nH]cc2cc1C C1(CC)(NC(c2ncc(C)cn2)=O)CCCN(C(=O)Cc2nn(C)cc2Br)C1 N1(C(CCCCCn2cc(C(C)(C)OC)nn2)=O)CC2CCOCC2C1 N1(C(Cc2ccc(C)cc2)=O)CCCC(C2CN(C(=O)C(CO)NC(N)=O)C2)C1 CC1(CO)CCN(C(C2CN(CC3CCC(F)(F)CC3)C2)=O)CC1O N1(C(c2ccc(CC)cn2)C(=O)NCCCN(C)C)CCC(N(C)C)C1C Cc1ccc(C(=O)NC2CC(CNC(c3c[nH]nc3C)=O)C2)cc1[N+](=O)[O-] C1(C(N2CCCC2c2ccc(F)c(Br)c2)=O)C2CCC(C2)N1Cc1cncs1 Cc1ccsc1CC(=O)NOCC(=O)N(CC(C)O)CC(C)O.NC S(=O)(=O)(c1cc(C(=O)N(CC(C)O)CCNC(=O)C2=C(C#N)CCC2)co1)NC C1(CNC(C(C)n2ccnc2)=O)Cc2ccccc2CN1C(=O)CSC(F)F N1(C(C2CC(=C)C2)=O)CCCC(F)(C(=O)N(CC(O)CO)CCO)C1 C(=O)(CCP(C)(C)=O)N(C1CCCCN(C(c2ncoc2-c2cccs2)=O)C1)C CC1(C)C2CN(C(=O)Cn3ccnc3)C(C(=O)NCC(F)Cl)C12 C(=O)(CC(C)(C)C(F)(F)F)N(C1CCN(C(=O)C(C)C(O)CC)C1)CC C1(CCNC(c2c(C)cno2)=O)C(C)CCCN1C(c1cnc(O)cc1C)=O c1(C(=O)NC2CCC(NC(C(COC)(F)F)=O)C2)cccc2ccncc12 c1(C(N(C2CCN(C(=O)C(C)n3cnnn3)CC2)CCC)=O)cc(C)c(CC)s1 C(=O)(C1=C(Cl)CCC1)NCC1C2CN(C(c3c(C)[nH]cc3)=O)CC21.c1(C)ccccc1 C1(C(N2CCCC(CNC(COC)=O)C2)=O)Cc2nnsc2S1 C#CCC(C)(C(=O)N1CCC(C(=O)OC)C1C)NC(c1cnccc1C)=O N1(C(C2N(C(N)=O)CCC2)=O)CC2CC2(NC(c2cc(C3CCC3)on2)=O)C1 c1(NCC2CCC(C(=O)Nc3ccccc3F)C2)cc(CO)ccc1[N+](=O)[O-] C=Cc1cncc(C(=O)NC2CC=CCC2C(=O)NCCCC(=O)NC)c1 CC1(C)CN(C(C2CC3CC(O)CC(C2)C3)=O)CC2(CN(C(=O)CNC=O)C2)O1 Cc1nc2cncc(C(=O)NC3CCC3CNC(=O)CSCCN(C)C)c2[nH]1 CCC(CC(C)CO)NC(=O)CCC1CCN(C)CC1 C1(CNC(c2cnc(CNC(C3C(C)CC3)=O)nc2)=O)CCn2nccc2C1 CCCC(C)(C)C(=O)N1CC(CNC(c2cc(OC)no2)=O)C(F)(F)C1 Cc1n[nH]c(C)c1C(C)C(=O)NCCOC1CCN(C(C2OCCC2(C)C)=O)C1 C1(C(=O)N)CCC2(CCC3(CC2)OCCO3)O1.C1(C(N)=O)CCCN1C c1(C(=O)NC2(N=[N+]=[N-])CCN(C(C(C)O)=O)C2)cccc2c1nc(O)n2C c1(C(=O)NC2CC(C)(NC(Cc3c(C)ccs3)=O)C2)ccc(C(F)(F)F)cc1O N1(C(C2CCCSC2)C(=O)NCCCC)CCC(C(N)=O)c2ccccc21 C1(C(N(CC(C)CNC(=O)CCOCC(F)(F)F)C)=O)COCCC1(F)F C1(C(C)C(=O)N(CCC#N)CCOC(F)F)(C(=O)O)CCCCO1 N1(C(C(c2ccccc2)NC(C(C)C(F)F)=O)=O)CC(CO)C2(CC2)C1 N1(C(c2n(C=C)ncc2)=O)CCn2ncnc2C1.C12CC(C1)OCC(=O)N2 C1(NCC=O)CCCC1.C(=O)(C(=O)NCCOC)NC1CC1.C12(CC1)N(C)C2=O Cc1cccc2[nH]cc(-c3cc(C(N4CCc5nncn5CC4)=O)n[nH]3)c12 C=CC1(CC(=O)NC(CN(C)C(C2CCCS2)=O)CC)CCCCC1 c1(OC)cc(C(=O)N(CCCCN(C)C(C2CCN(C)C2C)=O)C)cc(F)n1 N1(C(CCCCN(C)C)=O)CC2(CCCC2)C1C(N1CCC(F)C(O)C1)=O C(=O)(C1=CC(O)CCC1)NCC(C)NC(=O)CCN(CC(C)C(C)C)C C1(NC(c2cnn(C(C)C)c2N)=O)CN(C(=O)Cc2ccno2)CCC12CCC2 C1(C(C)NC(c2sccc2C2CC2)=O)CCCN(c2cc(Cl)ncn2)C1 C(=O)(C1CCCn2cncc21)N(CCCNC(C1C(=C)C1)=O)C(C)C C1(C(=O)NCC(C)N(C(C=CCC)=O)C)Cc2ccccc2OC1SC1CC1 C1(CNC(C2CC3CCC2O3)=O)CCCCN1C(=O)COCC1CCCC1 c1(CC(N2C(CC(=O)Nc3cc(Br)ccc3I)CCC2)=O)cc(F)ccc1F N1(C(c2c(C(F)(F)F)cn(C)n2)=O)C2CCC1CC(CNC(c1cn[nH]c1)=O)C2 c1(CNC(C(C)OCCn2ncc(CN)c2)=O)cc(C(=O)OCC=C)cs1.CC c1(CC)nc(C)cs1.c1(CCC)nc(-c2cc[nH]n2)n(C2CCC2)n1 CC1(CC(=O)Nc2cnn(CCF)c2)CCN(C(=O)CC2(CN=[N+]=[N-])CC2)C1 c1(CC)ccc(C2CCN2C(C(=O)OC)C(C2CCCC2)OC)cc1 C(=O)(C(C)CCCOC(F)(F)F)NCCn1cc(C2C(C)CCN2CC)nn1 c1(C(N2CC(N(C(Cc3c(C)non3)=O)C)C2)=O)cccc2c1NCCNC2=O N1(C(C=CCC)=O)CCC2CCC(NC(=O)Cc3cccnc3)C1C2 CCCCCCC(C)CC(=O)NCC(C)CNC(c1oc(CC)cc1C)=O CC1CN2CCN1C(NC(N1CCN(c3ccc([N+](=O)[O-])[nH]3)CC1)=O)C2 C=C(C)C(CC(=O)NCCC(C)(C)NC(c1ccnnc1C)=O)OCC N1(C(CCc2cc(C)[nH]n2)=O)CC2CC1CN(C(C1OCCOC13CCC3)=O)C2 c1(OC)cccc(CCC(=O)NCC2CCN(C(=O)CCSCC(C)C)C2)c1F CC1C(C(=O)N(CC(C)N(C)C(C2(C)CCC2)=O)C)C1C C1(NC(C2CCCC(O)C2)=O)CN(C(c2cccnc2O)=O)CC12CCC2 C(=O)(CCCC(F)F)NCC(C)(C)NC(C1CC(C)(F)C1)=O C1(C(N2C(COC)CCCC2)=O)COC2CN(C(=O)CC(C)(C)C(=O)OC)CC12 C#CCCCN=C(NCCCN(C)C)N(C)Cc1ccc(F)cc1 Cc1csc(COC(C)C(=O)NCC(C)NCCc2cnco2)n1 Cc1cc(=NCc2cccc(OCC(C)C)c2)nc(Cl)[nH]1 C1(C(N(CC#C)CCO)=O)CC12CCN(C(C1CCC3(CCC3)C1)=O)CC2 C1(C(=O)NCC(=O)N(C)C2CC2)CCNC(C2CC2)C1 C=CCCN=C(NCc1ccc(CSC)cc1)NC(C)C.c12nc(no1)C2 CCCCC(CC)CCC(=O)NCC(N1CCN(C(C2(OC)CC2)=O)CC1)=O CCC(C(N)=O)N(C(=O)C(C1CCCCC1)=O)Cc1cn(C(C)COC)nn1 C#Cc1cc(OC)ccc1C1OCCO1.C1(CC)(CCCC)c2nnnn2N1 N1(C(C2CC(N(C)C)C2)=O)CC(C)(C(N2CCC(CO)C(O)C2)=O)CC1(C)C c1(C(C)NC(CC(C)NC2CCN(C(CC)=O)C2)=O)ncccc1Cl CCC(C)C(CNC(C1COCCN(C(=O)Cc2ccc(C)cc2)C1)=O)CO c1(C(=O)NCCN(CCC)CCC)ccc(C(C)(C)C)[nH]1 C(CC(F)F)(C(=O)N(C1CC2(CC2)C1)C)NC(c1cc(C)no1)=O Cc1ccc(C=CC(=O)NCC(O)CNC(c2cnc3n2CCS3)=O)nc1 C1(NC(C2(OCC)CCC2)=O)CC2CCC1CN(C(C1CC=CC1)=O)C2 O=C(NNc1cc(Cl)cc(Cl)c1)C1CCC(O)(C2CC2)CC1 c1(C(N(CCOCCNC(C2CC(O)(CC#C)C2)=O)C)=O)ccc(CC)nc1 C1(NC(C(CO)OC)=O)CCC2CC1CN2C(=O)C(C)Sc1ccccn1 N1(C(c2[nH]c(C)c(C(=O)O)c2C)C)CCCC2(C1)OCCO2 C1(C(=O)OC)CN(C(=O)NCC(C2CCOCC2)(F)F)C2(CCCC2)C1 CC(=O)C(C)(C)CC(=O)NCC1CN(C(c2cc(C)nc(O)n2)=O)CC1C CCC(CC)=CC(=O)NCC=CCNC(=O)C(C)c1ccco1 N1(C(CCC(=O)NC)=O)CC(C(=O)NC2CC=CC2)C(F)(F)C1 C(=O)(C(C)CN(C)C)NCCN(C(C)=O)C.C(=O)NCC Cc1cc(C(N2CC(NC(c3cn[nH]c3)=O)C(C#N)C2)=O)cc(O)n1 C1(CNC(c2cncc(F)c2)=O)CN(C(=O)C=Cc2cccs2)CCO1 c1(CC(N2CC(C)C(NC(=O)C(C)CF)CC2)=O)ccc2ccccc2c1 c1(SC(C(C)C)C(=O)N2CCC(O)C2)ncc(Br)c(O)n1 N1(C(c2cnccc2Cl)=O)CC2OCCN(C(C3CC3C(F)F)=O)C2C1 C(=O)(C#CC1CCCO1)N1CCN(CC(C)NC(C2(C)CCCC2)=O)CC1 N1(N(CCC=O)CC=C)CCCNC(=O)C1C.c1(C=O)cn(C)cn1 CCC(CN=c1[nH]c2c(c(=NCCC3COCCO3)[nH]1)SCC2)OC C#Cc1cccc(C(=O)NCCCCCC(=O)N(C)Cc2cnnn2C)c1 S(=O)(=O)(c1cc2sc(=NCc3ccncn3)[nH]c2cc1Cl)N(CC(CCC)C)C C(=O)(CCCCCN(C)C(c1c[nH]ccc1=O)=O)NC(c1ccoc1)C C(c1ccc(Cl)nc1)=CC(N1CC(CNC(C2OCCN(C)C2)=O)OCCC1)=O Cc1nc(N2CCC(=CCNC(C34CCCN(CC3)C4)=O)CC2)[nH]c(=N)n1 N1(C(c2c(OC)scc2)=O)CCC(CC(=O)NCC(CO)C(C)C)C1(C)C N1(C(Cc2nc(C)sc2)=O)CCc2ccc(-c3ccnc(C#N)c3)cc2C1 C1(CCC(N2CC(C(N)=O)(CNC(C(=C(C)C3CC3)F)=O)C2)=O)CCCN(C)C1 S(=O)(=O)(c1cccs1)NCCC(=O)N(C)CCNC(=O)CC1CCCC12CC2 C1(C)(C(N(C2CCN(C(=O)C(C)SC)C2)CC)=O)CCCN1C(C)=O c1(C(C)C(=O)NCCCNC(=O)CCn2cc(Cl)cn2)cc2ccccc2o1 C1(C(C(=O)NCC)N(CCC#N)C2CC2)CC2CC(OC)C2C1 Cc1nc(N)cnc1C(N1CCC1CNC(=O)C(c1ccccc1F)(C)F)=O Cc1c(C(=O)NCC(C)NC(=O)C(C)N(C)C)cc(O)cc1N N1(C(c2nc(C)n(C)n2)=O)CCC(CO)(NC(c2coc(C3CCC3)n2)=O)CC1 C12(NC(c3cc(C)c(C)nn3)=O)CCN(C(c3cccc(F)c3C)=O)CCC1C2 C(=O)(CCNC(=O)Cn1cccn1)OCC(=C)F C12(C(=O)NC3C(CNC(C=CC=CCC)=O)CCC3)CC(C)(CO1)C2 c12nc(ncc1Br)NC2=O.CC1CCN(C(=O)C(=O)NC(CC2CC2)CO)C1 c1(C(N2CCC(NC(c3cc(Br)c(Cl)cc3F)=O)C2)=O)cncc2ccccc12 C1(N)CCCCCC1.c1(C(N2CC3CCC2C3)C(=O)NC)nn(CC(F)(F)F)cc1Br C1(CN(C(c2cn(CC(C)O)nn2)C(=O)NCC(C)C)C)CCCC(C)(C)CC1 C(CCCCCCN1CCCCC1)NC(CCCNC(C(C)C)=O)=O C1(C)(C(N(C)Cc2nc(CC)sc2)=O)CCCN(CCSCOC)C1 C1(C(=O)NCC2N(C(c3c(CC)con3)=O)CC2)(CC)CCCC1O CCCCCCCCNC(C1CCN(C(=O)C(C)OC(C)=O)C1)=O C#Cc1cc(C(=O)NCC(C2CC2)N(C(=O)C(CCC)NC(N)=O)C)ccc1Cl C12(C(N3C(CNC(CN4CC(C)(OC)C4)=O)CC(O)C3)=O)CC1COC21CCC1 Cc1ccc(=O)n(CC(N2CCC3(NC(=O)Cc4csc(C)n4)CC3C2)=O)c1 C1(CCNC(C2(CC3CCC3)CC2)=O)CCCN(C(=O)CN2CCOCC2)C1 c1(C(=O)NCCCCCCN(C(=O)C2=CCSC2)C)cc[nH]c2nccc1-2 c1(C(=O)NC(C(C)NC(C2CC(C#C)(O)C2)=O)C(C)C)cc(C)c(F)cc1Cl CC1CN(C(c2ccoc2Cl)=O)CCC12CCN(C(C1CCCCCC1)=O)CC2 c1(C(=O)NC2CC3CCC2(CNC(C24CC(CO2)C4)=O)C3)ccc2nn[nH]c2c1 c1(OC)cccc(CSC(C)C(N2CC(O)(C(C)NC(=O)CC3CCC3)C2)=O)c1 C=CCC(CNC(C1CC(n2ccnn2)C1)=O)NC(C1CCCSC1)=O c1(C(=O)OCC)ccc(NC(C2(C)CCN2c2nc(SC)ncc2Br)=O)cc1C C=CCC(C)(O)C(=O)NCC(C)=CC(=O)NCc1c(C)coc1C c1(C(=O)NCCN(CCCN(C)C)C(c2c(C)cns2)=O)nccc(C(F)F)n1 c1(C(=O)NCC2(C)CCN(C(C3(Cl)CC3(F)F)=O)C2)cccc2c1CCCC2 Cc1cc(C(=O)NC(CNC(c2ccc(Br)cn2)=O)CC(C)C)sc1Cl n1(CC)nc(C)cc1C(N1CC(CNC(c2ccnc(C3CC3)n2)=O)C(C)C1)=O c1(C(N(C(C)C(=O)NCC2(C(=O)OC)CC2)CCC)=O)cnn(C)c1C#N c1(CC(=O)NC2CCC(NC(C3CC(OCC)C3)=O)C2)c(C)nn(C)c1Cl C(=O)(CCCCC(N)=O)N1C(C(N2CCC(C)(O)C2)=O)CC1 CC1CCC(NC(c2csc(Cl)c2Cl)=O)CN1C(=O)CCCCCF C#Cc1ccc(F)c(C(=O)NCCCN(C)C(C2CC3(C)CCC2(C)O3)=O)c1 CCC(C)CC(C(=O)NC(C)CCSC)NC(=O)C(C)COC C(CCCO)(C(C)C)NC(C(C)N(C(c1nonc1C)=O)CC)=O c1(NC(=O)C(=O)N(CC(CN(C(C(=O)NC)C)C)O)C)ccc(C(C)(C)C)cc1 c1(NC(CNc2c(COC)onc2C)C)ccc(C#N)cc1 c1(C(CO)NC(c2cnn(C3CN(S(=O)(=O)CCCCl)C3)c2)=O)cccc(Cl)c1 Cc1nn(CC(=O)N(C2CCN(C(=O)Cc3c(O)ncnc3O)C2)C)c(=O)n1C N1(C(=O)Cc2csnn2)CCC2(CC1)CC(C(N1CC3(CNC3)C1)=O)C2 N1(C(c2cn(CC)nc2)=O)CCC2(CC(NC(c3ccnnc3Cl)=O)C2)C1 CC(C)(CS(N)(=O)=O)C(=O)N1CCCC2(NC(=O)CS(C)(=O)=O)CC2C1 CCC(C)(C)C(O)C(=O)N1CCC(c2cn(-c3cc(Cl)c(F)cc3Cl)nn2)C1 CC1=CC(C(=O)N(C(C)CN(C)C(c2cn(CC(N)=O)nn2)=O)C)SC1 C1(NC(c2cnc(C)[nH]2)=O)CC2CC1N(C(=O)CN1CCC(O)CC1)C2 N1(C(CC=CC)=O)CC2(CC(NC(=O)C(CCCC)N(C)C)c3nccn32)C1 CCCC(C)(O)CC(=O)NC(CNC(c1ccc(=O)n(CCO)c1)=O)C(C)(C)C c1(C(N)=O)nccnc1C(=O)NCC1CCCCN1C(=O)CCN1CCC(F)C1 c1(C(N2CC(N(C)C(c3csc(S)n3)=O)C(F)C2)=O)ccn(C)c(=O)c1 C(=O)(C1=C(Cl)CCCC1)NC1(CF)CCN(C(Cc2cc(C)sc2)=O)C1 c1(C(N2CCC(CNC(CSC)=O)C(C)C2)=O)cc2c(C(C)C)nn(C)c2s1 C12(CCNC(C(Br)=C(C)C)=O)CCC1CN(C(c1cnc(C3CC3)[nH]1)=O)C2 C1(CN(C(C(Cn2ccc(C)n2)C)=O)C)CN(c2nnc(C(C)(C)C)s2)CCO1 C(c1ccccc1C#N)=CC(=O)NCC12N(C(C=C(CC)CC)=O)CCC1CC2 CC1(C)CN(C(=O)Cn2c(O)nnc2O)CC1NC(=O)CNC(=O)C(=O)O C1(CN(C(CCCC)=O)CC)CCCN(C(c2ccccc2SC(F)F)=O)C1 CC1CCC(C)(C(N2CCCC(NC(=O)CCCN3CCCC3)C2)=O)CC1 c1(C(C(=O)NC(CN(C(C(CC)O)=O)CC)C)O)ccccc1C(F)(F)F CN1CCN(C2CCN(C(=O)CC(=O)N(C(=O)CCCn3ccnn3)CCl)C2)CC1 CC1(C)CC(NC(=O)C#CC2CCCC2)CN(C(C2CN3CCC2CC3)=O)C1 c1(CN2C(CN=[N+]=[N-])CCC2)ccc(-c2cccnc2O)cc1 C(=O)(C(C1=CCCSC1)N(CCCO)Cc1ccccc1)NCCCOC c1(C(N2CCC(CC=C)(NC(C3CC3(F)F)=O)C2)=O)c(C)nc2ncnn2c1C N1(C(c2cc(CCOC)on2)=O)CC(C2CCCN2C(C2(OCC)CCC2)=O)C1 Cc1cc(C(N2CCN(CCNC(=O)CC3CCC(C)(C)C3)CC2)=O)nn1C N1(C(C2CC(OCC)C2)=O)CCCC12CCN(C(c1cccc(CO)n1)=O)C2 C1(NC(C2(SCC)CC2)=O)COC2(C1)CN(C(C1C3CCCC13)=O)C2 c1(NC2C(C)(C)CN(C(C3CC(F)C3)=O)C2)ncnc2c(Br)cccc12 C1(NC(=O)CCCN2CCCC2)CCCN(C(c2sccc2C(F)F)=O)CC1 c1(C2CCC3(C(N4CCCN(CC)CC4)=O)C2CC3)cc(F)cc(N)c1N N1(C(C2C(C=C)OCC2)=O)CCOC2(C1)CN(C(C1CCCC1C(=O)OC)=O)C2 C#CCC(C)(CNC(=O)CC(C)C(=O)OC(=N)O)CO.O(C(F)(F)F)CC=O C(=O)(N=c1ccn(Cc2cccc(Cl)c2)[nH]1)c1c(C)ccs1 N1(C(C2(C#N)CCCO2)=O)C(CC(N2CCC(O)C(F)C2)=O)C2CCCC12 C1(SCC)CN(C(CC)C(=O)N2CC(C)(C(=O)N(CC)CC)C2)CCO1 c1(OC)nccc(C(=O)NC2CCN(C(=O)CC3CSCCS3)C2C)c1F CC(C)C(O)(C(=O)NC1CCC1NC(c1cnc(C2CC2)o1)=O)C(F)(F)F C(=O)(C1=CCCCC1C)NC(C1CC(NC(c2ccc(C)nc2O)=O)C1)C N1(C(C(CN(CC)CC)F)=O)CCC2(C1)CN(c1ncnc3sccc13)C2 c1(C(=O)NC)ccc(CN(CCCNC(C2C(C)CC2)=O)C2CC2)o1 c1(C(=O)OC)sc(NC(C)CCN2CCCC2)nc1Cl.C(C)(C)O CCCCC(CC(=O)N(C)CCn1cccn1)NC(C1CCC1CO)=O c1(C(N2C(CN(C(CC(C)SC)=O)C)COCC2)=O)cc(C)nc2c1CCCC2 C1(CCOC)CN(C(c2sccc2C)=O)CCN1C(=O)C(CCOC)OC C(=O)(C1=NOC2COCC12)NCC1N(C(C(CC)CN(C)C)=O)C2C(C1)CCC2 N1(C(COC(CC)CC)=O)CCCC(C)C1CNC(c1cccc(C(N)=O)n1)=O C(CC(C)(C)C)(C(=O)N(C(C(=O)NCC(C)CCO)C1CC1)C)OC N1(C(CCN(CCCCC)C)=O)CCN(C(c2cc(Cl)sc2Cl)=O)CC1CC C1(C(C)NC(C2CCS2(=O)=O)=O)CCCN(C(C2(CC3CC3)CC2)=O)C1 c1(CCCC=C)cn(C2(NC(C3C=CCC3)=O)CCOC2)nn1 C1(NC(=O)C(c2ccccc2)=O)CN(C(C2CSCCS2)=O)CC2CC12 C12(C(=O)NCc3n(C)c(Cl)nc3)CN(C(=O)OC(C)(C)C)CC1CCO2 C1(NC(c2nnc(CC)s2)=O)CC(C)N(C(=O)Cc2sc(C)nc2C)C1 C1(CC(=O)NC(COC)CO)CN(C(C2(OC)CC2)=O)CCO1 N1(C(C2CCC(CCCC)CC2)=O)CCN(C(c2cc(C)sn2)=O)CC1C(C)C CC1CN(C(c2ccc([N+](=O)[O-])s2)=O)CCC1C(=O)NCCCNC(N)=O C(C(C(C)(C)C)NC(=O)Cc1ccc(F)cn1)NC(C(C)SCCCC)=O C1(NC(=O)CCSCC2CC2)CS(=O)(=O)CC1NC(=O)C(F)(F)C1CC1.C(=O)(CO)N c1(N2CCOCC(=C)C2)nc(NCCc2ncccc2I)c2cnn(C)c2n1 Cc1nc(NCCCc2cn(C)cn2)cc(=NCC2C(C)(C)C2(F)F)[nH]1 c1(OC)cc(C(=O)NC(C)CO)c(NC(c2cc3sccc3s2)=O)cn1 C(C(CNC(c1cc2c[nH]nc2s1)=O)C(F)(F)F)NC(C(CC)(C)O)=O CN1CCN(C(=O)CC2CCNC2=O)C(CNC(=O)CNc2cccnc2)C1 CC#CCCC(=O)N1CCC(F)C(O)C1.C(=O)C(F)=CC C1(C(C)NC(=O)C(F)CC2CCOC2)CCCN(C(C2(C#N)CC=CC2)=O)C1 C1(C(=O)NCc2c(C(N(C(CC)CC)C)=O)n(C)nc2)CC2(CCC2O)C1 c1(OC)ccc(C=CC(=O)NC2(C3CCCN3C(c3cccc(Cl)c3)=O)CC2)s1 c1(CC(=O)OC)cc(Br)c(C)cc1NC(=O)CSc1nc(-c2cccs2)no1 C1(NC(c2c(C)c(C3CC3)on2)=O)CC2CC1N(C(=O)C=C1CCN(C)CC1)C2 N1(CC)CC(C(=O)NCCNC(c2cnn(C)c2C(F)F)=O)NC1=O c1(NC2CCN(C(=O)OCC=C)C2)ncnc(N2CCOC(CF)C2)c1C CCCCCC(O)CC(=O)NC1CCN(C(c2ccc(CSC)o2)=O)C(C)C1 N1(C(C(CCC)Cl)=O)CC2(CC(NC(c3ccc4cccnn34)=O)CO2)C1 N1(C(c2cccc(C(C)C)c2)=O)CC2(C1)CN(C(C1CC1F)=O)CC2CO C1(C(=O)N(C)CCOC2(C(=O)NC)CC2)CCCN(C(=O)C(F)OC(F)(F)F)C1 C1(NC(CC2(OC)CCC2)=O)CC2CCC1CN2C(c1coc(C2CC2)c1)=O Cc1cc(C2CCC2)ccc1C(=O)NC1CC(N(C)C(c2cncnc2)=O)C1 C1(CNC(C2N(CC)CC2)=O)CCN(C(c2ccccc2)=O)CC1.C(C)(=O)N c1(C(=O)Nc2cn(COC)nc2)cc(S(N)(=O)=O)oc1C c1(CCCC(=O)N(CCCNC(C2(CCC=C)CCOC2)=O)C)ccc(O)cc1 c1(C(=O)NCC2N(C(C=C(C)C3CC3)=O)CC(O)C2)cc(O)cc(O)n1 C1(CC(=O)N(C2CC(NC(C(C)OCCOC)=O)C2)C)CCC(C)(C)O1 Cc1nc(C(N2CCC(CN3CCN(C)CC3)CC2)C(=O)NCCO)c(Br)[nH]1 c1(C(N2CCC(C)(C(N3C(C#C)CCCC3)=O)C2)=O)cc2ccccn2c1 N1(C(c2cc(C)nn2C)=O)CC2CN(C(=O)C(O)CC(F)(F)F)CC2C1 Cc1oc([N+](=O)[O-])cc1C(N1CC2CC(NC(c3cc(Cl)c(Cl)[nH]3)=O)CC1C2)=O CCC(C(C)C)C(C(=O)NCC(F)F)N1CCc2sccc2C1 CCC(C)(C)C(=O)C(=O)NCC(C(=O)NC(c1ccc(O)cc1)C)N(C)C CN1CCC(C(=O)NC(CCO)C2CCCC2)(NC(=O)Cc2cscn2)C1 n1(C2C(C(=O)OCC)C2)cc(C(C)C(=O)NCCSC(C)(C)C)nn1 c1(C(=O)Nc2cccc(F)c2)cccc(S(=O)(=O)N2CC3CCC2CNC3)c1 C(=O)(C1CCc2ccccc21)N1CCC(C(N2CC(CC)NC(=O)C2)=O)(CC)C1 Cc1ccc(F)c(C(=O)NCC2CCCCN2C(=O)Cc2ccc(O)nc2)c1Cl c1(OC)ccccc1CN(C)C(C1CC2CC2N1C(=O)CCc1ccncn1)=O c1(C(=O)NC)ccc(OC)c2ccsc12.c1(C(C)CC)noc(CNC)n1 Cc1cscc1C(N1CCC(CN(C)C(C2(CN(C)C)CC2)=O)C1)=O C1(NC(C2(N)CCCNCC2)=O)CCOC2(CCCOC2)C1 C(c1cnn(C)c1C)=CC(=O)NC1CN(C(C(NOC)=O)=O)CC1SC C1(C(=O)NC2C(NC(CN(C3CC3)CC)=O)C2)CCN(C2CCCCC2)C1 C(=O)(C#CC(C)(C)O)NC(CNC(c1nn(C)c(O)c1)=O)C(C)(C)C C1(N(C(=O)Cn2nnc(C(C)(C)C)n2)C)CCN(C(c2cn[nH]c2)=O)CC1 N1(C(C2N(C)CCC2)=O)CCCC12CCC(NC(c1cc([N+](=O)[O-])n[nH]1)=O)CC2 c1(OCC=C(C)C)ccc(NC(C2CCN2C(c2[nH]c(O)nc2C)=O)=O)nc1 c1(N2CC3C(C)(C)C3C2)nc(=NCCC#CBr)[nH]c2ccsc12 C1(C(=O)NCC2CC(C)N(C(=O)CNC(=O)OC(C)(C)C)C2)CCCCN1N=O C(=O)(C1=CCC(C)CC1)n1c(N2CCN(CC)CC2)nnc1-c1cn(C)nc1C c1(C(N(CC(=O)NCCC(C)(F)F)C2CC2)=O)c[nH]ccc1=O CC1(C)CCCOC1C(N1CCOC(CNC(C2CC(F)(F)C2)=O)C1)=O C1(NC(C2ON=C(CC)C2)=O)CCN(C(c2ccc(OC)c(C)c2)=O)CC1F CCCC(C)C(=O)NC1CCCC(NC(=O)CN(C)Cc2ccc(C)cc2)C1 C1(NC(C(Cc2ccco2)NC(C(CCC)OCC)=O)=O)CCC(=O)N(C)C1=O Cc1ccc2sc(C(=O)OCC(c3ccc(Cl)cc3Cl)=O)nc2c1 N1(C(c2c(CC)noc2)C(=O)NC2CCC2)CCC2CCC(C1)S2(=O)=O N1(C(C2CC(NC(c3cccc4nccn34)=O)C2)=O)CCOC2(CCNC2)C1 c1(OC(C)=O)ccc(Br)cc1C(=O)NC1CCCC1NC(c1cnc(C)s1)=O c1(C(c2nnnn2C2CC2)NC(C2CCCCC2)CC)ccccc1SC(=O)OC c1(C(C(=O)NCCSCC)N(CCc2ccc(F)cc2)CC)ccnnc1C C1(Cn2cc(CC3CCCO3)nn2)CC2CCC(C1)N2Cc1c(C)ccc(C)c1 N1(C(C2(C)CC(=C)C2)=O)CC(O)(C2(CNC(c3cc4cnn(C)c4s3)=O)CC2)C1 N1(CC2(C(=O)OC)CC(=C)C2)CC(O)C(O)C1CO.c1(C(=O)N)nccc(C)c1F c1(C(N(C)CCNC(=O)CCc2cc(Cl)no2)=O)ccc(C(F)F)cn1 C1(OC)CC(NC(=O)COCC(F)F)CN(C(=O)C(N2CCNC2=O)C)C1 c1(C(=O)NC(C(CO)NC(C(CCC)O)=O)C)cc(C)n(-c2ccn(C)n2)c1C CCCC(C)(C)CC(=O)NCCCC1CCCN1C(=O)C(CCSC)OC c1(C(=O)NCC2CC(NC(C(CC(C)C)(C)O)=O)C2)nccc2ncccc12 C12(NC(c3c(C)nsc3)=O)CCCC(CN(C(=O)C(F)n3ccnc3)C1)C2 C1(NC(CCOCC#C)=O)CN(C(c2ccc(C3CC3)s2)=O)CC1S(C)(=O)=O C1(NC(C(C2N(C(c3cn(CC)nc3)=O)CCC2)(C)C)=O)CCCC(C2CC2)C1 C1(CNC(C(C)n2ccnc2)=O)CC(F)CN1C(=O)COCc1ccnc(O)c1 CC1CC=C(C(=O)NCC(c2ccccc2)NC(=O)Cc2nc[nH]n2)CC1 Brc1cccc(CCNCc2cn(C3CCCC3)cn2)c1 c1(OC)cnc(C(N2CCN(C(C3CC3(C)C(C)C)=O)CC2)=O)c(F)c1 CCN=c1[nH]c(C(=O)NC2CCCC2NC(c2ccc(OC(F)F)cc2)=O)cs1 N1(C(c2c(CC)ccs2)=O)CCC(C2CN(C(c3ccc(NC)cn3)=O)C2)CC1 CC(CN=c1nc2scnc2c(NC2CC2)[nH]1)C(C)(C)C c1(C(N(C2CCC2)CC#C)=O)coc(CNC(=O)COC2CCOC2)c1 N1(C(Cc2nn(C)c3c2cccc3)=O)Cc2ccccc2C2CC1C2 Cc1cc(C(N2CC3(CCN(c4ccc(C(F)(F)F)nn4)C3)C2)=O)c(C)cc1Cl C1(=CC(=O)NC2(CO)CCN(C(C3C=CCC3)=O)C2)CN2CCC1CC2 C(=O)(C(O)P(C)(C)=O)CCCN(CCCN(C(CC(OC)ONC(=O)NC(C)C)=O)C)C N1(C(C=CC)=O)CCC(NC(=O)C=Cc2cc(Cl)cc(Cl)c2)CC1C1CC1 C1(O)(C(N2C(C(=O)NC(C(=O)OC)C)CC(F)C2)=O)CCCCCC1 S(=O)(=O)(c1ccccc1)CCNC(=NC)NCC1COC1 N1(C(C2C(C)OCCO2)=O)CCC(O)(CNC(c2cc[nH]n2)=O)CC1 CC1CC(CNC(c2ccc(C(C)(C)C)o2)=O)CN(C(C2CCC(=O)O2)=O)C1 C(=O)(N1CC=CCO1)C1C(NC(CNC(c2ccc(C3CC3)o2)=O)=O)CCC1 N1(C(CCC=CC(C)C)=O)CCC(C)C1C(=O)NCCC1CCCCCC1 CC(C)CCCC(=O)NCCCCC1CN(C(c2cnc(N)cn2)=O)C1 CCCC(CNC(=O)Cc1cccc(O)c1)C(=O)NCC1CC12CCC2 c1(C(=O)NC(C(C)C)CNC(=O)C(c2cccn2C)=O)ccc(C#N)o1 C1(N(C)C)CCC2(C(=O)NC3CCCCC3C(=O)NC3CC(N(C)C)C3)CC12 c1(C2(C(=O)NCCC3CN(C(C(=O)NC)=O)CC3C)CC2)cccc(F)c1F c1(CCNC(=O)Nc2c(C)cc(C#N)cc2)cn(C)c2ccc(F)cc12 N1(C(C2CCC(C)O2)=O)CCC2(CCCN(C(c3nc(Br)cs3)=O)C2)C1 C(=O)(CCC(F)(F)F)NC(C)C(CO)NC(C1CC(=O)NC(=O)C1)=O CCCC(CC)CCC(=O)N1CCCC(C(=O)NC(C)CO)C1 CC(C)(O)C(F)C(=O)NC(C(=O)N(C1CC1)Cc1nc[nH]n1)C1CCC1 C1(C(=O)NC(CCOC)CNC(c2ccc(CN(C)C)o2)=O)CCN(C)S1(=O)=O c1(C(=O)NC23C(CN(C(C4C(=C)C4)=O)C2)CCOC3)c(O)cnc2ccccc12 C1(C)(OCC(=O)NCC2CC(CNC(c3ncn(CC)n3)=O)OC2)CCOCC1 Cc1cc(C(=O)N(C)CCN(C(=O)CC2CCC3CC23)C)ccc1[N+](=O)[O-] N1(C(c2cc(C)c(F)nc2)=O)CC2CCN(C(c3cc(I)c(F)cc3F)=O)C2C1 C1(NC(=O)NCCN(c2nc(Cl)nnc2Cl)C)CC2C=CCC(C1)C2 c1(C(=O)NCC2CC(NC(c3c(F)ccc(SC)c3)=O)C2)cc2nc[nH]c2cn1 N1(Cc2n(C)ccn2)CC2CN(C(c3cc(O)c(O)c(O)c3)=O)CC2C1 c1(C(N(CCCN(C(=O)CC2CC=CC2)C)C)=O)cc2ccsc2n1C O=C(C1=NN(C2CC2)C(=O)CC1)NCC1(F)CCN(C(C2CC23CC3)=O)C1 N1(C(c2cc(Br)ccn2)=O)Cc2ccc(-c3ccc(CN4CCCC4)s3)cc2C1 C1(NC(C=CSC)=O)CCOC12CCN(C(=O)C(=Cc1cccnc1)C)CC2 N1(C(CC(=C)C)=O)CCC(CO)C(NC(c2csc(COc3ccccc3)c2)=O)C1 N1(C(CC=CC)=O)CC2(CCC2NC(c2cc(C3CCOCC3)[nH]n2)=O)C1 Cc1cnc(C(=O)N(C2CC(NC(C3CC4CCC3O4)=O)C2)C)cc1Br C(=O)(N=c1nc(C)nc2[nH][nH]cc1-2)C1CC(=C)CN1Cc1cc(Cl)cnc1Cl n1(CC)cc(C(=O)N(C)CC2C3CN(C(=O)C=Cc4ccncc4)CC23)c(C)n1 Cc1cnc(C(=O)NC(CNC(c2ccns2)=O)C2CC2)cc1C c1(OC)ccc(S(=O)(=O)NC2CCCN(S(C)(=O)=O)C2)cc1NCC1(C)CC1 c1(NC2CN(C(C)=O)C2)ccc(S(=O)(=O)N2CCC3CC3C2)cc1C#N N1(C(C(=O)NC(C)C)=O)CCN(C(=O)CCC2OCCO2)CC2CCCCC12 C(c1ccccc1C)=CC(N1CCC(C(=O)N(C2CCSC2)C)(OC)C1)=O c1(C(=O)NC(C(C)NC(=O)Cc2cnns2)C)cccc(-n2cncn2)c1 CC(C)CCC(F)C(=O)NC1CC(C)(C(=O)NCC2CC3CCC2C3)C1 C1(C(=O)NCC(C)OCC)COC(CNc2ccccn2)C1 CC1C(NC(c2ncc[nH]2)=O)CC2CCC1N2C(c1cc2c([nH]1)CCC2)=O N1(C(c2ccc(C(C)C)o2)=O)CCC(C2CN(C(=O)CN3CCS(=O)CC3)C2)C1 C1(NC(CN(C(C)C)C)=O)CCOC(CNC(C23CC(C)(CO2)C3)=O)C1 N1(C(N(C)C)=O)CCC(C(=O)N(C)CCN(C(=O)CN2CCCC2=O)C)C1 c1(CN(C(C(C(C)C)NC(=O)Cc2cccs2)=O)C)ccc(Cl)c(Cl)c1 c1(C(=O)N=c2[nH]nc(C3CCC3)o2)cn2c(-c3ccc(F)cc3)cccc2n1 N1(C(C23CC(COC)(OC2)C3)=O)CCN2CCN(C(C3CC(SC)C3)=O)CC2C1 c1(N(C)C)ccc(NC(C2CCCN2Cc2cc(C(C)(C)C)n[nH]2)=O)c(O)c1 c1(C(=O)NCC23OCC(NC(CCCCC#C)=O)(C2)C3)cc(C)c(O)c(N)c1 N1(C(CCN(C)CC)=O)CCN(C(c2cc(-c3cnccn3)[nH]n2)=O)C(CO)C1 C1(OC)CC(C(=O)NCc2nc(C)sc2C)N(C(=O)CC2(n3ccnc3)CC2)C1 C=C(Cl)C(C)(C)C(=O)NCC1CC1NC(=O)CCCn1cc(C)cn1 c1(N2CCC(CNC(C(CC)(C)C)=O)C2=O)cc(F)cc(F)c1 CCC(O)C(C)(C)C(=O)NC1CCC(CC(=O)NCCCCF)CC1 c1(CNC(C2CSCCN2C(c2cccc(O)c2F)=O)=O)ccnc(Cl)c1F c1(C(N2CCC(O)(CCNC(C3(C)CCN(C)C3)=O)C2)=O)ncn2c1CCC2 C(=O)(C1=CCCCCC1)NC(c1ccc(F)cc1)CNC(c1c(C)onc1)=O c1(OC)cc(C(=O)NC2(CC3CN(C(=O)CCCSC)C3)CCC2)c(N)c(C)c1 C1(CC(N2CCC(CC(=O)NCC3CC(=O)NC3)CC2)=O)Cc2ccccc2O1 N1(C(c2cc(O)nc(O)c2)=O)CCC2(CCCN(Cc3cc(F)cnc3Br)C2)C1 c1(C(N2CCN(C(CC)CO)CC2)=O)cc(C)nc2ccc(OC)cc12 CS(=O)(=O)C1(C)CCCC1C(=O)NC(CNC(=O)CC1CCCC1)CC(F)(F)F CC1(C)C(C(=O)NCCC2(CNC(=O)CCc3ccc(N)cn3)CC2)C1(F)F N1(C(C(C(C)(C)C)SC)=O)CCCN(C(=O)Cc2c(C)cccc2C)CC1C CP(C)(=O)C(O)C(=O)N1CCN(C(=O)Cc2cncnc2O)C(CC2CC2)C1 C(CCC(=O)NCC1(F)CN(C(=O)CNC(C)=O)C1)OC c1(CCCC(N2C(CNC(C(c3ccccc3)C)=O)C=CC2)=O)ccc(F)cc1 N1(C(C(c2cnccn2)C)=O)CCC(C)N(C(=O)C(c2ccccc2)F)CC1 C(c1ccccc1Cl)=CC(=O)NCC1C(CNC(c2c(C)nc(C(C)C)o2)=O)C1 C(=O)(CC(C)C(C)(C)C)NC1CC2C(NC(CCCCOCC)=O)C2C1 CC1CCC(C(N2CC(C)(CCC(=O)N3CC(C(N)=O)C3)C2)=O)O1 CCC(CCOC)C(=O)NC1CC2CC(NC(=O)C=CC(C)(C)SC)C2C1 C1(CN(C(=O)C(=O)Nc2ncc(C3CCOC3)s2)C)CCCC12CC2 C(CCCN=c1[nH]cnc(NCC2COc3ccccc32)c1C)OC Cc1cccc(F)c1CC(=O)NCC(O)CCNC(c1ccc(F)cc1F)=O C1(C(=O)NC2CN(C(c3c(C)snn3)=O)CC2(C)C)C2C3CC4C1C1C2CC3C41 CC1=C(C(=O)NC2CN(C(c3scnc3Cl)=O)CC2C)CCS1(=O)=O C(=O)(C(C)(CO)NC1CC1C(C)(F)F)OCC C1(CC(=O)OC(C)(C)C)CCCC1NC(C1CC(n2cc(-c3csnn3)nn2)C1)=O C(=O)(CCC(C)S(C)(=O)=O)NCC1OCCN(C(c2cncc(SCC)n2)=O)C1 c1(NC(=O)Nc2ccsc2C(F)F)ccc(CC(F)(F)F)cc1 n1(CCN(C)C)ccc(C(=O)NCC2CC(NC(=O)C(C)(C)NS(C)(=O)=O)C2)n1 C1(C(=O)OCC)CC(NC(=O)NCc2nnc(CC)n2CCOC)C(O)C1 C1(C2(NC(=O)C=Cc3ccco3)CC2)CCCCN1C(c1ncccc1F)=O N1(C(c2ccc(C)cc2)=O)CCC(NC(=O)CC2CCCN(C(C)C)C2)C1(C)C c1(NC(N(CCCSC)C)=O)ccc(-c2nnn(C(C)(C)C)n2)cc1 C1(NC(=O)OC(C)(C)C)CCN(C(=NCCc2ccccn2)NC2CC2)C1 N1(C(C(C)=C(CC)C)=O)CCC2CCN(C(=O)C(c3cccnc3)C)CC12 C=C(C)CCCC(=O)NCC1CCN(C(C2CC(N(C)C)C2)=O)C(C)C1 C1(C(=O)NCCCCC(C)NC(C2(N(C)C)CC2)=O)CCCCC(=O)N1 C12(NC3CCC(n4cccc4)CC3)CCC(C(=O)OCC3COCCO3)(CC1)C2 C1(c2nnnn2C2CCCC2)(OC)CC(C)N(CCc2noc3c2COC3)C1 c1(C(=O)NC2(CNC(Cc3cnc(C)[nH]3)=O)CCOC2)cncc(N)n1 CC1(C)CCCCC1CCCONC(=O)NCCCc1ccccc1 c1(C(N2CC(C)(C)C(NC(c3coc(C4CC4)n3)=O)C2)=O)ncc2[nH]ncc2n1 c1(CCC(=O)NCC2N(C(C3(C)N(C)CCC3)=O)C3C(C2)C3)cc(F)cc(F)c1 C1(CNC(CN(C)CC)=O)CC2CC2N1C(C1CN(C2CCOCC2)C1)=O C12(C(=O)NCC3(CNC(C4C(OC)C4)=O)CCOCC3)CCCN1CCC2 C(=O)(C1=C(Cl)CCC1)NC1CC(C(N2C(CC(C)(C)C)CC2)=O)C1(C)C N1(C(c2cnn(C)n2)=O)CCCC(C2CCN(C(c3cnn(CCO)c3)=O)C2)C1 c12cc(C)cc(c1F)C(=O)N2C1CC2CC1CN2.C1(C(=O)OC)CCC(N)C1 c1(C(=O)OC)cc(C(N2CCN(C(C3CCCSC3)=O)CC2)=O)ccc1Cl C1(C(=O)NCC(CNC(C2(Br)CC2)=O)CO)CCC2(CC2)C1 Cc1cccc(F)c1C(=O)NC1(C)CCCN(C(c2ccc(=O)n(O)c2)=O)C1 c1(C(=O)NC2C(NC(C(CC(C)C)OC)=O)CC2)ccc(N)c2ccncc12 N1(C(C2CC(C(C)C)OCC2)=O)CCN(C(C2CC(N=[N+]=[N-])C2)=O)CC1C C(CCCCOC(C)(C)C)(c1nnnn1C1COC1)NC(COCC)C C1(COC)CCN(C2CC2)CC1.c12ccoc1C(=O)NC1CC(C1)NC(=O)C2 N1(C(CC(C)C2CC2)=O)CC2(CC(NC(c3ccnc(F)c3Cl)=O)CO2)C1 C1(C(=O)NC(COC)(C)C)CCCC12CCN(C(C1CCC(O)CC1)=O)C2 N1(c2nc(OC)c(F)c(C)n2)CCC2C(CCN2C(C2C3COCC23)=O)C1 c1(C(=O)NC2CCN(C(c3c(C)onc3)=O)CC2F)ccc2nnc(C)n2c1 c1(CCC(=O)NC2(C(N(C(CCSCC)C)C)=O)CCC2)cn(C)cn1 c1(OCCCN(CCOC(CN2C(C)CCC2)=O)C)nccc2oncc12.C1CO1 Cc1cccc(Br)c1C(C(=O)NCC1CCCN1C)NC(C1CN(C2CCC2)C1)=O C1(CNC(c2n(CCC)ccc2)=O)CCN(C(C2CC(C)N(C)C2)=O)CC1O C(N=c1cc(F)nc[nH]1)C1(NC(c2ccc(Cl)s2)C)CCCCC1 C(=O)(CCCCC(F)(F)F)NCC(CNC(CCCCNC(=O)OCC=C)=O)F c1(CN(CC(N2CC(N(C(=O)CCOCC(F)(F)F)C)C2)=O)C)cnnn1C c1(NC(=O)CN2CCN(c3ccc(F)cc3)CC2)c[nH]c2ccc(Br)cc12 CC(C(=O)NCC1CC2CCC1N2C(C1CCCCC1)=O)C(C)(F)F c1(NC(c2c(C)nco2)=O)cccc(NC(=O)CN2CCCC2C)c1 C1(CC(=O)NCCCN(C(=O)CC2CC(=O)NC2=O)CC)(COC)CCOCC1 N1(C(Cc2c(C)noc2)=O)CCCC(C2CN(C(=O)CSCC(F)(F)F)C2)C1 C1(C(N2CC(NC(=O)COCCF)C(F)C2)=O)CC2CCC(C1)C2 c1(C(=O)NC(C2(O)CN(C(c3cnc(Cl)cn3)=O)C2)C)cc(F)c(Cl)cc1F C(=O)(C1=CCCC1C)N1CC(F)(CNC(CC(C)c2ccco2)=O)C1 c1(C(=O)NC(C)(C)CCNC(=O)CSc2ccc(Cl)cc2)ccn2c1CCCC2 c1(N(CC=CCN(C(C2C(C(C)C)(CC)C2)=O)C)C(=O)C2CC2)nnn(C)n1 N1(C(Cc2ccc(CC)cc2)=O)CCCC12CCN(C(=O)CC1(O)CCC1)C2 N1(C(c2c(C)cc(CC)o2)=O)CC(NC(=O)C(C)(C)CN(C)C)CC1(C)COC CCC(C)(CNC(=O)COCCCF)C(=O)N(C1CC1)Cc1n[nH]c(C)n1 S(=O)(=O)(c1ccc(Cl)s1)N(CCOCC)CC1(O)CC(C(=O)O)C1 C1(C(=O)NC2CC(NC(=O)CCc3ccon3)CC2O)CCN2CCCC2C1 C1(O)(CNC(=O)NC(c2c(C3OCCO3)nccc2)C2CCOC2)CCCCC1 C1(C(=O)NCC(C(=O)NC(CC)C(=O)OC)N(C)C)CC2(CCO1)CC2 C(=O)(C1=CCCCC1)NCC1(NS(CCCC)(=O)=O)CCOC1.C1(C)C(=O)N1 c1(N2CCCC(COC)(CO)C2)nc(=NCCC(C)SC)[nH]c2ccsc12 c1(C(=O)NC2C(NC(C(CC)SC)=O)CCOC2)ncc(Cl)cc1O c1(C(N2CCCC(C)(NC(c3ccc(C)cn3)=O)C2)=O)cc(Cl)cc(Cl)c1N C1(N(C2COC(C=Cc3ccccc3)=[SH]2)C)CS(=O)(=O)C1(C)C C(C(O)CC(=O)NCCC1CCN(C(C2CC(OC(C)(C)C)C2)=O)C1)C1C(C)C1 C(=O)(CC(O)CCCC)NC(C1CC(NC(c2ccc(C=C)cc2)=O)C1)C C(=O)(CC(C)CC(C)(C)C)NC(C1CN(C(c2cnc(Cl)cc2F)=O)CCO1)C C1(CC=C)(NC(=O)Cc2cncnc2)CCCN(C(=O)COC)C1 c1(OC)ccc(-n2nnnc2C2CC2)c2ccccc12.c12cc(nn1C)NC2=O c1(CCCC)cn(CCN(C(=O)CCSCC)CC)nn1.C(C)C Cc1ccc(N)cc1C(N1CCC(C)C(NC(C2CC(S(C)(=O)=O)C2)=O)C1)=O N1(C(c2cc(C)c(C)[nH]2)=O)CC2(COC(CNC(=O)C(F)C(F)(F)F)C2)C1 Cc1ncn(C)c(=O)c1C(=O)N(C)CC1(O)CN(C(C2OCC2(C)C)=O)C1 c1(C(=O)NCC2CN(C(C3C(C=C)C3)=O)CC2O)ccc(S(N)(=O)=O)cc1 C1(NC(=O)CCCCN2CCCC2)C2CC(O)C1N(C(c1cn[nH]c1)=O)C2 N1(C(C(CN(C)C)NC(C(C)=C2CCCC2)=O)=O)CCC(O)CC1C1CC1 c1(C(=O)NCC(CNC(C(C)S(N)(=O)=O)=O)F)cc(F)cc(N)c1F c1(C(C)NC(C(=O)NC(C)C)=O)ccc(CNC(C2CC3(C2)CC3F)=O)cc1 C(C(C)(CC(C)C)NC(=O)CCn1ccnc1)NC(c1nc(C)sc1)=O CCCC(C)CCCC(=O)N(C1CN(C(=O)Cc2ccc(SC3CC3)cc2)C1)C CC(Cc1ccccc1)CC(=O)NCCC(C)NC(=O)C(Cl)=CCl C1(C(=O)NC(C)CCC2CC2)CN(C(=O)Cc2ccn(C(F)F)n2)CC12CCC2 C1(C(=O)NC(C)C(=O)NC(C)(C)C)CC2(CC(NC(C3(C)CCOCC3)=O)C2)C1 C(=O)(C(C)S(=O)(=O)C(C)C)N1CC(C2CN(C(Cc3ccc(OC)nc3)=O)C2)C1 c1(OC)cnc(Cl)cc1C(=O)NC(C)CNC(c1cnnc(C)c1)=O C1(NC(CN(CCCCCC)C)=O)CCN(C(=O)C(OC)OC)C(C)C1 C(CC(C)C)(C(=O)NCCOC(C)(C)CNC1CC(C)(C)CO1)NC(=O)OC C12CC3(CC(C3)NC1=O)C2.C1(C(=O)NC(CC)C)CC1(C)C CCCCC(O)C(=O)N1CCCCC1C1CCN(C(c2cncc(C)n2)=O)C1 C1(C(C)NCC2CCc3nccn32)CCC2(CC1)CC(C)(C)C2 Cc1nn(C)c(C)c1C(C)C(=O)N(C(C)CCNC(C1=NNC=CC=C1)=O)C C1(C(N2CCC(NC(C3(OCC)CCCC3)=O)CC2)=O)CCCS(=O)(=O)N1 C(=O)(C1CCSc2ccccc21)N1C(CCNC(COCC)=O)CCC1 c1(OC)ncnc(C(=O)NC2CC(NC(C3CC(=O)N(C4CC4)C3)=O)C2)c1F Cn1ccc(CCOC(C2CCN2C2CCCCC2)=O)n1 C1(CC(C)C)CCN(C(c2cc(CNC(c3coc(CO)c3)=O)[nH]n2)=O)C1 S(=O)(=O)(c1ccc(NC(=O)NC2CCOCC2N)cc1)N(CC=C)C CCCCC(C)(F)C(=O)NCCC1CC(NC(=O)Cc2cnc(C3CC3)[nH]2)C1 C1(NS(=O)(=O)CC)CC2CCC(C1)C2.N1(C)CCN1CCN(C)C.CC C(=O)(C(CC=C)CC(F)F)NC(C(C)(C)NC(C(CC#C)CC#C)=O)C c1(C(=O)NC2CCN(C(C3=C(C)OCC3)=O)CC2)ccn2ncnc2c1 N1(C)CC(C)C(F)(F)C1.c1(C(CC)N)ccc(OCC(F)(F)F)cc1 C1(C)(C(=O)NC(CNC(CCOC)=O)C(C)C(C)C)CCC(F)(F)CC1 C1(CNC(C(CC)CC)=O)CCC2CN(C(c3ccnn3C(C)(C)C)=O)CC12 c1(C(N2CCCC(C(=O)NCCSCc3n(C)ccn3)C2)=O)coc2c1CSC2 c1(C(=O)NCC(CC(C)C)NC(CC=C(C)C)=O)cnc2c(c1)NC(=O)CO2 c1(C(=O)NCC(C)CNC(C2CCCCS2(=O)=O)=O)cc2ccsc2s1 C(N=C(NCC1(F)CCOCC1)N1CCc2ccccc21)C1C(C)CCCC1 C(CC(N=c1cc(C)nc(N(C)CCc2cnc[nH]2)[nH]1)c1cccnc1)OC N=c1[nH]c2c(C(=O)NC3CC(NC(C4(F)CCCCC4)=O)C3)cccc2o1 C1(C(=O)NC2CN(C(c3ncc(NC)nc3)=O)CC23CC3)CC(C)(C)OC1(C)C C(=O)(C(O)C(C)(C)C)NCC(C)(C)CCNC(=O)C(F)CC1CCCCC1 C(=O)(C(C)(CO)NC(=O)NC(C)C(C)(C)Nc1ccccc1)OC C(C(CNC(C1CCC=CCCC1)=O)C(F)(F)F)NC(c1cnc(C#N)s1)=O CCCCC(O)C(C)C(=O)NCc1n[nH]cc1C(N1CCN(C2(C)CC2)CC1)=O Cc1c(C(N2CCC(F)(CNC(c3cccnn3)=O)C2)=O)cc(C2CC2)n1C C(N=C(NC1CCOC1)NC1CCS(=O)(=O)C1)c1n(C)ncc1.C1(C)OCCO1 N1(C(C2(NC(=O)OC)CCCC2)=O)CCC2CCN(C(c3n[nH]cc3C)=O)CC12 Cc1cc(C(C)(C)C(=O)N2CC(CNC(c3cncc(O)c3Cl)=O)C2)ccc1F C(N=c1nc(N2CCN(C=O)CC2)c2c([nH]1)CCCCC2)C1(CF)CC1 N1(C(Cc2ccn(CC)n2)=O)CC=CC1(C(N1CCCCC1)=O)COC C1(COC)(NC(C2CCCN2C(c2cnccc2N(C)C)=O)=O)CCOCC1 c1(CC)c(C(N2CCCC(CNC(C3CC(C)(O)C3)=O)CC2)=O)cccc1F CC1(C(=O)NCC(CC2CC2)C(=O)NCC(F)(F)C(N)=O)CC2CCC1O2 c12nonc1C(=O)N1CC(c3cn(nn3)CC2OC)C1.C1(CC)COC(=O)C1 c1(C(N2CCC3(CN(C(C4C(CC)C4)=O)C3)CC2)=O)cccc(S(N)(=O)=O)c1C c1(CCC(=O)NCCCN(C(c2cnn(C)c2F)=O)CC)cccc(C#N)c1 N1(C(=O)C=CC2CCCC2)CCC(C2OCCC2NC(=O)C(F)(F)CC2CC2)CC1 N1CCCC(C)(N(C(=O)CC=CC(C)(C)C)Cc2ccccc2)C1.Cc1cccnn1 C1(CNC(CC)=O)CC(C)CCN(C(c2cc(C(F)(F)F)cc(N)c2)=O)C1 CC(F)(F)C(F)C(=O)NCCCC(=O)NC1CC(C)(C(N)=O)C1 N1(C(c2c(C)nc(CC)s2)=O)CCC(C2CC2)(NC(=O)CC2COCCO2)C1 C(=O)(C(C)(O)CCN(C)C)NC(C1OCCN(C(C(F)=CC)=O)C1)C N1(C(C2OCCN(c3c(OC)c[nH]n3)C2)=O)CCC(C)C(N(C(C)=O)C2CC2)C1 C1(C(=O)NCc2ccc(C)s2)CCN(C(=O)CCCSC2CC2)CC1 CC1CCC=C1C(=O)NCc1cn(C2CN(C(=O)CC3CCCOCC3)C2)nn1 c1(OC)c(Br)ccc(C(N2CCCCC2C(=O)NCC2(F)CCC2)=O)c1F N1(C(Cc2c(C)n[nH]c2)=O)CC2CC2(C(N2CCC(C(C)C)C2)=O)C1 C1(C(=O)NC(c2cccnc2)CC)CN(C(=O)C(C)(C)CCF)CC1C1CC1 C1(C(N2CCN(C(C3CC(CC)OCC3)=O)C(CC)C2)=O)CN2CCN1CC2C c1(CNC(C2C(NC(=O)CC3(O)CCOC3)CCC2)=O)ncc(Br)cn1 Cc1cccc2ncc(C(N3CC(CNC(C4CC45CCC5)=O)CC3C)=O)n12 O=C(N=c1[nH][nH]c2ccc(C(F)(F)F)cc12)NC1C=CCCC1.C1COC1=O CCC(CCOC)C(=O)NCC12CC1CN(C(C1SCC=C1C)=O)C2 c1(OC)ccc(C(N2CCC(O)(CNC(C34CCC(CO3)C4)=O)C2)=O)cc1Cl C(=O)(C1CC=Cc2ccccc21)NCCCN(C(CCC(C)(C)OC)=O)C(C)C CN(C)NC(=O)CCC(=O)NCC(CNC(C12C=CC(CC1)C2)=O)CO C1(C(=O)NC(CC=C)CNC(c2c[nH]nc2C)=O)COc2c(Br)cccc2C1 CC(CC#N)C(=O)NCc1n[nH]cc1C(=O)NC1CN(C2CCC2)C1 CC1(F)CCN(C(C2CC2c2ccc(C#N)cc2)=O)CC1 c1(C(=O)NC2C(CNC(C=CC=CC)=O)C2)cccc(O)c1NC(C)=O Cc1c(Cl)ccnc1C(=O)N(CCC(C)(C)NC(=O)CCC(C)N(C)C)C CN1CCC(NC(C2(O)CCSC2)=O)C12CCCN(C(=O)CC1CCC(O)C1)C2 Cn1nnc2ccc(CN3CCN(C(CCNCCC(F)(F)F)=O)CC3)cc12 Cn1cnc2cc(C(N3CCC(NC(=O)CCc4ccon4)C(O)C3)=O)ccc12 C1(C(N(CCOCCN(C)Cc2c(C)noc2C)C)=O)CCc2nc[nH]c2C1 C(CCC(N)=O)(C(=O)N1CC(NC(=O)C(c2ccccc2F)O)C(C)C1)N(C)C C1(SCC)CCC(=O)CC1.Cn1cc(CN(CCO)CC2COCC2c2ccccc2)cn1 N1(C(CCCCC#C)=O)CCOC2(CCCN(C(=O)C(F)(F)C(C)OC)C2)C1 C(=O)(CCC1=NNC(=O)CC1)NC1C(NC(c2c(OC)n[nH]c2)=O)CS(=O)(=O)C1 c1(C(=O)NC(C)(C)CCCNC(c2ccc(F)cc2O)=O)ccc2c(c1)COC2 C1(CCC(=O)NCCCC(C)NC(c2cc[nH]c(=N)c2)=O)CC(C)(C)CO1 C1(CNC(c2c(CC)csc2)=O)CN(C(C2SCCCS2)=O)CC1(F)F C1(CNC(C2CC(O)(CC#C)C2)=O)CC(C)(C)CCC1NC(=O)C(F)F C=CCCCC(=O)NC(C)(COCC)CNC(=O)C(C)Cc1ccccn1 C(=O)(C#CC1(C)CC1)NC1CC(NC(c2c(CC)occ2)=O)C1 c1(C(N(C(C)CNC(=O)CN2CCC2)C)=O)ccccc1-n1ccnn1 N1(C(C2CC(SC)C2)=O)CC2CCC2(CNC(=O)CCCNC(C)=O)C1 Cc1cc(=NC(=O)C(=O)N2CC(CNC(c3sc4ncccc4c3Cl)=O)C2)[nH]o1 C1(CNC(C(CC=C)(F)F)=O)CC2(CO1)CN(C(c1ccc(Cl)cc1N)=O)C2 c1(C(=O)OC)ccc2cc(C)nc(N(CC(=O)OC)C3CC3)c2c1 C1(CC(=O)NCC2(OCC)CN(C(C3CCO3)=O)C2)CCC(=O)NC1 C1(C2CCN(C(C3CC34CCCC4)=O)C2)(NC(c2cnc3c[nH]nc3c2)=O)CC1 N1(C(c2c(CC)c[nH]c2)=O)CCC2CCCC12C(N1CCC(F)(F)C(O)C1)=O C1(C(=O)NC2CC(CCNC(c3c(CC)csc3)=O)C2)CC(=O)NC1(C)C C1(COC)(NC(C2CCC(C)=C(C)C2)=O)CCN(C(=O)C(C)(C)F)CC1 C1(NC(c2n(CC)nnc2C)=O)CC12CCN(C(c1cnoc1C(C)C)=O)CC2 C1(C(C)C)CCC(N=c2[nH]c(N3CCC(c4ccccc4F)C3)nc(=N)[nH]2)CC1 CCCCC(C(=O)N1CCC(CCOC)(NC(C2(C)CC3(CC3)C2)=O)C1)N(C)C Cc1cc(C=CC(=O)NC(C)CC(C)NC(c2ccc(=O)n(C)c2)=O)ccc1F c1(NC(C2CCN(C(C(CCC)OC)=O)C2C)=O)cnc(O)cc1C C1(NC(C(C=CC)O)=O)CN(C(c2cccc(C(=O)OC)c2)=O)CC1O O(NC(=O)C1=CCN(C(=O)C(n2cc(C)cn2)C)C1)CC(=O)NCC c1(C(=O)OC2CCN(Cc3nnnn3CCCF)C2)nc(Br)c2n1CCCC2 N1(C(C(c2c(C)nn(C)c2)O)=O)C2CCCC1CC(NC(=O)C=CCN(C)C)C2 C(=O)(CC(C)C(C)(C)C)NCCC(=C)CNC(c1ccnc(CO)c1)=O Cc1c(C(=O)NCC2CC(NC(=O)C(C)(C)CC3CC3)C2)cnn1C1CCCC1 c1(NC(=O)NC23CC(NC(C(C(C)(C)C)O)=O)(C2)C3)ccc(F)c2ccccc12 C1(C)(C(=O)NC(C(C)O)C(=O)NCc2n[nH]cc2C2CC2)CC2(CCC2)C1 c1(CC(=O)NC2(COC)CN(C(C3CN(C)C(=O)N3)=O)C2)ccc(O)cc1 C1(=O)CC(COC)COC2(C)CN1C2.C(CCNC(=O)CSCC)OC CCCN(OC)C(=O)C(CNC(C1CC=CCO1)=O)(CC)CC N1(C(C(CC(=C)C)C)=O)CCc2nc(CNC(C3C=CC=CC=C3)=O)sc2C1 c1(C(N2CCC(C(C)NC(c3ccco3)=O)C2)=O)cc2nnn(C)c2s1 N(C(=NCCCC(=O)N(C)C)NCC1CNC(=O)C1)C1CCCN(CC)C1 CCCC(F)C(=O)NCC(O)CN(C(=O)Cc1ncc(C)o1)C C1(CN(C(CC(=O)OC)=O)C)CCCC(NC(c2ccc(NC(N)=O)cc2)=O)C1 C1(C(=O)NCCCO)CCC2(CCN(Cc3c(I)ccnc3Cl)CC2)C1 C=CC(CCC)CC(=O)N1CC2=C(C1)CN(C(C1CC3CCC1CC3)=O)C2 c1(CNC(C(OC)OC)=O)nnn(C)c1C(=O)N(C)CC1CCOC1C c1(CCC)ncoc1C(=O)NC1CC(CNC(=O)C(C)OCC(C)C)C1 CCC(C)CC(=O)C(=O)N1CC(C(O)CNC(c2ccoc2C2CC2)=O)C1 N1(C(CNS(CCCC)(=O)=O)=O)CC(C)CN(C(C2CSCCS2)=O)CC1C C1(C(C(=O)NCCC23CCCC2C3)F)CCN(C(=O)Cn2cc(CO)nn2)C1 C=CCC(F)(F)C(=O)NCC(CO)NC(c1ccn(C2CC2)c1C)=O C1(NC(C(CCCC)O)=O)COCCN(C(c2cc(Br)cn(O)c2=O)=O)C1 c1(C(=O)NC(C(C(C)C)NC(c2n(CC)nnc2)=O)C)cc(C)c(C)c(C)c1 C(=O)(CS(=O)(=O)CC(F)(F)F)N1C2CC(NC(CCNC(=O)CO)=O)C1CC2 n1(CC(N2CC(C)C(NC(c3ccc[n+]([O-])c3)=O)C2)=O)cccc(N)c1=O Cc1cnc(C(=O)NC2CCC2NC(C2(C)CC=CCC2)=O)cn1 C1(NC(C2(C)CCN(C)CC2)=O)CN(C(=O)Cn2ccnn2)C2(CCOCC2)C1 C=CC1(CC(=O)NC(C)CCCCO)CN(C(C2CCCCC2C)=O)C1 C1(NC(=O)CC2CC2)CCC2(CC1)CC(NC(C1CCn3nccc3C1)=O)C2 C1(C(=O)NCC(c2ccccc2)CNC(=O)CC2CCSC2)CC2C=CC1O2 C(=O)(CC(C)COC)N1C(CNC(C=CC=CCC)=O)C=CC1 c1(NC(C2C(C)(C)CCN(C(=O)C3=COCC3)C2)=O)cnc2ccc(F)cc2c1 N1(C(c2nc(C(=O)OC)oc2)=O)CCCN(C(=O)C(C)(C)C(C)C)CC1C c1(-c2c(C(=O)NCC(CC)(C)NC(=O)CNS(N)(=O)=O)c[nH]n2)ccccc1Cl O=C(N=c1[nH]oc2nccnc12)C1CC1C(=O)NC1COCC1O C(=O)(C1=NN(CC)C2(CCOC2)C1)N(C)CC1OCCN(C(C(CC)=CC)=O)C1 Cn1ccc2c(-c3cncc(C(=O)Nc4cc(Cl)c(Cl)c(Cl)c4)n3)cccc12 c1(C(=O)OC2CCN(c3ccn(C)n3)C2=O)cccn2nccc12 C1(CCNC(CCCN(C)C(c2ccc(O)nc2)=O)=O)CCCCC1O CCCCC(=O)C(=O)N1CC2CC1C2NC(=O)CCc1cnc(O)[nH]1 C(=O)(CC1OCc2ncccc21)N1CC2C(NC(C3CCC(C)O3)=O)C(C2)C1 c1(OCC(=O)N(CC(CC)NC(C2(COC)CCNC2=O)=O)C)ccc(Cl)cc1 N1(C(CCC(C)SC)=O)CC2CC(NC(=O)CCn3cccc3)C(C2)C1 C1(O)(CNC(C2(OC)CC2)=O)CCCN(C(C2CCC(F)(F)C2)=O)C1 c1(C(N2CCC(N(C(c3cnccc3OC)=O)CC)C2)=O)cncc2nc[nH]c12 N1(C(c2cn(C(C)C)c(=O)cc2)=O)CCN(C(=O)C(=O)NCC(F)F)C(C)C1C c1(C(CNC(C2CC2OC(F)F)=O)NC(C2C(C)C2)=O)ccccc1 Cc1[nH]cc(C(=O)NC2CC3CCC2N3C(c2ccccc2Br)=O)c(=O)c1Cl C1(CNC(C(CCC)O)=O)CN(C(c2c(C)cccc2Cl)=O)C2(CCC2)C1 c1(CNC(c2occc2C(=O)Nc2ccccc2)=O)ccc(O)c(F)c1 C(=O)(CCCCC(C)(C)C)N(CC(=O)NCc1cccc(F)c1O)CC#C c1(SC)ccc(C(N2CCCN(C(=O)CC(C)n3cccc3)CC2)=O)c(Cl)c1 Cc1cccc(C)c1CNC(C1CCN1C(C1CC2CC1CC2=O)=O)=O C(=O)(C(C)(C)C(CC)CC)N1CC(CC(N(CC=C)OC)=O)C(C)CC1 Cc1cc(OCC(=O)NC2CCC(NC(=O)C(O)(C3CC3)C3CC3)C2)cc(C)c1 c1(C(N(CC(C)(C)NC(C(c2c(OC)cccc2)C)=O)C)=O)c[nH]cc(C)c1=O n1(C(c2nc(C(C)OCCO)on2)(C)C)cc(O)ccc1=O CCCCCC(=O)N1CCC(Cc2nc(C)cs2)C1.C1(=O)C(CC)N1C1CC1 C(=O)(C1=CCc2ccccc21)N1CCC(NC(c2c(C(C)C)c[nH]n2)=O)C(O)C1 C(=O)(C1=NN2CC(C)CN=C2N1)N1CCCC(NC(CCCCOCC)=O)C1 CCC(C)CCC(=O)NCC1CCN1C(=O)Cn1cc(-c2ccccc2)cn1 N1(C(CCc2ccc(C)cc2)=O)CC(NC(=O)CC2CCCOC2)C2CCCC12 c1(C(=O)NCC(C)N(C(CCCNC(=O)OCC)=O)C)cnc2[nH]cncc1-2 CN1CC(C(=O)N(C)Cc2cccc(CNC(c3csc(Cl)n3)=O)c2)NC1=O N1(C(C2CN(C(CCN(CCC)C)=O)CC(C)O2)=O)CCn2c(C)cnc2C1 C1(N(C(c2snnc2C)C(=O)NCC2CCOC2)C)(COC)CCN(C)CC1 N1(C(CC2=NNC(=O)C2)=O)CC2(C1)CN(C(C1NC(=O)C3CCC13)=O)CCO2 N1(C(c2c(CC)nn[nH]2)=O)CCC(C)C(NC(c2cc(C(F)(F)F)ns2)=O)C1 c1(CNC2CCC(CNC(c3ccc(F)cc3)=O)CC2)ncc(Cl)cc1Cl C1(C(N2CCC(CO)C2)C(=O)N(C2(C)CC2)CC2CCCOC2)C2CC=CCC12 CC1(C)CC(CC(N2CCC(OCC(N)=O)C2)=O)CN1C(C1CCC(=O)CC1)=O C(CC1CC1)(C(=O)NCCCC(N)=O)NC(C1C(=C)C1)=O C1(N(C(CC(=O)NCC)=O)C)CN(C(=O)CCc2ccccc2)CCC1C c1(C(N2CC(O)(CN(C(C3C(C)C3)=O)C3CC3)C2)=O)cccc2nccn12 CS(C)(=O)=Nc1ccc(C(N2CC(NC(=O)Cc3ccco3)CC(O)C2)=O)cc1 c1(C(=O)NCC2CC(CNC(CCCCN(C)C)=O)OC2)cnc2scnc2c1 N1(C(c2cnc(OC)s2)=O)CCC(NC(c2ccc(C(C)C)nc2C)=O)C(O)C1 c1(C(=O)NC2CN(C(CC3(N(C)C)COC3)=O)CC(O)C2)ccn2cncc2c1 N1(CC)CC(C(N2CC(CNC(=O)C(c3ccccc3F)O)(OC)C2)=O)CC1=O c1(CC)c(C(=O)NC(C)CNC(C2CCCC23CC3)=O)cnn1CC N1(C(=O)C(F)=C2CCC2)CCN(C(C2CC3C=CC2O3)=O)CC2(CC2)C1 C(=O)(CCS(=O)(=O)C(F)(F)F)N1C2C(CNC(CCCC#C)=O)(CCCC2)CC1 C1(NC(CCC(CC)CC)=O)CN(C(=O)CS(=O)(=O)NC)CC12CCCC2 C1(NC(CN(C(c2c(CC)c[nH]c2)=O)CCO)=O)(CSC)CCC(C)(C)C1 CCC(CC)(CO)C(=O)NC1CC2CC(NC(c3ncccc3SC)=O)C2C1 c1(C(=O)NC2C(NC(C3C(C(=O)OC)CCC3)=O)C2)ccc(C)cc1Br c1(NC(C(=O)NC(CNC(=O)OCC)C)=O)ccn(CC#N)n1 Cc1ncc(CCC(=O)NCC2CCN(C(c3nnn(CO)c3C)=O)C2)c(O)n1 N1(C(C2C(CC)OCC2)=O)CCOCC1C(=O)Nc1cccc(C)c1 N1(C(CCN(CCC)C)=O)CCC(F)(C(=O)N(C)CCOC(F)F)C1 N1(C(C2C(C(=O)OC)C2)=O)CCC(NC(=O)C(F)Cc2ccccc2)C1C C1(C(=O)NC(C(C)NC(c2ccc(SC)cc2)=O)(C)C)CCN(C)C(=O)C1 C=C(C)CC1C(=O)N1.c1(SCO)n[nH]cc1C(N1CC(OC(C)=O)C1)=O.C(C)(C)O N1(C(CSc2c(C)cccc2)=O)CCC2CCN(C(=O)C(C)CF)CC12 N1(C(c2ccc(C)s2)=O)CCCC2CN(C(=O)CCC3(C)CCC(=O)N3)CCC12 c12nc3ccccc3nc1NC1C(CS(=O)(=O)C1)N2.C1(C(N)=O)CCCCC1 C1(C#N)(NC(C2CCN(C)CC2)=O)CCN(C(c2ccc(O)cc2Cl)=O)C1 C1(C2(O)CCC2)(C(=O)NCC2(NC(c3c[nH]nc3C3CC3)=O)CC2)CC1 C(C(N)=O)(C(N)=O)NC(CNC(c1cnc(CC)s1)=O)=O CC(CC(N)=O)C(=O)NCC1(C)CC(NC(=O)COC2CCOCC2)C1 C(CN=c1[nH]c(N2CCC(c3nc[nH]n3)C2)nc(=N)[nH]1)c1c(C)cncc1 Cc1cc(C(=O)NCC2(CNC(C3CCOC3=O)=O)CC2)c(F)cc1F c1(C(CO)N(C(C2CCC2CCC(=O)Nc2nnsc2C)=O)CC)ccccc1 C(N=c1[nH]cncc1OC)C1(CNC(Cc2cccc(OC)n2)=O)CCCC1 Cc1ccc(C(=O)NC2CN(C(=O)C(F)C3CC3)CC2C(F)F)cn1 S(=O)(=O)(c1cccc(COCP(C)(C)=O)c1C)NCc1cn(CC(CC)O)nn1 c1(CN(CCOC)C(=O)NC(C)CC)cc(Cl)c(F)cc1Cl N1(C(C2(C(C)C)CCN(C(CCCCOCC)=O)C2)=O)CCC(F)C(O)C1 N1(C(C(C(C)C)C)=O)CC23CCCC2(C1)CN(C(=O)C(c1ccccc1)C)C3 N1(C(CC(C)CF)=O)CCN(C(=O)CC2CC=CC2)CC1CS(C)(=O)=O N1(C(CC(C(=O)OC)C)=O)CCCC(O)(CNC(c2c(C)nsc2C)=O)CC1 c1(C(N2C(CC(=O)Nc3ncc(Br)nc3Cl)CC2)=O)ncc(F)cc1F Cc1nn(C2CCC2)cc1C(=O)NCC1CN(C(=O)COCC(C)C)CCO1 C1(CN(CC(=O)NCC=C)C)CCCCN1C(c1nc(C)cn1C)=O C(=O)(C(CCF)NC(=O)OC(C)(C)C)OC.c1(NC=O)cccnc1C(F)(F)F c1(OCC)cc(N2CCC(CCNC(=O)C=Cc3ccccc3)CC2)nc(C)n1 c1(CCN(C(=O)C(C2CCC2)NC(=O)CN(C2CCCC2)C)C)cc[nH]n1 c1(OC)n[nH]c(C(=O)NCc2ccc(-c3cccc(I)c3)o2)c1C#N CCC(F)C(=O)NCC1CCC1NC(c1ncoc1-c1cnn(C)c1)=O C(C(C(=O)NC(c1ncc[nH]1)(C)C)NC(=O)C(C)OC)ONC(=O)OCC.C1(S)CC1 N1(C(C2NC(=O)OC2)=O)CCN(C(=O)Cn2nccn2)C(c2ccncc2)C1 CC1=C(C)CC(C)(C(N2C3CCC2CC(N(C)C(C2(F)CC=CC2)=O)C3)=O)CC1 O=C1CC2(CCC2)C(C(N2CCCN(C(C34CC(CO3)C4)=O)CC2)=O)CN1 c1(SC)cc(F)ccc1C(=O)NC(C(C)NC(=O)COC1CCOCC1)C(C)C c1(C(=O)NC2(C)CC(NC(c3n(CC)nnc3)=O)C2)cc2cnccc2cc1F c1(C(N2C(CNC(c3c(C)c(=O)cc[nH]3)=O)C(O)C(O)C2)=O)nnn2c1COCC2 c1(C(N2CC3(C(NC(CCSC)=O)CCS3)C2)=O)cn2c(n1)C(C)CCC2 c12ccc(cc1)S(=O)(=O)CC(=O)OC(=O)C2(C)C.C(C(O)CC)N(C(C=C)=O)C N1(CCC)CC(C(=O)NC(CNC(C2(CC3CC3)CC2)=O)C(C)C)CC1=O Cc1csc(C(=O)NCC(C)(CO)NC(=O)COC2CC=CC2)c1Br Cc1cnn(CC2CCN2C(c2sccc2C)=O)c1.c12cn(nn1)CCC21CC1 C1(C(=O)NCC(CNC(c2cc(C(CC)CC)no2)=O)OC)CCC(C)=C(C)C1 N1(CC)CCC(NC(=O)C(C)(C)CN(C)C(C2CCN2C(C)(C)C)=O)C(C)C1 C1(C(=O)NC2CC=C(C(=O)N3CC[Si](C)(C)C3)C2)Cc2ccccc2C1 C(N=c1[nH]c(=N)[nH]c(=NCc2cc3c(s2)CCCC3)[nH]1)C1CCCC(CC)C1 C(c1cn[nH]c1)=CC(=O)NCCN(C(=O)C(C)CSC(F)(F)F)CCC CCCC(C(=O)NCC1CC(C(=O)NC2CCC(CO)C2)C1)OC c1(C(=O)NC2(CC=C)CCN(C(=O)C(C3CC3)C3CC3)C2)cc2cnn(C)c2s1 C1(CNC(C(c2cccc(C)c2)=O)=O)CN(C(=O)CCCCCF)CCOC1 N1(C(Cc2cc(OC)c(C)cc2)=O)CCC(C2CCN(C(=O)C(C)(C)C)C2)C1 c1(NC(c2cc(-c3ccc(-c4ccc(F)cc4)cc3)n[nH]2)=O)cccc(O)c1Cl C(CCOCCO)(C(=O)NC1CCCC1(C)C)NC(CCC=C)=O Cc1cc(Br)cc(C(N2CCOCC(C(C)(C)C(=O)N(C)C)C2)=O)c1N Cn1nccc(C(N2CCCC(CNC(C3(C4(C)CC4)CC3)=O)C2)=O)c1=O Cc1cc(Br)c(NC(C23CC(C(=O)Nc4c(O)ccc(F)c4Br)(C2)C3)=O)cc1F C(=O)(C(F)(F)C(F)(F)C(F)F)N1CCC(NC(c2[nH]nc(S(N)(=O)=O)n2)=O)C1 N1(C(c2nc(CC)sc2)=O)C2CCC1CC(NC(=O)CC1CCCCC(=O)N1)C2 c1(N(CC(=O)NCC)C)nc(=NCC(C)(C)CSC)[nH]c2cccc(F)c12 C(=O)(CC(C)(C)C(F)F)NCC12N(C(C3N(C)CCCC3)=O)CC(C)(C1)C2 c1(CNC(CNC=O)=O)ccc(CNC(C2C3(CC3)C23CC3)=O)c(F)c1 N1(C(C2(CC#C)CCCCO2)=O)CCN(C(=O)Cc2csnn2)CC(CO)C1 Cc1cc(C(N2CC(NCc3cnccn3)C3(CC3)C2)=O)c(F)cc1F c1(CC(=O)NC(C2(O)CN(C(CC3CC(SC)C3)=O)C2)C)c(C)noc1Cl N1(CC(=O)NC2CC(CC(=O)NC(c3cn(C)nn3)C)C2)CC2CC2C1 CC(C)(C)C(C)(O)CNC(C1CC12CC(NC(c1cnccn1)=O)C2)=O C1(NC(C(C)=CC)=O)C2CN(C(c3cccc(Cl)c3)=O)CC12 N1(C(=O)C2CC2)CCN(C)C2(CC2)C1.C12(CCOCC1)C(=O)NOC(C)C(=O)N2 N1(C(C(CCC)O)=O)CCC(C(=O)N(CC(O)CO)CC)C1(C)C N1(Cc2c([N+](=O)[O-])cn(C)n2)CCn2c(nn(CC(=O)OC(C)(C)C)c2=O)C1 CN1CC2(CCN2Cc2cn(Cc3occc3C(=O)C(N)=O)nn2)C1 CON(C)C1CCN(C(=O)CCC2CCC(NC(=O)CCN3CCCC3)C2)C1 C(=O)(C(CCSC)NC(C1(F)CC1)=O)NC1CCN(CCC)C1 C1(CNC(C2(C)N(C)CCC2)=O)CC2(CC(NC(c3cnc4n3CCC4)=O)C2)C1 C(=O)(C(O)C1=CCCCC1)N1C(C(=O)NCC(C)(C)C(C)C)CC(OC)C1 C1(CNC(C2N(C)C(=O)NC2)=O)CN(C(c2cccc(=S)n2O)=O)C(C)(C)C1 N1(C(=O)C)CC2(CCC2)CC1CO.C#CC1CCCC(NC(=O)C(F)(F)F)C1 CCCC(C)C(=O)NC(C)CC1CCN(C(c2c(C)nsc2NC)=O)CC1 C(=O)(CS(=O)(=O)C1CCCC1)NC1C2(CN(C(C(CC)SC)=O)C2)CC1 C1(CC)CCCCC1C(=O)NCCNC(=O)Cc1ccc(NC(C)=O)cc1 C12(CNC(CSC(C)C)=O)CC1CN(C(=O)CC(Cl)Cl)C2 N1(C(COC(C)=O)=O)CCCC1(C)CNC(C1CCOC1c1ccc(Cl)cc1)=O Cc1nc2ccc(C(=O)NC3CN(C(c4csc(C)c4)=O)CC3C3CC3)cn2n1 N1(C(CSCC)=O)CSCC1C(=O)NC1CC(O)C1CC(C)C CC(CC(=O)N1CCN(C(=O)C(C)Oc2ccc(F)c(F)c2)CC1C)C(F)F N1(C(c2n(C)nnc2)=O)CCOC(C(=O)N(C2CC2C(C)(F)F)CC2CC2)C1 c1(-c2ccccc2)nnc(CCCCCSCCC2CCCO2)n1C1CC1 C(=O)(CC(C)(C)CCC)NC(CC(=C)C)C(=O)NCCc1nc(C)no1 c1(N(C2CC3CC4C(C3)C24)NC(c2c(C3(C)CC3)ocn2)=O)cc(=O)n(C)c(O)n1 C12(C(=O)NCc3c(C)cccn3)CCN(C(=O)Nc3ccc(F)c(F)c3)CC1C2 N1(C(c2c(C)nc(C)s2)C(=O)Nc2ccccc2Cl)CCC12CCSCC2 c1(C(=O)NC(CNC(C2CCCOC2)=O)CC(F)(F)F)nnn2ccccc12 C(=O)(N=c1cc(C#N)cn[nH]1)NCC1(C)CSCCO1 c1(C(N(C2CCCN(C(c3occc3Cl)=O)C2)C)=O)cnc2c(c1)ncn2C N1(C(C2CCC(=C)CC2)=O)CCC(NC(=O)CC(C)SC)C(F)C1 C1(CCC)(C(=O)N(CC(C)(C)NC(=O)C=CC2CCOC2)C)CCNC1=O C1(COC)CCC(NC(c2csc(Cl)c2)C)C1 C(=O)(C(CC)CC(C)C)NC1CCCC(NC(C2CC(C(=O)OCC)C2)=O)C1 C(=O)(C(O)CC(C)(C)C)NCCC(CNC(c1c(CC)con1)=O)O c1(NC(CN2CC(C)(OC)C2)=O)ccc(N)c2ccncc12 CC(C)CC(CNC(c1cc(-n2nnnc2C)ccc1Cl)=O)C(=O)O C1(C(=O)N2CCCCO2)C2CCC1CN(C(c1cn(C)nc1C(F)F)=O)C2 N1(C(c2cc(C)c(Cl)s2)C(=O)NCCCF)CCC(N=[N+]=[N-])CC1 n1(CC#C)c(C)cc(C(=O)NCC(C)NC(c2ccc(=O)n(C)n2)=O)c1C c1(C(=O)NC)cccc(OCC(=O)NC2(F)CN(C(C3COCC(C)O3)=O)C2)c1 N1(C(=O)CC=C(Cl)Cl)CC2OCCN(C(c3cnn4cc[nH]c(=O)c34)=O)C2C1 Cc1cc(C(=O)NC2CCCCN(C(=O)C(N)=O)C2)c(C)n1-c1ccccn1 Cc1ccc(N)cc1C(N1CC2CC(C1)C2NC(=O)C(c1ccccc1F)C)=O Cc1cc(C(N2CCN(C(c3cnn[nH]3)=O)CC2C)=O)cc(C)c1Br N1(C(C2(C3CCCO3)CCC2)=O)CC2CCC1CN2c1ncnc(O)c1Br c1(OCC(C)NC(=O)NCC2CSCCS2)ccc(F)cc1F CC1CCN(C(=O)C(C)N(C(=O)CC2CC(C3CC3)C2)C2CC2)CC1(C)C C1(O)(CN(C)C(C2COC(=O)N2)=O)CCN(C(=O)COC2CC=CC2)C1 C(c1cnc[nH]1)=C(C)C(=O)NC1CC(NC(=O)CCc2csc(Br)c2)C1 c1(C(=O)NC(CN(C(C(CC)(C)OC)=O)CC)C)cccc(OC)c1F C12(CC(N3CCC(N(C(c4c[nH]c(=NC)o4)=O)CCO)C3)=O)CCC(C)(C1)OC2 Cc1nsc2ncc(C(=O)NC3CN(C(=O)C(n4nccc4C)C)CC3C)cc12 c1(C(=O)NCc2c(C(N(CC(COC)O)C)=O)n[nH]c2)ccccc1O N#Cc1ccsc1C(N1C(C(=O)NC2(c3nc[nH]n3)CC2)CC2CC12)=O C(CCCCCNC(C1CC(O)C1)=O)NC(C1CC(N(C)C)C1)=O C(=O)(C1CCOc2ccccc21)N1CCC(CNC(C#CCC)=O)C1(C)C CN(CCCC(=O)N1CCC(=CCNC(=O)C=Cc2cscn2)CC1)N=O CCCCCCC(F)C(=O)NCC1CC(NC(c2cc3n(n2)CCCC3)=O)C1 c1(C(N(CCn2cc(CCCSC)nn2)C)=O)c[nH]ccc1=N C1(O)(CC)CCCN(C(C2CC(CCNC(=O)CCC(C)C(=O)OC)C2)=O)C1 C1(C(=O)NCC(CNC(C(C)OCCCC)=O)O)CN2CCCC2CO1 N1(C(c2nc(CC)oc2C)=O)CCCC(NC(=O)Cn2ncnn2)CC1 C1(C(=O)NCC23C(CN(C(c4c(C)con4)=O)C2)C3)Cc2ccccc2C1 c1(C(N2CC(OC)C(NC(c3cscc3F)=O)C2)=O)ncc([N+](=O)[O-])n1C N1(C(c2c(CC)sc(=N)[nH]2)=O)CC2CC(NC(=O)CC3CC=CCC3)C2C1 C1(C(=O)NCC(=O)NCC(C)(C)C)CCS(=O)(=O)CC1 CC1=C(C(=O)NCC2CCCCN(C(C3(C)CC3C)=O)C2)Cn2ncnc2N1C C1(CNC(CSc2cccc(C)c2)=O)CN(C(=O)C(C)S(C)(=O)=O)CCN1C C1(NC(C2CCOC2=O)=O)CC2(CCN(C(c3c[nH]c(Br)c3)=O)CC2)C1 C(=O)(C1=CC2C=CC1C2)NC1(C(N2CC(C)(CO)C2)=O)C(C)(C)C1 c1(C(=O)NC(CC(=O)OC)(C)c2cccc(F)c2)ccc2c(c1)C(=O)NCCO2 C(=O)(C(CC)(CC)CO)N1CCN(C(CC(=C)C)=O)C(CC2CCC2)C1 c1(C(N2CC(CC=C)(NC(c3cncn(C)c3=O)=O)C2)=O)cc2occc2n1C c1(C(=O)NCCN(C(=O)COCC2CCCCO2)C)[nH]c2ccc(C)cc2c1Cl N1(C(CCC2CCCN(C)C2)=O)CC(CO)C2(C1)CN(C(=O)C(=O)NC1CC1)C2 CC1(C)CN(C2CN(C(=O)N(S(=O)(=O)c3cccs3)CC3CC3)C2)C(=O)O1 C1(CN(C(=O)C2=CCOC2)C)CCN(C(c2ccc(Br)cn2)=O)CC1 c1(N2CCCC(CNC(CN(C(=O)OC)C)=O)C2)nc2c(C(N)=O)cccc2o1 C1(CC(=O)NCC(C2CCOC2)NC(c2cc(Cl)cs2)=O)COCCO1 C1(C(N(CCOC)C)=O)CN(C(=O)CCCC2(C)N=N2)CCO1 c1(N(CC(=C)C)C)nc(N2CC3C4CCC(C4)C23)nc2cc[nH]c12 c1(CC(=O)NCCN(CCOC)C(c2ncncc2Cl)=O)ccc(OC)c(F)c1 C1(CC(N2CC(C(=O)NCC3(CC)CC3)OCC2)=O)CCN(OC)CC1 C1(C(=O)NC2CCOC(C)C2)(CC)CCCN1C(=O)CCCc1cnn[nH]1 C1(NC(c2c(CC)n(C)nc2)=O)CCC2CN(C(=O)C=CC(=O)N(C)C)CC2C1 C1(NC(CCC)=O)CC=C(C(=O)NCc2cccc(F)c2)C1 N1(C(C(n2c(=O)oc3ccccc23)C)=O)CC2CCCN(C(C3CC3C)=O)C2C1 N1(C(C2(CCC)CC2)=O)CCCN(C(=O)C(C)SC)C(c2ccccc2)C1 C1(CC(N2C(C)CCCC2)=O)C2CCCC2N1C(=O)CNc1ncccn1 C1(C(=O)NCCCO)(CN(C)C)CCCC1 C#CCC(C)(C)C(=O)N1CCC(CO)(CNC(c2c(OC)ncnc2C)=O)CC1 CCCCC(O)C(C)C(=O)N1CCCC(NC(=O)Cn2nc(C)n(C)c2=O)C1C CCC(COC)C(=O)NCC(O)CCNC(c1[nH]c(C)nc1C)=O C(CCC(=O)N1CCC(CF)C1)(C(C)C)NC(CCCC(C)C)=O C(=O)(CCCC(=O)NC1CC(C)N(C(=O)Cc2c(C)nn(CC)c2C)C1)OCC N1(C(c2c(NC)cnnc2)=O)CC2(CCN(C(=O)CC3CCOC3)CC2)CC1C C1(NC(CCc2cc(OC)no2)=O)CCN(C(=O)OC(C)(C)C)C(C)C1 N1(C(c2c(C)snn2)=O)CC(O)CC1CNC(=O)C(c1cnn(C)c1O)=O C(=O)(NNC(=O)Cc1c(C)noc1C)N(CCCC)Cc1ccc(OC)cc1 CCCCC(C)(F)C(=O)NCC1COCCN(C(=O)Cc2cncc(OC)c2)C1 C1(C)(CC)C=C(C(=O)N(C2CN(C(c3cncc(F)c3)=O)CC2O)C)C1 N1(C(c2ncn(C)c2)=O)CCC2C(CCCN2C(c2cccc(CO)n2)=O)C1 CC(C)C(O)C(=O)N1CCC(OCCNC(c2ncccc2C(F)(F)F)=O)C1 N1(c2c(C)cncn2)CCC(O)(CNc2ccc(C(F)(F)F)[nH]2)CC1 O=C(C1=CC2C=CC1C2)NC1(CNC(C2CC3(C2)CC2(CC2)C3)=O)CCCCC1 N1(C(CCC(=C)C)=O)CCC(C2CC(NC(c3nc(C)c(C)nc3C)=O)C2)C1 C(=O)(C(C)C(O)C(C)CC)NCCN(C(c1cn(CCCC)nc1C)=O)CC C(C(=O)NNC(=O)c1cc(Br)ccc1F)OC(C1C(C)(F)CCC1)=O N1(C(C2(COCC)CC2)=O)CCC(NC(c2ccc(C3CC3)cc2)=O)C(F)C1 c1(C(N2CCN(C(C(C=C)CC)=O)CC(C)C2)=O)cccc2cnccc12 N1(C(C=Cc2n(C)ccc2)=O)CCCC(NC(c2cscc2Cl)=O)C(F)C1 C1(NC(Cc2c(C)noc2)=O)CN(C(=O)CC2CCC3(CC3)CO2)CC1N=[N+]=[N-] c1(OC)ccc(C(=O)NCC(C)NC(=O)CC(F)(F)Br)c(OC)c1 C1(CNC(CN(C2CC(C#N)C2)C(COCCC=C)=O)=O)CCCC(CO)C1 n1(CCOC)nccc1C(=O)NCC1CCC1NC(=O)CCC1CCCO1 c1(CC(=O)NCC2C(NC(C(C)(C)OC)=O)COC2)ccc2c(c1)COC2 C(=O)(N=c1[nH]c(Cl)ncc1C)c1nccc(C)c1.C1(C(C)C)CCC(=O)N1 Cc1c(-c2nc(C3CC3)nn2CCN(C)C)sc2ncc([N+](=O)[O-])cc12 c1(N2C(C(=O)Nc3cccc(OC)c3Cl)CC3CC32)ncnc2ncc(Br)cc12 N1(C(C(=O)C(C(C)C)OC)=O)CCCN(C(=O)N(C)C)CC1.CO Cc1nc(-c2ccc(C(=O)O)cc2)sc1CNSCC(c1cccc(F)c1)C=O CCCC(C)CC(=O)N1CCCC(NC(=O)COc2cccnc2)C1CC c1(C(N2CC(F)(CSCC)C2)=O)ccc(N2CCCC2)cc1.C12CC1C(=O)N2 C1(CC(=O)N(C2CC(C)C2)C)CN(C(c2cccc(OC3CC3)n2)=O)C(C)(C)C1 S(=O)(=O)(c1cnc2ccccn12)Nc1nc(-c2c(S(CC)=O)cccc2)n(C)n1 C1(CNC(c2n(C)cnc2)=O)CCC2(CN(C(c3cc(=O)n(C)o3)=O)C2)O1 Cc1ccn(C)c(=O)c1NC(=O)C(O)C1CN(C(C2CCCC2C(C)C)=O)C1 C1(C(=O)NCCC(=C)CNC(=O)CC2CC3(CCO2)CC3)CCC(F)(F)CC1 Cc1csc2nc(CC(=O)NC3CCCCC3NC(=O)CNC(N)=O)cn12 Cc1ccn2c(C(N3CCC(C)(NC(C4CC4C(=O)NCCO)=O)C3)=O)cnc2c1 C#Cc1c[nH]nc1C(N1CCCC(NC(C2CCN(C)C2)=O)C1)=O c1(CCN2CCCC(CC(=O)OCC)CC2)nc2cccnc2[nH]1 CCC(CNC(=O)CN(C(=O)C(C)CSC)CCOC)(CC)CC c1(C(N2CC(OCCNC(=O)C3=C(Cl)CCCC3)C2)=O)cnc2ccncc2c1 N1(CC2C(CNC(=O)OC(C)(C)C)C2)CCCC(c2ocnc2CC(N)=O)C1 c1(C(=O)NC2CC(NC(C(CC)C)=O)CC2O)c(Br)ccc(Cl)c1F c1(C(=O)NCC2(C(=O)NC3C(C)(O)CCC3)CCCCC2)ccc2cccnn12 c1(C(=O)NC(C2CCN(C(CNC(C(CC)C)=O)=O)CC2)C)c(Cl)nn(C)c1Cl C(CNC(c1cc(C(F)F)cc(F)c1)=O)(C(C)C(C)C)NC(COC)=O c1(CC)ccc(F)c(C(=O)NC(C)CCCNC(c2cncc(OC)c2C)=O)c1 c1(C(N2CCC(C(CNC(C(C=C)O)=O)C)CC2)=O)cc(N)ccc1Cl c1(C(=O)NCC(CC=C)NC(c2cnnn2C2CC2)=O)cc2ccsc2s1 C1(NC(C2(C=C)CCN(C(=O)C(c3cnn(C)c3)C)C2)=O)CN(C)C(=O)C12CC2 CCC(C)CCCC(=O)N1CCCC(CNC(c2c(C)noc2N)=O)CC1 Cc1c(Cl)ccc2c1CN(c1nccc(=NCC3CC4(CCC4)C3)[nH]1)CC2 N1(C(C2(C(N(C)C)=O)CC2)=O)CCC2(CCN(C(c3cc(Br)ccc3F)=O)C2)C1 CC(C)(C)CCC(=O)C(=O)N1CCC2(CNC(=O)Cc3ncno3)CCCCC12 c1(OC)c[nH]c(C(=O)NCC2CCCN2C(=O)Cc2ccc(C)nc2Cl)cc1=O CC(C(C)(C)C(=O)NC(C1CCC1)C1CCC1)NC(c1ccsc1Cl)=O CCCC(C(O)C(=O)Nc1scnc1CC)NC(C1CN(CC)C1)=O N1(C(C(C)(C)OCC)=O)C2CCC1CN(C(c1n[nH]c(C)c1F)=O)CC2 C1(CNC(CC(CN(C)C)O)=O)CC2CCC1N2C(c1cnsc1)=O Cc1nc(N2CC3CC3(C(=O)NCC(=O)NC3CCCCC3)C2)c2c[nH]nc2n1 CC1CN(C(C2(Br)CC23CCC3)=O)CCN1C(C1CC2(CC2)CO1)=O C1(C(=O)NC2C(NC(c3ccc(F)s3)=O)CCOC2)Cc2cccnc2C1 c1(C(N(C2CCCC2)CC(C)C)=O)cnc(CNC(=O)CC2CCC(C)O2)nc1 C1(C)(N(CC(C)SC)C(=O)COCCOCCO)CSC1.C=O N1(C(CCCC#C)=O)CC2CCCC1C2CNC(c1cnn2cccnc12)=O C(c1cccc(F)c1)=CCNC(C1C(NC(C2(C)CC(=C)C2)=O)CCCC1)=O C#Cc1ccc(C(=O)N(C2CCCC(N(C(=O)C3=NOCC3)C)C2)C)cc1Cl Cc1nc2ncnn2cc1C(=O)NC1CC(C)(NC(=O)CN2CCCCC2C)C1 Cc1cccc(C(=O)NC(C)(C)C(=O)NC2CCC3CC23)c1C#N N1(C(C(C)(C)NC(=O)OC)=O)CC(CNC(c2ccsc2Cl)=O)OC(C)(C)C1 Cc1ccccc1C(=O)NCc1cccnc1CNC(C1CC2CCC12)=O CCCCCCCCCC(CC(c1ccc(F)c2cccnc12)=O)CCCC N1(C(C2CC23CC3)=O)CCCNC(CO)C1 c1(C(N(C)CC2CCC(NC(C=CCCC)=O)CC2)=O)cc(O)nc(O)n1 c1(OC)cc(CN2CC3C(C(=O)NCCc4cnn(C)c4)C3C2)ccc1O c1(CC)c(C(=O)NC2CC2CNC(=O)Cc2csc(-c3ccoc3)n2)ccn1C C1(NC(C2(OC)CC2)=O)CCCC(C(=O)NCc2cccnn2)C1 C(c1cnn(C)c1)=CC(=O)NC(CN(C)C)C(=O)NCC#CCCO c1(C(N2CCCC(NC(CC(C)C3CC3)=O)CC2)=O)nc2ccccn2c1F c1(NC(C2(F)CC(NC(c3c(C)ccs3)=O)C2)=O)cnc(-n2cccn2)cn1 Cc1cccn2c(=O)c(C(=O)NC3CC(C(=O)NC4C5CCOCC45)C3)cnc12 c1(C(N2CC(C)(NC(=O)C(O)Cc3ccccc3)C2)=O)sc(Cl)cc1Cl c1(C(N(C2CCN(C(=O)CC3CCC(F)(F)C3)CC2)CC#C)=O)cc(=N)[nH]n1C Cn1cc(C(N2CCC(N(c3ccc([N+](=O)[O-])cc3)C3CC3)C2)=O)c(=O)c(Br)c1 C(=O)(CCCCN(C)C)N1C(C(C)NC(c2ccoc2C2CC2)=O)CCC1 C1(C(N2CCCC(O)(C(F)F)C2)C(=O)NCCCOC)CCS(=O)(=O)CC1 C1(NC(C(Cn2cncn2)NC(c2c(C)nc(C)s2)=O)=O)CC2(CCC2)C1O c1(SCC(=O)NCC2CCCN2C(C2CCC2)=O)nnc(S)s1 N1(C(c2c(CC)nco2)=O)CC(NC(=O)CCn2ccnc2C)CC(O)C1 C1(c2nnnn2CC(F)F)(NC(COC)C2CC2)CCCC1OC.c1nnc(Br)n1C N1(C(N2CC(c3ccc(Br)s3)C2)=O)CCCC1CCC1CCC1 C(=O)(C(F)C(C)C(F)(F)F)NC(CC)CNC(=O)C=Cc1ccc(Cl)s1 C1(NC(CC=CC=C)=O)CCCCCC1C(N1CC(CO)C2(CC2)C1)=O c1(NC(N2C(CC(=O)N(CC)CC)CCCC2)=O)c(-n2nccn2)cccc1F C1(NC(COCCC#C)=O)CC1C1CCN(C(C2CCOC2=O)=O)CC1 C(=O)(C1CCc2scnc21)N1C(CCNC(CCCCOC)=O)CCC1 C12(C(=O)NCC(CNC(C3(n4ncc(C#N)c4)CC3)=O)F)CCC(F)(CC1)C2 c1(C(N2CCCC(N(C(C3CC3(F)F)=O)CC)C2)=O)c(F)cncc1Br N1(C(C2CCCC(C(=O)OC)C2)=O)CCN(C(=O)CCC(C)=O)C2CC12 c1(CNC(C2(F)CCN(C(c3c(OC)ccs3)=O)C2)=O)cc(F)c(Br)cc1C C(CCCC(=O)NC(c1ccccc1C(=O)O)C(F)(F)F)N(C)C C1(C(F)F)(OCC2CC2)CCN(C(C(CCC)N(CCSC)C)C(=O)NC)CC1 N1(C(=O)OC(C)(C)C)CC2(CC(=O)OC2NC(C2(C#N)CCC2)=O)C1 N1(C(CCc2ccc(C)nc2)=O)CC(C(N2CC(C)C(O)C2)=O)CC(F)C1 c1(C(=O)NCCCCCNC(=O)CCF)c(Br)ccc2c1OCO2 N1(C(COC(C)(C)C)=O)CCC2(C1)CN(C(=O)C=CCC(F)(F)C(F)(F)F)C2 CCCC(C)(C)CC(=O)N1CCC(N(C(c2nccn3cnnc23)=O)CC)CC1 N1(C(CC2CCCC(OC)C2)=O)CC2CCCC(C1)N2C(C1(C)CC=CC1)=O c1(OC)cc(C(F)(F)F)nc(N(C2CN(C(=O)CCC3CCCCO3)C2)C)n1 c1(C(N2C(C)CC(CNC(c3cc(CC)c(C)o3)=O)C2)=O)cc(C)[nH]c(=NC)n1 c1(NCc2c(C)c(N)ccc2)cc(=NCc2cc(Cl)ccc2Cl)[nH]cn1 C(=O)(CC1CCc2ccccc21)N(CCNC(c1cscc1C(F)F)=O)CC C1(C(N2CCC(C(C)NC(=O)Cc3cnc(C4CC4)o3)C2)=O)CC2(CCC2)CO1 CC(C)(C)C(CNC(=O)CC1(O)CCCOC1)C(=O)NCc1ccncc1F c1(N2CCC(C)C(NC(c3scc(COC)c3)=O)C2C)nc2cccc(C)c2s1 c1(NCC(C(=O)NCC(=O)OC(CC)(C)C)(C)C)ccnc2c(Br)cccc12 C1(NC(Cc2cn(C(C)C)nc2)=O)CC2(CCN(C(C3CCC(C)(C)C3)=O)C2)C1 Cc1ccc(C(=O)NCCc2ocnc2CNC(C2CC(C)CO2)=O)cc1F C1(NC(=O)C=C(Cl)Cl)CCCC(CNC(c2cccnc2OCCO)=O)C1 c1(C(=O)NC2(COC)CN(C(=O)CO)C2)cccc2c1OCCO2 N1(C(=O)CC2CCCC23CC3)CC2(CCC(NC(C3(CF)CCOCC3)=O)CC2)C1 N1(C(C(CC)OCC)=O)CC(CO)C2(C1)CN(C(=O)CCn1nc(C)nc1C)C2 C1(C(=O)NCCOCCOC)CCCC(NC(c2cncc(F)c2)=O)C1 CC1CN(C(C2CN(C(=O)CC=C(Cl)Cl)CC2(C)C)=O)CCCO1 C1(C)(C(N2CCC(OCC=C)C2)=O)CN(C(c2ncccn2)=O)C(C)(C)C1 C1(NCCCCC2(NC(=O)Cc3c[nH]n(Br)c3=O)CC2)CCC2CC1CO2 CC(C)(C)C(CO)C(=O)NCC=CC(=O)NCC1CC2(CCO1)CC2 c1(COCC(=O)NCC(CC)NC(C2CCCCS2)=O)ccccc1C N1(C(C(C)NC(C2CCC2)=O)=O)CC2CN(C(=O)CC3CCOC3=O)CC2(C)C1 C1(NC(C(CC=CC)NC(=O)C=C(C)C)=O)(CO)CC2CCCC12 C(=O)(CCCCCCSC)N1CCCC(F)(CNC(C2(C#C)CCCC2)=O)C1 Cc1[nH]nc(Cn2cc(C(C)O)nn2)c1Br.c12cccc(c1)CO2 c1(C(=O)NC2(CO)CCN(C(C3CC=CCC3)=O)C2)c(OC(F)F)cccc1F c1(-n2cc(C(C)N(C)C(C3CC3(Br)Br)=O)nn2)ccc(F)nc1 c1(C(=O)NC2CN(C(c3n(CC=C)ccc3)=O)CC2C)nc2n(c1Cl)CCCC2 c1(Cc2nc(C(=O)NCCCNC(CCC#N)=O)sc2)cc2c(nn1)CCCO2 C1(C(N(CC(CN(C)Cc2cc(Cl)ccc2Cl)O)C)=O)CCC2CCCCN12 N1C(=O)NC(c2cc3c(s2)CCCC3)C2=C1C(Cc1nc(=N)[nH][nH]1)OC2=O c12ccc(c(Cl)c1)CCN2.c1(C(=O)OC)ncc(-c2cnccn2)s1 C12(C(N3C(CNC(=O)C(O)CC(F)(F)F)CCC3)=O)CC3CC(C1)CC(O)(C3)C2 C1(CCC)CCCC(NCN2CCC(CC(O)C(=O)OC)CC2)C1 C(C)(C)(C(=O)NC1CC(CNC(C2CCC(C(=O)OC)C2)=O)C1)SC C1(NC(c2nc(C(C)C)oc2)=O)CC(C(N2CCCC2)=O)C12CCC2 c1(OCCCC(=O)NCCN(C(C2CCCO2)=O)C2CC2)cccc(F)c1 c1(C(=O)NCC(CCOC)NC(=O)CCS(C)=O)ncc(C)cc1Br CC1(C)CN(C(=O)CC2(O)CCOC2)CC1C(=O)NCCN1CCOC1=O c1(C(CO)NC(C2CC(=O)N(CC3CCCO3)C2)=O)c(F)cccc1Cl c1(C(=O)NC(C)CC(C)NC(c2cnoc2-c2cccs2)=O)ncc(F)cc1F C=C=CCCC(=O)NCC(C)(C)CC1CN(C(C2COC(=O)C2)=O)C1 Cc1nnc2n1CC(C(N1CCN(C)C(CNC(=O)CN(C)C(N)=O)C1)=O)CC2 C(C(F)(C(=O)N(CC(O)CN(C)C)C)C(C)C)NC(C1(CC)CC(C)(C)C1)=O N1(Cc2cncc(C)c2)C2CCC1CC(NS(=O)(=O)c1cn[nH]c1)C2 C(=O)(C(F)(CNC(=O)CC1CSCCO1)C(C)C)NCCCc1c(C)n[nH]c1 c1(CC)ccccc1CSc1ccccc1-n1nnnc1C(N)CCCC C1(NC(c2ccc(CNC(CC3N(C)CC=CC3)=O)cn2)=O)CCC(=O)N(C)C1=O CCCC(CCCNC(=O)C(C)Cc1c(C)n[nH]c1C)NC(c1ccsc1C)=O c1(CSCC(=O)NC2CCC(NC(c3cnc(C(F)F)s3)=O)C2)cnccc1Cl CCC(COC)(CC)C(=O)NCC1CCCC1OC.c1(O)ccccc1F.C1(=O)CO1 c1(CC(=O)NC(CNC(C2CCCSC2)=O)C2CCC2)cccnc1Cl N1(C(CCNC(C)=O)=O)CCOC(CNC(=O)CCCNC(=O)C(C)C)C1 c1(C(=O)NCCCN(C(C(CCCC)C)=O)C)cccc2c1CCN2 N(C(=NCC1CCC1)NCC1CC1Cl)CC1CCCCC1 C(=O)(C1CCc2c(Br)cccc21)N1CCCN(C(C(C)C)=O)C(C)C1 CCCCC(C)(F)C(=O)NCCN(C(=O)C(C1CCC1)OC)CCC N1(C(C(C)CC2CCC2)=O)CC2CC1CN(C(=O)CCc1nncn1C)C2 C1(CCCOC(=O)CC2CCCC23CC3)CCC2(CC2)C(=O)O1 Cc1cc(O)c(C(N2CC3C(CNC(=O)Cc4csc(C)n4)C3C2)=O)nn1 c1(C(C(=O)NC2CCC(CNC(COC(C)(C)C)=O)C2)O)ccc(F)c(Cl)c1F CC1CN(C(=O)C=CCF)CC(C)N(C(=O)CCc2cn(C)nn2)C1 C(=O)(C(C)CCCC(C)C)N(CC(N1CCC(OC)(CO)CC1)=O)CC1CC1 C(=O)(C(CC)C(=O)OC)NC1C(NC(CC(=O)NCC#C)=O)CC1 N1(C(C2C(C)=CCS2)=O)CCN(C(c2nn(C)cc2Cl)=O)CC1C C1(OC)(OC)CC(C)(C(=O)NCC(C(C)C)NC(=O)Cc2ccccc2O)C1 c1(NC2C3CN(C(CC(C(=O)OC)(C)C)=O)CC32)ccc2c(ccn2C)c1 C123COC(C1)(C2)CNC3=O.C1(NC(CSC(C)C)=O)CCC1C(F)F C(C(CC(F)(F)F)NC(=O)CN(C)C(C)C)NC(C1C(=C)C1)=O c1(C(=O)NCCN(CCC)NC(C2(C)C=CCC2)=O)n[nH]c(C)c1[N+](=O)[O-].OC C1(NC(C=CCOC)=O)CCC(C)N(C(=O)CCc2ccc(C(=O)OC)nc2)C1 C(C)(N=c1cc(C)nc(-n2nc(C)cc2C)[nH]1)C1CCN(C(=O)OCC)CC1 C1(CNC(c2nccc(C(=O)OC)c2)=O)CC(NC(c2ccc[nH]2)=O)C12CCC2 c1(C(=O)OCC)ccc(C(=O)NCc2ccc(N3CCOCC3)cc2)cc1 n1(CC)nc(C)c([N+](=O)[O-])c1N1CCN(C)C(CNC(=O)C2=C(C)OCCS2)C1 C1(C2CCCC2)(CNC(C(=O)NCC(CCCCCCC)O)=O)CCNC1=O c1(C(C2(c3ccccc3)CCCCO2)=O)ccc(F)cc1F N1(C(CNC(C(n2c(C)ccn2)C)=O)=O)CCN(C(=O)CC(C)(C)C)CC1 c1(C(N2CCC(C(C)NC(C=CCOC)=O)C2)=O)n[nH]c2c(OC)cccc12 C(=O)(C1CCC(=O)c2ccccc21)NC1C(NC(CCS(N)(=O)=O)=O)C1 C1(CC)=CC=C(C(=O)NCC2C(C)CCN2C(=O)CC2(CC)CCC2)C=CCC1 C12CCC(CC1)C(=O)N2.c1(NC)scnc1C(=O)NCCN1CCC(CO)C1 C1(C2CCCN(C(c3noc4c3COCC4)=O)C2)(NC(CS(N)(=O)=O)=O)CC1 c1(NC(CC2N(C(C3CC(C(=O)OC)C3)=O)CC(O)C2)=O)cnc(Cl)c(C)c1 N1(C(C(C)n2cncn2)=O)CC2CCC1C(CNC(c1ccc(C3CC3)s1)=O)C2 C1(NC(c2cccc(N(C)C)c2)=O)C2CC3CN(C(=O)CC4(O)CCC4)C1C3C2 C1(C(C)C(=O)NC(Cn2cc(C3(CO)CCC3)nn2)C2CC2)CCC(C)(C)CC1 C(=O)(CC(O)C(C)C)NC1(CCNC(c2nc(COC)oc2)=O)CCC1 C1(C(=O)NCC2(C)CC(NC(C3CCC(F)(F)CC3)=O)C2)COCC2(CCC2)O1 Cc1c(C(N2CC(NC(c3cc(N)ccc3O)=O)CCC2C)=O)sc2cncn12 c1(CC)sc(C(=O)NCCOCCCN(C)C(C2(C)CC3CC3C2)=O)cc1C C1(C(=O)NCCOC2CCN(C(=O)C=C(Cl)Cl)C2)CC2(CSC2)C1 C1(Cc2nc(C)on2)CCCN(C(C2CCC(N)C2)=O)C1 O(N(CC)C(=O)CC1(C(F)F)CCCC1)C(=O)C CCC(C(=O)NCCCN(C(C1(F)CC1c1ccccc1)=O)C1CC1)NC(N)=O C1(C(=O)NCC2(O)CN(C(c3ccc(COC)[nH]3)=O)C2)CC12CCCOC2 C1(CNc2c(C)c(N3C4CCC3COC4)ncn2)(CO)CC2CCC1CC2 N1(CC(=O)NCC(CC)NC(=O)CS(=O)CC)CCc2ccccc21 c1(C(=O)NC(C)CNC(=O)Cc2cn(C)nn2)cc2ccc(C(C)(C)C)cc2[nH]1 N1(C(c2ccc(C(C)(C)C)cc2)C(=O)NC)CCC2CS(=O)(=O)CC2C1 c1(C(N(C(C)C)CCNC(C2(CO)CCC2)=O)=O)coc(C(F)Cl)n1 c1(O)cc(OC)c(F)cc1F.C(=O)(CCNC)OC C1(C2CN(C(c3ccc(F)cn3)=O)C2)(NC(=O)Cc2cscc2Br)CC1 N1(C(C2(C)CCCC2(F)F)=O)CCC(C2(O)CN(C(=O)CC3CCCC3)C2)CC1 c1(CNCC2N(C(c3ncc(C)c(Br)c3)=O)CCOC2)cccc2c1CCC2 Cc1ccsc1-c1cn(CC2CCCN2C(c2c[nH]nc2C)=O)nn1 Cc1cc2c(C(=O)NCC34CC(CN3C(C3(C)CC3(Cl)Cl)=O)C4)nccn2n1 Cc1cc(C(=O)N(CCNC(C2(C3CC3)CCC2)=O)C2CC2)c(F)cc1Cl S(=O)(=O)(c1ccsc1C(=O)NC1CN(C(C2CCC(=O)O2)=O)CC(F)(F)C1)NC CC(C)CCC(C(=O)N(C)CCOC1CC1)NC(=O)C#CC1CC1 c1(C(N2CCCC(CCNC(C(F)=CC)=O)C2)=O)noc2cc(Cl)ccc12 N1(C(CCC(C)O)=O)CC2(CC2)CC1CNC(=O)CCCN1CCCCC1 C1(O)(CC)CCN(C(C2(CNC(C3CCCO3)=O)CCCO2)=O)C1 N1(S(CC)(=O)=O)CCC(C(=O)NC2CC(NC(=O)CN(C)S(N)(=O)=O)C2)CC1 C(C(O)C(=O)N=c1cc(C)n(C2CC2)[nH]1)NC(CC(CC)(C)C)=O c1(C(=O)NC2CCCN(C(C(C)(C)COCC(F)F)=O)C2)csc2c(F)cccc12 CC(C)P(=O)(CC(=O)N(C(C)CCNC(=O)CC1SC(=N)NC1=O)C)C(C)C Cc1nc(NCC(C2CC2)NC(C2CCCC(C)(C)C2)=O)ccc1C#N C1(C(=O)NCCCCN(C(=O)CN2CCOC2=O)C)CC12CC2(F)F c1(OC)cc(C(F)(F)F)ccc1CNC(c1sc(C)nc1C)C(=O)NC1(CO)CC1 c1(SCC)ccc(C(=O)NCCN(C(=O)C(C2CCCO2)OC)C(C)C)cc1 n1(CC)nc(C(N2CCOC(C(=O)NC(C)C(C)(C)OC)C2)=O)cc1O CC(CC(C)(C)C)C(=O)N(CC(O)CNC(=O)Cc1c[nH]c2cccnc12)C c1(C(=O)Nc2cccc(NC(C3C(=C)CC3)=O)c2)cccc2c1CCCC2=O c1(C(=O)NCC(C)(C)NC(=O)Cc2nc(C(F)(F)F)n[nH]2)csc(F)c1 C1(NC(=O)CCOCCCF)CCCC1CN(C(c1cnco1)=O)C1CC1 CCC(CC)C(C(=O)NCC(C(=O)NC(CC)C(=O)N(C)C)OC)OC C(CC(=O)N1CC(CC(C)NC(=O)Cc2cc(C3CC3)no2)C1)(C(F)(F)F)OC N1(C(CC(CC)(F)F)=O)CCOCC2(COCCN2C(=O)C(C)CC(F)(F)F)C1 C1(NC(c2ccn(CC)n2)=O)C=CCN(C(C2COC(=O)O2)=O)C1 C1(C(=O)NCC2C(C(=O)NCCN3CCCC3=O)CCCC2)(CC)CC(C)(C)C1 C1(N(C(C=C(CC)C)=O)C)CCCCN(C(c2ccc(C)cc2C)=O)C1 C1(NC(c2cc(CC)oc2C)=O)CN(C(=O)CCNC(=O)NC)CCC1CO O=C1NC(=O)N2CCN(C(=O)C(=O)NCC3CC4OC3C3CC43)CC12 Cc1onc(CC(N2CCC(NC(=O)CC3(C)CC3)C(O)C2)=O)c1C#N C1(C(=O)NCCCN(C(=O)CC2(C)CCCCC2)CC)CCN(C2CC2)CC1 C1(CNC(c2c(CC)cns2)=O)CCC2(CN(C(=O)COC3(C)CCCC3)C2)O1 N1(C(c2c(C)cco2)=O)CCC2CCCC12CNC(=O)Cc1cc(C(C)C)no1 C(=O)(C(CC(=O)NCC(C)NC(=O)NC1CC(C)CC(C)(C)C1)C(C)=O)OCC C12(C(N3CCC(C(C)(C)NC(C(COC)C)=O)CC3)=O)CCCCC1OCC2 C1(C)(N(C(C(C)NCCc2ccnn2C)=O)C)CCS(=O)(=O)C1 c1(C(N2CC3C(CNC(c4scc(COC)c4)=O)(C3)C2)=O)nc(C)ncc1Cl c1(CN2C(C(N(C)CCO)=O)CSCC2)cccc(NC2CCCCC2)c1 C1(CC(=O)NCCC(C)NC(c2sccc2C)=O)C(=O)NN=C1C.C(C)(C)(C)O c1(OC)ccc(C#N)cc1CN1CC2CCC1CN2C(C1CC1F)=O CCC1CC(=O)N1C.c1(CC2CC2)cc[nH]c1C(=O)NC1CC(CSC)C1 c1(OC(C(=O)NC(CN(C(=O)Cc2nc[nH]n2)CC)C)(C)C)ccc([N+](=O)[O-])cc1 C(C(O)CC(=O)NC(C12CCC(CC1)C2)CNC(C1CCOC1=O)=O)N(C)C c1(C(N2CCCC(C)(NC(CC(CC)C(F)F)=O)C2)=O)cc2n(n1)CC1(CC1)C2 c1(C(=O)NCC2N(C(C3CCCCC3)C)CCC2)cc2c(Cl)cc(F)cc2[nH]1 C1(C(=O)N(C)CCC2CCC2)(CNC(C2C(Cl)(C(=O)OC)C2)=O)CCCO1 c1(C(N2C(C)CN(C(C(CC#C)C3CC3)=O)CC2C)=O)ccc2cncn2c1 C(=O)(C(F)(CNC(c1ncccc1N)=O)C(C)C)N1C(C(=O)NC)CCCC1 c1(C(N2CC(N(C(C3CCC(OC)CC3)=O)C)C(O)C2)=O)cccc(S(C)=O)c1 C1(NC(CC(=O)N(CC(C)C(=O)O)CC(C)C)=O)CCN(CSCC(F)F)CC1 C(=O)(CCCC(=O)NCc1cc[nH]c1C(=O)NCc1ncccn1)OCC c1(CC)ccc(C=CC(=O)NCC(O)CCNC(C2CCOCC2)=O)o1 c1(C(N2CCC(CN(C(C(CC#C)O)=O)C)C2)=O)cnc(O)c(F)c1 n1(CC(=O)OC)cc(CN(C(C(=O)O)c2cccs2)C)cn1 N1(C(CC(CC)C)=O)CC2=C(C1)CN(C(=O)CC1CCCS(=O)(=O)C1)C2 N1(C(c2ccc(OC)o2)=O)CCC(CN(C(=O)CCCC2CC2C)C)CC1 N1(C(c2c(C(C)C)nns2)=O)CCC(NC(C2(C)CSC2)=O)CC(C)(C)C1 N1(C(C=CC(C)(C)NC(C(C(CC)C)C)=O)=O)CCCC[Si](C)(C)C1 C1(NC(=O)Cc2c[nH]nc2O)CN(C(=O)C(F)CC2CC2)C2(CCCCC2)C1 N1(C(c2c(CC)ocn2)=O)CCC(CN(C)C(c2ncccc2C2CC2)=O)CC1 C=CCC(C(=O)N1CCCC1CNC(=O)Cc1nocc1CC)C(C)(C)C N1(C(c2cc(C)[nH]c2C)=O)CC2(CCC2NC(=O)C(N2CCOC2=O)C)C1 c1(C(C)C(=O)NCC(C2CC2)N(C(=O)CC2CC2)C)cc(F)cc(F)c1 Cc1ccncc1CC(=O)NC(C)C(C)NC(=O)CC=Cc1ccccc1 CCC(CC)(CC(=O)OC)C(=O)NCC(C1CC1)N(C(=O)C(C)c1cccs1)C N1(C(C(CC=C)CNC(c2cccc(C#N)c2C)=O)=O)CC2(CCC(=O)O2)C1 c1(C(=O)NCC(C)NC(c2cncc(N)n2)=O)cccc(Br)c1Cl c1(C(=O)NC2CCC(CNC(C34CCCC3C4)=O)CC2)cnc2n1CCCC2 Cc1nnnn1CC(=O)NCC1(F)CC(NC(=O)CNC(=O)NC2CC2)C1 C1(CNC(C2CCCC2(C)C)c2n(CCCOC)nnn2)CCCC2(CCC2)O1 C1(CNC(C(C)NC(N)=O)=O)CN(C(=O)CCc2cnoc2)CC12CC2 c1(CN2CC3C(NC(C4CC(=O)NC4)=O)(C3)C2)cc(Cl)cc(Cl)c1 CC1(C)OCc2c1n[nH]c2NC(=O)CNc1nccc(Oc2ccccc2)n1 CC(C)(C)C(O)CCC(=O)NCC1CCN1C(c1c(O)ccc2ccccc12)=O c1(CN2C(C(=O)O)(CC)CCC2)nn2cc(-c3ccccc3)nc2s1 C1(C(N2CC(O)(CNC(=O)CCC3NC(=O)NC3=O)C2)=O)OC2CCC1CC2 C1(C(=O)Nc2c(CC)scc2)CC(F)(F)CN1C(=O)C(c1ccoc1)OC C#CCC(CC(=O)NCCc1ccns1)NC(C12CCC(CC1)C2)=O Cc1cc(Cl)c(C(=O)NCC(F)CNC(=O)COC(=O)CO)c(Cl)c1 C1(CCC(=O)N(CC(CN(C(=O)C=CC2CCC2)C)O)C)CCCC(=O)N1 N1(C(CCc2n(C)cnc2)=O)CC2CC(NC(c3ccc(CO)o3)=O)C1C2 C(=O)(C1=C(C)OCCS1)NC1CC(NC(=O)C(CCOC)N)C1.C(CO)O c1(NC(C23C(CN(C(CSC)=O)C2)C3)=O)c(Br)cc(Br)c(C)c1Br Cn1cnc(C(=O)NCCC2(C(=O)NCCCN3CCCC3=O)CC2)n1 C1(C(=O)N(C(=O)CCCn2cccn2)C2CC2)CCc2nc(C3CC3)ncc2C1 C1(CNC(C23CCC(CC2)O3)=O)CCC2(CN(C(=O)CN3C(=O)CNC3=O)C2)O1 c1(OC)ccc(SCC2CCN2C(=O)NCC2CCCN2C2CCOCC2)cc1 Cc1ccnnc1C(=O)NCC#CC(=O)NCCCS(C)=O C1(CC(=O)NCC2CCC(F)(CNC(=O)C=C3CCC3)C2)CCCS1(=O)=O c1(CC)ccc2c(Cl)c(C(N3CC4(C3)CN(C(=O)CCC(C)SC)C4)=O)sc2c1 C(=O)(C#CC1(C)CC1)N1C(C)CC(NC(c2ncn(CC)n2)=O)C1 C=CC(CC)CC(=O)N(C1CCN(C(c2ccnn2CC2CC2)=O)C1)CCC CCCCC(C(=O)NCCc1nc(C)oc1C)NC(C1CCCN1C)=O c1(OC)cc(Cl)cc(Cl)c1NC(C1C(O)CCN1C(c1cccc(Br)n1)=O)=O c1(C(=O)NCC(=O)OC(C)(C)C)ccc(C#N)c(Cl)c1F c1(C(=O)NCC(C2CCN(C(CC=CCC)=O)CC2)C)cnc2c(c1)ncn2C C(=O)(CC(C)(O)C=C)N(CCC(=O)N(C)CC1CCOCC1)CC#C C12(NC(c3c[nH]c(=NC)s3)=O)CCCC1CN(C(c1ccc(C)c(F)c1)=O)C2 Cc1nnc2cc(N3CC(O)(C(C)NC(=O)Cc4ccc(F)c(F)c4)C3)ncn12 c1(CNC(c2c(C)ccs2)=O)cncc(C(=O)N(CC(F)F)CC(C)O)c1 Cc1cccnc1CC(=O)N(C(C)(CNC(=O)CP(C)(C)=O)C1CCC1)CCO C12(COC)CC(C(=O)O)(CO1)C2.c12cn(nn1)C2.C12CC(C1)CCC(=O)N2 C1(C(N(C(C(C)C)C)C)=O)CN(C)CCN1C(=O)C#CC1CC1 C1(CCNC(c2cc(C(=O)OC)on2)=O)CN(C(C2C3COCC23)=O)CCCO1 N1(C(CC=CCCCCC)=O)CCOC(Cn2cc(CCS(C)(=O)=O)nn2)C1 c1(C(=O)NCCC(C)NC(c2cccnc2)=O)cccc(-c2cc[nH]n2)c1 C1(OC)CC(NC(=O)Cc2cnoc2)CN(C(=O)COC(C)=O)C1 C=CCCCC=O.N1(C(C23CC(NCC=C)(C2)C3)=O)CCCC(C)C1 C(=O)(CC(CC)N(C)C(c1ccc(C(C)=O)o1)=O)NCC(CC)O C(CCCCCC(=O)NCCc1ccccc1C)NC(C1(C(=O)OC)CC1)=O c1(C(=O)NC(C2CCCC2)CNC(CS(C)(=O)=O)=O)cc2scc(Cl)c2[nH]1 C1(C(N2C(CNC(C(c3ccccc3)N(C)C)=O)CC2)=O)CCCC1(C)C N1(C(CC(C)C)=O)CC(C2CN(C(=O)CCS(C)=O)C2)C1 c1(C(=O)NC(C2(O)CCN(C(C(c3ccncc3)C)=O)C2)C)cc(Cl)cc(Cl)c1 C1(C)(C(=O)NC2C(C=C)C2)CN(C(c2n[nH]c(C(C)C)n2)=O)C(C)(C)C1 C1(CC)(NC(=O)Cn2nnc(C)n2)CCN(C(c2ccc(C(F)F)cc2)=O)CC1 C=CCC(CC(F)F)C(=O)N1CCC1CNC(=O)C=CSC CC(C)CC(CNC(=O)C(N1CCCC(CCF)C1)=O)OC(F)(F)F C12(C(=O)NCC(CNC(c3cn(C)nc3)=O)(C)O)CCCC(C)(C1)OC2 c1(NC2CN(Cc3c([N+](=O)[O-])cccc3)C2)ccc([N+](=O)[O-])cc1[N+](=O)[O-] N1(C(C(C)OCC)=O)CCC(NC(C2(COC)CC=CC2)=O)C(CC)C1 c1(CC)ncncc1NC(C1(CC)CN(C(C2CC(O)C2)=O)C1)=O N1(C(c2cncc(Cl)c2)C(=O)Nc2c(OC)cccc2)CCC(O)C(O)C1 C(=O)(C(C)N=[N+]=[N-])N1CC(C(C(=O)NC(CC(C)C)C)O)C1 Cc1ccc2oc(C(=O)NCC(C)NC(c3ccc(F)c(Cl)c3F)=O)cc2c1 C1(C)(C(N(CC(CC)NC(C2CC3(CC3)C2)=O)C)=O)C=CCCC1 Cc1ccc(C(=O)NC2(c3ccccc3)CCOC2)[nH]1 c1(OCC)ncc(S(=O)(=O)NCC2(CSC)CC3CC3C2)cc1C C1(C(N2CCCC(CNC(c3c(C(C)O)cccc3)=O)C2)=O)OCCN(C)C1=O C1(C(=O)NC2(CCCC(=O)NCC(C3CCC3)SC)CCC2)CCCCCC1C C12(NC(C(C=C=C)C)=O)CCOC(CNC(c3cncc(O)c3)=O)(C1)C2 C(C(C)(O)C(=O)N1CC(C(F)Cn2cc(CCN3CCCCCC3)nn2)C1)OC c1(NC)cnc(C(N2CC(C)C2C(=O)NCC(C)(C)O)=O)cn1 CCC(COC)C(=O)NCC(O)CNC(c1c(C)coc1C(C)(C)C)=O c1(C(=O)NCC(C)(C(C)C)NC(CC(COC)COC)=O)nc(Cl)cc(N)c1Cl C(C(C)C(=O)NCCC1(C(=O)NCc2nnc(CO)s2)CC1)OC c1(C(=O)NC2CN(C(C3CC3F)=O)CC2O)ccc(=O)n2c1CCCCC2 C1(CNC(c2ccccc2)=O)CC(F)CN1C(c1c(C(=O)OC)ccs1)=O c1(-c2nn(-c3nc(C)nn3C)c(C3CC=CCC3)n2)ccc2c(c1)OCO2 c1(C(=O)NCC(n2cc(C(C)OC)nn2)C)ccc2c(c1)C(=O)OCC2 c1(OCC)cccc(OC)c1CC(=O)N(CCCN(C)Cc1nonc1C)C c1(C(c2nnnn2CC2CCO2)NCCCC)sc(Br)c(C)c1C c1(OC)cc(C)sc1C(=O)NC1C2CN(C(c3cnn(C)c3)=O)CC12 CC1CCCC1(C)NC(=O)C(C1CC1)NC(=O)C(C)N=[N+]=[N-] c1(SC)ccc(C=CC(N2CCCC(NC(c3ccc(=N)[nH]c3)=O)CC2)=O)cc1 c1(C(N2CCC3(CC2)CC3C(=O)NC2CC3CC3C2)=O)nccc2[nH]ccc12 C(=O)(C1=C(C)C(C)(C)OC1=O)NCC(C)N(C(=O)C=CCCC(C)CC)CC C#CCCN=C(NCC1(C)CC(C)(C)C1)N1CN(C)C(=O)C1C C=CCC(C)C(=O)NCC(C)N(CC(O)COCc1ccccc1)C N1(C(CCCCN(C)C)=O)CC=C(C(=O)NC2CCCN3CCCC23)C1 C(=O)(CC(C)(C)C(F)F)NCC1(C(C)NC(=O)C=CC2CC2)CC1 c1(NC(C2C(C(=O)OC)C2)=O)cc(C(N2CCCC(O)C2C)=O)c(Br)cc1O N1(C(C(C)C)=O)CCCC(C2CCN(C(=O)CC3CCC(C)(C)CO3)CC2)CC1 C1(NC(C2C3CN(Cc4ccc(OCC)nn4)CC32)=O)CCN(C)C(=O)C1.C(=O)OC N1(C(C=CC=CC)=O)CC(C(=O)NOCc2ccc3c(c2)COC3)CCC1(C)C N1(C(c2ncc(C)o2)=O)CCC(n2cc(CCC3CCCO3)nn2)CC1.C(CO)O C1(NC(C(C)OCCOC)=O)CCC(C(=O)NC2(COC(F)F)CCCC2)C1 C1(C(=O)NC(CC)CCOC)CCCCC1(C)NC(=O)CC1CCC(C)CC1 N1(C(C2C(C(=O)OC)C2)=O)CC2CC1C2NC(c1sc(C2CCOC2)nc1C)=O C=CCC(CC)C(=O)N1CCC(OCCNC(=O)C=C2CCC(C)C2)CC1 C(C(C)(C)CN=c1cc(NCC2CCSC2(C)C)nc(C)[nH]1)SC Cc1cc(F)cc(C)c1C(N1CCC12CN(C(=O)C(C)NC(N)=O)C2)=O c1(CC)ccc(NC(C2CC(OC)CN2C(=O)CSC(C)C)=O)c(Br)c1 Cc1c(O)ccc(C(=O)NC2CC(C)N(C(=O)CCSc3ccccn3)C2)c1C c1(C(N2C(C(C)NC(=O)CSCC(F)F)CCC2)=O)nnn(C)c1N c1(C(=O)NC2CN(C(c3ccc(C)nc3O)=O)C(C)C2)cc(F)cc2nc[nH]c12 c1(C(N2CCC(CCNC(c3cccnc3O)=O)C2)=O)cnc2ccsc2c1 CC1CC(C)(C)CCC1NC(c1ccoc1CNC(c1n[nH]c(O)n1)=O)=O N1(C(c2ncccc2Br)C(=O)NC)CCC2CSCC2C1 N1(C(C=CCCC)=O)CCCN(C(=O)C(C)CCCc2ccccc2)CC1CO n1(CCC)cc(C(=O)NC2(CCNC(C3CNC(=O)C3)=O)CC2)c(C)n1 CCCC(C(O)C(=O)N1CCC12CCCSC2)NC(c1cccnc1C)=O CC1CCC(F)(F)CN1C(=O)CC(CC(N)=O)NC(c1ccccc1)=O C(C1=NOC2(CCC2)C1)NC(C(C(C)NC(c1c(CCC)[nH]cc1)=O)C)=O Cc1ncc(CN2CCC(=CC(N3CC4(CCC4)C3)=O)CC2)c(C)n1 Cc1cnc(C(=O)NCC2CCC(NC(C3CCN(C)C3)=O)C2)nc1 N1(C(C=CC=CCC)=O)CCCCC1CCCNC(c1scnc1Cl)=O C12(NC(C(CC3CC3)OC)=O)CCCC1N(c1nnc(-c3ccccc3)s1)CC2 Cc1nc(C)c(C(=O)N(C)CC=CC(=O)NCc2nc(N(C)C)n[nH]2)s1 N1(C(c2ccc(C#N)s2)=O)CC2CN(C(=O)CC3(O)CCC3)CC12 C(=O)(C1CCc2cc(Br)ccc21)NC1(CNC(=O)CCCC(F)F)CC1 C1(C(=O)NC2CCCC(NC(c3occ(C(N)=O)c3)=O)C2)CC2(C1)CC21CC1 C1(CNC(C(C2CCC2)OC)=O)CC2(CCN(C(=O)CC3CCC3)CC2)CO1 Cc1sc(O)nc1C(N1CC2C(NC(C3CC34CCC4)=O)C2C1)=O N1(C(c2cnc(C)s2)=O)CCC(CNC(C2CC(O)CN2C)=O)CC1 Cc1nc(CNC(C2CCC(n3cc(C4(N(C)C)COC4)nn3)C2)=O)co1 C(C)(CNC(=O)C(C1CCCCC1)N(C)C)(C(C)C)NC(C=C(C)C(C)(C)C)=O C1(CNC(C2(C=C)CC2)=O)CN(C(=O)CCCC2CCOCC2)CC(C)(C)O1 N1(C(C(C)(C)OCC)=O)CC(C(=O)NCC2(C)CC3CC3C2)CC(C)(C)C1 N1(C(CCc2onc(CC)n2)=O)CC(NC(C2CCCO2)=O)C2(CCOCC2)C1 C1(N(C)C)CN(C(=O)C(=O)Nc2ccnc(O)c2)CC12CC2 N1(C(c2cccc(OC)c2)=O)CCCN(C(c2ccns2)=O)C(C)C1 n1(CC(=O)NC2(CCNC(C(C)OCC)=O)CCC2)cc(OC)c(=O)cc1C c1(C(=O)NCCCCCC)[nH]c2cc(CN3CC(C)C3(C)C)ccc2c1C c1(CN2CCC(CC(=O)NCCC3CCC3)C2)cccc(Br)c1Br c1(C(N(C(CCNC(c2nc(CC)[nH]c2)=O)C)C)=O)cncc(-n2ccnn2)c1 C1(C(N2CCN(C(Cc3c(C)occ3)=O)C(CO)C2)=O)CC2(CCC2)CCO1 c1(CS(=O)(=O)C(C)NN2CC3CC3(CO)C2)ccc(C(F)(F)F)cc1 CC(CCC(C)(C)C)C(=O)NCC1CC(F)CN1C(=O)CC1=CCCC1 c1(-c2cn(CCC(=O)CCc3ccn(C)n3)nn2)cnn2c1NCC2 C1(CC(=O)NCC2OCCN(C(c3cnc(OC)nc3)=O)C2)CCC(F)(F)CC1 CC1(C)CCC(C(=O)NCCc2ccccc2F)(NC(=O)Cc2cnc[nH]2)C1 C1(NC(c2cnc(C)c(C#N)c2)=O)CCCC12CN(C(c1cn(C)c(O)n1)=O)C2 c1(OC)cnc2[nH]c(C(=O)NC3CC(N(C(=O)Cc4nccn4C)C)C3)cc2c1 C1(C(C(=O)NC2(CC)CN(C(CC3(C=C)CCC3)=O)C2)OC)CCC(F)(F)CC1 C(=O)(N=S(=O)(c1ccncc1)C(F)F)c1nn(CC)c(Cl)c1 c1(C(=O)NCC2N(C(C(=O)NCCOC)=O)CCC2(C)C)cc(F)c(F)cc1C c1(C(=O)NCC(C(C)C)NC(C2CCOC2(C)C)=O)cc[n+]([O-])cc1 C1(COC)CN(C(=O)CCCC(=O)OC)CCN1C(=O)C(O)CCSC C(=O)(C#CC1CCCOC1)Nc1ccc(C(N=c2ccn(C3(C)CC3)[nH]2)=O)o1 N1(CC(=O)NC2CC(CNC(C3(COC(C)C)CC3)=O)C2)CCCCC1C C12(C(N3C(C)CC(NC(C(CC)n4cccn4)=O)C3)=O)CCC(CO)(CC1)CC2 C(=O)(C(C)CC(=O)OCC)NC(COCC)C(=O)N1CCCC1CNC(O)C1CC1.C1CC1 C12(NC(C3C(OC)C3)=O)CCCN(C(C3(O)CCOCC3)=O)CC1C2 c1(C(N(C(C)C(=O)N(CCCOC(C)=O)C)CCC)=O)cccc(=O)n1C CCC(CC(C)C)C(=O)NCC1CCC1NC(c1cc(S(N)(=O)=O)co1)=O C1(F)(C(=O)NC2CCN(C(=O)CC3COCCO3)CC2F)CCC(F)(F)CC1 Cc1ccnc(C(=O)NCCN(C2CCCCC2)C(c2ccnc(Cl)c2)=O)c1N CCCC(C(O)C(=O)NC(CO)CCC)NC(c1ccnc(CO)c1)=O N1(C(C#C)=O)CC(C)CN(C(=O)Nc2ccnc(N3CCCC3)n2)C(C)C1 C1(C(C)C)Cc2cnn(C)c2CN1Cc1ccn(C2CCNCC2)n1 c1(C(C(=O)NCC2(C)CCN(C(=O)Cc3ccccc3)C2)O)ccc(F)cc1F CC1=C(C(=O)N2CCC(C)N(C(=O)Cc3cn(C)nn3)CC2)CCCO1 c1(C(C(=O)N(CCCN(C23CC(C2)C3)C)C)N(C)C)ccc(Cl)cc1 C1(O)(C(C)NC(C(C)=O)=O)CCN(C(=O)C=C(C)I)C1 c1(C(=O)NCC(CCC)NC(C2(C3CCCO3)CC2)=O)cnc2[nH]cncc1-2 CC1(NC(c2c[nH]nc2-c2ccccn2)=O)CCN(C(=O)COCCF)C1 c1(N2CCC(NC(=O)Cn3cc(C4CCOC4)cn3)C2)ccc(Cl)c(Cl)c1 C(=O)(C(C)N=c1cccc(S(=O)(=O)NCP(C)(C)=O)[nH]1)c1c(C)cccc1 CCCCCCC(C)C(=O)N1CCCC(C)(CNC(=O)COC(C)(C)CC)C1 C1(NC(c2nocc2Cl)=O)CCC(C(=O)NC2CCCC2O)C1 c1(C(=O)NCC2CC(NC(Cn3c(C)nc(C)n3)=O)C2(C)C)ccc(F)c(N)c1 c1(N2CCC(CNC(C)=O)CC2)nc2c(c(=NCCCC(C)CC)[nH]1)CCC2 C1(NC(Cc2nn(C)c(Cl)c2)=O)CC(CNC(c2n[nH]cc2F)=O)C12CCC2 c1(C(=O)NCC2C3CN(C(C4(C)CCNC4=O)=O)C2C3)ccc(F)c(Cl)c1F CC1CNC(=O)N2CCN(S1(=O)=O)CC2.C(=O)(CC#N)NC(C)C N1(C(=O)OC(C)(C)C)CCC2(NC3CC34CCC(=O)CC4)CCCC12 N1(C(c2c(OC)c(F)ccc2)=O)CCc2sccc2C1CNC(=O)CCC(N)=O C1(C(=O)NC(C(C(C)C)NC(CCN(C)CC)=O)C)CCc2ccccc2CC1 C1(NC(c2scc(C)c2Cl)=O)COC2(CNC(=O)C(C3CCOCC3)O)CC1C2 C1(CC(=O)NCCN(CCOC)C)CCC(NC(=O)C(F)n2cccn2)C1 C1(NC(C(C(C)C)OCC)=O)CC2CCC1CN2C(=O)CCC(C)(C)F Cc1cc(C(=O)NC(C)C(C(C)C)NC(=O)Cc2c(F)cccc2F)nc(O)n1 N1(C(CCC=C=C)=O)CCCC2(CC(NC(=O)Cc3csc(C)n3)CO2)C1 C(=O)(N=c1ncnc2[nH][nH]c(C)c1-2)c1ccc(OCCCCC)cc1.C(CC)N c1(C(=O)OC)cccc(C(N2CCCC(c3nnc(C4CCCCC4)o3)C2)=O)c1 N1(C(c2c(C)sc(-c3ccccc3)n2)=O)C2CCC1C(NC(=O)C=CC(C)C)C2 CC1(C)CC(NC(=O)Cc2ccccn2)CN(C(c2conc2C(C)(C)C)=O)C1 C(C(C)(C)Cn1cc(CCCO)nn1)N(CC)CC1(N(C)C)CCCC1 c1(C(=O)NC2CCC(C)N(C(c3c[nH]nc3F)=O)C2)cn2cnnc2cn1 c1(C(=O)NC2CN(C(=O)CCC3CCC3)CC2F)cc(Br)cc2cc[nH]c12 CC(=O)CCCC(=O)N1CCCC(CCNC(=O)CNS(=O)(=O)C2CC2)C1 C1(=O)CCN(OC)C(=O)C2CN1C2.c1(OCC)ccccc1CSC c1(NC(NOC)=O)cc(Oc2ccc(Br)cc2)ncn1 C=CCN=C(NCC1(CCOC)CCC1)N1CC2C3C=CC(C3)C2C1 C1(C(=O)NCCC2(NC(c3cc(C)sn3)=O)CC2)CCCC2(C1)NC(=O)NC2=O c1(C(C(=O)NC2C=CCN(C(C3OCCN(C)C3)=O)C2)(F)F)ccccc1C#N C(=O)(CC1=NN(C)C(=O)C1)N1C(CNC(C23C(C)OC(CO)(C2)C3)=O)COCC1 CC1Cc2c[nH]nc2C(C(=O)NCC2CCN(C(=O)C=CC3CC3)CC2)C1 C1(C(=O)NC(C)CN(C(=O)CCN2C(=O)CCC2=O)C)CCCCC1(F)F N1(C(c2c(Cl)cc(C)c(F)c2)=O)CCC2CCN(C(=O)C3=NOC(C)(C)C3)CC12 C(CC1=CCN(C(c2ccc3nonc3c2)=O)CC1)NC(C(C(C)C)SCC)=O c1(NC(=O)NC(CO)CO)cc(F)ccc1OCC1CCC1CO C1(CNC(C(C)Sc2ccccn2)=O)COCCN(C(C2(C(F)(F)F)CC2)=O)C1 CC1(C)CC(NC(=O)C=C2CCCCC2(C)C)CN(C(C2(C)CC2(C)C)=O)C1 N1(C(C(C)C(F)(F)F)=O)CCC(C(=O)NCC2(C#N)CC2)C(C)(C)C1 N1(C(C(C)=CC=C)=O)CC=C(CC(=O)N2CCC(F)(F)C(F)C2)CC1 C(=O)(CCCN(C)N=O)NCCC(CNC(=O)C(C)(C)C#N)OC C1(CNC(c2c(C)cns2)=O)CCCCN(C(c2c(O)cccc2F)=O)C1 C1(COC)CN(C(=O)CCSC2CCCCC2)CCN1C(=O)C1=C(C)OCC1 c1(OC)cccc(Cl)c1CC(=O)NC1CN(C(=O)C(F)=C(C)C2CC2)CCC1O N1(CC(=O)NCC(C)(C)NC(C2CCCCNC2=O)=O)CCS(=O)CC1 N1(C(C2(NC(=O)NC)CC2)=O)CCCC2CN(C(=O)C(CC)SC)CCC12.CCO O=C1OC2CN(C(=O)NC3(O)CCN(Cc4ccccc4)CC3)CC2O1 c1(CCC)ccc(C(=O)NCC2CCC(NC(=O)CCCC3CCCO3)C2)cc1 Cc1cc2sc(C(=O)NCCCOCCCNC(C3CC(C)(C)CO3)=O)cc2s1 c1(C(CC(=O)NC2CCN(C(C(CC)CC)=O)C2)C)c[nH]c2ccccc12 CC1CN(C(c2cnn[nH]2)=O)C(C)CN1C(c1ccc(OC(C)(C)C)cn1)=O N1(C(c2cn(CCC)nn2)=O)CCCOC(CNC(c2ccnn(C)c2=O)=O)C1 C1(CC(=O)NCC(=O)OC(C)C)CCCCN(C(=O)CCc2ccsc2)C1 C1(C(N(C2CN(C(c3cnn[nH]3)=O)C2)C)=O)CCN(c2ccccn2)CC1 c1(C(=O)NCC(=O)NC(C)CNC(C2CC2C(F)F)=O)cccs1 C(=O)(C1CCCc2ccnn21)NC1CCN(C(CCP(C)(C)=O)=O)C12CC2 C(=O)(C(F)CC(C)(C)NC(C1CCC2CC1CO2)=O)N(CCC1CC1)CC c1(OC)ccc(I)c(C(N2CC3CN(C(=O)C(=O)C(C)C)CC23)=O)c1 Cc1cc(C(=O)NCc2cc(C(=O)N(C3CCCC3CO)C)no2)c[nH]1 c1(C(=O)NCC23CC(NC(c4c(C)nn[nH]4)=O)(C2)C3)noc2cc(F)ccc12 c1(C(N(C)CC2N(C(CC=CC)=O)CCC2)=O)cccc2c1c(Br)nn2C c1(NC(C=CC(=O)OC(C)(C)C)=O)cc(C(=O)NC2CC(F)C2)ccc1Cl C1(C(=O)NCC23CC(OC)C2C3)CN(C(=O)OC(C)(C)C)C(C)(C)C1 c1(C(=O)NC(CCNC(C2(C(=O)OC)CC2C)=O)C)cncc2c(O)nccc12 C(=O)(CC(C(F)F)NC(c1ccsc1C#N)=O)NCP(C)(C)=O c1(C(=O)OCC)cnc(SC)[nH]c1=NCC(O)CNC(=O)C=Cc1ccccc1 C1(C(=O)NCc2nc(CNC(CCCOC(C)C)=O)sc2)CCCCC1F C1(C(=O)NCCCCC2CN(C(c3cncc(OC)c3)=O)C2)CCN2CCCC2C1 CC1(C)CCC(CNC(=O)CCC2NC(=O)NC2=O)(NC(=O)CC2CCOC2)CC1 C1(C(N(CC(C)CNC(=O)Cn2cccc2)C)=O)CCCOC1 c1(C(=O)NC(C2(O)CN(C(C3SCCS3)=O)C2)C)ncn(-c2ccccc2)n1 N1(C(C2(N(C)C(C3SCCS3)=O)CC2)=O)CCCC2CCCCC12 C12(CNC(c3cscc3C(F)F)=O)CCCC1N(C(c1sccc1F)=O)CCC2 c1(C2(C(=O)NCC3(NC(C(C)Cn4ccnc4)=O)CC3)CC2)c(F)cccc1F n1(CCCNC(C(c2ccc(F)cc2)C)CO)ncc(=O)c2ccccc12 C1(C(=O)NC2C3(CN(C(c4n(CCC)ccc4)=O)C3)CC2)CC2CCCC(C1)C2 C(C1=NOC2(CCC2)C1)NC(CC(CNC(C1CC(N(C)C)C1)=O)OC)=O CCC(C)(CO)C(=O)Nc1ccc(CCn2cc(C3(O)CSC3)nn2)cc1 c1(CNC(=O)Nc2c(C)nn(C3CCCCO3)c2C)c(C)c2ccccc2n1C CC1(C(=O)NC2C=CC(CNC(c3c[nH]c(C#N)c3)=O)C2)CCCc2ccccc21 C1(NC(CCC2CC(OC)C2)=O)CCN(C(c2cc(SC)ccc2C)=O)CC1O N1(C(C(C)(C)CC2CC2)=O)CC(NC(=O)CCC2CCCCCC2)C(C2CC2)C1 CON(C)C(=O)C(C)(C)CNC(=O)CCc1cccc(O)c1 c1(C(N2C(C)CC(CCNC(c3cnnn3C)=O)CC2)=O)c[nH]c2cccnc12 N1(C(c2c(C)nc(CCC)o2)=O)CCCOC(CNC(=O)COC2CCOC2)C1 C#CCC(O)C(=O)NCCNC(=O)C(c1ccc(F)cc1)Oc1ccc(C)cc1 c1(OCC)ccc(C(=O)N(C(C)CCNC(c2nccc(Cl)c2C)=O)C)cc1O c1(C(N2CC3(CC(NC(C45COCC4C5)=O)C3)C2)=O)cccc2cc[nH]c12 CC1CN(C(c2cnc(C3CC3)s2)=O)CCN1C(C1CC(C(=O)OC(C)(C)C)C1)=O c1(C(N2CC(C)C(CNC(c3ccccc3)=O)C2)=O)cccc(C#N)c1Br c1(C(=O)NCCN(CC(C)O)C(c2ccoc2Br)=O)c(F)cccc1F C1(C)(NC(CCCC)=O)CCCCC1C(=O)NCC(C)(C)COC C1(N(C(c2ncsc2Br)C(=O)NC)C)CCC2C3CCC(C3)C12 c1(C(=O)NCC=CCNC(C2(C#N)C(C)C2)=O)cc(F)cc2ccccc12 c1(C(N2C(C)C(NC(c3cc(CO)[nH]n3)=O)CCC2)=O)ccc(F)c2[nH]ccc12 C(=O)(CCC(C)(C)[N+](=O)[O-])NCC1C(CNC(C(c2ccc(F)c(Cl)c2)C)=O)C1 C(=O)(C(F)C(=O)N1CCCC(CNC(=O)C(F)(F)CO)C1)OCC C1(CNC(CCc2onc(C)n2)=O)CC(C)N(C(=O)C(C)c2ccco2)C1 C(=O)(C(CNC(=O)C=CC(F)(F)F)c1cc[nH]n1)N(CC(O)CF)CC C(=O)(CC(C(C)OC)NC(=O)Cc1ccoc1)NC1(C)CC(C(=O)OC)C1 N1(C(CCC(C)O)=O)CCC(C2CCN(C(c3cc(Cl)c[nH]3)=O)C2)CC1 Cc1ccc(Cl)cc1C(N1CC(NC(C2(O)CC2)=O)C(C)C1)=O c1(C(=O)NCC(N(C(c2nccc(C)c2F)=O)C)C2CC2)cnc2[nH]cnc2c1 C1(NC(C=C(C)C(F)F)=O)CN(C(C2SCCS2)=O)CC1C c1(C(N2CCC(NC(c3c(C)cc(F)s3)=O)C2)=O)ccc2nc(Br)nn2c1 c1(C(N2CCN(C(c3cnc(C)[nH]3)=O)CC2CCO)=O)cccc2c(C)coc12 c1(N2CC(O)CC(F)(F)C2)nc(N2CCC=C(Cl)C2)nc2c1CCCCCC2 C1(C(=O)NC(C=CC(=O)N(CC)CC2CC=CC2)C)CC(=O)N(OC)C1 C(=O)(CCC(F)(F)F)NC(C(C)(C)NC(C1N(CCC)CCCC1)=O)C c1(OCC)ccc(C)cc1C(N1CC(OC)C(NC(=O)CCC2CCCO2)C1)=O S(=O)(=O)(c1cccnc1N1CC2CCCCC2C1)N1C(C)C(C)(C)CC1 N1(CC(O)Cc2c(C)cc(C)cc2C)CCC2(CCC2c2cccs2)CC1 c1(CC)nc(=N)[nH]cc1C(=O)NCC1(C)CCN(C(c2ncc(F)cn2)=O)CC1 C(C(COC)C(=O)N1CCC(Cn2cc(-c3ccc(OC)cc3)nn2)C1)OC N1(C(C2C(C)C2C)=O)CC2(CCC2)CCC1CNC(=O)Cn1cnc(C(N)=O)c1 C(=O)(CC(O)C(C)(C)C)N1CC(CNc2ncn(C)c(=O)c2)OCCC1 CCCC(C(=O)NCc1nc(C(=O)NC2CCCSC2)c(C)o1)OC N1(C(C(CC#C)NC(=O)C(C)OCC)=O)CCC(C2CCC2)C1 N1(C(c2c(N)c(C)n(C)n2)=O)CCCC(C2CN(C(C3CCCC(O)C3)=O)C2)C1 c1(OC)cc(C)c(C(=O)NC(C)Cn2cc(CCc3ccccc3)nn2)cc1Cl C1(N(C(CC(C)N(C(C2CCN(CC)C2)=O)C)=O)C)CCCN(C)C1 CCC1=C(C(=O)NC2CN(C(c3ccc(OC)o3)=O)C3CCCC23)CCCO1 N1(C(C2(c3c(C)cno3)CC2)=O)CCCC2CN(C(c3ccnc(C)n3)=O)CC12 CC1NC(=O)C2=C1N(CCF)C(=O)NC2c1cc(Br)ccc1F c1(OC)ncc(C(N2CCCCC2CCNC(c2ccc(Cl)s2)=O)=O)cc1C CC1(C)CC(CNC(=O)C(C)(C)C)N(C(=O)CCC2NC(=O)NC2=O)C1 c1(CC(C)C)cccc(C(=O)N(C(C)CNC(=O)CC2CCCOCC2)C)c1 c1(-c2cn(CC3CN(C(c4cn(CC=C)nn4)=O)C3)nn2)c(F)cccc1F N1(C(CC2CCCC(C)C2)=O)CCCC12CCN(C(c1nonc1N)=O)CC2 CC1CCC(O)(C(=O)NCCCC(=O)NCCn2ccnn2)CC1 Cc1cc(C(=O)N(CCNC(=O)Cc2cc(C)no2)CC2CC2)nc(C)c1 Cc1nc2c(F)cccc2cc1C(N1CCC(NC(c2cc[nH]n2)=O)C1C)=O Cc1cc(C(=O)NC(C(N2CC(F)(CO)C2)=O)C2(C)CC2)nc(C)c1 Cc1ccccc1CC(C)C(=O)NC1CC1NC(=O)Cc1nc(C)c(C)s1 CCCCC(CCCC)NC(=O)CC1CN(C(=O)Cc2c[nH]nc2C)CC12CC2 Cc1ccccc1C(=O)NCC(CC(=O)NC1CC1(C)C(F)F)C1CCC1 C1(C(=O)NCCc2onc(C)n2)CN(C(=O)C(C)(C)F)CC1(F)F CCCCCCCC(C)CNC(C1CCC(OC)CC1)=O C1(C(N(CCN(C(=O)C2=CCC2)CC)CC)=O)OCCN(C)C1=O C1(NC(CN(C2CC2)CC)=O)CN(C(C)C(=O)NC(N)=O)CC2(CCC2)C1 CCC(C(=O)NC(c1cn(CC2CCC2)nn1)C)C(F)(F)F Cc1cc(OCC(=O)NCC2CN(C(C3(O)CCOC3)=O)CC23CC3)cc(C)c1 c1(N2CC(CNC(C(=O)NC(C)C)=O)OCC2)nc2cc(F)cc(F)c2s1 c1(C(=O)NC(CN(C(=O)CCS(C)=O)CC)C)cc(OC)c(Cl)cc1Cl C1(NC(c2[nH]nc3ncccc23)=O)CCCCN(CC2CN(CCOC)C2)CC1 CC1CCCCC1(CNC(=O)CSC(F)F)NC(=O)CCn1cnnn1 c1(N2CCC(C(=O)OCCCc3n(C)ncn3)C2)ccccc1F C1(C(NOCCCC=C)=O)CC2(CCN1C(=O)C=Cc1cscn1)CC2 C1(O)(C(=O)NC(CC=C)CNC(c2ncn(C)c2C)=O)CCCC(C)(C)C1 c1(C(N(C(C)C)CCN(C)C(C2CCSC2)=O)=O)cncc(F)c1Cl Cc1nn(CC(=O)NCC(F)CNC(C2CC2c2ccn(C)c2)=O)cc1Cl Cc1c(C(=O)NC2(CCCC(=O)NCc3ccc(O)nc3)CCC2)[nH]ccc1=O N1(C(C2CCCC2Cc2ccccc2)=O)Cc2ccc(Cl)c(F)c2C1 n1(C(C(=O)NC(CNC(CSCC#C)=O)(C)CO)C)nc(C)cc1C c1(C(=O)NCC2CCCC(NC(CCNC(C)=O)=O)C2)c(C)[nH]c2ncccc12 c1(C(=O)NC(CNC(CCC(CC)C)=O)C2CC2)cccc2c(C)ccnc12 C1(C(=O)NCc2c(C(=O)NCCCCOC)n[nH]c2)CC(C(C)C)=NO1 N1(C(CCCc2c(C)ccs2)=O)CCC(C)(CNC(=O)CC(C)c2ccco2)C1 C1(NC(c2c(C)onc2)=O)COC2(CNC(=O)C(C)OCC(F)(F)F)CC1C2 Cc1cc(NC(=O)C(O)CC2CCCCC2)ccc1NC(c1nc(C)c(C)[nH]1)=O C=CCCCCC(=O)N(C)CCOCCNC(C1CC1(CCOCC)CC)=O.CC CCC(C)CCCC(=O)N1CCN(C(=O)CN2C(=O)CCC2=O)CC1C(F)F c1(C(=O)NC2C(NC(C(C)NS(CC)(=O)=O)=O)C2)cc2c(C#N)cccc2[nH]1 C(=O)(C1CCCc2c1ncn2C)Nc1cc(-c2nc(CC)sc2)c(OC)cc1 C1(C(C)C)CCC(C(N2CC(C)(NC(=O)C=CCO)C2)=O)C(=O)N1 c1(CNC(C=C)CO)nnn(-c2ccccc2)c1C N1(C(CN(CCCCCC)C)=O)CCN(C(=O)C2=COCCO2)C(CF)C1 C(CC(C)(C)NC(=O)C(C1CC(C)(C)C1)O)NC(COCC(=C)C)=O C(=O)(C(C(C)(C)C)NC(N)=O)NCCCCN(C)C(c1coc(C(C)(C)C)n1)=O C(C)(C)(C#Cc1cn(CCC(F)(F)C(F)F)nn1)NC(C(C)NC(=O)NC)=O CCC(C)(C)C(=O)N1CCCC1CCC1CCN(C(=O)CS(C)(=O)=O)CC1 N1(C(=O)NC2CC(C)SC2)CCC(C)(N2CCOCC2)CC1 N1(C(c2ccn(CCCC)n2)=O)CCN(C(c2cccc(Cl)c2)=O)C(C)C1 C#Cc1ccc(C(N2CC(CCNC(=O)Cc3ccoc3)OC(C)C2)=O)cc1Cl C(=O)(C1CCc2ccccc21)N1CCC(CC(NOCCC(C)N=[N+]=[N-])=O)C1 Cc1sccc1C(=O)N(C)CC1(O)CN(C(=O)CC2CC(CF)C2)C1 CN1CCCCC1CC(N1CCC2CC12C(=O)NCCc1ccccn1)=O c1(NC(C(C2CCN(C(CC=C=C)=O)C2)F)=O)c(O)cccc1Cl N1(CC)C(=O)c2cccc(C(=O)NN(C)C(=O)NCCNS(=O)(=O)C(F)F)c2C1=O C1(C2CCCN(C(c3cccnc3S)=O)C2)(NC(CCCOCCOC)=O)CC1 Cc1ncc(C=CC(=O)NC2CCC(C)N(C(=O)C=Cc3cscn3)C2)c(O)n1 N1(C(CC2(OC)CC2)=O)CC(NC(c2ccnn2C2CC2)=O)C(n2cccn2)C1 c1(OC(C)(C)C)cnc(ONC(=O)NCC2C(NC(CCC)=O)COC2)c(C)c1 c1(C(N2CCOCC(CNC(C3CNC(=O)N3)=O)C2)=O)ccn2c1CCCC2 CC1CC(n2nc(COC(C)(C)C)nc2-c2ccc(Br)o2)CC(C)O1 C(CCCCC(=O)NCC(=O)N(C)O)NC(c1c(OC)cnnc1)=O c1(C(=O)NC23CN(C(C(F)OC)=O)C(C2)C3)occ2c1CCC2 C(=O)(C(C)CC(C)(C)C)Nc1c(C)cc(NC(C2(F)C(C)(C)C2(C)C)=O)cc1 N1(C(c2c(CC)onc2C)=O)CCC(F)(F)C(CNC(c2c(Br)nnn2C)=O)C1 C1(OC)CC2CCC1CC2C(=O)NCCCCCCNC(c1ccncc1Cl)=O CC1C(NC(c2cc(N)cc(F)c2)=O)CCCN1C(=O)CN(C)C(N)=O C(CCCC(CO)NC(=O)Cn1ncccc1=O)NC(C1(OC(C)=O)CC1)=O c1(CC(=O)NCC=CCNC(c2cc(Br)no2)=O)ccc(-n2cnnc2)cc1 c1(CN(C(C)Cn2cccn2)C)nn(C)cc1[N+](=O)[O-].c12cn(nn1)CCS2 CC1(C)NCCC1CC(=O)NCc1ccc(OC2CCOC2)cc1 N1(C(C2(C)CC2Br)=O)CCOC(c2cn(-c3ccccc3N(C)C)nn2)C1 Cc1ccc(N2CCCC2)c(C(N2CC(N(C)C(=O)NC3CCS3(=O)=O)C2)=O)c1 c1(C(C)C)ccc(CCC(=O)NCCC(C)NC(=O)Cc2cnccn2)cc1 N1(C(C(CSC)C)=O)CCC(C)(CNC(c2cc(Cl)ns2)=O)C1 C1(C)(C(=O)NCCC2(NC(CC3N(CC)CCC3)=O)CCCC2)CCC(=O)N1 C1(C#N)(C(N(CCN(C(C=C(C)CCc2ccccc2)=O)C)C)=O)CC1(C)C N1(C(=O)OC(C)(C)C)CCCC(C)(Cn2cc(C(=O)Nc3ccc(O)nc3)nn2)C1 C1(NC(c2cc(C)sn2)=O)CCS(=O)(=O)C12CN(C(=O)C(C)NC(N)=O)C2 c1(C(N(C2CCC(NC(c3nc(C)sc3)=O)CC2)C)=O)csc(S(N)(=O)=O)c1 CCCCC(O)C(=O)N1CCC(C)(C(=O)Nc2cc(OC)cc(C3CC3)c2)CC1 C(C(=O)N1CCC(C(=O)NCCC(O)C2CCC2)O1)OC(CC)(C)C c1(CNC(C2N(C(C(C)C)=O)CCC2)=O)nnccc1C(=O)O c1(SCC(=O)N(CCCNC(=O)C(c2cccs2)C)CC)ncccn1 CC(C)C(C(=O)N1CC(Cc2ccoc2)C1)NC(=O)CC1(O)CCOCC1 CCC(F)(F)C(C)(C)C(=O)N1CCN(C(=O)CC2CC2(C)C)C2(CCC2)C1 c1(CC(N2CCCCC2CC(C)O)C(=O)NC(C)C)ccc([Si](C)(C)C)cc1 C1(N(C(C(C2CN(C(CC(C)F)=O)C2)OC)=O)C2CC2)CCCCC1(C)C C1(N(C(CSCCN(CC)CC)=O)C)CCCN(C(c2ccnc(Cl)c2)=O)CC1 C1(NC(c2oc(CC)c(C)c2)=O)CN(C(=O)CC2CC23CC3)C(C)(C)C1 C=CCCCC=O.c1(CNc2ncc(CC)cn2)ccc(C(=O)NCC)nc1 C1(NC(C)Cc2ccc(N)cc2)CCCN(CC(F)(F)F)C1=O C=CCC(CNC(C1(CC=C)CCCN1C(=O)C(C)C1(O)CCC1)=O)CC(C)C c1(C(=O)NC2CCN(C(C3(C)CCCNC3=O)=O)C2)c(Cl)ccc2c[nH]nc12 N1(C(C(C)Sc2ccc(C)cc2)=O)CC2CC1CN(C(=O)C=CS(C)=O)C2 Cc1n[nH]c(C)c1C(C1C2COCC12)=O.C12CCCN(C1)C2.C1(C(=O)O)CCCCCC1 c1(C(=O)NCC2CC(C)N(C(=O)Cn3cnc(=N)[nH]3)C2)cc(F)ccc1C1CC1 c1(C(=O)NCc2scc(C(=O)NC(C(C)C)CO)n2)onc2ccccc12 C1(O)(CCNC(=O)C2CC2)CCN(CCCSC(CC)C)C1 N1(C(c2cccc(Cl)c2OC)C(=O)NCCCOC)CCC2(CNC(=O)C2)C1 N1(C(c2c(C(C)NC(C3CS(=O)(=O)C3)=O)noc2)=O)CCCC1(C)C(C)(C)C c1(CC)cc(F)c(C(N2CCCN(C(C3CCSC3)=O)CCC2)=O)cc1F c1(C(=O)OC2CN(Cc3cn(C)nc3OCC(F)F)C2)cnc2[nH]cnc2c1 c1(CCNC2C(SC)CCCC2)nnc2n1CCOC2 CC1CCC(C)N(C(=O)CCc2cn(-c3cccc(C(=O)O)c3)nn2)C1 C(CCCN=C(NCc1c(F)cccc1Cl)NC1CC1)c1cccc([N+](=O)[O-])c1 CC(N=c1cc(C2CC2)nc(Cl)[nH]1)C1CN(C(=O)CC2CC2)CCO1 c1(CNC(N(C(C2CCCCC2)C)C)=O)sc(Cl)cc1Cl C1(CC)CN2CC1C2=O.c1(NC(=O)CCc2nccs2)cnc(OC)nc1 c1(C(N2CC(C)N(C(c3ccc(=O)oc3)=O)CCC2)=O)c2c(nn1C)CCCC2 C1(CNC(C2(C#C)CC2)=O)CC2(CC(NC(c3cc[n+]([O-])cc3)=O)C2)C1 CN1CCN(C)C(C(=O)NCCCCCCN(C)C(c2cnn(C)c(=O)c2)=O)C1 c1(C(COC)NC(=O)CCCn2cc(C3CCC=CO3)nn2)cccc(C)n1 c1(C(N2CC(SCC)C(NC(C3CC3C(F)F)=O)C2)=O)cnc(C2CC2)nc1O N1(C(c2cnc(C)[nH]2)=O)CCC2(NC(C3CCOCC3)=O)CCCC12 c1(C(N(C(CC)C)CC)=O)cc(CNC(c2ccc(C)cc2)=O)nn1C C1(OC)CN(C)C(C)(C(=O)NCCCN(C)C(c2ccc(Cl)c(F)c2)=O)C1 C1(C(N(CCN(C(=O)C(C)C2CCCC2)CC)CC)=O)CCNC1=O CC(C)C(C#N)C(=O)NCC1CCC(C(=O)NCCc2cnco2)C1 C1(NC(=O)COCCOCCO)CN(C(C2(C)CCCNC2=O)=O)CC(C)(C)C1 Cc1cc(C(=O)Nc2ccnn2C(C)C(C)C)cc(F)c1 C(CN=c1[nH]c2c(c(=NCC3CCCC3C(C)(C)C)[nH]1)SCC2)N(C(C)C)CC CCC(CC1CCCCC1)C(=O)NC1CCC(NC(C2CC(F)(F)CS2)=O)C1 C=C(C)C1OCCC1C(=O)NC(C)(CNC(=O)CC(C1CC1)C1CC1)CO c1(NC(C2(F)CCN(c3ncccn3)CC2)=O)ccc(Br)c(F)c1 N(C1CC(C)c2ccccc21)C(c1cc2ccc(C)cc2s1)=O N1(C(C(C(C)(C)C)SC)=O)CCN(C(=O)CC2CC3(CC3)C2)C2CCC12 C1(C)(C(=O)NC(C(=O)NCC2OCCN(CC)C2)C(C)C)CC2CCC1C2 CC(C)CN=C(NC1CC1CF)N1CCCC(C(C)(C)C)C1 c1(C(N2C(C)C(NC(c3cc(Cl)sc3Cl)=O)CC2)=O)c[nH]c2cccnc12 c1(C(=O)NC2CCN(C(C(=O)NCC)=O)CC2O)noc2c1COCC2 C#Cc1ccc(CC(N2CCC(C=C)(C(=O)NC3CCCC3(C)CO)C2)=O)cc1 c1(CN=c2ccc(-c3ccc(C)cc3Cl)c[nH]2)ccc(C)c2ccccc12 c1(C(C(=O)OCCC(C(=O)OC(C)(C)C)F)(F)F)ccc(Cl)cc1Cl CCC(C)(C)C(=O)N1CCC(C(F)C(=O)NCCC(N)=O)C1 c1(C(=O)NC(CC=C)CNC(=O)CN2CCSCC2)ccc(C2(OC)CC2)cc1 Cc1ccncc1CC(=O)NC1CCCCC1CNC(=O)CN1CCCS1(=O)=O C1(NC(CCCCC)=O)CCC(C)(NC(=O)CN(C)C(C)C)CC1 CC1CC(N=c2[nH]c(N(C)Cc3nc[nH]n3)nc(=N)[nH]2)CC(C)(C)C1 C1C(C)(C)C(=O)N1.c1(CC(=O)N(C2CN(C(C)=O)C2)CCO)nnc(C)s1 N1(C(C(C(C)C)NC(=O)CCNC=O)=O)CCC(O)(CO)CC1 N1(C(=O)OC(C)(C)C)CC2(CC(NC(=O)C(=O)NC3COCCC3CO)C2)C1 C(=O)(CCCC(N)=O)N(CCC(C)NC(=O)COCc1cccc(Cl)c1)CC S(=O)(=O)(c1ccc(NCC=C(C)CN2CC(OC)C2)c(Br)c1)N1CCC(CCC)C1 c1(C(=O)NC(CNC(c2cncc(F)c2)=O)C2CCC2)ccc(Br)cc1[N+](=O)[O-] CC(C)CC(C(=O)NCC1(F)CC(CNC(c2ccc(F)cc2O)=O)C1)C(C)C C1(NC(C=CCN(C)C(c2cc(Cl)n(C)n2)=O)=O)CCN(C)CC1C#N N1(C(c2ccc(=N)[nH]n2)=O)CCC(C(=O)NCC2CC23CCCCC3)C12CC2 N1(C(C=CCCC)=O)CCN(C(C2CC3CCC2C3)=O)C(c2ccc(OC)cc2)C1 CCCC(CC(C)C)C(=O)NCCN1CCCN(C(C2CCC(CC)O2)=O)CC1 C1(NC(CC2C(NC(C(C)OCCN(C)C)=O)CC2O)=O)CCCCCC1 C12(CCC(C#N)(c3ccccn3)CC1)N(C)C2.C1(C(=O)O)CC(CCF)C1 N1(C(c2cnc(C)s2)=O)CCN(C(=O)C(C)(C)c2ccno2)CC(C)(C)C1 C1(NC(C(CCSC)O)=O)CN(C(=O)CSc2ccc(F)c(F)c2)C(C)(C)C1 N1(C(=O)OC(C)(C)C)CCC(NCC2CCCC(O)C2)CC1C1CCCC1 N1(C(CCc2scc(C)n2)=O)CCN(C(c2ccc(CC3CC3)s2)=O)CC1CO CCCCCCC(C)C(=O)N1CCOCC(CNC(c2nc(CC)no2)=O)C1 c1(C(=O)NCC2N(C(CCC=C)=O)CC=C2)nc(C(C)C)c(C)s1 CON1CC(C(N2CCC(CCNC(c3cncc(F)c3Cl)=O)CC2)=O)CC1=O C(=O)(CS(=O)(=O)N1CCCCC1)N(CCC(C)NC(=O)Cc1ccc(O)cn1)C N1(C(CCn2c(C)ncc2)=O)CCCN(CC(=O)NC(C)(C)C)CC1 C1(CCCNC(c2cn(CC3CC(F)(F)CO3)nn2)=O)CC2CCC1C2 C(=O)(C(C)(C)C(F)(F)F)NC1C2CN(C(CCc3nc(C)sc3)=O)C1C2 C1(C(=O)NCC(=O)NCC(N2CCC(CCOC)CC2)=O)CC(=O)NC(=O)C1 C1(CC(N2C(CN(C(Cc3nnc(C)o3)=O)C)CCC2)=O)CCC(=O)NC1 C1(C(N2CC(CC(C)NC(=O)C(F)(F)C(F)F)C2)=O)C2CC3CC(C2)CC1C3 N1(C(C(N2CCC(C)C2)=O)=O)CCC2CN(C(c3ncc[nH]c3=O)=O)CC2CC1 c1(C(N2CC(O)CC(NC(C3CCC(CC)CC3)=O)C2)=O)cc[nH]c2nccc1-2 c1(-c2cnc(C)s2)ccc2oc(C(=O)N(c3nnc(C)n3C)CCO)cc2c1 N1(C(c2nccc(C#C)c2)=O)CC2CCCC(C1)N(C(=O)CCC(=C)Cl)C2 C(CCCCCCC(=O)Nc1ccccc1)N1C(C)(C)C(c2ccccc2F)CC1 c1(C(=O)NCc2cc(COC)c(Cl)cc2)cc([N+](=O)[O-])c(C)c([N+](=O)[O-])c1 c1(NC(C=CCCC(C)(C)NC(c2cccnc2)=O)=O)cnc(O)c(F)c1 C1(OCC)CC2CN(C(c3csc(C)c3)C(=O)Nc3cc(F)ccc3F)CC12 N1(C(C2CC(OC)C2)=O)CC(F)(F)CC1C(N1CC2C(C1)C2(C)C)=O c1(C2C(C(=O)NC3C(CNC(CCS(C)(=O)=O)=O)C3)C2)ccc([N+](=O)[O-])cc1 N1(Cc2nc(C)[nH]n2)CCN(C(c2cc(F)ccc2Br)=O)CC1C(C)C CC1CN(C(=O)CCc2ccccn2)CC1CNC(=O)C(F)C1CCOC1 c1(C(=O)NCC(CC(C)C)(C)NC(C2CCCSC2)=O)cccc(P(C)(C)=O)c1 O=C(C1=NOCC1)NCCCN(C(c1cc(Cl)cnn1)=O)CC1CCCC1 C1(CCC(N2C(CNC(C(C)NS(CC)(=O)=O)=O)CC2)=O)CCCCO1 N(C1CCc2cccnc21)C(C1(CNC(CCC(C)OC)=O)CC1)=O N1(C(c2cccc(=O)o2)=O)CCC2CN(C(c3cnc[nH]3)=O)C2C1 C1(CNC(COCCCCCC)=O)CC2(CC2)CN1C(=O)COCC(C)C CCC(C)(Br)C(=O)N=S1(=O)CCC(CNC(=O)OCC)CC1.C(C)(C)(C)O CC1CCC(C)(C(N2CC(CNc3cc4nncn4cn3)(OC)C2)=O)C1(C)C N1(C(C(N)CC=Cc2cccs2)=O)CCOc2cccc(Cl)c2C1 Cc1nc(C(C2CC2c2ccccc2F)NC(=O)CC2CCCCN2C)c(C)s1 CC1(C)C(CC(N2CCC(C(N3CC(CO)C(O)C3)=O)C2)=O)C1(C)C c1(CC)c(C(=O)NCc2cn(CC(=O)N)nn2)nnn1C.N1(C)CCC(C)C1 C1(NC(c2ccccc2N2CCCC2)=O)CCCN(Cc2cncc(F)c2)C1 C1(C(N(C2CCCN(C(c3ccc(C(F)F)cn3)=O)C2)CC)=O)CCCN1C=O C12(C(=O)NCC3C(C=C)OCC3)CC(NC(=O)OC(C)(C)C)(C1)C(C)(C)O2 c1(C(N2CC(NC(Cc3ccc(C)cc3)=O)C(C)C2)=O)cccc2c1COC2 O=C(CCC1CCc2ccccc21)NC1CC(NC(C2CC23CCC3)=O)C1 N1(CC(N2Cc3c(nc(C)s3)C2)=O)C(=O)NC2(CC2(C)C)C1=O C(CCC(=O)NCC1CC1C(=O)NC(c1cnco1)C)OC(C)=O C(=O)(C1CCOc2ccccc21)N(C1CCN(c2ncnc3n[nH]c(Br)c23)C1)C C(=O)(C1=NOC2(CCN(Cc3nc4ccc(Br)cc4s3)C2)C1)NCC(=O)N(C)C c1(C(C)(C)C(=O)N2CC(NC(C3CCCCC3F)=O)C2)ccc([N+](=O)[O-])cc1F N1(C(c2c(C)cc(C)s2)=O)CC(C)OC2(CCN(C(=O)CC3CSC3)CC2)C1 N(C(=NCCC(C)C)NCc1csc(C(C)(C)C)n1)C1CC(OCC)C12CCC2 C1(CNC(CC2N(C)CCCC2)=O)CC2(CC2)CN1C(=O)Cn1ncnn1 c1(N2CC3C(C)(C)C(C3)C2)nc2c(c(=NCCc3ccc(Cl)s3)[nH]1)CCC2 N1(C(C(=O)NCC)=O)CC(C)CN(C(=O)C=Cc2cnn(C)c2)CC1C CC(C)(C#N)CCC(C)(c1nnnn1Cc1cccs1)NC1(C)CCS(=O)(=O)C1 C12(NC(c3c(SC)cccn3)=O)CCCC1CN(C(=O)C=Cc1cccs1)C2 Cc1cc(NC(=O)C(C)C2CCCC2)ccc1NC(=O)C=C1CCN(C)C1 CC1(C)OC(C(N2CCC2CNC(c2c(Cl)sc3nnsc23)=O)=O)C(C)(C)O1 C(=O)(C1=CC2CCCCC12)NCC(C)NC(=O)COc1ccc(F)c(F)c1 C=CC(C)C(C)C(=O)NC(C1CN(C(=O)CCCCCOC)C1)C Cc1ccccc1C(=O)NC(C)CCN(C(=O)Cc1ccc(CO)cc1)C C(CS(=O)(=O)CC(=O)NCC1(NC(=O)C2=CCC(C)CC2)CCC1)OC C1(C(=O)NC2CCN3CCCC23)CC2CN(C(C3CCOC3)=O)CC2C1 C1(CNC(C2CCN(C(=O)NCC)CC2)=O)CC2CCC(C1)N2C(C)=O C(=O)(CC(COC)NC(=O)CCC1CCCCC1)NCC(=O)NC N1(C(c2ccc(COC)o2)=O)C(C(=O)NOCC(O)CCC2CC2)CCC12CC2 c1(C(N2C(C)CC(NC(C3(Cl)CC3)=O)CC2)=O)n[nH]c2c1CC(F)(F)CC2 c1(CNC(=O)N(c2ocnc2Br)C2CC2)ccc(OCc2ccccc2)cc1 C#Cc1cn(C)nc1C(=O)N(C1CN(C(c2cccn2C2CC2)=O)CC1O)C c1(N(c2ccccc2)C(N2CCC(N(C)C)CC2)=O)cnc(C2CCC2)nc1O c1(CC(=O)NCC2CCCN(C(C=C(CC)C)=O)CC2)ccc(F)cc1[N+](=O)[O-] N1(C(C(C)(C)OC)=O)CCN(C(=O)C(C)CC2CCCCC2)C(CO)C1 c1(C(=O)NCC(C#C)CC2CC2)nc(CNC(=O)CN2CCCC2CC)oc1C c1(C(N2CCC(N(C)C(c3cc(C(F)(F)F)cs3)=O)C2)=O)cc(O)ncn1 C12(C(N3CCC(C)CC3)=O)COCC1CN(C(c1n[nH]c3c1CCCC3)=O)C2 C1(NC(CCc2ccc(C)s2)=O)CCN(C(=O)Cc2cccnc2)CCC1CO N1(C(=O)NCc2ccncc2Cl)CCOCC12CCS(=O)(=O)C2 CCC(C)C(C(=O)Nc1ccc(F)nc1)N(C)C(c1n[nH]cc1Cl)=O N1(CCC#C)CCC(C(=O)NCC2CC2NC(C2COC(=O)C2)=O)CC1 N1(C(C2(N(C)C)CCCC2)=O)CCCC(CNC(C2(Cl)CC23CCC3)=O)C1 c1(-c2nnc(Cn3nc(C)c(Br)c3)o2)cc(Cl)cc(Cl)c1 O=C(NNC(=O)CSCc1ccccc1)c1cnc(C2CCCO2)s1 C1(n2cc(CC=C)nn2)CC2CCC1(NC(=O)C(F)Cl)C2 C(C(CC1CCCC1)C(=O)NCC12CCCCC1C2)NC(Cn1c(C)ncc1)=O N1(C(CSC)=O)CC(CO)C2(C1)CN(C(=O)C(C)N(C)C)C2.C(C(C)C)O c1(C(N(CC(C)NC(=O)C(F)=C2CCC2)C)=O)ncncc1C#N N1(C(CCSCCC)=O)CCOC(C(C)NC(C2CC(O)CN2C)=O)C1 C(C1CCN(C(C2(F)C(C)(C)C2(C)C)=O)CC1)=CC(=O)N(C)Cc1cn[nH]c1 C(c1ccc(F)cc1Cl)=CC(=O)NCC1CC(C(=O)Nc2cncc(C)c2)C1 CCCCC(C)CCC(=O)NC1CCN(C(c2ncc(CC)cn2)=O)CC1O CCC(CC(=O)NCC(CC(C)C)C(=O)N1CCCC1CNC(C)=O)C(C)(C)C Cn1nc2ccccc2c1C(=O)NC1CC2CCCC2C1 C1(C(=O)NC2C(NC(c3c(C)cc(C)s3)=O)CCC2)CC(C2CCC2)C1 c1(C(N2CCC(N(C(C3CC4CCC4C3)=O)CC)C2)=O)cccc(OC)c1F C(=O)(C#CC1CCCCC1)N1CC(CN(C)C(C2CC2Br)=O)C1 Cc1ccc(=O)n(CC(=O)NC2CC(C)N(C(=O)C=Cc3cn[nH]c3)C2)n1 N1(C(c2c(CNC(c3ccc(O)cc3)=O)cco2)=O)CCC(F)(F)C(F)C1 C1(CNC(=O)C=CBr)CCC(NC(C2CCN(CC3CC3)CC2)=O)CC1 c1(C(=O)NCC(C)NC(C(C=C)O)=O)cccc(OCCF)c1 CC1(O)CCCC1NC(=O)C(O)C1CN(C(c2cc(O)ncn2)=O)C1 c1(CC)cc(F)ccc1C(N1CCSCC1C(=O)NCC1C=CCC1)=O c12cccn(c1=O)CC(=O)N2.N1(C(CCC2C(C)C2)=O)CC(C)(C)OC1=O N1(C(c2cnn(CC(F)(F)F)c2)=O)CCC2(CCCC(CO)O2)CC1 CC1CC(NC(c2ncsc2Br)=O)CCN1C(c1cc(Cl)no1)=O N(C1CCCn2nccc21)C(C1(OC)CCN(C(=O)CN2CC(C)(C)C2)C1)=O c1(CN2CC3(C(C(N4CCC(O)C4)=O)C3)C2)cc(O)cc(O)c1 C(C(=O)N(C1CCCC1)C)(C(C)C)SC.c12cn(nn1)CCC(=O)N2 C(=O)(C1=NOCC1)NCc1ccc(C(=O)NCCN(C(CC)C)C)o1 CC1(C(=O)NC(C)(C)CC2CCOC2)CN(C(C2CCCS2)=O)C1 c1(NC(C23C(CN(c4nccc(SC)n4)C2)C3)=O)ccc(C)cc1Br N1(CC(C)C)N=C(C(=O)N2CCC(NC(C34CCCC3OCC4)=O)C2)CCC1=O c1(C(=O)NCC2(F)CN(C(C(CC)SC)=O)C2)ccccc1S(=O)C(F)(F)F N1(C(=O)CNS(=O)(=O)C2CC2)CCC2(CCCN(C(c3ccon3)=O)C2)C1 C(C(C)(C)C#CC(=O)NC1CNC(=O)C1(C)C)NC(c1c(C)[nH]c(C#N)c1)=O c1(C(=O)NCC(c2ccccc2C)NC(C(C)=C2CCC2)=O)cc(Cl)cn1C N1(C(c2c(C)ocn2)=O)CCN(C(c2nn(C)cc2Br)=O)CC1CCO C1(C(=O)NCCCC(=C)Cl)CCN(C(C2CSC2)=O)C12CCC2 O=C(C#Cc1ccccc1)NCC1C2CN(Cc3c[nH]c4ncccc34)CC12 CC1CN(C(=O)CNC(=O)C2CC2)c2cc(C(F)(F)F)ccc2O1 N1(C(CNC(=O)NC)=O)CC(C)(C(=O)NCC2CC2C)C1 C1(N(C2CCC2)C(c2cnn(CC(F)F)c2)=O)C2CC3C(C2)C13.C1CN1 C1(C(=O)NCC(N2CCCC2)C)C=CCCN1C(=O)CN1CCNC1=O Cc1c(C(N2CC3CCC(C2)N3C(c2ccc(O)c(Cl)c2)=O)=O)sc2nccn12 C1(C)(OC)CN(CC(=O)NC2CC2CNC(C2CC3(CC3)C2)=O)C1 Cc1ccn2ncc(C(=O)NCC3CCCC(C)(C)C3)c2c1 c1(C(=O)NCC23CN(C(C(C)(F)F)=O)C(CC2)C3)cncc2[nH]ccc12 c1(NC(C(C(C)SC)O)=O)ccc(NC(=O)CCC2CCCCC2)c(C)c1 C(=O)(C1=CCCCO1)NCCC(C)(C)NC(=O)CCC1CCC1 c1(C(=O)NCC(C)OC)occc1CNC(c1cc[nH]c1)=O N1(C(c2ccc(C#N)cn2)=O)CC2CCC(CO)(C2)C1.C12CCCCC1NC2=O N1(C(CN(C)C2CC2)=O)CCC2(C1)CN(C(=O)CN(C)S(=O)(=O)N(C)C)CCO2 c1(C(N(CCC(=O)N(CC(C2CCC2)OC)C)C)=O)cc(O)ncc1F Cc1cc(C)c(C(=O)N(C2CCCN2c2nccc(C(CN(C)C)(C)C)n2)C)o1 c1(C(CNC(C)CC2CCC2)C)ccccc1 O=C1Cc2cc(S(=O)(=O)NC3CCC(C(=O)Nc4ccncn4)C3)ccc2N1 C1(CC(=O)NCC2CCCCN2C(c2ccc(CO)o2)=O)CC2(CCCC2)CO1 N1(C(CC(=O)NC)=O)CCC(CNC(=O)Cc2csc(C(F)(F)F)n2)(OC)C1 c1(SC)cc(C)c(C(N2CCN(CCN(C(=O)CC3COCCO3)C)CC2)=O)s1 n1(CC=C)ccnc1C(N1CC(O)(C2CCCN2C(=O)COCC)C1)=O C1(CNC(CC)=O)COC(C)(C)CN1C(=O)Cc1cn(Cc2ccno2)nn1 CC1CN(C(c2n[nH]cc2F)=O)CC1NC(c1ccc(OC2CCC2)o1)=O c1(C(N(C2CCCN(C(c3cnc(O)o3)=O)CC2)C)=O)ccc(O)c(Cl)n1 N#CC1(C(=O)NC2C=CC(CC(=O)NCCc3cnco3)C2)CC2CC2C1 c1(C(N(C2C(N(C(CCC=C)=O)C)CCCC2)C)=O)ccc(Br)c(C)c1F C(=O)(C1=CC2(CCOC2)C1)N(CCCCN(C(c1cc(C)nnc1)=O)C)C C(C(=O)N1CC(C)(O)C1)(C(C)O)NC(C=CC(CC)C)=O C1(c2ccccc2)(NC(=O)NCC(C(C)O)C)CCOCC1 C(=O)(C1=CCC2CCC1N2C(C1CNC(=O)N1)=O)N1CC(C(=O)OC)(CC)C1 c1(NC(=O)CC(Cc2cccs2)NCc2cccc(F)n2)cnc(Br)nc1 c1(C(=O)NC2C=CCN(C(C=COCC)=O)C2)ccc(S2(=O)=NCCC2)cc1 N1(C(C(CC)OC2CCCCC2)=O)CCC(C2N(C(=O)C3CC3)CC2(C)C)CC1 N1(CC(C)C)N=C(C(=O)N2CC(F)(F)CC2(C)CNC(C2CC2F)=O)CCC1=O N1(C(C(CC=C)(C)O)=O)Cc2[nH]nc(C(=O)N(C)CCN3CCCCC3)c2C1 c1(OC)cc2c(O)ncnc2cc1C(N1CCCC(c2cnc[nH]2)C1)=O N1(C(C2(F)CCCC2)=O)CC2(CCCN(C(C3CCC3c3nc[nH]n3)=O)C2)C1 c1(C(N2CCN(C(c3nc(C(C)C)sc3)=O)CC2)=O)cc2ccccc2[nH]1 C12(C(N(C)CC3CCN(C(C(CCSC)NC=O)=O)C3)=O)CCC(CC1)C(C)O2 C12(C(=O)NC3CN(C(C)=O)C3)COCC1CN(C(=O)Cn1ccc(C)c1)C2 N1(C(CCC#CC)=O)CCC2CN(C(=O)CC(O)CCC)CC2C1 C(=O)(CC(C)(O)C(F)(F)F)NC1C(C)CCN(C(c2csc(C)c2N)=O)C1 c1(C(F)(F)F)ccc(CN2CC3CC2CN3)cc1F c1(C(C)(C)C)cc(C(=O)NCCCn2cc(CSC3CC3C3CC3)nn2)on1 n1(CCC(=O)Nc2ccc(Oc3ccccc3Br)cc2)cnc(Cl)c1Cl c1(OC)c(Br)cc(NCCNC(=O)C(N)CCOC)cc1Br CC1(C)C(NC=O)CC1.C1(NC(C2(N3CCCC3)CCC2)=O)CC(F)(F)C1.N Cc1cccc(C(=O)NCC2CC(F)(CNC(=O)CC3(C)CCCO3)C2)c1F c1(C(N(CC(CN(C(=O)CN2CCOCC2)C)O)C)=O)cc2ccnc(Cl)c2[nH]1 C1(C(=O)NCC2(O)CC(NC(C(=Cc3cnc[nH]3)C)=O)C2)CC2(CCOCC2)C1 C1(NC(C2N(C)C(=O)CC2)=O)CC2CN(C(C3CCC(=O)NC3)=O)CC2C1 C(C)(C(CC(=O)NCC1(C)CC(C)(C)C1)NC(=O)C=CC1CCCN1C)OC c1(C(=O)NCCC2CCCN(C(CCCOC(C)=O)=O)C2)nc(O)nc(O)c1F c1(C(=O)NCC(CCNC(C23CCC(OC)C2C3)=O)OC)csc2nccn12 C(=O)(C1SCc2cccnc21)N(CC(C)(C)O)CC(C)(C)O Cc1ccc(I)cc1C(=O)NC1CCC(C(=O)NCc2ccccc2Cl)C1 C(=O)(C(F)CCC(C)C)NC1C(NC(c2cncc(C(C)=O)c2)=O)COC1 C1(NC(C2(COC)CC2)=O)C2CCCN(C(=O)CN3CC4C=CC3C4)C2C1(C)C c1(OC)cc(CC(N2CCN(CCNC(=O)CCn3cncn3)CC2)=O)ccn1 c1(C(=O)NCC23C(CN(C(CC(=C)C)=O)C2)C3)c(C(F)(F)F)nc2ccccn12 Cc1c(F)ccc(Cl)c1C(=O)NC1CCCN(C(c2cn(C)nc2Cl)=O)CCC1 C(=O)(C1=CCCO1)NC(C(C)C)CNC(=O)C(c1cncn1C)O N1(C(C2(C)CS(=O)(=O)C2)=O)CCC2(NC(c3ccc(C(N)=O)cc3)=O)CC2C1 C1(CC(=O)NCCCCN(C(=O)CNc2nccs2)C)C=CS(=O)(=O)C1 C#CC1(C(=O)NC2CC(C)CC(C)C2)CCN(C(C2CC2(F)F)=O)C1 C(C(=O)NC(c1c[nH]ccc1=O)C)(C(C)CC)NC(c1ccn(COC)n1)=O CC(CC(C)NC(c1cc(CF)on1)=O)NC(=O)CSc1cn[nH]c1 c1(C(c2cn(CC(C(C)(C)C)CO)nn2)O)ccc(F)c(F)c1F C1(CNC(CSC)=O)CC2(CCOCC2)CN1C(c1cccc2nccnc12)=O c1(C(=O)NC2C(CNC(C3C(CCC)C3)=O)CCC2)ccn(CC)c1C c1(C(c2n(C)nnn2)NCc2cc3ccccc3o2)ccc(F)c(Br)c1F C1(CC(=O)NC(C=C)C)CC(NC(=O)C(F)n2ccnc2)C1 c1(CC)cccc(C(=O)NC2CCCC2NC(C2CCCN2C(C)C)=O)c1O N#Cc1ccc(SCC(N2CCC(NC(=O)COC3CCC3)C2)=O)c(F)c1 c1(C(C(=O)NCCn2ccnc2)N(CCCF)CC)ccnn1COC C(C(F)C(=O)NCCC(=O)NCCN(CC(C)(C)C)C)C1CN(C(COC)=O)C1 C(C)(C(=O)N=c1ccn(C2CCC2)[nH]1)C1CCCN(C(Cc2c(C)ccs2)=O)C1 c1(SCC(N2C(c3cn(-c4c(C)ccc(F)c4)nn3)CCC2)=O)ccc(Cl)cc1F C(C(C)C)(C(O)C(=O)NCC1CN(C(=O)CC2(C)CC2)CC12CCC2)OC C1(C(=O)NCC(C)NC(=O)C(C)(C)c2cnsc2)Cc2cccc(F)c2O1 CCC(CNC(=O)COCc1cccc(C)c1)(CC)NC(C1CC2CCCC12)=O C12(C(=O)NCCN(C(C3CC4CCCCC34)=O)CC)CC1COC2(C)C c1(SC)ccccc1CC(N1CCCC1CCCNC(C1C2CCOCC12)=O)=O c1(COC)nc(C)c(C(=O)NCC2CCN2C(=O)CCc2ccc(F)cc2)s1 Cc1cccc2[nH]c(C(=O)NCCCCCCNC(C3(C)CCCC3C)=O)cc12 Cc1nc(CC(=O)NC(CNC(c2ccc(C(N)=O)o2)=O)CO)c(Cl)s1 c1(C(=O)NCC(N(C(=O)C=CCO)C)C2CC2)nc2c(s1)COCC2 C1(C#N)(C(N(CCCOCCN(C(CC2CC(=C)C2)=O)C)C)=O)CCCC(=O)C1 C1(CN(C(c2n(CC)c(O)nc2)=O)C)CCCN(C(C2CC3CC3C2)=O)C1 CC1CC(C)(C(N2CCCC(CNC(c3cn(C4CC4)nn3)=O)CC2)=O)CCO1 CC1(C)C(NC(C2CCN(CC(F)F)CC2)=O)CCN1C(C1CCS(=O)(=O)C1)=O C1(C(=O)NC(C2N(C(c3c(CC)ncs3)=O)CCC2)C)CN(S(N)(=O)=O)C1 C1(C(=O)OCC)CCC2(CC1)CC(C(=O)N(CC)Cc1c[nH]nc1C1=CCC1)C2 CCCC(C(=O)N1CCOC(CNC(C2CCN(C3COC3)C2)=O)C1)NC(N)=O c1(CSCC(=O)NCCOC)ccc2cc(C)[nH]c2c1 C1(C2CCN(C(c3c[nH]c(C#N)c3)=O)C2)(NC(CN(C2CCSC2)C)=O)CC1 c1(OC(C)C)c(C(=O)NC(CNC(=O)C=CS(C)=O)C(C)(C)C)cccc1N C(=O)(C(C)CCC(C)(C)C)N(CCC(N1CC(C)C1(C)C)=O)CC#C S(=O)(=O)(c1c[nH]c(C(N2CC(NC(c3cc(SC)oc3C)=O)C3CC23)=O)c1)NC CN1CC(O)CCC1C(N1CCCC(C(=O)NCC2CC23CC3)C1)=O C(c1ccc2c(c1)OCO2)=CC(=O)NCC(CNC(C#CC1(C)CC1)=O)(C)O N1(C(=O)CC2C=CCC2)CC(C2CC2)(C(=O)NOCCCCC2CC2)C1 c1(OCC(N2CCC(C)OCC2)=O)cc(Br)cc(F)c1F C(CCCC(=O)N1CC(CNC(c2ccc(NC(C)=O)nc2)=O)CC1C)SC c1(OC)cc(C)cc(C(=O)N(C2CCN(Cc3cnon3)CC2)CCO)c1C C(c1ccc(Cl)c(Cl)c1)=CC(N1CCN(C(CN2C(=O)CCC2)=O)C2C1C2)=O CC(C)C(O)C(C)(C)C(=O)N1CCCC(C(=O)NC2(C)CC(F)(F)C2)CC1 C1(CC(N2CCCC(CF)C2)=O)C2CCCC2N1C(C1(CF)CCOCC1)=O C=C(C)C(O)CC(=O)NCC(c1ccc(F)cc1)NC(c1cc(O)ccc1C)=O C1(NC(C2=CC(C)(C)C2)=O)C2CCCN(C(=O)COCc3nc[nH]n3)C2C1(C)C C1(CC=C)CCCN(C(=O)CCC2CCN(C(=O)COCC=C)CC2)C1 c1(C(N2CC(CNC(=O)CS(=O)(=O)CCO)C(O)C2)=O)cc2c(cn1)OCCO2 C1(NC(CCC(=C)Cl)=O)CCCC12CN(C(c1cn(C(C)C)nc1Br)=O)C2 N1(C(c2ccc(COC)o2)=O)CCN(C(=O)Cc2c[nH]nc2O)CC1CF N1(C(C(CC=C)OC)=O)CC2(C1)CN(C(C1CC(=O)NC1(C)C)=O)C2 c1(NCc2c(-c3ccc(COC)o3)cccc2)ccc2c(c1)C(=O)N(C)C2 C1(O)(C(=O)OC(=O)CC2CCCO2)CC(CN(C(C)(C)C)CCCl)C1 Cc1cc(N(C)C)cc(S(=O)(=O)Nc2ccccc2F)c1C.C12CC(C1)N2 N1(C(C(=O)NC(CC)(C)C)C(C)CC2CCCCC2)CCC2(C1)NC(=O)NC2=O C1(CC)C(NC(c2ccc(C(F)(F)F)s2)=O)CCN1C(=O)Cc1csc(C)n1 C1(CC(=O)NCc2ncsn2)CC(F)CN1C(c1ccncc1F)=O c1(OCOC)ccc(C(=O)NCC(C)(CO)NC(c2oc(C3CC3)nc2C)=O)cc1 C(CCC(C)C)(C(=O)N1CC(C(=O)OC)C1)NC(COCCOCC#C)=O c1(N(C)CC)nnc(C2(CO)CCOCC2)n1CC(C)(C)C CC1CC(C(=O)N(C2CC(NC(c3ccoc3)=O)C2)C)C1 N1(C(COc2c(OC)cccc2)=O)CCC2CC1CN2C(=O)C#CC1CCC1 C1(N(C(CCN(C)C)=O)CC2CCCO2)CNCC1(F)F C=CCC(CC=C)C(=O)NC1(C(=O)Nc2ccc3c(c2)CCO3)CC1(C)C CC(CC(=O)NCC1(C)CCCN(C(C23CCC(CC2)C3(C)C)=O)C1)P(C)(C)=O N1(C(COCC)=O)CCCOC(CNC(=O)COc2ccc(Cl)cc2OC)C1 Cc1ccc(C(=O)NC2CC2C(=O)Nc2ccc(F)c(C(N)=O)c2)cc1C C(=O)(CC1=CCOCC1)NC1CCCC(N(C(=O)CCn2ccnc2)CC)C1 CC(C)C(C(=O)NC1CCCCC1NC(=O)COC(F)F)n1cccc1 C(CNC(=O)Cc1nnc(O)s1)(C(C)C(C)C)NC(c1c(OC)ccs1)=O CC1=C(C(=O)NC2CN(C(c3cccnc3N(C)C(C)C)=O)CC2(C)C)CCO1 C1(C2CC2)(C(=O)NCC(CC)(CC)NC(=O)CCc2nncn2C)CC=CC1 C(=O)(CCC(=O)NC1CC(CNC(c2cncn2C(F)(F)F)=O)C1)OC c1(NC(C2CC3CC3N2C(c2ccnnc2O)=O)=O)cc(Cl)ccc1CO N(C1CCCc2cccnc21)(CCO)Cc1ccc(OC)c2c1cccc2 CC1CC(CNC2(C)CN(C(C3(F)CN(C(=O)OCC)C3)=O)C2)CCO1.C(C)(C)(C)O N1(C(C(CC=C)C)=O)CCCCC2(CCN(C(c3ccc(Cl)nc3N)=O)C2)C1 Cn1ncc2cccc(C(N3CCC4CN(C(=O)C(F)C(F)(F)F)CC34)=O)c12 c1(OC(C(=O)N(C(CCNC(c2c(C)n[nH]c2C)=O)C)C)C)ccc(Cl)cc1Cl C12(CNC(C(CC)CO)=O)CCCCC1N(C(=O)C(O)C1CC1)CC2 C(CC1CNC(=O)CO1)NC(C1(NCCOC)CC1)=O.C(CCF)OC O=C(C1=COCCC1)N1CCCC1CNCc1ccc(F)c(F)c1 CC1C(NC(=O)COCCN(C)C)CCCN1C(c1nc(C(F)(F)F)cn1C)=O c1(CN=C(NC(C)C)NCC23CCCC2CC(=O)N3)nc2c(s1)CCCC2 C1(NC(c2nnnn2CCSC)CCOCC=C)CC2CC(OC)C2C1 C(=O)(CCS(=O)(=O)c1ccc(OC)cc1)N1C2CC(NC(C=CC)=O)C(C2)C1 N1(C(C(C2CCC2)C2(CC(C)(C)C)CC2)=O)CCCC1CC(=O)NC.CO C1(C(=O)NCC2(CO)CC23CCC3)CCCCN(C(=O)Cc2ccns2)C1 Cn1nnc(C(=O)NC2CCC2NC(=O)C(O)c2ccco2)n1 C12(CC)CCC(C(=O)OCC(C)OC(C)C)(CC1)CO2 Cc1ncc(N)cc1C(N1CCC(C(C)NC(=O)CN2CCCC2)CC1)=O N1(C(C(CCC)OC)=O)CC(C(=O)N(C)CCC2OCCO2)CC1(C)C C=CCC(CNC(=O)C(F)(F)C(C)O)C(=O)NC1CCC(=O)N(CC)C1 c1(COC)nc(NCC2CNC(=O)C2(F)F)cc(=NC2COC(C)(C)C2)[nH]1 C1(C#N)(C(N2C3(CC(C#C)C3)CC2)=O)CC2CCC1CC2 N1(C(CN(C(=O)OC)C)=O)CCC(C)C(NC(=O)CCC(=O)N(C)C(C)C)C1 c1(C(N2C(C)(C)CC(NC(=O)CCn3cncn3)C2)=O)coc2c1C(=O)CCC2 c1(-n2c(CNC3CC(N)C3)nnn2)ccc(F)cc1.c1(CCSC)cn(C)cn1 c1(C(=O)NC(CNC(C2(C3CC3)CCC2)=O)C2CCC2)cc2cccnc2s1 c1(C(N2CCCC(C(=O)OCC)C2C)C(=O)NC)c(C)nn2ccccc12 c1(NC(CC(=O)OC)C)cccc(SC)c1 N1(C(CC(C)SC)=O)CCCCC12CC(NC(=O)Cn1ncc3ccccc13)C2 C(=O)(C(CC(C)C)C(N)=O)NC1CN(C(c2c(C(=O)OC)c(C)[nH]n2)=O)CC1C C1(CCNC(C(CC)OCC)=O)CCCN(C(c2ncsc2C(=O)OCC)=O)CC1 Cc1cscc1C(N1CC(c2ocnc2C(=O)NCCc2ccccc2)C1)=O C1(NC(C(C)(C)c2cc[nH]n2)=O)CC2CCC(C1)N2C(C1CC1C(F)F)=O S(=O)(=O)(CCC(=O)N(C)CCOCCCNC(c1coc(C(F)F)n1)=O)NC N12CCNC(=O)C1c1ccc(o1)C2.O=C1CCCN1Cc1ccccc1 C(CCC(C)(C)C(=O)NC1CC2CCC(C1)O2)NC(C(C(C)C)=O)=O c1(C(C)NC(=O)C(N2CC(CC3CC3)C3(CC3)C2)=O)cc(F)c(F)c(F)c1 N1(C(C2C(NC(c3ccc(C(N)=O)o3)=O)CCC2)=O)CC(CO)CC12CCC2 CC1CC(C(=O)NCC2C3CC2N(C(=O)CCC(=O)c2cccc(F)c2)C3)=NO1 C1(C(N(CC(=O)NCc2cccc(O)c2C)CC)=O)CC(=O)CC(=O)C1 c1(C(C(=O)OCC2CCOC2)(F)F)cccc(F)c1Br N1(C(C(COCC)C)=O)CCCC(CC(=O)NCCCOCCCO)C1 C1(CNC(C(C)C(C)(C)C)=O)CCC2(CN(C(=O)Cc3ccco3)C2)O1 c1(CC)cc(=NC(=O)C(C)C2CCN(C(=O)CC3CCN(C)C3)C2)[nH]n1C CN1CCC(OCCC(=O)NCC2(CNC(C3CCNC3=O)=O)CCCC2)CC1 C(=O)(C1=CCC(C)(C)CC1)N1C(C)CC(CNC(=O)C(F)C2CCCC2)C1 c1(C(=O)NC23C(CCN(C(CCC=C(C)C)=O)CC2)C3)cnc2ccncc2c1 c1(OCC(N2CC(NC(C)=O)C2)=O)cncc(C)n1.C(=O)(CCC(C)C)N N(C(=NCCCCl)NCc1cnn(C)c1)C1CCN(C2CCN(C)CC2)CC1 c1(CN(C(c2nc(C(=O)NCC=C)sc2)=O)CCOCCO)ccc(C)cc1C C1(N(C)C)CCC(C(=O)NC2CCC2NC(C2(c3ccc(Cl)cc3)CC2)=O)CC1 CC(C)(C)C(CNC(=O)CCc1ccncc1)NC(c1ccnc(C2CC2)c1)=O C1(O)(CNC(C2CCCSC2)=O)CCN(C(=O)CN2CCCC2CO)CC1 c1(C(=O)OC)c(F)cc(Cn2cc(-c3ccnc(Br)c3)nn2)cc1F C(=O)(C(O)P(C)(C)=O)N(C)Cc1cccc(CNC(=O)C(C)N2CCCC2)c1 C1(CC(=O)OC)CCC(NC(=O)C(N2CCC(C)(N3CCOCC3)C2)=O)CC1 Cc1cc(C(=O)NCC(CO)NC(C2C3CC4C(C3)C24)=O)nc(C)c1 Cc1cc(CCC(N2CC=C(CNC(c3ccn(C)n3)=O)CC2)=O)cc(C)c1 C1(O)(CNC(CC2(C)CCCO2)=O)CCCN(C(=O)Cn2cc(C3CC3)cn2)C1 c1(C(=O)NCCCOCCN(C(=O)CN2CC3CC3C2)C)c[nH]c2cccnc12 C1(NC(c2n(CC)cnn2)C(=O)OC)(CC)CCC(O)C1 C1(CC=C)(NC(C2CC3CCC(C2)S3)=O)CCCN(c2ncns2)C1 C(=O)(CC(C)C(C)C)NCCCN(C(c1ccc(C)c(Br)c1)C(=O)NCC)C C1(CC(=O)NC(C2(O)CN(C(c3cccn3C)=O)C2)C)CN2CCN1CC2 C1(CNC(CC(C=C)(C)C)=O)CN(C(=O)C(C2CCCCCC2)F)CCC1(F)F CC1CSCC1N=c1[nH]c(=NCCCc2nc(=N)[nH][nH]2)[nH]c2ncn(C)c12 N1(C(c2c(C)ncnc2)=O)CCC2CCC(NC(=O)CSC(F)F)C1C2 Cc1c(C(=O)OC(C)C(=O)Nc2ccccc2)cc(N)cc1O C1(C(N(CCCNC(c2c(C3C(C)C3)noc2)=O)C2CC2)=O)COCCC1C C(=O)(CC1COc2ccccc21)NC1CC(NC(c2cncn(C)c2=O)=O)C1 C(C(=O)N1OC2CCC1CC2)(C1CC1)NC(C1CC2CCC1CC2)=O c1(NC2CC(CNC(C(COC)OC)=O)C2)cc(C)ccc1[N+](=O)[O-] Cn1ccc2ccc(CNC(=O)CN3CCC(C)(C(=O)O)C3)cc12 c1(C(=O)NC2CC(C(=O)Nc3cnc(C(F)F)cn3)C2)cc2cccnc2[nH]1 CC(CC1CCCC1)C(=O)N1CC(O)(CCNC(=O)CCCC2CCC2)C1 c1(CCC(N2C(CCNC(c3cc(C)sc3C)=O)CCC2)=O)ccc(Cl)c(F)c1 C12(C(N3CCN(CC(N4CCC(CO)C(O)C4)=O)CC3)=O)CCCC1C2(F)F c1(C(=O)NCC(CC)NC(c2nccnc2Cl)=O)coc2cc(O)ccc12 N1(C(C(CC)O)=O)CCC2(CC1)CC(NC(c1cnc3c(c1)CCOC3)=O)CO2 c1(C(N(CC(O)CN(C(=O)C(=O)C(C)(C)C)C)C)=O)cccc2c1COCC2 c1(SC)nccc(=NC2CC3CN(C(=O)C(C)SC)CC23)[nH]1 c1(C(=O)NC(C2CCN(C(C3(P(C)(C)=O)CC3)=O)CC2)C)ccc(=O)n(C)n1 c1(C(=O)NC2CCC(NC(C=Cc3cn(C)nn3)=O)C2)ccc2c(c1)nnn2C c1(NC)cccc(-c2cnc(CC(N3CCC(C)(O)C3)=O)nc2)c1 N1(C(C2(C)N(C(c3ccc(OC)cc3OC)=O)CC2)=O)CCc2c(O)n[nH]c2C1 Cc1cc(C(N2CCC(CO)C(NC(c3ccccc3O)=O)C2)=O)c(O)nn1 C1(CC(=O)NCc2cccs2)CCCN1C(C1CCCC1Oc1ccccc1)=O C(CCCC(=O)NCc1cccc(C(=O)N(C2CCSCC2)C)n1)OCC Cc1cc(C=CC(=O)NC2CC(CNC(c3nn(C)c(C)c3Cl)=O)C2)c[nH]c1=N Cc1cc(COC(C2CCC=CO2)=O)n(C2CC2)n1 CC(C)C(C(=O)N1CCCC1C1(NC(C2CN(C)CCO2)=O)CC1)n1ccnc1 c1(C(=O)NCC2C(C)CN(C(=O)C(F)C(C)(F)F)CC2)nccc2ncccc12 C(=O)(CCCC(F)(F)F)N1CCC(C(C)NC(c2coc(N(C)C)n2)=O)CC1 c1(C(N2C(C)CC(NC(=O)Cc3cnc(C(F)(F)F)s3)C2)=O)ncn2c1CCC2 c1(OC)ccccc1C(N1CCCC(C(C)(C)C(=O)NC(CCO)C2CC2)C1)=O Cn1ccc(C(N2CCCC(CNC(=O)COCCF)C2)=O)c1-c1ccccc1 C(CN=C(NCCC1OCCC1(C)C)N(C)Cc1nnc(C)s1)OC N1(C(C(C)OC2CCCC2)=O)CCCCC1CCNC(=O)C(C)N1CCC1 N1(C(c2cc(CC)[nH]n2)=O)CCCC1(CNC(c1ccccc1)=O)COC Cc1cc2ccc(C(N3CCC(NC(=O)Cc4cnco4)C(C)C3)=O)cn2c1 c1(C(=O)NC2CCC(NC(C(CCC=C)(F)F)=O)C2)coc2c1C(=O)NCCC2 c1(OC)ccc(C(C(=O)NC(C)C)N(CC(C)C)C)c(Cl)c1.c1(C)ccco1 C=CC(C)(C)CC(=O)NCC1C2CN(C(C)C)CC12.c12ccc(cn1)NC2 C1(C)(C(N(CCCCCNC(C2CNC(=O)N2)=O)C)=O)CS(=O)(=O)C1 N1(C(C(C(C)C)OC)=O)CC2(CCCCN(C(=O)C=Cc3cccc(F)c3)C2)C1 c1(C(=O)NC2CCCN(C(c3c(OC)scc3)=O)C2)c(F)cccc1C#N N1(C(C=CCC)=O)CCN(C(=O)C2=C(C)CCC2)CC1CC(C)(C)C C1(CC(=O)NCC2CCCC2)CN(C(=O)CC2CCSC2)CCO1 C(=O)(C(C(C)(C)C)SC)N1CC(C(=O)NC(C2CCOCC2)C#C)OCC1 N1(CC(=O)NCC(CC)NC(C2(CC(F)F)CCC2)=O)CCC(C)(C)C1 N1(C(c2cncc(OCC)c2)=O)CC(C)N(C(=O)C2=CCCOCC2)CC1C N1(CC(C(=O)O)(F)C(=O)O)Cc2ccc(-c3ccccn3)cc2C1 C1(NC(CC(C=C)C)=O)CCC(C)(NC(c2cc(-c3csc(C)n3)c[nH]2)=O)CC1 c1(C2(C(N3CCN(C)C4C3C4)=O)CCC2)cccc(C#N)c1F CC(C)(C(=O)NCc1ccccc1CNC(=O)CCCCCF)C(F)(F)F c1(CC(=O)NCC2(O)CN(C(CCCC(N)=O)=O)C2)ccc2c(c1)NC(=O)CO2 CC(C)C(C(=O)N1CCC1CNC(=O)CC1CC12CC2)N1CCN(C)CC1 c1(OC)cc(O)ccc1NC(C1CC1C(N1CCNC(=O)C1C)=O)=O c12cc(Cl)ccc1NC2.CCCCC(CO)NC(C1CCN(CCC)C1)=O C1(CC(=O)NC(CCCNC(c2c(CCC)[nH]nc2)=O)C)CC2(CCC2)CO1 CC(N=c1[nH]c2c(c(=NC3CCC3)[nH]1)CSC2)c1ccnc(Cl)c1 CCC(CC(=O)N1CC(NC(=O)CC(C)(C)O)CCC1C)CC(C)C c1(CCC(=O)N(CC(N2C(C)CCCC2C)=O)CCCC(=O)NCCSC)nnc(O)nc1O N1(C(C(C)OCCNC(C2(CC#C)CC2)=O)=O)CCOCC(CO)C1 C1(NC(c2ccc(SCCC)cc2)=O)CN(C(c2csc(CO)n2)=O)CCC1C C(=O)(CC(CC(C)C)N(C(=O)C(Cl)Cl)C)N(C(CCCC)C)C N1(C(C=C(C)C)=O)CCCC(C)(C(=O)Nc2cc(C(=O)OC(C)C)ccn2)C1 N1(C(CNC(CCNC(=O)NC)=O)(C)C=O)CC2C3CCC(O3)C2C1.C(COC)N N(C1CCCOc2ccc(I)cc21)OC(c1ccc(N)c2c1CCCC2)=O c1(CC)cccc(C(=O)N(C)CC2C3CN(CCOCC4CC4)CC23)n1 Cc1cnc(C(=O)NC2(C(=O)NC3(C)CCCC3(C)C)CCOCC2)cc1C C(=O)(CC(C)(C)CC(=O)OC)NCC1CN(C(c2cccc(SCC#C)c2)=O)C1 c1(-c2cc(NC(c3n(C)cnc3)=O)ncc2)cnccc1C#N CC1(C)OCC2CC12C(N1C2CCC1(CNC(=O)Cc1nc[nH]n1)CC2)=O N1(C(C(N(C(Cc2c(C)ccs2)=O)C)C2CC2)=O)CC2(CCC(=O)O2)C1 C1(NC(c2cccc(Cl)c2)=O)COC2(C1)CN(CCc1c(Cl)cccc1Cl)C2 n1(C2CCN(C(c3nc(C)nc(I)c3)=O)C2)cnc2ccccc12 C(CC(C)(C)CC(=O)NC1(C)CCN(C(=O)CSc2n[nH]c(O)n2)C1)OC Cc1cc(C(=O)NCC(=O)Nc2cn[nH]c2)cc(C#N)c1 C1(NC(C(C)c2ccco2)=O)CC(C(F)F)(NC(c2csnc2Cl)=O)C1 c1(CC(C)C(=O)NC2CCN(C(c3nccn3C)=O)C2)ccccc1Cl C(C(C(C)(C)C)NC(c1cc[nH]c(=N)n1)=O)NC(CC(C)OC)=O C(C1=NOC2CCCC12)Nc1n(-c2ccccc2)nc(C)c1C CC(C)C(C(=O)NCC(F)CNC(C1CCSC1)=O)N1CCN(C)CC1 c1(CC(N2CC(C(C(=O)NCC(C)C(F)F)OC)C2)=O)ncccc1F C1(NC(C(C)(c2ccccc2)N(C)C)=O)Cc2ccccc2NC1=O c1(-n2cc(CSCCNC(c3cnc(CC)[nH]3)=O)nn2)cc(OC)ccc1F c1(C(N2CCN(C(C(CC)C)=O)C(CF)C2)=O)[nH]c2cc(F)ccc2c1C N1(CCC(=O)NC2CN(C(C3(C)CC3)=O)C2)CCc2ccccc2C1=O N1(C(C2(C)CC2(F)F)=O)CC(F)CC1C(=O)NC(C(O)CO)C1CC1 CCC(C)CCC(=O)N1CCC(C)(CNC(=O)CSc2c(C)n[nH]c2C)C1 C(C(=O)N1CC2CC1C2CO)(C(C)C)NC(C1C(OC)CCC1)=O c1(C(N2CC3C(CNC(=O)C=Cc4cnccn4)C3C2)=O)cc2cscc2s1 c1(C(N2CC(COC)C2)=O)ccc(C(F)F)c(OC)c1 Cn1cnc(C(=O)N(CCCNC(C2CC2(Cl)Cl)=O)C2CC2)n1 N1(C(C(CN(C)C)(F)F)=O)CC=C(C(=O)N2CC(C(C)(C)O)C2)C1 c1(C(=O)OC)cc(C)c(C(=O)NC(C)CN(C)C(c2cc(Cl)c(Cl)s2)=O)o1 Cc1nn(C)c(N)c1C(N1CCN(C(=O)Cc2cscn2)C(CCO)C1)=O c1(C(=O)NCC(CNC(C(CC)C#N)=O)C)cn2cccc(C)c2n1 C(=O)(CCCCC(C)(C)C)N1CCN(C(C(CCCOC)C)=O)CC1CCO c1(C(=O)NC2C(C)CN(C(C3CCC4(CC4)C3)=O)C2)ccc2c(c1)OCCO2 C(=O)(CCCC(N)=O)N.C1(N(C)CCO)CCN(C(=O)C(C)(C)NS(C)(=O)=O)C1 c1(OC)cc(CN(C)CCN(C)C(C2(F)COC2)=O)cc2c1OCO2 c1(C(N2CC(OCCNC(C(c3cn(C)nc3Cl)C)=O)C2)=O)cccc(CO)c1 CC1(O)CCCN(C(C23CC(NC(=O)CC4(C(F)(F)F)CC4)(C2)C3)=O)CC1 Cc1ccc(C(=O)NCC2CCC(NC(c3cc(C(N)=O)co3)=O)C2)c(F)c1 C1(NC(C=C(CCC)CCC)=O)CC(O)CN(C(=O)Cc2cc(C)ns2)C1 Cc1ccnc(C(N2CCC(OCCNC(c3cc(Cl)sc3Cl)=O)C2)=O)c1N c1(C(=O)NCC2(CNC(Cc3nnc(C)s3)=O)CC2)cnn2cccc(Cl)c12 c1(C(=O)NC2CN(C(c3ccc(C)c(C)c3)=O)CC2C)ccc2nnc(O)n2c1 C1(NC(C=CCOC)=O)CCC(NC(=O)COC2CC2)CC1.C1(C)CC(C)O1 C(=O)(CC(C)NC(CC)CN1CCCC1)NC1(CO)CC1 c1(N(C(N2CC(C)=C(C)C2)=O)C)nc2ccccc2[nH]1 C1(CC(C)NC(C=CCC)=O)CC2CCC(C1)N2C(C1OCCC1C(C)C)=O C(CN=c1[nH]c2cccc(F)c2o1)N(C(=O)C1c2ccccc2O1)CC Cc1cccc(C(=O)NC2CCN(C(c3cnsn3)=O)C(C3CC3)C2)c1F CC1C(C(=O)NC2CN(C(c3c(C4CC4)cnn3C)=O)C2)CCN1C Cn1c(O)ncc(C(=O)NCCCCC2CCCN(C(=O)CCC(N)=O)C2)c1=O CCCCC(C(=O)N1CCOC(C(N2CC(c3nc(C)no3)C2)=O)C1)C(C)C CC(C)CC(O)C(=O)NC1CC(C)CN(C(c2cccc(F)c2C(F)(F)F)=O)C1 c1(NC(C=CC)=O)ccnc(OC)c1.C1(C(=O)N)CC1C(=O)O c1(C(=O)NCCC2C(C)CN(C(=O)CNC=O)C2)ccnc(Br)c1N c1(C(N2C(C)CC(CNC(C3=C(C)CC3)=O)C2)=O)nn(C)c2c1CCC2 C12(C(=O)NC3C(NC(c4ccc(CN(C)C)nc4)=O)C3)CCC(CC1)CO2 N1(CCNC(COCCC(C)C)=O)CCC(N=c2[nH]c3ncc(Cl)cc3s2)CC1 Cc1cc(O)ncc1C(=O)NC1CCCC(C(F)(F)F)(C(=O)O)C1 CC(C)(CCCCNC(C1(C(C)(F)F)CC1)=O)NC(c1cncc(N)c1)=O C1(CNC(C2CSCCS2)=O)CCN(C(=O)Cc2ccc(Cl)nc2)CC1(F)F Cc1cc(N)c(C(=O)NCC2CN(C)CCN2C(=O)CN2CC(C)(C)C2)cc1C C1(CNC(C2(CCCC)CC2)=O)COCC1NC(C1(CO)CC1)=O C(CCCCCC(=O)C(CNC(CC(C)C)=O)=O)N.C1(N)CCCCN(C)C1=O C1(N(C)C(c2cc(Cl)n(C)n2)=O)CC2CCC(C1)N2C(=O)CCCn1ccnn1 c1(OC)cc(CN2CCC2(C)C(=O)NCCc2ccncc2)cc(C)c1 Cn1ncc(C(c2nnnn2C(C)(C)C)NCCSS(C)(=O)=O)c1Br CCC(F)(F)C(C)(C)NC(=O)CC(=O)C(C)n1cccn1 C(=O)(CC(O)CNC1(c2ccccc2)CC1)NCCNC(CSS(C)(=O)=O)=O Cc1c(Cl)ccnc1C(=O)NC(C1CCCCN1C(c1cc(F)n[nH]1)=O)C C1(C(N(CC(C(C)C)OC)C)=O)C=CCCN1C(=O)CS(C)(=O)=O c1(NC(=O)NC2C(OC)CS(=O)(=O)C2)nc(Cl)ncc1[N+](=O)[O-] C1(C(=O)NCCOCCCNC(COCC=C)=O)CCCC2(C1)CC2(F)F C12(NC(=O)CCc3cc(Cl)cs3)CCC(CC1NC(C1CC3(C1)CC3(F)F)=O)C2 c1(C(N2CCC(C(C)NC(c3cc(F)ccc3Br)=O)C2)=O)cc2cnccc2[nH]1 N1(C(c2ccnc(C)c2O)=O)CCC(CNC(c2cccn2C)=O)C12CCC2 C1(C(N(C(CC#C)C)C)=O)CC(O)C(O)CC1CNC(=O)CN(C(=O)COC)C c1(OC)ccc(NS(=O)(=O)CC2CCCS2)cc1C C1(C(C)NC(COCCCCCC)=O)CCN(C(=O)C(n2nccc2C)C)CC1 N1(C(C2C(c3cn(CC(C)C)nc3)C2)=O)CCC(COCC(C)C#N)CC1 c1(CC(N2CC3CN(C(c4cnc(C)s4)=O)CC3C2)=O)cccc2cnccc12 N1(C(C2=CCCC2C)=O)CCC2(NC(=O)CCc3nc(O)n[nH]3)CCCC12 C1(CCC(=O)OCC)CCN(C(=O)CCc2cnccc2C(F)(F)F)C12CCC2 c1(C(=O)NCCCN(C(C2CC(=S)NCC2)=O)C2CC2)cccc2ncccc12 C(c1cc(Br)ccc1F)=CC(N1CC2C(CN(C(CC(C)C)=O)C)C2C1)=O c1(C(=O)NC2CC(NC(c3c(OC)ccnc3)=O)C2)cc(F)cc(F)c1Br C12(CCNC(N(CC)CC3(O)CCC3)=O)CC(CCO1)C2 Cn1cnc2cc(C(=O)N)ccc12.C(=O)(CCCCCCCBr)C1C2CNCC21 c1(C(N2CCC(CNC(CN(C(C(C)C)=O)C)=O)C2)=O)cc(F)c(CO)c(F)c1 c1(C(N2CCN(C(=O)CCc3cccs3)C3C2C3)=O)ccc2c(Cl)ccnc2c1 C1(C)(C(=O)NCC(N(OCC)C)=O)CC(O)CN1C(=O)COCC(=O)OC C1(C(=O)NC(C(=O)NCCC23CCCC2C3)C2(C)CC2)CC(C)(O)C1 N1(C(c2ccc(C)[nH]2)=O)CCN(C(c2ccnn2CC(F)(F)F)=O)CC1CCO O=S(=O)(c1cccnc1N)N1CCSCC1CO.C12(CO)CCC(CC1)C2 c1(C(N2CCCC(NC(c3c(N)non3)=O)C2)=O)ccc2nc[nH]c2n1 C(=O)(C(CC1CCC1)NC(=O)CC1(O)CCC1)NCC(C)CN(C)C c1(CC(=O)N(CCC(=O)NC2CC(OC)C2)CC2CC2)cccnc1F c1(C(=O)NCCNC(C(CC)OC)=O)cc(-c2ccncc2)ccc1OC C1(NC(C(CC#C)O)=O)C2CC3CC(C2)CC1(CNC(c1ccsc1)=O)C3 c1(C(=O)NCCCN(C(=O)Cc2n[nH]c(C)n2)CC)cnc(C(F)(F)F)s1 CCCCCC(O)C(=O)N1CC2CC1CN(C(C1CCCC(F)C1)=O)C2 C(=O)(CC1OCc2ccccc21)NCC(C1CCC1)NC(CCCOC)=O C#CCCCCCCC(=O)NC1CCC2CCN(C(=O)CC(C)C(F)F)C12 C#Cc1cnc(C(=O)NC2C=CCN(C(c3ccc(CC)cc3F)=O)C2)c(C)c1 C1(CNC(C(=O)NCCOC)=O)CCN(C(=O)Cc2ccsc2Cl)C1(C)C Cn1cc2c(n1)CC(C(N1CC(CNC(C3CCCC(=O)CC3)=O)C1)=O)CC2 N(C1CCc2c(Br)ccc(Cl)c21)C(Cc1c(C(C)C)cccc1)=O c1(C(=O)NC2CN(C(c3c(C(N)=O)ccs3)=O)C2)ccc(F)c2cnccc12 C1(NC(=O)Nc2scc(-c3c(C(=O)OCC)csc3)n2)CC=C(C)CC1 C1(C(N2CC(O)(CCNC(CCSc3n(C)nnn3)=O)C2)=O)CC12CCCOC2 C1(CCCCC)CCC(C(=O)NCC=CCNC(=O)C(c2ccccc2)=O)O1 N1(C(c2nc(OC)oc2)=O)CCC(C(C)OC)(C(=O)O)C1 Cc1cc(C(=O)NCC2CN(C(C3CCCC3C)=O)C2)c(O)c(Br)c1 C1(CNC(C(C)=C(CC)C)=O)CC(O)(CNC(C2(CC)CC2(F)F)=O)C1 Cc1nnc2n1CC(C(=O)N(C1CCN(C(C3(Br)CC3)=O)C1)CCO)CC2 C1(CNC(c2cc(OC)cc(Br)c2)=O)C2=C(N(C)C1=O)CCCC2(C)C C1(NC(C(C)OCC)=O)CCOCC1NC(c1cn(C)nc1-c1cccnc1)=O C1(CC)CCC(C(=O)NC(C)CNC(=O)Cc2cnco2)O1 N1(C(CCC)C)CCc2nc(C(N3CC=CC3CO)=O)cn2CC1 CCCC(C(=O)NCC1CC2(CC2)CN1C(c1nccc(C(F)F)n1)=O)C(C)C C12(CCCCCC1)C(=O)N2.c1(SC)ncc(NC(=O)CC(C)n2ccnc2)cn1 C(=O)(CN=C(NC1CCC12CCC2)N1CCCC(n2ccnn2)C1)NCC=C c1(N(C2CCN(C(C(C)(CO)CO)=O)CC2)CCO)ncc2c(n1)NC(=O)C2 c1(CNC(CC)=O)cnn2c1CN(c1ccc(C(F)(F)F)c(C(C)C)n1)CC2 C(CCSC)(C(=O)NC(c1nc(C)cs1)C)NC(C=C(C)C(F)F)=O CC1(C)CC(NC(c2conc2C2CC2)=O)CN(C(c2nccc(N)c2Cl)=O)C1 CC(C)(CC(C(=O)NCCC#N)N1CC(F)C(F)C1)C(F)(F)F C(c1ccccn1)=CC(N1CC(CN(C)C(C2CC(n3ccnn3)C2)=O)C1)=O C1(C(=O)O)(NC(c2scnc2-c2cccc(I)c2)=O)CCCCCCC1 C12(C(N3CC(N(C(c4cc(C)ns4)=O)C)C(O)C3)=O)CCC(CF)(C1)OC2 C1(C(=O)NCCCNC(CCC=CC)=O)(Cc2ccccc2)CCCCC1 N1(CC(=O)N(CC(N2CCC(OC(CC)=O)C2)=O)C2CC2)CCCCCC1=O c1(C(=O)NC(CC)CNC(c2nsnc2O)=O)coc2c1C(=O)NCC2 C(=O)(C1=CS(=O)CCC1)NCC1C(CCC)C1 Cc1nc(C)c(C(N2CC=CC2C(=O)NCc2ncsn2)=O)o1 C12CC3CCCC(C1)N3C(=O)COC(=O)N2.C1(C(=O)OC)C(CN=[N+]=[N-])C1(C)C C1(C(N2C(C(=O)NC3CC(CCOC)C3)C=CC2)=O)CC2COCC2C1 C1(CC(=O)N(CCCNC(=O)Cn2ccc(Br)n2)C)CCC(F)(F)CC1 c1(C(=O)NCCC2(CNC(CC(=O)OC)=O)CC2)ccc(N2CCCC2)nc1 N1(C(C(N)=O)=O)CCC2(CCC(CNC(c3cc4ccsc4s3)=O)OC2)CC1 C(CNC(c1cc(F)cs1)=O)(CC(C)C)NC(c1cc(C)oc1)=O C1(C(=O)NCCCOCCN(C(=O)CN(C)C)C)CCCCC1n1ccnc1 N1(C(CN2CC(C)(C)C2)=O)CCCCC(C2CN(C(=O)C(=O)C(F)(F)F)C2)C1 C1(NC(c2c(CC)cc(F)cc2)=O)CCC(O)CN(C(=O)C(F)(F)CO)C1 C1(C(N(C2CC(F)(F)C2)C)=O)CN(C(c2cnn(C)c2Cl)=O)CCC1(C)C C(C)(CCCCNC(=O)C=C(CC)CC)NC(CC1(CCC#C)OCCO1)=O N1(C(c2c(C)n(C3CC3)cc2)=O)CC2C3CCC(C2C1)N(C(=O)C(C)N(C)C)C3 c1(CN2CC3N(C(c4ccc(F)c(F)c4)=O)C3C2)ccnc(Br)c1F C(=O)(C(CNC(c1ncccc1O)=O)CC(C)C)NC(CC#C)CC#C C(=O)(CC(CC(C)C)NC(C1CCC(N(C)C)C1)=O)NCc1cc(C)on1 c1(C(=O)NC2CC(NC(c3cccc(CCC)c3)=O)C2)ccc2c(c1)CCOC2 C1(C(=O)N(C(C)CO)C)(CNC(CC2ON=C(C)C2)=O)CC2(CC2)C1 Cc1ncoc1C(=O)N(C1CC(C(=O)N(C2CC(OC)C2)C)C1)C C1(NC(C(CC)C#N)=O)CCN(c2ccnc(C3CC3)n2)C(C)C1 c1(CC)oc(C)cc1C(=O)NC(CN(C)C(C1(CC2CC2)CCC1)=O)C c1(CNC(C2CCN2Cc2csc(C3CC3)c2)=O)cccc2cncn12 c1(C(=O)NCC#CCNC(C(CC#C)C2CC2)=O)ccc(C)c(C(F)F)c1 C1(C)(C(=O)N(C2CCOC2)C)CCC(C(=O)NCCNC(C2CC2)=O)O1.CC N1(C(COCCC(C)C)=O)CCCC(C(=O)NC2C=CC(C)(C)CC2)CC1 C(=O)(C1CCCc2nc[nH]c21)NC1CC2(CN(C(C3(CC)CCC3)=O)C2)C1 Cc1c(C(=O)N(C2CC2)CC2CCCN2C(C2CC(=O)N(C)C2)=O)cccc1Cl C1(C(=O)NC2(CCF)CC(O)C2)(SC)CN(C(=O)CCC2CCCOC2)C1 c1(C(=O)NCCC(C)NC(C(C)SCC)=O)cnnn1CC CC1C(CC(=O)NC2(c3ccccc3)CC(NC(C3CSC3)=O)C2)C1(F)F C(=O)(C1CCc2cccnc21)NC(CC=C)CNC(c1cc[nH]c1C)=O C1(O)(CCNC(C=C(C)C(C)(C)C)=O)CCCN(C(C2(C#N)CC23CCC3)=O)C1 c1(OC)cc(C(C)(C)C)cc(OC)c1OC.C12(CC1(C)C)CN(C=O)C2 CCC(C)(C(=O)NCC1CC(F)CN1C(=O)CC(=O)NC1CC1)OC Cc1cc2cc(NC(c3c4c(nn3C)CCC4)c3nnnn3C(C)C)ccc2o1 c1(C(=O)NC(CC(C)NC(=O)Cc2cncs2)C)c(S(C)(=O)=O)cnn1C CC1CCC(CC(=O)NC23CCCN(C(c4csc(O)n4)=O)C2C3)CC1C C1(C(=O)NCC2C(C)(C)OCC2)CCC2(CC2)N1C(C1C2CC3C(C2)C13)=O Cn1nc(C(F)F)cc1SCC(N1CCCC1C(=O)Nc1cnc(C#N)cn1)=O c1(OC)cnc(N2CCC2C(=O)NC2CCN(C(=O)C(Cl)(Cl)Cl)CC2)nc1 C1(C(N(CCC(C)NC(c2c(C)ccnc2O)=O)C)=O)CCc2ccccc2O1 c1(CNC(=O)CCn2cc(-c3cnc(C4CC4)o3)nn2)ccc(CF)cc1 C(c1ccc(Cl)cc1)=CC(=O)NCCC1CCN(C(c2cccc(OC)c2)=O)C1 N1(CC(=O)NCC(=O)N(C)Cc2c(C)cco2)CCCCC1=O.n12cc(nn1)C2 c1(C(N(C2CN(C(C(C(CC)O)C)=O)C2)C)=O)sc2ccc(C)cc2c1C NC(=O)CC(O)C(=O)NCC1CC(C(=O)NCc2nn[nH]n2)=NO1 C1(N(C(=O)Cn2cccn2)CC)CCCN(C(c2cccc(SC)c2)=O)CC1 CC(C)C(F)(F)CC(=O)N(C)CC1CCC(NC(C2CCC(C)C2)=O)CC1 C(=O)(C#CC(C)(C)C)NC1CCCC(CNC(Cc2c(C)noc2C)=O)C1 c1(C(=O)NCCCN(C(C)C(=O)OCC)CCC)c(CC)nn(C)c1Cl C1(CC)CCCCC1OCC(N1CC(NC(=O)Cc2cnns2)C(C)C1)=O N1(Cc2cccc(C)c2)CC2CCC(C1)C2NC(c1cc(Br)cs1)=O N1(C(C(C)NC(=O)C2CC2)=O)CCCC(CO)(CNC(C2COCC2(C)C)=O)C1 Cc1noc(C)c1NC(=O)CC1CN(C(=O)CCc2ccc(Cl)cc2)C1 C1(NC(CCC(=O)N(C(C)C)C)=O)CC2CCC(C1)N2C(=O)C(C)C(C)O CCCCC(C)(F)C(=O)NCCNC(=O)C(C)Oc1cccc(CC)c1 CC1CCN(C(=O)CCC2CCOCC2)CCN1C(=O)CCc1cocn1 N1(C(CCC(=O)N(CCC)CCC)=O)CCCCCC1CNC(=O)C(O)C1CC1 N1(C(c2c(C)c(F)c(F)cc2)=O)CCn2ncc(C3=CCS(=O)(=O)CC3)c2C1 c1(OC)cc(CC(=O)NC2CCC2CNC(=O)C(C(C)C)NC(N)=O)cc(Cl)c1 N1(CC(=O)NC23CC(CNC(C(C)(C4(C)CC4)OC)=O)(C2)C3)CC(=O)NC1=O N1(C(C(COCC)C)=O)CC2(CNC(c3cc4ccccc4s3)=O)CCC1CC2 C(F)(C(=O)NNc1ccc(Br)c(O)c1)=C(C)C N1(C(C(C=CC)O)=O)CCC(C)C(NC(=O)CCCSC)C1 C(C)(CC(C)(C)C)NC(c1cn(C2(C(=O)OC)CC2)nn1)c1nnnn1C(C)C C(C)(C)(CCC(=O)NC1CCCN(C(c2cncn2-c2ccccc2)=O)C1)OC CCCCC(C(=O)NC(C)(CC)CC)NC(=O)CN1CCOCC1=O CN1CCC(C(=O)NCC2CC(C)(C)CN2C(c2cc(Cl)on2)=O)CC1=O CN1Cc2ccccc2CC1C(N1CC2C(C1)N2C(c1c(O)cccc1O)=O)=O N1(c2cc(NCC(CC)(CC)SC)nc(C(C)C)n2)CCCC(C2(C)CC2)C1 C(CCc1ccccc1)(C(C)NC(C1CCC1(C)C)=O)NC(CC)=O c1(CC)cc(C)ccc1C(=O)NCC(COC)NC(=O)CC1CCCC12CC2 N1(C(C(c2ccccc2)C)=O)CCOC(C)(CNC(=O)Cc2ccc(Cl)cc2F)C1 C1(C(=O)NC2CC(C(C)C)OC2)CCN(C(c2cnsc2)=O)CC1(C)C C1(C)(C(=O)NCC2CN(C(CNC(CC)=O)=O)CC2(C)C)CCCNS1(=O)=O Cc1nc[nH]c(=NCCC2CC(NC(=O)CCc3c[nH]c(C(N)=O)c3)C2)c1Br N1(C(C2N(C(CN(C)C(=O)C3CC3)=O)CC=CC2)=O)CCOCCC1C1CC1 c1(C(=O)NCC2CC2CNC(c2coc(C3CC3)n2)=O)cncc(F)c1 C(=O)(CCS(=O)(=O)N(C)C)NCCN(C)CC1CN(C(=O)C=CC2CCOC2)C1 N1(CC(=O)OCC(C)N)CC2CCN(C(C)(C)C)C2C1.c1(C(CC)C)ccc(O)cc1 C1(NC(c2c(C(C)C)ocn2)=O)CCCC(C(=O)NCC(F)(F)C(C)(C)O)CC1 C1(C(=O)OC)CC(n2cc(C3(C)CSC3)nn2)CN1C(=O)CC1OCCC1(C)C c1(C(N2CCC(NC(CC=C)=O)C(C)(C)C2)=O)c[nH]c2cccc(F)c12 c1(C(=O)NC2CC(C)(NC(c3c(C)c(C4CC4)on3)=O)C2)ccc2nc[nH]c2c1 Cc1ccc(NC(=O)CCC2(C)CCCN2C(c2ccnc(C)n2)=O)c(C)n1 C1(CC)CCC(O)(C(=O)NC2CCC(NC(=O)Cc3ccc(C(C)=O)s3)CC2)C1 n1(CC)cnnc1CNC(N1CCC(c2cn(C3C=CCCC3)nn2)C1)=O C(=O)(C(C)(F)CCCC)NCCCCCN1CCN(c2ccnc(C#C)n2)CC1 CC(C)CC(C)CC(=O)NCC1CCN(C(=O)Cn2ncc(O)nc2=O)C(C)C1 C12(C(N3CCC(N(C(CN4CC(C)(OC)C4)=O)C)C3)=O)CCC(CC1)C(C)O2 N1(C(c2ncc(-c3cccc(C)c3)c(C)c2)=O)CCC2(CCCCC2)CC1 C1(CCNC(C2C(CC)C2)=O)CN(C(c2csc(-c3ccccn3)n2)=O)CCO1 c1(C)nnnn1C(C)(C)C.N1(C(C(C)SCCCNCC=C)C)CCCCC1 C12(CNC(C(C)n3ccnn3)=O)CC(NC(=O)CC3COCCO3)(C1)C(C)(C)O2 N1(C(c2ccc(C)nc2)=O)CCC2(CC1)CC(C(N1CCC1CO)=O)CO2 N1(CCNC(c2[nH]cc(C)c2)=O)CCCN(C(C2(Cl)CC2)=O)CC1 N1(C(c2cn(C(C)(C)C)nc2)=O)CCCC(O)(CNC(=O)CC(F)(F)F)CC1 N1(CCC=C)CC=C(CCNC(C2(COCc3ccccc3)CC2)=O)CC1 C1(CNC(C(CN(CC)CC)F)=O)C(C)CCN1C(=O)CN1CCC(O)CC1 c1(SC)ccccc1C(N1CCC1(C)C(=O)NCCN1CCOCC1=O)=O N1(C(CNS(NC)(=O)=O)=O)CCN(C(c2ccnc(C)c2N)=O)C2CCCCC12 c1(C(=O)NCC(CC=C)NC(c2cccc(CO)c2)=O)ccc(C)nc1O CC1(C)CCC(NC(=O)C(CC2CCC2)NC(=O)CCN2CCCC2=O)C1 N12CCC(CC1)C(=O)NC21CCCC1.C1(C#N)(C(=O)N)CC1C.C(=O)(NCC)NC N1(C(C2C(OC)CCC2)=O)CC2OCC(NC(c3cnn(C4CCC4)c3)=O)C2C1 c1(CC)cc([N+](=O)[O-])ccc1C(=O)NC(C)CCNC(=O)CC1CC(C)OC1C c1(C(=O)NCC2(O)CC(Nc3ncnc(Cl)c3CO)C2)cccc2nccn12 C12(c3nc(-c4ccc(C)cc4Cl)nn3-c3cnc(C4CC4)nn3)OCCCC1C2(F)F.C1C=N1 CCC(C)(C)CC(=O)NCC1(C(F)F)CCN(C(=O)C(C)S(C)(=O)=O)C1 N1(C(c2c(C)cno2)=O)CCC(C)(NC(=O)Cn2cc(C3CCC3)nn2)C1 C1(C(C)(C)C)CN(C(C2CCCS(=O)(=O)C2)=O)CCN1C(C1CC(=C2CC2)C1)=O c1(CN(C(=O)CCNC(=O)CC(C)C2CCCC2)C)cc([N+](=O)[O-])cnc1O C12(CCC(=O)OC)CCCCC1N(C(=O)CC1CCC1=O)CCC2 N1(C(C2c3nnc(C)n3CCC2)=O)CCC2OCCCC2(CO)C1 C1(CC(N2CC3CC2CC3C(=O)O)=O)CC2CCC1CC2.C12(CCC1)C(=O)NC2 C#Cc1cccc(C(N2CC(CNC(C3(Br)C(C)C3C)=O)C2)=O)c1F C1(C(=O)NC2C(NC(c3c(O)ccc(C(C)C)c3)=O)C2)CN2CCCN1CC2 CC1(C)CC(C(=O)NCC2CCOC2=O)CN(C(C2(C)CCC2)=O)C1 c1(CNCCC2(C(=O)NCCCCCC)CC2)nc(OC)c(C)s1 CN1CCC(C(=O)NC2(C)CN(C(=O)CC3CC4(CC4)CO3)C2)CC1=O c1(C(=O)OC)ccc2c(c1)C(C)CN2C(c1ccnc(N(C)C(C)=O)c1)=O C1(n2cc(C3(N(C)C)CCC3)nn2)CC2CCC1(NC(c1ccc(=O)n(C)n1)=O)C2 c1(C(N2CCS(=O)CC2c2cnn(C)c2)C(=O)NCC)cccc(S(N)(=O)=O)c1 Cc1nc(C(=O)NCCC2CN(C(C34CC(C)(C3)C4)=O)CCO2)cn1C Cc1sccc1CC1CN(CCCC(=O)NCCCc2nnnn2C2CC2)C1 c1(CNC(c2ccc(O)cn2)=O)ccc(Br)nc1[N+](=O)[O-] C(CCC(C)(C)C)(C(=O)NC(C)(C)CC)N1CCN(C(C#C)C2CCC2)CC1 c1(C(N2CC(NC(c3c(C)cnn3C)=O)C3(C2)CC3)=O)ccc2c(n1)CCOC2 C=CC(C(=O)N(CC(C)(C)NS(C)(=O)=O)C)c1ccccc1 N1(C(C(C)OCC#C)=O)CCCC1(C)C(=O)NOCCCOC c1(NC(C(=O)NC(C(C)NC(C#CC(=O)N(C)C)=O)CO)=O)cnc(O)nc1O c1(N(C(C)CO)C(=O)C=CCC2(NC(C)=O)CCC2)c(F)cccc1F CCC(C)C(=O)NCC(C(C)C)NC(=O)Cn1cc(C)cn1 N1(C(=O)OC)CCCCC1CN1CCC(n2cccn2)CC1 CC(C)CC(C)N=c1nc2sccc2c(NCc2ccnc(O)c2)[nH]1 N1(C(CC(CNC(CCOC(C)=O)=O)C2CCC2)=O)CC(O)C(C)(C)C1 c1(C(=O)NCC(C)NC(COc2c(C)cccc2)=O)cccc(F)c1I n1(CC(C)C)nccc1NC(=O)NCCc1nc(C2CC2)n[nH]1 C(c1cc[nH]n1)=CC(=O)NCC1CCCC1NC(=O)Cc1ccsc1Br N=c1nc(N2CCCC(C(N)=O)C2)[nH]c(=NCCc2nnc(CC3CC3)s2)[nH]1 c1(C(=O)NC(CNC(c2cccc(OC)c2)=O)CO)c(OC)ccc(Br)c1N C(=O)(CC(CC)SC)NCC1(C(C)NC(c2c(CC)noc2)=O)CC1 Cc1nnccc1C(N1CCCCC1C1CCN(C(C2(C#N)CC2)=O)C1)=O C=C(C)CN=C(NCC1CCC2(CCC2)CO1)NC(CC)CC c1(C(N2C(COC)C(OC)C(C(=O)OC)C2)=O)cc(Cl)cc(Cl)c1F C(=O)(C1=NN(CCO)C(=O)CC1)NC1C(NC(=O)CS(=O)(=O)C2CC2)CCOC1 N1(C(CNC(CCN(CCC)C)=O)=O)CCCC(C)(C#N)C1 C(=O)(CCCS(N)(=O)=O)N1CC(O)(C(C)NC(C2C=CCC2)=O)C1 C(=O)(C1CCc2c[nH]nc21)NC(C(=O)NC1(C(C)C)CCC1)c1ccoc1 c1(C(=O)NCCCN(C(C2CCC(C)S2)=O)C)coc2c1NC(=O)CCC2 C(=O)(C1CCCn2cncc21)N(CCNC(C(CC)OCC)=O)CCOC c1(-c2cc(OCC)cc(Cl)c2)cc(C(=O)NCc2nccn2C)c2[nH]ccc2c1 CCCC(CC)CCC(=O)N1CCCC(N(C(=O)Cc2cc(OC)no2)CC)C1 Cc1cc(N2CCCN(C)CC2)nc(N(C)CC2(F)CCC2)n1 C(=O)(CCC(=O)NC(C1CN(C(c2cn[nH]c(=O)c2)=O)CCO1)C)N(C)C Cc1cc(C(N2CCC(CO)(NC(C3CC=CCC3C)=O)CC2)=O)cc(O)c1 N1(CCNC(CCN(C)CC)=O)CCC(NC(C2CCOC2C)=O)CC1 C1(C(=O)NC(COC)CNC(C2CCC2COC)=O)CC2(C1)CC21CC1 c1(CCNC(=O)NCCc2cncs2)cc(Br)cs1 Cc1sc(C(F)(F)F)nc1C(=O)NC1CCN(C(C2CC2c2ccccc2)=O)C1 CCC(CNC(C1(c2ccccc2)CCN(C)C1)=O)(CC)NC(=O)CCCCl C1(C(=O)NCC2N(C(C3C(CC)CCC3)=O)CCC2)CCCCC(=O)C1 N1(C(Cn2c(C)ncc2)=O)CCn2ncc(CNC(=O)CN3CCCC3=O)c2C1 C1(CC(=O)NC2C(NC(c3ccn(C)c3)=O)C2)SC2=NCCN2C1=O N1(C(C2C(C(C)(C)C)CC2)=O)CCCC(CCNC(=O)C=Cc2cccs2)CC1 CC(C)C(CCC(=O)NCCC1CC(=O)N(C)C1)NC(c1ccc(O)cn1)=O CCC(O)CC(=O)NC(CCOCCO)C(=O)N1CCC(C(=O)NC)CC1 C(=O)(CCCC(F)(F)C(F)(F)F)NCC(CCNC(CC(C)C)=O)O c1(C(C(=O)NCC2CC2)N(CC(=O)NC)CCOC)ccc(OC)s1 c1(OC)ccc(CS(C)(=O)=O)cc1C(=O)NCc1cc(Br)cnc1OC c1(C(=O)NC(CCC)CNC(=O)Cc2csc(C)n2)c(C)nn(CC)c1C n1(CC)nc(Br)nc1C(c1nnnn1Cc1ccco1)NCCCc1nccs1 C1(C(N2CCC(C(C)NC(c3n(C(C)C)ncc3)=O)C2)=O)CC2(CCO1)CC2 C1(NC(Cc2c(C)occ2)=O)C2CN(C(=O)CC(C)C3CC3)CC12 N1(C(c2[nH]cc(CC)c2)=O)CCC2CN(C(C3CC3c3ccccc3F)=O)C2C1 CCC(CCC(=O)N(C(C)CC(C)CC)C)NC(c1ccn(C(C)C)n1)=O N(C1CSCc2ccccc21)CCn1nnnc1C(c1cnsc1)SC Cc1ccc(Br)c(C(=O)NC2CC(NC(=O)CC3CC(C(F)F)C3)C2)n1 C1(NC(CCN(C)CC)=O)C2CC3CN(C(C4CC(CC5CC5)C4)=O)C1C3C2 n1(CC)ncc(C(=O)NC2(CCC(N3C(CO)CC3C)=O)SCCS2)c1C N1(C(CN2CC(C)C2)=O)CCOC2CCN(C(=O)C(F)C3CC3)CC12 CCC(N=c1nc2ncn(C)c2c(NCC2CC23CC3)[nH]1)c1cccc([N+](=O)[O-])c1 C1(C(=O)NCC2N(C(CCC=C)=O)CC3(CC3)C2)Cc2c[nH]cc2S1(=O)=O CCCCC(CC)CC(=O)NC1(CNC(c2c(F)cc(C)cc2F)=O)CCCC1 C1(CN(C(=O)C(F)CC2CCOC2)C)CN(C(c2cc(F)c[nH]2)=O)CCO1 CCC(CC(=O)N1CCOC(CNC(=O)CCS(=O)(=O)NC)C1)C(F)F N1(C(C(CCCNC(C2(Cl)C(C(C)=O)C2)=O)O)=O)C2CCC1CC(F)C2 Cc1ncc([N+](=O)[O-])n1CC(N1CC(C)N(C(C23CC(F)(C2)C3)=O)CC1C)=O c1(CCC(N2CCC(CNC(Cc3n(C)ccn3)=O)C2)=O)nc2ncccn2n1 C1(C(=O)NCC(CC(C)C)NC(=O)CN=S(C)(C)=O)CC12CCC(C)(C)CC2 CCC(C)(C(=O)NCC(C(C)C)NC(C1CN(C(C)=O)C1)=O)C(N)=O C1(C#N)(C(=O)NCC(C)(C)CNC(=O)CC2C=CCC2)CC2CCC1CC2 C1(O)(C(C)NC(=O)CCCCC2CC2)CCN(C(=O)C(F)(F)C(C)O)CC1 N1(C(CC(CC)OC)=O)CC(NC(c2ccccc2)=O)CC2(CC2)C1 CCCC(C)(O)C(=O)NC1CCN(C2CCN(C(C3(C)CCCC3)=O)CC2)CC1 C1(N(C(c2ccn(C)c2)C(=O)NC(C)C)C)CCCCCC1F C(C(=O)NCC1(F)CCC(NC(=O)COc2cccc(Cl)c2)C1)(C(C)C)NC(C)=O N1(C(C=CC(=O)N2CCC2)=O)CCCC(C)C1.c1(CCCC)nc(CC)cs1 c1(OCC(=O)OC)cc(=NC(C)Cc2cccc(Cl)c2)[nH]c2ccc(Cl)cc12 CCCC(C)(C)CC(=O)NC(C)C(C)NC(=O)CSC(F)F c1(C(=O)NC2CCC(CNC(CNC(=O)NC)=O)CC2)cnn2cc(C)cnc12 c1(OC)ccc(CCC(=O)NC(C)CC(C)NC(=O)C2=NNC(=O)C2)cc1C Cc1nc(S(=O)(=O)NCC(=O)NCC=CCNC(C2CCC2(C)C)=O)cn1C N1(C(C(C(CC)C)NC(C)=O)=O)CC(=O)Nc2c(C#N)cccc21 N1(C(c2c(C)cccn2)=O)CCC(NC(=O)C=CC2(C)CCOCC2)C(C)(C)C1 N1(C(c2c(C)nn[nH]2)=O)CCC(F)(F)C(CNC(c2c[nH]c3nccc-3c2)=O)C1 C=C(Cl)CC(C(=O)NC(c1ccccc1C)C)NC(=O)C=C(C)C(C)(C)C c1(C(=O)NCC(CNC(c2c(C)cn(C)c2)=O)C)ccc(Br)c(Cl)c1F C1(CNC(c2cc[nH]n2)=O)CCN(C(C2CC(n3cccn3)C2)=O)CCC1(F)F CC1CC(NC(c2cn3ccsc3n2)=O)CCN1C(=O)CN1CCCOC1=O C(=O)(CCC(=O)NCC1CCC1NC(=O)C(C(C)O)N(C)C)NCCC Cc1nn(C)cc1CCNC(=O)C(C1(C)CC1)NC(c1ccccc1)=O c1(Nc2nccc(N(C)CC)n2)cccc(OC2CCCCC2)c1Br c1(CC)ccc(C(=O)NC(CO)C(=O)N2CCC2(C)CNC(C)=O)o1 Cc1cccc(CC2CC2)c1NC(c1c(C#N)cnn1-c1ccccc1Cl)=O c1(C(=O)NC(CCCNC(c2occ(C)c2)=O)C)[nH]c2ccc(Cl)cc2c1Cl c1(NC2CCC(CCNC(C3CS(=O)(=O)C3)=O)C2)cnc2ccccc2n1 N1(C(C(C)CF)=O)C2CCCC1CC(n1cc(C(O)Cc3ccccc3)nn1)C2 c1(CC)cnc(C(N2CC(CC(=O)NCCCN(C)C3CC3)C(C)C2)=O)nc1 C(C)(CC(=O)NC)NC(c1nnc(NC(CCC2CC(CC)C2)=O)o1)=O C=CCC(C(=O)NCCN(CC(C)O)C(=O)Cc1cnc(C)s1)C(C)C c1(C(C2CCSC2)C2CC2)nnnn1C1CCC1.C1(CCO)(N)COC1 O=C(C1=CCC(F)(F)CC1)NC1CCCCCN(C(c2nncn2C2CC2)=O)C1 C(=O)(C1COc2ccc(F)cc21)NCC1CCCN(C(c2ccc(C)o2)=O)CC1 CC1=CCC(NC(c2cn(C)nn2)c2nnnn2C2(C)CC2)CC1 C#CCC(C)(CNC(=O)CC1(NC(=O)C(C)S(C)(=O)=O)CCOC1)CO C(=O)(C#CC(C)(C)CNC(C1CCC(=O)O1)=O)NCC1CCC(C)C1 N1(C(Cc2cc(C(=O)OC)n(C)c2)=O)CCCCCC1CNC(=O)COC(F)F N1(C(C2C(=C)CC2)=O)Cc2ccccc2OC2(C1)CN(C(=O)COCCF)C2 n1(CC(=O)NC2(c3ccc(OC)cn3)CC2)cnc2ccccc2c1=O C1(O)(CN(C(CC(=O)OC)=O)C)CCCN(C(C2COC3CC2C3)=O)C1 C1(C(N2CC3CCN(C(C4CC=CCO4)=O)C3C2)=O)CCn2nnnc2C1 c1(C(CCC)NC(c2n(CC(=C)C)nnn2)C2CC2)c(F)ccc(F)c1Br N1(C(C(C2CCCN(C(c3cc4n(n3)CCC4)=O)C2)C)=O)CC2C=CC1CC2 c1(C(N2CCC(NC(CC3CC(=C)C3)=O)C2C)=O)ccc(Br)cc1NC C1(C)(OC(C)(C)C)CN(C(=O)CCCNC(=O)N)C1.C(CC(=O)OCC)=CC=C CC(C)C(C)C(=O)NCCC(C)N(C)C(C1CC1(Cl)Cl)=O c1(C(N2C(CNC(CN3CCC(NC)CC3)=O)COCC2)=O)cnc(C)cc1Cl C(C)(CN=c1nc(-c2ccccc2)nc(N2CCC(c3nncs3)C2)[nH]1)SC C1(NC(c2nn(CC)c(O)c2)=O)CC2(C1)CC(NC(C1CCOCC1(C)C)=O)C2 C1(CC(N2C(C(=O)NCCC(COC)O)CCC2)=O)CC2(CCC2)C1 CC(=O)CCN=C(NCC(F)(F)CO)NC(c1ccccc1F)CF c1(C(=O)NC2COCCN(C(C(CCC)CCC)=O)C2)ccc2c(n1)COCC2 C(=O)(CS(=O)(=O)NC=O)N(C(c1nc(NCC)sc1)=O)C.CCCCC(=O)N(C(C)CN)C C(=O)(CC(C)(C)C(C)(F)F)NC1C(C)CN(C(C2CC3(CC(C)=NO3)C2)=O)C1 N1(C(c2c(N)cc(Br)cc2)=O)CC2CCC1C(NC(C1CC1(F)F)=O)C2 N1(C(Cc2c(C)non2)=O)CCC(C(F)(F)F)C(NC(=O)Cc2cn(C)nn2)C1 C#CC(CC(C)C)NC(C1CCN1C(=O)C(O)C=C)=O c1(NC(COC2(C)CN(C(C(CC)=CCCC)=O)C2)=O)ccc(F)c(F)c1 C1(C(=O)NCC)C(C)CCN1C(c1ccc(CCOc2ncccn2)cc1)=O C1(Cl)(C(=O)OC)CC1C(=O)NCC1(NC(=O)COCC(F)(F)F)CC1 C(=O)(CC1C(=O)Nc2ccc(Cl)cc21)N1CCC(NC(CC=C)=O)C(C)(C)C1 CC1(C#N)CCN(C(C2(F)CCCN(C(C3CCC(CO)CC3)=O)C2)=O)C1 CC(C)C(F)(CNC(=O)CC1COC(=O)C1)C(=O)NCC1CCSC1 C1(C(N2CC(C)(NC(CCNC(COC)=O)=O)C2)=O)CCC2CC2C1 CCCCCC(=O)NC(C(=O)N(C)Cc1ccco1)C1CCCC1 C1(NC(c2cc(C)n(C)n2)=O)(CNC(=O)CCN2CCOCC2)CC2CCC1C2 Cc1c(C(=O)NCC2(C(=O)NCCc3cnc[nH]3)CCCO2)cncc1F n1(CC(=O)NC2C(NC(=O)CC3CC3(Cl)Cl)CCCC2)ccc(=O)c([N+](=O)[O-])c1 C1(C(=O)NC2CC(C(=O)Nc3c(C(=O)OC)nsc3)C2)CCC2(CC1)CC2 Cc1oc(C)c(C(N2CCOC(C(=O)Nc3cccc(O)c3)C2)=O)c1C C(=O)(C(CNC(c1ncccn1)=O)CC1CCCC1)NC(c1ccncc1)C N1(C(CC=CC)=O)CCCN(C(c2ccc(C)cc2CC)=O)C(C)C1 Cc1noc(CCCN(C2CN(C(c3ccccc3)=O)C2)C(c2ccco2)=O)n1 C1(C(=O)NCc2ccco2)CC(O)CN1C(=O)CCc1nncs1 c1(C(C)C(=O)NCC(C2CCCC2)NC(=O)C(C)CN(C)C)cccc(Cl)c1 C12(CCCC)CCN(CC1)C(=O)O2.C(CCCC1CCCC1)OCC N1(C(C(CCC)OCC)=O)CC(C)CN(C(C2C3CCC4C(C3)CC24)=O)CC1C c1(OC)cc(C(N2CC(NC(=O)CC(C)C)CC(C)(C)C2)=O)cc(OC)c1OC CCC(CC(=O)NC1CC(C)(C(=O)NC(C)CCC(C)C)C1)SC Nc1c(C(N2CC(NC(=O)Cc3ccc(F)cc3)C(O)C2)=O)ccnc1Br c1(NC(CCCN(C)C(C2CCCCNC2=O)=O)=O)cccc2c1OCO2 c1(NCCCCC(C)O)ccc(S(=O)(=O)NCCCCC(N)=O)cc1Cl c1(OC)cccnc1C=C1CCN(CC(F)(F)F)CC1 C(C(CNC(C1(C)CCOC1)=O)S(C)(=O)=O)NC(C=Cc1ncc(C)[nH]1)=O N#Cc1cc(CN2CCCC2CC(=O)Nc2ncc(I)cc2Br)ccn1 c1(C(N2C(CN(C(=O)C(F)F)C)CCC2)=O)ccc(Cl)c(Cl)c1 C(c1ccc(C)o1)=CC(=O)NC1(CC=C)CN(C(=O)Cc2ccccc2C)C1 c1(OC)cnc(C(N2CCOC(NC(=O)C3CC3)C2)C(=O)NC2COC2)nc1 C1(C)(CNC(c2nnn(CC)n2)=O)CCCN(C(=O)C=C2CCCCC2(C)C)C1 Oc1cccc2[nH]cc(CNC3(c4ccc(O)cc4)CCC3)c12 CCCC(CCC)CC(=O)NC1CN(C(=O)C(CC)C2N=N2)C2CCCCC12 C1(NC(C2(CNC(c3ncccc3O)=O)CC2)=O)CC12CCCC2 C1(CC)(CO)CCN(C(=O)C(N)=O)C1.C12CC13CC(C3)NC2=O C1(NC(C(C)OCCC=C)=O)COCC1NC(c1ccc(CC)[nH]1)=O c1(C(=O)NC2C(NC(C(CC)(C)CC)=O)CCCC2)cccc2nc(O)ccc12 CCC(CC(=O)NC(C1CCCCC1)C(N1CC(F)(C#N)C1)=O)C1CC1 O=C(C1=Cc2cc(Br)ccc2OC1)Nc1c(C(=O)O)cnc2c1cnn2C(F)F c1(NC(c2ccc(Br)o2)=O)ccc([N+](=O)[O-])cc1 CC1C(C(N2CCOCC(CO)C2)=O)CCCN1C(C1CC=CCC1)=O Cc1cnc(C=CC(=O)NC2CC(OC(=O)OC(C)(C)C)CC2SC(C)C)[nH]1 N1(C(CSC)=O)CCN(C(=O)C(C)Cc2cnc[nH]2)C(CC(C)(C)C)C1 Cc1ccc(OCCC(=O)N2CC(CNC(C3(C)CC=CCC3)=O)C2)c(C)c1 c1(C(N2CCC(F)(CNC(C3(CC)CC3)=O)C2)=O)cnc(OC)c(Cl)c1 N1(C(C2(C(C)C)CCCC2)=O)CCC2CCCC(C1)N2C(c1ccncc1Cl)=O Cc1cc(NC2CC3CN(C(c4coc(N(C)C)n4)=O)CC23)ccc1[N+](=O)[O-] C1(C(C)C)CN2CC1C2=O.C1(O)(CNC(CO)C2CCC2)CN(C)C1 C(=O)(C1CCOc2ccccc21)NCC(C(C)C)Oc1cc(Cl)cc(Cl)c1 c1(OC)cccc(C(N2CCC3C(NC(=O)CCC(C)SC)CC23)=O)c1F Cc1ccc2c(c1)CN(C(C1CC(F)CN(C(=O)CCN(C)C)C1)=O)C2 c1(N(C(c2ccc(Cl)nc2)C(=O)NCCOC)C)cccc(Br)c1C N1(C(C(c2cscn2)N(C)C)=O)CCC(O)C(C(=O)NCCC2CCOCC2)C1 N1(C(=O)COCc2nc[nH]n2)CCC2(CCCCN(C(c3ccsn3)=O)C2)C1 c1(C(N(CCOCCN(C(CCCC=C)=O)C)C)=O)ccc2ccoc2c1 O1NC(=O)C(C)(CC)NC(=O)C1CC(C)C.C1(CC)CC1CN(C)C N1(C(C2C(C)=C2)=O)CCC(NC(c2nc(Br)sc2C)=O)C(O)C1 C1(C(N2CC(NC(CCC)=O)C2)=O)CCCCC1.C1(NC(C)=O)CCS(=O)(=O)C1 C1(NC(C(C)N(C)C)=O)CCCC(NC(c2ccc(-c3cccs3)cn2)=O)C1 c1(C(=O)NCC(COC)NC(=O)C(C)C)ccc(OC(C)C)nc1 C(=O)(C(C)C(C)C(C)(C)C)NCc1nc(CNC(c2cccc(OC)c2F)=O)sc1 C1(NC(c2c(C)cncc2)=O)Cc2ccccc2N(C(=O)Cc2ccc(Cl)s2)C1 CC1CSc2ccccc2CN1C(c1cc(F)c(Br)cc1F)=O c1(N(C(=O)CC2(N)CC2)CCCN(C)CC2CC3CCC2O3)cc(O)nn1C c1(OC)cc(C(=O)NCC#CCNC(=O)CNc2ccccn2)c2c(c1)CCC2 CC(C)(C)C(CNC(=O)CC1CC1)C(=O)N1CC(O)(CO)C1 C1(NC(CC2(CC=C)CCCC2)=O)CC2(C1)CN(C(C1(C)CCCC1C)=O)C2 C1(C(=O)NC(C2CCCCC2)CC)N(C(c2cc(C#N)c[nH]2)=O)CCCC1(C)C c1(C(=O)NC(CCCC(=O)N2CCC(CCCC)C2)C)cnn2ccccc12 C12(NC(CNC(=O)OC)=O)CCCC1CN(C(=O)CCN1CCOCC1=O)C2 c1(NC(CN(C)C(CC(=O)O)=O)=O)ccc(-c2cn(CC(C)(C)C)nn2)cc1Br CC(N=c1[nH]c2cc(Cl)cc(F)c2s1)C(c1ccccc1)c1nnnn1CCF N1(C(C(C2CN(C(c3c(C)nn(C)c3C)=O)C2)OC)=O)CC2(C1)CN(C)CCO2 c1(C(=O)NCC(c2ccccc2)NC(CCOC(C)C)=O)cc(N)c(Cl)c(O)n1 C(C(C)C)(C(O)C(=O)NCC1CC(O)CN1C(C1CCC(C)(C)C1)=O)OC C1(C(=O)OCC)C(C(=O)NCc2nncn2C)C12CC2(F)F c1(C(=O)NCCN(CCC)C(c2csnc2OC)=O)cc(Cl)cc(C)c1N C1(C)(CNC(C(F)=CCC)=O)CC(OC)CN1C(c1cnc(C2CC2)nc1)=O C1(CCNC(CC(C)n2ccnc2)=O)CN(C(=O)Cn2ccccc2=O)CCO1 C1(CC)CC(C(=O)NC(C(=O)NCCO)C2CCCO2)C1.C1C(=O)N1 CN1C(=O)CC(C(=O)NCC2(CO)CCN(C(c3cnc(Cl)s3)=O)C2)C1=O N1(C(C(CCC)NC(C)=O)=O)CCC(NC(c2sccc2CC)=O)C12CCC2 Cc1cnc(NCCSCCO)c(S(=O)(=O)N2CCCC(C)(C(F)F)C2)c1 C(=O)(C1CCCc2nccn21)N1C2(CNC(C(C)CC3CCCC3)=O)CC(C1)C2 c1(CNC(C)(C)CNC(c2csc([N+](=O)[O-])c2)=O)cccn2ccnc12 c1(C(C)=O)cc(C(=O)Nc2cccc(NC(c3cnn(C)c3C)=O)c2)ccc1F c1(C(=O)NC(CC)CNC(C2CC(OC)(OC)C2)=O)cc(NC)cc(F)c1 c1(C(=O)NCCCCNC(C=CSC)=O)scc(C)c1OC C1(CNC(CC2C(C)CCO2)=O)CCC(C(=O)NC(C)C(=O)OC(C)C)CC1 c1(C(N2CCN(C(c3c(OCC)c(Cl)ccc3)=O)CC2)=O)cc(N)c(C)cc1C N1(C(C(C(=O)OC)C)=O)CC2CC1CN(C(c1c(F)ccc(OC)c1OC)=O)C2 C12(C(N3CC(COC)(CNC(C4CCOC4C)=O)C3)=O)C3C4C1C1C2C3C41C#N c1(CC(=O)NC2C(NC(Cc3ccn(C)n3)=O)C2)ccc2c(c1)CCCS2 N1(C(c2cc(OC)c(F)c(C)c2)=O)Cc2nccn2CC(NC(=O)C2CC2)C1 C1(C(N(CC)CC2CCCN(C(c3ccc[nH]3)=O)C2)=O)CN(C)C(=O)CCO1 c1(C(C)=O)ccc(C(=O)N(C2CC3CCC2C3)CC2CC2)cc1 N1(C(C(CCSC)NC(Cc2ccn(CC)n2)=O)=O)CCC(F)(F)C(F)C1 c1(CC)cc(NC(=O)C=CCN(C(=O)C(C)C(=O)OC)CC)ccc1F C(=O)(CCCCOC)NCCN(C(=O)C(F)C1CCCC1)CCC c1(C(=O)NC23CCC(CNC(CC(CC)C)=O)(OC2)C3)ccnn(C)c1=O c1(OC)ccc(O)c(C(N2CCN(C(=O)CC3(C)CCCO3)CC2C)=O)c1 N1(C(c2c(CC)ccs2)=O)CCC2CC2(NC(c2snnc2C2CC2)=O)CC1 C1(C(=O)NC(CC)(CNC(C2C3CCOCC23)=O)CC)CCCC(C)(C)C1 C1(C)(CNC(=O)C=CCOC)CC(OC)CN1C(c1cnc(C)o1)=O c1(SCC)ccc(C(N2CCC(CCNC(c3sccc3OC)=O)CC2)=O)cn1 c1(C(=O)NCCCNC(c2cc3occc3s2)=O)ccc2n[nH]cc2c1 C1(O)(CC)CCCN(C(C2(C)CCCN(C(=O)CC(C)(C)OC)C2)=O)C1 C1(C)(CNC(c2c(CC)n[nH]c2)=O)CN(C(c2[nH]cnc2C)=O)CCO1 N1(C(c2cn(C3CC3)nn2)=O)CCC2CN(C(C3CCS(=O)CC3)=O)C2C1 N1(C(c2c(C)cc(N)cn2)=O)CC(NC(c2ccccn2)=O)CC(C)(C)C1 C12(CNC(C(C)OCCC=C)=O)CC(NC(=O)C(C)N(C(CC)CC)C)(C1)C2 c1(C(=O)NC2CCC(CNC(c3n(CC)ncn3)=O)C2)cccc(Br)c1F c1(OC)cc(C(=O)N(CC(C)CNC(=O)CN(C)CCOC)C)ncc1Br C(CC(=O)NOC1CCCCC1)N(C(C(C1CCOCC1)C)=O)CCO N1(C(c2cc(CC(C)C)on2)=O)CCC(O)(CNC(c2cc(F)cs2)=O)C1 c1(CCNC2C3(CC(OCC)C3)C2)cn(C)c2c(C)cccc12 N1(C(COCCOC)=O)CCOC(C(=O)NCC(C2CCCC2)O)C1 Cc1c(C(=O)NCc2ccc(C(=O)NCCC3(C)CC3(F)F)o2)cccc1O Cc1cccnc1CCC(=O)NC(CNC(=O)C(C)n1cccc1)C1CC1 N1(C(c2c(C#N)ccs2)=O)CCN(C(C2C3CCC4C(C3)CC24)=O)C2COCC12 C1(NC(=O)CN2CC=CC2)COC2(CCN(C(C3CCS3(=O)=O)=O)CC2)C1 N1(C(CC2CN(C(c3cc(C)c(O)cc3)=O)C2)=O)CCc2cccnc2C1 N1(CC(=O)NC2CCCC2)CCN(CCC(F)(F)F)CC1 c1(C(=O)Nc2ncc(-c3ccc(C)cc3)nc2)nccc2occc12 C1(O)(C(C)C)CCCN(C(C2CC(NC(c3cc(C(N)=O)[nH]n3)=O)C2)=O)C1 c1(CC(=O)NCC(CCCC)NC(C=CC=CC)=O)c(C)nc(C)nc1O N1(C(CCOC(C)C)=O)CC2CCN(C(=O)Cn3nc(Cl)ccc3=O)CC2C1 N1(C(c2nn(C)c(F)c2)=O)CCC(NC(c2cc(C#N)c[nH]2)=O)C(F)C1 C1(C)(CC(=O)NC2C(NC(C3(CN(C)C)CC3)=O)COC2)CCCCC1 C1(CNC(CCCC)=O)CCC(C)CN1CCn1ncc(C(=O)OCC)c1C C1(NC(C2CCC(CC)CC2)=O)CC(C)CN(C(c2csc(C)n2)=O)C1 C1(C)(C(=O)NC(C(C)NC(c2c[nH]nc2-c2ccn(C)n2)=O)CO)C=CCCC1 Cc1cc(N)c(C(=O)NCC2CCN2C(C2CC(C)OC2=O)=O)cc1C Cc1c(CO)cccc1COC(C1COC2(CN)CC1C2)=O c1(C(C)C)ccccc1C(N1CCC(C)(NC(=O)CCC(C)N(C)C)C1)=O C1(NC(c2cnc(C)n2C(F)F)=O)CCN(C(c2c[nH]c(=O)cn2)=O)C(C)C1 CC1CN(C(=O)CCN2CCCC2)CC(C)CN1C(C1CCCC(F)C1)=O c1(C2N(C(C)C3CC3)CC2)ccccc1Br N1(C(C2CC(C)(O)C2)=O)CC(F)CC1CNC(=O)C=CI N1(c2ccc(C(=O)OC)cn2)CCCCN(S(C)(=O)=O)CC1 c1(C(C)C)ccc(NC(C2CC3CC3N2C(=O)C(=O)N(C)C)=O)c(Cl)n1 c1(CCNC(=O)NC23CC(C)(C2)OC3(C)C)ccc(S(C)(=O)=O)cc1 c1(C(=O)NOCc2cc(Br)ccc2C(F)(F)F)cc(Br)cc2cc[nH]c12 Cc1cnccc1C(C)C(=O)NCC1(NC(=O)OC(C)(C)C)CC1 C(C(C)CC(=O)N1CCCCC1CCCO)NC(CCn1c(C)ncc1)=O NS(=O)(=O)CC(=O)NC1(CO)CCN(C(=O)CCC2CNC(=O)N2)C1 N1(C(CC2CC(=O)C2)=O)CCC(NC(C2CC3COCC3C2)=O)C2(CCC2)C1 C#Cc1ccccc1CC(=O)NC1CCCC1NC(=O)CCCC(C)C S(=O)(=O)(c1cc(Br)c(F)cc1F)N1CCC(C(=O)NCC2COCCO2)C1 c1(C(N(CC=C)C2CC2)=O)ccc(Cn2cc(CC(C)(C)O)nn2)cc1 N1(C(c2c(OC)cccc2)=O)CCC=C(C(=O)NC2CS(=O)(=O)CC2O)C1 C1(C(N(C(C(=O)N(C)Cc2cn(CC)nc2)C)C)=O)CN(C)C(=O)N1 C(=O)(C(O)CC(C)C)N1CC2C(CCC(N(OC)C)=O)C2C1 C1(NC(C2N(C)CCC2)=O)CCCCC12CCN(C(=O)C#CC1CCOCC1)C2 C1(C)(C(=O)NC(C(C)NC(c2ccc(CO)s2)=O)CO)CCOC1C C(=O)(C(=O)Cc1cccs1)NC1C(NC(C=CCOC)=O)C1 C1(NC(c2ccc(-n3ccc(C)n3)cc2)=O)CCN(Cc2ccsc2)CC(O)C1 C1(CNC(c2n(CC#C)ccc2)=O)CCCN(C(=O)C(C)(C)C2CCCO2)CC1 N1(C(C2CC(=O)NC(=O)C2)=O)CC2CCN(C(=O)C#CC3CC3)CC12 C1(C(=O)NC2C(NC(c3cc(C)sn3)=O)C2)CCCCC12CC2 C1(C(N2CCC(NC(C)=O)CC2)=O)CC(F)(F)CN1C(=O)Cn1[nH]cnc1=N N1(CC)CCN(Cc2ccc(Br)c(OC)c2)CC12CCOC2 C1(NC(C(CCC)F)=O)CCN(C(=O)C(C)OC2CCCC2)CC1F C(C(C)N=c1nc(N(CC(C)C(=O)NC)C)c2c([nH]1)CCOC2)OCC CC1(C=CC(=O)NCCCN(C(=O)C=CSc2ccccc2)CCO)COC1 n1(CC)nc(C(=O)NC(CO)C(C)NC(=O)CCc2ncccn2)cc1C1CC1 CCCC(C(=O)N1CC(N(C)C)C(CNC(=O)C(F)CC2CCOC2)C1)N(C)C C1(NC(c2c(C)cc(CC)o2)=O)C2CC1CN(C(c1ccsc1CC)=O)C2 CC1(CNC(c2nccnc2N)=O)CN(C(C2CCOCC2)=O)CCO1 C1(C(=O)NCc2c(C)scn2)CCCN(C(=O)Cc2ccc(F)nc2)C1C C1(C(=O)NC23CC(CNC(C4(F)CC=CC4)=O)(C2)C3)CC2CCC1O2 CCC(CCC(=O)NCCOC1CCC1)NC(=O)C(C)n1ccnc1 C(CN=c1[nH]c(N2CCC(Cl)=C(Cl)C2)nc2c1COC2)N1CCN(C)CC1 CCC(C)C(O)C(C)C(=O)NCCC(C(=O)N1CCC(CCO)C1)OC CC1CC=C(C(=O)N2CCCC(C(N(C)CC34CCCCC3C4(F)F)=O)C2)CC1 N1(C(C2CC(NC(c3ccoc3)=O)CC2O)=O)CCC(O)(CO)CC1 c1(C(N(C2CCN(C(=O)CC34CCCC3C4)C2)CC)=O)ccc(C)c2c1CCC2 c1(N2C(=O)CC(C(=O)NC3(C)CC3)C2)ccc(F)c(Cl)c1.C12CCN(CC1)C2 C1(NC(C(CCC)(C)C)=O)CN(C(c2n[nH]cc2Cl)=O)C2(CCCOC2)C1 C(=O)(CC(O)C(Cl)(Cl)Cl)N(C)CCc1cn(C2CCCCC2(C)O)nn1 c1(N(C2CCN(c3cc(C)ns3)C2)C)cc(COC)cc(C)c1 c1(NCC2C(C)CN(C(C3CC4OC3C3CC43)=O)C2)ncnc2ccc(F)cc12 N1(C(C(CC)C#N)=O)CCCC(C)(NC(c2cn(C(C)C)nc2Br)=O)C1 c1(CC(=O)N(CC(C)NC(c2c(C)oc(Cl)n2)=O)C)ccc2c(c1)CCCS2 N1(C(C2CN(C(C)C)C2)=O)CCC(NC(=O)CC2COCCN2C)C(CO)C1 C1(N(C)C)CC2CC1CN2C(=O)Nc1ccsc1.C12CCN(C1)C2=O C(=O)(C1=CCCCC1)N1CCC(C(=O)NC(C)CCSC)(OC)C1 c1(OCCC(=O)NC2CC2NC(c2ccnc(C3CC3)c2)=O)ccccc1F C1(NC(CCCCOC)=O)CCN(C(c2cnoc2-c2cccs2)=O)CC1C c1(CN2CC(C(=O)OC(C)(C)C)OCCC2)cn2cccc(Br)c2n1 N1(C(c2c(C)nco2)=O)CCC(C(=O)NC(C(C)C)C2CC2)C12CCC2 CCCCCC(C)(CC)C(=O)NC1CC2CCC1N2C(c1c(C)coc1C)=O S(=O)(=O)(c1cc(C(=O)NC2CC(NC(C3CCCC34CC4)=O)C2)ccc1C)NC C1(CNC(c2ccn(C(F)F)n2)=O)CN(C(C2CCC(C(F)(F)F)O2)=O)CCO1 N1(C(C2N(CC)CCC2)=O)CC(C)CCC1CNC(c1csc(C)c1)=O C(c1cccc(F)c1)=CC(=O)NC1C(CNC(CCCOCCC)=O)C1 N1(C(c2n[nH]c(C)c2Cl)=O)CCC2CCC(NC(c3ccoc3)=O)C1C2 N1(C(C(C(C)C)O)=O)CCC2(NC(C3CC4(CCCCO4)C3)=O)CCCC12 C1(C(=O)NCCCCCNC(c2csc(-c3cnc[nH]3)n2)=O)CCCC12CCC2 C12(CNC(c3ncn(CC)n3)=O)CCC1CCN2C(=O)CCCn1ccnn1 CCCS(=O)(=O)C1CN(Cc2ccc(N3CCCC(O)C3)cc2)C1 CC(C)C(C(=O)NCC1CCCC1NC(=O)CS(N)(=O)=O)N(C)C c1(N(C)Cc2cscn2)nc(NCC2(C)CC3CC3C2)c2ccsc2n1 C1(C(c2n(CC=C)nnn2)NCC(C)(C)n2ccnc2)(CC=C)CCOCC1 Cc1[nH]c2ccnn2c(=O)c1CC(N1CCC(N(C(=O)C(F)C(C)(C)O)C)C1)=O C(=O)(CC(C)C(=O)N(CCC(=O)NCC1=CCCC1)C(C)C)OCC C1(C(N(CC(=O)N(CC(C)C#N)C)C2CC2)=O)CCC(C)(C)C1 C(CC(=O)Nc1cc(C)cc(C(N)=O)c1C)(C(F)F)NC(C(CC=CCC)C)=O N1(Cc2n(CC)ncc2)CC(C)C(Nc2nc3cccnc3s2)C(C)C1 c1(C(N(C)CC2CCCCN2C(C2CCCOC2)=O)=O)cc2ccc(F)cc2[nH]1 C(=O)(C(O)C1=CCCCC1)NCC1C(CNC(c2nn(C)c(Cl)c2)=O)C1 N1(C(C2C(CNC(c3cc(C(C)=O)on3)=O)C2(C)C)=O)CCC2(CCC2)C1 n1(CC(=O)NC2CC(CNC(C3CC(=O)N(O)C3)=O)C2)nnc2ccccc12 CC1(C)CN(C(c2cnn[nH]2)=O)CC1CNC(c1cn(CCC2CC2)nn1)=O c1(C(=O)NCC2CCC(NC(C3C(C=C)C3)=O)CC2)ccc2nsnc2c1 C(=O)(CC(C(F)F)c1cccc(F)c1)N1CCCC(NC(c2cn[nH]c2)=O)C1 c1(CN(C)CC2CCCN2C(=O)C(C2CCCCC2)=O)ccc(C(F)(F)F)cc1 C1(CNC(c2cnsn2)=O)CC(F)CN1C(=O)CCN1CCC(F)C1 C(=O)(C#CC1CCCCC1)N(CC(C)NC(=O)CCc1ccc(Cl)nc1)C c1(SC)cc(C(=O)NC2CCC(CCNC(=O)CSC(C)(C)C)C2)ccc1N c1(C(=O)NC2CC(NC(C3C(C)CCS3)=O)C2)ccc2c(c1)CCS2(=O)=O N1(C(C2(C#C)CCCCC2)=O)CCC2(CC1)CC2C(=O)NC1(C)CCC(C)C1 N1(C(c2ccc(NC)cn2)=O)CCC(NC(c2cnnc(C)c2)=O)CC(C)(C)C1 C1(O)(C(C)NC(C(F)=CCC)=O)CN(C(=O)COc2cc(C)on2)C1 c1(CNC(=O)N(C(C)C(c2ccccc2Cl)O)C2CC2)cccc2nc(O)oc12 c1(C(=O)NC2(CNC(C3CCC(C)CC3)=O)CCOC2)cc(F)c(F)c(F)c1N C(C)(CCCC(=O)NC1CC(n2cccn2)C1)NC(C1N(CCC)CCC1)=O C#CC1(C(=O)Nc2cnccc2N(C)C)CCN(C(C2CCCCNC2=O)=O)C1 C1(N(CC#C)C(C2(C)CC=CCC2)=O)CCN(C(c2c(C)csc2Cl)=O)CC1 N1(C(C2(N(C(C(NOC)=O)=O)C)CC2)=O)CCS(=O)CC1C N1(C(C2CCCN(CCC)C2)=O)CCN(C(=O)CCCSC)C2COCC12 O=C(NNc1cccc(Cl)c1)C(=O)c1c(O)cccc1Cl C(=O)(N=c1[nH]nc(C2CC2)s1)NCCC(C)NC c1(CCC)nc(-c2ccc(SC(C)C)cc2)n(C2CCCC2)n1 C1(=CC(=O)NC2(CO)CCN(C(c3cccc(Cl)c3)=O)C2)CN2CCC1CC2 C1(CNC(=O)CN2C(=O)CCCC2=O)CC(NC(c2sccc2Cl)=O)C12CCC2 C1(CC)CCCN(CC(=O)NCC(C)(C)NC(c2ccc(C3CC3)o2)=O)C1 C(C)(CCS(C)(=O)=O)NC(N(CCCN)C)=O.CO N(C(=NCCN1CCCC1)NCC1(C)CC1(C)C)CC1(CC)CC1 CC1(C)CC(C(=O)NC2CCC(NC(C3CC(O)C3)=O)CC2)=NO1 N1(C(C=Cc2n(C)cnc2)=O)CCCC2(NC(=O)CCS(N)(=O)=O)CC1C2 N1(C(C(CC(C)C)ONC(=O)COc2ccsn2)=O)CCCC2COCC12 C(=O)(CCCCNC(C12CC(n3cc(CCN4CCSCC4)nn3)C1C2)=O)OC c1(C(N2CC(C)(NC(=O)NCC(=O)OCC)C2)=O)ccc(Cl)c(C#N)c1 c1(CN2CC(C)(C)C2)ccc(F)cc1NC(C(=O)OCc1ccccc1)=O C1(C(c2ccccc2)=O)CCCN(CCC(N2CCC(SC(F)F)C2)=O)C1 CC1CN2CCN1CC2C(=O)NC1COCC1NC(c1cnc(O)o1)=O N1(C(C(C)C)=O)CCCC(C)(C(=O)N(C2CCC2)C2CCC2)C1.C(C)ON CCC(C)(C)C(=O)NC(C)CN(C)C(c1ccnc(OC)c1)=O Cc1ccccc1C=CC(=O)NCC(O)C(N1CCCC(CCCO)C1)=O CCC(C)CC(CC)(c1nnnn1C1CC1)NCc1ncnn1-c1ccccc1 c1(CC(N2CCCC(NC(c3cccc(NC(C)=O)c3)=O)C2)=O)cccc(Br)c1F c1(CNC(=O)NC(Cc2cccs2)C(=O)O)c(O)ccc2ccccc12 C(=O)(CC(CN(C)C)C(F)F)NCCC(C)NC(c1cccnc1C(F)(F)F)=O CCCC(CC)C(=O)N1CCCC(NC(=O)C=CC2(C)COC2)C1 C1(CCC)(C(=O)NCC(C)NC(c2ncccc2SC)=O)CCNC1=O CCC(C)CCCCC(=O)N1CC(NC(c2ccnnc2S)=O)CC1(CC)CC c1(SC)c(C(N2CCOCC(C)(CNC(C3(CF)CC3)=O)C2)=O)sc2ccccc12 C1(NC(C=CC(=O)N(C)C)=O)C2CC1N(C(=O)Cn1cnccc1=O)C2 C(=O)(N1CC(C)(O)CO1)C1(CNC(c2cc(COC)no2)=O)CC(=C)C1 c1(CN(c2cc(OC)ncn2)C2CNCC2F)c[nH]c2cc(F)cc(F)c12 c1(OC)ncccc1S(=O)(=O)N1CCOCC1CNC(c1cc(C)c(Br)s1)=O C1(CC)CCCC(c2nnnn2-c2cccc(OC)c2)(N(C)CC2(C)CCC2)C1 c1(C(=O)NCC2N(C(c3nc(N(C)C)oc3)=O)CCC2)c(F)cccc1F c1(C(=O)NCCN(C(C(CCCC)O)=O)C(C)C)cn(C)c2c(cnn2C)c1=O CC1CCCN(C(=O)CCOc2cccnc2)C1CNC(=O)C1=COCC1 Cc1cc(C(N2CCCC(CN(C(=O)CCNC(=O)CO)C)C2)=O)c(O)c(C)c1 Cc1ccc(NC(=O)CC2(C)CCN2C(c2cnco2)=O)cn1 CN(C1CC(F)(F)C1)N1CC2(CCCC2)CC1C(=O)OC N1(C(C2C(C)(C)CCO2)=O)CC2CC(C1)CN(C(c1ccnn3ccnc13)=O)C2 Cc1csc2ccc(CC(=O)NCC(C)CNC(C3(C)CCC(=O)NC3)=O)cc12 C1(N(C)C(c2cc(CNC(C3CCCS3)=O)[nH]n2)=O)CCC(N(C)C)CC1 c1(CNC(C(C)NC(=O)CN(C)CCO)=O)cnn(C(C)(C)C)c1 CC1CN2CCCN1N1CC3C(C3C1)N(C)C(=O)CC2=O.C(=O)CC1(C)CC1.N(C)C c1(C(N2C(C)CCC(NC(C(CC)(F)F)=O)C2)=O)ccc2c(c1)NC(=O)CO2 C1(C(=O)NC2C3CN(C(C4(F)C(C)C4)=O)C2C3)CCc2ccccc2C1 c1(C(C(=O)NCCN(C(=O)C(C2CC2)SC)CC)(F)F)ccccc1Br c1(CC)ncc(CNC(c2conc2CC(=O)NCC2(n3ccnn3)CC2)=O)s1 C12(C(=O)NCC3CN(C(CCC(=O)N(C)C)=O)C3)CCCC1CC(F)(F)CC2 c1(C(=O)NC(C)CNC(=O)COCC(N2C=NCC2)C)coc(S(C)(=O)=O)c1 N1(C(C2N(C(=O)C=Cc3cnccn3)CCC2)=O)CCC(CO)C12CCC2 C1(NC(C(C)(C)OC(C)=O)=O)CN(C(=O)C(F)C(C)C)CCC1C C(c1cc(Br)ccc1F)=CC(=O)N(C1CCC(NC(=O)CC2OCCO2)C1)C Cc1cc(N)cnc1C(=O)NCCc1n[nH]cc1C(=O)NCC1(O)CSC1 c1(C(N2CCC(C(=O)NC3CC4CCC(C3)C4)(OC)C2)=O)cc(C)cc(C#N)c1 c1(C(=O)NC(CC=C)CNC(c2cc(Br)ccn2)=O)cc(=N)[nH]c(Cl)n1 C1(NC(CCCC)=O)CCN(C(=O)Cc2cc(C)no2)C(C)C1 C1(NC(C2C(C)CCCC2)=O)CCCOC12CCN(C(C1CCC(=O)N1)=O)CC2 c1(CN(C2CN(C(C(C)CC3CCCO3)=O)C2)C)ccc(OCC(N)=O)cc1 Cc1oc(S(N)(=O)=O)cc1C(N1CC(CNC(=O)C=CCO)CC(C)C1)=O CCC(C)CCC(O)CC(=O)OCc1nccn2c(Br)cnc12 C=CCC(CNC(c1c(C)noc1N)=O)C(=O)N1CCCCCC1 c1(OC)cc(C)cc(C(=O)N(C)CCOCCNC(C2CCC(=O)NC2)=O)c1N c1(C(N(C(C)C)CCN(C(=O)COC2CCCC(C)C2)C)=O)cnn(C)c1C#N [N-]=[N+]=NCC(C(=O)N1C2CCC1COC2)NC(C1CC1Cl)=O C1(C(=O)NC2(CO)CN(c3ncnc4ccsc34)C2)CC2CCCCN2C1 C(=O)(C(C(=O)N1CC(C(C)NC(c2ccc[nH]2)=O)C1)C(C)C)OCC N1(C(c2c(SC)cccc2)=O)CCN(C(c2csc(C)n2)=O)C(CCO)C1 c1(C(=O)NCC(CC=C)NC(=O)COCc2scnc2C)ccc(C)c(C#N)c1 N1(C(c2cccc(SCCC)c2)=O)CCC(C)CC1CNC(=O)C(C)(C)C#N n1(CC)nc(C(=O)NCc2ccnc(C(=O)N(C)Cc3nnnn3C)c2)cc1O CC(CC#N)C(=O)NCc1cc(C(N2CC(O)C2)=O)n[nH]1 N1(C(C2C(C)OCCC2)=O)CCC2(NC(=O)Cc3cnn(C)c3)CCCC12 N1(C(C2CC(C#C)(O)C2)=O)CCC(C2CCN(C(=O)Cc3sccc3Cl)C2)C1 C(=O)(C(C)(C)S(C)(=O)=O)NC1(CNC(c2n(CC)cnn2)=O)CCOCC1 Cc1ccccc1CCNC(=O)CCC1CCCCN1C(c1ccns1)=O c1(-n2ncc(C(=O)NCC(C)N(C(=O)CC3CCCC3)CC)c2)cccc(O)c1 c1(C2(NC(C3C(C(=O)OC)C=C3)=O)CC2)c(F)cccc1F N1(C(C2CCN(S(CCCC)(=O)=O)CC2)=O)CCOC(C)(C)C1 c1(C(N2CCC(N(C(C3C(C)CCC3)=O)C)C2)=O)cccn2c(CO)nnc12 C(c1ccc(C#N)cc1)=CC(=O)N(CC(=O)N(CC(C(=O)OC)C)C)C C1(C(N(C)CC2(CNC(c3scnc3C(C)(C)C)=O)CC2)=O)CCCCS1(=O)=O c1(CCC)ncc(C(=O)N(C2CN(C(=O)CSCc3cccnc3)C2)C)s1 C1(S(N)(=O)=O)(C(=O)NCCN(C(=O)C(C)(C)C2CCCC2)C)CC1 c1(C(N2CC(N(C(=O)CC3CC3)C)C2)=O)coc2ccc(F)cc12 C(=O)(C(C(C)C)NC(C1OCCC1NC(c1cnc(N)cn1)=O)=O)OC N1(C(C(C)CN(C)C(C2CCNC2=O)=O)=O)CC2(CCCO2)C1 C1(C2(NC(C3CC(C(C)C)C3)=O)CC2)CCCCN1C(=O)C=C1CC1 c1(C(C)C)ccc(C#N)c(N(C)CC2CCCN(C(C3CCC(C)C3)=O)C2)n1 Cc1cc(C(=O)OC2CC3CN(C(=O)OC(C)(C)C)CC23)c(C)n1C1CCOC1 C(=O)(C(N)CCN(C(=O)CC1CCC1)C)NCCC(C)F c1(C(=O)NCCCN(c2cc(C(F)F)ncn2)CC)cccc2c(O)nncc12 n1(CC)nc(C)c(NC(=O)NCC(c2ccc(C)nc2)O)c1C c1(OC(CC)C(=O)NC2CCN(C(=O)C=CC(C)(C)C)C2)cccc(C)c1 C(C(=O)N=c1ccn(C2CC2)[nH]1)C1(C)CCN1C(C1CC2COCC(C1)C2)=O c1(C(=O)NC(c2ccccc2)CNC(C(F)=CC)=O)cnc2ccsc2c1 Cc1cc(F)ccc1C(N1CCC(O)(C(C)NC(c2cncn(C)c2=O)=O)C1)=O c1(C(=O)NC2C(NC(C3(C)CCC3)=O)CCCC2)c[nH]cc(Br)c1=N N1(C(CC(CC)O)=O)CCC2(CC1)OCCCC2NC(C1CCOCC1OC)=O c1(C(N(C2CCCCC2)C(C2C(C)(C)CNCC2)=O)=O)cc2c(F)cccc2[nH]1 C(C)(C(C(=O)N1CC(C(=O)OC)C2(CC2)C1)C(C)C)NC(C1CC(CCC)C1)=O N1(C(CC2CC(NC(c3c(C)n(C)cn3)=O)C2(C)C)=O)CC2(CCCN2C)C1 N1(C(c2c(C(C)(C)C)ncs2)=O)CCN(C(C2CCC2n2ccnc2)=O)CC1 c1(-n2c(C(CC(CC)C)NC3CCCC3C(N)=O)nnn2)ccc(Cl)cc1F C1(N(C(c2cnn(C3CCCCC3)c2)C(=O)NCCC)CC=C)CCN(C)CC1 C1(C(=O)N)CCOC1C(C)C.C(=O)(C(O)C1CC1)NCC1(OC)CC1 c1(C(=O)NCC23C(CN(C(C4CCC(=O)N4)=O)C2)C3)cc2[nH]ccc2s1 CC1OC(=O)NC1C(=O)NC1CN(C(c2cc(Br)sn2)=O)CC1C Cc1cc(C)c(NC(=O)C(N2CCC(C(O)C(F)(F)F)C2)C)c(C)c1 c1(C(=O)NC2CC2CNC(c2cc(C(F)F)oc2C(F)F)=O)cccc(CO)n1 Cc1ccc(F)c(CC(=O)NC(C)C(C)NC(c2cnc(C(C)(C)C)[nH]2)=O)c1 c1(CC(=O)NCCN(C(C(CO)N(C)C)=O)C2CC2)ccccc1N1CCCC1 N1(C(c2ccc(F)cc2Br)=O)CC2CCN(Cc3c(Br)ccnc3Cl)C2C1 c1(C(C(N2CC(CC)(CNC(=O)C(F)CC3CC3)C2)=O)(C)O)ccccc1F N1(C(C(c2ccc(OC)cc2)O)=O)CCC2(CC1)C(=O)Nc1cc(Br)ccc12 Cc1cc(C(=O)N(C)CC=CC(N2CCC(C(F)(F)F)C2)=O)nc(C)c1 Cn1ncc(C(=O)NCCC2CN(C(=O)CCC3CCCO3)C2)c1C(C)(F)F C1(NC(C(C(C)C)F)=O)CCN(C(c2ccc(OC(C)C)nc2)=O)C1(C)C N1(C(C(C(C)C)OCC(C)C)=O)CCCCCC1CNC(=O)C1=CCCCO1 CC1CN(C(=O)Nc2cccc3c2CCCC3)CC(C)S1(=O)=O c1(C(=O)NCCC2(O)CCN(C(C(COC)(C)C)=O)C2)nnn2c1CCCCC2 N1(Cc2cc(OC)c(OCc3ccco3)cc2)CCC2(CC1)NC(=O)C(C)(C)O2 c1(C(=O)NC(C2CCN(C(c3c(F)ccc(C)n3)=O)C2)C)cc2sc(C)cc2s1 C(CC)(CCCC(=O)N1CCC(OCCC)CC1)NC(C1(CC=C)CCC1)=O Cc1ccnc(O)c1C(N1CC=C(CNC(C2(F)CC=CCC2)=O)CC1)=O C1(N(C(Cc2nc(C)sc2)=O)C)CCN(C(C2CC(C)(C)CN2C)=O)CC12CC2 C(=O)(CC(C)(C)C)NC(C)C(N1CCC(c2nn[nH]n2)(OC(C)(C)C)C1)=O.C(=O)N CCC(C)CC(C)C(=O)N1CCOC(C)(C)C1C(=O)OC N1(C(C(c2ccccc2)OC(C)C)=O)CCCC(C)C1CN=c1[nH]nc(O)s1 c1(C(N(C2CCN(C(CCCCOC)=O)CC2)C)=O)cnc2sccn12 Cc1c(NCCN2CCN(C(=O)CO)CC2)ncnc1N(C)CCC1CCCCC1 c1(CC(=O)N(C2CCCN(C(CCS(C)=O)=O)C2)CCO)nc2c([nH]1)CCCC2 c1(C(=O)NC2C(C)CCN(C(c3c(C)cc[nH]c3=N)=O)C2)c(C)ccc(C)c1O C1(NC(c2ccncc2F)=O)CN(C(C23CC(F)(C2)C3)=O)CC1F N1(C(=O)CCN2CCCCCC2)CCC(F)C(NC(C2(F)CCC2)=O)C1 c1(OCCOC)ccsc1C(N1CCC(c2cn(Cc3cc(C)no3)nn2)C1)=O c1(CNC(C2CC(NCc3ccc(OC)nc3)C2)=O)sc2c(Br)cccc2c1C c1(C(C)C)cc(C(=O)OC(=O)NCCN(C)C)[nH]n1 CCC(C)(CC)C(=O)N1CC(CNC(c2cc(Br)c(C)s2)=O)C1 c1(COC2C(OC(=O)Cc3csc(Cl)c3)CC=C2)ccc(F)cc1Br c1(C(=O)NC(C2CN(C(=O)C=CCF)CCO2)C)cc2c(cc1F)OCC(=O)N2 C=CCC(C(=O)NC12CC(C(=O)Nc3cnn(CC)c3CC)(C1)C2)C(C)C C1(C(NNC(c2c(C)nc(Cl)s2)=O)=O)CC2CCC1C(N)C2 n1(CCC(N2CCC(F)(CNC(C3CCN(C)C3)=O)C2)=O)cc([N+](=O)[O-])cn1 N1(C(=O)CN2CC3CC3C2)CC2(C1)SCCC2NC(C1CCN(C2CC2)C1=O)=O Cc1nc(CNC(C2(NC(=O)CC3CC3(C)C)CCCC2)=O)c(C)s1 C1(C(=O)NCC(C)NC(c2c(C)cc(SC)o2)=O)CCc2nnnn2CC1 N1(CC(=O)NC(CNC(C(C)O)=O)CO)C(=O)Cc2ccccc2C1=O N1(C(c2ccc(CC)cc2)=O)CC2CCC1C(CNC(=O)CC1CC(C)=NO1)C2 C#CCC(C(N)=O)NC(=O)C(c1cccnc1)NC(C1CC2C=CC1O2)=O C(=O)(CCC(=O)N1CCC(O)CC1)NC1(C)CC(C(=O)NCC(C)CN(C)C)C1 c1(C(N(C)CC2CCCN2C(=O)C(=O)NCCC(N)=O)=O)cncc(N)c1 CC(N=c1nc2sccc2c(NCCC(CC2CCCC2)CO)[nH]1)c1cc[nH]n1 N1(C(C(CC)(C)C#N)=O)CC2(CCCN(C(c3ccc(N(C)C)cc3F)=O)C2)C1 c1(C(N(CCNC(C(C(CC)O)C)=O)C2CC2)=O)ccc(Cl)c(C#N)c1 C12(C(N(C3CN(C(CC(C)CN(C)C)=O)C3)C)=O)CCC(C1)C(C)(C)O2 c1(N2CC(C(C)NC(=O)C=C3CCC3)OCC2)nccnc1C#N c1(C(N2CCCC(CNC(C(C(C)(C)C)O)=O)C2)=O)ncn2cccnc12 c1(C(=O)NC(C)CCCNC(=O)C(=O)N(C)C)cc2cc(Cl)ccc2n1C CCCCCC(C)CC(=O)NC1CCC1NC(c1ccc(F)c(Cl)c1)=O c1(NC(=O)C(c2ccccc2)F)ccc(CC(F)(F)F)nc1 N1(C(c2cc(OCC)ncc2)=O)CCOCC(NC(C2CCCC2C2CC2)=O)C1 C1(C(=O)NCCN2CCOCC2=O)CCC(n2cc(-c3ccnc(F)c3)nn2)CC1 c1(CC)nc(C)ncc1C(N1CCCC(CN(C(c2c[nH]c(=N)s2)=O)CC)C1)=O c1(NC(=O)NCC2CCC(C(N)=O)CC2)ccc(OCC(F)(F)F)c(Cl)c1 c1(OC)ccc(C(CNC(C2C3CN(Cc4ncon4)CC23)=O)OC)cc1Br c1(C(N2C(CC)C(NC(C3C(F)(F)C34CC4)=O)CC2)=O)cc2cc(F)ccc2o1 C#CCC(C)(C)C(=O)NC(C1CCCN(C(=O)Cn2nnnc2C)C1)C C(C(C(F)(F)F)N1CCN(C(C2CC(CF)C2)=O)CC1)NC(C1N(CC)CC1)=O C1(C(N(C)Cc2ccc(CNC(C3C=CCS3)=O)cc2)=O)C2CCC(F)(F)C12 C1(NC(C2C3N(C(C4(C)C(C)C4)=O)C(CC3)C2)=O)CC2COCC(C1)C2 c1(OCC)ncccc1NC(C1(C)CN(C(=O)Cc2occc2C)C1)=O C#CC1(NC(C2CN(CCOc3cccc(OCC)c3)CCO2)=O)CCCOC1 CC(C(=O)NCC1(NC(c2cnn(C3CC3(F)F)c2)=O)CCCCC1)C(F)(F)F N1(C(C=CC(C)C)=O)CCC(CC(C)NC(=O)CCC2CCCN2C)CC1 C1(F)(C(N(C(C)C(C)(C)O)C)=O)CCN(C(=O)Cc2cccc(O)c2)C1 C1(C(N2C(CN(C(C3=C(C)CCC3)=O)C)COCC2)=O)CC2(CO1)CC(F)(F)C2 c1(C(N2C(CCC)COCC2)=O)cccc(C2(C(=O)O)CC2)c1 C1(C(=O)NCC(C(C)(C)C)NC(C2C(C)CCO2)=O)CC(C)(C)OC(C)(C)C1 C1(NC(CC2CC(OC)C2(C)C)=O)CC2(C1)CC(NC(c1nocc1C1CC1)=O)C2 c1(C(N(CC(O)CN(c2ccnn2C2CCC2)C)C)=O)cnn(C(C)(C)C)c1 N1(C(C(CC)(C)CO)=O)CC(C(=O)NCCCN(CC(C)C)C)CC(C)(C)C1 Cc1cc(C(=O)NCc2cn(C3CCCN(C(C4(C#N)CC4)=O)C3)nn2)cnn1 C(CCCCC(=O)NC1(CO)CC2CCCC12)N(C(c1cn(CC)nn1)=O)C c1(C(N2CCC(NC(c3cnc(Br)o3)=O)C2)=O)ccc(Br)cc1F C#CCCCCCC(=O)NC1(C(=O)NC(c2cn(C)nc2C)C)CC1(C)C c1(C(=O)NCC2N(C(CCC=C=C)=O)CC(C)(C)C2)ccc(S(=O)(=O)CF)cc1 CCC(F)(F)CC(=O)NCc1cn(CC(C)NC(C2CCC(C(N)=O)O2)=O)nn1 C1(CO)CC2CCC1CC2NCc1ccc(Oc2cccc(OC)c2)nc1 c1(C(N(C2CC(NC(CCCOCCOC)=O)C2)C)=O)cccc(OC)c1 C1(CNC(C(C(C)O)NC2CC2)=O)N(C(=O)CC2CC3CCC2O3)CCC1(C)C N1(C(C(F)=C(C)C)=O)CCN(C(c2cccc(CCC#N)c2)=O)CC1CO n1(CC(N2CC(NC(C(CCC)C(C)C)=O)C2)=O)nc2n(c1=O)CCCCC2 C(CC(O)C(=O)N(CCC(C)(C)NC(c1csc(C(C)(F)F)n1)=O)C)SC N1(C(C(N2Cc3c(nc(C)s3)C2)C(C)C)=O)CCC(C2CN(C(=O)O)C2)CC1 Cn1cc(NC(C2CCC(NC(C3(C)CCC3)=O)C2)=O)c(CO)n1 C(C(=O)Nn1ccccc1=O)C1CCN(C(C(c2cc(F)cc(F)c2)C)=O)C1(C)C S(=O)(=O)(c1c[nH]ccc1=NCCN1C(=O)CNC1=O)NC(c1ccncc1)C c1(CNC2CC(N3CCN(C)CC3)C(O)C2)cc(Br)c(O)c(Br)c1 N1(C(C)C)CCC(NC(c2csc(CNC(=O)CCOC3CC3)n2)=O)C1=O C1(CNC(COCCCCCC)=O)C2CN(C(=O)C(C)OC)CC12 CN1CC2CC1CN(C(C1COC3(C1)CN(C(c1cc(C#N)cs1)=O)C3)=O)C2 c1(OC)cc(C#N)ccc1C(=O)NCC1CCCN1C(=O)CCC1CCOC1 c1(C(=O)OCC)cnc(NC2(C)CC(NC(=O)CCNC(N)=O)C2)nc1C C1(CNC(C2CN(C)C2)=O)CN(C(=O)CCCn2cccc2)CCO1 c1(C(N2CC3N(C(c4n(C)cnc4)=O)C(CC3)C2)=O)cc2c(cnn2C)nc1O c1(C(N2CC(CC)N(C(=O)CC(C)C3CC3)CC2)=O)cccc2[nH]nc(O)c12 C1(C(C(N2CCC(O)(CN(C(=O)Cc3cnsc3)C)C2)=O)F)CCS(=O)(=O)CC1 C1(OC)CN(C(c2oc(CC3CC3)nc2C)=O)CC1NC(c1ccc(OC)o1)=O Cc1nn(C)c([N+](=O)[O-])c1N1CCC(OCC(N)=O)CC1.C1CCCCC1 N1(C(C(C#C)(C)C)=O)CCC2(C1)CN(C(c1occ(C)c1C)=O)CC(C)O2 c1(SCCNC(=O)CCn2ccnn2)noc(C(=O)NCCOC(C)(C)C)n1 c1(C(c2n(C(C)C)nnn2)NCc2cccnn2)cc(Cl)nc(Cl)c1F CCC(C)C(C(=O)NCc1cncnc1)N(C)C(c1cnc(Cl)s1)=O C1(CCNC(C2C(=C)C2)=O)CSCCN1C(c1cccc(Cl)c1)=O c1(C(N(CCCNC(C(C)OCC2CCCCO2)=O)C)=O)cnnc(O)c1 c1(CC)nn(C)cc1C(=O)NCCC(=O)NC(C)C(C)SC c1(C(N(C2CCCN(C(=O)CN3CC(=O)NC3=O)C2)C)=O)cccc2cnsc12 c1(OC(COC)C(N2CCCC2(C(=O)OC)COC(C)C)=O)ccc(Cl)cc1Cl C(C)(C)(CC(=O)N1CCCCC1NC(=O)CCC(=O)c1ccc[nH]1)N(C(C)=O)C O(NC(=O)C(CNC(C)=O)CC=C)C(C=C)C.C(=O)C(C)=CC(C)(C)C c1(NC(C2CCCCN2Cc2cnc(C3CC3)nc2)=O)ccc(Cl)cc1F c1(CCCC)ncc(C(=O)NCCC(Cc2ccccc2)NC(=O)CC=C)s1 c1(C(=O)NC(C2(C)CN(CCCC)C2)C)cc2ccc(OC(F)F)cc2[nH]1 N1(C(c2c(C)nn(CC)c2Cl)=O)CCCN(C(=O)COC2CCOC2)CC1 c1(C(CNC(c2ccn(C)n2)=O)NC(C2N(C(C)=O)CCC2)=O)ccc(F)cc1 C1(C(N2CC(CC(C)C)C2)=O)CC(F)CCN1C(C1CCCOCC1)=O C1(c2scc(C(=O)OC)n2)CCCCN1C(=O)CCCn1cc(CCO)nn1 c1(OCC(=O)NC2C(CNC(C=C(C)C3CC3)=O)CCCC2)ccc(Cl)c(Cl)c1 N1(C(c2c(CC)c[nH]c2)=O)CCN(C(c2cc(Cl)cn2CC)=O)CC1C(C)C c1(CC(=O)N(CCCCCO)C2CCOC2)cc(Cl)ccc1F c1(C(N2C(C(N(CCO)CC)=O)CCC2C)=O)n[nH]c2c1COC2 C1(O)(CNC(C2(C)CC2F)=O)CCN(C(c2cccc(O)c2Cl)=O)CC1 C(=O)(CC(O)CC(C)(C)C)N1CCC(=C)CC1C(=O)NCC1CCCC(C)(C)C1 N1(C(C(C)(C)C2CCN(C(c3nn(C)cc3Cl)=O)C2)=O)CCC2(CCO2)C1 C1(CC(=O)NCC(C)C(=O)NCCc2ncccn2)CC(=O)NC1=O C#Cc1cc(C(N2CCN(C(c3ccnc4[nH]ncc34)=O)C3CC23)=O)cc(F)c1 O=C1CCC(C(=O)NC2CC3CC2CN3C(=O)C=Cc2nccs2)=NN1 C1(C(N(C2CC(CO)C2)C)=O)CC12CCN(C(=O)CCC1(C#N)CCC1)CC2 N1(C(c2cc(C(C)=O)c(C)o2)=O)CC(NC(C2CCC2)=O)C2CCCC12 c1(C(=O)NCC23N(C(CCC#C)=O)CCC2CC3)c([N+](=O)[O-])cnn1CC(F)F c1(C(=O)NC(C2CCOC2)CNC(c2cnc(SC)s2)=O)cnn2c1OCCC2 c1(C(=O)OCC)cc(S(=O)(=O)N2CCC(C)(C)C2)ccc1C=Cc1cccs1 CC(CC(=O)OCC(=C1CCN(C)C1)F)C(=O)NC(C)Cn1cnnc1 C1(CNC(C2=NOC(C)(C)C2)=O)CC2(CCN(c3cccc(F)c3C#N)CC2)CO1 CC1=CC(C)CN(C(C2(CO)CCN(C(c3coc(N(C)C)n3)=O)C2)=O)C1 CCC(CC(C)O)N=c1nc2c(cnn2C(C)C)c(NCc2cc(Cl)cn2C)[nH]1 N1(C(C2CCC(NC(C=CC)=O)C2)=O)CCOC(C)(CC)C1 C1(NC(C(C=C=C)C)=O)CCN(C(=O)CCCn2ccnc2)CC12CCC2 C1(NC(c2cccnc2C2CC2)=O)CC(CNC(C2CCCSC2)=O)CC1O C1(C(=O)NC2CC3(CC(NC(C4CC(C)(O)C4)=O)C3)C2)COCC2(CCC2)O1 C1(C(N(C)CCOCCNC(=O)CCCCCN(C)C)=O)CCN2CCOCC12 C1(COC)(NC(=O)CCC2CCCN2C)CCN(C(=O)C(C)CC2CC2)CC1 Cc1cc(NC(C2CCN(C(c3cc(C)ccc3O)=O)C2)=O)cc(C)c1 c1(NC(=O)COC=CCl)cc(C(N2CCCC2C2(NC(C)=O)CC2)=O)oc1C c1(C(C(N)=O)N(C(=O)C(=O)Nc2cnn(C(C)(C)C)c2)C)cccc(F)c1 c1(C(=O)OCC)sc(NC(=O)CC2CN(C(c3cncc(C)n3)=O)C2)cc1C C1(C(N(C)CC2COCCN2C(c2nnc(O)cc2O)=O)=O)CCCC2(CC2)C1 Nc1cc2ccccc2c(C(N2CCC(OC(F)F)C2)=O)n1 N1(C(c2cc(C)c(O)cc2)=O)CC(NC(=O)CC2(O)CCCC2)C2CCCCC12 N1(C(C(CCN(C)C)NC(C2C(C)CCO2)=O)=O)Cc2ccc([N+](=O)[O-])cc2C1 N#Cc1cc(C(=O)O)cc(C(=O)NC(c2ccccc2)C2COCCO2)c1 c1(N2CC(C(C)NC(C3CCC(C)CC3)=O)OCC2)ncnc2c1cnn2C Cn1c(C(=O)NC2(C)CC2)ccc1-c1cn(CC(N2CCCCC2)=O)nn1 C1(C(N(C(C)CNC(c2csc(-c3ccco3)n2)=O)CC)=O)CC2C=CC1O2 CN1CCCC1C(=O)NCC(F)CNC(c1csc(-c2ccsc2)n1)=O c12ccc(F)c(c1)C(C)N(CC)C(=O)N2.c1(NC(=O)OCC)nnc(N)s1.OC C=CCCCC(C(=O)NC1CCC(F)(F)C1)NC(c1cc(CC)oc1C)=O N1(C(C(CC(C)(C)C)O)=O)CCCC2(CCN(C(C3CC3C(C)(C)C)=O)CC2)C1 N1(C(c2c(CC)ncs2)=O)CCC(CNC(c2cnn(CCF)c2)=O)(OC)C1 Cc1noc(C(C)C)c1C(=O)NCC1CC(C)N(C(=O)CSCCC#N)C1 N(C(=NCC(F)F)N1CCC(S(C)(=O)=O)CC1)CC(c1ccco1)OCC c1(C(=O)NCCC(C)NC(c2nc(C)oc2)=O)ccc(C2CC2(F)F)cc1 CCC(C)(C#N)C(=O)N1CCC(O)(CN(C(=O)COc2cc(C)cc(C)c2)C)C1 C(C(C)(C)C(=O)NCC1CCCC1NC(=O)C(c1cccc(C)c1)=O)NC(C)=O Cc1nc(C(=O)NC(C)(C(=O)N2CC(c3nc(=O)o[nH]3)C2)C2CCC2)co1 C1(C(=O)NCCSCC(=O)NCCn2cccn2)CC2CCC2C1 N1(C(c2ccc(C(=O)N(C3CC3)C(C)C3CC3)cn2)=O)CCN2CCCCC2C1.CO c1(C(N(C2CCCN(C(=O)CC3CCC3)C2)C)=O)ccc(CS(N)(=O)=O)cc1 c1(OCCOCC)ccccc1CN=C(NC1CC1)NC1C=CCCC1 CCC1=NOC(C(=O)NCCOC(C)C)C1.C1C(=O)N1 C1(C(N2CCC(C(=O)NCC=C(Cl)Cl)(OC)C2)=O)CC1C1(C)COC1 C1(=CC(=O)NCCOCCN(C)C(C2(C)COC2)=O)CCC(C)(C)CC1 Cc1nc(O)nc(C)c1CC(=O)NC1CN(C(c2cccn2C)=O)CCC1(C)C N1(C(c2cc[nH]n2)=O)CCC2(CC1)OCCC2NC(CN(C(C)(Cl)C1CC1)C)=O C(=O)(CC(C)CCC=CC=Cc1ccccc1)NCC1(O)CN(C(C=CC)=O)C1 C#CC1CC2(CC(C(=O)NCCC(C)NC(=O)CCC(C)(C)OC)C2)C1 C(=O)(CC(F)(F)C(C)C)N1CCC(CNC(C2(C=C)CCC2)=O)CC1C N1(C(CCCC#CC)=O)C2CCC1CN(C(C13CCC(OCC)C1C3)=O)C2 C1(C(NOCC)=O)CCC(C)CN1C(c1ccc(C2CC2)o1)=O.c1cc(CO)[nH]n1 n1(CC)ncc2cc(C(=O)Nc3c(C)nc(CO)nc3C)c(C)nc12 n1(CC)cnc2c(N3CCC(C)=C(C)C3)[nH]c(=NCCCc3ccnn3C)nc12 c1(C(=O)NCCNC(CC(C)(C(F)(F)F)N(C)C)=O)cccc2nc(O)n(C)c12 N1(C(C2C(=C)C2)=O)CCC(NC(c2ccn(CC(F)F)c(=O)c2)=O)C(F)(F)CC1 c1(C(=O)NC2(CNC(c3nc4ncccn4n3)=O)CC2)ccc(=O)n2c1CCC2 C1(C(=O)NC)CC12CCN(C(=O)CC1CC(OC)C1)C2.C1C(=O)N1CCC C1(CNC(C2(C)CC2(Cl)Cl)=O)CCN(C(=O)CC2=CCCC2)C12CC2 c1(C(=O)NC(C(=O)OC)CC2CCCCC2)cc2cc(C)ccc2nc1C C#Cc1cncc(C(=O)NC(CNC(=O)CC(C)CF)CC(F)(F)F)c1 CC(C(C)(C)C(=O)NCCc1ccncc1F)NC(C1CC(=O)NC1(C)C)=O Cc1ccc(C=CC(=O)NC2(CNC(=O)CCN3CCCCC3=O)CCC2)cc1 c1(CC)ccccc1CC(=O)NC(C)(CNC(=O)C(F)C(C)C)C1CCC1 Cc1cc(C(=O)NCC2(C(C)(C)C)CCN(C(c3ccnn3C)=O)C2)ccc1Cl n1(CC)cnc2c(NCc3ccc(Cl)o3)nc(N(C)Cc3ccccn3)nc12 c1(C(N(C(C(=O)OCC)Cc2ccc(Cl)cc2)C2CC2)=O)ccc(Br)c(C)n1 c1(C(N2CCC3CN(C(=O)C=CC4CCOC4)CC32)=O)cnc2ncnn2c1O O(NC(=O)C(C1(C)CC1)NC(=O)CC1CCC1)CCC=C C1(CCOC)CN(C(c2cccc(N(C)C)c2)=O)CCN1C(=O)CC(CC)OC c1(CC(C(=O)NCC2(NC(CCC(=C)C)=O)CCOC2)(C)C)ccc(C#N)cc1 c1(Cc2n(-c3cccc(C)c3)nc(CC3CC3)n2)cc2c(cc1Br)OCO2 N1(CCCc2ccc(OCCCCCCCC)cc2)CCc2cc(Cl)nnc2C1 C1(NC(C(C)N(C(=O)C(c2ccccn2)O)CCC)=O)CCC(C)(OC)CC1 N1(CC)CCCC1CN(C(=O)C(C1CCCC1)NC(=O)CCCn1ccnc1)C N1(C(C2(C(C)NC(c3cnc(CC)s3)=O)CC2)=O)CCC12CC(C)C2 c1(C(N(C)CC2CCN(C(C(COC)(C)C)=O)C2)=O)cc2nc(C)ccc2o1 C1(NC(c2c(CC)nc(C)nc2)=O)CCC2CCN(C(=O)C(F)(F)CO)C1C2 C1(S(C)(=O)=O)(C(=O)NCC(CN(C(C2(CCC=C)CC2)=O)C)C)CC1 CC(C)C(CCC(=O)NCC1CCCC12CCC2)NC(=O)C(C)(C)N(C)C c1(NC2CC2c2ccnc(Cl)c2)cc(S(=O)(=O)N)ccc1C#N.C=C1CC(N(C)CC)C1 CCC(CC(=O)NC1(CNC(C2CN(C)C2)=O)CCCCC1)C(C)(C)C C1(NC(COCCC#C)=O)CN(C(c2ccc(C(C)C)nc2O)=O)C(C)(CC)C1 c1(OC)c(C(=O)NC2CCN(C(c3ccn(C)c3)=O)C(C)C2)oc2ccccc12 C(=O)(CCN=c1[nH]ccs1)NC1(C)CCN(C(c2c(OC)oc(C)n2)=O)C1 C1(CC)CCC(C(=O)NCCCCCNC(C2COCCN2CC(F)F)=O)CC1 Cc1cccc(C(CNC(C2(c3nncs3)CC2)=O)NC(c2cc(C)sn2)=O)c1 N1(C(c2cccnc2-n2ccnc2)=O)CCCC2(CC1)CC2 C(C(C)(C(=O)NC1(C(N)=O)CCC1)NC(c1cc(=N)[nH][nH]1)=O)SC c1(NCC(=O)NC23CC(NC(C(CC)CC)=O)(C2)C3)ncnc2c1c(Br)cn2C C=C(C)C(C)(O)C(=O)NCC(C)(O)CNC(c1cccc(F)c1C1CC1)=O C1(N(CCO)Cc2nc(CCC)on2)CCCN(C(=O)C=C(C)C)C1 c1(C(=O)NCC2OCCN(CCC=C)C2)cnc2nc(Cl)ccc2c1 C(CC)(CC)C(C)C.c1(-c2ncc(-c3n(CC)ccn3)s2)c(C)cccc1C N1(C(=O)Cn2nnc(=O)[nH]2)CCC2CN(C(c3cc(C(F)F)on3)=O)CC2C1 C1(CNC(CN(C(=O)CCOCCOC)CC)=O)CN2CCC1CC2 C(c1ccccc1)=C(C(N1CCC(CCOC)CC1)C(=O)NCC=C)C c1(N2CCN(C(c3ccc(C(C)(F)F)cn3)=O)CC2)ccc2c(c1)NC(=O)C2 c1(CN2CC(n3ccc(NS(CC=C)(=O)=O)n3)C2)cc(C)cc(F)c1 N1(C(c2c(C)scc2)=O)C2CCCC1CC(NC(c1csnn1)=O)C2 C1(C(=O)NCc2ccc(C(=O)O)[nH]2)CCCCC1C.n1(CC(C)S)cc(CO)nn1 C(=O)(CC(CC)NC(c1cc[n+]([O-])cc1)=O)N(C(CC)CSC)C c1(C(N(CC(C)CNC(=O)CC(C)n2ccnc2)C)=O)cc[nH]c(=N)c1N CCC(CC)C(C)C(=O)N(C)CC1CCN(C(=O)COc2ccccc2F)CC1 C1(C(=O)OC)CN(C(C2CC2Oc2ccccc2)=O)CC1(C)OC(F)F O=C(C1=C(Cl)CCCC1)NC1CCN(C(=O)CCCn2cccn2)CC1F c1(C(=O)NCCC2CCCN(C(C3CC3(F)F)=O)C2)c(F)cc(F)cc1Br Cc1cc(C(=O)NC2COCCN(C(C3(C)CCCO3)=O)C2)c2c(O)n[nH]c2n1 N1(C(CCSCC)=O)CC2CS(=O)(=O)CC2(NC(C2CCSCC2)=O)C1 c1(NC(N2CC(N3CCCCC3=O)(O)C2)=O)sc2c(c1-c1nn[nH]n1)CCC2 C1(C(=O)NCC2N(C(C)(C)C)CC2)C2CC3C(C2NC(C2CCOC2C)=O)C13 C1(n2ccnc2)(C(N(C(CNC(=O)Cc2csnn2)C2CC2)C)=O)CCCC1 c1(C(N(CCC(=O)NCC(F)F)C(C)C)=O)cc(C2CC2)on1.C(C)(C)O C(=O)(CCS(=O)(=O)C(F)(F)F)N1CC(NC(C2(C=C)CC2)=O)C(CO)CC1 n1(CC(=O)N(CCC(N2CCC(CC(=O)OCC)C2)=O)CCO)ccccc1=O C1(CC(C)NC(=O)CC2=CCCC2)CC2CCC(C1)N2C(C1C(C)(C)C1(C)C)=O N1(C(c2c(CC)nn[nH]2)=O)CC2(CCC(CNC(c3cn(C)nc3OC)=O)O2)C1 N1(C(C2(C)CCN(C(=O)CC)C2)=O)CC2CC1CN2C(=O)C=CC(=O)OC.CN C1(CCNC(C2(CC)CC2)=O)C(C)CCCN1C(c1nccc(OC)c1C)=O C#Cc1cnc(C(N2C(C(N3CCC(C)(C#N)C3)=O)CCC23CC3)=O)c(C)c1 c1(C(=O)NCC(CN(C(=O)CCCn2ccnn2)C)O)nc(C(F)(F)F)cn1C c1(C(=O)NC(C(C)NC(c2sc(CC)c(C)c2)=O)(C)C)cc(OC)cnc1F Cc1cc(C(=O)NC2CCC2CNC(c2cn(C3CC3)nn2)=O)cc(C)c1Cl CN1CCC(n2nnc(C(F)(F)F)n2)(NC(c2ccc(C3CC3)cc2)=O)CC1 c1(C(N2CC(NC(c3cn[nH]c3)=O)C3C2C3)=O)n[nH]c2ccc(F)cc12 CC1(C)C(NC(=O)Cn2ccccc2=O)CCN1C(=O)C1=CCCCC1 c1(C(=O)NCc2ccc(C(=O)Nc3ccc(SC)o3)cc2)cc(N)cc(N)c1 Cn1c(C(=O)NCC(C)(C)CNC(c2c[nH]nc2-c2ccsc2)=O)cc(Cl)c1Cl C1(NC(c2cc(Cl)cc(Cl)n2)=O)CCSC12CN(C(c1cc(O)cc(O)n1)=O)C2 C1(CNC(C(CC)SC)=O)CCCCN(C(=O)CC2CCC2)C1 C1(CCC)CCC(NC(=O)C(N2CC(c3ccccc3)(C(F)F)C2)=O)CC1 C1(N(C(=O)C=CC=C(Cl)Cl)CCC)CCN(C(=O)C(C)O)C1 C1(C(=O)NC(CC)CCOC)CN(C(c2nnsc2C)=O)CC1(F)F CC12COC(C(=O)NCC(=C3CN(C(=O)CSCC4CC4)C3)F)(C1)C2 C1(CNC(c2cnc(OCC)nc2)=O)(CO)CCN(Cc2ncoc2C2CC2)CC1 C(=O)(C(C(C)C)N1CCCS1(=O)=O)NCCC1N(C(CC2CC(=C)C2)=O)CCC1 C(C(C)C(F)C(=O)NC(c1nc(=O)o[nH]1)C)NC(COCCSC)=O N#CC1(C(N2CCN(C(C3CCCN3N=O)=O)CC2)=O)CCCCC1 N1(C(C=CC(CC)C)=O)CCN(CCN(C)C(c2nc(C)oc2OC)=O)CC1 C1(CC(=O)N(C2CCN(C(=O)Cn3cccn3)C2)CC)CCCCCC1(F)F C(C1=CCN(C(C2CN(C(C)=O)CCO2)=O)CC1)NC(C1CCC(CC)O1)=O Cc1ccccc1C=CC(=O)NC(C1CC1C(=O)NCCCC(=O)NO)C N1(C(C(c2c(C)noc2C)(C)C)=O)C2CCC1C(CNC(=O)C(C)NC(N)=O)C2 C1(N2C(=O)CCC2)CCN(N2CCCC(c3noc(C(F)(F)F)n3)CC2)CC1 N1(C(C(CC)SC)=O)CCN(C(=O)COCc2cscn2)C(C(F)F)C1 C1(C(=O)NCC(CO)NC(=O)CC(Cl)Cl)C2CCC3C(C2)CC13 C1(C(=O)NCC=CCNC(c2n[nH]cc2[N+](=O)[O-])=O)Cc2ccc(F)cc2O1 C1(C(N2CC(C)N(C(c3ccc(O)nc3)=O)CC2)=O)CCn2c(O)nnc2C1 N1(C(C(C)SC)=O)CCC(C(=O)NCCCc2cnn(C)c2)C12CCC2 C1(CNC(C23C(C(N)=O)(CCC2)C3)=O)CC2CCC1N(C(C1CC(CF)C1)=O)C2 c1(OC)ccc(Cl)c(C(=O)NC(CO)CCCCNC(C2CCCCO2)=O)c1F N1(c2nnc(C)o2)CCOCC(C(=O)NCc2ccncc2C(F)(F)F)C1 C#CCC(CC#C)C(=O)N1CC(C)C(C)(CNC(=O)C=Cc2cncnc2O)C1 N1(C(Cc2c(C)noc2)=O)CCN(C(C2CC3C=CC2C3)=O)C(C2CCC2)C1 c1(C(N2C(C)(C(=O)NC)CC(O)C2)=O)ccc2ncccc2c1 CC(=NO)C1CC(C(N2CCC(C)(CNC(C3(C)CC3)=O)C2)=O)C1(C)C C1(CC(=O)NCC(N(C)C(c2ncccn2)=O)C2CC2)CN2CCN1CC2 n1(CC)nnc(C(N2CCC(CCCNC(C3(C)C=CCCC3)=O)CC2)=O)c1C Cc1cc(C(N2C3CCC2C(CNC(C2CC4(CCC4)CO2)=O)C3)=O)nc(O)n1 C12COCCC1NC(=O)NC1CCC(CC1)C(=O)N2.c1(C(O)C2CC2)ccccc1 N1(C(CSc2ccc(C)c(C)c2)=O)CCCC2(CCN(C(=O)C=CC3CC3)C2)C1 Cc1ccc(CC(=O)NC2CCN(C(C3CC3C(F)F)=O)CC2O)cc1Cl c1(COC)cccc(CC(=O)NCC2(O)CN(C(C34CCC(OC)C3C4)=O)C2)c1 N1(C(C(n2c(C)nnn2)Cc2ccccc2)=O)CC2CC(OC(C)C)C(C2)C1 c1ccc2c(-c3cn(Cc4cnoc4)nn3)csc2c1 C(=O)(N=c1cc(Cl)nc(CBr)[nH]1)N1C(C)CCC1C(=O)ON1CCCC1 Cc1c(C=CC(=O)NCC2CC(NC(c3cc(N)c(Cl)cn3)=O)C2)cnn1C N1(C(C(=C)C(F)(F)F)=O)CCOC2(CCC(NC(=O)C(=O)NCC3CC3)CC2)C1 c1(CC(=O)N(C)CC2(NC(c3cnn4c3CCC4)=O)CC2)cccc2c1OCC2 Cc1c(Cl)cn2c(=O)cc(CN3CCC(C)OC(C(F)(F)F)C3)nc2c1Cl C1(c2c(OC)nccc2C)CCC(=O)N(c2ccccc2)CC1 C(=O)(C1=CC2CCCCCC12)NCC1C2CN(C(C(CC(C)C)(F)F)=O)CC21 N1(C(COCCC=C)=O)CCC(F)(CNC(C2CCC2C)=O)C1 c1(OC)ccc(C)c(C(=O)NCC(CNC(=O)CNC(C)=O)S(C)(=O)=O)c1 O=C(CCCC(=O)C1CC1)NC1C2CCC1N(C(c1cnc(Cl)s1)=O)C2 Cc1oc(Br)c(C)c1C(N1CC(NC(c2cnc(O)n2C)=O)C(C)C1)=O c1(N2CCC3(C(C(=O)NC(C)CF)C3)C2)ncc2ccc(F)cc2n1 C12(NC(=O)Cc3cnc4cccnn34)CCCC(CN(C(=O)C(O)C3CC3)C1)C2 CC1(C)CC(NC(=O)CC(O)CNC(=O)C(=O)NCC2CC2)C(=O)O1 N1(C(c2c(C)nn(C)c2C)=O)CCCC1C1CCCN1C(=O)CCNC(=O)CO C=C(CC(CO)N=c1ccc(-c2ccc(Cl)s2)n[nH]1)C(=O)O c1(NC2CC(NC(=O)CSCC3CCCCO3)C(O)C2)c(Cl)cccc1[N+](=O)[O-] c1(CS(C)=O)cccc(C(=O)NCC(O)CNC(C2CC23CC3)=O)c1 C1(CNC(CC(C)OC)=O)CC2CCC(C1)N2C(c1n[nH]cc1C(C)(C)C)=O c1(C(=O)NC(CNC(C2C(C(C)(F)F)C2)=O)C2CC2)cc(C2(C)CC2)ccc1F C=CCCCCCC(=O)N(C)CC1CCCN1C(C1CC(C)(C)CN1C)=O c1(CCC)cccc(C(C)(C)N2CCCCN2CC2CC2)c1 C1(NC(=O)Nc2sc(N(C)C)c(C#N)c2)=CC2(Cl)C(=C1)N=CC=C2 c1(C(=O)NCC2C(C)CN(C(=O)COC3CCCOC3)C2)c[nH]c2cccnc12 C1(C(=O)NC(CC)(C)CCNC(=O)CC(C)C2CC2)CCC(=O)N(C)C1 C(C(=O)N=c1ccn(C2CCOCC2)[nH]1)C1(C)CN(C(=O)CCC(N)=O)C1 c1(N(C(C2CCCN2)=O)Cc2ccnc(OC)n2)c2c(nn1C)CCC2 NC(=O)CCCCC(=O)NCC(O)CNC(C1(C(=O)N(C)C)CCC1)=O CC(c1cccc(Cl)c1)=CC(=O)NCC(C)(F)CNC(C1(C)CCCO1)=O C1(NC(CC2N(C(CC)=O)CCC2)=O)CCN(C(=O)CC)CC1.C1CO1 CN1CCN(C)C(C(N2CCC(CC(=O)NCC(C)(F)F)C2)=O)C1 CCCC(c1nnnn1Cc1cccs1)(C1CCOC1)NCC1=CCSC1 CC1(C)OC2(C(=O)N(C3CCCCC3)CCNC(=O)C=CCN(C)C)CC1C2 C(=O)(CCCCCN(C)C)N1CCC(C)C1C(=O)N(C)CCO N1(C(c2cnc(C)o2)=O)CCC(C(=O)NCC2CCC(=O)N2)C(C)C1 C1(C(C(=O)NC(C)C)N(CC(C(=O)OCC)C)C)CCCOC1c1cn[nH]c1 CC(C)C(CNC(=O)CC1CC1)NC(=O)C(F)CC1CCC1 c1(C(=O)NCCN(CCC)C(c2cc(C)[nH]n2)=O)cnc(Br)s1 N1(CC(C(C(c2ccc(CC(C)C)cc2)C(C)C)=O)=O)CC2CCCOC2C1 C(C)(C(C)(C)NC(c1cn(CCN(C)C)nn1)=O)NC(C(C)OCCOC)=O C1(CC(N2CCOCC2C2CCOCC2)=O)CC(n2cc(C(=O)O)nn2)CCO1 O=C(C1=C(Cl)CCCC1)N1CCN(C(=O)CN2CC(F)(F)C2)C(C2CC2)C1 c1(C(=O)NC2CC(C)(NC(C3C(C)C(=O)C3)=O)C2)cccc2c[nH]nc12 c1(C2C(C(=O)NC3CCC(C(C)(C)C)C3)C2)cccc(O)c1Br c1(C(=O)NCC2C(CNC(C3C(C)(C)CCCC3)=O)C2)cc2c(cn1)OCCC2 c1(C(=O)NCC(C)NC(C(C=C)O)=O)cnn2c(C)ccnc12 N1(C(c2cn(CCCCF)nn2)=O)CCCCCC1CNC(C12CCC1C2)=O Cc1ccccc1-c1cccc(CC(=O)NC2(CO)CN(S(=O)(=O)CC3CC3)C2)c1 N1(C(CCOCCC)=O)CC(=O)CC1C(=O)NC1CCC2(C(C)C)CC12 c1(C(N(CCOCCN(C)Cc2onc(CCCC)n2)C)=O)c(Cl)cnn1CC c1(C(C)NC(c2ccc(OCC)c(OC)c2)=O)cnc(SCC)[nH]c1=NC(C)C C#CCCCC(C)C(=O)NC(C)(CSC)C(=O)NC(COC)CO Cc1nc2c(C(N3CC4(CCN(C(c5nonc5N)=O)CC4)C3)=O)cccc2o1 N1(CC(=O)NC(CNC(c2c(C(F)F)cccc2F)=O)CO)CCCCCC1=O c1(C(N2C(CNC(CCC)=O)CC2)=O)nc2ncccn2n1 c1(CNC(=O)NCCC(=O)NC(c2ccncc2)(C)C)cccc2nccnc12 c1(CC)onc(C)c1C(=O)NC1CC(NC(c2cnc(C)o2)=O)CC1O N1(C(C2(OCC)CCOCC2)=O)CCC2CCN(C)C2C1.n12cc(nn1)c(=O)[nH]2 C1(CC(=O)NCCN(C(c2cc(C(F)F)no2)=O)CC)CCc2nc(O)[nH]c2C1 c1(C(N2CC3CN(C(C4CC(OCC)C4)=O)C3CC2)=O)cccc2nccnc12 C1(NC(=O)CSC(F)F)CCC(C(=O)NCC(CNC(N(C)C)=O)(C)C)CC1 c1(C(N(CCCN(C(=O)C#CC2CCC2)C)C)=O)cncc(Cl)c1Cl c1(COC)cc(CNC2C3CC4COC2C4C3)ccc1OC c1(C(=O)NCC(O)C2(Cl)CC2)coc(CNC(C23CSCC2C3)=O)n1 C(CN=c1ccc(Br)c(S(=O)(=O)N(C2(CCO)CCC2)C)[nH]1)(CC(C)C)OCC c1(C(=O)NC2C(F)CCN(C(c3n[nH]c(CC)c3Cl)=O)C2)ccsc1S(N)(=O)=O CC1c2sccc2CCN1C(=O)Nc1cc(Br)ccc1O N1(CCC(=O)NCC(C)CNC(c2occc2Cl)=O)CCOC1=O C(=O)(C(CNC(C1(F)CCOC1)=O)C(C)C)NCCC(=O)NC C(=O)(C(C)C(C)C(C)(C)C)N1CC(C)(NC(c2cc(C)nnc2O)=O)C1 N1(C(C2(CC)CCCC2)=O)CCCC(O)(CNC(c2cc(C(F)(F)F)n[nH]2)=O)C1 c1(NS(=O)(=O)C2CC2)ccc(NC2CCCC(C(=O)NC(C)(C)C)C2)nc1 c1(CC(C)C(=O)Oc2ccc(N3CCC(C)(O)CC3)cc2)cnn2cccc2c1 C(=O)(CCCC(F)(F)CO)NCCC1CC(OC)CN1C(c1cc(C)cnn1)=O C1(c2ccccc2)(NC(C2C(CC)C2)=O)CCN(C(c2csc(CO)n2)=O)C1 c1(OC)cnccc1C(C)NC(=O)C(=O)NC(c1cn(C(C)C)nn1)C c1(C(N(CCN(C(=O)COC2CCCC2)C(C)C)C)=O)ncnc2ccsc12 c1(C(=O)NC(C2CN(C(c3ccc(N)c(C(=O)O)c3)=O)C2)C)csc2nccn12 CC1CC(NC(=O)OCC)CN1c1ccc(C(F)(F)F)cn1.C(=O)(C1CC1)NC c1(NC(C2(NC(CC3(CSC)CC3)=O)CC2(C)C)=O)ccc(O)cc1CO c1(CC)cc(C(N2CCCC2C(C)NC(c2ccc(Cl)o2)=O)=O)sc1C C(=O)(CCC(O)C(C)(C)C)N(CCCN(C(C(N1CCCC(C)C1)=O)=O)C)C C(=O)(C(=NO)c1csc(NC(=O)C(=O)NCC2CC(=C(F)F)C2)n1)OCC C(=O)(C(CC(C)C)C(C)C)NCCOCc1ccc(NC(C=C(C)Cl)=O)cc1 C(C)(CCOC(F)F)(c1nnnn1C1CCC1)NC1CC(OC(F)F)C1 C1(C(N(CCn2cc(-c3cn(C(COC)C)nc3)nn2)CC)=O)CCCCC(=O)C1 C(C(=O)NC1CC(NC(=O)C=NOC)C(O)C1)(C(C)C)N(CC)CC CC1(CNC(=O)COCCc2ccc(Cl)s2)CCC(NC(=O)CCCC2CC2)C1 C1(NC(CC(CC)CC)=O)CN(C(=O)CC(c2c(C)noc2C)C)C2(CCC2)C1 C1(NC(CS(C)(=O)=O)=O)CC(F)CN(C(c2cc(-c3ccc(O)cc3)[nH]n2)=O)C1 C12(NC(=O)CC3(CC4CC4)CC3)CCC(n3cc(C4CC4)nn3)(CC1)C2 N1(C(C=CCC)=O)CCCC(O)(CC(N2CCN(C)CC2CC)=O)C1 N1(Cc2scc(C)n2)C(C)C(=O)OCC1Cc1ccccc1 N1(C(c2nc3ccc(C)cc3s2)=O)C(C)CC2CN(C(C34CSCC3C4)=O)CC12 C1(C(N2C(C)(CCC)CC2)=O)CCCN(C(=O)C(C)(F)F)C1CC N1(C(C(F)OC)=O)CCC(C2CCCN(C(c3cnc(O)n3C)=O)C2)CC1 N1(C(c2c(N)sc(C)c2C)=O)CCC2(CCCC2CNC(C2CC2(C)Br)=O)CC1 CCC(CC(=O)NCC(c1ccccc1F)NC(C1(F)CCOCC1)=O)SC C(CN(C)C)(CO)(CO)NC(CN(C(c1cc(OCC)n[nH]1)=O)CC1CC1)=O C(CO)(CCC(C)C)NC(C1N(C(C2(OC)CCOCC2)=O)C(C)C1)=O C1(CNC(C(CC)N(C)C)=O)CC2(CCOCC2)CN1C(C1(C)CC(C#N)C1)=O C1(C(=O)NC2(C=C)CCCCC2)CC2(CCN(C(c3cnsn3)=O)C2)C1 C=CCCCCCN(C(=O)C=CC(C)NC(=O)CCCC1CC1C)C C1(C(N(C)CC2N(C(c3c(OC)ccs3)=O)CCCC2)=O)CCC2CC2CC1 C(=O)(CC(C)(C)N(C)C(c1cnns1)=O)N1C(C(CCC)C)CCC1 N1(C(CCCN(CCC)CCC)=O)CCC(NC(C2CN(C)C(=O)N2)=O)C(O)C1 N1(CC)CCCN(C(CCc2ccc(C)c(C)c2)C(=O)NCc2ccccc2)CC1 N1(C(C(C)C(C)C(F)(F)F)=O)CCCC(C2CCN(C(=O)CNC=O)CC2)CC1 C(=O)(C(C)(CC)CCC)N1CCC(NC(C2(C#C)CCC2)=O)C(F)C1 O=C(C1=COCCO1)NCCN(C(C1CC1C1CCCO1)=O)C1CC1 C(=O)(C(CNC(C1CC(O)CN1C)=O)CC1CCCCC1)OC Cc1ccc2c(c1)SC(C(=O)N(C)CCNC(C1CCn3nncc3C1)=O)C2 c1(C(N(C)CC2CCN(C(=O)CCc3cnoc3)C2)=O)cnn2cccc2c1 C1(C)(CC(N2CC(NC(c3n(C(C)C)ccn3)=O)C(C)C2)=O)CCS(=O)(=O)N1 C1(O)(CNC(Cn2ccc(C)n2)=O)CCN(C(=O)C(C)Cc2ccc(O)cc2)C1 C(C)(C(=O)N1CCC1C(=O)NCC1CC1c1ccco1)OCC N1(C(c2ccc3nc(N4CCCC4)oc3c2)=O)CCC(O)C2(CCCNC2=O)C1 C1(O)(C(=O)Nc2c(C(=O)OC)scc2)CCN(C(C2CC2c2ccccc2Cl)=O)C1 C12(NC(C(C)OCCC=C)=O)CCOCC1CN(C(=O)C(C)=C(C)CC)C2 CCCCC(O)C(C)C(=O)NCC(CO)NC(=O)CC(CC)CC C1(C(N2C(C3(C(N(CC(C)(C)CC4CC4)C)=O)CC3)CCC2)=O)COCCC1C N1(C(c2cscc2C2CC2)=O)CCN(C(=O)Cc2cccc(F)c2F)C(CF)C1 C1(C(NOC(C)(C)C)=O)CN(C(=O)C2CC2)CC1(F)F.C1(=O)CO1 C1(N(C(c2ccc(C)nc2)=O)C)CCCN(C(C2CC(C3CC3)C2)=O)CC1 N1(CCS(CC)(=O)=O)CCC(NC(c2cc(SC)ccc2O)=O)C(O)C1 N1(C(C2N(C(=O)OC)CCC2)=O)CCN(C(c2sc(OC)nc2C)=O)C(CF)C1 c1(C2(C(=O)NC3C(NC(C=CCC)=O)C3)CC2)ccc(OC)c(F)c1 c1(COC)n[nH]c(=NC2CCCCN(C(c3nc(O)c(C)s3)=O)C2)o1 c1(OC)ccc(C(=O)NC2(CF)CCN(C(=O)CN3CCCC3)C2)c(C(F)F)n1 c1(CCCC(=O)NC2CCCC(C(=O)O)C2)cccc(C(=O)O)c1 O=S(=O)(c1ccc(C(F)F)c(Br)c1)Nc1ccncc1N1CCOCC1 C(C(C)C(F)C(=O)N1CCC(CCCO)C1)NC(CN(CCC)C)=O.C(C)(=O)O N1(CC(N2C(C(C)C)C(NC(=O)CCC(C)N(C)C)CC2)=O)OC(C)(C)CC1=O C#CC1CN(C(c2cc(CC3CC3)on2)=O)CCN1C(c1ccc(=N)[nH]n1)=O c1(CCC(=O)NC2(C)CN(C(c3cnn(CC(F)(F)F)c3)=O)C2)cccc(F)c1 C1(NC(C2C(OC)CCC2)=O)CN(C(=O)Cn2cnc([N+](=O)[O-])n2)CC2(CC2)C1 c1(OCCC(=O)NC(CNC(C=CC=CC)=O)(C)CO)ccc(F)cc1F C1(C(N(C)C(N)=O)=O)CCC(C)(C)CO1.c12cc(ccn1)C(=O)NCCNC2=O c1(CC)ccc(C(C2CCN(C(=O)Nc3scnc3C)CC2)CO)cc1 C1(C(C)(C)C)CN(C(=O)CNC(=O)NC2CC2)CC1NC(=O)C=Cc1ncco1 CCC(CC)(C(=O)NCCCCSC)C(C)C.C12CC3C=CC1N(C3)C2=O Fc1cccc2c(N3CCCC4(CCCCC4)C3)ccnc12 C1(C(=O)NC(C(C)(C)C)CNc2cncc(Cl)n2)CCC(C2CCC2)NC1=O c1(C(=O)OCCC#N)ccc(NCC2CC(=O)N(CCc3ccccc3)C2)cc1 CN1CCN(C(=O)C(=O)Nc2ncc(CCO)s2)CC(O)C1 n1(CC)c(CC(=O)NCCC(c2nnnn2C)C(N)=O)cc2ccccc12 C1(C(=O)NC(CNC(c2cccc(C)c2)=O)C2CCC2)Cc2cc(F)ccc2O1 c1(CC)cc(C(=O)NCC2CN(C(=O)Cn3nccn3)CC2N(C)C)n(C)n1 c1(NCC2N(C(CC(C)(C)C)=O)CCC2)ncnc2c1nnn2CC1CC1 c1(NC(C(Cc2ncccn2)NC(=O)OC(C)(C)C)=O)cc2nc(Br)sc2[nH]1 C12CCCCN1C2=O.Cc1ccc(CNC(C2CC2c2ccoc2)=O)o1 Cc1cc(CCNC(c2conc2CNC(=O)CCCC2CC2C)=O)nn1C CCCCC(CC)C(=O)N1CCCC1CCNC(c1nc(C(F)(F)F)cn1C)=O N1(C(C(C(=O)OCC)CC)=O)CCC(C2(NC(C3(OC)CCSC3)=O)CC2)CC1 c1(N2CC(C)(COC)OCC2)nc2cc[nH]c2c(=NCc2ccoc2)[nH]1 c1(CCC(c2cn(C3C(OC)COCC3)nn2)O)ccc(C)cc1F C(=O)(C(C)(C)C(C)C)NC(C(C)NC(c1ccc(NC(=O)OC)cc1)=O)C c1(C(N2CCC(OCCNC(C3CN4CCC3CC4)=O)C2)=O)cc([N+](=O)[O-])c[nH]1 CCC(C)(C)CC(=O)NC(C)(CNC(=O)Cc1ccccc1F)C1CCC1 CC1(c2ccc(Br)cc2)CCN(CC(=O)NCc2csc(-c3ccccc3)n2)CC1 C(=O)(C1=CCCC1P(C)(C)=O)NC(CN(C)C(C1C=CCC1)=O)(C)C c1(N2CCCC(C)(CC)CC2)[nH]c(=NCC2(C)CCCCC2)nc2scnc12 N1(C(C(=O)NCCOC)=O)CCCC(C(=O)NC(C)Cc2ccccn2)C1 C1(C(N(CCCO)CCC)=O)CN(C(C2(F)CCCC2)=O)CC12CC2 C1(NC(CC(C)F)=O)CN(C(c2ccc(C3CC3)o2)=O)CCC1F C(C1c2ccsc2CCN1C(C1CCC(=O)N1C)=O)NC(CCC(=C)C)=O C1(CC(=O)N(CCCNC(c2coc(C(F)F)c2)=O)CC)CCCC1O C1(NC(c2ncc(NC)nc2)=O)CC2CN(C(=O)C(=O)NC(C)C)CC2C1 c1(C(N2CCN(C(COCC=C)=O)CC2C(C)C)=O)cc(N)cc2c1OCCO2 C1(C(=O)NCC2N(C(C3C=CCCC3)=O)CCN(C)C2)CCc2ccccc2C1 c1(C(c2n(CC=C)nnn2)NC(C)Cc2cccs2)ccc(N(C)C)cc1 C1(F)(CNC(=O)CC2COC(=O)C2)CCN(C(C2(CC3CCC3)CC2)=O)CC1 c1(C(=O)NC2(C)CCN(C(c3ccc(C#C)cc3)=O)C2)cc(C)nc(Cl)c1N C1(C(=O)NC(CC)(C)CC)CCN(C(=O)CC2C(=O)NN=C2C)C12CC2 c1(CC)c(C(=O)N(C2CCN(C(=O)C(C)C#N)CC2)CC(C)C)csc1C C1(CNC(C(C)n2cncn2)=O)CC2COCC2N1C(=O)C(C)(C)CCl C=C1CCN(C(=O)CCCCOCC)C(C(=O)NC2COC(C(F)F)C2)C1 c1(CNC2C(OC)CN(C(COC)=O)C2)ccc(-n2ccnc2)c(OC)c1 N1(C(c2ccc(CC)nc2)=O)CCN(C(C2CC(O)(C(F)F)C2)=O)C2CC12 c1(NC(C(c2ccccc2)C)=O)ccccc1-c1cccc(C(=O)N(C)C)c1 c1(NC(=O)NC(C2CC2C2CC2)C)ccc(C#N)c(Cl)c1 N1(C(C(C)SCC)=O)CC(NC(c2ccc(=O)n(CCOC)c2)=O)C(C)(C)C1 N1(C(C(C)OCC)=O)CCC2(CCCN2C(C2CC(=O)CCO2)=O)C1 C1(COC)(NC(=O)CCC)CCN(C(=O)CCC(=O)C2CC2c2ccsc2)CC1 Cc1cc(C(N2CCC3CN(C(C4(C)CCCC4)=O)CC23)=O)cc(F)c1C n1(C(C)(C)C)nnc(C(=O)NC(CNC(c2scnc2C(F)(F)F)=O)C2CC2)n1 C1(C(N2CC(CNC(COC)=O)C3C2C3)=O)C2(CCC2)C12CCC2 C(CCC(C)(C)OC(C1(CSC)CC1)C)NC(CN(C(=O)OCC)C)=O N#CC1=C(C(=O)NCC2CCN(C(c3ccncc3F)=O)C2)CCC1 C1(NC(C)=O)CC12CCC(NC(c1cc(-c3cccc(Br)c3)no1)=O)CC2 C1(C(=O)NC(CC(=O)NCC2(O)CCC2)C2CC2)CC2(C1)CC(O)C2 N1(C(c2c(C)ccc(OC)c2)=O)CC(NC(=O)C(C)CC(C)(F)F)CC12CCC2 c1(C(N2CCC(CNC(c3c(Cl)cc(Cl)nc3Cl)=O)C2)=O)c(F)cc(O)cc1F C(=O)(CN1C(=O)CCCc2sccc21)NCC(CN(C(c1c(C)nc[nH]1)=O)C)O c1(C(=O)NCC2(NC(C3C(OCC)CC3)=O)CCOC2)cncn(C)c1=O C1(CC)CN(C(=O)C(C)C2CCC2)CC1C(N1CC[Si](C)(C)C1)=O C12(C(=O)NC(C3N(C(c4cncc(C)n4)=O)CCCC3)C)CCC(CC1)C2(C)C c1(C(N(C)CC2CCCC2NC(=O)Cc2cnnn2C)=O)n[nH]cc1[N+](=O)[O-] C1(CC(=O)NC(c2ccccc2)CC)CCC(NC(=O)Cn2ccc(C)c2)CC1 CC(C)C(O)(C(=O)N1CC(C)(NC(=O)C(C)NS(C)(=O)=O)C1)C(F)(F)F c1(CNC(=O)NCc2c(C)nc(Br)o2)cn2cc(Cl)cc(C)c2n1 C1(COC)(NC(=O)Cc2csnn2)CCN(C(c2ccc(C3CC3)s2)=O)C1 c1(CCC)cc(C(=O)NCCN(C(=O)C=Cc2ccco2)C(C)C)ccn1 C(c1ccc(=N)[nH]c1)=CC(=O)NC1C(NC(C2CN(C(C)(C)C)C(=O)C2)=O)CC1 C1(C(=O)NCC(C)(C)OCC(=O)NCC(C(=O)OCC)(C)O)CCCCC1(C)C c1(C(=O)NCC2(C)CC(NC(=O)CN3CCSCC3)C2)cnc2[nH]nnc2c1 C1(C(=O)NC(CC)CO)(CC)CN(C(=O)C(C)CN(C)C(C)=O)C1 N1(C(c2c(C(=O)OCC)con2)=O)CCC(NC(=O)C(O)C(C)(C)C)CC1C C1(C(=O)NC2CC(CCNC(c3cncn(C)c3=O)=O)C2)CC(C2CCCC2)C1 S(=O)(=O)(c1cccs1)N(CC(=O)N(CCC(C)NC(c1ccc(F)o1)=O)C)C CC1(C)CC(O)(CC(=O)N(C2CC2)CC2CCCN2C(=O)C2=CCCSC2)CO1 n1(CCCNC2C(F)(F)C2)cccc1C(F)(F)F C1(C2C(NC(C(F)OC)=O)CCO2)CCN(C(=O)CCn2cccn2)CC1 C1(OC)CCC2(C(N3CCCCC3C3(NC(c4cccc(N)c4)=O)CC3)=O)CCC12 C(=O)(CCCCC(F)F)N1C(CN(C(COCCC=C)=O)C)CCC1 CC1CCN(C(c2nocc2C(C)(C)C)=O)C1CNC(c1coc(C2CC2)n1)=O N1(C(c2c(C)cns2)=O)CCC(NC(=O)CNC(=O)CN(C)C)C1C1CC1 CC1CCC(C)N1CC(=O)NCCOCCCNC(C1CC(=O)N1)=O C1(CNC(CC(CC)(F)F)=O)CCC2CN(C(=O)CCNC(=O)CO)CC12 O=C1OC2CCN(C(c3cn(C4CCC4)nn3)=O)CC2O1 N1(C(CSCC(C)=O)=O)CCCC12CCN(C(=O)C=CC1CCC1)C2 c1(NC2CC(CCNC(c3c(CC)nc(C)nc3)=O)C2)ncc2c(n1)CCCC2 c1(C(=O)NC2(CF)CCN(C(C3CC(C)C3)=O)C2)cnc2c(c1)CCOC2 C1(CNC(C2CCCC2)=O)CCC2CN(C(=O)CCc3cnc[nH]3)CCC2C1 C1(C#N)(C(=O)NC(C(C)NC(c2cc(CCC)on2)=O)CO)CC=CC1 CN1CCOCC1C(=O)NCc1ccc(C(N2CC(O)CC2C2CC2)=O)cc1 C(c1ccc([N+](=O)[O-])cc1)=CC(N1CCN(C(COC(CC)C)=O)CC1)=O Nc1ccc(C(N2CCC(CF)(NC(=O)Cc3sccc3Cl)C2)=O)cc1O Cc1cc(Cl)cc(N)c1C(=O)NC1CC1CNC(=O)C(C)CC(C)(C)C CC(C)(C(=O)NCCc1n[nH]cc1C(=O)NC1CCNC1=O)c1ccno1 C(C1=NOC2OCCCC12)N1CCC(=O)C(c2ccc([N+](=O)[O-])cc2)C1 C(C(CNC(c1ccc(OC(C)C)nc1)=O)S(C)(=O)=O)NC(c1cc(C)[nH]n1)=O C1(CNC(CCOC)=O)CCCCC1NC(=O)CC1(O)CCOC1 c1(NC(C(CC=C)c2ccccc2)=O)cnccc1C#N.C12CN(CCO1)C2=O Cc1coc(C(C)(C)C)c1C(N1CC(F)(CNC(C2(C)CC2(F)F)=O)C1)=O Cc1cc(N)c(C(N2CCC=C(CNC(=O)C3=C(Cl)CCC3)C2)=O)c(F)c1 C1(C(=O)NC(CCC)C)CN(Cc2ccc(OC)nc2)CC(F)(F)C1 N1(C(Cc2ccc(C#C)s2)=O)CCN(C(c2cnc(C(N)=O)cn2)=O)CC1CO c1(C(N2C(C)CC(NC(c3n[nH]c(C)c3C(F)(F)F)=O)C2)=O)ccc(O)c(F)c1 CN1CC(O)CC1C(=O)NCc1ccc(C(=O)NCC2CC2CO)nc1 CCCCCC(=O)NCC(=O)N(C1CC1)CC1CN(C(=O)CCS(C)=O)CCO1 N1(C(=O)C=Cc2ccccc2Br)CCC2CN(c3ncc4[nH]ncc4n3)CCC12 C1(CCCC)CN(C(c2n[nH]cc2OC)=O)CCN1C(C1C2COCC12)=O C1(NC(C(C2CCCN(C(c3cccs3)=O)C2)(C)C)=O)CCOCC1F C1(C(=O)NCCCNC(c2cc(CS(C)(=O)=O)on2)=O)CCCC1(F)F CCC(CC)(CO)C(=O)N1CCCC(NC(c2cccn2C2CCCC2)=O)C1 c1(C(=O)OC)c(C(N2CC(NC(C34CCC3C4)=O)C(C)C2)=O)n[nH]c1C c1(NC(c2cc(Cl)sc2Cl)c2n(CCCSCC)nnn2)ccc(F)c(CC)n1 N1(C(C(C(C)C)(F)CNC(C2(SC3CC3)CC2)=O)=O)CC(C2CCCCC2)C1 CC(C)CC(C)(O)CNC(C1CCC1NC(C1CC1[N+](=O)[O-])=O)=O c1(CCSCO)cc(=NC(=O)C2(N(C)C)CC(CF)C2)[nH][nH]1.C(=O)OC c1(OC)cncc(C(=O)NCC(C(C)(C)C)NC(C2CN(C)C(=O)N2)=O)c1 C(=O)(CC(C)C(C)(C)NC(=O)Cc1ccn(C)n1)NC(C)C(C)(C)C CC(C)(C)CC(O)C(=O)NC1CN(C(=O)CCc2ccccc2F)CC1O C1(C(N(CC(CNC(Cc2cc(C)nn2C)=O)(C)C)C)=O)CCCC(C)(C)C1 C1(CC(=O)NCC2CC3CCC2CC3)C2CCCC2N1C(c1ccc(F)c(F)c1)=O N1(C(c2c(C)ocn2)=O)CCN(C(=O)CSCc2ncc[nH]2)CC1C Cc1cccc([N+](=O)[O-])c1C(=O)NC(C)CNC(C1CC2CCCCCCC12)=O C1(CNC(C2(C#C)CC2)=O)CN(C(C2CC2(C)CC)=O)CC12CC2 CP(C)(=O)C(O)C(=O)NCC1(CNC(c2cccc(OC(F)F)c2)=O)CC1 N1(C(=O)COCC2CCC2)CCC(C2CCCN2C(c2cc(O)ncn2)=O)CC1 C(CC(C(=O)NCCc1ccncc1C)NC(=O)CC1CC2(CCC2)C1)=CC C1(C(=O)NCC2CCC2C(=O)NCc2occc2C(C)C)(OC)CCOC1 C1(C)(C(=O)NCC2CC(NC(CCC(=O)OC)=O)C2)CCC(C)=C(C)C1 C1(NC(c2n(CC)nnn2)CCc2ccc(F)cc2)CC2C=CCC(C1)C2 C1(OC)CN(C(c2cn(C)c(=O)n2C)=O)C(C)(CNC(=O)CCc2cc[nH]n2)C1 c1(C(=O)OCCc2ccccc2Br)ncccc1-c1ccncc1 Cc1ccc(Cl)cc1OCC(=O)NCC1CC2CCC1N2C(=O)Cc1cscn1 c1(C(=O)NC2CCC(CCNC(C3CC=CCC3)=O)C2)cncc2nc[nH]c12 N1(C(CNC(CC)=O)=O)CC(C2CCN(C(C3Cc4ccccc4O3)=O)CC2)C1 C=CC(C)(CC)C(=O)N1CCC(CO)C(NC(=O)CC2CCOC2C)C1 Cc1cccc2[nH]cc(C(=O)NC(CNC(=O)CC(C)O)C3CC3)c12 N1(C(CS(=O)(=O)NC)=O)CCCC12CCN(C(c1ccc(C#N)c(Cl)c1)=O)C2 CC1C(=O)NCC(=O)N1CCO.c1(C(F)(F)F)ncc[nH]1 c1(C(N(C2CCN(CCc3ccc(C(=O)OC)o3)C2)C)=O)noc2c1CCC2 C1(N)CCN(C(=O)CN(c2ccoc2)C)C1.C(=O)(CCNC)N(S(C)(=O)=O)C NS(=O)(=O)c1ccc(CC(=O)NCCN(C(C2CCCO2)=O)C2CC2)s1 C(=O)(C(CC)CCOC(=O)C(C)(C)C)NC1(CCNC(C(CCC)O)=O)CC1 N1(C(C#CC)=O)CC2CN(S(=O)(=O)C3CC3)CC2C1 N1(C(C(=O)NCCNC(C)=O)=O)CC(NC(C2CCCC(=O)CC2)=O)CC(C)C1 C1(C(=O)NCCCCCNC(CS(=O)(=O)NC)=O)C2CC3C(C2=O)C13 C(=O)(C(F)(F)CC=C)NC1CC2C(NC(C(C=C)C)=O)C2C1 CON(CCC(=O)NC1(C(F)F)CCC1)C(=O)C(C)CC(C)C(C)=O C1(C(=O)NCC2(CC(=O)OC)CCC2)(OC)CC(C)CC(C)C1 Cc1cc(C)cc(C=CC(N2CCCN(C(=O)C(c3cncnc3)C)CC2)=O)c1 N1(CC#C)CCN(C(=O)CN(C(C2(F)CCOCC2)=O)C(C)C)CC1=O c1(C(=O)NC2CCCC(CN(C(CC3(OC)CC3)=O)C)C2)ccc2c[nH]nc2n1 C1(CNC(c2c(C(C)C)nns2)=O)CN(C(C2COC2)=O)CC1C(F)(F)F N1(C(c2c(CC=C)cccc2)=O)CCN(C(c2ccc(OC)s2)=O)C(C)C1C C(=O)(C(C)C(C)(C)C)NCC(C1(O)CCN(C(C2SC3C=CC2CC3)=O)C1)C C(CNC(C1(C#N)CC1C)=O)(CCNC(=O)Cn1nccn1)OC N1(C(C2(OC)CCC2)=O)CCCC(C(C)(O)CNC(=O)COc2ccsn2)C1 S(=O)(=O)(c1c(F)cccc1F)NCC(=O)NCC(CO)NC(C1C(C)C1)=O c1(OC)cc(C)sc1C(=O)NCC1CN(C(=O)CNC=O)CC1O C1(CNC(c2c(C)noc2)=O)CCC(C)N(C(c2ccnc(Cl)c2F)=O)C1 C1(NC(CCOC)=O)CN(C(c2cnsn2)=O)CC1F C(C)(C(C(C)C)Nc1ccnc(C)n1)NC(C(c1cccc(Cl)c1)OCC)=O c1(C(N(C2C(NC(C=CC(=O)N(C)C)=O)CCCC2)C)=O)cnc(C(C)C)n1C c1(C(N2C(CN(C(c3n(CC)c(O)nc3)=O)C)CCC2)=O)cn2c(n1)CCC2 c1(C(=O)NCC2CN(C(C(C)N3CCCC3)=O)C2)ccc(C(F)F)nc1O CCC(O)C(C)C(=O)NC1CN(C(=O)CC2CCCC(OC)C2)CC1(C)C C1(C(=O)NCC(C(C)(C)C)OC)CCCN(C(C23CSCC2C3)=O)C1C N1(C(CC(C)(C)C2(C)CC2)=O)Cc2[nH]nc(-c3cnn(C4COC4)c3)c2C1 c1(C(C)(C)C)cc(C(N2CC3CC2C3NC(C2CC2[N+](=O)[O-])=O)=O)ccc1Cl c1(C(=O)NCC(C)NC(C(C)OC(=O)OCC)=O)cc(C)nc2[nH]nc(O)c12 C(=O)(C(C)(F)C(C)(C)F)NCC(C)CN(C(=O)CCS(=O)(=O)N(C)C)C C(=O)(CC(C)(F)F)N1CCC(C(N2CCC(N(C)C)C2)=O)C1 CC(CC(N)=O)C(=O)NCC1CN(C(=O)C=CC(C)(C)C)C2CC12 C12CCCC1NC(=O)CCOCCCNC2=O.C1(CC)COCC1O C1(CNC(c2c(CC(C)C)nc(C)s2)=O)CC2CCC(C1)N2C(=O)C(C)C(C)C C1(C(N(C2CCN(C(c3cnc(N)cn3)=O)C2)C)=O)CC(=O)N(O)C1 c1(C(N2CCN(CC)CC2)C(=O)NC(CC)(C)C)ccc2c(c1)C(=O)NCCO2 c1(OC)cccc(C(N2C(C(=O)Nc3ccc(CO)c(Cl)c3)CC3CC23)=O)c1F N1(C(COCC#C)=O)CC2(CCN(C(=O)C(C)Cc3ccccc3Cl)C2)C1 n1(CC(=O)N(CC(=O)NCC2CC(CF)C2)CC)nnnc1C n1(CCC)nccc1C(C(=O)NC(C)C1CC1)N(C(CC)CC)C1CC1 CC(C)(CS(C)(=O)=O)C(=O)NCC1(F)CCCN(C(c2ccc(Cl)cc2)=O)C1 c1(C(=O)NC2C(NC(c3cc(COC)no3)=O)CC2)cncc(F)c1 c1(C2(NC(C3CCCCC3)=O)C(C)C2)cccc(C2(C)CC2)c1 Cc1nc(-c2ccsc2)sc1C(=O)NCCC1(CNC(C2CCC(C)O2)=O)CC1 CC1CC(C(=O)N(C2CCN(C(=O)CC(C)C3CCCCC3)C2)CC2CC2)=NO1 c1(C(=O)NCC2(NC(c3c(C)noc3C)=O)CC2)ccnc(OCC2CC2)c1F N1(C(C2CC(SC)C2)=O)C2CCC1CC(CC(C)NC(c1cncc(C)c1)=O)C2 C1(CN(C(c2nc(CC)oc2)=O)C)C2CN(C(=O)Cc3csc(COC)n3)CC12 c1(C(=O)OC)c(C(N2CCCC2C(C)NC(=O)C=CC(C)(C)C)=O)cnn1C C(CN=C(NC1CC1c1ccsc1)N(C)CCN1CCOCC1)C1C(C)C1 N1(C(C(C(C)C)NC=O)=O)CC(C2CN(C(=O)C(C3CC3)SCC(N)=O)C2)C1 c1(N(C)CC2CCN(Cc3c(C)nccc3)C2)ncnn2cccc12 C1(OC)CC(CCNC(=O)CN(C)C)N(C(c2ccc(C3CCOC3)cc2)=O)C1 C1(Cc2cn(CC#CCC)nn2)CCCCN1.C(=O)CCCN1CCOCC1 CN1CC2(CN(C(c3cc(C(C)(C)C)cc(Br)c3)=O)C2)OC1=O C1(COC)CN(C(=O)C(F)=C(C)C)CCN1C(=O)Cc1c(O)ncnc1O NC(=O)CCCC(=O)NCCN1CCN(C(=O)Cn2ccc(C(F)F)n2)CC1 C1(NC(CC(C)(C)OC)=O)CC(NC(=O)CCC(CF)CF)C12CCOCC2 C1(NC(CC=C)=O)CC2C(NC(c3sc(F)cc3C)=O)C2C1 CC(CC(=O)NCCOCCOCCCNC(c1ccc(O)nc1)=O)P(C)(C)=O N1(C(C(CC#C)C)=O)CCC(CCNC(=O)CCc2n[nH]c(=N)s2)CC1C C=CC1CC(NC(=O)CCCNC(=O)C(C)NC(=O)NC)C1 c1(C(=O)NCCCN(C2CCCC2)C(C2CC3CC2C3)=O)cccc2ccoc12 C1(C(C(=O)NCCOCC2CC2)N(CC(F)(F)Br)C)CC1C1CC1 N1(C(C=C(C)Cl)=O)CCC2CCC(NC(c3cc(Cl)nc(Cl)c3)=O)C1C2 C1(NC(=O)NCc2cc(Br)c(F)cc2Cl)COc2ccccc2C1 N1(C(CCN2CCN(C)CC2)=O)CCC2(C1)CN(C(C1(C)CCC(=O)NC1)=O)C2 c1(C(N2CC3C(CNC(C(CC#C)O)=O)(CC3)C2)=O)coc(S(N)(=O)=O)c1 C(=O)(CCCC(F)(F)F)OCCOCCNC(CCC(C)N(C)C)=O C(=O)(C1=C(CC)OCCC1)NC(CC#C)C(=O)NCCOC1CCCCC1 Cc1cn2c(n1)C(C(=O)NCCN1CCN(C(=O)C=CC(F)(F)F)CC1)CCC2 Cc1ccn2nc(C(=O)NCC3CCN(C(=O)CC4C=CCC4)C34CC4)nc2n1 c1(C(=O)NCCC(C)NC(CC(CCC)(C)O)=O)ccc2nc(N(C)C)oc2c1 N1(C(C(CCC)C#N)=O)CCCC(C)(CNC(C2C3CC4C(C3)C24)=O)C1 N1(C(C(C)(C)C(N)=O)=O)CCC(NC(=O)CC2CC=CC2)C(CO)CC1 C(=O)(CC(CC)C(C)(C)C)NC1(CC=C)CCCN(C(C2C(C)(C)C2(F)F)=O)C1 CC1(C)OC2(CNC(=O)C=CC3CCC3)CC1(NC(C1CC3CCC(C1)S3)=O)C2 c1(CC(=O)NCC2CC(C)N(C(=O)Cc3nc[nH]n3)C2)cc(Cl)cc2c1OCC2 c1(NC(C(C)C)C(C)NC(=O)C=Cc2cnn(C)c2)ncc(C#N)cc1Cl C1(CNC(=O)CSCCNC(C2(C3CC3)CCCO2)=O)CCCC(F)C1 c1(OC)ccccc1C=CC(=O)NC1CC2CC(NC(=O)CCCCSC)C1C2 C12(C(N3CCC(O)(C(C)CNC(C4(C)CCCOC4)=O)C3)=O)CC(C)(C1)OC2C C1(C(C)(C)NC(=O)CC2CCCO2)CCN(C(=O)CCCc2csc(=N)[nH]2)CC1 CC(C)S(=O)(=O)C(C)C(=O)NC1CC(C)(NC(=O)CC2(C#N)CCCCC2)C1 N1(C(C2N(C)CCOC2)=O)CCC(NC(=O)CC#N)C(c2ccccc2)C1 C(CC(C(=O)Nc1ccc(NC(N)=O)cc1)NC(=O)CCC(C)C)=CC CC(C)C(O)CC(=O)NCC1COCCN(C(c2cnc(C(C)O)s2)=O)C1 c1(C(=O)NCC2C(CNC(Cn3c(C(C)C)nnn3)=O)C2)nccc2[nH]ccc12 C1(NC(C2(F)CCCC2)=O)CN(C(=O)Cc2ccc(Cl)cc2Cl)CC12CC2 C1(NC(Cc2cc(OC)c(C)cc2)=O)CN(C(C2CC2(C)C)=O)C2(CCCC2)C1 CCCCCCCCCC(C)CC(=O)NC1CCOc2ccc(Br)cc21 C12(NC(=O)CSCc3cccs3)CCN(C(c3ccc(N(C)C)cc3)=O)CC1C2 C1(C(=O)NCC2(O)CN(C(C3CCC(OCC)CC3)=O)C2)CC12CCOCC2 CC1(C)CC(O)(CC(=O)NC2CC(CNC(=O)C3=C(Cl)CCC3)C2)CO1 C12(CNC(C3CN(C)C3)=O)CCC(CN(C(=O)COc3c(Cl)cccc3Cl)C1)C2 C1(NC(C=C(C)Cl)=O)(CNC(=O)C=CC(=O)NCCOC)CCCCC1C c1(N(CCC(C)O)C)nc(=NCC2C(F)(F)C23CCCC3)[nH]c2c1CCCC2 c1(OC)sccc1C(=O)NCC(O)CNC(=O)CSCc1cscn1 c1(SC(CC=C)CC)cc(S(=O)(=O)c2nnco2)ccc1O CCC(C)C(C(=O)N1CCC(CF)C1)N(C)C(c1nnc(S)n1C)=O C1(CCNC(C2CC(C)N(C)C2)=O)CCCN(C(=O)Cc2ccnc(CO)c2)CC1 N1(C(C2(CC#N)COC2)=O)CCC2CN(C(c3cc(F)ccc3F)=O)CCC12 CC1=C(c2ccco2)CN(C(C23CC2COC3(C)C)=O)CC1.N12CCC(C1)NC2=O C(=O)(CC(CNC(=O)NCc1ccc(Br)s1)C(C)C)OC CC(C)(CS(C)(=O)=O)C(=O)NC1CC1CNC(=O)C(F)(F)C(C)(C)O C(=O)(C(F)CC(C)C)NCCN(C(c1cc(CCC)ncc1)=O)C C(CNC(=O)C1=CCCOC1)(C(C)C(C)C)NC(CCc1ccc(C)s1)=O C1(C(=O)NCC(C)N(C(CCc2cc(C)on2)=O)C)CCCCN(C)C1=O Cc1[nH]c2ccc(F)cc2c1CO.C12CCC1CC(=O)NCC2 CCC(C)(C(=O)NCCCC(N1CC(N(C)C)C(C)C1)=O)OC N1(C(c2c(C)nn(C(C)C)c2)=O)CCN(C(C2(N(C)C)CCCCC2)=O)CC1CO N1(C(c2ccc(C#C)cc2)=O)CC(NC(=O)C(c2ccccc2)C)CC2(CC2)C1 N1(C(C2(C)CC(NC(=O)CC3COC(=O)C3)C2)=O)CC(O)C(N=[N+]=[N-])C1 CC1(C)CN(C(=O)C=CC2CCOC2)CC1CNC(C1CC2CC1C2)=O C(=O)(C(C)N=[N+]=[N-])N(CCC(=O)NCC(COC)(F)F)C O(NC(=O)CCC1CCCN(C(=O)CNC=O)C1)CC#C c1(C(=O)NCCNC(c2nc(CC)sc2N)=O)ccc(C)c2cccnc12 CC1CNC(=O)CN1C(=O)CCCCNC(C1CSCC(=O)N1)=O c1(-c2cn(CC(C)C(N3CC=CC3(C)C)=O)nn2)ccnc(OC(C)(C)C)c1 C(=O)(C(C)(F)C(=O)N1CC(O)(C2CCCN2C(=O)Cc2cc[nH]n2)C1)OC S(=O)(=O)(c1ccc(C)c(C)c1)NC(c1ccc(=NCc2ccc(OC)o2)[nH]c1)=O CC1CN(C(c2cccc(N(C)C)c2)=O)CC1NC(C1CC(=O)CO1)=O c1(C(C(=O)NC(C2(O)CN(C(C3(C4CC4)CC3)=O)C2)C)=O)cnn(C(F)F)c1 C1(C)(CC)C=C(C(=O)N(CCCCCCNC(=O)C(C(C)C)NS(C)(=O)=O)C)C1 C1(CNC(CC(C)SC)=O)CN(C(=O)C(F)=CC2CC2)CC1(F)F c1(C(=O)NC(CC)CNC(=O)C(C)(C)C2CCCC2)ccc(=O)n2c1CCC2 N1(C(=O)NC(C)Cc2ccncc2)CCCCC(C)(F)C1 C(=O)(CC(C(C)(C)C)NC(=O)C(C)n1ccnc1)NC(C#C)CC1CCCC1 c1(CC)cc(N)c(C(=O)NC2CC2NC(c2ccc(OCCO)cc2)=O)cc1F Cc1cc(=O)c(C(N2CC3(CC3)CC2C(N2CCC(CN=[N+]=[N-])C2)=O)=O)c[nH]1 c1(CC)ncnc(Nc2ccc(OCC(C)C)cc2F)c1F c1(OCC(=O)NC(CC)(C)CNC(=O)CCC#N)cc(Br)ccc1Cl c1(NCCOC)ccc2c(c1)OCO2.n1(CCCOC)nnnc1CC(C)C N1(C(C=C(C)C)=O)CC2CC(C(=O)NC3(C)CS(=O)(=O)C3)C(C2)C1 CN1CC(O)CC1CNC(=O)C(O)C1CN(C(C2(C(N)=O)CC2)=O)C1 Cc1cnccc1C=CC(N1CC(C)C(C)(CNC(=O)C2=CCCCC2)C1)=O C1(NC(C=C(C)Cl)=O)CCN(C(c2ccc(=O)n(CC(C)O)c2)=O)C12CCCC2 C1(C)(NC(C2(N(C(=O)CN(CC(F)F)C)C)CC2)=O)CCCC1 CC1(C)CCCC(CCOC(c2ccc(F)c(C#N)c2)=O)O1 C1(NC(COCC(=C)C)=O)CCOC(C(=O)NCCN2CCOC2=O)C1 c1(C(=O)NC(CCC)CCCNC(c2ccoc2)=O)cccc2sccc12 c1(CNC(NC2CC(=O)N(c3ccccc3F)C2)=S)ccc(S(=O)(=O)CO)o1 c1(CC#N)cccc(C(=O)NC(CNC(C2CC23CCCC3)=O)CO)c1 N1(C(c2scc(C)c2)=O)CCOC2(C1)CN(c1ncc(F)cn1)C2 Cc1cc(C(N2CCCC(N(C)C(c3ccsc3Cl)=O)CC2)=O)cc(C)c1O CCC(CN(C(=O)CNC(=O)COC(C)=O)C)NC(=O)C(O)C1CCCC1 CC1CC(N=c2cc[nH]cc2C#N)CN1C(c1ocnc1C(F)F)=O CC1CC2(CCN(C(=O)CCNC(=O)C=CCl)CC2)CN1C(=O)Cc1cncs1 N1(C(c2nc(C(C)(F)F)cs2)C(=O)NCC(C)C)CCC2(CC=CCO2)C1 c1(C(N2CCCC(F)(CNC(C(C)C(C)(C)C)=O)C2)=O)cccc2[nH]ncc12 C1(C(=O)NC(C(=O)OCC)Cc2ccncn2)(CC)CCOCC1 N1(C(C(CC=C)C)=O)CC2CCCCC2(NC(=O)CCC2CC(F)(F)C2)C1 N1(C(c2cnn(C(C)C)c2N)=O)CCC(NC(c2cc3sccc3[nH]2)=O)C(C)C1 N1(C(C2(COC)CCCC2)=O)CC2CCC1CN2C(=O)CC1CCCCN1 C(CCCC=C)(C(=O)NCCC1(C)CCN(C)C1)NC1(n2cc(CN)cn2)CC1 C1(C)(C(=O)NC2CC(NC(CC3(C(=C)F)CCC3)=O)C2)CCC(O)CC1 C1(OC)CCCC1C(=O)NC1(C)CC(NC(=O)C=C(Cl)Cl)C1 C12(NC(C(CC)OC)=O)CCC(C1)N(C(=O)C=CC1CCCCC1)C2 CC1(C)CCC(CNC(=O)CCCC2CC2)N(C(=O)C=Cc2ccncn2)C1 c1(OC)cc(C(=O)NC2CC3(NC(=O)C(O)CCSC)COC2C3)cnc1O N1(C(COCCCOCCNC(COC)=O)=O)CCC(C(=O)N)CC1C.C(C)(C)O Cc1nn(C)cc1CC(=O)NC1(C(=O)NCC(O)Cn2cccn2)CCN(C)C1 N1(C(COC2CN(C(C)=O)C2)=O)CCCC(C)(C(=O)NC(C2CC2)C2CC2)C1 N1(C(CN(CC)CC)=O)CCCN(C(c2c(Cl)n[nH]c2C2CC2)=O)CC1 C1(NC(C(C2CC2)OCC)=O)CCC2CC1CN2C(=O)C(C)CCN(C)C N1(C(c2c(C)cccc2)=O)CCC(C)(C)C(NC(=O)C(O)C2CCCC2)C1 C1(C(N2CC(C)C(CNC(c3csc(Cl)c3)=O)C2)=O)CC2CC1C1CC21 C1(C(C)(C)C)(C(=O)N(C(CC)CNC(C2CC(CCO)C2)=O)CC)CCCC1 c1(C(N2CC(COC)(CNC(=O)CC3(C)CCC3)C2)=O)nc[nH]c2ncnc1-2 C(c1cc(Cl)c2c(c1)OCCO2)=CC(N1CC(C)C(NC(C2CC2C#N)=O)C1)=O C12(NC(c3c(F)ccc(C)n3)=O)CCCN(C(=O)C(=O)C(F)(F)F)CC1C2 c1(C(=O)N(CCCN2CCCC2)C)c(NCc2cc(O)cc(Br)c2)cccc1F C(=O)(CCC(CC)CC)NC(CC#C)C(=O)NCc1noc(C(N)=O)n1 N1(C(c2ncn(C)c(=O)c2)=O)CCC2(CC(NC(=O)CCC(F)(F)F)CO2)C1 n1(CCSC)nnnc1C(c1ncsc1C)NCc1ncnn1C(C)C C(c1ccc(C(=O)OC)o1)=CC(=O)NC1(CNC(C(CSC)C)=O)CCCC1 C(N=c1[nH]c(=NCc2ccn(C)c(=O)c2)[nH]c2c1CCC2)C1OCCN(C)C1 CCCC(C(=O)NC1CN(CC(=O)Nc2ccc(F)cc2F)CC1(C)C)C(C)C Cc1cnc(NCc2ncoc2C(C)(C)C)c(S(=O)(=O)N2CCCN(C)CC2)c1 c1(NC(CNC(CCOC)=O)C(C)C)nnc(C#N)s1 n12cc(nn1)CCCCN(C(N)=O)NC(=O)C2.c1(C(=O)NCC(C)C)cccs1 C=CCC(CC=C)C(=O)NCC1CN(C(=O)COCc2ccccc2)CCCO1 N1(C(C(CC)NC)=O)CCCC12CN(C(=O)Cn1ncc3ccccc13)C2 c1(C(N2CCC(NC(C(C)C)=O)C23CC3)=O)cc(Cl)c(N)cc1F N1(C(C(=O)NCCC(=O)OCC)C2CCC2CC)CC=C(C(C)(C)C=C)CC1 Cc1ccc(C(=O)NCC2CN(C(c3c(Cl)sc(C)c3C)=O)CC23CC3)nc1C C1(NC(c2cc(COC)on2)=O)CC12CC(NC(c1ccc(C(F)F)nc1)=O)C2 C(=O)(CC1CS(=O)(=O)c2ccccc21)NCC(CC(C)C)NC(C1(C#C)CC1)=O c1(C(=O)NCC2C(NC(c3cc(C)cc(O)n3)=O)C2)cnc2n1CCCC2 CC(CC(=O)NC1CC(NC(c2ccsc2C(F)(F)F)=O)C1)C(C)(C)C CC1CCC(C(=O)Nc2ccc(OCF)cc2)CN1C(c1c[nH]c(C(N)=O)c1)=O N1(C(C2CC(C(=O)NC(C3C(CC)OCC3)=O)C2)=O)CC=CC1(C)C C1(C(C)C)CN(C(C2CC(C)N(C(c3ccnn3C(C)C)=O)C2)=O)CCN1C C12CCCC1NC(=O)C2.C(C)(C)(C)OCCO.C=CCN(CCO)CC N1(C2CN(C(C3CCC(=O)C3)=O)C2)CCN(C(=O)Cc2ccc(C(=O)O)s2)CC1 C#CCC(CC#C)NC(c1ncoc1CNC(C1(Cl)CC1(F)F)=O)=O CC(C)CC(CNC(C1CC2CCCC2C1)=O)C(=O)NCCOC1(C)CCC1 N1(C(CCc2scc(C)n2)=O)CC2CC(NC(c3ccco3)=O)C(C2)C1 c1(NC(C(=O)N(C(C)CNC(c2cc(C3CC3)[nH]n2)=O)CC)C)ccccc1 C1(NC(C2CCc3c[nH]nc3C2)=O)CN(C(C2CSCCS2)=O)CCC12CCC2 C1(C(=O)NCc2n(CC)ncc2)COCCC1NC(=O)CC1(N(C)C)CCCC1 C1(CCCNC(c2c(OC)ccs2)=O)CCCCN1C(=O)CCCN(C)C(C)=O C1(C(C)C)CN(C(=O)Cc2cc[nH]n2)CC1C(=O)N(CCC(F)(F)F)C1CC1 CC12CN(CCCc3cccc(Br)c3)CC1(c1nc(C(F)(F)F)no1)C2 C1(O)(CC(=O)NC2(C=C)CCC2)CCN(C(=O)C(CC=C)NCNCC(C)=O)CC1 Cc1nccnc1C(=O)N(CC(C)O)CCNC(=O)C(C)(C)n1cnnn1 C1(OC)CN(C(=O)C#CC2CC2)CCC1NC(c1cc(C)oc1C)=O CC(=O)CCCC(C)C(=O)NCCCCCC(=O)NCCC1CCC1 C1(OC)CCN(CCn2cc(C(C)COC)nn2)C(C)C1 N1(C(COC2(C)CCC2)=O)CC2CCC(C1)N2C(C1CC1C1CCCC1)=O c1(C(=O)NCC2C(C)CCN(C(=O)CN(C)C(N)=O)C2)[nH]nc2c1COC2(C)C C=C(Cl)CC(C(=O)Nc1cnc(C)c(CC)c1)NC(=O)C(C)C(F)F c1(CNc2ncc(-c3cccc(SC)c3)s2)cnc(O)cc1O c1(C(=O)NCC(C)N(C(=O)CCC(C)(C)C)C)nc(Br)n2c1COCC2 Cc1c(C(=O)N=c2cncc[nH]2)cc(F)cc1[N+](=O)[O-].c1ccc(S(C)(=O)=O)c(F)c1 N1(C(C(C)S(N)(=O)=O)=O)CC2(C1)CN(C(c1ccn3ncccc13)=O)CC2CO c1(CCC(N2CCCC(C(F)F)C2)=O)ccc(COC(F)F)cc1 c1(C(=O)NC(CNC(c2cc(C)on2)=O)C)nnc2ccccc2c1O c1(CC)ccc(C(C)NC(c2nnnn2CCC2CC2)C(C)C2CC2)s1 C(c1ccc2occc2c1)=CC(N1C(CN(C(=O)C(C)(C)C)C)CCC1)=O C1(CNC(CCC2CC(OC)C2)=O)CN(C(C2CC(=O)C2(C)C)=O)CCC1C C=CC1(CC(=O)NCC(c2ccccc2)N(C(=O)CCC#N)C)CCOCC1 c1(C(N2CCC(C(C)(C)NC(c3c(CC)csc3)=O)C2)=O)ccc(OC)c(Cl)c1 C(=O)(CC(O)CCCCC)N(C1(CC#C)CCCCC1)CC(NOCC#C)=O N1(C(C2(CC)CC2)=O)CCOC2(CCN(C(=O)C(c3cccc(Cl)c3)(F)F)C2)C1 c1(CC(=O)NCC=CCNC(C2(CO)CCCO2)=O)c[nH]c2ccc(Cl)cc12 C1(NC(C(C)=CC)=O)CN(C(=O)Cc2cc(OC)ccc2F)CCC1C c1(NC(C2C(Cl)(C(=O)OCC)C2)=O)cc(C)cs1.C(COCCN(C)C(=O)C1CC1)O Cc1cccc(C(=O)NCC2(C(C)NC(=O)CCc3ccc(C)s3)CC2)c1 N1(C(CCOCCC)=O)CC(NC(=O)C(C)SC)C(C)C1 C12(CC)CCCN(C1)C(=O)C=CC(=O)N2.C1(C(=O)NC2CC2)CC2CCC(C1)S2 c1(C(=O)NCC2(F)CC(CNC(CCCNC(N)=O)=O)C2)cccn2nnnc12 N1(C(C(C=CCCC)O)=O)CCC(O)(C(C)NC(c2cc(C)nn2CCC)=O)C1 CCCCC(CC)C(=O)NC1CN(C(C2CC2C2CCC2)=O)C1 C1(C(N2C(C)CC(CNC(=O)Cn3cc(CO)nn3)C2)=O)CCc2nccn2C1 C1(NC(c2cc(=O)c(OC)co2)=O)COCCN(S(CCC=C)(=O)=O)C1 c1(CC(=O)N(CC(C)N(C(c2cc(C)[nH]n2)=O)C)C)c(O)ncnc1O N(C(=NCCc1ccc(OC)cc1F)NCCC(=O)NC)C(C#C)CN(C)C Cn1cc(I)c2c(NC(=O)CC3CCCN3Cc3ccc(O)c(Br)c3)ncnc12 Cc1ccc(NC(=O)C(CC2CCCC2)NC(=O)C(c2ccn(C)c2)C)cc1Cl C1(CC(=O)NCC2C3CN(C(=O)CCCCn4ccnn4)CC23)COCCOC1 CCC(C)C(C(=O)NC1CC1)N1CCC(CN2CCOCC2)CC1 C(=O)(C(CNC(C)=O)CO)NC1CC(F)(CNC(C2(C(=O)NC)CC2)=O)C1 c1(C(=O)NCCC(C)N(C)C(C2CCC2C)=O)cc(Br)c2cccnn12 C(c1ccc2[nH]ccc2c1)=CC(N1CCC(C)N(C(C2CC2[N+](=O)[O-])=O)CC1)=O c1(C(=O)NCC2C(C)CCN2C(=O)CC(C)C2CCCO2)noc2ccccc12 C1(CN(C(C(=O)N(C)CC)=O)CC)CCN(C(=O)CCCC2CC2)CC1 N1(C(C)=O)CCN(C(C2(CO)CCN(C(c3cnc(C4CC4)o3)=O)C2)=O)CC1C C1(C(N2CCC(CNC(c3cnn(CCC)c3Cl)=O)C2)=O)C2CCC1(C)C2(C)C CC1=NNC(=O)C1c1nc(-c2sccc2Br)no1 N1(C(CC(C(C)C)C)=O)CCCC2(C1)C(NC(C1CCCN1C)=O)CCN2C CC1=NN(C)C(=O)C1CC(=O)NC1(C)CC(NC(c2nnn(C)n2)=O)C1 c1(C(=O)OCC(c2ccc(Br)cc2)C)cccn(C2CCC2)c1=O C1(C2CCN(C(=O)Cc3cnoc3)C2)(NC(C2CC3CCC2O3)=O)CC1 N1(C(c2cnc(C)n2C)=O)CCOC2(C1)CN(C(C1CC(C)OC1C)=O)C2 C(=O)(N1CC(O)CO1)C1(F)CCN(C(COC2C(C)CC2)=O)C1 c1(OC)cc(N)c(C(N2CCN(C(=O)Cn3cc(Cl)cn3)CC(O)C2)=O)cc1O c1(C(=O)NC2CCN(C(C(C)C)=O)CC2CO)cc(Cl)c(N)c([N+](=O)[O-])c1 c1(OC)cccc(C(N2CCC(CNC(C3CCCN(C)C3)=O)(OC)C2)=O)c1 N1(C(c2cn(CC)nn2)=O)CC(NC(=O)C(N)=O)C(S(C)(=O)=O)C1 C1(CCCOC)CCCN(c2nnc(-c3cnn(C)c3)n2CCn2cccn2)C1 N1(C(C2=NOC(C)C2)=O)CC2CC(F)(F)CCC2(NC(c2ccc(=N)[nH]c2)=O)C1 O=C1CC(CC(N2CC(N(C(=O)COCC3CCOCC3)CCO)C2)=O)CN1 c1(SC)ccc(C(=O)NC2CC(F)(CNC(c3csc(C(F)F)n3)=O)C2)o1 CC1(C)CC(=O)N(CC(=O)NC2CCOCC2NC(=O)CC2SC(=N)NC2=O)O1 c1(C(N2C(C(C)NC(c3cc[nH]n3)=O)CCCC2)=O)ccc2nc(O)[nH]c2c1F C1(C(=O)NCC(CC=C)NC(C2(CC)CCCC2O)=O)CCC(CC)CC1 n1(CC)cc(CC(=O)NCC2COCC2NC(c2cnc(C(C)=O)s2)=O)cn1 c1(C(=O)NCCC2CC(NC(C(COC)O)=O)C2)cccc(S(C)=O)c1 C(=O)(CCCC(=O)NCC(C1CCOC1)NC(c1cnc(O)s1)=O)N(C)C C1(F)(CCc2c(NC(=O)NCN3CCC(OCC)CC3)ncs2)CNCC12CCC2 Cc1cn2ccnc(C(N3CC(F)CC3CNC(C3CCC(=O)NC3)=O)=O)c2n1 c1(C(=O)NCC2CC(NC(c3onc(CC)n3)=O)C2)cccc(F)c1F C1(NC(C=CC(C)NC(=O)CN2CSCC2=O)=O)C(O)C2CCOC12 O=C(O)C1c2ccccc2OCCN1CC(c1ccc2c(c1)OCCO2)=O C(C(=O)N(C(C)CCNC(=O)Cc1cnccc1C)C)(C(C)C)SC N1(C(=O)CSC(F)F)CCN(C2CCN(C(C3CC34CC4)=O)C2)CC1 C(=O)(C(C)(C)C(C)(F)F)NCC(c1ccc(F)cc1)NC(C(CSC)O)=O CC(C)CCC(=O)NC1C2CC1N(C(=O)C(C)OCC(F)(F)F)C2 C1(C(N(C2CCN(C(Cc3c(C)nsc3)=O)C2)C)=O)CCOCC1(C)C CS(=O)(=O)c1sccc1C(=O)NC1CC2CCC1N2C(=O)COC1CCCC1 C(=O)(C1=CS(=O)CCC1)N1CC2C(CNC(c3cc(N)nc(Cl)c3)=O)(CC2)C1 CCCCCS(=O)(=O)CC(=O)N1CCCC1C1CCCN1C(=O)CC(C)(C)F C(CCCCC(=O)NCC1CC(NC(C2CC2(C)Br)=O)C1)SC C(CN=C(NC1CCNC(=O)C1)NC1CCN(c2ncccn2)CC1)SC N1(C(CC2CC(NC(c3ccc(C(C)=O)o3)=O)C2)=O)CCc2nocc2C1 CC1(C)CC2(CCN(C(=O)NCc3coc4ccc(F)cc34)C2)CO1 C1(NC(Cc2cccc(OCCN(C)C)c2)=O)CCCN(Cc2ccccc2)C1=O C(=O)(C(C)(C)CCNC(C1CC(=O)C1(C)C)=O)NCCC(=O)NCC(C)C c1(CNC(C2(CC=C)CN(C(=O)CCN3CCC(F)C3)C2)=O)ncncc1OC c1(OCC)ccc(C(=O)CCC(=O)N(CC(F)F)C)cc1.c12ccccc1N2 c1(C(=O)NC2C=CC(C(N(CCC)C)=O)C2)nn(C)cc1C C(CS(=O)(=O)c1c(Cl)cccc1Cl)ONC(c1ccc(N=[N+]=[N-])cc1)=O c1(C(=O)NC2CC(CCNC(C3N(C)CCOC3)=O)C2)cc2ccc(F)cc2s1 N#Cc1ccc(N)c(C(=O)NC2CC2NC(=O)CC2CCCNC2=O)c1 N1(C(C(C2CC(F)(F)C2)OC)=O)CC(C)C(C)(CNC(C2(CF)CCOCC2)=O)C1 C(=O)(C(CCC)CC(C)C)N(CC)CC1CCN(C(c2csc(Cl)c2)=O)CC1 c1(C(N2CCC(CNC(C3CCCC(C)(C)C3)=O)C2)=O)coc2c(Cl)cccc12 C1(NC(c2cc(CCCC)oc2C)=O)CC(NC(=O)CC2=CCCC2)C12CCC2 c1(C(=O)NC(C(C)NC(=O)CC2COCC(C)(C)O2)(C)C)ccc(Cl)c(F)c1N c1(C(=O)NC2CCN(C(c3n(C)c(Cl)cn3)=O)CC2F)ccc2nnn(O)c2c1 N1(C(c2c(C)scc2)=O)CCC(C)(C)C(C(=O)NC(c2ccncc2)C)C1 CC(C)C(C(C)C)NC(=O)C(C1CCCC1)NC(c1cc(Cl)n[nH]1)=O C1(NC(C2(CC)CC(C(=O)OC)C2)=O)CCN(CCC(C)CC)CC1 N1(C(C(C(CC)O)(F)F)=O)CCCC(C2CCN(C(=O)CN3CCCCC3)C2)C1 C1(N(C(C(C)=C2CC2)=O)C)CCCC2CN(C(c3cc(CC4CC4)on3)=O)CC12 Cc1nc(Cl)sc1CNC(=NCC1CCC1)NCC(C1CC(F)(F)C1)O c1(C(=O)NC(c2cn(C)nn2)C(=O)NCC(C)OC)cnn(C)c(=O)c1 N1(C(C2CC(C)(C)O2)=O)CCC2(CCCN(C(=O)CCF)C2)C1 c1(C(N2CC(C)(NC(C3NC(=O)CC(C)C3)=O)C2)=O)cnc2nc(O)ccc2c1 c1(CC)nn(C)c(CC)c1C(=O)NCC1(NC(=O)CC2CCCC2O)CCOC1 C1(NC(c2cc(C)on2)=O)COC2(CCN(S(=O)(=O)c3ccc(F)cc3)CC2)C1 C=CC(C)(CCOC)C(=O)N1CCCC(NC(C2(C#N)CCCC2)=O)C1 C(=O)(C(CNC(C1CCOC1CC)=O)(CC)CC)NCC1N(CC)CC1.COC c1(C(=O)NC2C=CCN(C(c3c(C)n(C)nc3Cl)=O)C2)ccc2nnc(S)n2c1 c1(OCCCC)ccc(C(=O)NC2CC3(CCO3)C2)cc1OCC n1(CCCC)cc(C(=O)NCC(O)CNC(c2cnc(OC)s2)=O)nn1 C1(C(=O)Nc2ccc(C(F)(F)F)c(F)c2)CC2(CC2)CN1C(C(C)S)=O c1(C(C)C)ccccc1OCC(=O)NC(CNC(=O)C(C1(O)CCCC1)F)CO c1(OCC)cc(C(=O)NCC2CC2NC(=O)CN(S(C)(=O)=O)C)[nH]n1 n1(CC)nnnc1C(c1ncnn1CC(F)F)NCC(C1CCOCC1)(C)OC C1(CCN(C(c2nc(CCC)sc2)=O)CC)C(C)CCCN1C(=O)CCC1CC1 C(=O)(C(O)C1=CCCCC1)C(c1cc2c(s1)CCOC2)=O.C12C3CN(CC13)C2=O N1(C(=O)C(F)F)CCCC2(CCN(C(C34CCCC3C4(F)F)=O)CC2)C1 c1(C(N2CCC(N(C(C3CCCN(C(C)=O)C3)=O)CC)CC2)=O)cccc(F)c1Cl c1(CN(C)CC2CCCN2C(=O)CSc2cccs2)[nH]ncc1C#N C1(CNC(c2ccc(SC)o2)=O)COCCN(C(c2cc[n+]([O-])cc2)=O)C1 Cc1nn(C2CCCCO2)c(C)c1C(=O)NC(c1ncc(-c2ccccn2)[nH]1)C CC1CN(C(=O)CC2CCC=CCC2)CCCN1C(C1CC12CCOCC2)=O C(=O)(C(CNC(=O)C(O)Cn1cncn1)C(C)C)N(C(CC)C)CC c1(N(c2c(O)cccc2Cl)C(=O)NCCNC(C)=O)cccc(S(C)(=O)=O)c1F C#Cc1ccnc(C(N2CC(NC(=O)CN(C(=O)COC)C)C(C)C2)=O)c1 C1(c2ccncc2)(C(=O)NCC2CCC(c3ccccc3)N2)CCCCC1 c1(C(=O)NC2(CC)CCN(C(=O)C(C)C(=O)OC)C2)nc(C)n2ccccc12 CC(C)S(=O)(=O)c1ccc(-c2cccc(F)c2C#N)c(Br)c1 c1(NC(C)=O)ccc(C(=O)NCC#CCNC(=O)COC(C)C)cc1F c12ccccc1CC(=O)N2.c1(CCC)nnsc1CN(CC)CC.C1(C)CC1 N#CC1(N2CCC(NC3CCCCCC3)CC2)CCNCC1 N1(C(CSCCOC)=O)CCC(NC(c2cccnc2Cl)=O)C1(C)C CCC(CC(F)(F)F)C(=O)N1C2COCC1CC(NC(c1ccns1)=O)C2 CCC(C)CC(=O)N1CC(N(C)C(c2cnoc2-c2ccco2)=O)C1 c1(C(N2CCCC(NC(c3csc(Cl)c3)=O)C2)=O)ccc2nsnc2c1 CCC(CC(=O)Nc1ccc(CNC(=O)CC(=O)OC(C)(C)C)cc1)SC c1(C(c2n(C(CC)C)nnn2)NCCOCC(F)(F)F)ccc(OC)c(C#N)c1 N1(C(C(CCC)(C)C)=O)CC2CCN(C(=O)CN3CCCC3C)C2C1 CCC(C)(CCCNC(=O)NCc1ccc(F)cc1O)c1ccccc1 c1(CNC(c2ccc(-c3cnco3)cc2)C)ccc(N2CCCS2(=O)=O)cc1 n1(CC(N2CC(CNC(=O)C(O)C3CC3)C(O)C2)=O)cc([N+](=O)[O-])ccc1=O N1(C(=O)CCN2CCCCCC2)CCC2C(CCCN2C(c2ncccn2)=O)C1 C1(NC(=O)CCc2cnco2)CCCC12CN(C(C1(O)CCCCC1)=O)C2 N1(Cc2nc(-c3cc(OC)c(C)cc3OC)sc2)CC2CC(CO)CC(C2)C1 CC(=O)CCCC(=O)NCC1CCN(C(=O)CC2(O)CCCOC2)C12CC2 CC1CC=C(C(=O)NC2(C(=O)NCCc3nccc(O)n3)CC(O)C2)CC1 c1(C(N2C(C)CC(CC(=O)NCCn3cnnc3)C2)=O)ccc(F)c(O)c1 C12(CNC(C=CSC)=O)CC(NC(C3(F)CCOC3)=O)(C1)C(C)(C)O2 N1(C(c2nc(C)oc2)=O)CCC2(CO)CN(C(c3ccco3)=O)CC2C1 C1(NC(=O)C=CCC2(NC(C3CCSC3)=O)CCC2)CC(F)(F)C1 c1(C(=O)NC2C(CNC(c3nn(C)c(=O)cc3)=O)C2)cccc2c1COC2 c1(C(CC(=O)N(CC(C)NC(C(C)=CC)=O)C)NC(=O)OC)ccc(F)cc1 C1(NC(c2n[nH]c(CC)c2Cl)=O)CCC2(CCCN(C(=O)CCCC#N)C2)C1 c1(C(N2CC(CCNC(CN(C)C3CC3)=O)OCC2)=O)cnc2c(c1)COC2 N1(C(c2nc(OC)oc2)=O)CC2(C1)CN(C(=O)C(=O)NC1CC1)C2 N1(C(C(F)=C(C)C)=O)CC(NC(C2SCCS2)=O)C(CC(C)(C)C)C1 CC1(C)C(C)(C(N2CCC(C)(CNC(c3csc(Cl)c3Cl)=O)CC2)=O)C1(C)C c1(C(N2CC(CNC(C=CCOC)=O)(OC)C2)=O)cc2ccc(C)cc2nc1C C1(S(C)(=O)=O)(C(=O)NC2CN(C(C(CCC)C#N)=O)CC(F)C2)CCCCC1 c1(N(C(=O)Nc2c(C)nn(C(F)(F)F)c2)C)cc(C#N)ccc1F C(=O)(CS(=O)(=O)CC(C)C)N(C1CCCN(C(c2c(C)noc2C)=O)C1)CCF N1(C(c2c(C)c(Br)ccn2)=O)CC2CN(C(C3CCN(C)C3=O)=O)CC2C1 C1(=C(C(=O)NC(Cc2cnc[nH]2)CO)F)CCN(C(C2CC2c2ccco2)=O)CC1 c1(C(N2CCC(C(=O)Nc3ncc(I)cc3Br)C2)=O)ccc2cc(O)ccc2n1 c1(CCC)ccc(NC(=O)COC(=O)N(C)Cc2ccccc2)cc1 C#CC1(C(=O)NC(C)C)CCN(C(=O)C=Cc2cn(C)cn2)C1 C(=O)(C(C)CC(F)(F)F)N1C(CNC(Cc2cnc(C)[nH]2)=O)C(C)CC1 c1(NC(c2nc(-c3c(C)occ3)on2)=O)cc(Br)cc(Cl)c1F C1(NC(c2cncc(C)c2C)=O)CN(C(=O)C(CO)C(F)(F)F)CCC12CCC2 C1(C)(n2c(C(C)Sc3cccs3)nc(-c3ccc(OC)nc3)n2)CCS(=O)(=O)C1 c1(CCCC)cc(N)c(C(=O)NCC(C)NC(=O)CCCN=[N+]=[N-])c(F)c1 c1(OC(C(C)C(C)(F)F)=O)cc(Br)cc2c1OCO2 C1(C(N2C(C)CC(NC(c3c(CC)n(C)nn3)=O)C2)=O)CC(S(C)(=O)=O)C1 N1(C(c2cccc(C)n2)=O)CCC(C(=O)NC2CCCSC2)C(C)C1 c1(C(=O)NC2(COC)CN(C(=O)CNC3CCOCC3)C2)nnn(C(C)C)c1C N1(C(C2(CC=C)CCOCC2)=O)CC2COCCC2(NC(=O)CC#N)C1 CC1CCc2c(sc3ncnc(NC4CCCC4NC(C4CC5CCC4O5)=O)c23)C1 Cc1ncnc(O)c1CCC(=O)NCC1C=CCN1C(C1CCOC1C)=O Cc1c(NCCCc2cn[nH]c2)nc[nH]c1=NCc1c(C(F)(F)F)cnn1C C1(CC(=O)N(CCN(C)C)CCO)CCCCN1C(c1ccc(=N)[nH]c1)=O C1(CC(=O)N(CC(=O)NC(CN2CCCC2)CO)CCOC)CC2CC2C1 C1(NC(c2c(C)cccc2N)=O)CN(C(C2(F)CCS(=O)(=O)C2)=O)CC(C)(C)C1 N1(C(Cc2ccn(C)n2)=O)CCCCC1CCNC(c1cnn(CCO)c1N)=O C1(F)(CNC(CCn2c(C)nc(C)n2)=O)CCN(C(=O)C(C(C)O)N(C)C)CC1 c1(CC(=O)NC2C(C)CCN(C(c3c(C)n(C)cc3)=O)C2)ccc2sccc2c1 C1(N(C(c2n(CC)nnc2)=O)C)CN(C(=O)CCc2cc(C)sc2C)CC12CC2 Cc1nonc1CC(=O)NCC1(NC(c2conc2C2CC2)=O)CC1 N1(C(C2(C(=O)OC)CC2)=O)C2CCCC1CC(NC(c1ncc[nH]1)=O)C2 C1(CNC(C(CC#C)C)=O)CCC2(CCN(C(C3COC3)=O)CC2)O1 c1(C(=O)NC(Cc2cc(C)n(C)n2)C)cc(S(=O)(=O)N2CCCCC2)ccc1C C1(C(=O)NCC23CCC(CC2)C3)CC12CCN(C(=O)CN1CC3CC3C1)C2 CC1=C(C(=O)NCC2CC(F)CN2C(C2CCC(O)CN2C)=O)CCC1 C(=O)(C(C)CCC(C)(C)C)NCCC1(O)CCN(C(c2c(CC)[nH]cc2)=O)C1 CC(C)(CC(c1ccccc1)(C)C)CC(=O)NCCc1nc[nH]n1.C1(=O)CN1 N1(C(c2c(C)occ2)=O)CCC(C=CC(=O)NC2CCN(C(C)C)CC2)CC1 c1(C(C)OCCOCC)nnc(N(CC(F)F)C)n1CC1CC1(C)C c1(C(=O)NC2C(C)CN(C(=O)C(C)(CO)CO)C2)ccc(I)cc1C#N c1(C(=O)NC2CC(F)(CNC(C3CCC3C(F)(F)F)=O)C2)cc2ccccc2[nH]1 N1(C(=O)C(CC(F)F)NC(C2(F)CCCCC2)=O)CCc2ccc(F)cc21 c1(C(=O)NC2(C3CN(C(C4(C)C(C)C4)=O)C3)CC2)cnc2ncnn2c1O c1(C(=O)NCC(C)N(C(=O)CCSCCC(N)=O)CC)ccc(C#N)[nH]1 c1(NC(C2CC(=C)CN2Cc2ncc(Br)cc2Cl)=O)cccc(N(C)C)c1OC C1(CC(N2CC3C(NC(c4nn(C(F)F)cc4Cl)=O)C3C2)=O)CN2CCN1CC2 C1(NC(c2c(COC)cco2)=O)CN(C(c2cnc(N)c(Cl)c2)=O)CCC1CO N1(C(CC2C(CC)C2)=O)CCCC12CCN(C(c1cccc3[nH]ncc13)=O)C2 c1(C(=O)NC(CC=C)CNC(=O)CC(C=C)CCC)cc(F)c(F)cc1N C1(NC(c2c(CC)cns2)=O)CCN(C(c2cc(C)on2)=O)CCC1CO CN1CCCN(C(=O)CC2N(C(C3CC(=O)NC(=O)N3)=O)CCC2(C)C)CC1=O c1(CNC(C2CCN(C(COCC#C)=O)CC2)=O)c(C)cccc1C CC1CCC=C1C(=O)N(C(C)CCNC(c1cn(C)nc1-c1ccco1)=O)C c1(CN(CCC(=O)Nc2ccccc2C)CC=C)cccc(Br)c1C C=CCC(CNC(c1cc(C)n(C)n1)=O)C(=O)N1CC(CO)C2(CC2)C1 c1(C(=O)OC)cc(NC(=O)CCNC(=O)C=CC(C)=O)c(F)cc1C C(CNC(c1ncccc1F)=O)(C(C)(C)C)NC(c1cn(CCN(C)C)nc1)=O C(=O)(CC(C(=O)NCc1ccc(C(=O)OC)nc1C)NC(=O)OC)OC(C)(C)C C1(n2cc(CCS(N)(=O)=O)nn2)CCCCC1NC(=O)C(=O)Nc1ncc[nH]1 C1(C2(O)CN(C(C3CC(C4CC4)=NO3)=O)C2)(CNC(C2C(C(C)C)C2)=O)CC1 CC(C(=O)NCC1CCCN(C(c2cnoc2C2CC2)=O)CC1)C(C)(F)F Cc1ccc(C(=O)NC2(CNC(c3ccsc3C)=O)CC2)cc1S(C)(=O)=O CCCC(C)(CCC)C(=O)NC(C)CC(C)NC(c1ccnn1C(C)CC)=O C(C(CC(C)C)C(=O)OCC)NC(C1C(C(=C)C)OCC1)=O C1(N(C)C)(C(N)=O)CCCN(CCCC2CC(F)C2)C1 C1(C(N2CCC(C(C#C)C)CC2)=O)CCCN(C(=O)C(C)(C)C)CC1 c1(OC)ccc(C(N)=O)cc1C(=O)NCC(C)(C)CCNC(C12CCCCC1C2)=O Cc1ccc2cc(CN3C4CCC3CC(NC(C#N)C(N)=O)C4)c(Cl)nc2c1 n1(CC(=O)NC(C(=O)NC(CC=C)CC)CN(C)C)c(C)ccc1C C=C(Cl)CC(C(=O)Nc1cc(F)ccc1C)NC(=O)CC1CC=CCC1 N1(C(CC2CCCN(C)C2)=O)CC(CNC(c2n[nH]cc2Cl)=O)OC(C)(C)C1 CC1(C)CCC(CC(N2CCC(NC(=O)CSc3ccc(F)cc3)CC2)=O)OC1 c1(C(N2C(CNC(C(C=C)(C)CC)=O)CCC2)=O)cccc2ccn(C)c12 c1(C(=O)NC(CN(C(CCOC(CC(C)C)C)=O)C)C)ccc(C2CC2)cn1 C12(CNC(C(C=C)(F)F)=O)CCCC1CN(C(c1ccc3c(c1)NCC3)=O)C2 c1(C(N2C3CC(CNC(C(CSC)(C)C)=O)C2CC3)=O)c(O)cc(F)cc1F c1(C(N(CCNC(=O)CC2(C)CCCC2)CC)=O)cc2cnc(Cl)cc2s1 c1(N2CCC(N(C)C)CC2)nc(NCC2CCCO2)nc2c1cnn2C c1(CN2CC(C)(C(=O)Nc3nnccc3C(F)(F)F)C2)cc(F)ccc1[N+](=O)[O-] N1(C(c2nc(CC)sc2N)=O)CCC(NC(c2coc(Br)n2)=O)C1(C)C N1(C(c2cc(O)cs2)=O)CCCN(C(C2(C3CC3)CCCO2)=O)C(c2cn[nH]c2)C1 C1(CC)CN(C(C2CC3CC3N2C(c2cccc(CC#N)c2)=O)=O)CCO1 c1(CC(=O)NC(C(=O)NCC2CC(OC)CN2C(C)=O)C)ccc(Cl)c(Cl)c1 C=CC(C)(CCOC)C(=O)NC1CC(C)N(c2nc(OC)cc(C(F)(F)F)n2)C1 N1(C(C2C(C)C2)=O)CCC(OCCNC(=O)C(C)Cn2ccnc2)CC1 Cc1nn(C)c(Br)c1C(=O)NC1CC1CNC(c1cccc(Cl)c1Cl)=O N1(C(C(CC=C)(F)F)=O)CCC2CN(C(=O)Cc3cccc(F)c3O)CC2CC1 c1(C(N2CC(CC)N(C(=O)CC3CC(OCC)C3)CC2)=O)cc(F)c(F)c(F)c1 c1(C(=O)NC2(C)CN(C(C3(COC)CCC(=O)N3)=O)C2)cccc2ccncc12 C1(COC)(NC(=O)CC(C)SC)CCN(C(c2ccc(-c3cnc[nH]3)cc2)=O)C1 c1(C(=O)OC)sc(C2CCCN(C(C(=O)NC(=O)NC3CC3)C3CC3)C2)nc1C Cc1nc(O)c(C(=O)NCC(O)CNC(C2(C)CC2(C)C)=O)nc1C c1(OC)cc(CN2CC(C)(C(N3CC(F)C(F)C3)=O)C2)c(Br)cc1O CCCCC(=O)C(=O)NC1(CO)CCN(C(=O)C(CO)N(C)C)C1 c1(OC)ncc(F)c(N(c2ncc(C)cn2)C23CC(N)(C2)C3)n1 C1(N(C(c2c(C)nc(C)[nH]2)=O)C)CCN(C(=O)C(C)n2ccnc2)CC12CC2 c1(NC(CC2NCCN(C)C2)=O)ccc(F)c(C2CC2)c1 C(=O)(C(F)C(C)(C)O)NC(C1(O)CN(C(c2ccnn2CC2CC2)=O)C1)C c1(C(=O)NCC(C2(O)CN(C(C3CC4(CC4)C3)=O)C2)(C)C)cc(C2CCC2)[nH]n1 CC1CN(C(=O)Cc2c[nH]nc2O)CCC1NC(=O)CCc1nnc(S)nc1O N1(C(c2c(CC)[nH]cc2)=O)CCC(CN(C(=O)CCn2cnnn2)CC)CC1 CC(C)(O)CC(=O)N1CCN(CCCNC(=O)CC2CCSC2)CC1 C1(NC(C2CCCN(CCC)C2)=O)CC(C)CN(C(=O)Cc2sc(C)nc2C)C1 CC(C)C(C)C(CNC(c1ncsc1Br)=O)NC(c1ccn(C)c1)=O CC(C)C(O)C(=O)NCC1CCN(C(c2ccccc2Oc2ccccc2)=O)CC1 N1(C(CCC=CC(C)C)=O)CCN(C(=O)CCNC(C2CCCC(O)C2)=O)CC1 N1(C(c2ccc(C)s2)=O)CC2CCC1C2NC(C1CCSC1)=O C1(CNC(=O)Cc2csc(-c3nc[nH]n3)n2)COC(C(F)(F)F)C1 C=CCCCCC(=O)NC1CC(CNC(=O)COc2cccc(F)n2)C1(C)C c1(NC(CC)=O)cnccc1Br.C12CN(C1)C(=O)CO2 Cc1ncoc1C(=O)NCC(=O)N(C(CNC(=O)CC1(C)CC1)C1CC1)C N1(C(CC(CC)(F)F)=O)CC2CCCC(NC(C3(COC)CCC3)=O)C2C1 C(c1ccccc1)=CCNC(C1CCC(NC(C(CC)C2CCOCC2)=O)C1)=O c1(C(N(C(C)CNC(C2CC3CCC2O3)=O)C)=O)cccc2scnc12 N1(C(c2nc(COCC)sc2)=O)CCC(NC(=O)C(C)n2ccnc2)C(C)C1 c1(CC)nc(NC2CCN(CC3CCN(CC)C3)CC2)[nH]c(=N)n1 c1(C(=O)NCCN(C(=O)Cc2nnc(S)n2C)C)n[nH]c2c1CC1CC21 C=CCCCCC(=O)NCCCC(O)C(=O)NCC1(CC)CCCC1 c1(-n2cnc(C(=O)CC3CC3)n2)c(C)[nH]c2ccc(F)cc12.c1(C(=O)NCCOC(C)C)ccoc1C.N.C.NC CCC(C)CC(C(=O)NCC1CCCC1)NC(=O)C1=CC(C)(C)C1 N1(C(C)=O)CCC(C2CCN(C(=O)C(C(C)C)NC=O)C2)CC1.c1cccc(Cl)c1 C(=O)(C(C)C(=O)N1CC2C(C(=O)Nc3cccc(-n4cncn4)c3)C2C1)OC C(=O)(CC1C(=O)Nc2c(C)cccc21)NC(C1CCCCC1)CNC(C=CC)=O C(C)(CC(F)(F)F)N(C(C(Cn1cncn1)NC(C=C(COC)C)=O)=O)C CC1(C)C2CN(C(c3csc(Br)c3)=O)C(C(=O)NCc3ccncn3)C12 C12(C(N3CCC(CC#C)(C(=O)NCCCC4CC4=C)C3)=O)CC(C)(CCO1)C2 C1(CC)(NC(=O)Cc2cn[nH]c2)CCN(C(c2cn(CC)nn2)=O)CC1 CC1CC(NC(=O)C(=O)NCc2ccccc2)CN(C(=O)CCc2cn[nH]c2)C1 Cc1ccc2[nH]c(C(N3CC4CC(C3)C4NC(=O)COC(C)(C)C)=O)cc2c1 C(=O)(C1=C(Cl)CCOC1)NC12OCC(NC(CC(C)(O)C3CC3)=O)(C1)C2 C(=O)(CCC(C)(C)NC(=O)C(F)C(C)(F)F)NCC1(SC)CC1 CC1CCC(NC(c2n[nH]cc2[N+](=O)[O-])=O)CN1C(C1CCCC2(CC2)C1)=O N1(C(C)=O)CCC(C2(O)CCN(C(=O)CC(C)CCc3ccccc3)C2)CC1 CC(CCC(=O)NC(C(F)(F)F)C1CC1)NC(=O)Cc1cc[nH]c1 C1(CC)CN(C(=O)Cc2cnn(C)c2C)CC1C(=O)N(CCCO)C N1(C(C2CC(=C)C2)=O)CCN(C(C2CC3C=CC2O3)=O)C(CCCC)C1 c1(C(=O)NCC(c2cccc(OC)c2)NC(C2(O)CCC2)=O)cc(F)cnc1O C(C)(CCC(=O)N1CCCC1C=CC(=O)NCC1(OC)CCC1)OC C(=O)(C1COc2ccccc21)N1CCC(C2(NC(c3coc(Br)c3)=O)CC2)C1 C12(C(=O)NCCCN(C(C(CC)C(C)C)=O)CC)CCCC(=O)N1CCC2 CCCC(C)(C)CC(=O)N1CC(CNC(=O)Cc2c(C)cnn2C)CC1(C)C c1(N(C2CCC(NC(=O)C=Cc3ccnn3C)CC2)C)ccc([N+](=O)[O-])cc1 N1(C(C2(OC)CCSC2)=O)CCOC(CC(=O)NCCN2CCCCCC2)C1 C12(NC(CCOCC(C)C)=O)CCN(C(C3CC3c3ccccc3)=O)CC1C2 C1(CC(N2CCC(N(C(c3ocnc3C3CC3)=O)CC)C2)=O)CC2(CCC2)CO1 C#CCC(C)C(=O)NCc1cccc(CNC(=O)CCSc2nnnn2C)c1 N1(C(C2(C(=O)NC)CCC2)=O)CCCCC1CNC(=O)CCCCF c1(NCC(CO)OC)ccnc(N)c1 C1(c2n(CCCC)nnn2)(NCc2nc(C3CC3)no2)CCCN(C)C1 CN1CCCC(O)(CC(N2CCC(NC(C3CCC(=O)N3)=O)C(F)C2)=O)C1 n1(CC)nc(C(=O)NC(C)CCNC(=O)C(N2CCCCC2)C)c(C)n1 C1(NC(C2CCCCS2)=O)CC(O)C1CC(=O)NCCN1CCC(O)C1 C1(C(=O)NCC(CC)(C)Cl)CN(C)CCN1C(=O)Cn1cc(C#N)cn1 c1(OC)cccc(O)c1CN1CC(NC(c2nc(C)cnc2C)=O)C1 Cc1cc(C(=O)N(CC(C)NC(=O)CC2(C(F)F)CC2)C)ccc1S(N)(=O)=O N1(C(c2cc(OC)n[nH]2)=O)CCN(C(c2ccncc2N)=O)CC1C c1(NC(C(Cc2ccc(OCC)cc2)=O)=O)c(F)ccc(OC)c1Cl C1(OCC)(CNC(=O)C(n2ccc(C)n2)C)CN(C(=O)C(F)F)C1 C(CCCC(C)NC(C1CC1(C)C)=O)NC(c1nc(C(C)C)oc1)=O c1(C(N2C(C)(C)CC(NC(C3CCCC(C#N)C3)=O)C2)=O)ccc2c(c1)CCC2 CCCC(C(=O)N1CCN(CC(C)NC(=O)C(C)(C)CC)CC1)NC(C)=O N1(C(C2C(OCC)CC2)=O)CCN(C(=O)CCn2cc(C)cn2)CC1CCO c1(C(=O)NC(C(C)NC(C2(CC)CC2)=O)C(C)C)cc2c(nc1O)CCC(C)(C)C2 N1(C(C(C)N2CCCC2)=O)C2CC=C(C(=O)N3CCN(C)C(=O)C3)C1CC2 CCCC(C)(C)CC(=O)NC1(CNC(c2ccc(Br)c(N)c2)=O)CCOC1 N1(C(c2cccc(OC)n2)=O)CCCC(C2CN(C(=O)COCCSC)C2)C1 N1(C(C(C)=CC)=O)CC2CC(CNC(=O)C(O)CC(F)(F)F)CC1C2 c1(OC(C)C(N2CCC(CNC(c3cc(C(F)F)[nH]n3)=O)C2)=O)ccc(C)cc1 C1(C)(C(N(CCCNC(CC(CC)CN(C)C)=O)C)=O)CCC(=O)N(C)C1 CP(C)(=O)c1cc(C(N2CC3CC3(NC(C3CCCC3(C)C)=O)C2)=O)ccn1 C1(NC(c2occc2C2CC2)=O)CCN(C(c2cnnc(O)c2)=O)CC1O c1(C(=O)NCC(CN(C)C(c2ccon2)=O)(C)C)ncccc1Br n1(CC(=O)NCC2(NC(C(C3CCOC3)OC)=O)CCCC2)ncccc1=O c1(C(=O)NCC(CC)NC(=O)C(C)Oc2ccccc2O)ccc(F)cc1 C1(CNC(C=C(CCC)C)=O)CCN(C(=O)CC2COC(C)(C)CO2)C12CCC2 c1(CN(C(CCC(C)C)C)C2CC2)ccc(C(F)(F)F)c(Cl)c1 Cc1cc(C(=O)NCC2(C)CCCN(C(C3CS(=O)(=O)CCO3)=O)C2)cc(C)n1 c1(OC)cc(CCNC(=O)C(N2CCC(C(C)(C)O)C2)=O)c(NC(C)=O)cc1Br Brc1ccc2cnc(N3CCN(Cc4cscn4)C4CC34)nc2c1 c1(OC)nc(Cl)ncc1-n1cc(C(C)(C)N)nn1 Cc1cc(C(=O)NCCCC(C)NC(c2c(C)cccc2F)=O)cc(N)c1O N1(C(CC(C=C)C)=O)CCc2c(c(CNC(=O)C=CC3CCCN3C)nn2C)C1 CC1CC(C)(C)N1N1CCC(O)C(F)(F)C1C=O C1(CCC(=O)N(C(C(C)SC)C)C)CCCN(C(c2cc(C#N)c[nH]2)=O)C1 C(CC(C)C(=O)N1CC(NC(=O)CCc2csnn2)C(C)C1)OC c1(-c2nc(C(C)CC3CC3)nn2C2CCCC(C)C2)[nH]nc2ncccc12 C1(NC(C(=O)NC(C)C)=O)CC2CCC1N(c1ccc(C#N)cn1)C2 CCC(C(=O)N(C(C(=O)N1CC(C(=O)OCC)C1)SC)C)C(C)(C)CC C(=O)(C1=C(Cl)CCC1)NCc1oc(C(NOCC(=O)OC)=O)c(C)c1 c1(C(=O)OC)cc(Br)ncc1NC(=O)C(N1CCC(C2CCO2)C1)=O C1(NC(COCC)=O)C(CNC(=O)CN2CC3CC3C2)CCC12CCC2 N1(C(COCCC#C)=O)CCN(C(c2ncsc2C)=O)CC1c1cccc(Cl)c1 c1(CCC(=O)NC(CNC(C2(CC(C)C)COC2)=O)(C)C2CC2)ccc(O)nn1 C(C)(CCCCNC(=O)COc1nn(C)cc1Br)NC(C1C(C=C)C1)=O N1(C(CNC(CCC)=O)=O)CC2(CNC(=O)C(C)CO)CC1(COC)C2 C(=O)(C(C)C(C)S(C)(=O)=O)NC(CC1CN(C(c2c(OC)scc2)=O)C1)C C1(O)(CNC(=O)CC2CSCCO2)CCN(C(=O)CC(F)(F)Cl)CC1 c1(CC)c(N2CCN(C(C3CCCN3C(C)C)=O)C(C)C2)ncnc1Cl C12(CNC(C3OCC(C)(C)C3)=O)CC(C1)C(NC(=O)C(C)(C)C1CCCC1)CO2 C12(OC)CCC(C(=O)NC3CC3CNC(=O)CC3CCC4CC34)(CC1)CC2 c1(C(=O)NCC(C)NC(C2CC2c2ccc(F)cc2F)=O)ccc2c(c1)CCN2 CC1(C(=O)OC)CC2(CC(=O)C2)C1.N1(C(C2CC23CC3(F)F)=O)CCC(O)CC1 C1(NC(c2ccncc2Cl)=O)CS(=O)(=O)CC1NC(C1(c2cccnc2)CC1)=O C(=O)(C(CCN(C)C)NC(C1CC(C)CCO1)=O)N(CCOCC=C)C C1(COCCCNC(=O)OC(C)(C)C)CC2CC(C(F)F)C1C2 C1(C(N(CCSC)C)=O)CCN(C2CCN(C(=O)C(C)(C)C)C2)CC1 N1(C(C2(NC(CCC3C(C)(C)C3)=O)CCCC2)=O)CC(C)(C)CC1CO c1(CCC(=O)N(c2ccc(OC(F)(F)F)cc2)c2cnccn2)ccccc1I c1(C(=O)NCC(CNC(=O)C(C)Cc2ccco2)OC)cc2occc2n1C C(=O)(CC(C)(C)C(C)=O)NC(CCC(=O)NC(CSC)C(=O)OC)CC c1(C(N2CCC(OCC(=O)OC(C)(C)C)C2)=O)ccc(F)c(C(C)(F)F)c1 N1(C(C(C(C)C)n2cnnn2)=O)CCC2(CC1)CN(C(C1CCCOCC1)=O)C2 c1(CNC(C2CCN(CC)C2)=O)c[nH]c(=NCc2cnn(CCO)c2)s1 CCC(F)(C(=O)OC)C(=O)NC1CC(c2ccc(Cl)cc2C(F)(F)F)C(=O)N1 C(=O)(CC(F)(F)C(C)C)N1C(C)CC(CC(=O)OC)C1.C12(OC)CCC1NC2=O C(N=c1[nH]c(=NCc2csnn2)[nH]c2c1SCC2)c1nc(=N)[nH][nH]1 c1(C(=O)NC(C(C)NC(c2ccon2)=O)CO)cc2ncccn2n1 c1(C(=O)NC2CC(F)(CNC(Cn3ncc(C)c3)=O)C2)cc2n(n1)CCCC2O N1(C(CCCc2ccc(C)s2)=O)CC2CCC1C(CNC(=O)Cc1nccs1)C2 c1(NC(C)=O)ccc(C(=O)NC2CCC2NC(c2ncoc2C2CCC2)=O)nc1 CC1(C)CC(O)CCN(C(C2CCCCN(C(=O)CC3CCCC(=O)N3)C2)=O)C1 N1(Cc2nc(C)[nH]n2)CCCC(C(=O)N(C(C)C(C)C)C)C1 c1(C(=O)NCC2(F)CCC(CNC(C=CCOC)=O)C2)c(S(N)(=O)=O)cnn1C Cc1cc(C(=O)NC2CCC(CNC(C3CCC(C)O3)=O)C2)ccc1S(C)(=O)=O CC(C)(C)C(C(=O)NCC(O)C(=O)N(C)C)NC(c1cnccn1)=O C(=O)(C1=CCC(F)(F)CC1)N1C(CNC(C(C)OCC2CC2)=O)C(C)CCC1 C(=O)(CCC(C)(C)[N+](=O)[O-])NCC(CNC(C1CCCC(C)(C)C1)=O)O C(CCN=C1NCCC2CCN1C2)OC(=O)NC.c1(OC)cc[nH]n1 C1(NC(C2(C(=O)OC)CC2)=O)CC2CCCC(C1)N2C(c1cc(Br)cnc1F)=O c1(C(=O)NCC2(COC)CN(C(CN(C3CC3)CC)=O)C2)cccn(C)c1=O c1(C(=O)NCCCCCC(C(C(C(C)C)N)=O)COCC)cnn2ccncc12 Cc1cccc(C)c1NC(=O)C(C(C)(C)C)NC(=O)NC(c1ccccc1)C CCC(C)(F)C(=O)NC1CC(NC(=O)CCc2nncn2-c2ccccc2)C1 N1(C(c2cnc(C)s2)=O)CCCCC(CNC(c2occc2Cl)=O)C1 CC(CN1CCC1C1CC1)S(C)=O C#CCC(C)(C(=O)NC)NC(=O)COCCF.C(CC(C)CC=C)NC(=O)OC C(=O)(C(C)(O)CCN1CCCC(CN(C2CCC2)C(c2cc(Br)nn2C)=O)C1)OC N1(C(Cc2ccc(OC)cc2)=O)C2CCC(C2)C1C(N1CCCC(F)C1)=O c1(C(c2cc(F)ccc2Cl)NCc2n(CCCOC)nnn2)nccc(Cl)c1C N1(C(CC(CC(=O)OC)C)=O)CC2(CCN(C(=O)OC(C)(C)C)CC2)C1 c1(OC)ccc(C)cc1C(N1CC(S(C)(=O)=O)C1)=O Cc1cc(C)cc(C=CC(=O)Nc2c(Br)cnn2C)c1.C12(C(N)=O)CN(C1)C2 c1(C(=O)OC)c(C)ccnc1NCC(C1CC1)NC(c1cn(C(C)C)cn1)=O N1(C(C2C3C=CC(C3)C2C(F)F)=O)CCC2(CCC(O)CC2)CC1 CCC(C(=O)N1CCN(C(=O)COc2ccoc2)C(c2nccn2C)C1)C(C)C C(=O)(C(CNC(c1nnn(CC)c1C)=O)CC1CC1)N(CCCC)C C12(C(=O)NCC3(CNC(c4c(C)[nH]nc4Cl)=O)CC3(F)F)CCCCC1OCC2 C1(NC(C(C)N(C)C)=O)CC2CC1N(C(c1cc(Br)ccc1F)=O)C2 C1(C(C(C)C)NC(=O)CCNC(C2(C)COCCO2)=O)CCN(C(=O)CO)CC1 C(=O)(C(C(F)(F)F)C1CCC1)NCC12CC(NC(C(C)SCCC(C)C)=O)(C1)C2 c1(CNC(C(OC)OC)=O)cncc(C(=O)NCCc2c[nH]nc2C)c1 N1(C(C(C)Nc2ncccn2)=O)CC2CCN(C(=O)CN3CCC3)CCC2C1 C1(C(=O)NC(c2csnn2)C)C(O)CCN1C(c1ccc(C2CC2)nc1)=O c1(OC(C)C)cccc(C(N2CCCCC2CNC(=O)C(C)C2CCC2)=O)n1 C#Cc1cnn(C)c1C(N1CCC(C(=O)NCCCC2CC=CCC2)(CC)C1)=O c1(C(N2CCOCC(CNC(c3ccco3)=O)C2)=O)cc(F)c(F)cc1F Cc1cc(C(=O)NC2CCCC(NC(=O)C(C)C(F)F)C2)cc(C)c1O c1(OC)ccc(OC)c2c1CN(CCCCCC(C)C)CC2O C1(C(=O)NC(C)(C)CNC(=O)CC2SC(=N)NC2=O)CC2(CCC2)CCO1 C1(CC(=O)N(CC(O)CNC(=O)C(C)(Cl)Cl)C)Cn2ccnc2NC1=O N1(C(CC2CCN(C)C2)=O)CC2(NC(=O)CCc3ccccc3)CC1C2 N1(C(c2c(CC)c[nH]c2)=O)CCC(C)(CNC(C2(CO)CC2)=O)C1 C1(C(C)C)CN(C(C2CC(C3CC3)=NO2)=O)CCN1C(C1CC(C)N(C)C1)=O CC1(C)C(C(=O)NC2CC3(C2)CC3C(N2CC(c3cc(O)no3)C2)=O)C1(F)F C1(C(N2CCC(OCC(C)C)C2)=O)C2CCC(C2)C1NC(C1CC=CCC1C)=O C1(NC(C(C2CCOC2)OCC)=O)CCCCN(C(C2CCCN2N=O)=O)C1 c1(Sc2c(Cl)nc(NC(C(N3CCC(OC)C3)=O)=O)s2)cnc(O)n(C)c1=O C1(NC(C(=O)Nc2cccc(-c3nc[nH]n3)c2)=O)CCCC12CCCCO2 c1(-n2cc(C(N3C(C)(c4ccc(Br)cc4)CCC3)=O)nn2)cc(CO)ccc1N c1(C(=O)NC2(C)CCN(C(C(CCSC)O)=O)C2)ccc(C)c(F)c1N C(=O)(C(F)(F)CC)N(CC(C)NC(=O)CCC1CCC1)CC C1(CCC(=O)Nc2ccc3c(c2)CN(C(C)=O)C3)Cc2ccccc2NC1=O c1(CCC(=O)N(CCNC(=O)C(C)NC(N)=O)CC)cn(C)nc1C1CCC1 C1(C(=O)NCC(CNC(CC23CC(C)(OC2)C3)=O)O)CCC(N=[N+]=[N-])C1 C1(NC(C(CC)C(C)C)=O)CC2(CCC(CNC(C3C4CCCOC34)=O)CC2)C1 C1(F)(C(N(C(C)C)CCNC(=O)C=C2CCN(C)C2)=O)C2CCCCC12 N1(C(CCc2c(C)noc2)=O)CCC(F)(C(=O)NCc2ncccc2Cl)CC1 N1(c2nnc(Cc3nnc(C)s3)n2CC2CC2)CCc2ccnc(O)c2C1 C1(CC)CN(C(c2cccc(Br)c2OC)C(=O)NC2COC2)C(C)CO1 c1(CC(C)NC(=O)CSCCOC(=O)COC2(C)CCCC2)ncn(C)n1 C(CCCCCNC(c1ccncc1C(F)(F)F)=O)NC(=O)CC1CCC1(F)F C1(C(=O)NCC23CC(CN2)C3)C2CN(c3ncccc3Cl)CC12 N1(C(c2c(CC)scc2)=O)CCC(C)(CCNC(c2cn(C)nc2C)=O)C1 c1(CC(C(=O)NCC(C(C)C)NC(C2(COC)CC2)=O)C)ccccc1Cl c1(CN2CC3C(C(=O)NCC(F)(F)F)(C3)C2)ccc2ccnn2c1 c1(OCC(=O)N(CCC)CCNC(=O)CC2(O)CCCOC2)ccc(Cl)cc1F CC(C)C(C)C(C)CC(=O)N1CC2(C1)SCCC2NC(C1CC2CC2CC1C)=O C#Cc1c[nH]nc1C(=O)NC(c1nocc1C(=O)NCC1(Cl)CCC1)C C1(C(N(CCNC(CCCC(C)C)=O)C2CC2)=O)CN2CCCC1CC2 C1(C2N(OCC)C(=O)CC2)CCOCCN1CC(=O)Oc1ccc(Cl)cc1 c1(C(=O)NC2CC(CCNC(C=CCC)=O)C2)sccc1-n1ccnn1 C1(OC)CC(NC(=O)NCCCN(C2CC2)Cc2cnc(N(C)C)s2)CC1OC C(=O)(C(C)(C)C(F)F)N(CC(C)NC(=O)C(C)Sc1ccccc1F)C C1(NC(C2CC(C3CC3)=NO2)=O)CCC2CCN(C(=O)Cc3cscn3)C1C2 CC(C)C(N=[N+]=[N-])C(=O)N1CCN(C)C(C(=O)NCC(O)C2CC2)C1 CCCC(CCC)CC(=O)N1CCOC(CC(N2CCCC2(C)CC)=O)C1 CN1CCCC(NC(c2sccc2CNC(c2cccn2C)=O)=O)C1=O CCCCCCCCS(=O)(=O)NC1CN(C(c2nc(Cl)ccc2F)=O)CC1C#N C(=O)(C(CO)NC(C1(OCC)CCC1)=O)N(CC(CC)OC)C C1(C(N(CCCN(C)C)CC#C)=O)COCCC1NC(=O)COC1CC1(F)F c1(-c2cn(Cc3ccc(C)s3)nn2)ccc2c(c1)CCCN2CC1(C)CC1(C)C C1(C)(CNC(C2CN(CCC)C2)=O)CCCN(CC(C)CC(C)C)C1 c1(COCCOC)nc(-c2cccc(OC(C)(C)C)c2)n(CC2CCCOC2)n1 c1(CC)cc(COC(=O)C(C)NC(=O)C(C)NC(C)=O)n[nH]1 C(CCCCC(=O)N1CCCC(F)(F)C1)N(C(C1C(C)(COC)C1)=O)C C1(NC(C2(OC)CCC2)=O)CCCN(C(c2cc(SC)oc2C)=O)C1 c1(CNC(=O)NC(c2cccc(F)c2)CC(=O)OC)cccc[n+]1[O-] c1(NC(C2C(F)(F)CCN(C(C3C(C(C)C)CCC3)=O)C2)=O)cccc2c1ccn2C c1(C(=O)NCCN(C(C2(C)CCC(C)C2)=O)CC)cc2n(n1)CCO2 c1(CNC2CC(NC(c3c(C)ncs3)=O)C2)cc(Br)ccc1O N1(C(C(CCC)CNC(c2ccc(CC)s2)=O)=O)CCC2(COC(C)C2)C1 N1(C(c2c(C)nc(C3CC3)o2)=O)CCC2(NC(=O)CCc3ccon3)CC2C1 C1(C(=O)NC2(CNC(CCC(=O)O)=O)CC2)CCC(=O)NC1c1ccccc1 CCC(CC(F)F)C(=O)N(C1CCOCC1)CCOCc1ccccc1 N1(C(CCCC#C)=O)CCC2(CC1)CC(NC(C1CCCC1(C)C)=O)C2 C1(CN2C(c3c(C(=O)NCC(=O)OCC)c[nH]n3)CCCC2)CCC2(CC1)CC2 CC1CCCCC1(CNC(c1cn(CCO)nn1)=O)NC(=O)Cc1ccccn1 c1(CSC)cc(C(N2CCC(CC(C)C)C2)=O)ccc1C C(C1CC1)(C1CC1)=CC(=O)NCCCCNC(C1(Cl)C(C)(C)C1)=O c1(C(N2CC(O)CC(NC(c3cn(C(C)C)nn3)=O)C2)=O)cnc2c[nH]nc2c1 N1(C(C(c2ccc(Br)cc2)NC(C)=O)=O)CCC(C2(CO)CCOCC2)CC1 N1(C(CO[Si](C)(C)C)=O)CCC2(CCN(c3ncncc3F)CC2)C1 N1(C(c2nc(C)oc2)=O)CCC(C2CC2)C1CNC(c1cc(Br)sc1C)=O C(CCCCCN=C(NCCN1CCCC(C)C1)NCCCCO)SC N1(C(C(C=C)(F)F)=O)CCN(C)C(CNC(C2CC2c2ccccc2C)=O)C1 N1(C(C=Cc2ccn(C)c2)=O)CC2(CCN2C(=O)CN2CCNC2=O)C1 N1(C(C2OCCN(C(=O)C=CCN3CCCC3)CC2)=O)CCC2CCC(C1)S2 C(=O)(CC(O)C(C)CC)NCCn1ccc(C(=O)NCC(=C)C(F)(F)F)c1 N1(C(CC2N(C(c3n(C)c(Cl)nc3)=O)C3C2CCC3)=O)CC(CO)CC(C)(C)C1 CC(C#CC(=O)N1CCC(C)(C(=O)OC(C)(C)C)C1)NC(=O)NC1CC1 C(=O)(C(CC(F)F)c1ccccc1)NCC1CN(C(c2c(C)n[nH]c2)=O)CC1C c1(C(N(CCNC(c2cccc(C(C)(F)F)n2)=O)CC)=O)nc(C)c(C)nc1O N=c1ncc(C(=O)NC2CCN(C(C3C4CC5C(C4)C35)=O)CC2)c[nH]1 N1(C(c2c(OCC)scc2)=O)CC(NC(c2cccc(C3CC3)n2)=O)CC1C Cc1cc(C(=O)NCC2(CNC(=O)CCC3CCCO3)CC2(F)F)cc(C)c1O c1(C(=O)NC(CNC(C(CC)OC)=O)CO)cc2cccnn2c1 C(=O)(CC1=CCN(C)CC1)NCCC1CC(NC(CCC(CC)C)=O)C1 N1(C(=O)NCCCCCC=C)CC2(CN(C)C2)c2cc(C)ccc21 C#CCC(CC#C)C(=O)N(CCC)CCNC(C1CC(C)CC(C)(C)C1)=O C(=O)(C(C)(C)C(=O)NC1CCN(C(c2ccc(F)c(C(F)F)c2)=O)CC1O)NC c1(N2CCC(CCNC(C(C)OCCOC)=O)CC2)nc2cccc(C)c2o1 c1(N2CC(C)C(Nc3ccc(I)cc3O)C2)ncnn2cccc12 CC1=C(C(=O)N(C2CCCN(C(=O)CCc3cn(C)nc3C)CC2)C)SCCO1 c1(N(CC(=O)NCC2C(NC(C(C)SCCCC)=O)CC2)C)ccc(F)cc1 CC(CCCC(=O)N1CC(C(F)(F)F)CC1CNC(=O)CC(F)(F)F)C1CC1 CC(CCCCCO)NC(=O)C=CC(C)NC(C1CC2(CCO1)CC2)=O C1(NC(=O)Cc2csc(C(F)(F)F)n2)CCOCC1NC(c1coc(Cl)c1)=O N1(C(c2ccc(NC)cc2)=O)CC2CC1CCC2NC(=O)C1=CCSC1 CCC(CCOC)C(=O)NC1CC(C(=O)NCc2cnccn2)C12CCC2 C1(NC(C(C(C)C)n2cccc2)=O)CC2CC1CN(C(=O)C1=CCOC1)C2 c1(C(N(C2CCN(C(c3cc(N)nc(Cl)c3)=O)C2)C)=O)cccn2c(O)nnc12 N1(C(C(CC)(C)O)=O)CC2(C(=O)NCC(O)C3CC3)CCC1CC2 c1(CCNC(c2cc(Cl)nc(Br)c2)=O)nc2ncc(Br)cn2n1 c1(C(=O)NC(CC(C)NC(C2(S(N)(=O)=O)CC2)=O)C)n[nH]c2c1CCOC2 N1(C(CCC=C)=O)CCN(C(=O)CC(CC)C2CCC2)CC1CC(C)(C)O c1(C(N(C(COCCO)C(=O)NCCSC(CC)OC)CC)=O)ccc2nn[nH]c2c1 N1(C(c2c(F)cc(OC)c(OC)c2)=O)CC2(CCCN(C(C3CCSC3)=O)C2)C1 C1(C(C(=O)NCCCN(C(C2C(C)C2)=O)C2CC2)O)CCOCC1 c1(CN2CC(F)(C(=O)NC(C)C(F)(F)F)C2)c(C(=O)O)[nH]c2ccccc12 CC1(C)CCC(O)(CNC(C2CCCN(C(=O)C(C3CCOCC3)O)C2)=O)C1 N1(C(c2nccc(C)n2)=O)CCC(C)C(NC(c2cnc3n2CCS3)=O)C1 C(N=c1[nH]cnc(Cl)c1F)C1CCC(NC(CC(CCC)c2ccccc2)=O)C1 N1(C(C(CCC)OCC)=O)CCC(C)(C)C(CNC(=O)C(C)=C2CCC2)C1 N1(C(c2cc(C)no2)=O)CCC2CC2(C(=O)N(c2cccc(C#N)c2)C)CC1 c1(C(=O)OC)cc(NC(N2CCCC(O)C2)=O)c(I)cn1 C=CCCCCCNC(=O)C(CC1CCOCC1)NC(=O)CC(C)c1ccco1 c1(OC)ccc(-c2ccccc2)o1.C12(CC1)C(=O)N(CC(C)=O)CCCNC2=O C(=O)(C(C)(C)CC(C)=O)N1CC(C(=O)NCc2c(CC)noc2C)C(C)C1 N1(C(Cc2c(C)ocn2)=O)CC(C)CN(C(=O)C#CC(C)(C)C)C(C)C1 C1(C(N(CC(=O)OC)CC)=O)CCCC(NC(c2ccc(Cl)o2)=O)CC1 N1(C(CC(C)n2cc(Br)cn2)=O)Cc2ccccc2CC1C1CCCC1=O C1(CONC(CN2C(C(N(CC(F)(F)CO)C)=O)CC2)=O)CCCCC1 N1(C(c2ncn(CC)n2)=O)CCC(O)(C(C)NC(c2cnn(C(C)C)c2C)=O)C1 CC(C)C(=O)C(=O)NCC1CCCC1NC(=O)Cc1cncc(O)c1 C1(C(N(C(C)C)CCNC(=O)CCc2ccon2)=O)CCCS1(=O)=O c1(OC)ccc(O)c(C(=O)OCC2CC(C(N3CCN3)=O)C2)c1 C1(NC(C2CCC(C)CN2C(=O)CCC2CCC(=O)C2)=O)CCC2CCCC1O2 N#CC1CC(C(=O)NCC2CC(NC(c3c[nH]c(=N)o3)=O)C2)C1 C1(C(=O)NCC(CNC(c2cc(OC)no2)=O)OC)CCC(C2CCC2)CC1 C1(C(=O)NOCCCF)(CC=C)CCN(C(c2cnc(N)cn2)=O)C1 C1(O)(C(C)NC(=O)COc2ccsn2)CCN(C(c2cnoc2)=O)C1 CN1CCN(C(=O)CC2CCCN(Cc3ccn(C4CCCOC4)n3)C2)CC1 c1(C(=O)NCCCCC(C)NC(c2cc(CF)on2)=O)c(F)cc(F)c(O)c1F c1(C(=O)NC2CCN(C(C3(NC(C)=O)CC3)=O)C2)ccc2c(c1)NC(=O)CS2 c1(NC(C2(F)CCN(C(C(C)OC)=O)C2)=O)cc(Br)ccc1C N1(C(C=CC)=O)CCC(CNC(c2ccc(-n3cc(Br)cn3)cc2)=O)C(C)C1 C1(NC(C(CCN(C)C)O)=O)CN(C(=O)C=Cc2cscn2)CC1N=[N+]=[N-] N1(C(C2=C(C)CCC2)=O)CCC2(CCC2)C(CNC(=O)CCCF)C1 c1(NCCc2ccc(OC)nc2)cc(=NCc2cc(C)cc(N)c2)[nH]cn1 N1(c2snc(COC)n2)CCC2(CCOCC2)C(NC(c2conc2COC)=O)C1 c1(CN(C)C(C2CCCCS2)=O)cccc(CNC(c2cnccn2)=O)c1 C1(CNC(c2cnc(Cl)s2)=O)CCC(C(N2CCC(CCO)C2)=O)O1 CC(C(=O)N1CCC2CN(C(=O)C3=CCSC3)CCC12)S(=O)(=O)C1CCOCC1 C1(NC(CNC(C)=O)=O)CCC(C)(C)CC1CNC(c1nccc(F)c1Cl)=O N1(C(C(SC)SC)=O)CCCC(C2CCCN(C(c3csc(C)c3N)=O)C2)C1 C=CCC(CC)C(=O)N1CC(NC(=O)CCCc2ccc(F)c(F)c2)C(F)C1 C(C)(C)(CCC(=O)NCC(N1CCCCC1)C)OC.C1(C)C(=O)N1 CCCCCC(CC)C(=O)N1CCC2CCN(C(C3CCC3OCC)=O)C2C1 C(CC(C(C)(C)C)NC(c1cnsc1)=O)N(C(C(c1ccc(OC)cc1)C)=O)C CCCC(O)CC(=O)NCCCCCN(C(=O)C(C)NC(c1ccsc1)=O)C C(=O)(C1=NNC(=O)CC1)N1CC(C)C(N(C)C(c2ccn(C)c2)=O)CC1 c1(C(C(N2CC(C(=O)NCc3nccc(C)c3)C2)=O)=O)ccc(Cl)cc1Cl c1(C(=O)NCCN(CCC)C(C2(O)CC2(C)C)=O)ccc(Cl)cc1F C(N=c1[nH]cc(-c2ccc(OC)nc2C)cc1C)C(CCC)C(=O)OC Cc1nc(Cl)cc(=NCC(C)(C(C)C)NC(C2CCC(C)C(C)C2)=O)[nH]1 C(=O)(C(C)(C)C(=O)N1CC(NC(c2ccccn2)=O)C2(CC2)C1)OCC CCC(C)(C(=O)N(C1CCN(C(C23CC(C)(C2)C3)=O)CC1)CC1CC1)OC C1(C(=O)NC2CCCN(C(C3(C)CC=CCC3)=O)CC2)Cc2ccccc2C1 c1(C(N2CCC(NC(C)=O)C2)=O)nnc(COCO)n1C(C)C.C(C)(C)(C)S c1(C(=O)NC2C(N(C(CC(=O)OC)=O)C)CCCC2)cnc2cccc(C)n12 C1(C)(C(=O)NCC2(F)CC(CNC(CC(C)(C)C#N)=O)C2)CCCCCCC1 c1(C(=O)NCCOC2CCN(C(C3CCC4CC34)=O)C2)cc2c(=O)[nH]ccn2n1 Cc1c(C(=O)OC(C#N)C2CC2)cnn1-c1ccc(Cl)cc1 N1(C(C2(C)CCCN(Cc3ccc(SC)cc3)C2)=O)CCC12CCOCC2 C1(CC)CN(C(c2cnc(N(C)C)cn2)=O)CC12CC2.C12CN(C1)N(CC)C2=O C12(NC(C3CCCC(C)CC3)=O)CC3CC(C1)CC(NCc1cccnc1)(C3)C2 C(CC(C)C)(C(=O)NC1CCN(C(C2CCCN2C=O)=O)C12CC2)OC C(=O)(CC(O)C(C)C)NC(C(C)NC(CNc1cc(CSCC)on1)=O)(C)C c1(OC)cnccc1C(=O)NC(CC1CCC1)C(=O)NCCOCC(F)(F)F c1(N(C)CCO)ccc(S(=O)(=O)NC2CCCC(C)O2)cc1Br.C1CNS1 C1(CC=C)(C(=O)N(C)C(C)C)CCCN(C(C2CC23CCCCC3)=O)C1 N1(C(c2cc(C)[nH]c2)=O)CCC(CNC(=O)C(C)n2cnnn2)C(C)C1 C1(COCCC)CC(NC(CCCOC)=O)CN1C(c1cnc(OC)cn1)=O O=C(C#CC1CCOCC1)NCC12CC1CN(C(=O)CC1CCC(O)C1)C2 c1(CNC(C(CC2CC2)NC(C2CCN(CC)CC2)=O)=O)ccc(C)cc1F CC(CN=c1nc(C2CCOCC2)[nH]s1)N(C)C(c1cnc(CC2CC2)nc1)=O N12CC3(CCC3)CC1C2=O.N1(C(=O)OC)CCCC(CNC(=O)CS(C)(=O)=O)C1 CC12CCOC(C(=O)NC3CC4CC(NC(=O)CCC(F)(F)F)C3C4)(C1)C2 c1(NC(=O)OCC)c(C)c[nH]c1C(=O)NCC=CCNC(=O)CC1CCC1 c1(C(N2CCC(N(C(c3cc(C)c(C)[nH]3)=O)CCO)C2)=O)nc2cccnc2s1 c1(C(=O)NCC2CC(NC(c3c(C)n(C)nc3)=O)C2)cc2c(s1)CCC2=O N12CCCC1CN(C)C(C)C2=O.C1(NC(c2cncnc2)=O)(CO)CCCC1 CC(CC(C)(C)C)C(=O)NC(CNC(=O)CCn1ccnc1)CC(F)(F)F c1(CC(N2CC(CNC(C(F)=CC)=O)CC(C)(C)C2)=O)cc(F)cc([N+](=O)[O-])c1 n1(CC)cc(C(=O)NC2CCN(C(C34CSC(C3)C4)=O)CC2F)c2ccccc12 c1(CCC(=O)N(C2C3CN(C(C4CCCCC4O)=O)CC23)C)ccc(Cl)nc1 C(C(C)(C)C(=O)N1CCC(NC(N)=O)C1)NC(C=C(C)C(C)(C)C)=O N1(C(C(C)C)=O)CCCCC1C(=O)N(N1CCOC1=O)CC1(F)CCN(C(=O)CCCF)C1 C(C(C)(C)N=c1cc(Cl)nc(COC)[nH]1)N(C(C1CCC(C)(CC)O1)=O)C c1(C(N(CCC(C)NC(CCOC)=O)C)=O)cccc(N)c1C(F)F CCCCN=C(NCc1cncn1C)NCC1(C(C)(C)C)CCCO1 n1(CC)ncc(CN(c2cc(Br)c(C(=O)O)s2)C=O)c1F C(C(C)C(=O)N(CCCNC(=O)CC1(O)CCC1)C)OCC CC(C)CC(=O)C(=O)NC1CCC(CCNC(=O)C2=COCCC2)C1 CC(C)C(CC(=O)Nc1cnc(O)c(F)c1)NC(C1CN(C)C(=O)N1)=O CCC1=NOC(CC(=O)NCC2(O)CN(C(=O)C(CC#C)C3CC3)C2)C1 CCCCC(O)C(C)C(=O)N1CC(O)CCC1C(N1CC(F)(F)C1C1CC1)=O CC(=O)CCCC(=O)NCCCC(N1CCOC(C)CC1)=O CC12CC(CCO1)N(C(C13CCCC1N(C(=O)CNC(N)=O)CC3)=O)C2 c1(C(c2n(C(CC)C)nnn2)NCCc2nncs2)cscc1S(N)(=O)=O N(C1CSc2ccc(Br)cc21)C(c1n(CC=C)nnn1)C1CCC1 C1(NC(C(C(C)C)C)=O)C2CCC1CN(C(=O)C(C)(O)C(F)(F)F)C2 C#CC1(NC(=O)C(C2CCCO2)NC(=O)COCC(C)(C)C)CCCOC1 C=CCC(CC(C)C)C(=O)NC1CC2CN(C(c3ncsc3C(C)C)=O)CC12 Brc1ccc2c(c1)CCN(c1nccc(=NCC3C4COCC34)[nH]1)C2 c1(NC(c2cnc(C3CC3)nc2)=O)ccc2c(c1)S(=O)(=O)C=C2 c1(C(=O)NC(C)CCNC(C2CC(O)CN2C)=O)c[nH]c2ccc(O)cc12 C1(C(=O)NC2CCC(CNC(=O)Cc3ccsc3Cl)CC2)CC2CCC(C1)S2 C(CN=C(NCC1CN(Cc2ccccc2)CC1C)N1CCCC(C)C1)OC C(CCC(=O)N(CCNC(=O)C(C)N(C)C(C)=O)CCOC)OCCC Cc1nc(C(=O)NC2CCCCC2CNC(=O)CCc2cn(C)nn2)c(C)s1 C1(CC)CN(C(=O)Cc2nocc2C)CCN1C(c1cnccc1C(F)F)=O c1(OCC(=O)NCC2CCN2C(c2cnn(CCF)c2)=O)ccc(Cl)cc1Cl C1(CC(=O)N(CCCO)CCOC)C2CCCC2N1C(=O)CC1CCSCC1 c1(CC)cc(C(N2CCCC2CNC(=O)C(c2c(C)noc2C)C)=O)ncn1 C(CCCCC(=O)OCCSc1nccc(OC)c1)NC(=O)C(=O)O Cc1cc(C(N2CC3C(NC(C4CC5CCC4O5)=O)C3C2)=O)c2sc(=N)[nH]c2n1 c1(C(N2CCCC(n3ccnn3)C2)=O)ccnc(Br)c1 C1(NC(c2cc([N+](=O)[O-])c[nH]2)=O)CN(C(=O)COCCO)CC12CCOCC2 N1(C(C(COC)NC(C(C)=CCC)=O)=O)CCCC(OC2CC2)CC1 c1(C(=O)NCC2(NC(C(CC)CC3CCCC3)=O)CC2)cccc2c1NCC2 C1(NC(CC(=O)OCC)Cc2ccc(F)c(Cl)c2)CCOC12CCCCC2 N1(C(CCCOCC)=O)CC2CCC(C1)N(C(c1[nH]cnc1C#N)=O)C2 N1(C(c2ccncc2-c2c[nH]c3cccnc23)=O)CCC=C(c2ccccc2)C1 N1(C(c2n(CC#C)ncc2)=O)CC=C(C(=O)N(C2(C#C)CC2)C)C1 n1(CC)cc(C(=O)NCC(C)NC(C2CCCNC2=O)=O)c(C(C)C)n1 c1(C(N2CCCN(CCNC(C3C(=C)CC3)=O)CC2)=O)cc(Cl)c(F)cc1F c1(CC(N2CCN(C3CN(C(CC)=O)C3)CC2)=O)ccc(F)c(Cl)c1 Cc1cc(C(N2CCC(C3CCCN3C(=O)CO)CC2)=O)c2ccccc2n1 N1(C(C=CCOC)=O)CC(CNC(C2(CCN(C)C)CC2)=O)OC(C)C1 n1(C2CCN(C(c3cc(OC)c(Br)s3)=O)CC2)cnc2cc(OC)ccc12 C1(NC(C2C(CC)C2)=O)CC2CCC(C1F)N2C(C1(S(C)(=O)=O)CC1)=O c1(CC(=O)NC2COCCN(C(CC=CC)=O)C2)c[nH]c2ccc(Br)cc12 C(=O)(CCC(=O)NCC(F)(F)F)NC1CCC(CN(C(=O)OC(C)(C)C)CC)C1 C(C(=O)N(C)OCc1csc(Nc2ccccn2)n1)NC c1(OC)c(C(=O)NCCCCCC(=O)N(C2CCCC2C)C)cccc1F C(C)(C(C(=O)N(C)Cc1cnnn1C)C(C)C)NC(c1ccc(CC)o1)=O CC1CN(C(=O)C(C2(O)CN(C(C3CC4(CCC4)CO3)=O)C2)F)CCS1=O c1(C(=O)NCC2OCCN(C(C3(OC)CCOCC3)=O)C2)c(N)cc(Cl)cc1F O=S(=O)(c1cccc2nonc12)N1CCC2(CCCCN2)C1 N1(C(c2cc(C#N)sc2)=O)CCC(CO)C(NC(=O)CNC(c2ccsc2)=O)C1 c1(CC)c(C(=O)NC2CCOCC2C(=O)NC(CN(C)C)CO)cnn1C N1(C(C(=O)NCC(F)F)=O)CC2CCC1CN(C(C1C=CCS1)=O)C2 C1(NC(c2cccc(N3CCC(O)C3)c2)=O)COCCN(Cc2ccns2)C1 N1(C(c2c(C)c(N)cnc2)=O)CC2CC(C1)CN(C(=O)COCC1CCOC1)C2 N1(c2nccc(SC)n2)CC=C(CNC(=O)CN2C(=O)CN(C)C2=O)CC1 C1(CCNC(C(c2cncc(F)c2)C)=O)CCCN(C(=O)Cn2ccnn2)C1 N1(S(c2cccc(C(C)C)c2)(=O)=O)CCC2(CCCN2C)CC1 N1(C(C=CC(CC)=CC)=O)CCC(CC)(NC(=O)C(O)Cc2cn(C)cn2)CC1 N1(C(C(C(C)CNC(C23CCC(CC2)CC3)=O)F)=O)CC(O)(C2CCC2)C1 n1(CCOC)ccc(C(=O)NCCCCn2cc(C3CCCOC3)nn2)n1 C1(NC(c2c(CC)nns2)=O)CCCC1(C)CNC(=O)C(O)CCc1ccccc1 c1(N2CC(NCc3cccc(C)c3F)C(C)C2)ncnn2cc(Br)cc12 c1(C(F)(F)F)ccoc1CNC1CCCOC1 c1(OC)cccc(NC(=O)CCC2CC(NC(C3(CC4CC4)CCC3)=O)C2)c1 N1(C(CSCC(N)=O)=O)CC2CC1CN2C(=O)C(CC(F)F)c1ccccc1 c1(SCC(=O)NCCC(=O)NCCC(=O)OCC)cc(=O)n2nc(C)sc2n1 c1(C(=O)NCC(CCNC(CC(C(=O)OC)C)=O)(C)C)nc(C)n2ccccc12 c1(OC)cc(C)nc(NCc2ccc(=O)n(CCN3CCOCC3)c2)n1 N1(NC(NCC(CC)CO)=NCc2cc(C)on2)CCN(C(C)C)CC1 C1(C(=O)NC2C(OC)CCOC2)CN(C(=O)C=Cc2cncn2C)CC1C1CC1 C1(NC(c2c(C)cn(C)n2)=O)CC2CCC(C1)N2C(c1c(C)nc(C)nc1C)=O C1(CNC(C(Cn2cccn2)NC(CCC=C(C)C)=O)=O)C2CCCCCC12 C(=O)(C1=CCC(C)(C)CC1)N1C(=S)NC(C(=O)OCC)C2=C1C(C)(C)N(CC)C2=O Cc1cc(C(N2CC3C(NC(C4CCCCC4O)=O)C3C2)=O)cc2c1NCCC2 C(=O)(CC1=NNC(=O)C1)N(CC(C)CNC(=O)Cn1cc(C(F)(F)F)nn1)C C12(CNCC(CCCC)NC(=O)OC(C)(C)C)CCC(O)(CC1)CC2 Cc1ncc(CC(=O)NCC2COC(CNC(=O)Cc3cc(C)[nH]n3)C2)s1 C#CCC(CC#C)C(=O)NCCN(C(c1ccc(C(C)C)nc1)=O)CC1CC1 c1(C(C(=O)NC2C(NC(C(C(C)C)N(C)C)=O)CCC2)(C)C)cccc(Cl)c1F S(=O)(=O)(c1c[nH]ccc1=NCc1nccc(C2CC2)n1)NCCCCCCSC C1(CNC(C(CO)N(C)C)=O)CCN(C(c2csc(CO)n2)=O)C12CC2 c1(C(=O)NCC2(F)CC(CNC(c3n(CC)ccc3)=O)C2)c(F)ccc(F)c1O S(=O)(=O)(c1ccc(OC)c(C)c1)Nc1cc2[nH]cc(C(=O)NC)c2cc1 N1(Cc2nnc(-c3ccc(Cl)nc3)s2)CC2(c3nn[nH]n3)CCC1CC2 c1(CC(N2CC(C)C(NC(C3CCCC34CC4)=O)C2)=O)ccc(F)c(Cl)c1 CC(CS(C)=O)C(=O)NCC1(CNC(C2(F)CC=CC2)=O)CCCCC1 c1(N2CCCC(NC(c3cccc4cc[nH]c34)=O)C2)ncc([N+](=O)[O-])cn1 C(=O)(C(Cc1ccccc1)C(F)(F)F)NC1(C)CCN(C(=O)CCCF)C1 c1(C(=O)NC2C(NC(C3(C(=O)NC)CCC3)=O)CCC2)ccc([N+](=O)[O-])o1 N1(C(CCC=CC)=O)C(CNC(=O)CC2CCC(OC)CC2)CC2CCCC12 C12(C(N(CC(C)(C)CNC(=O)CCCC3CCCCC3)C)=O)CCCC1CC2 Cc1cc2cc(-c3ccc(NS(=O)(=O)CCCCl)cc3)ccc2nc1NC(C)C C(c1cccc(Cl)c1)=C(C)C(=O)NCC1(CN(C)C(C2OCCOC2C)=O)CC1 Cc1c(Cl)cnn1CC(=O)NC1CCCC1CNC(=O)COCc1ccncc1 Cc1ncccc1C(C)NC(c1cc(CO)[nH]n1)c1nnnn1CC1CCCO1 c1(CNc2ccc(NC(C)=O)cc2)c(F)cc(Br)cc1[N+](=O)[O-] C12(C(=O)NCC3(CNC(C(CC)COC)=O)CC3(F)F)CC3CC(CC1C3)C2 Cc1ccc(C)c(C(N2CCCC(CNC(=O)COc3ccon3)CC2)=O)c1 C1(CC(=O)N(C2CS(=O)(=O)C2)C2CC3CC2CN3)CCCC2(CC2)C1 C1(NC(C23CC(CN(C(C=C(CC)CC)=O)C2)C3)=O)CC(C)N(C)CC1C CCC(C)(C)C(O)C(=O)NCC(C)N(C)C(c1cccc(O)n1)=O c1(C(=O)NC(CNC(CC2(NC(C)=O)CC2)=O)CO)csc2ccccc12 C1(C(=O)NC(C)C(C)(C)CN(C)C)CC2CN(C(=O)CN3CCOCC3)CC2C1 C(=O)(CC(C)CN(C)C)NC(CCCNC(c1nc(C)[nH]n1)=O)c1ccccc1 c1(NC(N2C(C(C)OCCOCCOC)COCC2)=O)noc2c1COCC2 c1(C(N2CCC(NC(C(C)OCC)=O)C(O)C2)=O)cn(C)c(=O)c(C)n1 N1(C(C(C)CN2CCOCC2)=O)CCC(CO)(NC(=O)Cc2cc(Cl)n(C)n2)C1 Cn1c(S(=O)(=O)N2CCCC2)cc2ccccc12.C(CCOC(F)F)O N12C(C)=C3C=CC(=O)N(C=CC=CC=S13)CCC(C)N(CC)C2=O.CC.NC c1(CS(=O)(=O)N(C)C)ccc(C(F)(F)F)c(Cl)c1.c12ccccc1CNC(=O)N2 C1(CCC)(CNC(=O)CC2CC2COC)CCCN1C(c1ccco1)=O C1(F)(C(=O)NC2(CCCNC(CCSCC(C)C)=O)CC2)CCN(C)CC1 c1(OCC)cc(NC(=O)CCC2CCCN2Cc2cn(C)nn2)ccc1Cl C(c1cnccn1)=CC(=O)NC1CC(NC(=O)C(O)C2CC2)CC1O c1(C(=O)NC(CC#C)C(=O)NCc2cc(COC)no2)cc(C)c(F)cn1 N1(C(CCc2cnc(C)o2)=O)CCC(CNC(c2nnc(C)s2)=O)C12CC2 C1(C(=O)NCCC(O)C2CC2)(NC(C(C=C)O)=O)CCOCC1 n1(CCCC(NC(CC(C)C)(C)CCCl)CO)c(O)nc2cc(Cl)ccc12.c1(=O)c(=O)[nH]1 C1(NCc2c(C(OCC)OC)cccc2)CCS(=O)(=O)CC1 Cc1cccc(F)c1C(=O)NC1COCCN(C(c2cnn(C)c2C#N)=O)C1 CC1=NOC(C)(C(=O)NCC(CNC(c2cccnc2O)=O)CO)C1 C(C(CC(=O)N1CCC1C(C1CCC1)=O)C1CCC1)NC(c1n(C)ccc1)=O.C c1(C(=O)NC2CCN(C(C(CC)CC(C)C)=O)C2)cc(Cl)cc([N+](=O)[O-])c1 c1(C(=O)NCC(C)(C2CC2)NC(c2cnn(CC)n2)=O)ccc([N+](=O)[O-])c(C)n1 N1(C(CC2CCN(C(C3(C#N)CCCC3)=O)CC2)=O)CCC2(CC1)CC2 Cc1cc(=NC2COC3(CCC3)C2)[nH]c(NC2Cc3ccccc3C2)n1 c1(OC)ccc(C(N2CCC(CN(C)C(C34CC(C3)C4)=O)C2)=O)c(OC)c1 C(=O)(CCC(F)(F)F)NC(CN(C(C1(SC)CC(=O)C1)=O)C)C N1(C(C2(C)CC(C#N)C2)=O)C2CCC1CN(C(=O)CC13COC(CF)(C1)C3)CC2 C(=O)(C(C)C(O)C(C)C)N(C1CCC(NC(c2cnc(C)[nH]2)=O)CC1)CC c1(C(N2CCC(OCCNC(C(COCC)(C)C)=O)C2)=O)cc(Cl)ncc1O C1(O)(C(CNC(C(C)OCCC=C)=O)(C)C)CN(C(c2cnc(C(C)C)[nH]2)=O)C1 C(N=c1[nH]c(C)nc2[nH]ccc12)C1CCN(C(c2ccc(CCC)[nH]2)=O)CC1C N1(C(Cc2c(C)nn(C)c2)=O)CCC(C(=O)NCCC#CCO)C(O)C1 C1(CN(C(=O)CC(F)F)CC)CCCCN1C(=O)COc1ccc(Cl)cc1 C1(CNC(COC)=O)CC(O)(CNN(C(C2OCCC2CC2CC2)=O)C)C1 c1(C(N2CCC(C(C(=O)NCC(CCC)CCO)C)C2)=O)cccc(C#N)c1C C1(CCCNC(CN(C)CC)=O)CCCN1C(=O)CSC.C1=NC(=O)C1 c1(C(C(C)C)NC(CCC)C)cccc(C(F)(F)F)c1 C12(C(=O)OC)CN(C(c3ccc(F)s3)=O)C(CO)(C1)C2 CCS(=O)CC(=O)NCc1cccc(CNC(=O)Cn2nnc(=O)[nH]2)c1 c1(C(=O)NCC2(C(=O)NC3CC(C#C)C3)CC(C)(C)C2)cccc(C#N)c1C N1(C(CN(C(C(C)CC(F)(F)F)=O)C2CCC2)=O)CC2(CCC(O)CC2)C1 N1(C(C2CC(C)(C)C2)=O)CCN(C(=O)C=CCF)C(C2CC2)C1 N1(C(c2ccc(C#N)o2)=O)CCN(C(c2cncc(N3CCCC3=O)c2)=O)C2CC12 N1(CC(N2CCC(N(CCC)C(C3CC(C)(C)O3)=O)C2)=O)CCN(C)CC1 O=C(NNC(=S)Nc1ccc(I)cc1)C(F)CC(Cl)Cl C12(C)CC(C1)NC(=O)O2.C(=O)(CCC=C(C)C)OC(C=CC)=O c1(NC(CCC(C)NC(C2N(C(C)=O)CCC2)=O)=O)c(C)cc(C)nc1C c1(OC)cc(Br)c(CN2CCC(NC(c3ccc(Br)c(O)c3)=O)C2)cc1O O=S(=O)(c1ccc(Cl)s1)N1CCN(Cc2ccc(N3CCOCC3)cc2)CC1 c1(C(N2CCCN(Cc3ccc(C)nc3Cl)CC2)=O)ccc2c(c1)ncn2C C(=O)(CCCCCC(C)C)N(CC(C)(C)CNC(c1cc(SC)oc1C)=O)CC N1(C(C(C(=O)OCC)F)=O)CCC(NC(C2CC3(CSC3)C2)=O)C(O)C1 N1(C(c2c(O)ncc(CC)c2)=O)CC(NC(C2CCCS2(=O)=O)=O)CC12CCC2 c1(-n2cc(CO)nn2)ccc2cnc(C=O)n2c1C.N1(N(CC=C)CC)CC(F)C1 C1(NC(C2(CCC)CC2)=O)CN(C(c2cnn(C)c2Br)=O)CC1C(F)(F)F c1(C(=O)NC2C(NC(CCNC(COC)=O)=O)C2)cc(OC)cc(Cl)c1O C(CS(=O)c1ccccc1F)NC(=O)NC1(CC)CCOC1 c1(C(N2CCC(O)(CCNC(c3ccc(Cl)s3)=O)CC2)=O)cccc2nsnc12 CC1CCCN(C(C2(NC(c3ccc([N+](=O)[O-])[nH]3)=O)CCC(C)(C)C2)=O)CC1 c1(C2C(C(=O)NC3CN(C(C(CC)F)=O)CC3F)C2)ccc2c(c1)OCCO2 C1(N(C(=O)C(O)CN(C)C)C)CN(C(C2(F)CCOC2)=O)CCC1O Cn1cc([N+](=O)[O-])cc1C(N1CCCC(C)(NC(=O)CCCNC(N)=O)C1)=O c1(C(=O)NS(c2cccc(OC)c2)(=O)=O)cc2c(=O)[nH]ccn2n1 C1(NC(C=CC(=O)NC2CCCC2C(F)F)=O)CCC2(CC2)C1 C=C1CCN(C(C2CCCN(C(C)C)C2)C(=O)NC2CCCC2)CC1 c1(C(N2C(CNC(C=CC(CC)=CC)=O)CCC2)=O)cc(Cl)c(Cl)n1C N1(C(C(N2C(=O)CCC2=O)C)=O)CCCCC(CNC(=O)CN(C)C(N)=O)C1 C=CC1CN(C(=O)CC2CN(C(c3cccc(C#N)c3)=O)CC2C)CC1O c1(COC(=O)N(C)CC2CCCO2)ccc(CC2CCCN(N)C2)cc1 Cc1cc(O)ncc1C(=O)N(CC(C)O)CCNC(c1cscc1C#N)=O Cc1ccc(C)c(C(CCNC(=O)C(F)(F)CN(C)C)C(=O)O)c1 Cc1[nH]nc(I)c1C(N1CCC(NC(=O)CN(C)C)C1)=O c1(C(=O)NCCCCNC(=O)CC2CCOC2)cc2cccnn2n1 CC1CCCC=C1C(=O)NC(CC(C)(C)C)C(=O)N(CCCn1ccnc1)C CC(C(=O)N(C)CCOCCCN(C(=O)CCC1CC1(Cl)Cl)C)=C1CC1 c1(C(CC2CCC2)NC(c2n(C(C(=O)NC)C)nnn2)=O)ccc(C)cc1Br C(C#Cc1cccnc1)NC(CC1N(C(c2cc(=N)[nH][nH]2)=O)CC1)=O c1(CNC(CCCC#C)=O)nc(C)nc(Cl)c1C C1(CC=C)(C(=O)N(c2ccc(OC)cc2)C)CCN(C(=O)C=CCOC)C1 C(=O)(C(C(=O)N(C1(CC(=O)NCCC2CCCOC2)CC1)C)OC)OC C(=O)(C(F)(F)C(F)F)NCCC(C)CCNC(C1CCCC1C)=O Cc1cc(C(=O)N(C)CCNC(=O)Cc2cnnn2C)cnc1C c1(C(=O)NCC2N(C(CC(CCC)O)=O)CC(C)(C)C2)cnc2ncccc2c1 CCCCC(C(=O)N1CC(c2cc[nH]n2)C1)NC(c1ccoc1Cl)=O c1(OCC)ccc(C(=O)NCC2CC(F)(F)CN2C(=O)C(C)(C)O)cc1[N+](=O)[O-] N1(C(C2=CC(C)(C)C2)=O)CCC2CC2(C(=O)Nc2ccc(N=[N+]=[N-])cc2)CC1 C(=O)(C(C)(C)C(=O)N1CC2CC1CN2C(C1CCC=CCCC1)=O)OC(C)(C)C c1(C(=O)NC2(C3N(C(C(C)N4CCCC4)=O)CCC3)CC2)ccc2occc2c1 C(=O)(C=C1SCC(=O)N1C)NC1CC2(CN(C(C(C(CC)(C)C)O)=O)C2)OC1 c1(NC(C2CCCC(C(=O)O)CC2)=O)ccc(C(N2CCCC2)=O)cc1O C1(NC(=O)CC2CCCOCC2)CC12CCN(C(c1ccnc(O)c1)=O)CC2 N1(C(c2c(OC)c[nH]n2)=O)CCCC(C)C1CCNC(c1cn(C)c(=O)cn1)=O n1(CCCC)cc(C(=O)N(C2CCN(CC3CCCC(F)C3)CC2)C)c(C)n1 C(=O)(C(C)(C)C1=CCSCC1)NC(CC(C)C)(C)CNC(C1COCCO1)=O c1(C(N(C2CCCCN(C(c3ccnc(O)c3)=O)C2)C)=O)ccc(C#N)c(O)c1 N(C(=NCCCCN1CCCC1)NCCC1(C)CCCO1)C(C=C)C Cc1nsc(C)c1C(N1CCCC1C(C)(C)CNC(=O)C(c1cnn(C)c1)=O)=O C(C1CCCN1C(=O)CC1CCSC1)=CC(=O)NCCCC(=C)Cl CC1(C)CN(C(c2cscc2Cl)=O)CCC1NC(=O)C1=CS(=O)CCC1 c1(C2N(C(C3CC(C)(NC(C4CC(Cl)(Cl)C4)=O)C3)=O)CCC2)cccc(F)c1F c1(N2C(C)(CNC(Cc3cncc(C)c3)=O)CCC2)cc(C)nc2ncnn12 CC1(C(=O)NCC2CCCC2C(N2CC(O)(c3nn[nH]n3)C2)=O)CCC(=O)C1 Cc1nc(CN(CCN)CCC(C)(C)C)no1 C1(NC(C2N(C)CCC2)=O)CC2(C1)CC(C(=O)NCC(O)Cn1cccn1)C2 C1(NC(c2cn(CC)nc2C)=O)CCCCN(C(=O)C(CCOC)OC)CC1 c1(OCC)cc(C)c2cc(CNCC(C(F)(F)F)OC)[nH]c2c1 c1(OC)ccc(-c2ccccc2)cc1C.n12nc(CCO)nc1-c1ocnc1C2 c1(C(N(CC(CNC(c2c(CC)scc2)=O)C)C)=O)cc(C)c2n[nH]cc2c1 N1(CCCN(C(C)=O)CCO)CCN(C(c2n[nH]c(C3CC3)c2Br)=O)CC1 C1(NC(c2c(C)ocn2)=O)CC(C)CN(C(=O)CS(C)(=O)=O)C1 Cc1cc(COC(=O)CNS(=O)(=O)c2cccs2)cc(C)c1F C(=O)(C(C)C(=O)OC(C)(C)C)NC1C(NC(c2c(CC)[nH]cc2)=O)CCC1 n1(CC(=O)OC)cc(NCC2CCN(c3ccccc3C)C2=O)ccc1=O CC(=O)CCCC(C)C(=O)NCCCN(C)C(c1cnc2cc[nH]c2c1)=O N1(C(C(C(C)(C)O)(F)F)=O)CCC(CNC(C2C=CC=CC=C2)=O)C(F)(F)CC1 c1(NC(C2C(C(=O)Nc3scc(C)n3)C2)=O)nc(O)nc(O)n1 CCCCC(C(=O)NC(C)(C)CCCNC(=O)N(CCOC)C(C)C)C(C)C Cc1cc(Cl)c(C(=O)NCC2CCN2C(=O)C=Cc2cccs2)cc1Br N1(C(CCc2c(C)ncs2)=O)CCC(C)(NC(=O)CCSCc2ccccc2)C1 c1(CCC(=O)NCCC(C)NC(C2(C#N)CC3CC3C2)=O)cccc(F)c1F CC(C)C(CCc1ccccc1)C(=O)NC1CC2CCC(C1)N2C c1(NCC2C(C(=O)Nc3ccc(C(F)C(F)(F)F)cn3)C2)nc2ccccc2[nH]1 N1(C(CN(c2ncc(Br)cn2)C)=O)CCN(C(C2CCCCC2F)=O)CC1 N1(C(CC(C(=C)C)OCC)=O)CCC(C(=O)NCC2CCC(CC)O2)=C(F)C1 N1(C(C=C(C)Cl)=O)CC2(NC(=O)COCc3ncnn3C)CCC1CC2 Cc1cncc(CCC(=O)NC2CCC2NC(=O)COCCN(C)C)c1 c1(CC(=O)NC2CC(C)(NC(c3nc(C)oc3)=O)C2)c[nH]c2cnccc12 CCCS(=O)(=O)C(C)C(=O)NCC(C)NC(c1ccsc1OC)=O N1(C(C2(C)CC2Br)=O)CCC(NC(C2(C(C)(F)F)CCOCC2)=O)C(F)C1 c1(C(C)=O)cnc(CC(N2CCC(CNC(c3cc(Br)no3)=O)C2)=O)[nH]1 CC(CC(N)=O)C(=O)N1CC(C(=O)NCCNC(=O)CC2CCCCC(=O)N2)C1 c1(-c2cn(C(CNC(C(C3CCOCC3)OCC)=O)C)nn2)cc(C)ccc1C CC1CN(C(c2cc(O)nc(O)n2)=O)CCC1NC(c1cc(C#N)no1)=O C=C=CCCC(=O)NC(CNC(c1c[nH]nc1C)=O)(CC)CC c1(C(N2CCCC(NC(c3scc(C)c3)=O)C2C)=O)ccc2[nH]cc(C#N)c2c1 S(=O)(=O)(c1ccc2nc(Cl)ccc2c1)NC(C1(CCC)CCC1)=O c1(CC(N2CC(CC)(NC(=O)CCc3ccsc3)C2)=O)ccc(Br)cn1 N1(C(=O)OC(C)(C)C)CCC2(CC1)CC2CNC(=O)NCCc1cn(C)nc1Cl C(=O)(CCC(=O)NC1CCN(C(c2c[nH]nc2-c2cnn(C)c2)=O)C1)OCC C(=O)(CC(C(C)C)OCC)N(C(CCNC(C1(C#C)CC1)=O)C)C c1(N2CC3C(C(=O)Nc4ccc(C)nc4)C3C2)nc(Cl)c2c(n1)COC2 N12CCCC(C1)CC(=O)NC1(CCC1)C2=O.n1(CC)nc(C(=O)OC)cc1C C(=O)(C1=CCCOCC1)NC1CCN(CCNC(c2[nH]cc(C)c2C)=O)CC1 c1(C(N2CC=C(CCNC(C(F)=C(C)C)=O)CC2)=O)ccc2n[nH]c(C)c2c1Cl C1(NC(C2C(=C)CC2)=O)COCCN(C(=O)C(C)=C(C)CC)C1 N1(C(c2ncn(CC)c2)=O)CCC2CCCN(C(=O)CN3CC(C)C3)C2C1 C1(C(=O)NCC(C)(C)CC2CN(C(=O)CC3CCCOC3)C2)COCCC1(F)F C(=O)(CC(C)(C)C1CC1)NC1(C)CN(C(=O)COC2CCCOC2)C1 C1(NC(c2cccc(N(C)C)c2)=O)CC2(NC(c3ccoc3)=O)COC1C2 N1(C(CC=CCC)=O)CC2ON=C(CNC(c3c(Cl)nc4ccccn34)=O)C2C1 CCC(CC(=O)NCC(N1CCN(C(c2cccn2C(C)C)=O)CC1)C)C(C)C Cc1cccc(CC(=O)NCC2CCC(C)N(C(=O)C3=NOCC3)C2)c1C C1(CCOC)CN(C(=O)C(C)(O)C2CC2)CCN1C(c1cc(Cl)no1)=O C1(C(C)NC(c2ccc(-c3cccs3)s2)=O)CN(C(C2CC(O)C2)=O)CCO1 C(C(C)C(F)C(=O)NC1(C(F)F)CCC1)NC(c1c(CC=C)cccc1)=O C1(C(C)(O)CNC(C2CCO2)=O)CCN(C(=O)COC2CCC2)CC1 N1(C(c2cc(C(C)=O)on2)=O)CCOCC1CNC(=O)CCc1cnn(C)c1 CCCCCC(C)CC(=O)NCC(C(C)C(C)C)NC(=O)C(CC)NS(C)(=O)=O N1(C(c2c(CC)c[nH]c2)=O)CC(C2CN(C(c3sccc3Br)=O)C2)C1 C1(NC(c2c(C)csc2Cl)=O)CN(C(c2[nH]nc(C(F)(F)F)c2C)=O)CC2(CC2)C1 c1(C(=O)NC(C)CCCNC(C2CC2(Cl)Cl)=O)cccc2nsnc12 c1(C(=O)NC2CC(CNC(=O)COCc3cccnc3)C2)c(Cl)cccc1Cl O=C(C1=NNC(C(F)(F)F)C1)N1CCC(O)(CCNC(C2CC(O)C2)=O)CC1 Nc1c(C(=O)NC2CC2CNC(c2n[nH]c3c2CSCC3)=O)cc(F)cc1Cl c1(NC(C2C3CN(C(C4CN(C)C(=O)C4)=O)CC32)=O)cccc2cccnc12 c1(CC(C)NC(=O)CCNC(c2cscc2Br)=O)ccccc1F C(CC(N)=O)(C(=O)NC1(c2nc[nH]n2)CC1)NC(C=Cc1ccc(C)o1)=O c1(CSCC(C(=O)OCC)(F)F)nccc2ccc(OC)cc12 C1(OCC)CCCN(C(C2CC3CC3N2C(c2occc2CC)=O)=O)C1 C1(NC(CC(C)F)=O)(CO)CCCN(C(c2cnsn2)=O)C1 C1(CNC(CC=CC=C)=O)C2CN(C(=O)C(O)CCc3ccccc3)CC12 CN1CCC2C(CCN2C(C2CC(NC(=O)C=Cc3ccc[nH]3)C(O)C2)=O)C1 c1(C(N(C2CCCC(NC(C(=O)NCC)=O)C2)C)=O)cncc2cnccc12 c1(OCC(=O)NC2C(CNC(C(C)OCCCC)=O)CCC2)ccc(Cl)c(F)c1 C12(NC(c3c(C)onc3)=O)CCCC1CN(C(c1ccnn1C1CC1(F)F)=O)C2 C1(NC(=O)C2=CCCS2)CCC2CN(C(C3C4(CC4)C34CC4)=O)CC2C1 C#Cc1ccc(C)c(NC(=O)C(O)C(CCC)NC(=O)CC(O)C(C)C)c1 C1(C(=O)NCc2ccc(C)nn2)(COC)C=CCN1C(=O)CC1C(C)(C)C1(C)C c1(C(=O)NCC(C)NC(c2cc(OC)ncc2)=O)coc2c(F)cccc12 C(=O)(CCCCCn1cnnn1)NC(CC(C)C)CNC(=O)C=Cc1ccoc1 CC(CNC(=O)CSCc1ccncc1)(CO)NC(C1CC(C)(O)C1)=O CCCC(CNC(C1(C)CCOCC1)=O)C(=O)NCC(C)(O)C(C)C c1(C(=O)NC2CC(n3cc(-c4cc(OC)ncc4)nn3)C2)ccc(OC)cc1C C1(C)(C(=O)NCCN(C(c2c(C)n(CC(C)(C)O)nc2)=O)C)CCCCC1C c1(C(N2CCCN(C(C(C=CC)(F)F)=O)CC2)=O)csc(=NC2CCCCC2)[nH]1 c1(C(N2CC(F)CC(NC(C3C(C(=O)OCC)C3)=O)C2)=O)cn(C)c(C)cc1=O c1(OC)ccc(C(F)(F)C(=O)NC2CC(C)C2)cn1.c12cccc(c1)CNC2=O Cc1nnc2n1CCC(C(=O)NCC1C3CCCC1N(C(=O)C=C1CCC1)C3)C2 C=CC(CCC)CC(=O)N(C)CC1(O)CCCN(C(=O)CC2CC(=C)C2)C1 N1(C(C=C(CC)CC)=O)CCC(NC(c2cnc3[nH]ccnc2-3)=O)CC(O)C1 N#Cc1ccccc1CNC(=O)CC1C(NC(C2OC3CCC2C3)=O)CC1O C1(CNC(C(C)NC(C)=O)=O)CCCCN(C(C2COC(C)C2)=O)C1 Cc1nnc(CCC(=O)NCC(C)(C)NC(=O)C(C)CC2CC2)n1C CN1CCN(C(C23CC(CO)(CN2C(C2(C)CC(F)(F)C2)=O)C3)=O)C(CO)C1 c1(C(N2CC3C(NC(=O)C(O)C4CC4)C(C3)C2)=O)coc(=O)c2ccccc12 N1(C(CC(CC=C)NC(=O)C(SC)SC)=O)CCC(F)(F)C(F)C1 C1(NC(CCOCC#C)=O)CCC12CN(C(c1ccc(C)nc1C1CC1)=O)C2 C(CCCCC(=O)N(C)C)NC(C)=O.C1CCN(C(=O)COCCCF)CCN1 C12CCCN(CC1)C2=O.CCC(CC1CCCC1)C(=O)NCC(=O)NCC(F)(F)F C12(C(=O)NC(CNC(C=C(CC)CC)=O)(C)C(C)C)CCCN1CC(OC)C2 C1(NC(C(C)C)=O)CCN(C(c2csc(N(c3ccccc3)C)n2)=O)C1C(C)C C1(C(=O)NCC#CCNC(=O)COC(F)F)CCc2nn[nH]c2C1 C(C)(C(C)C(=O)NC(C)CCCCO)NC(c1cc(C)sc1)=O c1(C(=O)NCC2CC(NC(COCCCC)=O)CC2O)ccc2ncc(C)n2c1 c1(-c2cn(C3CCN(C(C(COC)N(C)C)=O)C3)nn2)c(C)cnn1C CC(C)C(CCN(C(=O)CN1CCC(C)CC1)C)NC(=O)CCn1ccc(=N)[nH]1 C(C(C)(C)N=c1[nH]nc(C(F)(F)F)s1)N(C)C(c1ccnn1C1CCCC1)=O C1(CNC(C=C2CCC(C)C2)=O)CC12CCN(C(=O)C(C)(C)C(C)(C)C)CC2 CCCCCC(CC)C(=O)NCc1ccsc1C(=O)N(c1ccccc1)C C(C(C(=O)NCC1C(C)C1(F)F)NC(=O)CCc1ncccn1)SCC c1(C(=O)NC2CN(C(C=CCC)=O)C(C)C2)ccc(=NCCOCC)[nH]c1 c1(C(C(=O)NCC(F)F)N(CCc2c(C)ncs2)C2CC2)cnn(C)c1C c1(C(=O)NCC2N(C(CNS(NC)(=O)=O)=O)CCCC2C)cc2c(ncn2C)[nH]1 c1(C(C(C)NC(=O)COCCc2cccs2)NC(=O)C(F)F)ccccc1 c1(C(N2CCOCC(NC(c3ccccc3Cl)=O)C2)=O)noc2c1CCCC2 c1(NC(CCCC)(C)c2nnnn2C2CCCC2)ccc(CC)cc1Cl Cc1ncc(Cl)c(NC(=O)NC23CC(C(=O)Nc4ccccc4C)(C2)C3)n1 N1(C(C2(CCCC)CC2)=O)CCC(F)(CNC(=O)C=CC(=O)OCC)CC1 CCC(CC(=O)N1CCC(O)(CNC(=O)CC2(CS(C)(=O)=O)CC2)C1)OC N1(C(C2(COC)CC2)=O)CCC2(NC(c3cc[nH]c3C)=O)CCCC12 N1(C(C(C)(C)SC)=O)CCCCC(CNC(=O)CC(C)C)CC1 N1(CC(C)C)CCOCC(C(=O)N(C)CC(C2CCCCC2)c2ccccc2)C1 C1(C)(CNC(C2(C)CCN(C(C)=O)C2)=O)CCCN(CCC2CCCNC2=O)C1 CN1CCC(C(=O)NCC2C3COCC23)(NC(=O)CC2OCCO2)C1 C(CC(C)C)(C(=O)N1CCCC(NC(C23CN(C(C)=O)C(C2)C3)=O)C1)NC(=O)OC Cc1cc(C)c(C(=O)NC(CNC(=O)CCCF)C(C)C)cc1C c1(C(N(C2CCN(C(CCCC)=O)C2)C)=O)cccc2c1C(C#N)C2 C1(CNC(C(C)OCC=C)=O)CC2(CCN(C(=O)CC3CCC(=O)N3C)CC2)C1 c1(CCCC(=O)NC2(N3CCC3)CC2)ccc(-c2nn[nH]n2)cc1 C(N=c1nc2ncn(C)c2c(N2CCOCC(C3CC3)C2)[nH]1)C1(OCC)CCC1 C1(CNC(C(CC)(C)CC)=O)CC2CCC(C1)N2C(c1cc(CSC)c[nH]1)=O C1(C(N(CC)CC)=O)CCN(C(c2oc(C(N)=O)cc2C)=O)C(C)C1 C1(CC(=O)NCCCCNC(c2ncn(CC)c2)=O)CCNC(=O)C1 CC(c1ccco1)=CC(=O)NC(CC(=O)NCC1CC1(CO)CO)C1CC1 c1(C(N2CC(NC(C(CC)(F)F)=O)(CO)C2)=O)cnc2ncnn2c1C c1(C(N2CC=CC(NC(c3ccc(CC)c(F)c3)=O)C2)=O)cccn2nnnc12 C1(CNC(CC=CCC)=O)CN(C(C2CC(F)(F)C2)=O)C2CCCC2O1 c1(C(=O)NC2C(CNC(=O)CSC3CC3)CCC2)cc(F)c(F)cc1Br CC1(C)CCN(C(C2(F)CCN(C(=O)C3=C(Cl)CCOC3)C2)=O)CCO1 c1(C(=O)NCC2Cc3ccccc3N2)ccc2nccnc2c1Cl c1(NCCC(C(C)C)NC(c2cn(CC)nc2)=O)ncnc2ccsc12 N1(C(CN(C)C(C2CC23CC3)=O)=O)CCN(C(=O)Cc2cccs2)CC1 Cc1ccc(C(N2CC(NC(=O)Cc3cc(Br)cs3)C(O)C2)=O)nc1C N1(C(c2c(OC)ccs2)C(=O)NCc2nnn(C)n2)CCC12CCCOCC2 Cc1c(Br)sc2ccc(NC(=O)CCC(F)(F)F)cc12 C1(CNC(C=CC)=O)CN(C(c2[nH]c(C)nc2C)=O)CC1C C1(COC)CN(C(=O)CCCNC(=O)C(C2CC2)OC)CCO1 C(=O)(C(F)(F)CO)N1CC(CCCCNC(C2C(COC)C2)=O)C1 CC1CC(C(N2CC(F)(F)CC2CNC(=O)Cc2cncs2)=O)CC(=O)N1 N1(C(CC(=C=C)C)=O)CCC2CCN(C(c3cc(SC(F)(F)F)oc3C)=O)CC12 c1(CC)[nH]c(=N)sc1C(N1CCC(O)(C(C)NC(=O)CN(C)CC)C1)=O c1(C(=O)NC(COCC=C)(C)C)coc(-c2ccccc2)n1 c1(C(N(C(CCNC(C2(CCCC)CCC2)=O)C)C)=O)ncnc(C)c1OC N1(CC(=O)NCC2CCCCN2C(=O)Cc2csc(Cl)n2)CSCCSC1 C1(CC)CC(C)CN1C(=O)C(C1(O)CCCCC1)NC(C1CCC(CC)O1)=O c1(C(=O)NCCN(CC(C)O)C(C2CC3CCC(C2)O3)=O)nc(O)nc(O)c1F C(=O)(C1CCCc2ccnn21)N1C(CNC(c2nc(Cl)c(Cl)s2)=O)CC(F)(F)C1 N1(C(Cc2cc(C)on2)=O)CC(C(=O)NCc2ncc(C)s2)OC(C)C1 c1(C(=O)NC2C(NC(c3c(OCC)cccc3)=O)CCOC2)coc2c1CSC2 C(=O)(n1cncc1CN1CCCC(C(=O)N(CCCCCO)C)CC1)NC(C)=O C(=O)(CCCC(F)(F)F)NC(C(=O)N(CCCCO)C)CO N1(C(=O)Cc2cnoc2)CCCN(C(=O)C(CC2CCOCC2)CC(N)=O)CC1 N1(C(CCC#C)=O)CCN(C(C2CCCN(C(=O)CC)C2)=O)CC1CCO N1(C(c2cccc(SCC)c2)=O)CCC2CCC(C1)N2C(=O)CCC1(O)CCC1 N1(C(C(CC)n2ccnc2)=O)CCCC(NC(c2cnn(CC)c2C2CC2)=O)C1 c1(N2CCC(NC(c3nccnc3Cl)=O)C(F)C2)ncnc2c1nnn2C1CC1 Cc1nnc(O)c(C(=O)NCC2(C)CN(C(=O)C(C)C3=CCCC3)CCO2)c1C c1(C(=O)OC)[nH]c(=NCC(CC(C)C)NC(C)=O)sc1C CC(C)(C)CC(C)(C)C(=O)NC1CCC1NC(=O)CNS(C)(=O)=O c1(NC2(C3CCN(C(c4cc(Cl)c(Cl)[nH]4)=O)CC3)CC2)ncc2cccnc2n1 N1(C(c2c(C)c[nH]n2)=O)CCCC(O)(CNC(=O)C(C)(C)n2cnnn2)C1 CCCCCN(CCC(=O)N(CCCCN(C(=O)CCC1CC1C)C)C)C.CC=CC C1(NC(C(c2cccc(OC)c2)O)=O)CC2CCC(C1)N2CCCCF C=CCC(CC(=O)NCCc1ccncc1)NC(=O)Cc1sccc1C C1(NC(c2n(C)ncc2)=O)CC2CC(C1)N(C(c1cc3ccsc3[nH]1)=O)C2 N1(C(c2ccc(C#C)cc2)=O)CCC(C)N(C(C2(c3oncc3C)CC2)=O)CC1 Cc1cccc(C)c1C(N1CCCC(C(=O)NCC2(O)CCC2)C1)=O c1(CC(N2CC(NC(COCC(=O)NC)=O)C3C2C3)=O)cc(C)ccc1O c1(C(=O)NC2(C3N(C(C4(C)CCCO4)=O)CCCC3)CC2)nsc2ccccc12 C1(NC(CNC(=O)OCC=C)=O)C=CCC(C(=O)NCCCOCCF)C1 N1(C(CC2(C)CC(F)(F)C2)=O)CCCC2(C1)CN(C(=O)COc1ccsn1)CCO2 Cc1[nH]nc2ccc(C(=O)NC(C(C)(C)C)c3ccccc3)c(Cl)c12 N1(C(c2ccc(COC)[nH]2)=O)CCC(O)(CCNC(=O)CC2CCOC2)C1 C(=O)(CC(CC(C)C)NC1CCOCC1O)OCC c1(C(N2CCN(C(C(C)CC3CCC3)=O)CC2)C)ccc(Cl)cc1Cl.C1C(=O)OC1=O C(=O)(CCCCC(=O)NCc1nc(C(=O)NC2CCCNC2=O)co1)OC c1(OC)ccc(N)c(C(=O)NCC2(C)CCN(C(=O)CNC(N)=O)CC2)c1 c1(C(=O)NCCC(C)N(C(COCC(=C)C)=O)C)cccc(C2CCOC2)c1 CCC(C)(F)C(=O)NCCN(C(C1CCOC(=O)N1)=O)C1CC1 c1(CNC(COCCNC(C(C)c2cc[nH]n2)=O)=O)ccccn1 CCC(C)(C(c1nnnn1Cc1ccccc1)NCCc1noc(C)n1)OC c1(C(=O)OC)ccc(C(N2CC3C(C2)N3C(c2ccc(C)s2)=O)=O)cc1F Cc1cc(C(=O)NCC(c2ccccc2)NC(=O)C(C)N(C)C)c(C)nc1C C(=O)(CCC(C)(C)[N+](=O)[O-])N1C2(CNC(COC(C)C)=O)CCC2CC1 c1(OC)ccc2c(c1)C(C(C)C)N(C(C1(c3ccccc3C#N)CC1)=O)CC2 N1(C(CCC(C)N(C)C)=O)CCOCC(F)(CNC(c2cc(F)cs2)=O)C1 c1(C(=O)NC2CN(C(c3c[nH]c(=O)cn3)=O)C2)c[nH]cc(Br)c1=O c1(C(=O)NC2C3CN(C(C4C(CCC)CCC4)=O)CC2C3)cscc1S(C)(=O)=O C1(n2cc(CNC(C(COCC=C)c3ccccc3)=O)nn2)CCCNC1=O N1(C(C(C)n2ccnc2)=O)CC2CCC(C1)N2C(=O)C(c1cccc(Br)c1)C C(=O)(CC(C)(C)C(F)F)N(CC(=O)NC(C(=O)NCC)(C)C)C Cc1nc2ccccn2c1C(=O)NC(C)C(CO)NC(=O)C(CN(C)C)C1CC1 c1(OCC)ccc2oc(N(C)Cc3cc(OC4CCOC4)ccn3)nc2c1 Cc1cc2ncc(C(N3CCC3CNC(c3cc(C)c(Br)s3)=O)=O)cc2[nH]1 C=CC(F)(F)C(=O)NC1CC(c2ccccc2F)(C(=O)OC)C1 C(=O)(CC(C)C(C)(C)NC(c1cnoc1C(C)C)=O)NC(CC#C)C CC(C(=O)NC(C)C=CC(N1CCN(C2(C)CC2)CC1)=O)C(F)F c1(OC)ncc(C(N2CCC(N(C)C(C3CCCC(CF)C3)=O)CC2)=O)cc1Cl N1(C(C2CC(NC(=O)OC(C)(C)C)C(O)C2)=O)CCN2CC3(CC3)CC2C1 N1(c2ccnc(N3CCN(C)CC3)n2)CC2CCCCC12 c1(C(=O)OCC2CN(C(C(CC)C)=O)C(=O)C2)cnc(Br)cc1C N1(Cc2n(C)nnn2)CCC2(CCN(C(=O)C3=CCCC(C)(C)C3)CC2)CC1 N1(C(c2ccc(=N)[nH]c2)=O)CC2(CCCC(CNC(=O)CC3CC=CCC3)O2)C1 C(=O)(C(CCC(C)C)n1nnnc1C1(NCCC2CC2)CN(C(C)=O)C1)OC N1(C(C(C)C)=O)CCC(CO)C(NC(=O)Cn2cc(F)ccc2=O)C1 C1(C(=O)OC)CCOCCC1NC(=O)CCc1ccc(-c2nn[nH]n2)cc1 c1(OC(C)C)cnc(C(=O)N(C(C)CNC(=O)Cc2ccccc2O)CCO)nc1 C(=O)(C(F)C(F)(F)F)NCC(N1CC=CCC1)C(C)C CON=C(C(=O)NC1COCCN(C(c2cccc(F)c2O)=O)C1)c1ccco1 c1(C(N2CC3CCC(C2)N3C(c2cccnc2Br)=O)=O)cc(O)ccc1[N+](=O)[O-] c1(CC)cc(C(=O)NC2CC(OCC(=O)NC3CCC3(C)C)C2)c(C)o1 c1(C(=O)NC(CC(C)NC(c2cc(C)[nH]n2)=O)C)cnc(C(F)(F)F)c(C)c1 C1(NC(C(c2ccccc2)OCC)=O)COCCC1NC(C1(C)CCOCC1)=O c1(C(N2CC(CN(C(C(C(C)O)(F)F)=O)C)C2)=O)nc2ccccc2nc1O c1(OC)cccc(-c2nc(C)c(C(=O)NCCOC3CCCCC3)s2)c1 N1(CCC=C)CC(NC(=O)C(COCOC(C)C)NC(=O)OC(C)(C)C)CC1=O.SC c1(NCC(c2ccc(Br)cc2)OC(C)=O)cc(Cl)c(F)cc1C#N C(C)(C)(CC(=O)N(CC(C)(C)CNC(C1CC1(C)C(F)F)=O)C)OC C1(OC)(CNCc2c[nH]nc2-c2cccc(Cl)c2)CC(C)(C)C1 c1(OC)ccc(NC(C2CCC(CNC(C3CCC3C)=O)CC2)=O)c(F)c1 C(=O)(C(CC)C(=O)N(C(Cc1ccc(Br)cc1C)CC)CC)OCC N#Cc1ccccc1N1CC(CNC(=O)NCC2(c3cncc(Br)c3)CC2)C1 c1(C(N(CCOC)CC)=O)ncoc1CNC(=O)C(O)CC CCC(CNC(=O)C(C(C)CC)NC(C)=O)N=c1[nH]c(Cl)ncc1C(N)=O CC1OC2(C(=O)NC3CC(CNC(C4(C)CC(F)(F)C4)=O)C3)CCC1C2 Cc1c(C(=O)NC(C)CC(C)NC(c2cnc(O)s2)=O)sc2cccc(F)c12 CC1CC(c2ccccc2)CC(C)N1CC1COCC(=O)N1C CCC(C)(C(=O)Sc1cn(C)nc1C)n1nnc(C(F)(F)F)n1 CCC(CO)CN=c1[nH]c2c(c(=NCc3cnc(OC)nc3)[nH]1)CCC2 c1(C(C)(C)C)ocnc1C(=O)NCC=CCNC(c1coc(C2CCOCC2)n1)=O N1(C(c2cc(C)c(C)[nH]2)=O)CCC(F)(CNC(c2cccc(C)c2O)=O)CC1 c1(Sc2cccc(N3C(=O)C(CC)N(C)C3=O)c2)cc(NC)c2ccccc2n1 N1(C(C=CC(C)NC(=O)OC(C)(C)C)=O)CCCN(C(c2ccsc2Cl)=O)CC1 c1(NC(c2c(NC(c3c(C)cno3)=O)cccc2F)=O)cc(O)c(Cl)cc1Cl NC(CC1CCCO1)C(=O)Nc1ncc(C(F)(F)F)s1 C1(c2c(C)n(C)nc2)C(C(=O)NC(c2csc(N(C)C)n2)C)CC(=O)N1C c1(SCC(=O)NCC(CC=C)NC(c2cnc[nH]2)=O)cccc[n+]1[O-] C1(C(=O)NC(CN(C(Cc2c(C)nc[nH]2)=O)C)C)COC2(CCC2)C1 C(CC(=O)N1CCN(C2CC2)C(=O)C1)(C(F)F)NC(c1cc(CC)[nH]n1)=O c1(C(=O)NC2COCCN(C(C3(O)CCOCC3)=O)C2)ccn2c1CSCC2 c1(CC)ncc(C(=O)NC(C)CCNC(=O)C(C2CCCOC2)OC)n1C c1(OC)cc([N+](=O)[O-])ccc1C(N1CCCC(CN(C)C(c2cnns2)=O)C1)=O N1(C(C(CCSC)O)=O)CCN(C(c2cc3nc[nH]c3cc2F)=O)CC(C)(F)C1 c1(C(N2CCSCC(CO)C2)C(=O)NCCC2CC2)coc2ccccc12 C(=O)(C1=CNC2=NCCCN12)NCC1(C)CCN(C(C(C)OCC)=O)C1 c1(C(=O)NC(C(C)C)CNC(=O)C(C#N)=CC2CC2)cn2c(n1)SCC2 N1(C(C(C(C)C)SCC)=O)CC(NC(C2(n3cccn3)CCC2)=O)C2(CC2)C1 N1(C(C(CCC)C)=O)CC(CNC(=O)CCCC2CCC2)C(F)(F)C1 N(C(=NCCC1CC1)N1CCC(S(C)(=O)=O)CC1)Cc1c(OC)cncc1OC CCCC(C(=O)NC1(C(=O)NCC=Cc2cccnc2)CCCCC1)NC(C)=O C1(C2CC2)(CC(N2CC(C(C)NC(C3(C(N)=O)CC3c3ccccc3)=O)C2)=O)CC1 Cc1cc(=O)oc(C)c1C(=O)NCC(CNC(=O)CSCc1csc(=N)[nH]1)CO CC(C)CC(C(N)=O)C(=O)NCC1(CNC(=O)CNC(=O)NC2CC2)CCC1.OC C1(C(=O)NC(C(C)N(CC=CC=CCOCC(F)(F)F)C)=O)CCCCC(=O)N1 O=C(C1=NOC(C2(O)COC2)C1)NCc1cc(C(=O)NC23CCCC2C3)n[nH]1 c1(C(N2CCC(O)(CNC(c3c(CC)cco3)=O)CC2)=O)ccc(C)c(C#N)c1 CCC(O)C(=O)N(CCNC(=O)C(F)CC1CCCC1)CCOC c1(C(=O)NC(C)(CNC(C2CC=CCO2)=O)C2CC2)cc(C(F)(F)F)ncc1Cl c1(NC(c2c(C(C)NC(C(C(CC)C)C)=O)noc2)=O)ccn2nccc2c1 N=c1[nH]c(-c2ccoc2)ncc1C(=O)NCc1csc(CNC(=O)C(F)F)n1 CCC(CC)C(C)C(=O)NC1CC(CNC(=O)C(Cc2ccccc2)OC)C1 C1(NC(=O)CC2CCCC2)CC2(CCN(C(=O)COC3CC3)C2)C1 Cc1nc(CC2CC2)oc1C(=O)NCCC(C)N(C(=O)CSc1ccncc1)C O=C(C(O)CCNC(C12CC1CNC2=O)=O)NC1CCN(C2CC2)C1 c1(C(=O)NC2C(OC)CN(C(c3ccc(C)s3)=O)C2)ccc(Cl)c2occc12 Cc1cc(Cl)cc(N)c1C(N1CCC(O)C(NC(c2c(C)ncnc2C)=O)C1)=O N1(C(C(C(CC)O)C)=O)CC2CCCC(C1)N2C(c1cc(C)ccc1OCC)=O C=CCC(C)(C)CC(=O)NCC(C)(C)CC(=O)NCC#CC#CCO C1(CCNC(CCc2ccn(C)c2)=O)CCCN(C(=O)Cn2[nH]cnc2=N)CC1 C1(NC(c2c(CC=C)cccc2)=O)CC2(CCN(C(c3nocc3CC)=O)C2)C1 c1(C(=O)NCCCNC(COCCCC)=O)ccc(CN(C)C)n1C N1(C(c2cc(C)on2)=O)CCCC2(CCCN2C(=O)C(C)C(C)S(C)(=O)=O)C1 O=C(C1COc2ccc([N+](=O)[O-])cc21)NCc1ccnc(N2CCCCCC2)c1 c1(C(=O)NC2CC3CC(NC(=O)C#CC4CC4)C2C3)cc2ccnc(Cl)c2[nH]1 CC(C)C(O)C(=O)N1CCC(O)(CCNC(c2cnn(C(C)C)c2Cl)=O)C1 C1(C(NOCC=C)=O)CC2(CC2)CN1C(=O)C=CC1CCCN1C N1(C(COC)C)CCC2(CC1)CN(C(C1CCN(C)C1=O)=O)C2 c1(COC)ccc(C(N2CC(=C(F)CNC(c3cc(CF)on3)=O)C2)=O)o1 c1(CC)c(C(=O)NC2CCC2NC(C)=O)cccc1F.C1C(C)(O)C(=O)N1 N#Cc1cncc(NCC(c2c(F)cccc2Cl)O)n1 C(C)(c1ccc(F)cc1F)=CC(=O)NC1C2CCN(C(C(OC)OC)=O)CN2C1 C(=O)(N=c1cc(C)n(C(C)C)[nH]1)C1N(C(C(CC#C)N(C)C)=O)CCC1C c1(C(=O)NC(c2ccc(O)cc2)C)ccc(NC2CNC(=O)C2)cn1 C1(C(C)C)C(=O)N1.C1=CCC2(CC2)N(C)C(=O)C1.CCOCC N1(C(c2cc(C(C)C)[nH]n2)=O)CC2CN(C(=O)CC(O)C3CCCC3)CC2C1 CCCC(C(=O)NC(C1(O)CCN(C(C2(OC)CCOCC2)=O)C1)C)NC(N)=O N1(C(c2cnc(CNC(C(C)CC(F)F)=O)nc2)=O)CCCN(C)C(=O)C1 C1(NC(C(C)(O)C2CCC2)=O)CCN(C(C2CN(C3CCCCC3)C2)=O)CC1F c1(NC(C2C(C(C)C)N(C(c3ncn4c3CCC4)=O)CC2)=O)cccc(F)c1O c1(C(N2CCC(C)(CNC(c3c[nH]c(Br)c3)=O)C2)=O)cn2ccccc2n1 c1(OCC)cc2c(cc1OC)CN(C(c1ccc(C#N)cc1)C)CC2 C1(N=c2cc(Cl)c(O)n[nH]2)(CNC(=O)CC2CCC(C(F)(F)F)O2)CCC1 c1(C(=O)NCC(CO)NC(c2nc(C3CC3)cs2)=O)cncc(OC(F)(F)F)c1 c1(NC(c2nc(CC)[nH]n2)C)cc(N2CCC(Nc3ncccn3)C2)nc(C)n1 C(CC(C)C(=O)NCc1ccc(C(=O)NC2CCN(C(C)(C)C)C2)s1)=CCC C1(C#N)(N(CCC)Cc2ccc(C(=O)OC)cc2)CCCC1C(C)(C)C c1(CN(C2CC3CCC(C2)N3)C(c2c(C(C)C)n[nH]c2)=O)ccc(Cl)c(C#N)c1 N1(C(C(c2cc(C)on2)NC(=O)C(C)CO)=O)CCC2(CO)CCCCC12 c1(OC)cc(-c2ccc(C3CC3C(=O)NCCc3cccc(Br)c3)s2)ccc1F c1(OCC(=O)OC(c2cccs2)C)ccccc1F Cc1cc(C)n(Cc2cn(CC(=O)NCCCCn3ccccc3=O)nn2)n1 C(=O)(C1CCCc2sc(NC(=O)Cc3nc[nH]c3Br)nc21)OCC C(CC(O)(CC)CC)NC(COCCNC(C1C(CC)OCC1)=O)=O C1(=O)CCCC(=O)NCC(C)CN1C.c12ccnc(c1)CNC2=O.CN c1(NC(C2CN(C(C=CC=CCC)=O)CC(C)C2)=O)cccn2nccc12 N1(c2nccc(OC)n2)CCCC(N(C)C(c2n[nH]c(C)c2Br)=O)CC1 C1(NC(C(C2CCOC2)NC(=O)CC(Cl)Cl)=O)CCC2CC2CC1 C1(C(=O)NCC=CCNC(c2ccc(Br)o2)=O)COCCOC1 c1(CN2CC(C(N=c3cc(OCC)o[nH]3)=O)OCC2)cc(O)c(O)c([N+](=O)[O-])c1 C(C(C(=O)NCCC1CC(NC(=O)CCC(CC)CC)C1)C(C)(C)C)OCC=C c1(C(=O)NC(CCCOC)C(=O)N)cc2ccncc2[nH]1.C(CF)OC(C)=O N1(CCCN2CC3C(C(C)NC(c4cnsn4)=O)C3C2)OC(C)(C)CC1=O CC1CC(NC(c2cnsc2)=O)CN1C(=O)CNS(C)(=O)=O S(=O)(=O)(CCCCS(=O)(=O)NC1CSC1)NC(CCC(C)=O)C c1(C(N2C3CCN(C(C4CCSCC4)=O)C(C3)C2)=O)cc2ccc(O)nc2s1 c1(COC)ccccc1CC(=O)NCC1CN(C(c2cc(F)n(C)n2)=O)CCO1 N1(C(C(C)NC(=O)OC)=O)CCN(C(c2cnc(CC3CC3)s2)=O)C(CF)C1 c1(C(=O)NCC(CNC(C(C=C)(C)C)=O)O)ccc(N2CCCC2)c(F)c1 N1(C(CCOC)=O)CCCC1(C)CNC(=O)C=Cc1cc[nH]n1 C1(NC(C2(C)CC(=C)C2)=O)CCCCCN(C(=O)Cc2ccc3c(c2)COC3)C1 Cc1nn(C)cc1CC(=O)NCC12CC1CN(C(c1cc(Cl)ccn1)=O)C2 C1(C(=O)NC(c2ccccc2F)CNC(C(C#C)(C)C)=O)CN2CCN1CC2 c12ccc(cc1Cl)C(=O)NC2.c1(C(=O)OC)cc(N(C(C)CCSC)C)ncn1 N1(C(c2cc(C)c(F)c(C)c2)=O)CCC2(CCCCN2C(=O)CC(C)P(C)(C)=O)C1 C1(NC(C2CC(C)(C)C2)=O)CCSC12CN(C(=O)CCN1CCC1)C2 c1(OC)c(C(=O)NC2CN(C(c3ncc(Cl)nc3Cl)=O)CC2C)nc(O)nc1O N1(C(C(OCC)OCC)=O)CCC(C(=O)Nc2conc2C)(C(C)C)C1 c1(OC)cc(F)c(NC(C2CC(F)CN2Cc2cccc(Cl)c2)=O)cc1OC C1(C2CCCOC2)(N(C(c2ncc(Br)cc2C)C(=O)NC)C)CC1 CN1CC2(CC2)CC1C(=O)NCCC(C)(C)NC(=O)CCC1CC(F)(F)C1 C12(CNC(C3CC(C)OCC3)=O)CCCC1N(CCC(F)(F)F)CCC2 N1(C(C2CC(=O)NCC2)=O)CC2CS(=O)(=O)CC2(NC(C2CC3(CCC3)C2)=O)C1 C1(CC)CC(C(=O)NC(C)CCN(C)C(C2CN(c3nncs3)C2)=O)C1 c1(C(=O)NCC2CC(O)(CNC(CCC=CC)=O)C2)cccc2ncnn12 c1(C(N(CCC)CCNC(=O)Cc2csc(C(F)(F)F)n2)=O)cccc(O)n1 N1(C(c2ncn(C)c2)=O)CCC2(CC2NC(C2CC23CCCCC3)=O)C1 N#Cc1nccc(N2CC(C(N)=O)(CNC(=O)CCC3CCC(O)CC3)C2)n1 Cc1cc(O)ccc1NC(=O)CC1CCC(NC(C2CCO2)=O)CC1 C12(NC(Cc3sc(C)c(CO)n3)=O)CCC(C1)N(C(c1cn(C3CC3)nn1)=O)C2 c1(CNC(C(=O)N(C)C)=O)cnn2c1CN(C(=O)Cn1nnc(=N)[nH]1)CC2 Cc1cc(=NCC(Cl)(Cl)Cl)[nH]cc1S(=O)(=O)N(CCC(C)(C)C)C C1(C(=O)NCC2C(NC(c3ccc(CC)o3)=O)C2)CC(=O)N(c2ccccn2)C1 C(C)(C)(C(C)CC(=O)NCc1ncccn1)NC(C(CC=CCC)C)=O c1(OC)ccc2c(c1)OCC(C(=O)N1CC3CN(C(c4ccc(C)o4)=O)C3C1)=C2 N1(C(c2nc(OC)oc2)=O)CCC(O)(CN(C)C(C2(OC)CCC2)=O)CC1 Nc1cc(F)c([N+](=O)[O-])cc1C(=O)NC1CCC1NC(C1(c2ncco2)CC1)=O c1(C(=O)NC(C)C(=O)NCCc2cc[nH]n2)cc(O)cc(=O)o1 N1(C(C2N(C(C)(C)C)CC2)=O)CCN(C(C2(C#N)CCCCC2)=O)CC1CO CCC(CNC(c1nnnn1C(C)CC)C1(NC(=O)OC(C)(C)C)COC1)(CC)CO n1(CC(=O)NC(C(C)NC(C(CC)n2cncn2)=O)CO)nc(C)cc1C(F)F O=C(C1=CCN(C(c2cccc3cc[nH]c23)=O)CC1)NCCN1CCC2CC12 c1(OC)cncc(CCC(=O)NC2CC(O)(CNC(=O)Cc3nccn3C)C2)c1 C(=O)(CC(=O)NC(CCC)C)N(CCNC(=O)COC(C)CC)CCC CCC(O)(C(=O)NC1CC(CCNC(=O)Cn2nnnc2C)C1)c1ccccc1 C1(C(=O)OCC)COCCN1C(=O)Nc1ccccc1OCC(=O)OC N(C(=NCc1c(Br)cnn1C)NC1CCN(c2ccccc2)CC1)C(C=C)C C1(C(=O)Nc2ccc(CC)cc2)CN(C(=O)Cc2ccn(C)c2)CC12CC2 Cc1cccc(C)c1C(O)C(=O)NC1CCC(CNC(=O)C2=CCNCC2)CC1 CCCCCC(O)C(=O)NCC1CCN(C(C2(CC)CCC(F)(F)CC2)=O)CC1 Cc1ccc(C)c(OCC(=O)Nc2c(OC(C)(C)C)csc2C)c1 C#CC1(C(N2CC3(CC3)C2)=O)CCN(C(=O)CSC(F)F)C1 C(=O)(C(O)C1=CCCCC1)NC12CCN(C(C(C)(C)C3CCCO3)=O)C1CCC2 C1(NC(CS(CC)=O)=O)CN(C(c2cc3c(nn2)CCOC3)=O)CC2CCCC12 c1(OC2CN(C(C3N(C(CC(C)C)=O)CCOC3)=O)C2)nc(=N)nc2[nH][nH]cc1-2 CCC(C)C(C(=O)NCCc1nccnc1C)N(C(=O)CNC(=O)NC)C CC1CN(C(c2occc2F)=O)CCC1NC(=O)CCCCN(C)C C(C(=O)OC)(C(C)C)NC(CCCOCC)c1nnnn1C(C)C.N1(C)CCOCC1 c1(OC)c(C(=O)NC2CC2CNC(=O)C(C)OC)cccc1F c12nccc(n1)CN2.C1(NC(C2CCCO2)=O)CCCC1C(F)(F)F c1(NC(C)=O)ccc(C(=O)NCC(CC(F)(F)F)NC(=O)C(C)O)c(F)c1 C(CCC(C(=O)NC(C)C(C)(C)CO)NC(=O)COC1(C)CCC1)OC C1(Nc2ccnc(SC)n2)CCN(C(c2cc[nH]n2)=O)CC1O Cc1ccc2c(c1)C(NC(=O)C(=O)N1CCC1c1ccccn1)C(C)C2 C1(C(N2CCOCC(NC(CCP(C)(C)=O)=O)C2)=O)CCC2(CC1)CC(O)C2 N1(CC2CCCC(C)C2)CCC2(CCCN2C(c2cnn(C(F)F)c2)=O)CC1 C1(NC(C2CC(CCC)OCC2)=O)COCCN(C(c2sccc2C)=O)C1 Cc1ncsc1SCC(=O)NCCC(O)CNC(C1CCN(C2COC2)C1)=O C12(CNC(=O)C=Cc3nccs3)CCC(CC1NC(=O)CN1CCCCC1)C2 Cc1cc([N+](=O)[O-])cnc1C(N1CC2C(N(C(=O)C=CC3CCCO3)C)C2C1)=O O([Si](C)(C)C(C)(C)C)C(C)Cc1ccc(CNC(=O)Nc2ccc(Br)o2)cc1 C12(NC(CC=C(C)C)=O)CCCC1N(C(=O)Cc1csc(C)n1)CCC2 c1(C(=O)NCCN(C(=O)CCC2CC2)CCOC)csc(C)n1 Cc1ccccc1C(=O)NC12CC1CN(C(=O)CSc1nnnn1C)C2 c1(COC)ccc(C(=O)NC2CCCC2CNC(=O)C(F)(F)c2ccccc2)s1 C=CCC(CNC(c1cn(C)nn1)=O)C(=O)N1CCC2C(C(N)=O)C2C1 c1(C(=O)NCC(c2cccc(C)c2)NC(C2CCCS2)=O)cc2n(c1)CCCC2 c1(C(=O)OC)cc(C)c(C(N2CC(O)CC2CNC(=O)CC2CC3CC3C2)=O)o1 CCC(C)CCCC(=O)N(C)CC1(O)CCN(C(c2cncc(C3CC3)c2)=O)C1 N1(C(CCCOC)=O)CCC2(CC1)CC2CNC(=O)Cc1cc(Cl)no1 Cn1ccc2[nH]c(C(N3CCCC3(C)CNC(C3CCCN3N=O)=O)=O)cc12 C(=O)(C(F)(F)C(F)(F)F)NCCOCCN(C(CCc1ccc(C)nc1)=O)C C1(NC(C2C(C)C2)=O)CCOC12CCN(C(=O)CC(C)(C)C#N)CC2 C1(C(=O)NC(C2CCCN2C(c2cc(C(C)(C)C)n[nH]2)=O)(C)C)CCCN1C=O [SH](=O)(=O)C1(C(=O)NCC2(C(N3CC(CC)C(C)C3)=O)COC2)CCCCC1 C1(C(N(CCC(=O)NCCc2cnc(C)o2)CC=C)=O)CCCCC1C N1(C(C(C)(O)CCc2ccccc2)=O)CC2(CCN(C(=O)C3=CCC3)C2)C1 C1(CCCNC(C(=C(C)C2CC2)F)=O)CCCCN1C(=O)C(C)C1CCCC1 CC(C)CC(CC(C)C)C(=O)NCC1(C(C)NC(C2CC(O)C2)=O)CC1 C12COCC1C(=O)N2.c1(CC(=O)NCC(=O)NCC2(OC)CCC2)ccccc1 N1(C(c2c(CNC(CCC(C)N(C)C)=O)cccn2)=O)CC2(C)CCC2(C)C1 Cc1nn2cc(CC(N3CC(CNC(=O)Cc4cnoc4)CC(F)C3)=O)nc2s1 c1(C(=O)Nc2ccc(C(=O)NCC(C)(C)C)nc2)ccc(O)c(I)c1 N1(C(c2cc(CC(C)C)[nH]n2)=O)CCC(C2CN(C(C3CCC3F)=O)C2)CC1 C1(N(C(C2N(C)CCCC2)=O)C)CC2CC1N(C(=O)CC1(C)OCCO1)C2 Cc1ccc(C(=O)NCCC2CN(C(C3CC34CCC4)=O)C2)o1 c1(C(=O)OC)cn2c(n1)CC(OCCNC(=O)CNC(=O)NC1CC1)CC2 CCCCCCCCCCC(=O)N1CCCC1CNC(=O)Cn1cccnc1=O C1(C(C)C)CN(C(=O)C=C2CCCCC2)CCN1C(c1ccnc(CO)c1)=O c1(COC(CNC(CCOCC)=O)C)nc(C(N2CC(OCCO)C2)=O)cs1 CC1(C)CC(=O)CC2(COCCN2Cc2cccc(-n3cncn3)c2)C1 C(=O)(CCCCC(C)(C)C)NC1C(C)(CN(C(C(COC)C)=O)C)CCC1 CN(C1CCc2ccc(Br)cc21)C(=O)CCCCCn1cnnn1 N1(CCC)CCCN(C(C2CCCCC2COC)C(=O)NCC(C)C)CC1 C1(NC(C(N2C(=O)CCC2=O)CC)=O)CCCC12CN(C(=O)CC13CC(C1)C3)C2 CCC(C(=O)N(C1CCN(C(C2(CC)CCC2)=O)C1)CC)n1ccc(C2CC2)n1 C1(C(C2CCC(n3ccnn3)CC2)c2nc(C(C)C)[nH]n2)COCCN1C(=O)NC N1(C(CC)=O)CC(CNC(c2nnn(C3CC3)c2C(F)F)=O)C2(CC2)C1 C1(CC=C)(NC(=O)COCC(C)C)CCN(C(=O)C=Cc2ccncc2)C1 c1(C(=O)NCC2C(C(F)(F)F)CN(C(C(C3CC3)SC)=O)C2)ccc(O)c(C)c1 N1(CC2CC(C)(C)OC2)CCOC(C)(C#N)C1 C1(C(N(CC#CC)C)=O)CC(=O)CN1C(=O)C(C)N(C)C c1(C(N2CC(C(C)NC(c3cnc(C)o3)=O)OCC2)=O)nccc2ccsc12 C1(CC)C(NC(=O)CCOCCCOC)CCCN1C(=O)CC1COCC1(C)C C(C)(CCC=O)NCC.c1(COC)c[nH]nc1C(=O)NC(C(=O)OC)C1CC1 CC(C)C(C)(C)C(=O)NC1CCN(C(c2ccc3c(c2)CC3)=O)CC1O C(=O)(C1Cc2ccc(Cl)cc21)N1CC(C(N(c2ccccc2)C)=O)C(C)(C)C1 Cc1ccc(C(F)C(=O)N(C)CC2(CNC(C3CC3F)=O)CC2)cc1 C(C1=NOC2CCCCC12)n1cc(CNC(=O)CC2CC23CCOCC3)nn1 c1(C(C(=O)NC2CCCN(C(=O)C=C(C)C(C)C)CC2)OC)c(F)cccc1F Cc1c(N)ccc(C(=O)NCC2CC(NC(=O)CC3CCOCC3)C2)c1C C1(C(=O)Nc2ccc(COC)cc2F)CCC2(CN(C(C)=O)C2)O1 C(CC(=O)NC(C)CC(C)(C)C)(CC(C)C)NC(C=C=C(C)C)=O C(CCC(C)C)(c1nnnn1-c1ccccc1)NCCC=CC C(=O)(C1=CC(O)C(NC(=O)CNC(=O)CC)C1)N(C(C=C)C)C c1(CC(=O)NC(CNC(C=CCC)=O)C(C)C)ccc(OCC)nc1 c1(C(=O)NC(C2CN(C(=O)C(C)CN(C)C)CCO2)C)cn(C)cc(Br)c1=O C(=O)(C1=COCCO1)Nc1cc(C2(C)CC2)on1.N12CCC(CC1)CCC=CC2=O n1(CC(=O)NC2(CC)CN(C(c3sccc3Cl)=O)C2)c(C)c(C)sc1=O c1(NC(C(=O)NC2(C(=O)OC)CCOCC2)=O)ccc(CS(C)(=O)=O)cc1OC C(CC(C)(C)C(=O)NCC12CC(NC(=O)CSC3CCCCO3)(C1)C2)SC C(=O)(C1=C(Cl)CCC1)NC1C(NC(Cc2c(C)cco2)=O)CCC1 C1(NC(C2CCC(C(C)C)CC2)=O)CN(C(=O)C(C)(C)C(N)=O)CCC1O C1(C(=O)NCC2(C(C)(F)F)CC2)CCCN(C(=O)NC2CCOCC2)C1 n1(Cc2nc(CCCC)nn2-c2cccnc2)c(=O)cnc2ccccc12 CC1CC(CNC(=O)CS(=O)(=O)N(C)C)CN1C(c1ncc[nH]c1=O)=O n1(CCC)nc(C)cc1C(=O)NC(C)(C)CCCNC(c1csnc1C)=O c1(COC)cccc(CC(=O)NCC(F)CNC(=O)C2=NOCC2)c1 N1(C(C)C)CCCC(CC(=O)NCC2(OC)CCN(C(c3ccccn3)=O)C2)C1 C1(C(=O)NCC2CC(NC(c3cnc4n3CCC4)=O)C2)CC2CC(O)C(C1)C2 C(=O)(CCCC(=O)N1CCN(C(=O)CNC(=O)C(C)CC)C(C(F)F)C1)OC C(=O)(CC1=CCCC1)NC(CC)CNC(=O)CC1CCOCC1 Cc1ccc(CC(=O)N(C)CC2CCCN2C(C2COCCN2C)=O)cn1 Cc1cc(C(N2CCCC2CC(=O)Nc2cnn(CCO)c2)=O)cc(Cl)n1 ClCCCN=C(NCc1cccc(-n2ccnc2)c1)NCC1CCCO1 c1(C(=O)NCC(c2ccc(F)cc2)NC(C(C)SC)=O)noc(C2CC2)c1C C1(C(=O)NCC2COCCN2C(=O)C=Cc2ncc[nH]2)CC2CCCC(C1)C2 CC1OCC2(CCNCC2)C1N(CC(F)(F)F)C(c1cnn2ccccc12)=O O=C(C1CCc2ccccc21)OCCc1csc2ccccc12 C1(CC)COCCN(C(=O)CC(C)NC(=O)CC2CCN(C)C2=O)C1 Cc1cc(O)nnc1C(N1CCN(C2CN(C(=O)C(F)CC)C2)CC1)=O C(C(C)CC(=O)N1CCN(CCCNC(c2ccc(C(C)C)nc2)=O)CC1)OC Cc1cccc2c1OC(C(=O)NC1CCCC1NC(c1cncc(Cl)c1Cl)=O)C2 CC1CC(CNC(=O)C=CSc2ccco2)CN1C(=O)CCc1cnn(C)c1 C(C(=O)O)(CO)(CC(=O)O)NC(Cn1cc(-c2nccc(C)c2)nn1)=O C(=O)(CCN(OC)C(=O)c1cccc[n+]1[O-])N(CC(C)(C)C)CCC N1(C(C(C)C(=O)OC(C)(C)C)=O)CCN(C(c2ccc(O)nc2)=O)C(CCO)C1 C12(CNC(C3CC(C)(O)C3)=O)CC1CN(C(c1ccc(C(F)(F)F)nc1)=O)C2 c1(CN2CCC(C)C(NC(c3cn(C4CCC4)nn3)=O)C2)c[nH]c2ccccc12 C1(C(=O)NCCC(=O)NO)(NC(C2CC2c2nn[nH]n2)=O)CC(CO)C1 C12(C(=O)NCC3C(NC(c4c(C)n(C5CC5)cc4)=O)C3)CCCC(=O)N1CCC2 N1(C(c2ncoc2C2CC2)=O)CC(O)CC1C(=O)N(CC1CCCC1)CC1CCC1 c1(C(=O)OC)ccccc1CN1C(C(=O)Nc2cnccc2Br)CC2CC12 C1(C)(C(=O)NCC(C2CN(C(C3(OCc4ccccc4)CC3)=O)C2)C)CNC(=O)C1 N1(C(C2(C(=O)NC3(C(=O)NC)CC3)CC2(C)C)=O)CCN(C)C2(CCC2)C1 S(=O)(=O)(c1cccc(NC(CCO)C(C)C)n1)N1CC(CC)OCCC1 C12(CNC(c3c(OC)nccc3)=O)CCC1CCN2C(=O)C(C)CSC Cc1cc(C(=O)N(CC(C)O)CCNC(=O)C=CS(C)=O)c2nccc(C)c2c1 CC1=C(C(=O)NC(C(=O)NC2COC(C)(C)C2)C2CC2)CCO1 C(=O)(C(C)(O)CC(F)F)N1CC(CCC)N(C(c2ccn(C(F)F)n2)=O)CC1 O=C(C1=CCCCCC1)NC1CN(c2ccnc(C(F)(F)F)n2)CC1F C1(N(C(=O)C(c2cccnc2)NC(C2CCC2(F)F)=O)C)CCCC(O)C1 c1(C(=O)NC(CN(C(C(COC)N(C)C)=O)C)(C)C)cnc2ccccc2c1C CC(C)C(C(=O)NC1CCCC1NC(c1nn[nH]c1Cl)=O)n1cncn1 c1(CCC(=O)N(C(C)CNC(C2CN(C)C(=O)N2)=O)CC)ccc(Br)cn1 N1(C(C(=O)Nc2ccc(Cl)c(F)c2)=O)CCC2CCCCC12 C=CC(C)(CCOC)C(=O)NCc1ccc(C(N2CCOC(CC)C2)=O)nc1 Cc1ccc(C(C)C(=O)NC2CCC(CNC(c3cnoc3)=O)C2)cc1 c1(N(C)C)nc(=N)nc(N(C2CCCC2)C)[nH]1 c1(C(N2CC(CNC(CCOCC)=O)OCC2)=O)ccc2nc(O)oc2c1 c1(NC(=O)C2CC2)ccc(-n2cc(C(=O)OCC)nn2)cc1 c1(CNC(=O)NCCCc2nc(C)c(C)o2)c(O)cccc1F C1(C)(CCC)CCCN(c2nnc(C3CC3)n2CCOC)C1 C(=O)(C(C)(C)NC(c1csnn1)=O)N(CCC(C)C)C c1(CC(=O)NCCc2cccs2)csc(=NCC2CC3(CCC3)C2)[nH]1 C1(CNC(C2CCCC2O)=O)CN(C(C2COCCO2)=O)CCO1 Cc1nc(NC(=O)COc2ccc(C(C)(C)C)cc2)n(C)c1C c1(C2(C=O)CC2)ccc(F)c(Cl)c1.C12CCN(C1)N1CC(=CC(=O)N2)C1 c1(OC)cc(C)c(C(=O)NCC(C)(C)NC(c2ccccn2)=O)cc1Cl N1(C(C2(CC(C)C)CCC2)=O)CC2CC(NC(c3cc(C4CC4)[nH]n3)=O)CC1C2 C1(CC)CN(C(=O)C(O)CN(C)C)CCN1C(C1CCC(CCOC)CC1)=O C(=O)(C1=COCCC1)NCCC1(NC(CC2(C)CC2)=O)CCC1 C1(C(=O)NCCC2CC(OC3CC3)C2)CCC(C(=O)NCC2CCC2)O1 N1(C(C=C(C)C)=O)C(C(N2CC(COC(C)C)C2)=O)CC2CCCC12 c1(OC)ccc(CCCC(=O)NCCN(C(=O)CC2CCC(=O)O2)C)cc1OC N1(C(CC2CC(NC(C3CCN(C)C(=O)C3)=O)C2)=O)CCC(C2(O)CC2)CC1 C1(C(N2CCC(N(CCC)C(C3CN(S(C)(=O)=O)C3)=O)C2)=O)CC(CC)=NO1 CCCC(C(=O)NCCc1cnccn1)NC(C1(C)CC(F)(F)C1)=O Nc1cc(C(N2CC3C(NC(=O)CC4CC(=O)NC4=O)C3C2)=O)ncc1Cl N1(C(c2c(C)sc(O)n2)=O)CC2(CCCC2NC(c2cccc3scnc23)=O)C1 O=C1NCC2(CCCN(C(=O)NC3C4Cc5ccccc5C34)CC2)O1 c1(C(=O)NC(c2onc(CC)n2)C2CC2)cc2cc(F)ccc2[nH]1 C(=O)(C1=CS(=O)(=O)c2ccccc21)NC1CC(NC(CC(=O)OCC)=O)C(O)C1 N1(C(C(C(C)C)n2cccc2)=O)C2CCC1CN(C(c1ncn(C)c1C)=O)C2 Cc1ccc(NC(C2CCC(NC(c3ccc(C)c(C)n3)=O)C2)=O)c(C)n1 S(=O)(=O)(c1c[nH]c(=NCc2csc3c(Cl)cccc23)cc1C)NCC1(CC)CC1 CC(C)CCC(C)NC(=O)CC1CCN(C(=O)CCCn2cccn2)C1 N1(C(c2c(C)noc2)=O)CC(NC(c2ccc(C3SCCS3)cc2)=O)CC1C c1(C(C(=O)NC2CCN(C(C)C)C2)N(CCC)C)ccc(OC)cc1 c1(OC)ccc(NC(C2CC(CNC(=O)CC(C)c3cccnc3)C2)=O)cc1 c1(OCCC)cccc(CC(=O)NCC2C(C)CCN2C(c2coc(C)n2)=O)c1 Cn1cc(C(N2CCCCC(Nc3ncnc(C)c3F)C2)=O)c(=O)n(C)c1=O C1(C(=O)NC(C2CCCC2)CNC(C2CCC(CC)O2)=O)CCC(C)(C)CC1 N1(C(C(C)N(CCC)C(c2c[nH]c(=N)o2)=O)=O)CC(C)=CC(C)C1 C1(C(N2C(CNC(c3n(C)cc(C(N)=O)c3)=O)CC2)=O)CCC([N+](=O)[O-])CC1 c1(C(=O)NC2CC(C)CN(C(c3cccnc3O)=O)C2)cn2cccc(Br)c2n1 C=CC1(O)CCN(C(=O)CC2CCCCN2C(C23CC(C#N)(C2)C3)=O)C1 C1(C(N(c2ccc(Cl)cc2)CC)=O)CN(C(C2(C#N)CCC2)=O)CCO1 S(=O)(=O)(c1ccc2c(c1)CCCC2)N1C2CN(C(C3CCCC(C)C3)=O)CC21 CCCCCCCC(=O)NC1CC12CCC(NC(C1COC3(CCC3)C1)=O)CC2 N1(C(C2CC2NCc2ccc(OC(F)F)nc2Cl)=O)CCc2cccnc2C1 c1(C(N(CC(C)NC(C2CC(C)CC(=O)N2)=O)C)=O)cc2ccccc2s1 C(C1CN(C(C2OCCC2(C)C)=O)CC1C(=O)NCCN(C)C(C)C)=CC C(=O)(CC(C)(C)C(F)F)N(C(C=CC(=O)N(C(COC)C)C)C)CC C1(F)(CNC(COCCC=C)=O)CC(NC(=O)C=CC(C)C)C1 C(N=c1[nH]c2cc(Cl)c(S(=O)(=O)NC34CCN(CC3)C4)cc2s1)C1C(CCC)C1 C(=O)(C(C)CCCC)NC1CC(C(C(NOCCCCC)=O)F)C1 C(CC(C(=O)N(CC)Cc1cnn(C)c1)NC(=O)C(C)C1CC1)OCC C1(C)(C(=O)NCC(CCNC(c2c(OC)cnnc2)=O)O)CCC2CC2C1 C=CCC(C(=O)N(C)C(c1cn(-c2ccc(C)c(I)c2)nn1)C)C(C)C N1(C(C2(C(=O)NC)CC2)=O)CCC2(CC(NC(=O)CC3=CCCCC3)CO2)C1 Cc1c(C(N2CCC(N(C)C(c3cnn(C)n3)=O)C2)=O)sc2ccccc12 C1(NC(CCC=C)=O)CC2CC1N(C(C1C3CC4C(C3)C14)=O)C2 N#Cc1ccccc1NC(=O)CN1CCC(NC(=O)CCCCO)C(O)C1 c1(CNC(c2cnc(CC)[nH]2)=O)cnn2c1CN(C(c1c(C)n[nH]c1C)=O)CC2 C1(C)(C(=O)NC2CN(C(CSC)=O)CC3C2C3)CCCCC1(F)F c1(C(N(C2CCN(C(=O)C=CCCC(C)C)C2)CC)=O)cnc2n1CC(C)CC2 Cc1nn(C)c(Cl)c1C=CC(N1CC(CCNC(C23CC(CO2)C3)=O)C1)=O C1(F)(CNC(c2c(C)csc2)=O)CCN(C(c2ccc(C)cc2O)=O)CC1 N1(C(CCC2N(C(c3cc(C)ncc3C)=O)CCCC2)=O)CCC2(CCSC2)C1 c1(C(N2C(C=CC(=O)NC3(C4CC4)CCC3)CCC2)=O)ccc2nncn2c1 C(=O)(C(=O)NNC(=O)N1CC(C)OC(C)C1)Nc1cccc(COCC2CC2)c1 CN(C1=NS(=O)(=O)c2ccccc21)CCNC(c1csc(NCCC(N)=O)n1)=O C(CCC(=O)NCCC(C)N(C)C(c1csc(C(N)=O)n1)=O)OCC C1(C(=O)NC2CC(C)(CC)C2)CC2(CCN1C(c1cc(Cl)ns1)=O)CC2 c1(C(N2CCC(N(C)C(c3nc(Cl)sc3Cl)=O)C2)=O)cc2cccc(Cl)c2s1 c1(CC)nc(C)ncc1Br.C12CN(Cc3ccccc3)CC1NC2=O N1(C(CCOCCC)=O)CCC2CCCN(C(c3c(N)sc(C)c3C)=O)C2C1 C1(CNC(CC(=O)OC)=O)CN(C(c2occc2-c2ccccc2)=O)CCCO1 C(=O)(CS(=O)(=O)C(C)C)NC1CCCCN(C(c2c(C)sc(Cl)n2)=O)C1 CCCCCCCC(=O)NCC1CC(NC(=O)C(F)=CC2CC2)C12CCC2 CN=c1cc(C(=O)NC2CCC(NC(C34CCC3CC4)=O)C2)cc[nH]1 CC1C(NC(C23CC(NC(=O)CC4(O)CCOCC4)(C2)C3)=O)C2CCN1CC2 c1(NC(=O)Nc2cccc(NC(CCSCC(=O)OC)=O)c2)ccc(F)c(F)c1 N(C1CC(C)n2ncnc21)CCC(c1nnnn1C)CC(c1ccccc1)C c1(NC(C(N2CCC(CN(C(C)=O)C)C2)C)=O)ccc(F)c(C)c1 C1(CC)CCC(CNC(=O)C(CNC(=O)CC2(O)CCCOC2)N(C)C)CC1 CCCC(CC)C(=O)NCC(C1CCCC1)NC(=O)COCCn1cncn1 NS(=O)(=O)C1CCN(C(=O)C(=O)NC2CC3CCC2CNC3)C1 C1(CNC(=O)CCc2cn[nH]c2)C2CN(C(C3CC4(C3)CC4F)=O)CC12 N1(C(C2=C3CC(C)NC3=N2)=O)CCN(C(c2cc(O)nc(O)c2)=O)CC12CCC2 N1(C(CC2(NC(c3c(C)nn(C)c3)=O)CCCCC2)=O)CCN(C)C2CC12 c1(C(=O)NCC(CC)NC(C2CN(CC(C)C)C2)=O)ccc(Cl)cc1OC C1(C(=O)NC2CN(C(c3cc(O)nc(O)n3)=O)C3CC23)CCn2nncc2C1 C(C(=O)N1CC(CCNC(=O)CCc2ccncn2)(OC)C1)(C(C)C)SCC Cc1ccc(CCC(=O)NCC2(NC(=O)C(C)S(C)(=O)=O)CCOC2)cc1Cl Cc1cncc2cc(C(=O)NC(C3CCCCC3)CNC(=O)CC3(C)CC3)sc12 c12cn(nn1)C(=O)N1CCC1CNC(=O)N2.c1(NC(=O)CC2CC2)cnc(O)o1 C1(OCC)CN(C(C)=O)CC1CNC(=O)CNC(=O)CCc1cn[nH]c1.C(C)(=O)N Cc1cc(C(=O)NCCN(C)C(c2ncnc3sccc23)=O)c2cnn(C)c2n1 CC1CCCC(OCC(=O)N(C(C)CCNC(=O)C(C)(O)C2CC2)C)C1 CN1C(=O)CCCC1C(=O)NC1CCCC1NC(c1cncc(F)c1Cl)=O C1(NC(c2c(C)con2)=O)COC2(CCN(C(C3(n4nccn4)CC3)=O)C2)C1 c1(NCC2OCCN(C)C2)[nH]c(=NCC2(CO)CC2(C)C)nc2scnc12 N1(C(CC(C)SC)=O)CC(NC(c2c(F)cc(F)cc2F)=O)C2CCCC2C1 N1(C(C2C(OC)CCC2)=O)CC(NC(CC2(OC(C)C)CCC2)=O)C2(CC2)C1 N1(C(c2c(-n3cc(-c4cnc(C)o4)nn3)ccs2)=O)CCOC(c2cnn[nH]2)C1 Cc1cccc(C(=O)NC2CC3(C2)CC3C(=O)NCCC(O)CC(C)C)c1 N1(C(C2N(C(CCCCSC)=O)CCC2O)=O)CCCC2COCC12 N1(C(C2(C)CCC2)=O)CCc2nc(C(=O)NCCN3CCCC(O)C3)cn2CC1 C1(C(N2CCC(C)(C)C2)=O)CC2(CC(NC(C3CCNC(=O)C3)=O)C2)C1 c1(C(N2C(C(C)(C)C)CC2)=O)cnc2[nH]nc(O)c2c1.C12C(C1(C)C)CNC2=O C1(NC(CCc2ncc(C)[nH]2)=O)CN(C(c2ccnc(S)c2)=O)C2CC12 C(=O)(C(C)(C)CC(=O)N1CCCCC(CNC(=O)CC(C)C(F)(F)F)C1)OC C1(C(=O)NCCCc2ncn(C)n2)CCC12CCCO2 C1(CNC(C(C)N2CCCC2)=O)CCCC(CN(C)C(c2cc[n+]([O-])cc2)=O)C1 C1(CNC(c2cc(C(C)(F)F)on2)=O)CC2CCC1N(C(C1CC1[N+](=O)[O-])=O)C2 N1(C(c2c(I)cnn2C)C(=O)Nc2c(C)cccc2C)CCC(O)C(C)(C)C1 N1(C(c2ncc(CO)[nH]2)=O)CCC(C(=O)NCC2CCCC2CC2CC2)CC1 Cc1cc(N2CCC(NC3CCCCC3)C2C)nc(N(C)C)n1 C=CCC(CC)C(=O)NCC(C1CCN(C(c2ccn(C(C)C)n2)=O)CC1)(C)O N1(C(c2c(C)cc(CNC(c3c(C#C)c[nH]n3)=O)o2)=O)CC(C2=NOC(C)C2)C1 c1(C(=O)NCC(C(F)(F)F)NC(c2nc(CCC)sc2)=O)cc(CC)ccc1C N1(C(CCOCC)=O)CC(C(=O)NCCC2CC(C)=NO2)C2(CCC2)C1 c1(OC)ccc(CN2CCCC(CC(N3CC4CC4C3)=O)C2)cc1C Fc1cc(Cl)cc(Cl)c1CN1CCCC(C(F)(F)F)C1 N1(C(c2cccc(C)c2Br)=O)CCC(C2CN(C(=O)Cc3cc[nH]n3)C2)C1 c1(C(=O)NCC23CC(n4cc(CCO)nn4)C2C3)csc2c(F)cc(Cl)cc12 C1(C(=O)Nc2c(C)nn(C)c2)CC12CCN(C(=O)C(=O)C(C)(C)C)C2 C(=O)(C1CCCc2ncccc21)NCC(CO)NC(c1n(C)c(S)nc1)=O c1(C(N2CCC3(NC(CCOCCOC)=O)C(C2)C3)=O)cc2c(Cl)ccnc2s1 O=C(C(=O)N=c1cc(C2CC2)o[nH]1)NC12CC1CN(C(c1cccc(Cl)c1)=O)C2 c1(OC)ccc(C)cc1N.C12CCC(O1)C(=O)NCCOCCNC2=O.C1(C)CC1.OC c1(CNc2cc(C(=O)Nc3n(C)ncn3)n(C)c2)c(F)ccc2occc12 CCC(CC(=O)N(C(CC(F)(F)F)C(=O)N(C)C)C)C(C)C C1(OC)CC(NC(=O)Cc2ccns2)CN(C(=O)C(C)C(F)(F)F)C1 C1(NC(c2ccc(C)o2)=O)C2CC3C(C2)C13C(=O)N(C1CCC1)C1CC1 C=C=C(C)CC(=O)NCc1ncccc1C(=O)NCC1CCC1CO C(C1CCN(C(C2CC(CCN(C)C)C2)=O)CC1)=CC(=O)N(CCCO)CC#C c1(CNC(COC(C)C)=O)nc(CNC(c2ccc(CC#N)cc2)=O)cc(O)n1 N1(C(c2ccc(CC)cn2)=O)CCN(C(=O)CC2CC=CC2)C2CC12 C(C)(CCC(=O)NCC1C2CN(C(C3CCC3(C)C)=O)CC12)OC C1(CNC(c2cc(C)n(C)n2)=O)CCC(C)(C)CN1C(c1cnc2sccn12)=O C(C(C(=O)N1CCCC1CCOC)C(C)(C)C)NC(CS(=O)(=O)NC)=O c1(C(C)C=O)c(F)cccc1F.c1(CC)ccccc1Cl c1(C(=O)NC2CN(C(C(c3cn(CC)nc3)=O)=O)C3C2C3)cc(F)c(F)cc1F C(C(C(=O)N(CCC(C)NC(=O)CCc1cc[nH]n1)C)NC(C)=O)OC C1(C(=O)NC(C)CCCNC(=O)C(C)n2cncn2)CC2(C1)CC1(CCC1)C2 c1(OCC)cccc2cc(C(=O)NC3CC(OC(C)=O)C3)oc12 c1(C(=O)NC(CNC(C(C)n2ccnc2)=O)CO)cc(S(=O)(=O)N(C)C)cn1C C1(C(=O)NCCC(C)NC(c2cn(CCO)nn2)=O)CCC(=O)N(C)C1 Cc1cc(C(N2CCCC(C)C2CNC(=O)Cc2cc[nH]c2)=O)cnc1C CC1=C(C(=O)N2CC(N(C)C(C3CCC(F)CC3)=O)C2)CCCC1 c1(C(=O)NC(C(C)NC(c2nn[nH]c2Cl)=O)C)ccccc1F Cc1ccc(C)c(OCC(=O)N(C)Cc2ccc(N(C)C)cc2)c1C Cc1ccc2ccccc2c1CN(c1ccncn1)C1CCNC1 c1(C(=O)NC2C(CC(=O)NC3CN(CCC)CC3C)CCC2)cc(C)cc(F)c1 N1(C(CCCC(=O)OC)=O)CC2CC(NC(=O)CC(F)(F)F)C(C2)C1 C1(CNC(N2CCC(C(=O)NC3CC3)CC2)=O)CS(=O)(=O)c2ccccc2O1 C1(O)(CNC(CC(=O)OC)=O)CCCN(C(c2cccc(I)c2Cl)=O)C1 c1(C(C)C)cc(C(=O)NCCOCC(N2CCC(SCC(F)(F)F)C2)=O)n(C)n1 C(=O)(C(C)CC(F)F)NCc1cc(C(=O)NC(c2cccc(C)c2)C)no1 N1(C(c2n(C)ccn2)=O)CCCC1(C)C(N1CC(N2CCNCC2)C1)=O CCC(C)(CC(=O)O)C(=O)Nc1ccccc1CC(=O)OCC c1(C(N(C2CCCN(C(=O)CSCC(F)F)C2)CC)=O)cnncc1O C(C1(C)CCC(C)C1(C)C)=CC(N1CCN(C(C(C)CF)=O)CC1)=O N1(C(CC(C)OC)=O)CCC2(CCC(CNC(c3scnc3C)=O)CC2)CC1 CCC(CC)C(C(=O)N1CC(NC(C2(CN(C)C)CC2)=O)CC1C)OC c1(C(N2CCC=C(C)C2)=O)n[nH]c2c1CN(C(C1CC3CCC(C1)C3)=O)C2 c1(C(N2CC(NC(C(CC)O)=O)C(C)CC2)=O)ccn2c1CSCC2 c1(C(=O)NC2C(NC(c3c(C(C)(C)C)ncs3)=O)C2)cc2n(n1)CCCC2 C1(C(=O)NC2CCN(C(CCC(C)(C)OC)=O)CC2)CCCC2(C1)CC2(F)F Cc1coc(CNC(=O)C=CCN(C(=O)Cc2cn[nH]c2)C)c1 N1(C(C(C(C)(C)O)F)=O)CCC2(CNC(c3csc(Cl)c3Cl)=O)CCCCC12 N1(C(Cc2cn(C)nc2)=O)CCCC12CCN(C(=O)CCP(C)(C)=O)C2 c1(C(N2CC(NC(C(=O)NCCOCCCC)=O)C(C)C2)=O)cc2ccccn2n1 CN1CCC(CCNC(=O)C=CCC2(NC(=O)CSC(F)(F)F)CCC2)C1=O N1(C(CC)=O)CCCC(C(N2CCCCC2CNC(=O)CCCOC(C)C)=O)C1 Cc1coc(CN2CCC(C(=O)NCCCC(=O)N(C)C)C2)c1 C1(C(=O)NCC(CC)NC(=O)Cn2nnc(C)n2)CCCC(=O)C1 Cc1ccc(C(C)C(N2CCCC2CN)=O)s1 N1(c2ccnc(C)n2)CC2CC1CN2C(C1(C(=O)N(C)C)CC1)=O C(=O)(CC(C)COC)NC(COC)C(=O)NCc1cn(C2CC2)cn1 C1(CNC(c2nc(C)oc2C)=O)CC2(CC2)CN1C(c1nccc(Cl)c1F)=O Cn1ccc2ccc(C(=O)NC3CC(CNC(c4cc(F)ccc4Cl)=O)C3)cc12 c1(C(N2CCC(NC(Cn3c(C)nnn3)=O)CC2C)=O)coc2c1C(=O)NCC2 c1(C(=O)NCC(=O)NCCC(=O)NCC(C)C(F)F)cnc(N)cn1 N1(C(C2C(C)SCCC2)=O)CC(C(N2CC3(CC(O)C3)C2)=O)C(C)(C)C1 c1(C(=O)NCC(=C)Br)conc1C(C)NC(=O)C(C)(C)C C(CC(=O)NNc1ccccc1[N+](=O)[O-])c1noc(C)c1Br c1(CC)cscc1NC(=O)CCN(C(c1ccns1)=O)C(C)C c1(C(N(CC(CC)NC(=O)C(N2CCC(C)CC2)=O)C)=O)cnc2c(c1)COC2 CC(C(F)(F)F)NC(C1CCN1C(=O)CN1CCSCC1)=O C1(C(=O)NC2CC(NC(C3(C(=O)NC)CCC3)=O)C23CCC3)CC2(C1)CC(C)C2 CC1CCCC1(C(=O)NCCn1cccnc1=O)NC(=O)CCCn1cccn1 C1(N(C(C(C)C2CC2)=O)C)CN(C(=O)CCC(=O)C2CC2)CC1(C)C C1(NC(CC(CC)O)=O)CCN(C(c2ccccc2O)=O)CC1C C#CCCCC(C)C(=O)NCCn1cnnc1C(=O)NCCCP(C)(C)=O C1(NC(COCC#C)=O)CC(C(=O)Nc2c(C)coc2CC)C12CCC2 C=CC1COCCN1C(c1cc(CNC(C2CCOC2)=O)nn1C)=O N1(C(CCC(C)NC(=O)CCCC(C)(C)C#N)=O)CCCC2(CCOC2)C1 c1(C(=O)NCCC(C)NC(c2ccc(CN(C)C)nc2)=O)cc(C#N)c(F)cc1F C(C)(C1Cc2ccccc21)N1CCC(CC(=O)Nc2ccc(C)c(C)c2)C1 C1(F)(C(=O)NCC(CC)(C)Cl)CCN(C(=O)CCCCC2CC2)CC1 C1(C(N2CCN(C(C3(OC)CCOC3)=O)CC2)=O)OCC2COCCC12 O(NC(=O)CCCC(C)(C)NC(=O)CCc1ccncc1)CC C1(C2(OC)CC2)CCCN1C(C1CC(F)(CO)C1)=O.C(=O)(C(F)n1cccn1)N CN1CCC(C(=O)NCCCCCNC(=O)CSc2nnc(S)s2)C1 C(CC(C)(C)CNC(=O)CCC1CCCC(O)C1)NC(CCCOC)=O CC(C)CC(C(N)=O)NC(C1CC(NC(C2CCO2)=O)C12CCC2)=O CON(CCC(=O)NCC1C2CCCOC12)C(=O)c1ccc(=O)n(C)c1 Cc1cc(C(=O)NCC2CC(O)CN2C(c2cc(C(N)=O)n(C)n2)=O)ccc1Cl O=C1NCc2cc(NC(C3CSCCN3Cc3ccncc3F)=O)ccc21 C1(CNC(c2n(CC#C)ccc2)=O)CCCCCN1C(c1ccc(CO)cc1)=O CC1=NNC(=O)C1CCC(=O)N(C)CC1CCCCN1C(c1ccsc1CO)=O c1(OC)nc(C(=O)NC(C2CCCN2C(=O)CCC2CC2(F)F)C)cc(O)n1 C(=O)(CC1CCc2ccccc21)OCC(CC(F)(F)F)OCC CC(CCCNC(=O)CNC(=O)Cc1ccccc1)NC(c1occc1Cl)=O N1(C(CC2CC(OC)C2)=O)CCCCC1C.C1(CCCO)(CNC=O)CC1 N1(C(C2(C)CC(=C)C2)=O)CCC(C)(CNC(=O)CCOCCN(C)C)CC1 Cc1nc2ncnn2c(N(c2ccccc2)CCNC(=O)COC(F)F)c1C c1(CN(CCN(C(C)C)C(C2CN(CC(F)(F)F)C2)=O)C)c(F)cccc1F C1(C(N2CC(NC(C3(CCC)CCC3)=O)C(F)C2)=O)CC(C)(C)CCO1 CS(=O)c1cccc(C(=O)NCC2CN(C(c3cncc(F)c3Cl)=O)CC2O)c1 N=C1NC(=O)C(CC(=O)NCCN(C2CCCC2)C(C2CCCCC2O)=O)S1 C=C1CCC(CNC(C2(N(C3CCN(C)C3)CC)CCC2)=O)CC1 c1(C(N2CC(N(C)C(C3CCCC(=O)N3C)=O)C(O)C2)=O)cc(O)cc(Cl)c1Cl c1(C(N2CCCC(C(C)NC(CCCSC)=O)C2)=O)cc2c(Cl)cncc2s1 C1(NC(CN(CCOC)C)=O)CC2CCC(C1)N2C(C1SCC=C1C)=O c1(C(=O)NC2CN(C(=O)C(F)(F)c3cncs3)C2)ccn2c1CSCC2 N(C1c2ccccc2CCC1CC)C(N(c1cccc(Br)c1)C)=O c1(CC)ccc(NC(=O)NCCC(=O)N(C)C(c2ccccc2OC)C)cc1 C1(C#N)(C(N2CCN(C(C34CC(CC)(OC3)C4)=O)CC2C)=O)CC2CCC1CC2 c1(CC)ccc(C=CC(=O)NCC2CC(OC)CN2C(c2sccc2SC)=O)o1 C(C(C(=O)NC(c1csc(C)n1)C)NC(=O)C(CO)NC(N)=O)OCC C1(N(C(=O)CC2CC(F)C2)C)CCCN(C(=O)CC2CCCS2(=O)=O)CC1 c1(C(N(CC(C)(C)CNC(=O)CC2CCC2)CC)=O)c(N)sc2c1CCC2 Fc1cc(-n2nc(-c3ccsc3)nc2Cc2ccoc2)cc(F)c1 Cc1cc(C(=O)N(CC(C)NC(=O)CCc2ccccc2)C)n(CC2CC2)n1 CC(C)CC(O)CC(=O)NC(C)C(C(=O)NC(c1ncc[nH]1)C)C(C)C c1(OC)cc(NC(=O)C(C)(C)Cc2cccs2)cc(OC)c1OC(F)F c1(C(C)C)noc2ncc(C(=O)NCCN(C)C(C3CCS(=O)(=O)C3)=O)cc12 c1(OCCC)ccccc1CCC(=O)NC1CC(CN(C)C(C)=O)C1 N1(CC(C)C)N=C(C(=O)c2ccc(CN3CCCCCC3)cc2)NCC1=O n12nccc1CC2.N1(C(=O)OC(C)(C)C)CC(C(=O)OCC(=O)OC(C)(C)C)C1 C1(C(=O)NCCn2ccc(C(C)(C)C)c2)N(C(c2cc(F)c[nH]2)=O)CC1(C)C C1(NC(C(C)OCCC=C)=O)CCCN(C(=O)C2=CCCC2)C1C c1(C(N2CC(CNC(C3C(C(C)C)C3)=O)CC2(C)C)=O)cnn2ccc(O)nc12 c1(NC(C2(CCF)CC2)=O)cc(F)cc(F)c1.n12cc(nn1)-c1cnn(c1)CC2 c1(OC)ccccc1CNC(=O)CC1(OC)CN(C(C2CC(CSC)C2)=O)C1 C1(NC(C(CCC)C)=O)CC2CCC1CN(C(c1cn(C)c(C)n1)=O)C2 c1(C(N2CCCOCC2)=O)cc(-c2ccccc2-n2ccnc2)ccn1 c1(SC)cn(C)nc1C(N1CCC(C)(CNC(C2CNC(=O)N2C)=O)C1)=O C1(CNC(c2c(C)ccnc2)=O)CCN(C(C2CC(=O)C2(C)C)=O)C12CC2 CC1CN(C(C2(C#N)CC2)=O)CCC1NC(c1cc(C(F)(F)F)cs1)=O C1(NC(C(C2(O)CN(C(C(CC)c3ccco3)=O)C2)F)=O)CCCN(C2CC2)C1 N1(Cc2c(F)ccc(C)c2)CCCn2nc(C(=O)Nc3nnc(Br)s3)cc2C1 c1(C(CO)NC(Cn2cc(C3CCC(=O)C3)nn2)=O)ccc(F)c(Br)c1 c1(-c2nnc(CCC(N3CC(C(C)=O)C3)=O)o2)ccc(C(=O)OC)cc1[N+](=O)[O-] Cc1cn(C)nc1CN1CCCC(CCNC(C2CC23CCOC3)=O)C1 C1(C(=O)NCCOCCOCC)CN(C)CCN1C(=O)CC1OCCCO1 C1(C(=O)NC2CC(NC(C(C)NC(C3CCC3)=O)=O)C2)CCSCC1 C(c1ccc(-c2cccs2)cc1)=CC(=O)N(C1CCN(CC(=O)O)C1=O)CC C1(NC(C=CC(CC)C)=O)CC(NC(c2cc(CCOC)on2)=O)CC1O C1(C(NCBr)=O)CC(F)CN1C(=O)CC1CC1F C1(CNC(C2(C(C)C)CN(C(C3(C)CCN(C)C3)=O)C2)=O)CC2CCCC2C1 c1(CC(=O)NCCC(C)N(C(C)=O)C)nc(C)sc1Cl N1(C(CCSCC)=O)CCN(C(=O)C(C(C)C)N2CCC2)CC(C)(F)C1.CC(C)C c1(C(N2CCC3(NC(c4n(CC)ncc4)=O)C(C2)C3)=O)ccc2nc(C)ccc2c1 Cn1ccnc1-c1cn(CCCC(=O)N2CCCC2C2(CO)CC2)nn1 c1(C(N(CC(CNC(C2C(C=C)C2)=O)O)C)=O)ccnc(O)c1Br N1(C(CCN(C)CC)=O)CCCC(NC(=O)C(N2CCSCC2)C)C1 C(=O)(CCCC(C)(C)C)N1CCC(N(C(Cc2n(C(C)C)ncc2)=O)C)CC1 c1(C(N2CCC(NC(=O)Nc3ccc(SC)cc3)C2)=O)ccc(Br)cc1[N+](=O)[O-] c1(C(=O)NC2CCCCN(C(c3ccc4c(c3)CC4)=O)C2)cccc([N+](=O)[O-])c1 c1(C(C(=O)OC)NCc2ccc(Br)cc2)cccc(Br)c1 c1(NC)cnccc1C(=O)NCc1occc1C(=O)NC1(C2CCCCO2)CC1 N1(C(Cc2ccc(C)cc2)=O)CCC(CNC(C2CCCO2)=O)C12CC2 N1(C(COCC)=O)C2CCCC1CN(C(C1CCC(=O)NC1)=O)C2 S(=O)(=O)(c1[nH]c(=NC2CC3C=CC2C3)ccc1Br)NCCOC1(C)CCCC1 S(=O)(=O)(c1ccc2nc(N3CCC(C)(CCO)C3)sc2c1)NC1(C)CCC1 N1(CC(=O)NCC(C)N(C(=O)Cn2ccnn2)C)CSCCSC1 C1(CNC(C(C(=C)Cl)(C)C)=O)CCN(C(c2cnn3ncccc23)=O)CC1(F)F Cc1ncccc1CC(N1CCC(CC(C)NC(=O)CCNC(N)=O)CC1)=O C1(O)(C(C)NC(C2(CF)CC(F)(F)C2)=O)CCN(C(=O)Cc2ccccc2)CC1 CCC(C)C(C(=O)NOCC#CC(F)(F)F)N(C(=O)C(O)CC(F)(F)F)C CCC(C)(CC)C(=O)N(C)CC1CN(C(=O)CCCn2c(C)csc2=O)C1 N1(C(C(c2cccc(Cl)c2)N(C)C)=O)CCCC(c2ccc(F)cc2)CC1 c1(C(=O)Nc2c(C(=O)NCCOC)cccc2)ccc2nc(O)oc2c1 C(=O)(C(C(C)(C)C)NC(=O)CCc1cnccn1)NC(C)CC1(O)CCC1 C(CCC(O)C(=O)NC(c1csnn1)C)NC(c1c(C)snc1)=O C=CC1(CC(=O)NC2CCCC(F)C2)CN(C(C2(C#N)CC(=O)C2)=O)C1 C(c1cccc(F)c1)=CC(=O)NC(C1CCCN(C(=O)Cc2nc[nH]n2)C1)C CC(=O)CCN=C(NCc1ccnc(-n2ccnc2)c1)N(C)CCC1CCCO1 C1(NC(C(=C)C(F)(F)F)=O)CN(C(c2ccc(C)nc2F)=O)Cc2nccn2C1 Cn1ncc2c(O)nc(CCC(=O)NC3CN(C(=O)CC4CC4)CC3(C)C)nc12 N1(C(c2nc(C)oc2)C(=O)NC(c2ccccc2)C)CC2CCCCC2C1C c1(C(=O)NC2(C)CC(NC(C3N(C)CC(O)C3)=O)C2)cc2cccnn2c1 C1(C(N(C(C)C)CC)=O)CN(C(C2CC(=O)CC(=O)N2)=O)CC1(C)C C1(CNC(C(CSC)OC)=O)CN(C(=O)C(C)CC(F)(F)F)CC12CCC2 N1(C(c2n(CCOC)ncc2)=O)CC(NC(c2ccc(F)c(F)c2)=O)C2(CC2)C1 O(NC(=O)C(C)(c1ccccc1Cl)N1CCOCC1)C(C)(C)C c1(CCC)cc(C(=O)NC(C)CCN(C(=O)COC2CCC2)C)n(C)n1 CC1CN(C(c2ccco2)=O)CCC1NC(c1ncn(C(C)(C)C)n1)=O C1(O)(CNC(C2(OCC)CCC2)=O)CC(NC(C2CCC(=O)C2)=O)C1 N1(C(C(CCCCC)O)=O)CC2CCCN(C(=O)CCc3ccon3)C2C1 C(=O)(CC(C)C(C)(C)C)NCCC(=C)CNC(=O)CN(c1ccncc1)C N1(C(c2c(SC)cccn2)=O)CCN(C(c2[nH]nc3ncccc23)=O)CC(O)C1 c1(C(N2CCOCC2CCO)=O)nccn2ccnc12 N1(C(c2cccc(-c3ccc[nH]3)c2)=O)CCOc2cc(Cl)ccc2C1 c1(OC)ccc(C(N2CCCC(CC(=O)NCC3COC(C)(C)C3)C2)=O)nc1 c1(CCC2CC(C)N(C(=O)CN3C(=O)CNC3=O)C2)ccc(F)cc1C(=O)N(C)C c1(OC)cc(CNCC2COCCN2C(c2cccc(O)c2Br)=O)cc(O)c1OC N1(C(C(c2cccc(Cl)c2)(C)C)=O)CCOC(CNC(C2CCC2CF)=O)C1 CCC(C)(COC)C(=O)N1CC=CC(NC(C2CC3(CSC3)C2)=O)C1 c1(C(=O)NCC23CC2CN(C(=O)CC(F)(F)F)C3)cccc2ccsc12 C(=O)(C(C)CCCC(C)C)N1CCN(C(C(COC)N(C)C)=O)C(CO)C1 CC1CCOC1C(=O)NCC1C(C(=O)NC2(N(C)CC3CC3)CC2)C1(F)F c1(CC)cccc(C(N2CCCC(N(C(=O)CP(C)(C)=O)CC)C2)=O)c1N N1(C(C(C)C#N)=O)CCC2(CCCN(C(=O)CNS(=O)(=O)c3cccnc3)C2)C1 CC#CC1CCN(C(C2OCCC2NC(=O)CC(=O)N(C)C)=O)C1 CS(=O)(=O)c1cccc(C(=O)OC(CCN(CCC#N)CCC#N)=O)c1 N1(C(C=CC=CCC)=O)CC2CCC(C1)N(C(c1cnn(C)c1Cl)=O)C2 C1(NC(CN(C(c2cnccn2)=O)C2CC2)=O)(CN(C2C(C)CC2)C)CC(C)(C)C1 C(=O)(C(CCC)C(C)C)NC(CCC=C)C(=O)NCCn1ccc(=O)cc1 C1(CCOC)(C(=O)Nc2ccc(C(F)(F)F)[nH]2)CCN(C(=O)C=C2CCC2)CC1 CC1C(NC(=O)Cc2cccc(Cl)c2)CC2CCC1N2C(C1CCC1)=O c1(CC(=O)NC(C(C)NC(=O)C=Cc2ncc[nH]2)(C)C)ccc([N+](=O)[O-])cc1 C(=O)(CCS(C)(=O)=O)NCC1CCCC(NC(C2CC(OC)C2)=O)C1 c1(C(N(CCOC)CCNC(=O)C(C2CCOCC2)F)=O)ccc(C(C)O)cc1 Cc1nn(C)cc1NC(=O)CC(CC1CC1)NC(c1ccc(Cl)cc1)=O c1(C(=O)NC2(CNC(c3ccc(SC)[nH]3)=O)CC2)cccn2c(C)nnc12 Cc1cc(C(N2CCC2CNC(=O)C(N2CCCC(C)C2)=O)=O)cnc1C(F)F C(=O)(C(C)C(O)CC)NCCN(CCC)C(c1cccn(C)c1=O)=O Cc1cnc(C(=O)NC2CC2CNC(=O)Cn2nnnc2C)cc1C N1(C(CC(C=C)(C)C)=O)C2CC=C(C(=O)N3CCn4nncc4C3)C1CC2 c1(CCN(C2CCCC(C)(C)C2)C(C)Cc2ccccc2OC(F)F)ccc(F)c(Cl)c1 CCCCCCC(CC)C(=O)NCC1C=CCN1C(=O)COc1ccc(F)cc1 CCCCCCCCC(=O)NCCCN(C(C1CC1CCC)=O)C(C)C c1(-c2nc(-c3nccc(C)c3C(F)(F)F)on2)cc(F)c(F)c(F)c1 C1(CC(=O)NC(CNC(c2c(CCC)[nH]cc2)=O)CCOC)CCCC(C)(C)O1 Cc1ccc(C(N2CC(NC(=O)C(C)(C)C3CCOCC3)C2)=O)o1 c1(CC)ccc(F)cc1C(=O)NCC(C)CNC(C1CC1C(C)C)=O C(=O)(C(C)(CO)NC(c1nc(Cl)oc1C)=O)N(CC=C)CCOC C(c1ccc(OC(F)F)cc1C(=O)O)=CC(N1CCC(C2(C)N=N2)CC1)=O N1(C(c2nc(C(C)OC)oc2)=O)CCN(C(=O)CC2(C)CC(F)(F)C2)CC(O)C1 c1(C(N2CCCCCC(NC(C(C(C)C)C)=O)C2)=O)ccc2c(c1)CN(C)C2 c1(C(=O)NC2CCN(C(CN(C)CC)=O)CC2C)cc(Cl)c(F)cc1N c1(C(N2CCC(C(C)NC(c3cccnc3)=O)C2)=O)nc2n(c1Cl)CCCC2 c1(OC)ncc(C(=O)NCC#N)cc1C1=CCC(C(F)(F)F)CC1 C1(Nc2c(Br)cc(Cn3ccnc3)cc2)CC2(CCCNC2)C1 N1(C(C(CCCC)NC(c2coc(OCC)n2)=O)=O)C2CCC1CN(C)C2 C(C1Cc2ccccc21)NC(C(C(C)C)CNC(=O)Cc1cccnc1F)=O C(=O)(CCOC1CN(C(=O)CNC(N(CCC)C)=O)C1)OC Cc1coc(Cl)c1C(N1CC(NC(=O)CC2CNC(=O)C2)C(C)C1)=O c1(C(C(=O)NCC(F)F)NC(c2cc(Br)ccn2)C)ccc(O)cc1 CC1CCC(NC(C2(c3ccnc(Cl)c3)CC2)=O)CN1C(=O)CC1CC1(C)C N1(C(C2=CC(C)(C)C2)=O)CCC(O)C(C(N2CCn3nccc32)=O)C1 N1(CCC(=O)NC(CNC(=O)CCc2cnc(O)[nH]2)CO)CCS(=O)CC1 c1(N2CC(C(F)(F)F)(OC)C(F)C2)nc(=NCC(C)C(C)(C)C)[nH]c2cccnc12 c1(C(=O)NC2C(C(=O)NCc3c(OC)nn(C)c3)COCC2)ncc(N)cc1C C1(NC(c2ncc(C)nc2)=O)CN(C(=O)COC2CCCC2)CC2(CC2)C1 N1(C(Cn2cnc(C#N)n2)=O)CC2CCCC(CNC(=O)COC3CCC3)C2C1 C(C)(C)(C(=O)NC1CC(CCNC(=O)C(F)(F)C2CCOCC2)C1)OC Cc1cc(C=CC(=O)N(C2CCCCN(C(c3nnsc3C)=O)C2)C)c[nH]c1=N C12(NC(COCCC=C)=O)CC(CN1C(=O)CCC(C)O)C2 Cc1ccc(CCC(=O)NCC=CCNC(=O)CCC=CBr)cc1C N1(C(C2(COCC)CC2)=O)CC(NC(=O)CC2CCCO2)C1 c1(C(c2nnnn2C)NC(CC)C2CC2)c(F)cc(Cl)cc1F C1(O)(CC(C2CCC3(CCC3)C2)=O)CCCN(C(C2(F)CCOC2)=O)C1.C N1(C(C2(C)CC(C)C2)=O)CCN(C2CN(C(=O)C(c3cccnc3)C)C2)CC1 C1(NC(c2c(CC)onc2C)=O)CCN(C(c2cc(C)sc2C)=O)CC1C c1(CN2CCOCC2)ccc(-c2ccc(C(=O)NC3(C)CCCC3)nc2)cc1 c1(C(=O)NCC2CC3CC3N2C(C2CC23CCSCC3)=O)cc(Cl)c([N+](=O)[O-])[nH]1 C1(C(=O)NC(C2CN(C(=O)CC3CC(F)C3)C2)C)CCCC1(F)F C1(N(C(C(C)CN(C(=O)CCn2cccc2)C)=O)C)CNC(=O)C12CC2 c1(C(N(C)CC2N(C(C(CC)OCC)=O)CCC2)=O)cccc(C2(O)COC2)c1 c1(C(N(CCC)CCNC(=O)C#CC2(CC)CC2)=O)cc(Cl)c(F)cc1Cl C(CCN=c1[nH]c(=NCc2ccc(C(N)=O)s2)[nH]c2c1COCC2)=CC c1(C(N(CC(C)CNC(c2cnc(C(C)O)s2)=O)C)=O)cnc2c(Cl)cccn12 CCCCCCOC(C)C(=O)N(C)CCOC.C(=O)(CC(C)N(C)C)N(CCCCN)C c1(C(=O)OCC)cc(=NC(=O)c2n[nH]cc2C2CC2)[nH]c(Cl)n1 c1(C(C)=O)ccc(=NCc2nc(C)c(-c3ccc(F)cc3)o2)[nH]c1Br C1(NC(Cc2cnc(C)s2)=O)CC2CC1N(C(=O)CN1CC(C)C1)C2 c1(C(=O)NC2C(NC(COC(CC)C)=O)C2)ccc2c(c1)CCC(=O)N2 CC1CCC(CNC(c2cnc(O)c(F)c2)=O)CN1C(c1cc2c(s1)CCC2)=O C1(CC(=O)N(CC(N2CC(CC(C)NSCC#N)C2)=O)C)CC=CCC1 C(N=c1[nH]cc2ncnc-2[nH]1)C1(NC(=O)Cc2cnnn2C)C(C)CCCC1 CC1CN(C(c2cc(CO)n(C)n2)=O)CCC1NC(C1CC(n2cnnc2)C1)=O N1(C(c2ccc(C#N)[nH]2)=O)CCC2(CNC(=O)CCCN=[N+]=[N-])CCCCC12 C(=O)(C(O)C(F)F)N(CCOCCCN(C(c1c(C)ncs1)=O)C)C c1(CC)[nH]nc(Cl)c1C(=O)NCC(C(C)(C)C)NC(=O)CCc1cncs1 c1(C(N2CC(C)C(NC(=O)COC3CC3)CC2)=O)cc2scc(Br)c2[nH]1 N1(C(CN(c2ccc(Cl)cn2)C)=O)CC(NC(c2ccc(N)cn2)=O)C(C)(C)C1 CN=c1cc(C(=O)NC2(CNC(=O)C(C)C3CCOC3)CCCCC2)cc[nH]1 C1(C(=O)NCC(C)(C2CC2)NC(c2coc(Cl)n2)=O)Cc2ccccc2S1 C#CCCCCCCC(=O)N(CC(=O)NC(C1CCOC1)C)C(C)C C(N=c1[nH]cncc1I)C1(CCN(C(=O)CCc2cccnc2Cl)C2CC2)CC1 c1(C(N2C(C3(C(=O)NCc4c(CC)c[nH]n4)CC3)CCC2)=O)cncc(C)n1 O=C(CCS(=O)(=O)C1CCCC1)NC1CCN(C(C2OCCCO2)=O)CC1F c1(C(=O)NC(CNC(c2c(Cl)cc(C)nc2)=O)C2CC2)cnc2c(c1)CCOC2 CCC(CCC(=O)N(C)Cc1cncn1C)NC(=O)C(O)CC1CCCC1 C(CCCCCC(=O)NCC1CCN(C(=O)C2=CC(C)C2)CC1)SC C1(C(=O)NC(C(=O)NCc2nc(CC)oc2)C2CC2)CCC(F)CC1 CCC(CC(=O)N1CCN(CCNC(=O)C=C(C)c2ccsc2)CC1)C(F)F c1(NC(CCC(CC)CC)=O)c(C)c(C)nc2ncnn12 c1(C(C(=O)NCCC(C)NC(=O)C(N2CCSCC2)C)(F)F)ccc(F)cc1 c1(C(N2CCC(NC(COC)=O)C(C)C2)=O)cc2c(s1)-c1ccccc1OC2 C1(C(N2CCCCC(NC(C3C4C5CCC(C5)C34)=O)C2)=O)CC2(CCOC2)C1 N1(C(c2nscc2Br)=O)CCCC2(C1)CN(C(C1CC1(F)F)=O)CCO2 C1(C(N2CC(CCC=C)(C(=O)NC3(C4CCC4)CC3)C2)=O)CC1C1CCCC1 c1(CCC(=O)NC2(CO)CN(C(c3csc(O)n3)=O)C2)cc(F)ccc1F Cn1ncc2ncnc(N3CCN(C)CC3)c12.c1(C)ccc(C(=O)O)[nH]1 N1(C(C2N(C)CC(O)C2)=O)CCC2CCCC12C(N1CCC1CC1CC1)=O N1(C(c2cc(CC)sn2)=O)CC(CNC(c2ncccc2C)=O)C(F)(F)C1 c1(C(=O)NCCCCN(C)C(C2CN(c3nncs3)C2)=O)cnn(CC2CC2)c1 N1(CC(=O)Nc2c(CC)cccc2)CCCN(C)C(=O)C1 O=[N+]([O-])c1ccnn1SC12CCCCC1C2 C1(O)(CCNC(c2ncn(CC)n2)=O)CCN(C(C2(OC)CCCCC2)=O)CC1 N1(C(C2(CCC)CC2)=O)CCCC1CNC(C1CC1c1ccncc1)=O C1(NC(=O)Cc2cnc[nH]2)CCN(C(=O)Cn2cnnc2O)CC1CO c1(C(=O)OCC(c2ccc(OC)cc2)OC)cc(O)nc2c(F)cc(C)cc12 c1(CC)cc(C)ccc1C(=O)NCCC(C)(C)NC(c1csc(CC)n1)=O C(=O)(CCCCC(=O)NC)NCC1CCC(F)(CNC(C=C(CC)C)=O)C1 C12(NC(CC(CCC)C)=O)CC(C)(C1)OC21CN(C(=O)CCC2CC2)C1 c1(C(N2CCCCC(NC(CC(CCC)C)=O)C2)=O)c(F)cc(C)cc1Cl N1(CC(=O)OCC(C)C)CCN(C(C2(F)CC2C(=O)NC(C)C)=O)CC1 N1(C(c2c(C)oc(Cl)n2)=O)CCN(C(c2ccccc2F)=O)CC1CC(C)(C)C CCCCC(C)C(=O)N(CC(C)NC(=O)CC1CCOC(C)(C)C1)C C(=O)(CC(C)C(=O)N1CC=C(C(=O)N2CCC(OC(F)F)C2)C1)OC C1(C(N2CCCC(n3cc(C4CC4)nn3)C2)C(=O)NCCC)CCCC(C)(C)C1 C1(NC(C=Cc2n(C)ncc2)=O)CC(F)CN(C(=O)CSc2cccs2)C1 C1(CC(=O)NC2CCN(C(CCOCC(C)C)=O)CC2)CC(C)(C)CCO1 S(=O)(=O)(c1cccs1)NCC(N1CCC(CC=C)(NC(=O)C=CS(C)=O)C1)=O c1(OC)ccc(C(N2CC=CC2C(=O)NC(C)CCC2CC2)=O)s1 C1(C(=O)NCC(Cl)Cl)C2CC(O)C(C2)N1C(=O)C=Cc1cccnc1 CC(CC(=O)N1CCC(CO)(NC(C2CCCCC2OCCO)=O)CC1)C(F)F C1(C(=O)NCCSCCC=C)CCCN(C(=O)CC2CC2CC)C1.C(C)(=O)O c1(C(=O)NCCC2CCN(C(c3c(C)noc3)=O)CC2)cc2n(n1)CCCC2O C1(NC(C(N(C)C(c2cccc(CO)c2)=O)C2CC2)=O)CC12CCCCC2 C1(C(c2nnnn2C2CCOCC2)NCCc2ncoc2)CC2(C1)OCCO2 N1(C(=O)NC2(C(=O)NCC)CCC2)CCSCC1c1ccc(OC)cc1 c1(NC(N2CC(C)C(Cc3ccccc3)CC2)=O)ncc2c(n1)CCC2 N1(C(C(C)OC2CCCCCC2)=O)CC(NC(=O)Cn2cccn2)C(C)C1 C(C)(CC(C)CC)OC1CN(C(C)=O)C1.C1CC(=O)N(C)CCOCC(=O)N1 C1(C(N2CCC(CCC(=O)NCC3CC(OCC)C3)C2)=O)CCN(C)C1=O c1(CNC(C(C(C)NC(c2c(CC)ocn2)=O)C)=O)ncc(C)cc1C C1(CNC(C(C)CF)=O)CCN(C(c2cn3ccnc3s2)=O)C12CC2 c1(NC(CN(C(c2cn(C)nc2OC)=O)CC)=O)ccc(C)cc1F C1(C(C)C)CN(C(=O)C(N2CCOCC2)C)CC1C(=O)NCC1(C#N)CCC1 C=CC1OCCCC1C(=O)N(CC(C)O)CCNC(c1ccc(C#N)o1)=O C1(NC(c2cc(C)oc2C)=O)CC2CN(C(=O)CC3CCC(=O)C3)CC2C1 c1(C(N2CC(OC)C(NC(=O)C(F)C3CC3)C2)=O)cc(Cl)cc(Cl)c1O CCC(CC(F)(F)F)C(=O)NC1CC(F)CN(C(c2ccc(C)o2)=O)C1 CC1CC(N(C)C(C2(NC(c3cnn(C)c3Cl)=O)CC2)=O)CC(C)C1 C1(CC#C)CCCN1C(=O)COC(C)(C)CNC(C1(COC)CC1)=O C(=O)(CCP(C)(C)=O)N(CCCNC(=O)C(C)CC1CCCC1)CC CS(=O)(=O)CCCC(=O)N1CC2(CCCC2NC(C2CC2C2CC2)=O)C1 N1(C(CC)=O)CC(C2CN(C(=O)CC3(C)CCCC3)C2)C1 C(CS(=O)(=O)CC(=O)N1CCN(C(c2cccnc2OC)=O)C(C(C)C)C1)OC C1(C(C(C)N)=O)CCCCC1.n1(C2CN(C(=O)CC(C)F)C2)cc(C(C)C)nn1 C1(NC(C=CCOC)=O)CCN(C(c2c[nH]cc2C(C)(C)C)=O)CC(C)(C)C1 N1(C(C2(SCC)CC2)=O)CCC(O)(CC(NC(=O)C=C(C)c2ccco2)CC)C1 c1(NC(C2N(C(CC=CC)=O)CCC(C)C2)=O)cnc(C)c(C#N)c1 c1(C(=O)NCC23C(CN(C(CCCCC=C)=O)C2)CC3)cccc([N+](=O)[O-])c1C C1(C(N(C2CN(C)C2)C)=O)CCCN1C(C1CC1F)=O C(=O)(C(O)CCC(C)C)NC(C(=O)N(CC)CC)CC1CCCC1 C(=O)(CCP(C)(C)=O)N1C(CNC(CC2(C(=O)OC)CCOCC2)=O)CCC1 CCC(C)C(C(=O)N(C1CN(C(=O)CN2C(=O)CNC2=O)C1)C)NC(C)=O C12(CNC(C(C)(C)CCOC)c3n(CC)nnn3)CC1COC21CCC1 c1(NCc2ncn(C)c2)cc(N2CC3C(C(N)=O)C3C2)nc(C(F)(F)F)n1 N1(C(CSCC(=O)OC)=O)CCCC1C1CCCN1C(=O)C(C)n1cccn1 N1(C(C2(C)C(C)CCC2)=O)CC2CCC(N(C(=O)C(F)=CC3CC3)C)C2C1 N1(C(CCC(C)=O)=O)C(CNC(c2cc(Cl)cc(Cl)n2)=O)CC2COCC12 c1(CC)ccc(CC(N2CC3CC3(NC(c3coc(C(=O)OC)n3)=O)C2)=O)cc1 c1(OCCC(=O)NCC2CCN(C(C3CCC(=O)N3)=O)C2)ccc(Br)cc1 C(CC(=O)NCC1COCC(=O)N1C)(C(F)(F)F)NC(c1c[nH]c(=NC)o1)=O Cc1ccccc1C1(CO)CCCCC1.n1(C)cc(CC(C)C2CC2)nn1 C1(C(=O)NCc2[nH]nc(COC)n2)CC(C)(C)CCN1C(c1ccnnc1C)=O C(C(=O)NC1(CNC(c2nncs2)=O)CCC1)(C(C)C)NC(C)=O N1(C(Cn2cc(C(C)=O)nn2)=O)CC2OCCN(C(=O)Cc3csc(C)n3)C2C1 c1(CC(=O)NCCn2cc(C(N(C3(CO)CC3)C)=O)nc2)ccnnc1O C1(C(C)C)CCC(C(=O)NCC2(O)CC(O)C2)N1C(=O)C=CC1(C)COC1 C1(C(=O)NCC(CN(C(c2ccc(CC)cn2)=O)C)O)CCC2(CC1)CC(O)C2 N1(C(=O)Nc2ccc(Cl)nn2)CC2CC(C1)CN(C(C1(Br)CCC1)=O)C2 c1(CN(C2CCC(O)C2)CCO)noc(-c2ccccc2)c1Cl Cc1cccc(C(O)C(=O)N(C)CC2CN(C(=O)CC3(O)CCOCC3)C2)c1F c1(C(N2CCCC(CCNC(=O)Cn3cnnn3)C2)=O)cc2c(s1)CCC2=O c1(NC(C2N(C(c3c(OC)scc3)=O)C(C)CC2)=O)ccc2ccoc2c1 N1(c2cc(CC)ncn2)CCC2(CC1)CC(NC(=O)Cn1nnc(=O)[nH]1)CCO2 C1(NC(c2cnn(CC)n2)=O)CC2(C1)CC2NC(c1cnc(SC)[nH]1)=O N#Cc1cc(C(=O)NC2CC(NC(C3Cc4nnsc4S3)=O)C2)c(F)cc1F N1(C(COC)=O)CC(NC(=O)COCCOC2CC=CC2)C(C)(C)C1 C1(CNC(c2cnc(O)s2)=O)CN(C(=O)CCn2cccc2)CC1(F)F C1(C)(C(=O)NCCN(C(c2occc2C)=O)CC)CCCN1C(C)=O N1(C(CC(=O)NCC#C)=O)CC2CCC1C(CNC(=O)C(CC(C)C)N(C)C)C2 c1(NCC2CC(C)C2)ccc(S(=O)(=O)NCC2(C)CCCCO2)cc1Br C1(C(=O)NC(CCCCNC(CCC)=O)C)C2Cc3ccccc3C12 C1(CC)CN(C(=O)C(=Cc2cn[nH]c2)C)CCC1CNC(c1cc(C#N)cn1C)=O C(CN=c1cc(NCc2ccc3c(c2)OCO3)nc(C)[nH]1)C1CCC(OC)C1 C=C(Cl)CC(C(=O)NCC1CN(C(N)=O)C1)NC(=O)C1=CCCC1 C=CCC(C(=O)N1CCC(C(F)C(=O)NCc2ccn(C3CC3)n2)C1)C(C)C C12(C(=O)NCCOCCNC(c3cc(-c4ccncc4)on3)=O)CCOCC1C2 c1(C(=O)NC(c2ccc(C)cc2)C(O)C2CC2)ccc(C)c([N+](=O)[O-])c1 C(=O)(C#CC1(C)CCCO1)NCC(C)(C)OCCNC(c1ccc(C)c(C)c1)=O Cc1cccc(F)c1CC(N1CC(NC(C2(O)CC2)=O)CC(O)C1)=O Cc1ccnc2ccc(C(=O)NC3CN(C(C4CCCNS4(=O)=O)=O)C3)cc12 c1(C(=O)NCC(c2ccc(C(F)(F)F)cc2)NC(C)=O)cc(C)c(F)cn1 C1(OC)CCC(C(N2CCC(C(=O)NCCC3(C)CC3)C2)=O)C1 C12(C(=O)NC3CN(C(C=COCC)=O)CC(C)C3)CCCC(C)(C1)OC2 CC1(NC(c2cnncc2O)=O)CCN(C(C2CCC2C(F)(F)F)=O)C1 C(=O)(CCCCC(C)(C)C)NC(CCNC(c1cc(C)c(F)cn1)=O)C C1(C(N2C(C(N(CC(C)SC)C)=O)C=CC2)=O)CCC(C)(C)C1 C(C#Cc1cn(C2CCOCC2)nn1)NC(CC(C)Cc1cccc(F)c1)=O N1(C(C2N(CC)CC2)=O)CCN(C(c2coc(CSC)c2)=O)C(CF)C1 O=C(CC1CCCc2ccccc21)NC1CC12CCN(C(c1csnn1)=O)CC2 C=CC(C)(CC)C(=O)NC1CCC(CNC(=O)C(C)(C)CCC)CC1 C1(CC(=O)NCC(F)F)CCN(Cc2cncnc2)CC1 CCCC(CCCNC(C1(SC)CC(O)C1)=O)NC(=O)C(N)=O N1(C(S(c2c(C)cccc2)(=O)=O)=O)CCCCCC(S(C)(=O)=O)C1 Cc1cccc(C(CNC(C2(N(C)C)CC2)=O)NC(c2cnc(O)o2)=O)c1 c1(C(N2C(C(=O)Nc3cnn(C(F)(F)F)c3)CCC2)=O)ccc(Br)nc1[N+](=O)[O-] c1(CCNC(CN(C)C)=O)ocnc1CNC(=O)CC1CCC2CC12 C1(NC(COCCCC)=O)CN(C(c2cscc2Cl)=O)CC1N=[N+]=[N-] N1(C(CC2(NC(C3CC34CC4)=O)CC2)=O)CCC2(CC2)C1 N1(CC)CCOCC1C(=O)NCCC1CCN(C(=O)CSc2nccn2C)C1 C=CCC(C)(C)CC(=O)N1CC(CN(C(=O)CC(=O)OC(C)(C)C)C)C2(CC2)C1 c1(C(N2CC(C)N(C(C3CCC(F)(F)C3)=O)CCC2)=O)cc2cnc(Cl)cc2s1 Cc1cccc2c1c(CN1CC(C(=O)NCc3cccnn3)C1)cn2C C1(NC(CC(C=C)CCC)=O)CCC2(CC1)CN(C(C1CCC1)=O)CCO2 C1(C(=O)NCC(C)CN(C)C(c2ccccc2SC(F)F)=O)CCCCN1C CC(C)(CC(=O)NC1COC2(C1)CN(C(=O)CSCCC#N)C2)C(F)(F)F c1(C(N2CC(NC(CC=CCC)=O)C(O)C2)=O)ccc(C)cc1C1CC1 Cc1nnc2n1C(C(=O)NC(CNC(=O)Cc1cncn1C1CC1)C1CC1)CC2 N1(c2nnc(C)s2)CC2C(CN(C(=O)CC3CC34CC4)Cc3ccccc3)C2C1 C1(C(=O)NC(CNC(CCN(C)CC)=O)C2CCC2)CC12CC(C)(C)C2 C1(CC=C(C)C)CN(C(=O)COC(=O)CO)CCC1NC(=O)CCC(C)C C(=O)(CC(C)(C)C)NCCOC(C1C(NC(CNC(=O)OC)=O)CCC1)=O N1(C(c2nccc(C)c2)=O)CCC2(CC2NC(C2CN(C)C2)=O)C1 c1(OC)nccc(C)c1NC(C1CCCCCN(C(C2CC(C)(C)CO2)=O)C1)=O N1(C(C2(F)CCCCC2)=O)CC2(CCCCN2C(=O)C(C2CCOCC2)O)C1 c1(N(CCCC2(C)C(CCCCC3C(C)C3)C(=O)N2)C)nc(C(F)F)nc(=N)[nH]1 C=Cc1cc(C(N2CCN(C(=O)CC3CC=CCC3)C(CO)C2)=O)cc(F)c1 CC(C)CC(O)C(=O)NC1CC(C)(CNC(c2cc(C3CC3)[nH]c2C2CC2)=O)C1 c1(C(C)NC(CN(CC(C)C)C(=O)C=CCO)=O)ccncn1 c1(C(=O)NCC(C)CN(C)C(C2(CF)CC2)=O)cccc(Br)c1Cl c1(C(=O)NCC2CN(C(c3cccc(=O)o3)=O)C3CC23)cnc2n1CCS2 C1(C(=O)NCC2C(NC(c3cc(C)ncc3)=O)C2)CN2CCN1C(C)C2 C(=O)(C(C)C(C)NC(c1cccc(NC)c1)=O)NC(CCC)C1CCC1 CC(C)C(C(=O)N1CCCC1CC(=O)NCCC(C)(C)C1CC1)n1cccc1 N1(C(=O)CCc2cncnc2)CCC2(CC1)CN(c1ccnc(Br)n1)C2 c1(CNC(=NCCC)NC2CCC(C)(C)CC2)nn(C)c(C)c1S(N)(=O)=O C=CC(C)CC(=O)NCC1CCC1NC(=O)C(C)(C)Cc1cnn[nH]1 n1(CC(=O)NC(C2CCN(C(CN(CCC)C)=O)CC2)(C)C)cc([N+](=O)[O-])cn1 N1(C(C(C)n2ccnc2)=O)CCC(c2cn(-c3ncc(Br)cn3)nn2)CC1 N1(C(N(CCC)OC)=O)CCC2CCN(C(=O)CC(=O)OC)CC12 O=C(C1CCCn2nc(C)nc21)Nc1cccc(NC(c2sccc2Cl)=O)c1 C1(NC(c2ccc3oc(O)nc3c2)=O)CC2(CCC(NC(C3CC3Cl)=O)CC2)C1 N1(C(C2(N)CCC2)=O)CCCCC1C(c1cn(C2(C(N3CCCC3)=O)CC2)nn1)O N1(C(C(C)C)=O)CCC(C)C1CNC(C12CCC(CC1)C2)=O N1(C(C(S(C)(=O)=O)C2CC2)=O)CCC2(C1)CN(C(C1CC(=O)C1)=O)C2 CCC1=NOC(CC(N2CCC(C(=O)NCc3csc(C)c3C)C2)=O)C1 c1(NC(=O)NC2CCN(CCCC)CC2)cnc2[nH]c(C)nc2c1 c1(CNC2CN(C(n3ccc(CC)n3)=O)CC2(F)F)ccc2ncsc2c1 C1(NC(c2c(C)nc[nH]2)=O)CN(C(=O)CCCCCc2cccs2)CC1(C)C c1(C(=O)NCC2CCCN2C(=O)CC2CCCOCC2)nsc2ccccc12 N1(C(c2cc(C)nc(O)c2)=O)CC(CO)C2(C1)CN(C(c1csc(Cl)n1)=O)C2 CC1COc2c(C(c3ccccc3)Nc3nc4cc(Br)cnc4[nH]3)cccc21 CC1=NS(=O)(=O)N(C)C=C1C(=O)OCc1nnc(C2CCCCC2)s1 C1(CC(N2CCCC(CNC(C=Cc3ccn(C)c3)=O)C2)=O)CCC(=O)NC1=O N1(C(c2cn(C)nc2Br)=O)CC2CC(C1)N(C(C1COCC(C)(C)O1)=O)C2 C(C(C(C)C(C)C)NC(=O)CSc1n[nH]c(=N)s1)NC(CCCOC(C)C)=O C(=O)(C1=NN(C)C(=O)CC1)N1CC2C(NC(c3ccc(C)c(C)c3)=O)CC(C2)C1 C1(C(C)C)CN(CC2CC2C)CCN1C(=O)CC=Cc1ccccc1OC c1(C(=O)OC)cc(C(=O)N(C(C)CCNC(C2(C)CCCO2)=O)C)[nH]n1 C12(NC(c3cc(C)oc3C)=O)CCC(C1)N(C(=O)CC1NC(=O)NC1=O)C2 c1(C(=O)NC2CCC(N(C(=O)Cc3ccco3)C)C2)c(N)cc(F)cc1F c1(CC)ccc(C)cc1.C(=O)(NNC(=O)SC(F)F)OCC C1(C#N)(C(N2CCC(CNC(c3ccc(SC)cc3)=O)CC2)=O)CC2(CC2)C1 CCC(C(=O)N1CCN(C(c2cc(C3CC3)[nH]n2)=O)C(C2CC2)C1)C(C)(C)CC N1(CC)CCC(N(C(=O)C(N2CCC(c3nc[nH]n3)CC2)=O)C)CC1C C(c1ccc(Cl)cc1F)=CC(=O)NC1CCC(NC(C2(SC)CC2)=O)C1 N1(C(C=COCC)=O)CCOC2(CCN(C(=O)C3=C(Cl)CCC(C)C3)C2)C1 O=C1Nc2ccc(F)cc2C1NCC1NCCC12CCC2 c1(CC)cc(C(N2CCC(NC(C3CC(OC)C3(C)C)=O)C(C)C2)=O)ccc1F Cc1[nH]c2ccnn2c(=O)c1CC(N1CC(CNC(C2CCOC2)=O)C(C)C1)=O c1(C(=O)Nc2c(C)nc(-c3ccc(C)c(C(F)(F)F)c3)s2)cccc2c[nH]nc12 N1(C(C(=O)NCC)=O)CCCC(CC(=O)Nc2ccc(C3CC3)nc2)C1 C1(C(N2CC(O)(CCNC(C(C(C)C)F)=O)C2)=O)CC(=O)OC1(C)C N1(C(c2ccc(C(C)(C)C)cn2)=O)CCC2CN(C(C3CC4CCC3O4)=O)C2C1 C(CC(=O)OC)N(C1CN(C(=O)C(C)=C(C)C)C1)CCC c1(NCC2(CCC)CC2CO)cn(C2CCC(CC)C2)nn1 c1(OC)cc(N)c(C(=O)NCC2(C)CCC(NC(=O)Cc3ccco3)C2)c(F)c1 CS(=O)(=O)C1CN(C(=O)C(c2cccc(Cl)c2)N)C2(CCOCC2)C1 C12(C(c3nnnn3C3CCCC3)NCC3CC(O)C(O)C3)CCC(CC1)OC2 c1(OC)cc(CC(=O)NCCC(C)N(C(=O)COC2(C)CCC2)CC)ccc1O C1(C)(C(=O)NC(C#C)C)CN(C(=O)CCCNC(N)=O)CC1C CC1C(C(=O)NCC(C)NC(c2nccc(Cl)c2F)=O)=NOC1C N1(C(C(CCC)F)=O)CCC2(CC(NC(=O)CC3CC3c3ccccc3)C2)C1 C1(C(=O)NCc2c(C)nn[nH]2)CCN(C(=O)CCOC2CCC2)C(C)(C)C1 C(=O)(CCCCCC(C)(C)C)NCC1CC(NC(c2c(OC)nsc2)=O)C1(C)C C(=O)(C(C(=C(COc1ccc(F)cc1)C(C)C)OC)N(C)CCOC)OC C1(NC(c2cc(CC)n(C)n2)=O)CCN(C(=O)C2=CCCCC2)CC1F C1(CNC(C2C(C#N)C2)=O)CC2CN(C(c3ccc(-c4ccccn4)s3)=O)CC12 C1(NC(c2c(C)noc2)=O)CN(C(c2nncs2)=O)CC1C1CC1 C1(C(N2CCC(N(C(C=CCOC)=O)CC3CC3)C2)=O)CCC2CCCCC2C1 Cc1ccc(Br)c2c1C(C)(C)CN2C(c1ccc(C(C)(C)C)s1)=O C1(C(N2C(C(=O)NC3CC(CN(C)C)C3)C(O)CC2)=O)CC(=O)C12CCC2 Cc1cn(CC(N2CCCC(N(C(=O)CC3CC3(C)C)C)C2)=O)c2ccccc12 c1(C(N2C(COC)SCC2)=O)cc(O)nc(SC)n1 N1(C(=O)C=CSc2ccccc2)CCN(C(=O)NC2CC2c2nc[nH]n2)CC1 c1(C(=O)NC(C)(C)CCNC(=O)CC2CCCC(F)(F)C2)cncc2c[nH]nc12 c1(C(N2CCC(CC(C)NC(c3cnc(S)nc3)=O)CC2)=O)cc(N)ccc1Cl c1(C(N2CC(N(C(C(C)N(C)C)=O)C)C2)=O)cc(C2CC2)cc(F)c1 N1(C(C(C)n2ccnn2)=O)CCCC1CN(C(=O)Cc1cnn(C(F)F)c1)C C1(NC(c2c(Cl)ccc(C)c2)=O)CC2CN(C(=O)C(C)(O)C(C)C)CC2C1 C#CCCCCCC(=O)NC(CC(=O)N(c1ccccc1F)C)C(F)(F)F C(=O)(CCC(C)(C)F)N1CCC(N(C(C2CCC2)C)Cc2nnc(CC)o2)C1 N1(C(C(CCC=C)NC(C)=O)=O)CCN(C(=O)C(O)COC)C2(CCC2)C1 c1(N2CCC(NC(=O)CCCc3ccccc3)C(F)C2)cc2ncnn2cn1 c1(C(=O)N(CC2N(C(C=CC)=O)CC(OC)C2)CC)cc(C)n(-c2ccon2)c1C C(=O)(C1=CC(O)C(NC(=O)CC2=CCOCC2)C1)NC1(C(=O)OC)CC1 C1(CNC(C2C(C)(C)C2)=O)COCC1NC(c1cn(C(C)(C)C)nn1)=O Cc1cc(CC(N2CCC(NC(=O)C=CCOC(C)(C)C)C2)=O)cc(C)c1 C12COCCN1C(=O)c1cn(cn1)CCN(C)C(=O)CS2.C(=O)(C1CC1)N(C)C C1(C(=O)NCCc2cc(CC)no2)CC(C)(C)CCN1C(=O)CCCC(C)CC c1(C(CC(=O)NCC=CCNC(CC(C)n2cccn2)=O)O)ccc(Cl)cc1 C(CNC(C1(NC(C2CC(F)C2)=O)CC1(C)C)=O)(C(C)C)OC c1(CC(N2CCC(C(C)NC(C3C(CC)CCC3)=O)C2)=O)nnc2n1CCOC2 c1(C(=O)NCCNC(c2ccccc2)=O)cccc(C2CC2)c1F.c1(N)cccnn1 c1(C(N2CCCC(O)(CNC(CNC(C)=O)=O)CC2)=O)cnc2n1CCC(C)C2 C1(NC(=O)COc2cccc(F)c2)CCN(C(=O)COC2CCCC2)CCC1CO C1(N(C)C(c2cc[nH]n2)=O)CC2CC1N(C(c1nnn(C3CC3)c1C(F)F)=O)C2 N1(C(c2c(SC)csc2)=O)CC2COCC(C1)C2NC(=O)CCn1ccnn1 c1(COC)nc2ccccc2c(C)c1C(=O)NCCN(C(=O)C(C)C(C)O)C N1(C(CC2C(C)OCC2)=O)CC2CCC1CC2NC(=O)CCC(C)(C)C Cc1ccc(CCC(=O)NCC2(C)CN(C(=O)CNS(C)(=O)=O)C2)cc1C C1(C(C(C)C)NC(C2CC(OCC)C2)=O)CCN(C(c2ccc(=O)oc2)=O)CC1 C(CCCCCCCF)N(CC(C)C)C(N1CCOC(N)C1)=O CCC(C)C(O)C(=O)NCC(C(=O)NCC1CCCC1)n1cc(COC)nn1 C1(C(N)=O)(c2ccon2)CCN(N2CCCC23CCS(=O)(=O)CC3)CC1 c1(NC(C)=O)cnc(O)c(C(N2CC(CO)(NC(C3CCC(=O)N3)=O)C2)=O)c1 Cn1nc(C(N2CCC(CO)C(NC(=O)Cc3ccc(O)nc3)C2)=O)c(Cl)c1Cl C(=O)(C1=CC2CCCC12)Nc1ccccc1.CC1CN(C)C(=O)C2CN(C1=O)C2 C(=O)(C(CO)C(F)(F)F)N(C)CC1C2CN(C(c3ccc(=O)n(C)c3)=O)CC12 c1(C(=O)NC2(CO)CN(C(CCOC(CC(C)C)C)=O)C2)cn2ncccc2n1 C=CC(CCC)CC(=O)N1CCC(C)(C(=O)NCc2cc(F)ccc2F)C1 N1(c2ncc(C)cn2)CC(NC(=O)C=Cc2cncn2C)CCC1C c1(C(=O)NCC(C(N2CCC(C#N)C2)=O)OC)[nH]ccc(=O)c1C c1(CC(=O)NCC(C)NC(C2(C#N)CC(=O)C2)=O)c[nH]c2cc(Cl)ccc12 C1(C(N2C3(C(N4C(CN=[N+]=[N-])CC4)=O)CC3CC2)=O)CC(C2CC2)=NO1 Cc1cc(N)c(C(=O)NC(C)CCNC(=O)CCc2ncccc2C)c(F)c1 Cc1c(C(=O)NC23CCCN(C(=O)Cn4cncn4)CC2C3)sc2nccn12 C1(C(N2CCC(N(C)Cc3nnc(C)n3C)CC2)=O)CCC2(CCOC2)O1 N1(C(C2(OCC)CCOC2)=O)CCC(CO)(CNC(c2nocc2C)=O)CC1 Cc1nc(-c2cn(C3CCC(C(N4CC(O)(CO)C4)=O)C3)nn2)cs1 CCC(C)C(O)CC(=O)NCCN(C(c1coc(C)c1)=O)CC1CC1 C1(C(N2C(C(N(CCCCC=C)C)=O)COCC2)=O)CC2(C1)CC(O)C2 c1(C(=O)NCCC2(O)CN(C(C3CC(C(=O)OC)C3)=O)C2)c[nH]c(=N)nc1C c1(C(=O)NCC23CN(C(C4(C)CC4)=O)C(C2)CO3)cc([N+](=O)[O-])cnc1C1CC1 CC1CN(C(=O)COc2ccn(C)n2)CCC1N(C(=O)C(C)(C)CC#N)C N1(C(c2c(COC)scc2)=O)CCCC12CCN(C(c1cc(C)cc(F)c1)=O)C2 c1(C(N2CCC(C3N(C(C(C)C4CCC4)=O)CCC3)C2)=O)ccn2nccc2n1 c1(C(=O)NCc2cccc(NCCC(C)SC)n2)cc2ccncc2[nH]1 C(CC(C)(C)C(=O)NC(C1CCN(C(=O)C(C(C)C)NC(C)=O)CC1)C)OC c1(N2CCC(CC(=O)N(c3ccccc3C)CCC)CC2)ncnc(Cl)c1Cl n1(CC)nc(C)c(C(=O)NC2CCC2NC(c2cnc(O)cc2OC)=O)c1C CS(=O)(=O)CCCCCNC(=O)C(O)Cn1cncn1 N1(C(CCC=CC#N)=O)CCC(Cc2ccccc2)C(O)C1 c1(OCC)ncccc1CC(=O)NCC(C)CN(C(=O)CCc1nncs1)C C12CCC(O)CN(C1)C(=O)CN2.C1(C(N(c2ccccc2)CC)=O)CCOCC1 c1(C(N2CC3C(CCNC(CC(CC)(F)F)=O)(CC3)C2)=O)ccn2ccccc12 C1(NC(CCC(=O)N(C(C)C)C)=O)CCN(C(=O)C(C)(C)c2cncs2)CC1C C#CC1(C(=O)N(C)CC2CCC(NC(=O)C(C3(O)CCCC3)F)CC2)CC(=O)C1 CC1(C)C2CC1CNC(=O)C(=O)N2.C1(CC(=O)NCC(F)F)CSCCO1 c1(NC(CC2N(C(CC(C)N(C)C)=O)CCCC2)=O)cc(F)c(F)cc1Cl n1(CC)nnc2c1C(C(=O)NC(c1cc[nH]n1)C)CN(C(C1CC1(F)F)=O)C2 N1(C(C(COCC)NC(=O)CCN2CCCC2=O)=O)CC2CCN(C)C2C1 C1(CO)CN(C2CC2)CCC1(F)F.C(c1ccc(OC)c(Cl)c1)=CC(=O)OC(C)(C)C C(=O)(C(=O)C(C)(C)C)NCc1cncc(C(=O)Nc2cccc(C(C)C)c2)c1 c1(CC(=O)NCCCN(C(C=C(C)C)=O)C2CC2)cc(F)cc2c1OCOC2 C(=O)(C1=CS(=O)CCC1)NC1CCCC(CN(C)C(C2(C)CC2)=O)C1 Cc1cc(C(=O)NC2CCC2CC(NCP(C)(C)=O)=O)c(C)nn1 C1(NC(c2c(Br)ccc(C#C)c2)=O)CC1C1CCN(C(=O)C2=COCC2)CC1 c1(CN(CC(C)C)C)nc(C(C)(C)C)c(Br)s1 N1(C(c2nnc(-c3ccncc3)o2)=O)CCC(O)C2(CC2)C1 C(c1ncccc1C)=CC(N1C(CNC(C(C#C)(C)C)=O)C(C)CC1)=O Cc1c[nH]c(C)c1CCC(=O)NC1CC1C(=O)Nc1cn(C)nc1C(F)(F)F N1(C(C(CO)NC(C2C(C)(C)C=C2)=O)=O)CCCC(N=[N+]=[N-])C1 c1(C(N2C(C)CCC(CO)C2)=O)cnc2ccccc2c1 CC1Cn2nccc2CN1C(c1sc(Cl)cc1Cl)C(=O)NCC1CCOC1 Cc1ccc(OCCCC(=O)NC2CN(C(C3CC3F)=O)CC2(C)C)cc1C C1(NC(Cc2ccn(CC)n2)=O)CCN(C(C2CCC=CCCC2)=O)C(C)C1 c1(C(N2C(C)(C)C(CNC(=O)C3=CCCO3)CC2)=O)cc2ccc(F)cc2o1 N1(C(C(C)(CO)OC)=O)CC(C2CCCN(C(c3ccnc(CO)c3)=O)C2)C1 O=C(NNc1ccc(Br)c2ccncc12)c1ccc(Br)cc1Cl Cc1cc(C)c(C(=O)NCC2CC2CNC(=O)C(N2CCCCCC2)C)s1 C12(C(C#C)NC(=O)C(C)=CCNC(=O)COC3CCOC3)CCC(CC1)C2 c1(OC)ccsc1C(=O)N(CCNC(c1coc(-c2cccnc2)n1)=O)C(C)C N1(C(c2c(NC(C)=O)sc(Cl)c2)=O)CCCC(C(=O)NCCN2CCCC2)C1C C1(CC(N2CCCCS2)=O)CCCN(CCCc2nn[nH]n2)C1 Nc1ccc(C(N2CCC(NC(=O)CC3CC3)C3(CCC3)C2)=O)c2cnccc12 c1(C(=O)NCC(CNC(C(=Cc2cccs2)C)=O)(C)C)cncc(S(C)(=O)=O)c1 C(=O)(C1CCCc2n[nH]cc21)NC(CNC(c1cc(OC)ncc1Cl)=O)C(C)C N1(C(C2CC(C)(C)C2)=O)CC2CN(C(C3CC(C(=O)OC(C)(C)C)=NO3)=O)CC2C1 Cc1cn2cccc(C(N3CC(NC(=O)CCCc4cncs4)CC3C)=O)c2n1 C(C(=O)N1CCCc2ccnn21)(C(C)(C)O)NC(C1C(C)C2CCC1C2)=O c1(CCC)cc(C(N2CCCC(CN(c3nnc(SC)s3)C)C2)=O)n(C)n1 C1(C(=O)NC2C(CNC(C3(CC)CCCC3)=O)CCC2)CCC2(CCC2)CO1 C1(CNC(c2nc(C(C)=O)sc2)=O)CC(C)(C)CN1C(c1csc(Cl)c1OC)=O C1(CNC(CC(COC)C)=O)CC2CCC1N2C(=O)CC(=O)NCC1CC1 C1(C)(c2ccc(Br)cc2)CC(NCCCc2cncs2)S1.n1(CC)nnnc1.SC CC1CCN(C(=O)C(C)(C)NC(c2nccs2)C)CC1 n1(CCOC)cc(NC(=O)C(Cc2ccco2)NC(=O)Cc2cc[nH]n2)cn1 C1(N(C(CCCOC)=O)C)CCCN(C(=O)CC(C)(C)c2ccc(C)cc2)CC1 C1(OC)CCC(C(=O)NCC2CCN(C(C3CCCCS3)=O)C2)CC1 C(c1nc(C)cs1)=CC(=O)N(C)CC1(CNC(C(CC)F)=O)CC1 c1(C(=O)NCC(C)CNC2(CC=C)CCC2)ccc(-n2ccnc2)cn1 CCC(C)CCC(O)CC(=O)NCC(C(C)C)NC(c1cc(OC)ccc1C)=O N1(CC)CCC(CNC(c2n[nH]cc2CNC(c2cc(OC)n[nH]2)=O)=O)C1 CCC1=NOC(CC(=O)NCC2(CCNC(=O)CC(C)n3ccnc3)CC2)C1 C1(N(C(=O)Cc2cn[nH]c2)C)CCN(C(C2(C)CCNC2=O)=O)CC12CC2 N1(C(C(=O)NCCOCC)C2CCC2)CCC(C(=O)OC)C(C)(C)C1 CC1=NS(=O)(=O)N(C)C=C1C(=O)NC1COCCC1NC(=O)C=CC(C)C C1(NC(c2c(-c3cc(C)no3)ocn2)=O)CN(C(=O)CCCC#N)CC12CCC2 N1(C(CN(CC(C)C)C(=O)CC2CCCOCC2)=O)CCC2(CCOC2)CC1 C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)NCCC(C)CCNC(C12COCC1C2)=O C(CC(=O)NC(c1ncccc1F)C)(C(F)(F)F)NC(CCc1cc(C)on1)=O C1(CC(=O)NCC(=O)NCC2(ONN)COC2)CCC(=O)N1.C1(C)CCCO1 C12(NC(CC=CC)=O)CCN(C(c3nn(CCC)cc3Cl)=O)CC1C2 C1(CNC(CCCC#CC)=O)C(C2CC2)CCN1C(C1CCCC(F)C1)=O N1(C(C2C(C)OCCC2)=O)CCN(C(=O)CCC2CCC(=O)C2)CC12CC2 c1(CNC(C=CC(CC)C)=O)cc[nH]c1C(=O)NC1(c2ccccn2)CC1 c1(C(N2CC(C)C2(C)C)=O)cc(OC(F)F)cc(SC)c1.C(C)(C)(C)O N1(C(c2nc(NC)sc2)=O)CC23CCCC2(C1)CN(C(C1(C)CCCCC1)=O)C3 C1(C(N2CCOCCC2C(N2CCC(CC3CC3)CC2)=O)=O)CC(O)C12CCC2 c1(NC(CO)=O)ccc(OC)c(OC)c1.c1(-n2c(OC)ccn2)ccc(C)cc1 CC1COCC(C(=O)NCc2ncccc2CNC(=O)CCc2nc(=N)[nH][nH]2)O1 Cn1cc(C(N2CCCN(C(C3(C)CC3(F)F)=O)CC2)=O)c(=O)n(C)c1=O Cc1cncc(CNC(C2CCC2NC(=O)C(n2nccc2C)C)=O)c1 c1(OC)cc(CNC(=O)C(F)ONC(=O)C(C)=O)cc(OC)c1OC.C(C)(C)(C)O CC(C)C(CO)NC(=O)C(c1ccccc1)NC(C1CC12CCC2)=O c1(C(=O)NC(c2ccccc2)C(=O)NCC2CCSC2)ccc(F)cc1F C(N=c1[nH]c(=NCCC(C)O)c2ncccc2[nH]1)c1cccc(CC)c1 C1(NC(c2nc(Cl)cs2)=O)CC2C(NC(c3cc(F)c[nH]3)=O)C2C1 N1(C(C(C#C)(C)C)=O)CCC2CC(C1)CN(C(c1cncc3sccc13)=O)C2 N1(C(CC(CC)C2CC2)=O)CCCC2(C1)CN(C(c1nnsc1C)=O)CCO2 Cc1cc2n(n1)CCN(C(=O)C1=CC(O)C(NC(c3ccc(C4CC4)o3)=O)C1)C2 c1(NC(c2cccc(COCCO)c2)=O)cc2cc(F)cc(F)c2[nH]1 C(=O)(CC(C)(C)C(F)F)N1CC(CC(=O)NCCc2cc(C)no2)OCC1 N1(C(C2N(C(C)=O)CCCC2)=O)CCN(C(=O)C=CC(=O)NCC2CC2)CC1C C1(COC)(NC(c2occ(C)c2C)=O)CCCN(C(c2cccn2C(C)C)=O)C1 C(=O)(C(CNC(C1(N2CCCC2)CCC1)=O)N(C)C)NCC(c1nccs1)C N1(CC)CC(NC(C2(C)CCN(C(=O)C(C3CC3)C3CC3)C2)=O)CCC1=O CC(C)P(=O)(CC(=O)NCC(F)CNC(c1cc2n(c1)CCC2)=O)C(C)C c1(C(=O)NC23CC(NC(Cc4scc(C)n4)=O)(C2)C3)coc2c(F)cccc12 C(=O)(C1COc2ccc(Cl)cc21)NC1(C)CN(C(c2cc3n(n2)CC(F)C3)=O)C1 N#Cc1c[nH]c(C(N2CC(CNC(C3CC3C3CC3)=O)C2)=O)c1 c1(-c2cn(CCCN(C(C(C)P(C)(C)=O)=O)C)nn2)ccc(F)c(C#N)c1 C1(C(N(C2CCN(C(=O)CCOCC(F)F)C2)CC#C)=O)CC12CCOCC2 C(=O)(CC(C(F)F)N1CCOCC1)NCC(CCCC)NC(C1CSC1)=O C1(CNC(C2(F)C(C)C2)=O)CCC2CN(C(C3(C)COC3)=O)CCC2C1 c1(NC(C2CCN(Cc3cc(O)nc(O)n3)CC2)=O)cnc2cccnn12 N1(S(c2ccc(NC3C(OCC)COC3)nc2)(=O)=O)CCC2(CCN(C)C2=O)C1 c1(C(N2CCCC(n3cc(C4CCCC(C)C4)nn3)C2)=O)ccc([N+](=O)[O-])n1C N1(C(CSC)=O)CCC2(CCCCC2NC(=O)C(C)C2CCCC2)CC1 CCC(CCC(=O)N1CCCC(C(=O)NCc2cnc(OCC)cn2)C1)OC CC1(C)CC(=O)NC1CNc1cc(CN2CCCCC2)cc(Br)c1 C1(NC(c2ccc(F)c(C(F)(F)F)c2)=O)CN(C(=O)C2CC2)C2(CCC2)C1 c1(NCC(CNC(c2c(CC)n[nH]c2)=O)C)ncc(C#N)cc1C(=O)OC C(CC(=O)N1CCC(C(N)=O)C1)(C(F)(F)F)NC(c1c(COC)cco1)=O c1(C(=O)NC2CC(CNC(CC=C=C)=O)C2)scc2c1CCCC2 N1(C(c2[nH]c(=NC)sc2)=O)CC2CCN(C(=O)C=C3CN4CCC3CC4)CC12 C1(NC(c2c(C)nco2)=O)CCC2CC1CN2C(C12C3C4C1C1C2C3C41C)=O Cn1cccc(C(=O)NOCC(N2CCC3(CC3)C2)=O)c1=O c1(NC(CNS(CC(CC)C)(=O)=O)=O)ccc(Br)c(S(N)(=O)=O)c1 C12(C)CCN(C1)C(=O)C1CC1CNC(=O)C2.c1(C(C)=O)cc(C(C)C)no1 c1(C(C)C)ccc(C(=O)COC(C2CCC=CO2)=O)c(C(F)(F)F)c1 N#Cc1c(F)cc(-c2cncc(F)c2C(=O)Nc2cncnc2Cl)cc1F C1(OC)(CNC(c2[nH]ccc2C2CC2)=O)CCN(C(c2c(C)ncn2O)=O)CC1 C1(OCC(=O)NCC(C)N(C(=O)CC2CCCC2)C)CCCCC1C C(C(CC1CC1)C(=O)N(C(C)C(C)(C)O)C)NC(C=C(C)C)=O c1(SCC(=O)NCCCCCF)ccccc1-n1cc(C2CCC=CO2)nn1 c1(C(=O)NCC(C)CNC(C2(C)CCC(F)(F)C2)=O)c(N)cc(F)cc1F CCC(CCCC(=O)NCC1CC2CCC2C1)NC(C1CC(N(C)C)C1)=O CC(=O)CCCC(=O)N1CCCOC(NC(=O)COCP(C)(C)=O)C1 N1(C(C(CCC)CC)=O)CCC2(C1)CN(C(C1CCCC(=O)CC1)=O)CCO2 c1(C(C)C)cc(C(=O)NC2CCNC2C(C)C)c2cn[nH]c2c1 Cc1cc(OCC(=O)NCC(CNC(C2CC(CC3CC3)C2)=O)CO)no1 Cc1nc(CC(=O)Nc2cnn(C(C)(C)C)c2)sc1NC(=O)OC(C)(C)C CC1CCCCN1CC(=O)NC1CC(NC(=O)C(O)Cc2cnc[nH]2)C(O)C1 c1(C(N(CC(CC)NC(C(CC=CC)CC)=O)C)=O)cc(OC)cc([N+](=O)[O-])c1 c1(C(N2CC(CC)N(C(c3cc(C(N)=O)c[nH]3)=O)CC2)=O)ccnn2ccnc12 CCC(C(=O)NCC1CCCN1C(C1C2CN(CC(F)(F)F)CC12)=O)C(C)C C1(F)(SCC(F)(F)F)CCC(NC(C2(NC(N)=O)CC2)=O)C1.C1(=O)CN1 c1(OC)cc(CNC2CCN(c3ncnc(O)c3Br)CC2C)ccc1Cl C1(C(N(CC(CNC(C2(CC)COC2)=O)(C)C)C)=O)CCc2cnn(C)c2C1 C(CCCCCNC(c1c[nH]nc1C(F)(F)F)=O)NC(c1cc(COC)no1)=O CC12CCCC(C(N3CCC(CCNC(=O)Cc4csc(Cl)c4)CC3)=O)(CO1)C2 c1(C2CN(C(C3C(C(C)O)C3)=O)C2)cn(Cc2nocc2C(C)(C)C)nn1 C1(CC)CN(C(=O)Cc2ncc(C)[nH]2)CCN1C(c1cc(F)n[nH]1)=O C1(NC(C2(C(C)C)CCC2)=O)CCCN(C(c2ccccc2C#N)=O)C1C N1(C(CC2(C)CCOC2)=O)CC(O)CC1C(N1CC(CO)C(O)C1)=O c1(OC)c(C(=O)NC2(C3CN(C(=O)C(O)CCSC)C3)CC2)cccc1F C(=O)(CCC(C)CC)N1C(C(N(CCC)CCN(C)C)=O)(CC)CCC1 C1(C(N)=O)CN(C(C2(NC(=O)COCC3CC3)CC2(C)C)=O)CCO1 N1(C(C2CC3(CC3)CN2C(c2cocn2)=O)=O)CCc2nnnn2CC1 Cc1cccc(CCNC(=O)CN(C(=O)COCP(C)(C)=O)C(C)C)n1 C1(N(C(CC2CCC2)C(=O)N(C)CCOC(F)F)C(C)=O)CCN(C(C)=O)CC1 N1(C(C(C)NC(C2CC2(F)Cl)=O)=O)CCC(C(C)(C)C)C1 Cc1nc(C(C)C)ccc1C(=O)NC1CC(NC(=O)C(C2CCOCC2)C)C1 C(C1CCCC1)=CC(=O)N(C(C)C(=O)NCCCNC(N)=O)CCOC N1(C(CN(C(C2CC(C)OCC2)=O)C2CC2)=O)CC2CC2C2CC12 C1(O)(CNC(c2cc[nH]c2)=O)CCN(C(c2cc(C3(C(=O)OC)CCC3)[nH]n2)=O)C1 C(C(CC(C)C)C(=O)NCC1CCCN1C(=O)CCc1nc(C(C)C)no1)OC N1(C(C2CCCCCN2C(=O)CN2CCC(F)CC2)=O)CC2CCC(CC2)C1 N1(C(c2c(C)nsc2)=O)CC2(CCN(Cc3c(Cl)ccnc3Br)C2)C1 C(N=c1[nH]c(=NCCC2CC2(Cl)Cl)[nH]c2c1CSC2)C1N(C)CC1 Cc1cc(C#N)c(C(=O)NCC2COCC(NC(=O)OC(C)(C)C)C2)s1 N1(C(c2cccc(C)c2)=O)CC2CCN(C(c3ccsc3C)=O)CCC2C1 N1(C(C(C=C)(C)C)=O)CCC(C(N2CCC(C)(CCO)C2)=O)C(C)(C)C1 Cc1cnc2ccccc2c1C(N1Cc2cnc(C(C)C)nc2C1)=O c1(OC)nc(NCC2CNCCN2C(=O)C(C)NS(C)(=O)=O)nc2[nH]cnc12 c1(C(=O)NC2CN(C(C=C(CC)C)=O)CC2C)cnc2c(c1)c(C(C)C)nn2C N1(C(C2C(C)C2)=O)CCCC(C)(C)C1CNC(=O)CCOCC(F)(F)F c1(CC(=O)NC2C(CNC(C(CC)n3ccnc3)=O)C2)c[nH]c2cnc(Cl)cc12 C12(CNC(C3(C)C=CCCC3)=O)CCC(CN(C(c3cncc(C#N)c3)=O)C1)C2 N1(C(CCSC)=O)CCN(CCNC(=O)CC2C=CCC2)CC1 C12(NC(c3oc(C)c(CO)c3)=O)CCN(C(=O)C(C)(C)C)CC1C2 c1(C(=O)NCC(CO)OC)c[nH]nc1CCNC(=O)Cc1ccnn1C C1(C(=O)NCCC(=C)CNC(=O)CCC(C)(C)C)CC2CCC1CC2OC CC(C(C)(C)C)=CC(=O)NCC(C(C)C)NC(=O)C=CC(C)C c1(C(=O)NC2(C)CCCN(C(=O)C3=COCCC3)C2)cccc2oncc12 N1(C(C(C2CCN(C(c3ccc(F)c(F)c3)=O)CC2)C)=O)CCC2(CCCO2)C1 C1(C(=O)NCCn2cncn2)C2CC1N(Cc1cccc(O)c1)C2 C(C(CC1CC1)C(=O)N(C)Cc1ccncc1)NC(C(C)SC)=O N1(C(C=CSC)=O)CCC2(NC(c3cc4ccnc(Cl)c4[nH]3)=O)CCCCC12 c1(C(C(=O)NCCC)N(C)CCOC)cc(C(=O)OC)c(CC)o1 c1(S)ccc(C(=O)O)o1.c1(CN)ccc(Br)s1.c12n[nH]cc1NC2=O c1(C(c2nnnn2C2(C)CC2)NCC2(COCC)CC2)cncc(C)c1 N1(C(C(CC)N(C)C)=O)CC2(C(=O)NC3CC3C(F)(F)F)CCC1CC2 C1(COC)CCCC1NC(c1csc(C)c1)=O.c12cc(on1)CNC2=O.C(C)(C)(C)O Cc1ccn2ncc(C(=O)N(C)CCN(C(=O)CC3CCC3C3CC3)C)c2c1 Cc1nn(C)c(Cl)c1C(N1CC(C)OC(C)C1)C(N1CCC(CCNC)CC1)=O c1(-n2c(C(C)C)nc(-c3ccsc3)n2)ccc(C#N)cc1 N1(C(CC=C(C)C)=O)CCCC2(N(C(=O)CCc3ccc(Cl)nc3)C(C)C)CC12 C1(NCC(=O)OC)CCN(C(c2cc3n(c2)CCC3)=O)CC1C Cc1ccc(S(=O)(=O)N(C)C)cc1C(=O)NC1CC1NC(c1ocnc1C(F)F)=O C1(SC)CCN(C(=O)C(CC2CC2)NC(=O)CC(=O)NC2CC2)C1 CC(CC(=O)NC1(CO)CN(C(C2CNC(=O)C2)=O)C1)CC(C)(C)C C(CCNC(=O)C=Cc1cscn1)(C(=O)N1CCCC1CN=[N+]=[N-])OC C1(CN(C(=O)CCCNC(C2(C(N)=O)CCC2)=O)C)CCCCNC1=O NCC1CCCn2ncc(C(N3CCCC3c3ccc(F)c(Cl)c3)=O)c21 c1(NC(N(CC=C)C2CC2)=O)ccc(N(S(C)(=O)=O)C)cc1C.C(C)(C)N C(=O)(C(C)(C)C(C)O)NCC(C)CN(C)C(c1ccc(CO)c(F)c1)=O N1(C(C(C=C)(C)O)=O)CC2(CNC(=O)C=CCNC(=O)OC(C)(C)C)CCC1CC2 C1(CNC(C2C(=C)C2C(=O)OC)=O)CN(C(=O)C(C)CC2CCC2)CCO1 C1(NC(c2ccc(OCC)cc2)=O)CCN(C(c2cc(C)nc(C)c2)=O)C(C)C1 C(=O)(C(C)(C)CCCNC(=O)CCNC(=O)CO)NCC(C(C)C)(C)F.O Cc1cc(C#N)c(F)cc1NC(C1C2CC1N(Cc1cccc(F)n1)C2)=O c1(N2C(CN(C(C(CC)F)=O)C)CCC2)cc(C)ccc1[N+](=O)[O-] C12(C(=O)NC3(C)CCN(C(CS(CC)(=O)=O)=O)C3)CCC(OC)(CC1)CC2 N1(C(C(C(C)(C)C)O)=O)CCC2(COCCN2C(C2CCC(F)(F)C2)=O)C1 c1(CN2CC3C(C(=O)NC4(CC(C)C)CCC4)(C3)C2)nc2ccc(F)cc2[nH]1 c1(CC(=O)NCC(C)(C2CCC2)NC(c2nc(CC)sc2)=O)ccc(C)nc1 C(=O)(CCCCN=c1cc(C)nc(N2CCCOC(C)C2)[nH]1)NC N1(C(CN(C)CC)=O)CC(NC(=O)Cc2ccc(C)cc2)C2CCCC12 c1(C(=O)NC2CN(C(CCC=CCC=C)=O)CC2C)cnn2c(O)cc(C)nc12 N1(C(C2CC(OC)C(OC)C2)=O)CCC(C)(C)C(NC(c2ccnc(C)c2)=O)C1 CC(O)C(C)(C)C(=O)N1CC2CC(C(=O)NC(CN(C)C)CO)(C2)C1 Cc1ccc(CC(=O)N(C(N)=O)Cc2ccc(C#N)cc2)cc1C c1(CCC)nc(C(=O)NCC2CCN2C(c2csc(-c3nc[nH]n3)n2)=O)co1 Cc1nn(CCC(=O)N(C(CNC(C2CCCC2)=O)C2CC2)C)c(C)c1[N+](=O)[O-] NC(=O)CCC(C(=O)NCCC(=O)N1CCCC1)n1cc(-c2cncs2)nn1 C12(C(=O)NCC(=C3CN(C(c4cncc(SC)c4)=O)C3)F)CC3CC1C2C3O CCC(CC(=O)N(CCCNC(c1ccncc1F)=O)CCO)C1CC1 c1(OC)cccc(SCC(=O)N(C2CCN(C(=O)Cc3c[nH]nc3O)CC2)C)c1 n1(CC)cc(C(=O)NCCC2(CNC(C3CC4CC4C3)=O)CC2)c(C(C)(C)C)n1 Cc1cc(C(N2CCCCC2CC(=O)NCc2cn(C)cn2)=O)cc(C#N)c1 N1(C(C(F)=C(C)C)=O)CCN(C(C2COC(=O)C2)=O)C(CCO)C1 N12CCC(=O)N(C1=O)Cc1ccc(cc1)C2.N1(N(CC)CC)CCCC(CF)C1 c1(CC)cnc(C(=O)N(C2CCCCC2)CCNC(=O)CC(C)OC)nc1 Cc1cc(CC(=O)N(C)CCNC(C2NC(=O)OC2C)=O)c(C)s1 N1(C(c2[nH]cc(C)c2)=O)CCC(NC(=O)CCc2ccnn2C)CC(C)(C)C1 C1(NC(c2nnnn2C2CC2)(CSCC)C)CCC(S(C)(=O)=O)C1 Cc1ccc(C)c(C(=O)NC(C)CCN(C)C(C2(CF)CCC2)=O)c1 c1(N2CC(C)SCC2)ccc(S(=O)(=O)NCC2CCCC23CC3)cc1Cl C12(CNC(c3n[nH]c(C)c3C)=O)CCC(CN(C(=O)CN3CCC(O)CC3)C1)C2 n1(CCCN(C(CNC(C(C)SC(F)(F)F)=O)=O)C)cc(CO)nn1 C1(C(N2CC(C)(NC(C(COC(C)C)(C)C)=O)C2)=O)CCN(C)C(=O)C1 c1(N2C(C)CC(CNC(C(C(CC)C)C)=O)C2)ncnc2c(Cl)cc(Cl)cc12 C(=O)(C#CC1CCCCC1)N1CC(C)C(NC(C2CCC3(CCOCC3)O2)=O)C1 C(=O)(C(=O)NOC)NCCCC(=O)NC(CC)CO c1(C(N2CC(CNC(C(C(C)C)F)=O)C(O)C2)=O)cccc(Cl)c1Cl O=C(CC1C2CCC1CN(Cc1ccccc1)C2)N=c1cc[nH]cc1OC(F)F Cc1ccc(C(=O)NCC2C3CN(C(c4cnncc4N(C)C)=O)CC23)c(C)n1 C1(CNC(C2(COC)CC2)=O)(CO)CCN(C(C2CCCCC2(C)C)=O)CC1 N1(C(C(CC)OCC)=O)CCOCC1CN(C)C(c1nc(C)sc1C)=O Cc1ncnc(C(=O)NC2CN(C(=O)Cc3csc4nccn34)CC2F)c1C N1(C(CC2(CSC)CC2)=O)CC(NC(=O)C(C)(C)NS(C)(=O)=O)CC1(C)C CC1(C)C2CCC1(C(N1CCCCC1C1CCN(C(C3CCCS3)=O)C1)=O)CC2 CC(C)C(C(=O)N1CC(C(C)NC(c2cnn(C3CC3)c2)=O)C1)C1CCC1 c1(CC(=O)N(C(C)(C(=O)NCCN2C(=O)CCC2=O)C2CC2)C)cccnc1O C(CC(C)C(=O)NCCOC1CCN(C(c2cc(COC)cn2C)=O)CC1)=CC N1(C(C2OCCN(C)C2=O)=O)CC2(CCCC2NC(=O)CC2CSCCS2)C1 C(=O)(C(C(C1CCOC1)OC)N(C1CCCCC1)C1CC(OC)C1)NCCCC C1(NC(C(C)(C)c2ncco2)=O)CCOCC1NC(=O)C1=CCSC1 c1(C(N(CCCNC(=O)Cc2nocc2Br)C)=O)c(F)ccc(F)c1Cl c1(NC(C#C)CC)cc(NC(=O)OC(C)(C)C)c2c(c1)COC2 C1(C(=O)NCC(C(=O)NCC2COCC(C)O2)N(C)C)CCC2(CCC2)O1 C1(NC(C(COC)COC)=O)CC2(NC(=O)C3=COCCC3)COC1C2 c1(OC)n[nH]c(C(=O)NC2CCC(NC(=O)Cc3csnc3C)C2)c1Cl CCC(C)C(CC(=O)NC1CCC(CC)CC1)NC(C1CC1(F)Cl)=O C12(CCNC(=O)COCC3CCCO3)CCC1CN(C(C1(O)CCC1)=O)C2 c1(CNC(C(=O)N(CCCC)CC)C)ccnc(F)c1Cl C1(C(=O)Nc2cn(CC)nc2)CN(C(=O)CC2COCCO2)CCC1(C)C CC(C)CC(CNC(=O)CC1(N2CCCC2)CC1)NC(=O)Cc1cccc(F)c1 C1(CC)CN(C(=O)CC2CC2C2CC2)CCC1CNC(c1csc(O)n1)=O C1(C)(C(=O)NCC(C)(C2CCC2)OC)C=CCN1C(=O)CCOCC(C)C C1(C)(C(=O)NC(CC(C)C)CNC(=O)CC2CCCC2C)CC(C2CC2)=NO1 CC1CC(NCC23CC(C2)C(C(F)F)O3)CN1C(N(C)C)=O C1(NC(C2(C)CC(=C)C2)=O)CC2CC(C1)CN(C(C1(COCC)CC1)=O)C2 C1(C(C)C)N(C(=O)CCC2(C)N=N2)CC12CCN(C(=O)COCC1CC1)CC2 C1(C(=O)NC2(CO)CCSC2)(NC(c2ccnn2CCF)=O)CCSC1 c1(C(COCC)CNCC(c2ccc(F)cc2)(C)C)ccc(F)cc1F c1(C(=O)NC2CC3CC2N(C(C24CCC(C2)C4)=O)C3)cc2ccccc2[nH]1 c1(C(N)=O)cc(CC(=O)NCCCNC(c2csc(-c3ccncc3)n2)=O)cs1 c1(NC(c2ccccn2)CCc2ccc(OC(F)(F)F)cc2)ccc(OC)c(Br)c1.CO C1(CN=c2[nH]cc(C(=O)OC)s2)CCCN(C(CCCc2ccccc2)=O)C1C C1(NC(=O)C=Cc2cncs2)CN(C(=O)CC=C(Cl)Cl)CC12CCOCC2 C1(NC(C2(C)CCOC2)=O)CN(C(=O)CCCC(F)F)CCC1C(F)(F)F C(=O)(CC1=CCCCC1)NCC1C(NC(COc2ccc(C#C)cc2)=O)CCC1 N1(C(C2C(CCC)CCC2)=O)CCC(C(C)(C)C)(CNC(c2c[nH]c(=N)s2)=O)C1 c1(C(=O)NCCC2CCN(C(C(CC)=CC)=O)CC2)cc(O)cc(F)c1 CN1CC=C(CC(=O)N2CC(CN(C)C(C3(F)CCOCC3)=O)C2)CC1 c1(OCC(=O)NC2C3CN(C(C=CC)=O)CC32)ccc(F)c(F)c1 C1(C(=O)NCC(C=C)O)(CNC(c2ncn(C(C)C)n2)=O)CC2(CC2)C1 C=CCCCCCC(=O)NCC(C)(C1CCC1)NC(C1CC12CCOCC2)=O CN1CCN(C(=O)CC2(C)OCCO2)CC1CNC(C1CC(=O)C1(C)C)=O c1(NC2CC(C)N(C(=O)Cc3cnnn3C)C2)ncnc2cccc(F)c12 CCC(C)CCC(=O)N(CC(O)CNC(C1(Cc2ccccc2)CC1)=O)C C12(NC(C(CC=C)C)=O)CCC(NC(=O)CCc3cccc(OC)c3)(C1)OC2 C1(NC(CCCc2scc(C)n2)=O)CN(C(=O)C(N2CCOCC2=O)C)CC1C CN=c1[nH]cc(C(=O)NC(CCC2CC2)C(=O)N2CCCCC2CC2CC2)s1 C1(C(N2C(C3CCN(C(C=NOC)=O)CC3)CCCC2)=O)CCc2nn[nH]c2C1 C1(C(=O)NCC2CCN(CCC)C2)CN(C(c2ccco2)=O)CC(C)(C)C1 N1(C(c2c(CC)scc2)=O)CCC(OCCCNC(=O)CC2CCCC2)CC1 C1(CNC(CC)=O)CC(C(=O)NCCN(CCN(C)C)CC)=NO1.CCC(C)SCC C1(NC(CSCCC)=O)CCCCC12CCN(C(=O)Cn1cc(C#N)cn1)C2 C1(NC(c2cc(OCC)ncc2)=O)CN(C(=O)C(O)C(C)C)CCC12CCC2 CCC(CNC(=O)C(=O)NCCC(c1cccc(C)c1)=O)CC(=O)OC C1(CN(C)Cc2ccc(C(F)F)cc2)CC2(CCC2)CO1.C12CCN(C1)C2=O Cc1cccc(OCC(=O)NCC23CC2CN(C(C2(N(C)C)CC2)=O)C3)c1F C1(C(N2CC3C(NC(=O)Cc4ccc(F)cc4F)C3C2)=O)CC2CCC1C21CC1 C#Cc1ccc(CC(N2CCC(CCNC(=O)C(C)P(C)(C)=O)CC2)=O)c(F)c1 CCC(C(=O)NC1CCCC(NC(=O)Cc2nc[nH]n2)C1)C(F)(F)F c1(C(N2C(CNC(c3ccc(C)cc3C)=O)CN(C)CC2)=O)cc(C)c(=O)n(C)c1 C1(CCC)CN(C(c2nn[nH]c2Cl)=O)CCN1C(=O)C=Cc1ccc(C(N)=O)o1 C12(CCNC(c3c(C)scc3)=O)CCC(C1)N(C(C1CC1(Cl)Cl)=O)C2 c1(C(=O)NC2CN(C(C(CN(C)C)O)=O)CC23CCC3)ccc2cnccc2n1 N1(C(c2c(C#C)c[nH]n2)=O)CC2(NC(=O)CCn3ccnc3C)CCC1CC2 CC(CC(=O)N(CCN(C)C)C1CC1)C(C)(C)CCNC(=O)CCCF C(C1c2ccsc2CCN1C(=O)CCC1CC1)NC(=O)C(C1CCOCC1)F Cc1ccc(CC(N2CC(NC(=O)C=Cc3ccco3)CC2C)=O)cn1 n1(CC#C)cccc(-c2ccc(NCc3ccc(SC)cc3)nc2)c1=O C#Cc1ccc(Cl)c(C(=O)NC(CNC(c2cc(C#C)ccc2Cl)=O)CC)c1 c1(NC(C2CCN(C(c3sc(C)c(Br)c3)=O)C2)=O)cc(C(N)=O)cc(F)c1 N1(C(c2c(I)ccc(C)c2)=O)CCC2(CCCC2C(N2CCC(OC)CC2)=O)C1 C(C(=O)N(C(C)C(F)F)C)(C(C)(C)C)NC(c1nnn(CC)c1C)=O C1(C(=O)NCCN2CCN(C(CN(C3CC3)CC)=O)CC2)CCC(C)(C)CC1 N1(C(Cc2ccc(C)o2)=O)CCCOC(CNC(c2nncs2)=O)C1 C1(CNC(c2[nH]cc(CC)c2)=O)C2CC1N(C(=O)C(C)C(C)n1cccn1)C2 c1(C(=O)NC(C(C)NC(C2CN(C(C)C)C2)=O)CO)ccc(CO)c([N+](=O)[O-])c1 N1(C(c2c(C)cccn2)=O)CCCC(C)(NC(=O)C(c2cccnc2)C)C1 C1(C(=O)N(C(C)C(=O)NCC2CC23CCC3)C2CC2)(OC)CCSC1 C(C)(C)(CCN(C(=O)CC1CCCN1C)C)NC(CSCC#C)=O C1(C(=O)NCC2N(C(Cc3cccc(OC)c3)=O)CC2)CC(=O)CC12CCC2 c1(C(=O)OC)ccc(C(=O)NC2CC(NC(C3CC3(C)C(C)C)=O)C2)cc1Cl Cc1nn(C)cc1CCC(=O)N1CC(OCCC(=O)NC2(CO)CCNC2=O)C1 C12(C(N3CC(CCC)C(CO)C3)=O)CCCC1CCN2C(C1CCCN(C)C1)=O N1(C(c2c(C)nc(-c3ncc[nH]3)s2)=O)CCC(NC(c2coc(O)n2)=O)C1(C)C C1(CC)CN(C(=O)CC2C(=O)ON=C2C)CCC1NC(c1cc(Cl)nc(Cl)c1)=O Cc1[nH]nc(C(F)(F)F)c1C(=O)NCCC1CCN(C(C2CC2Br)=O)C1 C1(OC)CCCC1C(=O)NCC1CCC1NC(=O)Cc1n[nH]c(=N)s1 CN=c1ccc(C(N2C(C(N3CCC3(C)CCO)=O)CC3CC23)=O)c[nH]1 C1(C(N(CC(C)NC(=O)Cc2cnoc2)C)=O)CN(C)CC1C(F)(F)F c1(C(=O)NC(CC)CNC(c2cc(N)cnc2Cl)=O)cnc2[nH]cncc1-2 Cc1c(Br)ccc(C(=O)N(CC(C)CNC(=O)CS(N)(=O)=O)C)c1N N1(C(CCC(=C)Cl)=O)CC2CCCCC2(CNC(c2cc(C#N)ccc2C)=O)C1 C1(NC(C2(CCC)CC2)=O)CCC2CCN(C(=O)Cc3ccccc3Cl)C12 C(=O)(C1=NOC2(CCC2)C1)NC(C)CCCC(=O)N(C)Cc1ccncn1 C#Cc1cccc(C(=O)N(C(C)CNC(=O)C(CC2CCCC2)OC)C)c1Cl N1(C(CC(CC)C)=O)CCc2nc(C(=O)NCC3(COC)CCCC3)ccc2C1 C1(CC(=O)OCC)CN(C(=O)CS(=O)(=O)CC)CCN1C(c1ccc(O)nc1)=O C12(NC(c3cc(CC)ncn3)=O)CCN(C(c3sc(C)cc3C)=O)CC1C2 N1(C(=O)CC(c2ccccc2)n2ccnn2)CCc2c(O)n[nH]c2C1 C1(C(=O)NC2CN(C(CC3CCC(C)(C)CO3)=O)C2)CCC2CCCCN12 C=CCC(C)(CNC(=O)CC(C)N(C(=O)C=Cc1cocn1)C)CO C1(NC(=O)CCCC2OCCO2)(CO)CCN(C(=O)C(F)=C2CCC2)C1 c1(C(=O)NCCC2N(Cc3cn(CC)nc3)CCC2)nn(C)cc1Br c1(CN2C(C(N3CCCC(O)C3)=O)CC(C)C2)ccc2ncnn2c1 N1(C(C2(C#N)CCCCC2)=O)CC=C(C(=O)NOCc2cccnc2)C1 C(=O)(C(C)(O)Cn1ccccc1=O)NC(C)CN(C)C(c1cccnc1)=O c1(N(C)C)c(-c2ccc(C(N3CC(O)CC3CO)=O)s2)cccc1[N+](=O)[O-] C1(C(=O)NC(C)CCC(=O)NC(CC2CCC2)CO)CCC2(CCC2)C1 c1(NC(N2CCC(=C)C2)=O)cc(Br)c(OC)cc1F C(c1nc2ccccc2n1C1CCCC1)=CC(N1CC2CCC1CS2(=O)=O)=O Cc1cn2nc(N3CCC(C)(NC(=O)C(O)C4CCCC4)C3)sc2n1 C1(C(N(C)CC2(C(=O)NC)CC2)=O)(CN2CC(C#N)(CN(C)C)C2)CC12CCC2 N1(C(C2(OCC)CNC2)=O)CCCCC(NC(=O)CCCOC)CC1 C1(O)(CN(C(CCCC#C)=O)C)CCCN(C(c2occc2C(=O)OC)=O)C1 C(=O)(C(C)(C)CCCc1ccccc1)NCC1CC1C(=O)NC(COC)C(C)C C(C(C)CN=c1[nH]nc(O)s1)NC(c1ccc(OC(CC)C)cc1)=O C(=O)(C1=NOC(C)C1C)NCCC(=C)CNC(=O)CN(S(C)(=O)=O)C CN1CC(C(=O)NCCCCCC(=O)N2CCC2C(C)(C)O)CCC1=O c1(CC(=O)NC(C)(CS)C2CC2)ccc(OCC(N)=O)cc1.CC(C)(C)OCC(F)F c1(CC(N2CCN(C(=O)C(F)=C3CCCC3)C3CC23)=O)ncc(Cl)cc1F C1(C(N(CC(C)N(C(CCc2ccc(C)nc2)=O)C)C)=O)CCCCCS1(=O)=O Cn1cc(C#N)cc1NC(C1CCCCN(C(C2CCCOCC2)=O)C1)=O N1(C(c2cc(C)no2)=O)CCSCC1C(=O)Nc1cccc(SC(C)C#N)c1 C1(NC(c2cc(Cl)ncc2O)=O)CC2(CCN(C(=O)CCOCC(F)F)CC2)C1 N(S(C)(=O)=NC1CC1)C(CSc1ccccc1)=O.CC12CCN(C1)C2=O FC1(F)CN(Cc2sccc2Br)CCOC12COC2 Cc1c(C(=O)NCCC(C)N(C)C(C23CC(C)(C2)C3)=O)nnn1-c1ccn(C)n1 C1(NC(C2(CCCC)CC2)=O)CCN(C(=O)CC2(C3CC3)CC2)CC1C C12CCN(C3(CCCC3)C1)C(=O)C(=O)OC2=O.C(C(C)S(N)(=O)=O)NC(=O)OCC N1(C(c2ncoc2C2CCCO2)=O)CCC2(C1)CN(C(=O)CC=C(Cl)Cl)C2 C=C1CCN(C(=O)C=Cc2cc[nH]c2)C(C(=O)NC2CCCCC2O)C1 c1(CC(=O)NCCNC(c2nn(C)c(C3CCCO3)c2)=O)ccc(O)c(F)c1 C(=O)(C(F)(F)CC1CC1)NCCCO.C1(C(N)=O)CC1C(=O)NCC c1cc(S)nc(NCC2(COC)CC2)n1.n1(CCNSCC)ncc(C)n1.CC c1(C(C(=O)NCCC)N(CC2CCOC2)CC2CCC2)ccc2n[nH]cc2c1 c1(C(=O)NCC2CCN(C(C3CCC(C)S3)=O)C2)cc2n(n1)CCNS2(=O)=O c1(C(N2CCCC(c3nc(CNC(CSC)=O)[nH]n3)C2)=O)ccc(Cl)c(F)c1 C(C)(C)(CCCNC(C1CCC(c2ccccc2)O1)=O)NC(C(CC)OC)=O Cc1nc(C)c(C(N2CCC(NC(c3scnc3C(C)C)=O)C2C)=O)[nH]1 Cc1nn(C)c(Cl)c1C(=O)NCC1CN(C(=O)CC(C)F)C1 C(=O)(C(O)CCCNC(c1cc[nH]c(=N)n1)=O)N(C1CCC2CC12)C c1(OC(C)C)nc(C(=O)NC2CCCC2NC(C2(C)CC2(F)F)=O)cc(O)n1 c1(C(N2CC(C=C)C(NC(c3cc(C)n(C)c(=O)c3)=O)C2)=O)ccc([N+](=O)[O-])s1 n1(CC)cc(C(N2CCC2CNC(=O)CC(C)n2ccc(C)n2)=O)cn1 c1(C(C)(C)C)ccc(C(N2CCOC(CNCc3occc3Br)C2)=O)cc1Br c1(C(=O)NCC(CCC)NC(C2CC(C)(C)CO2)=O)cc(C)c(CC)nc1O c1(C(=O)NCC2N(C(c3cccc(NC)n3)=O)CCCC2)ccc(F)c(F)c1F N1(C(C2C=C(C)CS2)=O)CCC(C(=O)NCCCN2CCCC2=O)CC1(C)C C1(NC(C(COC)NC(C)=O)=O)CC12CCN(C(c1cnc3n1CCS3)=O)CC2 CS(=O)(=O)C1(C(=O)NC2CCC(CNC(C3CSC3)=O)CC2)CC(O)C1 c1(C(N2CCCC(NC(c3ccc(Cl)o3)=O)CC2)=O)ccc2[nH]c(=O)cnc2c1 C(C)(C)(CCC(=O)NCC(C)(C)CNC(c1cc(Cl)on1)=O)OC c1(NC(c2ccc(=NCc3ncc(C)nc3)[nH]c2)=O)ccc2c(c1)NC(=O)C2 N1(C(C(C=CC)O)=O)CCC2(CCOCC2)C(NC(=O)CCCOC)C1 N1(C(C2CN(C(C(n3ncc(C)c3)C)=O)CC2(F)F)=O)CCC2CCCC2CC1 c1(CNC(CSC(C)(C)C)=O)ccn(-c2ccccc2)n1 c1(CC(=O)NC(C(C)NC(C2N(CC)CC2)=O)C)ccc(F)cn1 C1(CC)CN(C(C2(CCOC)CCC2)=O)CCN1C(C1CCCS(=O)(=O)C1)=O C(=O)(C(C)(C)C(=O)NCC1CC(NC(=O)Cc2ccc(F)cc2F)C1)OC CC(C)(C)S(=O)(=O)CC(=O)NCC1C(C2CC2)CCN1C(c1n[nH]c(=N)[nH]1)=O N1(C(CCNC(=O)NC)=O)CCC(C(=O)NC2C=CC(COC)C2)C12CC2 c1(C(=O)NC2C(CNC(C3CCC(=O)NC3)=O)CCC2)snc2ccccc12 c1(OC)ncccc1S(=O)(=O)N1CCCC(C(=O)Nc2ccsc2C(N)=O)C1 C1(C(=O)NCC(C)(C)NC(C2(Cc3c(C)ocn3)CC2)=O)C(C#N)C1(C)C O=C1CC(C(=O)NC2CCN(C(C3CCCC3C3CC3)=O)CC2O)=NN1 c1(C(N2CC(O)(CNC(C(CC)C)=O)C2)=O)cc2sc(S(N)(=O)=O)cc2s1 Cc1ccc(C(=O)NC2(CN(C)C)CN(C(=O)Cc3c(C)noc3Cl)C2)cc1C C=CC(C)(C)C(=O)N1CC(NC(=O)C=Cc2cocn2)C(n2ccnn2)C1 c1(CNC(=O)CC2CC2)ccc(C(F)C(F)(F)F)cc1 c1(CC(=O)N(CC(C)(C)CNC2CC2)C)ccnc(Br)c1.n1(CC=O)cccn1 C1(NC(CCC(=O)NC)=O)CCN(C(=O)Cc2n[nH]c(=NC)s2)CC1F CC(CC(N)=O)C(=O)NC1(C2CN(C(=O)CCn3cnc(=N)[nH]3)C2)CC1 c1(CC)noc(CC)c1C(CCSC)C(=O)Nc1csnn1.C1C(C2CC2)N1C C1(C)(C(=O)NC2C(N(C(=O)CC3CC3C(F)(F)F)C)COC2)CC2CCC1O2 c1(SC)ccc(Cl)c(C(N2CCCC(C)(NC(c3ccnn3C)=O)C2)=O)c1 N1(C(C(CC)OC)=O)CCC(c2n[nH]c(=N)o2)CC1 c1(C(N(CC(=O)NCC2CC(C(N)=O)C2)CC)=O)csnc1Cl CN1CCC(C)(CNC(=O)C(C)(CO)NC(c2ccon2)=O)C1 c1(N2CC3(CCN(C(CCC(C)SC)=O)C3)C2)cnc(C#N)c(C#N)n1 C(=O)(C1CCc2cc(F)ccc21)N(C)CCN1CCN(C(C2CCO2)=O)CC1 N1(C(C(COCC)C)=O)CCCC1(C)CNC(c1cncc(-n2cccc2)c1)=O CC1CN(C(=O)CC2CCSCC2)CC(C)N(C(C2CCC(F)C2)=O)C1 Cc1c(C(=O)NCC(CC(=O)N(C2CCC2(C)C)C)C2CCC2)nnn1C C1(F)(CNC(CC2(C)CCC2)=O)CN(C(C2(CO)CCCO2)=O)C1 c1(C(N2CCC(C)(CCNC(CN(C3CC3)CC)=O)C2)=O)ncn2c1CCC2 C1(C(C)C)CN(C(C23CC(C)C2C3)=O)CCN1C(=O)CC1(c2ccccc2)CC1 C1(C(=O)NCC(C)(CNC(=O)Cc2ccoc2C)OC)CCCCC1O N1(C(C2CN(C)C(=O)N2)=O)CC2(CCC(CNC(=O)CC3CCN(C)C3=O)O2)C1 c1(OCC(=O)NC(CNC(C(CC)COC)=O)(C)C2CCC2)ccc(C)c(C)c1 c1(CC)ccnc(C(C)NC(c2sc(COC)nc2Cl)=O)c1 C1(CCNC(c2cnc(CC)o2)=O)CCCN(C(c2ocnc2C(C)C)=O)C1 c1(OCC)ccc(N)c(C(=O)NCCN(CCC(C)O)C(C2(C)CCOC2)=O)c1 N1(C(C(C)CC2CCC2)=O)CC2(CCN2C(=O)CCCC2CCCC(=O)N2)C1 Cc1nc(C(=O)NC2(C(=O)NCC(O)C3(Cl)CC3)CCCC2)c(C)o1 C1(C(=O)NC2C(CNC(=O)Cc3cccc(O)c3)CCC2)CCC(F)(F)CC1 N1(C(Cc2cc(OC)c(Cl)cc2)=O)CCC2CCN(C(=O)C(O)CC(C)C)C2C1 C1(CCNC(c2ncc(C)cn2)=O)C(C)CCCN1C(=O)CCCn1ccnn1 c1(C(=O)NCC2CC(O)CN2C(C2CC2C2CC2)=O)cnc2ncccc2c1 C(=O)(CC1COc2ccccc21)NCC(CN(C(=O)C#CC1(CO)CC1)C)O N1(C(c2c(C)nc(CO)s2)=O)CCC(N(C)CCO)C(F)C1.C(=O)(CC(C)CN(C)C)N C1(C(N2CC(OC)CC(CC)C2)C(=O)NCC(F)F)CCn2cncc2C1 N(C(=NCCc1ccccn1)NCCc1cccc(C)c1)C(C(COC)C)C N1(C(c2cnc(C)[nH]2)=O)CCC(C(C)NC(c2ccc(=N)[nH]n2)=O)CC1 N1(C(C(CC)O)=O)CCCC2(CCCN2C(c2ncc(C)cc2C)=O)C1 c1(CCCC)nc(-c2ccc(OCC(C)C)cc2)n(C2CCCC(C)C2)n1 N1(C(C2(C)CCOCC2)=O)CC2(C(N3CCOC(C(C)(C)C)C3)=O)CC1CO2 c1(C(=O)NC2C(CNC(CCCCNC(N)=O)=O)CC2)cnn2c1OCC(F)C2 C1(OC)CN(C(=O)C(=O)NC2CC2)CC1C(=O)NCC1CCCC1OC CCCCC(O)C(C)C(=O)NNC(=O)c1cc(C(=O)OC)cc(N)c1 C1(C(=O)NCCC#C)CCN(C(c2cnn3c2OCC3)=O)C(CC)C1 c1(CC(=O)N(CC(CC)NC(c2occc2C)=O)C)cccc(C)c1Br N1(C(C=CCN(C)C(C2CC2C2CCCO2)=O)=O)CCCCC1CCCO Cc1nc2c(C(=O)NC(CNC(=O)CC3CCCCC3)CC(C)C)cccc2o1 c1(C2(C(=O)NCCCN(C(=O)C(C)CF)CC)CC2)ccc(Br)cn1 C1(NC(CCOCCC)=O)CC2CCC(C1)N2C(=O)CCc1nnc(C(C)C)o1 C1(C(N(C2CCN(C(c3c[nH]cc3Br)=O)C2)C)=O)CCCCC(C)(C)C1 c1(C(N2C3CC(CNC(C4CN(C(C)=O)C4)=O)C2CC3)=O)cc2ccncc2[nH]1 Cc1csc(C(=O)NCc2nnn(C)c2C(=O)NCC2CCOC2C)c1C C1(NC(C2C(C(C)C)CCC2)=O)CC2CC1CN(C(c1cnsn1)=O)C2 C1(C(=O)NCCOCC(=O)NCc2ccc(F)cc2F)CCC2(CC1)CC2(F)F C1(NC(c2cncc(C)c2)=O)CN(C(=O)CC2(O)COC(C)(C)C2)CC12CC2 N1(C(c2ccc(C)s2)=O)CCCC(C(=O)NCCc2ccccc2)C1 C1(c2nnnn2C)(NCc2c(C)ncnc2C)CCC2(CC1)COC(C)(C)C2 N1(C(C2CCC(C)O2)=O)CC(NC(c2csc(-c3ncc[nH]3)n2)=O)CC1C C1(CCC)CN2CC1CC1(CC2=O)CC1.c1(SC(=O)OC)ccccc1 C(=O)(CC1=CCN(C)CC1)NCC(CC=C)C(=O)NC(C)CCCN=[N+]=[N-] C1(NC(C(CC#CC)NC(=O)CCc2nc(O)n[nH]2)=O)CC=C(C(C)C)CC1 C1(O)(CNC(CN(C(CCOC)=O)C)=O)CCN(C(C2CC2Br)=O)C1 c1(C(N2CCC(NC(CC3CC(OCC)C3)=O)C2)=O)n[nH]c(CC)c1C C1(N(C(C(=O)OCC)CCSC)CCOC(F)(F)C(F)(F)F)CC2(CCC2)CO1 C1(CNC(C2(C)CCOC2)=O)CN(C(=O)CC2CCCSC2)CC1(C)C CC1(C)CCCCC1=CC(=O)NCCCNC(=O)Cc1cnccc1C(=O)O C1(CNC(c2c(C)cncc2)=O)CCN(C(C2CN(C)C(=O)N2)=O)CC1C Cc1ccc(C(=O)NCCC(O)CNC(C2CCS(=O)CC2)=O)nn1 C(=O)(C(O)C(C)(C)CC)N(CC(N1CCCN(CCC)CC1)=O)C CC1CC(C)CN(CCC(=O)N(O)Cn2cc(CCN(C)C)cn2)C1 CC1=NOC(C(=O)NC2CN(C(C)C)CC2N2CCCC2)C1C N1(c2cc(C#N)cc(Cl)n2)CCc2sc(-c3ccc(OC(F)(F)F)cc3)nc2C1 C(=O)(CC(C)(C)CNC(=O)CC(O)C(C)C)N(C1CCN(C)C1)CC N1(C(c2cccc(CNC(N)=O)c2)=O)CC(NC(=O)CCC2CCOC2)CC(F)C1 c1(NCC2(C)CC2)ncccc1S(=O)(=O)NCC1CCC(=O)NC1 N1(C(C2C(C)N(C(c3nn(C)cc3Cl)=O)CC2)=O)CCC(F)(C#N)C1 C1(C2CCCO2)(C(=O)NOCc2cn(CC3COC(=O)C3)nn2)CCCO1 N1(C(c2n(CC#C)ccn2)C(=O)NCCOC)CC(C)=CC(C)C1 C(=O)(C(C)(F)C(=O)NCC(C1CCCC1)NC(c1cnccc1C)=O)OC c1(C(=O)NC(n2ccc(-c3c[nH]nn3)n2)CC)cccnc1OCC.CC(C)C C(=O)(C(C)(C)C(F)F)NCC(CCOC)NC(=O)CCc1ccncc1 C(=O)(C(O)CC[S+](C)C)N(CCCNC(c1ccnn1CC(F)(F)F)=O)C C1(CNC(C(=O)Nc2ccc(Br)cc2Cl)=O)CCC2(CCC2)N1 CC1(CNC(=O)CC2CC=CCC2)CCN(C(C2CCCCS2)=O)CC1 c1(NC(=O)NC2CC(c3n[nH]c4ccc(Cl)cc34)C2)ncnc2[nH]c(Br)nc12 C(=O)(C(CNC(c1c[nH]nc1CC)=O)CC(C)C)NC(CCC)C(=O)NC Cc1nc(CO)ncc1C(=O)NCC1(F)CCC(CNC(C2CCC2C)=O)CC1 C1(NC(CC2C(C)OCC2)=O)CC=C(C(=O)N2CCN(CC(N)=O)CC2)C1 C1(C(N(CCNC(c2n(C)ncc2)=O)C2CC2)=O)CC2CCC(C1)N2C1CC1 C1(CC=C)(NC(=O)CSC(F)(F)F)CCN(C(C2CC=CCC2C)=O)C1 C1(CNC(C(=O)N(C(CC)C(=O)NO)CC)=O)CCCOC1c1cn(C)nn1 C1(C(=O)NCC(C(C)C)NC(=O)CCc2cnn(C)c2)CN2CCN1CC2 c1(OC)cc(C)ccc1C(=O)Nc1nc(C)ccc1CO c1(NCC2(OC)CCCSC2)nccc(=NC(C)c2cncc(F)c2)[nH]1 c1(C(N2CCCCC(NC(C3C(C)(C)CCC3)=O)C2)=O)ccnc2cc[nH]c12 C[Si](C)(C)C1(C(N2C(C(=O)NCC(O)C(F)F)CCC2C2CC2)=O)CC1 c1(CC(=O)NCC23CC(NCc4cnc(OCC)s4)(C2)C3)nnc2n1CCCC2 C1(CNC(C(N2CCSCC2)C)=O)CN(C(=O)CCC(F)F)C2(CCOCC2)C1 C(CN=c1[nH]c2c(cc1C#N)c(C)nn2C)(C1CC1)NC(C1C(C)=C1)=O C(c1c(F)cccc1F)=CC(=O)NC1COCCC1NC(C1CC12CCC2)=O.C(O)CF c1(C(N2C(c3cn(CC)nc3)CCC2)C(=O)NC2CC2)cc2c(Cl)cccc2s1 CS(=O)(=O)c1ccc(CNC(c2ccc(N3CCNC3=O)cc2)=O)cc1Cl C1(C(=O)NCC2(F)CC(NC(c3ccon3)=O)C2)CCS(=O)(=O)C1 c1(C(N2C(CNC(C(C)OCC#C)=O)CN(C)CC2)=O)cc2ncc(C)cn2n1 CCC(CC(=O)NCc1nc(C(=O)NC(C2CCCC2)CO)c(C)o1)C(F)F C1(C(=O)NC(C(C)NC(CCCOCC)=O)C)(OC)CCC(F)(F)CC1 CCC(CCCC(=O)N(C)CCc1cccnc1)NC(c1cc(C2CC2)no1)=O CCC(CO)C(=O)N1CCN(CC2CCCN(C(C3CC(=C(F)F)C3)=O)C2)CC1 C1(S(C)(=O)=O)(C(=O)NCC(C2CC2)NC(CC(C(=C)C)OCC)=O)CCCC1 C#CCCCCCC(=O)NC(c1nc(C(=O)NCC2(OCC)CCC2)co1)C C(CCCCCC(=O)N(CC1CC1)CC1CC1)NC(c1nn(C)c(=O)cc1)=O c1(N(CCN(C)CCO)C)ncc(S(=O)(=O)NC2(C)CC3(CCC3)C2)cc1Cl N1(C(CCCC=C)=O)CCC2CN(C(c3ccccc3Br)=O)CC12 c1(CCC(=O)NCC(C)CNC(=O)C(C)C2(O)CCC2)nnc(C(F)F)o1 CC(C(=O)Nc1cccc(NC(c2cc(C3CC3)on2)=O)c1)C(F)F Cn1cnc2nc(N3CCCC(OCCO)C3)nc(NCCCCC(F)(F)F)c12 C=CCC(CC)N=c1[nH]c2c(c(=NCC3OCCOC3(C)C)[nH]1)SCC2 c1(NC(C2CC(NC(CNC(=O)OCC)=O)CC(C)C2)=O)ccc2nncn2c1 C1(CC)C(NC(=O)C(n2cc(C)cn2)C)CCCN1C(c1ccccc1Cl)=O C1(O)(C(=O)NCCOCCCN(C(=O)C(O)c2cnc[nH]2)C)CCCC(C)(C)C1 c1(C(=O)NC2CCCN(c3nc(C4CC4)ns3)CC2)cccn2nncc12 c1(OCC(=O)N(CCC)CCNC2(C(=O)N(C)C)CC(O)C2)c(F)cccc1F C12(CNC(CNC(=O)NC)=O)CCC(CC1)CN2C(=O)Cc1cccc(O)c1 c1(OCC)cc(C(F)(F)F)n[nH]c1=NC(=O)Cn1cnc([N+](=O)[O-])c1 C1(C)(C(N2CCC(C(CNC(CC(=O)N(C)C)=O)(C)C)C2)=O)CS(=O)(=O)C1 c1(C(C)C)ccc(S(=O)(=O)N(C2CC3CC2CN3)Cc2ncon2)cc1 Cc1c(C=CC(=O)NCC23CCC(CC2)N3C(C2CCSC2)=O)cnn1C N1(C(CCNC(c2cc(C(=O)OC)n[nH]2)=O)=O)CC2(CCCN(CCOC)C2)C1 C(=O)(C1=C2CCCN=C2NN1)N1C(C)CC(CNC(CCC(=O)NCC)=O)C1 N1(C(Cc2cc(OC)no2)=O)CCC2(CC1)CN(C(=O)CCN1CCC1)C2C(C)C CCC(C(=O)NC1CC=C(C(=O)N2CC3(C2)CN(C(C)=O)C3)C1)C(C)(C)CC N1(C(C=CCC)=O)CCOCC(NC(=O)C(Cc2ccccc2)C2CC2)C1 N1(CCOC)CCC(N=c2[nH]c(=NCCc3nnc(C)s3)c3sccc3[nH]2)CC1 C(=O)(C(CC(F)(F)F)c1cccc(F)c1)NC1N(C(C(C)CC2CCCC2)=O)CC1 O=C1CCCC(C(=O)NC(CC2CC2)C(=O)NC2CCNC(=O)CC2)CC1 C1(C(=O)NCC2CCN(C)C2=O)C2CCCC1CN(C(c1nocc1Cl)=O)C2 c1(NCCC(C(F)(F)F)OC(C)(C)C)ccc2oc(O)nc2c1 Cn1nnc2c(C(=O)NC3(CCNC(=O)C(F)=C4CCC4)CC3)cccc12 c1(N(CC(CC)(C)OC)C)ncc(C)cc1S(=O)(=O)NCCc1ccc(C)cc1 c1(C(=O)NC(C2(O)CN(C(c3cc(C)ns3)=O)C2)C)cnc2n1CCCC2C C(=O)(C1=Cc2cc(F)ccc2OC1)N(CC(C)CNC(=O)CC(C)(C)C)C Cc1ccoc1C(=O)NC(C1CCCC1C(=O)O)C c1(CNC(CC#N)=O)ccc(N2CCN(C(=O)Cc3cscc3Br)CC2)cc1 c1(OC)cccnc1C(N1CC=CC(NC(c2cccc(C3CCC3)c2)=O)C1)=O C12(NC(C(Br)=C(C)C)=O)COC(C1)C(NC(c1scnc1C1CC1)=O)C2 c1(CSCC(=O)N(C(C2CC2)=O)CC2COC(C3CNC3)C2)ccccc1 C1(O)(CNC(CC2C(C)(C)CC2)=O)CCCN(C(c2ccc(C3CC3)cn2)=O)C1 C1(C)(NC(c2oc(C)c(Br)c2)=O)CCCN(C(C2Cc3nccn3C2)=O)C1 N1(C(C(CC(C)C)N)=O)CC2(CCC2)OC2(CCC2)C1 N1(C(CCc2c(C)ncs2)=O)C2CCCC1CN(C(=O)C(O)C(C)(C)C)CC2 C1CN=C(NCC(C)(F)F)N1.c1(C)ccc(N2CCOCC2)c(Cl)c1.CCS N1(C(c2nc(COC)oc2)=O)CC(C(=O)NCCN(CC(C)O)C)CC(C)(C)C1 c1(CC)cc(F)c(C(=O)NCC2CC2CNC(=O)Cc2nc(=N)[nH][nH]2)c(F)c1 Cc1ncc(C(=O)NCC(C)CC(=O)NCCC(F)CN=[N+]=[N-])c(C)n1 c1(C2(C(=O)NC3C(CNC(=O)Cn4nc(Cl)ccc4=O)C3)CC2)ccc(Cl)c(Cl)c1 n1(CC(F)F)nnnc1C(C1CC(n2cncn2)C1)NCC1(C(F)(F)F)CC1 N1(C(CC2(OC)CCC2)=O)CC2CC1(CNC(=O)CSc1c(C)n[nH]c1C)C2 C(=O)(CC(C)CC(F)(F)F)NC(CNC(c1c(C#C)cnn1C)=O)(C)CO Cn1cnnc1CCCC(=O)NCC(O)CNC(C1(C)CC1(F)F)=O N1(C(=O)CCN(CC(=O)NC(C)C)C)CCC(CNC(=O)CCCC2CC2)C1 c1(C(=O)NCCC(C)CCNC(=O)CC(C)(C)C#N)ccc2ncccc2n1 c1(C(N(CCCNC(C=CC)=O)Cc2ccccc2)=O)c(C)ccc(Cl)c1F c1(C(=O)NC23CC2CN(C(=O)CCCN2CCCC2)C3)cc(Cl)ccc1Cl c1(NCC=C(C)C)[nH]c(=NCC2CCCC(F)C2)nc2c1ncn2C CC(C)CC(C(=O)N1CC(C)C(NC(=O)CCNC(=O)OC(C)C)C(C)C1)C(C)C Cc1ncc2n1CC(C(N1CC(NC(=O)Cc3cn[nH]c3)C3(CCC3)C1)=O)CC2 c1(OC)cc(CCC(N2CC(F)(CNC(c3ocnc3C)=O)C2)=O)ccc1O c1(OC)cc(O)cc(CN2CCOCC2CC(=O)Nc2nc(O)nc(O)n2)c1O C1(NC(C(CC)n2nccc2C)=O)CCOCC1NC(c1ccccn1)=O Cc1cc(NC(c2ccc(COc3ccccc3)[nH]2)=O)cc(C)c1F N1(C(=O)NC(CCCCCO)C2CC2)CCc2ccc(Br)cc2C1C(F)F c1(C(N(CCN(C(C2(CCC)CC2)=O)C)C(C)C)=O)ccnn1C(F)F N1(CC(=O)N(C2CCN(C(c3ncn(CC)c3)=O)C2)C)CCN(C)C(=O)C1 C1(C(=O)NCC(C)NC(c2ccc(F)nc2)=O)CC1C1CCCCC1 C1(OC)CCN(C(c2cc(CNC(=O)C(F)OC(F)(F)F)[nH]n2)=O)CC1(C)C c1(OCC)cc(NC2CCCC2NC(=O)CN(C2CCSC2)C)ccc1[N+](=O)[O-] N1(C(C(CCC)N(C)C)=O)CC2(CC(CNC(=O)CC(C)N3CCCC3=O)C2)C1 C1(C(=O)NCC2CN(C3C(C)C3)C2)CN(C(=O)CSC(F)F)CC1(C)C C1(NC(c2c(C)noc2C)=O)Cc2ccccc2N(C(=O)CCc2ncc[nH]2)C1 C1(NC(C(N)Cc2ccc(Cl)cc2F)=O)Cc2ccc(Br)cc2C1 C1(NC(CN(CC(=O)NC(C)C)C)=O)(NC(=O)CN2CC=CC2)CC(F)(F)C1 N1(C(c2nc(C)nc(O)c2)=O)CCN(C(=O)CSC(F)(F)F)C2COCC12 N1(C(CN(C)CC)=O)CCN(C(c2cc(OC)ncn2)=O)CC1CC(C)(C)C c1(CC(=O)NC2CCN(C(C(CSC)O)=O)C2)ccccc1NC(C)=O C(=O)(CC(C)(C)C(F)F)NCCC1N(C(C2N(C)CC(O)CC2)=O)CCCC1 C1(NC(c2cccc(CC)n2)=O)CN(C(=O)CC2CC(C)(C)CO2)CC12CCC2 Nc1cc(-c2cccc(C3CC3OCC(N3CC(F)(F)C3)=O)c2)c(F)cc1F N1(C(c2[nH]cnc2-c2cccnc2)=O)CC2OCC(C(N3CC4CC4C3)=O)C2C1 c1(C(C(=O)NC)N(C2CC(F)(F)C2)C)ccnc(NC(C2CCN(CC)C2)=O)c1 N(C1CCc2cccnc21)C(CC1C(NC(CCNC(=O)NC)=O)CCC1)=O c1(N(CC(C)C)C)ccc(C(=O)NC2COCCC2NC(C2(F)CC2C)=O)cn1 C1(C(=O)OCC2CCC(C(F)F)CC2)CC12CCS(=O)(=O)CC2 N1(C(C2(SC)CC2)=O)CC(CO)C2(CCN(C(=O)CC3CCCC3)CC2)C1 O=C1CCN(Cc2ccc3occc3c2)C(=O)N1Cc1cc2c(s1)CCCC2 C1(OC)CC(CNC(=O)Cc2cc(C)cs2)N(C(=O)C(=Cc2cnc(C)s2)F)C1 c1(CC)oc(C(=O)NC(CNC(C2(c3cc(C)no3)CC2)=O)CO)cc1C c1(C(CC(=O)NC(C)CNC(C2CS(=O)(=O)C2)=O)C2CC2)ccccc1[N+](=O)[O-] C(C(C)(C)C(=O)NCc1cncc(C(=O)NC2CCOCC2)c1)NC(C)=O CC(C)CC(C)C(=O)NCCCC(=O)NC1(c2ccnn2C)CC1 N1(CC(c2ccccc2)Nc2c(C(=O)OC)cnn2C)CCCCCC1C C(C1=CCN(C(c2conc2C(C)NC(=O)C(=Cc2ccco2)C)=O)CC1)OC N1(C(c2ccc(CC)cc2C)=O)CCC2CCN(C(=O)C(CC(C)C)OC)C2C1 CC(C)CC(C(=O)NCC1CCCC1NC(=O)CCN(C)C)c1ccc(Cl)cc1 C(CC(C)(C)CC(=O)NC1CCCC1C(=O)NC12CC(C)(C1)C2)OC c1(CC)noc(CCC(=O)NCCC2(O)CCC2)n1.C12(CCO)CN(C1)C2=O N1(C(C2(C#C)CCC2)=O)CCC2(CCCCC2NC(c2cncc(SC)c2)=O)C1 CC(C)C(CC(=O)N1CC(NC(c2cccc3sccc23)=O)CC(O)C1)C(C)C CN=c1nc(N2CCCC2)[nH]c(=NCc2ccc(Br)o2)[nH]1.C(CC#N)NC C1(NC(CC=CC)=O)CCCC12CCN(C(c1cccn1CC)=O)C2 c1(OC)cc(C(N2CC3CC(NC(c4cscn4)=O)C2C3)=O)cc2cn(C)nc12 Cc1ncoc1C(=O)NCC(C)CNC(=O)C(=O)NCC1CC1 c1(C(=O)NCC2(CN(C(C3CC(C)OC3)=O)C)CC2)cc2ccsc2s1 c1(C(N(CC(C)NC(=O)CCc2ccccc2)C)=O)cc(F)cc(F)c1O c1(C(N2C(CNC(c3cn(CC=C)nn3)=O)C=CC2)=O)cc2c(cn1)OCCO2 c1(CC)oc(C(N2CCC(C(=O)NC(c3cccn3CC)C)C2CC)=O)cc1C CCCC(O)CC(=O)NC1(C2CCCN2C(=O)C=Cc2cc(C)no2)CC1 N1(C(CCN(C(CN(C(=O)OCC)C)=O)C)=O)CCCN2CCCC2C1 C(=O)(CCC(C)CC)N(CCN(C(c1nc(CC)oc1)=O)C(C)C)C Cc1ccc2c(C(=O)NCC3C(C)CCCN3C(=O)COCCF)c[nH]c2c1 C#CCCCCCCC(=O)NC(C(=O)NCC12CCCC(CO1)C2)C(C)C C1(O)(CNC(C2(CC#C)CCC2)=O)CCN(C(C2(CF)CCC2)=O)C1 C1(CNC(C2(CC)CC2)=O)CCN(C(c2scc(C)c2C)=O)C1(C)C C=CC(C)(CC)C(=O)NCCCOCCCNC(c1conc1CC)=O C1(CNC(C(CC)OC)=O)CN(C(c2cncc(NC)c2)=O)CCC1(C)C c1(NC(C(=O)N(CCCC(N2CCN(C(C)(C)C)CC2)=O)C)=O)ccc(Cl)cc1O c1(SCC)cncc(C(=O)NC(CNC(=O)Cc2cccc(Cl)c2)C2CCC2)n1 c1(C(=O)NC(CCCC)CNC(=O)CCSC)cnc(C)nc1OC c1(C(=O)NCC(CC)NC(=O)CSc2cccc(C)c2)ccc(C(F)(F)F)cn1 c1(C(N2CCC(CNC(CCCc3onc(CC)n3)=O)C2)=O)ncc(N)cc1Cl N1(C(C2C(C(=O)OCC)C2)=O)CCN(C(=O)CCF)CC1 N1(C(CCN(CC)CC)=O)CC2(CC2)CC1CNC(=O)CCC1CCOC1 C1(C(N2C(C#C)CC2)=O)CSCCN1C(C1CCCCN1C)=O c1(NC2CCN(c3c(C(=O)OC)ccs3)C2=O)cc(Cl)ncc1F c1(CCC(N2CC(N(C)C(c3n[nH]cc3F)=O)C2)=O)ccc(Br)cc1 Cc1ccc(O)c(CN2CCC(N(C(=O)C(CO)c3ccccc3)C)CC2)c1 N1(C(C2(C(C)C)CCCO2)=O)CC2(CC(NC(=O)CC(O)CN(C)C)CO2)C1 c1(NC23CC(C(=O)NCc4ccc(F)cc4)(C2)C3)cc2cc[nH]c2cn1 C(=O)(C1CCCn2ccnc21)N1CC2C(CNC(=O)CC3CCC3)(CC2)C1 N1(C(C2C(CCC)C2)=O)CCC(F)(CNC(c2cnn(C(C)C)c2)=O)C1 c1(C(=O)NCC2(O)CC(C(=O)NCC(=C)Cl)C2)cccn(C)c1=O C(C)(C)(CCCC(=O)NC(Cc1ccccc1)CCO)C(C(C)C)C(=O)N(C)C c1(C(N2CC(C)C(CNC(=O)COc3cccnc3)C2)=O)ccc2c(n1)CCO2 CC1CC(CC(=O)N(CC(=O)N(C)C)C2CC2c2ccccc2)C(C)O1 N1(C(C(=O)N(CC(c2ccoc2)C)C2CC2)=O)CCCC2(CC=CCO2)CC1 c1(C(=O)NC2CN(C(C3C(CCOC)C3)=O)CC2C)ccc2ncc(=O)[nH]c2c1 C1(C(N(CCNC(CCC=C)=O)CC)=O)CN(C(=O)CC(C)(C)C)CCO1 n1(CC(=O)NC2CC(C)(C)N(C(=O)C=CC(F)(F)F)C2)ncn2nccc2c1=O c1(C(=O)NCC2(F)CCC(NC(COCC#C)=O)C2)c(C)ccc(C)c1C CCC(CCCC(=O)N(C1(C)CC2C=CC1C2)C)NC(c1cccn(C)c1=O)=O N1(C(C(C)N(C)CC)=O)CCC2(CCCC2NC(c2cc(C)cc(C)n2)=O)CC1 C(CC(O)C(=O)NC1CC(CCNC(c2onc(C)c2C)=O)C1)SC C(=O)(C(C)CNC(=O)C(C)=CCNC(c1cc(C)cs1)=O)NC CCCCCCC(C)(CCC)C(=O)NCC(CCOC)NC(c1nn[nH]c1Cl)=O S(=O)(=O)(c1cnc(NCCS(=O)(=O)C2CC2)c(Cl)c1)NC1C(CC)CCCC1 C1(CC)C(=O)NCCCN1C(=O)C(Cn1cncn1)NC(=O)CCc1cnoc1 C(c1ccccc1)=C(C(N1CCC(C(C)NC(=O)NC2(CF)CCC2)C1)=O)OC C12(CNC(C(CC)C)=O)CC(NC(=O)CC(C)C)(C1)C(C)(C)O2 c1(C(=O)NCC(C)(C2CC2)NC(c2cnc(C3CC3)[nH]2)=O)sccc1C1CCC1 CC(C)(C)C#CC(=O)N1CCC(NC(c2cc3c([nH]2)CCC3)=O)CC1C N(C(=NCCCN(C)C(=O)N(C)CC)NC1CCC1)CC#CC c1(C(=O)NCC(CNC(C2CCC(CCCC)CC2)=O)C)ccnc2ccnn12 CC(C)(C)CC(O)CNC(c1coc(CNC(c2ccccc2)=O)n1)=O CC1CC(NC(=O)CN2CCCNS2(=O)=O)CCN1C(c1cncc(O)c1Cl)=O C1(SC)CCN(C(=O)CC2CCCCN2C(=O)C(C2CCCCC2)C)CC1 C1(C(=O)NCCN(CC(C)O)C(c2cc(CN(C)C)c[nH]2)=O)CSCC(=O)N1 CCC(C)CCCC(=O)N1CC2C(CNC(c3cc(C)ncc3C)=O)C2C1 c1(-n2c(-c3ccc(Br)nc3)ncn2)nc2ccccc2n1C.Cn1cncc1C c1(C(N(CC(C)OC)C(C)C)=O)cc(N2CCCC2)cc(C)c1 c1(C(N2C(CN(C(C3(CSC)CC3)=O)C)CCCC2)=O)cc(C)ccc1C CCCCCC(O)C(=O)NCC#CCNC(c1ccc(NC=O)cc1)=O C(CCN=c1[nH]c(=NCCn2cnc3sccc3c2=O)[nH]c2c1CSC2)OC N1(C(CNC(N)=O)=O)CCC2CN(C(=O)C3=CCC(F)(F)CC3)CCC2C1 CCC(C)CN=c1nc2ncn(C)c2c(NCc2c(S(C)(=O)=O)cnn2C)[nH]1 C(N=c1[nH]ccc(C#N)c1[N+](=O)[O-])C1CC(NC(COc2cccc(C)c2)=O)C1 N1(C(C2(C)N(C(CC=C(C)C)=O)CC=C2)=O)CCC2C(C(N)=O)C2C1 c1(C(N2CC(CNC(CC=CC=C)=O)C(C)C2)=O)c(F)ccc(F)c1OC C=CC(C)(C)C(=O)N1CCC(C2CCCN2C(=O)C(C)(C)COCC(F)F)C1 C1(CN(C)C(C2CC(c3ccc(Cl)cc3)(O)C2)=O)CCCN(C(C2(Cl)CC2)=O)C1 Cn1cnc2ccc(C(N3CCC(Cn4cc(C5(C)CCCO5)nn4)C3)=O)cc12 C1(OC)CN(C(c2cncc(N)n2)=O)CC1NC(C1(C(F)F)CC(F)(F)C1)=O Cc1c(C(N2CC(NC(=O)CCCN=[N+]=[N-])C(C3CC3)C2)=O)ccc(F)c1F C1(CCOC)CN(C(=O)C=C2CCSCC2)CCN1C(c1cnc(O)n1C)=O CCCC(C(=O)NCC(CCOC)NC(C1(SC)CC1)=O)S(N)(=O)=O.NCC C1(CC(=O)NC2(C)CN(C(C3CCOC3)=O)C2)CC2CCC1CC2 Cc1ccc(C(C)(C)CNC(=O)NC(c2ccccc2)c2ccncc2)nc1 N1(C(C2CCC(C)CC2)=O)CCCC2CN(C(c3csc(C(F)F)n3)=O)CCC12 C1(O)(CN(C(C(C)Cc2ccccc2)=O)C)CCN(C(=O)CCOCC2CC2)C1 N1(C(C(C)OC(C)C)=O)CC(C(N2CCC3(CCC3)CC2)=O)CC12CCC2 C=CCC(C(=O)NCC1(C(N2CCC2C(C)C)=O)CC=CC1)C(C)C O=C1CCC(C(=O)OCCc2nc(-c3ccccc3)no2)CN1 n1(CCCC)nnnc1C(C(C)(C)N(CC)CC)NCCCC1CC1 C(CNC(=O)CC(C)SC)(C(C)(C)C)NC(C(CC)n1cccn1)=O C(=O)(CCCC(=O)NC1CC(F)CN1c1ccnc(C2CCCC2)n1)N(C)C C1(C)(CNC(CCCOC)=O)CN(C(=O)C(C)C2=CCCC2)C(C)(C)C1 c1(CNC(CC#C)C(=O)O)ccc2c(c1)CC(C)(C)O2 CC1CN(C(=O)CCCOc2ccc(F)cc2)CC1NC(=O)C(C)NC(N)=O Cc1cc(C(=O)NCC2CN(C(=O)CC3CCC(=O)NC3)CC2(C)C)nc(C)n1 N1(C(C(C)c2ccsc2)=O)CC2CC2(CN2CCOCC2)C1.C12CC1CNC2=O c1(C2C(CNC(CC=C)=O)C2)cccc(Br)c1C.C12CCCN1C(=O)C21CC1 c1(C(N2CC=C(CNC(C=C(CCN(C)C)Cl)=O)CC2)=O)ccsc1S(N)(=O)=O N1(C(C2(OC)CCSC2)=O)CCN(CCOCCCN2CCNC2=O)CC1 C1(NC(C2C(C)CC2)=O)CCCC(C(=O)N(C)Cc2ncnn2C)CC1 CC1(C)CC(C(=O)NC2CN(C(c3cccnc3N)=O)CC2F)CCO1 C1(OC)CCC2(C(=O)NCC3CCCN(C(=O)C=C(Cl)Cl)C3)CCC12 Cn1ccc2nc(N(C3CC(N)C3)C(C3CNC(=O)C3)=O)ncc12 CCCCCC(O)C(=O)NC12COC(CNC(c3cc(C(F)F)cs3)=O)(C1)C2 N1(C(C=C(CCC)C)=O)C2CCC1CN(C(=O)C(C)(F)CCCC)C2 C1(CC(N2CC(C3(NC(C4=NOC(C)C4)=O)CC3)C2)=O)CC(c2ccccc2)=NO1 C1(CNC(CC(C)O)=O)CC(C)N(C(=O)CNC(c2ccccc2)=O)C1 C1(CC(=O)NC(c2nc(C(C)C)[nH]n2)C)CC2(CCOCC2)O1 CC(C(=O)N1CCC(C)(CNC(c2cnn[nH]2)=O)C1)C(C)(C)O Cn1cc([N+](=O)[O-])cc1C(N1CC2CC1C2NC(=O)CN1CCCCCC1=O)=O N1(C(COCC(C)C)=O)CC(NC(c2ccc(Cl)c(Cl)c2)=O)CC1(C)C c1(C(=O)NC2CC3(C2)CN(C(c2ccnc(Cl)c2Cl)=O)C3)cnc(Cl)c(F)c1 C1(CC(=O)NC2CCC(NC(C3CC(F)C3)=O)C2)(COC)CCCC1 N1(C(c2c(C)nn[nH]2)=O)CCCCC2(C1)CN(C(=O)C1CCc3c[nH]nc31)C2 O=C(C1CCc2c[nH]nc21)NC1CC2(C1)CC2C(=O)NCC1(CCCO)CC1 N1(C(C(C)SCCCC)=O)CCCN(CCNC(=O)COCCF)CC1 c1(NC(=O)CCC2CC(NC(c3cccc(Cl)n3)=O)C2)cc(F)cc(F)c1 N1(CCC(C)(C)C#N)CCC2(CC1)CC(n1cc(C(=O)OCC#N)nn1)CCO2 c1(C(=O)NCC(C(=O)NC(C2CCOC2)C#C)(C)C)c(C)cccc1C Cc1oc(C)c(CNC(C2CCCN2c2ccc(Cl)cc2)=O)c1C C(=O)(C(F)(F)C(F)(F)C(F)(F)F)NC(C1CN(C(=O)CCOC2CCCC2)C1)C c1(C(N(CC(C)NC(c2c(SC)cccn2)=O)C)=O)cc(F)cc2nc[nH]c12 C1(NC(=O)Nc2cn(CS(C)(=O)=O)nc2)CC2CCC(C1)N2C(=O)OC(C)(C)C c1(CC(N2CCCCC(NC(C3C(C(N)=O)C3)=O)C2)=O)ccc([N+](=O)[O-])c(N)c1 C1(C(=O)NCC(c2nccs2)C)COC2(C1)CN(C(C1CN(C)CC(C)O1)=O)C2 N1(C(C(C)SCC)=O)CC(NC(=O)C(C)(C)COC(C)C)CC(O)C1 C(=O)(N=c1ccn(CC2CC2)[nH]1)C1C(CC)CCN1C(=O)C(CO)OC c1(NC(=O)NC(c2cccc(OC)c2)CC)cc(S(=O)(=O)N(C)C)ccc1F N1(C(CC)=O)CCC2(CC1)CC2CNC(=O)C(c1ncccc1C)(F)F C1(NC(CN(C)C(N)=O)=O)CC12CCC(NC(=O)CCn1ccnn1)CC2 c1(C(N2C(C#N)CN(Cc3cc(Br)ccc3Br)CC2)=O)cc([N+](=O)[O-])ccc1Cl CCCC(CC1CCCC1)C(=O)NCC1(C)CCCC1NC(=O)Cn1cccn1 C1(CNC(CN(C)CC)=O)CC2(CCN(C(C3COCCC3(F)F)=O)CC2)CO1 c1(C(NOCC(=C)Cl)=O)cn(CCNC(=O)Cc2cocn2)cn1 N1(C(CCOc2c(C)cccc2)=O)CCC(O)C(NC(C2CCC(=O)NC2)=O)C1 c1(C(=O)NC(C2CN(C(c3n(CC)ncn3)=O)C2)C)c(C)oc2ncnc(O)c12 S(=O)(=O)(c1ccc(Br)c(F)c1)N1C(C(=O)Nc2ccnnc2)CC(OC)C1 c1(C(N(CCN(C(c2ccc(OC)nc2)=O)C)C)=O)ccc2[nH]c(C)c(C)c2c1 c1(C(N(CCC)CCNC(C2CCC(C(=O)C3CC3)C2)=O)=O)cccc(F)c1 C(=O)(CCCCCNC(c1cnc(N)cn1)=O)N1CC(CC(C)(C)C)C1 C(=O)(C(O)CC(C)C)NC(CCC(=O)NC(CC=C)C(=O)NC)C N1(C(C2CCCO2)=O)CCOC2(CCN(C(C3(Cl)CC3(F)F)=O)C2)C1 C1(NC(C2C(C)N(C(C3CC4C(C3)C4(C)C)=O)CCC2)=O)CCC(=O)NC1(C)C C(=O)(CS(=O)(=O)C(C)C)NCC1(F)CCN(C(C2C(C(=O)OC)C2)=O)CC1 C(=O)(C1=COCCC1)NCCC(C)CCNC(c1ccc(C(N)=O)o1)=O c1(C2N(C(c3ccc(C)s3)C(=O)NCCOCC)CC2C)nncn1C CC1CN(C(=O)CCN(C(=O)C2=C(Cl)CCOC2)C)CC(C)(C)O1 c1(C(=O)NC2CC(NC(c3ccc(C)c(N)c3)=O)C2)cn2ccc(C)c(C)c2n1 C(=O)(C(CNC(c1cnc2ccccn12)=O)C(C)(C)C)N(CCCO)CCC Cc1nc(C(C)C)ncc1C(=O)NCC1(F)CC(NC(C2CCSC(C)C2)=O)C1 N#Cc1ncccc1N(C1CC2CNC1C2)C(=O)Cc1ccc(Br)c(F)c1 C1(CC(=O)NCC(N2CCN(C(C3(C)CCC3)=O)CC2)C)CCCC2(CCC2)O1 C1(NC(CCOCCC)=O)CN(C(c2ccc(F)c(C(C)C)c2)=O)CCC1F Cc1ccccc1C=CC(=O)NCCC(C)N(C(=O)C=Cc1cscn1)C Cc1ccc(Cl)c2[nH]c(C(N3CC(NC(=O)CC(C)CN(C)C)C(C)C3)=O)cc12 N#Cc1cnc2ccnn2c1C(=O)N(c1ncc2[nH]cc(I)c2n1)C1CNC1 N1(C(C(C=CC)O)=O)CC2(CCCN(C(=O)CNC(=O)CNC(C)=O)C2)C1 c1(C(N(C2CC(NC(=O)C(F)CC3CCCC3)C2)C)=O)cnc2sccc2c1 CC(C)(CCCNC(=O)Cc1cc(Cl)sc1Cl)NC(C1CC1F)=O c1(CN2CC(C(=O)Nc3cccc(Cl)c3)C(F)C2)ccnc2ccccc12 C(C(=O)NOC1CCCCC1)O.c1(C)cn(C2CCC2)nn1.CC(C)(C)N1CC1=O C1(C(N2CC(C=C)(CC(=O)N(C)Cc3cnn(C)c3C)C2)=O)CC(=O)NC1(C)C CC(CC(=O)N1CC2CC1C2CNC(=O)Cc1cncs1)CC(C)(C)C CCCCC(C)CCC(=O)N1CC=CC(NC(=O)CC2CCC2C)C1 C(CC(C)(C)CC(=O)N1CCCCC1CCNC(=O)C1=NNC(=O)C1)OC C(CC(N)=O)(C(=O)NC(C#C)CC1CCCO1)NC(CCCCC)=O CCC(C)CCCCC(=O)NCC1CN(C(C2CN(C)CCO2)=O)C1 CC(C)C(C)C(=O)NC(C(=O)OC(C)C)c1ccsc1 CC1CCC(C)N1C(C1CC(NC(C2CC2(F)Cl)=O)C1)=O C(C(CC1CC1)C(=O)NCC1(O)CCC1)NC(c1cc(CC)on1)=O Cc1cccc2c(CC(=O)NCCNC(C3CN(C)CC3C)=O)c[nH]c12 C1(C)(C(=O)OC)CCC(NC(=O)Nc2ccc(NS(=O)(=O)C3CC3)cc2)C1 N1(C(c2c(N)c(C)n(C)n2)=O)CC(NC(=O)C=Cc2ccncc2)C2(CCC2)C1 C(C(=O)NC1COC1)(C(C)C1CCCOC1)N1CCC(CC)C1 C(=O)(C(C)S(C)(=O)=O)N(C(c1ccc(F)cc1)CC)C(C)C c1(C(C)(C)NC(=O)CNC(=O)Cc2ccccc2)ccc(Cl)cc1 C1(C(N(CCN2CCCC2=O)CC)=O)CCn2c(C(F)(F)F)nnc2C1 C(C(C)(C)CNC(=O)CC1CCCO1)N(C(=O)CCn1cc(Cl)cn1)C c1(NC(C2C=CC(NCc3ncc(Br)cc3[N+](=O)[O-])C2)=O)cnnc2ccccc12 N1(C(C(C=CC)O)=O)CCC(CC(=O)Nc2ccc(OC)cc2C)C1(C)C N1(C(c2cccc(C#C)c2C)=O)CCN(C(=O)C(F)CC(C)(C)C)C2(CCC2)C1 N1(C(c2cc3cc(Cl)cnc3[nH]2)=O)CCCC2(CCCN2C(c2ccsn2)=O)C1 Cc1cc(Cl)cc2cc(C(=O)NC3CCN(c4cc(O)ncn4)C3)[nH]c12 C1(NC(CCCCC)=O)CC2CC(NC(=O)Cn3cnc4c3CCCC4)CC2C1 N1(C(C(CC)(F)F)=O)CCC(C2CCCN(C(=O)CC3COCCO3)C2)C1 c1(C(=O)NCCC(CCNC(C(=O)NCC)=O)C)cc(O)cc(O)n1 c1(CC)occ(C)c1C(=O)NC1CCC(CCNC(=O)C=Cc2ccc(C)o2)C1 c1(C(=O)NC(C)C(CO)NC(=O)CNC=O)nn(CC(F)F)cc1[N+](=O)[O-] CCC(CC)CC(=O)NC(C(C)NC(=O)C(=Cc1cnc[nH]1)C)C(C)C c1(C2(C)CC(Cn3nc(C4CCC4)cc3C3OCCO3)C2)nsc2ccccc12 O=C1CN(CC(=O)NCC(=C2CN(C(c3nc[nH]c3C(F)(F)F)=O)C2)F)CCN1 c1(CC(=O)NC)ccc(S(N)(=O)=O)s1.C12(CO)CCN(C1)C(CC)C(=O)N2 CCN=c1cc(-c2nc(CC3CC(CC)C3)n(C(=O)C3=COCCO3)n2)cc[nH]1 N1(C(C(CC)C)=O)CCN(C(C2CC(O)C2)=O)CC1c1cccc(Cl)c1 C(=O)(CC1=CCN(C)CC1)N1CCCC(C(=O)NC(c2nc(C)on2)(C)C)CC1 Cc1ccc(O)c(C(N2CCC(NC(=O)C(C)(C)C3CCCCC3)CC2)=O)c1 C(=O)(C(F)(F)C(F)F)N1CCCC(C(C)NC(=O)CC2(C(F)(F)F)CC2)C1 Cc1ncc(C#N)c(N2CC(F)(C(=O)Nc3cnc(O)c(Br)c3)C2)n1 C(=O)(C#CC1CCOCC1)N1CC(CC)C(NC(=O)Cc2n[nH]c(=NC)s2)CC1 C1(C(N2CC(OCCNC(C3C(C)=C3)=O)C2)=O)CCc2n[nH]c(C)c2C1 c1(CN2CC(NC(CCSC)=O)CC(F)(F)C2)cc2cc(C)ccc2[nH]1 N1(C(C(C)OCC=C)=O)CCN(C(=O)C(F)(F)c2nccs2)CC1C1CC1 n1(CC(=O)NCC2(O)CC(NC(=O)CCC3CCC3)C2)ncc(O)nc1=O C1(c2n(CCCC)nnn2)(NCCc2cc(Cl)ccc2Br)CCOCCC1C C1(O)(C(CNC(C2(C)C(C)C2)=O)(C)C)CN(C(C2CC(c3ccccc3)C2)=O)C1 C1(NC(CCCCNC(C2C=C(C)CS2)=O)=O)CCCCC12CC2 C1(C(=O)Nc2cncc(OC)c2)CCN(c2nc(C)cc(C)n2)CC1O N1(C(C(CCCC)N(C)C)=O)CCC(C2(NC(C3CC(C)OC3C)=O)CC2)C1 c1(C(C(CC(C)CO)=O)NC)oc2ccccc2c1Br.N1(CCNC)CCOCC1 C1(CCC(N2C(NC(CN(C(CC)=O)CC3CC3)=O)CC2)=O)CCOCC1 CC1CN2CCN1C(C(N1CC3CN(C(C45CC(C)C4C5)=O)CC3C1)=O)C2 C(=O)(CC1=NNC(=O)C1)NC1C(CNC(c2cc(CC)on2)=O)CC1 c1(C(=O)NCCC2(OC)CN(C(=O)CSCc3cc(C)on3)C2)c(C)noc1C c1(CC)ccc(C(=O)N(C2CCCN(C(=O)C(C)NC(C)=O)C2)CC)cn1 C(=O)(CCCCCC(C)O)N1C(CNC(COCC(=O)OC)=O)COC(C)(C)C1 c1(CN2CCCC(NC(C3=C(C)OCC3)=O)C2)cc(Cl)c(Cl)c(Cl)c1 N#Cc1cc(CN2CCN(C(c3cc(F)c(F)c(F)c3)=O)C(CO)C2)cc(Cl)c1 C#CCC(CC(=O)N(C)CC1OCCC1(C)C)NC(c1cnc(C)cn1)=O c1(C(N2C(C)CC(NC(=O)Cn3ccc(=N)[nH]3)CC2)=O)ccc(O)c([N+](=O)[O-])c1 Cc1cc(O)n2ncc(C(=O)NCC3CC(NC(C4(C(F)F)CCC4)=O)C3)c2n1 c1(OC)cc(C(=O)NCC2CCOC(C3CC3)C2)ccc1Sc1ccccn1 C(=O)(C1CCc2scnc21)NCC1C(C)(C)C(NC(c2ccccc2F)=O)C1 c1(-c2c(C)occ2)nc(C(C)CCC23CC(C(F)F)(C2)C3)n(-c2nc(Br)nn2C)n1 C1(NC(C(C#C)(C)C)=O)CCCCN(C(c2cc(C)c(Br)s2)=O)C1 C12CCN(C1)C2.c1(NC(C(c2cnn(C)c2)C)=O)cn(-c2cccnc2)nn1 C(=O)(C1CCCc2sc(C)nc21)N1CC(CCNC(C2N(CC)CC2)=O)(OC)C1 N1(Cc2ccc(-c3c(C)noc3)s2)CCC2(CC1)CC2NC1CCCC(F)(F)C1 c1(C(=O)NCCCN(C(=O)C=Cc2scnc2C)CC)cc(C)c2[nH]nnc2c1 C1(F)(CNC(c2cccnc2)=O)CCN(C(=O)C(F)CC2CC2)C1 c1(NCc2c(Cl)ccc(OC)c2F)ccc2c(c1)CCC2=O Cc1nn(C(C)C(=O)NCCNC(c2c(C)noc2C(F)F)=O)c(C)c1[N+](=O)[O-] C1(C(N2CCC3N(C(C(C(C)C)O)=O)CC(C3)C2)=O)C2C3CC4C1C1C2CC3C41 N1(CC(COC(C)C)O)CCC2CCC(C1)N2C(c1ccccc1)C C1(CNC(C(C)O)=O)CC2CCC1N2C(=O)CCCc1csc(=N)[nH]1 N1(C(C2(c3cc(C)no3)CCOCC2)=O)CCCC(C(=O)NC2CC2)CC1 N1(CC(N2C(C)CCCC2)=O)CCC(N(C(C2CCCS(=O)(=O)C2)=O)CC)C1(C)C C1(CNC(=O)CCc2nc[nH]n2)CN(Cc2ccc(O)nc2)CCO1 C1(CC)CN(C(=O)NC(=O)NC2(NC(C)C)CSC2)CC(C2CCC2)O1 CC1=NS(=O)(=O)NC=C1C(=O)NC1Cc2ccccc2CN1c1ccnc2c(OC)cccc12 N1(C(C(c2ccccc2F)(C)OC)=O)CCC2(CCN(C(C3CCCO3)=O)C2)C1 N1(C(C2CCCN(C)C2)=O)CC(NC(=O)Cn2cnc(=N)[nH]2)C(C2CC2)C1 Cc1nn(C)c(C)c1C(=O)NCC1CN(C(c2ccc(C3CCOC3)cc2)=O)C1 C=Cc1cncc(C(=O)NC2CC(CO)N(C(C3CC(SC)C3)=O)C2)c1 c1(C(=O)NC(CN(C(C(C2CCCCC2)C)=O)C)(C)C)c[nH]nc1F C1(CC(=O)NC2(C(=O)OCC)CC2)CCC(NC(=O)CC2CC2(C)C)CC1 N1(CC)CCCC(C(=O)NCC2(C)CCCN2C(c2cocn2)=O)C1 C1(CNC(c2ccn(CC)c2C)=O)CN(C(c2csc3nccn23)=O)C(C)(C)C1 N1(C(C(C=C)(C)O)=O)CCC(C2(Nc3ncc4ncnc-4[nH]3)CCC2)CC1 Cc1cc(Br)ccc1S(=O)(=O)N1CCOC(CC(N2CCCC(C)CC2)=O)C1 N#Cc1ncccc1-c1cc(CNC(=O)Cc2ccc(F)cc2)ccn1 C=C=CCC(=O)N(CC(C)N(C)C(c1n[nH]cc1C)=O)C C1(C)(CC(=O)NCC(C(=O)NCC2CN3CCC2C3)OC)CCOCC1 N1(C(C(C)Oc2ccc(Cl)s2)=O)CC(CO)CC(F)(F)C1 c1(C(c2nnnn2C2CC2)NC(c2cccc(I)c2)C)cccc(S(C)(=O)=O)c1 c1(CCC(=O)NCCOCCNC(C=CC(CC)=CC)=O)ccc(C)s1 N1(C(C2COCCN(C(C(CCCC)F)=O)C2)=O)CCc2sccc2C1 C(=O)(CS(=O)(=O)C1CCCC1)NCC(CNC(c1n(C)nc(CC)c1Cl)=O)(C)C C1(C(=O)NC(C2CN(C(=O)CN(C)S(=O)(=O)N(C)C)C2)C)CCCC2(CCC2)C1 c1(-c2n(C)c(N3CCCc4sccc4C3)nn2)cc2ccc(O)cc2o1 Cc1cc(F)c(N)cc1C(=O)NCCOCCOCCNC(=O)C=CCOC c1(NC)cncc(C(=O)NC2(CO)CN(C(=O)CC3CCCOC3)C2)c1 Cc1cc(C(=O)NCCCN(C)C(C2CC2C2CCOC2)=O)nn1C C(=O)(CC(C)NC(=O)CN(CC)CC)NCCCC C12(C(N(CC(=O)NC)CC)=O)CCC(CN(C(=O)CC3CC(C4CC4)C3)C1)C2 c1(OCC)cc(Br)cc2c(CNCC3CCCCN3CC(C)C)c[nH]c12 CCCC(C(=O)N1CCN(C2CN(C(=O)C(C)=NOCC#N)C2)CC1)NC(N)=O c1(C2N(C(=O)NC(COC)(C)CC(C)C)CCC2)nc2ccccc2[nH]1 CC1(C(N2CCC(C)(C(N3CCCC3)=O)C2)=O)CC2CCC1O2 N1(C(c2cnc(Cl)cn2)=O)CCC=C(C(=O)NCC2N(C)CCC2)C1 CCC(CN(C)C)C(=O)NC1CC(NC(=O)C(O)Cn2cncn2)CC1O C1(CNC(C2CC(C(C)C)C2)=O)CC2(CO1)CN(C(c1cc(F)n(C)n1)=O)C2 C1(C)(C(=O)NCCNC(CCCC=C)=O)CCCN(C(=O)OCC=C)C1.C(C)(C)(C)O C1(=O)NNc2cccc(c2)N(C)N2CCC12.C1(C=O)CCCOC1 c1(NC(=NC)NCC(=O)OC2CC(C)CN(C(C)C)C2)ccc2nc(C)[nH]c2c1 N1(C(C2(COC)CC(=C)C2)=O)CC2CC(OC)C2C1.C1(C)CCC(=O)N1 C(=O)(C1=C(C)OCCC1)NC(CCC#C)C(=O)N(C(CO)C1CC1)C CC(C)(CCNC(=O)C=CCO)NC(=O)CC1CC1(C)C C1(CCNC(CNC(C)=O)=O)CCN(C(c2cnn(C(C)C)c2)=O)C(C)C1 N1(C(c2cc(C)oc2)=O)CC(O)CC1(C)C(=O)NC1CCCSCC1 c1(Cc2cn(CC(=O)NCC(COC)(C)C)nn2)cc(OC)c(OC)c(OC)c1 C1(CC(N2CCC(CN(C(C3(C(C)C)CCC3)=O)C)C2)=O)CCCCC1O CCC(C)CCCC(=O)N(CC(C)CNC(C1(Cl)CCC1)=O)C C=C1CCC(C(N2CC(OCCC(=O)NCCOCCCO)C2)=O)CC1 C1(N(C(c2cc(C)ns2)=O)C)CCN(C(=O)C(C)OCC2CCCCO2)CC1 N1(C(C(c2ccc(O)cc2)C)=O)CCC(O)C(NC(C2CC23CCCCC3)=O)C1 C#CCC(C(=O)NCC1CCC1(F)F)NC(=O)C=CCOCCOC C1(CC(=O)OC)CN(C(c2ncccc2Br)=O)C2CC12 C=CC1(C(N2CCC(O)(CN(C)C(C34CCCC3C4)=O)CC2)=O)CCOCC1 c1(C(=O)NC2C(NC(C3CCC(CC)C3)=O)COCC2)cnc(OC)cc1OC C1(NC(CN(C)CC)=O)CN(C(=O)Cc2nc(-c3cccs3)oc2C)CCC1F N1(C(C(CC#C)C)=O)CCC2CCC(NC(C3(CCOC)CCC3)=O)C12 C1(N(C)C)(C(=O)NC2CC(NC(C3(C)CC(C(F)(F)F)C3)=O)C2)CCCC1 c1(C(N(CC(CC)NC(C2CCCC2CF)=O)CC)=O)nc2ccccn2c1F CC(C)(CC#N)C(=O)N1CCCC(CCC(N2CCCC2C(C)(C)CO)=O)C1 C1(C(=O)NC2COCCN(C(c3c(C)cc(CC)o3)=O)C2)CCCC2CCCN12 C1(C(N2C(C(CNC(CC3(C#N)CC3)=O)(C)C)CCC2)=O)CSC2(C)CCC(=O)N12 CS(C)(=O)=NCC(=O)N1C2CCC1C(CNC(=O)C=CC1CCCCCC1)C2 C(=O)(C1CCc2ccccc21)NCC1(CNC(CCC=CC)=O)CC12CCC2 c1(CC)oc(C)cc1C(=O)NC(CCSC)C(=O)NCC1CC12CCC2 C(=O)(CCS(=O)(=O)Cc1ccncc1)NC1(C)CN(C(c2ncn(C)c2)=O)C1 N1(C(C)C)CCC(C(C)(C)CNC(=O)CS(C)(=O)=O)CC1.N12CCC(CC1)C2=O N1(C(C(C(CC)(C)C)O)=O)CC2CC(N=c3[nH]nc(C(C)C)o3)C2C1 N12CC(C)N(CC1C)C(=O)c1c(COC)ccc(c1)C2=O.C1(OC)CCCCC1 c1(NC(CN(CC(C2CC3CCC2C3)(C)O)C)=O)cc2ccccc2s1 C(c1ccccc1Cl)=C(C)C(=O)NC1CC(NC(C2CCC(=O)N2)=O)C(O)C1 C1(C(=O)NC2CCCCN(CC3(O)CCOCCCC3)C2)CC2CC1C1C2C1(F)F Cc1cc(C(N2CCCC2C(C)NC(C2CCCCNC2=O)=O)=O)cnc1O C1(NC(C2CC23CCOC3)=O)CN(C(=O)C2=CCCOCC2)CC2(CCC2)C1 Cc1cc(C(=O)NC2CCCCC2NC(C2CCCN(C(C)C)C2)=O)cc(N)c1 c1(OC)nccc(C(=O)NC(C)(CNC(c2cc(O)nn2C)=O)CO)c1F c1(C(=O)NCCN(C(COC)=O)CC(C)O)cc(C(C)C)ccc1F O=C(CCC1CC1(F)F)NCCC1CC(NC(=O)CCC2CC2(Cl)Cl)C1 C1(C(=O)NCC(C2CCC2)NC(c2occ3c2CCC3)=O)C2CCC(F)(F)C12 CC1(C)CCC=C1C(=O)NCCN1CCN(C(=O)CCCCN2CCCC2)CC1 N1(C(c2nnn(C)n2)=O)CCC2(CC1)CC2NC(=O)Cc1ccc(S(C)=O)cc1 Cc1nc(NCC2(NC(c3cnco3)=O)CCCCC2)cc(SC(C)C)n1 CCCCCC(F)C(=O)NCC1(OC)CN(C(C2CC2(F)Cl)=O)C1 N1(C(C(c2c(OC)cc(Cl)cc2)=O)=O)CC2CN(C(=O)C(F)C(C)C)CC2(C)C1 c1(C(N2CCC(O)(CN(C)C(C3(C)CC(C)(C)C3)=O)C2)=O)ccc2ccsc2c1 C(=O)(C(C(C)(C)C)NC(=O)CN1CCC(=O)CC1)N(C(C)CC(N)=O)C c12ccc3c(c1)N(CCC3)C(=O)Nc1ccc(nc1)N2C.C(C(F)F)OC C1(NC(N2CCCCC2)=O)CCCC1CNc1ncsc1-c1ccccc1 C12(C(=O)NCCC(C)NC(c3ccnc(F)c3N)=O)CCCN(CCC1)C2 C1(CC(=O)OC)CCN(N2CCCCC2C(C)O)CC1 C(=O)(C1=CCOCC1)N1CCC(F)(C(N2C(CC(N)=O)CCCC2)=O)C1 c1(C(=O)NCC(F)CNC(c2cccn2C2CC2)=O)c(Cl)ccc2c[nH]nc12 C1(O)(Cc2nc(NC(C3C(C=C)C3)=O)sc2N)CCN(C(=O)OC(C)(C)C)CC1 Cc1nc(C(=O)N(C(C)CCCNC(=O)OC(C)(C)C)C)c2n1CCCC2 C=CC(F)(F)C(=O)NC(C)(C)CN1CCN(C(=O)Cc2n[nH]c(C)n2)CC1 C1(C)(CCC(=O)NCC(C2CC2)SC)CN(C(C2C3COCC23)=O)C1 C1(OC)(CNC(C2COCC2C(N)=O)=O)CCN(C(C2CC2(Cl)Cl)=O)C1 C1(SC)CN(C(=O)C(F)C2CC2)CC1n1cc(CC(C)O)nn1 CCC(O)C(C)(C)C(=O)N1CCC(N(C(=O)CCn2ccc(C)n2)CC)CC1 C1(C(=O)NCCCC(=O)NCC2C(C)(C)COC2)OCCCC1(C)C N1(C(C=CC=CCC)=O)CC2CCC(NC(c3ccc(OC)nc3C)=O)(C2)C1 N1(C(CCOCCOCC)=O)CCOC(CNC(c2cnn(CC(F)F)n2)=O)C1 N1(C(C2C(COC)(COC)C2)=O)CCN(C(c2ccc(C(N)=O)o2)=O)CC1CO C1(NC(C2(Br)CC2)=O)COC2CN(C(C3CCC4(CCC4)CO3)=O)CC12 CCCCCC(C)(CC)C(=O)NCCN(C(=O)C(C)Cc1ccc(Cl)c(Cl)c1)C c1(C(N2CC3CN(C(C(C)(C)SC)=O)CC3C2)=O)nnn2c1C(=O)NCC2 C1(F)(CNC(C2C(=C)C2)=O)CCN(C(C)=O)C1.C1(=O)C(COC)N1CC.C(C)(C)(C)O c1(C(=O)NC(CC)(CNC(C2CC2C2CCCO2)=O)CC)ccc(C)c(C)c1Cl C1(C(=O)NCC(C2CCC2)NC(C(CCC)(C)C)=O)CCOC2(CCOCC2)C1 c1(N2CCC(CCC#N)CC2)nc(N(CC(Cl)Cl)C)c2ccccc2n1 C1(C(=O)NCCCN(C(=O)C(F)C2CCOC2)CCO)CS(=O)(=O)C1 c1(C(=O)NC2(C3CCN(C(C(C)C#N)=O)C3)CC2)ccc(OCCF)cc1 Cc1c(C(N2CCCCC2C(=O)NCCc2ncccc2F)=O)nnn1C N1(C(C=CC(=O)NCC)=O)CCC(C)C(NC(c2ncccc2OC(C)C)=O)C1 c1(C(=O)NC2CC(N(C(COC)=O)C)C2)cc(F)cc2nc(C)c(C)nc12 c1(NC(C)=O)ccc(C(N2CCN(C(c3ccc(F)nc3C)=O)CC2)=O)cc1C c1(OC)c(Cl)nc[nH]c1=NCC1CN(C(=O)C=Cc2cn(C)nn2)CCC1C O=C(CCS(=O)(=O)c1ccc(Br)cc1)N1CCOC(c2ccc(C(=O)O)cc2)C1 C1(NC2(c3nnnn3C3CC3)CCC(CC(F)(F)F)C2)CCC12CCOCC2 c1(N2C(=O)CC(C(N(CC#N)CC3CC3)=O)C2)ccc2c(c1)CCC2 C1(CC(=O)NC(CNC(C(c2cccc(Cl)c2)(C)C)=O)C2CC2)CC=CCN1C C(CCC(=O)N1CC(C(C(=O)NC(c2ccon2)C)N(C)C)C1)=C(C)C C1(CC(=O)NCC(N)=O)CC2(C1)CN(CC1CCCSC1)C2 N1(C(c2ccc(OC)o2)=O)CCN(C(C)CNC(C2CCCN(C)C2)=O)CC1 N1(C(C2CC(C)(CC)C2)=O)C(C(=O)NCCC2(C)CCCO2)CCC12CC2 C1(C(C(=O)NCC(F)F)N(CC(=O)OCC)CC2CC2)CC12CCCCC2 C1(N(C(=O)COC(C)(C)C)CC)CCN(C(=O)C(c2ccn(C)n2)C)CC1 N1(C(CC2CCN(C)CC2)=O)CCCC2(CCN(C(C3COC(=O)N3)=O)CC2)C1 N1(C(CCC=C)=O)CCN(C(c2csc(Br)n2)=O)C(CC)C1 CC(C)(C)C#CC(=O)NCC(C1CCOC1)NC(=O)CCOc1ccc(N)cc1 CCC(CC(=O)NCc1nccc(O)n1)NC(=O)CCc1nc(C)no1 CN1C(=O)C(N2CC3COCC(C2)C3NC(=O)OC(C)(C)C)Cc2ccccc21 N1(C(c2c(C)cco2)=O)CC2CN(C(=O)C=CC3CCOC3)CC(F)(F)C2C1 C=CCCCC(C(=O)NC1CCCC1)N1CCC(C(=O)OC)C1C Cc1[nH]c2ncccc2c1C(=O)NC1CCN(C(c2occc2F)=O)CC1O N#Cc1cccc(OCC(=O)NC2(F)CCCN(C(=O)COCOCCF)C2)c1 N1(C(C(C(C)C)NC(C)C)=O)C2CCCC1CN(C(c1cocn1)=O)C2 C1(C(=O)NC(C2CCN(C(C3(SC)CC3)=O)CC2)C(C)C)CC2(C1)CC21CCC1 c1(C(=O)NCCN(C(C(F)OC)=O)C2CC2)ccc(-c2cn[nH]c2)cc1 c1(C(=O)NCC=CCN)ccc(OC2CC2)nc1.c1(CC2CC2)nc(C(=O)CC)cs1 C=CC1(CC(=O)NCC2(O)CCOCC2)CN(C(C2CC(CC)C2)=O)C1 CC(C)(CCNC(=O)CC1CCCC1)C(=O)NC1CC2(CCC2)C1 N1(C(c2cnc(C)[nH]2)=O)CCC2C(NC(c3cc(Br)sc3Cl)=O)C12 Cc1nc(N(C(C(=O)NCC(N2CCCCCC2)=O)C2CC2)C)cc(N(C)C)n1 CC1OC2(C)CC1(C(=O)NC1CC3CC1N(C(=O)CCn1cnnn1)C3)C2 n1(CCC#N)c(NC2CCOC2)nnc1CC(N1CCC(N2CC=CC2)CC1)=O c1(CC(=O)NCC(C2CC2)NC(C2C(C(=O)OC)C2)=O)cn(C)nc1C C1(C(=O)OC)C(C)CCN1C(C1CCC1CNC(c1cncnc1)=O)=O C=CCCCCCCCC(=O)NC1(CCNC(=O)COC2(C)CCCC2)CC1 C(CC(C)(C)CNC(=O)C(C)=C1CCCC1)OCC C1(NC(C(=O)Nc2c(OCC)c(C#N)c(F)cc2)=O)CCC2C3C=CC(C3)C12 c1(CNC(C23CC(NC(C(=O)N(C)C)=O)C(C2)CO3)=O)cn2ccccc2n1 C1(CC)CCCN(C(C2CC(O)CN2C(=O)CC2CCOC2(C)C)=O)C1 CCCCC(C(=O)NCC1CN(C(=O)CCOC2CCC2)CCCO1)C(C)C Cc1cc(CN2CC3(CC(CC(=O)N(C4CCCC4)CC(C)C)C3)C2)cnc1F C1(=O)C(CC)C(=O)O1.O(NC(=O)Cc1cnc(C)o1)CCCC N1(C(C2(CNC(c3cc(OC)no3)=O)CC23CCC3)=O)CCC2CCC(C1)N2C c1(C(N(CCCCNC(c2cccc(F)c2)=O)C)=O)ccnc(Br)c1N CC(c1ccccc1F)=CC(N1CCOC(CN(C)C(c2ccon2)=O)C1)=O N1(C(C(C(F)(F)F)OC(C)=O)=O)CCN(C(c2nc(C)oc2C)=O)CC(O)C1 N1(C(COCC=C)=O)CC2CCC2(NC(=O)C(c2ccc(OC)cc2)=O)C1 C=CC(C)(CCOC)C(=O)N(CCNC(c1cnn(CC2CC2)c1)=O)C1CC1 c1(C(=O)NC(CNC(C(C(C)C)SCC)=O)(C)C(C)C)nn(C)c2c1CCCC2 N1(C(C(=O)NCCCOC)CCC2CCOCC2)CCCSCC1C1CC1.C1CS1 C1(C(N2CC(O)C2)=O)CCN(C(c2csc(-c3ccsc3)n2)=O)C(=O)C1 CC(C)(CC(=O)NC1CCN(C(C2CC(F)C2)=O)C12CC2)CC(F)F C(=O)(C(C)(F)C(C)(C)F)N1C2C(CNC(C(C)CN3CCCCC3)=O)C(C2)C1 CC12CCC(C(=O)NC3CCC(C(N4CCC(O)C4)=O)C3)(CO1)C2 C(=O)(C1CCc2c(Cl)cccc21)NC(CNC(C(C)Cc1ccncc1)=O)(C)C C1(OC)(CNC(c2cnn(CC3CCC3)c2)=O)CN(C(C2CC2C)=O)C1 c1(C(=O)NCC2(NC(COc3cccc(C)c3)=O)CC2)n[nH]c2c1CC1CC21.OCC CC1CCCC(CC(N2CCC(NC(C3CCCCC3)=O)CC2)=O)C1 N1(C(Cc2ccc(OC)cc2)=O)CCCC1C1CCCN1C(c1cncs1)=O N1(C(=O)Nc2c(OC)cc(OC)c(Br)c2)CCN2CCCCC2C1 C(CCN=c1cccc(S(=O)(=O)NCC2CCC(C)C2)[nH]1)OCC=C C1(C(=O)NC(CC)CC)CCCN(C(C2CCCN(C)C2)=O)C1 c1(C(=O)OC)coc(C(C(=O)NCCNc2cn(CC)cn2)N(C)C)n1 c1(C(=O)NC2CC(NC(COC3CCCC(CO)C3)=O)C2)cc(O)cc(F)c1 C(=O)(C1OCCc2ccccc21)NCC1CCC(NC(C2(CC)CC=CC2)=O)C1 c1(NC(CN(CC(C)OC)Cc2cnn(C)c2C)=O)c(C)cc(C)cc1C C1(C(=O)Nc2c(C(c3nn[nH]n3)(C)C)ccc(C)c2)CCCC2(CCNC2)O1 C1(CNC(=O)NCC2C(=C)CCC2)(OC)CCCC(C)(C)C1 c1(C(=O)NC2C(OC)CN(C(c3ccc(SC)o3)=O)C2)cc2c(Cl)cccn2n1 c1(CC)ccc(C(=O)NCC(C2CC2)NC(c2cc(O)nc(C)n2)=O)cc1OC CC1(C)COC(C(=O)NCC(C2CCC2)NC(=O)C(c2cccc(Cl)c2)(F)F)C1 Cc1ccc(C)c(SCC(=O)NC2CCN(C(=O)C=CC3(C)CCOCC3)C2)c1 C(C)(CNC(=O)CCn1cc(C)cn1)(CC)NC(C1C(C=C)C1)=O N1C(=NCCCF)N2CC(OC(C)C2)C(=O)NC1=O.C1(OCCOC)(CO)CC1 C(=O)(C(C)(CC)CO)N1CC(OC)C(NC(c2cc(C)c(C)o2)=O)C1 C(=O)(CCCCCCN=[N+]=[N-])N1C(CCNC(C(CCC)(C)C)=O)CSCC1 c1(N(C23CC(C2)C3)C(c2scc(C(N(CC)CC)=O)n2)=O)ccc(Cl)cc1 C1(O)(C(C)NC(c2n(CC)cnn2)=O)CCN(C(=O)C2=CCOCC2)CC1 c1(NC(C2C(C(=O)Nc3cccc(C)n3)C2)=O)cc(C#N)ccc1Cl N1(C(CCCCC)=O)CCC2(CC1)CC2NC(c1cc(Cl)cc(Cl)c1)=O N(C1c2ccccc2CC1NC(C1CC2(C1)CC2F)=O)C(C#CC1(C)COC1)=O C1(C2CCCN(C(c3ncsc3C)=O)C2)(NC(C(C)NC(COC)=O)=O)CC1 Cc1cc(C(=O)NCC2C3CN(C(c4nccnc4C(N)=O)=O)CC23)cc(N)c1 c1(-n2c(N(n3ccnc3)C)nc(CCC(C)(C)C)n2)ccc(F)c(F)c1.C(N)=O CC(C)(C)C(O)C(=O)NCC=CCNC(=O)C=Cc1sc(Cl)nc1Cl C1(C)(CNC(c2c(C)nccc2)=O)CC(F)(F)CN1C(C1C(C(F)F)C1(C)C)=O N1(C(CC2CC(C(C)(C)C)C2)=O)CCCC(C)(C)C1C(=O)NOC1CCCC1 Cc1nc(CC(=O)NCC(C)CN(C(=O)C(O)C2CCCC2)C)oc1C C1(NC(c2cnn(CC)n2)=O)CC2CC1N(C(=O)CCC(C)(C)N(C)C)C2 CC1CCc2n[nH]cc2C1C(=O)N1CCC(CNC(c2ccoc2)=O)C12CC2 N1(C(CC=CCCCCC)=O)CCC2(CC2NC(c2nn(C)cc2Cl)=O)C1 N1(C(CNC(c2c(C)occ2)=O)=O)CCOC(CCNC(c2coc(Cl)n2)=O)C1 CN1C(=O)CSC1=CC(=O)NCC1CCC(NC(c2cc3ccccn3c2)=O)C1 c1(CC)c[nH]nc1C(=O)NC(C1(C(=O)NCc2cnc[nH]2)CC1)C CC(O)CC(C)(C)CNC(C1CC(CNC(=O)COC2CCC2)C1)=O c1(C2N3CCC(C3)CNC2=O)ccc2c(c1)CCCC2.c1(CC)ccc(OC)cc1 C(=O)(C1CCCn2nccc21)NCCCCN(C)C(C1CCc2nn[nH]c2C1)=O N1(C(CC2CCN(C(C(C)OCCC=C)=O)C2)=O)CCOC2(CCC2)C1 CC1(C)OCCOC1C(=O)NCC1CCN(C(c2cnn3c2OCC3)=O)C1 Cc1nnc2n1CC(C(=O)NC1CC=CCC1)N(C(=O)C1CC1)C2 N1(C(C(C)(C)n2cc(CNC(C3(C(N)=O)CC3)=O)nn2)=O)CCCC(N2CCCC2)C1 c1(CC(N2CCC(C)(NC(C3C(C)OCCO3)=O)C2)=O)csc2nccn12 C12(C(=O)NC3C(C)CN(C(=O)CCc4cncs4)CC3)CC(CO)(C1)OC2(C)C N1(C(c2ccnc(C)c2N)=O)CC2CC1CN(C(c1cc(Cl)sc1Cl)=O)C2 C1(C(=O)NCCC2(CNC(=O)CCNS(C)(=O)=O)CC2)(CC)CCC(O)CC1 C(=O)(C1=C(C)OCCC1)NC1C(CNC(c2ccc(C=C)cc2)=O)CCCC1 C(c1cc(Cl)cc(Cl)c1)=CC(=O)NCC(CO)NC(c1ncc(Cl)cc1F)=O Cc1cn2cc(C(=O)N(C3CCCCC3)CC3CC3)nc2s1 C1(C)(CN(C)Cc2scnc2-c2ccc(Br)cc2)CC(=O)C12CCC2 c1(C(C)C)[nH]nc(C(N2CCC2CNC(=O)Cn2ncnn2)=O)c1[N+](=O)[O-] N#CC1(CC(=O)NCC2(F)CN(C(c3nc[nH]c3C(F)(F)F)=O)C2)CCCCC1 C(=O)(C1=COCCC1)NCCC(CNC(c1c(CC)ncnc1)=O)O CS(=O)CCCCNC(C1(SC)CN(C(C2CN(C(N)=O)C2)=O)C1)=O N1(C(CC=CC=C)=O)CCC2(CC2NC(c2ccc(C(F)F)nc2)=O)C1 c1(C(=O)OC)cnccc1C(=O)NCC(C)(C)CNC(c1cc(C)sc1N)=O N1(C(c2ccc(OC)cc2)=O)CCC(C)(C)C1C(=O)NCCC(C)c1cn[nH]c1 N1(C(C2(NC(c3cc(C)oc3C)=O)CCC2)=O)CCC2(CCOC2)C1 c1(C(C)C)csc(CNC(=O)NCC2(O)CCNC2)n1 C1(C(N(CCCC=C)CC)=O)CC=CCN1C(C1CCC1(OC)OC)=O C12(C(=O)NCCCN(C(Cc3ccc(C#N)cc3)=O)C3CC3)CCCCC1OCC2 c1(C(=O)NCC(CNC(Cc2c(C)nccc2)=O)F)ccc2nccn2c1 C1(CNC(C(C)Cn2cccn2)=O)CN(C(c2cnc(S)[nH]2)=O)CC(C)(C)C1 C12CCN(C1)C(=O)c1ccc(s1)O2.C(C(=O)NCCC)OCCC c1(COC(C)=O)cn(-c2nnc(-c3ccccc3)s2)cn1.C1CNC(=O)N1 C(=O)(CS(=O)(=O)CC1CCCO1)NCCC1CN(C(C(=O)NCCOC)=O)C1 C(=O)(C#CC1CCCO1)N(CC(CN(C)C(C1(O)CC(C)(C)C1)=O)O)C c1(C(=O)NC2CCN(C(C(C)C(F)F)=O)C2(C)C)cc2cccnc2s1 C1(C(=O)NCC2(O)CN(C(=O)Cc3csc(C)n3)C2)(OC)CCCCCC1 C1(NC(CC(C)SC)=O)CCC(C)N(C(=O)CC=Cc2ccccc2F)C1 C1(C(N(C(CN(C(COCCSC)=O)C)C)C)=O)CCOC1c1ccncc1 S(=O)(=O)(CCCCF)NCCC1CCC(NC(=O)OC(C)(C)C)CC1 CC1CN(C(c2cc(C3CC3)ncn2)=O)CCC1NC(C1CCCCS1(=O)=O)=O N1(C(c2cc(C)[nH]c2C)=O)CC(O)CCC1C(=O)N(C)Cc1ccsc1 C(CO)(CC(C)(C)C)NC(CN1CCN(C(C2(C)CCN(C)C2)=O)CC1)=O C1(C(=O)NCCN(C(CC2CC(C)C2)=O)C)C(C)C1(F)F c1(CN2CCC(CNC(C3CC3(F)F)=O)CC2)cc(F)c(O)cc1F c1(C(N2CCC(OC)CC2)=O)cnn2ccc(-c3ccc(O)c(C)c3C)cc12 CCN=C(NCc1cc(C2CC2)no1)NC1CC1c1cccs1 C(=O)(C1=COCC1)NCCC(=C)CNC(=O)C(O)Cc1ccccc1Cl c1(C(=O)NCC2CC(NC(C(COC)O)=O)C2)ccc2nc(N(C)C)sc2c1 n1(CCOC)nccc1C(N1CCC(CN(C)C(C23CC(C)C2C3)=O)C1)=O N1(C(c2ccc(-c3c(OC)nccc3)cc2C)=O)CCOC2(CCOC2C)C1 c1(-c2n(C(=O)N=c3[nH]nc(C(F)(F)C(F)(F)F)s3)ccn2)ccc2c(c1)OCCO2 CC1CCCC(C(=O)NCC2CCCCC2NC(C2CC3CCC2C3)=O)C1 Cc1ccc(C)n1CC(=O)N(CCCN(C)C)CCNC(C1(F)CC1C(F)F)=O CCC(CNC(=O)CCC(C)NC(=O)C(C)NC=O)C(C)(F)F CC1(C)CCCN(C(c2cc(CCO)on2)=O)C1CNC(c1ncc(Cl)s1)=O N(C(=NCC(C)(C)c1ccccn1)N1CCC(OC)C1)C(COC)C CC1CCCN(C(c2cn(CC(N)=O)nn2)=O)C1CNC(c1ccc(O)cc1)=O Cc1nc(Cl)cc(NNC(=O)C=Cc2cnc3n2CCCC3)n1 C(=O)(C(C)CC(N)=O)N(C1CCN(C(CC=CCC)=O)C1)C c1(C(=O)NCC(C)NC(c2cc(OCC)ncc2)=O)ccccc1C#CC1CC1 C(CC(C(=O)N(C)Cc1ccoc1)NC(c1ccn(C2CC2)n1)=O)=CC C1(NC(C2=NOC(CNC(C3(SC)CCC3)=O)C2)=O)CC2CCC(C1)C2O C1(SC)CN(C(C2CCCC2)=O)CC1NC(c1cnc(-c2ccccc2)[nH]1)=O N1(CCc2cccc(C)c2)CCC(NC(C2CCCCO2)=O)CC1C S(=O)(=O)(CC(=O)NC1(C2CCN2C(C2CCS(=O)CC2)=O)CC1)NC(C)(C)C N1(C(c2ncc(OC)nc2)=O)CCC2CN(C(=O)C(=Cc3cccs3)C)C2C1 CCCC(CC)C(=O)NCC1C=CC(NC(c2cn(C)nc2C2CCOC2)=O)C1 N1(C(c2cc(OC)cc(Cl)c2)=O)CCCC2C1CCN2C(c1cnc(Br)s1)=O C1(NC(=O)NC(CCCC)CC)CC2C=CC1CC2 C1(CN(C(c2c(C(C)C)c[nH]n2)=O)C)CCCCN1C(c1cc(C2CC2)no1)=O C1(C(=O)NCC(=O)OC(C)(C)C)CC12CN(C(=O)C(c1ccc(Br)cc1)(C)C)C2 N1(C(c2ccc(OCCN(CCNCCCC)CCO)cc2)=O)CC2C3COCC3C2C1 N1(CC)CCCC(C(N2CC(OCCC(N3CC(C)(CC)C3)=O)C2)=O)C1 c1(CC)cccc(C(=O)N(C2CCCN(C(=O)CC(C)CF)C2)CC)c1N O=C(CCc1cnco1)NCCC1(C(=O)NCCCCc2cnc[nH]2)CC1 C(=O)(C(C)(C)C(=O)NC1CC1)N(CC(F)(F)Br)C N1(C(Cc2nc(C)oc2)=O)CCC(NC(=O)C2=NOC3COCC23)C(F)(F)CC1 CCCC(C(O)C(=O)NCc1cnc(N(C)C)nc1)NC(=O)CC1CNC(=O)O1 C1(CC(=O)NCCOCCC#C)CC(NC(c2cn[nH]c2)=O)C1(C)C c1(CC)cnn(CCNC(C2(N(C)C(c3coc(CO)c3)=O)CC2)=O)c1 C1(C(N2CCC(N(C)C(c3nccnc3C(N)=O)=O)C2)=O)CC(C)(C)CN1C c1(C(=O)NC(C)CN(C)C(c2cc(C(F)(F)F)on2)=O)cncc(Cl)c1 C1(NC(C(C=C)C)=O)CN(C(=O)C=Cc2csnc2C)C2(CCC2)C1 c1(C(N2CC3C(NC(C4(C#N)CC=CC4)=O)C3C2)=O)c(Cl)cccc1Cl Cc1cnsc1C(=O)NC1CCCC1OC1CCCCC1 CC(C)CC(O)C(=O)NC1CCN(C(c2cccnc2OCC(C)C)=O)CC1O N1(C(C(c2c(C)noc2C)C)=O)CC2(NC(c3ccn(C)c3C)=O)CCC1CC2 C1(CNC(c2cc(C)nc(O)n2)=O)CC2CCC1N(C(C1CC13CC3)=O)C2 C1(C(NOCCCOC)=O)CC2CCCC2N1C(=O)COCc1nc[nH]n1 C1(CCNC(C2CC23CCSCC3)=O)CCCN(C(=O)Cc2csnn2)CC1 C1(C(=O)NCCC2CN(C(C(C)(C)C3CCCC3)=O)C2)CNC(=O)CC12CCC2 Cc1nc(C(N2CC(CNC(C3CCCS3)=O)C(C)C2)=O)ccc1Br C1(CN(C(=O)C=C(C)C)CC)CCCN1C(C1CCCC1)=O c1(CCNC(C(=O)Nc2n(CC)nnc2C)=O)ccc2c(c1)OCO2 C1(NC(c2ncccc2Br)=O)CC(CO)N(C(=O)CSc2n[nH]c(O)n2)C1 C(=O)(CCP(C)(C)=O)N(C1CC(CCNC(=O)C=CC2CCCCC2)C1)C C(CC1=CCCCC1)NC(CCC1(NC(CC(C)C2CC2)=O)CCCC1)=O N1(C(c2c(CC)n(C)cc2)=O)CCC(C)(NC(C2(C3CCCO3)CC2)=O)CC1 C#Cc1ccc(C(=O)NCC2COCCN2C(=O)C(n2ccc(C)n2)C)cc1C C1(C(=O)NCC2CCCN(C(c3cncc(O)n3)=O)C2)CCn2ncnc2C1 N1(C(C(C)C2CC2)=O)CCCC(Cc2cn(CCSC3CC(=O)NC3=O)nn2)C1 c1(C(N2C3CN(C(c4cccc(OC)c4OC)=O)CC32)=O)cc(O)ccc1[N+](=O)[O-] CCC(C)C(O)C(C)C(=O)N(CC(=O)NCC(CC)C1CCC1)C c1(CNC(CCC2(C)CC2)=O)cccc(CNC(=O)CC(c2ccc(F)cc2)C)c1 c1(C(C(=O)OC)N(C2CCC(C)(C)C2)C)cccc(C(=O)N(C)C)c1 C1(C)(CNC(CC2CN(C)C2)=O)CCCN1C(=O)CC(C)C1CCCCC1 N1(C(=O)C(F)=CC2CC2)CC2OCCN(C(C3SCCCS3)=O)C2C1 c1(OC)cc(C(=O)NC(C2CN(C(C3CCN3S(C)(=O)=O)=O)C2)C)ccn1 c1(C(=O)NCCC(CNC(CC(C)(C)OC)=O)O)ccc([N+](=O)[O-])cc1[N+](=O)[O-] C1(CNC(CC(CC)OC)=O)CC2(CCN(C(=O)C3=NNC(=O)CC3)CC2)C1 c1(C(=O)NC2C(NC(C3CN(C(N)=O)C3)=O)C2)ccncc1-c1ccccc1 c1(C(N2CC=CC(C(=O)NC3(C)CC(=C)C3)C2)=O)ncc(N)cc1C N12CCC3(CCCC13)C2=O.C1(COC(C)=O)CC2CCC1CC2 CC1CC(CNC(c2snc(O)c2Cl)=O)CCN1C(=O)C1=CCCSC1 C1(CNC(c2sccc2Cl)=O)CN(C(=O)C=Cc2ccsc2)CCCO1 c1(NC(C2(C)N(C(CCN(C(C)=O)C)=O)CC2)=O)cc(Cl)c(F)c(Cl)c1F c1(CNC2CCC(C(=O)Nc3onc(C)c3C)C2)cccc2c1CCC2 Cn1nccc1CCCNC(C1(CNC(c2cc(C(N)=O)c[nH]2)=O)CCCC1)=O CCC(C(=O)NCc1ccc(CNC(C2(C)COCCO2)=O)cc1)C(C)O C1(CNC(C(C)OCOC)=O)CCC(C)(C)CN1C(c1sc(CO)nc1C)=O CCCCCCCCCCCCC(O)C(=O)NCC1OCC2CCCC12 CCC(C(=O)NC1CC2CC(C1)N(C(c1nc(C(C)C)oc1C)=O)C2)C(C)(C)CC N1(C(C(C)(C2(C)CC2)OCC)=O)CCC(F)(CNC(=O)CC(CC)OC)CC1 N1(C(CN2CC(CC)C2)=O)CC2ON=C(CNC(c3ccc(=O)oc3)=O)C2C1 C12(C(N3CC(CNC(CCNC(=O)CO)=O)C4(C3)CC4)=O)CCC(=O)N1CCS2 c1(COC)cc(C(=O)NCC2(F)CC(NC(c3cn(C(F)F)cn3)=O)C2)n(C)c1 C12(C(N(CCNC(=O)CC3CC(SC)C3)CC)=O)CC(CO)(C1)OC2C c1(OC)cc(C)nc(N2CCC(C#N)C2)n1 CC(C)(C(=O)N1CCC1CNC(C1CC1C(C)(C)O)=O)N1CCOCC1 c1(OC)ccc(Cl)c(C(=O)NCCNC(C2COC(C)C2)=O)n1 c1(OC)cccc2c1CN(C(=O)NCCCN1C(=O)CCCCC1=O)CC2 C1(C2CN(C(C3CCCCNC3=O)=O)C2)(NC(=O)COc2ccc(O)cc2)CC1 c1(C2CN2)ccccc1Cl.C1(CC(C)(c2nnnn2C(C)C)OC)CC(F)(F)C1 C1(NC(=O)CSCc2cccnc2)CCN(C(=O)C(O)c2ccsc2)CC1O c1(NC(c2scc(C)c2)C)nccc(N2CCCC(n3[nH]c(C)nc3=O)C2)n1 CC1CCCn2cc(C(=O)NCC3CC4CCC3N4C(c3sccc3Cl)=O)nc21 c1(CC(=O)NCCC(C)N(C)C(c2cc(-c3ccccc3)no2)=O)cncn1C Cc1ccc(Cl)cc1C(=O)NCCCOCCCNC(=O)C(F)C(C)(C)O c1(C(N2CCN(C(=O)OCC=C)CC2)=O)ccc2[nH]c3c(c2c1)CNCC3 c1(C(N(CCC)CCNC(C2(C)CCCC2)=O)=O)cncn(C)c1=O N1(C(C(C)OCC#C)=O)CC2CC1C2NC(c1cnn(CC(F)F)c1)=O c1(CC)nc(C)c(C(N2CCCOC(CNC(=O)COC(F)(F)F)C2)=O)c(C)n1 C12(C(=O)O)CC(c3nc(C4CCC(C)O4)no3)(C1)OC2C.CC(C)(C)OC(=O)N Cn1ccc(-n2cnc(C(=O)NC3COCC3NC(=O)C(F)(F)C3CC3)c2)n1 CCCCC(CN(C(C1CN(C)C(C)(C)C1)=O)Cc1nc(CC)no1)CCC N1(C(Cc2c(C)n[nH]c2)=O)CC2OCCN(C(c3cccc(Br)c3O)=O)C2C1 C(CC1CC1)(C(=O)NCC(F)Br)NC(C(C)OC(C)(C)C)=O N1(C(c2c[nH]nc2C(F)F)=O)CCC(NC(=O)CSCC2CCCCO2)CC1 c1(C(N2C3CC(NC(C4(OC)CCC4)=O)C(C3)C2)=O)cnc2nc(C)[nH]n2c1=O C1(NC(CCC(C)C)=O)CC2CN(C(=O)C(=O)Cc3ccc(Cl)cc3)CC12 CCCC(C)CCCC(=O)N1CC(CNC(=O)C(C)=C2CCCC2)CC1C C1(CNC(C2CCN(C(C)=O)C2)=O)CC(F)CN1c1nnc(C2CC2)s1 C(C(C)(C)C(=O)NCCN(C(c1ccc(Cn2ccnn2)cc1)=O)C1CC1)SC N1(C(C(c2cccc(O)n2)C)=O)CC2(C1)CN(C(=O)C=CC1CCOC1)C2 c1(CSCC(=O)N(C2CCN(CC)C2)CC)ncc(NC(N)=O)c(C)n1 c1(C(=O)NC(C(C)C)(C)CNC(c2ccc(C#N)s2)=O)c(F)ccc2c1OCC2 N1(C(CC2(N(C)C)COC2)=O)CC2(C1)SCCC2NC(C1CC2CCC2C1)=O CC12CN(CC(O)COc3ccccc3)CC1C1CC2C1 C1(NC(C2CCC3(CC2)CC3)=O)CCCC12CCN(C(C1SCCCS1)=O)C2 Cc1cc(=NCC2CNC(=O)CO2)[nH]c(NC2CCc3ccccc32)n1 C1(CC(=O)NC(C2(O)CCC2)C)CCCCN1C(c1cnccc1Cl)=O C(=O)(C(O)C(C)CC)NC(C1N(C(C(C)OCC#C)=O)CCC1)(C)C Cn1ccnc1CCC(=O)NCC(C)(C)OCCNC(=O)C(O)C1CCCC1 c1(C(N(CCCNC(C(C)CC(N)=O)=O)C2CC2)=O)cccc2oc(=N)[nH]c12 CC(C)(F)CCC(=O)NC(C)(CNC(=O)CCN1CCC(O)CC1)CO Cn1cccc(C(=O)NC2CCC2CNC(=O)Cn2nccn2)c1=O C1(C(C)(C)O)(NC(CC2C(OCC)C2)=O)CN(C(C)=O)C1 N1(c2nccc(C)n2)CC2CC1CN(C(c1cc(CC(C)C)on1)=O)C2 c1(-c2cn(CC(=O)N(C(c3conc3C)=O)CC)nn2)ccc(NC)cc1 C(=O)(C(CC(=C)Cl)NC(=O)CCCCCN(C)C)NC(COCC(=O)OC)C c1(OC)cccc(C(=O)NCC2CCC(NC(c3c[nH]c(Br)c3)=O)C2)c1 N1(C(C(CC)C)=O)CC2(CC(C(=O)NCc3cc(C)cc(C)c3)CO2)C1 c1(OC)ccc(C(N2CCNC(C(=O)Nc3ncc(F)cc3C)C2)=O)c(O)c1 CC(C)(C)C(C(=O)N1CCCC(NC(CC(=O)NC2CC2)=O)C1)NC(=O)C1CC1 C(=O)(CC(C(F)(F)F)N(C(c1c[nH]c(C#N)c1)=O)C1CC1)NC(CC)(C)COC c1(C(N2CC(C)C(NC(c3cccn4nccc34)=O)C2)=O)ccc2ncccn12 C1(=CCN=[N+]=[N-])C(=O)Nc2ccc(-c3ccc(CCO)cc3)cc21 C1(C(=O)NC2C(CNC(c3c(CC)nn[nH]3)=O)C2)CCCOC1c1cn(C)nn1 c1(SCC(N2CC(C)(NC(C3CCN(CC)CC3)=O)C2)=O)nc2ccccc2s1 C1(CC)CN(C(c2ccc(C3CC3(F)F)cc2)=O)CCN1C(c1cnsn1)=O C(=O)(CC(COC)COC)NCC(CN(C(=O)CC(C)OC)CC)(C)C c1(C(N(C2CCN(C(C3N(C(C)=O)CCC3)=O)C2)C)=O)cn2c(n1)CCC2 C1(CCC(N2CCC(CSC)C2)=O)CCCC(NC(=O)CSc2ncccn2)C1 c1(OC)ccc(CN(C)C(=O)Nc2cccn(C)c2=O)c(OC)c1OC C1(C(=O)NC)Cc2ccccc2N1C(=O)C(=O)NC(c1ccccc1)C1CC1 N1(C(C#CC2(CC)COC2)=O)CC2(C)CN(C(=O)C(C)(C)CC)CC2(C)C1 N1(C(c2ccc(OC)s2)=O)CCN(C(c2c(C)cccc2F)=O)CC(O)C1 N1(C(c2ccc(SC)cc2)=O)CC(C2(NC(=O)CS(=O)(=O)N3CCCC3)CC2)C1 C1(C(N2C(CNC(c3scc(C)c3)=O)CC3CC32)=O)Cc2cncn2C(=O)N1 C12(CC(=O)NCC(C)N(C(=O)Cc3ccon3)C)CCCN1CCC2 c1(C(C(=O)NC2CCCC2)N(CC(C)(C)C#N)C)sc(=O)n(C)c1Cl C(=O)(CC(C)(C)CCOC)N1C(C)CC(CNC(CNC(CC)=O)=O)C1 Cc1cccc(CC(=O)NCCN(C(c2cscc2C(F)F)=O)C(C)C)c1F C1(C(C)O)CCCN(C(C2(NC(=O)C=CCN3CCC3)CC(O)C2)=O)C1 CC12CCC1CN(C(=O)CCCCCNC(=O)CCCc1cnn[nH]1)C2 C1(C)(NC(C(CCNC(=O)CN2CCC(=O)CC2)OC)=O)CC(C)(C)OC1=O Cc1cn2[nH]c(=NC3COC4(CCN(C(C5(O)CCSC5)=O)CC4)C3)sc2n1 C1(NC(C(C=CC)O)=O)CCC2CN(C(=O)C3=CCCO3)CC2C1 c1(C(N2CCN(CC(C)NC(=O)CC(C)CF)CC2)=O)cccc2cncn12 c1(OC)ccnc(C(=O)NCCN(C(c2ncccc2Br)=O)C2CC2)c1 c1(CNc2occ(C)n2)ccc(Nc2nnnn2-c2cccc(Cl)c2C)c(C)c1 CCCS(=O)(=O)CC(=O)NC1CCC(CCNC(C2(Cl)CC2(F)F)=O)C1 c1(C(=O)NC2CC2CNC(C2OCC3CCCC23)=O)cnc2nccnc2c1 N1(C(CC(C=C)CCC)=O)CCC2(CCCN2C(=O)COCC(C)C)C1 C(=O)(CC(C)c1cnn(C)c1)NCC(C)CNC(c1cncn1C(F)(F)F)=O Cc1ccc(C(N2CCCN(S(C)(=O)=O)CC2)C(=O)NCCC#N)c(C)c1 C=CCCC(F)(F)C(=O)NCC1CC1CNC(=O)C=Cc1cncc(O)c1 C1(CNC(C2C(OCC)C2)=O)CCC(NC(=O)CCN(S(C)(=O)=O)C)C1 c1(C(N2CCCC(n3cc(C4CCOC4)nn3)CC2)=O)cc(F)c(F)cc1Br C12(C(=O)NC3CC(CCNC(C=CC(CC)C)=O)C3)CCC(=O)N1CCS2 N1(C(CC(CC)C2CC2)=O)CC(C)C(C)(C(=O)NCCCOC)C1 C#Cc1ccc(C(=O)NC2CN(C(=O)C(C)NC=O)CC2C(F)F)c(OC)c1 N1(C(c2c(F)cc(Br)cc2F)=O)CCCC12CCN(C(C1CC1F)=O)C2 c1(C(N2CCC(O)(C(C)NC(c3cnsn3)=O)CC2)=O)cnc2ccccc2c1 CC1(SC(F)F)CCN(CC(=O)NCC(F)F)C1 n1(C(C)C)ccc(C(=O)N(CC(C)NC(=O)CC(O)CC2CC2)C)cc1=O c1(S)ccccc1.C(=O)(C(C)n1cccn1)NCC(C(C1(C(=O)N)CC1)C)C1CC1 C(=O)(C(F)(F)C(F)(F)C(F)F)N1CCC(C(C)NC(c2cc(Cl)ncc2O)=O)C1 C=C1CC2(C1)CN(C(C1CN(C)CCN1C(C1CCN(CC)CC1)=O)=O)C2 CC(O)CC(C(=O)O)NC(c1ncoc1C(=O)OC(C)(C)C)=O c1(C(=O)NC(C)CN(C)C(C2CN(S(C)(=O)=O)C2)=O)cccc(C(=O)N(C)C)c1 c1(NCC2(C(=O)Nc3ccc(CC)cc3C)CC2)cnc(C#N)c(C#N)n1 c1(OC)c(CN(C2CC2)CC2(C)CCOC2c2ccccc2)c(C)nn1C n1(CC)cc(Cl)cc1C(=O)N(CCCNC(=O)Cc1nnc(C)o1)C(C)C C(=O)(CCCCCF)NC1(CN(C(c2c(C)onc2CC2CC2)=O)C)CC1 N1(C(CCC)=O)CCN(C(c2cnn(C)c2Cc2ccccc2)=O)CC(O)C1 N1(C(C(C(C)C)OC)=O)CC2OCCN(C(c3ccc(C(F)F)s3)=O)C2C1 C1(C(=O)NC(C(C)C)(C)CNC(=O)CCNC(N)=O)Cc2ccccc2C1(C)C Cc1cnc(C(=O)NCC2CCN(C(c3cc(F)ccc3N)=O)CC2C)c(C)c1 C(=O)(CC(C)C(=O)N1CC(=O)NCC1C(=O)NCC1CCCO1)OC c1(C(=O)NCC2N(C(CC3CCC(C)(C)O3)=O)CC=C2)cc(Br)cnc1O c1(CCC(=O)N(CCCCN(C(=O)C(C)(C)C#N)C)C)ccc(OCCF)cc1 Cc1cccc(Br)c1C(C(=O)N1CCC1C(C)C)NC(=O)C(F)n1ccnc1 Cc1ccc(C2=CCN(C)CC2)c2nc(C(N3CCCC3C)=O)cn12 C1(F)(C(N2CCC(NC(c3sc(CC)c(C)c3)=O)C2)=O)CS(=O)(=O)CC12CCC2 c1(OC)ccc2cc(C=CC(N3CCN(c4ncncc4C)C4CC34)=O)ccc2c1 N1(C(CN2CCC(C)(C)C2)=O)CC2(CC(NC3CCOCC3)C2)C1 C1(C(N(C2CC(NC(=O)Cc3c(F)cccc3F)C2)C)=O)CC2(CCCCO2)C1 N1(C(C2=CCN(C(C(COC)COC)=O)C2)=O)CC2CC(C)(C)C2C1 Cc1ncncc1C(=O)N(CCCNC(c1cn(Cc2cccs2)nn1)=O)C c1(OC)ccc(Cl)cc1C=CC(=O)NCCC(C)NC(=O)C(C)N(C)C N1(C(c2c(C)n(C)cn2)=O)CC(F)(F)CC1CCNC(=O)CCSCC(C)C c1(CNC(=O)NC(c2cccnc2)CC=C)ccc(Cl)c(O)c1 Cc1cc(NC(=O)NCC(CN(C)C)N(C)C)cn2ccnc12 C1(CC(N2CCN(C(C(CC(=C)C)C)=O)CC2CC)=O)SC2=NCCN2C1=O N1(C(C2COCCN(C)C2)=O)CC(NC(=O)CC2CSCCO2)CC2(CCC2)C1 c1(C(=O)NCC2CC(NC(C=CCOC)=O)C2)cccn(C2CCC2)c1=O c1(C(N2C(CCNC(C3(SC)CCC3)=O)CSCC2)=O)cc(C)cc(C)c1O c1(OCC(=O)OC)ccc(C(N2CC=CC2CNC(=O)CC2(C)OCCO2)=O)cc1 N1(C(C)C)CCCC(C(N2CCOCC2CNC(=O)CC2(C)CC2)=O)C1 O=C(C1=NOC2(CCC2)C1)N1CC2CC(C1)N(C(c1cccc[n+]1[O-])=O)C2 C(C(C)C(=O)N1CCC(CN(C(=O)Cc2cnn(C)c2)C)C1)OC N1(C(c2ccc(CC)[nH]2)=O)CC2CC2(NC(=O)Cc2cc(Br)cs2)C1 N1(C(c2cnco2)=O)CCN(Cc2cc(-c3ccccc3)ccn2)C(CO)C1 Cc1ccc2nc(CCCNC(=O)C=CC(N3CCOCC3)=O)[nH]c2c1C N1(C(C(C)NC(C)(C)C)=O)CCCCCC1CNC(c1cc(CCCO)on1)=O C1(CCNC(c2cnc(O)s2)=O)CN(C(=O)C(c2ccccn2)O)CCCO1 c1(CC)cc(C(N2CCC(CNC(=O)Cc3cccc(C)c3)CC2)=O)cc(O)n1 C1(NC(Cc2cccc(OC)n2)=O)CCC(C)N(C(c2cccs2)=O)C1 c1(SC(CNC(CC2C(CNC(=O)CN3CCNC3=O)C2)=O)O)ccc(F)cc1 C1(CC=C)(C(=O)NC2CN(C(=O)CCCCC3CC3)CC2C(F)F)CCOCC1 c1(C(=O)NCC(C)N(C(=O)Cc2nc[nH]n2)CC)cc2cccnc2[nH]1 N1(C(COCCC(C)C)=O)CC2CC2(CNC(=O)CC2CCNC2=O)C1 C(=O)(C1=CC2CCCCC12)NC1CC2(C(NC(c3ccc(C#C)cc3)=O)C2)C1 c1(C(=O)NCCC2CCN(C(CC3CC(CC)C3)=O)C2)c(C)sc2ccccc12 C1(C)(NC(C2CCC(C)O2)=O)CCN(C(c2cn(CCCF)nn2)=O)C1 C1(F)(C(NOCC2CC(=C)C2)=O)CCCN(C(c2cnc(CC)s2)=O)C1 CC(CCC(=O)NCC1(CO)CC=CC1)NC(=O)Cc1cncs1 CCCCCCCCCC(C)CC(=O)N(CCCCCNC(=O)C(C)C(=O)OC)C N1(C(c2sc(F)cc2Br)=O)Cc2ccccc2OC2(CCOC2)C1 N1(C(Cc2nc(C)[nH]n2)=O)CCCC2(CNC(=O)CC3CCC(O)C3)CCCC12 C1(NC(C(c2cccnc2)NC(=O)Cc2nocc2C)=O)CCC2CC12 Cc1nc(C)n(CC(N2CCN(CCNC(C3C(C)C3C)=O)CC2)=O)n1 C#CCC(O)C(=O)NC(C)C(C)(C)NC(=O)C(CO)NC(=O)C(C)C CCCC(CCCNC(C12CCCCC1C2)=O)NC(c1cncc(N)c1C)=O C(=O)(CCN(C(C1(n2nccn2)CC1)=O)C1CC1)NC(c1cccs1)C C1(CC(=O)NC2CC(NC(Cn3c(C)nnn3)=O)C2)CC(O)C1(C)C.C1(C)CC1 c1(SC)nc(C(=O)NC2CC(CNC(C3CCCN3C(C)=O)=O)C2)cs1 N1(C(NC(NCC(C)Oc2ccco2)=S)=O)Cc2[nH]nc(Cc3ccco3)c2C1 N1(C(C2CC(O)(CC#C)C2)=O)CC2(C)CC1(C(N1CCN(C3CCC3)C1)=O)C2 N1(C(C(F)=CC)=O)CC(CNC(c2oc(C)cc2C)=O)C(C)C1 N1(C(COCCCC)=O)CC2CCN(C(c3ccc(OC)c(C)c3)=O)C(C2)C1 Cc1ccccc1CC(N1CCC(CF)(NC(c2csc(F)c2)=O)C1)=O C(CC(=O)NCC12CC(CN1C(c1ccc(Cl)c(C)c1)=O)C2)(C(C)C)OCC N1(C(C2CCN(C(C)N(C)C)CC2)C(=O)NC2CCC2)CCCC(C)(CSC)C1 CC1=C(C(=O)NC(C)C(C)NC(=O)C#CC(=O)N(C)C)SCCO1 c1(C(N2CC(NC(Cc3c(C)nc(C)s3)=O)C(O)C2)=O)nccc(C#N)c1F c1(C(N2C(C(=O)Nc3cncc(OC)c3)CC2)=O)cnc2[nH]ccc2c1 C1(F)(CNC(=O)CCc2cncs2)CN(C(c2cnn(-c3nccs3)c2)=O)C1 c1(N2C3CN(C(c4ccc(Cl)c(C)c4F)=O)C(C3)C2)nc(Cl)c2c(ccn2C)n1 C1(NC(c2cc(F)cc3cc[nH]c23)=O)C2CC3CN(C(C4CC4F)=O)C1C3C2 C(CC(=O)NCC1CCCCN1C(c1ccsc1Cl)=O)(C(N)=O)NC(C)=O Cn1ncc2c(NC(C3(O)CCN(C(C4CCC45CCC5)=O)CC3)=O)ncnc12 C1(C(=O)NC(C)CCCCNC(=O)CCP(C)(C)=O)COc2ccc(F)cc2C1 Cn1cc(I)c2c(C(=O)NCc3ccncc3N3CCCC3)ncnc12 c1(C(=O)NCCNC(CC2N(C)CCCC2)=O)ccc2[nH]c(=O)c(=O)[nH]c2c1 C1(C(=O)NCCCC(C)(C)NC(CCCOCCC)=O)CCCC(F)(F)C1 c1(C(=O)NCCC2CCN(C(C(C=C)c3ccccc3)=O)C2)cccc[n+]1[O-] c1(C(=O)NC2CCCC(C(N3CCC(C(C)C)CC3)=O)C2)cnc(OC)c(F)c1 O=C1CCCC(C(=O)NC2CCCC(NC(=O)CSc3cn[nH]c3)C2)C1 C(=O)(C1=Cc2ccccc2C1O)NCC(CO)NC(c1c(N)cncc1)=O CC1CN(C(C2SCCS2)=O)CCN(C(=O)C(c2cnn(C)c2)O)C1 c1(C(=O)NC2C=CC(CNC(C(C)(C)c3cnco3)=O)C2)ncccc1F CC1CN(C(c2cn(CCO)nn2)=O)CCC1NC(=O)C(F)C1CCCC1 N1(C(CC2(OCC)CC2)=O)CC(C)CN(C(c2cc(C)sc2C)=O)C(C)C1 c1(CC(=O)N(CCC)CCNC(=O)C=CSc2ccccc2)cccc(Cl)c1F C=C1CC(C(=O)NCCC(=O)NC(C(=O)N(CCCC)CCCC)C)(C(F)F)C1 c1(N2CCC(C=C)C2)nc2c(c(=NC(C)CC(C)C)[nH]1)CCC2 N1(C(C2C(COC)(CNC(C3(C)CC3)=O)C2)=O)CC2CC1C2CO C1(C(=O)NC2CC(C(N)=O)OCC2)CCC(F)(F)CC1 C=CC(CCC)CC(=O)N1CC2C(NC(c3c[nH]c4nccc-4c3)=O)C2C1 Cc1c(Br)cnn1CC(=O)NC1CC(NC(C2CCCSC2C)=O)C1 CN1CCC(NC(C2(CO)CCN(C(=O)CCOCC(F)F)C2)=O)C1=O C(=O)(C#CC(C)(C)C)NC(C(=O)NCC(C)OCC=C)CCSC c1(CC)[nH]nc(C(=O)NC2CCC(C)N(C(=O)CCc3nncs3)C2)c1[N+](=O)[O-] S(=O)(=O)(c1ccc2cc(Br)ccc2c1)NC1(CN(C)C)CCCC1 C12(NC(C3CCN(C(C(C)NC=O)=O)C3)=O)CCCCC1C2 N1(C(c2c(C)ncs2)=O)CC2CCCC(NC(=O)CC(C)n3ccnc3)C2C1 Cc1cccc2c(N3CC4C(C(N5C6CCC5CNC6)=O)C4C3)ncnc12 C1(COC)CN(C(c2nc(=O)n(C)[nH]2)=O)CCN1C(=O)C(O)Cc1cnc[nH]1 N1(C(CC2N(C(c3cc(C(C)C)no3)=O)CCCC2)=O)CC(C)OC(C)(C)C1C C1(CNC(CCOCCN(C)C)=O)CN(C(c2cn(C3CC3)cn2)=O)CC1C Cc1cc([N+](=O)[O-])ccc1C(N1CC(C)(c2cn(-c3ccc(CO)cc3)nn2)C1)=O C(CC(C(C)(C)C)NC(C1CC2CCC1CC2)=O)N(C(C(SC)SC)=O)C CN1C(=O)NCC1C(N1CCCC(CNc2nccc(C(F)(F)F)n2)C1)=O C(=O)(C(F)(F)C(O)CC)NCC1N(C(c2cn(CCC=C)nn2)=O)CCCC1C c1(C(=O)NCCN(C(C2CC3CCC23)=O)C2CC2)ccnc(OCC(F)(F)F)c1 N#CC1CCN(C(=O)CCC2CCCN2Cc2cnc(O)c(Cl)c2)CC1 N1(c2cc(C)ncn2)CCN(C(C2(c3cnccn3)CC2)=O)CC1C(C)C C(=O)(C#Cc1ccccc1)Nc1ccc(Oc2ccc(C)c(C)c2)c(F)c1 c1(CN2CCNCC2)ccc(CN(C(=O)C(=O)NC2CC23CC3(F)F)CC)cc1 C12(C(=O)OC)CC3CC(C1)CC(F)(C3)C2.C12CC3CCC1N(C3)C2=O C1(C(=O)NCCC2CCCCC2)(CNC(=O)CCc2ccco2)CCCO1 c1(N2CCC(CN(C(=O)C=CC3CCC3)C(C)C3CC3)C2)nccc(S(C)(=O)=O)n1 C1(CC(=O)N(C2(C(=O)OC)CC2)C)CN(C(C2CCC(C)C2)=O)C(C)(C)C1 Cc1ccc(C(N2CCC(C)C(NC(=O)CC3CCCC3C)C2)=O)c(C)c1 N12CCC3(CC1)CC3N2Cc1cc(C)nn1C.C(=O)CC(C)C(F)(F)F.C(C)=O CC(CC(N)=O)C(=O)N1CCC(C)(C(=O)NC2(CO)CC2)C1 N#Cc1cccc(CC(=O)N(CCNC(c2ccc(O)nn2)=O)C2CC2)c1 N1(C(=O)Cc2ccco2)CCCC2(C1)CN(C(=O)C(=O)N(CC(F)F)C1CC1)C2 N1(C(CC2(C=C)CCC2)=O)CCC2(CC1)CC(C)N(C(C1CC(C)CO1)=O)C2 c1(C(=O)NCC2COCCN2CC(F)F)nnc(O)cc1O CC1(C)CC(C(=O)NCC2CC[Si](C)(C)C2)CN1C(c1n[nH]c(O)n1)=O N1(C(C2(C#C)CN(C(=O)C=C3CCC3)C2)=O)CC2(CCC2)OCC1C c1(NC(c2n(C(CC)(C)C)nnn2)(C)CSC)ccc(O)cc1OC c12cc(nc(C)c1)S2.c1(CC)cccc(Nc2ccc(C(N)=O)nc2)c1 CC(CC(F)F)C(=O)N1CC2CC(NC(=O)CCN3CCCC3=O)C1C2 c1(CN2CCC(C(=O)NC(C(C)C)CCO)C(O)C2)ccc([N+](=O)[O-])c(O)c1 C1(C(=O)NCC(C)(CO)NC(c2ccc(OC)nn2)=O)CCC(C2CC2)CC1 c1(N)ncoc1C1CN(C(=O)CCNc2ccccc2)C1.CC(C)C(=O)NCC N1(C(CCc2c(C)n[nH]c2C)=O)CCC(C)(C)C(NC(=O)Cc2cnco2)C1 C1(NC(c2cc(C)c(C)nn2)=O)CCN(C(C2CN(C(C)C)CCO2)=O)CC(O)C1 C(CCCCC(=O)NC(CO)CCF)N(C(c1cc(C2C(C)C2)[nH]n1)=O)C C(=O)(CC1=CCN(C)CC1)NCCCN(C(Cc1ccc(C)nc1Cl)=O)C c1(NC(C2N(c3c(OC)cncn3)CC(F)C2)=O)ccc(O)c(Br)c1 N1(C(C2CN(C(C3C(C)CCOC3)=O)CC2CO)=O)CCCN(C=O)CC1 N1(C(CC2(COC)CC2)=O)CCOC2(C1)CN(C(C1CCn3nccc3C1)=O)C2 CCCCCCC(=O)NC(CO)C(C)NC(=O)CC12COC(CF)(C1)C2 c1(C(=O)NCCCCCCN(C)C(C2CCOC(=O)N2)=O)cccc(N)c1F Cc1ccc(C(=O)N(CCC(C)NC(C2(c3ccccc3C)CC2)=O)C)cc1O N1(C(C(C)=C2CC2)=O)CC2CC1CC2NC(=O)C(C(C)C)n1ccc(C2CC2)n1 C1(OC)CC(NC(=O)C(C)SC)CN(C(c2scnc2C(C)C)=O)C1 C(C(=O)NOCC1CCOC1)NC(COCC#C)=O.C(C(C)(C)C)=C Cn1cc(C(=O)NC2COCC2NC(=O)CC2CCCCCO2)cc1Br N1(C(C=C(CC)C)=O)CCCC2(C1)CN(C(=O)CCc1ccc(Cl)c(C)c1)C2 c1(C(=O)NCC2C(CNC(C3C(C(C)C)(CC)C3)=O)C2)c[nH]c2cccc(Cl)c12 N1(C(c2cnc(C)nc2)=O)CC2CCN(C(C34CC(C(F)(F)F)(C3)C4)=O)CC2C1 CCCCCCC(F)C(=O)NCC(O)CNC(=O)C(C)(C)O c1(C(N2CCCN(C(C3CC(OC)C3)=O)CC2)=O)cc(C)c2c(c1)CCCN2 CS(=O)CCCCNC(C1CCCCC1)c1nnnn1C1(C)CC1 c1(C(=O)NC(CCNC(c2[nH]cc(CC)c2)=O)C)ccnc(C2CC2)n1 C1(C(C)C(=O)NCCCCNC(c2cc(C3CCC3)no2)=O)CCCCCC1 C1(NC(=O)OCC)CC2CCC1CC2NC(c1ccc(C(=O)C(C)(C)C)cc1)=O c1(OC)ccccc1C(CNC(=O)CO)NC(=O)C(c1ccc(Br)s1)C Cc1ccc(Cl)c(N)c1C(N1CCCC1C(=O)N(C1CC(O)C1)C)=O C1(NC(C(C)CN(C)C(C23CCCCC2C3)=O)=O)CCC(=O)N(C)C1=O CC1=C(C(=O)NC2CC(CC(=O)NCC3(CC4CC4)CC3)C2(C)C)CC1 N(C(=NCCSC)NC(c1ccc(CSC)cc1)C)C(CC=C)C C(=O)(C(C)(C)CC(C)C)NCCNC(c1c(C)nncc1)=O C1(n2cc(-c3cc(OC)ns3)nn2)CN(C(c2cc(C)cc(Cl)c2)=O)CCC1C N1(C(C(CC)OC2CCCCC2)=O)CCC(OC2CCCCN2)CC1.C1CS1 c1(OC)cc(C(=O)NC(C2CN(C(c3ncccc3Cl)=O)C2)C)ccc1Br N(C)(C(=NC)N(C)C)CC(F)(F)F.CCCNC C1(NC(=O)NC(CC)(C)Cc2ccccc2)CN(C(=O)OC(C)(C)C)CC1N=[N+]=[N-] N1(C(c2cncc(C)c2)=O)CCC(C)(NC(=O)CC2CC2(Cl)Cl)CC1 C1(CC(N2CC(CC(C)NC(=O)Cc3ccnc(O)c3)C2)=O)CCCS1(=O)=O N1(C(c2cc(OC)nn2C)=O)CCC2C(C1)CN2C(c1ccoc1Br)=O C1(CC=C)(NC(C2CCCCN2CCC)=O)CCN(C(c2cccc(C)c2)=O)C1 N1(C(C(CC)C)=O)CCC(F)(CNC(C2CCCNCC2)=O)CC1 C1(NC(c2c(COC)noc2)=O)CC(C)CN(C(c2csc(CC(C)C)n2)=O)C1 C(=O)(CCCCCN(C(=O)COC(C)(C)CNC1CC(C)OC1=O)C)OC N1(C(c2cscn2)=O)CCC2(CCN(C(c3cc(C(F)F)ccc3F)=O)CC2)C1 N1(C(c2c(C)noc2C)=O)CC(NC(=O)CCc2nncn2C)CC(C)(C)C1 c1(C(N2CCC(O)(C(C)NC(CCCCNC(C)=O)=O)C2)=O)cc2c(s1)CCC2 N1(C(c2cn(C(C)C)nc2)=O)CCC(CNC(C2CCC(C)(C)OC2)=O)CC1C c1(CN(C(C2C(=C)CC2)=O)C)ccc(CNC(c2nnsc2CC)=O)cc1 c1(C(=O)NC2CN(C(Cc3cc(C)ns3)=O)CC(O)C2)nccc2occc12 c1(C(N(C2(COC)CCCC2)C)=O)nc(CNC(c2cnncc2O)=O)oc1C C(=O)(C(C#N)C(C)C)NCCN(C(=O)COCC(C)C)CCOC CC1CC(CNC(=O)CCCn2ccccc2=O)CN1C(=O)CNC(=O)C1CC1 c1(C(=O)NC2(CCOC)CN(C(CSCC=C)=O)C2)ccc2cc[nH]c2c1 Cc1ccc(Br)c(C(=O)NC23CC(CNC(C4(O)CCC4)=O)(C2)C3)c1 c1(C(C(=O)NC2CC(CO)C2)N(C2CCCC2)C2CCCC2)ccc(F)c(Br)c1F C(CC(C)(C)C(=O)N1CCCC(NC(c2cnn(C)c2C(F)F)=O)C1)OC Cc1cccc2cc(C(=O)NCCCCN(C(=O)CCC(C)(C)F)C)[nH]c12 c1(C(C(=O)NC(CC)C)(C)C)ccc(CNC(=O)C(C)NC(C)(C)C)cc1 N1(C(C=C(CC)CC)=O)CCSCC1CCNC(=O)C(C1CCC(=O)N1)C C(=O)(C(Cc1cc[nH]n1)NC(c1coc(C2CC2)n1)=O)N(C1CC2(CC2)C1)C c1(C(N2CCOC(C3CCC3)C2)C(=O)NC2CC(F)(F)C2)ccc2c(c1)CCO2 C1(C(N(CCCC)CC(N)=O)=O)COC2(C1)CN(C(c1cnnn1C(C)C)=O)C2 N1(C(CCC(C)NC(c2c(C)cc(CC)o2)=O)=O)CCC(C)CC1C c1(C(=O)NC2CN(C(C3=CCCC3C)=O)C(C)(C)C2)ccc(N)c([N+](=O)[O-])c1 N1(C(CC2CC(C(=O)OC)NC2)=O)CCNC(=O)CC1(C)C C(=O)(C(CC(F)(F)F)c1ccccc1F)OC.CN1CCC(F)(c2c[nH]nn2)CC1 O=C(CCC(=O)N1CCCC(c2nn[nH]n2)C1)c1cccc(O)c1.Cn1cnn(C)c1=O C=CCC(C)(C(=O)N(C(C)CCNC(=O)CC(c1c(C)n[nH]c1C)C)C)N(C)C c1(CCN(C(C(=O)OC)C2CCCC2)C(C)C)c(C)[nH]c2c(C)cccc12 C1(F)(C(=O)NCCCSCC)CCCN(C(=O)CCCN(C)C(C)=O)C1 c1(C(=O)NC(C(=O)N(CC(CCC)O)C)c2ccoc2)nccc2[nH]ccc12 N1(C(C(C)S(C)(=O)=O)=O)CCC2CN(C(C3CC3C3(C)COC3)=O)C2C1 C1(C)(c2nc(C(N(CC)CC)=O)no2)CCCN(C(=O)NC2CC(F)C(=O)N2)C1 N1(C(c2cccc(CNC(C(C)(C)CCCF)=O)n2)=O)Cc2ccc(O)cc2C1 CC(C(C)(C)NC(C1C=CCS1)=O)NC(=O)CCNC(N)=O Cc1c(C(NC2COc3ccc(F)cc32)=O)oc(=O)c2ccccc12 c1(C(=O)NC2C(NC(=O)CCc3cnoc3)CC2)cc2ccc(Cl)cc2o1 Cn1nc([N+](=O)[O-])cc1C(N1CCN(C(C2C=CCCC2)=O)CC1C(C)(C)C)=O n1(CC(=O)NC(CNC(C2(OC)CCSCC2)=O)CC(C)C)ccc([N+](=O)[O-])n1 N1(CC)CCN(C(=O)CC2C3CCC(C3)N2C(=O)Cn2cnc(C#N)n2)CC1=O CN1CCCCC1CC(=O)NCCCOC1CCN(C(c2ccns2)=O)CC1 N1(C(Cc2c(C)ocn2)=O)CC(C)CN(C(C23CC4CC2C3C4(F)F)=O)C(C)C1 CCCCCC(C)(C)C(=O)NC1CCCC1CNC(c1ccc(NC=O)cc1)=O N1(C(C=CC=CCC)=O)CC2CCCC2(NC(c2ccc(SCCC)cc2)=O)C1 N1(C(CCCCOCC)=O)CC(O)CCC1C(=O)NC1C=CCCCC1 C1(C(N2CCC(NC(CC)=O)C2C)=O)Cc2cc(Cl)ccc2O1 Cc1cc(C(N2CCCC2(C)CNC(=O)C2=CCCCCC2)=O)cc2ccoc12 N1(C(c2nn(C)c(C(N)=O)c2)=O)CC2(CCCCN2C(C2CCC(O)C2)=O)C1 C1(C(=O)NCCC2N(C(COCCSC)=O)CCC2)CS(=O)(=O)CC(=O)N1 C(C1=CCN(C(=O)C(c2ccc(Cl)cn2)(F)F)CC1)NC(c1cnn(C)c1F)=O c1(C(N2C(C(C)C)C(NC(=O)CCCNC(N)=O)CC2)=O)cc(F)cnc1O c1(C(=O)NC(C)CC(C)NC(C2(C3CCCO3)CCCC2)=O)ccc(N)cc1F CC1CN(C(=O)CNC(c2ccoc2)=O)CC1NC(=O)C(CO)N(C)C C(=O)(C1=NNC(C(F)(F)F)C1)N1CC(C)C(NC(=O)C(C)(C)c2cnco2)C1 C1(COC)(CNC(C23CC(F)C2C3)=O)CCCN1C(=O)CCN1CCOCC1 c1(C(=O)NC2C(NC(c3cc(C)sc3C)=O)CC2)csc2c1CCCCCC2 C(CC1=CCN(C(C2(n3cncn3)CC2)=O)CC1)NC(c1nccc(C#C)c1)=O c1(C(=O)NCc2cc(O)ccc2Cl)ccc2c(c1)CN(Cc1cc(I)c[nH]1)CC2 C(CC(C(=O)NCC1CCC(=O)N1)NC(=O)CC(Cl)Cl)OCC CC(CC1CC1)C(=O)N(CCCOCCNC(=O)C(c1cnn(C)c1)C)C C1(O)(CN(C(C2(NC(C)=O)CCC2)=O)C)CN(C(C2CC(C(F)(F)F)C2)=O)C1 N1(C(=O)Cc2ccoc2)CCC(C2CCCN2C(c2ccc(Br)o2)=O)C1 c1(C(=O)OC)cccc(C(N2CCOC(CNC(C3CN(C)CCO3)=O)C2)=O)n1 c1(NC(=O)NC2C3CN(C(CC(C)=C(C)C)=O)C2C3)cc(F)ccc1F c1(CC(=O)NCC(C)N(C(c2cccc(COC)c2)=O)C)cccc(C)c1F N1(C(CC23C(CN(C(C(CC)NC)=O)C2)CC3)=O)CCC2CNC(=O)C2C1 c1(C(C(=O)NCC=CCNC(C(c2cccc(F)c2)(C)O)=O)O)cccc(Cl)c1 C1(C(=O)NC(CC)CCOC)CCOCCN1C(c1cc(F)ccc1OC)=O N1(C(=O)C2=NOCC2)CCNC(C(=O)NCC(O)Cc2ccc(F)cc2)C1 N1(C(CCCCCC)=O)CCC2(CCC2NC(=O)C(CC2CCC2)OC)CC1 C(CC(CC)C(=O)N1CC(CO)(NC(c2nc(Cl)sc2Cl)=O)C1)=CC n1(-c2cc(C)on2)c(C)cc(CNCC(Cc2cccc(Cl)c2)CO)c1C Cc1c(NC(C2(F)CCN(Cc3cc4ccccc4s3)C2)=O)cccc1[N+](=O)[O-] CC1CN(C(c2ccccc2CC(C)(C)C)=O)CC1NC(C1(C)CCC(C)C1)=O c1(CNc2ccc(C(=O)NC(C)(C)C)nc2)cc2cnn(C(C)(C)C)c2nc1Cl CN=c1nc(N2CCC(C(C)(C)OC)C2)[nH]c(=NCC2CCC(SC)CC2)[nH]1 C1(C(N2CCC(NC(CCOCCOCC)=O)C2)=O)CCC(CCCCC)CC1 N1(C(c2nc(C)[nH]n2)=O)CC(C)N(C(=O)Cn2cccc(O)c2=O)CC1C N1(C(C2N(C(C)=O)CC(O)C2)=O)CCCC(C)(C)C1CNC(=O)CC1C=CCC1 C1(Cc2cn(CC3CC(O)(CO)C3)nn2)CN(Cc2c(C)cccc2)CC1(F)F C1(CCNC(c2n(CCC)ccc2)=O)CN(C(=O)CC2C=CCC2)CCS1(=O)=O C1(C(=O)NCCN(C(c2n[nH]cc2C)=O)CC)CC2CCCC(C1)C2=O Cn1ccc(C(N2CCSCC2C(=O)NCCN2CC3CC3C2)=O)cc1=O c1(CN(CC)Cc2ccc(OCC)cc2)cc(I)cc(I)c1Br c1(N2CCC(OC)C(C)C2)nc(=NC)nc(N(CC2=CCSC2)C)[nH]1 C1(C(=O)NCc2ccc(C)nn2)CCN(C(=O)C(C)c2ccn(C)n2)O1 C(=O)(CCN(CC(C)C)N1CCCC1C(=O)NC)Nc1ccc(C)cc1 c12cc(cc(F)c1)C(=O)NCC1CCN1C2=O.C1(C(=O)OC)CCC(C(N)=O)C1 CC1CN(C(c2sccc2CNC(c2cnccn2)=O)=O)CC1(C)CO CCN=C(NCC1CCN(c2ccccc2)C1)N1CC2C(C(F)F)C2C1 N1(C(CCC(=O)NCC)=O)CCC2(CCN(C(c3[nH]cnc3C)=O)C2)C1 CC1OC23CC1(C2)NC(=O)C3(C)C.C1(OC(C)(C)C)CCC1 C1(NC(C(C)=C(CC)C)=O)CN(C(c2ccc(CC)cc2)=O)CC1OC C12(CNC(c3cn4ncccc4n3)=O)CCCC(CN1C(c1csc(Cl)n1)=O)C2 C1(OC)CC(NC(c2ccc(O)nc2C)=O)CN(C(C2(OC)CCCCC2)=O)C1 Cc1cccc(C)c1C(N1CCN(CC(N2CCOC(CF)C2)=O)C(=O)C1)=O c1(SC)cc(N2CCCCC2CNC(c2cc[n+]([O-])cc2)=O)ncn1 CCC(CC)C(C)C(=O)N1C(C(=O)NC2CCCC23CC3)CCC12CC2 Cn1ccc2c(C(=O)NCC(c3ccno3)O)cccc12 c1(OCCC(=O)NC2CCCN(C(C3CCCCS3)=O)CC2)ccc(Cl)c(F)c1 c1(OC(C)C)cnc(C(=O)NCCSC2CCN2C2CCCC2)c(Cl)c1 C=C(C)CC(C(=O)NCC1CC(NC(c2ccncc2)=O)C1)NC(C)=O c1(NC(c2scc(C(N)=O)c2)=O)cc(Cl)ccc1I CN1CC(C(=O)NC2COCC2NC(C2(CF)CC2)=O)CC1=O C=CC(CC)CC(=O)NC(C1CCCN(C(=O)C(C)NC(=O)C2CC2)C1)C N1(C(CSCCC)=O)CCC(N(C(=O)COCCCF)CCC)C1 N1(C(CC2CCC(NC(c3cc(C)nc(O)c3)=O)C2)=O)CC(O)C2(CCCC2)C1 S(=O)(=O)(c1ccc(Cl)cc1)NCC(N1CCN(C(C2CC2Cl)=O)CC1)=O Cc1cc(C(=O)NC(C)(C)CN2CCN(C(C3(F)CCC3)=O)CC2)cnc1O C1(C(N2CC(CNC(c3cn(CC(=O)OC)nn3)=O)C2)=O)CCCC2CCCN12 C1(NC(C2C(=C)C2)=O)CC(NC(=O)C(C)(C)CSC)CC1O C1(C(=O)NCC(C)N(C)C)C(C2CCOCC2)C1(C)C c1(OC)cc(NC(C2CCN(C(=O)C(C)C(=O)OC)C2)=O)ccc1F C(=O)(C(O)C(O)C(=O)O)N1CC(c2cn(CC(=O)OC)nn2)C1 c1(NC(C23CC(C(N4CCC5(CC4)CC5)=O)(C2)C3)=O)ccc2nncn2n1 c1(C(=O)NCCNC(C(CC)CC2CCCC2)=O)cnn2c(Cl)cccc12 Cc1cc2cccc(C(=O)NC3CC(CC(=O)Nc4nccc(C)c4Br)C3)c2[nH]1 C1(NC(C2N(CC)CCC2)=O)CCN(C(c2cnn3ccn(C)c23)=O)C12CCC2 N1(C(c2cnc(OCC)s2)=O)CC(NC(c2cc(C)n(C)c2C)=O)C2(CCC2)C1 C1(N(C(C(CC#C)O)=O)C)CCCN(C(=O)Cc2nc(C)sc2Cl)CC1 C1(CNC(c2cc(-c3cccs3)on2)=O)CC2(CCN(C(=O)CCF)C2)CO1 C(=O)(C1=NOC2COCC12)N1CCC(NC(C2C(CC)OCC2)=O)C(C)C1 Cc1cc(F)cnc1C(=O)NC(C(N1CC(CO)C(O)C1)=O)c1ccco1 CC(C)(O)CC(=O)NCc1c[nH]nc1C1CCN(C(=O)CC2CCCO2)C1 N1(N(C(=O)C(N2CCC(CCC#N)CC2)=O)C)CC(SCC)Oc2ccccc21 C1(COC(=O)CCc2nnc(-c3cncc(Br)c3)o2)CCC2(CCCCCC2)O1 c1(C(N2CC(N(C(c3cccc(OC(F)(F)F)c3)C)C)C2)=O)ccnc(SC)c1 c1(C(=O)NCC2CC(NC(C3(OCC)CC3)=O)C2)cnccc1C(F)F CCC(C)C(O)C(=O)NC1CN(C(=O)Cc2csc(-c3ccoc3)n2)CC1C C12(NC(C=C(COC)C)=O)CCC(C1)N(C(c1cc(SC)oc1C)=O)C2 C(CCC(=O)NC(C)CCCNC(c1coc(C(=O)OC)n1)=O)OCCC CC1(C)CC(CNC(C2CC(C)(C)C2)=O)N(C(c2cccn2Cc2cccs2)=O)C1 c1(C(=O)NCC(CC=C)NC(=O)CCc2cccs2)ccc(OC(C)C)cc1C C1(C(C)NC(=O)C(n2cc(Cl)cn2)C)CCN(C(C2CC2(Cl)Cl)=O)CC1 n1(CC)ccc(C(=O)NCCn2cc(C(=O)NCCS(C)(=N)=O)nn2)n1 C(COC)(C(=O)NC(C)C)N(CCNC(CSC)=O)C.C1CS1 C=CCCCCCCC(=O)N1CCCC1C1(C(=O)Nc2cnn(CCOC)c2)CC1 Cc1ncn(C)c(=O)c1C(=O)NCC(C1CCC1)NC(=O)COC(F)(F)F c1(C(=O)NCCCN(C(CCCC2C(C)C2)=O)CCO)occ2c1CCC2 c1(C(C(=O)NCCCC2CC2)N(CC(=O)OC)C2CC2)ccc(C)c(Br)n1 c1(C(N2CCC(C(C)NC(c3cnn(C)c3C(F)F)=O)C2)=O)ccc(N)c(F)n1 C1(C)(CC)CCN(C(C2COCCC2NC(=O)CC2(N(C)C)CC2)=O)C1 C1(NC(=O)Cn2ncnn2)COC2CN(C(c3cnc[nH]3)=O)CC12 N1(C(c2scc(C)c2)=O)CC2CCN(C(=O)CCC3CCN(C)C3)C2C1C CN(C(C)c1cnn(C)c1)N1CCC(F)(F)C(C#N)C1 C1(OC)COCCC1(c1nnnn1C)NCCCSc1ccc(OC)cc1 C(C(C)(C)C(=O)N1CCC(C(O)CNC(c2cc(Cl)ns2)=O)CC1)OCC CCC(C)(C(=O)NCCC(C)NC(=O)CC1(NC(C)=O)CC1)C(N)=O c1(C(=O)OC2C(C)CN(C(=O)OC(C)(C)C)CC2)cc(Br)cc([N+](=O)[O-])c1 C(=O)(C1=CCCCO1)NC(CNC(c1nc(C(C)OCC)sc1)=O)CC N1(C(C(C)(C)c2ccccn2)=O)CC2CCCC(C1)N2C(=O)CC#N CCCCC(C)C(=O)NCCCCC1CCN(C(C2OCC2(C)C)=O)CC1 C(=O)(CCCCCN(C(=O)C(CC1CC1)OC)C)NC(CCC=C)C c1(C(=O)NC2CC3(CCOCC3)O2)cccc2c1CCO2 c1(C(=O)O)ccnc(N2CCN(Cc3cccnc3O)CC2)c1 CON1CCC(C(=O)N(CC(O)CN(C)C(C2(F)CCOC2)=O)C)CC1 N1(C(c2c(C)n(C)cc2)=O)CCCC(C)(C(=O)NC2CCOCC2F)C1 c1(OC)c(CN2CCCC(N3CCC3)C2)ccc2ccccc12 C(C(O)C(CC)CC)NC(CC1N(C(C(CC=C)NC(C)=O)=O)CC1)=O C(C)(CCCC(=O)NCC1CC12CC2)NC(Cc1c(C)cccc1)=O CN1C(=O)OC2CN(C(C3(NC(=O)C4=NOCC4)CCC(C)(C)C3)=O)CC12 N1(C(C(CN(C)C)(C)C)=O)CCC2(NC(=O)CSS(C)(=O)=O)CCCC12 C1(C(=O)NCCC2CC(O)C2)(CC)CCN(C(=O)CCC2CCCOC2)C1 NS(=O)(=O)N1CCC(C(=O)NCCn2cc(Cc3nncn3C(F)F)nn2)CC1 N1(C(CCc2c(C)n[nH]c2C)=O)CC2(CCN(C(C3CC(=O)C3)=O)CC2)CC1C N1(C(C(CC2CCC2)NC(=O)COC2CCCC2)=O)CCc2ncsc2C1 N1(C(CSCC)=O)CCC(C(C)NC(=O)CCc2c(C)noc2Cl)CC1 C1(C(=O)NCCCOC2CCN(C(C(C(C)C)O)=O)CC2)CC2OC(=O)OC2C1 c1(OCC)cccc(-n2c(-n3nc(C)nc3C)cnc2NC(CO)CCCN)c1 C(C(C)C(C)C(=O)Nc1cnn(CC(N2CCC(O)CC2)=O)c1C)OC C1(C(=O)N)CCC(C(CCCCCNC(=O)C=C2CCCC2)C2CC2)CC1.CO C1(C(N(C)CC2CC2)=O)CN(C(=O)C(C)(C)n2cccn2)CC1F c1(OC)ccnc(NC(C2C(CNC(c3cc(CO)ccn3)=O)C2(C)C)=O)c1 O(NC(=O)CNC(=O)CC(C)SC)CCOCC#C.C1(=O)CN1CC C(=O)(C(O)C(F)(F)F)N(C)CC1CCN(C(C2(CC)CCOC2)=O)CC1 c1(C(N2CC(NC(COC(CC)C)=O)(COC)C2)=O)cc(C(N)=O)ccc1C c1(C(=O)NCC2CCN(c3ncnc4cnccc34)C2)cccc2nccnc12 Cc1nn2c(C(=O)NC3CCCCC3NC(=O)CC3OCCCO3)c(C)nc2s1 C1(C(=O)NCCCCCN(C(CCCOCC)=O)C)CCCN2CCCC12 c1(C(N2C(C)COCC2)=O)n[nH]c2c1CN(C)CC2 n1(CC)c(C(=O)NC2CN(C(c3onc(C)c3C)=O)CC2C)cnc1O c1(C(=O)NC2(C3N(C(c4nc(SC)sc4)=O)CCC3)CC2)ccc2ncnn2c1 C1(OC)CC(CNC(c2ccc(CSC)o2)=O)N(C(=O)C(C)Sn2ccnn2)C1 C1(CC(=O)Nc2cncc(CNC(COCCOC)=O)c2)COC(C)(C)CO1 c1(C(N(C2CCCN(C(=O)CCc3cccnc3)C2)CC)=O)cc(Br)cnc1O C1(C(=O)NCC2OCCN(C(c3ccc(OC)nn3)=O)C2)C2CCC3C(C2)CC13 C1(CNC(C2CCCN(C)C2)=O)CC2CCC1N2C(=O)CCc1cccnc1 C1(CN(C(CCOCC)=O)C)CCCCN1C(=O)CC(C)n1cccn1 c1(CN(CCOC)CCO)cc(Cl)ccc1Cl.C1(=O)C(OC)CN1 N1(C(COCC)=O)CCC(CCNC(=O)Cc2cccc(Cl)c2F)CC1C Nc1cc(F)ccc1C(=O)NC1CCN(C(C2C(Cl)(Cl)C23CC3)=O)CC1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(C)(C)CC(=O)Nc1cccc(C(F)F)c1 C1(NC(c2ccc(-c3cn(C)nc3)o2)=O)C2CCCC1COC2 N1(C(C(C=C)(C)O)=O)CCn2ncc(C(F)(F)F)c2C1 C1(NC(CCCCC)=O)CN(C(C23CSCC2C3)=O)Cc2nccn2C1 Cn1nc(C(N2CCC(C)(CNC(C3CCCSC3)=O)C2)=O)cc1Br C#CC1(NC(c2cc(CNC(c3csnn3)=O)nn2C)=O)CCCCC1 n1(CC=C)cc(C(=O)N(C(CSC(C)(CC)C2CC2)C(=O)NC)C2CC2)nn1 CC1CC(NCc2ccsc2)CN(C(c2cccc(O)c2)=O)C1 c1(C(=O)NC(c2ccc3c(c2)CCCC3)C(=O)OC)c[nH]c2c(Cl)cc(Cl)cc12 N1(C(COCCC=C)=O)CCN(C(=O)CC(C)OCCCC)CC1CC N1(C(c2cc(C)n(C)n2)=O)CC(NC(C2CCC3(CCC3)O2)=O)CC(O)C1 c1(C(N2CCC(CCNC(C3(N(C)C)CC3)=O)C2)=O)cc(Cl)nc(Cl)c1 N1(C(c2ccccc2CC(F)(F)F)C(=O)NC(CC)C)CC2CCC2(OC)C1 c1(C(=O)NCC2(O)CN(C(C3(CC#C)CCCCO3)=O)C2)coc(S(N)(=O)=O)c1 C1(C)(CNC(CCSCCC)=O)COCCN(C(=O)C2=CCC(C)CC2)C1 N1(CC)CCCC(N2CCC2)C1.C1CCC(=O)N2CC(C)(C2)C(=O)N1CC Cc1ccc(-c2ccc(C(=O)NCc3cc(Cl)ccc3I)nc2)c(CO)c1 c1(CNC2C(C(=O)Nc3ccc(C=C)cc3)C2)cc(OC(C)C)c(OC)c(F)c1 c1(C(N2CCC(C(C)NC(CC=CC)=O)C2)=O)cnc(Cl)cn1 CN1CCc2nc(C(N3CCCC(CNC(C4C=CC=CC=C4)=O)C3)=O)sc2C1 C(=O)(CS(=O)C(F)(F)F)N(CC(C)NC(=O)CCn1cnccc1=O)C N1(C(CCNC(C2C(C)C2)=O)=O)CC2(CC(NC(=O)CC3COCCO3)C2)C1 c1(OC)ccc(C(=O)NCC(CNC(C2(C)COC(=O)C2)=O)CO)c(F)c1F N1(C(C(=O)NCCOCCCC)=O)CCC2(CCC2CNC(=O)C=CCF)CC1 Cc1ncnc(C(=O)NCC2CCN(C(=O)C=CC3CCC3)C2(C)C)c1C n1(CC(=O)NCC(O)CNC(=O)CSC2CCS(=O)(=O)C2)c(O)nnc1O CC(CC(F)(F)F)C(=O)NCCOC(C)(C)CNC(=O)CSC(C)C CC1(C)CN(C(=O)C2=COCCO2)CCC1NC(c1cc(Cl)cc(F)c1N)=O C(=O)(C(O)(C(F)(F)F)c1cn(C2CCOCC2)nn1)N(CC(=O)O)C1CC1 c1(OC)c(C(=O)NC2CCCN(C(=O)CO)C2C)ccnc1F C=Cc1ccc(C(=O)NC2CCC(C(=O)Nc3sncc3C#N)C2)cc1 c1(C(=O)NC(C(C)NC(CC2(NC(C)=O)CC2)=O)CO)cccc(C)c1F C1(CC#C)(C(=O)NCCCOCCCNC(C2CC(C(F)(F)F)C2)=O)CCOC1 c1(OC)ccc(C2(NC(=O)NCC3CC34CC4(F)F)CC2)c(OC)c1OC C1C(C(C)(C)C)C(=O)NCC2(O)CN(C2)Cc2cscc2O1.C=CCOCCC C(CN=c1[nH]cnc(F)c1C)n1cc(C=CC(=O)OCC)nn1 C1(C)(NC(C(CC)(O)c2cccc(Cl)c2)=O)CCN(C(=O)C(O)C(F)(F)F)CC1 C1(COC)(CNC(=O)C(C(C)C)NC(C)=O)CCN(C(=O)Cc2ccoc2)C1 Cc1noc2ncnc(N3CC(C)(C)CC3CNC(c3ccc4n[nH]cc4c3)=O)c12 c1(C(N2CCC(c3n(CC)cnn3)CC2)=O)ccc(OC)c(Br)c1OC N1(C(=O)Cn2cc(N3CCCCC3)nn2)CCOC(c2ccccc2Cl)C1 C(=O)(CC(C)P(C)(C)=O)N1CCN(C(COc2ccc(C)cc2)=O)CC1CCO N1(Cc2ccc(CC(C)C)cc2)CCN(CC(=O)Nc2ncc(C#N)s2)C(=O)C1 c1(C(=O)NCC(CC)NC(=O)COC2(C)CCC2)cc(C(F)(F)F)cc(F)c1 c1(C(N(C)CC2CN(C(c3ccnn3C(F)F)=O)C2)=O)nccc(C#N)c1F CCCC(CNC(C1CC(C2CC2)C1)=O)C(=O)N(C1CCCC1)C1CC1 C1(NC(c2ccc(CO)o2)=O)CCCC(NCc2coc(C3CCCCC3)n2)C1 C1(NC(C(CCO)N(C)C)=O)CC2CCC(C1)N2C(=O)Cc1cccc(Cl)c1 c1(SCC(N2CC(O)(C3CCCN3C(c3ccncn3)=O)C2)=O)nnc(S)s1 c1(C(=O)NCCCN(C(c2cn(C)c(C)n2)=O)CC)cnc2c(c1)CCC2 c1(C(N2CC(CCNC(=O)CC3C=CCC3)OCC2)=O)cc2ncccn2n1 CC(F)CC(=O)NC1CCC(CNC(c2ncoc2-c2ccon2)=O)C1 c1(NCc2c(CC)con2)ccc(S(=O)(=O)N2CCC3(C)C(C2)C3(Cl)Cl)cc1Br C(=O)(CC(F)(F)CNC(c1nnnn1CNCc1ccccc1)C1CCCOC1)OC C1(C(=O)NCC2(F)CN(C(c3ccc(C)nc3C)=O)C2)CCCCC12CCC2 C(=O)(C1=CC2(CCN(C(C3CCC(OC(C)=O)CC3)=O)C2)C1)N(CCCC)CC C1(OC)CC(NC(=NC)NC2CC(OC(C)C)C2)C12CCC2 CC1(C)OC2(CNC(C3CCOC3)=O)CC1(NC(=O)CCC#N)C2 C=C1CCC(C(=O)N(CC(O)CN(C)C(c2cscc2SC)=O)C)CC1 N1(C(CNC(CN(CCC#C)C)=O)=O)CC2CCCC2C12CC2 C1(CNC(CNS(CC)(=O)=O)=O)CCCC1C(C)(C)C c1(C(=O)NC(C=CC(=O)NCCNC(c2ccc(Br)cc2)=O)=O)cccc(Br)c1 CCC(N=c1[nH]c(=NCCOCCC2CC2)c2sccc2[nH]1)c1ccccn1 c1(NC(C(=O)NC(c2nc(C)on2)c2ccccc2)=O)cc(Cl)ccc1C C(=O)(C(O)C(F)(F)F)NC1(C)CCN1C(=O)C=Cc1ccncn1 Cc1cc(-c2nnc(N3CC(C)CC(C)C3)n2CC2CCCO2)c(C)cn1 CN1CCNC(c2cn(CC3CC34CN(C(=O)CC(=O)OC(C)(C)C)C4)nn2)C1 C(=O)(CC(C)(C)CN(C)C)NC(C(C(=O)NC1(c2cc(C)no2)CC1)C)C C#CC1CN(C(=O)C(C)CC=C)CCN1C(=O)COCCC(C)C Cn1cc(NC(c2ccccc2Cl)CCO)cc1C(=O)NCc1cncs1 C(=O)(C(CCC(N)=O)N(C)C)N(CCNC(C1N2C(C)CN(CC2)C1)=O)C1CC1 c1(C(N(CC(C)CNC(c2cnn(C)n2)=O)C)=O)coc2c1CSC2 Cc1noc2ncc(C(=O)NCC(CC(C)C)NC(=O)C3=COCCO3)cc12 c1(C(=O)NC2CCN(C(C3C(C=C)OCCC3)=O)C2)cc2c(=O)[nH]ccn2c1 CCCC(C)CC(=O)N1CCC(Cc2cn(-c3cccc(Cl)c3Cl)nn2)C1 N1(CC)CCCC(C(=O)NCCOCCN(C(=O)CSCCOC)C)C1 C=CC1OCCC1C(=O)NC1CCC(C(=O)NC2(C)CCCC2O)C1 C(C)(C(C)(C)CN(C)C)NC(CC1N(C(C=CCN(C)CC)=O)CCC1)=O c1(C(N(CC(C)N(C)C(C2(CF)CCC2)=O)C)=O)ccc(Cl)c(F)c1F N1(CC(=O)N(C2CCN(C(Cc3c(C)non3)=O)C2)CCO)CCCS1(=O)=O N1(CCC2(C)CC2)CCCC(C)(C(N2CCC(CS(N)(=O)=O)C2)=O)C1 C(=O)(CC(C)C(F)(F)F)N1CC(CNC(C2CCC(CCC)CC2)=O)C2(C1)CC2 C(=O)(CCC(=O)NN(C)C)NC(C1CN(C(c2cc(Cl)sc2Cl)=O)CCO1)C C1(COC)CCC(C)N(C(=O)Cc2cn(CCCc3ccccc3Cl)nn2)C1 C12(C(=O)NCC(C3CCC3)NC(=O)CCc3cnco3)C3CC(CC13)C2(F)F C1(CC(=O)N(CCCCN(C)C(C2CC3(CC3)C2)=O)C)CCOC(C)(C)C1 c1(C(=O)OC)ccc(CNC(=O)Nc2cc(C(F)F)ccc2C)nc1O C1(C(=O)OC)(NC(C)C)CC1(C)C.C1(=O)C(=O)N(CCCO)CCN1 N1(C(c2nnc(C)s2)=O)CCCN(C(c2[nH]nnc2-c2ccccc2)=O)CC1C C(=O)(C(CC(C)C)NC(C1CN(C)CC(C)O1)=O)NCC1CC(=C)C1 N1(C(C(C)NC(=O)NC)=O)CCCC12CCCN(C(=O)CC1OCCC1(C)C)C2 N1(c2ncc(CCOCCOCC(=O)OCCC(C)C)s2)CCN(C)CC1.C(=O)O c1(N(CCCOC(C)C)C)nccc(=NC2CCCSCC2)[nH]1 c1(C(C(=O)NC2CN(C(CC)=O)CC2C(F)F)C)ccc(F)c(F)c1 c1(C(=O)NC2CCC(CCNC(C(C)CN(C)C)=O)C2)ccnnc1S CC(C)(O)C(F)(F)CNC(=O)CCOC1CN(C(=O)C(O)CN(C)C)C1 C1(NC(C2CCCCC2C(F)(F)F)=O)CC2CCC(C1)N2CC1CCOC1 c1(C(N(C(C)CNC(=O)Cn2cc(Cl)cn2)C)=O)c[nH]c2ccccc2c1=O C1(C(=O)NCCCCN(C(C2(C(C)C)CCCO2)=O)C)CCc2ncnn2C1 C1(NC(C2(O)CC2)=O)CCC(NC(C2(CC(F)F)CC2)=O)CC1 c1(C(=O)NC(CCN(C(C2(CC#C)CC2)=O)C)C)nc(C)n2c1CCCC2 c1(C(N2CCN(C(=O)Cc3nc[nH]n3)C3C2C3)=O)cc(Br)cc(C(F)(F)F)c1F N1(C(C(C)C)=O)CCC(C(N2CC=CC2CNC(=O)C=CC2CCC2)=O)C1 CC1(CS(=O)(=O)NCC2CCS(=O)(=O)C2)COCCN1 C(CC(C(=O)N1CCN(CCO)CC1)NC(C)=O)SC.c1(C2C(C)C2)cccnc1 N1(C2CCC(NC(C)CC(C)(C)O)CC2)CCN(C(=O)OC(C)(C)C)CC1=O Cc1ccc(Cl)c2ccc(NC(=O)Nc3cccc(OCC(=O)OC(C)C)c3)nc12 c1(CNC(C2CC(NS(CC)(=O)=O)C2)=O)ccc(C#N)cc1F C1(CNC(C=C(C)C)=O)CC(F)CN1C(=O)C(F)CC1CCC1 C(=O)(C(CNC(=O)CCCCC1CC1)CC1CC1)NCC1CN(C(N)=O)C1 C1(N(C(CCOCCCOC)=O)C)CCCCN(C(C2CNC(=O)N2)=O)C1 c1(CNCC2CC3(CC(NC(=O)Cn4cc(Br)cn4)C3)C2)nc2ccccc2[nH]1 c1(CNC(c2ccccc2)COC)ccc(C2=CCOCC2)nc1 O=C1NC2(CO1)CC(C(N1CCCC1CN(C(C1COCCO1)=O)C1CC1)=O)C2 C(=O)(CC(F)(F)CC)NC(CC)CNC(=O)CC1CCN(C)C1=O S(=O)(=O)(C=Cc1ccccc1)NCC1CN(C(c2ccnnc2O)=O)CC1O c1(C(=O)NC2C(CNC(c3ccc(NC(N)=O)cc3)=O)C2)cccc(F)c1Br c1(C(=O)NCCC(Cn2cc(C(COC)(C)O)nn2)(F)F)c[nH]c2cccnc12 C=C=C(C)CC(=O)NCc1cc(C(=O)NCC(CSC)OC)co1 c1(C(=O)NC2(CC=C)CCN(C(C3CC3F)=O)C2)cnn2c1CC(C)CC2 CCC(C#N)C(=O)N1CCC(C(=O)NCCc2ncoc2C)CC1 N1(C(c2n(CC)ncc2)=O)CC2(CC(NC(=O)C(C)(C)n3ccnn3)CO2)C1 CC1(C)CCC(O)(CNC(C2CC=CCC2NC(=O)Cc2ccns2)=O)C1 c1(C(=O)NC2(CNC(=O)COC3CCC3)CC2)cccc(-c2ccsc2)c1 c1(NC(CNc2sc(CC(=O)OCC)c(C)n2)=O)cccc2c1C(=O)N(C)C2 c1(CC(=O)NCCN(CCC)C(c2cc(C(N)=O)n(C)n2)=O)ccc(C)c(F)c1 c1(OC)ccc(CN2CCN(C(c3cc(C4CC4)n(C)n3)=O)CC2)cc1[N+](=O)[O-] Fc1ccc2[nH]cc(SCc3ccc(I)cn3)c2c1 C(CNC(=O)CC1CC=CCN1C)(CC(F)(F)F)NC(c1c(CCC)n[nH]c1)=O C1(NC(C2CNCCO2)CC)CC2(C1)CC(CN)C2 C=CCC(CC)C(=O)N1CC(O)(CNC(C2CCC2(C)C)=O)C1 c1(OCC)ccc(CNC(=O)Cc2ccc(CSc3ccccc3)cc2)c(Br)c1 c1(C2(N(C(C(=O)N(CCCF)C)C3CC3)C)CC2)cccnc1 c1(Cc2scc(C(=O)N(C3CCN(C(=O)C(F)F)C3)CCO)n2)ccc(F)cc1 C(=O)(CC(C(C)(C)C)NC(=O)Cc1cn[nH]c1)NC1CCN(CCC)C1 N1(CCN(C(CC(N(C)CCC2CC2)=O)=O)Cc2ccccc2)C(=O)CNC1=O CCCCCC(O)C(=O)NC(C1CCN(C(c2cccc(CO)n2)=O)CC1)C c1(C(N2CCC(C(C)NC(=O)C(C)(C)F)CC2)C)ccc(F)c(Cl)c1 CC1CN(C(C2CS(=O)(=O)C2)=O)CCC1NC(c1cncc(-n2ccnc2)n1)=O c1(N(C)C)ccnc(C(N2CC(C(N)=O)(CNC(=O)CC3CC4CC4C3)C2)=O)c1 N1(C(CCC2CCN(C(c3cn(CC)nc3)=O)C2)=O)CCS(=O)CC1C C(=O)(C1=CC2(CCN(C(=O)Cc3ncoc3C)C2)C1)NCc1ccc(CC)s1 C1(C(C)C)(C(=O)NCCN=S(C)(C)=O)CCN(C(C2CCC(=O)O2)=O)C1 Cc1cc(C)c(C(N2CC(NC(C3(C)CC3(F)F)=O)CC3(CC3)C2)=O)c(O)n1 C(=O)(C(COC)(CC)CC)N1CC(CC)C(NC(=O)Cn2cc(OC)cn2)CC1 CC1=CCC(C)(C(N2CC(CNC(=O)CCc3cccc(O)n3)C(C)C2)=O)CC1 c1(OC)c(C(=O)NC2CC(CC(=O)Nc3ccnc(O)c3)C2)cccc1C CC1Cc2c[nH]nc2C(C(=O)N2CC3(C2)CN(C(=O)CN2CC4CC4C2)CCO3)C1 c1(C(=O)NCC(CCCC)NC(c2cnc(Cl)c(C)c2)=O)nc(C)c(N)cc1C N1(C(=O)C(O)C2CN(C(=O)C(O)CN3CCCC3)C2)Cc2cncnc2C1 N1(C(CSCCN(C)C)=O)CC2(CCN(C(C3(C)CCC(C)(C)CC3)=O)CC2)C1 N1(C(c2ccc(OC)s2)=O)CC(NC(=O)CN2CC3CCC2C3)CCC1C Cc1cc(N2CCC(C3CN(C(=O)OC(C)(C)C)CCO3)C2)c([N+](=O)[O-])cc1C CC#CCCC(=O)NC1CN(C(C2CN(S(=O)(=O)C(F)F)C2)=O)CC1C Cc1cccc(N)c1C(=O)NCC1CCN(C(c2cc(Cl)cs2)=O)C1 CC1(C)CN(C(C2(NC(=O)CCN3CCOC3=O)CCCC2)=O)CCO1 c1(C(=O)NC(CCC)CCCNC(=O)CC(C)CC)ccc2ccccc2c1 C1(C(=O)NC(CC=C)CNC(=O)Cc2cc(CC)on2)CCC(N(C)C)CC1 CCCCCCCC(=O)NCC1(F)CCCN(C(=O)CCOCC)C1 CC1CCCN(C(=O)CN(C(=O)C=Cc2cn[nH]c2)CC2CC2)C1CO c1(CCNC(C2C(CNC(c3cnn(C(C)C)n3)=O)C2)=O)ccnc(C)c1 c1(OC)cc([N+](=O)[O-])ccc1C(=O)NC1CC2CC1CN(C(c1cnsn1)=O)C2 c1(CC)ccc(CCC(N2CCC(C)(CNC(C3(C)CC=CCO3)=O)C2)=O)cc1 C(N=c1[nH]c(N2CCC(F)C(F)C2)nc2c1CCC2)C1(OC)CCSC1 C(CCCCC(=O)N1CC(N(C(=O)Cc2ccn(C)n2)C)C1)OC N1(C(C=CC)=O)CCCC(NC(C2(COC)CCCO2)=O)C1C C1(C(N2CC(CCC)C2)=O)C2CC3C(C2NC(c2ccc(=N)[nH]c2)=O)C13 c1(C(=O)NC(CCNC(C2(COC)CC=CC2)=O)(C)C)cc(C#N)cc(C)n1 N1(C(C(CC)NC(C)=O)=O)CCC(C(=O)NCCc2ccnn2C)=C(F)C1 c1(CN2C(C(N3CCCN(CC)CC3)=O)CC(C)(C)C2)c[nH]c2ccncc12 N1(CCN(C(C2C(NC(c3cocn3)=O)C2)=O)CC2CC2)CCCCC1 C(C)(N=c1[nH]c(=N)[nH]c(=NCC(C)C)[nH]1)c1cc(C)sc1C C1(NC(C(CC)=CCCC)=O)CCN(C(=O)CC(C)c2cnn(C)c2)C1C(C)C Cn1cc(C(=O)NC2C=CCN(C(C3(C)CCCC3(F)F)=O)C2)n(C)c1=O CC1(C)CCCC(CC(=O)NC2(CNC(=O)CC3(C)CC3)CCCCC2)O1 N1(CCNC(C2CCN(C(C3(Oc4ccccc4)CC3)=O)C2)=O)CCC(O)CC1 c1(SCC(=O)NCCC(=C)CNC(c2cccnc2N)=O)ccccc1C CCC(C)CCCC(=O)N1CC2C(CNC(C3(c4ncccc4F)CC3)=O)C2C1 C1(NC(c2ccc(Cl)s2)=O)C=CC(CNC(c2cnn(C3CCCCC3)c2)=O)C1 N1(C(=O)Nc2c(=N)c3c([nH]c2)cccc3)CC2(CCC2)c2ncccc21 c1(OCC(=O)NC2CCC2NC(C2CC2F)=O)ccccc1Cc1ccccc1 C(C(C)(O)CCCO)NC(c1c(C(C)C)nccc1)=O.C1=C2CN(C(=O)CC1)C2 N1(C(Cn2c(C)c(Cl)cn2)=O)C2CCC1CC(NC(C1CCCCC1F)=O)C2 C1(C2CCOCC2)(C(N2CC(CCNC(C(C)OCCCC)=O)C(C)C2)=O)CC1 N1(c2nc(OC(C)C)cc(C)n2)CCC2C1CCCN2C=O.C(CCC(=O)O)NCN N1(C(CNC(CC(C)(C)C)=O)=O)CC2CCC(NC(c3cnc(O)o3)=O)CC2C1 C(=O)(C(F)C(C)CNC(c1ncccc1F)=O)N(C(C(=O)OC)C)C C1(C(=O)NCC(CCNC(C=CC(C)(C)SC)=O)O)COCC1(C)C N1(CC(C2CC2)NC(C2(C)CC2)=O)CCN(C(=O)CC2(CO)CC2)CC1 c1(C(=O)NCCCN(C(C(C(=C)C)(C)O)=O)C)ccc(Cl)c(Cl)c1N C1(COC)CN(C)CCN1C(=O)C(=O)Nc1ccc(-n2nncc2C)cc1 c1(CCN(C)CCNc2cc(NC3CCCC34CC4)ncn2)ccc(F)cc1F CC1(C)COCC1C(N1CC(O)CC1C(N1CC(F)(CF)C1)=O)=O Cc1nn(C)c(Cl)c1CN(C)C(N1CCCC(c2ncc[nH]2)C1)=O c1(N(C(c2ncccc2Br)C(=O)NCCCSC)CCC)ccc(C)cc1OC C(c1ccc2c(c1)CCO2)=CC(=O)NC1CN(C(C2CC3(CC(C)(C)C3)C2)=O)C1 C1(CCCNC(C(C)C2CCOC2)=O)CCCCN1C(=O)CC1CC(=O)C1 C(=O)(C(C#N)CCC)NC(CCC)C(=O)NCC1CC12CCCCC2 Cc1ccn(CC(C)C(=O)NCCC2(NC(C3CC3C)=O)CCC2)n1 c1(CC(=O)NC2CCN(C(C3C=CCCC3)=O)CC2O)n[nH]c2c1CCCC2 N1(C(=O)Nc2c(C)ccs2)CCCN(C(C)C(=O)NCCOCCOC)CC1 C(=O)(C1Cc2ccccc21)CCN(C)CCOC1CN(c2ncc3ncnc-3[nH]2)C1 C12(CNC(C=C(C)C(C)(C)C)=O)CC1CN(C(=O)Cc1csc(Cl)c1)C2 N(C(=NCc1ccco1)N1CCOC(Cc2nncs2)C1)CC1(OCC)CCOC1 N1(C(c2ccc(CC)[nH]2)=O)CCCC(CC(=O)NCCc2cc(C)on2)CC1 C1(C(=O)NC2C(C)N(C(=O)CCCC(N)=O)CCC2)CCc2nncn2C1 C1(C(=O)NCCCCCC)CN(CCC2CCCC2(F)F)CC1(C)C c1(C(=O)NC(C2CCCN(C(c3cnn(C)n3)=O)C2)C)cccc2nccnc12 C1(CNC(=O)C(N2CCCC2)C2CC2)(NC(=O)Cn2ccnn2)CCCCCC1 C(CCCC(C)NC(c1ccc[n+]([O-])c1)=O)NC(c1c(C)cno1)=O C1(NC(Cc2c(C)noc2C)=O)CCC2(CCN(C(C3(O)CC3)=O)CC2)C1 C1(CN2CC(NC(CCOCCOC)=O)C2)(CNC(=O)C2CC2)CCCC1 c1(CC(=O)NC(C2CCN(C(CCCCC)=O)C2)C)cccc(OCC)c1Cl N1(C(C2CCN(C(C(CCC(C)C)F)=O)C2C)=O)CCc2nc(O)[nH]c2C1 CCCCC(CNC(C1(C)CCOCC1)=O)NC(c1cc(C2CC2)on1)=O C1(CNC(c2ccccc2Cl)=O)CC(NC(=O)CC2(CO)CC2)C12CCC2 c1(OC)ccc(C(N2Cc3c[nH]nc3C2)C(=O)NCCNC(C)=O)c(Cl)n1 N1(C(=O)NCC(CCC=C)CCC)CCC(COC)CC12CCC2 C(CC(C(=O)NCCF)NC(C1COC(=O)N1)=O)OCC c1(C(=O)NC2CCC(CNC(c3c(CC)ccs3)=O)C2)ccc(F)cc1C c1(C(=O)NC2C(NC(COC(CC)C)=O)CCOC2)sc2nccn2c1C C1(NC(c2c[nH]nc2-c2ccncc2)=O)CCN(CCF)C1=O C(=O)(C1=Cc2ccccc2C1)NC(C1CCCCC1)C(=O)NC(C(C)(C)C)CO C1(OC)(CNC(=O)CC(C)CF)CCN(C(=O)CS(=O)(=O)NCC2CCCO2)C1 c1(C(N2CCCC(NC(C3(C)CCNC3=O)=O)C2)=O)cc(F)cc2nn[nH]c12 CC1CN(C(c2ccc(C3CC3)cc2)=O)CCC1N(CCC(N)=O)C(=O)CCF N1(C(c2nc(CCCC)sc2)=O)CCCCC(NC(c2ccc(CF)cc2)=O)C1 N1(C(C(C)OC)=O)CC(C)(C)OCC1CNC(=O)C(C)(C)c1cnc[nH]1 N1(C(COCCC)=O)CCOCC(CNC(=O)CC2COCC(C)(C)O2)C1 C(N=c1[nH]cnc(NCCCc2cnn[nH]2)c1C)c1c(C)c(C2CC2)ccc1 N1(C(Cc2ccn(C)n2)=O)CCOCC(C(=O)Nc2ccc(N)cn2)C1 N1(C(C(COC)OC)=O)CCC(C)C1CNC(=O)CNS(C)(=O)=O N1(C(CC(C)(C)C)=O)CCN(c2nnc(Cc3c(F)cccc3F)s2)CC(O)C1 C(C1CCCN1C)=CC(N1CCC(C(C)NC(C2(C)CC2)=O)C1)=O C=Cc1cncc(C(=O)NCC2CN(C)CCN2C(c2ccc(C)c(C)n2)=O)c1 C(=O)(C(O)C1=CCCCC1)NC(CC(=C)C)C(=O)NCC12CC(C1)C2 C1(SC)CCCN(C(c2ccc(Br)nc2)C(=O)NCCCOCC2CC2)CC1 C=C(C)C(C)(C)C(=O)Nc1cccc(SCC2CC(C)(C)CN2C(=O)C2CC2)c1 CC1C(C(N2CCN(CC3CN(C(C45CSCC4C5)=O)C3)CC2)=O)CCN1C c1(C(=O)NC2CCN(C(C(C3CCOC3)OCC)=O)CC2)cc2sccc2s1 Cn1cncc1CCCc1c(C(=O)NC=O)con1.C(=O)(CCCNC1CC1)N O=C1CC(CC(=O)NC2CC3CCC2(NC(C2CCC2)=O)C3)CCCN1 CCC(C)(C#N)C(=O)NCc1cc(C(=O)NCC(O)COC)cs1 C(=O)(CC(C)(C)C1CC1)NC1C(C(C)NC(=O)CC2(CN(C)C)CCC2)C1 N1(C(CNS(NC)(=O)=O)=O)CC2CN(C(=O)Cn3ccc(Br)n3)CCC12 c1(CNC(CCNC(C)=O)=O)cc(C(=O)NCc2ccc(=N)[nH]c2)n(C)n1 Cc1ccc(C(CNC(=O)CCc2nccs2)NC(c2cn(C)cn2)=O)cc1 CC1CCCCC1CC(=O)NC1CCC(NC(=O)CN(c2ccncc2)C)C1 N1(Cc2c(OCC)cccc2)CCC2(CCCC2C(N2CCC(F)(F)CC2)=O)C1 c1(OC)ccc(F)c(NC(C23CCN(C(C4CC5CCC(C4)O5)=O)CC2C3)=O)c1 c1(C(N2CC(C(N)=O)(CNC(C(C)SCC)=O)C2)=O)nn(C)c(=O)cc1C Cc1nccn1CCNC(C1CCCC1NC(=O)Cc1ccn(C)c1)=O N1(C(=O)NC2CCN(c3ccn(C)n3)C2=O)CCC(P(C)(C)=O)C1 n1(CCOC)ccc(C(=O)N(C2CCN(C(C3(N(C)C)CC3)=O)C2)C)n1 c1(OC)ccc(Br)cc1C1CN(C(C2(CN(C)C)CCCCC2)=O)C1 N1(Cc2ccc(COCC)s2)C(=O)CCN(CC23CCC(CC2)O3)C1=O N1(C(Cc2c(CC)cccc2)=O)CCC(N=c2[nH]nc(CC3CCC3)s2)C1 C(=O)(C(C)CC(N)=O)N1CC(CNC(c2c(CC)nn[nH]2)=O)OCC1 C1(CO)CC(OC)N(C2c3ccc(s3)C(=O)OC2=O)C1.C1(C)CCC1.C1(COC)CC1 C(CC(C)C(=O)NC(C)CSc1ccccc1)OC c1(NC(C2CCN(CC(F)(F)F)C2)=O)ccc(NC(C)C)nc1 CC1OC2CCC1(C(N1CCN(C)C(C(=O)NC(CCO)C3CC3)C1)=O)C2 n1(CCCC)cc(C(=O)N(CC(O)CNC(=O)C=CC(C)(C)C)C)nn1 C(=O)(C1CSc2ccccc21)NCC=CCNC(COCc1cc(C)on1)=O C(C)(CNC(C1CC=CCO1)=O)(C(C)C)NC(C1CC(CC(=O)OC)C1)=O C1(NC(CSCCC)=O)CCC2(CC1)CC(NC(c1ccc3ccnn3c1)=O)C2 c1(CC)oc(C)cc1C(N1CCOCC1CN(C(=O)CC1C=NN(C)C1=O)C)=O n1(CCC)nccc1C(=O)N(C(C)(C(=O)NCC(C)CC1CCC1)C1CC1)C CCC(C)(COC)C(=O)NCCCCCN(C)C(c1cc(C)cc(Br)c1)=O C1(NC(CCC)=O)CC(CC(N)=O)N(C(c2cccc(CSC)c2)=O)C1 C(=O)(C(C)(C)CCCF)NCC(CC)NC(=O)Cc1ccc(Br)cc1C N1(C(C=C(C)c2ccco2)=O)CC2COCC2(C(=O)NCC(CC2CC2)CO)C1 N1(C(C(C)(F)F)=O)CCC2(CCCC2NC(c2ccn(O)c(=O)c2)=O)C1 N1(C(c2ccc(NC(c3c(SC)cccc3)=O)cn2)=O)CCCC2CCCCC12 C1(CC(=O)NCCc2ccn(CCNC(CCC=C)=O)c2)CCC1C1CC1 C1(CNC(c2n(C(CC)CC)ncc2)=O)CCCN(c2ncc(Cl)cn2)C1 Cc1cc(C)n(C(C)C(=O)NC2CN(C(C3(C(F)F)CCC3)=O)CC2C)n1 Cn1cc(C(=O)NCC(CNC(=O)CCOCC(F)(F)F)CO)ccc1=O N1(C(C2C(NC(c3csc(C)c3C)=O)COCC2)=O)CC(C)N(C)C(C)C1 C(=O)(C(CCCC)C(C)C)N1CCC(C#C)(C(=O)N(C2CN(C)C2)C)C1 c1(CCC(=O)NC(C(=O)NCCCCC)c2ccco2)conc1C c1(NC2CCN(C(=O)C=CC3CCCC3)C2)ncnc2ccccc12 CCCC(C)(O)CC(=O)NC(CC1CC1)CC(N1CCCN(C=O)CC1)=O Cc1c(NC(C2CCC(CNC(=O)CCC(C)(C)C)C2)=O)cccc1F CC(CCO)N=c1[nH]c(=N)[nH]c(=NCC2Cc3cc(Cl)ccc3O2)[nH]1 N1CCC2(C1)CC2(F)F.c1(N(C)C)ccc(CN2CC3C(C(=O)N)C3C2)cc1 n1(CC(N2CC(CNC(C3CC(CC)OCC3)=O)C2)=O)ccc(=O)n(C)c1=O O=C1CCN(CC2CCCN2N2CCCC2)C(=O)N1Cc1ccc(Br)cc1Cl S(=O)(=O)(c1cccc(C(N2CCC(NCc3ncc[nH]3)CC2)=O)c1)N(C(C)C)C N1(C(COC)C)CCC2(CC1)COC(C(=O)NCCC(N1CCOCC1)C)C2 Cc1cc(-c2nn[nH]n2)ncc1C(F)(F)F.C1(=O)C(=O)NCC2(CC(=O)N1)CC2 CC(C)(C(=O)NC1CCCC1CNC(=O)COCc1nc[nH]n1)C(F)F c1(NC(C)CCCCO)nccc(=NCC(CO)C2CCCC2)[nH]1 c1(OC)cc(OC)[nH]c(=NCCCN(C)C(C2C3CCC(C3)C2(C)C)=O)n1 c1(C(=O)NCC(CC)NC(C2(C(F)(F)C(F)(F)F)CCC2)=O)ccnn(C)c1=O c1(C(N2CC3C(CNC(C4(C#N)CCC4)=O)C3C2)=O)ccc2c(c1)CCOC2 C1(NC(C2CC(=O)NC2)=O)CCCCC1C(=O)NC1(c2ncc[nH]2)CC1 CCC(C#N)(CC)C(=O)NCC(C)(F)CNC(C1CCCNC1=O)=O c1(N(C)CC2CCN(C(c3ocnc3C3CC3)=O)C2)c(F)cc([N+](=O)[O-])cc1F C1(NC(CC(C)SC)=O)CC2(CCN(C(=O)CSc3ccc(F)cc3F)CC2)C1 N1(C(C=C2CCC(C)C2)=O)CCCC(C)(C)C1CNC(c1cc(O)ncc1F)=O N1(C(CC(CNC(C(C(=O)OCC)F)=O)(C)C)=O)CCC2(CCCC2)C1 C(C(=O)N(CC(CC)NC(c1nc(C)c(C)s1)=O)C)(C(C)C)SCC N1(C(CSCCC#N)=O)C(CNC(c2cccc3nonc23)=O)CC2COCC12 c1(OC(C)C)cccnc1C(=O)NCCN(C(=O)CNS(N)(=O)=O)C(C)C C1(CN(C(c2cc(C)sc2)=O)C)CN(C(=O)C(F)CC2CC2)CC12CC2 Cc1cc(C(N2CC(O)(C(C)NC(=O)C(C(C)C)NC(=O)C3CC3)C2)=O)cn1C CC1C(C)N(C(=O)C=Cc2c(F)cccc2F)CCN1C(=O)CNc1cccs1 C1(C(=O)NCC=CCC(=O)NCCCCSC)CCC(=O)NC1 N1(C(c2cc(OC)ns2)=O)CCCCC(CNC(C2CC(CF)C2)=O)C1 N1(C(c2c(C)[nH]cc2)=O)CCC(C)(CC(=O)NCCN2CCCCC2C)C1 Cc1cc(CNC(C2CC=CC(NC(=O)C=CCF)C2)=O)ncn1 N(C1CCc2ccc3c(c21)CCO3)C(=O)NCCc1ccc(OCCCC)cc1 c1(C(=O)NCCN(C(c2nc(C3CC3)oc2C)=O)CC)cc(Cl)c(Cl)[nH]c1=N N1(C(=O)CC2CC3CCC2C3)CC2CCN(Cc3cncc(F)c3)C2C1 C1(C(=O)NCC(CCC)OC)CCN(C(c2cccc[n+]2[O-])=O)C12CCC2 N1(C(C(CC=CC)CC)=O)CCCN(C(=O)Cc2cnc(Cl)cc2C)C(C)C1 c1(N2CCC(OC)(CO)C2)nc2ccsc2c(=NC(C)C2CCC2)[nH]1 S(=O)(=O)(CCC(=O)NCCOCCNC1CCCC1C)NC C1(C2CN(C(=O)CC3CCCC3(F)F)C2)(NC(CC2C(C)OC(C)C2)=O)CC1 C#CC1COCCN1C(C1(NC(c2ccc(C3CC3)o2)=O)CCC(C)(C)C1)=O CC(C)C(O)C(F)(F)C(=O)NCC1CCCC1NC(=O)CC(C)C(F)(F)F c1(C(N(C2CC2c2csc(C#N)c2)C)=O)nc(Br)sc1C1CC1 c1(C(=O)NCc2cn(C(C(=O)N(CCOC)C)C)nn2)cncc(OC(C)C)c1 c1(C(=O)NC2C(N=[N+]=[N-])CN(C(c3ccsn3)=O)C2)c(F)ccc(F)c1Cl N1(C(C(CCCC)n2ccnc2)=O)CCn2ncc(CO)c2C1 c1(C(=O)NCC2CN(C(C3(COC)CCC3)=O)C2)cc(=O)n(C)c2ccccc12 CCC(C)(COC)CNC(C1CC(O)(CNC(=O)CCCCNC(C)=O)C1)=O Cc1cc(C(=O)NCC(C2CC2)NC(=O)C(C)C(C)O)cc([N+](=O)[O-])c1O CCCC(CNC(C1CC1C(C)(C)C)=O)C(=O)N1CCCN(C2CC2)CC1 C1(C(C(=O)NCC2(C)CC2)N(C(c2ccccc2)COC)C)CC2CC1C1CC21 c1(OC)cc(C(=O)NCC(C)NC(=O)CSCc2ccncc2)ccc1C#N c1(NC(CC(N)=O)C2CC2)[nH]c(=NCCc2conc2Br)nc2scnc12 N1(C(C(C)CC2CCC2)=O)CCCC(C2CC2NC(C2CCC(=O)O2)=O)C1 N1(C(C)=O)CCOCC1CC(N1CC(NC(C2CCCS(=O)(=O)C2)=O)C1)=O c1(OC2(C(=O)NC(CNC(Cc3ccc(C)cc3)=O)C)CC2)ccc(Cl)c(Cl)c1 c1(C(=O)NC2C(CNC(C3(COC)CCC3)=O)CCCC2)nc(Cl)ccc1Cl C(=O)(C(CC(F)F)N(C(=O)C=Cc1cncn1C)C)NCC(C(C)C)(C)C c1(-c2c(C)onc2)ccnc(N2CCN(C(C3(C(C)C)CCC3)=O)CC2)c1 S(=O)(=O)(c1c(Cl)cc(Cl)cc1[N+](=O)[O-])N1CC(C(=O)OC)C(c2ccccc2)C1 c1(OC)ccc(F)c(C(=O)N(C2CN(C(=O)C(C)CC(F)(F)F)C2)C)c1N c1(C(N2CCC(CN(C(C(c3ccccc3)OC)=O)C)C2)=O)sc(C#N)cc1Cl N1(C(C2OCC(C)C2)=O)CC(CO)C2(C1)CN(C(c1c(F)cccc1F)=O)C2 C#CC1(C(N2CC3(CCC3NC(c3ccc(Cl)cc3O)=O)C2)=O)CCCCC1 Cc1ncc(Cl)cc1C(=O)NC1CCCC1NC(C1(C2CCCCO2)CCC1)=O C(=O)(CCCCCF)NC1CCCC(CNC(CCN(CCC(C)(C)C)C)=O)C1 C1(NC(CC(=O)OCC)=O)CCN(C(=O)CC2CC=CC2)CC1C c1(-c2cn(CCCCNC(C3CCn4ccnc4C3)=O)nn2)cccc(Cl)c1Cl c1(N(C(c2cnc(C)[nH]2)C(=O)NCCCOC)CC)cc(C)cc(Cl)c1 c1(C(=O)NC2CC(NC(CC3CC(OC)C3(C)C)=O)C2)nsc2c(Cl)cccc12 c1(OCCC#C)ccc(CS(N)(=O)=O)c(F)c1.C1CCCNC1 N1(C(C2C(C=C)C2)=O)CCN(CCCCCNC(C2CC(SC)C2)=O)CC1 C1(C(N2CCC(C(C)(C)NC(CCCC#C)=O)C2)=O)CCc2c[nH]nc2C1 N1(C(CSCCC#N)=O)CC(NC(c2ccc[n+]([O-])c2)=O)CCC(O)C1 c1(N(CC(=O)NCC(C)(CO)NC(C2CC23CCC3)=O)C)ccc(Cl)cc1 c1(NC(c2cc(-c3ccc(F)cc3)no2)=O)ccc(C2=CCCCC2)cn1 CCC1=NOC(CC(N2CCCCC2C(N2CCC(C3(C)N=N3)C2)=O)=O)C1 O=C(N=c1cc[nH]cc1Cl)c1csc(=NCc2cccc3c2CCCC3)[nH]1 C1(CNC(C2CCC=CCCC2)=O)CN(C(c2ccsc2Cl)=O)CCC1CO c1(C(=O)NC2CN(C(CCC=CC)=O)C(C)CC2)ccc2c(c1)B(O)OC2 C#Cc1ccc(-c2nc(-c3ccccc3)no2)cc1OC c1(C(=O)NC(CC)(C)c2nn[nH]n2)n[nH]c(C)c1[N+](=O)[O-].C12=CC=C(C=C1)C2 N1(C(C(CC)(C)C)=O)CCCC(C2CN(C(c3cc(S(N)(=O)=O)ccn3)=O)C2)C1 CN1CCCCC1C1(NCc2ncc(-c3ccccc3)s2)CCC1 N1(C(C2CCN(CC(C)C)C2)=O)CC(NC(c2cnc(OCF)s2)=O)C(O)C1 c1(-c2c(N3C(C(CC)CO)CC3)csc2)ccc(C)cn1.C(=O)O c1(C(=O)NC2(CNC(c3cc(CC)on3)=O)CC2)cccc(-c2ccccc2)n1 C1(NC(CNS(CCOCC)(=O)=O)=O)CN(C(=O)COCCF)CC2(CCC2)C1 CCC(C)CCCCC(=O)NC(CC(=O)N1CCC(O)C1)C(C)C c1(C(N2CC(O)(CN(C(C(COC(C)=O)C)=O)C)C2)=O)ncc2ccccn12 Cc1cc(C(=O)NCC(CC(=O)NC2CC(N3CCC3)C2)C2CCC2)cn1C c1(C(=O)N(C)C)cn(C)c2cc(C(=O)NCC(c3ccno3)C)[nH]c12 N1(C(C(C)=CC2CC2)=O)CC2(CCC2)CC1C(=O)N(C)CC1CCCC2CC12 C1(O)(CCNC(C(C=C)c2ccccc2)=O)CCN(C(=O)CC(=O)OC)C1.OC CC1CN(C(=O)C(Cl)=CCl)CCC1CNC1CC(OC(C)(C)C)C1 c1(N(C(C(=O)NCCSCc2ccon2)C2CC2(Br)Br)C)ccccc1Cl c1(OC)ccc(C2CC(C)N(C(=O)NC3CC3c3ccccc3CCO)C2)cc1 N1(C(C=C(C)C)=O)CC2CC(C1)N(C(=O)Cc1cc(Br)ccc1F)C2 N1(CCCOC)CCN(CCNCc2c(C)noc2C)CC1 c1(C(=O)NCCCC(C)NC(=O)C(C)CO)cc(Cl)cnc1O C1(C(=O)N)COC2(CCC2)CO1.C(CC)(C(=O)NCCOCCOC)OC.CCCC=O.CN C(=O)(C(C)CC(F)(F)F)NC(CNC(C(C(CC)O)C)=O)C c1(C(=O)NCCCCN2CCCCCC2)ccc2c(c1)N(CC(F)F)C(=O)CS2 C(C)(C)(CCCC(=O)NCCc1nnc(C)n1C)NC(C(CCCC)O)=O Cc1nn(C(C)(C)C)c(C)c1C(=O)N(C)Cc1ccc(C(=O)N=S(C)(C)=O)cc1 C(c1ccc(F)c(F)c1)=CC(=O)NC1CCC1NC(c1cnn(C(F)(F)F)c1)=O c1(C(=O)Nc2cc(Cl)ccn2)cc2n(n1)CCCN(C(c1occc1Br)=O)C2 CC(F)(C(=O)N1CC(O)(C(C)(C)CNC(c2ccnc(CO)c2)=O)C1)C(F)(F)F c12ccc3c(n1)CN2CC3.C1CC2C=CCC(C1)C2.O=CO Cc1cnc2cc(C(=O)NCCC3COCCN3C(C3CCOC3=O)=O)nn2c1 C12(COC)CC(CNC(C3(O)CCC3)=O)(CN1C(=O)C=C(C)c1ccco1)C2 CC1CC(C)N(C(=O)Cn2cnc(Br)n2)CCN1C(c1cc[nH]n1)=O C(N=c1[nH]c(C)cc(=NC(COC)c2ccccc2Br)[nH]1)C1(CC=C)CCCC1 Cc1ncc(C(N2CC(NC(C3OCCCO3)=O)C2)=O)c(=N)[nH]1 N1(C(C2C(=O)NCC2)=O)CCC2(CCN(C(=O)CC3CCCC3O)C2)C1 N1(C(C2CC(C)C2)=O)CCN(C(C2CN(S(N)(=O)=O)C2)=O)CC12CCC2 c1(C(N2CC(NC(C(C)C(F)(F)F)=O)C(F)CC2)=O)c(F)cccc1[N+](=O)[O-] N1(C(C(=O)NC(C)Cc2ccc(Br)cc2)=O)CCS(=O)(=O)CCC1C c1(COC)ccccc1NC(=O)C(O)CNC(=O)COc1ccsn1 N1(C(c2c(C)cns2)=O)CC2COCC2(C(N2CC(C)C(F)C2)=O)C1 C1(CNC(C2CCN(C)C2)=O)CCC(C)(C)CN1C(c1ccc(N)c(F)c1F)=O C1(CNC(=O)Cn2cnc(-c3ccccc3)n2)CN(C(C2CCC2)=O)CC1O c1(N(CCC(=O)N(CCCNC(C(C)OCC=C)=O)C)C)ccncc1 C1(C(N2CCC(NC(CC3(OC)CC3)=O)C(F)C2)=O)CC12CCCCCC2 c1(C(=O)NCCNC(C2CC(SCC)C2)=O)ccn(CCN(C)C(C)=O)c1C c1(C(=O)NC2CCN(C(c3ncn(CC)c3)=O)C2)ccc(N)c(O)c1 CCC1=NOC(CC(=O)NC2CCCC(NC(c3nc(O)sc3C)=O)C2)C1 c1(OCC)ccccc1C(=O)NCCCN(C)C(c1ccc(CSC)o1)=O C1(COC)CCCN1CC1CCCO1.C1(C2COC2)C(=O)N1 N1(C(C2C(CC)CCC2)=O)CC2CCC(C1)N2C(=O)CC(C)c1cccnc1 N1(C(CC(C)(C)SC)=O)CCCC2CN(C(c3ccc(C)c(F)c3)=O)CCC12 C=Cc1cncc(C(=O)NCC(CC(=O)NCC2(C#N)CCOCC2)OC)c1 C(c1ccccc1C#N)=CC(=O)NC(CN(C(CCC=C=C)=O)C)C C1(C2CCN(C(c3noc4ccccc34)=O)CC2)(NC(CCOCC)=O)CC1 CC1CCCC(C(=O)NCCCC(=O)NC2CCNC(=O)C2)C1 c1(C(=O)NC(CNC(c2nn(C)c(Cl)c2Cl)=O)C2CC2)ccc2ncncc2c1 C1(NC(c2cccc(F)c2Cl)=O)CN(Cc2c(F)cc(Br)cc2Br)CC(F)(F)C1 CC1C(C)N(C(C23CC(C)(C2)OC3(C)C)=O)CCN1C(c1cnc(O)cc1O)=O C1(C(CNC(c2[nH]cc(C)c2)=O)(C)O)CCCN(C(=O)Cc2csc(S)n2)C1 C(=O)(C1OCCn2ccnc21)NC1C(NC(c2ccn(C)c(=O)c2)=O)C1 C1(CC(=O)N(C)CC2(C)CC2)(OC)CN(C(=O)C(C)N2CC(C)C2)C1 N1(C(C(C(C)(C)O)(C)C)=O)CCC2CCN(C(c3cc(Cl)c(Cl)s3)=O)CC2C1 C1(CNCc2ccc(OC)cc2)CN(C(c2[nH]ccc2C2CC2)=O)CC12CC2 c1(N2CC(C)CNC(=O)C2)nc2c(c(=NCCC#CBr)[nH]1)CCCC2 C(CCCCC(=O)NC1CCC(CNC(C23CCC(C2)OC3)=O)CC1)SC c1(C(N2CC3CN(C(CC(=O)OCC)=O)CC3C2)C)cn(C)c2cccc(C)c12 C(=O)(CCCC(C)(F)F)NCC1CCCN(C(CCOCCCC)=O)C1 N1(C(=O)Cn2ccc(O)nc2=O)CCC2(CCCN(C(C3CNC(=O)O3)=O)C2)C1 N12CCC(O)(C1)NC2=O.CC(CCO)NCCCCC1CCCC1 Cn1cnc2c(NC(=O)CCC3(C)CN(C(=O)OCC(C)(C)C)C3)ccnc12 CC(CNCc1ccc(C(=O)OC(C)(C)C)c(C)n1)CC(F)(F)F C(=O)(CCCCC(=O)N1CCCOC(CCNC(c2cncs2)=O)C1)OC Cn1c(=O)n(C)c2cc(C(=O)NC3CC4(CNC(=O)C4)C3)ccc12 c1(C(N2CCC(NC(c3c(C)noc3Cl)=O)C2)=O)cccn(C(C)(C)C)c1=O c1(C(=O)NCC2N(C(CCC#C)=O)CCC2C)cc2ccncc2s1 c1(C(=O)NC2CC(NC(C3(C)CC(F)C3)=O)C2)cc2ncccc2o1 c1(NC(C)=O)nc(CC(=O)NC2CC2NC(=O)CC2CC2(C)C)cs1 C1(CN)CCCCC1.c1(OC)cccs1.C12CC1C(C)(C)CN(C(=O)C1CC1)C2=O c1(C(N2CC(SC)C(NC(c3csc(COC)n3)=O)C2)=O)nnn2c1CCCC2 c1(CC(=O)NC2(CNC(CCC=CC)=O)CC2)c(CC)noc1CC C=CCCCCCCCCC(=O)NC(C)CNC(=O)CNC=O C(C(F)(F)Cn1cc(CCO)nn1)NC(C(C)SCCCC)=O C(=O)(CC(O)C(C)C)N1CC(NC(C(c2ccccn2)C)=O)(CO)C1 C1(O)(C(CNC(C2CN(C(C)=O)C2)=O)(C)C)CCCN(C(c2ccc(F)s2)=O)C1 N1(C(CSc2n(C)ccn2)=O)CCCC(CCNC(=O)CCCC#N)C1 C12(NC(C(CCC=C)NC(c3ccn(C(F)F)n3)=O)=O)CCC(C1)C(O)C2O c1(C(=O)NCCCN2CCN(C(CN(C)C)=O)CC2)cc(=N)[nH]cc1Br CC(C#N)C(=O)NC(c1cnn(C)c1)C(=O)NCCNS(C)(=O)=O C(C)(C)(CC(C)NC(=O)C(C)(C1CCC1)NC(=O)C=Cc1cscn1)OC O=C(CC1(c2nn[nH]n2)CC2(CCC2)C1)N=c1ccn(-c2ccccc2Cl)[nH]1 CCC(CC)C(C(=O)NC1(CC(=O)NC2CCCCC2(C)C)CC1)OC C1(C(N2CCC(C)(CO)C2)C(=O)NCCCOC)CCSC1(C)C C12(C(=O)NCC3(F)CC(NC(CCC(C)OCC)=O)C3)CCC(OC)C1CC2 c1(C(=O)OC)cnc(NCC2(C)CCC(NC(C3(C(F)(F)F)CC3)=O)C2)c(Cl)c1 Cc1ccc(N)c(C(=O)NCCC(C)NC(=O)C(C)(C)C(F)F)c1 N1(C(c2oc(CC)c(C)c2)=O)CC2(NC(=O)C=Cc3cscn3)CCC1CC2 c1(C(=O)NC2C(NC(C3(OC)CCC3)=O)CCC2)c(C)cccc1O C1(NC(C2CCC(CC)CC2)=O)CCCC12CCN(C(=O)C(C)(C)COC)CC2 N1(C(=O)OC(CC(C)C)C)CCCCC1CNC(=O)CCC(C)O C(CC(CC)C(=O)NCC1C2CC1N(C(c1ccc(OC)c(OC)c1)=O)C2)=CC C12(NC(c3c(OC)ncc(Cl)c3)=O)CC(N=c3nc[nH]n4c(Br)ccc34)(C1)C2 c1(SCC)ccc(CC(=O)NCC2(C)CN(C(c3[nH]nnc3C)=O)C2)cc1 C12(NC(C3CC4CCC3O4)=O)CCCC1N(C(c1cccc3c1COC3)=O)CC2 C1(NC(c2c(CC)ocn2)=O)CCCN(C(c2nc(OC)cc(OC)n2)=O)CC1 C1(CC(=O)NCCCOC(C)(C)C)CC2(C1)CN(C(=O)Nc1nnc(C)o1)C2 C1(CC)(NC(C2CCN(C)C(=O)C2)=O)CCCN(C(=O)C(C)(C2CC2)OC)C1 c1(OC)nc(C(=O)NC2(C(=O)NC(c3cn[nH]c3)C)CC2(C)C)co1 c1(CNC(c2ccc(CC)s2)=O)nn(C)c2c1CN(C(c1c[nH]c(=N)o1)=O)CC2 N1(C(=O)NC2CCCN(C(=O)OC)C2)Cc2cccc(C)c2CC1(C)C c1(C(N(CCCOC(N(C)C)=O)C)=O)cccc(F)c1OC(F)F c1(C(=O)NC2C(NC(CCOCCOCC)=O)CCOC2)cccc2ncnn12 C=CC1CCCN(C(=O)CC2CC(C(=O)NCC)C2(C)C)C1.C12CC(C1)C(=O)O2 C=CCCCCC(=O)NCC1(NC(c2cc(C)cnc2C)=O)CC(F)(F)C1 c1(C(C(=O)NC(=O)Cn2cc(CC3(CO)CC3)nn2)O)ccc(F)c(Cl)c1 C(=O)(CC(CC1CC1)NC(=O)CC12CCCC1C2)NCC1CC(=C)C1 c1(C(N(C2CCC2CF)C)=O)cc(F)c(CNC(C2(C)CC2Br)=O)c(F)c1 C1(C(N2C(C(=O)NCC(C3CCCC3)O)CCCCC2)=O)CC2(CCC2O)C1 c1(OC)cccc2c(CNCCC(C)(C)CN)cccc12 C(CN=c1ccc(C(C)C)c[nH]1)NC(=NCC)NC1CCOCC1C N1(C(C(C2CCOCC2)C)=O)CC(C(N)=O)(NCCCC2CCC2)C1 C1(NC(=O)CC(F)(F)F)CN(C(C2CC2C(F)(F)F)=O)CC2(CCOCC2)C1 c1(C(=O)NCCC23CN(C(C=CC=CC)=O)C(CC2)C3)[nH]nc2c1COC2(C)C C1(C#N)(C(N2CC(CCNC(C(CC)(C)C)=O)C(C)C2)=O)CCCOC1 CCCCC(=O)NC1CC(CCNC(C2(CCF)CCC2)=O)C1 Cc1cccc(C(COCCNCC)C2CCC2)c1.C(C(=O)OC)OCC(=O)C(=O)O COn1cnc(C)c1C(N1CC(NC(C2(n3cccn3)CC2)=O)C(COC)C1)=O c1(-c2n(C(C)C3CC3)nc(C(C)O)n2)cc(F)c2[nH]nnc2c1 C1(CNC(C2N(CC)CCCC2)=O)CC(C)(C)CN1C(C1CCCN1N=O)=O C12(C(=O)NC3C4CN(C(c5cc(C)[nH]c5)=O)C3C4)CC3CC(CC(C3)C1)C2 C(=O)(CC1=CCCCC1)NCC(C)(O)CNC(c1cnc(C2CCC2)o1)=O Cc1cc(NC(=O)CCC2CC(NC(=O)C(C3CCOCC3)F)C2)cs1 c1(C(C)C(=O)N2CC(CC(n3cc(-c4cnn(C)c4C#N)nn3)=O)C2)cc2ccccc2o1 Cc1cc(-n2nc(-c3nccs3)nc2C2CC2(F)F)ccc1C(C)(C)C c1(CC(=O)NCC2(NC(C=CCCC)=O)CCC2)cc(F)cc(F)c1 N1(C(=O)CC2(C(F)(F)F)SCCS2)CCN(C(C2(C3CCCCO3)CC2)=O)CC1 c1(CNC(C)Cc2cccc(F)c2)cnc2c(c1)CCC2.C(CF)OCCO C12(NC(c3c(OC)nsc3)=O)CCOCC1CN(C(c1cn3ccnc3s1)=O)C2 C1(NC(CNC(C2C(C)C2)=O)=O)CC2(C1)CN(C(c1c[nH]c(C(F)(F)F)c1)=O)C2 C1(NC(C=CC(CC)=CC)=O)CN(C(C2CN3CCCN2CC3)=O)CC2(CC2)C1 N1(C(C(N2CCC(C)C2)=O)=O)CCN(CC(=O)NCc2ccc[nH]2)C(=O)C1 C1(NC(C(C)(O)C2CC2)=O)CC2(CCCN(c3snc(Cl)c3C#N)C2)C1 c1(N2CCCC(CC#N)C2)nc2c(c(=NCC3CC(CC4CC4)CO3)[nH]1)CSC2 c1(C(=O)NC(C2CCOC2)CNC(c2c(C)nc(C)o2)=O)nccc(Cl)c1Cl c1(C(=O)NC2C3(CC(NC(c4cccs4)=O)C3)C2)cnn2c1S(=O)(=O)NCC2 c1(CCC)nc(C)c(C(N2CCC(C)(N(C(=O)COC(CC)CC)CC)C2)=O)s1 c1(C(N2C(CNC(c3ccc(F)cn3)=O)CC2)=O)n[nH]c2c1COC2 c1(CNC(=NCC)NCCCn2ccnc2C)cc2cc(F)ccc2o1 c1(C(=O)NC2(C(=O)NCCC3CCN(C)CC3)CCCCC2)cc(O)ccc1F CCC(CC)C(F)C(=O)N1CC(C(=O)N(C(C)CC)C)CCC1(C)C CC1CC(NC(=O)C(C)(C)NS(C)(=O)=O)CCN1C(C1CCCN1C)=O N1(C(C(CC)COC)=O)CCCCC(N(C)C(c2cc(Cl)c(Br)[nH]2)=O)C1 c1(CC(N2CC(CCNC(Cc3cn(C)nc3)=O)C2)=O)ccc(O)cc1 C=CCC(F)(F)C(=O)NCCC1CC(CNC(c2cc(O)nc(O)c2)=O)C1 CC(F)(F)C(F)C(=O)NC(CC(N1CC2(CC(OC)C2)C1)=O)C1CC1 C(=O)(N=c1[nH]nc2[nH]ccnc1-2)c1ccc(-c2ccc(C)cc2C)cn1 C#Cc1ccccc1CC(N1CCC(C)(CNC(c2cccc(OC)c2)=O)C1)=O c1(NCC2N(c3cccc(C)c3)CCC2)nnc(C)c(C)n1.N12CCCCC1C2 c1(OC)cccc(NCCC(=O)NC2(CNC(=O)CC3CC(=O)NC3=O)CC2)c1 c1(C(N(C)CC2CCCN(C(C(C)P(C)(C)=O)=O)C2)=O)cc2c[nH]cnc-2n1 c1(CC)nc(C)n(C)c1C(N1CCCC(O)(CN(C(=O)CC(C)(C)C)C)C1)=O C1(O)(CCNC(C(CC=C)C)=O)CCCN(C(c2ccnc(C)c2C)=O)C1 c1(OC)cccc(C(=O)NCC(C)(F)CNC(c2c[nH]nc2[N+](=O)[O-])=O)c1C N(C(=NCCC(C)N(C)C)NCc1ccnn1C)C(c1ccc(OC)nc1C)C C(C(=O)NCCC1(NC(=O)Cc2cn(C(C)C)nn2)CCCC1)(C(C)(C)C)SC C1(NC(CCC=C)=O)CN(C(C2CC2F)=O)C2(CCC2)C1 C1(C(N(C(CC(C)C)C)C)=O)C(C2CC2)CCN1C(=O)Cn1nccn1 C(C1=CCN(C(c2ncc[nH]c2=O)=O)CC1)NC(c1cc(OCC)no1)=O c1(C(=O)OCC)cnc(N2CCC(NC(C3CCCCC34CC4)=O)C2C)cc1C Cc1cc(C)c(CC(=O)OCC2CC(=O)N(CC3CC3)C2)c(C)c1 C(=O)(C1CCCn2ccnc21)NCC1C2N(c3c(C#N)cnc(C)n3)CC(CC2)C1 C1(N(C(CCOCCC)=O)C)CN(C(c2cc(C3CC3)no2)=O)CC12CC2 C1(CCN(C(C(C)CN(C)C)=O)C)CCCCN1C(c1cnn(C2CC2)c1)=O N1(C(C2N(C(C(CCC)F)=O)CCCC2)=O)CCn2nc(C)cc2C1 C1(C(=O)NC23CC(NCc4ccc(NC(C)=O)s4)(C2)C3)Cc2ccccc2CO1 Cc1ccc(C)c(C(=O)NC(CNC(C2CC3CCC3C2)=O)C2CC2)c1C Cc1ncc2cc(C(=O)NCCC3CCN(C(=O)C=C4CCC(C)C4)C3)ccn12 N1(C(c2sc(CC)c(C)c2)=O)CCC(C2CC2)(CNC(c2c(C)ncn2O)=O)C1 c1(OC)cnc(C(N2CC(NC(=O)C(C)c3cncs3)C2)=O)cn1 c1(-c2ccc(C(=O)NC(CNC(C(COC)OC)=O)C3CC3)o2)ccccc1C C1(CNC(CCC#N)=O)(CNC(=O)CC(=O)NC2CC2)CC12CCC2 N1(C(CC(COC)COC)=O)CC2(CCC2)CC1C(=O)NCCN(C)OC c1(C(C)NC(=O)NCc2cccnc2)ccc(-n2cncn2)cc1 C1(C)(C(=O)OC)CCN1C(c1coc(C(C)NC(=O)CC(C)F)n1)=O C1(C(=O)NC2(C)CCN(C(C(C)c3ccsc3)=O)C2)CCC(C)(C)CC1 c1(OC)ccc(CNCC2CCCCN2C(c2cccc(F)c2C)=O)cc1CCO Cn1cnc(C(=O)NCCCN(C(C2CC23CCC3)=O)Cc2cccnc2)c1 C=C(C)C(CC(=O)NC1CCCC1NC(=O)COc1ccsn1)OCC Cc1noc(C)c1C(N1CC(NC(C2CC(=O)N(CC3CC3)C2)=O)C(C)C1)=O C=CC1(C(N2CC(N3CCN(C(C4CC4C#N)=O)CC3)C2)=O)CCOCC1 c1(C(=O)NCC23CC2CN(C(=O)C(F)C2CCCC2)C3)ccn2nnnc2c1 c1(C2CCN(C(CC3C(C)CCO3)=O)CC2)c[nH]c2cc(Cl)ccc12 C(=O)(CCC(=O)NCC(CO)NC(c1coc(N(C)C)n1)=O)N(CC)CC C(CC(C(=O)NCCc1ccon1)NC(C1C=CCS1)=O)OC Cc1ccc(C(=O)N(C)CC2CC(F)CN2C(=O)CCC2CNC(=O)N2)nc1C N1(C(c2c(COC)noc2)=O)CCC(F)(CNC(C2(C)CC2(F)F)=O)C1 CC(CC(=O)N1CCCCC(C)(F)C1)C(C)(C)NC(=O)C1=C(C#N)CCC1 c1(C(=O)NCC2C(NC(c3ncccc3Br)=O)C2)cc2c(nn1)CCCO2 c1(C(=O)NC(C)CN(C(=O)Cn2ccnc2)C)ccc(N(C)C2CC2)cc1 C1(C)(CCNC(C(C)C2CC2)=O)CCN(C(=O)CN(C2CCSC2)C)C1 C1(C(=O)NCC2(COCCO)CCCC(C)(C)C2)CCC2(CCOCC2)CO1 c1(NC2(CO)C(C)CCC2)nccc(=NCc2ccnc(-c3ccncc3)c2)[nH]1 c1(C(=O)NCCN(C(=O)Cn2cnc(=N)[nH]2)CCC)ncnc(C)c1C C(CCC(C)NC(=O)C(c1cnn(C)c1)C)NC(CC1CC(C(=O)OC)C1)=O C(C)(CCC(=O)N(C1CCN(C)CC1)C)NC(COC(CC)C)=O C1(NC(c2cccc(N)n2)=O)CN(C(c2cc(O)cc(O)n2)=O)C2(CCOC2)C1 c1(CNCC(c2cccs2)C)cc(Cl)c(F)cc1[N+](=O)[O-] C(C1Cc2ccccc21)NC(CC1C(NC(c2ccn(C)n2)=O)CCCC1)=O C1(N(c2nnc(CCCOC)n2C)C)CCCN(C2CC2C)C1=O c1(CNC(C2CC(CNC(c3cnn[nH]3)=O)OC2)=O)ccncc1Cl N1(C(=O)Nc2ccc(C)cc2)CCC2CN(C(c3ccoc3)=O)CC12 Cc1ncn2ccc(C(=O)NC34CCCN(C(=O)CCS(C)=O)CC3C4)cc12 n1(C2CC(N)C2)cc(C2CN(C(=O)CCNC(N)=O)C2)nn1 C1(NCc2c(C(=O)OCC)ccs2)CC2CCC(C1)N2C c1(C(=O)NCC2C(NC(C(C)C3(O)CCC3)=O)CC2)ccc2n[nH]cc2n1 N1(C(c2scc(C)c2)=O)CCCN(C(=O)COC2CCC(F)(F)CC2)C(CO)C1 CCCC(CCC)=CC(=O)NC(COC)C(=O)NC1C(O)CC1O n1(CCC)cccc1C(=O)N(C)CC1CCCN1C(c1csc(C(C)=O)n1)=O n1(CC(=O)NCC(CC)NC(c2cc(C)cc(O)n2)=O)c([N+](=O)[O-])cnc1C c1(C(=O)NC(CC)CNC(c2conc2C2CCCO2)=O)csc(Cl)c1OC N1(CC(=O)NCCC(C(C)C)NC(=O)CC(C)C(F)F)Cc2ccccc2C1=O Cn1c(C(N2CC(C)(NC(=O)C(C3CCCCCC3)O)C2)=O)ccc1C#N N1(C(CC(C=C)CC)=O)CCC2(CCCN(C(C3CC3C(=O)OC)=O)C2)CC1 N1(C(C(CN(CC)CC)F)=O)CCC(C)(CCNC(=O)C=CBr)C1 N1(C(C2C(Nc3nc(SC)c(Br)cn3)CCC2)=O)CCn2c(C)nnc2C1 C1(N2CCCC(C)(C(N(C)Cc3csc(C4CC4)n3)=O)C2)CC2(CCNCC2)C1 c1(C(N2C(C)CN(C(=O)C3=CCCS3)CC2)=O)cc2ccc(F)cc2[nH]1 C=CC(CCC)CC(=O)N(C)CCNC(c1cc(Cl)c([N+](=O)[O-])[nH]1)=O c1(C(=O)NCCN(CC(C)O)C(=O)C=CC2CC2)cc2c(cn1)OCCC2 n1(CC)c(-n2nc(C)cc2C)cnc1S(=O)(=O)Cc1cnn(CC(F)(F)F)c1 C1(C(N2CCC(C3N(c4snc(CC)n4)CCC3)C2)=O)CC(=O)NC2CCCCC12 n1(CC)c(C(=O)N(C)Cc2ccc(CNC(=O)C(C)(C)CF)cc2)cnc1O CC1CCOCC1C(=O)NC1CC(CCNC(c2ccc(C#N)[nH]2)=O)C1 N1(C(C(C#C)(C)C)=O)CCCC(C)(NC(c2ccc3c(c2)CC3)=O)C1 N1(C(C(C)(C)CF)=O)CCCC(F)(CNC(C2(O)CCOC2(C)C)=O)CC1 N1(C(c2ccc(F)cn2)=O)CCCCCC1C1CCCO1 N1(C(Cn2c(C)cnc2)=O)CC2=C(C1)CN(C(=O)CCC(C)(C)N(C)C)C2 C=CCC(CC(=O)NCCCC1CCOC1=O)NC(c1ccc[nH]1)=O c1(C(=O)NCC2CCN(C(c3ccc(C(C)C)o3)=O)C2)ccc(Br)cc1N c1(CC)ncccc1C(=O)NC(CCSC)C(=O)NCC1(C)CC=CCC1 CCC(C)(C)C(=O)NC1CCCCC1CC(N1CCC(Cc2ccccc2)C1)=O Cc1c(C(F)(F)F)cccc1CNC(=O)C(=O)NC1(C)CC1C1CCN(C)CC1 C=C1CCN(C(c2cn(C)c(C)n2)=O)C(C(N2CC(OC)CC(C)C2)=O)C1 C1(C(=O)NC(C(C)C)CCNC(c2cccc[n+]2[O-])=O)CCc2cncn2C1 c1(C(=O)NCC=C(C(=O)NCCC(C)C)C)ccc(=N)[nH]c1 CC1CCN(C(=O)C(N2CCCCC2CNC(=O)CCC2(C)CC2)=O)CC1 Cc1cc(C#N)ccc1CC(N1CCSCC1C(=O)NCc1nccc(O)n1)=O c1(C(N2CC(NC(C(=O)N(C)C)=O)C3(C2)CCC3)=O)cc2cccnc2cc1F Cc1cc(C(=O)NCCC2(O)CN(C(=O)C(C)OCC(C)C)C2)nnc1C Cc1ccc(C(=O)NC2CC(CCNC(=O)C(C(C)C)N(C)C)C2)c(O)c1C c1(C(N(CCNC(=O)CCc2nnc(C)n2C)CC)=O)ccc2ncncc2c1 N1(C(c2ncc(C)c(Cl)c2)=O)CCCN(C(=O)C=CC2CCCO2)C(C)C1 c1(NC(=O)NC)ccc(Cl)c(C(=O)NC(CC(C)C(C2(C3CC3)CC2)=O)C)c1 CN1C(=O)CCCC1C(N1CCC(NC(=O)CC2CCCSC2)CC1)=O c1(N(C)Cc2cc(Br)cs2)ccnc(NC2(c3cccnc3)CCC2)n1 N1(CC(=C)Cl)CCC2(CC1)CC2(C)C(=O)NC(C)C(C)C CC1CN(C(=O)Oc2ccccc2C#N)CCCO1 c1(C(C)C(=O)NCCC2(C(=O)N(C3CC3)CC3(O)CCC3)CCC2)ccn(C)n1 C1(C(NOCCOCC#C)=O)CC(NC(=O)Cn2cnnc2O)C1(C)C C12(COC)COC(CC(c3nc(C)[nH]c3Br)c3nnnn3C3(C)CC3)(C1)C2.NC C1(NC(CSC)=O)CC2(C1)CN(C(c1cnc(Br)c(N)c1)=O)C2 C1(CCC(=O)NC(C2(CNC(CN(CCOC)C)=O)CC2)C)CCCCO1 c1(N(C2CCNCC2O)Cc2c3ccc(C)cc3[nH]c2)ncnc2c(Br)csc12 N(C(=NCCCF)N1CCC(O)CC1)CC.N12CCCC(C1)C(C)NC2=O C(C)(C(=O)NC(C(=O)NCCCF)c1ccco1)OCCOC C1(NC(=O)CN2CC=CC2)CCCC2CN(C(C3CCCCC3O)=O)CC12 n1(CC(=O)NC2C(NC(c3scc(C)c3)=O)CCC2)cc(C#N)cn1 c1(C(N2CCC(N(C(=O)CC3(C(F)(F)F)CC3)C)C2)=O)cccc(C(F)F)c1F N1(C(C(COCC)N=[N+]=[N-])=O)CC2C3CCC(C2C1)N(C(c1n[nH]c(C)n1)C)C3 c1(NCC2CCC(C)C2)ccccc1C(=O)NCC(C)(C)CCO c1(C(N)=O)ccc(Br)cc1CS(=O)(=O)Nc1cc(C(=O)O)on1 C(C)(C)(CC#Cc1ccccc1)c1n(CCC(C)(C)C)nc(C2CC2)n1 c1(OC)cc(CNC(c2sc(I)cc2Br)=O)c(C2CC2)cc1C CC(CCCC(=O)NCC1([Si](C)(C)C)CC1)NC(=O)Cc1cnns1 C(C(=O)NCC(C)=CC(=O)NC1CC(CO)C2CC12)(C(C)C)SC Cc1ccnc(NC(c2cscc2-c2cccnc2NC(C)(C)C)=O)c1F CC1CCN(C(c2cnn3cc[nH]c23)=O)C(CNC(=O)CSCc2cscn2)C1 C1(C(=O)NC(C)CN2CCCCC2)CC(C)CN1C(c1csc(C#N)c1)=O c1(C(C)(C)C)ccc(C(=O)NC2C=CCN(Cc3cn(CCO)nn3)C2)cc1Cl Cc1c(C(N2CCC(O)(NC(C3CC(O)C3)=O)CC2)=O)cccc1Br c1(OC)c(C)csc1C(=O)NCC(O)CN(C(=O)C(C)N(C)C)C c1(C(C(=O)N(C)Cc2ccco2)O)cc(F)c(F)cc1F.C12CCN(CC1)C2=O C(=O)(CCCCCC(C)(C)C)NC(C1CCCN(C(c2cn(C3CC3)cn2)=O)C1)C C(C)(c1ccco1)=CC(=O)NCC1(C(=O)NCC(CC)N(C)C)CC=CC1 C12(C(=O)NC3CCC(O)C3)CC(CO)(CN1C(c1n[nH]c(O)n1)=O)C2 c1(Oc2nccc(CNC(=O)C(=O)OC)c2)ccc2c(COC)csc2c1 C1(C(=O)NCCCC(CC)C)CN(C(C2(O)CC2)=O)CC1(C)C CC(C)(C)C(O)C(=O)N1CC2(NC(=O)CSc3cccc(F)c3)CCC1C2 n1(CC)c(C)nn(CC(=O)NC(C)C(C)(C)NC(=O)C(C)CSC)c1=O CC(C)CCC(C)N(C(=O)C(F)C1CC(NC(=O)Cn2cc(C#N)cn2)C1)C CN1CC(CC(=O)NCC(O)CNC(C2CC2C(F)(F)F)=O)c2ccccc21 c1(C(N2CCCC2)CNC(C2CC2(F)F)C)nc2ccccc2s1 N1(C(C2C(CC)N(C)CC2)=O)CCCN(C(=O)CN2CCCCC2)C(C)C1.CCF Cc1c(C(N2CCC(NC(=O)CCOC3CCCOC3)C2)=O)cncc1Br Cc1cc(Cl)cc2cc(C(=O)NC34CC(NC(=O)Cc5csnn5)(C3)C4)[nH]c12 N1(C(c2ccc3ccccc3c2)C(=O)NC2CC2)CCOCCC12CCC2 N1(C(CCSCC)=O)CCC2(CC1)CCN(C(C1(C)CC1)=O)CC2 c12ccc(cc1)CN(CC1CC1)C2C.C1(C)(C(=O)OCC)COCCO1 C#CCCCCC(=O)NC(C)CNC(=O)C(c1ccc(F)c(Cl)c1)C N1(C(CCC(=O)NCCC)=O)CCN(C(=O)CC(C)(F)F)C2COCC12 CC1CC(C(=O)NCCSC(F)F)N(C(c2ccc(Cl)o2)=O)C1 c1(C(=O)NC2CN(C(c3cc(C)c(C)nn3)=O)CC(F)C2)cccc2nccn12 c1(C(=O)NC(C(C(=O)NC(COC(C)=O)CO)C2CC2)=O)cc(Cl)c(F)cc1C C1(NC(N)=O)CCN(C(=NCc2ccns2)NC2CCC2)C1 CC(CC(F)F)C(=O)N1CC(n2cc(-c3cncc(C#N)c3)nn2)C1 c1(OC)ccc(CC(=O)NC2CCN(C(C3CCN(C)C3C)=O)C2C)nc1 N1(C(CCCCN(C(C)=O)C)=O)CC2CN(C(c3ccc(C)cn3)=O)CCC12 C(CC)(CC)(CCNC(C)=O)N(C(CC)CC)C(C1CC(OC)(OC)C1)=O C(=O)(C(C)C(C)S(C)(=O)=O)N(C(C)CNC(c1ccc([N+](=O)[O-])cc1N)=O)C n1(CC(N2CCN(C(CC(C(C)C)OC)=O)CC2)=O)ccc2ncc(Br)cc12 CC(C)(CC(F)(F)F)C(=O)NCCCCCn1cccn1 c1(C(=O)NCC(C)S)ccc2c(c1)nc(O)n2-c1cn[nH]c1 C12(n3cccn3)CCN(CC1)C2=O.c1(C(N(C)C)=O)cccc(O)c1 N1(C(c2c(C)nc(C)o2)=O)CCN(C(=O)C(CO)c2ccccc2)C(C)C1 CN1CCN(C)C(C(N2CCC(NC(=O)CC34COC(C)(C3)C4)C2C(C)C)=O)C1 C(C(=O)NC1CC1OC(C)=O)(C(C)C)N(C(C)CC(=O)Oc1ccccc1)CC N1(C(C(C)OCC(C)C)=O)CCCC1C(=O)N(C1CC2CC2C1)C Cc1c(Cl)c(C(=O)NC2CCC(NC(c3cc(Cl)c[nH]3)=O)C2)nn1C c1(N2CC=CC(OC)C2)nc(N2CCC(CCN(C)C)C2)nc2c1SCC2 C1(C(=O)Nc2cnc3cccnc3c2)COc2cccc(Cl)c2O1 N1(C(CCC(CC)O)=O)CCN(C(c2cc(C)cnc2F)=O)CC(O)C1 C1(CN(C(=O)C=Cc2nnn(C)n2)C)CCCN(C(=O)CCCn2cccn2)C1 C1(C(=O)NC(C2(O)CN(C(C3CS(=O)(=O)C3)=O)C2)C)CC2CC2C1 Cc1ccn(C(C)C(=O)NC(CNC(c2cnsn2)=O)CO)n1 c1(CCC(=O)N(C(C(=O)N(C(C)C(=O)NC)CC#C)C)C)cnc(O)[nH]1 N1(C(c2n[nH]c(C)c2N)=O)CC(C)CN(C(=O)CC(C)(F)F)CC1C c1(C(N2CCC(NC(c3nc(C)oc3C)=O)C(C)C2)=O)cc(=O)n2nccc2[nH]1 CC1=NOC(C)(C(=O)NC(c2nocc2C(=O)NCC2CCCC2CF)C)C1 c1(CCC(=O)NC2CC(CCNC(COC)=O)C2)cnc(C2CC2)o1 C1(C(=O)NCCOc2ccccn2)CC2CCC1N2C(c1cccc(=O)n1O)=O Cn1ncc2c1CCCN(Cc1ccnc(-n3ccnc3)c1)C2 c1(C(N2C(CC(=O)N(CC3(CO)CCN(C)C3)CC)CC(O)C2)=O)cc(O)ncc1F N1(C(c2[nH]ccc(=N)n2)=O)CCC2(CC1)CN(C(C1CCCCS1(=O)=O)=O)C2 c1(NCC(C)OC(F)F)cc(=NCC(c2ccsc2)N2CCCC2)[nH]cn1 N1(C(C(C)CS(C)=O)=O)CC2CCN(C(c3coc(-c4ccccc4)n3)=O)CC12 Cc1cccc2c1CCOC2C(=O)NC(C)CNC(c1cc(C(C)C)[nH]n1)=O N1(C(C(COC)O)=O)CC2CC(C1)CN(C(=O)CCNC(C1CCCCC1)=O)C2 c1(OC)cccc(O)c1C(=O)NCC(C)(C1CC1)NC(C1CCCC(C)(C)C1)=O C1(n2cc(-c3csc(C)c3)nn2)CCCN(c2ccc(F)c(C)c2)C1=O.CCO c1(C(N2CC(CCNC(COCCOC)=O)OCC2)=O)cncc2cnccc12 c1(CNC2CC(C(=O)Nc3ccc(C)c(O)c3)C2)c(F)ccc(O)c1F C1(C(C)O)CCCN1C(=O)CC1CCCN1C(c1cncs1)=O C1(C(=O)NCC(C)(O)C2CCCC2)COCCN(C(=O)CCn2ccnc2)C1 C1(C(N2C(C(=O)OC)CC(F)C2)C(=O)NCc2cccs2)CCCC(C)(C)C1 C1(CN(C(c2ccc(-c3cccc(O)c3F)cn2)=O)CC)Cc2ccccc2O1 C1(C)(COC)CC2CN1N1CC(C1)OCC(=O)O2.C1CC(C#N)C1.C(=O)C1CC1 c1(C(=O)NC(C(=O)N(CCC)CCSC)C2CC2)ncc(C#N)cc1C C1(NC(C2C(NC(=O)OC(C)(C)C)C2)=O)CC(NC(c2nncs2)=O)C1 N1(C(C2C(=O)NCC2)=O)CC2CN(C(c3ccc(N4CCOCC4)nc3)=O)CC12 C1(C(N(C2CC(O)C2)C)=O)CCCC(NC(=O)CC(C)(C)C)C1 N1(C(C2C(OCC)C2C)=O)CCOC2(CCN(C(=O)C=CC(C)(C)SC(CC)OC)C2)C1 c1(NC(CSC)=O)sc2c(c1C(N1CCC3(CC1)CC(O)C3)=O)CCCC2 c1(C(=O)NC(C)CCNC(c2nnn(C)c2N)=O)n[nH]c2c1COCC2 Cn1nncc1NNC(=O)C1(c2cc(Cl)ccc2Cl)CCC1 C(c1cccc(F)c1Cl)=CC(=O)NC1CCN(C(C(CC)=CC)=O)CC1O c1(C(=O)NC(C(C)(C)NC(C2(SCC)CC2)=O)C)cc(F)cc2ccncc12 c1(OC)cccc(O)c1C(=O)NCCC1(OC)CN(C(c2n[nH]c(C)c2C)=O)C1 N1(CC(=O)NCC2(O)CC(CNC(c3ccc(COC)o3)=O)C2)CCOCC1=O N1(C(C(C(C)C)OCC)=O)CCC(C)(C)C(NC(=O)C(CC)CC(F)F)C1 C1(NC(Cn2c(C)cc(C(F)F)n2)=O)CCCN(C(=O)CNC(=O)C2CC2)CC1 C#CC1(O)CC(c2nc(C3CC3CS(C)(=O)=O)no2)C1 C1(F)(C(=O)NCCN(CCOC)C(C2(C)CC2C(F)(F)F)=O)CCCC1 Cc1cc(C(N2CCC(NC(=O)CSc3c(C)n[nH]c3C)C(O)C2)=O)cc(C)c1 C(C(Cc1cn(CC(O)CO)nn1)C(=O)O)NC(c1cc(C(=O)O)n[nH]1)=O C1(NC2CCC(N(C(=O)C(=O)SCC(F)F)C)CC2)CSC(c2ccccc2)=N1 c1(N2CCCCC(SC)C2)ccncc1S(=O)(=O)NCC(O)Cn1cccn1 N1(C(C(COC)OC)=O)CC(CNc2ccco2)C2(C1)CN(C(=O)C1=CSCS1)C2 CCC(C)C(C(=O)N(CCCCNC(c1sccc1CC#N)=O)C)NC(C)=O Cc1cc2nccnc2cc1C(N1CCN(C(=O)C(C)C(C)O)CCC1C)=O C1(C(=O)NCC2CC(C)N(C(C3CC3(Cl)Cl)=O)C2)CCC2(CC1)N=N2 Cc1ccc(OCC(=O)NCCCSC)cc1C.C1(C(C)C)CC(C)CCC1C(C)C C(=O)(C1=C(Cl)CCOC1)N(CC(N1CCC(C)C1CC1CC1)=O)C N1(C(COCCC=C)=O)CCC(CNC(=O)COCC2CCCO2)CC1C N1(C(CCC(C)(C)OC)=O)CC2CCCC2(CNC(c2ccnnc2)=O)C1 N1(C(CC(CN(C)C)O)=O)CCCC(CNC(=O)Cn2nnc(=O)[nH]2)CC1 C12(N(C)C(=O)NCC3(C)CCCCO3)CC3CC(C1)CC(c1ccccc1)(C3)C2 C(C(C)(C)C#CC(=O)NCC1CCC(O)CC1)NC(c1cc(CC)sn1)=O CCC(F)(F)CC(=O)NC(CC(=O)N(C)CCc1cccs1)C(F)F N#Cc1cncnc1N1CC=CC(NC(c2cccc(-c3ccoc3)c2)=O)C1 C1(CCNC(CC2(OC)CCC2)=O)CN(C(=O)COC2CC=CC2)CC1C Cc1csc(C=CC(=O)NCC(C(C)(C)C)NC(=O)C(n2nccc2C)C)n1 C1(C(=O)NCC(CNC(=O)C=Cc2ccncc2)OC)CCCCC1N=[N+]=[N-] C1(C)(CNC(C(CC)F)=O)CCN(C(c2c[nH]cc2-c2csc(C)n2)=O)CC1 C(C)(CNC(=O)Cc1cc[nH]n1)(C(C)C)NC(C(c1scc(C)n1)(F)F)=O C12(NC(=O)C3=CCCCC3)CCCC1CN(C(=O)CC1C=CCC1)C2 N1(C(COCC(C)C)=O)CCC(C(F)C(=O)NCCc2cn[nH]c2)C1 c1(-c2cn(CC3S(=O)(=O)CCC3)nn2)ccc(O)c(F)c1 c1(CC(=O)N(CC(C)NC(C(CC)N(C)C)=O)C)ccc(C)c(Cl)c1 c1(OC)cc(F)c(-c2ccc(C(N3CC(O)C(O)C3)=O)nc2)cc1OC Cc1[nH]c(=NC2(CNC(c3cc(Cl)c4c(c3)OCCO4)=O)CCC2)ccc1C#N c1(CCNC(=O)Nc2ccc3cnn(C(F)F)c3c2)cccc2cccnc12 c1(OCC(N2CCC(CNC(=O)CCCF)C2)=O)ccc(F)cc1O C1(CNC(COCC)=O)(CNC(=O)C=Cc2ccc(SC)s2)CC2CCCC2C1 C=C(Cl)CCC(=O)NC(C(=O)NC1(CO)CC(C)C1)C(C)O CN1CCC(C(N2CCCCC2CNC(c2ccnn2C2CC2(F)F)=O)=O)CC1 c1(CC#N)ccc(C(=O)NCC(CNC(c2ccnc(C3CC3)n2)=O)CO)cc1 c1(N2CCC(NC(CCOC)=O)C23CCC3)ncnc2cc(C3CC3)nn12 c1(C(C)C)cc(F)c(C(N2CCOC(CNC(=O)CC3CCCO3)C2)=O)cc1F C1(NC(C(CCC)N(C)C)=O)CC2CN(C(c3ccccc3C)=O)CC2C1 C(c1ccc(F)cc1F)=CC(=O)Nc1scc(-c2cc(COC)c(Cl)cc2)n1 C1(CC(=O)NC)CN(C(=O)C=CC2CCOC2)CCN1C(=O)Cn1cncn1 CCC(CCOC)C(=O)NC1(CCNC(=O)Cc2cc(C)cc(C)c2)CCC1 Cc1cc(-c2cn(CCN(C)C(CC(C)O)=O)nn2)oc1Br c1(CNC(=O)CCn2ccnn2)csc(CNC(C2CC2C2CC2)=O)n1 c1(CC(=O)N(CCCNC(C2CC2(Cl)Cl)=O)C)coc2cc3c(cc12)CCC3 Cc1coc2ccc(C(=O)NCC3COCCN3C(C3C(C)C3C)=O)cc12 O=C1CC2(CCN(C(=NCCCCl)NC(=O)CSc3ccccc3)C2)CN1 c1(C(N2CCN(C(C(CCC)C)=O)C(CC(F)F)C2)=O)ccc(C)c([N+](=O)[O-])c1 c1(CC)ccc(C(=O)NCCC2CN(C(c3nnn(C)c3N)=O)C2)c(C)n1 c1(C(N(CCCNC(c2c(C)cc(SC)o2)=O)C2CC2)=O)cc(O)cc(Cl)c1 c1(C(=O)NC2(CC=C)CN(C(=O)C(C)N(C)C)C2)nnc2ccccc2n1 C1(C#N)(C(N2CC=CC(NC(c3cncc(C)c3)=O)C2)=O)CCN(C)CC1 C1(C(N2CC(OC)C2)=O)CCC(C)(C)OC1.C12OCCC1NC2=O Cc1nc[nH]c(=NCC2CC2(F)F)c1NC(C1CCCN1C(N)=O)=O N12CCC(CC)(CC1)CNC(=O)CCC1CC(C1)C2=O.C(C(O)C(C)C)N(C)C N1(C(C)C)CCCC1C(=O)NCC1CC(NC(c2cnc(C(C)(C)C)s2)=O)C1 C1(N)CCC(=O)NC1.C1(NC(CN(C(=O)OCC)C)=O)CC(O)C1 C(=O)(CC(C)C(C)(C)C)N1CC(NC(c2c(Cl)cnc(C)n2)=O)C(F)CC1 C1(C(=O)NCc2ccnc(Br)c2F)CN(Cc2cccc(CO)c2)CCC1(F)F N1(C(c2c(C)n(C(C)C)nc2)=O)CC(C)Oc2c(F)cccc21 N1(C(Cc2ccn(CC)n2)=O)CC2C(CNC(=O)CCc3scnc3C)C2C1 Cc1cc(CN(CCO)CC)cc(C)c1N.C(CCO)SNCCO n1(CC(=O)N(C)C)cc(C#CCNC(c2cccc(OC(C)(C)C)c2)=O)nn1 C1(NC(C2CC(=C)C2)=O)CN(C(C2CCCS2)=O)CCC12CCC2 Cc1nc2c([nH]1)CN(C(=O)C(C)(C)C1CCN(C(C3CC3(C)C(F)F)=O)C1)CC2 c1(CC(=O)NC2CN(Cc3c(Cl)ccc(C(=O)O)c3)C2)ccc2ncnn2c1 C1(C(=O)NCCC(C)N(C(=O)Cn2cnnn2)C)CN(C)CCO1 C1(N(C(C2CCN(C)CC2)=O)C)CCCN(C(=O)C(C)(C)c2ccn(C)n2)CC1 c1(C(C(=O)NC2CCC(NC(CC(=O)OC)=O)C2)C)cc2ccccc2s1 C(=O)(CC1OC(=O)c2ccccc21)N(C(c1cn(C2CCN(C)CC2)nn1)C)C c1(OCC#C)cc(C(N2CC(NC(=O)C#CC(C)(C)C)C2)=O)cc(Br)c1 c1(C(=O)NCC(C)(C(C)C)NC(c2ccc(OC)o2)=O)cc(F)c(F)cc1F CC1(NC(=O)CCCCCNC(=O)Cc2ccccc2)CCCCCC1 c1(C(N2CCN(C(C)C)C(C)C2)C(=O)NCC)cc2cccc(Cl)c2o1 C1(C(N(C)Cc2ccc(C)nc2)=O)C2CCN(C(C3CC4CCC3CC4)=O)CC12 N1(C(C(C)CN(C)C(C2CC(Cl)(Cl)C2)=O)=O)CCC(CC2CC2)CC1 C(=O)(CC(C)(O)C(F)(F)F)NCC1CCC2(CN(C(CCCCCC=C)=O)C2)O1 CP(C)(=O)CN1CCC(C(=O)NCCCCCCCn2cc(C(O)CCl)nn2)C1 c1(C(=O)NC(CC)CN(C)C(c2ncc(C(F)F)s2)=O)cncn(C)c1=O N1(C(CC2(C)CCCO2)=O)CC2CC1CC2CNC(c1cccnc1S)=O C12(NC3C(C)CCN(C(=O)C(F)(F)F)C3C)CC3CC(F)(C1)CC(F)(C3)C2 c1(C(=O)NCCCOCCN(C(C2C(OC)C2)=O)C)c[nH]nc1-c1cnn(C)c1 C1(C(=O)NC2CC(CNC(C(CC)CC)=O)C(O)C2)CCc2c[nH]nc2C1 C#CC1(C)CCCN(C(C2CC(CNC(=O)C=CC(=O)N(C)C)C2)=O)C1 C12(C(=O)NC3CC(CSC)C3)CCC(CC1)N(C(=O)CC1CCCCN1C)C2 C1(C(=O)OCC)CN(C(c2ccc(C(C(F)(F)F)NC)cc2)=O)CC1n1cccn1 C1(C(=O)NC(CCOC)CNC(c2ccsc2C(F)(F)F)=O)CC2(CCC2)C1 N1(C(C2(CNC(C3C(C)=CCS3)=O)CC23CCC3)=O)CCOCC2(CCC2)C1 Cc1ncc(C(N2CCN(C(c3sccc3CO)=O)C3CC23)=O)c(=N)[nH]1 c1(CN(C(CC)C)CCOCc2ncn(C)n2)ccc(-c2ccccc2CC)cc1 c1(NC(C(N2C(CCC)CCCC2)C2CC2CC)=O)c(C)cccc1C CC(C)(C(=O)N1CCCCC1CNC(C1CN2CCN1CC2)=O)C(N)=O C(=O)(C(CC(C)(C)C)OC)Nc1ccc(NC(C(C)NC(CC)=O)=O)cc1C C(=O)(C(C)(CO)NC(C12CSCC1C2)=O)N(C1CCC1O)C C1(CNC(CC(C)OC)=O)CN(C(c2cnn(C)c2F)=O)CC2(CCC2)O1 Cc1ccc(OCC(=O)NC(C)CCNC(COCC(C)C)=O)c(C)c1 C1(C)(C(=O)NC(C)CCCNC(C23COCC(C2)C3)=O)CCN(C)C1=O C1(C(=O)NC(CC(C)C)CNC(c2nc[nH]c2C(F)(F)F)=O)CC(S(C)(=O)=O)C1 C=C(C)CC(C(=O)NCC1CC2(CC2)CN1C(C1COC(=O)O1)=O)OC CCCC(CCCNC(c1nc(C)sc1C)=O)NC(c1ccc(C)cc1Cl)=O C(=O)(CC(C(F)(F)F)NC(c1ccc2cccnn12)=O)NC(CC(C)O)C C(=O)(C(O)C(F)(F)F)NC(C1CCN(C(=O)C=Cc2ccoc2)CC1)(C)C C1(NC(c2cnc(CC)[nH]2)=O)CN(C(=O)C=CBr)CCC1C c1(C(N2CCOCC(NC(C3CON=C(C)C3)=O)C2)=O)cn(C)c(=O)n(C)c1=O C1(C(=O)NCC(CNC(C2NC(=O)C(F)C2)=O)CO)CC2(C1)CC(O)C2 N1(C(c2c(C)nc(CC)o2)=O)CCCN(C(c2cc3ccsc3s2)=O)C(CO)C1 c1(CC)cc(C(=O)NCC2(C(=O)N(CCC(=O)N(C)C)C)CCCO2)n[nH]1 N1(C(c2cc(CCC)[nH]n2)=O)CC(NC(=O)C(CC)C(C)O)CC1(C)C C(=O)(CC(C)C(=O)c1ccccc1)N(CCC(C)NC(COC(CC)C)=O)C C1(NC(C2C(C=C)C2)=O)CCN(C(c2cn(C3CC3)cn2)=O)C1 CCCCC(=O)C(=O)NC(c1cnn(C)c1)C(=O)NC1CC12CCCCC2 S(=O)(=O)(c1cccc(F)c1)NC12CCC(NC(c3cccc(CO)c3)=O)(CC1)C2 Cc1ccc(-n2nc(C3CC3)cc2C(=O)NCCN(C(C2CCC2F)=O)CO)cc1.N CCC(C)C(C(=O)NCCc1ocnc1CNC(=O)CN1CC2CC2C1)OC N1(C(C2(C)CC2)=O)CCC(C2CCN(C(C3(n4cc(C#N)cn4)CC3)=O)CC2)C1 c1(C(=O)NCC(C)(F)C(=O)N2CCCCC2OCF)cc(C#N)ccc1O CC1(C)CC(NC(C2CCC2CNC(c2coc(C(F)F)n2)=O)=O)CO1 Cc1cnc(COCC(F)(F)F)c(S(=O)(=O)NCC(C)(C)C(F)F)c1.C1(C)CN1 N1(C(CSCCC)=O)CCCC2(NC(c3cccc(C)c3Cl)=O)CC2C1 c1(NC(C(C(C)C)NC(CC(COC)(C)O)=O)=O)ccc2ccoc2c1 N1(C(C(CC#C)O)=O)CC(NC(=O)Cc2coc(C(F)F)n2)C(C)(C)C1 c1(CNC(C2COCCN2C(=O)COC2CCCC2)=O)cncc(Br)c1 C1(NC(c2cc(OC)c(O)nc2)=O)CC2(CCN(C(C3OCCOC3C)=O)C2)C1 c1(C(=O)NC2CCC(NC(c3cc(Br)ccn3)=O)C2)cc2c(cn1)OCCO2 c1(C(=O)NCC(CCC)C(=O)NCC2(COCC)CC2)cnc2cc[nH]c2c1 c1(C2CN(c3n(CC#C)c(-c4nnc(C)s4)nn3)CC23CC3)cc(Br)ccc1Br O(C=CC(=O)NC(C)CC(C)NC(=O)CN1CCC(C)C1)CC C12(NC(c3csc(CC(F)F)n3)=O)CCC(CNC(C3CCSC3)=O)(CC1)OC2 c1(C(=O)OC)cc2c(s1)CN(C(=O)NC1CC(SC)C(n3ccnn3)C1)C2 CC1CC(F)(F)CCN1C(=O)CCCCNC(c1ncnc(O)c1F)=O C#Cc1cncc(C(N2CC(C(=O)N(C(CSC)CC)C)C(C)C2)=O)c1 C(C(C(=O)NOCC1CCCO1)N(C)C)NC(C(n1c(C)ccn1)C)=O c1(C(=O)NC2(C3CCN(C(c4cc(C)no4)=O)C3)CC2)ccc2c(c1)CN(C)C2 C1(CN(C(c2n[nH]cc2C)=O)CC)CCN(C(=O)CC2CNC(=O)O2)CC1 c1(CCCC)ncc(C(=O)NC2(CNC(C3(CC)CCC3)=O)CCC2)s1 S(=O)(=O)(c1cccs1)NC(C)C(N1CC(NC(C2(CCF)CCC2)=O)C(O)C1)=O c1(C(=O)NCC2(Nc3ncc(O)cn3)CCCC2)ccc(=O)n(CCF)n1 C(C(C)(C)CC(=O)NC1(C)CSC1)NC(c1cccc(CC)n1)=O c1(C(C(N2CC(NC(c3cncc(OCC)c3)=O)C2)=O)C)cccc(Br)c1C c1(NC(=O)CC2(OCF)CN(C(=O)CCc3cccc(O)c3)C2)ccc(F)cc1 C1(NC(C(=O)NCc2c(C)n3c(s2)ncc3)=O)CCCCC12CCOCC2 N1(C(CCC(=O)OC)=O)C2CCCC1CN(C(C1(C3CCCCO3)CCC1)=O)C2 C1(C(N(CCN(C(=O)CCCOc2ccccc2Cl)C)C)=O)CC12CC2(F)F CN=C(NCC1CCCSC1)NC1CC(OC)C1(C)C.C(C)(C)(C)O c1(N2C(c3n(C(CC)C(N)=O)ccn3)CCC2)c(Br)cc(F)cc1[N+](=O)[O-] C1(CO)CC2CN(N3CCOC(C4CC4F)C3)CCN2C1 N1(C(C(CC)C)C(=O)NCCOCC2CC2)CC2NC(=O)C(=O)NC2C1 N1(C(C2CCC(C)CC2)=O)CCc2cccc(C(N3CCCNC(=O)C3)=O)c2C1.NCC Cc1ncc2n1CC(C(N1CC(OCCNC(=O)CCF)C1)=O)CC2 c1(C(=O)NCC(O)CNC(C23CCC2CC3)=O)cc2cccc(Br)c2cn1 CCC(C(c1nnnn1C)(c1ccccc1)NC(C)(C)COC)C(C)C C1(C(=O)NC2(CC(C)C)CC2)CC(C)(C)CCN1C(=O)C(F)n1ccnc1 C1(C(N2C(CNC(Cc3c(C)scc3)=O)CC2)=O)CC2C=CC1C2 Cc1ccc(NC(=O)CC(C)(C)CNC(=O)CC2CCC(C)O2)c(C)c1O CCC(CN=c1[nH]c2c(c(=NCCc3cc(F)cc(F)c3)[nH]1)CCC2)CC(C)C C1(NC(c2c(CC)cccc2)=O)CCN(C(C2(C)CCC2)=O)CC1CC c1(C(N2C(CC(=O)NC(COC)C)CC2)=O)cc(C)ncc1C c1(OC)cc(C)c(NC(=O)CC(C)CNC(=O)C(C)n2cccn2)cn1 C(C(=O)N1CCCC1CC(=O)N(C)Cc1cn(C)nn1)(C(C)C)OC c1(C(=O)NCC(CC=C)NC(c2c[nH]nc2C(C)C)=O)cc(C)ccc1OC N1(C(C(CC#C)C)=O)CCC2C(CCN2C(c2cc(Cl)c([N+](=O)[O-])[nH]2)=O)C1 c1(OC)cc(NC(=O)C2CC2)ncn1.C1C(OC2(c3nc[nH]n3)CC2)CC(=O)N1 CS(=O)CC(c1ccccc1)C1CC1.n12cc(nn1)C(C)(C)CN(C)C(=O)CC2 C1(C(=O)NC(C)CN(C)C)COCCN1C(c1cnc(N(C)C)nc1)=O c1(C(C(N2C(C)C(NC(=O)COC3CCCCC3)CC2)=O)O)ccc(C#N)cc1 N1(CC)C(=O)CCC1C(=O)NC(C)CC1CN(C(=O)C(C)NC(=O)OC)C1 c1(CN(S(=O)(=O)CC2COC(C)(C)C2)C)cc(F)ccc1C(F)(F)F C(=O)(C1CCN(C(=O)NCCn2cccc(C)c2=O)c2ccccc21)N.CO CC(C)CC(C(=O)NC1CCCN(O)C1=O)ONC(=O)Cc1cn[nH]c1 C=CC(C)(C)CCCNC(C1C=CCCN1C(c1cc(C2CC2)no1)=O)=O c1(C(=O)NCCCCCNC(C(C)(C)F)=O)cc(Br)cc2c1OCO2 CC(CN(C)C)CCC(=O)N(C(C)CNC(c1ccc(OCCO)cc1)=O)C C1(C(N2C(CC)C(NC(=O)C(CO)C(C)C)CCC2)=O)CCC2CC1C2(C)C C1(C(=O)NCC2OCCN(C(c3c(CC)non3)=O)C2)CC1C1CCCCC1 c1(CN(C(CCCOCC)C(=O)NCCCOC)C)nccc2ccn(C)c12 CN(C(=NCCF)NCC1CCC(C(N)=O)O1)CCC1CCCC(C)C1 C(C)(N=c1ccc2ncc[nH]c-2n1)C1CCN(C(C2(C)CC(C)=C(C)CC2)=O)C1 C1(C(=O)NCc2cc(CC)[nH]n2)COCCC1NC(c1c(C)nsc1C)=O S(=O)(=O)(c1[nH]c(=NCCSC2CCCC2)ccc1Br)N(CC(CC)CC)CC c1(OC)cc(C(=O)NCC2CC2CNC(c2cnnc(C3CC3)c2)=O)ccc1F CC(C)(C)CC(CO)NC(C1CCN(C(C2CC2Cl)=O)CCO1)=O C1(NC(C(=O)NCC)=O)CN(C(c2c(-c3ccccn3)noc2C)=O)CCC1C N1(Cc2cc(C(=O)OCC)[nH]c2)CCN(C(=O)CCCCCBr)C(C(=O)NC)C1 C(C1CN(C(=O)C(O)C2CCCC2)CC1C(=O)NCCCc1cncnc1)=CC c1(OC)ccc(CCN2CCCCC2=O)cc1NC(=O)Cc1csc(C#N)c1 Cc1ccc2[nH]cc(CC(N)C(=O)NCn3cc(Br)nn3)c2c1 c1(OCC)ccc(CNc2ncnc(NC(c3ccccc3)C)c2C)cc1OC CCCCCCCCNCC(=O)N(C)Cc1cccs1 C1(CNC(C=Cc2nc(C)sc2)=O)(CO)CC12CCN(C(=O)Cc1cn[nH]c1)CC2 C1(C(N2CC(CNC(c3[nH]c(=NC)sc3)=O)C(C)C2)=O)C(O)C(=O)N(C)C1C N1(C(c2c(CC)nccn2)=O)CCCC(CO)(CNC(=O)Cn2ncnn2)C1 C1(CC)CN(C(=O)C(CN(C)C)NC(c2ccnc(C)c2)=O)CC1F Cc1cc(C)c(C(=O)NC2C3CN(Cc4ncccc4O)CC23)c(C)c1 C1(C(N(C(CCNC(C2(CC#C)CCOC2)=O)C)C)=O)CCC(C)(O)CC1 c1(CC(=O)NCC2CC(C)N(c3nc(-c4ccccc4)ns3)C2)cc(O)nc(O)n1 C1(CNC(C2N(C)CCC2)=O)CC(C)(C)CN1C(=O)C1=COCC1 CCCC1CNC(=O)C2(CCC2)C(=O)NC2(O)CCN(C1=O)C2.N(C)(C)CC CCCC(C(=O)N1CCC2C(NC(=O)COC3CCCC3)C2C1)C1CC1 c1(C(C)C)ncncc1C(=O)N(CC(O)CN(C(=O)CCn1cnnn1)C)C N1(C(C2CCC(C(N)=O)C2)=O)CC2(CC(NC(c3cc4sccc4s3)=O)C2)C1 N1(C(CC2CC(NC(C3C4CCC(F)(F)C34)=O)C2(C)C)=O)CCc2ccsc2C1 N1(C(CC(CNC(C(CC)COC)=O)C2CCC2)=O)C2CCC1CC1(CC1)C2 c1(C(=O)OC)nsc(N2CC(OCCNC(=O)C(C3CCCO3)C3CC3)C2)n1 c1(C(=O)NC(CNC(c2ccccc2)=O)C2CCC2)cc(N2CCCC2)ccn1 C1(C(=O)N(C2CCC2)CC2(CNC(c3c(CC)ocn3)=O)CC2)CC2(C1)CC(C)C2 c12nccc(c1F)CN(CCOCC)CC(C)NC2.C(C)(C)(C)OC(=O)CC.O c1(C(N2C(CNC(C3CC(OC)C3)=O)CC(OC)C2)=O)cncc2ccsc12 c1(CNC(C23CCC(CC2)OC3)=O)cnn2c1CN(C(C1CC1F)=O)CC2 C1(NC(c2nccc(C)c2)=O)CC2CC1N(C(c1cc3c(s1)CCC3)=O)C2 c1(C(N2CCN(C(=O)COC3CC(F)C3)CC2)=O)cn(CCO)c(=O)nc1O C(C#Cc1cn(Cc2ccc(O)cc2)nn1)NC(C1C(C)(C)C1(F)F)=O C1(n2c(CC3(NC4CN(C)C(=O)CC4)CC=CC3)nnn2)CCCCCCCC1 C1(N=c2cc(-c3cccc(C(F)(F)F)c3)n(C)[nH]2)(c2n(CCOC)nnn2)CC1 c1(C(=O)NCC(C)N(C)C(c2conc2C(F)(F)F)=O)csc(C(C)(F)F)n1 C1(C(N2C(C(C)NC(C3CSC3)=O)CCC2)=O)CC(=O)OC1(C)C Cc1nsc(C)c1C(=O)NCCOCCN(C(=O)C(C)C(C)C)C N1(C(C2(OC(C)=O)CC2)=O)CCN(CCCNC(=O)CN2CC3CC3C2)CC1 c1(C(=O)Nc2ccc(C)c(C(=O)NC3CC3)c2)cc(C)c(Cl)c(C)c1 c1(CC#N)ccc(C(=O)NCC2CCN(C(C34COC(C3)C4)=O)C2)cc1 C1(N(C(c2cccc(CC)c2)=O)C)CCCN(C(C2CCC(C(N)=O)O2)=O)CC1 N1(C(c2cc(C)c(C)s2)=O)CC(C(=O)N(C)CCOC(F)F)C(C)(C)C1 Cc1c(C(N2CCC(N(C)C(c3scnc3C3CC3)=O)C(C)C2)=O)cccc1N C1(C(N2CCCC(N(C)CCO)C2)=O)COCCN(c2ccnc(C3CCC3)n2)C1 N1(C(C(CC#CC)NC(c2c[nH]c(C#N)c2)=O)=O)CCC(C)C(F)(F)C1 CCC(CC(=O)NCCC(CNC(=O)CCCNC(N)=O)OC)CC(C)C N1(C(C2C(C)(C(F)F)C2)=O)CCCC(CC(=O)NC2(C)CCSCC2)C1 CC(=O)CCCC(=O)N1CCC(C(=O)NCCc2ncccc2F)C(O)C1 Cc1coc(C2CC2)c1C(=O)NCCCOCCNC(C1CN(C(N)=O)C1)=O.OC C1(C(N2CCC(NC(=O)COc3ccc(C#N)[nH]3)C2)=O)(CC)CCC(F)(F)CC1 C1(CNC(c2c(CCC)occ2)=O)CN(C(=O)C(C)(C)n2cnnn2)CCC1C c1(CC(=O)NC2CCCC2CNC(C2CC(O)C2)=O)noc2ccc(O)cc12 C1(=O)C(C(C)C)N1.C1(OC)(CN(C(=O)CN(C2CCC2)C)C)CC1 C(CC(=O)NCC(C1CC(C)(C)C1)O)(C(F)(F)F)NC(C=CC(C)C)=O CN1CC(O)CC1C(=O)NCc1cccc(NC(C2(C3CCCO3)CC2)=O)c1 CC1CCCCC1(CNC(C1CCCCC1(F)F)=O)NC(C1CC=CCO1)=O N1(C(c2ccc(-c3ccc(F)cc3)o2)C(C(CC)(C)C)=O)CCCCC1C(F)F Cc1ccc(C(N2CCC(C(C)C(=O)NCC3(CO)CCC3)C2)=O)c(C)c1 Cc1ccc2c(c1)C(N(C)C(=O)C(N1CCC3(CC1)NC(=O)NC3=O)=O)CC2 N1(C(C(CCCOC)C)=O)C(C)CN(C(c2cn(C)nc2OC)=O)CC1C C(C1=CCN(C(=O)CCc2nncnc2O)CC1)NC(C(COC)O)=O CC1=NOC(C)(C(=O)NCCCCN(C)C(C2(c3ncccc3F)CCC2)=O)C1 N1(C(CCC(CC)C)=O)CCC(C(=O)NC2CCOC(C)C2)=C(F)C1 N1(C(C2C3CN(C(C(=C)Cc4ccccc4)=O)CC32)=O)CCN2CCCCC2C1 N1(C(CN(CC(C)C)CCO)=O)CC2(CCC(CNC(=O)C(C)C3CCC3)O2)C1 c1(C(N2CCC3CN(C(C=NOC)=O)CC3C2)=O)cc2c(F)cc(Cl)cc2[nH]1 C1(CC(=O)NCC(CN(C(C2CC(OC)C2)=O)CC)(C)C)CCCCC1(C)C C12(C(N3CC(NC(C(COCC)(C)C)=O)C(O)C3)=O)C3CC(CC13)C2(F)F N1(C(C(=O)NCCOC)C(C)(C)C)CCCC2(C)COCCC12 CC(C)C(O)C(F)(F)C(=O)NC1CC(CNC(c2ncn3cc(Cl)ccc23)=O)C1 C=C1C(NC(N2CCC(Nc3cccc(Cl)c3)C2)=O)CC2CC1C2(C)C N1(C(c2c(C)cco2)=O)CCCC2(NC(=O)Cn3ncc(Br)n3)CCCC12 c1(C(=O)NC2(C(=O)NCC(F)C(C)(C)O)C(C)(C)C2)ccc(N=[N+]=[N-])cc1 Cc1cc(CO)oc1C(=O)NC(c1ccnn1C)C(N1CCCC1C)=O c1(CC(=O)NCCC(O)CNC(c2cnn[nH]2)=O)c[nH]c2cc(Cl)ccc12 N1(C(C(CC)(C)CC)=O)CC2CN(C(=O)CCc3cn[nH]c3)CC2C1 c1(CN(C2CCCN(CC(F)F)CC2)C)cnc2[nH]ccc2c1 C1(O)CCC(C)CC1.c1ccc(COCCNC(C2CC3(CC3)C2)c2nc[nH]n2)nc1 C1(CN(C(=O)C=Cc2ccc(Cl)s2)C)CN(C(=O)CCc2ncccn2)CCO1 C1(C(N(CC(C)NC(C(c2ccccc2)C)=O)C)=O)CN2CCCC2CO1 CCN=C(NCC(C)Oc1cccc(C)c1)NCC1CN(C)CCO1 C(=O)(CC(C)(C)C1CC1)N(CCCNC(C1CCN(C)C1)=O)C1CC1 C(=O)(C1CCc2nccn21)NCCC1CC(C(=O)NCC2CCC(C)(C)C2)C1 C1(CNC(CC(C)OC)=O)CC2(CCN(C(c3cccc(N)n3)=O)CC2)C1 c1(NC(C(=O)NCCC2C(C(=O)OC)C2)=O)ccc(O)nc1 N1(C(C(CC)OC)=O)CC2CN(C(c3cc(N)c(Cl)c(O)n3)=O)CCC12 C1(C(=O)NC(C)Cc2cccs2)CC2CCC(C1)N2C(=O)CC(Cl)Cl c1(CCC(=O)NCC2N(C(CC(=O)OCC)=O)CCC2)ccccc1OC c1(C(N2CCC(NC(Cc3c(C)noc3C)=O)CC2C)=O)ccc2ccccc2c1 Cc1cc(C(N2CCC(F)(c3cc(F)cc(F)c3)CC2)C(=O)NC(F)F)ccc1Br n1(CC)cc(C(=O)NC2CC(C)N(C(=O)CN3CC(C)(C)C3)C2)c(C(C)C)n1 C(=O)(C1=CCC(C)CC1)NCc1c(C(N(CCC)CCC)=O)n[nH]c1 c1(OCCC(=O)NC2C(NC(=O)CCc3ccncn3)CC2)ccc(Cl)c(F)c1 N1(C(c2ccc(F)cn2)=O)CC2CCC(Nc3ncncc3Br)CC2C1 C1(F)(C(=O)NCC2CN(C(CC(C)(C)O)=O)C(C)(C)C2)CS(=O)(=O)CC12CCC2 C=CCCCC(=O)N1CC(CNC(=O)CC2CCCN(C)C2)(COC)C1 CC1(C)CCN(c2cc(NC3CC(C(N4CCCCCC4)=O)C3(C)C)ncn2)C1 c1(C(N2CC(CCOC)N(C(=O)CCOC(C)C)CC2)=O)c(C)ccc(C)c1C c1(N2CCC(S(=O)(=O)NC)C2)nc(=NCc2cc(C)on2)[nH]c2c1CSC2 C1(CNC(c2c(CC)nccc2)=O)CCCN(C(=O)CC2CCC(=O)N2C)CC1 c1(CC(N2CCC(NC(c3c(C)ccc(CC)c3)=O)C2)=O)ccc(C)c(F)c1F C1(NC(COC)=O)CCC2CN(C(c3nnc(O)nc3O)=O)CC2C1 c1(N(C2CC3(CNC3)C2)C(C2(C(=O)NC)CC2)=O)cc(C(=O)OC)[nH]c(=N)n1 N1(C(c2nc(CC)sc2N)=O)CCC(NC(=O)C(=O)NCCC(N)=O)CC(C)(C)C1 c1(CC)ccsc1C(=O)NC(C)CN(C)C(c1csc(C2CC2)n1)=O C1(O)(CNC(c2c(C)c(C(F)(F)F)n[nH]2)=O)CCCN(C(c2ccns2)=O)C1 C#CCCC(O)C(=O)NCCC(C)(C)CNC(c1cc(N)c(F)cn1)=O O(N1CCC(CC(=O)NC2(C)CN(C(=O)CC3CC(OC)C3(C)C)C2)CC1)CC CC1CCN(CCCc2ncns2)C1(C)C C1(C)(C(NOc2c(COC)cccn2)=O)CN(C(=O)CC(F)(F)F)C(C)(C)C1 C(CC(=O)NC1CC(=O)N(C)C1)(C(F)(F)F)NC(c1nc(CCC)oc1)=O c1(C(=O)NCC(CNC(c2cc(OCC)no2)=O)F)cccc(=O)o1 C(C(C)NC(=O)C1=CCCC1)(C(C)C)NC(c1c(C)scc1)=O c1(OC)ccccc1OC(C)C(=O)Nc1cn(-c2nccs2)nn1 C(=O)(C(F)C(F)(F)F)NCC1CC(NC(CC(C)(C)c2cccs2)=O)C1 c1(C(=O)NCCCC2(CC)CCCC2)ccc(CNc2ncc(Cl)cn2)cc1F c1(C(N2CC3C(CNC(C4C(C(=O)OC)CC4)=O)C3C2)=O)cc2cccnc2o1 C12CC(C1(C)C)CC(=O)N2.N1(C(c2cn(CC=C)nn2)=O)CC(=O)N(CC)C1 c1(C(=O)NCC2CCC(F)(CNC(C3C(C(=O)OC)C3)=O)C2)ccc2cncn2c1 CCC(CCCC(=O)NCCCc1nc(C)no1)NC(c1cnsc1)=O Cc1cc(Cl)c([N+](=O)[O-])cc1NC(C1CCCCN1S(=O)(=O)CCCl)=O C(=O)(C=C1SCC(=O)N1C)NCc1cccc(NC(C(CC)(CC)CC)=O)c1 N1(C(C2CC(=O)C(OC(F)(F)F)N2)=O)CCN(C(C)(C)CO)CC1 Cn1c(O)ncc(OC(=O)NCOC(C)(C)C)c1=O.C12(C#N)CN(C1)C(=O)C2 C1(COC)CCCN1C(=O)CC1CCN(C(=O)CCc2ccccn2)C1 C(C(O)CNCC1CC1)OCCc1cnsc1.C12(CC1)N(C)C2=O.C(=O)(N)OC N1(CC)CC(C(=O)NCC2CCC2C(=O)NC2(C(C)(F)F)CC2)CC1=O c1(C(=O)OC)cc(C)cnc1N1CC(C)(C(=O)NCc2cc(C)ccc2O)C1 c1(C(C(=O)NC2(CNC(c3c(C)con3)=O)CCC2)C)ccccc1Cl N1(C(c2ccccc2C(F)F)=O)CCCOCC12CCC2 S(=O)(=O)(c1c(Cl)cccc1Cl)NC(C)N(C)N(C)CC1CCCCC1 C1(CNC(C(CC#C)C2CC2)=O)CC2CCC(C1)N2C(=O)C(F)(F)CCCC C1(C(=O)Nc2c(OC)ccc(NC(=O)NC3CC3F)c2)CC2COCC(C1)C2 CC1CCC(NC(c2c[nH]nc2-c2cccnc2)=O)CN1C(=O)CC1(O)CCC1 C(C)(CC(F)(F)F)NC(C(CNC(C(CC)N(C)C)=O)C)=O n1(CC(=O)NCC2N(C)CCN(C(=O)C#CCF)C2)cnc2ccccc2c1=O C(=O)(C1=CCC(NC(=O)CC2CCCCC2)C1)NC(CC#C)CO N1(C(c2nccc(C)n2)=O)CCC(NC(=O)COc2c(C)occc2=O)CC1C S(=O)(=O)(c1ccc(F)c(NC(=O)NC(C2CCCO2)CN(C)C)c1)N(CC)CC N1(C(=O)C2CC2)CCc2c(C(C)=O)csc2C1 C(=O)(C(F)C(=O)N1CCC(c2ccon2)C1)OCC.C(CC(=O)N)NCC1CC1 c1(CNC(NC2CCN(C(=O)NCC)C2)=NC)cc(Br)ccc1C#N c1(CC(=O)N(CCCNCCC(O)CC=O)CC)ccc2c(c1)NC(=O)C2 c1(C(N(C2CCN(C(c3c(C#C)c[nH]n3)=O)CC2)C)=O)cc(Cl)cc(Cl)c1F CC1CCN(C(C2(NC(c3cnc(O)c(F)c3)=O)CC2)=O)CC1(C)C C(=O)(C(C)(O)CCC1CCCC1)N(CCC(=O)O)C C1(C(=O)NCC(CCOC)O)CN(C(c2oc(C)nc2C)=O)CC12CCC2 c1(-c2ccc(CN3CC(OC)C(OC)C3)cc2)ncnc(C)c1C C1(C(N2CCC(C(=O)OC)C2)=O)CCN(C(=O)C(C)CCc2ccccc2)CC1 c1(C(N2CC(=C(CNC(c3cccc(Cl)c3)=O)F)C2)=O)cc(O)ncc1F N1(C(C2OCCN(C(C)=O)C2)=O)C2CCC1CN(C(=O)C(C)N(C)C)CC2 C1(NC(C2CCSCC2)=O)CCCC(NC(C23COC(CF)(C2)C3)=O)CC1 C(C[Si](C)(C)C)(C(=O)OC)NCC1(COC)CCOC1 c1(CC)ccccc1C(=O)NC(CC(N1CCOC(O)C1)=O)C1CC1 Cc1cc(C2CCN(C(=O)OC(C)(C)C)CC2)c(C)cn1.C1(C(=O)N2CC2)CC(F)C1 C(=O)(CCCCCCSC)NC1CCC(C)N(C(=O)CCCCN(C)C)C1 S(=O)(=O)(c1cccc(=NCc2ccc([N+](=O)[O-])cc2)[nH]1)NCCC1CCN(C)C1 c1(C(N2CCCC(N(C(=O)C=Cc3cnc[nH]3)CCO)C2)=O)ccc(O)c(O)c1 C(=O)(C1=CCN(C(c2cnc(C3(C)CC3)nc2)=O)C1)NC12CCC(CO1)C2 n1(CCC(=O)Nc2nccc(CN)c2)c(=O)nc(O)c2ccccc12 S(=O)(=O)(c1ccc(NCCCS(C)(=O)=O)c(C#N)c1)N(CCCN(C(C)=O)C)C N1(C(c2c(C)scc2)=O)CCC(F)(F)C(NC(C2CCCC2C)=O)C1 C=CCCCC(=O)NCCC1CCN(C(c2c(C)noc2C)=O)CC1 O=C(C1=CCCSC1)NC1(CO)CCCN(C(=O)CCCc2nccs2)C1 c1(OCC)cncc(N2CCN(C(C3(OCC)CC(F)C3)=O)CC2)c1 C(=O)(C(CC)C(C)O)NC1(CNC(c2cn(CCCC)nn2)=O)CCOC1 c1(SC)nccc(N(C(=O)CC2CCCN2CC(=O)NC(C)(C)C)C)n1 c1(CCC(=O)N(C(CCNC(C(c2cnn(C)c2)C)=O)C)C)ncccn1 c1(C(=O)NC(CC)(CNC(C2CCCCC2O)=O)CC)cc(C)cc2c1CCC2 C1(NC(c2cc[nH]n2)=O)C2CCC1CN(C(=O)CCCCc1ccccc1)C2 N1(C(c2cnc(C)[nH]c2=N)=O)CC2CCC1C(CNC(=O)CC1(C)CC1)C2 CC1C(C)N(C(c2cnc(-c3ccccc3)[nH]2)=O)CCN1C1CC1 c1(CC)oc(C(=O)NC(C)CC(C)NC(c2cccnc2)=O)cc1C Cc1cc(Cl)ccc1NNC(=O)c1ccnc(-c2cccnc2)n1 C(=O)(C(C)(C)CC1CCN(C(=O)OCC2OCCO2)CC1)OCC CON(C(=O)C1=C(F)CN(C(c2cc(C)cc(C)c2)=O)CC1)C1CCCC1 C(=O)(CCC(C)CCCC)N1CCCC(CC(N2CCC(CC=C)CC2)=O)C1 c1(C(N(CC(=O)OC)C)=O)ncccc1F.C12CCC(CC1)C(=O)NC2 C1(CNC(C=CC=CCC)=O)CCCCCN1C(c1scnc1CC)=O S(=O)(=O)(CCC(=O)N1CCN(C(C2CCC(CC(C)C)CC2)=O)CC1)NC C1(C(N2CCC(C)(C(N3CCN(CC=C)CC3)=O)C2)=O)CC(=O)NC1(C)C c1(C(N2CC(c3ccccc3)(NC(C(C=C)O)=O)C2)=O)cc(N)c(F)cc1F c1(C(N2CC=CC(OCC)C2)C(=O)NCC(=C)C)nn(C)c(CC)c1Cl Cc1ccc(CCNC(=O)C(C2CCN(C(=O)C=Cc3cc[nH]c3)C2)F)cn1 c1(C(N(C2CCC(NC(C(C(=C)Cl)(C)C)=O)C2)C)=O)cccc2[nH]ccc12 C1(C(=O)NCC(C)O)CN(C(c2ncoc2C2CC2)=O)CC12CC2 N1(C(C(CC(C)C)O)=O)CC2CC(NC(c3cnn(-c4nccs4)c3)=O)CC1C2 c1(OC)ccc2c(c1)OCCC2C(=O)NCCNC(c1cccc2c1NCC2)=O Cc1cc(=O)c(C(=O)NC2CC(NC(C3CCCCC3O)=O)C2)cn1C1CC1 N1(C(C(C2CN(C(c3cc(O)n(C)n3)=O)C2)OC)=O)CCOCC2(CC2)C1 C#CCC(CC(=O)NC12CC1COC2(C)C)NC(=O)CCN1CCCCC1 C1(CC(=O)NCC(C2CC2)OC)CCN(C(=O)CSC)C1 C1(C(N(C2CC(NC(c3c[nH]nc3C3CCC3)=O)C2)C)=O)CCC1(F)F C1(C(=O)NCC2CC2NC(=O)C(C(C)C)NC(C)=O)(OC)CCCCC1 C=CC1(C(=O)N(CCCF)C)CCN(C(=O)CC2=CCCC2)C1 c1(C(N(C2CCC(NC(c3ccc[nH]3)=O)C2)C)=O)cncc2[nH]ccc12 C(=O)(CCCCNC(c1c[nH]nc1C(C)(F)F)=O)N(C)CCSCC#N C1(CC(=O)N(CCCNC(=O)C(C)NC(c2ccoc2)=O)CC)CC2CCC1O2 O=C(C1=NOC2CCC3(CCN(C(c4cocn4)=O)CC3)C12)NCCCBr C#Cc1ccc(OC)c(C(=O)N(C(C)CNC(=O)CCS(N)(=O)=O)C)c1 c1(CC)ncc(C(N2CCCC2CNC(c2ccnc(Cl)c2N)=O)=O)c(O)n1 N1(C(CSCc2cccc(C)c2)=O)CCC(NC(C2CC3(CC3)C2)=O)C(O)C1 C#CC1CN(C(c2cnncc2OCCC)=O)CCN1C(=O)COCC C(CC(=O)NCCN(C(=O)CCC1CC1COCCSC)C1CC1)(C(F)F)NC(N)=O c1(OC)ccc(C(O)CNC(c2cccc(Cl)c2F)C)cc1F c1(CNC(C2CC(O)CCN2C(C2CS(=O)C2)=O)=O)cccn2nccc12 N1(C(c2ccc(C)nc2)=O)CCCC(O)(CN(C(=O)C=CC2CCC2)C)C1 c1(C(N(C(C)CNC(C2CC3(CC3)C2)=O)CC)=O)ccc2c(c1)CCCO2 CN1CCC(C(N2CC(O)(C3CCCN3C(c3ccc(Cl)o3)=O)C2)=O)CC1 Cn1ccc2cccc(C(=O)NCC(CO)NC(c3cnc(O)n3C)=O)c12 CC1=C(C(=O)NC2(C(=O)NC3CC3C3CC3C)CCN(C)C2)CC1 c1(C(=O)NCC(C)(CNC(=O)C2=CCSC2)OC)ccc(Cl)c(Cl)c1 c1(C(N(C)CC2(O)CCN(C(C3C(C)C3)=O)C2)=O)cc2cc(F)ccc2[nH]1 C#CCCCCCCC(=O)N1CCC(C)(C)C1C(=O)Nc1ccc2c(c1)OCO2 C1(N(C(C(C)O)=O)CCO)CCCN(C(c2cc(-c3ccccn3)ns2)=O)C1 C1(C(=O)NC2CC3CCC(C2)O3)(CC)CCN(C(=O)Cn2nccc2C)CC1 c1(CC)c(NC(c2cnoc2C)=O)cnn1C1CCCC1.C1CO1.C(C)(=O)N c1(NC(C2C(CC)N(C(c3snc(C)c3N)=O)CCC2)=O)cc(C)c(O)cc1C c1(CC)c[nH]cc1C(N1CC(C)(CN(C(=O)C(C)C)C)C1)=O.C(=O)(CNC)NC N1(C(c2c(OC)cc(N)cc2)=O)CCC2(CCCN2C(C2CCCC(F)C2)=O)C1 CCCCCCCCS(=O)(=O)N1CCC2(CC1)CN(C(=O)CC(F)(F)F)C2 CC1=C(C)CC(C(N2CCN(C(c3nc(Br)c(C)s3)=O)CC2CF)=O)CC1 C1(N(C(c2c[nH]nc2C2CC2)C(=O)NCCCSCC)C)CCCC(C)C1 C(=O)(CCC(=O)NC1(CNC(=O)CN2CCCC2=O)CCOC1)c1ccc(C)s1 N1(C(CC(C)C2CC2)=O)CC2CCC(CNC(c3ccn4cncc4c3)=O)(C2)C1 c1(CC(N2C(CNC(C34CC(F)C3C4)=O)CC2)=O)ccc(Cl)c([N+](=O)[O-])c1 C1(C(=O)NCC(C)(C2CCC2)NC(COCCC)=O)C2CCCC12 C(=O)(CCC(C)NC)N1CC(C(CC)C)(NC(=O)COC)C1.c1(O)ccccc1NC C1(F)(C(=O)NC2C(OC)CN(C(=O)CCOCC(F)(F)F)C2)CCCCCC1 N#Cc1cc(Br)ccc1C(=O)NCCCCCOCCOCCOCC.C(CCN)O c1(CNC(C2C(NC(C(CC)SC)=O)C2)=O)ccc([N+](=O)[O-])cc1[N+](=O)[O-] c1(CC)ccnc(C(=O)NCCC2CC(NC(=O)C=CC3CCCO3)C2)c1 C1(C(=O)NC2(C)CC2)CCC(CNC(=O)C=CCF)CC1 Cc1ncc(S(N)(=O)=O)cc1C(=O)NC(C)CNC(c1ccc(F)c(CO)c1)=O CC1=C(C(=O)N(CC(O)CN(C)C(c2cnccc2Cl)=O)C)CCC1 c1(CNC(CC(=O)OC)Cc2ccc(Br)cc2)c(F)cc(O)cc1F c1(NC(C)=O)cnccc1C(N1CC(NC(C2(C)COC2)=O)C(C)C1)=O c1(OC)ccsc1C(=O)N(CC(C)C(=O)NCC(c1ccco1)O)C c1(CN2C(C(=O)Nc3c(Cl)ccc(C(=O)OCC)c3)CC2)c(F)cc(F)cc1F CN1CCC(C(=O)NCC2CCC(NC(C3CC(C)(C)CCO3)=O)C2)CC1=O c1(C(=O)NC(c2cccc(C(=O)OC)c2)C)cnc2[nH]nnc2c1 Cc1nn(C)c(C)c1C(c1nnnn1C(C)(C)C)NCCSC(C)C c1(C(N2CCC2C(F)F)=O)cncc(-n2cc(C3CCCO3)nn2)c1 C1(C(=O)NC(C2CCN(C(C3C4CCCC34)=O)C2)C)(C(F)F)CCOCC1 C(=O)(C(CN(C)C)N(C)C)NCCCN(C(C)C)C(c1ccon1)=O c1(N(C(CCOC(C)=O)=O)C)ccc(CNC(=O)CCSc2nnnn2C)cc1 N1(Cc2cc(OC)c(Cl)cc2)CC2C(C1C(=O)NC(C)CC(F)(F)F)C2(C)C C1(NC(c2c(OC)n(C)nc2)=O)CCN(C(C2(CC(C)C)CC2)=O)CC1O C1(NC(c2cnc(C(C)C)n2C)=O)CCC12CN(C(c1ncn(C)n1)=O)C2 c1(CC(=O)NC(CCCCNC(C2CC(CC)C2)=O)C)c(F)cccc1Br N1(C(C(C)SCCCC)=O)CCCC(N(C(=O)CCC(=O)NCCOC)C)C1 C(CC(C(=O)NC1CCCCC1NC(c1cc(C)co1)=O)NC(N)=O)SC N1(C(CCC(C)(C)C)=O)CCC2(CC1)CN(C(=O)C(C)(C)CC#N)CCO2 c1(CC(N2C(C(CNC(CS(CC)=O)=O)(C)C)CCC2)=O)c(C)nn(CC)c1C C1(CC)CCN(N2CCC2(CCC)C(N)=O)CC1 c1(C(=O)NCC(C)CN(C(=O)C(C)COc2ccccc2)C)cocc1C(N)=O S(=O)(=O)(c1ccc(N2CCN(CC3COCCO3)CC2)cc1Br)NC(CC)C c1(C(=O)NCCCc2cn(-c3ccc(CO)cc3)nn2)cc(F)cc2nc[nH]c12 C12(C(=O)NCC(CSC)OC)CCCC1CCN2C(c1ccc(O)nc1C)=O N1(C(c2n(CC)ccc2)=O)CCN(C(C2CCCC(C)(C)O2)=O)CC1C1CCC1 c1(C(=O)OCc2ccc(Br)cc2C(F)(F)F)cc(Br)c2cccnn12 C(=O)(C(CC1CCOCC1)NC(=O)C(C)Cn1ccnc1)NC(c1ccn(C)c1)C c1(C(N2CC(OCCC(C)C)C2)=O)ncoc1C(=O)NCC1CC1c1ccsc1 CC(C#N)C(=O)NCC(C)NC(c1nccn1C)=O c1(C(C)NC(C2CN(C(c3sccc3Br)=O)CCO2)=O)cc(Br)cc(Br)c1 C1(NC(C=C(C)C)=O)CCCC12CCN(C(c1cc(F)c(C)cc1Cl)=O)CC2 Cc1cc(C(=O)NCC(C)(C)C(N2CC(O)C(C)(C)C2)=O)ncc1F n1(CC(=O)NC(C2CN(C(=O)CSCc3cccs3)C2)C)cnnn1 C1(C(=O)NCc2cn(CC(C)NC(c3[nH]cc(CC)c3)=O)nn2)CC2(CC2)CN1C C1(NC(c2c(N=[N+]=[N-])ccs2)=O)CN(C(C2CCCO2)=O)CCC12CCC2 c1(C(N2CCC(NC(c3c(CCC)nco3)=O)CC2)=O)c(C)ncnc1O C=CCCCCCC(=O)N1CC(C2CN(C(=O)C(=O)NC3CC3)C2)C1 c1(CCCOCC)nc(-c2scnc2C)nn1-c1ccc(C(C)(C)C)cc1 CC1=NC(C)(CNC(=O)C(CCC2CC2)NC(=O)Cc2ccc(O)cc2)CS1 C(CC)(CC(C)CO)NC(CC1C=CC(NC(c2c(OC)cnnc2)=O)C1)=O C1(NC(c2c(C(C)C)cco2)=O)CC2CCC(C1C)N2C(C1(C(F)F)CCC1)=O CCCC(C)(O)CC(=O)N1CCN(CCCCCNC(=O)C(C)S(N)(=O)=O)CC1 C1(NC(c2c(C)nn(C)c2)=O)CN(C(C2(CS(C)(=O)=O)COC2)=O)CCC1C C(C#Cc1cn(-c2cc(C)cc(C)c2)nn1)NC(C1CCCC(OC)C1)=O C(C)(C)(C(=O)N1CC(O)(CCC(N2CC(C)(C(N)=O)C2)=O)C1)OC(C)=O Cc1c(C(N2CC(NC(c3conc3C(C)C)=O)C3CC23)=O)ccn1C C1(CC)(NC(C(=O)NC(c2ccc(Br)s2)C)=O)CCCN(C(C2CCCCO2)=O)C1 Cc1ccc(CC(N2CCCC2c2cn(-c3cccnc3)nn2)=O)c(C)c1 c1(CN(C2CCN(C(CC)=O)CC2)C)c(Cl)cc(C)nc1Cl N1(C(CC2(CNC(c3c(C)cnnc3O)=O)CC2)=O)CCC(N=[N+]=[N-])CC1 N1(C(C(CC(C)C)OC)=O)CC(C(=O)NCCc2ccns2)C(C2CC2)C1 N1(C(C(=O)NCCC2CCCCO2)=O)CC2CC1CC2Sc1ccc(Cl)cc1 C#CCCCCC(=O)NCC1CCC1NC(c1nn[nH]c1C(F)(F)F)=O C(CC1CCC1)(C(=O)NC(C)C(=O)NCc1cc(C(N)=O)co1)OC n1(CCC)nc(C)cc1C(=O)NC1CC1CNC(C12CC(C)C1C2)=O N1(C(CC2C(C)CCO2)=O)CCC(O)(CNC(C2CCSCC2)=O)CC1 c1(C(CNC(C2(OC)CC2)=O)NC(CN(CCOC)C)=O)ccccc1Cl n1(CC2CC2)cc(C(=O)N(C2CN(NC(C3C(COC)C3)=O)C2)C)cn1 c1(CN2CCN(C)C(CNC(c3cccc(F)c3Br)=O)C2)ccc2cc[nH]c2n1 C(=O)(CC1=CCOCC1)C1CN(C(=O)CCCC)CCC1C(F)(F)F.O=CO c1(NCc2cc(C)nn2C)[nH]c(=NC(C)C(C)F)nc2c1ncn2C(C)C c1(C(=O)NCC2C(NC(c3cn(CCOC)nc3)=O)C2)cncc2[nH]ccc12 N1(C(C(C(C)C)C)=O)CCCC2(NC(=O)C(C)c3ccsc3)CC2C1 C(=O)(CCC(CC)NC(=O)CCC1CC(C)C1)NC(CC#CC)CO c1(CC)ccc(OC)c(C(=O)NCC2(CNC(=O)COC(F)F)CCC2)c1 CC1OC(C)CC1C(=O)NC(C)CC1CCN(C(c2[nH]ncc2C#N)=O)CC1 C#CCC(C)(CC)C(=O)NCC1CC1CNC(=O)CSc1cccnc1 Cc1cc(C(O)CNC(CCC2=CCOCC2)=O)ccc1F C(c1ccccc1)=CCCC(=O)NC1CC(C)(NC(c2coc(C(=O)O)c2)=O)C1 C1(CCC(=O)NCCC(=O)N(CC)CC)CCCCN(C(=O)CC(C)(C)CC)C1 c1(C(N2CC(CN(C(C(C)CO)=O)C)OCC2)=O)cc2n(n1)CCN(C)C2 c1(C(=O)OCC)ccc(C(N2CCC(C(=O)Oc3ccc(OCC)cc3)C2)=O)cc1 Cc1c(Br)cnn1CC(N1CCCC1(C)CNC(=O)CC1CC2CC2C1)=O c1(C(=O)NC2CC(F)(CNC(C3CC(N(C)C)C3)=O)C2)cnn2ccn(C)c12 N1(C(C(=O)N(C)CCN(c2ccc(F)cc2Br)C)=O)CCc2nc(Cl)ccc2C1 C1(CNC(C2CC2C2CC2)=O)CN(C(c2ncc(Cl)cc2F)=O)CC12CCC2 c1(OC(C)C(=O)NC(C2CCCN2C(=O)CSC2CCCCO2)C)ccccc1 N1(C(C2N(C(=O)C(C3CCOCC3)=O)CC2)=O)CCCC2(CC1)CC2 c1(C(=O)NCC2(NC(C(CC)OC3CCCC3)=O)CC2)cc(Br)c(C)cc1F N1(C(c2c(OCC)cccn2)=O)CCN(C(=O)OC(C)(C)C)CC1CC(C)(C)C c1(C(N2CCCN(C(C(C=C)O)=O)CCC2)=O)n[nH]c2cc(C)ccc12 C1(NC(c2c(C)cns2)=O)CC2CC(NC(=O)CC(=O)NC3CC3)C2C1 c1(OCCC)ccc(C=CC(N2CC(CNC(c3cc[nH]c3)=O)C(C)C2)=O)cc1 c1(OCCCOC2CCN(C(=O)C(=O)NCC(F)F)CC2)ccc(N=[N+]=[N-])cc1 c1(C(=O)NC2CCCN(C(=O)CC3CCCO3)CC2)cc(Cl)cc2c1OCC2 C12(CNC(c3c(C)cc(O)nc3)=O)CCCC(CN1C(=O)C(C)SC(C)C)C2 Cc1ccc(CCC(=O)NCC2CN(c3ncccn3)C2)cc1Cl N1(CC)CC(C(=O)NC2C3CC2N(C(c2ocnc2C)=O)C3)CC1=O C=CC(C)(O)C(=O)NCC(C)(F)CNC(=O)Cc1cc(C)cs1 C1(C(=O)NCCCCNC(C(CCOC)C)=O)CSC(c2ccccc2O)=N1 C(CC(C)(C)C(=O)N(C1CCCOC1)C)NC(c1cc(C)on1)=O C(=O)(C#CC1CCCCO1)NCC(CC)NC(c1cocc1C)=O c1(CNC(C(C2CN(C(CN(C(C)=O)C)=O)C2)O)=O)nn(C)c(=O)n1C C(=O)(C1=CCC2CCC1N2C(=O)C(O)C(C)(C)CC)NCC(CCC)O c1(C(=O)NCC(COC)O)ccc2[nH]c3c(c2c1)CN(C(C1CCCC1)=O)CC3 c1(CN(C(C(C)SC(F)(F)F)=O)C)cccc(CNC(C2(C)CCNC2=O)=O)c1 c1(OC)cc(F)c(C(=O)NCC2CCN(Cc3cccc(Cl)n3)C2)c(F)c1 C=CC1CN(C(=O)CCC(C)(C)NC(=O)C(CCC)OC)CC1COC C(CCCCCNC(c1nocc1Br)=O)OCCC(=O)NCC1CC1 c1(CC(=O)N(CC(CO)(CO)NC(CSCC#C)=O)C)cc(F)c(F)cc1F C(CCS(=O)(=O)C(C)C)N1C2CC(NC(CC=C)=O)CC1CC2 C1(NC(CCc2c(C(=O)OC)c(C)[nH]c2)=O)CCCC1P(C)(C)=O C(=O)(C(C)CC(C)C(C)=O)NC(CC(N1CCC(C#CC)CC1)=O)CC c1(C(N2CC3C(C(N4CCC(F)(F)C(O)C4)=O)C3C2)=O)cc(I)c(O)c(I)c1 c1(C(N(C2CCN(C(CC(=C)Br)=O)C2)CC2CC2)=O)cccc(OC)c1C C(=O)(C(C)(C)CCCO)NCC1C2CN(C(C3C(C(=O)OC)CCO3)=O)C1C2 c1(C(N(CCCCN(C(C(C)OCCOC)=O)C)C)=O)cccc(Cl)c1[N+](=O)[O-] C1CSc2ccccc2O1.CN1CN(C(=O)OC(C)(C)C)CC1COC(=O)C1CC1 c1(C(c2n(C3CC(C(=O)OC)C3)nnn2)NC2CC(CF)C2)cccc(Br)c1 Cc1c(C(N2CCN(C(=O)CC3COCCO3)C(C)C2)=O)cccc1S(N)(=O)=O c1(C(=O)NCCNC(=O)CC2CC2C(F)(F)F)cnsn1 C(=O)(C1=CC2CCCCCC12)NCCCNC(c1c(CC)non1)=O N1(C(c2c(C)cccc2N)=O)C2CCC1CN(C(=O)C(C)C(C)n1cccn1)C2 c1(OC)cc(NC(N2C3CN(C(c4cccc(F)c4C)=O)CC23)=O)cc(O)c1O N1(C(c2nc(O)[nH]c(=O)n2)=O)CCC2(CCCN2C(c2ccc(F)c(Cl)n2)=O)C1 c1(OCCOC)ccc(NC(=O)CCC)cc1.c12ccc(cc1)CNC2 C(CC(=O)NC1CC=CCC1C)(CC(C)C)NC(c1nc(C(C)C)oc1)=O CON(CCC(=O)N1CCCC(C(N)=O)C1)C(=O)c1cccc(C)c1O c1(C(=O)OC)ncnc(N2CCCC2)c1Nc1cccc(C(=O)NC2CC2)c1 C1(NC(=O)Cc2ccsn2)CCCC(NC(=O)Cn2ccc(Br)n2)C1 Cc1cc(NC(C23CCC2CCN3C(=O)C2=CCCCCC2)=O)c(C)c(C)c1 c1(C(=O)NCCC2CCN(C(=O)C=CC3CC3)C2)c(O)nnc2c1CCCC2 CC(C)CCCCCC(=O)NC1CN(C(=O)Cn2cnc(C#N)n2)C2CCCC12 c1(OC)nc(Cl)c(-c2nc(Cc3ccc(OC4CCOC4)nc3)no2)s1 C(=O)(C(C)CC(C)C)NCc1c(C(=O)NCc2c(C(=O)OC)nccn2)occ1 c1(C(C)NC2CN(C(C3CC3C(F)(F)F)=O)CC2C)ccc2c(O)nccc2c1 CC(CNC(=O)CCC(=O)C1CC1)C(F)C(=O)N1CCC(C)(CCO)CC1 CC1(C)CC(NC(c2cscc2C(N)=O)=O)CO1 C12CCN(C(=O)C3(OC)CCN(C3)C1=O)O2.C1(NC(C)=O)(CO)CCC1 N1(CC)C2CCC1CC(NC1CCCN(C(SC(F)(F)F)=O)C1)C2 C1(C(=O)OC)C2CC(NC(C3(c4ccc(CN)cc4)CC3)=O)(C2)N1C(C)=O C1(NC(Cn2c(C)cc(C(F)F)n2)=O)CC2CC1CN(C(C1C(C)C1C)=O)C2 C1(NC(C=C(CCC)C)=O)CCC(O)CN(C(C2CCCC2(F)F)=O)C1 CCC(CC)(C(=O)NCc1ccc(C(=O)NCC2CCC(C)(C)O2)cn1)C(C)C C12(CNC(C(C)CF)=O)CCCC1N(C(c1cccc(S(C)=O)c1)=O)CCC2 c1(C(=O)NCC(CNC(C(CC=CC)C)=O)F)ccc(S(=O)(=O)NC)o1 c1(CN2C(C)(C(=O)Nc3nccs3)CCC2)cccn2ccnc12 C1(CC)(NC(=O)COCC(F)(F)F)CCCN(C(C2CCOC2C2CC2)=O)C1 C(=O)(C1Cc2ccc(Cl)cc21)N1CCC(CCNC(C(C)(C)C2CC2)=O)C1 C1(NC(C(C(F)(F)F)OC(C)=O)=O)CC2CC(C1)N(C(c1cc(Cl)no1)=O)C2 c1(C(=O)NCC(CNC(C2(C)C(C)(C)C2(C)C)=O)CO)cccc2c[nH]nc12 Cc1nc(=NC(C)CC(C)NC(=O)CCCCN2CCCC2)s[nH]1 c1(CCC(=O)NCC2N(C(C3C(C)C3)=O)CCOC2)ccc(C#N)cc1 CCCC(C(=O)NCC1COCCN1C(c1cccc(C(=O)OCC)n1)=O)OC N1(C(CN(S(CCCC)(=O)=O)CC)=O)CCC(S(=O)(=O)c2ccc(C)cc2)CC1 c1(-c2scc(C(=O)NCC(C3CC3)NC(C(C)CC3CC3)=O)n2)ccc(F)cc1 N1(C(C(C(CC)C)OC)=O)CC2CC(C)N(C(c3csc(C)n3)=O)C2C1 C1(=CC(=O)N(C(CNC(c2ccccc2)=O)Cc2ccccc2)C)CCN(C)C1 C(=O)(C1CCCc2n[nH]cc21)NC(C1CN(C(c2nc(=O)n(C)[nH]2)=O)CCO1)C c1(C(N(C)CC2CCCN(C(=O)CCCCN=[N+]=[N-])C2)=O)ccc2cc[nH]c2n1 C1(CC)(CC)CCN(C(C2CC(OC)CN2C(=O)Cn2cccn2)=O)C1 C1(NC(c2c(CC)nn(C)c2)=O)CCC2CCN(C(c3coc(C)c3)=O)C1C2 Cc1ccc2oc(C(=O)NC(CNC(c3ccc(Br)cc3)=O)CO)cc2c1 N1(C(CC(n2ccc(C)n2)C)=O)CC2C(CNC(=O)CN(C)C(N)=O)C2C1 c1(C(=O)OC)cc(I)cnc1NC(C1(C)CCN1C(c1cccc(C#N)c1)=O)=O CC(C)C(C(=O)NCC(Cl)=CCl)C(C)NC(c1c[nH]c(C(N)=O)c1)=O Cc1ccc2c(c1)C(C(=O)N1CCN(C(=O)CCc3ccncc3)C(CO)C1)C2 C(=O)(C(C)(C1CCC1)NC(=O)CCc1cnc[nH]1)N(C(CC)C)C c1(CNC(=O)NCc2nc(C)[nH]n2)c(C)nn(C)c1C(N)=O C1(CC(C)C)(C(N2CCC(N(C(=O)C(C)NC(N)=O)C)C2)=O)CCOCC1 N1(C(C2(OC(C)=O)CC2)=O)CCC(C)(CCNC(c2ccnc(Cl)c2)=O)C1 C1(NC(c2ccco2)=O)CC12CCC(NC(c1ccnn1C1CCC1)=O)CC2 N1(C(c2ncn(C(C)C)n2)=O)CC(CNC(C2CC2(F)F)=O)CC1(C)C CCCCC(CCCC)NC(=O)C(C)C(C)NC(=O)Cc1ncoc1C c1(CCNC(N(C)Cc2onc(C)n2)=O)ccn2ccnc2c1 C1(CNC(c2cc(C)oc2)=O)CN(C(=O)CCC(C)(C)C)CC12CCC2 C(=O)(C(O)C1=CCCCC1)NCC1(NC(=O)CN2C(=O)CCCC2=O)CCOC1 CC1CN(C(=O)C=CC2CCCO2)CC(C)CN1C(c1cccc([N+](=O)[O-])c1)=O CC1CCC(NC(C2(C)CN(C(C3(n4cccn4)CC3)=O)C2)=O)C1 Cc1ncnc(C)c1CC(N1C2CCC1C(CNC(=O)C=CCN(C)CC)C2)=O C1(CNC(CC2ON=C(C)C2)=O)CN(C(N)=O)CC1O.C1(=O)CCCN1 c1(C(=O)NCCC(C)NC(C2OC3CCC2CC3)=O)cc(C#N)ccc1F N1(C(C(C)(C)F)=O)CCC2(CC1)CN(C(=O)C=CSc1nc[nH]n1)C2 N1(C(C(CC=C)N(C)C)=O)CCC(O)(CNC(=O)CC2CC=CCC2)CC1 C1(C(=O)NC2(C(=O)NCc3cnc(C)s3)CCCC2)CC(=O)CC12CCC2 Cc1cccc(Cl)c1OCC(N1CC(NC(C2CCCO2)=O)C(O)C1)=O CCCC(C(=O)NCC1C(O)C(O)CN1C(=O)CCc1cn[nH]c1)S(N)(=O)=O CC1CCC(CNC(C23CC(C(F)(F)F)(CO2)C3)=O)CN1C(c1ccn(C)n1)=O C1(NC(C2(C)CC2(F)Cl)=O)CCCCN(C(=O)CC2CC3(CC3)C2)C1 CC1(CNC(=O)CCC2CCCN(C(=O)CCCC#N)C2)CC2(CCC2)C1 N1(C(CCc2c(OC)ccc(F)c2)=O)CC2CC(C1)N(C(c1nocc1Cl)=O)C2 C(c1ccc(O)cc1)=CC(=O)NCC1CC2(C1)CN(C(=O)CC1CC1(Cl)Cl)C2 Cc1cc(C(N2CC3(C2)CN(C(=O)CC2CCCCC2O)C3)=O)ncc1Cl C12(C(N(CC)CC3CCCN3C(=O)CNC=O)=O)CC1COC2(C)C C(=O)(C(C)C(O)C(C)CC)NCC1(c2ccccc2)CC(=C)C1 CP(C)(=O)C1(C(=O)Nc2cccc(CNC(c3ccc(F)cc3)=O)c2)CC1 c1(C(N(CCC)CCNC(=O)C(C)(CC)CO)=O)cc([N+](=O)[O-])nn1C C1(NC(c2cc(OC)ncc2)=O)(CO)CCCN(C(C2(C#N)CC(C)C2)=O)C1 c1(OCC)ccc(C)nc1C(=O)NCC(O)CN(C)C(c1cc2n(c1)CCC2)=O c1(C(F)(F)F)ccc(Cl)c(Br)c1.N12CCC(CC1)n1nc(-c3ccco3)nc12 C(N=c1ncc(F)c[nH]1)C1(C)CCC(NC(C2CCCS(=O)(=O)C2)=O)C1 C1(C(=O)NCC(CNC(c2c(OCC)cccc2)=O)OC)CC(F)(F)C1(C)C c1(C(N(C(C)CNC(c2cnn(C(C)C)n2)=O)CC)=O)sccc1OC N1(C(C2N(C(=O)OC)CCC2)=O)CC2CCC(C1)C2NC(c1n[nH]cc1I)=O C1(NC(=O)CC2C3CCC(C3)N2C(C2CCCSC2)=O)CC2(C1)CC(O)C2 C(C)(C)(CC(=O)N1CCC(C(C)CO)CC1)OC1CCN(C(COC)=O)C1 Cc1nn(C)c2sc(C(=O)NC3CCC3NC(=O)C(F)(F)C(C)O)cc12 C(CC1=CCN(C(=O)CCC#N)CC1)NC(C1N(C)CC(O)C1)=O C1(C(=O)NCCCSCC)CN(C(C2(O)CCOC2(C)C)=O)CC12CC2 C(=O)(C#CC(C)(C)C)NC12CC(CNC(c3c(C)onc3CO)=O)(C1)C2 N1(C(C(COC)(F)F)=O)CCCC2(CCN(C(=O)CCc3scnc3C)C2)C1 c1(C(=O)Nc2cccc(CNC(C(CCOC)(C)C)=O)c2)ccc2n[nH]cc2c1F CC1CCC(NC(c2cc(C3(C)CC3)n[nH]2)=O)CN1C(c1cc(F)cnc1O)=O C(=O)(C(C)(F)C(=O)NCC(C)(C)NC(c1sc(CC)nc1C)=O)OCC c1(C(=O)NCC2(NC(C3CN4CCN3CC4)=O)CC2)ccc(C(F)(F)F)cc1N C(CN=c1nc(N2CCCC(C(C)C)(CO)C2)c2cccc(F)c2[nH]1)=CCOC S1(=O)(=O)c2cc(nc(Cl)c2)-c2nnc(SC(C)C)n2CC1CC N1(C(C2(COC)COC2)=O)CCCCC(NC(=O)C(=O)C(F)(F)F)C1 C(C(CC(=O)Nc1cc(C)c(Cl)c(N)c1)CC(C)C)NC(=O)OC(C)(C)C C1(C2CCN(C(C(=O)NC(CC#C)(C)C(=O)O)=O)C2)(c2ccc(Cl)cc2)CC1 CC1(C)CCCN(C(=O)Cc2ccon2)C1C(=O)NCc1ccc(O)cc1F C1(CC=C)(NC(C2(COC)CC2)=O)CC2CCC(C1)N2C(C1CCNC(=O)C1)=O CCC(CC)(CO)C(=O)N1CCC(CCC2CCCN(C(=O)CCOC)C2)CC1 C1(CNC(c2c(COC)noc2)=O)CC2(CC2)CN1C(c1cnc(COC)s1)=O C1(C)(C(=O)NCCOCCN(C)C)CC(O)CN1C(C12CCC(C1)C2(C)C)=O C1(OC(CC)C)CCN(C(=O)NCCCCN2CCCC(O)C2)CC1 C(CN=C(NCC(=O)NCCc1ccc(Br)cc1)N1CCCC(C)(C#N)C1)OC N1(C(C2(O)CC(C)(C)C2)=O)CC2CCN(C(c3sccc3CO)=O)CC2C1 c1(C(C(=O)NC(C)CC)N(CCCC)C2CC2)nn(C)c2c1COCC2 C1(n2cc(N(C(C(C)N3CCC3)=O)C)nn2)COc2ccccc2C1 CC1CCn2c(C(=O)NCCCNC(=O)CCC3NC(=O)NC3=O)cnc2C1 c1(C(N2CC(NC(C=CC(CC)C)=O)C(n3ccnn3)C2)=O)c(C)[nH]c(C)c1C c1(CC)cc(C(=O)NCCCCC(C)NC(=O)CCCCCNC(C)=O)ccc1C N1(C(C(CCCNC(c2c(CC)[nH]cc2)=O)O)=O)CC2(CCC2)C12CCC2 C1(NC(c2cnc(COC)s2)=O)CCC(F)(CNC(=O)CC2CCCN2C)C1 C(=O)(C(CCF)NC(c1ccc(C(N)=O)o1)=O)NCC(C)OC(F)F C(=O)(C1COc2ccccc21)N(C1CN(C(c2cn3cc(C)sc3n2)=O)C1)C C1(C(N2CC(CC)(NC(=O)CN3CCCC3=O)C2)=O)COCCC1(F)F C(C(=O)NC(CNC(C1(C(F)F)CCC1)=O)C(C)C)(C(C)C)NC(CC(C)C)=O N1(C(C(SC)SC)=O)CC2CC1CN(C(c1cc(F)ccc1F)=O)C2 CCC(CC)C(=O)NCC(=O)NC1CC(CNC(=O)CCOC2COC2)CO1 N1(C(C(CC)C)=O)CCC(C2(O)CCN(C(=O)CCCCC(=O)OC)C2)CC1 O=C(CC(C(F)F)c1ccccc1F)NC1CC(NC(=O)CN2CC3CC3C2)C1 Cc1cc(N2CCC(NC(C3CCCO3)=O)C2)ncn1 C(CC(O)CC(=O)N1CCCC1C(C)NC(c1ccsn1)=O)SC Cc1nc(CN2CCC(NC(C3OCCC3C(=O)O)=O)C2)cs1 N12CC3(CC3)CC1C2=O.c1cnc(Cl)cc1C(=O)NC1N(C)C(=O)CC1.C(N)=O c1(C(C(C)NCc2cc(-c3c(F)cccc3F)on2)O)c(F)cccc1F c1(CN(C(C2(NC(CC3CC(=C)C3)=O)CC2)=O)CC)c(C)cccc1C C12(C(=O)NC3CCN(C(=O)CCc4ccc(Br)s4)CC3)CCCC1C2(F)F C(CCN=c1ccc([N+](=O)[O-])c(O)[nH]1)N1CC(C(=O)Nc2c(C)cc(=O)n(C)c2)C1 N1(C(C2(C#N)CCOC2)=O)CCN(C(=O)CC2CCSCC2)C(CF)C1 CC1(C)C(CC(=O)NC(c2ccccc2F)CNC(=O)C=CC2CCOC2)C1(C)C C12(CNC(c3cc(C(=O)OC)ncc3)=O)CCCC1CN(C(=O)CC1OCCO1)C2 C1(CNC(C2CN(CCC)C(=O)C2)=O)CN(C(C2CCCN2C)=O)CCC1(F)F N1(CCC)CCC(C(=O)NC(C)(CNC(c2cc(C)sn2)=O)C2CCC2)CC1 Cc1c(C=O)cnn1C.C1(C)(NCC2(O)CC(CO)C2)CCN(C(=O)OC(C)(C)C)C1 C12(CNC(C3C(=O)NCC3)=O)CN(C(=O)CSc3ccccc3O)CC1CCO2 c1(OC)cc(C)c(C(=O)NC(C2CN(C(=O)CNC(N)=O)CCO2)C)cc1OC Cc1nc(C(C(=O)Nc2ccccc2)N(c2ccccc2)C)sc1Br C(N=c1[nH]c(=NCC(C)CO)[nH]c2c1CCC2)C1(c2c(OCC)cccc2)CC1 C1(C(=O)NC(CC)C(C)CN(C)C)CN(C(=O)Cc2cccnc2)CCC1(C)C C1(CC)C(NC(=O)COC2(C)CCC2)CCCN1C(C1CC(S(C)(=O)=O)C1)=O C12(NC(C(CC3CC3)NC(=O)C=CCOC3CCCC3)=O)CCC(CC1O)C2 C1(C)(C(=O)NC(CCC)C2CC2)CN(C(=O)Cc2cccnc2F)C(C)(C)C1 C1(C(=O)NCC(c2ccsc2)C)(CNC(=O)CCN(C)C)CC12CCC2 c1(C(N(C(CNC(C(CC(C)=O)(C)C)=O)C)C)=O)c[nH]c2cc(Cl)ccc12 C12(C(N3C(CNC(CC(c4c(C)noc4C)C)=O)CC3)=O)CC(C)(C1)OC2=O CC1c2c(F)cccc2CCN1C(=O)NC1CC(N(C)C)C12CCC2 N1(C(C2C(C)(C)C2C#N)=O)CC(C(=O)NCC2CC23CC3(F)F)C2(CCC2)C1 Cc1cncc(C(N2CCC(N3CCN(C(c4cc(C#N)no4)=O)CC3)C2)=O)n1 Cc1n[nH]c(C)c1SCC(=O)NC1CCC1NC(C1CCS(=O)(=O)C1)=O C1(C(=O)NC(C(C)CCNS(=O)(=O)N(C)C)=O)CN(C(N)=O)CC1(C)C C#CCCCC(=O)N1CCCC1C1(NC(=O)COc2ccccc2C)CC1 C1(OC)CCN(C(=O)COC2(C3CC3)CN(C(=O)C(C)=CC3CC3)C2)CC1(C)C c1(C(=O)NCCSCC(=O)N(C)CC)cc(C2CC2)on1 Cc1cccc(C)c1C(O)C(=O)NC1C2CN(C(c3ccsn3)=O)CC12 N1(C(CCC#C)=O)CC2CCC2(CNC(C2CC3C(C2)C3(C)C)=O)C1 C1(N(C(C(C(C)C)F)=O)C)CN(C(=O)COc2ccsn2)CC12CC2 c1(C(=O)NC2(CNC(C(F)=CCC)=O)CCCC2)c(C)ccc(F)c1O Cc1ccc(Cl)c(N(c2cccn(C3CCSC3)c2=O)CC2CCC2)c1 C=CCC(C)(CC)C(=O)N1CCC(NC(=O)CCc2cccc(O)n2)C(F)C1 C(C(C)(C)CC(=O)N1CC(CCNC(=O)CSc2ccc(F)cc2)(OC)C1)OC CC1(C)OCC2CC12C(=O)N(c1cc(Cl)ccn1)CCNC(=O)C1CC1 N1(C(c2ccc(C#C)cn2)=O)CC(C)C(NC(=O)CCC(C)(C)OC)C(C)C1 CCCCCC(C)(C)C(=O)NCCCC1CCCN1C(c1cn(C(C)C)cn1)=O C1(C(c2n(-c3c(CC)cccc3)nnn2)NCCF)CCCC(=O)CC1 C#CCCCCCCNC(C(C)(C)OC)c1nnnn1CCCSC N1(C(c2cncc(C3CN(C(C(C(C)(C)C)O)=O)C3)c2)=O)CCC(O)C(F)CC1 C1(CC(=O)N(CC(F)Cl)C)CCCCN1C(c1ccnc(O)c1)=O C1(NC(C2(COC)CCCC2)=O)(COC)CCN(C(=O)CN2CC3CC3C2)CC1 Cc1ccn(C)c1C(=O)NC1CC(NC(=O)C)C1.c1(SCC=C)ccccc1Cl CC#CCC(C(=O)NCCc1c[nH]nc1C)NC(c1cccn1CC)=O C1(NC(C2(C)N(C(CNC(C3C(C)C3)=O)=O)CC=C2)=O)CCCCC1N=[N+]=[N-] Cc1nn(CC(N2CCOCC(NC(=O)CN=S(C)(C)=O)C2)=O)c(=O)nc1C Cc1cnc2c(c1)N(C(=O)CC1(N(C(=O)Cc3coc(C)n3)C)CC1)CC2 c1(NC2C(C)CN(C(=O)C=CC3CCCC3)C2)ncc2c(n1)CCCCC2 c1(NC(c2ccc(CNC(C=C(C)C(F)F)=O)o2)=O)ccc[n+]([O-])c1 C1(C2CCCN(C(=O)C#CC3CCCO3)C2)(NC(=O)CC2CCCCC2)CC1 c1(N2CCC(=CCC)C2)nccc(=NCc2ccc(F)cc2C)[nH]1 N1(C(c2cnn(C)c2N)=O)CCCCCC1CNC(C1(n2cccn2)CC1)=O CCCC(C)C(=O)NC(Cn1cncn1)C(=O)N(CCC(C)C)C N1(CC(C(CC)C)(C)O)CCCNC(=O)C12CCC2 CC(C)C(O)CN(C(=O)C(CO)NC(c1cocn1)=O)C N1(C(c2c(CC)cno2)=O)CC(NC(=O)C(F)CC2CCC2)CC2(CCC2)C1 c1(C(N(C(CO)CO)CC)=O)snnc1C C1(NC(CC(COC)C2CCC2)=O)(CO)CC2CCC1C2.C12CN(C1)C2=O c1(-c2cc(OC)c(C)cc2)cncc2sc(C(=O)NC(CO)C(C)C)cc12 N1(C(c2ccc(OCC)c(C)c2)=O)CC2CC1CN2C(C12CC(F)C1C2)=O C(C(=O)N(C)Cc1ccnn1C1CC1)(C(C)C)SCC.C1CCC(=O)N1 C(C(CC1CC1)C(=O)NCCCCC(=O)NC1CC1)NC(=O)C=CCF C(=O)(C1Cc2c(Cl)cccc21)N1C2CCC(CN(C(CCNC(=O)NC)=O)C2)C1 C1(N(C)C)(C(N)=O)CN(C(C2CC(n3ccnc3)C2)=O)C1 N1(C(CC(C)n2cccc2)=O)CCC(NC(=O)CC2CCC23CCC3)CC1 C1(NC(Cc2cc(CC)nn2C)=O)CC2CCC(C1)N2C(=O)C=CC1CCCO1 c1(C(N2C(C(=O)NCc3n(C)ncc3)C3CCC2C3)=O)c[nH]c2cccnc12 C=C1CC(C(=O)N(CC(N2CCCC2)C)C)(CNC(C2(CCO)CC2)=O)C1 N1(C(C(c2c(C)cncc2)C)=O)CCN(C(C2(C)CC2)=O)CCC1C c1(CC)cc([N+](=O)[O-])ccc1NC1(C)CN(C(=O)C2=C(Cl)CCOC2)C1 c1(C(N2CC=CC(NC(C3(C)CC3(F)F)=O)C2)=O)cc2c(cc1Cl)OCO2 c1(C(N2CCN(C(C=C3CCN(C)C3)=O)C(CO)C2)=O)c(F)ccc2n[nH]cc12 c1(N(C)C)cccc(C(N2CC(OCCNC(=O)CC3CCC(=O)C3)C2)=O)c1 C12(CNC(=O)CCF)CC1CN(C(C1CCC(CN3CCCCC3)O1)=O)C2 N1(C(C(CNC(c2c(OC)cnnc2)=O)C)=O)CC(=O)NC(C(C)C)C1 C1(CNC(CC=CCC)=O)CC2(CCN(C(=O)C(C)(C)F)C2)CO1 Cc1nc(C=CC(=O)NCC2CCC(NC(=O)CCc3ccn(C)n3)C2)[nH]c1C N1(C(C(C(C)O)(F)F)=O)CCC2(CCN(C(=O)CCC(C)(C)C)C2)C1 C(=O)(C(C)C1OCCc2sccc21)N(CCOC(CC)(C)C)C CCC(CC(F)(F)F)C(=O)C(C#N)C(=O)Nc1cccc(S(C)(=O)=O)c1 C=CC(CCC)CC(=O)NC(C)(C)CC(=O)N1CCCC1CC1CC1 n1(CCCC)nc(CSc2nnc(SC)n2C2CCC2)c2ccccc2c1=O Cc1cn2ccccc2c1C(=O)NCC1(F)CCC(NC(C2(F)CC2)=O)C1 C1(CC(=O)NCC2CC2CNC(c2cn[nH]c2)=O)CCCCO1 c1(C(N(CCNC(CCCSCCCC)=O)CCOC)=O)cc(SC)oc1C N1(C(C(CC)F)=O)CCOC2CN(C(=O)COc3ccc(Cl)cc3F)CC12 c1(CC)cc(C(=O)NC2(C)CCCN(C(C34CC(C3)C4)=O)C2)ccc1F CON=C(C(=O)NCCOCCNC(=O)CCCc1ccccc1)c1ccco1 c1(C(=O)NCC(C)(C)NC(C2(F)CC2(F)F)=O)cccnn1 N1(C(COC(CC)CC)=O)CCC2(CC(NC(c3ccc(C(C)=O)[nH]3)=O)C2)C1 N1(C(C2C(C=C)OCC2)=O)CC2(CC(NC(=O)C(C3CCCC3)OCC)C2)C1 c1(-c2n(C3CCC(C)C3(C)C)nc(C3CSC3)n2)ccc2c(c1)C(=O)NCCO2 N1(C(C(CCCC)O)=O)CC2CC(NC(=O)CCCC3CCCC3)CC2C1 Cc1c(C(=O)NC(C)Cn2cc(C(C)(O)CCO)nn2)cc(Br)cc1F Cc1cc(C(=O)NC2CCC(NC(=O)CCCCn3ccnn3)CC2)nc(O)c1 C1(CC(=O)NCC2CCCCN(c3snc(C)n3)C2)CCc2ccccc2N1 c1(CC(=O)NCC2(OC)CCN(C(CCC=C)=O)C2)ccc(C#C)cc1F c1(C(N2CCC(N(C(=O)Cc3cccc(F)c3)C)C2)=O)cnc2n(c1=O)CCS2 N1(C(CNC(C=CC=CCC)=O)=O)CCCC(O)(Cc2cccc(OC)n2)C1 C(c1cccc(Cl)c1)=CC(=O)N(C1CCN(C(c2ccon2)=O)CC1)C C12(NC(c3cc(SC)c(C)o3)=O)CCN(C(=O)Cn3ncc(O)nc3=O)CC1C2 c1(C(=O)NC(C#C)(C)C2CCOC2)coc(CNC(C2CC23CCC3)=O)n1 C(C)(C(O)C(=O)NCCN1CCN(C(=O)C(c2ccccc2)C2CC2)CC1)SC c1(CC(=O)NCCCCNC(C2(C)C(CC)CCC2)=O)ccc2c[nH]nc2c1 CC1CC(NC(c2sccc2Cl)=O)CN1C(c1cccc(O)n1)=O c1(CNC(CC(C2CC2)NC(C2C=C(C)CS2)=O)=O)cccc(C)c1O Cc1cc2n[nH]cc2cc1C(=O)NCC1CCN(C(=O)C(C)CF)CC1C N1(C(c2nc(C)sc2)=O)CC2CCC(NCc3nnnn3CC(F)(F)F)CC2C1 C1(CNC(C2(C)CC2F)=O)(CNC(=O)C=CCF)CCOCC1 C12(C(=O)NCC(C)CNC(=O)CC(F)(F)C(F)(F)F)CC3CC(CC(C3)C1)C2 c1(CCCC(=O)NCC2CN(C(C3CC4(C3)CC4F)=O)CCO2)ccccc1Cl Cc1cc(Cl)ccc1C(=O)NCCN1CCN(C(=O)C(C2CC2)C2CC2)CC1 c1(CC)cc(C(N2CC(NC(=O)CN3CC(C)C3)C(C)C2)=O)oc1CC c1(C(=O)NC2(CC=C)CCN(C(=O)CCC(C)(C)F)C2)nc(C)ncc1Cl c1(C(N2CCCCCC2)C(=O)N(C2CC2)CC2CCOC2)nc(F)ccc1Br c1(C(=O)NCCCNC(=O)CC(=O)NCC(F)(F)F)ccc(C2CC2)nc1 C1(NC(Cc2cccc(SC)c2)=O)CC2CC1N(C(c1cnc(N)c(Cl)c1)=O)C2 C1(C(N(CCCC)CCO)=O)(OC)CCN(C(=O)CC2CCCNC2=O)C1 c1(C(C)OC)nc(C(=O)NC(C2CCN(C(C3COC3)=O)C2)C)cs1 CCCC(O)CC(=O)NC1CCN(C(=O)Cc2ccc(C)s2)C(C)C1 CC1(C#N)CCCN(C(=O)CC2CCN2C(c2cc[nH]n2)=O)C1 C1(C)(C(N2CCN(C(C(CSC)OC)=O)C(CF)C2)=O)Cc2ccccc2C1 c1(CNc2c(CC(=O)Nc3cnc(I)c(Cl)n3)cccc2)cccc2c[nH]nc12 c1(N2CCC(C)(OCC)C2)nc(N2CCC(CCCC#N)CC2)c2ccsc2n1 c1(C(N2CC(O)CC(NC(CCCC#C)=O)C2)=O)cc2cc(F)ccc2[nH]1 C1(C#N)(CC(N2CCC(COC)(NC(=O)CN(C)C)C2)=O)CCCCC1 C1(C(=O)NC2(C#C)CC2)CC(C)CN(C(c2cc(CSC)c[nH]2)=O)C1 C1(C(N2CCC(CC3CCCC3)C2)C(=O)NC)CCCN1CCNC(=O)N(C)C N1(C(c2sc(Cl)cc2Cl)C(=O)NCCCF)Cc2ccc(O)cc2C1 N1(C(C)C)C(=O)COCC1C(=O)OCC.c1(C(=O)N)cc(C(c2ccccc2)=O)c[nH]1 c1(CNC(c2cnc(C)s2)c2nnnn2CC2CCCO2)ccc2nc(O)oc2c1 C1(NC(c2cccc(S(=O)(=O)N(CC=C)C)c2)=O)CCc2c(nnn2C(C)C)C1 CCCCC(C)C(=O)N(CC(C)N(C)C(c1nc(C)ccc1F)=O)C c1(COC)nn(C)cc1C(=O)NC(C)CCNC(C1CCC(=O)N1C)=O N1(Cc2c(C)cc(C)[nH]2)CCN(C)C(C(=O)NC(c2ccccc2Br)C)C1 CC1CCCCCN1C(=O)Cn1cc(-c2cccc(C3CC3)n2)nn1 c1(OCCN(C2CC2)CC)ccc2cc1-2.N1(C)CC(C2CCCO2)C1.C(C)(C)(C)O C(=O)(C1=CC(O)CCC1)NC1CCC(NC(=O)Cc2csc(S)n2)C1 C1(CC)CN(C(=O)C=Cc2ccc(OC)cc2)CCC1NC(=O)CC(O)C(C)C C=CC1(C2(C(=O)NCCC3(c4ccccc4)CCCC3)CCC2)CCC1 N1(C(c2cnn(C)n2)=O)CCC2(CNC(c3cnccn3)=O)CCCCC12 C(=O)(C(CC(C)C)NC(C)=O)NC1CN(C(c2noc(CC)c2C)=O)CC1SC C1(C#N)(NC(CC=CCC)=O)CCN(C(c2ccc(N3CCOCC3)cc2)=O)C1 CCCCCC(O)CNC(=O)C=CCN(C(=O)CC1CC2(CC2)C1)C N1(C(CC(CC)C)=O)CCCC12CCN(C(C1CCCCC13CCC3)=O)C2 Cc1cc(O)ncc1C(N1CCC(NC(c2ccc(OCCN(C)C)cc2)=O)C1)=O C(CCF)(C(=O)NCCOCc1nc[nH]n1)NC(=O)CC1CC1C1CC1 C1(CNC(C=CCCC)=O)CC(NC(c2ccnc(-n3ccnc3)c2)=O)C(O)C1 N1(C(C2N(C(C)C)CCCC2)=O)CCCCC2(CCN(C(=O)C3=CCC3)C2)C1 N1(CC2C(CC)CCC2)CCCC(Cn2cc(-c3cccc(O)c3F)nn2)CC1 N1(C(CCC2CC(NC(C3C4CCC(F)C34)=O)C2)=O)CCC(F)CC1 N1(C(CC(=O)NCC#C)=O)CCCN(C(=O)Cc2cnc(C)s2)CCC1 Cc1ncc(Cl)c(C(=O)NC(CO)C(C)NC(c2ccc(F)c(Cl)c2)=O)n1 C1(C(N2CC3(CN(C(CC4CC(C)(C)OC4)=O)C3)C2)=O)CCC([N+](=O)[O-])CC1 C123CC1CN(C2)C(=O)N3.n1(CC=C)cc(CNC(C)(C)C)cn1 C1(CNC(C(C)SC)=O)CCN(C(=O)CCn2cc[nH]c(=O)c2=O)C12CC2 c1(CNC2CC(CC(=O)NC3(c4cc(C)[nH]n4)CC3)C2(C)C)c(C)cccc1F CCC(C)C(C(F)(F)F)NC(=O)NCC(c1cccc(C)c1C)O C1(C(=O)NC(c2nc(C)sc2)C)CC(F)(F)CN1C(c1cn(C)cn1)=O C1(C(=O)NC(CCOC)(C)C)CCN(C(=O)CCc2cccc(O)c2)O1 c1(NCC(CN(C(c2cn[nH]c2)=O)CCO)O)ncc(C(F)F)cn1 Cc1nc2cccc(C(=O)NCC34CCCC3CN(C(=O)C(N)=O)C4)c2[nH]1 N1(c2snc(C)n2)CCC2(CCN(C(=O)NC3CCn4c(C)nnc4C3)CC2)C1 N1(NC(C2CCC(NC(C3CCCC(C)C3)=O)C2)=O)CCC(C)(C)CC1 C1(NC(C(CC)C)=O)CC(C)N(C(c2ccc(C3(F)COC3)cc2)=O)C1 C1(NC(CN(C)C(=O)C2CC2)=O)CN(C(C2(C#N)CCCC2)=O)CC1CO C1(NC(c2c(OC)n[nH]c2)=O)COCCN(C(=O)CN(c2ncccn2)C)C1 c1(C(C)C(=O)N2CCC2CC(C(C)CCCO)=O)ccc(Cl)cc1.C(C(C)(C)O)N C1(C)(C(N(CCC(C)NC(=O)CN2CC=CC2)C)=O)CCCNS1(=O)=O N1(C(C2CCN2Cc2cncc(C(F)(F)F)c2)=O)CCCC1c1cc[nH]n1.C1CC1 N1(C(COCCOC)=O)CCC(C)C(N(C)C(c2cc3n(n2)CCC3)=O)C1 CC(C)(C(=O)NC1CC(CNC(C2CS(=O)C2)=O)C1)C1CCCCC1 N1(C(c2nc(CCOCC)oc2)=O)CCC(C)(CNC(=O)C2=CCOCC2)CC1 c1(NC(N2C(C)CC(CO)CC2)=O)cccc2nc(O)ccc12 CC1CCN(OC2CCN(C(=O)C(N3CC4C=CC3C4)=O)CC2)CC1 c1(C(=O)NCC2CC(C)N(C(c3cnc(C(C)C)[nH]3)=O)C2)cc(Cl)c(N)c(Cl)c1 CC(CC1CC1)C(=O)N(CC(C)NC(c1occc1-c1ccccc1)=O)C C(=O)(CC1OCCc2sccc21)NCCC(C)N(C(Cc1c(C)cccc1)=O)C C12(C(c3ccc(F)cc3)NC(C(=O)N(CCC(C)F)C)=O)CCCN1CCC2 C1(C(N(C)CCOCCC(=O)NCC(C)(O)CO)=O)CCCN1C1CC1 CC(C(O)C(=O)N1CC(N(C(=O)C(F)=C2CCC2)C)C1)c1ccccc1 C#CCC(N)=O.c1(CCN2C(C3CCOC3)C(=O)O2)cocn1 Cc1cc(C)c(C(N2CC(NC(c3ccc(O)c(F)c3)=O)C(C)C2)=O)c(C)c1 C1(N(C(C(C=C)C)=O)CC)CCN(c2cc(OC3CCOCC3)ncn2)CC1O N1(C(C=CC)=O)CC2CCCC1C2CNC(c1ncc(Cl)cc1F)=O C1(CN(C)C(C2CCOC2(C)C)=O)CCCN(C(=O)C=Cc2ccoc2)C1 C1(C(=O)NCC2OCCN(C(C=Cc3nc(C)sc3)=O)C2)CC(S(C)(=O)=O)C1 N1(C(C(C)(O)C2CC2)=O)CCC(NC(=O)CSCC#N)C2(CCC2)C1 C1(NC(=O)C=Cc2ccc[nH]2)CCCCC12CCN(C(c1conc1C1CC1)=O)C2 c1(C(=O)NC2C(F)CCN(C(CNC(N)=O)=O)C2)ccc2cc(O)ccc2n1 c1(OC)cc(CN2CCC2CNC(C2CC3CCC2C3)=O)ccc1C(F)F N1(C(c2cccc(N(C)C)n2)=O)CCC2(CCOC2)C(CNC(C2(O)CC2)=O)C1 C1(C(N(CCCSC)C)=O)CC2CCC1C2.C12CC(C1)NC(=O)CO2 C1(N(C(C)=O)CC)CCCN(C(c2ccoc2)C(=O)NCCC2CC2)C1.C(COC)S c1(OC)cnc(C(=O)NCCC2CCC(NC(c3csc(C)c3)=O)C2)c(Cl)c1 c1(C(C(N)=O)N(C)C(c2conc2C2CCN2)=O)cccc(F)c1 c1(NC(CC2(C)N(C(Cn3c(C)ncc3)=O)CC2)=O)ccc(Cl)nc1Cl CCC(CCC(=O)N1CCCC(OC)C1)NC(c1nscc1C)=O N1(C(C(CC)n2cccn2)=O)CCC2C(NC(=O)CCc3ccc[nH]3)CC12 Cc1ccc(-c2cn(CC3CN(C(=O)CCC(C)(C)C)CCO3)nn2)c(C)c1 C1(C(=O)NC(COC)(C)C)Cc2cc(O)ccc2CN1c1ccc(C(C)=O)cn1 Cc1cc(NC(=O)NCC(O)CNC(=O)OC(C)(C)C)cnc1Cl c1(CC)onc(C(=O)NCC2CCCCC2NC(=O)CCCOCCOC)c1C C1(NC(=O)COC(F)F)CN(C(c2ccno2)=O)C1 C1(NC(C2(OC)CC(C)C2)=O)CC2CN(C(C3CC(F)(F)C3)=O)CC2C1 C1(CC)CCN(C(=O)Cn2cccnc2=O)C(C(=O)NCCC(C2CC2)C2CC2)C1 c1(C(=O)NCCC2CC(OC)CN2C(=O)C2=CCC2)ccc(F)cc1C#N C1(C(=O)NC2CCCC2CNC(=O)C(C)(C)NC(C)=O)CCC(COC)CC1 c1(CNC(CCSCCC)=O)ncccc1C(N1CC(C(N)=O)C(CCC)C1)=O C1(CNC(C(COCC)C)=O)C(C)CCN1C(c1ccnn1COC)=O N1(C(c2cccc(OC)n2)=O)CCC(C)C(NC(=O)Cc2cc(C3CC3)on2)C1 N1(C(CC(C(C)(F)F)(F)F)=O)CC(C2CCCN(C(c3ccc[n+]([O-])c3)=O)C2)C1 C1(N(CCC#C)CC(=O)O)C2CCOC2C12CCCC2 C#Cc1ccc(C(N2CCCC(C)(C)C2C(=O)NCc2csnc2C)=O)cc1C c1(C(N2CC(NC(c3ccc(Cl)cc3CO)=O)C(F)C2)=O)c(F)cc(Cl)cc1Br C1(NC(c2c(COC)noc2)=O)(CF)CCN(C(C2(F)CCOC2C)=O)C1 c1(NCC(=O)NC(C)CNC(c2cc(Cl)c[nH]2)=O)ccc(C(C)(F)F)cc1 Cc1cccnc1C(=O)NCC1CCCCC1NC(=O)C(F)OC(F)(F)F c1(C(=O)NCC23OCC(NC(CCC)=O)(C2)C3)c(Br)ccc2c1OCO2 C(C)(CCC(=O)NC1CCCSC1)NC(c1n(CC)ncc1)=O Cc1cccc2c1CCC2NC(c1ccc(F)c(OCF)c1)C(=O)NCC(F)F n1(C(C)C)ncc(C(=O)NCC(C2CCOC2)NC(c2coc(Cl)n2)=O)c1N C=CCCCC(C)(C)C(=O)NC1CC2CC(C1)N(C(c1cc(Cl)n[nH]c1=N)=O)C2 C(=O)(CCC(CC)NC(c1cscn1)=O)N1C(CC(=O)OC)CCC1 C1(C(=O)NC2CCC(CCNC(CCCNC(C)=O)=O)C2)C(C)(C)C1(F)F C(=O)(CCCCC#CC)NCCC1(CC(=O)NC(c2ccccc2)C#C)CCC1 c1(C(=O)NC(C)C(C)NC(C2(C)CCOCC2)=O)cc([N+](=O)[O-])n[nH]1 CC(C)CC(CNC(=O)C=CC(N1CCCC1)C)C(=O)N1CCC2(CCCO2)C1 C1(CN(C(=O)Cn2cncn2)C)CCCN(C(c2cc[nH]c2C(F)F)=O)C1 c1(C(C)C)cccc(C(=O)NC(C)(C)CCCNC(=O)CCF)n1 c1(NC(C(C)OCCOCC)=O)ccccc1CNC(=O)C=Cc1cn[nH]c1 C1(C(=O)NC(C)CNC(=O)C=C2CCCCC2(C)C)CC2(CCCCC2)C1 c1(C(=O)NCCNC(C2CC2C2CCC2)=O)ccc2cc(Br)ccc2n1 N1(C(c2ncc(Br)s2)C(=O)NC2CCOC2)CCCCc2sccc21 C(C(C)(O)CNC(=O)C=CCn1cncn1)NC(C(c1cccs1)SC)=O C1(CC(=O)NC(C)C(C)NC(c2ccccc2NC(N)=O)=O)COCC(C)(C)O1 n1(CCOC)nc(C(=O)NCC(C(C)C)NC(=O)Cc2n[nH]c(=N)s2)ccc1=O c1(C(N2CC(C)CC(C(=O)NC)C2)C(=O)NCCSC)c(F)cc(F)cc1Br C=C1CCN(C(=O)C(C)N(C)C(C)=O)C(NC(=O)NCC(O)(CC)CC)C1 C1(NC(C2(COC)COC2)=O)CCN(C(c2cnn(C3CC3)c2Cl)=O)C(C)C1 CC(C)(C)CCCC(=O)NC1CC2(CCN(C(=O)Cn3ccc(=N)[nH]3)C2)C1 C1(C(=O)OCC(C)(C)C(F)F)CCCC(=O)CC1 C1(C(N(CC(CN(C(=O)CSC(F)F)C)O)C)=O)(CCN2CCCC2)CCCC1 C(=O)(CC(CN(C)C)C(F)(F)F)N1CC(OCCc2cn(CC(C)CO)nn2)C1 N1(C(C2C(CCOC)C2)=O)CC2CN(C(c3cc(F)ccc3OC)=O)CCC12 c1(OC)ccc2nc(SCCC(=O)NCC3CCCC(C)C3)cn2n1 c1(C(N(C)CC2CCN(C(C(CC)F)=O)C2)=O)cc(F)c(F)c(F)c1N C1(NC(C(C)C(F)(F)F)=O)CN(C(c2nc(Cl)ccc2N)=O)CC2(CCC2)C1 C12(n3cc(C(C)OC4CC4)nn3)CCC(NC(=O)CCN3CCC(O)CC3)(CC1)C2 C1(CC(=O)NC(C(=O)OCC)(C)C)CCCC(NC(=O)Cc2ccccc2O)C1 c1(OCC(=O)NCC(C)CNC(=O)CCC(=O)NN(C)C)ccc2c(c1)CCCC2 C1(C(=O)NC(CNC(C2CC(CC)(CC)C2)=O)C(C)C)CCCCC12CC2 CCCCCC(C)(C)C(=O)NC1(C(=O)NC(C)Cc2ncn(C)n2)CC(O)C1 C(=O)(CC1NC(=O)c2ccccc21)NCC1N(C(C2(OCC)CCCC2)=O)CC1 c1(C(N(C(CNC(C(CC)=CCCC)=O)C)C)=O)cccc(C2CC2)c1 C1(N(c2ccncc2)CC)CC(COC)N(C(=O)C(C)N(C)C)C1 C(=O)(CC(C)O)N(CCC(=O)NCC=CCOC)C(C)C c1(C(=O)NCC2C(C(=O)NC(CC=C)C)C2)cc2cccn2cn1 N1(C(c2ccc(C#C)cc2)C(=O)NC2CCCC2)CCc2ccccc2C1 C1(c2ccc(OC)cc2)(NCc2c(COCC)noc2)CC2(CCC2)C1 c1(CCC(=O)NCC2CCSCC2)nncnc1O C1(S(N)(=O)=O)(C(=O)NCC2CC(NC(Cc3ncc(C)s3)=O)C2)CCCC1 c1(C(=O)NC2C(NC(c3c(C)nn[nH]3)=O)COC2)sc2cc(F)ccc2c1C C1(NC(CN2CCC(C)C2)=O)CN(C(=O)CCCCC2CC2)C2(CCOCC2)C1 CC(c1cnn(C)c1)=CC(=O)NCC(C)(C)CNC(c1c(Cl)cnn1C(C)C)=O c1(C(=O)OC)cccc(N2CCN(C3CCOC3)C2=O)c1.C1C(=O)O1 C1(NC(C(=O)NN(C(C)COCCCC)C(C)=O)=O)CC2(C1)CC(CO)C2 N1(CCNC(C2CC3COCCC23)=O)CCS(=O)(=O)CC1 C1(C(=O)NC2CCCC2CSC)(NC(C(C=CC)O)=O)CCOCC1 Cc1c(Br)cnc(O)c1C(=O)NCC1CCCC1NC(C1(CO)CC1)=O n1(CC(=O)NC2CN(C(C3(CC#C)CC3)=O)CC2C)ccc(=O)c(O)c1C N1(C(CSc2n(C)ncc2)=O)CC2(CC(NC(C3CCOC3=O)=O)CO2)C1 c1(NC(=O)NCc2ccc(CC(=O)OC)cc2)ccc(Cl)c(I)c1F CC1(C)CCC(C(N2CC3CC2(CNC(=O)CC2CC2)C3)=O)CO1 CC1(C)CC(CO)CN1C(C1CC(CCNC(C23CC(C#N)(C2)C3)=O)C1)=O c1(C(=O)NC2CN(C(c3ncncc3Cl)=O)CC2O)cn2cc(Cl)cnc2n1 C1(C(=O)Nc2cncnc2)C2CC1N(C(c1cncc(O)c1)=O)C2 C1(C(N2CCC(O)CC2CC)=O)(CC)CCCN(C(C2CSC2)=O)C1 C1(n2c(C(=O)NCC(CNC(C(C)(C)N(C)C)=O)O)cnn2)CCS(=O)(=O)C1 c1(C(N2CC(C)CC(CNC(CCCC#C)=O)C2)=O)cccc2c1ncn2C c1(C(=O)NCC(CCC)O)ccnc(CNC(=O)CCOCC2CCC2)c1 Cc1conc1C(N1CCCC1C(=O)NCc1cn(C2CC2)cn1)=O C(CC(O)CNC(C1(O)CC1)=O)NC(c1cnc(Cc2ccccc2)s1)=O O=C(CCC(F)(F)C(F)F)NC1CC2CC(C1)N(C(=O)C=CC1CCCO1)C2 N1(C(c2cc(CC)n(C)n2)=O)CC2CCC(C1)C2CNC(C1CCCS1)=O N1(C(c2cn(CCO)nn2)=O)CCC(OCC(=O)NC(CCO)C2CCCC2)C1 CC(CC1CC1)C(=O)N1CCC1CNC(c1cc(Cl)on1)=O N1(C(C2CCC(C)O2)=O)CCC(CO)C(NC(=O)CCC23CCC(CC2)C3)C1 c1(NC(C2(NC(CC3CCCC(C)C3)=O)CC(O)C2)=O)ccc(F)cc1C1CC1 c1(NCC2(OCCOCC)CC2)ccc(C(N2CC(O)C(F)C2)=O)cn1 N1(C(CSC(C)(C)C)=O)CCN(C(c2ccn(CCF)n2)=O)C(CCO)C1 c1(CC)ccc2nc(Br)[nH]c(=NCCC3CCS(=O)(=O)CC3)c2c1 CCCC(C(=O)Nn1cnn(CC)c1=O)NC(=O)C=Cc1ccsc1 O=C(C1=NOC(CNC(c2conc2C2CC2)=O)C1)NCCC1CCCO1 C1(N(C(C)=O)C)CN(C(C2CC23CCSCC3)=O)CC1(C)C C1(C(N2CC(CCC)C2)=O)(CC)CCN(C(=O)Nc2ccc(C)nc2O)CC1 c1(C(=O)NCC2C=CC(NC(C3(OC)CC3)=O)C2)nccc(Cl)c1Cl CC1(C)CCC(CCNC(=O)C(C2CC2)NC(=O)COCC2CC2)C1 c1(C(=O)NC2CCC(CNC(C3(C=C)CC3)=O)C2)ccc(Br)c(F)c1 N1(c2ncc(C)cn2)CCC(C2CC2)C1CNC(=O)C=CCF C1(C2(O)CN(C(=O)CCn3ccnn3)C2)(CNC(Cc2nc(C)[nH]n2)=O)CC1 c1(C(=O)NC(c2nn[nH]n2)CC)sccc1CNC(c1cccn1C(C)C)=O C1(NC(CC2(C)CCOC2)=O)(CO)CCCN(C(C2CC3(CCC3O)C2)=O)C1 CC(C)S(=O)(=NC(=O)c1cnn(CCn2cccn2)c1)C(C)C C1(CONC(c2cc(CF)on2)=O)CCCCN1C(c1cc(CC2CCC2)on1)=O Nc1cc(C(=O)NC2CC(NC(C3CCCCNC3=O)=O)C2)cc(Cl)n1 c1(CC)cc(C(N2CC(CCNC(C34CCCC3C4)=O)C(C)C2)=O)ccc1C CC(C)(C(=O)OC)C1=CCN(C(c2cc(C(F)F)[nH]n2)=O)C1.C12CCN1C(=O)C2 c1(OC)cc(C(N2CC(N(C)C(c3cnc(C)nc3)=O)C2)=O)c2ncccc2c1 C1(C2CC2)(C(=O)Nc2ncc(C(=O)OCC)nc2)CCN(C(=O)CCS(C)=O)C1 CC1CC2CN(C(=O)CCc3cccnc3F)CC2N1C(C1CCCCO1)=O c1(C(N2CCN(CC(C)NC(CCCCCC)=O)CC2)=O)cc(C#N)ccc1O C1(OC(CC2C(C(=O)OCC)CC2)=O)CC(C)CN(C(=O)OC)C1 Cc1coc(C(N2CCC(Oc3ccccc3F)C2C)=O)c1C C(N=c1[nH]c(N(CCC(C(C)CC)OC)C)nc(=N)[nH]1)c1c(CC)n[nH]c1 CC(C)S(=O)(=O)CC(=O)NC1CCOC1C1CCN(C(C2(CCO)CC2)=O)CC1 N1(C(c2c(OC)n(C)nc2)=O)CC(NC(=O)CCC(=O)c2ccsc2)CC(C)C1 CC(C)C(C(=O)NCc1coc(C(C)C)n1)NC(=O)CCC1CCCOC1 N1(C(C(C)S(C)(=O)=O)=O)CCC2(CC1)CC2CNC(c1cc(F)cc(F)c1F)=O C=CCC(CC=C)C(=O)NC1CCCN(c2ncnc(O)c2Br)CC1 C(=O)(C1=NOC2(CCCN(C(=O)C(F)Cl)C2)C1)Nc1ccc(NC(C)=O)cc1C c1(CNC2CC(C(N(CCC)CCO)=O)C2)cnc(OC)c(Cl)c1 C(=O)(C1=CCCCO1)NCCOC(CNC(Cc1nc(C)sc1)=O)(C)C CC(C)C(COC)C(=O)N(C)CC1CN(C(=O)CCOC2COC2)CCO1 C1(O)(CC)CCN(C(=O)C(CNC(C2CN(C)C(=O)N2)=O)N(C)C)CC1 C=CC1CCN(C(c2ccnc(CNC(=O)Cc3ccccc3O)c2)=O)C1 Cc1cccc(C)c1CN(C(=O)CN1CCNC(=O)C1)CC(C)C Cc1cnc(C(=O)NCC2CCN(C(C3(C)CCC(=O)NC3)=O)C2)c(F)c1 C1(C(C)NC(c2ccnn2CC#N)=O)CN(C(=O)CCOCCN(C)C)CCO1 CC1CN(C(c2ccsc2)=O)CC1CCNC(=O)C=CC1CCOC1 C1(NC(=O)CO)C2CC3CC(C2)CC1(CNC(C1(n2cccn2)CCC1)=O)C3 C(CC(C(C)(C)C)NC(=O)Cc1csnn1)N(C(=O)CP(C)(C)=O)C Fc1cc(F)c(Cc2nc(-c3cccnc3)nn2-c2ccnnc2)cc1F CC1(C)CN(C(=O)CCCn2cccc2)CC1CNC(=O)CN1CC=CC1 CCC1=C(C(=O)NCC2CC3CCC2N(C(c2cocc2C)=O)C3)SCCO1 C1(CC(=O)N(C)Cc2ccncc2)COCCN1C(=O)CC1CC(F)(F)C1 c1(COC)cc(C(=O)N(CCCNC(c2c[nH]c(Br)c2)=O)C(C)C)no1 C1(C(N2C(COC)(CNC(=O)CCS(C)(=O)=O)CCC2)=O)CC(C)CC(C)(C)C1 C1(NC(c2c(C(C)NC(C3(CCO)CC3)=O)noc2)=O)CCCOCC1 CC(C)C(CC(=O)N1CC(NC(C2(C(F)F)CCCCC2)=O)CCC1C)C(C)C c1(CC)ccc(Br)c2nc(NC(C3CC(C)C3)=O)sc12 CCCCCCCCC(C)CC(=O)NCCCCCNC(c1cc(C)[nH]c1C)=O c1(N(CCNC(C2CCN(C(C)=O)C2)=O)C2CC2)c(C(F)(F)F)ncn1O c1(SCCCC)cccc(NC(=O)OCC)c1.C1(CC(=O)OC)CN1 C1(C(=O)NCC(C2CCCC2)NC(c2[nH]cc(CC)n2)=O)CCCCCCC1 Cc1ncnc2c1CC(C(=O)NCC1(O)CN(C(C3CCNC(=O)C3)=O)C1)CC2 c1(C(=O)NCC2(CNC(C(CC=CCC)C)=O)CCCCC2)cc([N+](=O)[O-])n[nH]1 Cc1cnc(C(=O)NC2(C)CC(NC(=O)Cn3ncn(C)c3=O)C2)cc1Br C=C(C)CCC(C(=O)N1CCC(c2cccc(Cl)c2Cl)C1)N1CC(=O)NCC1(C)C c1(C(N(CC)CC2CCCN2C(=O)CCS(C)=O)=O)n[nH]c2cc(C)ccc12 c1(Cc2ccncc2)cn(CCCF)nn1.C1(C(F)F)(C)CC1 Cc1ccc([N+](=O)[O-])cc1NC(=O)CCc1ccc(C(F)(F)F)cc1 c1(OCC(=O)NCC2CC(C(=O)NCC(C)(O)CN(C)C)C2)cccc(F)c1 c1(C(=O)NC2CC3(C2)CN(C(=O)CC2CCOC2)C3)ccc(=O)n2c1COCC2 C1(CN=C(NC(C)C)NCC2OCCCC2(C)C)CCC2(CCC(C)(C)CC2)O1 C12(C(N3CC(CCO)(OC)C3)=O)CCC(CC(=O)NC(C)C)(CC1)C2 N1(CCCC)CC(C(=O)Nc2cnn[nH]2)CC1=O.C12CCCN1C(=O)C21CC1 Cc1cccc(CC(N2CC(CNC(c3c(C)cnn3C)=O)C(C)C2)=O)c1Br CN1CCn2nc(C(N3CC4CC4(CNC(=O)Cn4ccnn4)C3)=O)cc2C1 CS(=O)(=O)CC(=O)NCC(O)CCNC(C1C2(CC2)C12CC2)=O N1(C(C(C)=C2CC2)=O)CCCC1C1CCCCN1C(c1ccc2c(n1)CCC2)=O CC(C(=O)NC(CN(C)C(C1(O)CCC1)=O)CO)N(C)NC(=O)OC(C)(C)C Cn1c(O)nc2cc(NC(c3cccn(C4CCC4)c3=O)=O)ccc12 c1(CNC(C2OCCN(C(c3cc(C)n(C)c3)=O)C2)=O)c[nH]cc(Cl)c1=O C(=O)(CC(CCCC)NC(=O)C(C)(C1(C)CC1)OC)N1C(CCCC)CCC1 C(C(N=[N+]=[N-])C(=O)NCC(C)CC(=O)NCCOC(F)F)OC.C1(C)CCC1 c1(NC(C2C(O)CCN2Cc2cc(Br)cnc2Br)=O)ncc(Br)cc1Br c1(CC)cc(C)c(C(=O)NCCCN(C(C2CC2c2ccc(C)cc2)=O)CC)o1 S(=O)(=O)(C1CC2C=CC1C21CC1)C(C(C)CC1CC1(F)F)=O C1(CNC(COCCCC)=O)C2CCCC1N(C(C1(O)CCSC1)=O)C2 CC(C(=O)N(C)CCN1CCCC1)S(N)(=O)=O.c12cc(ncn1)OC2 c1(C(=O)NCC(C)CNC(=O)C(C)(C)NS(C)(=O)=O)cc2c(s1)CCC2=O CCC(C)C(C)C(=O)NCCCN(C(=O)CCc1ccccc1O)C1CCCC1 C(C)(C(CC(=O)N(OC)C(C)C(=O)Nc1cc(C)nn1C)SC)OC c1(NC(C2CC(NC(=O)CSc3ccccc3)C2)=O)ccc2ccccc2c1Cl c1(C(=O)NC23CN(C(=O)C=CC(F)(F)F)CC2COC3)cc2cncc(Br)c2s1 C1(NC(c2c(C)c[nH]n2)=O)CCCC2CN(C(c3snnc3C)=O)CC12 C1(C(C)C)(C(=O)NCCN2CCOCC2)CCCN1C(c1ncn(C(C)C)n1)=O N1(c2n(CC(=O)NCCO)c(C(C3CCCCO3)OC)nn2)CCn2ncc(Br)c2C1 N12CC3CN(C3C1)C2=O.c1(NC(c2c(C)cco2)=O)ccccc1C(F)(F)F c1(C(=O)NCCCC(C)NC(=O)CC(C)(C)F)n[nH]c2ccc(O)cc12 N1(C(N2CC=CC(O)C2)=O)CC2CCCC1C2 C1(N(CCC)C(c2cnn(CCF)c2)=O)CCCN(CC(=O)NC(=O)NC)CC1 C1(C(N2CC(CCn3cc(CC(C(C)(C)C)O)nn3)C2)=O)COC2CCCCC12 CCC(C)(C)C(C)CC(=O)NCC(C1CC1)NC(=O)CN1CC(C)(C)C1 CC1CCC(C)(C(N2CCC(n3cc(CNC(=O)CCC#N)nn3)C2)=O)C1 c1(C(N2C(C(=O)NC3CCC(CC)CC3)C(C)(C)CC2)=O)c[nH]c2ccccc12 CC1CN(C(C2(C)CCN2Cc2cccc3cc[nH]c23)=O)Cc2ccc(Cl)cc21 c1(C(=O)NC2(CC)CCCN(C(=O)CO)C2)cncc2c1CCNC2=O c1(C(N2C(CNC(C3N(CC)CC3)=O)CC3CC32)=O)cc(C)cc(C)c1C N1(C2CCN(C(=O)C=CC3CCCO3)C2)CCS(=O)(=O)CC1 CCC(CC)C(C)C(=O)NCC1(OC)CCN(C(c2ccc(C#N)c(C)c2)=O)C1 N1(C(C(C)(C)C2CCOC2)=O)CCOC(CC(=O)NCc2cncc(F)c2)C1 c1(C2(C)CC2SCC(Cl)Cl)ccccc1F N1(C(CCOc2cccc(C)c2)=O)CCCOC(CNC(c2csc(C)n2)=O)C1 c1(C(N2CCC(NC(CSCCC)=O)C(C)C2)=O)nn2c(c1C)CCCC2 C1(CNC(CCOCC)=O)CC2CCCCC2N1C(C1CNC(=O)N1)=O N1(C(C(C)SCCC(C)C)=O)CCCCC1CCNC(=O)C(=O)N(C)C N1(c2c(C)c(NCC(=O)NCC(F)(F)F)ncn2)Cc2ccccc2C2(CC2)C1 N1(C(c2scc(C)c2C)=O)CCN(C(c2cccc(C(F)F)c2)=O)CC1CF N1(C(CS(C(C)C)(=O)=O)=O)CCC2(CCCC2CNC(=O)CN(C)C2CC2)CC1 N1(C(=O)C=CCOc2ccc(F)cc2)CCC2CN(C(C34COCC3C4)=O)CC12 CCCC(CCC)CC(=O)N1CCC2CN(C(C3CCCCO3)=O)CC12 n1(CCC(N2CC(C)N(C(=O)CN(C)CCO)CC2)=O)ccc2cccnc12 C1(C(=O)NC(c2ccnn2C)C(N2CC(OC)C2)=O)C2CCCCCC12 c1(OC)ccc2ccccc2c1NC(c1cn(C2(Cc3cc(C)[nH]n3)CC2)nn1)=O N1(C(C2N(C(C3CC(=C4CCC4)C3)=O)CC(=O)NC2)=O)CCCC(CO)CC1 N1(C(CC2C(C)C2)=O)CCCC2(CC(NC(=O)CCC3(C)CC3)C2)C1.C1CO1 C(c1cccc(C(F)(F)F)c1)=CC(=O)N(CC(C)NC(=O)Cc1ccccc1)C C1(NC(c2c(SC)cccc2)=O)CC(NC(=O)C=Cc2ccccc2)C12CCC2 Cn1cnc(C(=O)NCCCOCCC(=O)NCC2(O)CCOCC2)cc1=O Cc1cc(C)c(C(=O)N(C(C)CCNC(C2CC2c2nc[nH]n2)=O)C)cc1N C1(NC(C(n2cc(Cl)cn2)C)=O)CC2CC(NC(=O)CCCN3CCCC3)C1C2 C(=O)(CCC(C)(C)F)NCC(C(=O)NC(c1cn(C)nc1)CO)(C)C C(=O)(C(O)C1=CCCCC1)NCCCN(C(=O)CC(C)(C)O)C(C)C c1(OCC)c(OC)cc(C(=O)NCCCCCNC(C2CCC(C)C2)=O)cc1Cl c1(OC)ccc(C(=O)NC(C)CCNC(=O)CC2(CO)CC2)c(C(F)(F)F)c1 C1(CNC(C2CC=CCC2)=O)CC2CCC(C1)N2C(=O)Cc1cn[nH]c1 c1(C(=O)NC2C(CNC(c3cn(CCC)nc3C)=O)C2)cc(Cl)c([N+](=O)[O-])[nH]1 c1(C(N2CCC(C)(CNC(CC(C)N(C)C)=O)C2)=O)nn2c(c1Br)CCC2 N1(C(c2cc(CCC)[nH]n2)=O)CC=C(C(=O)Nc2cccc(CO)c2)C1 C(C1=NOC2CCCC12)NC(C1CC(NC(=O)C2=COCC2)C1)=O C(c1cc(C)ccc1OC)=CC(=O)NCC(CC)OC(=O)CC1CC1N N1(C(c2cc(C(C)C)no2)C(=O)NCC=C)Cc2cc(Cl)ccc2C(C)C1 c1(CC(=O)NCC2CN(C(C(C)(Cl)Cl)=O)C2)ccc2c(c1)OCO2 N1(C(c2ccc(N)cc2F)=O)CCC2(CCCN(C(C3(O)CCCC3)=O)C2)C1 Cc1ccnc2c(C(=O)NC3(CNC(c4cnc(S)nc4)=O)CC3)cnn12 C1(N(C(c2cc(C(N)=O)[nH]n2)=O)CC2CC2)CCN(C(=O)C=C(Cl)Cl)CC1 Cc1c(Br)c(C(=O)NCC(C)(CC(C)C)NC(C2CC23CC3)=O)nn1C C1(C(=O)NCC2C(NC(c3cc(C)no3)=O)C2)CCC(C)(C)CO1 Cc1ccc(C(N2CCC(C(C)NC(C3(C(F)(F)F)CC3)=O)CC2)=O)cn1 CN1CCCN(CCC2CCN(C(=O)CC3CS(=O)(=O)C3)CC2)CC1 c1(CC)ccccc1NC(=O)C(c1cccc(F)c1)N(CCC#N)C(C)C c1(C(=O)NC2CCN(S(=O)(=O)CCCCl)CC2F)ccc2c(Cl)ccnc2c1 c1(CN(CCN(C)C)Cc2cc(C(F)F)ccn2)cccc(CN)n1 C1(N(C)C(C2CCCOC2)=O)CC2CCC(C1)N2C(C12CCC(CC1)C2(C)C)=O N#Cc1ccccc1CCC(N1CCCC(O)(CNC(=O)CSS(C)(=O)=O)C1)=O C(=O)(C(O)(C(F)(F)F)C1CC1)N1CC(CNC(c2cc(F)cs2)=O)OCC1 c1(OC)cc(C(=O)NC2CN(C(=O)CCCC(C)=O)CC2F)ccc1OC(F)F c1(N(C(=O)C(c2ccccc2)O)C)cnc(N(C)CCC2CCNCC2)cn1 Cc1cc(Cl)cc(C)c1C(=O)NC1CC(CNC(C2CC(CC3CC3)C2)=O)C1 CC1CN(C(C2(C)CCCS2)=O)CC1CNC(c1ccc(C(F)F)nc1)=O c1(OCC(=O)NC2CCCN(C(c3n(C)nnc3)=O)C2)ccc2c(c1)CCC2 N(C(=NCCc1nc2ncccc2[nH]1)NC1CCc2sc(Cl)cc21)C1C(C)C1 C1(C)(CN(C)C)CCN(C)C1.c12nocc1C(=O)NCC1(CC1)C(=O)NC2C c1(C(=O)NCC(C)N(C(=O)C(C)C#N)CC)coc2ccc(Cl)cc12 C1(NC(c2cc(CCC)[nH]n2)=O)CCC(O)CN(C(c2nccc(Cl)c2F)=O)C1 CC1CC(=O)NC(C(N2CC(CNC(=O)CC3CCOC3=O)C(F)(CO)C2)=O)C1 c1(C(N2CCC3CN(C(C4C(=C)CC4)=O)CC3C2)=O)c[nH]c2cc(C#N)ccc12 N1(C(CC2(C#N)CCCCC2)=O)CC2(C1)CN(C(=O)Cc1csnn1)CC2CO C1(NC(c2nc(C(C)C)sc2)=O)CN(C(=O)C(C(C)C)NC(N)=O)CC1F N1(c2ccc([N+](=O)[O-])cn2)CCC2C(CCCN2C(=O)CC2CCCC2)C1 c1(OC)ccccc1C(C)N(C)C(C1CCN(C(=O)Cc2nc(O)n[nH]2)CC1)=O c1(C(N(CC(CC)NC(c2nc(CCC)sc2)=O)C)=O)ccc(N)cc1C c1(C(=O)NC(C(C)NC(c2cc(OC)n[nH]2)=O)C)cc(O)ccc1Cl Cc1ccc2c(C(=O)NCCC3CCCN3C(=O)C3=C(Cl)CCCC3)csc2c1 CC(=O)CCC(=O)NC12CC(NC(c3sccc3C)=O)(C1)C2 C=CCCC(C)C(C(=O)NC1(C)CC1)N(C)Cc1ccccc1Br C1(O)(C(C(=O)NCC(C2CC2)NC(C2C(C=C)OCC2)=O)(F)F)CCCCCC1 c1(C(C(=O)NC)N(c2c(OCCC)cccc2)C)cc(F)cc(Br)c1 N1(C(C2=CCN(C(c3ncc(OC)nc3)=O)C2)=O)CCOCC(C)(F)C1 c1(C(N2CC(NC(=O)C=CC3CCC3)C2)=O)cc(Cl)sc1Cl c1(C(C)(C)SC)cn(CCC(=O)Nc2cc(-c3ccccn3)on2)nn1 n1(C(C(=O)NCC(C)NC(C2CC3CC3C2)=O)C)cnc(C#N)n1 N1(N(C(C(C)SC)=O)C)CCOC(C)C1.c1(C)cn(CC(O)CC)nn1 c1(C(N2CC(N(C(c3ccc(COC(C)C)cc3)=O)C)C2)=O)nn(C)c(Cl)c1Cl N1(C(CCN(CCCCC)C)=O)CC2(CCC2NC(=O)Cn2cccnc2=O)C1 CC(O)(CNC(=O)COCCNC(C1CC(=C2CC2)C1)=O)C(F)F CC1CC(NC(c2cc[nH]n2)=O)CCN1C(=O)CCn1ccccc1=O C1(C(=O)NCc2nc(C(N)=O)on2)CCC2CCC1N2C(c1ccns1)=O C(CCN=c1cc(CCc2ccc(Cl)cc2)nc[nH]1)N(C)C(C1CC2CC2C1)=O Cc1ccc(SCC(=O)Nc2sc(C3CC3)nc2C)cc1.C12CN(CC1C)C2=O c1(CNC(CCC=C)CO)ccc2c(c1Br)OC(F)(F)O2 C(N=c1[nH]c2cc(F)ccc2o1)C1(NC(C(C)=C2CCCC2)=O)CCCCC1C Nc1cc(Cl)ncc1C(N1CC(F)(F)CC1CNC(C12CCCC1C2(F)F)=O)=O c1(CNC(C2C=CCCC2)=O)ccc(C(=O)NC(CC2CC2)C2CC2)cc1 C1(C2CC2)(CNC(CC(C)CN(C)C)=O)CCN(C(=O)CCc2ccsc2)C1 C1(CCOC)(NC(C2CCC(=O)NC2)=O)CCN(C(=O)CN2CC=CC2)C1 Cc1csc(CCCC(=O)NCCCN(C(=O)CCC2CCCOC2)CCO)n1 C1(NC(C(C)OCCOC)=O)CCCCN(C(=O)COCP(C)(C)=O)CC1 c1(OC)cccc(C(C)=CC(=O)NCC(C)N(C)C(c2cc3n(n2)CCC3)=O)c1 c1(C(N2CC(SC)C(NC(=O)Cc3nnc(O)s3)C2)=O)cc(NC=O)nc(Cl)c1 N1(C(CCNC(=O)NC)=O)CC2(C)CN(C(C3CC(C)CO3)=O)CC2(C)C1 Cc1cc(=O)oc(C)c1C(=O)NCC1CN(C(=O)COCC(C)C)C2CC12 N1(C(CC(C)CN(C)C)=O)CCCC(NC(=O)COc2cncc(Cl)n2)C1C c1(C(=O)NCC(C)(C2CC2)NC(CCCC#C)=O)ccc(C)cc1Cl Cc1cc(CNC(=O)COC2CN(C(=O)CC3CCC3C)C2)nn1C C1(C(N(CCNC(C(C(C)C)OCC)=O)C)=O)CCc2ncccc2C1 C1(OC)CCN(C(=O)CCCNC(=O)C(F)=CC2CC2)C1C(C)C C1(C(=O)NCCSCCC=C)CCCCCN1C(c1ccc(F)cc1C)=O Cc1noc2nc(-c3ccccc3)c(Cl)c(C(=O)NCC(O)CN3CCCC3)c12 O=C1NCC2CCCN(C(c3cc(-c4cccc(Cl)c4)no3)=O)C12 N1(CC)CCN(CC(=O)NN(C)C(C2(C(=O)NC)CCC2)=O)CC1.C12CC(C1)CC2 c1(C(=O)NC2CC(CCNC(c3cc(C(C)=O)sc3)=O)C2)n[nH]c2c1CC1CC21 C1(C(N(CCNC(C2N(S(CCC)(=O)=O)CCC2)=O)C)=O)CCOCC1(C)C c1(C(=O)NC2CC3(C(NC(c4ccc(CC)s4)=O)C3)C2)cc2cccc(Cl)c2o1 C1(NC(c2nc(OCC)sn2)=O)CC(NC(c2ccc(C3CC3)o2)=O)C(O)C1 N1(C(Cc2ccc(C#C)cc2)=O)C2CCC1CN(C(=O)CN(C1CCSC1)C)C2 C=CCC(CC(C)C)C(=O)NCC1CC1NC(c1cc(C)c(C)c(F)c1)=O N1(C(N)=O)CCCC(C(=O)NCCN(C(C2CC23CC3)=O)C2CC2)C1 C(N=c1cc(C)nc(N(CCCS(C)(=O)=O)C)[nH]1)C1CCC(COC)O1 C(CC(C)(C)NC(=O)CCc1ccc[nH]1)N(C)C(C1CC1C#N)=O n1(C(CC)C)ncc(C(=O)NC(CNC(c2cnc(C(F)(F)F)s2)=O)CC)c1C N1(C(C2CCC(C)C2)=O)Cc2occ(C(=O)NC3(CO)CCCCC3C)c2C1 c1(CC(=O)NCC2CCC(N(C(C)=O)C)CC2)cn(C)c2ccccc12 CCC(CC)CC(F)C(=O)NC(C(=O)NC1CCCC(O)C1)C1CC1 Cc1c(Cl)ccnc1C(=O)NCCC1CCCN(C(C2CCC2(F)F)=O)C1 CC1=C(C(=O)NCC2(NC(=O)CCc3cccc(O)n3)CCC2)CCC1 Cc1cc(C(=O)NCC#CCNC(c2occc2C(C)C)=O)ccc1[N+](=O)[O-] c1(C(=O)NC(C2CN(C(C3CCCN3C=O)=O)CCO2)C)ccc2cc[nH]c2c1 CCCCC(CC)CC(=O)NC(CC(=O)NC(C)(CO)CCF)C(F)F N1(C(C(C(C)O)C)=O)CCCCC(NC(C2CC=CCO2)=O)C1 c1(C(=O)NC(C2CCCN(CCOc3ccc(C)cc3)C2)C)cc2n(n1)CCOC2 c1(NC(c2c(CNC(CC3(C(=C)F)CCC3)=O)ocn2)=O)cc(OC)cc(O)c1 c1(C(=O)NCC2(NC(C(CC(CC)C)C)=O)CC2)ccc2c(c1)OCCNC2=O c1(CC(N2CCC(F)(CNC(c3ccsc3Cl)=O)C2)=O)ccc2c(c1)CCC2 C(=O)(CCC(=O)c1cccc(SCC2CC(C(N(C)C3CC3)=O)C2)c1)N.C1(OC)CC1 C1(S(C)=O)(CNC(C(C)N(C(=O)CC(Cl)Cl)C2CC2)=O)CC1 C1(CN(C(Cc2cc(C)sc2)=O)C)CN(C(C2CCCC(=O)N2)=O)CCO1 C#CCCCCCCC(=O)NC1CCC(CC(N2CCC(C(=O)OC)C2)=O)C1 C#Cc1ccc(C(=O)NCC2CCOC2C(=O)NCC2(C)CC=CCC2)nc1 CC1OC2(C(=O)NCCC3CCCS3(=O)=O)CC1(NC(=O)OC(C)(C)C)C2 N1(C(C2C(CC)N(C(=O)C(C)=C3CCCC3)CCC2)=O)CCCOC(C)(C)C1 C1(NC(c2cc(C3CC3)no2)=O)CCC(CNC(CCNC(=O)OC)=O)C1 N1(C(C2N(C(C)=O)CCC2)=O)CC2CCC1CN2C(c1ccc(C)c(F)c1F)=O C(C(CC(C)C)NC(=O)Cc1ccc(C(C)=O)s1)NC(c1ccc(CC)s1)=O c1(C(N(CC(CO)(CO)NC(c2c(C)ccnc2)=O)C)=O)ccc([N+](=O)[O-])s1 N#Cc1cc([N+](=O)[O-])cc(Cl)c1NC(C1CC12CCN(C(c1ncsc1Br)=O)C2)=O C1(NC(=O)C(F)CC2CC2)CN(C(=O)CN2CCS(=O)CC2)CC12CCC2 c1(CNC(C2CCC(NC(=O)Cc3csc(C4CC4)n3)C2)=O)cc(F)ccc1F C12(C(=O)NCC3CC(NC(=O)CC(c4ccc(Cl)cc4)O)C3)CCC(CC1)CO2 N1(C(C2CCC(C(C)C)CC2)=O)CCCC2CN(C(=O)C(C)(C)C)CCC12 C1(O)(C(C)NC(C2CCC(=O)O2)=O)CCN(C(C2(CO)CCCCC2)=O)CC1 CC1COCC(C(=O)NCc2ccc(C(=O)NCC3(Cl)CC3(F)F)nc2)O1 C1(NC(C(C2CC(C)(C)C2)NC(=O)Cc2ccccc2F)=O)C2CCCCCC12 Cc1cc(C)c(C(=O)NC2CN(C(C3CC3c3cnnn3C)=O)C2)c(C)c1 C(CC(=O)NC(c1csnn1)C)(C(C)C)NC(Cn1ncc(C)c1)=O C1(C(=O)NCC(CNC(C2(C)COCCO2)=O)OC)CC2(C1)CS(=O)(=O)C2 C1(C(=O)N(C(C)CCSC)C)(CC)CCCN(C(C2OCCC2(C)C)=O)C1 N(C1CCS(=O)(=O)c2ccccc21)C(C1=NOC(c2ccc(N)cc2)C1)=O C1(NC(c2c(C)n(CC(F)F)nc2)=O)CN(C(C2CCC2(C)C)=O)CCC1(C)C CCCC(CCC)C(=O)N1CCC(C(C)NC(=O)C(C)c2ccsn2)CC1 CC1(CNC(c2ccc(C3(F)COC3)cc2)=O)CN(C(C2CCCC2)=O)CCO1 c1(C(N2C(C(N(C)CC3CCCN3C)=O)C=CC2)=O)cc[n+]([O-])cc1 c1(C(C(=O)NCC(C)C)N(CCCC(C)C)C2CCCCC2)cc2n(n1)CCC2 c1(C(=O)NC2C(NC(c3ccc(C)o3)=O)C2)cn(-c2cccc(Cl)c2)nc1C c1(C(N(C(C)CN(C)C(c2cnn[nH]2)=O)C)=O)cccc2cncn12 c1(CC(=O)NC(C(=O)OC)Cn2cccn2)cc(NC(=O)CC#N)n(C)n1 c1(C(=O)NCC2ON=C(C)C2)ccc(OC(F)F)cc1F C(CN=c1nc[nH]s1)C1CN(C(c2cc(CC)ncc2)=O)CC1C C(N=c1[nH]c(=N)[nH]c(Cl)c1[N+](=O)[O-])C1C(C)CN(C(=O)CN2CCCNS2(=O)=O)C1 N1(C(C2CC3(CC(C#C)C3)C2)=O)CC2CS(=O)(=O)CC2(NC(=O)CC)C1 c1(C(N(C)CC2(OC)CCCC2)=O)cc2c(F)c(F)c(F)cc2[nH]1 CCCCCCCCNC(=O)C(C)C(C)NC(=O)Cc1ccc(O)cn1 CCC(CCC(=O)N1CCC(C(=O)NC2CCC(O)C2)O1)OC CCC(C)(C)C(O)C(=O)NC(c1cccc(C(F)F)c1)C(=O)Nc1cncc(Cl)c1 N1(C(c2cc(C)c(O)cc2)=O)CCCC(NC(=O)CC2CC2(C)C)CCC1 c1(C(N(CC(C)NC(C(COCC)C)=O)CC)=O)cc(Br)c(Cl)s1 N1(C(C(C)OCc2ccc(C)cc2)=O)CCC(NC(C2(C)CC(F)C2)=O)C(F)C1 N1(C(C2CN(C)C2)=O)CCC(NC(=O)Cn2cc(C#N)cn2)C(F)(F)CC1 N1(C(c2c(OCC)nccc2)=O)CCOC(C)(CC)C1.c12cc(n[nH]1)C(=O)NC2 c1(OC)cc(C)c(NC(C2CCN(C(=O)C(c3ccccn3)=O)C2)=O)cn1 c1(C(=O)NCC2CC(NC(C(C)N(C)C)=O)C2)ccc2nnn(O)c2c1 C1(NC(Cc2n(C)cnc2)=O)CCC(NC(=O)CCc2cscn2)CC1 C1(NC(=O)CCc2cccnc2)CC2CN(C(c3cc([N+](=O)[O-])n[nH]3)=O)CC2C1 c1(C(N2CC(=C(CNC(C3N(CC#C)CCC3)=O)F)C2)=O)ccc(C)nc1 C1(NC(C(CSC)C)=O)C2CCN(C(=O)COc3cccc(O)c3)CCC12 c1(CC)cnc(Cl)[nH]c1=NCCC1CCN1C(=O)C(C)CN(C)C N1(C(Cn2nc(C)oc2=O)=O)CC(NC(=O)C(C)C2CCOC2)CC2(CC2)C1 c1(CC)ccccc1C(CNC(=O)Cc1cnc[nH]1)NC(c1cc(Cl)n(C)n1)=O CC1(C)CC(C(N2CCC(=CCNC(C3CC3C(F)(F)F)=O)CC2)=O)CCO1 C1(CC)CN(Cc2cc(C)cc(Cl)c2)CCN1C(c1ccc(OC)c(I)c1)=O N1(CC(N2CC(CNC(C3(O)CC3)=O)CC23CCC3)=O)Cc2ccccc2C1 N1(C(c2n(CC)ncc2Cl)=O)CCCC(CNC(C2(C)CC2C(F)(F)F)=O)CC1 C(=O)(C(CC(C)C)C(N)=O)N(C1CCCN(C(=O)CCc2cc(C)[nH]n2)C1)CC C(=O)(CC(C)C(F)(F)F)NCc1occ(C(N(CCC)CC)=O)n1 N1(C(c2ccc(C)o2)=O)C2CCCC1CN(C(=O)CC1COC3CC1C3)CC2 C1(NC(CC2ON=C(C)C2)=O)Cc2ccccc2C1NC(c1ccc(Br)s1)=O Cc1c(Cl)ccnc1C(=O)N(C)CC1(NC(=O)C(C#N)C(C)C)CC1 c1(C2C(CNCC(C)CC3CC3)CC2)cccc(Cl)c1Cl C(=O)(C(C(CC)CC)OC)NC1CN(C(CCCC)=O)CC(C)C1 C1(NC(c2nc(C(C)C)sc2)C)CCC2(CC2)C1 Cn1cnc2ncc(C(N3CCC(CNC(=O)CC4=NNC(=O)C4)CC3)=O)nc12 CN1CCC(C)(C(=O)NC2CCCC(NC(c3cnoc3CC(N)=O)=O)C2)C1=O c1(OC(C)(C)C)ccc(-c2nc(-c3cscc3Cl)n(C3CS(=O)(=O)C3)n2)cn1 N1(C(c2cocc2Br)C(=O)NCCCC)CCOC(CN(C)C(C)C)C1 C1(C(N(C2CCNC2=O)C)=O)C2CC2CN1C(=O)CCn1ccnc1 N1(C(Cn2c(C)c(Cl)cn2)=O)CCC2(NC(c3cocn3)=O)CC2C1 c1(OC(C)C)ccccc1CSC(C)C(C)C.c1(S)nnc(-c2ccccc2)n1C Cc1c[nH]c2ccccc2c1=NCCN(c1cnn(C)n1)C C12CCC(=O)N(C1)C(=O)NCCCN2C.c1(OC)cccc(CC2CCCO2)c1 C1(O)(CNC(C(C=C)O)=O)CCCN(C(=O)CNC(=O)Nc2cccc(Cl)c2)C1 C1(C(N(CCN(C(C=CC(C)C)=O)C)C(C)C)=O)CCc2[nH]nc(O)c2C1 c1(C(N2C(CCNC(c3c(C)cccn3)=O)CCCC2)=O)ccc2ccoc2c1 N1(C(CC2(C=C)CC2)=O)C2CCC1C(C)C(NC(=O)CC(C)(C)CC(F)F)C2 N1(C(c2n(CC)ccn2)=O)CCC(C(C)NC(c2ocnc2C)=O)CC1 N1(C(COCC)=O)CCC2(CC1)CN(C(c1csc(C(F)F)n1)=O)CC2CO c1(C(=O)NC2(CN(C)C)CCC2)cnc(CNC(C2CCC(=O)NC2)=O)nc1 N1(C(c2ncn(C(C)C)n2)=O)CC(NC(C2(CC3CC3)CCC2)=O)CC(C)C1 C(=O)(C(C#N)C(C)(C)C)N1CC(C)(C(=O)NCC2N(C(C)=O)CCCC2)C1 c1(N(CCCNC(C(C)OCCC=C)=O)C)ccc2c(n1)CCC2=O CC(F)(F)CCC(=O)NCC(C)(C)NC(=O)CC1CNC(=O)C1 c1(C(N(C(C)CCNC(c2cnc(O)o2)=O)C)=O)ccc(F)c2cccnc12 C1(NCc2cc(C(=O)OC)[nH]c2)C2CCC(NC(C3CCCC34CC4)=O)C12 C1(NC(=O)C2=CCCC2)CCC2(CCN(C(=O)Cn3ncccc3=O)C2)C1 C1(NC(C(CCC)OC)=O)CN(C(C2CCC2)=O)CC1(C)C C(=O)(C1=Cc2ccccc2C1)NC(CN(C(=O)C1=CCCC1)C)(C)C C1(OCC#N)CCN(N2CCC2Cc2ccccc2Cl)C1 CCC(C(=O)N(C(C)CSC)C)Nc1ccccc1 N1(C(Cn2c(C)ccn2)=O)C(C)CN(CC2CCCC2(F)F)CC1C C1(O)(CNC(=O)Cc2cocn2)CCN(C(=O)COCCN2C(=O)CCC2=O)C1 n1(CC)nc(C)c(Cl)c1C(N1CCC(C)(CSC)C1)C(=O)Nc1ccccc1C Cc1cc(CC(N2CC(NC(C3C4CCOCC34)=O)CC2C)=O)cc(F)c1 N1(C(CSCC=C)=O)CCC(C(=O)NC2CC(C)OC2=O)C(C)C1 c1(CN(C(c2sccc2NCc2cccc(OC)c2)=O)CC)ccc(F)c(Cl)c1 N12CCC3(CC(C3)C1=O)CN2C(=O)Cn1cc(C)cn1.C(COC)OCC C1(C(=O)NCCOCCNC(C2CC23CCOC3)=O)OCC2CCCC12 Cc1cccc(N)c1C(=O)NCC1CCN(C(c2cc3sccc3[nH]2)=O)C1 N1(C(C(CC)=CCCC)=O)CCC(NC(c2cc(C(F)F)cc(F)c2)=O)C(O)C1 N(C1CCCc2c[nH]nc21)C(=O)NCc1ccc(N(C)CC)cc1 N1(C(C2(NC(CCC(C)SC)=O)CCSC2)=O)CCC(C)(C)C(CO)C1 c1(C(N2C(C(C)NC(=O)C3=COCCC3)CCC2)=O)cccc2c1COCCN2 CC1(CNC(=O)C(F)OC(F)(F)F)CC2(CCN2C(C2(CN)CC23CCC3)=O)C1 N1(C(C(C(C)C)NC(c2ncn(CC)n2)=O)=O)CCN2C(=O)NCC2C1 C1(NC(C(C)NC(N)=O)=O)CCC2CN(CCNc3ccc(Cl)c(Cl)c3)CC2C1 Cc1cc(C(N2CCC(NC(C3CN4CCC3CC4)=O)C(F)C2)=O)c(C)cc1Cl C=CCCCC(C)(C)C(=O)NOC(CC(C)C)C(=O)N1CC(=C)C1 c1(C(=O)NCCC(C)O)ccnc(CNC(C2CC2c2ccncc2)=O)c1 C1(COC)CN(C(c2sccc2CNC(C2OCCOC2C)=O)=O)C1(C)C C1(CC(N2CCC(OC3CN(C(C(C)OC)=O)C3)CC2)=O)CCN(OC)CC1 c1(C(=O)NCC(CNC(CC2CC(OC)C2)=O)O)cccc2ncn(C)c12 C1(C(N(C2CCOC2)CCOCCC)=O)COCCN(C(c2ccccc2)C)C1 CCCCC(C)CCC(=O)NCc1cc(C(=O)N(CCCC)CCC)n[nH]1 C1(NC)Cc2ccc(C)cc2S1.C1(CN(CC=C)C)CCN(C=O)C1 c1(COC)cccc(Oc2ccccc2)c1.C12CC1C(C)NC2=O C1(C(=O)NC2CC3CCC2N3C(=O)C(F)F)CCCC(F)(F)CC1 C=C(C)CCC(=O)N1CCCC1C(C)NC(=O)COCCCN(C)C C1(NC(c2nnn(C(C)(C)C)n2)=O)CC(C)N(C(=O)Cc2ccns2)C1 Cc1cccc(C)c1C(O)CNC(=O)C(F)Cc1ccc(Cl)c(F)c1 C12(C(=O)NC3CC(CNC(c4c(CC)cccc4)=O)C3)CCC(C(F)F)(CO1)C2 C1(OC)CN(C)C(C)(C(=O)NC2CN(C(C3(S(N)(=O)=O)CC3)=O)CC2C)C1 N1(C(C2(C)CS(=O)(=O)C2)=O)CCCN(C(C2CC23CC3)=O)C(CO)C1 Cc1cnc(C(=O)NCC2CC(O)CN2C(C2CCCCCC2)=O)c(C)c1 C(=O)(CCc1cnc[nH]1)N(CCNC(=O)COC1CCOC1)CC C1(CNC(CN(C(C)=O)C2CC2)=O)(CO)CCCN1C(c1cocc1C)=O c1(C(N(C2CCN(C(c3coc(C(F)F)n3)=O)C2)CC)=O)cc(C(C)C)on1 Cc1cscc1C(=O)NCC1CCC(NC(C2CC2c2ccncc2)=O)C1 C(=O)(C1=CCCCCC1)NC1C(NC(c2nc(OC)oc2)=O)CC1 C12(CC(=O)NCC3(CCNCc4nc(CCC(=O)C5CC5)on4)CC3)CCCC1C2 C(=O)(CCC(N)=O)N(CC(C)C(=O)N1CCC(OCCF)C1)C c1(C(=O)NC2CCC(F)(C(=O)OC)C2)cc2c(Br)coc2cn1 Cc1ncc(NC(C2CSCCN2C(c2cnc(C(N)=O)cn2)=O)=O)c(C)n1 C(=O)(C(F)(F)C(F)(F)F)N1CC(C)(C)C(CNC(c2ccn3cncc3c2)=O)C1 C(=O)(C(C)(C)C1=CCN(C(c2ccoc2)=O)C1)NC1CCN(OC)CC1 CC1(COC(C2CNCC2OCc2ccccc2)=O)CCCOC1 C(=O)(CCCCC(F)(F)F)NCC1N(C(C(CCCOC)C)=O)CC2(CC2)C1 Nc1ccc(O)c(C(=O)NC2CCCCN(C(c3ccc(C4CC4)cn3)=O)C2)c1 C(CS(=O)(=O)c1ccccc1)NC(=O)NCc1oc2ccccc2c1Br N1(C(C23C(CN(C(c4sccc4F)=O)C2)COC3)=O)CCC2(CCCOC2)C1 c1(CC)nc(C)c(C(=O)NCC2C(C)CCN2C(=O)Cc2ccn(C(C)C)n2)s1 c1(N(C(C)CNC(=O)CC2(N(C)C)CC2)C)nccc(-c2ccccc2)n1 c1(C(N2CC(NC(=O)CCP(C)(C)=O)CC(OC)C2)=O)cnc2[nH]ncc2c1 c1(C(=O)OC)c(NC(N2CCOCC2C(c2cccc(C)c2)O)=O)cccc1F C(c1ccc2c(c1)OCO2)=CC(=O)NC(CCNC(CN(C(=O)OC)C)=O)C C1(NC(=O)CCNc2ccccc2)CN(Cc2cc(Br)c[nH]2)CCC1F c1(C(N2CCC(NC(C34CC(C)C3C4)=O)CC2C)=O)cc(Cl)c(Cl)cc1O c1(C(=O)NCC2CCCN(C(CC3ON=C(CC)C3)=O)C2)ccc2nn[nH]c2c1 c1(C(N2CCC(NC(Cc3cc(C)[nH]n3)=O)C2)=O)nccn2c(C)nnc12 c1(C(=O)NC(CC)CNC(c2sc3ccccc3c2C)=O)cc2c(C)cccn2c1 C(=O)(C(C)CC(=O)OC)NC(CC#C)C(=O)NC(C)CC(C)C CCN1CCCCC(=O)NS(=O)(=O)C2CCN1C2.c1(NC(C)C)cccnc1 CC1CN(C(=O)C(C)P(C)(C)=O)CC2(CCN(C(=O)C(C)(C)CS(C)(=O)=O)C2)O1 c1(OC)ccccc1-n1ncc(NC(=O)C(C)C2CC2)c1C1CC1 C1(NC(c2ccc(CSC)o2)=O)CC(C)CN(C(=O)C(C)=C2CCCC2)C1 c1(OC)cccc(C(=O)C(=O)NCc2noc(-c3ccc(Cl)cc3)c2C)c1 c1(C(=O)NCCCNC(C(c2ccccc2)SC)=O)c(O)cnc2ccc(Cl)cc12 N1(C(c2n(C)nc(C)c2Cl)=O)CCOC2(CCN(C(=O)CCCC(C)C)C2)C1 c1(C(=O)NC2CCN(C(C(CC)(C)CC)=O)CC2CO)scc2c1OCCO2 S(=O)(=O)(c1[nH]c(=NC2CN(CCN(C)C)C2)ccc1Br)N(C(CC)C)C C1(NC(C23CC(C(=O)OC)(C2)C3)=O)CCCCN(C(=O)C(C2CCCCC2)=O)C1 c1(C(=O)NCCOCCCNC(c2c(CC)ocn2)=O)ncccc1C(=O)OC c1(C(=O)NCCc2cn(-c3ccc(C)nc3Cl)nn2)cccc2c(Br)cccc12 C1(C(C)CNC(C2(F)CC2)=O)CCN(C(c2ccnn2C2CCC2)=O)CC1 C1(O)(CNC(C(CNC(c2ccnn2C2CC2)=O)OC)=O)CCOCC1 c1(C(=O)NCCC(COC)O)ccnc(CNC(c2[nH]nnc2C)=O)c1 C1(C(N2CCC(C(=O)NC)CC2)=O)C(C)OCCN1C(=O)CSc1cn[nH]c1 CN1CCCC(O)(CC(=O)NC(C)(C)CCCNC(c2ccnn2C2CC2)=O)C1 C(=O)(CS(=O)(=O)CC)NCC1(C)N(C(c2c(CCC)[nH]cc2)=O)CCC1 c1(C(=O)NCC(CN(C(C(C)Cn2ccnc2)=O)C)O)cc2c(nn1)CCCO2 c1(C(=O)NC2CCC(NC(C3CN(C)C3)=O)C2)cccc(SC(F)(F)F)c1 C(C)(C(=O)NCC(CO)NC(c1csnn1)=O)N(C(C)=O)C N1(C(CC(C=C)(C)C)=O)CCC2(CC1)CC(CNC(=O)CC(=C)Br)C2 C1(NC(COC(CNC(c2c(CC)cncc2)=O)(C)C)=O)CCC2CCCC1O2 Cc1ccc(C(=O)NCC2CCN2C(c2sc(C)c(C)c2C)=O)cc1F c1(CN=C(NC(C)C)NCC2CC(CC3CC3)C2)c(OC(F)F)cccc1Cl N1(C(Cc2c(C)cccc2)=O)CCC2CN(C(=O)CC3CC3)CCC2C1 c12nc(co1)C(=O)N2.C1(NC(CSCCN(CC)CC)=O)CC(CC(F)F)C1 N1(C(c2c(C)ncc(N)c2)=O)CCC(C)N(C(C2CCC(C(F)(F)F)O2)=O)CC1 n1(CCN(C(=O)NCC(=CC(=O)OCC)C)C)ncc2ccccc12 c1(C(=O)NC2CCC2NC(c2csc(CO)n2)=O)cnc(O)c([N+](=O)[O-])c1 CCCC(C)(O)C(=O)NCCC1C(C)CCCN1C(c1sc(C)cc1OC)=O C1(NC(c2ncccn2)=O)(CO)CCN(C(c2cc(Cl)nc(Cl)c2)=O)CC1 c1(N2C(C)CC(NC(c3csnn3)=O)C2)c([N+](=O)[O-])ccc2nsnc12 Cc1nc2ccccn2c1C(=O)Nc1nc(C(F)(F)F)ccc1Cl C1(N(C(C=CSC)=O)CCOC)CCN(C(=O)CCCc2ccccc2)CC1 C(=O)(C1=COCC1)NCC.C(C(C)(O)COCCNC(C1CC(OCC)C1)=O)N c1(C(=O)NC(C(=O)N(CC(O)C(F)(F)F)C)Cn2ccnn2)cc(F)cnc1O Cc1cnc(C(=O)NC2CC(CNC(=O)C(C(C)C)NC(N)=O)CC2O)cc1Cl CC(C)CCC(=O)NOCC(=O)N(C)Cc1ccn(C)n1 c1(C(N2CC(CCNC(C(C(C)(C)C)CO)=O)C2)=O)cc(N)cc(S(C)(=O)=O)c1 C(C1CCCN1C)=CC(=O)NCC(C)CN(C(=O)Cn1nnnc1C1CC1)C1CC1 c1(C(=O)NC2CC(NC(c3cc(C)c(Br)o3)=O)C2)cncc2c1CCC2 N1(C(C(C2CC2)OCC)=O)CCCC(C2CCN(C(c3cnsn3)=O)CC2)C1 c1(CC(=O)NC23CC2CN(C(C2(CF)CCOCC2)=O)C3)cnc2cccnn12 C12(C(N3CC4(CC(=O)N4)C3)=O)CCCC1N(C(c1csc([N+](=O)[O-])c1)=O)CC2 C1(C)(CC)C=C(C(=O)NC2CC(NC(c3cccc(OC)c3Cl)=O)C2)C1 C1(CNC(=O)OC(C)(C)C)Cc2c(F)ccc(F)c2CN1C(CC(CCC)(C)O)=O N1(C(Cn2c(C)ccn2)=O)CC2CCC(C1)N2C(=O)CC1CC(OC(C)(C)C)C1 CN1C2CCC1CN(C(C13CC(NC(=O)CCCC(F)(F)F)(C1)C3)=O)C2 c1(CSc2n(CC)c(C)nc2)cc(Br)ncc1F N1(c2ccnc(CC)n2)CCCC(CNC(C2C3COCC23)=O)CC1 C(=O)(C(CC(=C)C)NC(=O)NC)C1(F)CC(NC(CSCC=C)=O)C1.C1(N)CC1 C(CC(C)C(=O)NCCOCCCN(C)C(c1ccc(C(C)F)cc1)=O)OC Cc1ccc2sc(C)c(C(N3CC(CNC(C4(C)CC4)=O)C4(CCC4)C3)=O)c2c1 CCCC(CC(C)C)C(=O)NC1C=CC(C(=O)NCCOc2ncccn2)C1 N1(C(CCCNC(CC2(N(C(C)=O)C)CC2)=O)=O)CC(C)(C)C1CN(C)C c1(NC(C2CC(NC(C3C(C)(C)C3)=O)C2)=O)ccc(C(F)(F)F)nn1 C1(CNC(=O)CCNC(C2CCC2)=O)CC(C)N(C(c2nc(C)sc2)=O)C1 C1(NC(C2CCN(C)S2(=O)=O)=O)CN(C(=O)CO)C2(CCCC2)C1 c1(N(C(C(C)(C)NC2CC(OC)C2)c2nn[nH]n2)C)ccc(C)c(C(N)=O)c1 c1(NC(C)=O)ccc(-n2nc(-c3ccc(C)o3)nc2Cc2cccc(Cl)c2)cc1 c1(OC)cc(N)cc(C(N2CC(C)C(NC(=O)CCC(N)=O)C(C)C2)=O)c1O CC1(C)CCCN(c2ccc([N+](=O)[O-])cc2)C1CNC(=O)CCCC1CCCC1 N1(C(C2(CCNC(CC3(C)CCC3)=O)CCC2)=O)CCCN(CCN(C)C)CC1 c1(NC(C2CCCN(C(c3nc(Br)cs3)=O)C2)=O)c(I)cc([N+](=O)[O-])cc1I C=CCC(CNC(=O)CC1COCCO1)C(=O)NCC(CC)(CC)OC C1(C(=O)NC(CC)C(F)(F)F)CCN(C(=O)C=C2CCOCC2)CC1C N1(C(COC(C)C)=O)CC2CC(NC(=O)C(C)NC(=O)OC(C)(C)C)C2C1 CC1CCCCC1N=c1[nH]c2c(c(=NC3CCN4CCCC34)[nH]1)COC2 N1(C(CC=C)=O)CCCC(O)(CNC(c2sc(=N)[nH]c2CC)=O)C1 C(=O)(N=c1ccc(N2CCN(C)CC2)n[nH]1)Nc1n(CC)nc(C)c1Cl N1(C(C(C(C)C)C)=O)CCC(NC(=O)C=Cc2ccccc2Cl)C(C)C1 c1(SCC(=O)NC2C(CNC(C(C)(C)N3CCOCC3)=O)C2)c(Cl)cccc1Cl CC#CCCC(=O)NC1CN(C(c2occ(C)c2C)=O)C1 c1(OC)ccccc1CC(=O)NCC(C1CCN(C(=O)CCCSC)CC1)C N1(C(C2(C)CCSCC2)=O)CCC2(CC1)CC2C(=O)NC1CC(C#N)C1 N1(C(C2(C)CC3(CC3)C2)=O)CCCCC(NC(=O)Cc2nc[nH]n2)C1 CC1(C)CC(NC(c2ccnnc2)=O)CN(C(C2CCS(=O)CC2)=O)C1 c1(OC)sccc1C(=O)NC(C(=O)NCCCc1nncs1)c1ccoc1 N1(C(Cn2c(=O)sc(C)c2C)=O)C2CCC1CC(CNC(c1cc(F)c[nH]1)=O)C2 CCC(CC)CCC(=O)NCC1CCC(C(N2CC(O)CC(O)C2)=O)CC1 S(=O)(=O)(c1cc(Cl)ccc1C#N)NCC(C)CNC(N)=O CC1CN(C(c2cc(C(N)=O)no2)=O)CC1CCNC(c1cnn(C2CC2)c1)=O c1(C(=O)NC2C3CN(C(=O)C=Cc4cscn4)CC23)cccc2nccn12 c1(NC(C(COC)NC(=O)C(c2ccn(C)c2)C)=O)ccc(CO)nc1 N1(C(c2c(CNC(c3c(CC)ocn3)=O)c[nH]n2)=O)CC(C)C12CCOCC2 C1(CNC(C2C(NC(CCNC(C3C(C)C3)=O)=O)C2)=O)CCCC(C(C)(C)C)C1 CC1CCCC(CNC(c2cc(CNC(c3cocn3)=O)cs2)=O)CC1 c1(C(=O)NCC(C)CNC(C2(C)CC(=O)N(C)C2)=O)ccsc1S(C)(=O)=O c1(C(=O)NC2(C)CC(NC(c3ccc(CC)o3)=O)C2)ccc(-n2cncn2)cc1 C(=O)(CCC(C)(C)C#N)NC(C(C)NC(CCc1onc(C(C)C)n1)=O)C(C)C C1(NC(C=Cc2n(C)ncc2)=O)CN(C(=O)Cc2ccsc2Cl)CCC1CO C1(CCNC(c2c(COC)ccs2)=O)C(C)CCCN1C(c1ccnn1C)=O c1(CNC(=O)NC2CN(C)C(=O)C2)ccc(Br)c(Br)n1 c1(C(C(=O)NCCN(C(C2(C)CC2C(F)(F)F)=O)CC)=O)cc(Br)co1 C(=O)(C#Cc1ccccc1)N1CCC(Nc2ccnc(SC)n2)C1 C1(NC(=O)Cc2ccccc2Cl)CCCC(NC(=O)CN2CCCCC2=O)C1 Cc1nc(C=CC(=O)NC(C)C(C)NC(C2(C(C)(F)F)CCOCC2)=O)[nH]c1C C(=O)(CC(C)N1CCCC1=O)NC1CCN(C(n2cc(C3(O)CCC3)nn2)C)C1 N1(C(c2c(OC)ccs2)=O)CCCC1(C(=O)NC1C(C)CCC1C)C(C)C N1(CC)CCCC(C(N2CCC(CNC(=O)CO)(OC)C2)=O)C1 N1(C(c2cn(CC)nc2)C(=O)NCC2CCOCC2)CCC(C2CCOCC2)C1 CC1CC(C(=O)NCC2(C(N)=O)CCCC2)CN(C(c2ccnc(O)c2F)=O)C1 N1(CC=C)CCC(C(N2CCC2CNC(c2[nH]c(C)nc2C)=O)=O)CC1 C1(O)(CNC(c2c(C)nco2)=O)CCCN(C(=O)C2=CCCCC2)C1 C1(CN(Cc2n(C)ncc2)CC2CCCCC2)CCC(C)(C)O1 c1(C(C(=O)NCC(N2C(C(C)F)CCC2)=O)(C)C)ccc(Br)cc1 N1(C(C2CN(CC)C(=O)CC2)=O)CCC(O)(N(C)C(C2CN(CC)C2)=O)CC1 c1(OC)c(Cl)cc(C(N2CC(Cc3ccc(C#N)nc3)C2)=O)cc1Cl C(C1=CCN(C(=O)C(C(C)C)c2cnn(C)c2)CC1)NC(C(COC)O)=O c1(C(=O)NCCCNC(C2(COC)CC2)=O)cc(C(F)F)cs1 CC12CCCC1N(C(=O)C1=CCCS1)CCN(C(c1cnc(C3CC3)o1)=O)C2 c1(C(CNC(C2CC(O)C2)=O)NC(c2nc(CCC)sc2)=O)ccc(C)cc1 c1(C(=O)NCC2CC(NC(C=CC)=O)C23CCC3)c[nH]c2cc([N+](=O)[O-])ccc12 Cc1cc(F)ccc1C(=O)NCC1CN(C(=O)C(C)(C)CN(C)C)CCC1C N1(C(c2noc(CC)c2C)=O)CC2(CCN(C(=O)CCc3ccccc3O)C2)C1 N1(C(c2cn(C(C)C)nc2)=O)CCC(CN2CC(Cc3ccco3)C2)C12CC2 C1(C(=O)NC23C(=O)NCC2C3)CN(C(=O)C(O)C2CCC2)CC12CCC2 N1(C(c2cncc(COC)c2)=O)CC(NC(=O)C(C)(O)C(C)C)CC12CCC2 c1(N(CC(=O)NCC=C)C)nc(N2CCC(C)C(C)C2)nc2ncn(C)c12 C(=O)(C(C)(C)CCCO)N(C1CCCN(C(c2ccc(C(F)F)o2)=O)CC1)C CN1C(C(N2CC(F)CC2CNC(=O)COc2ccccc2O)=O)CCS1(=O)=O C1(C(N(CCCNC(=O)C(O)C(C)(C)C)CC)=O)CCCCN1S(N)(=O)=O c1(C(N2C(C)(C(=O)NCC(C)(C)CO)CC2)=O)ccc2nccnc2c1 c1(C(=O)NC2CCC(CNC(C3(C=C)CCC3)=O)C2)cc2c(F)ccc(Cl)c2[nH]1 CC(C(F)(F)C(F)(F)F)=CC(N1CC2CCCC2(NC(c2csc(C)c2)=O)C1)=O c1(CNC(N2CCCC(c3ncc(C(=O)OC)s3)C2)=O)cn2cc(Cl)ccc2n1 C1(C(=O)NCCCNC(=O)CC)(NC(=O)OC)CCC(Cc2ccccn2)CC1 C1(O)(C(C)NC(C(C(C)C)C)=O)CCN(C(C2CNC(=O)O2)=O)CC1 c1(C(=O)NC2CCCN(C(CC3C(C)(C)C3(C)C)=O)C2)nccc(C#N)c1F CCC(CNC(c1ccc(C#N)s1)=O)(CC)NC(=O)C(F)CC1CCC1 C1(CC(N2CCC(C)C2)=O)CCC(=O)CC1.C(CN)(C1CCC1)N(C)OC N1(C(C(C)N2CCC2)=O)CCC2(CCOCC2)C(CNC(=O)C(C)N(C)C)C1 C1(CC)(CNC(C2(CCNC(=O)CC(C)N(C)C)CCCC2)=O)CCCO1 C(CCCOC)(C(=O)Nc1cncc(O)c1)NC C1(CC2N(CC3CCC(C)N3C)CC2)CCCCN(C(=O)C(c2ccco2)C)C1 N1(C(CCc2cc(C)no2)=O)CCN(C(=O)CCN(C)CCO)CC1C(C)(C)C c1(-c2nc(CCCOC)nn2Cc2cc(F)ccc2Cl)cn(C)c(=O)n1C c1(CCC)cc(=NC(=O)C(=O)N2CCCCC2C)[nH]o1 CC(CC(=O)N(C(=O)C(F)Cc1ccccc1)C1CCC1)c1cnc(=N)[nH]n1 C1(CNC(c2cc(C(C)=O)on2)=O)CN(C(C2(CO)CC2)=O)CCC1C(F)(F)F C#Cc1cc(Br)ccc1NC(=O)CCCSC1CCCC1(F)F C1(C(=O)OC)CC12CCN(C(=O)C=CC(C)(C)SC)C2 C(=O)(NNc1c(Cl)cccc1Br)C1C(CC(C)C)CCC1 S(=O)(=O)(c1cc(Cl)cnc1N)NC(c1cccc(C(=O)OC)c1)C Cc1ccc(CC(=O)NC(C)C(C)(C)NC(C2CC(F)C(=O)N2)=O)cc1Br C(=O)(C1Cc2ccccc21)CC(O)CF.c1(NC)ccc(Br)c(S(=O)(=O)N)n1 C(=O)(C1CCCc2scnc21)NC1CN(C(c2ccc(C#N)[nH]2)=O)C2(C1)CCC2 N1(C(C2(C#N)CC2)=O)CC(NS(=O)(=O)CCCCCl)C(F)(F)C1 CCC(C)CC(C(=O)N(C(C)C(=O)NC(C)C)C)NC(=O)C(CCOC)OC c1(CC)nc(O)c(C(=O)NCC2(O)CN(C(=O)C(O)Cc3cnc[nH]3)C2)cc1C C1(CC)C(NC(C2CCC(=O)N(C)C2)=O)CCCN1C(c1ccnnc1)=O c1(CCC)ccc(C(=O)CCC(=O)N(C)CCNC(C2C=CCC2)=O)cc1 c1(NC(c2cc(C#C)cc(Cl)c2)=O)nc2cc(C)cc(C)c2[nH]1 CC1(C(N2CCCC(Cn3cc(-c4cncnc4O)nn3)C2)=O)COCCO1 c1(C(=O)NCC(C)(C)CNC(C2CCC3CC3CC2)=O)cc(Br)cnc1N N1(C(C2(C)CN(C(C(CO)OC)=O)C2)=O)CCc2ccccc21 CC1(CO)CC(NC(C2CCN(C(C3(C(=O)NCC4CC4)CCC3)=O)C2)=O)C1 N1(C(C2OCCN(C(c3n(C=C)ncc3)=O)C2)=O)CCC2CCCC12 c1(NC(c2n(CCC)nnn2)c2ccccc2)ccc(OC(C)C)c([N+](=O)[O-])c1 C(=O)(CC(O)CC(C)C)N(CC(=O)NCc1cccnc1O)CCC c1(OC)cc(C(=O)NC2CC2C(N2CCC(O)C2)=O)cc(OC)c1Br C(CCC(C)(C)C(=O)N1CC(C)(C)C1)n1cc(C2CN(C)CCO2)nn1.CS Cc1ccccc1Cc1nc(C2CSC2)nn1-c1ccccc1 C1(COC)CN(C(=O)CCCCN(C(=O)C(C2CCCCC2)O)C)CCO1 c1(NC2(c3n(CCC)nnn3)CC(C[Si](C)(C)C)C2)cccc2c1OCCC2 N1(C(CC(=C)Br)=O)CCC(SC(C(=O)NC(C)C)C(C)C)CC1 CC(CS(N)(=O)=O)NC(=O)C(=O)NCC1CCCN(Cc2cccnc2)C1 C1(C(=O)NC2CCC(NC(=O)C(C)OCC3CC3)C2)(CC)CC(C)(C)C1 Cc1cc(C(N2C(C(=O)NCc3ccc(Cl)cc3F)CC3CC23)=O)cc(C)c1F C1(CCNC(CC)C(C)c2nnnn2C2CCCCC2)CCCC12CC2 Cc1ccc(CSCC(=O)NCCC(C)NC(=O)C=Cc2ccccn2)cc1 c1(C(=O)NC2CC(CNC(c3c(C)cnn3C)=O)C2)cnc2scc(C)n12 N1(C(C(C(C)C)C)=O)CC2(C1)CN(C(=O)C=Cc1nnc(C(C)C)o1)CC2CO C(=O)(C(O)(C(F)(F)F)C1CC1)NCCCN(C(C(CC)NC(N)=O)=O)C(C)C N1(C(CCCOC)=O)CCC(Cc2cn(C(C)(C)C)nn2)C(F)(F)C1 C1(C(=O)NCc2cccc(I)c2)CC2(C1)CC(n1cc(-c3cccnc3)nn1)C2 c1(CC)ccoc1C(=O)NC(C)CC(C)NC(c1cc(C)co1)=O C1(C(=O)NCC2CCCC(NC(C(C=C)(F)F)=O)C2)CC2(CC2)CN1C N1(C(c2cc(CCC)[nH]n2)=O)C2CCC1CN(C(=O)Cc1ccn(CC)n1)CC2 N1(C(CCC(C)C)C(N)=O)CCCOCC1(C)C C=CC1(C(=O)NC2C=CCN(C(=O)COCCCOC)C2)CCCCC1 N1(C(C2N(CC)CC2)=O)CC2CC2(C(=O)NC2COC(CN(C)C)C2)C1 C1(C)(CNC(c2onc(C)c2C)=O)CCCN(C(=O)CCC2CC2(C)C)C1 C1(C(=O)NC2CCC(O)CC2)(CC)CCN(C(c2cc(Cl)no2)=O)C1 C12(NC(CC(CC)NC(=O)CN3CCOCC3=O)=O)CC1COC21CCC1 C1(C2(N(CCC(=O)NS(C)(=O)=O)C)CC2)CCCCO1 C1(C(=O)NCC(c2cccnc2)O)(CC)CCN(C(C2CCOC(CC)C2)=O)C1 c1(OC)ccc2c(C(=O)Nc3[nH]nc([N+](=O)[O-])c3Cl)c[nH]c2n1 N1(C(Cc2cc(C)sc2)=O)CC(CCNC(C2CC3(C2)CC3F)=O)C(C)C1 C1(CNC(c2cncn(C)c2=O)=O)N(C(=O)CC2(C(F)F)CC2)CCCC1(C)C CC1(C)C(O)C2CCCN(C(c3ccncc3)C(=O)NC3CCC3)C12 C1(CC)CN(C(=O)Cn2nc(O)ccc2=O)CCC1NC(C1(CC)CCCC1)=O C(=O)(C(CN(C)C)N1CCC1)NC(CN(C(COCC)=O)C)C.C1(N(C)C)CC(CF)C1 c1(OC)ccc(CO)cc1NC(=O)CC1COCCN1C(=O)CCCCBr C=CCCC(C)(C)C(=O)NCCC1CC(NC(c2cc(N)c(F)c(F)c2F)=O)C1 c1(C(=O)NC2CC(NC(C3C(COC)C3)=O)C2)cccc2c1OC(F)(F)O2 C1(NC(=O)C2=CSCS2)CCOC12CCN(C(C1CC(C3CCCC3)C1)=O)CC2 C1(CC(=O)NCC2CCCC2NC(c2cc(Cl)cs2)=O)CCCS(=O)(=O)C1 N1(CC(=O)NCC2CCN(c3nc(SC)nc(N)c3)CC2)C(=O)NC(C)(C)C1=O c1(OCC(=C)C)cccc(CN2CC3C(C(=O)Nc4nc(C#N)cs4)C3C2)c1 c1(OCC)nc(C)ccc1C(N1C(CNC(=O)CC(C)(C)F)CC2CC12)=O C(=O)(CC(C)(C(F)F)N(C)C)N1CCC(CNC(C(c2ccc(CC)s2)=O)=O)C1 C#CCC(C(=O)NCc1ccc(C(=O)NCCC(=O)NC2CC2)s1)C1CC1 C1(C(N(CCOCC#C)C)=O)(CC)CCCN1C(=O)CC1CC1C1CC1 N(C1CCCc2occc21)C(c1c(CNC(CC2CCN(C)C2)=O)cc[nH]1)=O C12(CNC(CN(c3ccncc3)C)=O)CC1CN(C(c1n[nH]cc1C1CC1)=O)C2 c1(CCCO)ccc(-c2cnn(C(=O)NCCn3c(C)ncc3)c2)c(F)c1 C(C(C)C(=O)NC(C1CN(C(c2c[nH]nc2C(F)F)=O)C1)C)OC C1(COC)(NC(=O)C=C2CC2)CN(C(c2ccccc2)=O)C1 C(c1cc(F)c(O)c(F)c1)=CC(=O)NC(CNC(C(C(CC)O)C)=O)(C)C(C)C Cc1ccc(C(C)C)cc1C(=O)N(C1CCN(C(=O)C=Cc2ccccc2)C1)CC N1(C(CCC(CC)OC)=O)CC2(CCC2)CC1CNC(=O)C(CC)SC C1(C2(O)CN(C(c3nn[nH]c3Cl)=O)C2)(CNC(=O)CC2CCOC2)CC1 C(C)(C)(CCCNC(=O)Cn1c(C)csc1=O)NC(C(c1cc(C)sc1)(C)C)=O C=CC(CC)CC(=O)N(C(C)C(=O)N(C)CCc1cccnc1)C1CC1 C=C(C)CC(C(=O)NCC1(OC)CCC(C)C1)NC(=O)C(C(C)C)SCC C1(C(N2CCC(N(C(c3scc(C)c3)=O)CCO)C2)=O)C(C)(C)OC1(C)C CCC(C)(C(=O)NC(CNC(c1cnc(CC(C)(C)C)s1)=O)C(C)C)C(N)=O C1(C)(NC(C(CCOCCO)NC(C2(F)C(C)(C)C2(C)C)=O)=O)CN2CCC1CC2 c1(C(CC)C(=O)NCC(O)CCNC(c2cncn2C)=O)c(C)noc1C C(C)(CN=c1[nH]cnc2[nH]ccc12)(CC(C)C)NC(Cn1ncc(C)c1)=O N1(C(c2cc(CC)ncn2)=O)CC2CCN(C(=O)C=C=C(C)C)CC12 CC1=C(C)CC(C(=O)N(CC(C)(C)CNC(c2cnnc(O)c2)=O)C)CC1 c1(C(=O)Nc2ncc(-c3c(C)ccs3)s2)ccc(C(C)O)cc1 CN1CC(C(=O)NCC2CCN2C(=O)CCc2cc(Br)sn2)OCCC1=O c1(COC)ccccc1NC(=O)N(C(C)Cc1ccccc1F)C S(=O)(=O)(c1cccs1)NCC(=O)NCC1N(C(c2c(OC)c(C)sc2)=O)CCC1 c1(C(=O)NCC2N(C(C(C)N(C(C)=O)C)=O)CCCC2)ccc2ncccc2n1 c1(C(=O)NC2CC(F)(CNC(=O)COC(F)(F)F)C2)ccccc1-n1cncn1 CC(C)C(F)C(=O)N1CCC(C)(NC(=O)Cc2cncn2C)C1 C1(NC(C2CCN2C(c2cccnn2)=O)=O)CC12CCCCCC2 Cc1c(C(=O)NC2CC3(C2)CN(C(C24CCCCC2C4)=O)C3)nn2c1OCCC2 c1(CC(N2CCC(C)(CNC(c3ccnn3CC#N)=O)C2)=O)cc(O)nnc1O C(=O)(C1=CS(=O)(=O)CCC1)NC(CCNC(C(C)Sc1nncn1C)=O)(C)C C1(NC(C(CCSC)O)=O)CCSC12CN(c1nc(C)cc(C)n1)C2 Cc1ncc([N+](=O)[O-])n1CC(=O)NC1CC(NC(=O)C(C)P(C)(C)=O)C1 c1(C(=O)NCC2(NC(c3ccn(C(F)F)n3)=O)CCCC2)c(Cl)cccc1Cl C(C(F)(F)F)=CC(=O)NC(CNC(COCC=C)=O)C c12ocnc1C(=O)N1CCCC1C2.c1(C2C(C(C)(F)F)C2)cn(CC(C)(C)O)nn1 C1(F)(C(=O)NC(c2c(C)ccnc2)C)CCN(C(C2(C)CC(C)(C)C2)=O)CC1 N1(C(CNC(c2ccsc2)=O)=O)CCC2(CCCCN(C(c3csc(O)n3)=O)C2)C1 N1(C(CN(c2ccccc2)C(C)=O)=O)C(CNC(=O)CCSC)CC2COCC12 N1(C(C(C=CCCC)O)=O)CCC(O)(C2CCN(C(C3CN(C)C3)=O)CC2)CC1 C1(CNC(=NCC)NC2CCN(C(C)=O)CC2)CCc2nnc(NC(C)=O)n2C1 C1(C(=O)NCc2cnc(C)s2)CC(O)CCN1Cc1cccc(F)c1Br C1(CNC(CN(CCC#C)C)=O)CCCC1C(=O)NCCCc1ccncc1 N#CCS(=O)c1ccc(C(=O)NCC(O)CNC(c2csnc2Cl)=O)cc1 C(CC(C)C)(C(=O)NCc1nn(C)cc1C)N(C(COC)=O)C C(=O)(C1=CCCCCC1)NC(CC(C)C)C(=O)NCCCC(C)(C)O N1(C(c2snc(C)c2N)=O)CCC(C(=O)NC(c2ccccn2)CO)C(C)C1 C1(NC(c2nc(C)oc2)=O)CC2CC1N(C(C1(CO)CCC1)=O)C2 c1(OC)ccc(Cl)c(C(N2CCC2CNC(c2cscc2F)=O)=O)c1N N1(C(c2ccc(C#C)cc2C)=O)CCC2(CCC2)C(NC(C2CCOCC2)=O)C1 c1(C(N(CCCNC(CC(C)(C)SC)=O)CCO)=O)cnc2cc(C)nn2c1 N1(C(C2C(c3ccc(C)o3)C2)=O)CCC2CN(C(=O)C3=COCCO3)C2C1 c1(C(=O)NCC(C(=O)NC(C(=O)NC)CC2CC2)C)nc(C)ccc1C c1(C(=O)NCC(CC)(C)NC(C2CCC=CCC2)=O)ccc(CO)nc1 c1(C(C23N(C2)C3)=O)cccc(C(N)=O)n1.C1(C(=O)OCC)CC1(Cl)C(=O)NCC c1(OC)ncc(C(=O)N(C2CN(C(=O)C=C3CCC(C)C3)CC2O)C)cc1Cl C1(O)(c2cc(C(=O)OCC)on2)CCN(C(=O)C(C(C)C)C(F)(F)CN)CC1 Cn1cc(NC(c2c[nH]c(C(N)=O)c2)=O)cc1C(=O)NCC1CCC(=O)NC1 c1(C(C(=O)NCc2cn(C3CN(C(CCCOC)=O)C3)nn2)C)ccc(C)cc1 c1(C(=O)NCC2(NC(C(F)OC)=O)CC2)ccc(N(C)C)c(F)c1 N1(C(c2c(C)cccc2)=O)CCC(O)(C2(NC(c3cnnc(Cl)c3)=O)CC2)CC1 C1(C(N2CC(=C(CNC(c3c(C)nccn3)=O)F)C2)=O)CCCC2CCCN12 C1(COC)CCN(C(=O)Cc2cc(C)on2)C1.C(=O)(C(F)OC(F)(F)F)OCC C1(NC(C2N(C(C3(Cl)C(C(C)=O)C3)=O)CC(O)C2)=O)CC2C=CCC(C1)C2 c1(C(N(CCOCCCN(C(Cc2cnc(C)s2)=O)C)C)=O)csc2cncn12 C1C(C)(C)CN=C2C=CNC=C2S(=O)(=O)N1.C1(COCC)CCCC2(CCC2)O1 C1(CC(=O)OCc2c(CC)nco2)CCCC(NC2CCOC2=O)C1 c1(C(=O)OCC(c2c(N(C)C)cccc2)=O)cc(Br)cnc1O c1(CC(=O)N(C2CCN(C(c3csc(C(F)(F)F)c3)=O)C2)CC)ncc(C)s1 C(=O)(C(CCC(N)=O)n1cc(-c2ccc(N)c(N)c2)nn1)N1C(C(C)C)CC1 c1(C(N2CC(CCCCN)OCC2)=O)cc(F)c(F)c(F)c1F C1(C(=O)NC2CCCN2C(=O)C(C)(C)C)(NC)CC(O)C1 C(C(C)(C)C(=O)N1CCC(CNC(c2cc(CN(C)C)on2)=O)CC1)OC N1(C(CCOC(C)=O)=O)CCC2(CC1)CCN(C(C1CCS(=O)(=O)C(C)C1)=O)C2 CC1CC(C(=O)NN2CCCC2C(N2CC(=O)NCC2C)=O)=NO1 c1(NC2N(C(C(C)OS(CC)(=O)=O)=O)CC2)cc(C#N)cc(Br)c1CO N1(C(CN(C)C)=O)CC=CC(C(=O)Nc2cccc(NS(C)(=O)=O)c2)C1 CC(C)CCCCCCNC(C1(C)CCCN1C(=O)C=Cc1nccs1)=O C(=O)(C(CCCC)C(C)C)N1CCC(F)(C(=O)NC(C=C)C)C1 C=CCCC(C(=O)N(C)Cc1cccc(C)n1)NC(=O)C=C(C)C c1(CC)cc(Cl)ccc1C(=O)NC1CN(C(=O)Cc2cn(C)nc2C)CC12CC2 C12(C(N(CC(CNC(CCC(=C)C)=O)O)C)=O)CCCN(C1)S(=O)(=O)C2 c1(C(=O)Nc2cc(C(=O)O)nn2-c2cc(F)cc(F)c2)nnc2ccc(Cl)nn12 c1(OC)cc(F)c(Cl)cc1C(=O)NC1CN(C(c2nnccc2C)=O)CCC1F CC(C(=O)NCC1(C)CCCN(C(C2(c3ccc(F)cn3)CC2)=O)C1)S(N)(=O)=O C1(C(=O)OC)CC12CCN(c1nnnn1C1C3COCC13)CC2 CC1=NOC2(C1)CC(C(=O)NC1CC(F)(CNC(=O)C(F)CC3CCC3)C1)C2 C=CCC(CC)C(=O)NC1CCC(N(C(=O)Cc2cnnn2C)C)CC1 CC(C)C(C#N)C(=O)N1CCN(C(=O)CCC(C)(F)F)C(c2cccc(Cl)c2)C1 C1(OCO)C2CC(O)C(C2)N1C(=O)C=Cc1ccoc1.C(C)(C)C.CN1C(=O)NC1 n1(C(C)(C)C)ccc(NC2C(C(=O)C3CC3)C2)n1.C1(C(=O)N)(CCCC2CC2)CC1 C(=O)(C(F)CCC(C)(C)C)N1CCCC(F)(CNC(C(C)C(F)(F)F)=O)C1 N1(C(CCCN(C(C)C)C)=O)C(C(=O)NCCC(O)C2CCC2)C2CCCC12 C1(CC(=O)Nc2c(OC)ncc(C)c2)CCCC12CN(C(=O)CN(C)C(C)=O)C2 Cc1cc(C(=O)NCC2(C)CCN(C(c3cc(C4CC4)no3)=O)C2)nc(CO)n1 Cc1cc(NC(C2CC3(CC3)CN2Cc2ccc(C(C)C)nc2)=O)cc(Br)c1C c1(CCC)cccc(C(=O)NC(C)CCCNC(C2CCCC(=O)N2)=O)c1 N1(c2nnc(C#N)s2)CCC(NC(C23CCCC(CO2)C3)=O)C12CCC2 O=CN=c1nc2ccccn2[nH]1.C1(C(=O)O)CCCC1C(c1cn(C)nn1)O c1(C(=O)OC)ccc(NCc2[nH]c(=N)ccc2C)cc1F c1(CC(=O)N(CCNC(C=CC)=O)C)ccc(-c2ccccc2)cc1 C#Cc1ccc(C(=O)NC2CC(C(=O)NC(C=C)CO)C2(C)C)cc1C c1(C(=O)NCC2CC(NC(c3ccc[n+]([O-])c3)=O)C2)ccn2nccc2n1 C=CC(C)(C)CC(=O)N1CCC(O)(C(C)CNC(c2ccc(OC)cc2F)=O)C1 N1(C(C2CC(C#N)(F)C2)=O)CCOC2(C1)CN(C(=O)CC1CCC3CC13)C2 C1(CNC(COCC(=O)NC)=O)(OC)CCCN(C(C2CCN(C)C2=O)=O)C1 c1(C(c2n(C(CC)(C)C)nnn2)Nc2cncnc2C)c(O)ccc(F)c1F C(=O)(C(C)C(O)CC)N1CC(C=C)(CC(=O)N(CCCCCO)C)C1 O=C(CC(O)CC1CC1)NCC1CC1CNC(C1CC1c1ccccc1)=O C(=O)(C1=Cc2ccccc2C1)NC(C1CC1C(=O)NC1CCCC1)C C1(C2(C)CC2)CC(NC(N2CCCC(Oc3cnccn3)C2)=O)CCO1 CN=c1[nH]c(NC(c2ccc(OCC(C)C)cc2)C)ncc1Cl C1(C#CC(=O)NC(C)C(C)C(=O)N(C)CCOC(C)=O)(CC)COC1 N1(C(CCC=CCC=C)=O)CCCN(CCNC(=O)C(C)CC(N)=O)CC1 C(C(O)CN=c1nc2scnc2c(NCCn2ccccc2=O)[nH]1)OC(C)C CC(C(=O)N1CCC(C(=O)NCc2ccccc2F)(CO)C1)S(N)(=O)=O c1(C(=O)NCCCN(C(=O)CCC2CC2)C(C)C)cn2c(n1)CCC(C)C2 C(CC(C(C)C)NC(=O)C(c1ccc(Cl)s1)=O)N(C(C(CC)OCC)=O)C CC(C)C(C)(C)C(=O)NCC1CN(C(=O)CC2CCCCCO2)CCCO1 N1(C(CCc2cnc(C)nc2O)=O)CCCC2CN(C(=O)C3=NOC(C)C3)CC12 Cc1ccc(NC(=O)C(CCSCC(C)O)NC(=O)OC(C)(C)C)c(F)c1C c1(-c2c(CNCc3c(OC)ccs3)c[nH]n2)ccc(Cl)c(Cl)c1 C1(NCC2(C)CC(C(N3CCC3C3CCCC3)=O)C2)CC(=O)NC(=O)N1 c1(C(=O)NC2CCC(CNC(=O)Cn3cnnc3O)C2)[nH]nc([N+](=O)[O-])c1Cl Cc1cc(=NC(=O)CC2C3CN(C(C4C5CC(=O)CC45)=O)CC23)[nH]n1C1CC1 N1(C(Cn2ncc(CC)c2)=O)CCC2(CC2C(=O)NCc2cccnc2)C1 c1(C(N(C)CC2N(C(c3c(C)coc3)=O)CCOC2)=O)cnn2c(Cl)cccc12 O=C(CCC(F)(F)Cn1cc(-c2cccnc2)nn1)NC1CC2CCCC2(O)C1 CC1CCC(C(=O)NCCN(C(c2ccc(-c3cccs3)o2)=O)CC2CC2)S1 c1(CNC(CCC(=O)OCC)C)ccc2cc(OC)ccc2c1 C=CC1(C(=O)NCc2sc(C)cc2C)CCN(C(=O)CCC(C)OCC)C1 C(=O)(C(CCC)CC(C)C)N(CC(CC)NC(C)=O)C.C(=O)(C=C(Cl)Cl)N C1(OC)(CNC(=O)CC2CCC(F)(F)C2)CCN(C(=O)C=CC2CCC2)C1 C#CCC(C)(CC)C(=O)NC(CN(C)CCC)CO.C1C(=O)NCCS1 C(C(=O)N(CC(C)N(C)C(c1cnc(Cl)n1C)=O)C)(C(C)C)NC(=O)OC(C)C N1(C(c2cc(C)no2)=O)CC2(CCCC2)C1C(=O)NCCc1ncc[nH]1 C(=O)(C#CC(C)(C)CNC(C1COC(=O)N1)=O)N1CC(C)SCC1 C(=O)(C(O)CCS(C)=O)NC(c1ccc(OC)c(OC)c1)C1CC1 C1(CNC(c2nc(C(C)C)oc2)=O)CN(C)CCN1C(=O)CCOCC(C)(C)C c1(OC)cc2cc(c1)-n1cc(nn1)CCO2.C1(OC(C)C)CC1(F)F C(C(O)CC(c1nnnn1CCCF)NC1CC(OC)C1(C)C)OCCC S(=O)(=O)(c1c(F)cc(OC)cc1Br)NC(C1CC(CC(=O)OC)C1)=O C1(C(=O)NC(CNC(c2ncn(C)c2)=O)(C)C)CC12C(=O)Nc1ccccc12 N1(C(CC(=O)NC2CC2)=O)CC2CCC1C1CN(C(C3COCCO3)=O)CC21 C1(CNC(CNS(N(C)C)(=O)=O)=O)CN(C)CCN1C(=O)CCCn1cccn1 c1(C(=O)NC(CNC(C=CCOC)=O)(C)C)ccc(Br)cc1N1CCOCC1 C1(C(N(C)CC2CCCN(C(c3c(CC)non3)=O)C2)=O)CC(C)(C)CN1C C1(C(=O)NC(c2n[nH]c(=N)s2)C)CNCC12CCS(=O)(=O)CC2 Cc1c(CC(=O)NC(C)CN(C(=O)CSCC(F)F)C)cnn1C CC1=CCC(C(=O)NCC(C2CC2)NC(C2(C)CCOCC2)=O)CC1 CN(C1CCOCC1)N1CCC(CCc2cnccn2)C1 C(=O)(C1=Cc2ccccc2C1O)NC(C)(C)CNC(c1cc2n(n1)CC1(CC1)C2)=O C(=O)(C(CC(C)C)NC(c1csc(=N)[nH]1)=O)N(C1C(NC(C)=O)CCCC1)C C1(CNC(c2ccc(Cl)o2)=O)CC(CNC(=O)CCc2cccs2)CO1 Cc1nccc(C(=O)NCCC2(C)CCN(C(=O)C(C3CCOCC3)C)C2)n1 C1(C(N(CCN(C(=O)C(F)C(F)(F)F)C)C)=O)CC2OC(=O)OC2C1 Cc1cccc(C(=O)NC2CCC(CC(=O)NC(c3ccsc3)C)CC2)c1C#N C1(C)(CN(C(Cc2c(C)non2)=O)C)CCCC1NC(=O)CC1CCCC1O C12(NC(CCc3ccn(C)n3)=O)CCCC1CN(C(C1CCCCC1(F)F)=O)C2 N1(C(=O)COC2CCN(C(c3ccn(CCC)n3)=O)C2)CCC(F)(F)C1 C(CN=c1[nH]c2c(c(=NCC(F)C3CC3)[nH]1)CCC2)(c1cccc(Cl)c1)OC C1(C(N(CCC(=O)OC)CC2CC2)=O)CCCN1C(c1cccnc1)=O c1(OCC)ccc(NCC2CC(c3cnc(C(F)(F)F)nc3)C2)c(S(=O)(=O)O)c1 C(=O)(CC(F)(F)C(F)(F)F)N1CC2CC(NC(c3c(C)ccc(OC)c3N)=O)C2C1 C1(CNC(c2csnn2)=O)CN(C(=O)COC2CC=CC2)CC1(F)CO CCCCC(C(O)C(=O)Nn1ccnc1)NC(C1CCC(C)CC1)=O c1(C(N2CC(NC(c3c(COC)cc[nH]3)=O)C3(C2)CC3)=O)ccc(F)c(C)c1N Cc1cc([N+](=O)[O-])ncc1C(N1CCC2CN(C(C3CNC(=O)N3)=O)C2C1)=O CC1CN(Cc2cccc(-c3ccc(Cl)cc3)c2)C2(CC2)C1 C(=O)(C(C)(C)C(C)NC(=O)C(C)N=[N+]=[N-])NC(c1nccc(O)n1)C c1(CC)ccc(CNC(C2C3CCC(C3)N2C(=O)C(C)(C)F)=O)c(O)c1 C(=O)(C(C(C)(C)C)NC(=O)OC(C)(C)C)NCC=CC(=O)OCC.CC(C)O Cc1cc(=O)n(C)nc1C(=O)NC1CCC1CNC(=O)C1=NOC(C)C1 N1(CCC)CCCCC1C(=O)NCCCNC(c1ccnn1CCF)=O C(=O)(C#CC1(CC)COC1)NCCN(C(=O)CC(C(F)(F)F)OC)CCCCCC N1(C(c2c(CCC)ocn2)=O)CCC2(CC1)CCN(C(=O)C1CC1)CC2C c1(OC)cc(C(N2CC(NC(=O)C(F)(F)C(C)O)CC2(C)C)=O)cc(F)c1C#N C12(OC)CCC(C(=O)N(C)CC3CC(F)CN3C(C3CC3(C)Br)=O)(CC1)C2 c1(C(=O)NC2CCN(C(=O)CO)C(C3CC3)C2)cccc([N+](=O)[O-])c1 C=C(C)C(C)(O)C(=O)NCC1CCN1C(=O)Cc1cccc(OC(F)F)n1 Cc1ccc2cc(C(=O)NC(CO)C(C)NC(c3scnc3C)=O)ccc2n1 C1(C(=O)NC(C(N)=O)C2CC2)C2CCC(C2)N1C(C1(CF)CC1)=O n1(CC(C)O)cc(C(=O)NC2CCCC(NC(=O)C(C)(C)O)CC2)ccc1=O C(=O)(C(C)(F)C(=O)NC1CC1CCCCNC(=O)Cc1c(C)cnn1C)OCC C1(C(N(CCOCCCNC(c2c(C)cco2)=O)C)=O)CC2CCCCN2C1 N1(C(c2c(CC)cco2)=O)CCCCCC(N=c2nc(C3CCCCC3)[nH]s2)C1 N1(C(C=CC=CCC)=O)CCC(C(N2CCCC(C(C)C)CC2)=O)C(C)(C)C1 n1(CC(F)(F)F)nnnc1C1(NCC2CCC2CO)CC(CC(F)(F)F)C1 CCN(OC)C(=O)CNC(=O)C(c1cccs1)NC(=O)C=CC1CCCC1 c1(CC(C)C)cc(=NCCC2CCN(C(=O)C(CO)NC(N)=O)CC2)[nH]cn1 C1(C(N2CC(CC(C(=O)N(C)Cc3ncco3)F)C2)=O)CCOC1(C)C N1(C(C2CS(=O)(=O)C2)=O)CCOC2(CCN(c3ncnc(Cl)c3Br)C2)C1 C(=O)(C#CC1(C)CC1)NCC(C1CCCCC1)NC(C(C(C)C)NC(C)=O)=O C(=O)(CC(C)CC(C)C)N1CC2C(C(N3C(C#C)CC3)=O)(C2)C1 c1(C(C)NCc2cccnc2F)cc(-c2cccc(C3(C#N)CC3)c2)ccc1Cl c1(CC(=O)NC2(C)CC(NC(C(CCC)N(C)C)=O)C2)c[nH]c2cc(F)ccc12 c1(C(N(CC(C)O)CCNC(C(n2cnc(C#N)n2)CC)=O)=O)ccc(Cl)cc1Cl c1(NC(c2cc(C)ncc2Cl)=O)ccc(OCF)c(C#N)c1 c1(C(=O)NC(c2nc(C(N3CC(O)(c4nc[nH]n4)C3)=O)co2)C)cnc(C2CC2)o1 C1(NC(C(N2CCCCCC2)C)=O)CN(C(c2cc(Cl)ns2)=O)CC2(CCC2)C1 C1(NCn2cc(C3(O)CN(C(=O)CC4CC=CCC4)C3)nn2)CC2CC1CC2O n1(CCOC)cc(C(=O)NCC2CCC(NC(=O)CCN(S(C)(=O)=O)C)C2)cn1 c1(C(N(CCC)CCNC(c2cnns2)=O)=O)cnccc1OC c1(OC)cc(C(=O)NC2CC2NC(=O)C(F)n2ccnc2)cnc1Br C(=O)(C(CNC(c1cc(Cl)n[nH]1)=O)N(C)C)N1CC(CCC#C)C1 N1(C(C2(OC)CCOC2)=O)CC(C)(C)CCC1CNC(=O)Cn1ccnn1 C(=O)(C(C)CC(=O)N1CCCC(CNC(c2ccc(C)cc2SC)=O)CC1)OC C1(CNC(C(COC)COC)=O)COCCN(C(=O)COC2(C)CCC2)C1 c1(CCC(=O)NCC2C(NC(C(C)SCC)=O)C2)cc(F)cc(F)c1 C1(NC(c2c(NC(N)=O)cncc2)=O)CCCN(C(C2(CO)CCCO2)=O)CC1 C1(C)(CC(=O)N(C)CC2CCCO2)CCN(C(c2ccnnc2)=O)C1 C12(C(N(CCCC=C)C)=O)CC(CO)(CN1C(=O)CC1CCCOCC1)C2 c1(C(=O)NC2C(NC(C3C(COC)(COC)C3)=O)CC2)cc(C2CC2)ccc1O c1(-n2c(C3C(CC)OCC3)nc(C(O)CC)n2)ccc(Cl)c(Cl)c1.C C1(NC2CC(NC)C2)CCc2nc(O)c(C#N)cc2C1 N1(C(c2cc(C)n(C(C)C)c2)=O)CCC(C)C(NC(C2CCCCC2(C)C)=O)C1 CC(C)C(C(=O)N1CC(CNC(=O)C(O)C2CC2)C(C)C1)NC(S(C)(=O)=O)=O n1(CC(C)C)cc(CNC23CCC(C)(C2)C3)c(-c2ccccn2)n1 N1(C(c2cc(Br)c3c(c2)OCO3)=O)CCC(C2CCCNC2)C1 c1(CN2C(C(=O)NCC(C)N(C)C)CCC2)c(F)cncc1F Cc1nc(C)c(C(=O)N(CC(N2CCCC2CC2CC2)=O)CC(C)C)s1 c1(C(N2CCC3C(NC(C(CC#C)O)=O)C32)=O)ccc([N+](=O)[O-])nc1 c1(C(=O)NC(CCNC(C(CC(C)C)=O)=O)C)ccc2c(ccn2C)c1 C=C(Br)CCC(=O)NC(C)(C)CN(C)C(c1cncc(N(C)C)c1)=O c1(-c2nc(C)[nH]n2)cccc(NC(=O)C(=O)NCc2ncccc2C(C)C)c1 c1(CC)cc(NC(c2ccc(O)nc2)c2nnnn2C2CCCC2)ncn1 Cc1cc(NC(=O)C(=O)NC(c2cccc(Br)c2F)CO)cc(C)c1Br c1(C(=O)NC(CNC(c2cccc(OC)c2)=O)C2CC2)cc(C(N)=O)ccc1C C#Cc1cnn(C)c1C(=O)NC(CNC(C1CC(C)OC1C)=O)CC(C)C C(C(N=c1cc(N)nc(Cl)[nH]1)c1ccco1)c1c(OC)ccc(C)c1 N1(C(C2C(=C)C2)=O)CC(OC)CC1CCNC(c1cccc(C2CCC2)c1)=O C1(CNC(C2CC2(F)F)=O)CCN(Cc2ccc(CO)cc2)CC1(F)F c1(C(N2CC(C)N(C(C3CC4CCC(C3)O4)=O)CC2)=O)ccc(=O)n2c1CCC2 N1(C(C(C)C)=O)CCC(C(C(=O)NC(C)C)N(C2CCOC2)C)CC1 C1(NC(C2CC(OC(F)(F)F)C2)=O)CCC2CN(C(C3C=CCC3)=O)CCC2C1 c1(OCC)cc(C(=O)NCC2(O)CCCN(C(c3nnc(C)s3)=O)C2)cc(F)c1 C(=O)(C1=CCCC1C)N(C1CCN(C(c2cnn(C(C)C)c2Cl)=O)C1)CCC C1(C(=O)NCC(C2CC2)NC(c2c(CS(C)(=O)=O)n[nH]c2)=O)C2C3CCC(C3)C12 N1(C(C(CC)OC)=O)CCCCC(CNC(=O)C(C)N(C)C)C1 N1(C(CN(C(C=C)=O)Cc2cccc(Br)n2)=O)CC2CCCC(C1)C2C(=O)OC N1(C(c2c(C)ocn2)=O)CCC2(CCCN2C(c2cn(C(F)F)cn2)=O)C1 CCC(O)C(F)(F)C(=O)N1CCC1CNC(c1occc1Br)=O c1(C(=O)NC2CCCCN(C(C(CCC#C)O)=O)C2)cc(F)cc(C#C)c1 N1(C(C2(NC(C)=O)CCC2)=O)C2CCCC1CC(CNC(C(C1CC1)OC)=O)C2 CC1(CNC(C)(CCc2ccncc2)c2nnnn2C2CC2)CC2CC2C1 C(=O)(C(C(C)CC)N(C)C(C1CCC(CC)CC1)=O)N(CCCC)C c1(C(=O)NC2CCN(C(c3cc(CCC)nn3C)=O)C2)c(C)cc(C)nc1C c1(CC)cccc(CC(N2CCC(F)(CNC(=O)C(F)C3CCCC3)C2)=O)c1 N1(C(C(C)NS(C)(=O)=O)=O)CCC(CNC(=O)CCC2(N)CCCC2)C1(C)C c1(-c2c(C(=O)NCC(N(OC)C)=O)c[nH]n2)cc(F)cc(F)c1O C1(CNC(c2cncc(OC(F)(F)F)c2)=O)CC(F)CN1C(C12CC(C1)C2)=O CC1CC1C1CC1C(=O)NCCC1CSCCN1C(=O)COc1ccccc1F Cc1cn2cc(C(N3CCCN(C(=O)Cc4cc[nH]n4)C(C)C3)=O)cc(C)c2n1 c1(OCC=C)ccc(C(N2CCCC2CNC(c2ccc(C(N)=O)cn2)=O)=O)cc1 N1(C(C2CN(OC)C(=O)C2)=O)CCC2(CC1)CC2C(=O)NCC1COC(C)(C)C1 N1(C(c2scc(C#N)c2)=O)CCC2(CCN(C(c3c(F)ccnc3F)=O)CC2)C1 Cc1cc(=NCC2(C)CCC(F)(F)CC2)[nH]c2ccc(Br)cc12 C1(NC(C(CNC(C2N(CC)CCCC2)=O)O)=O)CCCC(C)(C)C1 S(=O)(=O)(c1cccc(Cl)c1Cl)N1CCC2(CN(C(c3c(C)nn(C)c3)=O)C2)CC1 N1(C(c2cc(OC)c(O)nc2)=O)CCC2(CCCN2C(=O)CC2CC2C)CC1 Cc1ccc2cccc(C(N3CC(O)C(O)C3CNC(=O)CC(F)(F)F)=O)c2n1 CN1CCCC(CC(=O)NC2CC(CC(=O)NC3CCN(C(N)=O)CC3)C2)C1 C1(CNC(c2[nH]cc(C)c2)=O)CC(C(C)C)CCN1C(c1cc(=O)n(C)cn1)=O c1(C(=O)NCC=CCNC(C2C(C=C)OCC2)=O)cccc(=S)n1O c1(C(=O)NCCOCC(N2C(C#C)CC2)=O)ccc(C)nc1 c1(CNC2C(C)CN(C(CN(C(C)=O)C)=O)CC2C)cc(Cl)c2c(c1)OCCO2 CCC(C)(CCNC(C1CCCC1SC)=O)NC(c1ocnc1C(C)C)=O C1(N(C)C(c2ccoc2C2CC2)=O)CCC(n2cccc2)CC1.C(=O)(CC(F)F)N Cc1cccc(C(N2CC(O)CC2C(=O)NC(C)CO)=O)c1C Cc1c(Cl)cnn1CC(=O)NC1CCC(NC(=O)CS(=O)(=O)N(C)C)CC1 N1(C(c2c(CC)noc2)=O)CCC(C(C)(C)NC(=O)C=Cc2cnccn2)CC1 Cc1nc(C(N2CCC(C(=O)NC3CCN(C)C3=O)(CF)C2)=O)c(C)o1 c1(CC)ccc(C(=O)NC2CCCN(C(=O)CC3=CCCC3)C2C)c(OC)c1 c1(C(N2CCC(C(=O)OC)(COC)CC2)C(=O)NC)cnn2c1CCC2 C(=O)(C1CCCc2nncn21)N(CC(C)NC(c1sccc1C(C)(C)C)=O)CC C1(C(N2CC3CC(C)C3C2)=O)CC2(CCN(C(=O)C(C)(F)F)C2)C1 C1(O)(CCNC(C2CN(C3CCC3)C2)=O)CCN(C(=O)C=C2CCCCC2)C1 S(=O)(=O)(c1cc2c(cc1Br)OCO2)N(CC)Cc1ccc(C(F)(F)F)s1 C1(C(=O)NCC(C2CCCC2)NC(C=CC(CC)=CC)=O)(CC2CC2)CC1(F)F C1(COC)CN(C(c2cccc(C3CC3)c2)C(=O)NC(OC)OC)CCO1 C1(NC(=O)CC2CC2)CN(C(C23COC(CF)(C2)C3)=O)CC1c1ccc(F)cc1 c1(CS(=O)(=O)NC(CC)Cn2cncn2)cnc2ccccn12 CCCCC(CNC(=O)C(C)NC(=O)NC)NC(c1cnn(C2CC2)c1CC)=O C1(N(CCOCC)C)COCCN(C(=O)C(C)(C)C(O)c2cc(Cl)cc(Cl)c2)C1 Cc1cnnc(O)c1C(=O)NCCC(O)CNC(=O)CCc1cccn1C c1(C(N(CCCNC(c2coc3c2CSC3)=O)C)=O)cc(F)c(F)c(F)c1N C1(CC(=O)NC(C)CN(C)C(c2cc(C#N)cn2C)=O)CCC(C)C(C)C1 c1(C(=O)NCCN(C(C2CC3CC3C2)=O)CC2CC2)cc2cc(Cl)ncc2[nH]1 C1(C(=O)OCC)CCCC(C(=O)N(C)Cc2cn(Cc3cnc(O)nc3)nn2)C1 CC(C)(C)CC(O)C(=O)NC(C1CCN(C(c2cccc(O)c2F)=O)C1)(C)C c1(C(=O)NCC2CC(OC)CN2C(c2ccc(Cl)o2)=O)ccc2cc[nH]c2n1 C1(NC(C(C(C)C)NC(C2CC(=O)NC(=O)C2)=O)=O)CCN(C)CC1(C)C CCCCCCCCC(=O)N1CC2(COC(CNC(c3ccccn3)=O)C2)C1 Cn1nc(C(=O)N(CCNC(c2cn(CCCC#N)nn2)=O)C2CC2)cc1F N12CCCC1C1CCCN1CC2=O.Cc1ccc(-c2cc[nH]n2)cc1C c1(C(=O)NC2CC(N(C(CC3CC(C)C3)=O)C)C2)cc2c(Br)cccc2[nH]1 c1(C(=O)NCC(C(=O)NCC2CC(O)C23CCC3)OC)ccc2occc2c1 C1(CC=C)(NC(=O)C=CBr)CCN(C(C2CCCOC2)=O)C1 N1(C(CC(=C=C)C)=O)CCN(C(=O)Cc2ccsn2)CC1CS(C)(=O)=O Cc1cc(N2CCC(NC(=O)Cc3ccsc3)CC(C)(C)C2)ncc1[N+](=O)[O-] C1(NC(=O)CC2CC=CC2)CN(C(=O)C(O)C2CC2)C2(CCOCC2)C1 C(=O)(CC(CNC(C1CC12CCC2)=O)C1CCC1)N(C1CCSCC1)C Cc1cnc(C(N2CCOC(CNC(=O)CNC=O)C2)=O)cc1C#N c1(OC)nccc(C)c1C(=O)NC(C)CN1CCN(C(C2CCC2CF)=O)CC1 C1(NC(C(CSC)(C)C)=O)CC2CN(C(=O)COC3CCOCC3)CC2C1 C1(N(C)C)CCCN(C(=O)CC2COCCN2C(C23CCC(C2)C3)=O)C1 c1(CCC(=O)N(CCCNC(C(CC)SC)=O)CCO)ccc(OC)cc1F N1(C(CC(C)c2ccco2)=O)CCN(C)CC1C(N1CCCC1CF)=O c1(CC(=O)NCc2cn(C3CCCC(C)C3)nn2)cccc2[nH]ncc12 c1(OC)cc(F)ccc1-n1nc(CC2CCCC2)nc1C1CC1F c1(C(=O)NCCCC(C)NC(COC(C)C)=O)ccc([N+](=O)[O-])o1 C1(NC(C(CCF)NC(C2CCC(=O)C2)=O)=O)CC2(C1)CC21CCC1 c1(C(N2CC(CCNC(C3C(C=C)CC3)=O)OCC2)=O)cc(N)cnc1Cl c1(C(N2CC3CC(NC(CSC)=O)CC3C2)=O)nc2ncccc2cc1C N1(C(c2c(OC)c[nH]n2)=O)CC2(NC(c3cn(C)cc3C)=O)CCC1C2 N1(C(C)C)CC(C(N2CCC(CCNC(C3(C)C=CCC3)=O)CC2)=O)CCC1=O C1(NC(CCC(=O)NC)=O)CCCN(C(c2ccc(C)c(O)c2)=O)CC1 CC(C)CC(CNC(c1ccnnc1)=O)C(=O)N1CCC(C)CC(C)C1 C1(CC)CCCN(C(=O)CCCc2cnn[nH]2)C1C(=O)NC1(CC)CCC1 c1(C(CC)=O)ccc(NC(=O)C(=O)NC(c2ncccc2C)C)cc1 C1(C(N(C(CNCS(C)(=O)=O)C2CC2)C)=O)C2CC3C(C2=O)C13 C(F)(c1ccccc1)=CC(=O)OCCCCc1cccc(Br)c1 N#Cc1ccc(N2CCCCC(CNC(=O)C=CI)C2)nc1C(F)(F)F c1(C(=O)Nc2ccc(C(N(C)Cc3ccsc3)=O)cc2)ccccc1OC(F)F Cc1c(C(=O)NC(CNC(=O)COC2CC=CC2)CO)sc2nccn12 CC1(C)CCN(C(=O)OC(C)(C)C)CC1NC(=O)CCc1ccc(N)c(F)c1 Cc1noc(Cl)c1CCC(=O)N(C1CCN(C(=O)C(C)(C)C2CCOC2)C1)C c1(C(N2CC3CN(C(C(CCC)C#N)=O)C3CC2)=O)sc2ccccc2c1Cl c1(C(N2CC(N(C(CCCOC)=O)C)C(C)(C)C2)=O)cc2cccnn2n1 c1(OC)cc(OC)c(F)c(C(N2CCC2C(=O)NCc2cc[nH]n2)=O)c1 c1(NC(CN(C(C)=O)C)=O)ccc(NC(C2CC2C(N)=O)=O)c(C)c1 N1(C(C2(C)CC(F)C2)=O)CCC(NC(c2cc[nH]n2)=O)C(c2ccccc2)C1 C1(C)(P(C)(C)=O)CCC(CC(=O)OC)OC1.C(CCC)=CC C1(NC(=O)CCc2ccsc2Br)CCCC12CN(C(=O)CO)C2 C(C(C)C)(C(O)C(=O)NC1(C(=O)O)CC(O)CCC1)OC c1(C(=O)NC(C(C)NC(C(C)N2CCC2)=O)C)nn(C)c2c1CCC2 C(=O)(C(C)CCN(C)C)NCC(C(N1CC(C)(OCC)C1)=O)N(C)C C1(CNC(c2c(C)noc2C)=O)CCN(C(=O)CCCC(=O)C2CC2)C12CC2 CCC(CC)(CCC(=O)NCC(O)CNC(C12C=CC(CC1)C2)=O)[N+](=O)[O-] Cc1nc(C2CCCOC2)sc1C(N1CC(CNc2cccnc2)C1)=O C(CCCCNC(C1C(C)CC1C)=O)N(CC(=O)OC)C(c1nnnn1C1CC1)=O C#Cc1ccc(C(=O)NCC2CC2NC(C2CCC(C(=O)OC)CC2)=O)cc1C CC(C)CC(CC(=O)NOC1CCC1)N(C(=O)CCC1OCCO1)C1CC1 C1(NC(c2ccc(F)cn2)=O)CCCC(N=c2ccn3nccc3[nH]2)C1 C1(C)(CNC(C2C(C)OC(C)C2)=O)CCCN(C(C2(CC(F)F)CCC2)=O)C1 C1(C(N(C2CCN(Cc3ccccc3Cl)C2)CC)=O)CC(=O)N(c2cn[nH]c2)C1 c1(N(C(CC(=O)O)Cn2cncn2)C(c2csc(Br)n2)=O)cc(F)ccc1F CC1C(NC(=O)CCC[N+](=O)[O-])CCCN1C(=O)C(c1ccc(F)cc1)F C1(NC(C(CCSC)NC(N)=O)=O)CC2CC1CN(C(=O)CN(C)C1CC1)C2 Cc1sc(C(=O)N(C2CCN(C(=O)CNc3ccccc3Cl)C2)CCO)c(C)c1C N1(C(C(=O)N(c2ccccc2)C(CO)C2CC2)=O)CCC2(CC=CCO2)CC1 C1(O)(CC(N2C(CN(C)C(c3cc(C4CC4)sn3)=O)CCC2)=O)CCCCC1 C1(C(=O)NCCCNC(C=C(CCC)C)=O)(CCF)CCOCC1 Cc1nc(C)c(C(=O)N(C2CCCCC2NC(=O)CCc2cnn(C)c2C)C)o1 C1(CNC(C2(CSC)CC2)=O)CCN(C(C2OCCC2C(C)C)=O)C1 C1(NC(c2nccc(C)n2)=O)CCOC12CCN(C(c1ccc(Cl)cn1)=O)CC2 N1(C(c2c(OC)oc(C)n2)=O)CC2(CCCC(CNC(=O)CC(C)C(C)(C)C)O2)C1 c1(C(NNC(C(=O)NCC(C(=O)OC)(C)O)=O)=O)nc2c(C)cccc2o1 C1(N(C)C(C2CCCN2C(=O)C=C2CCC2)=O)CCN(C(C2(C)COC2)=O)CC1 c1(C(N2CCC(NC(C(C)SC)=O)C(O)C2)=O)cnc2ccnn2c1N C1(NC(CC(CC)NC(c2cnc(OC)nc2)=O)=O)CCCCC1C#N C1(NC(CCN(CC)CC)=O)CN(C(C2(C(F)F)CC2(F)F)=O)CC(C)(C)C1 Cc1ccc(-c2ccco2)cc1.c1cn(CC2C=CCN2C(=O)C(C)C)nn1 c1(OC)c(NC(C)=O)ccc2[nH]ccc12.n12cc(nn1)CC(=O)NCCCC2 c1(C(C(=O)NCc2c(CCNC(C=C(C)Cl)=O)ocn2)(C)C)ccc(F)c(F)c1 C1(C(=O)NCC2CN(C(=O)CCNS(=O)(=O)C(F)(F)F)C2)CC2CC(O)C(C1)C2 N1(C(CC(=O)OC)=O)CCN(C2CC2)C(=O)C1.n12cc(cn1)C(=O)NCC2 Cc1nc2ncc(C(N3CCN(C(C4(CF)CCC4)=O)CCC3C)=O)c(=O)n2[nH]1 c1(C(N(CCCNC(C2C(CC)C2)=O)CC2CCCC2)=O)ccc(F)c(N)c1 C1(C)(C(=O)NCCN2CCN(C(c3n(C)[nH]c(=N)c3)=O)CC2)CCCCCC1 C1(NC(C(C)(C)n2cccn2)=O)CCC2(CC1)CCN(C(=O)CC1(CO)CC1)C2 c1(CC)cnccc1C(=O)NC1CCC(NC(C2(CCO)CC2)=O)CC1 N1(C(CSCCN(C)C)=O)CC2(CC(NC(c3cc(Cl)no3)=O)CO2)C1 C1(CC)CCCN(C(C)=O)C1C(=O)NC1CCCN(C(=O)C=CCOC)C1C C(CN=c1nc(N2CCSCCC2)c2c([nH]1)c(C)nn2C)c1c(C)nc(C)s1 CCCC(C)(C)C(=O)N1CC(C(=O)Nc2cccc(C(C)O)c2)C(O)C1 Cc1ccc2oc(C(N3CCC(NC(c4nc(C)sc4C)=O)C3)=O)cc2c1 c1(C(N2CC(C(N3CCC(CNC(COC)=O)C3)=O)C2)=O)cc2cccc(C)c2o1 C1(O)(C(C(=O)NC2C(CCC)C2)F)CN(C(=O)C(N2CCC(C)C2)=O)C1 N1(C(C2(C)CC(F)C2)=O)CCCCC(NC(=O)CNC(C2CCC2)=O)C1 N1(C(C2CCCCO2)=O)CC(NC(C2(F)CCOCC2)=O)C(F)C1 C1(CNC(c2c(C)ccc(Cl)c2)=O)CN(C(c2cc(Cl)sc2Cl)=O)CCC1(F)F N1(C(C(COC)C)=O)CC2C(C(=O)NCc3nc[nH]n3)C2C1 N1(CCC(c2cc(CC)no2)OC)CCCC(O)(Cc2ccc(F)c(F)c2)CC1 C(=O)(CCC1(CCSC)CCC1)NCCN(C(COCC(=O)OC)=O)C1CC1.N(C)C Cc1cc(C(=O)N(CCC(C)NC(c2ccc(N(C)C)nc2)=O)C)ccc1Cl CC1=C(C(=O)N(C(C)CNC(=O)C2=CC3(CCOC3)C2)C)Cn2ncnc2N1C N1(C(C(CC)F)=O)CC2CCC1(CCC(=O)CC(C)(C)O)CC2.N C1(C(N(C2CC(OCC)C2)C)=O)CC12CCN(C(=O)CSc1cnn(C)c1N)C2 N1(C(CCCN(C)C)=O)C2CCC1CN(C(=O)Cn1cncn1)C2 c1(C(N2CC(CC(C)NC(=O)CCF)C2)=O)ccc(C2CC(F)(F)C2)cc1 Cc1ccc(C#N)cc1C(=O)NC1CCN(C(=O)CC23CCCC2C3)C(C)C1 NC(=O)C(O)C(CC1CCC1)SC1CCC(NC(=O)Nc2cccc(Cl)c2F)C1 c1(C(=O)NCC(CNC(CN(CCOC)C)=O)(C)C)c(N)ccc(C)c1F Cc1c(Br)ccc(C(=O)NC2CN(C(c3ncccc3Br)=O)CC2F)c1C Cc1cc(C(=O)N(C)CC2(O)CN(C(c3c[nH]c(Br)n3)=O)C2)cc(C)n1 CC(C(=O)NC1(CO)CCCN(C(c2cc(N(C)C)cnc2F)=O)C1)C(F)(F)F CCC(CC)CC(=O)NCC(c1ccc(CO)cc1)NC(c1ccc(F)cc1)=O c1(CSCCNC(=O)C=Cc2cscn2)c[nH]c2ccccc12 N1(C(C2(CC(=O)OC)CC2)=O)CC2CC1CN(C(=O)C(C)=C1CC1)C2 C1(C(=O)NCC2(NC(C3C(CCC)C3)=O)CCC2)CC12CC(O)C2 CCC(C)(C(=O)NCCNC(=O)CCCN(C(C(=O)OC)C)C(C)C)OC N1(C(CCCC(=O)NC)=O)CCC(C2CC2)(NC(=O)C=C2CCC(C)(C)CC2)C1 Cc1ccccc1C(C)NC(C1(C)CN(C(C2CC2(Cl)Cl)=O)C1)=O c1(OC)cccc(S(=O)(=O)N(C(=O)Cc2cccc3cccnc23)CC2CC2)c1 c1(C(=O)NCC2OCCC(NC(c3[nH]cc(C)c3)=O)C2)cc(Cl)c(C)cn1 c1(CCC(=O)NC(C)CCN(C(=O)CO)C)cccc2ccccc12 C(=O)(C1CCCc2ncnn21)N1CC(C)CN(C(C(COC)O)=O)C(C)C1 C#Cc1ccc(C(=O)NCC2C(C)CCN2C(c2cc(C(N)=O)co2)=O)nc1 c1(NC(C)Cc2ccccn2)nc(N2CCC(C)(C)C2)nc2c1cnn2C C12(CNC(c3cnn4c3CCC4)=O)CCC1CCN2C(c1c[nH]cc1Br)=O CCCC(C(=O)N1CC(N2CC(NC(C3(CC)COC3)=O)CC2=O)C1)OCC C(C(CO)(CO)NC(C1CCCS1(=O)=O)=O)N(C(=O)CCCc1cnn[nH]1)C Cc1cc(Cl)ccc1CC(=O)NC(C)(CNC(=O)CCN1CCCCC1C)CO C1(C2(NC(c3cnc(C4CC4)[nH]3)=O)CC2)CCCN1C(C1CC1CF)=O CCS(=O)(=O)CC(=O)N1CCC(COC)(NC(=O)Cc2csc(Cl)c2)C1 c1(C(N2CCC(CCCCCNC(C=CC)=O)CC2)=O)cc2n(n1)CC1(CC1)C2 N1(C(c2c(CCC)nns2)=O)CCOC(CNC(=O)CCn2cncn2)C1 N1(C(C=CC(C)C)=O)CCC2CN(C(=O)CSn3cncn3)CC2C1 n1(CC(=O)N(CC(=O)NCC(COCC)C)CC)c(O)nnc1O N1(C(c2cn(C3(C)CC3)nc2)C(=O)NCc2ccco2)CCC(F)(F)C1 C1(NC(CCN(C(CC)CC)C)=O)CCC(C(=O)NC2(C(=O)OC)CC2)C1 c1(C(C)C)nc2c([nH]1)CC(C(=O)NC1CN(C(c3ccncc3)=O)CC1C)CC2 C1(CC)CN(C(C23CC4CC2C3C4O)=O)CCC1NC(=O)CCc1nccs1 C(=O)(CCC(CC)NC(C1CC1C(F)F)=O)N1CC(OCC)(CO)C1 Cc1cc(C(=O)NC2CC(CNC(=O)CC3CC3)CC2O)c(C)nc1C Cn1nc(C(F)(F)F)c(I)c1CNCCC(=O)Nc1ccc(F)cc1Cl C1(O)(CC)CCN(C(=O)C(C2CC2)N(C(=O)CCc2ccnn2C)C)C1 N1(C(C2(O)CC(C)(C)C2)=O)CCCC(CNC(=O)C=CC(=O)NC2CC2)CC1 C(=O)(CC(F)(F)CC12CCCC1C2)N(C(c1cnn(C)c1)C)C CCCC(C)(O)CC(=O)NCC1COCCN1C(=O)C=C(C)C(C)(C)C CC1CC(NC(=O)C(CC2CC2)NC(C2CCCCCN2C)=O)CC(C)(C)C1 c1(C(CC(=O)N(CC(C)CNC(C2(C(N)=O)CC2)=O)C)C)ccc(C#N)cc1 c1(CNC(COCC=C)=O)ccccc1CNC(C1CC(C)C1(C)C)=O C1(CC(=O)N(C)CCOCCNC(c2nc(Br)c[nH]2)=O)CCC(C)CC1 N1(C(c2ccc(OC)cc2C(C)C)=O)CC2CC(C1)CN(C(=O)CC(C)(C)O)C2 c1(OC(C)C(=O)NC2CCN(C(=O)C(c3cnn(C)c3)=O)C2C)cccc(F)c1 C#Cc1ccc(C(N2CC3CC2CN(C(=O)CC2COCC2O)C3)=O)cc1Cl c1(NC(C(CC)NC(c2cn(C)cn2)=O)=O)cncc(OC)c1 C1(NC(C(S(C(C)C)(=O)=O)C)=O)CC2(C1)CC2N=c1[nH]nc(C(F)(F)F)s1 c1(C(N2CCN(C(c3c(CC)[nH]c(=N)s3)=O)CC2C)=O)csc2ccc(F)cc12 N1(C(CSCCCC)=O)CCCC2CN(C(=O)C#CC3CCCCC3)CCCC12 N#CCCCC(=O)N1CC2CC2(C(=O)NCCc2ncccc2F)C1 CCCC(CNC(c1cccn(C)c1=O)=O)C(=O)NC(CC)C(C)C C1(CNC(C(CC)NC(C)=O)=O)CC2CN(C(c3ccc(F)cc3O)=O)CC12 C1(OC(C)C)CCN(C(C2CCN(C(=O)C#CC3CC3)C2C)=O)CC1 N1(CC=Cc2cc(C)cc(C)c2)CC2C3CC(CC3C2)C1.c12cc(ncn1)N2 CC(C)(C)C(CC(=O)NC1C(NC(C2CN(C(N)=O)C2)=O)CC1)C(F)F c1(-c2nc(-c3c(C)occ3)on2)cnn2cccc(Cl)c12.C1(N)C(C)CCC1C CCC(C)(O)C(=O)NC1CCCCC1CC(=O)NC1CCOC(C)C1 N1(C(COC)=O)CCN(C(c2cnc(N)c(Br)c2)=O)C(C(C)C)C1 c12nc(c(C)o1)C(=O)NCC(C)(CO)NC2=O.c1(CC)ccc(N2CCC2)nc1 c1(C(N2CC3C(NC(c4c(CC)scc4)=O)(C3)C2)=O)cc2c(nc1O)CCCCC2 Nc1c(Cl)c(C(N2CCCC(c3cn(CC(F)(F)F)nn3)C2)=O)cc(F)c1Cl C1(C(=O)Nc2nnc(C3N(CC#C)CCC3)s2)CCC(C(=O)OC)CC1 CCC(C)(CCC(C)C)C(=O)N1CC(NC(=O)C(C)(C)C)CC(C)C1 c1(C(N2CCC(CC=C)(NC(=O)C(COC)N(C)C)C2)=O)cccc2scnc12 C1(NC(C2CCCC(NC(CC=C(C)C)=O)C2)=O)CCc2n[nH]cc2C1 N1(C(C(CC)O)=O)CCOC(c2cn(Cc3cccnc3)nn2)C1 C(=O)(C1=CC2C=CC(C1)C2)N1C2(C(N3CCC(C(N)=O)C3)=O)CC2CC1 C1(S(=O)(=O)c2ccc(Cl)cc2)(C(=O)NCCNC(=O)CC2CC=CC2)CC1 C(=O)(C1=CN(CC)CCC1)Oc1cc(COC)cc(F)c1 N1(C(C(C2CCCN(C(c3c(C(C)C)ocn3)=O)C2)C)=O)CCC(F)(F)C(F)C1 c1(C(N2CCC(N(C(CCNC(C)=O)=O)C)CC2)=O)ccc(N)c(Cl)c1 O=S(=O)(c1ccc2c(c1)CCO2)NC1CC2CCC(C1)N2S(=O)(=O)CC1CCC1 c1(CNC(CC(C)N(C)C)=O)ccc(C(=O)NC2(C)CC2(C)C)nc1 CC(C)C1=NOC(C(N2CCCC(F)(C(=O)NC34CC(C3)C4)C2)=O)C1 c1(CC(=O)N(C)CCOCCNC(C2CCC(C)(C)O2)=O)ccc(Br)cc1F c1(C(=O)NC(C2CN(C(Cc3cc(C)on3)=O)C2)C)ccc2c(c1)N(C)CCO2 N1(C(c2c(C)occ2)=O)CCC(NC(=O)C(F)(F)C2(O)CCC2)C(C)C1 C1(C)(C(=O)NCc2c(SCC)nccn2)CC12CCN(c1ncccc1Cl)CC2 N1(C(C(CCCC)O)=O)CC(NC(c2cnc(C3CC3)s2)=O)C2CCCC2C1 c1(C(N(CC(=O)NCC(=O)N(C)C)CC#C)=O)cccc(C)c1C c1(CCC(C)C)nc(C(O)C(C)NC(C)=O)n(-c2cccc(C(N)=O)c2)n1 c1(C(=O)NC2CCC(C(=O)NCC3CCC(C)C3)C2)noc2ccc(F)cc12 CC1=NOC2(C1)CC(C(=O)NC1CCCN(C(C3CC(C)OC(C)C3)=O)C1)C2 CC(C)C(O)Cc1cn(CCCCCNC(=O)CSC(C)(C)C)nn1 c1(C(=O)NC23C(CN(C(C=C(C)C)=O)C2)COCC3)cccc2cnnc(O)c12 c1(C(=O)NCC(CNC(=O)C=C(C)C(C)C)OC)ccc(Br)c(N)n1 Cc1nc(C(N2CCN(C(c3ccnnc3O)=O)CC(O)C2)=O)c2n1CCCC2 c1(C(=O)NCc2ccncc2)cccc(NC(=O)NC2(CC(=O)OCC)CC2)c1 Cc1cc(F)ccc1C(N1CCCC(N(C(=O)C=Cc2ccc(Cl)s2)C)C1)=O c1(C(N2CC(C)(NC(c3ccc(SC)o3)=O)C2)=O)cncc(NC(C)C)c1 Cc1cc(C=CC(N2CCCC2CN(C(=O)CCCC(N)=O)C)=O)c[nH]c1=N CC(C)C(C(=O)N1CCC(CNC(c2ncccc2C(F)F)=O)C1)NC(N)=O C1(C(N(C2CN(C(C3(OC(C)C)CCCC3)=O)C2)C)=O)CCCC(C2CC2)O1 C(=O)(C(C)(C)C(C)NC(c1ncnc(O)c1F)=O)NC1(c2onc(C)n2)CC1 n1(C(C)C)ncc(C(=O)NC(CO)C(C)NC(C2(O)CCOC2)=O)c1C(F)(F)F N1(C(=O)NCC(CC)(C)C(C)O)Cc2ccccc2CC1CC CC1CCC(NC(c2ccc(C3CC3)cn2)=O)CN1C(C1CCC(C)CC1)=O C1(NC(CSCCC=C)=O)CC(CO)N(C(=O)COCC2CCC2)C1 n1(CC#C)cccc1C(=O)NCCC(C)N(C(=O)CC1(COC)CC1)C Cc1oc(C)c(C(=O)NCC(C)NC(=O)CCCc2cccc(Cl)n2)c1C c1(C(=O)NCC2CC(CNC(C3C(C)=CCS3)=O)C2)cc2c(cn1)COCC2 C1(C(=O)NCC2CC(O)C23CCC3)CCCCCCN1C(=O)CC1CCOC1=O Cc1ccc(O)c(C(N2CC3CC3(NC(=O)C=CSCc3ccco3)C2)=O)c1 c1(C(=O)NC2CC(C(=O)Nc3n[nH]cc3[N+](=O)[O-])C2)cccc2ncsc12 C(=O)(C(C)(C)CCCNC(c1ccnc(O)c1)=O)N(CC(c1nn[nH]n1)C)C C1(NC(C(C)(F)F)=O)CN(C(c2csc(Cc3cccc(Br)c3)n2)=O)CC1F N1(C(CCCC)=O)CC(NC(c2nccn2CC)=O)CC12CCCCCC2 Cc1cc(O)ccc1CC(=O)NCC1CC(NC(C2CSCCS2)=O)C1 N1(CC(c2noc3c2COCC3)=O)CCOc2cc(Cl)c(Cl)cc21 c1(C(c2nnnn2CCC)NCC=C)c(F)cc(C(=O)O)c(Br)c1F C12(NC(c3c(CC)nns3)=O)CCOCC1CN(C(=O)CC(CC)C(F)F)C2 c1(C(=O)NC2CCCN(Cc3ccc(F)c(O)c3)C2)cccc2c1OCO2 N1(C(=O)Nc2n(CC)cnc2)CCCCC1CC(=O)N(C1CCN(C)CC1)C C1(NC(c2c(C)nn(C)n2)=O)CN(C(=O)C(C)N2CCCC2)CC1(C)C c1(C(=O)NC2C(C(=O)Nc3ccc(CC)cn3)C2)ccc2scnc2c1 c1(C(=O)NCCN(C(CC2ON=C(C)C2)=O)C)cc(S(=O)(=O)C(C)C)ccc1F C(=O)(CCC(=O)NCC1(C)CC(NC(C2CC(C(C)(C)C)C2)=O)C1)NC N1(C(C2C(OC)CCCC2)=O)CCC(C(N2CC(CO)(CF)C2)=O)CC1(C)C N1(C(C2CC(C#C)(O)C2)=O)CC2CCC(CNC(=O)CNC=O)C2C1 c1(C(=O)NC(CC=C)CNC(c2ccnc(CC)c2)=O)ccc2nc[nH]c2n1 N1(C(C(=O)NC(CC)(C)C)C2CC2c2ccsc2)CCN2C(=O)NC(=O)C2C1 C1(C(C)C)CC=C(C(C(=O)OCC2CCOCC2)N2CCCC3(CCC3)C2)CC1 c1(C(C)C(=O)OCC(c2nnc(Br)s2)=O)ccc2c(c1)OCCO2 C1(CNC(C(c2ccoc2)NC(C2C(CC(C)C)C2)=O)=O)CCC(CO)O1 CCC(CC)C(=O)NCC(C1CCOC1)NC(=O)C=Cc1ccsc1 N1(C(=O)OC(C)(C)C)CC2C(C1)C2(C)COC(C1CCC(=O)CC1)=O C=C=CCCC(=O)N1CCC(C2OCCCC2NC(C2CCCNC2=O)=O)CC1 N1(C(C2C(C)=CCS2)=O)C(C(N2CCCN(C)CC2)=O)C2CC(O)C1C2 C(CCCCC(=O)NC1CCCN(C(=O)CC2CN3CCC2CC3)C1)N(C)C1CC1 c1(OC)cc(C(N2CCC(C)(CCNC(=O)CC(C)SC)C2)=O)ccc1C N1(C(c2c(C)nccn2)C(=O)NCc2ccc(F)cc2)CC2CNC(COC2)C1 N1(C(c2cc(C(C)=O)sc2)=O)CCCC(N(C(=O)CC2CCOCC2(C)C)C)C1 c1(C(=O)NC2CCN(C(c3cncc(NC)c3)=O)C2)ccc(S(N)(=O)=O)cc1Cl C1(c2ccccc2)(C(N2CC(OCCNC(C=CC(C)(C)C)=O)C2)=O)CC1(Cl)Cl C1(CC(=O)OC)CCCC12CCN(C(=O)CCc1cn(C)cn1)C2 Cc1ncnc(NC23CCC2CN(C(c2ccc(C(F)(F)F)cc2C)=O)C3)c1F C(C(=O)NC(C)CCCNC(c1c(-c2ccn(C)n2)noc1C)=O)(C(C)C)OC CC1(C)CC1(O)C(N1CCC(OCCNC(c2ccc[nH]2)=O)C1)=O C(C(C)C(C)C(=O)NC1(CO)CCCN(C(=O)C=CCOCCOC)C1)OC C1(C(=O)NC23CC(NC(C(C4CC4)OC)=O)(C2)C3)CC(=O)N(C2CCCCC2)C1 N1(C(C2CCS(=O)CC2)=O)CCC2CN(C(c3cc(O)ncn3)=O)C2C1 N1(C(C(c2c(OC)cccc2)(F)F)=O)CCNC(=O)C(F)(F)C1 N1(C(CC#N)=O)CCCC2(CCN(c3ncnc4ccc(Br)cc34)C2)C1 C1(C(N2CC(O)(C(C)NC(CCCn3c(C)ncc3)=O)C2)=O)CCC12CCC2 N1(C(CCc2c(C)cccn2)=O)CCC2(CCN(c3ncc(Br)c(C)n3)C2)C1 C1(C(=O)NC(CC)CN(C(=O)CCc2cn[nH]c2)C)CCCC(C)(C)O1 c1(CC(=O)NCCC(C)NC(C2CCOCC2)=O)ccnc(Cl)c1F Cc1noc2ncc(NC(=O)C(C)OC3CCOC3)cc12 c12cnc(nc1C(F)(F)F)NC2.c1(CCC#N)cncnc1O C1(OC)CC(NC(c2ccc(Cl)c(F)c2)=O)C12CCN(C(C1(O)CCC1)=O)CC2 CN1CC2(CCN(C(C3CC4C=CC3N(C(=O)CC3CC3C3CC3)C4)=O)CC2)C1 C(=O)(C1=CCCCO1)NC12CC(CNC(c3n(C)cc(Br)c3)=O)(OC1)C2 C=CCC(C)(CC)C(=O)N1CCC(OC(=O)C(F)(F)F)CC1 N1(C(c2ccc(CCC)cc2)=O)CCC2CCC(NC(=O)C(C)(C)F)C1C2 CCCCN=C(NCC1CCCCC1)NCC1(N(C)C)CCSC1 c1(NCC(C)Cn2ccnc2)cc(Br)ccc1S(=O)(=O)N1CCCC1 N1(C(C2(CO)CC2)=O)CC(C)OC2(CCN(C(=O)CCCC#CC)C2)C1.C#CCN C(CCC1CC1)(C(=O)N(C(C)C(C)(C)O)C)NC(C(C)SC(C)C)=O N1(C(C2CN(C)CC(C)O2)=O)CC(NC(C23CC2COC3(C)C)=O)CCC1C N1(C(c2c(CC)noc2)=O)C2CCC1C1CC1(NC(C1CN(C(N)=O)C1)=O)C2 C1(CC(=O)NC(CNC(Cc2scc(CC)n2)=O)CO)C=CS(=O)(=O)C1 CC1CN(C(=O)CC(C2CC2)NC(C2(C)CCCO2)=O)C1(C)C C1(NC(C(C)SC)=O)C=CCN(C(=O)CCOCC(F)(F)F)C1 c1(C(=O)NCC(c2cccc(OC)c2)F)cc(Cl)c(Cl)cn1 c1(C(=O)NCC(C)NC(C2(C(C)C)CCC2)=O)cc(Cl)c(F)c(Cl)c1 C(=O)(C#CC1(CC)CC1)NC1(CNC(c2nc(C(C)OC)sc2)=O)CC1 C1(CNC(C2C(C)CCC2)=O)C(C)CCN1C(=O)CC1CCS(=O)(=O)C1 c1(CNC(C)=O)ccc(NC(N2CCCC2c2ccn(C)n2)=O)cc1 N1(C(CCN(C)C(c2cccn2C2CC2)=O)=O)CC2CCCCC1C2 c1(C(N2C(C(C)NC(C3CCCC3O)=O)CCC2)=O)ccc(C2CC2)nc1O N1(C(C(C)=CC)=O)CCOC(CN(C)C(C2CCN(c3ccncn3)CC2)=O)C1 C(C(CC1CC1)C(=O)NCCCc1cccnc1)NC(CC1CC(=C)C1)=O Cc1c(N)ccc(C(=O)N(C)CC2CN(C(=O)C(C)CO)CCO2)c1C Oc1ccccc1Cn1cc(C2(O)CCOC2)nn1 C=C(C)CC(C(=O)N1CC(O)(CO)C1)NC(=O)CC(C)=C(C)C C1(C)(CNC(C2(C)CC(C)C2)=O)CN(C(=O)C2=NOC(C(C)(C)C)C2)CC1C C(=O)(C1CCCc2ncnn21)N(CCCCN(C(=O)C1=CS(=O)(=O)CCC1)C)C N1(C(C2(F)CCN(C(c3cc(COC)no3)=O)CC2)=O)CCCC(F)(F)CC1 CC1(C)C(NC(c2ccccc2F)=O)C2CCCN(C(c3cccnc3)=O)C12 C1(C(=O)Nc2ccc(C=C)cc2)CCc2nc(-c3cncc(OC)c3)sc2C1 c1(C(=O)NC2CCN(C(CNC(=O)OCC=C)=O)C2)cc2cc(F)c(Cl)cc2[nH]1 C(=O)(CCCS(N)(=O)=O)N1C(C(C)(C)NC(C=Cc2nc(C)c(C)[nH]2)=O)CCC1 C12(CNC(C(=O)N(C)Cc3ccsc3)=O)CC(C(F)F)(C1)C2 CC(C)C(C)C(CNC(c1ccon1)=O)NC(c1ccc(N)c(O)c1)=O c1(Nc2c(COC)cccc2)c(C)ncnc1C Cc1cc(C)n(C(N2CCC(=CC(=O)Nc3ccccc3C)CC2)C)n1 c1(C(CC)OCC)nc(-c2cnn(CC3CCCCC3)c2)n(C(C)C)n1 c1(CNC(C2COCCN(Cc3ccco3)C2)=O)ccc(F)cc1Cl C1(C(N(C2CC(NC(=O)CC3(n4cncn4)CC3)C2)C)=O)C2CC2C2CC12 N1(C(C(C=C)O)=O)CCC(CNC(=O)CC2CCC(C(F)(F)F)O2)CC1 C(=O)(CS(=O)(=O)CCC(F)(F)F)NC1(CNC(C2C(C(C)O)C2)=O)CCC1 C(CC(C(=O)N(CC(C)C)C)NC(C1CCN(C)C1)=O)OC c1(CNC(c2ncccn2)CO)nc(Cl)ccc1Br c1(-c2c(C(C)O)cccc2)ccc(C#N)cc1.c1nc(Cc2ncc[nH]2)no1 C1(C(C)(C)NC(C2CCC(C)O2)=O)CCN(C(=O)Cc2cnc[nH]2)CC1 n1(CC)ccc2cc(CNC(CCO)CCC(F)(F)F)ccc12 c1(CCN(c2nnc(C(=O)OC(C)(C)C)n2CC(=O)NC)CC)ccc(C)c(C)c1 CC1N(C(C2CCC(NC(=O)CCc3ncccn3)CC2)=O)CCCC12CCC2 C1(C)(NC(C2C(c3cn(-c4c(C)c(F)ccc4)nn3)C2)=O)CN(S(N)(=O)=O)C1 C1(C(=O)NCCOCCCNC(CCCOCCC)=O)OCCN(C)C1=O N1(C(C2(CO)CC2)=O)CCC2(CC1)CC2CNC(C1CC(F)(CO)C1)=O C1(C(N2CCC(CCC(=O)NC(C(=O)NC)C3(C)CC3)C2)=O)(CC)CCOCC1 CC(C)(C)C(O)C(=O)NC1CCC1NC(c1c[nH]nc1-c1cccc(Cl)c1F)=O C1(CNC(CN(CCOC)C)=O)CCN(C(C2C(c3ccncc3)C2C)=O)CC1 C(=O)(CS(=O)(=O)N1CCOC(C2CC(CNC(=O)OCC)C2)C1)OC(C)(C)C C12(NC(Cc3ccc(SCC)cc3)=O)CCC1CN(C(=O)CCC(F)F)C2 CONC(=O)C(=O)NC1CC(N(C(=O)C=Cc2ccncn2)C)C1 c1(NC(=O)CCC2CCCN2Cc2ccccc2F)cccc(F)c1Br c1(C(N2CCCC2c2cccs2)C(=O)NC(C)(C)C)nc(CBr)sc1Br C1(C(=O)NCc2c(C(=O)NC(C)(C)CC3CC3)con2)CC2(CCCO2)C1 O=C1Nc2ccccc2CC1SCC(N1CCC(C(=O)O)C1)=O C1(C(=O)OC)(COC)C=CCN1C(c1ccc(Cl)cc1)C(=O)OC n1(C(C)C)cnc(C(=O)NCCSCC(=O)N(CCO)C2CC2)c1 c1(CC(N2CCCC(N(C(CC(C)n3cccn3)=O)C)C2)=O)cccc(C#N)c1 c1(CC)ccc(C(C)CC(=O)N2CSCC2CNC(=O)CNS(C)(=O)=O)cc1 CCCCCC(C)(CC)C(=O)NC1CCN(C(=O)C(C(C)C)SC)C1 c1(C(N(C)CC2(O)CN(C(C(C)OC3CCCC3)=O)C2)=O)occ2c1CCC2 C#CC1CN(C(C2(CNC(c3cc(C#N)n(C)n3)=O)CC23CCC3)=O)CCO1 C(=O)(C(CCC)C(=O)OCC)N(C(C(=O)NC(CC#C)CC)C)C1CC1 Cc1ncc(C(=O)NCC2CCC(NC(=O)C(C)(C)c3cnco3)C2)[nH]1 n1(Cc2nc(C)sc2)nnc(C(N2CC(NC(=O)C(C)(C)OC(C)C)C2)=O)c1C c1(CNC(=NCc2cc(C)nc(C)n2)NC2CCCC2)cc(F)c(Cl)cc1F C(CC(C)CC)(C(=O)N1CCC(CC(N)=O)CC1)NC(CC=CC)=O N1(C(C23C(CN(Cc4nc(C)on4)C2)COC3)=O)CCCc2ccccc2C1 C(=O)(CCCC1CCCO1)NCCN(C(=O)C(C)C1CC1)C(C)C N1(C(C2(C)CCOC2)=O)CCCC(F)(C(=O)NC2CC(c3ncc[nH]3)C2)C1 C(=O)(CC(C)(C)C(C)(F)F)N1CCN(C(C(C=C=C)C)=O)C(CCOC)C1 C1(S(C)(=O)=O)(CN2CC(=O)N(CC(C3CCCC3)OC)C2=O)CCOCC1 C(C1CCc2cccnc21)NC(C1C=CCCCC1)=O O=C(C1CCc2c(Cl)cccc21)NC1C2CC1N(C(C1CCCC(O)C1)=O)C2 C12(C(=O)NCC(C(C)C)=O)COCC1CN(c1ccccn1)C2 C(=O)(C(S(C)(=O)=O)C1CC1)NCCN(C(c1[nH]c(C)cc1C)=O)CC S(=O)(=O)(c1ccc(Cl)s1)N(C1CCS(=O)(=O)C1)CC1CCC2(COC2)O1 C(=O)(CCCc1cn(CC2CCCN2C(=O)C(C)NC(=O)CC)nn1)OCC c1(C(N2CCC(F)(CF)C2)C(=O)NCCC(=O)OCC)csc([N+](=O)[O-])c1 N1(C2C(c3cn(-c4ccc(C=O)nc4)nn3)CC2)CCC(C2CCCNC2)CC1 C(=O)(C1SCc2cccnc21)NC1CCN(C(CSCCC(C)C)=O)CC1O C1(CC)CN(C(c2cc(C)sn2)=O)CCC1CNC(=O)C(O)c1ccsc1 C1(CCNC(C2CC(=O)N(O)C2)=O)COCCN1C(c1ccc(O)cc1)=O c1(C(=O)NC2(CNC(CCN(CC)CC)=O)CC2)ccncc1 c1(C(=O)NC(C)(C)CCNC(=O)CCC2CCOC2)ncc(Cl)cc1F C1(NC(C2C(CNC(C(C)(C)NC(=O)OC)=O)CCC2)=O)CCOCC1(C)C C=C(C)CC(C(=O)NC(CCC)CCO)NC(C1CCCCO1)=O c1(CC)nocc1C(=O)NCCC(C)(C)NC(=O)C(C)OCCN(C)C CCCCCCC(C)CC(=O)NCC1CN(C(=O)CCc2cc(C)on2)C1 C(=O)(C1=C(C)CCCC1(C)C)NCC1OCC2(CN(C(C3C(CCC)C3)=O)C2)C1 N1(C(c2ccc(Cl)o2)=O)CC2CCN(C(=O)CCCOc3ccc(Br)cc3)C2C1 c1(OCC)cc(NCCCNC(c2coc(Cl)n2)=O)ncn1 c1(CC(CN(C)C(c2cccs2)=O)NC(C2(Cl)CC2(F)F)=O)ccccc1 c1(CC)ccc(OC2CCCC(NC(=O)Nn3cnnn3)C2)cc1 c1(C(=O)OC)cc(CN(C)C(c2nc(CN3CCCCC3)no2)C)no1 c1(C(N2C3C(NC(C(C)C)=O)C(C3)C2)=O)oc2ccccc2c1CO N1(C(c2cnc(SC)n2C)=O)C2CCC1C(C)C(NC(=O)CCn1ccnn1)C2 CC1=C(C(=O)NC2CCC(NC(=O)CCCOc3ccc(F)cc3F)C2)CCC1 c1(OC)cc(C(N2CCCCC2c2cccc(O)c2)=O)cc(OC)c1OC CC1(C)CCC(CO)N(C(c2c[nH]nc2CNC(=O)CCCC2CCC2)=O)C1 c1(C(=O)NC2C(CNC(c3c(C4(C)COC4)noc3)=O)CC2)ccc(=O)oc1 Cc1cccc2c(C(=O)NC(C34CC(CO3)C4)C)coc12 C1(C(N(CCCNC(c2onc(CC)n2)=O)C(C)C)=O)CCc2nc[nH]c2C1 CC1(C(N2CC(NC(c3cc(O)cc(O)n3)=O)C(O)C2)=O)CCC(=O)NC1 C1(C(N(C)CC2CCCCN2C(=O)Cn2ncnn2)=O)CC12CCCCC2 N1(C(CCCCC#C)=O)C(CNC(c2cc3n(c2)CCC3)=O)CC2CCCC12 N(C1CCc2cc(CNC(c3nn(C)nc3C)=O)ccc21)C(C=C(CCC)C)=O N1(C(c2ncc(C)cn2)=O)CCCC(F)(CNC(c2cnn(CC(F)F)c2)=O)C1 N1(C(C(C)NC(CC)=O)=O)CCC(COC)(CNC(=O)C(F)(F)C(C)O)CC1 Cc1cc(C(=O)NCCCCCCNC(c2cnc(Br)s2)=O)c(C)o1 C1(NC(=O)NC(CC(=O)OC)C2CC2)CCN(CCC(C)F)CC1 C1(NC(C(COC)OC)=O)CCCCN(C(c2ccncc2C)=O)C1 N1(C(CC(C)C)=O)CC2CCC(C1)N2C(c1c[nH]c2ccccc12)=O Cc1cc(CC(=O)NC(C)CN(C)C(C2OCCCO2)=O)no1 c1(C(=O)NCC2CCN(C(C(CC)(C)CC)=O)CC2O)cnn2c1CC(F)(F)C2 N1(C(CCC(=O)OCC)=O)C2CCC1C(NC(=O)C(CC)n1cncn1)C2 c1(C(N(CC(CC)NC(COC2CN(C(C)=O)C2)=O)C)=O)coc(S(C)(=O)=O)c1 C=CC(CC)CC(=O)N1CCC(C)(NC(=O)Cc2cc(O)nc(O)n2)C1 c1(NC(C(N2CC(c3cn(CC)nc3)OCC2)=O)=O)cc(O)cc(O)c1 c1(OC)ncc(Cl)cc1C(=O)NCC12CC(NC(=O)Cc3cccs3)C(CO1)C2 c1(C(=O)NC2CN(C(C3(C(CC)(F)F)CC3)=O)CC2O)ccc(F)c(C(C)C)c1 C(CC(O)CC(=O)NC12CC1CN(C(=O)C=CC1CCCN1C)C2)SC CCCCCCC(=O)N(C1CCCN(C(c2ncn(C)c2C)=O)CC1)C N1(C(c2cnn(CC3CC3)c2)=O)CC2CN(C(c3ccn(C4CC4)n3)=O)CC2C1 N1(C(C2N(C(C3N(C)CC3)=O)CC(F)(F)C2)=O)CCC2(CCOC2)C1 N#CC1CC(c2nnnn2C2CCC2)(NCCCN2C(=O)CCC2=O)C1 c1(CC(=O)NCC#CCNC(C23CCCC2C3(F)F)=O)ccc(Cl)cc1F C(=O)(C1=COCC1)NC(C1(CNC(c2ccc(N3CCOCC3)nc2)=O)CC1)C C1(O)(C(N(CCNC(C(C(C)C)N(C)C)=O)CCOCCO)=O)CCCCCC1 C1(C(=O)OCC)CCC2(CCN(C(C)CC3CCCOC3)CC2)O1 N1(C(c2ccn(C)n2)C(=O)NC2(C)CC2)Cc2ncsc2C1 C(C)(C(CC(=O)N(C1CC(O)C1(C)C)C)NC(=O)C(C)(F)F)OC c1(CC(=O)OC)cc2c(s1)CCOC2=NC(=O)C1(N2CCC(C)C2)CC1 N1(C(C2(CCNC(C3(C#N)CCOC3)=O)CC2)=O)CC(=O)N2CCCC2C1 c1(CC)cnc(C(=O)NC2CCCCC2CNC(C2CC(C)CO2)=O)cn1 c1(NC(=O)NCCCc2ccc(Br)cc2)ccc(I)c(Br)n1 N1(C(Cc2ccc(C(C)(C)C)cc2O)=O)CCN(C(=O)C(Cl)=CCl)CC(O)C1 C(=O)(C(C)(C#N)CC)N1CCCC(N(C(c2c(CC)oc(C)c2)=O)C)C1 c1(C(=O)NC2(C)CN(C(C3C(CCOC)C3)=O)C2)ccc(CCN(C)C)cc1 Cc1ncc([N+](=O)[O-])n1C(C)C.C(=O)(C(C)C)N(CC(=O)N(C)C(=O)NCCCC(=O)C)C=O C1(CNC(C(Cc2ccc(OCC)cc2)C)=O)CN(C(=O)CO)CCN1C C1(C)(NC(COC)=O)CCCN(C(c2n[nH]c(C)c2Br)=O)C1 C1(CCC)CN(C(=O)CN2CCNC(=O)C2)CCN1C(=O)C(CO)OCC C1(NC(c2c(C)csc2)=O)CCCCC1CNC(C1CS(=O)(=O)C1)=O CC1(C)CC(O)CCN(C(C2CC3CC2CN(C(c2cncc(F)c2)=O)C3)=O)C1 N1(C(C(C)(C)C2CCCN2C(=O)C=CC(F)F)=O)CC[Si](C)(C)CC1 C1(N=c2cncc(Cl)[nH]2)(CNC(c2ccc3c(O)ncnc3c2)=O)CCCC1 Cc1nn(C)cc1C(=O)N(C1CN(C(=O)C(C2CCCO2)OC(C)C)C1)C N1(C(CCC)=O)CCCC(C(N2CCN(C(=O)CCn3cncn3)CC2)=O)C1 C1(NC(C(C)OCCCC)=O)CCC2(CCN(C(=O)CC(C)(F)F)C2)C1 c1(CC(=O)NCC2CCN(C(C34CCC(OC)C3C4)=O)C2)ccc2c(c1)CCC2 c1(C(=O)NCC(C(=O)NCc2c(OC)n(C)nc2)C(C)C)cc(C)cc(C#N)c1 C1(C(=O)NCC(C)NC(c2cnsc2)=O)SCCCN1C(=O)OC(C)(C)C N1(C(CNC(=O)Cn2cccn2)=O)CCN(C(C2CCC(=O)O2)=O)CC1 c12cc(n(C)n1)OC2=O.N1(C(COC)C)CCCC(OC)C1 Cc1ccccc1OCC(N1CCCC1CNC(=O)Cc1c(C)cnn1C)=O C=CCN=C(NCCC(C)(C)C(=O)OC(C)(C)C)N(C)CC1CCCO1 N1(C(CN(CCC#C)C)=O)CCC(NC(=O)CCCN2CCCC2)CC1C C1(OC)CN(C)C(C)(C(N2CCC(C(C)NC(c3cccnc3F)=O)C2)=O)C1 N1(C(CCNS(CC)(=O)=O)=O)CCCC(C)(C)C1CNC(C1CCCS1)=O N1(C(C(C)NS(CCCC)(=O)=O)=O)CCN(C(=O)CNC=O)CC1CO C1(C2=CCNCC2)(CN(C(C)(C)C)Cc2c(OC)cccc2)CCOCC1 CC1(C)C(C(=O)NCC2(O)CSC2)CCN1C(=O)C1=COCC1 c1(C(N2CCC(Cc3ncc(Br)cc3Cl)C2)C(=O)NCC)nccc(Cl)c1Cl CS(=O)(=O)CCCCC(=O)NC1CC2CC(C1)N(c1ncnc(=N)[nH]1)C2 C(C(C)(C)C(=O)NCC(c1ccccc1)NC(C1CCCC(O)C1)=O)SC N#Cc1cc(F)cc(NNC(=O)NC2CC2NC(=O)OC(C)(C)C)c1 Cc1cc(N2CCCC(NC(=O)C(c3ccccc3C)C3CCCC3)C2)n(C)n1 CC1(C)CN(C(=O)C2=CCC(F)(F)CC2)CC(CNC(c2sccc2F)=O)O1 C=CC1(C(=O)NC(c2scnc2C)C)CCN(C(c2ccc(O)cc2F)=O)C1 C1(C(NOCc2cn(-c3cc(C)c(Cl)cc3)nn2)=O)CCC(=O)CC1(C)C CC1C(NC(=O)CCCCc2ccccc2)CCCN1Cc1ccccc1 N1(C(CC(=O)NCC#C)=O)CCC(C(=O)NCCN(C)CCF)CC1CC C1(CC)CC(O)CCN1C(=O)CN1CCN(C(C2CCCC(=O)N2)=O)CC1 C1(CN(C(C2(CC=C)CN(C(C3CCCC3OC)=O)C2)=O)C)CCCN(C)C1 CC1CC(NC(c2ccccc2)=O)CCN1Cc1ccccc1C(F)F C#Cc1cccc(CC(=O)NCCNC(c2ccc([N+](=O)[O-])s2)=O)c1 c1(C(=O)NCCC(=O)NC(C#C)COC)nonc1N n1(CC)nc(C(C)C)cc1C(=O)N(C)CC1(NC(C23CCC2CC3)=O)CC1 c1(CC(=O)NCCN(C(C2CCOC2C(F)(F)F)=O)CC)ccc(F)cc1 C12(NC(CN(C3CC3)CC)=O)CCC(CC1NC(c1ccc(C#N)cn1)=O)C2 Cc1ccc(C(=O)Nc2cccc(C(C)(F)F)n2)cc1 c1(C(=O)NC2CC(C)(CNC(=O)CS(N)(=O)=O)C2)ccc(F)c2ccccc12 c1(C(N2CCCC(N(C(=O)C(C)C#N)CC)C2)=O)cccc2c1OCCCO2 Cc1c(CN2CCC(c3ccccc3)C2)sc2ccc(F)cc12 c1(C(=O)OC)cnn2c(C(=O)NCC(CC)(CC(C)C)SC)ccnc12 Cc1cnccc1CCNC(=O)CC1CC1CNC(=O)C=CC1CCOCC1 c1(C(=O)NC2(C#N)CCN(C(c3ccccc3Br)=O)C2)ccc([N+](=O)[O-])cc1 N1(C(C(C=C)(C)CC)=O)CCc2ccccc2C(N(C)C(=O)CCC2CCC2)C1 NC(=O)C(CO)NC(=O)CO.C1(=O)C(F)CC2CN1C2.C1(=O)CCN1 C1(C(=O)NC2CC(CNC(C(C)NS(CC)(=O)=O)=O)C2)CC2(CC2)CO1 CCCCCCC(=O)N1CCN(C(=O)CNC(C2CC2(Cl)Cl)=O)CC1 C(=O)(CCCC(F)F)N(C)Cc1c(CNC(COCCN(C)C)=O)cccc1 Cc1nn(C)cc1SCCN1CCC(NC2CCC(C(F)(F)F)CC2)CC1 Cc1cc(C(=O)NCC(C)CNC(=O)CSc2ccc(C)c(C)c2)c(N)cc1F N1(C(C=C(CC)C)=O)CC(C)(C)C1C1CCN(C(c2nnc(C)s2)=O)CC1 C1(C(N2CCC(=CCNC(c3c(OC)noc3C)=O)CC2)=O)CCCNS1(=O)=O Cc1ccc2c(ccn2CCC(=O)N(C(C)CN(C)C(c2cscn2)=O)C)c1 CCCC(C)CC(=O)N1CCC(NC(c2cccc(-n3cnnn3)c2C)=O)CC1 N1(C(c2nc(Cl)cc(N)c2Cl)=O)CCCC12CCN(C(C1CCCOC1)=O)C2 C(CN=c1[nH]c2cc(F)cc(F)c2o1)C1CCC(NC(C(CC)(C)CC)=O)C1 C1(CNC(=O)C=Cc2cc[nH]n2)CCCC1NC(c1c[nH]nc1F)=O c1(C(=O)NCC(C)(C2CC2)NC(CN(C(C)=O)C)=O)cnc(C2CC2)cc1C c1(OC)ccc2sc(-c3nc(C(=O)Nc4cccn5ncnc45)c(C)s3)cc2c1 C(C(=O)N1CCCCC1CNC(c1csc(C(=O)OC)c1)=O)(C(C)C)NC c1(OC)cc(C=CC(=O)NCC2CC2CNC(c2ocnc2C)=O)sn1 CCC(O)C(C)(C)C(=O)N1CC(NC(c2cc(C)c(C)o2)=O)C(F)C1 C1(C(=O)NCC2(O)CN(C(=O)C=C3CC3)C2)CCC2C1C2(F)F c1(C(=O)NCCOC2CCN(C(C(C(=O)OCC)(C)C)=O)C2)cccc2ccoc12 C=C(Cl)CC(C(=O)NC(C)C(C)(C)OC)NC(=O)CC1OCCC1(C)C c1(NCC2(CNC(c3cnc[nH]3)=O)CC2)nc(Cl)[nH]c2ncnc1-2 c1(C(=O)NC2CCCCCN(C(CC(=O)N(C)C)=O)C2)c[nH]c(=O)c2ccnn12 c1(C(=O)NCC(CC)NC(C2CCCC2(C)C)=O)cnc2ccnn2c1O C=CC(C)(CC)C(=O)NC(CC)CCC(=O)N1CCC(F)C(F)C1 N1(C(c2ccn(C)n2)=O)CC(F)CC1CC(=O)NC1CCC1 CC(C)C(C)CC(=O)N(C1CCCN(C(C2CCC3(CC3)C2)=O)C1)C c1(C(C(=O)NC2(COCC=C)CCC2)=O)ccccc1OC(C)C(=O)OC CCC(C)(CC(=O)NC(CO)C(C)NC(c1c(C)cc(C)cc1C)=O)C(=O)OC C1(NC(C(CCC)C(C)C)=O)CC2CCC1CN(C(=O)Cc1ncn(C)c1C)C2 C(=O)(CC(C)CC(C)C)NCC1CCCC(NC(CNC(=O)OCC=C)=O)C1 CCC(C)C(C(=O)N(CCNC(c1cc(C(F)F)n(C)n1)=O)C1CC1)NC(N)=O CC1CCCn2cc(C(N3CC4CCC3C4NC(=O)CCC(N)=O)=O)nc21 c1(C(N(CCC(=O)N(C(C)C(N)=O)C)C2CC2)=O)cncnc1 c1(NC(COC)=O)ccccc1SC.c12[nH]ccc1[nH]c(=O)[nH]2 n1(C(C=C)C)ncn(CCN(C)CC)c1=S C(=O)(CC(F)(F)C(C)(F)F)N1CCN(C(c2ccc(C)cn2)=O)CC1 C1(NCc2cc(C)[nH]n2)CC(NC(C2CC(=O)NC(=O)C2)=O)C12CCC2 N1(C(c2nc(CC)oc2)=O)CC2COCC2(C(=O)N(CC(F)Cl)C)C1 N1(CCOC)CC2CCC1C1CN(C(=O)COC(c3ccccc3)C(C)C)CC21 Cc1cc(C(N2CC3C(CN(C(=O)CC4CSC4)C)C3C2)=O)c(C)o1 c1(CS(C)=O)cccc(C(=O)NCC=CCNC(C2(C)C=CCC2)=O)c1 C#Cc1ccc(CCC(N2CCOCC(NC(=O)C=CS(C)=O)C2)=O)cc1 c1(C(=O)NCC(CO)NC(C(CC(C)C)F)=O)ccc2[nH]c(=N)oc2c1 C(=O)(C1=C(C)OCCS1)N1C(C(N2CC3C(C(=O)OCC)(CC3)C2)=O)CCOCC1 c1(C(=O)NCC(CNC(CN(C(=O)OC)C)=O)O)cc2c(F)cc(C)cc2[nH]1 C#Cc1cccc(CC(N2CC(N3CCN(C(C4CC4F)=O)CC3)C2)=O)c1 N1(C(CCC2C(C)=NNC2=O)=O)CC2(C1)CN(C(=O)CN(c1ccncc1)C)C2 c1(C(=O)OC)cc(C(=O)NCC2CCC(NC(=O)CCC3CC3)C2)ccc1F C(=O)(CCC(=O)N(C(C)CC)CC)NC1(C(=O)NCC)CC1C C1(NC(c2ccc(OC)s2)=O)CC2CC(C1)CN(C(=O)Cc1ccn(C)n1)C2 C1(=O)C(C(C)C)NC(=O)c2coc(n2)C(C)N1.C1(C(=O)OC)(CSC)CC1 c1(C(=O)CC2(C(N3CCC(CC(=O)OC)C3)=O)CCCCC2)cc2cccnn2c1 CCCC(C(=O)NC1CN(C(c2ncccc2CSC)=O)CC1F)S(N)(=O)=O Cc1cc(C(=O)NC2CCN(C(C3CNC(=O)C3)=O)C2)cnc1Cl CC1CN(C)CCN1C(c1cnn(C)c1C(F)(F)F)C(=O)NC(F)F C1(CCOC)(NC(C(C)=CC)=O)CCN(C(c2ccnc(C3CCC3)c2)=O)C1 c1(C(=O)O)cccc(S(=O)(=O)NC(c2ccc(=NCc3cnc(Cl)s3)[nH]c2)=O)c1 C(=O)(CCCS(=O)(=O)c1ccc([N+](=O)[O-])cc1)N1CCC(CN(CC)CC)C1C C(=O)(C(C)(C)C1=CCN(C(C2CC2(C)C(F)F)=O)C1)N(CC(C(=O)OC)C)C c1(C(=O)NC(C)CCCCNC(=O)Cc2cccn2C)cc2c(nn1)CCOC2 N1(C(CNC(C(C)(C)C)=O)=O)CCC2(CCCC2Nc2ncnc(Cl)c2F)C1 C1(C(=O)NCCCN2CCN(C(C3(CF)CC3)=O)CC2)(OC)CCCC(C)C1 N1(C(CC2N(C(c3ccn(CC)c3C)=O)C3C2CCC3)=O)CC(C)(C)OCC1C CCC(C)CCCC(=O)N1CCC(C(=O)Nc2cccc([N+](=O)[O-])c2)O1 c1(C(=O)NCC2CC(CNC(C)=O)OC2)cc(S(N)(=O)=O)cs1 C(=O)(C1=CC(C)(C)C1)N(C1CCN(C(C2CCN(CC(C)C)C2)=O)C1)CC N12CCC(CF)(C1)C(=O)NCC(C)C(=O)OCC2=O.CCC(C=O)SC CC(C)C(F)(CNC(C1CCOC1C(C)C)=O)C(=O)N1CCCC(O)(CO)C1 Cc1ccc(Cl)cc1-n1cc(C2(NC(=O)CN(C)CCO)CCC2)nn1 C1(CC)CN(C(=O)CCC(C)NC(c2cc(F)cc(F)c2)=O)CCCO1 c1(CC(=O)NC2CCC(NC(c3cnc(O)s3)=O)C2)cccc2nonc12 N1(C(CC2CC(=C)C2)=O)CCN(C(c2nocc2CC)=O)CC1CC Cc1cc(C(=O)NC(C2CCN(C(c3coc(Cl)c3)=O)C2)C)sc1Br C12(C(=O)NC(CNC(C3CC3(F)F)=O)C3CC3)CC3CC(C(=O)N1)C2C3 C1(CCNC(=NC)NC(C)CCC(=O)OC(C)(C)C)CCCN(C)C1 O=C(CS(=O)(=O)C(N1CCCC1)=O)N1CCOC(C(C2CCCC2)O)C1 c1(C(=O)NCC2(NC(CCCCSC)=O)CCCCC2)cc(C)cc2c1OCC2 S(=O)(=O)(c1ccc(OC(C)C)c(F)c1)NC1C(C(=O)OCC)CC(O)C1 c1(C(N2CCC(C)(NC(COC)=O)C2)=O)ccc(N)cc1C N1(C(C(CCC)O)=O)CC=C(C(=O)Nc2ccc(Cl)c(O)c2)C1 c1(NCC(C)(C)OCC)ncc(C)cc1S(=O)(=O)N1CCCC(OC(F)F)C1 c1(C(=O)Nc2ccc(C(=O)NC(c3cccc(F)c3)C)cn2)cccc(Br)c1O Cc1cc(C(=O)NCCc2cn(CC3CCS(=O)(=O)C3)nn2)c(C)cn1 C1(C(N2CC(CC(=O)OCC)C2)=O)CC2CC2N1C(=O)C(C1CCCCC1)F C(N=C(NC(C)C1CC1)N1CC=C(F)C1)c1c(COC)c(F)ccc1 CC1CN(C(c2ccnnc2)=O)CCN1C(=O)CC(=O)OC(C)(C)C N1(C(c2ncn(C(C)C)c2)=O)CC(C)CN(C(c2cnccc2C#N)=O)C(C)C1 CC1C(NC(=O)CCC2CC2(F)F)CCCN1C(C1CCC(C(N)=O)C1)=O Cc1cc(=NC(CNC(c2csnc2Cl)=O)C(C)C)[nH]c(Cl)n1 c1(C(=O)NC2CC(CNC(=O)C#CC3CCCO3)C2)ccc2c(c1)C(=O)NC2 C=CCC(CC)C(=O)NCC12CC(CN1C(=O)C(C)CCCc1ccccc1)C2 C(=O)(CC(CC)CC(C)C)N1CCC(C(=O)NC(CC#C)CCOC)CC1C C(N=c1[nH]cc(Br)o1)C1(CC#N)CCCC1 c1(C(=O)NCC(C(=O)NCC#CC)C)cccc(CC)n1 C(=O)(C1=C(C)OCCS1)NCCCN(C(CCC1C(C)=NOC1=O)=O)C CC1CCC(NC(c2cc(C3CC3)on2)=O)CN1C(=O)Cc1cn(C)nc1Cl c1(C(=O)NCC2(CNC(C3(C)CCNC3=O)=O)CC2)cc2c(nn1)CCOC2 C1(NC(CCC(C)C)=O)CCN(C(c2cnn(CC(F)(F)F)n2)=O)C(C)C1 c1(C(N2CCCC(CN3CCC(CO)CC3)C2)=O)cc(Br)cnc1Cl C1(NC(CCC(=O)OCC)=O)CCCC(NC(c2ncnn2CC)=O)CC1 N1(C(C2CCOCC2)=O)CC2CN(C(C3CC(F)(CO)C3)=O)CCC12 C1(NCCc2sc(C(=O)OC)c(C)n2)CCN(C(=O)OC(C)(C)C)C1C.OC C1(NC(CN(C(CN2CC(C)(C)C2)=O)C2CCC2)=O)CC(=O)NC1=O S(=O)(=O)(c1ccc(C)c(C)c1)Nc1cncc(C(=O)Nc2ncc(OC)nc2)c1 c1(C(N(CC(C)NC(=O)Cn2ccc(C)n2)CC)=O)nc(C2CC2)sc1Br N1(C(c2cc(C(C)(F)F)ncc2)=O)CCC(F)(F)C(CNC(=O)CS(C)(=O)=O)C1 C(N=c1cc(C)c(C#N)c(C)[nH]1)C1(CCC(N2CCCC(O)(CO)C2)=O)CC1.CO C1(C(N2C(C)CN(C(=O)Cn3cnc4ccccc34)CC2)=O)CC1C1CCCCC1 C1(CNC(c2c(Cl)cnc(C)n2)=O)CN(C(=O)C(F)CC2CC2)C2CCCC2O1 c1(C(N2C3CCC(CCNC(CCC4C(C)C4)=O)(C3)C2)=O)ccn2nccc2n1 c1(CC)nc(C(=O)NCc2cc(C(=O)NCc3ccoc3C)no2)cs1 C(C)(CC(=O)NCCC1(C(=O)NC2CC(CC(C)(C)C)C2)CCC1)OC CN1CC(C)(C)CC1C(=O)NCC1CCCN(C(c2cnoc2)=O)CC1 N1(C(=O)OC(C)(C)C)CCC(C2CC2)(C(=O)Oc2ccc(OCC(F)F)cn2)C1 c1(C(N2C(CC(=O)NCC=CCOC)CC2)=O)cnc(O)c(F)c1 N1(C(C2C(C)(C)C2)=O)CCC(CCC(=O)NCCCCCCO)C1 C(=O)(CC(C)Cc1cccc(F)c1)NCCN(C(c1c(C)noc1)=O)C(C)C C12(CNC(CS(CC)=O)=O)CCC1CN(C(c1cn(C(C)C)nn1)=O)C2 c1(CN(C)CC2CCN(C(c3nnn(C)n3)=O)C2)cc(S(C)(=O)=O)cs1 C(=O)(CCCCC(=O)NC)NC1C2N(C(C(C)OCC#C)=O)C(CC2)C1 N1(C(C2(C=C)CCOCC2)=O)CCc2c(CNC(=O)C(C)(O)C=C)cccc2C1 CCC(CN=c1[nH]c(N2CCN(c3cccnn3)CC2)nc2cc[nH]c12)OC C1(C(=O)NCC(C(=O)OCC)C)CCN(C(C2(CSC)CC2)=O)C1 N1(C(c2c(C)ccc(C)n2)=O)CCCC(C)(C)C1C(N1CCOCC(C)(C)C1)=O N1(C(CC2CCCN(C(CC3CCCC(C)O3)=O)C2)=O)CCCC(F)(F)C1 Cn1nnc(Br)c1C(=O)NCC(C1CCC1)NC(C1(CC2CC2)CC1)=O C1(C(F)(F)F)(C(=O)NC(CNC(C(C)NC(C)=O)=O)(C)C)CC=CCO1 CC(C)C(C(=O)NCC(C)(C)CNC(c1cc(CO)[nH]n1)=O)c1cccnc1 C(=O)(C(COC)(CC)CC)NCCNC(C1(COC)CCCOC1)=O c1(C(N(C(C)CNC(c2ncn(C)n2)=O)CC)=O)cn(C)c2ncccc12 c1(CC(=O)NCC2CC2CNC(c2ccncc2F)=O)ccc(F)cc1F Cc1cc(C)c(NC(=O)NC(CO)CCSC2CC2)c(=O)o1 N1(C(C(C2CN(C(CC(=O)OC)=O)C2)O)=O)CCOCC(C)(C)C1 c1(CC(C)NC(C2CCC2(F)F)=O)ccc(CNC(c2ccnn2C)=O)cc1 c1(COC)ncc(C(=O)NCC2(O)CCCN(C(c3ccsc3C)=O)C2)c(=N)[nH]1 c1(Oc2c(-c3n(CC(C)C)nc(C(N)=O)n3)nnn2C)c(C)cc(Br)cc1C c1(C(CC)=O)ccc(N2CCOC(C)C2)c([N+](=O)[O-])c1.c12ccc(cc1)[nH]2 Cc1cccc(O)c1C(=O)N(CCCOCCNC(C1CC2CC2C1)=O)C Cc1cc(NC(=O)CC2CCCN2C(c2c(Br)ccnc2Cl)=O)cnc1F N1(C(C2(C)CCN(C)C2)=O)CCC(O)C(N(C)C(C2CC(F)C(=O)N2)=O)C1 C(=O)(C(CCC(C)C)OC)N1CCCCC(CC=C)C1.C12CCCC1NC2=O c1(CC)ccc(CNC2CN(C(c3ccc(N4CCCCC4)nc3)=O)C2)cc1 C(c1ccccc1Br)=CC(=O)NCCCN(C)C(C1(C)C=CCC1)=O C1(CC=C)(C(N2CC(F)(F)C2)=O)CN(C(=O)COCCC)C1 N1(C(CCN(C)CC)=O)CCN(C(c2ccc(C(F)F)cc2F)=O)C(C)CC1C C1(O)(CNC(C(=Cc2ccncc2)C)=O)CCCN(C(c2nc(C)oc2C)=O)C1 N#Cc1cn[nH]c1C(=O)N(C1CCC=CCC1)C1CCN(CCF)C1 C1(N(C)C)CN(S(=O)(=O)N2CCCCC2CN)CC1OC c1(C(=O)NCCC(C)NC(c2cc(C)on2)=O)ccc(C(F)(F)C(F)F)cn1 c1(C(=O)NCCCN(C(C2CCN(C(C)=O)C2)=O)C)ccc(C)c(N)c1 C12(CNC(CCc3nc(C)sc3)=O)CC1CN(C(c1scnc1C(F)(F)F)=O)C2 N1(C2CCC(OCC(=O)NCC)C2)CC2CN(C(C3CC3(F)Cl)=O)CC2C1 c1(CC(=O)N(CCNC(C(C)=C(C)C)=O)C(C)C)csc(Cl)n1 CC1CC2CN(C(=O)CCCC(=O)NC3CC3)CC2N1C(=O)CC1COC(=O)N1 C12CCOCC1NC(=O)C2.CNS(=O)(=O)NCC(=O)NCCN(C1CC1)CC C1(CC=C)(NC(C2(F)CCOCC2)=O)CCCN(c2nccc(CSC)n2)C1 c1(CN(C(=O)C(Cn2cccn2)NC(=O)C(Cl)Cl)C(C)C)ccnn1C c1(NC(C2CC(NC(Cc3scc(C)n3)=O)C2)=O)ccc(C(F)(F)F)c(Br)c1 CCCS(=O)(=O)C(C)C(=O)NC(C)CN(C(=O)COc1cccc(C)c1)C Cc1ccc(C(C)NC(=O)CNC(C2CCCC2O)=O)cc1 C#Cc1ccc(C(=O)NCCN(C(=O)CCC(C)(C)C)C2CC2)c(C)c1 C(CCC(C)CC(=O)NCc1ccc(Cl)c(C(F)(F)F)c1)=C(C)C C1(COC(=O)NC)CCCCN1C(c1c(Br)cnn1C)=O c1(COC)ncc(CNC(c2nnnn2C)CSc2nc(C(F)(F)F)cc(Br)c2)[nH]1 CP(C)(=O)C1(C(=O)NCC2(NC(=O)C(F)C3CCC3)CC2)CC1 C(=O)(C(F)C(F)(F)F)N1CC(C(N)=O)(CNC(C(C)(C)OCC)=O)C1 C1(NC(CC2(OC)CC2)=O)CCCCN(C(=O)C=Cc2cccc(Cl)c2)CC1 c1(CC)[nH]nc(C(N2C3CCC2CC(NC(=O)CCCCF)C3)=O)c1[N+](=O)[O-] N1(C(C2(C#C)CC2)=O)CCC2(CC1)CN(C(C13CCCC1CCC3)=O)C2 c1(OC)ccc(C#N)cc1CNC(=O)C(=O)Nc1c(F)ccc(OC)c1F C1(NC(c2ccc3sncc3c2)=O)CN(C(=O)Cc2ccoc2)C2(CCCC2)C1 C#CC1(C(N2CCCC2CC(=O)NCC(c2nccs2)C)=O)CCCC1 c12ccc(cc1)NC(=O)C2N.c1(C(C)OCC)nc(C(F)(F)F)n[nH]1 Cc1ccc(C(N2CCCC(CNC(C3(C)CC3)=O)C2)=O)c2ncccc12 CCCC(C)(O)C(=O)NC1CCCC1NC(c1ccoc1CC(N)=O)=O C12(NC(CCC)=O)CCCCC1CN(C(c1sc([N+](=O)[O-])cc1Cl)=O)C2 Cc1sccc1C(=O)NC(C(=O)NCCOCCN(C)C)C1CCOC1 c1(NC(C(C)(N(C(c2cc(OC)n[nH]2)=O)C)C2CC2)=O)cncc(SC)c1 C1(C(=O)NC2C(CC(=O)NOCc3nn[nH]n3)C2)CC2CC1CC2O Cc1ccc(F)c(-c2cn(C3COCC3NC(=O)CCCN(C)C)nn2)c1Br CS(=O)(=O)CC(=O)N1CCCC(N2CCN(C(c3cccnc3)=O)CC2)C1 Cc1c(O)ccc(C(=O)NCC23CC2CN(C(=O)C(C)P(C)(C)=O)C3)c1C C1(C(=O)NC(C2CN(C(=O)C(C)(Cl)Cl)CCO2)C)CCCCCCC1 c1(CCC(=O)N(C2CCN(C(C(C)n3cncn3)=O)C2)CCO)ncc(F)cn1 C(N=c1[nH]c(NN(C)C)nc2c1COCC2)C1CC(C)C1.c12ccnc(c1)N(C)C2 C#CCCC(O)C(=O)NCC(C(F)(F)F)N1CCN(C(=O)C(C)(F)F)CC1 c1(CC(N2CCC(NC(c3n(COC)ncc3)=O)C2C)=O)ncn2c1CCCC2 C12(NC(CNC(NOCCSC)=O)=O)CCOCC1C2 N1(C(CC2CCCN(C(CC3(CC)CCC3)=O)C2)=O)CC(C2CC2(F)F)C1 c1(C(N2CC(NC(c3c(OC)cc(F)cc3)=O)C3C2C3)=O)ccc(Cl)c(F)c1O C1(C(=O)NCC(COCC)C)CCC(O)CN1C(=O)CC1CC(C)=NO1 N1(C(C(C2CC2)NC(c2ccccn2)=O)=O)CCC(F)CC1 Cc1ccc(N2CC(C(=O)NNC(C3CCC3C3CC3)=O)CC2=O)cc1 C(=O)(C(O)C(C)SC)N(CCNC(C1(COC)CC1)=O)C c1(C(C)C)cccc(CC(N2CCCC(N(CCO)C(C3CC=CCO3)=O)C2)=O)c1 O=S(=O)(c1ccc(Cl)c(C(F)F)c1)NC1CCCC1CF N1(C(C2(CC(C)C)CC2)=O)C2CCC1CC(O)(CNC(C1CCCSC1)=O)C2 C1(O)(CCNC(CCCN(C(C)C)C)=O)CCCN(C(=O)CCC2CC2(F)F)C1 c1(C(N2CC3CN(C(c4cc(Cl)cnc4Br)=O)CC32)=O)cnc2[nH]ncc2c1 C1(C(N2CCN(CCOC)CC2)=O)CCCN(C(=O)C(C)n2cccn2)CC1 C(=O)(C(O)CCC(F)(F)F)N1CCC=C(CNC(c2cc(C(C)C)no2)=O)C1 c1(OC)cc(C)ccc1OCC(N1CC(CO)C(c2ccccc2)C1)=O N1(C(CC(C)OC)=O)CCC(=CCNC(=O)C(C)(C)c2cccs2)CC1 CC(C)CN=C(NCC1C2CCCCC12)N(C)CCC1CCCO1 C1(CC(=O)NCCN(C(=O)CSc2n[nH]c(O)n2)C2CC2)CC2CC2C1 C(=O)(C(F)(F)CCn1cc(-c2ccc(F)cc2Br)nn1)NC1(C)CCOC1=O C1(C(N2CCC(CNC(C3COC(=O)N3)=O)C2)=O)(COC)CCOCC1 N1(C(C(C)NC(COC)=O)=O)CCN(C(c2ccnc(OC)c2Cl)=O)CCC1C C1(C)(CNC(Cc2cc(C)ns2)=O)CCCN(C(c2n[nH]c(C3CC3)n2)=O)C1 c12nc(c(Cl)cc1Br)CN2C.CCC(C)CC(C)NC c1(C(=O)NCC2CCCN(C(C(CO)OC)=O)C2)c(C)ncnc1C N1(C(C(C)c2cc[nH]n2)=O)CCOC(Cn2cc(Cn3ccccc3=O)nn2)C1 c1(OC)ccc(C)c(C(=O)NCC2(O)CN(C(c3sc(C)nc3C(C)C)=O)C2)n1 c1(C(N2CCC(N(C(=O)Cn3ccc(=O)cc3C)CC)C2)=O)ccc(Cl)nc1N C1(C)(CNC(C2(C)C(C)(C)C2)=O)CC(F)(F)CN1C(c1ccc(C(F)F)cc1)=O C1(CCNC(C(CC)OC)=O)CC2CCC(C1)N2C(c1nn[nH]c1C(F)(F)F)=O Cc1nc2cc(C(=O)NCC3(NC(=O)CNC(=O)CC(F)(F)F)CC3)ccc2s1 Cc1c(F)ccc(C(=O)NCCNC(=O)C(F)(F)C2CCCC2)c1C CN(C)N=Nc1ccccc1C(=O)NC1CN(C(C2CCOC2)=O)CCC1CO c1(OC)ccc(CC(N2CCC(CCNC(=O)C(CCSC)OC)C2)=O)cc1 N1(C(COCCCOC)=O)CCCOC(CNC(c2cccc[n+]2[O-])=O)C1 C1(CNC(CCc2cc(OC)no2)=O)C2CN(C(=O)Cc3cc(CC)no3)CC12 C1(C(=O)NC2CC(C)(NC(=O)CSc3ccccc3Cl)C2)(CO)CCCCC1 N1(C(C2CC(OC)C2)=O)CCC(C)(C)C1C(=O)NCCc1ccns1 Cc1cc(Cl)cc(C)c1C(=O)N(CC(O)CNC(c1ccsc1C#N)=O)C N1(C(c2ccccc2Cl)C(=O)NC2C(C)C2)CCC2(CCCC2)CC1 c1(C(N2CCC(CC(N3C(C)(CO)C=CC3)=O)C2)=O)nc(Br)ccc1Cl N1(C(=O)C2=CCC2)CC2CC(C1)CN(C(=O)Cc1ccc(OC(F)F)c(Cl)c1)C2 C1(CNC(=O)CCN2CCCC2)CCCCC1NC(c1cnoc1C1CCC1)=O c1(CC2(C)CC2)ccc([N+](=O)[O-])cc1.N12C(CO)CSC1CC2=O N1(C(CNS(CC)(=O)=O)=O)CC2CC1CN(C(=O)C(C)(C)NCS(C)(=O)=O)C2 c1(C(N(C2CN(C(C(CCCC)=O)=O)CC2F)C)=O)ccc2c(c1)C(C)(C)CO2 N1(C(c2nnn(Cc3cc(C)on3)c2C)=O)CC(C)N(C(=O)CC2CC2)CC1C CC(C)(C#N)CCCC(=O)NC1CC(CCC(=O)NCc2cccc(Cl)c2)C1 Cc1ccc(C(=O)OCCOC2CC(C)C2)cc1I CC1(CNC(=O)Cc2ccc(O)cc2)CCCN(C(C2CCO2)=O)C1 C1(NC(c2ccn(CCC)n2)=O)CCOCC1C(=O)NCC1(OC)CC1 c1(CCCN(C(=O)NC(C(C)C)C2(C)CC2)C2CC2)nc(-c2ccncc2)no1 C1(CC(=O)N(CC(=O)OC)C2CC2)CN(C(c2ccc(O)cc2)=O)CC1C N1(C(Cc2c(S(C)(=O)=O)cccc2)=O)CCC(C2=NOC(C(=O)O)C2)CC1 C1(c2c(C(=O)NCCC#N)c[nH]n2)CCCCN1C(c1ccc(Cl)cc1)=O C1(CCOC)CN(C(C2(CCOC)CC2)=O)CCN1C(C12CCCCC1C2)=O CC1=C(C(=O)N2CC(C)C(C)(CNC(=O)Cc3cc(C)cc(F)c3)C2)CCCC1 CCC1=C(C(=O)NC2CC2CNC(c2cnc(O)n2CC)=O)SCCO1 c1(C(=O)NC2(C)CCCN(C(Cc3c(C)cccn3)=O)C2)cc2ccccn2n1 c1(CC)ccc(C(N2CCN(C(c3cnn(C)c3CO)=O)C(CC)C2)=O)cc1F N1(C(C(C)CF)=O)CCC(O)(CNC(c2ccc(CC#N)cc2)=O)C1 C=CC1(CO)CCN(C(C2(C(C)C)CCCN2C(=O)C(O)C(C)(C)CC)=O)CC1 CC(C)(CCCNC(=O)C(C1CCCCCC1)F)NC(=O)C=CC1CCCCC1 C(C)(C(=O)NC1CCC(NC(c2coc(-c3ccccc3)n2)=O)C1)(C1CC1)OC C1(NC(=O)C=Cc2cc[nH]c2)CC2CC1N(C(c1ccccc1Cl)=O)C2 C1(C(N2CC(CN(C(COC(C)C)=O)C)OCC2)=O)CC12CCSCC2 c1(CC)nccnc1C(=O)NC1CN(C(C2(C(=O)N(C)C(C)C)CC2)=O)CC1C c1(N2C(CCNC(C(C)(C)O)=O)CCC2)ncnc2ccc(C(F)(F)F)cc12 CCCCC(C(=O)NC)NC(=O)CONC(C1CCN(CC)C(C)C1)=O C(C1CCCN1C)=CC(=O)NC1(C(=O)NC2(C(N(C)C)=O)CC2)CC(CO)C1 C1(N(c2ccnc(C)n2)C)CC2CCC(C1)N2C(c1ccc(=O)n(O)c1)=O C#CC(CNC(=O)C(F)(CNC(=O)Cc1cnn(C)c1)C(C)C)CC(C)(C)C N1(C(c2c(C)ccc(C)c2)=O)CC2(COC(=O)C2)C1.n12cc(nn1)C(=O)NOCC2 N1(C(=O)C2=COCC2)CC2CCN(C(c3cc(F)c(F)cc3O)=O)CCC2C1 Cc1cc(=NCC(F)(F)C(C)C)[nH]cc1S(=O)(=O)N1CCCC(NCCO)C1 CC(C)CC(C)CC(=O)NC(C(N1CCC(CN=[N+]=[N-])CC1)=O)c1cccs1 c1(CC)cc(=NCC2OCCC2NCCn2cccn2)[nH]cn1 C(=O)(C1CCCc2c[nH]nc21)N1CC2(CC(NC(CC(C(C)C)OCC)=O)C2)C1 N1(C(CCCC=C)=O)CCCC(CNC(=O)CC2CCCC(OC)C2)CC1 c1(C(N2CC(N(C)C(C3CC3(C)C)=O)C(F)C2)=O)occ2c1CCC2 c1(C(=O)NCC(C(C)C)NC(=O)CC2CCCN2C)cc(O)nc2c1CCC2 C(=O)(C1=C(Cl)CCOC1)NCC1C(C(=O)NC2C(C)(CO)CCC2)CC1 C=C(C)CCC(C)N=c1[nH]c2c(c(=NCCCc3ccccn3)[nH]1)CC(C)CC2 c1(SCCC)ccc(C(=O)NCC2(F)CCN(C(=O)C(C)c3ccsn3)C2)cc1 c1(C(C)(C)C#N)cncc(NC(C2(C)CCCN2Cc2cccc(O)n2)=O)c1 Cc1cccc(C(O)C(=O)NC2C=CCN(C(=O)Cc3coc(C)n3)C2)c1 c1(C(C)C)ccc(C(=O)NC(C)(CNC(=O)C(=O)NCC(F)F)C(C)C)cn1 c1(C(=O)NCC2(CNC(c3ncc[nH]c3=O)=O)CC2(F)F)cc2ccccc2s1 CC(CC(C)NC(C1CCCN1C1CC1)=O)NC(=O)C(C)NC(c1ccco1)=O Cc1cc(C)c(C(N2CCC3C(NC(C4CCCC(=O)N4)=O)C3C2)=O)cn1 C(C(C)(C)C(=O)NC1C2CC1N(C(c1ccc(O)cc1)=O)C2)OC.C(C)(C)OC(C)C Cc1oc(C)c(S(N)(=O)=O)c1C(=O)NCC1CC1CNC(=O)CC1CC1 c1(CN(C)C)nnsc1CNC(C1(CC)C(CCCC)CC(O)C(=O)N1C)=O C(=O)(C(CCC(C)C)NC(C1CN(C)CCO1)=O)N(C)Cc1c(CC)noc1 Cc1ncnc(C)c1C(N1CCN(C(=O)C(=O)NC(C)C)CC1C1CCC1)=O Cc1cc(C(=O)NC2CCN(C(c3ccccc3N(C)C)=O)C2)c(Br)s1 CC(C)C(C)(CNC(=O)Cn1nnnc1C(C)C)NC(C1(O)CC1)=O N1(C(CCNC(C(c2cccnc2)C)=O)=O)CCC(O)C(CO)C1 Nc1ccc(Cl)nc1C(=O)NCC1(CCNC(c2cc(C3CCC3)on2)=O)CC1 c1(C(=O)NC2CC(N(C(CCC(=O)NC)=O)C)C2)cc(O)cnc1Cl c1(C(N2CC3C(NC(C(CCSC)(C)C)=O)(C3)C2)=O)cnn2cccnc12 N1(C(c2cc(OC)ns2)=O)CC(C)N(C(=O)Cc2ccsc2C)CC1C C(=O)(C1=C(C)CCCC1)N1CC(CCC)N(C(=O)CCc2ccc(C)o2)CC1 Cc1c(O)c(=O)ccn1CC(N1CCC(OCCNC(=O)C#CC2CC2)C1)=O c1(C(=O)NC2C(C)CN(C(C3CCC(=O)N3)=O)C2)c(F)cccc1[N+](=O)[O-] CCCCCC(O)C(=O)NCCOCCCN(C)C(c1c(C)cc(C)nc1O)=O Cc1cc(=NC(=O)c2ccccc2-c2ccc(C)c(F)c2)[nH][nH]1 C1(C(N(CC(=O)N(C)Cc2ccnn2CC)CCC)=O)CCC(CO)CC1 C1(N(C(C(=Cc2cccnc2)C)=O)C)CCCN(C(=O)C(C)(C)CC2CC2)CC1 CC(CNC(=O)NCCn1ccnc1)Cn1ccnc1 N1(C(C(C)(C)O)=O)CCC(CO)(NC(=O)CCN2CCC(F)C2)C1 Cc1oc(C(N2CCC(C(C)NC(c3cnsc3C)=O)C2)=O)cc1CO CC#CCC(C(=O)NCC=CCl)NC(c1cn(CC)nc1C)=O c1(C(=O)NC2CCN(C(Cc3nc(C)sc3)=O)C(C)C2)coc2c1C(=O)NCC2 C1(NC(=O)Cc2c[nH]nc2O)CC(O)CN(C(c2c(F)cccc2Cl)=O)C1 c1(C(=O)NC2CC3CN(C(C(C)NC(CC)=O)=O)CC32)cccc(S(N)(=O)=O)c1 C12(C(=O)NCC(CNC(C3(C(=O)OCC)CCC3)=O)O)CCCN(CCC1)C2 C(=O)(C(C)(C)CC1CC1)N(CC(C)(C)CNC(C1CCC1F)=O)CC c1(NC2CCN(C(c3c(C)cc(OC)nc3)=O)C(C)C2)nc2cc(Br)cnc2s1 C1(C(N(C2CCCN(C(=O)CNS(N)(=O)=O)CC2)C)=O)CCC(C2CCC2)CC1 CC1C(C)N(C(c2cnc3n2CCCC3)=O)CCN1C(=O)CSc1nccn1C N1(C(C(C)=CC)=O)CCOC(CCCNC(=O)C(C(C)C)NC=O)C1 C(N=c1[nH]c(=N)[nH]c(=NC(C)C2CCCCC2)[nH]1)C1N(CCCC=C)CC1 C1(Cn2c(N3CCCC(C)(C)C3)nnc2Cn2nccn2)CCn2nccc2C1 N1(C(c2cccc(C(=O)NC)n2)=O)CC(NC(c2cc(CO)[nH]n2)=O)CCC1C C(=O)(C1=CC2CC(C1)CC2O)N1CCC(CCNC(CN(C)C)=O)C(F)(F)CC1 C1(CNC(C(c2cc(C)cc(F)c2)C)=O)CC2COCC2N1C(c1ccon1)=O C1(F)(CNC(CCCC#C)=O)COCCN(C(c2cc(C)ccc2C(C)=O)=O)C1 C(CCCCC(=O)N1CC(N(C)C(C2CC2C2CC2)=O)C2(CC2)C1)SC c1(CC)oc(C)cc1C(=O)NCCCC(C)(C)NC(C1CC1c1ccccc1)=O C1(NC(C(F)OC)=O)CCN(C(c2ccc(Cl)nc2N)=O)C12CCC2 C(CCN(C)C)(C(=O)NCc1ccc(OCF)cc1)NC(C(C)OC1CCCC1)=O CC#CCC(C(=O)NC1CN(C)CCC1O)NC(c1oc(C)nc1C)=O Cc1cc(C(=O)NCC2COCCN2C(c2ccc(Br)o2)=O)ccn1 c1(C(N2CC3C(CNC(c4c(C)nsc4)=O)(C3)C2)=O)nc(Br)cnc1N C1(NC(c2ccc(CC(C)(C)O)s2)=O)(CO)CCCN(C(=O)CN(C)C2CC2)C1 C(=O)(CCCC(C)=O)NCC1C(CC(N2CCCC(CC=CC)C2)=O)C1 C12(NC(C(CC)NC(C)=O)=O)COC(CC3CC3)(C1)C2.C1(=O)C=CC(=O)N1 N1(C(C(CC)OC)=O)CCC(C2(NC(=O)CC(C)(C)OC)CCC2)CC1 CC1(C)C2CCC(C2)C1C(=O)NCC1(Cn2cc(-c3cn[nH]c3)nn2)CC1.OCC C(CC(C)C(=O)N1CCC=CC1C(=O)N(C)Cc1cscn1)=CCC C1(NC(C(N2CCCC(N3C(=O)CCC3)C2)=O)=O)C2CC3CC(C2)CC1C3 c1(CC)nc(C)[nH]c1C(=O)NC(C)(C)CN(C(=O)CSCCOC)C Cc1cc(C#N)c(NCC2NCCC2C2CC2)cc1F Cc1cc(C(N2CCOC(C(C)NC(c3ccc(CO)o3)=O)C2)=O)nn1C Cc1ccc(Br)c(C(=O)NC2C3CCN(C(C4CC(N(C)C)C4)=O)CC23)n1 C1(CC)CN(C(C2CC(NC(c3ccc(F)cc3)=O)C(O)C2)=O)CC1O C1(CCNC(CSC)=O)C(C)CCCN1C(c1cnc(O)c(C)c1)=O N1(C(CN(C(COC)=O)C)=O)CC2CCN(C(=O)C(C)S(N)(=O)=O)CC(C2)C1 c1(C(N(CC(C(=O)NCC=CCC(=O)OC)C)C)=O)ccc(C#N)o1 c1(COC(N2CC(O)(C(C)C3CC3)C2)=O)cc2ccsc2n1C n1(C(C)C)ncc(=NC(=O)C2CC(=O)CN2C(C2C3CCC(F)C23)=O)[nH]1 N1(C(C2(C)C=CCC2)=O)CC2(COC(CNC(c3cc(C4CCC4)no3)=O)C2)C1 CC(CCc1ccccc1F)C(=O)NCC#N C1(C(C)(C)C)CCC(=CC(=O)NCC2CC(C)N(C(C3CC=CC(O)C3)=O)C2)CC1 C1(CC(C)C)CCCN(c2nnc(C(C)(C)C3CC3)n2CC2CC2)C1 C(=O)(C1=CC2C=CC1C2)NCC(CCC)C(=O)NCCC(=O)NC C(=O)(CCCN=[N+]=[N-])NC(CNC(C(c1cccs1)SC)=O)(C)Cn1cccn1 c1(C(N2CCC(OCCNC(C3CSCCS3)=O)C2)=O)cc(F)cs1 CCC(CC)C(C(=O)NCC1CCN(C(=O)C(F)(F)c2ccncc2)C1)OC N1(C(CS(=O)(=O)NCC)=O)CCC(NC(C2(CO)CC2(F)F)=O)C(CC)C1 c1(C(=O)NC2C(C)N(C(=O)CC3CC34CC4)CCC2)ccc2ncsc2c1 C(CCO)(C(C)(C)CN(C)C)NC(N1CCCC(c2cccs2)C1)=O C1(CC#C)(Oc2ccccn2)CCN(C(=O)NCCN(C)CCC)CC1 N1(C(C(c2ccco2)NC(C2CC3(CC3)CO2)=O)=O)CCCN(C2CC2)CC1 Cc1nc2ncccc2cc1CC(=O)N(CC(O)CN(C)C1CC1)C N1(C(CCCNC(C)=O)=O)CC2(CC(C(N3CCC(C)(C(N)=O)C3)=O)CO2)C1 CCC(CC(F)F)C(=O)N1CCC(C(N2CC3(C2)CN(C)C3)=O)CC1 c1(OC)ccnc2c1CCN(C(=O)Nc1cc(C)ncc1C#N)C2 c1(NC2(C)CC(NC(C(Cc3ccccc3)OC)=O)C2)ncnc(C)c1Br C1(C(=O)NCCCC=C2CN(C(c3ccc(F)cc3F)=O)C2)CC2C(C1)C2(F)F c1(OC)cc(C(=O)NCC2CN(Cc3cc(F)c(F)cc3C)C2)ccc1C#N Cc1nc2ccc(-c3cn(CCNC(c4cnccc4N(C)C)=O)nn3)cc2s1 C1(C(N(CC(CN(C)C(c2ccc(O)c(N)n2)=O)O)C)=O)CCC2(CC1)CC2 N1(C(=O)CCOCC(F)F)CCCC(F)(CNC(C2(N(C)C)CC2)=O)CC1 c1(C(=O)NC2C(NC(Cc3cc(C)[nH]n3)=O)CCC2)cccc(Br)c1N c1(OC)ccc(Cl)cc1CC(=O)NC(CNC(C1CCC1(C)C)=O)C1CC1 C=C(C)CCCC(=O)NCC1(NC(=O)Cc2cnn(C)c2)CCC1 C(c1ccccc1C#N)=CC(=O)NC1CC(C)(NC(c2c(C)oc(Br)c2)=O)C1 CC1=NOC(C(=O)NC(C2CCN(C(=O)CSc3nncs3)CC2)C)C1C N#CCCCCC(=O)NC1CCCCC1CNC(c1cn(C2CCCC2)nn1)=O Cc1ncc(C(N2CCC(C(N3CCC(C)(O)C3)=O)C2)=O)c(C)n1 C1(NC(c2cc(C3(C(C)(C)C)CC3)n[nH]2)=O)CC2CC1N(C(=O)Cc1ccsc1)C2 c1(C(N2C(C)CC(NC(C3CC(=C4CCC4)C3)=O)C2)=O)cc(S(N)(=O)=O)c[nH]1 C1(C(=O)NC(c2cnn(C)c2)CC)CC(NC(C2CCC3(CC3)C2)=O)C(O)C1 c1(CC)nc(C)c(C(N2CCC(CNC(=O)CN3CCNC(=O)C3)C2)=O)c(C)n1 CC1CN(C(=O)Cc2cn[nH]c2)CCC1N(C(=O)COC1(C)CCC1)C CCCC(O)CC(=O)NC1CCC1NC(c1ccc(N)cc1F)=O N1(C(CCNC(C)=O)=O)CC(CO)C2(CCN(C(=O)C=C3CCC3)CC2)C1 c1(N2CC(NC(c3nn(CC)c(C)c3)=O)(CO)C2)ncc(C)c(O)n1 c1(OC)ccc(CN2CCC2C2CC2)c(OC)c1 C1(NC(C(C)(CO)NC(C(C)C)=O)=O)CC2(C1)CC(CO)C2 c1(C(=O)NC2CC2)ccc(-n2cc(Cn3cc(C4CCC=CO4)nn3)nn2)cc1 C1(C(=O)NC2CC(CNC(c3c(CC)cno3)=O)C2)CCC(N=[N+]=[N-])C1 C(=O)(C(C)CC(C)(C)C)Nc1c(C)nc(C(F)F)o1 C(=O)(C1CCCc2ncnn21)N1CCCC(NC(=O)COCCO)C1 c1(C(N2CCC(O)(CNC(c3csc(Cl)c3Cl)=O)CC2)=O)nc2ncccn2n1 CC(C)C(CNC(c1nnnn1C1CC1)c1ccsc1)CCO c1(CC(=O)NC(CN(C(C(c2scc(C)n2)C)=O)C)(C)C)cnccc1C C12(N(CCn3cc(Nc4ccccc4F)cn3)CC)CCCCC1OCC2 C12(C(=O)NC(C3CCN(C(C4(C)CCC(=O)N4)=O)C3)C)CCC(F)(CC1)C2 c1(C(C(=O)NCCCC)N(CC)CC2CCCOC2)nc(C)sc1C N1(C(c2c(CC)nc(C)[nH]2)=O)CC(NC(c2cn(C)nn2)=O)C2(CC2)C1 C1(CNC(C=C2CCN(C)C2)=O)CCCN(C(=O)CC2CCC(=O)CC2)C1 N1(C(C(C=C)C)=O)CC2CC(C1)N2C(=O)Cc1c(C)noc1C C1(C(=O)NCCCNC(=O)C(F)(F)CC2CCCO2)CC2CC(O)C(C1)C2 Nc1ccc(C(=O)NCC2CC2NC(=O)CCN2CCC2)c2c1CCCC2 c1(C(=O)NCCC(C(=O)NCc2nnc(O)n2C)OC)cccc(C)c1O C1(CNC(CSCCCC)=O)C(C)CCCN1C(c1cc(Cl)cn1C)=O C(CCC(=O)NCC(=O)NC(C12CC(CO1)C2)C)NC(C)=O C1(CNC(c2ccc(C)cn2)=O)CCN(C(c2cc(C)on2)=O)C12CC2 CS(=O)(=O)c1ccc(N2CC3CCCC2C3CNC(=O)CN2CCC(F)C2)nc1 c1(CNC(CN(CCC)C)=O)ccc2c(c1)CCCC2NC(=O)C(F)C1CC1 C(c1ccc(F)cc1F)=CC(N1C(C)(C)CC(CNC(C2CCCS2)=O)C1)=O N1(C(C2C(C)OCC2)=O)CC2(CC(NC(=O)C=CC(=O)NCC3CC3)C2)C1 C(C(=O)NNC(=O)C(=O)Nc1ccc(Oc2ccc(Cl)cn2)cc1)(C(C)C)SC N1(C(C(C2CCC2)NC(c2ccc(C)nn2)=O)=O)Cc2ccc([N+](=O)[O-])cc2C1 c1(OCC)cnc(C(=O)NC2CC(C(=O)NC3CC(CN(C)C)C3)C2)cn1 C(CC(C)C(F)(F)F)NC(C(CC1CC1)NC(C(C)=C1CCCC1)=O)=O CCC(O)C(C)C(=O)NC(CNC(c1ccc(Cl)cc1N)=O)CO N1(C(C(C)c2cccs2)=O)CCC2(CC1)CCN(C(=O)CC(C)C1CC1)C2 C12(C(N3CC(CCNC(C4CC(=O)N(O)C4)=O)C3)=O)CC3CC(CC1C3)C2 Cc1ccc(S(=O)(=O)CC(C)NC(=O)C(N2CCC(C)C2C)=O)cc1 c1(C(=O)NCCCN(C)C(C2(Cl)CC23CCC3)=O)ccnnc1O N1(C(C2CCC(N(C)C)C2)=O)CCCC(CO)(NC(c2cc3n(n2)CCC3)=O)C1 c1(C(=O)NC(C(=O)N2CC(N3CCC3)C2)C2(C)CC2)cnccn1 c1(CCNC(N(CCC#CCC)c2ccco2)=O)c(F)ccc(F)c1F c1(C(N2CC(F)(C(C)(C)CNC(=O)CNC=O)C2)=O)cc(Cl)cc(F)c1N N1(C(c2c(C)csc2)=O)CCC(C)(C)CC1C(=O)NCc1ccoc1C C(=O)(C#Cc1cccs1)N(c1cccc(C)n1)C1CC1 C(=O)(CC(C)(C)CSC)N1CC(CNC(c2c(SC)cccc2)=O)C(C)C1 N1(C(CCNC(CC(C)C)=O)=O)CCCC(C(=O)NC2CC2c2cncs2)C1C c1(NC(CNC(C(CC)OC)=O)C(C)C(C)C)c(F)cc([N+](=O)[O-])cc1F N1(S(CC=C)(=O)=O)CCn2cc(C(=O)Nc3[nH]nc4cnccc34)nc2C1 Cc1ccc([N+](=O)[O-])c(N2CCOCC(CNC(c3cc(F)c(F)cc3Cl)=O)C2)c1 C(=O)(CCC(F)(F)F)N(C1CCCN(C(c2ccc(C(=O)OC)n2C)=O)C1)C CCC(C)(CNC(c1cc(CNC(C2(CC3CC3)CCC2)=O)ccn1)=O)C(C)O C1(C(=O)NC2C(C)(C)C2C(=O)N(C2CCCCC2)CCO)CC2(CSC2)C1 C1(C(N2CC3CN(C(C45CCCN4CCC5)=O)CC3C2)=O)CCc2c[nH]nc2C1 c1(Nc2cc(C(N3CCCC(C)(O)CC3)=O)n(C)c2)nccc(S(C)(=O)=O)n1 C12(CNC(N3CC(N4CCN(C(C)=O)CC4)C(C)C3)=O)CC3CC(CC(C3)O1)C2 C1(CNC(c2nc(CC)[nH]n2)=O)CCN(C(c2nc3ncccn3n2)=O)CC1C CCC(CC)C(=O)NCC(N1CC2C(CNC(c3cn(C(F)F)cn3)=O)C2C1)=O c1(NC(c2c(CNC3C=CC(C(=O)OC)C3)noc2)=O)c[nH]c2ccc(Cl)cc12 C(=O)(C(F)(F)C(F)F)NC1CCN(CCNC(C2N(C(C)=O)CC(O)C2)=O)CC1 C1(C(N(CCCCCCNC(C(CC)(C)O)=O)C)=O)CCCCCC1(F)F c1(C(=O)OC(c2ccc(I)cc2)C(=O)OCC)ccc(O)nc1 C=CC(C)(C)CCOC(=O)NCCC(C)NC(=O)NCCl.C(C)(C)(C)O CCC(C)C(O)C(=O)N(C)CC1CCC(CNC(C2CCC(C)(C)C2)=O)CC1 c1(C(=O)NC(C(=O)NCC2CC2)C2(O)CCC2)cccc(CO)c1 C(=O)(CN=c1cc[nH]cc1)NC(CC(C)NC(C1CC2(CCOC2)C1)=O)C C1(CNC(CC=CC=C)=O)CC2CC1CN2C(=O)Cc1nnn(C(C)(C)C)n1 Cc1cc(C(=O)NCC2C(C)CCCN2C(=O)CN=S(C)(C)=O)cc2ccoc12 N1(CC(COC)O)CCC2CCC(C1)N2C(=O)CCc1ccn(C)n1 N1(C(c2sc(C)c(Br)c2C)=O)CCN(C(=O)C2CC2)C2CCCCC12 C(=O)(C(CCOC)OC)NCCC.C1(C2c3nnnn3N2)CCOC1(C)C c1(N(CCNC(C(C)N(C(C)=O)C)=O)C(C)C)cccc(F)c1[N+](=O)[O-] C1(NC(CSC)=O)CCC(C)N(C(=O)CC2CCOC2(C)C)C1 N1(C(C=Cc2n(CC)ncc2)=O)CCC(C)C(CNC(=O)Cc2ccc(Cl)s2)C1 C1(NC(c2c(CC)n(CC)nc2)=O)CCN(C(=O)CCSC(F)(F)F)C(C)C1 c1(OC)ccc(F)c(C(=O)NC2CCN(C(=O)Nc3ccc(F)cc3)CC2)c1F N1(C(C(F)=C(C)C)=O)CCC(C(=O)NC2CCN3CCC2C3)C1(C)C C1(F)(c2cn(Cc3ccc(OCC(N)=O)cc3)nn2)COCCN(C(=O)C(Cl)Cl)C1 C1(C(=O)NCC2CC(NC(C3C(C)CCO3)=O)C2)CCn2c(O)nnc2C1 C=CC1(CC(=O)N(CC(C)C)CC)CN(C(=O)C2COC2)C1.C(C)OC S(=O)(=O)(c1ccc(NCC(C)(C)OC(C)(C)C)c(Cl)c1)N1C(C(C)C)CC(O)C1 N1(C(C=CC(=O)N(C)CC2CC2)=O)CC2CN(S(=O)(=O)C(Cl)(Cl)Cl)CC2C1 n1(CC)cc(C(=O)NCC2CN(C(C3(F)CCOC3)=O)C2)c(C(F)(F)F)n1 Cc1cnccc1C(=O)N(CCNC(=O)Cc1ccnc(O)c1)C1CC1 C1(CNC(C2(CC#C)CCC2)=O)CC(C)(C)CN1C(c1ccc(F)c(C)c1)=O c1(CCC(=O)NC(C)C(C)NC(=O)Cc2nccn2C)cnccn1 c1(C(=O)NC2(CN(C)C)CC2)cc(CNC(C2CC2(F)Cl)=O)cs1 c1(CCN(C(C(C)SC)C2CC2)C)ccccc1Br CC(C)(C)C(O)C(=O)NC1CCCN(C(c2ccccc2C2CC2)=O)C1 C1(C(=O)NCCCC(=C)Cl)CCC(NC(=O)Cn2nnc(C)n2)CC1 C1(NC(=O)CSc2ccccc2)CC2CN(C(C3SC4C=CC3CC4)=O)CC12 N1(C(C#CC)=O)CCCCC(NC(C2SCCCS2)=O)C1 c1(C(=O)NCC2CC(NC(C(C)=CCO)=O)C2(C)C)ccc2c(c1)CCC2=O CC1(NC(=O)CC2CCCCC2(C)C)CCCN(C(C2CCC23CCC3)=O)C1 N1(C(C(C2CCCCC2)OC)C(=O)NC2CC(F)(F)C2)CCCC2CN(C)CC12 C12CCCN(C1)CCC(=O)NCC2.c1(C(C2CCOCC2)=O)cccnc1Cl C(=O)(CCC(=O)NC1CC1)NC(C(=O)N(C)Cc1n(C)ccn1)C1(C)CC1 C1(C)(NC(CN(C(C(c2ccnn2C)C)=O)CC(N)=O)=O)CCOC1C C1(C(=O)OC)CCCCN1C(=O)CC1CCN(C(=O)CCCn2cccc2)C1 C1(C(=O)O)CN(C(=O)CC2CCOC2)CCO1 N1(C(C2C(C)C2c2ccccc2)=O)CCC(CNC(=O)C(=O)Nc2ncc[nH]2)C1 Cc1ncccc1C=CC(=O)NCC1CCC(C(=O)NC23CCCN(CC2)C3)C1 C(=O)(C1=CC2C=CC(C1)C2)NC(CCCNC(COCc1nnc(C)s1)=O)C c1(C(=O)NC2CCN(C3(C(N(CC)OC)=O)CC3)C2)cncc(C#N)c1 C1(NC(C(CC)(C)F)=O)(COC)CCN(C(=O)CCc2scnc2C)CC1 c1(CC)oc(C)cc1C(=O)NC1(CCC(=O)NCC(O)C(C)C)CCC1 N1(C(c2scc(C)c2)=O)CC2CC1CN2C(C1CCC(C(C)C)CC1)=O C1(ONC(=O)N(C(CC2CCCO2)C(F)(F)F)C)CCCCCCC1N CC1CC2CN(C(c3ncc(F)cn3)=O)CC2N1C(C1CC1c1ccccc1)=O CC(C)CC(C(=O)OC(C)(C)C)N(C)Cc1cncc(C#N)c1 C1(CC(=O)N(CCC)C)COCCN1C(=O)CNC(=O)COCCCF C(=O)(C(C)(F)C(C)(C)F)NC1CN(CC(=O)N(C)Cc2ccccc2)C(=O)C1 c1(CNC(c2cc(C)cc(C)n2)=O)cc2n(n1)CCN(C(c1ccoc1Br)=O)C2 n1(CCC(=O)NCC(Cc2ccoc2)CO)cc(Br)cn1 c1(OC)cc(C(N2CCCC2CN=c2[nH]nc(C(N)=O)s2)=O)ccc1F c1(OC(CC)C)cc(CNC(=O)NCC2CCCC(CC(F)(F)F)C2)ccn1 N1(C(CC2C(NC(C(C(C)C)OCC)=O)CCCC2)=O)CCCC(C)(C)C1 N1(C(CC(C(C)C)C)=O)CCCN(C(c2occ3c2CCOC3)=O)CCC1 C1(C2CCN(C(c3nc(=N)[nH][nH]3)=O)C2)(NC(C2ON=C(C)C2)=O)CC1 c1(C(N2CC(C)(CNC(C(C=C)O)=O)OCC2)=O)cc2c(cc1N)CCC2 C1(CC(N2CC(NC(c3c(F)cccc3F)=O)C(O)C2)=O)Cc2ccccc2O1 C1(CCC)CN(C(=O)CNC(C2CCC2)=O)CCN1C(=O)C(C)c1cncs1 C1(C2CC2)(NC(C(C)OCC)=O)CCN(C(c2csc(Cl)n2)=O)C1 c1(C(=O)NC(C2N(C(C(C)NC(=O)NC)=O)CCC2)C)cnc(SC)n1C Cc1cc(CC(N2CCN(C(=O)CCCC#N)CC2)=O)c(C)n1-c1ccon1 C1(C(N(CC(C)C#N)C)=O)CCN(C(=O)Cc2ccc(O)cn2)C1(C)C N1(C(C=Cc2ccc(C)cc2Cl)=O)CCOC2CCN(C(C3C(C)C3C)=O)CC12 c1(N2CCC(OC)(CO)C2)[nH]c(=NC2C=CCC2)nc2c1ncn2C(C)C c1(CC)cc(C)ccc1C(N1CC(N(C)C(C2CC2CC)=O)C(O)C1)=O C(=O)(C1=COCC1)NC(C1CCCCN1C(c1ccc(Cl)nc1)=O)C c1(C(=O)NCCC(=C)CNC(C2(CC(F)F)CCC2)=O)ccc(OC)c(F)c1 N1(C(CC(CC)C)=O)CCC(C=CC(=O)NCCCc2c[nH]nc2C)CC1 c1(OC)c[nH]c(C(N2CCCCC2c2cnco2)=O)cc1=O C1(Nc2cc(OCC)ncn2)CCC2CN(C(c3ccc(Cl)nn3)=O)CCC2C1 C(C)(CO)(C(F)(F)F)NC(c1c(CNC(c2c(C)scc2)=O)n[nH]c1)=O Cn1cc(Br)c(CC(=O)NC2(CNC(C3CN(CCF)C3)=O)CC2)n1 S(=O)(=O)(c1ccc(NCC(c2cccs2)O)cc1Cl)NCC1(CC#N)CC1 C(=O)(C1CCCn2c(C)nnc21)NC1CCN(C(C(C(CC)C)O)=O)CC1F C(=O)(CCN=c1ccc(C)c[nH]1)NCCN(C(C(CCC)CC1CCCC1)=O)C N1(C2CC2)CC(F)(C(=O)NC)C1.C(=O)(COCCF)NC(C1CC1OC)C N1(C(COC)=O)CCCC(C(=O)NCCn2ccnc2C)C1C CCCS(=O)(=O)CC(=O)N1CCCN(C(=O)CC2CCC(C)O2)CC1 c1(C(c2n(C(CC)C)nnn2)NC(C)C)cc(Br)c(OC)cc1OC N1(C(C(C)N(C(C(n2c(C)ncc2)C)=O)C2CC2)=O)CCC(C2(C)CC2)C1 c1(C(=O)NC2CC(NC(CCCOCCC)=O)C2)cnc(S)nc1 N1(C(c2nn(CC)c(C)c2)=O)CCN(c2ccc(OC)cc2F)CC1CC#N c1(SCC2CCN(OCc3c(Br)c[nH]n3)C2)ccc(F)cc1 CC1CCCC(O)(CNC(C23CC(NC(=O)CCc4cn(C)nn4)(C2)C3)=O)C1 C1(C)(NC(CCc2cc(C)n(C)n2)=O)CCCN(C(=O)C#CC2CC2)C1 C(=O)(N(CCO)OC)N(C1CCN(C(=O)C(C)Cc2ccccc2)C1)CCOC c1(C(=O)OCCSC(C)(C)C)cccc(-n2cccc2)c1 C1(CCOC)(NC(c2cn(C3CC3)nn2)=O)CCN(c2ncc(C)cn2)C1 C(C(C)(O)CNC(=O)CN(C(c1ccn(C(C)C)n1)=O)CC1CC1)OC N=c1nc(C(=O)NCc2cc(C(=O)NCC#CC3CC3)co2)cc[nH]1 CCCCN=C(NCCCN1CCN(C)CC1)N1CCC2(C)C(C1)C2(Cl)Cl c1(C(=O)NC(C)CNC(c2ccc(C(C)(C)C#N)cc2)=O)cn2ccsc2n1 c1(C(N(C(C)C(=O)Nc2ccc(O)cc2Cl)CC)=O)ccc(C)c(C#N)c1 c1(C(=O)NC2CN(C(c3c(CC)ncs3)=O)C2)cccc2nncn12 c1(NC(=O)CNC(c2ccc(-n3cccn3)cc2)=O)cccc([N+](=O)[O-])c1 S(=O)(=O)(c1ccccc1F)N1C(C(=O)Nc2c(C(=O)OC)nccn2)CCC1 C=CCCCCC(=O)NC1CC(CC(=O)NC(CN(C)C)C(C)(C)C)C1 C1(=O)C#CC2CCCCN2C(=O)O1.c1(OCC)ccc(C(=O)OC(C)(C)C)cn1 c1(C(=O)OCC)nc2cc(F)ccc2o1.C1(=O)C(C(O)c2ccccc2)O1 N1(C(C(C(C)C)CO)=O)CCC2CCN(C(c3cc4cc(O)ccc4[nH]3)=O)CC12 CC1(C)CC(NC(c2cc(C3CCC3)on2)=O)CN1C(=O)CCSC(F)(F)F N1(C(C2N(C(N(C)C)=O)CCC2)=O)CCN(C(c2cc(F)n[nH]2)=O)C(CCO)C1 C(=O)(C1=NN2CCCN=C2N1)NC(C)CC(C)NC(C1COCCO1)=O Cc1ccc2c(c1)C(NC(=O)C(C)(O)C(F)(F)F)CN2C(c1ccc[n+]([O-])c1)=O c1(C(=O)NC(C2CCCN(C(=O)C=C3CCOCC3)C2)C)ccc(CO)c(Cl)c1 CCCC(C)CCNC(N1CCC(Oc2ccc(CNCCC)cc2)C1)=O N1(C(C2(C)CCOCC2)=O)CCC2(CC2NC(=O)C(=O)NCCC(N)=O)C1 c1(CNC(C2C(CNC(c3c(COC)occ3)=O)COC2)=O)c(C)cnnc1O C1(NC(CC(c2cccc(OC)c2)C)=O)CC2CCC1N(C(=O)C(C)C(C)O)C2 c1(Cc2ccc(C(N3C(C)C(O)CCC3)=O)cc2)cccc2c1OC(F)(F)O2 C(CC(C(C)(C)C)NC(=O)CN1CCCC1)N(C(C(CCSC)OC)=O)C c1(OC(CC)C(=O)NCCNC(=O)CCCN2CCCC2)ccccc1F c1(C(=O)NC(CCC)C2CCC2)cccnc1CNC(c1cc(C(N)=O)on1)=O C#CCC(C(=O)N1C=CCCC1C(=O)N(CCF)CC1CC1)C1CC1 c1(SC)cc(=NC(=O)c2ccn(C(F)F)n2)[nH]o1.c12ccccc1S2 N1(C(C(COCC)NC(c2n[nH]c(C)c2O)=O)=O)CC2CCC(C1)C2O C(=O)(C1=CCCOC1)NC1C(CC#N)COC1 CCCC(C#N)C(=O)N1CC(OC)C(C(=O)NCC=CC(C)(C)C)C1 c1(CC)ccc(NC(=O)CCSC)c(C(=O)N(C2CCNCC23CC3)C)c1 C1(NC(CC23CC(C)(OC2)C3)=O)COCCN(c2ncc(C(F)F)cn2)C1 c1(-c2onc(C(=O)NC(CNC(=O)CC3CCC(O)C3)CO)n2)cccc(F)c1 Cc1cnc2cc(C(=O)NC3CN(C(c4cncnc4)=O)CCC3CO)nn2c1 c1(C(=O)NC(CC)CNC(=O)CCc2ccc(F)nc2)ccc(Br)nc1O Cc1c[nH]nc1CNC(=O)CCC1CCCN1C(=O)CCCC1CC1C CCC(C)CCC(=O)N1CCC(C(=O)NOCC(=O)OC)O1 C1(C(=O)NC2CC(O)(CNC(C(C)(C)c3ccccc3)=O)C2)CC(F)(F)C1(F)F C=CC(C)(C)CC(=O)NC12CC(NC(=O)Cn3ccc(Br)n3)(C1)C2 C(c1cncc(C)c1)=CC(=O)NCCCNC(CCNS(CC)(=O)=O)=O N1(C(COCCC(C)C)=O)CCC(C2CN(C(=O)CCn3cncn3)C2)CC1 N1(C(C2N(C(c3c(C)nc(C)s3)=O)CC(O)C2)=O)CCC2(COC(C)C2)C1 c1(-c2cncc(C(=O)Nc3c(OC)cc(F)cc3)n2)cc(O)c(F)cc1F c1(C(=O)NC(CCNC(C(C)=CC2CC2)=O)C)cc2cccc([N+](=O)[O-])c2[nH]1 C(=O)(C(C)(C)C(C)C)NCC1(O)CCN(C(c2ccc(CCCC)cc2)=O)C1 N1(C(c2ccc(C(C)(C)C)nc2)=O)C2CCCC1CN(C(c1cncnc1)=O)C2 c1(C(=O)NC2C(NC(c3ccc(C#C)o3)=O)C2)cc2ccccc2[nH]1 C1(C(N2CCCC(OCCC)C2)=O)CC(C)(C)CN1C(=O)CC1OCCC1(C)C C1(NC(C2C(C)COCC2)=O)CC2(CCN(C(=O)CSc3ccccc3)C2)C1 O=C(C(C1CCCC1)NC(C1CC12CC2)=O)NOCC1CCCO1 CN1CCN(C(c2cccc(F)c2Cl)=O)CC1CNC(=O)C=C1CCSCC1 C12(C(N(CCNC(CC3C(C)(C)CCO3)=O)C3CC3)=O)CC1COC2(C)C Cc1ccc(F)c(OCC(=O)NC(CO)C(C)NC(=O)CN2CC3CC3C2)c1 C1(NC(C(C)c2ccsc2)=O)CN(C(=O)Cn2cc(CO)nn2)CCC1(C)C C1(NC(c2cc[nH]c2)=O)COCCC1NC(=O)C(c1ccccc1)F c1(C(=O)NC2CN(C(c3ccc(F)s3)=O)CCC2O)ccc2n[nH]cc2n1 C1(C2N(CCCC(C)N3CCCC3)CCC2)CCN(C(C)=O)CC1.C(=O)(COCCF)N n1(CC(=O)NCC2(NC(CC3CCC(C)O3)=O)CC2)nc(C2CC2)n(C)c1=O C1(CNC(C2C(C(C)NC(=O)COC3(C)CCC3)C2)=O)CCCNS1(=O)=O c1(OC)ccc(C(=O)CCC(=O)NCCCC(C)(C)NC(=O)CC2CC2)cc1 C12(CCNC(=O)CC(=O)Nc3nccs3)CCC1CN(C(C1C=CCC1)=O)C2 c1(C(=O)NCC2CCCN(C(C(C)OC(C)(C)C)=O)C2)nccn2nccc12 CC(C)CC(CC1CCCCC1)CC(=O)NC1(C)CN(C(=O)C(C)CC(N)=O)C1 CC1CCc2sc(C(=O)NCC3CCN3C(c3cc4sccc4cn3)=O)cc2C1 c1(C(N(CCOCCCN(C(C(C2CCC2)OCC)=O)C)C)=O)cnc(Cl)s1 N1(C(CCOCC)=O)CC2CCC1CN(C(c1cccc3nc(C)cnc13)=O)C2 C(CCCCC(=O)N1CCC1C(=O)N(C)Cc1nnnn1C)OCC C1(C(=O)NC2CC(NC(=O)CSC3CCOC3)C2)(CO)CC1(F)F C1(CC(=O)NC)CC2CCC(C1)N2C(=O)C(C)(C)C1(C(=O)OC(C)(C)C)CCC1 c1(N2CCC(N(C(C3CCc4nncn4C3)=O)CC)C2)ccc([N+](=O)[O-])cc1 CC1CC1C1CC1C(=O)NCC1COCC1NC(=O)C(N)=O c1(CC(=O)NC(C(C)C)CNC(=O)C(C)(C)O)cnn2ccccc12 CCCCC(C(=O)NCC1CC(CC)C1)NC(=O)C(C(C)C)N(C)C(=O)OCC N1(C(c2ccc(C)c(O)n2)=O)CCC2CC2(NC(c2cnc(C(C)C)s2)=O)CC1 c1(C(C)(C)C)nnc(CC(=O)NCCCNCC=CCNC(=O)C=C2CCC2)o1 N1(C(C(C)=C2CCC2)=O)CCC(C(=O)NOCC(O)CO)C1C c1(-c2n(-c3cccc(CC)c3)nc(COC(C)C)n2)cnc(SC)c(C)c1 C=CCCC(C)C(C(=O)NCC(=O)OCC)N(CCCNCCC#N)C.C(C)(C)(C)O Cc1nnc(CN(CC(=O)NCCC2CCN(C(C3(C(N)=O)CC3)=O)C2)C)n1C C1(NC(CCCN(C(C2CN(CC)C(=O)C2)=O)C)=O)C=CC(C)(C)CC1 c1(CC)nc(C)cc(=NCC2(NC(=O)CSCc3cccnc3)CCOCC2)[nH]1 C=C1CC(CC(=O)NC2(CNC(C3CC(CCO)C3)=O)CCC2)C1 c1(-c2ccc(Nc3ncc(C(=O)OC)nc3C#N)cc2F)cccc2c1OCC2 c1(CN2CCC(NC(c3cn(C)nc3C(F)F)=O)CC2)cccc2occc12 C12(C(N3C(C)C(NC(C4CC4F)=O)CCC3)=O)CCC(N=[N+]=[N-])C1C2 c1(C(N2CCC3(NC(c4cccc(OC)n4)=O)C(C2)C3)=O)ccc2cnnn2c1 c1(C(=O)NC(CNC(C(CSC)O)=O)C)cc(S(C)(=O)=O)ccc1Cl c1(NC(=O)NC2C(C(=O)Nc3cncc(C)c3)C2)cccc2c(Br)cccc12 N1(C2CN(C(c3coc(Cl)n3)=O)C2)CC(NC(C2CCC(=O)N2)=O)CC1=O C#CC1(CNC(=O)CC2CCCC(NC(=O)C(C)CC(F)F)C2)CCOCC1 c1(CCC(=O)NC2C=CC2CO)ccc2ccccc2c1 C1(C(=O)N(C2C(OC)CN(C(C3C4CC5C(C4)C35)=O)C2)CC)CCC(=O)N(C2CC2)C1 c1(NC(CC2N(C(c3cc(C)oc3C)=O)CCOC2)=O)ccc(C#N)c(O)c1 c1(C(=O)NC(CCCOCCOC)=O)cncc(NCCC(C)(C)C2CC2)c1 N1(C(=O)NCc2c(C)nn(CC(=O)OC)c2C)CCC(C2CC2(F)F)C1 c1(C(=O)NC(C(C)C#N)c2ccccc2)ccc(OCC(F)(F)F)nc1 c12ccc(C(C)C)cc1NC1C(COC1)O2.c1(COCC)ccc(C(C)(C)C)s1 c1(C(N(C2CCC(NC(CNC(CC)=O)=O)C2)C)=O)cc(OC)cc2c1CCC2 C12(C(=O)NCCN(C(c3cnsc3)=O)C3CC3)CC(C(F)(F)F)(CO1)C2 N1(C(CCSC)=O)CC(CNC(c2cc(C3CCC3)[nH]n2)=O)CC1(C)C n1(CC(C)C)cc(N=c2scc(-c3cc(F)c(F)c(F)c3)n2C2C=CCC2)cn1 C12CCCC(C1)CC(=O)Nc1cn(nc1)CC(=O)N2.N1(C(=O)CO)CCCC1 CC1(F)CN(C(c2sccc2C2CC2)=O)CCN(C(C2CCC23CCC3)=O)C1 C1(C(=O)NC(CC=C)CC(F)F)CC2(CCC2)CN1C(C1C2CC3C(C2)C13)=O C1(NC(C(C=C=C)C)=O)CC2CCC1(NC(c1ccnc(OC)n1)=O)C2 CC(C)C(O)C(=O)NCC(C1CCCC1)NC(c1cccc(C2CCCC2)n1)=O C12(NC(C3C(OCC)C3)=O)CCCN(C(=O)Cn3nc(C(C)=O)cc3C)CC1C2 C1(NC(C(C)SC(F)(F)F)=O)CCC2CN(C(C3(C)CC3(F)F)=O)CC2C1 N1(C(CS(C(C)C)(=O)=O)=O)CCC2C(CCN2C(c2cc(Cl)cn2C)=O)C1 N1(C(C=NOC)=O)CCCC(C2CCN(C(c3coc(C#N)c3)=O)CC2)C1 C(=O)(C1=CCCCC1C)N1CCC(CNC(CCn2c(C)cc(C)n2)=O)CC1 Cn1nc(C(=O)NC2COCC2NC(C2CCC3(CCC3)O2)=O)c2c1CCC2 S1(=O)(=O)c2ccc(cc2)N1CC=C.N1(C(C2CC2c2cccs2)=O)CCN(C)CC1 N1(C(C=NOC)=O)CC(CNC(C2(C)CCCCCC2)=O)OC2COCC12 c1(C(=O)NC2(CC=C)CCN(C(CCCC#CC)=O)C2)coc2ccc(F)cc12 C1(N(C)C(C2CCS2(=O)=O)=O)CCN(C(=O)COc2cccc(F)c2)C1(C)C C1(c2ccno2)(C(=O)NCC(CC)NC(c2c(CC)nns2)=O)CCOCC1 N1(C(C2(C)CCCC2)=O)CCc2nc(-c3ccc(CC#N)cc3)sc2C1 c1(C(=O)NC2CC(NC(=O)CCC3CCCCO3)C2)ccc(CO)cn1 C(=O)(C(O)C(F)(F)F)NC1CC2(C(C(=O)NCC3(CC)CCOC3)C2)C1 c1(CN2C(C(=O)Nc3cc(F)c(F)cc3Cl)C=CC2)c(Cl)c[nH]c2nccc1-2 C1(C2CC2)(CNC(c2c(CC)onc2C)=O)CCN(C(C2CCN(C)C2=O)=O)C1 c1(N(C)CC2OCCN(C(c3cc(C)sn3)=O)C2)ncnc2scc([N+](=O)[O-])c12 N1(C(C(CC=C)N(C)C)=O)CC(CNC(=O)Cc2ccn(CC)n2)CC1(C)C C1(C(=O)NCCCCN(CCCNC(=O)C(N)=O)C)CCCCCS1(=O)=O N1(C(CC2ON=C(C)C2)=O)CCCN(C(=O)CS(=O)(=O)C(C)C)CC1CO Cc1ccnc(C(=O)N(CC(C)CNC(c2ccc(C(F)F)nc2)=O)C)c1O Cc1cc(C(=O)NC(CCF)C(=O)NC23CC=CC(C2)OC3)nc(C)n1 CCC(CCC(=O)Nc1ccc(F)cc1CO)NC(=O)CC1(O)CCOC1 CCC(CC(F)(F)F)NC(=O)C(C)(CC1CC1)NC(=O)NC(C)C c1(NC(C2CCCN(C(C(c3cccc(Cl)c3)C)=O)C2)C)nc(C#N)c(Cl)s1 C(=O)(CC(C)n1ccc(C)n1)NCCC1CN(C(CCNC(=O)OC)=O)C1 C1(F)(CNC(c2cc(Br)c[nH]2)=O)CCCN(c2cc(C3CC3)nc(Cl)n2)C1 N1(C(C2C(O)CCN(Cc3ccc(C)cc3O)C2)=O)Cc2cc(O)ccc2C1 C1(CCNC(C2(n3cc(CC)nn3)CC2)=O)CCN(C)C(=O)O1.C1CC(=O)N1 c1(-c2ccc(C(=O)NCCC3CCC(NC(CC(C)O)=O)C3)s2)cccc(Cl)c1 CC1CN(C(=O)COc2cccc(Cl)c2)CC1NC(c1n[nH]cc1Br)=O C1(C)(CC(=O)NCCCN(C(c2c(CC)nn(C)c2)=O)C)CCCCCC1 N1(C(C=Cc2cnc(C)s2)=O)C2CCC1CN(C(c1cnc3n1CCS3)=O)C2 N1(C2CN(C(c3c(SCCOC)nccc3)=O)C2)C(=O)CCN(C2CC2)C1=O C(=O)(CCCCC(=O)NCC(C1CC1)N(C)C(C1CC(F)C(=O)N1C)=O)NC c1(CN2CC(NC(C=C3CCN(C)CC3)=O)C2)ccc(F)c(O)c1 CC(C)C(C)(F)F.c1(-c2cn(C(C(=O)OC)C)nn2)cc(N2CCCC2)ccn1 Cn1cc2c(n1)CCCC2C(=O)NCC(O)CCNC(=O)C(C)(C)C(N)=O c1(NCCCC)ncnc2nc(N3CCCC(N4CCOCC4)CC3)sc12 CC1(C)CCOC1CC(=O)NC1(C2CCCCN2C(=O)CCc2cncs2)CC1 C(=O)(CC1=NNC(=O)C1)NCC(C)CNC(c1cnn(C(C)(C)C)c1N)=O N1(C(CN(C(=O)OC)C)=O)CC2CCCC1CN(C(=O)CCCC(F)(F)F)C2 N1(C(=O)C(F)(F)F)CCC(Oc2c(Br)c(OC)n(C)n2)C(F)(F)C1 O=C(CCCC#Cc1ccccc1)NCC1CC(CNC(c2ccc[nH]2)=O)CO1 N1(C(=O)CC2CCC2)CC2(CCCN2C(c2cccc(-c3cn[nH]c3)c2)=O)C1 O(NC(=O)C1=NOC(CNC(c2ccc(O)c(F)c2)=O)C1)C(C(=O)OC)(C)C CC1(C)CCC(CNC(c2ccsn2)=O)N(c2cnc(F)cn2)C1 c1(C(N2CCCC(CC(C(=O)OCC)N)C2)=O)cc2n(n1)CC(C)NC2=O c1(CC)cc(C(=O)NC2CCCCC2NC(C2(CS(C)(=O)=O)CCC2)=O)n(C)n1 c1(-c2nc(-c3cc(C)nn3-c3ccccc3C)on2)cnnc(O)c1Br Cc1nn2ccccc2c1C(N1CCCN(C(=O)COCCF)C(C)C1)=O c1(CNC(=O)CSC(F)F)ccc2c(c1)CCC2NC(c1cccc(=O)o1)=O N1(C(CNC(c2cc(C)c(C)nn2)=O)=O)CC(C)(C)OC(C)(C)C1 c1(C(=O)NC2CC(NC(C(C)(C)OCC)=O)C2)ccc(F)c2ncccc12 C1(OC)CN(C(=O)C(C(C)C)N(C)C)CC1NC(=O)Cc1coc(C(F)F)n1 c1(C(N2C(C(=O)NC(C(C)C)C)CC(=O)C2)=O)cccc(O)c1F C(N=c1nc2scnc2c(NCC2(c3ccc(F)cc3)CC2)[nH]1)C1CCC(C)N1 N1(C(C(C)N(C)C(C2CC23CCCCC3)=O)=O)C2CCCC1CN(C)C2 Cc1cc(Cl)nc(N)c1C(=O)NC1CC1NC(c1cccc(CS(C)(=O)=O)c1)=O C1C(CO)CCc2occ(c2)C(=O)N1.CC(C(=O)NC)OC(C)(C)C C1(CNC(c2cn(CC(C)C)nc2C(F)F)=O)CCC(C)CN1C(=O)CC1CC1 C(C(F)(F)F)CN(C(=O)NC1CN(C2CCC2)C1)CC c1(OC)cc(CNC2(c3ccc(C(=O)O)c(F)c3)CC2)c(F)cc1Br C1(C(=O)NCCC2CCN(C(CCNC(=O)CO)=O)C2)CCCOCC1 CN1CCC(C(C(=O)Nc2ccccn2)N(C)CCc2cccc(Br)c2)CC1 C=CC(C)(CCOC)C(=O)N1CC(C(C)NC(c2ncoc2CSC)=O)C1 c1(-n2cc(CC3CCN(C(C4COCOC4)=O)C3)nn2)ccc(Br)cc1 c1(C(N(CCNC(c2ccc(CN(C)C3CC3)cc2)=O)CC)=O)ccc(Cl)c(C)c1 Cn1cc2c(n1)CC(C(=O)N(CCNC(C1(C3CCCO3)CC1)=O)C1CC1)CC2 Cc1cccc(C(O)C(=O)NCC2CC(NC(c3cccc[n+]3[O-])=O)C2)c1F Cc1ccccc1C(=O)NC(Cc1ccco1)C(N1CCC(CC(C)O)CC1)=O CN1CCCCC1CCC(N1CCC(O)(CN(C(=O)C=C2CCC2)C)C1)=O c1(C(N2C(CNC(CCC)=O)CCC(C)(C)C2)=O)cc2c(cc1Cl)NC(=O)C2 c1(C(=O)NC2CC(NC(c3n(CCC)ccn3)=O)C2)ccnc(C)c1O c1(C(N(CCNC(C2CC(=C3CC3)C2)=O)CC)=O)cc(C2CC2)[nH]n1 C1(NC(CNC=O)=O)CCN(C(c2cccc(C3CCC34CCC4)c2)=O)CC1O N1(C(CCCS(C)(=O)=O)=O)CC2CC(NC(=O)C=Cc3cscn3)CC(C2)C1 c1(CNC(N(CC(C)C)Cc2ccc(F)cc2F)=O)cc(Cl)cnc1O C12(C(=O)NCCCN(C(=O)C(O)Cn3cncn3)C)CCC(CC1)CO2 c1(C(c2ccccc2)C(=O)NCC2(CO)CN(C(C(C)C)=O)C2)nn(C)cc1Cl C1(C(=O)NC2CCC(F)(F)C2)CCCN(C(=O)CCn2cccn2)CC1 c1(C(=O)NCC(CCC)NC(=O)CCC(C)(C)C)cc([N+](=O)[O-])c(C)s1 C1(C(=O)NC(C)C(=O)NCC2CCCCO2)C(C)(C)C1(C)C c1(C(N2CC(C)C(CNC(C3CCCOC3)=O)C2)=O)cc(F)ccc1S(C)(=O)=O c1(OOCNCc2cncc(OCC)c2)sc2ccccc2c1Br.c12cccc(c1)O2 c1(C(C)(C)OC)nnc(N(C2CCCC2)C)s1 Cc1nn(C)c(Cl)c1C(=O)NCCN1CCN(C(=O)CCCC2CC2)CC1 Cc1c(C(=O)NCC(C)CN(C(=O)C(F)CC2CC2)C)[nH]c2cc(F)ccc12 c1(NCCCCCC)nc(=NCc2ccnc(C)c2)[nH]c2c(C)nn(C)c12.C1(N)CC1 c1(C(=O)NC(CC)CNC(C2CC(=O)N(CC3CC3)C2)=O)cccc([N+](=O)[O-])c1 c1(C(C(=O)NC2CC(F)(CNC(c3c(CC)nc[nH]3)=O)C2)OC)ccccc1F c1(C(=O)NCC(CC)NC(c2c(CC)oc(C)c2)=O)cc2c(F)ccc(F)c2s1 c1(C(=O)NC(CC(C)C)CNC(C2CCCC2CF)=O)cc2cccnc2cn1 N1(C(Cc2nnc(C)s2)=O)CCC(NC(C2CC23CCC3)=O)C1C N1(C(c2c(NC)c(N)ccc2)=O)CCCC2(C1)CN(C(=O)C(C1CC1)OC)C2 N1(C(C(N2C3C(C(=O)OCC)C(C3)C2)=O)=O)CCOc2ccccc2C1C(F)F Cc1cc2c(cc1C(N1CCC3CN(C(=O)CC#N)CC3C1)=O)OCCO2 C1(CNC(C2(N(C(=O)C(c3ccccc3)O)C3CC3)CCC2)=O)CCCCS1 C1(NC(=O)CC2CCCC23CC3)CN(C(c2cccc(Br)c2)=O)CC2(CCC2)C1 C(CCF)(C(=O)N=c1ccn(C(F)F)[nH]1)NC(c1c(CC)n[nH]c1)=O C(C1CCC(C)CC1)=CC(=O)N(CC(CNC(C=C(C)Cl)=O)O)C C(=O)(CCC(C)S(C)(=O)=O)N1CC2CN(C(c3cc(C)n(C(F)F)n3)=O)CC2C1 CC(C)C1=NOC(C(=O)N(CCC(=O)N(C)C)CCO)C1.C1(C)C(=O)N1.OCC c1(NC(c2csc(C3OCCO3)c2)=O)cccc(F)c1C(=O)O N1(CC(=O)NCC(C)(C2CCC2)NC(C(C)NC(C)=O)=O)CC(=O)NC1=O CC(C)(CNC(=O)CCC1CCCC1)CC(=O)NCCC(O)C(F)(F)F N1(C(COCC(C)(C)C)=O)CCN(C(=O)C(C2CCCCC2)F)CC(C)(C)C1 C1(c2ccccc2)(CC(=O)NCC(CNC(c2[nH]nnc2C)=O)OC)CCCC1 C1(CNC(CC)=O)CCC2(CCN(C(c3coc(N)n3)=O)CC2)CO1 C(=O)(CCCCCN=[N+]=[N-])N1C2(C(=O)Nc3c(OC)ncnc3)CCCC2CC1 Cc1cccn2c(C(=O)NC3(CO)CCN(C(C4OC5CCC4C5)=O)C3)cnc12 c1(C(N2CCC(NC(C3CCCN(C)C3)=O)(CF)C2)=O)c[nH]c2cc(O)ccc12 N(C(=NCC(C)OC(F)F)NCC1(C)CC1)Cc1ccc(OCC)cc1 CC(C)C(C#N)CS(=O)Cc1cccc(NC=O)c1 c1(NCCCCN(C)C)ccc(S(=O)(=O)N2CCC(OCCF)C2)cn1 Cc1nc(C(=O)NCCC2(NC(=O)C(C3CCOCC3)C)CCCC2)cc(O)n1 c1(C(=O)NC2C=CCN(C(c3ccc(C#C)cc3)=O)C2)ccc2nc(O)[nH]c2n1 Cc1cc(=O)oc(C)c1C(=O)NC(C)C(C(C)C)NC(=O)CC1(O)CCCC1 C(=O)(CC(C(F)F)NC(=O)CCCCCn1cc(C(C)N(C)C)nn1)OC n1(CC(=O)NCC2(CN(C(C(CC)COC)=O)C)CC2)ccc(C)cc1=O c1(CCNC(c2sccc2Cl)=O)ocnc1CNC(C1(C2CCCO2)CC1)=O N1(C(CC(C)Sc2cn(C3CC4C=CC3C4)nn2)=O)CCC(OC2CC2)CC1 Cc1nn2c(C)c1OC2.C(C(C)(C)C)OCCNC(=O)OC(N)=O N1(C(C2(CC#C)CC2)=O)CC(NC(C2(C(F)(F)F)CC2)=O)CC(C)(C)C1 Cc1nc(C)c(C(=O)N(C2CCCC(N(C(=O)C(=O)N(C)C)C)C2)C)[nH]1 C1(C(N2CC(CCNC(c3sccc3Cl)=O)(OC)C2)=O)CC2CCC1NC2=O Cc1cc(CCC(=O)NCC(C)CNC(c2cc(CN(C)C)on2)=O)on1 C(=O)(CC1=NNC(=O)C1)NC(CC(C)NC(C1CC2CCCC(C1)C2)=O)C C(=O)(C(F)CC1CC1)NCC(C)OCC=C.C1(=O)C(C)(C2CC2)N1C C1CC(NC(C)=O)C(=O)N2CC(C2)C(=O)NCCN1C.c1(C)nn[nH]c1Cl.CS Cn1cc(C(=O)NCCNC(c2ncoc2CCC(F)(F)F)=O)c(O)n1 N1(C(C2CC2F)=O)CCN(C(c2ccco2)=O)C(c2ccc(F)c(F)c2)C1 C1(NC(CCCC)=O)CN(C(C2(C)CCCS2(=O)=O)=O)CCC1F c1(C(N2C(CN(C(c3cnco3)=O)CC)CCC2)=O)cc(N)cc(F)c1 N1(C(c2ccc(C)[nH]2)=O)CC(C(=O)N(C2CCN(C)C2=O)C)CC1(C)C c1(C(N2CC(C(C)NC(C3CCC(=C)CC3)=O)C2)=O)c(F)cc(F)cc1F CCCCC(C)CCC(=O)NC1(C(=O)NC2CC(C)CC(C)(C)C2)CCCC1 CC1CCN(C(=O)C(=O)NCCN(C(=O)Cc2nccn2C)C)CC1 C1(C)(NC(C23CC(NC(=O)OC(C)(C)C)C2C3)=O)CCCC1O c1(C(=O)NC(CN(C(=O)CC2CCCOCC2)CC)C)ncccc1Br C12(CC)COC(C(=O)NCC3CC(F)CN3c3ncc(Br)cn3)(C1)C2 C#Cc1cc(C(N2CCCC(C)(CNC(=O)C(F)C(C)C)C2)=O)cc(F)c1 CC1CC(C(=O)NC2COCCN(Cc3cccnc3)C2)CCN1C n1(CC(=O)N(C2CN(C(=O)CC3CC3)CC2F)C)cc([N+](=O)[O-])cn1 Nc1ccc(F)c(C(=O)NC2CC(F)(CNC(=O)CSc3ccc(F)cc3)C2)c1 C1(c2cc(C(=O)OC)[nH]n2)CCCN(C(=O)Nc2[nH]c(C)nc2-c2nn[nH]n2)C1 C(=O)(C1=CC2CCC=CCCC12)NC1(CNC(=O)OC(C)(C)C)CC2CCCC12 C12(NC(C(C(C)C)C3CCC3)=O)CCCC1CN(C(=O)CCC(C)C)C2 CC1(O)CCN(C(=O)CCC2CCCN(C(c3cc(O)cc(F)c3)=O)C2)CC1 n1(CC(=O)NCC2OCCN(C(CC(C=C)C)=O)C2)nc2n(c(=O)c1=O)CCC2 N1(C(C2(C)CC2)=O)CC2(CC1CNC(c1ccn3ccnc3n1)=O)CC2(F)F c1(NCC2C(C)C2)cc(=NCCOCCc2ccccc2)[nH]cn1 c1(CC(=O)NC(C)CCNC(C2CC2c2ccncc2)=O)cccnc1O CCCC(C(=O)N1CC(n2cc(CC(=O)Nc3ccccn3)nn2)C1)NC(C)=O CC1CC(NC(c2sccc2F)=O)CN1C(c1ccc(SC(F)(F)F)o1)=O c1(-c2c(CNC(c3ccc(N(C)C)s3)=O)ccnc2)cncc(C2CC2)c1 CC(CNC(c1n[nH]cc1CNC(=O)C(C)(Cl)Cl)=O)CC(F)(F)F c1(C(=O)NCCOC2CN(C(C3(C)CC3(F)Cl)=O)C2)ccc(S(N)(=O)=O)cn1 S(=O)(=O)(c1[nH]c(=NCCC2(CO)CCC2)ccc1Br)N(C)CC1C(C)CCCC1 CN1CCN(C(=O)NC23CCC(C(=O)OC(C)(C)C)(CC2)C3)C(CO)C1=O C1(C)(C(N(CC(C)C)CCC)=O)CCCN(c2nccc(C(F)(F)F)n2)C1 c1(C(=O)NC(CC(C)NC(c2ccc(C#N)c(F)c2)=O)C)cc2c(o1)CCCC2 C=CC1CN(C(=O)CC2CCCOCC2)CC1NC(c1cnc(C)cc1C)=O C=CC(C)(CCOC)C(=O)N1CCN(C(=O)CN2CCCNC2=O)C(C(C)C)C1 Cc1ccncc1CC(=O)NC(C1CCCC1)CNC(=O)Cn1ccnc1C C#Cc1c[nH]nc1C(N1CCCC1C1(C(=O)NC(CC=C)CC=C)CC1)=O N1(CCC(=O)OC)CCC(NC(=O)CCN2CCCCC2C)C(O)C1 c1(N(C)C)ccc(C(=O)NCC2CC(O)CN2C(=O)C(O)CF)cc1 c1(CC)nnc(NCC2C(C)CCCN2C(=O)CN2CCC2)c(C#N)c1CC C1(C(=O)NCC2CN(C(CC(C)O)=O)CC2C(F)(F)F)CSc2ccccc2O1 N1(C(C(CNC(c2c(C)ncnc2)=O)CC2CC2)=O)CC2CCC(C1)C(=O)O2 C#CC1CC2CCC1N(C(=O)C(C1CCCC1)NC(C1CC3(CCC3O)C1)=O)C2 Cc1ccnc(C)c1C(=O)NC1CN(C(c2ccc(Br)cc2F)=O)C2CC12 C(=O)(CC1=CCCCC1)NCCN(C(=O)CN1CCCCC1)CC N1(C(C2(SC)CC2)=O)CCCC(C(=O)N(C)CC2CCCCC2)CC1 C1(NC(=O)CC2CC2(Br)Br)CC2(C1)CC2NC(=O)CC1OCCO1 C=CCC(CNC(c1nonc1N)=O)C(=O)NC1CC2C=CC1C2 C#CCC(CC(F)F)C(=O)N1CCN(C)CC1C(=O)NC(CO)C1CCC1 C1(C(N(CC#C)CC)=O)C(CNC(=O)C(C)NC(=O)CC)C1(F)F Cc1[nH]c(C#N)cc1C(N1CCOCC1CCNC(c1cnc(Br)s1)=O)=O C(=O)(C(O)C(C)CC)N(C1CCN(C(c2n[nH]cc2C)=O)CC1)CC#C c1(C(=O)NCCCN(C(C=Cc2ccc(CC)o2)=O)C2CC2)ccc(O)c(F)c1 C1(NC(C(CC#C)C2CC2)=O)(CC)CCCN(C(C2CCC(CC)CC2)=O)C1 N1(C(C(CC)CN(C)C)=O)C(CC(=O)NC2CCN(CC)C2C)C2CCCC12 N1(C(C2(OC)CC(C)(C)C2)=O)CC(O)(C2(CNC(C3CN(C)CCO3)=O)CC2)C1 N1(C(Cc2nc(C)sc2C)=O)CC(CNC(c2ccccc2F)=O)OC(C)(C)C1 N1(C(CCC=CC(C)C)=O)CCOC(C)C1C(=O)NCC1CCCO1 C1(NC(c2ccc(CC)cc2)=O)CCN(C(c2ccncc2F)=O)CC1O c1(C(=O)NC2CN(C(C(C)(C)NC(=O)OC)=O)CC2O)cc2ccsc2s1 Cc1cc(CC(N2CCC(C(C)(C)C(=O)N3CCC(C)C3)C2)=O)cs1 C1(C(N2CCC(CC)(CC)C2)=O)C2CCCC2CN1C(=O)CCOC(=O)NC C1(NC(C(Cn2cccn2)NC(c2ccc(O)cc2)=O)=O)C2C=CC(C2)C1CO c1(C(N2CCC(CN(C(c3cc(SC)c(C)o3)=O)C)C2)=O)cn2ccsc2n1 C(=O)(C1=CCc2ccccc21)N1CCCC(CNC(C(CCC)C#N)=O)C1 c1(C(=O)NC2C(CNC(CCCOC)=O)C2)cc2n(n1)CCNS2(=O)=O N1(C(Cc2cccc(CC)c2)=O)CCC2(CC2NC(=O)CCC(C)C)C1 C(=O)(CS(=O)(=O)CCO)N1CC(C(=O)NC2C(CCOC)C2)C(C)C1 c1(C(=O)NCC2CN(C(C3CSC3)=O)CC3(CCC3)O2)ccc2nc(O)oc2c1 C1(NC(c2nc(COC)oc2)=O)CCN(C(=O)C(C)CN(C)C)CC(O)C1 CCC(C(=O)N1CCC(C)C(NC(=O)CN(C)CC)C1)C(C)O C(=O)(C(CC(C)C)C(C)C)N1CC(C(=O)NC(CC#C)C)(Cc2ccccc2)C1 C#CC1(C(=O)NC2(COC)CCCCC2)CN(C(=O)CCCCC2CC2)C1 O=C(CCC(=O)c1ccncc1)NCCCC1CCCCN1C(=O)C(F)C1CC1 C(=O)(C(C(C)(C)C)NC(=O)C(C)CCOC)NCC(CC)(C)CO Cc1cccc(C(N2CC(C(=O)NCCC(C)C)C3(CC3)C2)=O)c1C#N N1(C(C(CC#C)C)=O)CCC2CN(C(=O)C=C(C)C(C)(C)C)CC2C1 C1(NC(C(c2nnnn2Cc2nnn(C)n2)SC)(C)C)CCC2(CC2)C1 C1(CC(=O)NCc2ccc(NS(=O)(=O)c3cccs3)cc2)CC(O)C12CCC2 C1(NC(CCN(C(=O)C(c2ccnn2C)C)CC=C)=O)CCCC(C)C1 c1(C(N2CCN(C(CNC(CCSC)=O)C)CC2)=O)cnc2ccnn2c1 N1(C(C=Cc2cnc(C)s2)=O)CC(C)CN(C(C2CCSCC2)=O)CC1C C1(C2CCCN(C(c3ccc(Cl)cc3)=O)C2)(NC(CC(CC(C)C)C)=O)CC1 C1(C)(CNC(C(C)OCC)=O)CCCN1C(c1oc(CO)cc1C)=O C1(NC(C2CCC(CNC(CCC(=C)Cl)=O)C2)=O)C2CCC3C(C2)CC13 c1(OC)cnc(C(=O)NCC(C2CCOC2)NC(=O)CNC(C)=O)nc1 C=CC(C)(CC)C(=O)N1CC(F)(CNC(c2ccc(CNC(C)=O)c(F)c2)=O)C1 C12(NC(C3C4CC4C4CC34)=O)CCC(CC1)N(C(=O)CS(=O)(=O)CC1CCCO1)C2 c1(C(=O)NC(C)CNC(C2CCCC(O)C2)=O)cccc2c1NCCNC2=O Cc1cc2ncc(C(N3CCCCC3Cc3cn(CCCF)nn3)=O)c(C)n2n1 CC(O)(CC(=O)NC1(CNC(C2(C3CCCO3)CCC2)=O)CCCC1)C(F)(F)F Cc1cc(CNC(=O)C(CC(C)C)N(C(=O)CCCCNC(N)=O)C)cc(C)c1 N1(C(Cc2c(C)nc(C)s2)=O)CCCN(C(=O)CC(F)(F)C(F)F)C(C)C1 N1(C(C2CC(C)C2)=O)CC2CC(NC(=O)C(C)(C)COCC(F)F)CC(C2)C1 c1(C(N2CCCC(N(C(=O)Cc3cccs3)C)C2)=O)sc2cccc(F)c2c1Cl C(=O)(CCCCN1CCOCC1)NCC(CO)NC(C1C(COC)C1)=O c1(C(C(=O)N(CC(C)(C)NC(=O)CCC2CCC(=O)N2)C)OC)ccccc1F C1(NC(c2cnn(C)n2)=O)CN(c2nc(C(N)=O)ns2)CC2(CCOCC2)C1 C(CC1=CCN(C(c2ccc(Cl)c(C)c2O)=O)CC1)NC(C(CCN(C)C)O)=O N1(C(CNC(c2ccccc2)=O)=O)CCOC(CNC(=O)Cc2cnccn2)C1 CCCC(C(=O)OC)C(=O)N(C)CC=CC(N1CCC(O)(CC)C1)=O C1(NC(c2ccn3ccccc23)=O)CCN(C(C2CC23CCC3)=O)CCC1(F)F c1(C(=O)NC2CN(Cc3c(C)cc(O)cc3)CC2C#N)cc(Cl)c(Cl)c(Cl)c1Cl C1(C(N2CC(CCNC(C3(O)CCCC3)=O)C2)=O)CC(C2CC2)=NO1 c1(NC(C2C3CN(C(=O)NCC(=O)OCC)C2C3)=O)cc(Cl)cc(I)c1 C1(CNC(CN(CCC#C)C)=O)CC(C)CN(C(C2CC3CCC2O3)=O)C1 C(=O)(C(C)C(C)(F)F)NCC12C(CN(C(c3[nH]cc(OC)c(=O)c3)=O)C1)C2 C1(NC(c2cccc(-c3cnco3)c2)=O)CCN(C(c2cc(CO)[nH]n2)=O)CC1 C(C1=NOC2CCCC12)NC(C12N(C(C3OCCN(C)C3)=O)CC(C1)C2)=O N1(C(c2occ(C)c2)=O)CCCC(C2CCN(C(=O)CC3=CCCC3)C2)C1 N1(C(CC)Cn2ccnc2-c2cccc(-c3ccc(C)nc3)c2)CC2CCC1C2 c1(C(C)=O)ccccc1C(N1CC(C(C)NC(=O)C(F)OC(F)(F)F)C1)=O C(=O)(C(C)(F)C(F)(F)F)NC12CC(CNC(C(C=C=C)C)=O)(OC1)C2 N1(CC)CCN(C(C2(F)CCCN(C(C3CC=CCC3)=O)C2)=O)CC1=O c1(C(N2CCN(C(C3C4CC5C(C4)C35)=O)CCC2C)C)cc2ncccc2[nH]1 c1(C(N2CC(CN(C)C(C3SCCCS3)=O)C2)=O)cccc(C(C)(F)F)n1 C(c1ccc([N+](=O)[O-])s1)=CC(=O)NCC1(C(C)NC(c2cc(Br)no2)=O)CC1 Cc1cncc(C(=O)NCC(CC2CCCC2)C(=O)NC(C2CCCCC2)C)c1 C1(C(C)NC(C(C)C2CCOC2)=O)CCCCN1C(=O)CCOCCN(C)C Cc1nc(C(=O)C(=O)NCC(O)CN(C)C(C2CCCO2)=O)cs1 C1(C(N2CC(C3(NC(Cn4nnc(C)n4)=O)CC3)C2)=O)CCC2C(C1)C2(F)F c1(CNC(C2C(CC)C2)=O)ccc(-n2cc(COc3ccccc3N)nn2)cc1 C1(C(=O)NCCc2cccs2)CN(C(c2cccc(I)c2)=O)CCC1O C(CCCCC(=O)N1CC(NC(=O)CC2OCCCO2)C(C)(C)C1)N(C)C N1(C(c2c(C)noc2C(F)F)=O)CCN(C(C2CCC(=O)N2C)=O)CC(O)C1 c1(OC)cc(F)ccc1C(=O)NCCN(C)C1CC1 N1(C(Cc2c(C)con2)=O)CCN(C(=O)C(N2CCNC2=O)C)C(CC(F)F)C1 CCCCCC(C)CC(=O)NCC1(NC(=O)COCC(=O)OC)CC1(F)F C1(NC(c2cncc(CO)c2)=O)C2CCC(C2)C1C(=O)NOC1CCOCC1 C1(NC(C=CC(C)(C)C)=O)CN(C(c2ncccc2O)=O)CCC1O n1(CC(=O)NCCN(C(C(C)OC)=O)C2CC(C(=O)OC)C2)cc(Br)c(C)n1 Cc1nc(-c2nc(C3CCOCC3)nn2Cc2ccncc2)sc1C N1(C(C(CCCOC)NC2C3CC4C(C3)C24)=O)CCCC(O)(C(F)(F)F)CC1 C(=O)(CCCCCS(N)(=O)=O)N1C(C2(NC(=O)C=CC3CCCC3)CC2)CCC1 NS(=O)(=O)CCC(=O)NCC(O)CNC(C1COCCO1)=O c1(C(=O)NCC2(C)CN(C(=O)Cc3cnsc3)CCO2)cc(Cl)c(F)c(Cl)c1 C1(C(N2CC(O)(CNC(C3(Br)CC3(F)F)=O)C2)=O)CN2CCN1CC2 Cc1ccc(C(=O)NCC2CC(OCC(=O)NC(C(O)CO)C3CC3)C2)n1C C12Cc3ccccc3N1C2=O.c1(COC(=O)OC(C)(C)C)cc2ccccc2s1 CC1(C)C2CCC13CCN(C(=O)NCc1cccc(Cl)c1)C3C2 N#Cc1cc(C2(NC(C3CC4CC4N3S(=O)(=O)CCCl)=O)CC2)ccc1F Cc1cc(F)ccc1C(=O)NC1CCN(C(=O)OC(C)(C)C)C1C1CC1 c1(OC)cc(C(N2CC(CC(N3CCC(C)(O)C3)=O)C2)=O)cc(Br)c1Cl CC1CC2(CCN(C(c3ccc[n+]([O-])c3)=O)CC2)CN1C(C1CC1C(F)F)=O N1(CCN)CCc2sccc2C1C.c12cc(ncn1)N2C.N1(C(C)=O)CCC(C=O)C1 C(=O)(C1=CCCOC1)NCC(CNC(C(c1ccccc1O)C)=O)(C)O C1(C)(CC)CCN1C(C1CC(CCNC(=O)C(C2CCCC2)OC)C1)=O c1(C(=O)NC(c2cn(-c3ccc(C)cc3)nn2)C)cc2c([nH]1)CCC(C)(C)C2 NS(=O)(=O)CCCC(=O)N(C1CCN(C(c2cc(F)c(N)c(F)c2)=O)C1)CCO c1(NC(C2C(NC(CCC(C)C)=O)CCC2)=O)cc2ccccc2[nH]1 c1(C(=O)NCCC(C)NC(=O)C(=O)NC2CC2)cc(OC(F)F)cc(F)c1 CC1CCC(CCNC(c2cncc(CNC(C3CCC(F)(F)C3)=O)c2)=O)CC1 c1(NC(N2CC(C(C)C)C2)=O)cc[n+]([O-])cc1.C12C(C1(C)C)C2OC c1(CC)ccc(OC)cc1F.c12cccc(c1)CC(=O)NCc1nnc-2o1 N1(C(c2c(C)ncn2C)=O)CCCN(C(=O)CC2CC3CCC2O3)C(C)C1 Cc1ccc(C(=O)NC2(CO)CCN(C(c3cnn(CCF)c3)=O)C2)c(N)c1C c1(C(=O)NCCC(C)(C)NC(c2n(CC#C)ccc2)=O)cn(C)c(=O)cc1C C12(C(=O)NC(C)CCC(=O)OC(C)(C)C)CCCCC(=O)N1CCC2 CC1(C)CCN(C(=O)Cc2cncs2)CC1NC(=O)COc1ccc(F)cn1 Cc1ncc(CNC(C2CC(C)N(C(c3nccs3)=O)C2)=O)n1C C1(C(=O)Nc2cccc(O)c2)(CNC(C=CCCC)=O)CCCC1C CCC(C)(C(=O)NC(CNC(C1(CC(F)(F)F)CC1)=O)CO)OC n1(CC)nc(C(=O)NC2(C)CN(C(C3(N4CCOCC4)CC3)=O)C2)c(C)n1 C1(NC(C2ON=C(C)C2)=O)CCOC12CCN(C(c1ccc(C)c(O)c1)=O)CC2 C1(NC(=O)COc2cccc(F)c2)CC(Nc2nccn3nnnc23)C12CCC2 C1(C(=O)NC(CCN(C(c2c(C(C)C)noc2)=O)C)C)CCn2ccnc2C1 C1(CCNC(CN(C)C)=O)CCCN(C(c2ccnc(C(F)F)c2)=O)C1 C12(C(N3CCC(NC(c4n[nH]c5c4CCC5)=O)C(F)C3)=O)CCOC1CCOC2 c1(C(=O)NCC(CNC(C=CC(=O)OCC)=O)C)ccc(OCCOC)cc1.C1CC1 N1(C(COCCC)=O)CC2CCC(C1)N2C(C1(Cc2ccccc2F)CC1)=O c1(N(C)C)cc(Br)cc2cncc(N3CCCC(C)(O)C3)c12 N1(C(=O)NCC(=O)NCC(C)(O)C2CC2)CCC(OCC(F)F)C1 C1(NC(c2c(Br)ccc(OCC)c2)=O)CC2CCC(C1)N2C(C1(C)CCC1)=O Cc1nc(N2CCCC(NC(=O)CCC3CCCN3C)C2)cc2nncn12 C(CC(C(=O)N1CC(NC(C)=O)C1)NC(c1cnc(OC)s1)=O)OCC CCC(C)(C)CC(=O)NCC1(C)CCCN1C(=O)CCn1cnccc1=O N1(C(c2c(NC)cccc2)=O)CCCC2(CCCN2C(=O)CCCCCOC)C1 C12(C(N(CCCc3nn[nH]n3)C)=O)CCC1CN(C(=O)CNC(N)=O)C2 CCC1=C(C(=O)NC2(C(=O)N(C)CC3(N(C)C)CCCC3)CC2)SCCO1 S(=O)(=O)(c1cnn2ccc(=NCc3cc(C4CC4)nn3C)[nH]c12)N(CCCC)C CCCCC(C(=O)N1CCC2(CC2NC(=O)CCc2cc(C)on2)C1)C(C)C N1(C(CC(C)CCc2ccccc2)=O)CCC2(C1)NC(=O)N(C)C2=O N1(C(C(C(C)NC(C=CCCC)=O)C)=O)CC2(C1)NC(=O)NC2=O N1(c2snc(COC)n2)CCC2(CCCC2NC(c2nccc(Cl)c2F)=O)CC1 N1(C(CCN(C(CCCC(=C)C)=O)CCO)=O)CCC12CCCOCC2 c1(C(C(N2CCC(C)C2=O)C)=O)ccc(-n2cncn2)cc1 C12(CCOC1)C(=O)N2CC1(CNC(COC)=O)CCCO1.C1(CC2CC2)CC1 C12(NC(C=Cc3c(C)cc(C)c(C)c3)=O)CCCC1N(C(=O)C1CC1)CCC2 C1(CNC(C(C(CC)C)O)=O)CN(C(=O)Cn2nc(Cl)ccc2=O)CC12CCC2 C1(C(=O)NCC2CCC(OC)C2)CC(NC(C2(C(=O)NC)CCCC2)=O)C(O)C1 C1(NC(C(c2ccc(F)cc2)(C)C)=O)CN(C(c2ccnc(F)c2)=O)CCC1(F)F c1(-c2scc(CN(CC(=O)N(C34CC(C3)C4)CC)C)n2)ccc(C)cc1 C1(NC(C2(CC)CCOC2)=O)CC2CC(NC(c3cc4c(s3)CCC4)=O)C2C1 C1(N(C(=O)Cc2nc(=N)[nH][nH]2)C)CC2CCC(C1)N2C(C1CCCS1)=O C#Cc1cncc(NC(C2CN(C(=O)CN3CCOCC3)C2)=O)c1 n1(CCNC(C2(CF)CCC2)=O)cc(-c2ccncc2)nn1 c1(CC(=O)NCC(CNC(=O)CCSCC(N)=O)OC)cccc(SC)c1 N1(C(CC2(CC(=O)OC)CC2)=O)CC(C(N2CC(C(C)OCCO)C2)=O)C(C)(C)C1 N1(C(CC(C)OC)=O)CCC(C2CC2)C1C(=O)NCC1CCC1 C(=O)(C1=COCCC1)NC1CC(C(N2CCC(SC)C2)=O)C1 c1(OC)ccc(Cl)c(S(=O)(=O)N2CCCCC2C)c1 CN=C(NCC1CC12CCC(F)(F)CC2)N1CCC(SC)C1 C(=O)(CN=c1cc[nH]cc1)N1CC(CCC)C(C(N2CCC(C(C)(C)O)C2)=O)C1 C1(C)(C(=O)NC(C)Cn2cc(CNC(C3CCOC3)=O)nn2)CCNC1=O c1(C(N2C(C3CCCN(C(C4C(=C)C4)=O)C3)CCCC2)=O)cc(C)ccc1F c1(N(CCCNC(c2n[nH]c(C)c2Cl)=O)C2CC2)cnc2ccccc2n1 C(=O)(C#CC1CCC1)N1C(C(=O)NCCN(c2ccccc2)C)CC1 c1(SC)nccnc1C(=O)NCC(C1CCN(C(=O)Cc2csnn2)CC1)O C1(CC(=O)NC2C(NC(Cn3ncc(C)c3)=O)C2)CCCN(CC(F)(F)F)C1 c1(OC)cc(C=CC(=O)NC(C)C(C)NC(C2CC=CCC2)=O)ccc1F N1(C(C2C(C)(C)C2)=O)CCC(CNC(c2cc3ccccn3n2)=O)C(F)(F)CC1 N1(C(CCCC2(CNC(CC3N(C)CCC3)=O)CCC2)=O)CCCCC(C)(F)C1 Cc1cc(-c2csc(C(N3CCCC(F)(F)C3)=O)n2)ccc1F c1(C2(C(=O)NCC(C)NC(C34CC(OC)C3C4)=O)CCC2)ccc(C#N)cc1 C1(NC(C(CN(C)C)O)=O)CN(C(c2cccc3c2OCC3)=O)C2CCCC12 C1(C(=O)NC(CCCNC(c2cc(C)ns2)=O)C)CN2CCC1C2 C1(NC(CC2(NC(C)=O)CC2)=O)CCN(C(c2cc(O)cc(O)n2)=O)C(C)C1 N1(C(C2(CCOC)CC2)=O)CCC(CC(C)NC(C2CC2(Cl)Cl)=O)CC1 N1(C(CN(C(C(C)C)=O)C)=O)CCCC(C)C1CNC(=O)CNC1COC1 C=C1CCC(C(=O)NCc2cc(C(=O)Nc3ccccc3F)ccn2)CC1 CC1(C(N2CC(O)(CNC(c3ccnc(O)c3)=O)C2)=O)COC(=O)C1 C1(C(C)C)(C(=O)NC2CCCC2F)CCN(C(c2ccc(O)cn2)=O)C1 c1(N(C2CC3CC2CN3)C(Cc2cnc(C)s2)=O)cc(Cl)cc(Cl)c1 c1(C(=O)NC2C(NC(c3cc(-c4ccn(C)n4)on3)=O)CC2)cncc(Cl)c1Cl c1(C(=O)NC2CC3CC2CN(C(c2ccc(Cl)s2)=O)C3)cccc2c1CCOC2 N1(C(CC=CCC)=O)CCCC(N(CCF)C(C2CCC(C)(C)O2)=O)C1 N1(C(CCOCC)=O)CC(C)OC2(CCN(C(=O)CSc3ccccn3)C2)C1 c1(C(N2CCC(C(C(=O)NC(CCC=C)C3CC3)C)C2)=O)cccc2c1CCC2 CC1CC(N2CCOCC2)CN1C(=O)C(C1CCCO1)C1CC1 CCCCCCC(CC)NC(=O)C(CCSC)NC(C1CCCCC1)=O c1(NC(C)C(F)(F)F)ccc(C(F)(F)F)cc1S(=O)(=O)Nc1cccc(Cl)c1Cl C1(F)(CNC(C(COC)(C)C)=O)COCCN(C(=O)C(O)CCN(C)C)C1 C(=O)(CC(C)C(=O)OC)NC(CCC)C(=O)N(C)CCc1noc(C)n1 C1(C)(CC(=O)N(CC=C)CC2CC2)CCN1C(=O)C(C)(C)O C1(NC(CNC(CN(C)CCO)=O)=O)CCOCC1NC(=O)C1=CSCS1 n1(CC)nc(C)cc1C(N1CCC(C(=O)NCC2CC23CCC3)(CO)C1)=O N1(C(C(C2CCCC2)NC(C)=O)=O)CC2CC(NC(=O)Cn3nccn3)C1C2 N1(CCC(N2C(C)C(NC(=O)C(=O)NCC3CC3)CCC2)=O)Cc2ccccc2C1 C1(CNC(c2c(C(C)C)nns2)=O)CC2CCC(C1)N2C(C1(C#N)CC1(C)C)=O CCC1=NOC(C(=O)N(CC(C)NC(c2ccc(C3CC3)o2)=O)CC)C1 c1(C(=O)OC)cccc(C(N2CCC(C)(CNC(=O)CC3CC=CCC3)C2)=O)n1 CC(C)CC(C)C(=O)NC(C1CCCC1)CNC(c1ccnc(C(C)(F)F)c1)=O Cn1nc(C(N2CCCCC2C(C)(C)C(=O)NC(C2(CO)CCCO2)=O)=O)cc1CO C(=O)(C(CN)CC(=O)Nc1ccnc(OC)n1)OC N1(C(c2c(OC)cncc2)=O)C2CCC1CN(C(c1scc(OC)c1Cl)=O)C2 N12CCC(C)(CC1)C1(CC1)C2=O.C1(C(O)CC)(CCC)CC1 N1(Cc2nnc(CC)s2)C2CCC1CN(C(C1CC(=O)NC1(C)C)=O)C2 CCC(CCC(=O)NC(c1nccnc1C)C)NC(=O)C(F)CC1CCOC1 N1(CC)CC(NC(=O)C(C)NC(c2coc(CO)n2)=O)C(C)(C)C1 Cn1cc(N)c(C(N2CCCC(N(C(=O)CN3CC4CC4C3)C3CC3)C2)=O)n1 C1(NC(c2c(CC)n(-c3ccc(C)cc3)nc2)=O)CCNCC(C)(C)C1 C1(C(=O)NC(C)C(C)(C)NC(N)=O)CCn2nncc2C1.C12CCN(CC1)C2=O N1(C(c2ccc(C#C)cc2)=O)CCCC(C2CC2NC(c2cc(C)ns2)=O)C1 c1(CSC)noc(CC(=O)NCCN(C(=O)C(F)C2CCOC2)C(C)C)n1 c1(OC)ccc(C(N2CCCC2CC#N)C(=O)NC(C)C)c(Cl)c1 C=CC(C)(CC)C(=O)NCC1CC2(CC2)CN1C(c1cc([N+](=O)[O-])n[nH]1)=O C(CCC(=O)NC1(CCNC(C2CN(C3CCOC3)C2)=O)CCC1)=CCC=C CCC(C)C(C(=O)NC(COC(C)C)C(=O)NC1COCC1O)OC c1(CC(=O)OC2(C(=O)NCc3ccsc3)COC2)ccc(Br)c(O)c1Br C1(CCNC)=CCC(N=[N+]=[N-])CC(S(C)(=O)=O)=N1.C1(O)CC1 C1(NC(c2cn(CC(F)F)cn2)=O)CCN(C(=O)CCc2cocn2)C1 N=c1cc(-c2cnc(C(=O)NCCC3CC3)nc2)cc[nH]1 C(C)(C)(CC(F)C(=O)NCC1CCN1C(C)(C)C)NC(C(CSC)C)=O CCC(O)(CNC(=O)CC(C)CNC(=O)COc1cnn(C)c1)CC N1(C(c2cc(OC)n[nH]2)=O)CC(C)CCC1CNC(=O)C=Cc1ccoc1 C1(NC(CCSCCCC)=O)CN(C(C23CCCCC2C3)=O)C2(CCOCC2)C1 c1(C(N2CC(NC(C3(CC#C)CCOC3)=O)C2)=O)ccccc1CC1CC1 Cc1ccc(C(N2CCC2Cn2cc(-c3cccnc3C)nn2)=O)cc1 C1(c2nn[nH]n2)(NC(CC)(C)C2CCCO2)CCC2OC(C)(C)OC12 C1(C(=O)NC2(C)CC(NC(COCCN(C)C)=O)C2)Cc2ccccc2S1 C1(C(=O)NCc2csc(O)n2)(CNC(=O)CC2CSC2)CC12CCC2 N1(C(C)=O)CCN(C(=O)CS(=O)(=O)NC2CC2N)C(C)CC1C.C(CCO)SC c1(CNC2CC(NC(c3ccc(OC(F)F)cc3)=O)C2)ccc(Cl)cc1 C1(CNC(c2c(C)cc(C)o2)=O)CN(C(=O)CCC(F)F)CCCO1 c1(C(=O)NCCC2N(C(CC=C=C)=O)CCCC2C)cnc2c(c1)NC(=O)CS2 c1(C(N2C(C)(CNC(C3CCC(=C)CC3)=O)CCC2)=O)cc(N)c(F)cc1C C(N=c1[nH]c2c(C)cc(C)cc2s1)c1nnc(C(C)=O)n1C C(=O)(C1=CCCC1)NCC=C(C(=O)NC1(CC=C)CCOC1)C CCC(CC(=O)N1CC(C2CN(C(c3c[nH]c4ccncc34)=O)C2)C1)C(F)F C(=O)(CC(C)(C)C=C)N1C(C2(C(=O)NC(C#C)C(C)OC)CC2)CCC1 N1(C(C2(C)CCN2Cc2cc(C(=O)O)ccn2)=O)CCC2(CCCC2)CC1 c1(C(=O)NC2C(C)CN(C(C3CCOCC3)=O)CC2)nn(C)c2c1CSCC2 CC12CCC(C(=O)NCCC3CCN(C(C4CC4F)=O)C3)(CC1)C(C)(C)O2 c1(N(C(=O)CCC(C)N(C)C)CCN(CCC)CCC)ccc(C)cc1O c1(C(C)=O)cc(C(=O)NCCCCC(C)NC(=O)Cc2ccc(F)cc2)oc1C c1(COC(C2(CC#C)CCCO2)=O)cccc2c1OC(C)(C)O2 n1(CC)nc(C(=O)N(C(C)CNC(c2ccc[n+]([O-])c2)=O)C)c(Br)n1 N1(C(C2(C)CC2(F)F)=O)CC2CCN(C(c3ccc([N+](=O)[O-])cc3)=O)CC2C1 C(=O)(CC1CCc2ccccc21)NC(c1ccc(OC(C)=O)cc1)CC CCN=c1ccc(C(=O)NC2CCCCN(C(C3Cc4nnsc4S3)=O)C2)c[nH]1 CCCC(C)(O)C(=O)N(C)CC1(O)CN(C(=O)C(CN(C)C)c2ccccc2)C1 c1(N(C)CC2CCCN(C(c3ccc(C(C)=O)[nH]3)=O)C2)cc2nnc(C)n2cn1 C1(N(C(=O)CC2CC3(CCC3)CO2)C)CC2CC(NC(=O)Cn3cccn3)C1C2 C(C(C)(O)C(=O)NC(C)CCNC(C1(c2ccc(C)cc2)CC1)=O)OC C1(NC(c2n(C)cc(Cl)c2)=O)CN(C(=O)CC(C)(C)C)CC2(CC2)C1 c1(OC)cnc(CN2CCC(C(N3CCC(C)(NC(C)=O)CC3)=O)C2)c(F)c1 Cc1ccsc1C=CC(=O)N(C)CC1CN(C(=O)CN(C2CCCC2)C)CCO1 N1(C(c2cc(O)ncn2)=O)CC2(C1)CN(C(c1ccn(C(F)(F)F)n1)=O)C2 C(=O)(C(F)C(F)(F)F)NCC1C(C)CCN1C(=O)COCCN(C)C c1(C(N(C(C)C(=O)NC2CCN(CC)C2)CC)=O)cccc(CO)n1 Cc1cc(C#N)ccc1C(N1CC(CNC(=O)Cc2cccnc2)CC1C)=O C1(N(C(c2c(C)nn(C)c2)=O)C)CN(C(=O)COc2ccc(Cl)cc2)CCC1C N1(C(C=CC)=O)CCC(CNC(c2ncc(C(F)F)s2)=O)C(F)(F)C1 N1(C(CSCCCC)=O)C2CCC1CN(C(c1n[nH]c3c1CCC3)=O)C2 C1(NC(C23CN(C(C4CNC(=O)N4)=O)C(C2)CO3)=O)CC1C1CCOCC1 CC1(C(=O)NCCNC=O)CCN(C(=O)C=CC(F)F)C1 C(CCCOC)(C(=O)N(C1CCCCC1)C)NC(C1C(CC)CCC1)=O C1(C(N(CC(C(=O)NC(CCCC=C)C)(C)C)C)=O)CC(C)CC(=O)N1 C(=O)(C1CCCc2nnn(C)c21)N(C1CC(C)C1)C(c1cc2n(n1)CCOC2)=O C1(C)(CN2CC3C(CNC(=O)OC(C)(C)C)(C3)C2)CCCCCC1 C1(C(C)NC(c2n(CC)ncc2)=O)CN(C(=O)CCN2CCC(F)C2)CCO1 C(C(=O)NC1CCCC(NC(=O)Cn2cc(C)cn2)C1)(C(C)C)OCC(C)C C1(CC(=O)OC(C)C)CCN(C(=NCC2CNC(=O)C2)NC2CCCC2)CC1 C(=O)(C(C)CS(C)(=O)=O)NCC1(C)OCCN(C(c2c(F)ccc(C)n2)=O)C1 c1(CC(=O)NCCN(C(=O)CCc2cc(OC)no2)CC)ccc(Cl)c(F)c1 CCC(F)(F)CC(=O)N1CC(C(C)NC(c2ncc(OC)cc2F)=O)C1 Cn1ncc2ncc(C(N3CC(NC(=O)CC4CC4)CC(O)C3)=O)cc12 C1(=CC)CCN(C(C2CC(NC(C3(OC(C)(C)C)CCCC3)=O)C2)=O)C1 C1(OC)CN(C(=O)C(C)(CO)OC(=O)Nc2ccccc2)CCNC1=O N1(C(C2CC(N)C2)=O)CC(=O)N2CCCCC2C1.CC(C)CC(O)c1cn(CO)nn1 N1(CCCC)CCC(CNC(=O)N(c2noc(C)n2)Cc2cc(C)cs2)C1 C=C(Cl)CC(C(=O)Nc1nccn1CC)NC(=O)CSC1CC1.C(=O)(C(C)CC)N N1(C(C(C(=O)NC)(C)C)=O)CC=C(C(=O)N(CC(C)(O)C2CC2)C)CC1 C1(CCNC(CC(C)c2ccco2)=O)CCN(C(=O)CCC2(C)CC2)CC1 N1(C(C=CCOC)=O)CC(NC(c2cc(F)ccc2F)=O)CCC(O)C1 C(=O)(CCC1=CCCCC1)NCCC1(C(=O)NC2(C(COC)O)CC2)CCC1 C1(NC(CCCC(=C)C)=O)CC(NC(c2ccc(CC)o2)=O)C12CCOCC2 N1(C(c2nc(C)oc2)=O)CCN(C(=O)CCc2ccc(CO)cc2)C2CCC12 Cc1ccc(Cl)c(OCC(N2CC=C(CNC(C3CCCC3(F)F)=O)CC2)=O)c1 CC1=C(C(=O)N2CC3CC3(NC(=O)CC3(O)CCCCC3)C2)CCC1 C1(C)(CN(C(=O)CSS(C)(=O)=O)C)Cc2ccccc2C1 C(CCC(C)NC(C1(C)CCCC1)=O)NC(C1C(C=C)C1)=O c1(CNC(C(C2(C)CC2)NC(C(SC)SC)=O)=O)ccnc(C)n1 CCC(F)(F)C(C)(C)C(=O)N1CC(C)CN(C(=O)CCC(C)OC)C(C)C1 Cc1ccc(-c2cnc(CN3C(C(=O)NC)CC4(CC4)C3)[nH]2)cc1F c1(OCC(=O)NC(C2(O)CN(C(=O)C(F)F)C2)C)ccc(Cl)c(F)c1 c1(OC)cc(C#N)ccc1CNC1CC(C(=O)Nc2ccc(F)c(C)c2)C1 CN1CCC2(CC1)CC2NC(=O)NCC1CN2CCCN1C2 c1(CC(N2CCN(C(c3cnns3)=O)CC2C2CC2)=O)ccc2ccccc2c1 N1(C(C(CC)OCCC)=O)CSCC1C(N1CC(CC(=O)OC)C1)=O c1(C(N(C2CC(O)CN2C(CCO)C(F)F)CC)=O)ccc(O)cc1F C(=O)(CCCCC#N)NCCN1CCN(C(Cn2c(C)cc(C)n2)=O)CC1 c1(C(=O)NCC2OCCC(NC(CC(C)C)=O)C2)cnc2c(c1)NC(=O)CO2 c1(C(C(=O)NCC(F)F)N(C)Cc2ccc(C)cc2)cccc(C(F)F)c1F C12CC3CCC(C1)N3C(=O)CCNC2=O.C=CC1CC1C(=O)NCC1CCC1 C1(CCNC(c2cc(C3CCCC3)no2)=O)CCN(C(c2cc(Cl)ns2)=O)CC1 c1(C(=O)NCc2ccncn2)n[nH]c2c1CCN(C(c1cnc(O)nc1O)=O)C2 C1(C(=O)NCc2cccc(C)c2)CN(C(C2(C)CCOC2)=O)CCN1C c1(CC(=O)NCCOCCn2cc(-c3cccc(C)n3)nn2)ncc(Cl)cc1Cl CC1(OCC(=O)NCC2(O)CC(CNC(=O)CC3OCCO3)C2)CCCC1 c1(C(=O)NC(CC)CN(C(=O)C=Cc2ccsc2)C)cc(C)c(F)cc1N c1(C(=O)NC(CNC(COCCC=C)=O)CCCC)ccc(=O)n(CCSC)n1 CCC(C)(C(=O)N(C)CC1CN(C(=O)CC2CCC(F)(F)C2)CCO1)OC C(=O)(CCC(C)(C)C(=O)OCC)NC(CC(CNC(C(CC)(C)CO)=O)C)C CC1(C)CCCCCC1NC(=O)CCCCNC(=O)CN1CCCC1=O c1(SCC)cncc(C(=O)N(C)CC2CN(C(=O)Cn3nnc(C)n3)CCO2)n1 N1(CC(=O)NCC(C)(C)OCC(=O)NCC2CC2Cl)CCOCC1 N1(C(CC2N(C(C(C)SC(C)C)=O)CCOC2)=O)CCC(O)C(C)C1 c1(C(=O)NCC2CCN(C(c3c(CC)c[nH]n3)=O)C2)cnn2c(N)ccnc12 c1(C(=O)NC(C)CCCCNC(C2COCCN2C)=O)cc2c(Cl)ccnc2s1 CN1CCOCC1CC(=O)NC1COCC1C(=O)NCc1ncc[nH]1 c1(OC)ccc(C=CC(=O)NCCN(C)C(c2ccnc(C)n2)=O)cc1OC C#CC1CN(C(c2ccnc(OC)n2)=O)CCN1C(C1OCCN(C)C1=O)=O C1(NC(CC2CCC(C)O2)=O)CCCCCCC1NC(=O)Cn1cnnc1 C(=O)(C1=CC12CC(NC(=O)OC(C)(C)C)C2)N1CCC(NC(=O)OC)C1 C1(C(N2CC(n3cc(C(N4CCCC4)=O)nn3)C2)=O)(OC)CCCC1 C1(CNC(CC)=O)CN(C(=O)Cn2nc(O)ccc2=O)C2(CCOCC2)C1 n1(COC)ccc(=NC(=O)c2ccc(S(=O)(=O)N3CCN(C(C)=O)CC3)o2)[nH]1 C(CCN=C(NCc1ccco1)N(C)CC1OCc2ccccc21)OCC c1(C(N2CC(C#N)C(NC(=O)Cn3ccnc3)C2)=O)cc(Cl)c(O)cc1O c1(C(=O)NC(CCCC)CNC(c2ccc(CC)cn2)=O)cn2cc(C)sc2n1 c1(NC2C3(CN(C(C4C(C)(C)CC4)=O)C3)CCC2)ncnc2cc(F)c(F)cc12 C1(N(C(C(CO)NC(C(C)(C)OC(C)C)=O)=O)C)CCCCC1C(N)=O c1(CCN(C(=O)C(=O)NCC2NC(=O)NC2=O)C2CCC2)cccc(Br)c1 CC(C)CCCC(=O)N1CCN(C2COCC2NC(=O)CCc2cn[nH]c2)CC1 C(C(=O)NCCCC(C)(C)NC(C1CCCC(OC)C1)=O)(C(C)C)OC C=CC1(C(=O)NCCCc2nncs2)CCN(C(=O)Cc2c(C)noc2C)C1 c1(NC(c2n(C)ccn2)C(C)(C)C)nc(=NC2CC(CO)C2)[nH]c2c1CCC2 C(CN=C(NCc1cc(C)nc(N2CCCC2)n1)NCC1CC1Cl)OC C1(C(=O)NCCCC2(CNC(C(C)N(C)C)=O)CCCC2)CC2C=CC1C2 CC1(O)COCCN(C(C2COC(CNC(=O)C(O)CN(C)C)C2)=O)C1 c1(CN2CC(NC(c3c(F)cc(Cl)cc3Cl)=O)C(O)C2)ccc(Cl)c([N+](=O)[O-])c1 C1(N(CC(N2CC(CNC(C3CCCO3)=O)C2)=O)C)CCN(CC(F)(F)F)CC1 c1(SC)ccc(-c2cccc(C(O)CN3CCCC3)c2)cc1 C1(NC(C2CC(C(F)F)C2)=O)CN(C(c2ccc3c[nH]nc3c2)=O)CC12CCC2 c1(N2CC3(C)C(C2)C2CCC32)nc(C(c2cccs2)(C)C)nc2cccnc12 C(C)(C)(CC(=O)N1CC(NC(=O)CO)CC1C)n1cc(-c2n(CC)ccn2)nn1 C(CC(C(=O)NCC(c1ccccc1)C)NC(c1ccnn1CCF)=O)=CC C1(N(C(=O)Cc2ccsc2)C)CN(C(=O)CN2CCCCCC2=O)CC12CC2 C(N=c1[nH]nc(CO)s1)C1CC(C)N(C(C2CCCCS2(=O)=O)=O)C1 N1(C(c2ccc(O)cc2F)=O)CC2CCN(Cc3cn4ccccc4n3)C2C1 c1(C(C(=O)CS(=O)(=O)CS)=O)cccc(O)c1N.c1(OC)cnc(C2CC2)s1 c1(C(=O)NC(CN(C(=O)C=CCF)CC)C)cc(OC(F)(F)F)c2ncccc2c1 c1(OC)c(C(=O)NC2CC(F)CN(C(=O)CC(=O)OC(C)(C)C)C2)cccc1Cl c1(C(C(=O)NC(C(=O)OCC)C)N(C2CCCCC2)C)ccc(C#N)cc1 c1(CCC(=O)NCC(CC=C)NC(C2CC2C2CC2)=O)ccc(F)c(F)c1 N1(C(c2nc(CC(C)C)sc2)=O)CCCCC(N(C)C(C2(CC(C)C)CC2)=O)C1 C1(CNC(c2cnn(C3CCCCO3)c2)=O)CN(C(c2cc(F)cs2)=O)CCO1 N1(C(C2C(C(=O)NCC#C)C2)=O)CC2C(CNC(c3nnsc3N)=O)C2C1 c1(OC)cscc1NC(C1CC(C)(NC(=O)CCCN(C)C)C1)=O c1(-c2cccc(C(=O)NCC3CNCC(C)C3)c2)cccc(C#N)c1 c1(C(=O)NC2(CCNC(C3C(C)OC(=O)N3)=O)CCC2)ccc(Cl)c(F)c1 C1(CC(=O)N(CCCOC)COC(C2CSCCS2)=O)CCCCC1(C)C c1(C(C)C(=O)NC2CC(N(C)C(C3CC4CC3C4)=O)C2)ccc(C#N)cc1 C(=O)(C(F)(F)C(O)C1CC1)N(C)CC1(O)CCN(C(C2CC(N(C)C)C2)=O)C1 C(CC(C)(C)C(=O)NCC1CCN1C(c1csc(-c2cccs2)n1)=O)OC c1(C(N(CC(C)NC(=O)CNC(N)=O)C)=O)ccc2c(Br)cncc2c1 c12ncccc1NC2=O.c12nc(co1)C(=O)NCC2N(C)C.C(C)(=O)N.CC N1(C(Cc2n(C)cnc2)=O)CC2(CNC(=O)COc3cccc(F)c3)CCC1C2 N1(C(CC2(CSC)CC2)=O)CC(O)CC1CNC(C1(c2nccn2C)CC1)=O CC1(C)CC(NC(=O)CC2CCN(C(=O)Cn3cncn3)C2)C12CCC2 c1(C(N2CC(O)(C(CNC(C(CC)SC)=O)(C)C)C2)=O)cc2c(cn1)OCO2 C1(CNC(C=C2CCN(C(CC(C)(C)C3C(C)C3)=O)CC2)=O)CCCC(C)(C)O1 c1(C(=O)NCCOC2CN(C(C(CC(C)C)OC)=O)C2)ccc(C)c(C)c1Cl C1(C(=O)NCCCN(C(CC(=O)NCC#C)=O)C)CC(=O)N(CCN(C)C)C1 c1(C(N(CC(C)NC(=O)CCC2CCCC2)C)C)ccc(F)c(F)c1 C(C)(C(O)C(F)F)NC(C1CC(CCNC(c2c(C)ocn2)=O)C1)=O CN=c1[nH]cc(C(N2C(C(=O)NC(C)(CC)CCO)CCC2C2CC2)=O)o1 O=C1CC2(CCN(C(c3ccnc(Oc4ccccc4)c3)=O)CC2)CN1 c1(C(N(C(C)CNC(c2cn[nH]c2)=O)CC)=O)ccc(Cl)c(Cl)c1C CN1CCCCC1C(N1CCCCC1CNCc1cccc(C(F)(F)F)c1)=O c1(C(=O)NCC2CC(F)CN2C(=O)C=Cc2cocn2)nnn2c1COCC2 c1(CNC(C2C(O)CCN(S(CCC)(=O)=O)C2)=O)n[nH]c2ccccc12 C1(NC(C(C)=C(C)C)=O)CCCN(C(c2cc(Cl)ccc2Cl)=O)CC1F C(=O)(C(C(C)O)NC(=O)CCc1cncs1)N1C(CN(C)CC)CCC1 CC1(C#N)CCN(C(C2CN(C(c3ccon3)=O)CC23CC3)=O)C1 c1(CC(N2CC(C)(NC(c3nc(C(C)=O)sc3)=O)C2)=O)cccc(S(C)(=O)=O)c1 C1(C)(COC)CC(NC(=O)CCF)CN1C(=O)CCc1ccnn1C C(=O)(CC(C)O)N(CCC(=O)N(CC(C)OC)C)C(C)C C=CCC(CC)C(=O)NCC(C)(C)NC(c1cnc2n1CCS2)=O c1(C(N2CC(C)C(NC(c3cocn3)=O)C2)=O)cc(O)nc2cnccc12 c1(C(N2CC3C(CNC(C=CC(C)(C)C)=O)(C3)C2)=O)c(F)cc(Br)cc1F C(CCC(C(=O)N1CC2(CCCC2)C1)NC(=O)CC1CCCCC1O)OC C1(CCNC(=O)NCCCc2ccc(C)cc2Br)CC2(CCOCC2)CO1 C1(NC(C2CCCOC2)=O)CC2CN(C(c3cc4ccncc4[nH]3)=O)CC2C1 c1(C(=O)NC(C2CCOC2)CNC(c2ccncn2)=O)cc2scc(Cl)c2[nH]1 C1(C(=O)N(CC(C)CNC(c2cnn(C(F)F)c2)=O)C)(OC)CCCOC1 c1(CC(=O)O)ccc(S(=O)(=O)N2CCN(Cc3cccc(I)c3)CC2)cc1.CCO C(CCC(C)C(=O)NCC1(C)CCCN1C(c1ccc(C)cc1OC)=O)OCC c1(NCCN2CCC(CSC)CC2)ccc([Si](C)(C)C)c(C(=O)O)c1 N1(C(C2(CF)CCN(C(C34CCC(OC)C3C4)=O)C2)=O)CCOC2(CCC2)C1 N(C(=NCCN1CCCC1)NCc1ccco1)CC1CC(C(F)(F)F)C1 c1(C(N(C2CC(NC(c3c(OC)ccnc3)=O)C2)C)=O)ccc2c(c1)COC2=O C1(C(=O)NCC2(C)CCN(C(c3ccc(O)nn3)=O)C2)CC1C1CCCCC1 c1(C(=O)NCC(CC(C)C)(C)NC(=O)CC(=O)N(C)C)cccc2nccn12 c1(C(=O)NCC2C(C(F)(F)F)CN(C(CSSC)=O)C2)cnc2c(c1)ncn2C C1(C(=O)NC2C(NC(c3ccc(Br)cc3)=O)C2)Cc2cccnc2C1 CC(C)(C(=O)N1CC(O)(CNC(=O)CC2CSC2)C1)C1CC1 Cc1csc2ncnc(NC(C3CC3c3cccc(C(F)(F)F)c3F)=O)c12 c1(C(N(CCCNC(C(C=CC)O)=O)C)=O)cc(O)nn1C c1(NC(C2CCCCN2C(=O)C(C)(C)N(C)C)C)nc(Cl)ncc1F C(=O)(CS(=O)(=O)C1CC1)N(C)CCC1CCCCN1C(C1(c2ccno2)CC1)=O c1(NC(=NCCCCl)NCC2CC2)ccc2oc(=O)ccc2c1 C1(NC(CC=C=C)=O)(CC)CCCN(C(=O)C2=NOCC2)C1 Cc1ccc(C#N)cc1C(=O)Nc1ccc(N2CCCC2)c(F)c1 C12(C(=O)NCCN(C(C3C4CCCOC34)=O)CC)CC(C)(CN1CC)C2 S(=O)(=O)(c1cnccc1C#N)N1CCCC(C(C)O)C1 CCC(N=c1nc(N2CCC3(CC3)C2)c2ncn(CC)c2[nH]1)c1cccs1 c1(CC)nn(C)c(CC)c1C(=O)NC(CCN(C)C(C1OCCC1C)=O)C(C)C CC(C)C(C)C(=O)NCC12CC(NC(c3cn(C(C)C)nn3)=O)(C1)C2 N1(C(C2OCCC(C)C2)=O)CC2(CCNC(=O)C(O)CC(C)(C)C)CCC1CC2 CC(CC(=O)N1CCCC1C(C)(C)NC(=O)CCc1ncc[nH]1)C1CC1 c1(C(N2CCC(CNC(C3C(C#C)C3)=O)C2)=O)ccccc1N1CCCC1 C1(C(=O)NCCC(CCNC(c2c(C)cno2)=O)C)CC2CC(F)(F)C2C1 C1(C(C)(F)F)(C(=O)NCC(CN(C(c2cncnc2)=O)CC)O)CCOCC1 C=CCCCCCCCC(=O)N1CC2C(C(=O)Nc3cccc(Cl)c3F)C2C1 Cc1ccc(C(=O)CCC(=O)NC23CC(NC(C4CC4(F)Cl)=O)(C2)C3)cc1 CC(O)(CC(=O)NCC(C)(C1CC1)NC(c1cncc(F)c1)=O)c1ccccc1 C(=O)(CCC(C)(C)[N+](=O)[O-])NCCN(CCC)C(c1cc(Cl)ccc1F)=O C(=O)(CCSCCNC(C1CCCO1)=O)NC(c1cc[nH]n1)C c1(OC)cc(CC(=O)NC2(CNC(=O)C(O)c3ccsc3)CC2)cc(OC)c1O CCCCC(CC)C(=O)N1CC(NC(c2ccc(CO)s2)=O)CC(F)C1 CN1CCN(CC(=O)N(C)CC2COCCN2C(c2scnc2Cl)=O)CC1 C=C(C)CCC(c1nnnn1CCC(=O)OCC)NCC(C)(COC)OC CCCN=C(NCCOC(C)C)NCC1(N2CCOCC2)CCSC1 C1(CNC(Cc2c(C)nc(S)s2)=O)CCC2(CCN(C(C3CC3CF)=O)CC2)O1 C(=O)(CC1=NNC(=O)C1)NCCN1CCC(NC(c2n(C)c(S)nc2)=O)CC1 CC(C)CC(=O)N(C1C(c2ccccc2)OCC(COC)N1)C(c1ccco1)C C(=O)(C(C)(C)C(=O)N1CCC1CNC(=O)CC12CCCC1C2)NC c1(C(N2CCC(NC(c3cnc(CC)[nH]3)=O)C2)=O)cc(F)cc(Br)c1 c1(-c2cn(CCC(=O)OCC)nn2)ccccc1CN(C)C(C1CC12CC2)=O c1(C(=O)NC2C(NC(Cc3c(C)cccc3F)=O)C2)cnc2ccccc2c1 CN1CCC(C(=O)NC2CC(NC(C3(C#N)CCC3)=O)C2)(C(F)F)CC1 c1(C(N2CC(CNC(C3CCC=CO3)=O)OCC2)=O)cc2c(o1)CCCC2 Cc1cc(C(N2CCCC2CNC(=O)CC2CCC(C)C2)=O)cc(C)c1F C(=O)(CC(C)CC(F)(F)F)N1C(CNC(c2cccc(C)c2)=O)CCC1 C1(C2CCCO2)(C(N2CC3CN(C(CC4(C)CC4)=O)CC3C2)=O)CCCO1 C#Cc1ccccc1CC(N1CC(C)CC1C(=O)NCc1occc1C)=O C1(n2cc(C(=O)Nc3snc(CC(C)C)n3)nn2)CCCN(C(=O)OC(C)(C)C)C1 N1(C(c2nc(COC)oc2)=O)CCCC2(CC(NC(=O)CN(C)C(C)=O)C2)C1 c1(CNC(C(C)CNC(=O)CCN2CCOC2=O)=O)c[nH]c2cnccc12 C1(C(=O)NCC2N(C(c3nc(CCCC)sc3)=O)CCC2)Cc2nccnc2C1 N1(Cc2cc(C)no2)CC2CC2(C(=O)NCCc2cc[nH]n2)C1 C1(NC(=O)CC2CC=CC2)CC(O)CN(C(c2cncs2)=O)C1 Cn1ccc2nc(N(C3CNCC3F)Cc3ccc([N+](=O)[O-])cn3)ncc12 c1(C(=O)NC2C(CNC(=O)Cc3ccc(F)cc3)C2)csc2ccccc12 S(=O)(=O)(c1ccc(NC2CCC2O)c(Cl)c1)NC1CCCC(CC(C)C)C1 C1(NC(Cc2cn(C(C3(O)CN(C(C)C(=O)N(C)C)C3)C)nc2)=O)CCCCC1C c1(NC(=O)CN)cccc(C2CC2)c1.c1(OC2(Cn3nccn3)CC2)noc(OCC)n1 C(c1ccccc1)=CC(=O)NCCN(CC)CC.C(C)(C)(C)OC(=O)N(C)C CC1(C)OCC2CC12C(=O)NCC1CC1NC(c1cc(Br)co1)=O c1(C(N2C3C(C(=O)Nc4c(C)cc(Cl)nc4)C(C3)C2)=O)c(C)cc(O)cc1C C1(C(N(C2CCC2)CC)=O)CCCC(NC(=O)CC2CC3C=CC2C3)C1 c1(CC(N2CC(NC(c3c(C)onc3)=O)C(O)C2)=O)cc2cc(Br)ccc2o1 C12(CNC(C3OCCC(NC(=O)CC4CC4)C3)=O)CCC(CC1)O2.c1ccccc1 C1(NC(C(C2CN(C(C(CC)(C)COC)=O)C2)OC)=O)CCN(C)CC1C#N C(=O)(CCC(C)(F)F)N1CC(C=C)(CC(=O)NCC2COCC(C)O2)C1 c1(CC(=O)NC2CC(CNC(C(CC)N(C)C)=O)C2)nc2c([nH]1)CCCC2 N1(C(CCN(CCC(C)(C)C)C)=O)CCC2(C1)CN(C(=O)C1=C(C#N)CCC1)C2 c1(C(=O)NCC2CC(NC(c3cc(F)ccc3F)=O)C2)cc2n(n1)CCCC2O C(C(=O)N=c1cc(C)[nH][nH]1)NC(=O)NC(c1ccc(F)cc1)(C(=O)OC)C C1(CN(C(CC(C)NC(=O)C2CC2)=O)C)OCCN(C)C1c1ccccc1 c1(C(N(C)CC2COCCN2C(c2cocn2)=O)=O)ccc(N)c2cnccc12 c1(C(N(C(C)CNC(=O)C(C)CF)C)=O)ccc(Cc2cscn2)cc1 c1(NC(c2ccc(C)s2)C)ccnc(N2CCC(c3ccn(C)n3)CC2)n1 CCCC(CNC(c1conc1C1CC1)=O)C(=O)NCCCN(C)CCOC S(=O)(=O)(CCC(=O)N1C2CCC1C(CNC(C1CCCS1)=O)C2)N(C)C c1(C(C)NC(=O)NCC2(CC)CCOC2)cc(Cl)cc(Br)c1 c1(C(=O)NC2CN(C(CN(C)C(N)=O)=O)C(C)(C)C2)cc(F)c(F)c(C#N)c1 c1(NCC2C(CNC(COCCC(C)C)=O)C2)[nH]c(=O)n(C)c(=O)c1C#N N1(C(C(C2CN(C(C3COCCC3(F)F)=O)C2)O)=O)C(CO)C2CC(O)C1C2 CC1(CNC(C2CC=CC2)=O)CCC(NC(C2(c3ccsc3)CC2)=O)C1 N1(C(=O)C=C2CCOCC2)CC2(CCN2C(=O)C(F)C2CCOC2)C1 N#Cc1ccc(CC(N2CCOC(CNC(C3CCC3(F)F)=O)C2)=O)cn1 Cc1cc(Cl)c(C(N2CCCC(C(C)NC(=O)CCC3CCC3)C2)=O)cn1 N1(C(C23CCC(CNc4c(C)cnc(C)n4)(OC2)C3)=O)CC2CCC(CO)(C2)C1 N1(C(C(C)OCCN(C)C)=O)CCCC(C)C1CCNC(=O)CS(N)(=O)=O C1(c2cn(CCC3(C)CC3)nn2)CCCCN(C(=O)C(C)(C)N2CCCC2=O)C1 c1(C(=O)NCC(C2N(C(c3n(C)nnc3)=O)CCC2)(C)C)cc2sccc2s1 N1(CCNC(=O)Nc2cn(C)nc2C(N)=O)C(=O)C2C3C=CC(C3)C2C1=O C12(C(N3CCC(C(=O)NCCCC(F)F)C3)=O)CCC(F)(CC1)C2 N1(C(=O)NCc2c(C)con2)CCOC(c2ccccc2)(C2CC2)C1 c1(NC)ncccc1C(=O)NCCOCCCNC(c1cc(SC)c(C)o1)=O c1(C(=O)NC2CC(NC(C(C)(C)c3ccns3)=O)C2)ccncc1O c1(C(=O)NC2(CCNC(C3(OC)CCOC3)=O)CC2)ccc(N=S(C)(C)=O)cc1 C12(CNC(C(c3cccs3)SC)=O)CC1CN(C(=O)C=Cc1cocn1)C2 n1(CC(=O)NC(CNC(CN(CCC#C)C)=O)C(C)C)nc(C)n(CC)c1=O c1(N2C(CN(C(c3n(CC#C)ccc3)=O)C)CCC2)ccnc(-c2nccs2)n1 C=CCC(CC)C(=O)NC(CNC(c1ccnc(O)c1Br)=O)C1CC1 C1(NC(=O)C2=CCCCC2)CN(C(C2CCOC2=O)=O)CC2(CC2)C1 C1(C(=O)NCC(c2ccccc2F)NC(C(COC)O)=O)CN(C)C(=O)N1 N1(C(c2c(C)cc(OC)c(Br)c2)=O)CCc2c(Br)ccc(Cl)c2C1 C12(CNC(c3ccc(CC)s3)=O)CC1CN(C(c1cnc(C(F)F)nc1)=O)C2 N1(C(CCSC(C)(C)C)=O)CC(C(=O)NCCCON)C1(C)C C1(NC(C=Cc2cnc(C)s2)=O)CC(NC(=O)C=Cc2ccnn2C)C12CCC2 Cc1cc(NCC(C)(CC(C)C)NC(=O)Cc2ccco2)c(F)cc1[N+](=O)[O-] c1(C(=O)OC)cccc(O)c1NC(C1CCN(Cc2cncc(Br)c2)CC1)=O C1(NC(COCC=C)=O)CCN(C(=O)Cc2ccc(C)c(NC)c2)CC1C c12ccc(nn1)[nH]c2=O.C(C)(C)(C(C)NC(=O)C(C)C)NC(CNC(=O)NC)=O CC(CC(F)(F)F)C(=O)N1CCC(CCCNC(=O)CN2CC3CC3C2)CC1 C1(CNC(=O)NC(COc2c(C)cccc2C)C)CC(C)(C)OC1(C)C N1(C(CC(C)C2CCCC2)=O)CCC2(C1)CN(C(=O)Cc1ccnn1C)CCO2 C1(CCN(C)C)CCN(C(=O)CCN(C(=O)C2=NOCC2)CCO)CC1 C1(C)(C(=O)NCC=C(C(=O)NC2CC(CCC)OCC2)C)CCCN(C)C1 CC(CC(=O)NCCCCCN(C)C(c1cc(C2CCC2)no1)=O)CC(F)(F)F N1(CC(=O)NC(CC)COC)CCOCCC1C(C)C N1(C(c2cnc(O)cc2O)=O)CCc2cnccc2C1 N1(C(C(C)OCC2CCCCO2)=O)CC2CN(C(c3cccs3)=O)C2C1 C(=O)(C(CC(CC)CC)NCC)Nc1ccccc1N(CC(C)CC1CC1)C CC1CN(C(=O)CCC2CCC(C)O2)CCN(C(c2sccc2F)=O)C1 C=C1C(C(=O)OC)C1C(=O)NC1CC1c1cncs1 N1(C(CNC(C(CC)C)=O)=O)CCC(CC(=O)NCC2=NOC(C)C2)C1(C)C c1(C(=O)NCC2CCN(C(C(c3cc(F)cc(F)c3)C)=O)C2)cc(O)cc(O)n1 c12ccc(nc1)[nH]c2=O.C1(CC=C)(C(N)=O)CN(C(=O)CCC2CC(OC)C2)C1 c1(C(=O)NCC=CCNC(=O)C2=CCCOC2)c(F)ccc2c1OCO2 N(C(=NCC(F)(F)c1ccccc1)NCc1ccccc1)CC1C(C)C1 c1(CN2CC2)cc(F)cc(F)c1O.N1(C(=O)COc2ccccc2)CCCCC1 N1(C(CCOC)=O)CCCC2CN(CCNC(C3CCC(C)CC3)=O)CC12 N1(C(Cc2c(C)nc[nH]2)=O)CCCC2(CC(NC(C3CCCC(CF)C3)=O)C2)C1 C1(NC(c2cn(CC(F)F)cn2)=O)CN(c2nc(Cl)ncc2Cl)CC2(CC2)C1 CN1CCN(C(=O)C(N2CCCC2COC(C)(C)C)=O)CC1.C1(=O)C=CCN1.COC C1(C(C)NC(c2cnc(CC)o2)=O)CN(C(c2nonc2N)=O)CCO1 CCC(CNC(=O)CCCCN(C)C)(CC)C(=O)NCC1CC1Cl c1(C(N2CC(CCNC(CCSC)=O)C(C)C2)=O)ccc2[nH]ccc2n1 N1(C(C2OCCN(CC)C2)=O)CCOCC(NC(=O)COCc2ccncc2)C1 c1(C(=O)NCCCC(C)NC(C(CC2CC2)OC)=O)ccc2c(c1)C(=O)CCC2 N(C1CCc2c1ccc(Cl)c2Br)CC(=O)NC(c1ccc(F)cc1)=O C1(C(=O)NC2CCC(F)C2)CCN(C(=O)CCOCC(F)F)CC1 n1(CC)nc(C(=O)N(CCC(C)NC(c2ncnn2CC)=O)C)c(C)n1 C1(CC(=O)OCC(CC#C)(C)C)OCc2ncccc2NC1=O N1(C(C2N(S(C)(=O)=O)CCC2)=O)CCN(C(c2cncc(N)n2)=O)C2COCC12 N1(C(=O)Cc2ccc(Cl)cc2)CC2(CCN(C(=O)CCNC(=O)C3CC3)CC2)C1 N#Cc1ccnc(C(=O)NCCC2(O)CCN(C(c3ncc(F)cn3)=O)C2)c1F C1(NC(C(C(C)C)S)=O)CC2CCC(C1)N2C(=O)CS(C)(=O)=O c1(NS(c2cn(CC)nc2C)(=O)=O)ccc2c(c1)OCCS(=O)(=O)C2 N1(C(CCC(=C)C)=O)CC2CCC1C(CNC(=O)CNS(C)(=O)=O)C2 c1(C(=O)NCC2(F)CC(CNC(C3(C4CC4)CCCO3)=O)C2)ccc2n[nH]cc2c1 Cc1ccc(C)n1CC(=O)NC1(c2nn[nH]n2)CCSCC1 C(CC(=O)NC(c1nncn1C)CO)(C(F)(F)F)NC(C1C(CC)N(C)CC1)=O C1(CNC(Cn2nnc(=N)[nH]2)=O)CCCCC1NC(=O)Cc1ccsc1 c1(-c2ccc(C3(C(=O)NCCC#C)CC3)cc2)ccc2sc(C)nc2c1 C12(NC(C(C)SC(F)(F)F)=O)CCC(CNC(c3cnc(C4CC4)s3)=O)(C1)OC2 C1(C)(C(N(CCCOCCN(C(CCCSC)=O)C)C)=O)CCCC1C N12CCN(CC1)c1ccc(cc1)NC2=O.N1(S(CC#N)(=O)=O)CCC(F)(CO)C1 c1(NC(CS(C)(=O)=O)CO)ncc(S(=O)(=O)N2CC(CO)C3(CC3)C2)cc1Cl CC1=C(C(=O)N2CCC(C)(CNC(=O)Cc3nncs3)C2)Cc2ccccc2O1 C1(C(=O)NCC2(F)CCCN(C(=O)CNc3ccccn3)C2)CC2CCC(C1)O2 C1(NC(c2ccc(C(C)C)cc2)=O)CCCC2CN(C(C3CCC(=O)O3)=O)CC12 N1(C(CC(CC)CC)=O)CCCC2(CCCCC2NC(c2cnc(OC)s2)=O)C1 c1(N(CC=C)C)ccncc1S(=O)(=O)NCC(N1CCOCC1)C c1(C(=O)NC(C2CCCCC2)C(=O)N(C(CC)C2CC2)C)cccc(O)n1 c1(C(N(CC(CNC(CC=CC)=O)C)C)=O)n[nH]cc1F c1(C(=O)NCC2CCCN(CC3CCC(C)O3)C2)c(Cl)ccc2c[nH]nc12 C1(CNC(C(c2ccc(F)cc2)OC)=O)CC(F)CN1C(c1cccnc1S)=O n1(CCC(=O)NCCc2ccc(CNC(CC)=O)cc2)ncc2ccccc12 N1(C(c2cnc(CCCC)s2)=O)CCN(CC(C)NC(=O)CCC(C)OC)CC1 C1(C2CCN(C(=O)CC(F)(F)F)C2)(NC(C(c2ccccc2)N(C)C2CC2)=O)CC1 c1(NC(c2cc(C3CCC3)n[nH]2)=O)cc(C(F)(F)F)ccc1O c1(NCCn2c(C(C3CCN(C(=O)OC)C3)OC)nnn2)ncc(C)cc1F CC1C(NC(=O)CSC(F)F)CCN1C(c1ccoc1)=O CC1CC(C(=O)N2CCOC(C(=O)N(C3COCC3O)C3CC3)CC2)=NO1 Cc1cnnc(O)c1C(=O)NC1CC(C)N(C(c2ccc(Br)cc2O)=O)C1 c1(CC(=O)NC2CN(C(CCOC)=O)CC2(C)C)c(O)nc2[nH]nc(O)c2c1C N1(C(c2c(C)cncc2)=O)CCN(C(=O)C(C)C2CCCC2)C(CC(F)F)C1 C1(C2CC2)(C(=O)NC2CN(C(COC(CC)C)=O)CC(C)C2)CCOCC1 C(CNC1(C2CCSCC2)CC1)(CCS(C)(=O)=O)OC N1(C(CNC(N)=O)=O)CC2(CCN(C(C3(c4cccc(O)c4)CC3)=O)C2)C1 CC1(C)OCCC1CCNC(=O)C(c1ccco1)NC(=O)CCn1cncn1 C1(NC(C2CCC(C(=O)OC)C2)=O)CCC(C)N(C(=O)Cn2cccnc2=O)C1 c1(NC2CCN(C(c3ccccc3C3CC3)=O)C2)ncc(C(F)(F)F)cn1 C(=O)(C(O)CCNC(C1CCNC1=O)=O)N.c1(C(N)=O)cc(CN)on1 C(CCCC(=O)NCCC(C)(C)NC(c1[nH]nnc1C1CC1)=O)N(C(C)=O)C CC1CCCCC1(NCC1CN(C(=O)OC(C)(C)C)C(C)(C)C1)CO.C C12(CNC(C3(C(C)=O)CC3)=O)CCCC1CN(C(C1CCOCC1(C)C)=O)C2 C1(C(=O)NC(C)CN(C(=O)C(N2CCOCC2)C)C)(CC)CC1(F)F Cc1cc(CCC(=O)NCC(=O)N(C2CCOC2)Cc2cn(CC(=O)O)nn2)on1 c1(NCC2CC(NC(c3c(OC)nccn3)=O)C2)ccc(I)cc1Br c12cccc(c1)C(=O)N(C)C(C)CN(C)C2=O.c1(C(=O)NCC)c[nH]ccc1=O C1(C(=O)NCc2c(C)occ2)CN(C(=O)CC2(CN(C)C)CC2)CC(C)(C)C1 C1(CC)CN(C(=O)CCN2CCCC2)CCN1C(c1cccc(C#N)c1)=O C12(C(N3C4(C)CC4CC3)=O)CC(CO)(CN1C(=O)CCC(F)(F)F)C2 C1(CC(=O)NCC2CN(C(=O)Cn3nnnc3C3CC3)C2)CCCOCC1 c1(N(c2ccc(-c3cnc(C4CC4)nc3)cc2)CCCC)cncc(C#N)n1 c1(CNC(c2n(C(C(=O)OC)C)nnn2)C2(COC)CC2)cnn(C)c1C CCCCC(O)CC(=O)NCCC(C)NC(=O)Cn1cc([N+](=O)[O-])nc1C S(=O)(=O)(CCC(=O)N1CCC(NC(=O)CSCC2CCCO2)C(F)C1)NC CC1CC(NC(c2ccc(-c3ccccc3)s2)=O)CN(C(c2ccn(C)n2)=O)C1 N1(C(C(CC)NC(C)=O)=O)CCn2nc(C(N3CCCC(C)(C)CC3)=O)cc2C1 C1(C(=O)NCCC(CC)C)(CO)CCN(C(=O)Cn2cncn2)C1 c1(C(N(C2CCCN(C(C3CCCC3CF)=O)C2)C)=O)cc(F)cc(Cl)c1O c1(NC2(COC)CC2)cc(Br)ccc1S(=O)(=O)NCC1CCCC(CC2CC2)O1 N1(c2snc(CCC)n2)CCC(NC(=O)C(C)(C)COC)C(O)C1 C1(CCC(=O)NCc2nc(C)sc2)CCCN(C(=O)CCc2nc(O)n[nH]2)C1 c1(N2CCC(SC)C2)ncnc2c1ncn2C1COCC1(C)C N1(C(CC2(OC)CCCCC2)=O)CCC(NC(C2CSC2)=O)C(C)C1 C(C(CC)(CC)C(=O)NCc1cccc(F)c1F)NC(C(C1CC1)OCC)=O C(CC1=CCN(C(c2cc(F)c(F)cc2F)=O)CC1)NC(c1c(C)nn(C)c1)=O c1(CC(=O)NC2CN(CC3CCCN3)CC2F)ccc(C(F)(F)F)cc1C(F)(F)F N1(C(c2ccnc(Cl)c2)=O)CCCC2(C1)CN(Cc1cccc(O)n1)CCO2 C12(C(=O)OC)CC1CN(C(C1CCCN(C(=O)CC3COC(C)(C)C3)C1)=O)C2 C1(C(=O)OCC)CCCN1C(=O)C(C1CC1)N(C(=O)CC1(C)CCC1)C C1(N(C)C(c2cc(C#N)c[nH]2)=O)CCC2CN(C(C3CCCC(C#N)C3)=O)CC12 c1(OC)nccnc1C(=O)NC1CC(n2cc(CSC3COC(C)(C)C3)nn2)C1 C1(C(N2CCC(NC(c3ccn(C(F)F)n3)=O)CC2)=O)CC12CCS(=O)(=O)CC2 N1(C(CSCC)=O)CCN2CCN(C(=O)CCC3CCCN(C)C3)CC2C1 C12(C(=O)NCCC3CCC(NC(c4c(C)noc4)=O)C3)CCC(CF)(CC1)CC2 C1(C(N2CCC(NC(CCSCCC)=O)C(C)C2)=O)CC2(C1)CC1(CC1)C2 C(=O)(C(C)(C)C(C)O)N1CC2C(C(N(CC(C)(C)CO)C)=O)C2C1 CCC(C)(CNC(=O)C(C)CC(C)C)C(=O)N1CCC(c2ccco2)C1 c1(C(=O)NCC2(CNC(C(C)(C)C3CCCO3)=O)CCC2)cccc(O)c1 CCC(CC)CC(F)C(=O)N(CCC(C)NC(C1CS(=O)(=O)C1)=O)C C(=O)(NNc1ccc(OC(F)F)cc1[N+](=O)[O-])c1c(C)[nH]c(=N)nc1O C1(CC(=O)NC2(C(=O)NC(c3ccccn3)CC)CC(F)C2)COCC(C)O1 CN1N=C(C(=O)NC23CCN(C(c4c[nH]cc4C4CC4)=O)CC2C3)CCC1=O c1(C(C)NCC(C)(O)Cn2cc(Br)cn2)ccc(O)nc1 c1(C(N2C(CNC(C3(CC#C)CCCO3)=O)CC2)=O)ncc(F)cc1F c1(NC(CCC(CC)C)=O)ccc(C(N2CCCC2)=O)c([N+](=O)[O-])c1 c1(C(N2CC(CC(C)NC(C3CC(C4CC4)=NO3)=O)C2)=O)c(F)ccc(O)c1F c1(C2C(C(N3CCC(NC(C(C)Cc4cnc[nH]4)=O)C3)=O)C2)ccccc1Cl N1(c2nnc(-c3n(C)cc(Cl)c3)n2CCC#N)CCN2CC3(CC3)CC2C1 c1(CCC(=O)NCCN(C)C(c2cccc[n+]2[O-])=O)ccc2c(c1)NC(=O)CO2 c1(NC(CN(C(=O)CNC(=O)CCn2cc(C)cn2)CCC)=O)cccc(C)n1 n1(CC)ccc(=NC(=O)c2ccnc3[nH]ncc23)[nH]1 C(C)(C(=O)NCCOCCCCN(C)C(C1(C(F)(F)F)CCC1)=O)OCCOC C1(NC(C2(NC(=O)CCc3cn[nH]c3)C(C)CC2)=O)CC2CCC1C2 C1(NC(C(C)(C2CCC2)NC(Cc2n(C)ncn2)=O)=O)C2CCC(C2)C1CO N1(C(Cc2cc(C)on2)=O)CC2CC1CC2N1CCC(C)C1CO C1(C(=O)NC2CCCC(NC(COCC=C)=O)C2)CCCC1P(C)(C)=O O=C(C1=CCCC1)NCC1COCCN1C(c1ccc(-c2ccccc2F)[nH]1)=O C=CC1CN(C(=O)CCc2cnc(C)s2)CC1NC(=O)C(CC)c1ccccc1 C1(C2CN(C(C3CCCC3C)=O)C2)(NC(c2cc(C)sc2)=O)CC1 N1(C(c2cncc(C)n2)=O)CC(C2CCCN(C(c3ccc(Br)nc3F)=O)C2)C1 c1(C(=O)NC(c2cncc(O)c2)C)ccc(-c2cn(CC(=O)O)nn2)cc1 c1(OC)nccc(CNC(C2(C)CN(C(C3CC4(CC4)CO3)=O)C2)=O)n1 c12cc(cc(C)c1)S2.c1(C(COCC(=O)N(CC)CC)C)cn(CC(=O)O)nn1 C=CCC(C(=O)N1CCCC1C(=O)NCCc1cncc(C)n1)OC N1(C(=O)NCCCCCc2cn(C3CCC3O)nn2)CCc2ccnc(O)c2C1 N1(C(CC2(OC)CCCCC2)=O)CC(CNC(C2(C)CCCS2)=O)C2(CCC2)C1 c1(CC)cccc(CC)c1C(N1CCCC1C(=O)OC)=O.C(=O)(N(CC)CC)NCC.OC Cc1ccc(Cl)cc1C(=O)OCC1CCN(C(C2CC3(CCC3)C2)=O)C(=O)C1 C1(CC(N2C3CCC(NC(c4nc(OC)oc4)=O)(C3)C2)=O)SC2=NCCN2C1=O N1(C(c2c(OC)ccs2)=O)CCOC(CNCc2ccnc(SC)c2)C1 C12(CNC(c3cn(C(C)C)nc3)=O)CCC(C1)N(C(C1CCCCNC1=O)=O)C2 c1(OC)ccc(Cl)cc1C(C)OC(=O)C(C1CCN(Cc2cccs2)C1)C C1(C(NNC(c2c(C)cc(NC(C)=O)s2)=O)=O)COC2(CCC2)CO1 c1(C(=O)OC)ccc(C(=O)N(C(C)CCNC(c2cccc(C)c2)=O)C)c(C)c1 C1(COC)(CNC(=O)C=C(C)c2ccco2)CCCN1C(=O)CC1(C)CCC1 CC1CCC(CC(N2CCC=CC2C(N2CCC(OCCOC)C2)=O)=O)OC1 N1(C(c2cc(C)c(O)nc2)=O)CCC(C(=O)N(C(C)CO)C)C(C)(C)C1 C1(C(=O)NC2CCN3CCC2C3)(NC(c2c(CC)cno2)=O)CCC(C)(C)C1 c1(CC(=O)NCCC(C)(C)NC(C=CC(C)C)=O)ccc2c(c1)CCCC2 c1(-c2scc(C)n2)cccc(C(=O)NC2CC(NC(c3[nH]cnc3C#N)=O)C2)c1 C1(CNC(CN(C(=O)CCOCC(F)F)C2CCC2)=O)CC2CCC(C1)C2 c1(C(N(CC)CC2CCCN2C(c2n[nH]c(=N)s2)=O)=O)cc2n(n1)CCO2 c1(C(N2CC(C)C(NC(c3nn(C)c(Cl)c3Cl)=O)C2)=O)coc2c1C(=O)NCC2 N1(C(C(C)=CC)=O)CCC2C(CCCN2C(c2nc3ccccn3n2)=O)C1 C1(C(N2CC(N(C)C(c3ccc(CC4CC4)s3)=O)C(F)C2)=O)CC2(C1)CC2(F)F C(CC(CNC(C1CCCN1C(c1ccccc1)=O)=O)NC(=O)CCF)OC C1(C)(CNC(C2(CC=C)CCC2)=O)CN(C(=O)C(COC)N(C)C)C(C)(C)C1 c1(OC)noc(C2CC2)c1C(=O)NCC1CC(NC(=O)C(C)=C2CC2)C1 C12(c3n(-c4c(C)noc4C)nc(CCC(C)C)n3)CCCCC1C2(F)F n12cc(nn1)CNC(=O)C2.CC(C)C(=O)N(C(c1ccon1)=O)CC1CC1 N1(C(C(CC)C#N)=O)CC2CC(NC(=O)Cc3c(OC)cccc3F)C2C1 C1(C(C)CNC(c2cccn2C)=O)CCN(C(c2coc(Cl)c2)=O)CC1 C1(NC(CC2C(C)CCC2)=O)CC2(CCN(C(c3cnn(C)c3N)=O)C2)C1 C1(NC(C(CCC)(C)CC)=O)CC2(CCN(C(=O)CCCCC#N)CC2)C1 Cc1c(C(=O)NC2(CCO)CN(C(C3CCCOC3CC(C)C)=O)C2)ccn1C C1(NC(C2CC3CCC2O3)=O)CN(C(c2ncccc2F)=O)CCC1F c1(C(=O)Nc2ccccc2-c2ccccc2)cc2[nH]ccc2nn1 CC1CCC(=CC(=O)NC2CCN(C(C3CC(n4cccn4)C3)=O)CC2)CC1 N1(C(=O)NC2C(NC(=O)OC(C)(C)C)CCC2)CCCC(CCC2CC2F)C1 O=C(CCC1CC(OC2CC2)C1)N=c1c(Cl)c[nH]cc1I N1(C(C2(C#C)CCC2)=O)CCC2CCCN(C(=O)CC3CC(=O)NC3=O)C2C1 CC1(C)CN(C(c2csnc2Cl)=O)CCC1NC(=O)C(F)(F)CC1CCCO1 c1(C(=O)OC)cccc(C(=O)NC2CCCC2NC(c2cnc(C3CC3)o2)=O)c1 CC1CCN(c2ncccc2S(=O)(=O)NCc2nc(=N)[nH][nH]2)CC(C)O1 N1(Cc2c(C(N(C)CC)=O)cccc2)C(=O)CCN(CCC2CCCOC2)C1=O c1(C(N2CCN(C(C3N(CC)CCC3)=O)CC2CO)=O)coc2c(F)cccc12 N1(C(C(CC)C)=O)CC2CC1CN2C(=O)COCc1cccnc1 c1(C(=O)NCC2CCCC(NC(=O)CC3CCCS3(=O)=O)C2)ccc2c(c1)CC2 C(C(F)(C(=O)N1CC(CC(F)(F)F)C1)C(C)C)NC(C1(C)CC(=C)C1)=O C12(NC(=O)Cc3cccnc3)CCCC1CN(C(c1c(F)ccc(F)c1Cl)=O)C2 Cc1nc(C(=O)NC2CC2NC(C2(O)CCCC2)=O)nn1-c1nc[nH]n1 Nc1ccc(C(N2CCC(C(CO)NC(c3c[nH]nc3F)=O)CC2)=O)nc1N C1(S(C)(=O)=O)(C(=O)NCCCN(C(c2cc(O)n(CC)n2)=O)CC)CC1 N1(C(C(COCC)C)=O)CCCCC(CCC(=O)NC2CCC2N(C)C)C1 c1(C(N2CCC(c3ccccc3)C(O)C2)=O)ccc2ncnn2c1 c1(C(=O)Nc2cccc(-c3ccsc3)n2)cccnc1NC(c1cnccn1)=O N1(Cc2c(C)scn2)CCC2(CCCC2C(N2CCC(N3CCCC3)CC2)=O)C1 C(=O)(C1=NOC2(CCOC2)C1)N1CC(CN(C(=O)Cc2cnn(C)n2)C)C1 C(C(=O)NCC1CC(C)(O)C1)(C(C)(C)C)NC(C(c1ccccc1)OC)=O C1(CC(=O)N(CCC)CCO)CN(C(=O)CC2(C#N)CC2)CCO1 C(=O)(CCCS(C)(=O)=O)NCC12CC(NC(c3c(C)ncs3)=O)(C1)C2 Cc1nc(-c2ccccc2F)sc1C(N1CC2CC2(NC(c2cnco2)=O)C1)=O N1(C(c2cccc(OC)n2)=O)CC(NC(c2ccc(Br)c(F)c2)=O)CC(C)C1 C1(NC(=O)NC2CCN(S(C(CC)CC)(=O)=O)CC2)CCn2ccnc2C1 CN1CCN(C(=O)Nc2cc3cc(-c4cnsc4)ccc3o2)CC12CCOC2 Cc1ccc(OC(F)F)c(NC(N2CCC(Br)CC2)=O)c1 C1(NC(CC2CC(OC)C2(C)C)=O)CCC2(CC1)CN(C(c1ccc(Cl)s1)=O)C2 C(=O)(C(CC(C)CC)NC(=O)CCCC1CC1)NC1(C(=O)NCCC)CC1 C1(CCC(=O)N(C2CCN(CCOCC(F)F)CC2)CCO)CCCCCC1 CC(C)C(C(=O)NCC(c1ncc[nH]1)N(C)C)C(C)NC(=O)CCCC1CCCC1 C1(CNC(c2cnsc2)=O)COCCN(C(c2cc(F)ccc2C(F)(F)F)=O)C1 c1(-c2nccc(C(N(c3c(C)ccnc3)C)=O)c2)ncn2c1CNCC2 Cn1cnc2cncc(C(N3CCC(CNC(c4cccc(N)c4O)=O)C3)=O)c12 C12CC(C1(C)C)CC(=O)N2.n1(CC)nc(C(=O)NC2(C(C)(F)F)CC2)c(C)n1 Cc1ccc2scc(CC(=O)NC34CC(NC(=O)C(F)=CC(C)C)(C3)C4)c2c1 c1(C(=O)NCCC(C)NC(=O)CC2CC(CF)C2)cc(Cl)c[nH]1 c1(C(=O)NC(C2CCN(C(C(CC)SC)=O)CC2)(C)C)n[nH]c2cccnc12 c1(N(C)Cc2cnc(OC)c(Cl)c2)cc(OC)c(OC)cc1C Cc1cc(C(N2CCN(CCCCCNC(=O)C3=CCC3)CC2)=O)c(C)o1 N1(C(C(C2CN(C(CC3(OC)CCC3)=O)C2)OC)=O)CCCC(C)(F)C1 N1(C(c2ccc(CC)cc2C)=O)CCN(C(=O)CS(=O)(=O)N(C)C)CC(O)C1 N1(C(C=Cc2c(C)coc2C)=O)C2CCC1CN(C(C1CCCC(C)C1)=O)C2 c1(C(=O)NCCC(C)(C)NC(C=C(C)Cl)=O)cnc2c(Cl)cccn12 CC1CC(CN2CCN(c3ccc(C(N)=O)cn3)CC2)CCO1 C(C(C)(C(=O)NCCN1CCCC(O)C1)NC(=O)C(F)OC(F)(F)F)SC C1(C(=O)NC(CC)CNC(c2cnn(C(C)C)n2)=O)Cc2ccccc2N1C c1(CNC(=O)NC2CCCCO2)cc(CN2CCOCC2)ccc1F Cc1c[nH]c(C(=O)NC2CC(CNC(C3CCCN3CC(C)C)=O)C2)cc1=O c1(C(N2CCCC(c3onc(C)n3)C2)=O)ccc(NC(=O)OC(C)(C)C)c(Br)c1 Cc1ccc(F)cc1C(=O)N(C)CC1(O)CN(C(c2ccnc(CO)c2)=O)C1 CN1CC(O)CCC1NC(C1COCC1NC(=O)CCN1CCC(O)C1)=O Cc1nc(N2CCCC2CCCNC(=O)C(C)C2CCC2)cc(C#N)n1 N#Cc1cnccc1N1CCN(CCCNC(c2c(F)cncc2Br)=O)CC1 C1(C(N2CCC(N(C)C)C2)=O)(NC(C2CC(CC)C2)=O)CCC(C)(C)C1 c1(OCC)cc(C(N2CC(OC)C(NC(=O)C(F)CC3CC3)C2)=O)oc(=O)c1 CC(CC#N)C(=O)NC1CC(CC(=O)N(C)CC2(C)CC2)C1 c1(CC(=O)N(CC(C)O)CCNC(C(F)=CC)=O)cnn2c1OCCC2 C1(C(N2C(C(=O)NC3CC(CC)C3)CC2C)=O)CC(=O)CCO1 N1(C(C(C)=C(CC)C)=O)CC2CC2(CNC(=O)CCNC(=O)OC2CCC2)C1 N1(C(C)C(=O)N(c2cccs2)C2CC2)CCCC(C)(C(N2CCNC(=O)C2)=O)C1 c1(C(N2CC(CNC(c3cnn(CC)c3C)=O)C(C)C2)=O)cc[nH]c(=NC)c1N C#Cc1cc(C(=O)NCCC2CCN(C(C3CCC34CCC4)=O)C2)cc(F)c1 C1(C(N2CCC(N(C(C)=O)C)CC2)=O)CCCC1C1CC1 c1(C(N)=O)cocc1C(N1CCC(CCNC(=O)COCC2CC2)C1)=O C123CCC(CC1)(CO2)NC3.Cc1cncnc1C(=O)N(C(C1C2CC3C(C2)C13)=O)C c1(C(N(C2CCCN(C(c3cscc3Cl)=O)C2)C)=O)ccc(Cl)cn1 c1(C(N(C2CN(C(COCC=C)=O)CC2F)C)=O)nccc2nn[nH]c12 N1(C(c2cccc(OCCC)c2)=O)CCC2CN(C(C34CCC(C3)C4)=O)C2C1 CCC(CC1CCCC1)C(=O)N1CCN(C(c2c[nH]c(=N)s2)=O)CC1 c1(C(=O)NC(C)CCN(C)C(C2(C3CCCO3)CC2)=O)ccc(F)c(C2CC2)c1 c1(CNC(C2N(C(=O)OC(C)(C)C)CC2)=O)cc(-c2ccncc2)[nH]n1 c1(C(=O)NC(c2c(C)cccc2)C)ccc2n[nH]c(C)c2c1 c1(C(N2C(CNC(=O)CC3CCCC3)CC(OC)C2)=O)cncc(S(C)(=O)=O)c1 c1(C(N2CCN(C(C3CC3C(F)F)=O)CC2)=O)nc(Br)sc1Cl CC1(C(=O)NC2CCN(C(=O)C#CC3CCCOC3)C2)CCn2ccnc21 C(C1=NOC2CCCCC12)NC(CCCCCSc1c(C)nn(C(C)C)c1Cl)=O N1(C(C(C)SC)=O)CCC(C)(NC(=O)CC23CC(C2)C3)C1 N1(C(C2(C#C)CCC2)=O)CCN(C(=O)C(C)CC2CC2)C(CF)C1 c1(C(=O)NCC(C)N(C)C(C2(C)CCCCNC2=O)=O)ccc2c(c1)C=CCC2 N1(C(CCC(C)CN(C)C)=O)CC(NC(=O)CCOCC2CC2)C2CCCCC12 c1(OCCC)cccc(NC(=O)OCC2CC2c2ccc(O)cc2)c1 CC#CCC(C(=O)NCc1ccc(F)c(O)c1)NC(c1cnsn1)=O C1(NS(=O)(=O)CC2CC2)CCCC(c2ccccc2)C1 c1(C2(C(=O)NC(C3CCCC3)CNC(C(C)CF)=O)CC2)cccc(F)c1F Cc1ccc2nc(C)cc(C(N3CC(NC(=O)C(N)=O)C(C)(C)C3)=O)c2c1 c1(C(N2CC(C)(NC(c3cn(CCCC)nn3)=O)C2)=O)c(N)cc(Cl)cc1F N1(c2cc(C(=O)OC)on2)CCOC(COC(c2cnn(C)c2C)=O)C1 Cc1nc(C(=O)NCC(C)CN(C)C(c2nc(=O)n(C)[nH]2)=O)nn1C C1(C(=O)NC(CCC)(C)CC)CN(C(=O)CC2(COC)CC2)CC(C)(C)C1 N1(CC2CC(OC(C)(C)C)C2)CCOC2(CC1)CCS(=O)(=O)C2 c1(C(=O)NCC2(C)CCN(C(C3CCC(=O)C3)=O)C2)cc(Cl)c(F)cc1Cl N1(C(C2CC(CNC(c3c(C)nn(C)c3N)=O)C2)=O)CCOCC(C)(O)C1 c1(C(N2CC(NC(C3(C(F)(F)F)CC(=C)C3)=O)C2)=O)cc(O)c2ccsc2c1 c1(OC)ccnc(C(=O)NC(CNC(=O)COC(C)=O)C(C)(C)C)c1 C1(CNC(C2(C#C)CCC2)=O)CC2CCC1N2C(=O)C(C)(C)OCC C(=O)(C(CC1CCOCC1)NC(C1CCCCS1)=O)N(CC(CN(C)C)O)C C1(NC(c2cnc(C)nc2)=O)C2COCC1CN(C(c1cc(C#N)ncn1)=O)C2 N1(C(C)=O)CCCC(C(=O)NCCCN2CCN(C(=O)C(C)(Cl)Cl)CC2)C1 C12(CC(N3CCC(C)(CNC(c4noc(C)c4Br)=O)C3)=O)CCCCC1C2(F)F C1(C)(CC)CN(C(C2CCN2C(c2cn[nH]c2)=O)=O)C1 c1(C(N(C)CC2(O)CN(C(C(C)OCC(C)C)=O)C2)=O)cc(=O)cc[nH]1 C1(C(N(CCNC(C(CC=C)CC)=O)C)=O)CCc2nc(CC)ncc2C1 C1(C(=O)Nc2c(OCC(C)C)cccc2)CCCCC(C)(C)C1 N1(CC(c2ccccc2)(C)F)CCC2CCCC(C2)C1 N1(C(C(CSC)O)=O)CC2C(CC(N3CC(O)(c4cnn[nH]4)C3)=O)C2C1 C(=O)(C1=CC2(CCN(C(=O)CCc3cncnc3)C2)C1)N(CC=C)CC1CC1 c1(C(C)NC(=O)CC2(F)CN(C(C3CNC(=O)C3)=O)C2)ccc(O)cc1 CC1(C)CC(CNC(c2nn(C(C)(C)C)cc2Cl)=O)CN1C(=O)CCF Cc1nn(C(C)C)c(C)c1C(N1CC(NC(C2CCC(=O)NC2)=O)C(O)C1)=O c1(OCC)ccc2c(c1)OCC(CN1CCC(c3[nH]cnc3C)CC1)=C2 C1(CNC(CSCCC(C)C)=O)CC(C(=O)N2CCOC3CC23)=NO1 N1(C(CC2C(NC(c3n[nH]c(O)n3)=O)CC2O)=O)CCC(F)(F)C(O)C1 N1(C(C2CCCC3C2C3(F)F)=O)CCC2CCC(C1)N2C(=O)CCF C12(C(=O)NC(CCOC)CNC(c3csc(C)n3)=O)CCCC1(C(=O)OC)C2 c1(OC)nn(C)cc1C(=O)OCCC(O)c1cccs1 N1(C(C=C(C)C2CC2)=O)CCC(CO)CC1C(=O)NCC1([Si](C)(C)C)CC1 N(C1c2ccccc2CC1NC(c1nc(=O)n(C)[nH]1)=O)C(CC=CC)=O c1(NC(C2CC2C(N2CCC(O)(CO)CC2)=O)=O)cc(F)c(Cl)nc1Cl c1(C(N(C(C)CNC(C2CCN(C)CC2)=O)C)=O)cccc2nccn12 c1(C(=O)OC)c(C)[nH][nH]c1=NC(=O)c1csc(NC(c2ccccc2C#N)=O)n1 C1(n2c(-c3cc(C)n(CC)n3)nc(C(C3CC3)OCC)n2)CCCC(C)(C)CC1 Nc1ccc(C(N2CCC(NC(=O)C(C3CCS(=O)(=O)CC3)O)CC2)=O)cc1F N1(C(CCN(C)CC)=O)CCC(C2CC(NC(c3cccnn3)=O)C2)CC1 N1(C(CCCNC(C)=O)=O)CCC(C)(C(=O)NC2CN(C)NC2=O)C1 C(=O)(CCC(=O)C(C)(C)C)N1CCC(C(=O)NC(C)C)C12CCC2 NS(=O)(=O)c1cc(C(N2CC3CCN(C(C4(F)CC4)=O)CC23)=O)co1 c1(N(CCNC(C2CN(CC)C(=O)C2)=O)CCOC)cc(C)c(C#N)cn1.OC S(=O)(=O)(c1ccc(N(C)CC2(F)CCC2)nc1)NC(c1nccn1C)C C1(C(=O)NCCN2CCN(C(CCc3cc(C)on3)=O)CC2)C(F)(F)C12CCC2 Nc1ccc(F)cc1C(=O)NCCCCC(CO)NC(C1CC(CC2CC2)C1)=O CCC(CC)(CCNC(C1CC(O)CN1C)=O)NC(=O)C(F)C(C)C C(c1ccc(C)nc1)=CC(=O)NC1(CC=C)CN(C(=O)CCCSC)C1 CC(C(=O)NC1CCC1CNC(=O)C(c1csc(C(C)(C)C)n1)(F)F)C(F)F C1(OC(CC(C)F)=O)CC(CCN(C)C)N(C(=O)CCOc2ccc(Cl)cc2)C1 C1(C(C)(F)F)CCCCN1C(c1cnn(C2CNC2)c1C(F)(F)F)=O C1(NC(C(c2ccccc2F)OC)=O)CCN(C(C2(Cl)CC2(F)F)=O)CC1 c1(C(=O)NCC2CC2NC(c2cnnn2C(Cl)CO)=O)cccnc1OCC(F)F N1(C(CCC2N(C)CCC2)=O)CC(O)CC1C(=O)NCCCc1nccn1C N1(C(c2c(CC)ocn2)=O)CCC(C)CC1CNC(=O)C(C)(C)C(=O)NC Cc1ccc(F)c(CC(N2CCC(NC(c3scc(C)c3Br)=O)C2)=O)c1 C1(CNC(C(CC)Cc2cccc(C)c2)=O)N(C(=O)CC2CC2)CCCC1(C)C N1(C(CC=CC)=O)CCN(C(c2ccc(CC3CC3)s2)=O)C(C)CC1C N1(C(=O)Nc2cc(Br)c(F)cc2F)CCC2CCC(O)C1C2 c1(C(N2CC(NC(c3cncc(C)n3)=O)C(O)C2)=O)c(Br)ccc(N)c1F C1(CC=C)(NC(=O)COC)CCN(C(c2nccnc2C(N)=O)=O)C1 c1(OC)ccnc(C(=O)NC2CCCCN(C(=O)C(F)(F)c3nccs3)C2)c1F c1(CC)cc(NC(c2ccc(Br)c(OC(F)F)c2)=O)cc(N)c1 N1(C(c2nc(C)cn2C)C(=O)NCC=C)CCC(Br)=C(C)C1 C(=O)(NNc1ccc([N+](=O)[O-])c(C)c1)n1c(C2CCOC2C)nc(C)n1 c1(CNC(C(c2cn(C)nc2)(C)C)=O)nnc2n1CCN(C(=O)CC=C(Cl)Cl)C2 C1(C(=O)OC)CC2(CCOCC2)CN1C(=O)CCS(=O)(=O)Cc1ccccn1 C1(CNC(CC=C)=O)CN(C(c2cnc(-c3ccccc3)s2)=O)C2CC12 Cc1ccc(C(C)C)cc1C(=O)Nc1ccc(NC(=O)CSC(F)F)c(C)c1 c1(C(N(C(CNC(C(CCC)N(C)C)=O)C)CC)=O)cccc2nc(CO)[nH]c12 C(=O)(C(C(C)C)C(C)C)NC1C(CNC(c2c(C)nc(C3CC3)[nH]2)=O)CC1 C(=O)(C1CSc2ccccc21)NCCCC(C)NC(c1c(O)ccc(C)n1)=O c1(C(N2C(CN(C(CCOC)=O)C)CCC2)=O)cnn2c1OCC(OC)C2 C(C(O)C=O)NC(C=C(CC)CC)=O.C(CO)NC(C)=O C(=O)(C1=CN2CCS(=O)(=O)N=C2C=C1)NC(CN(C(C(CCC)CC)=O)C)C CN1CCC2(CCN(C(C3CCCCN(C(C4(C)CC5CCC4O5)=O)C3)=O)C2)C1 CC(CC(=O)NCCCN(C(=O)CNC=O)CCO)C(C)(C)C C(=O)(C(C)C(C)CC)NC1CN(CCC)CC1C.C123CC(C1)(C2)C(=O)N3 N1(C(C(COC)C)=O)CC2C(CN(C)C(c3sccc3CC#N)=O)C2C1 Nc1cc(Cl)nc(C(=O)NCC2CCCC2NC(c2cnn[nH]2)=O)c1Cl C1(NC(CC=CC)=O)CC2CC1CN(C(c1cc(CO)c(C)o1)=O)C2 C1(C(C)NC(c2c(C)cno2)=O)CN(C(c2nc(C)sc2C)=O)CCO1 c1(CC)ncnc(N2CC(CNC(c3conc3C)=O)CC2C)c1F c1(SC)nc(N2C3CC2CN(C(c2c(O)cccc2F)=O)C3)cc(C(F)(F)F)n1 N1(C(=O)Cc2cnoc2)CC(CO)C2(C1)CN(C(c1cccnc1S)=O)C2 C(=O)(CCC(=O)N1CC(OCCC(N2CC(C#N)C2)=O)C1)NCCC Cc1cc(C(C)N(C)C(C2(CCNC(=O)CC3CC(F)(F)C3)CC2)=O)no1 CC1(C)CC(=O)CCC1C(N1CC=CC(NC(c2ncccc2Cl)=O)C1)=O c1(CN2CCC(NC3CCC(C)N3)CC2)nc(O)c2c(N3CCC3)csc2n1.C(=O)OC Cc1ccc([N+](=O)[O-])cc1C(N1CCC2(CCN(c3cnc(C#N)cn3)C2)C1)=O C(=O)(CCC(C)(C)[N+](=O)[O-])N1CCN(C(CNC(CCSCC)=O)C(F)(F)F)CC1 C12(CNC(C(C(C)C)C(C)C)=O)CCCCC1CN(C(C13CCC(C1)C3)=O)C2 Cn1cnc2c(C(N3CCCCC(CNC(C4(C)CC4(F)F)=O)C3)=O)ccnc12 c1(N2C3CN(C(c4ncc(OC)cn4)=O)C(C3)C2)ncnc2onc(C)c12 C1(NC(C2COCC(C)O2)=O)CC(C)CN(C(c2ccccn2)=O)C1 Cc1cc(F)c(C(N2CCCC(CNC(C3CCOCC3)=O)C2)=O)cc1F CCC(C)(C)CC(=O)NC(C(C(C)C)NC(=O)C1=NOCC1)c1ccccc1 C1(C(=O)NC(C2CCCC2)CNC(CC(C)c2ccco2)=O)CC(=O)N(C)C1 c1(SC)cc(N2CCN(C)CC2CNC(=O)CN2CCC2)nc(SC)n1 C1(C(=O)NCC2C(c3cn(C)nc3)C2)COCCN(C(=O)CCC2CCCC2)C1 c1(C(C(=O)NCC2C(C(=O)OCC)CCC2)(F)F)cc(Cl)ccc1Cl CC(C)(CCCO)C(=O)N1CCOC(CNC(C2CCCC23CCC3)=O)C1 CC1(C)CN(C(=O)C=Cc2cccc(Cl)c2)CC1NC(c1nncn1C1CC1)=O N1(C(CC=CCNC(c2cc(CCC)on2)=O)=O)Cc2cnn(C)c2C1 CCC(O)C(F)(F)C(=O)NCC1CC(NC(=O)C2=NOC(C3(O)COC3)C2)C1 O=C(C1CCc2c[nH]nc21)NCC1(F)CCC(NC(=O)Cc2sc(O)nc2O)C1 c1(-c2cccc(COC)n2)c[nH]c2cc(C(=O)NCCC(F)(F)F)ccc12 C1(C(c2ccccc2)NCCCN2CC(=O)NCC2)C2Cc3cc(Cl)ccc3C12 c1(C(N(CCN(C)C(c2cc(O)cc(O)n2)=O)C)=O)nnn2ccccc12 N1(C(c2nnsc2OC)=O)Cc2[nH]nc(C(=O)Nc3ccnc(CC)c3)c2C1 Cc1scc(C(N2CC(NC(=O)C3=NOCC3)C3CC23)=O)c1N N1(C(C2C(C)CC=CC2)=O)CCC(O)C(NC(=O)Cc2ccns2)C1 c1(CC(=O)N(CC(C)NC(=O)C=CC2CCCO2)C)cncc(Br)c1 c12ccc(cc1)c(=O)n2C.N1(CCCCO)CCOCC1C1CCCOC1.OC#N N1(C(CCCSC)=O)CCN(C(c2coc(Br)c2)=O)CC(C)(C)C1 C1(NC(C2(CC)CC(C)(C)C2)=O)CC12CCN(C(=O)CC1CC3(CC3)C1)CC2 c1(CC(N2CC(CCNC(CC=C)=O)OC(C)C2)=O)cn2cc(F)ccc2n1 C(CCN(C)C(C1C(C)C1C)=O)(C(C)(C)C)NC(c1cc(C)ns1)=O c1(C(CC)NC(C)(CCBr)c2nnnn2CCCC2CC2)cccc(C)c1 c1(N2CCC(NC(C3N(CC)CC3)=O)C(CO)CC2)cc(C)nc2ncnn12 C(CCCC(=O)NCc1nc(C(N2CCC2(C)C(C)C)=O)co1)OC c1(C(=O)NC(CCCNC(C(C)c2ccco2)=O)C)cc[n+]([O-])cc1 CC1=C(C(=O)NCC2(NC(=O)C(O)CC3CCCC3)CCC2)SCCO1 c1(CC2C(C(F)(F)Cl)CC2)ccccc1CNc1ccccc1F Cc1cc(Br)oc1C(N1CCN(CCNC(C2C(C)C2C)=O)CC1)=O N1(C(C2CC(NC(C3N(C)CC(O)C3)=O)C(O)C2)=O)CC2(COC(C)(C)C2)C1 C1(C(=O)OC)CCN(C(=O)C(C(C)C)NC(C2CC(=C3CCC3)C2)=O)O1 CC1(C)CCN(C(=O)CCCC(F)(F)F)CC1CNC(=O)Cc1cccs1 C1(C(=O)Nc2c(C)cc(NC(c3cncs3)=O)cc2)CC2CCC(C1)S2(=O)=O c1(CN2C(C(=O)NCCN(C)CCC3CCS(=O)(=O)C3)CCC2)cnc(Cl)c(F)c1 CCC(CN=c1[nH]cnc2ccc(OCC)cc12)NS(=O)(=O)c1ccc(Cl)nc1 C=CCN=C(NCc1ccc(C)c(F)c1)NCCC(C)(C)C(F)(F)F C(=O)(C(C(=O)NC1CC(F)(F)CC1NC(c1nccnc1N)=O)C(C)C)OCC N1(C(CC(CC)C)=O)CC2CCC(C1)N2C(=O)C(O)C1CCC1 O=S(=O)(c1ccc(C#N)c(NCCC(O)C2CCC2)c1)N1CCC(F)C(O)C1 C1(CNC(C(C2CC2)OC)=O)CN(C(=O)Cc2ccc(Cl)cn2)C2CCCC2O1 Nc1cc(C(N2CCC(O)C(NC(c3cccc(Cl)c3)=O)C2)=O)cc(F)c1 C1(C2CC2)(NC(C2C(c3ccc(C)cc3)C2)=O)CCN(C(=O)C(F)(F)CO)C1 N1(CC(C)(C)NC(C(N2CCC(O)CC2)C)=O)CCN(C(C2CC(O)C2)=O)CC1 C1(NC(CCSCC)=O)CCCCCN(C(c2ccnn2CS)=O)C1.C1(C)CCC1 N1(C(C2CC(OC)C2)=O)CC2CS(=O)(=O)CC2(NC(c2cc(C(N)=O)no2)=O)C1 c1(NC(=O)NC(C)CCCCO)ncnc2c(Br)nn(C)c12 c1(NCC(C)C(F)(F)F)ccc(S(=O)(=O)NCC2(F)CCCCC2)cc1Br CCC(CC(C)C)C(=O)NCC(C)CNC(c1cc(OC)ccc1N)=O N1(Cc2ccc(C(=O)O)s2)CC2(CCC(NC(c3cnccc3C#N)=O)CC2)C1 N1(C(c2ccc(C(C)C)cc2F)=O)CC2(COC(CNC(C3CC3(F)F)=O)C2)C1 CC1(C)COC(C(N2CCC2C(N2CC(C(C)(C)C#N)C2)=O)=O)C1 C(C(=O)NCC(C1CCCC1)NC(c1ccc(C(C)C)o1)=O)(C(C)C)OC C1(C(N2C(C(N(C)CCOCCCO)=O)CC=CC2)=O)OCCCC1(C)C c1(C(=O)NC2C(NC(Cc3c(COC)cccc3)=O)C2)cc(Cl)c(Cl)n1C C1(CNC(C2(C)CC(=O)C2)=O)C2CN(C(C3(O)CCSC3)=O)CC12 c1(C(=O)NC2CCCC(CN(C(C3CN(C(C)=O)C3)=O)C)C2)c(Cl)ccnc1C c1(N(C2CC(CS(=O)(=O)NC(C)=O)C2)C(C)C)ccc(Br)cc1F N1(C(CC=CC=C)=O)CCCCC12CN(C(c1cnsc1)=O)C2 O=C(Cc1ccc(O)cc1F)NNc1cccc(O)c1 C=CCCCCCCC(=O)NCC(C)N(C(=O)C(N1CCSCC1)C)C N#Cc1cc(CN2CCN(C(c3ccncn3)=O)CC2C#N)ccc1Cl C(=O)(C(CNC(c1cn(-c2cc(CC)no2)nn1)C1CC1)(CC)CC)N(CC)CC C1(CCCNC(CC(C)n2cccn2)=O)CCN(C(=O)CNC=O)CC1 C1(CNC(C(C)(C)F)C)COC2(CCCC2)O1 N1(C(c2nc(C(C)C)oc2)=O)CCC2CC12C(=O)NC(CC1CC1)C1CC1 CC1OC(C)C(C(N2CCC(C)C(CNC(=O)C(C)(C)CN(C)C)C2)=O)C1C C12(C(=O)NC(CC=C)CNC(C3(OC)CC3)=O)CC3CCC(CC(C3)C1)C2 c1(OC)ccc(CN2CCSCC2C2CC2)cc1-c1ccc(C(=O)O)s1 N1(CCC(=O)NC2CCN(C(c3cc(C)sn3)=O)CC2F)C(=O)NC(C)(C)C1=O c1(OC)cc[n+]([O-])c(C(=O)NC2CN(C(c3occc3C(C)C)=O)CC2O)c1 c1(NC(Cc2cc(C)no2)C(=O)O)cc(Br)ccc1S(=O)(=O)N(C)C c1(N2CCC(CC#N)C2)cc(CO)nc(N2CCCC(N3C(=O)CCC3=O)C2)n1 C1(C(N(CCC)CCNC(C2(SC)CCC2)=O)=O)CCCN(C(=O)C(C)=O)C1 c1(CNC(C(C(CC)C)C)=O)nc2c(s1)CN(C(c1cc(Br)n[nH]1)=O)CC2 C1(C)(CNC(C(C)OC2COC2)=O)CCN(C(C2CC(=O)N(C)C2)=O)CC1 C(=O)(NNc1ccc(C(F)(F)F)s1)NCC(CC#C)C1C(SC)CCC1 N1(C(CCCCNC(C2C(=C)C2)=O)=O)CCc2nc(O)[nH]c2C1 CN1CCC(N2CC(NC(=O)NC3CCC(SC4CC4)CC3)CC2=O)CC1 c1(C(CN2CCN(OC(C)C(N3CCNCC3)=O)CC2)O)cccc(SC(F)F)c1 CC1CCN(C(=O)CC(=O)NC2CC2)C1CCCNC(=O)Cc1ccco1 N1(CC(=O)NC2CCN(C(C(CCSC)O)=O)CC2F)CCc2ccccc21 C(CNC(c1ccoc1C(C)C)=O)(CC(C)C)NC(C1C(C=C)C1)=O N1(C(C2CCC3(CC3)C2)=O)CC2(C=C(C(=O)N3CC(CO)C3)CO2)C1 C(=O)(C1=CCN(C(=O)C(C)CC2CC2)C1)N1C(C(=O)OC)CC(O)C1 CC1CCC(C(N2CC(N3CCN(C(c4ccccc4N)=O)CC3)C2)=O)CC1 c1(C(=O)OC)ccc(C(=O)NCc2c(F)cccc2Br)c(F)c1 N1(C(Cc2c(C)nc(S)s2)=O)CCCCC2C(NC(C3(N4CCCC4)CC3)=O)C12 C1(CNC(=O)COCC2CCC2)CCC(NC(C23CCC(CO2)C3)=O)CC1 C(C(C)(C)CC(=O)NC(C)(C)CCCNC(C1(CF)CCC1)=O)N(C)C N1(C(C(=O)NCC)=O)CCC2(CC1)CC2NC(c1cnc(C2CC2)[nH]c1=N)=O N1(C(COCCC)=O)CCCC(C2CC2NC(=O)Cn2nc(C)cc2C)C1 N1(C(c2n(CC)nnc2)=O)CC(C(=O)NC23CC=CC(C2)OC3)CC(C)(C)C1 c1(N2CCOCC(NC(C3CCc4cncn4C3)=O)C2)ccc(Cl)cc1[N+](=O)[O-] C(=O)(C1SCCc2sccc21)N1CCC(F)(CNC(=O)C#CC2CCCC2)CC1 C1(C(=O)NCC2CCCN(Cc3ccc(Br)o3)C2)CC(=O)N(c2ccccc2F)C1 C1(CNC(=O)CCc2ccccc2Cl)CCCN(C(C2CC(=O)N(O)C2)=O)CC1 C1(NC(C(Cc2ccoc2)NC(CC2C=NN(C)C2=O)=O)=O)CCC(O)C(O)C1 CCCC(CNC(C1(C#N)CC1)=O)C(=O)N1CC2CC2(C(=O)OC)C1 c1(C(N2CCN(C(C(C)(C)S(C)(=O)=O)=O)C3(C2)CC3)=O)cc2c(Cl)nccc2o1 Cc1ccc(Cl)c(F)c1C(N1CCOC(CCCNC(=O)CC2CCCO2)C1)=O CC1CC(CNC(c2ccc(OC)cc2)=O)CN1C(C1CC(N2CCCC2)C1)=O c1(N2CCC(CN(C(=O)C(C)(C)C3CCCO3)CCC)C2)ncc(CC)c(C)n1 C1(C(=O)NCCN(C2CC2)CC)CCN(C(c2cccc(C)c2N)=O)CC1O N1(C(=O)CC23CCCC2C3)CC2COCC2(C(=O)NCCC2CCCCO2)C1 Cc1ccnc(N2CC3C(C(=O)Nc4nc(C(F)(F)F)cs4)C3C2)n1 C1(N(C(c2cn(C(C)C)nc2C)C(=O)NC)C)COC(C)(C)OC1 c1(CC)ncc(C(=O)NCC2COCC2NC(=O)Cc2cccnc2)s1 N(C1CCc2ccccc21)NC(C1C2CC1N(S(=O)(=O)c1cccnc1)C2)=O N1(C(C(C)(C)NC(=O)OC)=O)CCCC(C2CC2NC(=O)CCS(C)(=O)=O)C1 Nc1cc(C(N2CCC2CNC(c2cnn3ccsc23)=O)=O)ccc1Br C#Cc1cccc(C(=O)NCCNC(c2cnn(C3CC3)c2)=O)c1 CC1CN(C(c2cn(C)nc2C(F)F)=O)CC1CNC(c1ccn(CCF)n1)=O C(=O)(C(O)CC(F)(F)F)NC1CC(CNC(C(c2ccccc2Cl)OC)=O)C1 C1(N(C(CNC(C(C(=O)OCC)OC)=O)=O)C)CCCCC1CO.C(CCN=[N+]=[N-])O C(=O)(CCCCCC#N)N(C1CN(C(c2c[nH]nc2[N+](=O)[O-])=O)CC1(C)C)C c1(NC2CC2)nc(Cl)ncc1F.c1(OC)ccc(C(C)C(=O)NC2(C)CC2)cc1 C(=O)(CC1CCc2cc(Br)ccc21)N1CCN(C(CC(=O)NCC)=O)C(C)C1 CCCC(C)C(=O)NC1CC(CNC(c2ccncc2C(F)F)=O)C1 N1(C(C(C)C)=O)CCC2(CC1)CCN(C(C1Cc3ccccc3N1C)=O)C2 c1(C(CNC(C2CC(CS(N)(=O)=O)C2)=O)F)cc(F)cc(F)c1 S(=O)(=O)(c1cnn(C)c1)NCC(=O)N(C1CN(C(=O)CNC=O)CC1F)C Cc1cc(C#N)cc(C(=O)NC(C)(C)CCNC(=O)CNC(=O)CC(F)(F)F)n1 CC1(CNC(=O)CC2CC=CCC2)CC(F)(F)CN1C(=O)CCCC1CCCC1 N1(C(COC(CC)C)=O)CCN(C(=O)CCC2CCCCCC2)C(CC)C1 C(=O)(C(N)C(C)(C)C)Nc1cn(CC2(C)CCC2)nc1 C#CCC(C(=O)NCC1CCN(C(=O)OC)C1)NC(=O)CCc1nncs1 c1(C(=O)NC(C2CCN(C(c3c(C)nccn3)=O)C2)C)cc2cnccc2[nH]1 c1(C(C)C)cnc(O)c(C(=O)NC2C=CCN(C(=O)C(c3cnn(C)c3)O)C2)c1 C1(CNC(Cc2n(C)ncn2)=O)C2CN(C(=O)C(c3ccc(F)cc3)(C)F)CC12 N1(C(C(COC)N(C)C)=O)CCCC(C2CN(C(=O)Cc3csnc3C)C2)C1 Cc1ncc(N)cc1C(=O)NC1CN(C(=O)CC=Cc2cccc(F)c2)CC1C Cn1nc(C2CC2)cc1CC(=O)NCCC1CCCN(C(=O)CCOC2CC2)C1 Cc1sccc1C(=O)N(CC(O)CN(C)C(C1CC(C)(F)C1)=O)C C1(C(=O)NCC2CCCN(CC)C2)(NC(=O)CCc2cnoc2)CCC(C)(C)C1 c1(C(N(CCC(=O)N(C(C)(C(=O)NC)C2CC2)C)CC)=O)cnncc1O C#Cc1ccc(F)c(C(N2CCN(C(=O)CCn3cc(Cl)cn3)CC(C)C2)=O)c1 C1(C(=O)NC2CCN(C(C3(C=C)CCOCC3)=O)CC2)CC(C(C)=NO)C1(C)C Cc1n[nH]c(C)c1SCC(=O)NC1CC(F)(CNC(=O)CC2CC(=O)NC2=O)C1 CC(C)CC(O)C(C)C(=O)NC1CC(OCC(N2C3C=CC2CC3)=O)C1 C1(NC(C2(CC=C)CCCC2)=O)CC2(CCN(C(c3nccn3C)=O)C2)C1 C1(SCCn2c(C(C3(COC)CC3)NC3CCOCC3)nnn2)CCCN(C)C1 C(=O)(C(CCC(C)C)CC(=O)OC)NCC1(CNC(C(CCC)C)=O)CCCC1 c1(N(C(CS(=O)(=O)N(CC)CC)=O)CCCNC(C)=O)cc2nnc(C)n2cn1 Cc1c[nH]cc(C(=O)N(CCCOCCNC(=O)CC2(O)CC2)C)c1=O c1(C(=O)NCC(CCNC(c2cn(SC(C)(F)F)nn2)=O)O)ccnc(O)c1F c1(C(=O)NC2CN(C(C(C)CC(N)=O)=O)CC(F)C2)ccc2cnoc2c1 C=C(Cl)C(C)(C)C(=O)NC1CC(F)(CNC(=O)CN2CCCCS2(=O)=O)C1 n1(CC#C)ncc2cc(C(N3CC(C)N(C(=O)C(C)=CCCC)CC3C)=O)cnc12 Cc1ccn2ncc(NC(N3CCN(C(=O)CC4CC4)C4CC34)=O)c2c1 N1(C(CCCOC(C)=O)=O)CCC(C2(NC(=O)CN3CCC3C)CCC2)CC1 c1(C(=O)OC)cc(Br)cnc1NC(N1CCC(O)C1C(=O)O)=O c1(CC)ncnc(N2CCN(C(C3CCCC(C)CC3)=O)CC2)c1F c1(C(CS(C)=O)NC(=O)C(F)(F)c2cnccn2)ccc(Cl)cc1 C(=O)(C(C(C)(C)C)C1CCC1)N1CCC(N(C(c2cnn(C)n2)=O)CCO)CC1 C(c1ccc(C#N)cc1)=CC(=O)N(CC(C)NC(C1(N(C)C)CC1)=O)C C#CC1CN(C(=O)C(CC)OCC)CCN1C(=O)C=Cc1cc[nH]c1 CC(C)(C)CCC(=O)NCC(C1CCCC1)NC(=O)CC1CC2CCC1O2 C1(CNC(C(C)SC(C)C)=O)CCCCCN1C(c1csnn1)=O Nc1c(O)ccc(Cl)c1C(=O)NCC(O)CNC(=O)CSc1ccsc1[N+](=O)[O-] N1(C(C(CCOC)C)=O)CCC(F)(CNC(C2CN(C)C2)=O)CC1 C1(CNC(c2cncc(F)c2)=O)CC2(CCN(C(=O)COCCCF)CC2)CO1 C1(NCc2cc(CCCC)no2)CCN(c2ncncc2Br)CC1F C1(NC(C(=O)NCCOC)=O)(CNC(=O)C(CC)NC(C)(C)C)CCC(C)(C)C1 C1(C)(NC(CCC2CC(OC)C2)=O)CCN(C(=O)CC2CC(C)(C)CO2)CC1 C=C=C(C)CC(=O)N1CCOC(CNC(c2cc(C)n(-c3ccccc3)n2)=O)C1 C#Cc1c[nH]nc1C(=O)NC(C)CC1(C)CCN(OC(CNC(=O)COC)=O)C1 c1(CNC2C(n3cc(C=CC)nn3)CCCC2)ccc(C)cc1OC c1(NC(C)=O)ccc(C(=O)NCc2cc(NC(=O)N(C)C)ccc2Br)cc1F CCC(CC(=O)NC1(CF)CN(C(=O)COC2(C)CCC2)C1)C(C)C CC1(C)CCN(C(=O)C2CC2)CC1CNC(=O)CC(F)F Cc1ocnc1C(=O)NC1(CO)CN(C(=O)C(C)(O)C2CCC2)C1 c12cccc(c1)OC(=O)COC2.C#CCOCCOCC#N N1(C(C2=C(C)CCC2)=O)CC2(C1)SCCC2NC(c1ccc2ccnn2c1)=O N1(C(=O)Cc2csc(C3CC3)n2)CCC(NC(=O)COCC2CC2)C(CO)C1 CCCCCCC(CN1CC(=O)N(Cc2cc3ccccc3s2)C1=O)CC C1(CC(=O)N(CCCC(=O)NCCC2CCC2)C2CC2)CC(C2CC2)C1 C1(CNC(CNS(CC)(=O)=O)=O)C(C)CCN1C(=O)CNC(N)=O CC(CN=c1nc2sccc2c(N2CCCC(COC3CCCC3)C2)[nH]1)C(F)F C#CCCCCCCC(=O)NCC1CN(C(c2nnnn2C)(c2ccccc2)C)CC12CC2 N1(C(C(COC)(C)C)=O)CC2(C1)C(NC(=O)C1Cc3ccccc31)CCS2(=O)=O C1(NC(C2CCCC2)=O)CCC(C(=O)NCC(c2nn[nH]n2)C)C1 c1(OC)cc(C(=O)NCC2(C)CN(C(c3coc(Cl)c3)=O)CCO2)cc(F)c1F C1(C(=O)NCC(C2CC2)SC)CCN(C(=O)CC2CCC(C)(C)C2)CC1 C1(CNC(C2CC(CCNC(C(COC)(F)F)=O)C2)=O)CCCN(C)C1=O c1(Cc2nc(CCCC(C)(C)C)on2)cc(Cl)ccc1Br N1(C(c2c(C)scc2)=O)CC(C(=O)NCC2COCCO2)CC1C C1(C(N(CCNC(c2nccnc2C)=O)CC)=O)CCCC2(CC2)C1 N1(C(CC(C)(C)OC)=O)CCC2(C=C(C(=O)N3CCC3c3ccccc3)C2)C1 c1(C(N2CC(O)(CCNC(c3cnn(C)c3Cl)=O)C2)=O)c(N)ccc(F)c1F CC(C)CC(C)C(=O)NCC1CC(C(N2CCN(C)CC2C(C)C)=O)CO1 C1(C(=O)NC2(CC=C)CN(c3cc(O)nc(C)n3)C2)Cc2cccc(C)c2O1 C(=O)(CCCCC(C)(C)C)NCC1CC(NC(c2c(C)c(N)ccc2)=O)C1 C(=O)(CCCCC(=O)NC1CCN(C(c2cn(CCO)nn2)=O)C(C)C1)OC C1(NC(c2nccnc2Cl)=O)CCCC12CN(C(C1CCC3C(C1)C3(F)F)=O)C2 c1(OC)ccc(C(=O)NCCC2CCCN2C(=O)CCCC2(C)N=N2)c(Cl)c1 C1(CNC(CCCOC(C)C)=O)CCN(C(=O)C(N2CCCCCC2)C)C12CC2 c1(C(N(C)CC2CCCN2C(c2cn(C)nc2C(F)F)=O)=O)cc2n(n1)CCC2 O=C1CC(C(=O)NCC2CCCC(NC(=O)C(N3CCCC3)C3CC3)C2)=NN1 Cc1ncc(C(=O)NC2CN(Cc3ccc(F)nc3)CC2(C)C)c(C)n1 N1(C(C(C)=C2CCC2)=O)CCC2C(CCCN2c2ncncc2C#N)C1 C1(C(NOCC(C)OC(F)F)=O)CCN(C(=O)CCN2CCCC2)C1 CC(C)CC(CC(=O)NCCn1ccnc1)NC(C1CC=CCC1C)=O C1(C(=O)NC(C)CN(C(=O)CCN2CCC(F)C2)C)CC2CC(O)C(C1)C2 c1(CC(=O)NCC2CCN2C(=O)CSC2CC2)ccco1 S(=O)(=O)(c1cccc2c1NCCC2)NC(c1cccc2cccc(Cl)c12)=O N1(C(CC2CN(C(C(n3ccc(C)n3)C)=O)C(C)(C)C2)=O)CC2OCCOC2C1 N1(C(c2cc(SC)oc2)=O)CC(C)CN(C(C2CN(C(N)=O)C2)=O)CC1C C(=O)(CCC(C)NC(=O)COC1CC1)NCC(C(=O)OC)C C1(NC(C(C(=O)NC)C)=O)CC=C(C(=O)NCCOCCOC)C1 CC1CN(C(=O)C(C)Cc2cnc[nH]2)CCCN1C(c1ccn2nccc2n1)=O C12(NC(c3[nH]nc4ncccc34)=O)CCCC1N(C(C1(O)CCOCC1)=O)CC2 C(C)(C(C(=O)NCCN1CC=CC1)NC(C1CC2(CC2)CO1)=O)OC C1(NC(C2(C)CC2)=O)CCCC(CNC(C2CC(n3cnnc3)C2)=O)C1 N1(C(CC(CC)OC)=O)CCN(C(C2(N(C)C)CCCC2)=O)C2(CC2)C1 C1(NC(CC)=O)CN(C(=O)C(F)(F)C(C)O)CCC12CCC2 c1(C(N(C(C)CNC(c2nocc2C)=O)CC)=O)cn(CCO)nc1C CC1=C(C(=O)N2CCC(=CCNC(=O)CCc3cnc[nH]3)CC2)SCCO1 C1(C(=O)NCC2CCC(NC(c3cnc(CC(F)(F)F)s3)=O)C2)CCCOCC1 CC1CC2CCN1C2.C(=O)(C(C)NS(C)(=O)=O)N.C1(C(=O)NC)CC1F C1(NC(=O)C=CBr)CC2CN(C(=O)CSc3ccc(Cl)s3)CC2C1 N#Cc1cccc2cc(NC(C3CCCCN3C(c3cnc(Br)s3)=O)=O)cnc12 N1(C(c2cnn(C)n2)=O)CC(C)(C)OCC1CNC(c1c[nH]nc1Br)=O N1(C(CC(CC)O)=O)CCC2(CCCN2C(c2cc3cccn3cn2)=O)C1 C(N=c1[nH]cnc(Cl)c1CO)C1C2CN(C(c3nc(C(C)C)oc3)=O)CC21 c1(-c2ccc(C)cn2)ccc2c(c1C(=O)NC(C(=O)OCC1(CN)CC1)C)OCO2 Cc1ccc(O)cc1C(=O)N(C(C)C(=O)NCC1CCCC2(CC2)C1)C Cc1cc(CNC(c2n[nH]cc2Nc2cnccc2C)=O)c(F)cc1Br C12(CNC(C(C)CN(C)C)=O)CCC(NC(=O)Cc3ccc(O)nc3)(CO1)C2 c1(C(=O)OC)cc(C(N2CCC(O)C2)C(=O)NC2CCCC2)n(C)n1 C(c1ccc(F)c(F)c1)=C(C(N1CCC(NC(c2cnc(SC)s2)=O)C1C)=O)C C1(C(N(CC(=C)C)C)=O)COCCC1NC(=O)CC12CCC(CC1)C2 N1(C(C(C)N(C)CC)=O)CC(CNC(=O)C(COC)OC)C2CCCCC12 C1(CCNC(Cc2ccc(C)s2)=O)CN(C(=O)CC(C)C)CCO1 c1(CC)ccncc1NC(=O)CCCN(C)C(c1csc(CC)n1)=O N1(C(C(CC)CCOC)=O)CCCC2(CCCCC2NC(C2C=CCC2)=O)C1 c1(C(C)=O)ccc2cc(C(=O)NCc3cnc(C)c(C#N)c3)[nH]c2c1 c1(CC(N2CCC(CCNC(C(C)(C)SC)=O)C2)=O)ccc(C)nc1Cl CC(N=C(NC1CSC1)N1CCCC(Oc2ccccc2)C1)c1ccccc1 CCCC(O)(CCC)CC(=O)N1CCC(c2nc(Cl)c(=O)[nH]c2N)CC1 C1(NC(CC(CN(C)C)O)=O)CN(C(c2c[nH]nc2C(F)F)=O)CC2(CCC2)C1 n1(CC)cnc2c(Sc3ccc(Cl)nc3)nc(N3CCC(Cl)=C(Cl)C3)nc12 C1(NC(CC)C(=O)OC)COC2CN(C(=O)C(C(C)C)NS(=O)(=O)CCC)CC12 c1(C)cn(CCN(CC(=O)N(C2CC2)N)C)nn1.c1(CS)ccon1.C1(C)CC1 C(=O)(C1CCC(=O)c2cccn21)NCC1CN(C(C=C(C)C(C)(C)C)=O)C1 C1(C(N2C(CN(C)C(c3ccc(O)cc3F)=O)CCC2)=O)COC2(CO)CC1C2 C1(NC(C=C2CCC(C)CC2)=O)CCC2(CCCN(C(=O)Cn3ccnn3)C2)C1 C1(C(=O)NC(C(=O)NC(c2ccccc2)C#C)CC2CC2)CC(C(C)C)=NO1 CCC(C)C(O)C(C)C(=O)N1CCC(CC(=O)NCCCC2CC2)C1(C)C c1(C(=O)NC2CCC(NC(=O)Cn3ccccc3=O)CC2)nccc2[nH]ccc12 c1(CC(=O)NCCCC(C)NC(C(C2CCCC2)OCC)=O)cn2ccsc2n1 C(CC(C)(C)NC(c1csc(C(C)C)n1)=O)NC(C(C1CC1)OCC)=O C=CCCCCCN1CCC(C(C)(C)O)C1.c12ccc(cc1)NC(=O)C2 N1(C(C)=O)CCCCC(NC(c2cccnc2OC2CCCOC2)=O)C1 c1(CC(=O)NCC2(C)N(C(c3c(C)ncs3)=O)CCC2)csc2ccccc12 C1(C(=O)NC2C(CN(C)C(C3(C)CC3)=O)CCC2)CCCCN1C(=O)CC1CC1 n1(CCC)cc(C(=O)NCC(F)CNC(c2cc(C)oc2C)=O)c2ccccc12 c1(C(=O)NCCC(C)NC(CSCC(C)C)=O)ccccc1C(N)=O N1(C(CC2C(CNC(C(CCC)OC)=O)C2)=O)CCCC(C#N)C1 Cc1cc(C(=O)N(CC(C)NC(C2(C3CCC3)CCC2)=O)C)c(O)c(C)c1 Cc1ccc(C(=O)NCC(C)(C(C)C)NC(=O)CC2CCC2(C)C)c(F)c1F C1(C2CN(C(CCC=CC)=O)C2)CN(C(c2cscc2Cl)=O)CCO1 C(C(C)(C)CC(=O)N(C)CC1C2CN(C(=O)C(C)OCC3CC3)CC12)OC CC1CCCN(C(=O)OC(C)(C)C)C1CC(=O)N(CC(Cl)C(F)(F)F)C1CC1 C1(CNC(C(CC)Cc2ccccc2)=O)CC2CCC1N2C(c1scnc1Cl)=O Cc1cc(C(=O)NC(CNC(=O)CSc2nccn2C)C(C)C)ncc1C(F)F N1(CC(c2cc(C(=O)OCC)no2)=O)CCc2ccccc21 C(=O)(CN=c1ccc(Cl)n[nH]1)N1CC(C)C(CNC(C2(C)CC(F)(F)C2)=O)CC1 c1(C(N(CCOC)CCNC(=O)CC2CCCSC2)=O)nn(C)nc1C C1(NC(CC2C(=O)NC(=N)S2)=O)CC2CCC1N(C(C1(Br)CC1)=O)C2 N1(CC=C)CCN(C(C2CCCN(C(C3(CC)CCCC3)=O)C2)=O)CC1 c1(NC(=O)NC(C(C)F)C(=O)NC(C)(C)C)ccc2c(c1)COCC2 c1(C(N2CCCC(C(C)(C)O)C2)=O)c[nH]c2nc(F)ccc12 c1(C(=O)NCCCC(C)NC(=O)Cc2coc(C(F)F)n2)occ2c1CCCC2 c1(C(=O)NCC2(C)OCCN(C(C(C)C(C)O)=O)C2)cc2cc(F)ccc2cn1 N1(S(C=Cc2ccc(C)o2)(=O)=O)CC2CC(NC(C3CC(O)C3)=O)CC1C2 c1(OC)ccc(C(N2CC(NC(c3cccc(Cl)n3)=O)CC(C)C2)=O)cc1O C(=O)(CC(CC)C(=O)OCCC)NCC(=O)N(CCCC(C)SC(C)C)C.C(C)(C)(C)O N1(C(c2c(C#C)c[nH]n2)=O)C2CCC1CC(NC(=O)C(=O)NC(C)C)C2 Cc1ccccc1-c1nc(C(N2CCC2CNC(C2CC(=O)N(C)C2)=O)=O)cs1 N1(C(COC(CC)C)=O)CCC2(CCCN2C(=O)C2=NN(CC)C(=O)CC2)CC1 N1(C(c2c(-c3ccc(SCC)cc3F)cncn2)=O)CCc2cnn(C)c2C1 N1(C(C2(CNC(c3[nH]cc(C)c3)=O)CCCO2)=O)CCn2nncc2C1 N1(C(C(CC)C)=O)CCSCC1CCNC(=O)Cc1cc(C)no1 CCCC(CCCNC(=O)C(C)c1ccsn1)NC(=O)CNC=O N1(C(C(CC)N(C)C)=O)CCC(N(C(=O)C(c2cnn(C)c2)C)CC)CC1 C1(N(C(C(C2(O)CN(C(CC)=O)C2)F)=O)C)CC(O)C1(C)C C1(C(N2CCCN(CC)CC2)=O)CN(C(=O)C(C)CC(C)(C)C)C2(CCC2)C1 CC1(C)CCCN(C(C2CC3CC3C2)=O)C1CNC(c1c(F)cc(F)cc1Cl)=O C(=O)(CCC(C)(C)C#N)NCC=CCC(=O)NC(CCCCC)C1CC1 CCC(CC(=O)NCC(C)(C)CC(=O)NCCC1CCOC(C)C1)C(F)F C(CCCCC(=O)NCC1CCCC1NC(=O)CNS(N)(=O)=O)N(C)C c1(C(C)C)cccc(CC(N2CCCC(N(C(=O)C(O)CN(C)C)C)C2)=O)c1 C1(CC)CC(CNC(=O)C(c2ccoc2)NC(=O)C=CC2CC2)C1 N1(C(c2cccc(C)c2Cl)=O)CCC2CN(C(C34CCCC3C4)=O)CC2CC1 c1(C2C(c3ccc(OC)cn3)C2)ncc(Cl)cc1Br C12(NC(COCCSC)=O)CCN(C(c3cc(C(F)F)cc(Cl)c3)=O)CC1C2 c1(CSC(COC)C)cccc(C(=O)CCNSc2nnnn2C)c1.OC C1(CNC(c2c(OC)ccnc2)=O)CN(C(=O)C2=CCCCC2)CC1(C)C c1(C(=O)NC23CC(C(N4CC5CCNCC5C4)=O)(C2)C3)ccc2ncncc2c1 c1(CC(=O)NC(CC(C)C)CNC(=O)CC2CCC3CC23)ccc(C#N)nc1 C12CC3(COC1C3)C(=O)N2.C1(=O)CCC(=O)NCCN1.CC1(OC(C)(C)C)CCC1 Cc1nc(Cl)sc1CNc1cnn(-c2ccccc2OC(C)C)c1 C(C#CC(=O)N(CCNC(C1CCOC1)=O)CCOC)(OC)OCC1CC1 c1(N2CC(NC(CCC)=O)CC3(C2)CCC3)nc(C)nc2c1cnn2C c1(CCNC(c2ccc(OCC(F)(F)F)cc2)=O)c[nH]c2cccc([N+](=O)[O-])c12 Cc1cc2ncn(CCC(=O)NCC3CN(C4COC4)C3)c2cc1C C1(C(=O)NC(C2CN(C(C(n3ncc(C)c3)C)=O)C2)C)CC(O)(C#N)C1 C1(C(=O)NCC2CCN(C(C3=NNC(=O)C3)=O)C23CC3)CCC(C2CCCO2)O1 c1(C(=O)NC(C(C(C)C)NC(C=C(CCC)C)=O)C)nc2c(s1)CN(C)CC2 C1(CNC(C(COC)O)=O)COCCN1C(=O)COCc1ccc(OC)nc1 c1(C(c2n(CCCCCC)nnn2)NCC2(CO)CCC2)ccncc1Cl C1(c2n(CC)nnn2)(N2CCCC2c2cccc(C(N)=O)c2)CCCN(C)CC1 c1(C(N(CCCNC(CC2(C(=C)F)CCC2)=O)CC)=O)ccc(Cl)cc1C c1(C(N2CC(NC(Cc3cc(C)no3)=O)C(O)C2)=O)cnc(Cl)c(N)c1 c1(Cc2nc(C(CC)C)nn2-c2ccnc(Cl)c2)ccc(Br)cc1Br C1(CNC(c2c[nH]c(=NC)o2)=O)CCC(C)CN1C(c1cc(C(C)C)oc1C)=O C(=O)(CCC(=O)c1cccc(Cl)c1)NCCC(CNC(c1[nH]cc(CC)c1)=O)O c1(C(CC(=O)N(C2CN(C(C3CC4(CC4)CO3)=O)C2)C)C2CC2)ccccc1F C(=O)(CCCCCC(C)O)N(CCOC)CCNC(=O)C(C)CC(F)(F)F C1(CNC(Cc2cc(C)no2)=O)CN(C(=O)CN(C)C)C2CC12 C1(CNC(CNC(CC)=O)=O)COCCN(C(c2ccc(OC)cn2)=O)C1 c1(C(=O)NCC2N(C(CN(C(=O)OC)C)=O)CCN(C)C2)ccc2ncsc2c1 c1(C(=O)NCC2CC(CNC(CC(C=C)CCC)=O)C2)cnc2sccn2c1=O N1(C(C(C(C)C)SC)=O)CCN2CCN(C(C34CCCCN3CCC4)=O)CC2C1 c12ccc(cn1)NCCNC(=O)C(=O)N2.c1(OC)cscc1C(C)(C)C C1(CNC(c2c[nH]c3c(F)cccc23)=O)CNCCC12CCOCC2 CN1C(=O)NCC1C(=O)NCC1CN(C(C2(N(C)C)CCC2)=O)CC1O CC12CCN(C(c3ncc(F)cc3N)=O)C1CN(C(c1cncs1)=O)C2 c1(OC)cccc(S(=O)(=O)NC2CN(Cc3ccnnc3O)CC2F)c1 c1(C(=O)NCC2C3(CN(C(=O)OC(C)(C)C)C3)CC2)cc(Cl)cc2c1CCC2 C#CC1(NC(=O)CN(CCOC)C(C2CS(=O)(=O)C2)=O)CCOC1 C1(C(N2C(CNC(c3cc(C)n(CCO)n3)=O)C=CC2)=O)CC2(COC(=O)N2)C1 Cc1nc(Cl)ccc1NC(C1CC2CC2N1C(C1CC1(C)C)=O)=O C#CC1(C(=O)NC2CCSC2)CCN(C(=O)C(F)CCCC)CC1 Cc1nc(=N)[nH]c(C)c1C(=O)NCC1CN(C(C2CCC3CC23)=O)CC1(F)CO C12(C(=O)OC)CCCCC1CC(N1CC(OC)C(NC(=O)C3CC3)C1)CC2 C1(CNC(CSCC=C)=O)CCC(C(=O)N(C2CC(C)C2)C)CC1 c1(C(NNC(=O)C2CC(C(=O)NCCCOC(C)C)C2)=O)ccc2c(c1)OCO2 c1(CC(N2CCN(C(C3SCCS3)=O)C(C3CCC3)C2)=O)ccc(Cl)cc1F C12(C(=O)NC3CN(C(CCC=CC(C)C)=O)C(C)CC3)C3CCC(CC13)C2(F)F CCCCCCOCC(=O)NCCC(C)(C)NC(c1coc(CO)c1)=O C(CC(N)=O)(C(=O)N1CC(CCO)C1)NC(C1CC=C(C)CC1)=O N1(c2n(C)nnn2)CCC(N(C(=O)CCc2ccc(O)nn2)CC2CC2)CC1 C1(C)(CC)CC(NC(c2cscn2)=O)CN1C(=O)CNC(c1ccnn1C)=O C1(NC(Cc2nc(C)sc2C)=O)CCCCN(CCC2CCCO2)C1 Cc1ccc2c(c1)CCN(CC(c1ccc(C)s1)O)C2 C=CCC(C)(C)CC(=O)NCC1CC(F)CN1C(C1COCCC1(F)F)=O C1(C(=O)NC2CCCCC2(C)O)(CC)CCCN(C(c2ccc(C(C)=O)o2)=O)C1 C(C(=O)Nn1cncn1)(C(C)C)NC(C(CC)(CO)OC)=O C=CC(C)CC(=O)NC(C1CCN(C(c2cc(C)c(Br)s2)=O)C1)(C)C Cc1cc(N2CCCC(C)C2CNC(=O)CS(C)(=O)=O)nc(C)c1C#N C1(NC(C(c2ccccc2Cl)OC)=O)(CNC(=O)C=C(C)Cl)CCOCC1 S(=O)(=O)(c1ccc(C)c(Cl)c1)N1CC2CCN(C(c3ncc(C)s3)=O)CC2C1 c1(C(C(=O)NCCN(C(=O)Cc2csc(SC)n2)CC)=O)cc(OC)cc(OC)c1 N1(C(c2ccc(C)cc2)=O)CCCN(C(c2ncc(C(N)=O)cc2Cl)=O)C(C)C1 CCCCC(CNC(C1(CO)CC1)=O)NC(c1csc(CS(C)(=O)=O)n1)=O N1(C(C(C)S(N)(=O)=O)=O)CC2OCC(NC(=O)C(=Cc3c[nH]cn3)F)C2C1 c1(OC)cc(C(N2CCC2CNC(c2ccc(C)cc2C)=O)=O)cc2ccoc12 C(=O)(C(C(C)(C)C)N(C)C)N(CCNC(CCc1ccc(OC)cc1)=O)C(C)C CCCCC(=O)C(=O)N1CC=CC(C(=O)NCC(C)SC)C1 N1(C(Cc2ccc(OC)cn2)=O)CC2CC1CC2NC(c1cc(C2CC2)[nH]n1)=O N1(C(CCC=C(C)C)=O)CC2(CCN(C(c3cnc(C4CC4)nc3C)=O)C2)C1 N1(C(CCCOCC)=O)CCC(C)C(NC(=O)CCC2CC2(C)C)C1 C(=O)(CCCc1ncc(C)o1)N(CC(CC)NC(C1C(CCOC)C1)=O)C N1(C(C(n2ncc(C)c2)C)=O)CCCN(C(c2ccnc3[nH]nnc23)=O)C(C)C1 N1(C(CCSCCC)=O)CC2CCC(C1)N2C(=O)CCc1cscn1 Cc1oc(C)c(C(=O)NC2CCCN(C(=O)CCn3ccccc3=O)C2C)c1C C#Cc1ccc(C(=O)N(C(CC)CC(=O)NCC2CC2(C)C)C)nc1 c1(OC)cc(I)c(Cl)cc1NCC(C)SC C1(NC(c2c(OC)nccc2)=O)CN(C(c2nc(C)c(C)s2)=O)CC2(CCC2)C1 n1(CC)cc(Cl)c(C(=O)NC2CCN(C(=O)CS(=O)(=O)NCCOC)C2CC)n1 C#CC(C(C)C)NC(=O)NCCCN(c1ccccc1)C c1(OC)c(NC(CNC(c2cnc(O)cc2C)=O)C(C)C)ncnc1Cl S(=O)(=O)(c1cccc(Br)c1F)NC(C(C(=O)OCC)C(C)C)=O C(=O)(C(C(C)C)C1CCCCC1)NCC(C)NC(C(C)=C1CC1)=O CCC(COC)C(=O)NCCCCCCNC(c1cccc(C2(C#N)CC2)c1)=O C12(COC)CCCC1CN(C(=O)Cc1ncn3c1CCC3)C2 C(C(C)(CO)NC(c1cncn1C)=O)NC(C1CC(C(C)C)C1)=O C1(CNC(c2nnc(CC)s2)=O)COCCN1C1COC1 C(=O)(C(C)(C)CCCO)NC(C1N(C(c2c(F)ccc(OC)c2)=O)CCC1)(C)C c1(CCC(N2CCC(CNC(c3c(CC)onc3C)=O)C2)=O)c(Cl)cccc1Cl C(=O)(C(C(C)CC)OC)N1CCC(C(=O)NCCC(C=C)(C)C)CC1 C(=O)(C(C)(C)S(=O)(=O)C1CC1)N(c1cc(C(F)(F)F)c2c(c1)CCO2)CC CCCCCCCCCCC(=O)NC1CC(NC(=O)C=COCC)C1 C1(C(=O)NC(C=C)(C)C)CCN(C(=O)C(C2CC2)OC)C12CC2 c1(CC(=O)NCC(C)(O)CNC(=O)Cc2ccnc(Br)c2)cccc(O)c1 c1(COC(c2c(OC)cc(Cl)c(C3CC3)c2)=O)ccc([N+](=O)[O-])c(O)c1 c1(C(N2CC3CCN(C(C4CN(C)C4)=O)C3C2)=O)cccc(Cl)c1[N+](=O)[O-] C1(NC(CCc2nnc(C)n2C)=O)CN(C(=O)CSC2CC2)C2(CCOCC2)C1 Cc1ccccc1CC(=O)NC1CC(C(=O)NC2CCC2O)C1 c1(C(C)=O)ccc(OC(C)C(=O)N(C(C)CCNC(=O)Cc2cccs2)C)cc1 O=C1CC(C(=O)NCCn2ncnn2)N(C(C2(C(=O)C3CC3)CCC2)=O)C1 CC1CN(C(C2(O)CCC2)=O)CCC1NC(c1cnn(C)c1Cl)=O c1(NC(CCc2ccc(C(N(C)Cc3cnc(SC)s3)=O)[nH]2)=O)ccccc1I C1(CCC(=O)NCC(CNC(=O)C(CSC)OC)OC)CCCCCC1 CC1C(C(=O)N2CC=CC(NC(=O)CCN3CCCC3=O)C2)=Cc2ccccc21 C1(CNC(=O)CC2CCCC2)C=CCN(C(=O)COC2CCCC2)C1 Cn1cc([N+](=O)[O-])cc1C(=O)NC(C)(C)CNC(c1cc(Cl)cnc1O)=O CS(=O)C=CC(=O)NCC1CCN(C(=O)CCc2cccc(Br)c2)C1 Cc1cc([N+](=O)[O-])ccc1C(=O)NCCC1CC(NC(c2ccnnc2S)=O)C1 c1(C(=O)NC2CC(C)(NC(c3c(O)ncc(CC)c3)=O)C2)cn(C)c(=O)c(C)n1 C1(C(N(CC(CC)NC(C(CC)=CC)=O)CC)=O)CCc2nc(CC)ncc2C1 c1(OC)ncc(C)cc1C(=O)NC1CC(CNC(=O)CC(C)C)C1(C)C C1(C(=O)NCCC(C)(C)CNC(=O)Cn2cnnc2)CNC(=O)CC12CCC2 C1(CNC(c2c(C)cc(C)o2)=O)CN(C(=O)C(c2ccc(F)cc2F)C)CCCO1 c12cn(nn1)CCC(=O)N(CC)CC2.C1(OCC)CCOC1 C#Cc1ccc(F)c(C(=O)NC2CCCC2CNC(C2(C)CCCCC2C)=O)c1 c1(CN(C(c2ccccn2)CC)CC)cc2c(C)cc(Br)cc2[nH]1 c1(CNC2CC(CC(=O)Nc3ncc(Cl)cc3O)C2)cc(Cl)ncc1Cl c1(C(=O)NC2C(NC(c3nc(C)c(C)s3)=O)C2)cc(=O)c2cc(F)ccc2o1 C#CCC(C)(C)NC(C1C(C)CN1C(=O)CC=C)=O CC1C(NC(c2occc2Br)=O)CC2CCC1N2C(c1cc(C#N)on1)=O C1(C#N)(C(=O)NCc2cc(C(N(C3CC(F)(F)C3)C)=O)n[nH]2)CC=CC1 c1(C(c2nnnn2CCNc2csc(C)n2)OC)cnc(C2CCC2)o1.C1C(=O)N1 Cc1nnnn1CC(=O)NCC1CC(CNC(c2c[nH]nc2F)=O)CO1 c1(-c2cn(CCCC(=O)N(CCCCCC)C)nn2)ncn(C)c1C O=C1CCC2(C(=O)NC3CCCC3NC(=O)C(c3ccccc3)O)CCCC2C1 C1(C(=O)NCCC2CC(NC(c3cc(CC)c(CC)o3)=O)C2)CCN(C)C(=O)C1 C(c1ccc(C)nc1)=CC(=O)NC(CNC(C(c1cccc(Cl)c1)SC)=O)C c1(SCC2C(CC)C2(C)C)cc(OC(F)(F)F)ccc1C c1(SC)ncc(N)c(C(N2CCC(C)(NC(C3CC(SC)C3)=O)C2)=O)n1 C(CN=[N+]=[N-])(C(=O)C(C1C(C)=CCS1)=O)N.C1(CN)CCC1 C(N=c1nc2sccc2c(NCCc2ncco2)[nH]1)C1C(C(C)C)C1 c1(C(N(C)CC2CCCN2C(=O)COC2(C)CCC2)=O)ccnc2c1CC(=O)N2 S(=O)(=O)(c1cnn(C)c1)CN1CC(NC(C(c2ccc(CC)s2)=O)=O)C(F)C1 c1(C(=O)NCC2C(NC(c3ccn(C(C)C)n3)=O)C2)ncccc1OC(F)F C(=O)(CCCCC(C)=O)N1CCC(=C)CC1C(=O)NC(C)CCCC C1(CC(=O)OC)(C(=O)NCC2(C)CC(NC(C34CCC3CC4)=O)C2)CCCC1 CC(CN(C(=O)CC1(C)CCN(C(c2nccn2C)=O)C1)C)C(F)(F)F N1(C(CCCCN(C)C)=O)CCC(C)(C(N2CCC(CO)C(O)C2)=O)CC1 C1(CNC(Cc2c(C)nccc2)=O)CCN(C(=O)C2=COCCO2)CC1C c1(C(=O)NCC2(O)CC(NC(C(C)CC3CCCO3)=O)C2)cc2c[nH]cnc-2n1 C(=O)(C1=C(C)OCC1)N1C(C(C)NC(C(c2cccc(F)c2)OC)=O)CCC1 CC(CS(=O)(=O)c1ccc(Br)cc1)C(=O)N(C1CCOCC1)C c1(C(N2CCC(CCC)(NC(CCC=CC)=O)CC2)=O)ccc([N+](=O)[O-])cc1O c1(OCC(=O)N(C2CCC(NC(c3ccc(C)cn3)=O)C2)C)c(C)cccc1C C(C)(CCC(=O)NCc1nocc1C(=O)N(C)CC1CCCN1C)OC N1(C(C2(CC=C)COC2)=O)CCCC(CCNC(C2CCCC(C)(C)C2)=O)CC1 Cc1cc(F)c(C(C)C)cc1C(=O)N(CC(=O)NC(C)(C)C)C N1(C(c2n(C)cnc2)=O)CC(NC(=O)CC2(O)CC2)C(F)C1 C=CCC(CC)C(=O)N(C)CC1CCN(C(=O)Cc2cccc(Cl)c2F)C1 N1(C(c2ccc(=N)[nH]c2Cl)=O)CCC2OCCN(C(C3CCCCO3)=O)C2C1 C1(C2CCOCC2)(NCCCSc2c(F)cccc2)CC1 Cc1nnc(C2CCCN2C(=O)CN2CC2=O)o1.c1(C(=O)N(C)C)ccccc1 C1(C(F)(F)F)(OC)CC(C(=O)N(C)CC2(O)CN(C(=O)C(C)N(C)C)C2)C1 CC(C)(CS(N)(=O)=O)C(=O)NC1CC(NC(=O)Cn2cc(Cl)cn2)C1 C1(CNC(C2CC(O)(CC#C)C2)=O)CCCC2CN(C(C3(CC)CC3)=O)CC12 C(=O)(C1=CCN(C(=O)OC(C)(C)C)C1)Nc1cccnc1.C1C(=O)N1CC C(=O)(C1=CCC(F)(F)CC1)NCC1(CNC(C(C(COC)C)C)=O)CCC1 Cc1cc(N2CCCC(N(CC(F)(F)F)C)C2)nc(C(C)C)n1 CCCCC(C(=O)NCCCN(CC(C)C)C)NC(C1CCOC1=O)=O Cc1ccc2sc(C(=O)NC3CCN(C(C4CC(=O)NC4(C)C)=O)C3)cc2c1 N1(C(C(C2CC2)OC)=O)C2CCC(C2)C1CC(=O)NOCC1CCOC1 C(CCCOC)(C(=O)NC(c1ccc(C)cc1)C)NC(c1cc(CCC)on1)=O C1(CC)CN(C(=O)Cc2csc3nccn23)CCN1C(=O)Cc1ccc(Cl)s1 N1(C(c2sccc2Br)=O)CCC2(CC1)CN(C(c1coc(Cl)n1)=O)C2 C1(C(N2C(CC(=O)NCC3C(C)CCC3)CC2)=O)C2CC3C(C2=O)C13 c1(C(N2CC(NC(C(CC)NC(C)=O)=O)C3(C2)CC3)=O)cccc2c(C)[nH]nc12 c1(-c2cc(C(=O)NCC3CCCN3C(C3CC3(F)F)=O)sn2)ccc(Cl)cc1 C1(NC(COC)=O)CCC(NC(C2CCCC2OC(F)(F)F)=O)CC1 C1(C(N(CCNC(CSCC)=O)C)=O)CCOC1c1ccnn1CC1CCC1 c1(C(C)Cc2ccncc2)nc(-c2cnn(C)c2)nn1C1CCCCC1O C1(CNC(C(COCC)C)=O)CN(C(c2nc(O)c(C)s2)=O)CC1C(F)(F)F C=CCC(C)C(=O)NCC1(NC(=O)Cc2ccon2)CCCC1 CC(C(=O)NC(c1nocc1C(=O)NCCc1cccc(F)c1)C)C(F)F C1(C(N(CC#C)CC2CC2)=O)C2CCC(C2)N1C(=O)C(C(C)CC)N(C)C C1(C(=O)NCC(F)F)CCN(C(c2occ(C(=O)NCCO)c2)=O)C1 CC(C)CC(CN(C)C)NC(c1[nH]nnc1C1CC1)=O N1(C(CC(=O)NCC2CC2)=O)CC(NC(=O)CCN2CCC(O)CC2)C2(CCC2)C1 Cc1cc(C2(NC(=O)CCCNC(=O)C=Cc3ccncn3)CC2)cc(C)c1 c1(NC(COCCNC(C2(CCC)CC2)=O)=O)cncc(SC(C)C)c1 Cc1cc(C(=O)NCc2ccc(O)cc2)cc2c[nH]nc12.N12CC3C(C3C1)C2=O C1(C(N(C)CC2(N(C)C)CC2)=O)C=CCCN1C(=O)CCC1CC1 N1(C(C2(CNC(C(CC)(CC)OC)=O)CCCO2)=O)CC(CC)OC(C)(C)C1 c1(C(=O)NCCCCN(C(c2cc(C)on2)=O)C)c(C)nn(CCCC#N)c1Cl C1(NC(C(CCC)O)=O)CCC12CN(C(=O)CCCCCc1cccs1)C2 CCS(=O)(=O)CC(=O)N1C(C(=O)Nc2ccc(Br)c(Cl)c2)CC2CC12 C1(C(N2CC(O)(CCNC(C(C)(C)OC(C)C)=O)C2)=O)CCC12CCC2 Cc1ccc(CC(=O)NC(C2CN(C(=O)COc3cccnc3)C2)C)cc1 c1(C(=O)NC2CN(C(c3n[nH]cc3F)=O)CC2CC2CC2)cc2ncccc2o1 c1(C(=O)NC2CCC(NC(COCC#C)=O)C2)cc(OC)cnn1 C1(NC(C2C(C)OC(C)C2C)=O)CCCCC12CCN(C(C1CC1(F)F)=O)C2 c1(NC(C(CC)F)=O)c(C)cccc1C.C12CN(CC1O)C(=O)COC2 C1(C)(C(N2CCC(Cc3n(C)ncc3)CC2)=O)CCN(c2ccccc2)S1(=O)=O c1(C(C(=O)NCCOC)N(C(C)C(=O)OC(C)(C)C)C(C#C)C)cnn(C)c1F c1(C(=O)NCC(C)N(C(=O)C(F)CC2CCCC2)C)cccc(C(N)=O)c1F Cc1ncccc1CC(=O)NCC(C)CN(C(=O)CCCc1nnc(C)n1C)C c1(C(=O)NCC(CCCC)NC(c2cc(Cl)cc(Cl)c2)=O)ccc(C)c(C)n1 N1(C(COc2cccc(C)c2)=O)CC2OCC(NC(=O)C(CO)C(C)(C)C)C2C1 N1(C(CCCCOC)=O)CCCC(NC(c2nccc(N)c2Cl)=O)CC1 N1(C(CC(N)C(=O)O)=O)CCOC2(CCSC2)CC1 C1(NC(C(C)SC(C)C)=O)CCC(C)(CNC(=O)Cn2ccccc2=O)CC1 c1(C(N2CC(O)(C(C)NC(C(C3CCOCC3)C)=O)C2)=O)cnn2cnnc2c1 C1(CN(C)C(C2COC(=O)N2C)=O)CCN(C(C2CCN(C3CC3)C2=O)=O)CC1 c1(C(=O)NC2CN(C(CN(C(C)=O)C)=O)CC2C)cc(C)c2c(c1)CCC2 N1(C(C#CC2(CC)CC2)=O)C2CCC1CN(C(C1CCC1C(C)(C)C)=O)C2 c1(C(N2C(C(C)NC(c3c(C)nc(O)[nH]3)=O)CCC2)=O)cccc(Cl)c1O C1(CNC(c2ccc(C)c(O)n2)=O)CCC2CN(C(=O)C(F)C3CC3)CCC2C1 N1(C(C2CCC(C)N(C(=O)CC3CCCC4CC34)C2)=O)CC2(CCC2(C)C)C1 CCC(C)C(O)C(=O)NC(C)(C)C=CC(=O)NCc1cc(C)cs1 C(C(CN(C(=O)CC(C)(C)C#N)C)C(F)(F)F)NC(Cc1cccc(C(C)=O)c1)=O c1(C(N(C)CCn2cc(CO)nn2)=O)cccnc1S.C12(CCCO1)C(=O)NC2 CCS(=O)(=O)c1ccc(OC)c(C(N2CC3CC2C3NC(C2CCOC2)=O)=O)c1 CC1(C)CC(CNC(c2ccc(Cl)cc2N)=O)CN(C(=O)CCc2ncc[nH]2)C1 c1(C(=O)NC2CC(CNC(C3CCN(CC(C)C)C3)=O)C2)ccncc1N CCC(F)(F)CCNC(=O)CC(C)N(C)C(C1(F)CCCCC1)=O CC(c1cccnc1)=CC(=O)NC1CCCC(CNC(C2CCC(C)(C)C2)=O)C1 C=C(C)CC(C(=O)NC(c1nc[nH]n1)CC)NC(=O)CC(C)(C)SC C(C(C(=O)N(C(CC1CC1)CO)C)C(C)C)NC(C1(CC#C)CCC1)=O n1(CC(=O)N(CCCNC(C2CC2CC(C)(C)C)=O)CC)cnnc1 c1(C(N(CC(C)N(C(=O)C(c2cnn(C)c2)O)C)C)=O)cc(O)ncn1 c1(NCc2cc(CC)on2)ncccc1S(=O)(=O)N1CCCC1C1CCCO1 C12(CCC(C)(C)C1)C(=O)N2.c1(C(C)=O)csc(C(=O)NC(c2cnn(C)c2)C)c1 N1(C(C(NOC)=O)=O)CC2(CCC2)CC1CNC(=O)C(C)(C)CC1CC1 C(c1ccc(F)cc1)=C(C)C(=O)NC1C2CN(C(=O)C(C)=C3CCCC3)CC12 N1(C(c2ccn(C)c2)C(=O)NCCOC)CCCC2(CC1)CNC(=O)C2 N1(C(c2cccc(C(=O)OC)n2)=O)CC(C)(C)OCC1CNC(C1CC1C)=O c1(C(=O)NCC2(NC(C(CC#C)C3CC3)=O)CC2)cc2ccc(F)cc2nc1O CC1(C)Oc2cccc(S(=O)(=O)N3CC(CS(C)(=N)=O)C3)c2O1 c1(C(=O)NC2C(C)CN(C(c3cnnn3C)=O)CC2C)ccc(Cl)c2occc12 C1(NC(=O)CC2CCCS(=O)(=O)C2)CCCCN(C(c2cc(Br)c[nH]2)=O)C1 N1(C(C(C2CCOC2)OC)=O)CCC(C)(CCNC(c2cccc(C)n2)=O)C1 C1(C(N(CCC(C)NC(C2(C#N)CCN(C)CC2)=O)C)=O)CCCCCS1(=O)=O N1(C(C2(S(N)(=O)=O)CC2)=O)CCC(O)(CNC(c2ccc(CO)cn2)=O)CC1 C(c1cc2ccccc2o1)=CC(N1C(C)CN(C(C2CC3CC3C2)=O)CC1)=O Cc1cccc(CCC(N2CC3C(CNC(=O)C=Cc4ccco4)C3C2)=O)n1 O=C(CCCCC(F)(F)F)NCC1CCN(C(c2ccc3ccnn3c2)=O)CC1 CC(C)C(F)(CNC(=O)C(C)SCC(C)(C)n1ccnc1)C(=O)NC(C)(C)C N1(C(c2[nH]nnc2C2CC2)=O)CC2(C(N3CCC34CC(O)C4)=O)CC1CO2 c1(C(=O)NCCOCCN(C(=O)Cc2nc[nH]n2)C)ccc(C(F)F)o1 CC#CCC(C(=O)NC(c1csc(C)n1)C)NC(C1C2CCCOC12)=O N1(C(C(n2c(C)ccn2)C)=O)CC(CNC(c2ccc(C(C)(C)C)[nH]2)=O)C(C)C1 c1(C(=O)NCc2ncc(C)o2)ccc(C(=O)NCC2CCCC2F)cc1 N1(C(=O)C(C)SCCN(C)C)CCC(C)(CNC(C2(COCC)CCC2)=O)C1 c1(N(CC#CC)C(C2COCCN2C(c2ccccc2)=O)=O)c(Br)cc(C)cc1Br c1(NC(C#CCNC(c2nc(CC)oc2)=O)=O)ccc(F)cc1 C1(NC(Cc2nnc(C)o2)=O)CC2CC1CN2C(=O)COC1CCOCC1 c1(C(N2CC(NC(C3CCC(CO)CC3)=O)C2)=O)ccc(N2CCCCC2)cc1 c1(CC)ccc(C#N)c(NC2CC3CN(C(c4c(OC)ncnc4C)=O)CC23)n1 C(=O)(C(C(C)(C)C)OC)N.c1(CC)occc1C(=O)NOCC=CCl Cc1nn(C)c(C)c1S(=O)(=O)N1C2CCCC1CN(C(C1CC3CCC1O3)=O)C2 C=CCC(CNC(=O)CCC)NC(C1(OC)CCSC1)=O N1(C(c2c(C)cn(C)n2)=O)CC(C(=O)NCc2nonc2C)C(C)(C)C1 C12(C(C)=O)CCC(C(=O)NCC3CCCN(C(c4nonc4N)=O)C3)(CC1)CC2 CCCC(C(O)C(=O)NC1CCC2CC1C2(C)C)NC(=O)CCCC(C)CC CCC(CC)CCC(=O)NCC1CN(C(C2(N(C)C)CCCC2)=O)CCN1C c1(C(N)=O)ccccc1C(N1CCC(O)(CNC(=O)Cc2ccccc2Cl)C1)=O N1(C(C(c2cccc(OC)c2)O)=O)CC2CC(NC(c3cnoc3C)=O)C1C2 C1(C(=O)NC(CNC(=O)CCc2ncc(F)cn2)CC(C)C)(OC)CCCOC1 C1(C(=O)NCC2N(C(CCCNC(C)=O)=O)C3C(C2)C3)CC2(C1)CC21CCC1 c1(C(N2CCC(C(C)NC(C3(CSC)CCC3)=O)C2)=O)ccc(Cl)cc1Cl O=C(CCc1cn(Cc2cccnc2)nn1)CCO.C12CN(CC1CO)C2=O C1(C(=O)NC2(C(=O)OC)CC2)C(C2CC2)CCN1C(C12CCC(C1)OC2C)=O C1(NC(CC(CN(C)C)O)=O)CCC2CN(C(=O)C=Cc3cnc[nH]3)CC2C1 N1(C(CC(C)OC)=O)CCOC(C(C)NC(=O)CCc2ccc(C)cc2)C1 N1(C(c2c(CC)nc(C)[nH]2)=O)CC(NC(c2cc(Br)sn2)=O)CCC1C CC1C(NC(c2cc(Cl)c(Cl)n2C)=O)CC2CCC1N2C(=O)C(F)(F)C1CC1 S(=O)(=O)(c1ccc(Cl)cc1F)N(C1C(C)CC1)CCc1nc2ccccc2[nH]1 N1(C(c2c(C)ncnc2O)=O)CCCC2(CCCN2C(C2CNC(=O)N2C)=O)C1 c1(CC)cc(C(=O)NC(C2(CNc3nc(C(=O)OC)co3)CCOC2)=O)sc1C N1(C(n2c(C)cc(C(=O)O)n2)=O)CCN(C2CCOCC2)CC1C Cc1ccc(C(=O)NC2CCC2NC(=O)CC(n2nc(C)cc2C)C)nn1 c1(CC(=O)NC2CN(C(c3nc(C)nn3C)=O)CC2C)cnc2c(C)cccn12 c1(NCC(C)NC(=O)OC)nccc(=NCCc2c(Cl)cccc2Cl)[nH]1 C1(C)(C(N2CCC(CC)C2)=O)CN(C(c2cc(CO)on2)=O)C(C)(C)C1 Cn1ccc2cc(CNC3CC(NC(c4nc[nH]n4)=O)C3)ccc12 C#CC1(CN2CCCC(n3cc(C(=O)O)nn3)C2)CCCC1 C1(C(=O)NC(C#CCC)(C)C)CN(C(=O)C(n2nccc2C)C)CC12CCC2 CC(C)C(O)C(C)(C)C(=O)N1CC2(CC(CC(=O)N)C2)C1.N1(CCO)CCCOCC1 Cc1oc(Br)cc1C(N1CCCC1C1(C)CC1)=O N1(C(CC(C)OC)=O)CCN(C(C2COCC2C(N)=O)=O)CC12CCC2 n1(CC(N2CCOCC(NC(C3OCCO3)=O)C2)=O)nnc2c1CCCC2 C#Cc1cn(C)nc1C(=O)N(CCCNC(c1cc(Br)n[nH]1)=O)CC C(c1ccc(O)c(O)c1)=CC(=O)NCC(C1CC1)NC(C(c1ccccc1)C)=O c1(CS(C)(=O)=O)cccc(C(=O)NCCCCNC(=O)C=Cc2ccc[nH]2)c1 CCC(CC(=O)N1CC(NC(C2(C)CCCCO2)=O)CC2(CC2)C1)C(F)F N1(C(Cn2c(=N)nc[nH]2)=O)CC2(CCC2)CC1C(=O)NC1CCCN(O)C1=O c1(CC)ccc(NC(C2(NC(=O)CSC(F)F)CCCC2C)=O)c(C)c1 C1(OC)CC(O)C(O)CC1C(=O)OCC1(C)CCN(C(=O)OC(C)(C)C)CC1 N1(C(Cc2nc(C)sc2C)=O)CCCC(NC(c2cc3occc3[nH]2)=O)CC1 c1(NC(N2CC(C(N(C)C)=O)C2)=O)cccc2cc(N)ccc12 Cc1ccc(CCNC(C2(c3nccs3)CCCC2)=O)c(Br)c1 C12(C(N3CCCC(NC(C45CCCC4C5(F)F)=O)C3)=O)CCCN(CCC1)C2 N1(C(CCOC(C)C)=O)CCC(CNC(=O)C#CC2CCCO2)C(F)(F)C1 C(CO)(CC(F)(F)F)NC(C(COCC)NC(=O)C(=O)C(C)C)=O Cc1nc(Cl)cc(=NCCC2C(C)CCCN2C(C2CCCN2C(N)=O)=O)[nH]1 c1(C(N2CC(C3CN(C(C4(C)CCC4)=O)C3)C2)=O)ccc2c(c1)C(=O)CCCC2 O(NC(=O)C(CC1CC1)NC(C1CC1Cl)=O)C(COC)COC C1(C(CNC(CCCN(CC)CC)=O)O)CCCN(C(=O)CCCCOCCO)C1 CC(C)(C#N)CC(=O)N1CCC(C(N2CCC(C)(CCO)C2)=O)C1(C)C C1(NC(C(CC)c2cccnc2)=O)COC2(C1)CN(C(=O)C=Cc1ccco1)C2 c1(C(=O)NC23CC(C(N(C4CC(F)(F)C4)CC)=O)(C2)C3)ccc(F)cc1Cl Cn1cc(C(N2CC3CC3(NC(=O)C(=Cc3cccnc3)F)C2)=O)ncc1=O c1(NC(C(CC#C)NC(=O)CCC(C)=O)=O)cccc(C#C)c1C CC(C)(CN(C=O)CCC12CCCC1C2)C(N)=O c1(C(=O)NCC(C)(C2CCC2)NC(=O)CCc2cn[nH]c2)ccc(F)c(CO)c1 O=[N+]([O-])c1ccc(I)c(NCCCc2cccc(O)c2)c1 C1(NC(c2ccc(OC)nn2)=O)CC2CCC1(NC(C1CC1c1cnc[nH]1)=O)C2 C(=O)(C1(NC(N)=O)CCc2ccccc21)NC1CC(=O)N(C)C1=O N1(C(C(C)(C)N2CCCC2)=O)CC2(CCC2)CC1CNC(=O)C(F)(F)CO c1(C(N2CCC(CCOC)CC2)C(=O)NCC(F)F)ccc2ncccc2c1 C1(NC(Cc2ccc(OCC(C)C)cc2)=O)CC2(C1)CC(N)C2 C(C)(C)(C(C)(C)CO)C(=O)NCC1(CC(C)C)CC1.C1CC(=O)NCCCO1 C(=O)(C(F)C(C)(F)F)N1CCC(C(=O)NCCCOCCCC)C1C C(C1=NOC2(CCC2)C1)NC(C(N1CCCCC(C)C1)=O)=O n1(CC)nc(C(=O)NC2(C(N3CC(C)(C)C3C3CC3)=O)CC2(C)C)cc1C CC(C)C(C(=O)N1CCC(O)(C(F)F)C1)NC(=O)C(C)CC1CCCC1 N1(C(C(C(=C)Cl)(C)C)=O)CCCC(C2CCN(C(=O)C(C)(C)c3ccno3)C2)C1 CC1(C)CC(C(=O)NCCC2COCCN2C(=O)Cc2ccco2)CCO1 C12(CNC(C(CC=C)(F)F)=O)CC(CCO1)N(C(=O)C(C)CCOC)C2 c1(C(=O)NCC2(O)CN(C(c3c(CC)cno3)=O)C2)cccc2cc[nH]c12 N1(C(c2c(Cl)ccc(N)c2)=O)CC(=O)NC(=O)C12CCCCC2 N1(C(Cc2cnn(C)c2C(F)F)=O)CCC2(C1)CN(C(c1csnc1Cl)=O)C2 C1(C(=O)NC2CCCC(NC(C(C)(C)C(F)F)=O)C2)COC2CCCCC12 C=CCC(CC)C(=O)NCC1CCCCN(C(=O)C(C)(C)CCSC)C1 C(CC(F)F)(C(=O)NCC1CC[Si](C)(C)C1)N(C(C(C)OCC)=O)C c1(CC)ccc(C(=O)NC(C)CNC(c2cc(-c3ccc(C)s3)[nH]n2)=O)c(C)n1 N1(C(c2nccc(CC)c2)=O)Cc2occ(C(=O)NC3CCCC3C#N)c2C1 C(=O)(C(C)(C)CCNC(c1ccncc1)=O)N(C)CCc1cnc[nH]1 C1(C(=O)NC(COC)CNC(=O)C(C)C2CC2)CC2CCC1CC2 C(=O)(C(C)(O)CC)NCCNC(C1CCN(c2ncc(C(=O)OC)s2)C1)=O CCC(C)(CNC(=O)C(=O)NC1CC1)C(=O)NC.C1C(O)C(=O)N1 c1(CC)cc(C(N2CCCC2CCC(=O)NCC2CCC2C)=O)ccn1 C(CC(C)(C)CC(=O)N1CC2CCN(C(=O)C(CC)c3cccnc3)C2C1)OC C1(NC(C(=O)NC2CC2)=O)CN(C(=O)Cc2ccccc2Br)CC2(CCC2)C1 N1(C(C=C(C#N)C(F)(F)F)=O)CC2(C1)CN(C(=O)C=CBr)CC2CO C(=O)(C1CCc2nnc(C)n21)NCCCC(CCC)NC(c1csc(C)c1)=O Cc1ccc2c(c1)C(C(=O)NC1CCN(C(c3cc(C4CC4)on3)=O)CC1)C2 Cc1cc(CNCC2CC(C(=O)N(C)C3CC3)=NO2)cc(C)c1F c1(C(N(C(C)CNC(=O)CN2CCOCC2=O)C)=O)nn(C)c2c1CSCC2 N1(C(C=CC(C)NC(C2CCOC2C)=O)=O)CCC(C)C1(C)C c1(C(N2CCC(CNC(C(C3CC3)OCC)=O)C2)=O)cnc(C)c(C)c1 C(=O)(C(C)(C)Cc1ccccc1)NC(CCN(C(C(COC)C)=O)C)C N1(C(C(C(=O)OC)(C)F)=O)CCC(C2(NC(=O)C(C)N(C)C)CC2)CC1 C1(NC(C2(CC#C)CCC2)=O)CN(C(c2ccco2)=O)C2(CCCOC2)C1 c1(CNC(C2(C)CCCC2)=O)ccc(C(N2CCC(CCO)C2)=O)cn1 Cn1nc(I)c2cc(C(N3CC(NC(c4csc(Cl)n4)=O)CC(F)C3)=O)ccc12 N1(C(C(=O)N(CCNC(=O)C=CC2CCC2)CC)C)C(C)CCC1C N1(C(c2c(O)ccc(C(C)C)c2)=O)CCC(NC(C2SCCS2)=O)C(F)(F)CC1 c1(NC(C)C)ccccc1C(=O)NCC1(O)CN(C(=O)C(C)(C)C2CCCC2)C1 c1(C(C)=O)cnc(NC(=O)COC(c2nnc(C3CCC3)o2)=O)[nH]1 CC1(CNC(=O)CCC2CCCN(C(c3cn(CCO)nn3)=O)C2)COCCO1 C1(C(=O)NC2(C)CN(C(C=CCOC)=O)C2)Cc2ccccc2S1 Cn1c(Cl)nc2nc(Cl)nc(N3CCCC(C)(NC(C4CC(C)(F)C4)=O)C3)c12 n1(CCC(=O)NCC2N(C(c3nc(C(C)OC)oc3)=O)CCC2)c(C)csc1=O c1(C(=O)NC(CCCCNC(CSCCOC)=O)C)cc2c(s1)CCCCC2 c1(N(C)CC2COCCO2)cc(NCc2cccnc2)nc(C(F)(F)F)n1 c1(C(=O)NC(=O)C2CC2)ccc(CCN)cc1.N1(C=O)CCC(N2CCCCC2)C1 C1(CC)CN(CC)CCN1C(C1CCCCCC1NC(c1c(C)noc1N)=O)=O c1(CC=C)ccc(CNC(=O)Cn2cc(C(C)O)nn2)cc1 C(=O)(C1=CC2(CCOC2)C1)N1C(C(=O)NCc2cccc(C#N)n2)(COC)CCC1 c1(NC(c2c(CC)cc(Cl)cc2)=O)n[nH]c2c1CN(C(c1ncccc1Br)=O)C2 N1(C(C(c2c(C)cc(F)cc2)O)=O)CCN(C(c2sccc2C)=O)C2CSCC12 C1(=O)C(C(C)(C)C)CN1.O(NC(=O)CC1CCCOC1)C(COC)COC C(C(=O)N1CC(NC(c2ccc(Br)o2)=O)C(O)C1)(C(C)(C)C)NC(C)=O c1(OC)c(F)cc(F)c(C(N2CC3CC2(C)CC3)=O)c1Br N1(C(C2=CC(C)(C)C2)=O)CCCC(C2CCN(C(=O)CC(C)(C)C)C2)C1 N1(C(C2C(C)=C2)=O)CCCCC1C1(NC(=O)Cc2csc(C)n2)CC1 C1(CN(C(=O)C(C)(C)n2cccn2)C)CN(C(=O)C(C2CC2)C2CC2)CCO1 C1(CNC(CC2(OCC)CC2)=O)CC2CCCC2N1C(=O)Cc1cnn(C)c1 c1(C(=O)NCCCCN(C(C2C(C)CC2)=O)C)cccc2cccnc12 c1(C(=O)NC2(CNC(C(C)OCC=C)=O)CCCC2)n[nH]c(C)c1Br C1(C(=O)NC(c2ccccc2F)CNC(C=C(C)C(C)C)=O)CC2(CCOC2)C1 C1(NC(CCC(C)N(C(CC2CC(=C)C2)=O)C2CC2)=O)CN2CCC1CC2 c1(N2CCC(CCC#N)CC2)ncccc1S(=O)(=O)N1CCCCC1C1CC1 C1(CNC(C=C2CCN(C)C2)=O)CN(C(=O)CC2(N(C)C)CC2)CCCO1 c1(C(N(C(C)CNC(=O)COCC2CCC2)CC)=O)cc2scnc2[nH]1 CC1Cc2ccccc2N1C(=O)CC1CCCCC1NC(c1cn(C)cn1)=O N1(C(Cn2c(C)cnc2)=O)CC2CC2(CNC(c2nocc2Cl)=O)C1 C(C(C(=O)NC(C)(C)C(F)F)C(C)(C)C)NC(C(C)(C1(C)CC1)OC)=O CN1CCC(=CC(=O)NC2(CNC(=O)CCCNC(=O)C3CC3)CCOC2)C1 c1(C(=O)NC23C(CN(C(C(CC=C)(C)CC)=O)C2)CC3)ccc(Cl)c([N+](=O)[O-])c1 N1(CC(=O)N(C2CCN(C(=O)COc3csnn3)C2)C)CCCCCCC1=O C(c1cccc(OC)c1)=CC(=O)NC(CCN(C(CCC(C)OCC)=O)C)C C1(C)(CNC(C(COC)(C)C)=O)CN(C(c2cccc(NC(N)=O)c2)=O)CCO1 C1(NC(C(N2CCC(C)CC2)=O)=O)CCN(C(=O)CC2CC(F)(F)C2)C1(C)C N1(C(c2ncc(C)nc2)=O)CCCC(F)(C(=O)NCCOC2CCCC2(C)C)C1 C1(NC(CCSc2cc(C)on2)=O)=CC=CN=CS1 c1(OC)cc(C)c(C)cc1C(=O)NC1CC1C(=O)Nc1nc(C)c(F)s1 C(c1cc(F)c(F)c(F)c1)=CC(N1CCCC(NC(C(C)S(C)(=O)=O)=O)C1)=O CC(CC(=O)NC1CCCC1CNC(C1CC2(C1)CC21CC1)=O)C(F)(F)F C12(CNC(C3CC(C)(C)C3)=O)CCC(CC1)N(C(=O)C(C)(C)CC1CC1)C2 N1(C(C(N)CCF)=O)Cc2ccccc2C(c2cccs2)C1 N1(C(C2N(C(C3(C)CSC3)=O)CSC2)=O)CCOC2CC12 C(=O)(CCCCC1CC1)N(C(C)CNC(C1CSCCS1)=O)C c1(C(=O)NCCC(C)N(C(=O)Cn2cccc2)C)ccc(-c2ccccc2)[nH]1 CC1CC(C(=O)NCC(C)(Cn2cccn2)NC(C2(C)CNC(=O)O2)=O)CCS1 CP(C)(=O)CN1CC(C(=O)NCC(C)(C)NC(C23CCC(=O)N2CCS3)=O)C1 c1(C(=O)NCC2CCN(C(c3n(CC)nnc3)=O)C2)ccnc(C(N)=O)c1 C1(C(N(C)CC2COC(=O)N2)=O)CCCC(NC(=O)C2=CCCC2)C1 c1(C(=O)OC)cnc(NC2CN(C(=O)OC(C)(C)C)C2(C)C)c(Br)n1 c1(C(N2CC3C(Br)C3C2)=O)cc2c(Br)cncc2s1 N1(C(C(C(CC)C)O)=O)CCC2C1CCN2C(c1ccc2ncnn2c1)=O Cc1nn(C)c2sc(C(N3CC4(C3)CN(C(C3CCCC(C)C3)=O)C4)=O)cc12 c1(NC(=O)NCCN(c2cnc(C3CNC3)o2)C)coc(-c2ccsc2)c1 c1(C(=O)NCCCC(C)(C)NC(c2cncc(OC)n2)=O)c(C)cc(F)cc1C C1(C(=O)Nc2ccsc2)Cc2cc(O)ccc2CN1C(=O)CCc1ccco1 N1(C(=O)COCC2CCCC2)CCCCC1C1CCN(C(C2(F)CCCC2)=O)C1 S(=O)(=O)(c1cc(F)c(Br)cc1F)N1C(C(=O)NCC2(CO)COC2)CC(C)C1 C(CC1CCCC1)(C(=O)NC(c1csc(C)n1)C)NC(C1CN(C(C)=O)C1)=O C(C)(CCCC(=O)NC(CO)C(C)(C)CO)NC(C1(C(=O)OCC)CC1)=O C1(CNC(COc2c(C)cccc2C)=O)C(C2CC2)CCN1c1nnc(C(N)=O)s1 C1(O)(CNC(CC=C)=O)CCCN(C(c2ccc(C3CCC3)cc2C)=O)CC1 Cc1sc(Br)c(C(N2CCC23CN(C(c2ccc(F)cc2)=O)C3)=O)c1C C(C(=O)NC(C)CNC(=O)CC1(C)CC1(F)Cl)(C(C)C)OCC(C)C C12CC(=NO1)C(=O)NC2.C(C1CCOC1)=CC(=O)NC1C(C(C)(C)C)C1 C(CCC(C)(C)C(=O)N(C(CCO)C(F)F)C)NC(CCCCC)=O C1(CNC(C(C)=CC)=O)CN(C(C2CN(C(N)=O)C2)=O)CC1(C)C c1(C(N2CC(CNC(C(C(C)C)NC(C)=O)=O)C2)=O)cncc2c(F)cccc12 N1(C(C2CC(OC)C2)=O)C(CNC(C2CC(C)C2)=O)CC2CCCC12 CCC(c1ccccc1)=CC(=O)N(CC(C)(C)CNC(=O)Cn1nccc1C)C c1(NC(c2ccc(NC3=NCCC3)cc2)=O)cc(-c2nn[nH]n2)cc(Br)c1 CCCC(C(=O)N1CC(O)(CCNC(=O)C(C)C(F)F)C1)OCC c1(C(N(C(CCNC(C(=O)NCCNC(C)=O)=O)C)C)=O)ccncc1O c1(C(COC)(C)C)cc(=NC(=O)C(=O)NC2CCCCCC2c2ccccc2)[nH]o1 C1(C(N2CC(N(C(=O)C(C)(F)F)C)C2)=O)CCc2ccccc2N1 C(=O)(CCC(C)S(C)(=O)=O)N1CCC(CC=C)(NC(C23CC=CC(C2)OC3)=O)C1 C1(COC)(CNC(c2cccn2C(C)C)=O)CCN(c2nnn(C)n2)CC1 C1(C(=O)NC(CC)CN(C(=O)C(C)SC)C)CC2(C1)CC2(F)F N1(c2c(Br)cnc(OC)n2)CCN(C(=O)Cc2c(C)n[nH]c2C)C(C)(C)C1 C12(C(=O)NCC(CNC(c3cccc(C(C)=O)c3)=O)(C)O)CCCC(C)(C1)OC2 CCC(C(=O)N(CCC(=O)NCCn1ccnc1)C)C(F)(F)F CCCCC(O)CC(=O)NC(C1CCCN1C(=O)Cc1nncn1C(C)C)C C1(CC(=O)NC(CCC)CO)C2CCC(C2)N1C(=O)Cc1ccon1 c1(C(=O)OC)cnc(N2CCCC(C)(NC(c3nnc(O)nc3O)=O)C2)cc1C CCCC(CCC)C(=O)N1CC(CCC)(C(N2CC(O)CC2COC)=O)C1 Cc1ccc(-c2nc(CC(=O)NC3CCC(N(C(=O)CC(F)F)C)C3)cs2)o1 C1(C(N2CCC(NC(=O)CCn3cccn3)C23CC3)=O)CC12CCS(=O)(=O)CC2 C(CC(O)CNC(c1ccn(CCC#N)n1)=O)NC(C1(CCC=C)CC1)=O N1(C(C=C(CC)CC)=O)CCC(C)C(CC(=O)NCCN2CCCCC2=O)C1 O=C(CCCC(F)(F)C(F)(F)F)NC1CC2CC1N(C(C1CC1F)=O)C2 C#CCCCCC(c1nnnn1Cc1ccccc1)NCCN1C(=O)CCC1=O N1(C(Cc2scc(C(C)(C)C)n2)=O)CCC(NC(C2CC2F)=O)C1(C)C C1(OC)CC(C(=O)N(C)Cc2ocnc2C)N(C(C2CC2(Cl)Cl)=O)C1 Cc1ccc(-c2cc(C(=O)NCC=CCNC(c3cc(CF)on3)=O)on2)cc1 C(=O)(CCCCN=[N+]=[N-])NCC1CC(OC)CN1C(C1CC12CCCC2)=O N1(c2nnc(CC)o2)C2CCC1C(C)C(NC(c1cc(C)no1)=O)C2 c1(C(CC)C)ccc(C(N2CCC2Cn2cc(CCC(C)(C)O)nn2)=O)cc1 CC1(C)CCC(CC(=O)N(c2cccc(Cl)c2)CC(C2CCOC2)O)CC1 C(C(CC(=O)N(C)CC1(NC(=O)CS(=O)(=O)N(C)C)CC1)CC(C)C)NC(C)=O C(=O)(CCC1CC1)NC(C1CCOC1)C#C.C12(CC1)C(C)(C)N2 c1(C(N2CCCC2c2cccc(F)c2F)C(=O)NCC2CC2)cccc(Br)c1F CC1CC(NC(=O)Cc2cnccn2)CN1C(c1csc(C#N)c1)=O N1(C(C(=C(C)C2CC2)F)=O)CC2CCCC2(NC(=O)Cc2cc(C)ns2)C1 C1(CC)CCOCCN1C(=O)CN1CCN(CC(C)(C)O)CC1 CC1CCC(Cl)=C(C(=O)N2CCC(CNC(c3ccc4c(c3)NCCC4)=O)C2)C1 C(CCCCC(=O)Nc1ccccc1F)NC(C=CC1(C)COC1)=O N1(C(C2CC23CCOCC3)=O)CCC2(CC1)CN(C(c1ccsn1)=O)CC2CO Cc1nc(CO)sc1C(=O)NC1CCCCC1CNC(=O)Cc1ccnnc1O N1(C(C(C=C)CC)=O)CCC(C=CC(N2CC[Si](C)(C)CC2)=O)CC1 C1(C(N2CCN(C(c3c(C)c(Br)cs3)=O)CC2)=O)CCCCC12CCC2 CC(C)(C(=O)N1CC(O)(C2CCCN2C(C2C3CC4C(C3)C24)=O)C1)C(F)(F)F CN1CCC(NC(=O)C(=O)CCc2cn(CCC(=O)N3CCCC3)nn2)C1(C)C C1(CCC(=O)NCCC2(OC)CN(C(c3ncc(C)s3)=O)C2)CCC(O)CC1 C(c1cn(C)c2ccccc12)=CC(=O)NC(C1CN(C(c2n[nH]cc2Cl)=O)C1)C C(=O)(C1(C)CCc2ccccc21)N1CCCC(N(C(=O)C2=CCSC2)CC)C1 N1(C(C(C)(C)SC)=O)CC2CCCCC2(CNC(c2ccncc2C(F)F)=O)C1 C1(NC(c2n(CC)ncc2Br)=O)CCCC12CN(C(C1CC13CC3)=O)C2 c1(C(=O)NC(CN(C(C2(COC)CCOC2)=O)C)C)ccc([N+](=O)[O-])c(SC)c1 C1(N(C(CCOC(C)=O)=O)C)CCCC2CN(C(C3COC(=O)C3)=O)CC12 c1(COC)nn(C)cc1C(=O)Nc1cccc(NC(=O)C=Cc2nccn2CC)c1 c1(C(=O)NC2CN(C(C3CCCS(=O)(=O)N3)=O)CC2F)ccnc2ncnn12 c1(OC)ccc(C(=O)N(CC(=O)NCC2(C(C)(F)F)CC2)C)s1 Cn1nc(C(=O)NCc2cc(C(C)(C)C)no2)cc1C(F)(F)F Cc1[nH]cc(C(=O)NCC2CCC(C)CN2C(=O)Cc2cn[nH]c2)c(=O)c1Cl N#Cc1cc(C(=O)NC2(c3nc4ccccc4s3)CCC2)ccc1O N1(C(C2CC(=O)NC(=O)N2)=O)CCC2(CC2)CC1C(=O)NCCCN1CCCC1 C1(CC(=O)N(C)CC2(OC)CCC2)CN(C(c2cc(C)nn2C)=O)CC1C c1(C(N2C(CNC(=O)CC=C(Cl)Cl)CC2)=O)cc(Cl)c(Br)cc1F C1(C(COC)NC(C2CN(C(c3n[nH]c(C)n3)=O)C2)=O)CCCN(C(C)=O)C1 c1(C(C(C)C)NC(=O)C(N)C2CC2c2ccccc2)ccc(F)c(F)c1 c1(OC)nc(C(N2CCCC2CNC(=O)N(CCCO)CCO)=O)ns1 C1(S(C)(=O)=O)(C(N2CC(CNC(C3N(CC)CC3)=O)N(C)CC2)=O)CCOCC1 Cn1nc(CC(=O)Nc2cc(C(C)(C)C)no2)cc1C(F)F C1(CNC(C2CCN(C(CC)=O)C2)=O)(OC)CCN(C(=O)C(C)O)C1 C1(C(=O)NCC(C)C)COC(CNC(=O)C(c2ccccn2)C)C1 C1(NC(Cc2c(C)nsc2)=O)(CO)CCN(C(=O)C(C)(C)C2CCCCO2)CC1 C(C)(CCN=c1ccnc(NCCCc2cccc(Br)c2)[nH]1)OC N1(C(C=CC(C)C)=O)CCN(C(=O)C=CC2CCOC2)C(CF)C1 CCC(C(=O)NC(C1CN(C(=O)Cc2ccccn2)C1)C)NC(C)=O C1(NC(=O)COC2CCOCC2)CN(C(c2cnc3n2CCS3)=O)CC1C1CC1 C1(C(C)C)CN(C(c2ccon2)=O)CC1C(N1CC(CF)C1)=O c1(C(N(C)CC2CC2CNC(=O)C(O)CC(N)=O)=O)ccc2nccn2c1 c1(CC(=O)N(C2CC(C)N(C(=O)CN(C)C)C2)CC)ccc(C#N)cc1.C1(=O)CN1 C1(CC)C(NC(C2CN(C(C)=O)C2)=O)CCN1C(=O)CN1CCCC1=O.C(C)(C)(C)O c1(C(N2CC(OC)(CNC(=O)C(F)=C(C)C3CC3)C2)=O)cc2n[nH]cc2cc1C N1(C(C(CC=C)(C)N(C)C)=O)C2CCC1CN(C(=O)C1=NN(C)C(=O)CC1)CC2 C(=O)(CC(C)(C)COC(C)=O)N1CCC(COC)(CNC(c2coc(C)c2)=O)C1 C1(C)(CNC(C(C(C)C)OC)=O)CN(C(c2ccsc2C#N)=O)C(C)(C)C1 C1(C(C)(C)CO)COCCN1CC(=O)NCCCSc1cccc(F)c1 c1(C(=O)NCCN(C(=O)CCCn2ccnn2)CCOC)ncsc1C C1(CN(C(=O)C(C)(C)CC2CCC2)C)CCCC(NC(c2ccncc2F)=O)C1 c1(C(=O)NCC(C(C)C)NC(C2(C=C)CCOCC2)=O)cnc2ncc(Cl)cn12 c1(C(=O)OC)n[nH]c2ccc(C(=O)Nc3cccc(C4CC4(F)F)n3)cc12 C(=O)(C(C(C)NC(c1sccc1C#N)=O)C(C)C)NCC(C1CC1)SC N1(CCNC(=O)NC2N(C)C(C(N)=O)CC2)C(=O)NC(C)(C)C1=O N1(C(c2nccc(CC)c2)=O)CCC2(CC1)CC(Nc1nc(C#N)c(Cl)s1)CO2 N1(C(C(CC)(C)O)=O)CC2=C(C1)CN(C(=O)CCCc1ncc(C)o1)C2 N1(C(CC2(C(=C)F)CCC2)=O)CCCCC(CNC(c2ccc(O)nc2C)=O)C1 C1(NC(c2nc(C)oc2)=O)CC2CCC(C1)N2C(=O)CCn1ccnc1C C1(NC(c2ccc(C#N)s2)=O)CC2CCC(C1)N2C(=O)CSCCC#N C1(=O)CCCCN1.C(C)(C(=O)NCCNC(=O)N(C)C)N(CCC)C C(=O)(CCCC(OC)OC)NC12CC(CNC(CCC(=C)C)=O)(C1)C2 C12CC13CC(C3)NC(=O)CCSCC(=O)N2.N1(S(CC)(=O)=O)CCCCC1 c1(C(=O)NCC2CCN(C(C3C(=C)CC3)=O)C2)csc2c(Br)cccc12 C1(COC)CN(C(c2cc(N(C)C)ccn2)=O)CCN1C(c1cnnc(O)c1)=O C(=O)(CCCCCC(C)C)N1CCC(C(=O)NC2CC(F)(C(=O)OCC)C2)C1 c1(C(N2C(CC)CN(C(C3(Br)CCC3)=O)CC2)=O)ccc2ncnc(O)c2c1 c1(COC(c2ccc(N3CCC(OC)C3)o2)=O)cc2nc(Cl)ccc2o1 c1(C(C)(CNC(=O)OC(C)(C)C)NC(C2C=C(C)CS2)=O)ccccc1F c1(-c2c(C)ccc(OCC)c2)cnc(Cl)c(C(=O)Nc2ncc(C)nc2Br)c1 c1(CC(=O)NC(C2CCN(C(C=CCN(CC#C)C)=O)C2)C)cccnc1O C1(NC(C(=O)NC2N(C)CC(C)(C)C2)=O)Cc2nc3ccccc3n2C1 c1(NC2(C)CC(NC(CCC(=O)NCCC)=O)C2)nc(C)c(C#N)cc1Cl C1(CC=C)(NC(=O)CC2CCSC2)CCN(C(C2(C(F)(F)F)CC(F)C2)=O)CC1 C1(CC(=O)NC(c2cc(-c3ccccc3)n[nH]2)C)CS(=O)(=O)CCN1C C1(C(=O)C(c2sccc2S(C)(=O)=O)C#N)CCC2CC1CN2C(=O)OC(C)(C)C c12cc(c(C)c([N+](=O)[O-])c1)C(=O)N1CCC1CN2.n1(CC)ccnc1CNC Cc1nn(CCC(N2CCC(NC(c3nccs3)=O)C(C)C2)=O)c(C)c1C C12(CNC(c3c(CC)n(C)nc3)=O)CCCC1N(C(=O)Cn1cnnn1)CCC2 Cc1ccc(NC(c2nnnn2C(C)(C)C)C2CC2(Br)Br)cc1F C12(C(=O)NCC3N(C)CCOC3)CCN(C(=O)CCc3ncn(C)n3)CCC1C2 N1(C(c2c(N)cn(C)n2)=O)CCC(C(F)(F)F)C(CNC(=O)CCCCC#N)C1 N1(C(c2n(C)c(S)nc2)=O)C(CNC(C2CCC2C(F)(F)F)=O)CC2CCCC12 N1(C(c2cnn(C(C)C)n2)C(=O)NCCSC)CCC(C)(C)CC(C)(C)C1 N1(C(C2CN(C(C)C)C2)=O)C2CCC(C(N3CC(F)(CO)C3)=O)C1CC2 C(=O)(N(OC)C(C)C)C1CCC(CNC(C2(C)CC(=C)C2)=O)CC1 CC1CC(NC(c2cn(C)nc2Cl)=O)CCN1C(c1cncc(C(N)=O)c1)=O C(=O)(C(CN(C)C)C(C)C)N1CCCC(NC(C2(COC)CC2)=O)C1C C#CCC(C)C(=O)NCCC1CCCN1C(=O)C(O)C1CCCC1 N1(C(CC2C(=O)CCCC2)=O)CCN(C(=O)C(CC2CC2)CC2CC2)CC(O)C1 C1(CNC(c2c(CC)ocn2)=O)CN(C(=O)CSc2nnnn2C)C(C)(C)C1 N1(C(CCC=CC)=O)CCN(C(c2ccc(Br)c(C)c2)=O)CC1C1CC1 n1(CC(=C)C)nnnc1C(c1cnc(-c2ccccc2)o1)NC1CC1F c1(NC(C2CCN(C(C(CC)NC(c3ccccc3)=O)=O)C2)C)ncc(O)cn1 CC1(C)CCC(C(=O)NC(CC2CC2)C2CC2)CN1C(C1(O)CC1)=O c1(NC(c2c(OC)ccs2)=O)ncc(-c2ccc(OCCN(C)C)nc2)cn1 c1(C(=O)NC2CCCC(NC(C(C(C)C)N(C)C)=O)C2)ccc2c(c1)NC(=O)C2 C1(F)(C(N(C(c2nccc(C(F)F)n2)=O)C)C2CC2)CCNCC1.C(=O)(C(F)(F)F)N C1(COC)CCN(C(=O)OC(C)(C)C)CC1.c12nsc(n1)C(C)OC2=O c1(NC(C2N(C(CSc3cn(C)nc3)=O)CC(F)C2)=O)ccc2c[nH]nc2c1 C(=O)(CC(F)(F)CC)NC1C(CC)N(C(=O)C2=CCCCO2)CC1 C(C)(C(CC(=O)NCCc1ccsc1)NC(c1cnc(O)c(C)c1)=O)OC c1(C(C)CNC(=O)CNC(=O)CCc2ccc(N)cc2)cc(F)cc(F)c1 C1(CNC(c2occ(C)c2C)=O)CCN(C(c2ncccc2CO)=O)CC1C c1(NC(C(CC(C)C)NC(c2ncccc2Cl)=O)=O)cn(C)c(=O)nc1O CS(=O)(=O)CCC(=O)N1CCC(C(c2cn(CC3CCC4CC4C3)nn2)C2CC2)C1 C1(CNC(C(C2CCCOC2)OCC)=O)CN(Cc2ccc(C)s2)CCO1 C(=O)(CCC(C(C)C)NC(c1ccnc(CO)c1)=O)N1CC(C#C)(F)C1 C1(C(=O)NCCC=CC)CSCCN1C(c1ccc(CO)o1)=O O=C(C1=C(Cl)CC1)NCC1C2CC1N(C(c1cc[n+]([O-])cc1)=O)C2 C1(CNC(c2oc(C(=O)OC)c(C)c2)=O)(CO)CCN(C(C2CC2C#N)=O)CC1 C(=O)(C(F)(F)CC1CCCO1)N(CC(C)CNC(c1n[nH]c(C2CC2)c1Cl)=O)C c1(OC2CN(C(c3c(C(=O)OC)cco3)=O)C2)ccccc1O N1(C(CCNC(=O)OC)=O)CC(N(C(=O)Cn2cncn2)C)C(F)C1 C(=O)(C1CCCc2ccnn21)N1CC(OCCNC(CCCCCC#C)=O)C1 c1(CC(=O)NCC2CCN(C(=O)CC3CS(=O)(=O)C3)C2)ccc(C(F)(F)F)nc1 S(=O)(=O)(C1CCN(C(C)(C)C)C1)Nc1c(C)cc(C(=O)OC(C)(C)C)o1 C1(C(=O)NCc2nc(C)c(C(=O)N(C)C(C3CCCC3)C)o2)CC(C2CC2)=NO1 C(C(=O)NCc1nnn(C)c1C(N1CC2C=CC2C1)=O)(C(C)C)SC O=C(CC1=CCN(C(c2ccc(O)nc2)=O)CC1)NCC(F)Cl c1(C(=O)NC(C(=O)NCCS(C)(=N)=O)(C)C2CCC2)ccc(C#N)n1C c1(N(C(C(=O)OC)C)C)ncoc1C1CN(C(N2CCCCC2)=O)C1 CS(=O)c1ccc(CC(N2CCC(C)C(NC(=O)Cc3nc[nH]n3)C2)=O)cc1 N1(C(C(=O)NC2C(c3cncc(C)c3)CCC2)=O)CCC(O)C(C)(O)C1 c1(C(=O)NC2CCN(C(C3CC(C)C3)=O)CC2F)cc(Cl)cc(Cl)c1O CC(CC(=O)NC1CN(C(c2ccc(=N)[nH]n2)=O)CC12CC2)C(F)(F)C(F)(F)F c1(CC(=O)NCCC2(NC(=O)CCC3CCCOC3)CC2)nnc(O)s1 Cc1nc(NCC2(C)CCCS2)cc(=NCC2CC(O)C2)[nH]1 c1(C(=O)NC2C(NC(Cc3c(C)cc(Cl)cc3)=O)CC2)ccn2cnnc2c1 Cc1cn2c(n1)CC(C(=O)NC(C(=O)NC1CC1c1ccco1)C1CCCC1)C2 C=CCC(CC(C)C)C(=O)NC1CN(C(c2cnn(C)c2)=O)CC1CC(C)(C)C Cc1cccc(N2CCN(C(=O)C(=O)N3CC(C4CCC(F)C4)C3)CC2)c1C.CO N12CCOC(C)(C1)C(c1cn(C3CCOC3)nn1)NC(=O)C2.CC(C)(C)C(=O)O c1(C(N2CCC(C(N(CC(C)O)C(C)C)=O)C2)=O)ccc2c(c1)CCC2 c1(CSC)n[nH]c2ccnc(OCCCN(C=O)Cc3cccc(OCC)c3)c12 C(C(C)(CO)CO)N(C(=O)C(c1cccs1)NC(=O)CC1NC(=O)NC1=O)C C=CCC(C)C(=O)NC1CCOC(C(=O)Nc2cnccc2C)C1 c1(CCC(=O)NC(C(=O)OC)C)ccc(Cl)cc1F C1(CC(NOCC(=O)OC)=O)CCCN(C(=O)CC2CCC2)C1 C1(C)(CNC(CC=C=C)=O)CN(C(=O)Cc2ccc(OC)c(OC)c2)C(C)(C)C1 N1(C(c2c[nH]c(=NC)o2)=O)CC(NC(C2CCCN2C(C)=O)=O)CCC1C C(CCC(=O)N(C)CCNC(=O)CO)N(C(C(COC)C)=O)C c1(CC(=O)NC2CC(=O)N(C3CC3)C2)c[nH]c2ccccc12.C12CC1CNC2=O C(=O)(C(C)CC(N)=O)NCC1(C)CCN(C(c2csc(C)c2C)=O)C1 c1(CN(C(=O)CC2(O)CCC2)CCNC(C(C2CC2)SC)=O)ccccc1 C(C)(CCC(=O)N1CC(O)CC1C(=O)N(C1CC1)Cc1cnn(C)c1)OC c1(C(=O)OCC)ccc(NC(C2CCCOC2CCN2CCSCC2)=O)nc1C C(C(CC(F)(F)F)NC(=O)C(C1CCCCCC1)C)NC(C(CSC)(C)C)=O c1(C2C(NC(C(=O)NCC(N3CCOCC3)=O)=O)CN2)cccc(Cl)c1 Cc1cc(Br)cc(C)c1C(N1CCCCC(NC(=O)CCF)CC1)=O C(CCN=C(NCCOCCO)NCC1CC1)N(C)C.C1(C)CC2(C1)CC21CCC1 C1(CNC(c2cc(C)c(C)o2)=O)CN(C(C2CCC(N(C)C)CC2)=O)CC1(F)F C1(CC(=O)N(CCCNC(=O)CCc2cnco2)CC)COCCOC1 C1(OC)CC(CNC(C2CCC2(C)C)=O)N(C(=O)CCOC2CCOCC2)C1 C(=O)(C1=NNC(=O)CC1)N(C)CCN1CCN(C(c2cnco2)=O)CC1 CCC(CNC(c1cccc(C(N)=O)n1)=O)(CC)NC(C1CCS1(=O)=O)=O CC(C)C(C)CC(=O)NC1C=CCN(C(=O)C(C)Oc2ccccc2F)C1 c1(C(=O)NC(CNC(C(CC=C)CC)=O)C(C)C)cccc([N+](=O)[O-])c1O n1(CC)nccc1C(=O)NC(C(=O)NCCS(N)(=O)=O)C1CC1 n1(C(CC)C)nnnc1C(c1cnc(C)o1)NCCCCOC(C)(C)C c1(C(=O)NCC2(OC)CCN(C(=O)CCC3CC3(C)C)C2)ccc(C)c(Cl)c1F C1(NC(C2C(NC(Cc3c(C)nccc3)=O)CCC2)=O)CCCCC12CC2 c1(NCc2cc(O)c(C(F)(F)F)cc2)ccc2ncccc2c1 n1(C(=O)NCC2N(c3snc(CC)n3)CCC2C2CC2)[nH]cc2c(=O)ncnc1-2 c1(OC(C)CNC(=O)CCN2CCCCC2C)ccccc1C#N c1(CNS(C)(=O)=O)cccc(C(=O)NC2CCC(NC(c3cscn3)=O)C2)c1 c1(OCCCC(=O)NC2(C)CN(C(C3N(C)CC3)=O)C2)cccc(C#N)c1 N1(C(C(CC=C)CC(C)C)=O)CCC2(C1)CN(C(c1sncc1C)=O)CC(C)O2 N1(C(c2cn(CCOCC)nc2)=O)CC2CC1CCN2C(=O)CC1(CO)CC1 CC1CC2CC2CC1Nc1ncc(C(C)NCCC2CC3CCC2O3)cc1Cl Cc1cccnc1CC(=O)N(C(C)(C(=O)NCCn1ncccc1=O)C1CCC1)C N1(C(CCc2ccc(C)s2)=O)CCOCC1CN(C)C(c1ncn(C)c1C)=O C1(CNC(CCC#C)=O)CN(C(=O)Cc2nnc(S)n2C)CC1C C(=O)(CCCCC(N)=O)NC1CCC(CCNC(C=CC)=O)C1 N1(C(Cc2c(CC)n[nH]c2CC)=O)C2CC1CN(C(c1cc(C(N)=O)c[nH]1)=O)C2 CC(C)C(C(C)NC(c1cn(C)nn1)=O)NC(=O)CCCCc1cnc[nH]1 Cc1cnc(C(=O)NC2C3CN(C(=O)Cc4n[nH]c(=N)s4)CC23)cc1C c1(C(=O)NC2COCCN(C(c3c(C)n(C)nc3Cl)=O)C2)cc2n(n1)CCCC2 c1(C(=O)NCC2(OC)CN(C(c3nnn(C)c3C)=O)C2)ccc2c(c1)COC2 C1(NC(=O)CC2CCCC23CC3)CC2CC(C1)N(C(=O)C=Cc1cc[nH]c1)C2 N1(N2CCCC(C(C)(C)C)C2)CC2CC(C(C3CCC3)=O)C(C2)C1.C(=O)N c1(C(N2C(C3CCN(C(C4C(C)OCC4)=O)C3)CCC2)=O)cccc(Br)c1 CCC(C)CCC(O)CC(=O)NCC(C)N(C(C1CC(F)C1)=O)CC C1(C(=O)NCC(CO)NC(=O)C=Cc2ccccn2)(OC)CCCCCCC1 c1(N2CCC(C)C2CNC(C2(O)CC2)=O)cc(Cl)c(O)nn1 C#CC1(NC(=O)CC2CCCCC2C(=O)O)CCCC1.c12cnccc1NC2=O CN1N=C(CC(=O)NC2COC3CN(C(=O)C=CC=C(Cl)Cl)CC23)CC1=O C1(C(=O)NC2C(CNC(CC3(OCC)CCC3)=O)C2)CCCC1F N1(CC=C)CCC(C(C)(O)CNCC(CCOC)N(C(=O)NCC)C(C)C)CC1 CCC(CC(F)(F)F)C(=O)NCC1CCN1Cc1cccn(CCOC)c1=O C1(CCNC(C(CC)(C)C)=O)CCN(C(=O)CCOCCOC)C(C)C1 N1(C(COC(C)=O)=O)CCC2CC2(NC(c2c(C)nn3c2CCC3)=O)CC1 C(=O)(C1=C(C)C(C)(C)OC1=O)NC(C1CCOC1)CNC(CCSCC)=O N1(C(CC2(N(C)C)COC2)=O)CC2CCC1CN2C(C1CC=CCC1)=O N1(C(c2c(C)n(C(C)C)nn2)=O)CC(NC(=O)CC(C)(C)O)C2(CCOCC2)C1 Cc1cnc(CNC2(C)CCN(S(=O)(=O)Cc3ccc(F)cc3)C2)cc1Br n1(CC(=O)NCC2(C(C)NC(C3CCN(C)C3=O)=O)CC2)nc(Cl)ccc1=O N1(C(C2C(C)(C)OCC2)=O)CCCC(O)(CCNC(C23CNC(=O)C(C2)C3)=O)C1 C(=O)(C1=COCCC1)Nc1cccc(NC(CC2C(C)(C)C(O)C2)=O)c1 O=C(NNc1nc2cnccc2s1)C1CC2OCCC2NC1 Cn1c(CNC2CC2C(=O)Nc2ccc(O)cn2)nc2ccccc12 c1(OCC)nccc(C)c1C(N1CC(NC(=O)C(O)C(F)(F)F)C1)=O N1(C(C(CCC)F)=O)CC2CN(C(C3CCCOC3C)=O)CC2(C)C1 CC(C)C(C)C(=O)NCC1CC(O)CN1C(=O)C(C)Oc1ccc(O)cc1 Cc1ccc(C(=O)N(CC(C)C#N)CC(=O)NCC2CC(C(C)O)C2)cc1O c1(C(=O)NC2(C)CCN(C(C(CO)OC)=O)C2)ccc(O)cc1F C1(C(=O)NC(C2(OC)CCC2)C)CC2CC1CN(C(=O)C(Cl)Cl)C2 N1(C(=O)NCCCCc2onc(CCC)n2)CCc2c(OC)cccc2C1 C1(CC(=O)OCC)Cc2ccccc2CN1C(=O)C(C)Sc1ccccc1F C(C)(C(C)C(=O)NCCCCCCF)NC(COC(C)C)=O N1(C(COCC(=O)NC)=O)CCN(C(=O)CC2CCCN2C)CC1C1CCC1 C1(O)(C(CCNC(C(C)n2cccn2)=O)(C)C)CN(C(=O)CC2CC2C(F)(F)F)C1 C1(OC)CC2C1CCN2CC(CO)SC c1(CC)ccc(C(=O)NCC2CCCCN(C(=O)CN(CC)CC)C2)c(Cl)c1 C12(C(N(CC(C)N(C(C(F)=C(C)C)=O)C)C)=O)CC3CCC(CC(C3)C1)C2 Cc1ccc(C(c2nnnn2C(C)C)NCCCC2CCOC2)cc1C C1(NC(C2CN(C(C)=O)C2)=O)CC2CCC1CN2C(C12CC1CNC2=O)=O Cc1ccc(Cl)c(F)c1CNCC(O)Cc1ccc(F)cc1F Cc1cc(C(=O)NCC(CNC(c2cc(-c3ccco3)on2)=O)CO)cs1 C(=O)(CCCCCNC(C)=O)N1C(C)CCC(CNC(CCC(=C)C)=O)C1 N1(CC(=O)NCC2CCN(c3nc(C#N)c(Cl)s3)CC2)Cc2ccccc2C1=O c1(C(N2CCC(C(C)NC(CCC(CC)C)=O)CC2)=O)cc(F)c(N)c(F)c1 C1(C(N2CC(c3ccccc3)(NC(C(CC)C)=O)C2)=O)CC(C2CCC2)C1 n1(CCC)cc(C(=O)NC2COCC2CNC(C2CCN(C(C)=O)C2)=O)nn1 N1(C(CCc2cccc(OC)c2)=O)CCN(C(=O)CCC(C)C)CC(C)(F)C1 C1(C)C(C)C(=O)N1.c1(CC)oncc1C(=O)N(C(C)=O)Cc1ccccc1 N1(C(CCN(C(=O)CCS(N)(=O)=O)CC)=O)CCC2(CCCO2)C1 c1(CC)cccc(C(=O)NC2CC(CCNC(C3CN(C(N)=O)C3)=O)C2)c1 C1(C(=O)OCc2cc3occc3s2)CC2CCC1(C(F)(F)F)C2 CC1CC(CNC(=O)COC2CCCOC2)CN1C(=O)Cn1cc(N)cn1 N1(C(CC(C)C(C)(C)NC(=O)CCCC(C)(C)C)=O)CCCCC2(CCC2)C1 c1(-c2cccc(CN3CCC(c4c(C(N)=O)c[nH]n4)CC3)n2)ccc(Cl)c(Cl)c1 C(=O)(C(C)(F)CC1CCCC1)NC(C)CN(C(=O)COCC1CCCC1)C1CC1 N1(C(C=C(C)C(C)C)=O)C2CCC1CC(NC(=O)C(F)CC(C)C)C2 C(=O)(CC(F)(F)C(F)F)N1CCC(N(C(=O)CC(F)(F)F)CC)C1 N1(C(C(C(COC)C)C)=O)CCCC12CCN(C(C1(S(N)(=O)=O)CC1)=O)C2 c1(C(N2CC(NC(CSC(C)C)=O)C(C)CC2)=O)ccc2cc[nH]c2n1 Cc1sc(O)nc1C(=O)N(C)CC=CC(=O)NCC(C)OCCO C1(CNC(C2C(OCC)C2C)=O)CC(C)N(C(C2CN(C)C(=O)N2)=O)C1 C1(CNC(=NC)NC(c2cccnc2)C)CC2CCC(C1)N2Cc1cccs1 c1(C(=O)NC2(CNC(C(C3CCCO3)OC)=O)CC2)c[nH]c(Br)c1 C1(C2CCCO2)(C(=O)NC2C(C)CN(C(c3nscc3N)=O)C2)CCCO1 Cc1nn2c(C(=O)NC3CN(C(c4cccc(F)n4)=O)CCC3C)c(C)nc2s1 C(C(C)(C)CNC(=O)CN1CC2CC2C1)NC(C(C)OC)=O CC1CCC(CNC(C2CCN(C(N)=O)CC2)=O)CN1C(C1CC(O)C1)=O CC(C)(C)CCC(=O)C(=O)N1CC(NC(=O)C2=COCCC2)CC2(CCC2)C1 c1(C(=O)NC(C2CCCN2C(C2CC(CC3CC3)C2)=O)C)cnn(CC(F)F)c1 c1(C(=O)NC(c2cn(CCCCC)nn2)(C)C)cccc2[nH]cc(Cl)c12 C1(C(=O)NC(CC)(CC)CO)CC(C)CN(C(C2C3CCC(F)C23)=O)C1 CC1CC=CCC1N=c1[nH]c2c(c(=NCC34CC(CCO3)C4)[nH]1)CCCCCC2 N1(C(C2C3(CC(C)(C)C3)C2)=O)CCCC12CCN(C(=O)CCc1nc(=N)[nH][nH]1)C2 c1(C(=O)NCC2N(C(CN(CCC)C)=O)CC(O)C2)ccnc(C)c1C C1(CNC2CCN(C(c3ccc(Cl)cn3)C)C2)CCc2nn[nH]c2C1 C1(CNC(c2nc(CC)sc2N)=O)CN(C(=O)Cc2cnc(C)s2)CC12CCC2 CCC(CCC(=O)NC1(CCC(=O)NCC(O)C(F)F)CCC1)OC Cc1cc(C)c(C(=O)NC2CN(C(=O)C(C)CCCc3ccccc3)C2)cc1N N(C(=NCCCC(F)F)NC1CCOCC1)Cc1c(OCC(F)F)cccc1OC C1(O)(CC(=O)NC2CC(NC(C(C)Cc3ccccc3F)=O)C2)CCCCCC1 C1(CC(=O)NCc2ccc(F)cc2)Cc2cccc(F)c2O1 N1(C(C(C)CF)=O)CCC(C2N(c3ncc(Br)cn3)CC2(C)C)CC1 N1(C(CSCC=C)=O)CCC(C)C(CNC(c2c[nH]c(C(N)=O)c2)=O)C1 N1(C(C2(OC)CCCOC2)=O)CCC(C)N(C(c2cnc3n2CCS3)=O)CC1 N1(C(=O)COC2COC2)CCC2(CC1)CCN(C(c1ncncc1Cl)=O)CC2 C12(CCC(=O)NC3(C)CC(NC(c4nc(C(F)(F)F)cs4)=O)C3)CCC(CC1)C2 c1(CCC)cc(C(N2CCC(C(C)NC(=O)C(C)(C)c3cscn3)C2)=O)c(C)o1 C=CC1(CC(N2CCCCC2CNC(C2C(C3CC3)C2(C)C)=O)=O)CCCCC1 C(=O)(C1=CC2(CCOC2)C1)N1C(CCC)CN(C(=O)CN2CSCCSC2)CC1 c1(CC)ccc(C)c(C(N2CC(CNC(C3(O)CCOC3)=O)C(C(F)F)C2)=O)c1 C1(NC(c2cnccn2)=O)CCC2CN(C(c3cccc(C(F)F)c3)=O)CC2C1 n1(CC)cnc2nc(N3CCCC(F)(F)CC3)nc(N(C)Cc3cccnc3)c12 N1(C(CCOC(C)C)=O)CCCCCC(NC(=O)C#CC2(C)COC2)C1 c1(C(=O)NCC2CN(C(=O)Cc3cnc[nH]3)C3CC23)ccc2cnccc2c1 CC(C)CC(CNC(C)C)CC(=O)OCC1(COC(C2CCC=CCC2)=O)CC1 N1(CC(C(=O)O)NCc2ccc(-c3c(C)n[nH]c3)cn2)CCc2ccccc2C1 Cc1ccc(C(=O)NCCS(C)=O)c2c1CCCN2 C=CCCN=C(NCC1(C)CC1)N(C)CC1CCC1 C1(NC(N)=O)CCC(C(N2CC(=C(F)CN(C(=O)C3=CCSC3)CC#N)C2)=O)CC1 C1(C(=O)O)C2CCCC2CN1Cc1ccccc1[N+](=O)[O-] Nc1ccc(C(=O)NCC2CCCC2NC(C2(c3ccccc3)CC(O)C2)=O)nc1 N1(C(COC(C)=O)=O)CC(C)(C)CCC1CNC(=O)C(CC1CCCCC1)C(C)C CCCCC(C)C(=O)NC(C1CCCCC1)CNC(=O)Cc1nc(C)cs1 CN=c1nc(N2CCN(CCS(C)=O)CC2)[nH]c(=NCC(C)(C)C(N)=O)[nH]1 c1(C(=O)NC(C(C)NC(C=CC(CC)=CC)=O)C(C)C)cc2c(cc1N)OCO2 c1(OCC)nc(C(=O)N(CCC(C)NC(C2CC2c2ccsc2)=O)C)co1 CC1(C)CC(CO)(NCCOc2c(F)cccc2Br)CO1 C1(C(=O)NCC(CC)(C)Cl)CCCN(C(c2cnc(=N)[nH]c2)=O)C1C N1(C(C(C)Cn2cccn2)=O)CC(CNC(=O)CN2CCNC(=O)C2)CC1(C)C OCC(Cc1ccccc1)CN=c1[nH]n(Cc2ccccc2)cc1[N+](=O)[O-] n1(CC(=O)NC(C2(O)CN(C(c3c(CC)cco3)=O)C2)C)cc([N+](=O)[O-])c(C)n1 C#CC1(C(=O)NCC(C)C(C)O)CCN(C(C2CC2CC)=O)C1 c1(C(N2CCN(C(C(CCSC)NC(N)=O)=O)CC2)=O)csc2cncn12 N1(C(c2cn(CC=C)nc2)=O)CC(NC(=O)CN2CCCCC2=O)CC1(C)C C1(NC(c2cc(C)on2)=O)CC2(NC(=O)CC3COCC3O)COC1C2 c1(C(N2CCC(NC(C3C4COCC34)=O)C2)=O)c(F)ccc(Cl)c1F N1(C(C2CC(C(C)C)C2)=O)CCC(NC(c2ccc([N+](=O)[O-])[nH]2)=O)C(F)C1 C1(N(C(CN(C)CC2CC(O)C2)=O)C)CN(C)CC1c1ccsc1 Cc1c(C(=O)NCCC(O)CNC(=O)CCn2cnccc2=O)cnn1C1CC1 CC(CN=c1[nH]c2c(c(=NCc3ccc(C#N)cn3)[nH]1)CSC2)c1cccc(Br)c1 c1(N(CCC#N)C(N(C2CCN(C)CC2)C)=O)ccccc1S(C)=O N1(C(C(C)Cc2ccccn2)=O)C(C(=O)Nc2cncc(Br)c2)CC2CC12 CC1CCN(C(=O)CCC2NC(=O)NC2=O)CC1NC(C1(C)CNC(=O)C1)=O N1(C(Cc2c(C)scc2)=O)C2CCC1CC(N(C)C(C1(C3CCC3)CC1)=O)C2 c1(C(=O)NCc2cn(CCN(C)C)nn2)ccccc1CN(C)S(N)(=O)=O c1(CNC(COCCC=C)=O)nc2c(s1)CN(C(=O)CC1(COC)CC1)CC2 N1(C(c2cc(OC)ns2)=O)CC2C(NC(=O)CCCN3C(=O)CCC3=O)C2C1 Cc1ccc(C(=O)NCC2CCC2NC(c2cnc[nH]c2=N)=O)c(F)c1F c1(C(c2nnnn2C)NC(C2CCCCC2)CC)cc2ccccn2n1 CC(O)C(C)C(=O)N(C)CCOCCNC(c1ccn(C(F)(F)F)n1)=O N1(C(c2nc(OC)oc2)=O)CC(C(=O)NCC2(C)CCCS2)CC(C)(C)C1 N1(CCNC(C(C)Cn2cccn2)=O)CCN(C(=O)Cc2ccon2)CC1 c1(C(=O)NC2CN(C(C3CC4CCC34)=O)C2)ccc(S(=O)(=O)N2CCCC2)cc1 c1(C(=O)NCCC(C)N(C(CCC(=O)NC)=O)C)cnn(C)c(=O)c1 N1(C(=O)OC(C)(C)C)CCC(C2CC2NC(C2CCC3(CC3)C2)=O)CC1 c1(CSCCC)ccc(C(=O)NC2(CO)CC2)cc1.C1(C(=O)N)CCC1OC(C)C.C N1(C(c2cccc(OC)n2)=O)CC2(CNC(C3(C)CCNC(=O)C3)=O)CC1CO2 c1(C(=O)NC2(CC=C)CCC2)c[nH]nc1CCNC(=O)C(N)=O N1(C(CC(C)OC)=O)CCC(C(N2CC(O)(C(C)C)C2)=O)C12CCC2 c1(C(C)OCCCNC(CC)C)ccc(C)cc1 N1(C(C(C)NC(CC)=O)=O)CCCN(C(c2ncn3cccnc23)=O)C(CO)C1 C1(C#N)(C(N(CCNC(c2cnc(CC)nc2O)=O)C2CC2)=O)CC2C=CC1C2 N1(C(CCCCSC)=O)CC(NC(=O)CN2CCN(C)CC2)CC12CCCCC2 c1(C(=O)NC(CCN(C(c2c(C)nccn2)=O)C)C(C)C)ccc(N)cc1F CCC(CN(C)C)CC(=O)NCCOCCN(C)C(C1CCCO1)=O C1(COC)CN(C(=O)C(=CC2CCCCC2)F)CCN1C(=O)C=CC1CCCO1 CN1C(=O)OCC1C(=O)NCC1C=CC(NC(c2cnn(CCF)c2)=O)C1 C1(N(C(=O)C=CC2(C)COC2)C)C2CN(C(=O)CCc3nccs3)CC12 C1(=O)C(C)(C)C(=O)N1CC(CC(F)(F)F)C.n1(CCCC)cc(CCN)nn1 C(=O)(C(C)(C)CNC(=O)C(C)(C)C1CCCN1C(=O)CCOCC1CC1)NC C1(CCCC(=O)OC(C)(C)C)CCCC(=O)N1.c12ccc(cc1)OC2C C1(C)(C(N2CCC(=C)CC2)=O)CCCN(Cc2ccn(C)c2C)C1 c1(-c2cc(C)[nH]n2)nc2c(s1)CCN(C(=O)CCNC(c1ccncc1)=O)C2 CN1CCCC2CN(C(=O)Nc3cnn(C4CC4(F)F)c3)CCC12 c1(C(=O)NC2C(NC(CC=C=C)=O)CC2)cccc(F)c1C C1(C(N(C2CCCC2)CC=C)=O)CCCN(C(=O)C(O)C2CCCC2)C1CC c1(CC(=O)NC(CCNC(c2cc(C)ns2)=O)(C)C)cccc(C(F)(F)F)c1 c1(OC)ccc2c(c1)CCC(N=c1[nH]c3c(c(=NCCCF)[nH]1)CCCC3)C2 Cc1cccn2nc(C(N3CC(NC(=O)Cc4cccs4)CC3C)=O)cc12 c1(OCC(=O)NC2C(NC(C(CC)(C)C)=O)CC2)cc(C)ccc1Cl O=C1CCN(CC2CCC=CO2)C(=O)N1CC1CC(O)C12CCC2 N1(C(c2cc(COC)no2)=O)CCN(C(=O)CC2SC(=N)NC2=O)CC1 C1(C(N2C(CNC(C3CC(N(C)C)C3)=O)CC(OC)C2)=O)CCC2(CCC2)CC1 C1(OC2(c3cn(CC(=O)NOCC(F)(F)F)nc3)CCC2)C(=O)OCC1CO c1(C(N2CC(CNC(C(C)OC3CCCC3)=O)C2)=O)ccncc1C(F)(F)F C(=O)(C1=Cc2ccccc2C1)N1CC2C(CNC(C(=Cc3ccco3)C)=O)(C2)C1 C1(NC(=O)Cc2cccc(Br)c2)CC2CC1N(C(C1CCCC(=O)O1)=O)C2 c1(OC)cc(C(=O)NC2(CNC(=O)COC3CCCCC3C)CCC2)cc(C)n1 CC1C(C(=O)NCC(O)CNC(=O)OC(C)(C)C)C1C CC1(C)Cc2cc(CNC(=O)C(N)CO)ccc2O1 N1(C(c2cccc(C)c2F)=O)CCC2(CC1)CC2CNC(C12CCC(C1)OC2)=O C(C(C)CC(=O)N1CCC(F)(F)C1)NC(C1(OC)CC1)=O c1(N2CC(C)CS(=O)CC2)ccncc1S(=O)(=O)NCC(O)C1(Cl)CC1 C(=O)(C(CN(C)C)C(C)C)NCC1(NC(c2c(C)nccc2)=O)CCC1 Cc1cccn2nc(C(=O)NCC3(NC(C4CC45CCOCC5)=O)CCC3)cc12 c1(C(N(CC(CC)NC(=O)C(O)Cn2cncn2)CC)=O)ccc(CSC)cn1 C1(C(N2CC(C)C(CNC(c3cccc(Cl)c3)=O)C2)=O)CCCC(C#N)C1 C(C)(C)(C#Cc1cn(Cc2cccnc2)nn1)NC(C(CC)OCC)=O C1(C)(C(=O)NCC(C)N(C(C2N(C(C)=O)CCC2)=O)C)CC2CC2C1 C(CCC(CCC)NC(=O)C(C(C)C)c1cnn(C)c1)NC(COCC#C)=O C1(CCOC)(NC(=O)C(C)OC)CCN(C(=O)C(C)(C)n2ccc(C)n2)CC1 N1(C(C(CC=C)(C)C)=O)CC2CCC(C1)C2NC(c1ccnc(C)n1)=O C1(NC(c2cnc(C(C)C)s2)c2nnnn2C2CCCCC2)CCOCC1(C)C c1(C(c2nnnn2CC(F)F)NC(CC)CCC(C)C)nnc2n1CCOC2 C(=O)(CCC(C)(C)N(C)C)NCc1c(C(=O)NC(CC)C2CCC2)scc1 C=CC(C)(CC)C(=O)NCCCC1(CNC(c2cc(C(C)C)sn2)=O)CCCC1 Cc1nn(CC(=O)NCCCNC(C2(C)CC(F)C2)=O)c(C)c1C N1(C(C(CSC)C)=O)CCN(C2CCCN(C(=O)C(C)C(C)C)C2)CC1 C(=O)(C(F)C(F)(F)F)N(C)CC1CCCN(C(C(C)(C)NC(=O)OC)=O)C1 C1(C(C)C)C(=O)N1.C1(C(CNC(C)=O)(C)C)CCCN1C(C1CC1C(C)O)=O C1(C(=O)NC(C)CF)CC2CC1CN(C(c1cc(O)n(C)n1)=O)C2 C1(NC(C2CC(C)(F)C2)=O)CN(C(c2ccc(NC(N)=O)c(Cl)c2)=O)CC1(C)C N1(C(CN(C)CC)=O)CCC(F)(CNC(c2cc(C)ccc2F)=O)CC1 N1(C(CONC(C(CSC)C)=O)=O)CCCC2(CCCC2)C1 C1(NC(c2cc(C)c(O)nn2)=O)(CNC(C2CC(C)CO2)=O)CCC(C)(C)CC1 CCCC(O)CC(=O)N(C1CCN(C(=O)CCCOC(C)=O)C1)CC1CC1 c1(OC)ccc2c(c1)OCC(C(=O)NCC1(NC(=O)C(C)=C3CC3)CCOC1)C2 CCCC(CCCC(=O)OC)NC(=O)CC(CC)C(C)(C)C N1(C(CNC(=O)CCc2nc[nH]n2)=O)CCC(C2CCCC2)C1 C1(C(=O)NCCCN(C(=O)CCCCNC(N)=O)CCC)C(C)(C)C1(F)F C1(CCCC)CCCN(C(C2CC23CC(NC(C24CCN(CC2)C4)=O)C3)=O)C1 C12CC3CN(CC13)C1CC(C1)C(=O)NC2.c1(C(=O)O)cn(CC)nn1.C1(O)CCCC1 N1(C(c2[nH]cc(C)c2C)=O)CC(C2CC2)(C(=O)NCCC(C)(O)C(C)C)C1 C1(C(=O)NCCC2CN(C(c3c(C)ccs3)=O)CC(C)O2)Cc2ccccc2C1 c1(C(C)(C)C)c[nH]c(C(=O)NCC2CCCN2C(=O)CCCn2cccn2)c1 C1(C)(CNc2ccc(C(=O)NCC(=O)NC)cc2)CS(=O)(=O)CCO1 c1(CC(C(=O)NC(C2CC(OC)C2)C=C)NC(=O)CN)ccc(Cl)cc1Cl C(=O)(C1=CC2CCCCCC12)NC1CN(C(C2(C)CC2Br)=O)CC12CCC2 C1(C(N(C2CCCC(NC(=O)C(C)(C)CC3CC3)C2)C)=O)C2(CCC2)C12CCC2 Cc1[nH]nc2c1CN(C(C1CC1NC(c1c(F)cc(Cl)cc1Br)=O)=O)CC2 Cc1ccncc1CC(N1CCOC(CCCNC(C2CCCSC2)=O)C1)=O C(C)(C(C(=O)N1CCC1C(N)=O)NC(=O)C(C)=C(C)C)OC C(C)(C)(CC(=O)N1CCCC(CCC(=O)NCC2([Si](C)(C)C)CC2)C1)OC C1(NC(=O)NC2(CC=C(C)CN3CCOCC3)CCC2)CCCC2(CC2)C1 C1(C(N2CC(C(N)=O)(CNC(=O)CCn3cc(Cl)cn3)C2)=O)CC2CC1CC2O Cc1ccc2c(c1)C(C(=O)NCCC1CCCN(C(c3ccoc3)=O)C1)C2 c1(C(N2CC(CCC=C)(C(=O)N)C2)=O)cc2ccccc2[nH]1.C1(COC=C)CC1Cl c1(NC(C23CN(C(CCC(C)(C)C)=O)C(C2)CO3)=O)cc2n(n1)CCCO2 N1(Cc2cc(Br)c(-n3ccnc3)cc2)CC=CCC2(CCOCC2)C1 C1(CC(N2CCCC(C(C)NC(COCCC#C)=O)C2)=O)CC2CCC1CC2 c1(C(=O)NC2CN(C(C3C(C)C3(F)F)=O)CC(O)CC2)ccc2[nH]ccc2c1F C1(C(C)NC(C2(C)COC2)=O)CCCN(C(C2(C)CC2(F)F)=O)C1 Cc1nccnc1C(=O)NC(C)(C)C(=O)N(C)CC1CCCC2CC12 CCCCC(=O)C(=O)N1CCCC(N(C(=O)Cc2[nH]cnc2C)CC)C1 C(=O)(CCC(=O)CC)N1CC(C=C)(CC(=O)N(C(C)CN(C)C)C)C1 c1(N(CCc2ccc(OC)cc2)C)cc[nH]c(=NCCC2CCS(=O)(=O)CC2)n1 C1(CC)CN(C(=O)C(c2cscn2)N(C)C)CCC1NC(c1ncc[nH]1)=O C1(NC(c2cnoc2)=O)CCSC12CN(C(c1c(F)ccc(F)c1Cl)=O)C2 C1(C(=O)NC(CCOC)CNC(=O)CCNS(C)(=O)=O)CC1C1CCCCC1 c1(C(=O)NC2CCC(NC(C3CCS3(=O)=O)=O)C2)nc[nH]c2nccc1-2 c1(C(C)C(=O)NCC2CC(c3nn[nH]n3)NC2=O)c[nH]c2ccccc12 N1(C(CCC(CC)C)=O)Cc2[nH]nc(C(=O)N(C)CCN3CCOC3=O)c2C1 C(N=c1[nH]cc([N+](=O)[O-])cc1CO)C1(NC(c2cc(Cl)c(Cl)[nH]2)=O)CCCC1 C1(CNC(CCCN(C)C)=O)C2CCC(C2)N1C(=O)CC1OCCCC1(C)C CC(C)CC(CNC(=O)CN1CCCC1C)C(=O)N(C(C)CC1CC1)C c1(-c2n(C(C)C(F)(F)F)nc(CSC)n2)ccc(Cl)c2ncccc12 c1(C(CNC(C2CC2(F)F)=O)NC(c2ccncn2)=O)cccc(Cl)c1 C(=O)(CCCCCC(C)O)NC(CCCC)CC(=O)NC12CC(CO)(C1)C2 C=CC(F)(F)C(=O)NCC(C)(C)NC(c1oc(CC2CC2)nc1C)=O O=C(NNC(=O)C1CCCOC1)c1csc(-c2ccc(Cl)cc2)n1 c1(C2C(NC(C3CN(Cc4ccccc4)C3)=O)CC2)ccc(Cl)c(Cl)c1 C1(CNC(CC2OCC(C)(C)C2)=O)(CO)CCN(C(=O)COCCO)CC1 C1(NC(c2ccc(C(C)(C)C)[nH]2)=O)CCC2(CC1)CN(C(=O)C(C)(C)O)C2 Cc1c(C(N2CCC(C(N3CCS(=O)CC3)=O)C2)=O)cccc1C1CC1 c1(C(N2CCCC(C(C)NC(c3cccnc3F)=O)C2)=O)cccc(O)c1Cl C(CC(=O)N1CCC1C(=O)NCC1(CC(=O)OC)CCC1)OC.C(C)(=O)OC Cc1nc2cccc(C(N3C4CCC3C(CNC(=O)C(C)O)C4)=O)c2[nH]1 C1(C(N2CCC(C)(NC(=O)CC3CC4CCC3O4)CC2)=O)CCc2nncn2C1 N1(C(c2nc(OCC)oc2)=O)CCC2(CC2C(N2CC(O)CC2(C)CO)=O)C1 N1(C(c2c(C)cc(O)nn2)=O)CCCC2CN(C(c3cn(C)cn3)=O)CC12 c1(OC)cc(C(=O)NCCOC2CCN(C(=O)C(c3cnn(C)c3)O)C2)ccn1 N12CCN(C(C)C1=O)CCC2.C1(OCC)(CN(C)SC2CC2)CCSCC1 c1(C(N2CC(C)N(C(=O)CC3CCC(=O)NC3)CC2)=O)noc2c1CCCCC2 c1(C(N2CCC(CNC(C(C)(O)C3CC3)=O)CC2)=O)nc(C(F)(F)F)ccc1F N1(C(CCC=CC)=O)CCC(N(C(=O)C(C=C)CC)C)CC1 C1(C(=O)NCC2N(C(c3nc(C)c(C)s3)=O)CCC2C)CCC2(CC1)CC2 C1(CNC(CCc2cc(C)n(C)n2)=O)CC(C)N(C(c2cccc(=S)n2O)=O)C1 CC1CC(C)(C)c2cccc(NC(=O)NCC3CCC4(CC4)C3)c21 N1(C(C(=Cc2ccccc2)CC)=O)CCC(C2CC2)(NC(=O)CCC=C(C)C)C1 c1(C(N2C(C(C)C)CN(C(=O)C(F)C3CCCC3)CC2)=O)cc(O)cc(C#N)c1 C1(CNC(C2(c3cccs3)CCCC2)=O)CCCN1C(=O)CN1CC2CC2C1 C1(C)(OC)CC(NC(c2cc(CNC(=O)C(C)NC=O)on2)=O)C1(C)C C=CCC(CC(F)F)C(=O)N(CC(C)CNC(=O)C(C)C1CCCC1)C C12(CNC(=O)Cc3cncs3)CC1CN(C(C1COCCO1)=O)C2 N1(C(c2cc(-c3cccs3)on2)=O)CCC(COC)C1.C12(CC1)C(C)NC2=O.CN n1(CC(C)C)ncc2cc(C(=O)NC(C)CCNC(=O)Cc3cccs3)cnc12 C1CC(CNC2C(CNC(=NCC3CC3)NC3CC3)C2)OC2(CCC2)C1 N1(C(C(CCN(C)C)O)=O)CCC(NC(c2csc(CO)n2)=O)C(F)C1 Nc1cc(F)c(C(=O)NC2CC2CNC(c2ccc3c(n2)CCC3)=O)cc1Cl c1(CC(=O)NCC(CO)NC(=O)COC2CC=CC2)cccc(CC(F)(F)F)c1 C12(C(=O)NCC3(NC(c4cc(CC)ncn4)=O)CC3)CCCC1C2(F)F C(CCOC(C)CCC(=O)N(C)C)(C(=O)N=c1ccn(C(C)C)[nH]1)NC(C)=O C1(C(N(C2(CN(C)C)CC2)C)=O)CCC2(CC2)N1C(C1CCS1(=O)=O)=O C12(C(=O)NC(CCC)CCC)CCCC1CN(C(C1CC3(CC3)CO1)=O)C2 Cn1cnc2ncnc(N3CC(C(=O)Nc4cc(Cl)cc(Br)n4)CC(F)C3)c12 N1(C(C(OC)OC)=O)CCC(N2CCN(C(C)=O)CC2)CC1 N1(C(C2(CC)CCC2)=O)CCCC2(NC(=O)CC3CCCOCC3)CC2C1 c1(OC)ccc(OC)c(C2CCC(CNC(=O)N(c3cc(C)cc(C)n3)C3CC3)C2)c1 c1(C(N2CC3CCCC(NC(C45CC(C)(C4)C5)=O)C3C2)=O)ccc2cccnc2c1 C(CCC(=O)NCC1(F)CC(CNC(C2CCCS2)=O)C1)=CCC=C c1(CC(N2C(CNC(C(Br)=C(C)C)=O)COCC2)=O)cc(Cl)cnc1C N1(C(C2CCCC2F)=O)CC2(C(=O)NC3CCc4c[nH]nc4C3)CCC1CC2 C1(NC(CC(CC)(C)C)=O)CCC12CCCN(C(=O)C=CCOCCOC)C2 CC(C)(C)C(=O)CCc1cn(CCCC(=O)NCc2nc(O)[nH]c(=O)n2)nn1 C1(NC(c2ccsc2)=O)CC(F)CN(C(c2cccnc2S)=O)C1 n1(CC)nnc2c1C(C(=O)N=c1cc(C)n(Cc3ccccn3)[nH]1)CNC2 C1CCCN(C(=O)COC)C1.C1(C(=O)NN(C)CCOCCO)CCCO1 c1(C(=O)OC)ccc(C(=O)NC(CNC(=O)CN(C)C(C)C)CO)nc1 C1(CC(=O)NCC2CCN(C(c3cc(-c4ccc(Cl)s4)c[nH]3)=O)C2)COC(=O)C1 c1(C(=O)NCC2C3CN(C(C4C(c5n(C)ncc5)C4)=O)CC32)ccc(O)c(N)c1 c1(C(N2C(CC)C(NC(=O)C=CC3CCOC3)CC2)=O)cc(Cl)ccc1N c1(C(N2CCCC(CNC(=O)Cn3cncn3)C2)=O)n[nH]c2c1CCCCC2 CCCCCC(C)(CC)C(=O)NC1CC2(CCN(c3nnc(C(C)C)o3)CC2)C1 CC1CCc2sc(C(=O)NCCNC(c3cc(C(F)(F)F)no3)=O)cc2C1 Cn1cc(C(=O)NCC2CCN2C(C2CC2c2ccccc2)=O)c(Br)n1 C1(c2nc(Cc3n(C)ccc3)[nH]n2)CCN(C(=O)N(CCO)C(N)=O)CC1 C1(CNC(c2ncn(CC)n2)=O)CNC(=O)CO1.C12(CC1)C(=O)NC2 C1(c2n(CCN(c3ccc(C(N)=O)cc3)C3CC3)nnn2)(OC)CCN2CCCC12 c1(C(c2n(C(CC)C)nnn2)NCCCn2cc(CO)nn2)cncc(Cl)c1 C1(CCNC(c2cnc(C)o2)=O)COCCN1C(=O)C(c1nc(C)cs1)C Cc1cc(C(=O)NC2CC(O)CN(C(C3(F)C(C)(C)C3(C)C)=O)C2)c(F)cc1F C(=O)(CC(O)CC(C)(C)C)NCCOC(CNC(c1cccc(C)n1)=O)(C)C N1(C(c2c(C)ccs2)=O)CC2CCC(NC(=O)Cc3cc(O)nc(O)n3)(C2)C1 c1(Oc2cn(NC(CCNC(N)=O)=O)nc2)cc(I)cc(I)c1 C1(C(=O)Nc2c(C)ccnc2)CC2CN(C(C3(C)C=CCC3)=O)CC2C1 C1(CC(=O)NCC2CCN(C(c3n(C)ccn3)=O)C2)Cc2ccc(Cl)cc2C1=O C1(CNC(C(C)SC)=O)CCC(C)(C)CN1C(c1cnn2ccccc12)=O c1(CC(=O)NC(CNC(c2c(OC)ccs2)=O)CO)ccccc1N1CCCC1 c1(C(N2C(C(C)NC(c3occc3F)=O)CCCC2)=O)ccc(N)c(Cl)c1 C(=O)(C1CCCn2cnnc21)NC(CC1CN(C(C=C(C)C(C)C)=O)C1)C N1(C(CN(C2CC2)CC)=O)CCC(C)C1CNC(C1(F)CCCCC1)=O C(C)(C)(C(=O)NCC(C1(O)CN(C(=O)CSc2ccccc2)C1)(C)C)OC(C)=O N1(C(Cc2c(C)nn(C)c2)=O)CC2CCCC2(NC(C2CC(=O)NC(=O)N2)=O)C1 c1(C(N2CCC(CNC(C(C)n3cccn3)=O)C2)=O)cccc(I)c1 Cc1sc(Br)nc1S(=O)(=O)NC1CCNC12CCC2 c1(N(C(C2CCC(NC(CC=C)=O)CC2)=O)C(C)C)c(O)cccc1C#N C1(C(N(CC(C)NC(=O)C(c2cncnc2)C)CC)=O)(CC)CCCCC1 c1(C(C(=O)NCC2CC(NC(C(C)CO)=O)C2)(F)F)ccc(Br)cc1 CS(C)(=O)=Nc1ccnc(C(N2CC3CC3(CNC(=O)CCOC3CC3)C2)=O)c1 c1(CC(=O)NCC(C)CN(C)C(C2(F)C3CCCC23)=O)ccccc1CC#N c1(CC(=O)NC2(C)CCN(C(c3c(C)oc(CO)c3)=O)C2)cc(F)cc(F)c1 c1(NC(C2N(Cc3cn(CCC)nc3)CC2)=O)ccc(Cl)c(O)c1 C1(NC(CN(C)Cc2cccs2)=O)C2CC1N(C(=O)CCc1nccs1)C2 C=CCC(CNC(C1(C#N)CC1)=O)NC(=O)C(C)c1ccco1 Cc1nnc(C(=O)NCC2COC(CNC(=O)C(c3cccn3C)=O)C2)s1 Cc1c(Cl)ccnc1C(=O)NCC(C1CCCC1)NC(c1cccn1C(C)C)=O CC1c2ccccc2OC1CC(=O)NC(C)CNC(c1c(F)cc(Cl)cc1F)=O c1(N2CC3C(N(C)C)C3C2)nc(C)cc(=NC(CCCN(C)C)c2ccccc2)[nH]1 c1(C(=O)NC(CNC(CC(C=C)C)=O)CC)cc(C#N)c2n1CCCC2 N1(C(Cn2c(C)cc(C)n2)=O)CCCCC(C(N2CC3CC2CC3O)=O)C1 Cn1nc(Cl)c(C(N2CCC(NC(=O)C=CC3CCCO3)CC2)=O)c1Cl c1(OC)ccc(C(=O)NC23CC(CNC(=O)Cn4nc(C)cc4C)(C2)C3)cc1C C(C)(C)(CCC(=O)OC)NC(=O)NC1CN(C(CC)CC)C(=O)C1 N1(C(c2cc(C(C)C)no2)=O)CC(NC(c2cnn(C(C)(C)C)c2)=O)CC1(C)C C(=O)(CCS(N)(=O)=O)NC(CC(C)C)CNC(=O)CC(O)CC1CC1 C1(OC)CC(CCNC(C2CC3CC3C2)=O)N(C(=O)Cc2csc(C(C)=O)c2)C1 C(CCCC(=O)NCCC1CN(C(=O)CO)C1)n1c(C)ncc1 Cc1ncccc1CC(=O)NCC=CCNC(=O)COC1CCC1 N1(C(c2c(C)nn(CCO)c2)=O)CCCC(C)(NC(c2ccc[nH]2)=O)C1 c1(C(C)NCC(O)C(O)C(F)(F)CBr)ccc(F)c(F)c1F Nc1ccc(C(O)C(=O)NCCCCNC(=O)COC2CC2)cc1 N1(C(C(=O)NC(C2CCCCO2)CC)=O)CC(CC)CC1C C1(NC(c2ccc(OC)s2)=O)CC2CC(C1)N(C(=O)CCCc1ccccn1)C2 C(CCCOC)(C(=O)N=c1cc(OC)n(C)[nH]1)NC(C(C=C)CC)=O n1(CC(C)C)ccc(C(=O)NC2CCC(CCNC(C3(C4CC4)CC3)=O)C2)n1 C1(NC(C=CC)=O)CN(C(=O)CCc2cc(Cl)cc(Cl)c2)C(C)(COC)C1 c1(C(=O)NC2CCC(NC(C=Cc3nnn(C)n3)=O)CC2)nnc(Cl)cc1N c1(C(C(N2CCC(O)(CN(C(CC=C=C)=O)C)C2)=O)C)cccc([N+](=O)[O-])c1 c1(CC(=O)NC(CNC(c2cn(CC(C)C)nc2)=O)C)cc(O)nnc1O C1(CCC)CC(C(=O)NC2(C)CN(C(=O)Cc3cnccn3)C2)CCO1 N1(C(CN(c2ccc(Cl)cc2)C)=O)CCC(NC(=O)C(C)(F)c2ccccc2)CC1 C12CN(C1)C(=O)C(C)N(C)C(=O)C1(CC1)C2.c1(C(=O)N)ccco1.CC(CN(C)C)O CN=c1[nH]cc(C(N2CC=CC2(C)C(N2CCC(C(=O)OCC)C2C)=O)=O)o1 c1(NC(C2CNCCN2S(=O)(=O)C(F)(F)F)=O)c(Br)cc(F)cc1[N+](=O)[O-] CCCN=c1[nH]c(N(C)CC2CCc3nc(CC)cn3C2)nc2cc(C)ccc12 Cc1cc(C(=O)NCC(=O)NCC2C=CCN2C(C2CC(C#N)C2)=O)c(C)o1 c1(NC)cccc(C(N2CCC(O)C2C(=O)NCCC23CCC(CO2)C3)=O)c1 CC1C(NC(=O)CCCCN(C)C(C)C)CCN1C(C1COC(C)C1)=O N1(CC)CCOCC1CC(=O)NCC(CNC(=O)CCc1ncc(C)[nH]1)CO CCC(CC)C(C(=O)NC(C)(C)CNC(c1cnc[nH]c1=N)=O)OC N1(C(c2c(C)cco2)=O)CCC2(CC1)CCN(C(=O)C(C#N)=CC(C)C)CC2 c1(NC(C(C=C)O)=O)cccc(NC(C2(C(N)=O)CC2)=O)c1C c1(C(=O)OC(C)(C)C)cccc2cncn12.C1CC(=O)N2CC(C2)CCC(=O)N1 Cc1ccc(C)c(C(=O)NCC(CNC(=O)Cc2csc(C)n2)CO)c1 C(N=c1[nH]c(C)ncc1C)C1C(C(F)(F)F)CCN(C(CC(=O)NCC#C)=O)C1 C1(C)(C(N2CCC(N(C(C(C)(C)OC(C)C)=O)CCO)C2)=O)CC2(CCC2)C1 CCCC(C(=O)NC1(C)CN(C(=O)C(C)C2CCOC2)C1)NC(=O)C1CC1 CCC(C)(F)C(=O)NCC(N1CCN(C(=O)CP(C)(C)=O)CC1)COC C1(N(C(c2ccnc(CC(C)C)n2)=O)C)CN(C(=O)CC2CCCO2)CC12CC2 N1(C(c2ccn(CCC)n2)=O)CCCOC(CNC(C2(CC3CC3)CCC2)=O)C1 N1(C(C(C)C#N)=O)CCCC(O)(CN(C)C(c2cccc(F)c2)=O)C1 c1(C(=O)NCC(C)(C2CCC2)NC(c2cnc[nH]2)=O)ccc2n[nH]cc2n1 C(=O)(CCC(C)(C)C(=O)N1CCCC1CNC(c1cnn(CC(F)F)n1)=O)OC c1(CCC(N2CC(O)CC(NC(=O)C(Cl)=CCl)C2)=O)cnc2n1CCCCC2 c1(OCC(=O)NC2C(CNC(c3cc(CC(C)C)on3)=O)CC2)ccc(F)cn1 N1(C(C(c2cccc(C)n2)(F)F)=O)CC2CCN(C(=O)CSC(F)F)CCC2C1 N1(C(C2C(OC)(OC)CC2)=O)CCC(CNC(=O)Cc2cccs2)C(C)C1 C(c1ccc(F)c(F)c1)=CC(=O)OC(c1ncccn1)C C1(CN=[N+]=[N-])CN(C(=O)C(Cc2ccoc2)NC(=O)CCc2ccco2)CCO1 C1(NC(=O)CCOC2CN(C(=O)Cn3ccnc3)C2)CCC2(CC1)CC2 CC1(C)CC(C(=O)NC2(CCC(=O)Nc3ccc(F)cc3)CCC2)=NO1 CCC1=NOC(CC(=O)NC(C(=O)NC(c2cccc(C)c2)C)c2ccco2)C1 c1(CCC(=O)NC(CNC(CCOCCCOC)=O)C)ccc(C(C)(C)C)cc1 CC1CN(C(=O)CCC2CCC(O)CC2)CCN1C(=O)CCc1cccc(O)c1 c1(CC)nn(C)c(C(N2CCCC2CN(C)C(c2nnn3c2CCC3)=O)=O)c1Cl C=CC(C)(CCOC)C(=O)NC1CC2CCC1C(NC(c1cnc(CC)[nH]1)=O)C2 c1(C2C(C(=O)NC(CN(C(=O)CCSC)CC)C)CC2)ccc(F)cc1 Cc1ccc(Cl)c(F)c1C(N1CC(NC(=O)C(C)(C)CO)CC(O)C1)=O C(=O)(C(C#N)(CC)CC)NC1(CNC(C(CCCC)N(C)C)=O)CCC1 c1(CNC(Cc2ncc(-c3c(SC)cccn3)cn2)=O)ccc(O)cc1Br c1(NC2CN(C(c3nnc(C)s3)=O)CC2(C)C)ncnc2c1cnn2C(C)(C)C C(C(C(=O)NCC(=C1CN(C(C2(O)CC2)=O)C1)F)N(C)C)OC C(C(CC(C)C)C(=O)NC1CN(C(c2cc(Cl)c(F)cc2O)=O)CC1OC)OC O=S(=O)(C1CC12CCC2)NC1CCN(Cc2ccc(Cl)cc2)C1=O CC(C)C(C)(CN=c1ccc(-c2ccncc2)n[nH]1)NC(c1csnc1Cl)=O CC1CCCN(C(=O)C(N2CCC(C(=O)NC(=O)CSc3cnn(C)c3)C2)=O)C1 C1(CCCC)(C(=O)NC(C)CC2CN(C(=O)CN3CCCC3CO)C2)CCCC1 C(=O)(C(C)(C)C(=O)N1CC(NC(c2coc(C(C)(C)C)n2)=O)C(F)C1)OC N1(C(C(c2cn(CC)nc2)=O)=O)CCCC(NC(c2cnco2)=O)C1C Cc1nc(C)c(C(=O)NC(c2ccccc2)C(C)Nc2ccnc(CO)n2)[nH]1 Cn1cnn(CC(N2CCSCC2CCNC(=O)CC2CCCCC2O)=O)c1=O c1(CC)ccc(C(N2CC(CNC(=O)CC3CN(C)C3)C(C)(C)C2)=O)c(C)n1 c1(C(=O)NC(c2ccncc2Cl)CN)cnc2c(c1)CNCC2 Cc1cc(Br)ccc1-n1nc(C(C)C)nc1C1C2CC2C2CC12 C1CCCC(=O)N1.C1(NC(c2cc(C(C)=O)sc2)=O)CCCC1(C)CN(C)C C(=O)(C(CO)c1ccccc1)NC(CC)CNC(=O)CCC1(O)CCC1 C(CCC1CC1)(C(=O)NCCSC)NC.CN=[N+]=[N-] N1(C(C(C)O)=O)CC2(CCC2CNC(c2cccc(SCC#N)c2)=O)C1 c1(CCC)nc(C)c(C(=O)NCc2ccc(OC(C)(C)C)nc2)s1 N1(C(Cc2c(C)noc2)=O)CCCC1(C)C(=O)NCCOC1CC1(F)F c1(CC(=O)OC)ccnc(N2CCC(C(C)NC(c3csc(C4CC4)n3)=O)C2)n1 c1(CN(CC(C)C#N)CC)nc(CC(C)(Cc2ccccc2)C2CC2)no1 C#CCCCCC(=O)N1CCC(C)C(CNC(c2cnn(C3CC3)c2)=O)C1 C1(CCNC(Cn2c(C)ncc2)=O)CN(C(=O)C(=O)Nc2ncc[nH]2)CC1C CC1CN(C(=O)COc2c(F)cccc2F)CCC1NC(c1ccnc(O)c1)=O CC1CC(CCNC(=O)CC2CN3CCN2CC3)CCN1C(=O)Cc1cn[nH]c1 c1(C(N2CCN(C(C(COC)COC)=O)CC2CO)=O)cc2ccccc2nn1 Cc1cc(C(=O)NCC(C)(C)C(N2CCN(C)C(C(C)C)C2)=O)cc(C)c1 N1(C(c2cnc(C)nc2)=O)C2CCC1CC(O)(CNC(=O)CCCCF)C2 CC1OC(C)C(C(N2CCC(C(C)NC(c3cccn3C)=O)C2)=O)C1C c1(C(=O)NC23CCCN(c4ncc(Br)cn4)CC2C3)noc2c(F)cccc12 c1(C(=O)NC(C)C)ccc(C2CCC(NC(C3(C(=O)NC)CC(=O)C3)=O)C2)cc1 C(C)(C)(C(=O)NCC1CC1NC(c1[nH]cnc1C)=O)NC(=O)NCC C1(NC(c2n(C=C)ncc2)=O)CN(C(=O)CC=CC=C)CCC12CCC2 C1(NC(COCCC#C)=O)CCCN(C(C2(COC)CC(=C)C2)=O)C1 Cc1cccc(C2=CCN(C(=O)C(N3CCCC4(CNC(=O)C4)C3)=O)CC2)c1C c1(C(N2CC3C(NC(C4CC(SC)C4)=O)(CC3)C2)=O)c(C)cc(C)nc1O C1(CN(C(=O)Cc2cnn(C)c2)C)CCCN(C(=O)C=Cc2ccncn2)C1 C=C(C)CCC(=O)NCCCCC(C)NC(c1ccc(NC(=O)CC)cc1)=O CC1CCCCN1CC(=O)NC1CCC(NC(=O)CCCN2CCCC2)C1 C(CCC1CC1)(C(=O)NC1CCSC1)NC(=O)CNC(=O)C1CC1 Cc1c(C(=O)NC(C)C(C)NC(c2cc(C3CC3)nn2C)=O)sc2ccsc12 c1(CNC(C2CN(C(CN(C(=O)OC)C)=O)C2)=O)csc(=N)[nH]1 C1(CNC(CCC(=C)C)=O)CCN(C(C2(n3cnnn3)CC2)=O)C12CC2 c1(NC2(CC)CC2)ccc2nc(CC)nc(N3CCC(N4CC(C)(C)C4)C3)c2c1 n1(CCC)ccc(C(=O)NC2(CNC(c3sccc3C(F)F)=O)CCOC2)n1 Cc1cc(Cl)ncc1CC(=O)N(C)CC1CN(C(C2(C)CCNC2=O)=O)CCO1 N1(C(C=C(CCC)C)=O)CC(C)N(C(=O)CC2(NC(C)=O)CCCCC2)CC1C N1(C(C(c2nccc(C)c2)(F)F)=O)CCC2CC2(NC(=O)CCCF)CC1 N1(C(C=CC(C)(C)SC)=O)CCC(F)(CNC(C2CCCC3(CC3)C2)=O)CC1 C(=O)(C1CCCc2ccnn21)NCC12OCC(NC(C3CCCO3)=O)C(C1)C2 C1(C(N(C2CCCCC2)CC(=O)OC)=O)CCCC(NC(c2ncsc2CN)=O)C1 c1(C(=O)NC2CCC(CNC(COC(C)C)=O)CC2)c(F)ccc2ccncc12 C(=O)(C(CC(=O)N1CCCN(C(c2csnn2)=O)CC1)C(C)=O)OCC N1(C(c2c(CC)nn(C)c2)C(=O)NC(C)CC)CCC2(CC1)COC(=O)N2 n1(CC=C)ncc2c(O)nc(=NCC(C3CC3)N(C(=O)CCCCOC)C)[nH]c12 C1(CNC(COCCCC)=O)CN(C(c2cc(C)c(O)nn2)=O)CCN1C C(=O)(CC(CC)C(C)(C)C)N1CCC(C(C(=O)N(CCCC#C)CC)C)C1 C1(C(=O)NCC(=C)Br)CN(C)CCN1C(C1CC(C)CO1)=O C1(C(N2CC(NC(C3=C(C)OCCS3)=O)(CO)C2)=O)CCC(S(N)(=O)=O)CC1 N1(C(CC=CC=C)=O)CCN(C(=O)CC2(OC)CC2)C(c2cccc(OC)c2)C1 C1(NC(Cc2onc(C)n2)=O)C2CCC1CN(C(c1cccn3cncc13)=O)C2 c1(C2C(C(=O)NC3(CCNC(CC4CC(=O)C4)=O)CC3)C2)ccncc1F C1(C(=O)NC(c2cccnc2)C(N2CCC(C(=O)OC)C2)=O)CC2(CCC2=O)C1 c1(C(=O)OC(C)C)nnn[nH]1.C1(NC(C2C3COCC23)=O)CCC(O)C1 C(C(=O)N(C(C)CN(C(=O)CN1CC(C)C1)C)C)(C(C)C)OC c1(C(N2CCC(C)C2CNc2ccc(=O)n(O)c2)=O)cnc(C#N)cn1 C1(C(N2CCCC(CC)(NC(=O)CCC(N)=O)C2)=O)CCc2cc(F)ccc2O1 N1(C(C2CC(=C)C2)=O)CCC(C2CC2)C1CNC(=O)CNS(C)(=O)=O Cn1cnnc1CCCC(=O)NC1(C)CC(NC(C2(C)C=CCC2)=O)C1 n1(-c2ccc(-c3onc(C)n3)cc2)cc(N=c2cc[nH]cc2C#N)cn1 C(=O)(CC(O)CC(C)C)N1CCCC(C(C(=O)N(CC#C)CC)C)C1 C1(NC(C2(CC)CCC2)=O)CC2(C1)CC(C(=O)Nc1ccc(Cl)nc1)C2 C1(CC)CN(C(C2CC(F)CN2C(C2CCOC2)=O)=O)CC(=O)N1 CC1CC(=O)NN1S(=O)(=O)CC1CC(=O)CC(=O)C1 CCCCC(O)C(=O)NC1(C2CCCN2c2nnc(C(N)=O)s2)CC1 N(C1CCCc2c1cnn2C(C)C)C(=O)NCC1=C(C)OCCS1 C1(NC(C2(CC)CCCN(C(C3CC3(C)C(F)F)=O)C2)=O)CCCN2CCCC12 C1(CC(=O)N(CCCC(F)F)C)CCCN(C(C2CC(C)(O)C2)=O)CC1 C1(N(C(CC2(OC)CCC2)=O)C)CN(C(c2coc(C(C)(C)C)n2)=O)CC1F C1(NC(Cc2ccc(C)s2)=O)CN(C(c2nc(C(C)(F)F)cs2)=O)CCC1(C)C C1(NC(c2cc(OC)ncc2)=O)CCN(C(=O)C(C)Oc2ccccn2)CC1O N1(C(CC(C)NC(N)=O)=O)CC2CC1C2NC(=O)C(c1ccc(F)cc1)(F)F C12(CCN(C)C1)C(=O)N2.CC(C(=O)NCCSCCO)N1CCCC1 C1(CC)(NC(c2cc(C(F)F)no2)=O)CCCOC1 c1(C(N2CC(C3(NC(c4cc(OC)n[nH]4)=O)CC3)C2)=O)cc(F)c(Cl)cc1F CC(CC(C)(C)C)C(F)C(=O)NC1CCN(C(c2csc(Cl)c2)=O)CC1C(N)=O C(CCCC(=O)N1CC(NC(c2cnn(-c3ccc(Cl)cc3)n2)=O)C(C)C1)OCC O=C(C(O)CC(F)(F)F)NC1COCC1CO.C12(CCCC1)C(=O)N2 N1(CC(=O)NCC(CC(F)(F)F)NC(C(CC)C)=O)CCc2ccccc21 c1(C(=O)NCC(CC)NC(=O)C(C)SC(F)(F)F)nn(CC)nc1C Cc1cc(C(=O)NCCC2COCCN2C(=O)CC(C)F)c(C)n1NC(N)=O CN=C(NCc1cnc(-c2ccco2)s1)NC1CC=CC1 N1(C(C2C(COC)C2)=O)CCC2(C1)CN(C(c1[nH]ccc1-c1ccccc1)=O)C2 N12CCOCCC1C2=O.N1(C(C2N(CC)CC2)=O)CC(C)(C(=O)OC)C1 c1(C(N2CCCCC2CNCc2nc(Cl)cs2)=O)cccc(F)c1Cl N(C)C(=NCCO)NC1CSC1.Cc1csc(C(c2ccccc2)O)n1 N1(C(CCCCCOC)=O)CCCCC(NC(c2cnc(N(C)C)nc2)=O)CC1 C12(CNC(CN(CCC)C)=O)CC(CO1)N(C(=O)C(CO)c1ccccc1)C2 CCCCCC(O)C(C)C(=O)NCC1CC(C)N(C(=O)Cc2cc(C)no2)C1 Cc1cc(C(=O)N(C)CC2CCCC(NC(c3nocc3Cl)=O)C2)cc(C)c1 c12cccc(c1)CNC2=O.C1(CNC(C2C(C)=CCC=C2)=O)CC2C=CC1C2 c1(CN2CC3(CC(CC(=O)Nc4ccc(Cl)nc4)C3)C2)cc2c(Br)cccc2s1 N1(C(c2c(O)ncc(C(C)C)c2)=O)CCC(NC(=O)C2=CCSC2)C(CO)CC1 c1(CC(=O)N(CC(C)(C)NC(=O)C=CC2CCC2)C)cc(F)cc(Br)c1 N1(C(C)=O)CC(SC(C)C(=O)NC2CC2)C(F)(F)C1.C12(CCC1)C(=O)N2 Cc1cccc(CNC(C2CC=CC(NC(=O)C=CCO)C2)=O)c1F C(C(CC)(CC)C(F)(F)F)N(CCCC)C=O.C=O CC(c1cccc(Cl)c1)=CC(=O)NC1CCN(C(=O)Cc2nonc2C)CC1C C1(C(N(CCCC(=O)OC)C)=O)CN(C(=O)Cc2ccoc2C)CC1C(C)C c1(C(=O)NCC(C)N(C)Cc2ncn(-c3ccccc3)n2)cncc(F)c1 C(=O)(CC(C)(C)c1cccs1)N1CC(CC(C)NC(C2(C3CCCO3)CC2)=O)C1 C(C(C)CC(=O)NC1(CC2CCC2)CC1)NC(C1(COC)CC=CC1)=O c1(C(c2nnnn2C(C2CCCCC2)C)NC2CC(OCC)C2)cccc(Br)c1 CC(C)(C)C(=O)C(=O)N1CC(CNC(C2(C)CC3CC3C2)=O)C(F)(F)C1 C(=O)(C1=NOC2(CCN(C(c3cc4c(C)cccc4o3)=O)C2)C1)N(CCO)CC CC1CN(C(=O)CCC2CC2)CCCN1C(c1cccc(OCC(F)F)n1)=O C1(C(=O)NCC23CCC(NC(CCC=C)=O)(C2)CO3)CCC([N+](=O)[O-])CC1 c1(CC)cc(NC(=O)C(CC(C)C)ONC(=O)C2CCO2)cc(C)c1 c1(OC)ccc(C(F)(F)F)c(C(F)(F)F)c1.c12cnc(o1)CC1CCN(C1)CC2 N1(C(c2cc(C(C)C)n(C)n2)=O)CCC(NC(C2OCC2(C)C)=O)C(O)C1 C1(CC(=O)NC2(C3N(C(CCCC=C)=O)CCC3)CC2)OCCCC1(C)C c1(C(N2CCC(CCNC(=O)CNC(=O)C3CC3)C2)=O)csc2nccn12 N1(C(C(C)n2ccnc2)=O)CC2CC(NC(=O)Nc3c(F)cccc3F)CC1C2 C1(c2cn(CCC(=O)OCC)nn2)C(C)CCCN1C(C1(F)CC(CN)C1)=O c1(C(=O)NCC=CCC(=O)NCCCc2ccncc2)ccc(O)cc1F c1(CC(=O)N(C2CC2)CC2(C(=O)NC(C(N)=O)C3CCCC3)CCC2)cccnc1O C12(C(=O)OC)CC(N=[N+]=[N-])C1C2.c1(NC)ccc(-c2nc(C(=O)NCCOC)cs2)cc1 C1(NC(c2nc(Cl)cs2)=O)CCN(C(=O)Cc2cc(Br)ccc2Cl)CC1F CC1C(NC(c2cc(CO)[nH]n2)=O)CCCN1C(c1cc(Cl)ncc1N)=O c1(OC)ccc(F)c(NCC2CCC(F)CN2C(=O)OC(C)(C)C)c1F c1(C(=O)NCC2(NC(c3cc(Cl)no3)=O)CCCC2)c(F)ccc2[nH]ccc12 c1(CC)ccc(C(=O)NC2CCCC2(C)NC(c2n[nH]cc2C)=O)nc1 C1(NC(=O)Cc2cc[nH]n2)CC(CNC(=O)CSCC2CCCO2)CC1O CC(C)(C)CCCNC(C1(C(F)F)CCCO1)=O c1(CN2CC(CNC(C3(N(C)C)CCOCC3)=O)OCC2)ccc(O)c(F)c1F N1(C(CCCC#C)=O)CCN(C(c2nnsc2SC)=O)CC1CS(C)(=O)=O c1(CNC2(C(N)=O)CCCCC2)cc2c(nc1Cl)CCCC2 OCC1=CCN(c2nnc(C3CCC(=O)NC3)n2CC2CCC=CO2)CC1 CC1(C)CCC(C(N2CCS(=O)C2)=O)CN1C(=O)C(O)CC(F)(F)F c1(C(N2C(CNC(C3CC=CCO3)=O)CCCC2)=O)onc2c1CCCC2 CC1ON=C(C(=O)NCc2cccc(NC(=O)C(C)(C)CN(C)C)c2)C1C CC(C)CC(C)(C)CNC(C1CCC(CNC(C2CCCC(C#N)C2)=O)CC1)=O Cn1cc(CC(N2CCC(C(=O)N=c3[nH][nH]cc3Br)C2)=O)c2ccccc12 N1(C(COC)=O)CCC2(CC1)OCCCC2NC(C1CCNC(=O)C1)=O c1(SC)cc(C(=O)NCCC2CN(C(=O)C(F)CC3CCOC3)C2)ccn1 C(=O)(C(CCOCCO)C(c1scnc1C)C)Nc1ccsn1.C1(=O)CO1 c1(OC)cc(C)c(C(=O)NC2CN(C(=O)CNS(C)(=O)=O)C(C)(C)C2)c(C)c1 CCCCCCCCCCCC(=O)N(C1CN(C(c2ccoc2)=O)CC1F)C C1(CNC(CCCC)=O)N(C(C2CCCCC2C(N)=O)=O)CCCC1(C)C c1(C(N(C)CC)=O)ccc(CSC(C)C)cc1.c1(S)ccc(C(=O)N)cc1 C(=O)(C#CC1CCC1)N1CC(NCc2cccc(OC)c2)C(C)C1 C#Cc1ccc(CC(=O)NC2CC(NCc3ccc(OCC)cc3)C2)cc1 C1(O)(C(C)N(C(C2CC23CCCC3)=O)C2CC2)CCN(C(C2CCC(C)O2)=O)CC1 C1(CC(=O)NCC23CC(NC(C(C)CC4CCOC4)=O)(C2)C3)CCCC1(F)F N1(CCN(C)C(C2CCSC2)=O)CCN(C(C2CC3C=CC2C3)=O)CC1 CC1=C(C(=O)NCC2COCCN2C(C2CC(F)(F)CS2)=O)CCC(C)(C)C1 c1(NC(C2N(C(Cc3cnc(C)s3)=O)CC(F)C2)=O)cc(O)cc(Br)c1 C1(C)(CNC(C2C(CCC)C2)=O)CCN(C(c2cc(C(C)=O)c(C)o2)=O)C1 C=CCC(C)(C)COCCNC(OC(CC)CC)=S c1(C(N2CCC(CC=C)(NC(=O)CCC(C)C)C2)=O)c[nH]c2ccncc12 C(=O)(C(C(C)(C)C)N(C)C)NCC(C1CCC1)NC(c1ccc(C)cn1)=O C1(C2N(C(c3n(CCOC)ncc3)=O)CCC2)CCN(C(C2(OC)CC2)=O)CC1 C1(NC(COCC)=O)C2CC1CN(C(=O)CC1C(C)(C)C1(C)C)C2 CCCS(=O)(=O)CC(=O)N1CCCC(F)(CNC(C2(N(C)C)CC2)=O)CC1 N1(C(c2ccn(C)c2)=O)CCCCC1C1CCCN1C(c1cc(Cl)n(C)n1)=O N1(C(=O)CCCCn2cc(C(O)C3CC3)nn2)CCC2CCCC(C2)C1 c1(C(=O)NC2C3CN(C(C(C)N(C)C)=O)CC2C3)ccc2ccccc2c1 C1(CC)CN(C(=O)COc2cc(C)on2)CCC1NC(=O)CCOCC1CCCO1.O C1(CC(=O)NCCN(C(=O)C#CC(=O)N(C)C)CCCCCC)CCC(F)(F)C1 N1(C(c2c(NC(C3CC(=C)C3)=O)cnc(F)c2)=O)CCc2ccccc2C1C c1(C(N2CCC(F)(CF)CC2)=O)ccc2nc(CNc3nccc(Br)n3)[nH]c2c1 c1(N2CC3C(CO)(C3)C2)ccnc2cc(Br)nn12.C(=O)NCC N=c1ccc(C(N2CCC(F)(CNC(c3nn[nH]c3Cl)=O)C2)=O)c[nH]1 C1(OC)CCC2(C(N3CC(O)(C(C)NC(C4CCCN4S(C)(=O)=O)=O)C3)=O)CC12 C1(NC(CC=CC(C)(C)C)=O)COCCN(C(C2CC3CCC2O3)=O)C1 N1(CCNC(C2(NC(C(C)CC3CC3)=O)CC(O)C2)=O)CC2CCC1C2 C#CCC(C)(CNC(=O)C(C(C)OC)NC(=O)C=Cc1ccccc1)CO C(=O)(C(O)CC(N)=O)NCC(CCC)NC(=O)C(CC(C)C)N(C)C c1(C(N(CCN(C(=O)C(C)C2CCC2)CC)CC)=O)ccc2nn[nH]c2n1 N1(C(C2N(CC)CC2)=O)CCC(C)C1CNC(=O)C(c1ccc(F)cc1)(F)F C1(C(=O)NC2(CC=CC(=O)NCc3cc(CC)[nH]n3)CCC2)CCCCC1(C)C C1(CN(C(=O)CC2CCC2)C)CN(C(c2ccnc(O)c2)=O)CCO1 c1(CC)occ(C(F)(F)F)c1C(=O)NCC1CCCC1NC(=O)C(C1CC1)OC CCCCS(=O)(=O)CC(=O)NC(CNC(=O)CCCO)C1CCC1.SCC Cc1nc(C(N2CC(O)CC2CC(=O)NC(c2ccc(O)cc2)C)=O)sc1C C(CCC(N)=O)(C(=O)N1CC(NC(=O)C=Cc2ncc[nH]2)CCC1C)NC(C)=O C1(C(=O)NCC(c2ccncc2)N(CC)CC)CCC(C)(CC)CC1 C1(F)(C(=O)Nc2cc(C)sc2)CCN(C(c2cc(CO)ccn2)=O)CC1 N1(C(C2CCC(Cn3cc(CCCCC)nn3)C2)=O)CCC(O)C(O)C1 C1(NC(C(C)=C(CC)C)=O)CCN(C(c2ccc(Cl)c(O)c2)=O)C(C)C1 c1(CC)nc2ccccn2c1C(N1CC2CC(NC(C3CCOC3)=O)C1C2)=O c1(C(=O)NC2CC3CN(C(CCOC)=O)C(C2)C3)cnc([N+](=O)[O-])cc1C c1(Cn2cc(C3(C)N(C(C(C)OC)=O)CCC3)nn2)ccc(Cl)cc1Cl C1(C(N2C(CC)COCC2)=O)CC(O)CCN1C(c1cnc(SC)nc1)=O C(=O)(C1Cc2ccc(F)cc21)NCC1(F)CC(NC(C(CC)(F)F)=O)C1 C1(CN(C(C(C)C2CCCC2)=O)C)CCN(C(C23CC(C(F)F)(CO2)C3)=O)CC1 C=CCC(C)(CNC(C1CCC(O)CN1C(=O)CCCN1CCCC1)=O)CO C(C)(CC(=O)NCC12CC(CN1C(=O)CC1=CCCCC1)C2)(C(F)(F)F)N(C)C C(=O)(C#CC(C)(C)CNC(=O)CC(O)CN(C)C)NC1CCC(CC(C)C)C1 N1(C(C2(C#N)C(C)(C)C2)=O)CCC(NC(=O)CCNC(=O)CO)C2(CCC2)C1 Cc1c(NC(=O)COc2cc(Br)cnc2Cl)ccc(Br)c1Br N1(C(C(CCSC)(C)C)=O)CCS(=O)(=O)C(CCNC(c2cscc2C)=O)C1 C1(C(N(CC(C)O)CCNC(=O)C(Cl)=CCl)=O)CCCC2(CCC2)O1 c1(OC)ccc(SCC(=O)NC2CN(C(=O)Cc3cc(Cl)n(C)n3)CC2O)cc1 C1(C(C)C)CN(C(=O)C(=CC2CCCCC2)F)CCN1C(=O)C(F)=C1CCC1 C1(C(=O)NCCCCC=C)CN(C(=O)C(C(C)CC)N(C)C)CCC1(C)C N1(C(C(n2cc(CN(C)C(c3cccnc3CO)=O)nn2)C)=O)CCP(C)(=O)CC1 C1(CNC(CCCOCC=C)=O)CCC2CN(C(c3ccnnc3O)=O)CC12 Cc1ccnc(NC(C23C4C5C2C2C3C4C52C(C)C)=O)c1C Cc1c(-n2cc(C3(C)CN(C(=O)C(C)(C)O)C3)nn2)cccc1Cl C1(NC(C(CNC(c2c(C)snc2)=O)N(C)C)=O)CCCC1(F)F N1(C(CC(C(=O)OC)C)=O)CCN(C(=O)C=Cc2cn(C)cn2)CC(C)(F)C1 N1(C(Cn2nnc(C)n2)=O)CC2(C1)CN(C(c1cc(Cl)n(C)n1)=O)C2 c1(N(C)C)cc(C(=O)NC2CN(C(c3ncn(C)n3)=O)CC2CC2CC2)ccn1 C1(NC(C2CCCCCC2CC(F)(F)F)=O)CC2(CCN(CC3CCC3)CC2)C1 N1(C(C2C(CC)N(C(=O)CCC(=O)C3CC3)CCC2)=O)CCN2C(=O)NCC2C1 CC1(C)CC(C(N2CCC3(NC(=O)CCOCC4CC4)CCCC23)=O)CNC1=O C#CC(C)(C)C(=O)NC(C1CCCCC1)C(C)Nc1nccc(C)n1 c1(C(C)C(=O)N2CCCC2)ccc(S(C)(=O)=O)cc1.c12cn(cn1)CC(=O)N2 C(CNC(=O)CCc1ccc(CO)cc1)(C(C)C(C)C)NC(C)=O c1(CC(=O)NC(CNC(C(CC=CC)C)=O)C(C)C)ccc2cnccc2c1 C(CCC(=O)NC(CNC(=O)C=CCF)Cc1ccccc1)N(C)C c1(-c2occ(C(N(C(C)C)CCNC(=O)C(C)(C)C)=O)n2)cccc(Cl)c1 c1(C(N2C(C)CN(C(c3ccoc3Cl)=O)CC2)=O)cccc2c1nnn2C c1(C(N(CC(CNC(c2cn(CC=C)nc2)=O)C)C)=O)c(C)nn(CCO)c1C c1(CC(=O)NC(C)CCN(C)C(C2C3COCC23)=O)cccc(N(C)C)c1 N#Cc1c(CNC2CC(F)(CNC(C3CCC4CC34)=O)C2)cccc1F Cc1coc(C)c1C=CC(=O)NC1CN(C(c2ccc(C3CC3)nn2)=O)C1 Cc1sc(C(=O)NC2CN(C(=O)Cn3cccc3)C(C)(C)C2)c(Br)c1C C=CC(C)CC(=O)N(C1CCCCCC1)CCNC(c1ccc(Cl)s1)=O C1(CCNC(C=C2CCN(C)C2)=O)CN(C(C23CC(C2)C(C(=O)O)O3)=O)CCO1 C(=O)(C1CCc2cccc(F)c21)NC(CCCC)CNC(=O)C1=CC(C)(C)C1 c1(NC(N2CCC(C)C2C(=O)O)=O)ccc2c(c1)CCCN2 CC(C)CCC(=O)C(=O)N1C2CCCC1CN(C1CCNC1=O)C2 Cc1cc(CC(=O)NC2CCN(C(C3CCC(F)(F)C3)=O)C2)nn1-c1ccccc1 N1(C(C2CC3(CC(=C)C3)C2)=O)CC(NC(C2(C)CCCCO2)=O)CC2(CCC2)C1 C=CC(F)(F)C(=O)N(CCCC(=O)NC1CC(O)C1O)C C1(OC)CCOCC1NC(C1(NC(=O)Cc2nccn2C)CC1)=O c1(C(=O)NCC23CC2CN(C(c2ccsc2Cl)=O)C3)cn2ccccc2n1 CCC(C)(C)CNC(=O)CC1(NC(=O)Cc2ccoc2)CCC1 N(C(=NCCN1CCOCC1)N(C)C)C(c1cccc(C#C)c1)C1CC1 C(=O)(C(F)C(C)CNC(=O)Cn1ccccc1=O)NCC(C)C1CC1 c1(NC(C(CCCC#C)N(C)C)=O)ccc2c(c1)OCCO2 CCC1=C(C(=O)N2CCN(C(=O)C=Cc3ncc[nH]3)C3CC23)CCCO1 C1(NC(C(CC)n2nccc2C)=O)CCN(C(c2cnoc2C)=O)CC1F c1(C(=O)NC2CC(N(C)C(C3CC4C=CC3C4)=O)C2)ncnc2c1ccn2C c1(CCNC(=O)Nc2occ(C)n2)ccc2c(c1)C(C)C(C)O2 Cc1nn(C)c(Cl)c1C(=O)NC1CCCN(C(c2cnnc(O)c2)=O)C1C CC1(C#CC(=O)NCC2C3CN(C(=O)CCOC4CCOC4)CC23)CC1 c1(C(=O)NCC(CNC(CN(CCCCCC)C)=O)F)cc(C)ccn1 c1(C(C)C(=O)NC2CC2CNC(c2ccoc2Br)=O)cnn(C)c1C(F)F c1(C(=O)Nc2cccc(NC(C3CC3F)=O)c2)ccc2c(c1)CCCO2 N1(C(C=C(CC)CC)=O)CSCC1C(=O)NC(C1CCCC1)CNC(C)=O CCCCC(C)C(=O)NC1CN(C(=O)CCCc2csc(C)n2)CC1(C)C c1(C(N(CCC(C)NC(c2cc(Cl)cc(Cl)c2F)=O)C)=O)ccn2nccc2c1 c1(CNC(=O)CCNC(C2CC2C2CCCO2)=O)ccc2c(c1)CCN2 c1(C(=O)N(CC(=O)N(C2CCC2)CCO)CC(O)C2CCC2)cc(SC)co1 c1(SCCC(N2C(C(=O)Nc3n(CC)nc(C)c3)CC2)=O)cc(F)cnc1Cl C(=O)(C1=CCCCCC1)NCC1N(C)CCN(C(C2C(OC)CCC2)=O)C1 Cc1nc(C(=O)Nc2cccc(C(C)F)c2)ccc1-c1cccs1 Cc1ccc(C(N2CCC(CCNC(=O)CN3CC4CC4C3)CC2)=O)c(=O)n1C c1(CC)ccc(C)c(C(N2CCCC(Cn3cc(C4(COC)CC4)nn3)C2)=O)c1 Cc1cc(C)c(CC(N2CCCCC2CNC(c2ncn(C(C)(C)C)n2)=O)=O)s1 c1(C(C(=O)NCC2(O)CC(NC(c3cnc(COC)s3)=O)C2)O)cccc(F)c1 Nc1cc(C(N2CCC3C(NC(=O)CN4CCSCC4)C3C2)=O)ccc1F c1(N(C(=O)CC2CCN2C(=O)OC(C)(C)C)C)cncc(Br)c1 C1(NC(C2CCC(=C)CC2)=O)CCCN(C(c2cc(N)ccc2Cl)=O)C1C N1(C(C2OCCN(C(C3CC4(CCC4O)C3)=O)C2)=O)CC(F)(F)C(F)(F)C1 c1(C(=O)NCC2(O)CCN(C(C(CC)F)=O)CC2)ccc2c(c1)CCC2(C)C C1(NC(C#CC(C)C)=O)C2CC3CN(C(=O)CCc4cncc(F)c4)C1C3C2 Cc1ncc(N)cc1C(N1CC2(C1)CN(C(=O)COC1CC1)C2)=O N1(C(C2(C(=O)OC)CC2)=O)CCN(C(=O)C(CO)C(C)C)C(c2cn[nH]c2)C1 CC(CC(=O)NCC1(C)CCCCC1)C(C)(C)NC(c1cc[nH]c(=N)n1)=O CCC(CC)(CCNC(=O)C(C)OCC(C)(C)C)NC(C1(c2ccsc2)CC1)=O Cc1ncc(F)c(N2CCC(C)(C(=O)Nc3cnns3)C2)n1 C(=O)(CCCCCCc1ccccc1)N1CC(C)(NC(CC=CC)=O)C1 c1(CN(c2cc(Nc3c(C)ccc(Br)c3)ncn2)C)cn2cc(Cl)cc(C)c2n1 C(=O)(C#CC1CCC1)NCCC(C)NC(c1cc(C)n(C(C)(C)C)n1)=O N1(C(C(COCCOC)C)=O)CCC2(CC1)COC(C)C2N1CCC(OC)C1 CCCN(Cc1ccc(F)cc1)N1CCCC(OC)C1 Cc1noc(C)c1C(C)NC(NNC(=O)Nc1ccccc1)=O c1(NC)scnc1C(=O)N(CC(O)CN(C(=O)C(C)Cn1cccn1)C)C C(N=c1[nH]c(Cl)ncc1Cl)C1(C)CCN(C(=O)CC2CCC3(CCC3)O2)C1 c1(C(N2CCN(C)CC2CNC(c2sccc2Cl)=O)=O)cc2nc(=O)ccn2[nH]1 C(CNC(=O)C(C)=CCNC(=O)C(C)N1CC(C)C1)(C(F)(F)F)OC c1(C(C2CCCN(C(c3ccc(Br)s3)=O)C2)O)cc(F)c(F)c(F)c1 N1(C(C2(CC#C)CCC2)=O)CCC2CN(C(=O)Cc3cnccn3)CC2CC1 C(=O)(C(C(C)C)C(C)C)NC1C(OC)CN(C(c2ccc(Cl)cc2)=O)C1 N1(C(c2c(CC)scn2)=O)C(C)C2CC1C2NC(c1ccc(F)cc1)=O C1(NC(C2(C(C)NC(c3c(C)n(C)cn3)=O)CC2)=O)CCN2CCC1C2 N1(C(C(CC)Oc2ccccc2)=O)CCN(C(c2snnc2C)=O)CC1CF Cc1noc(C)c1CC(N1CCC(NC(C2CC(C)(C(C)C)C2)=O)C1)=O N1(C(C2N(C(CC)=O)CSC2)=O)CCCC(CNN(C)C(C23CC(F)C2C3)=O)C1 C1(C(N(CC)CC2CCCN2C(=O)Cn2nccn2)=O)NC(=O)OC1C c1(CC)sccc1S(=O)(=O)N(C1C(C(=O)OC)CCCC1)C.C12(O)CN(C1)C2=O C1(NC(=O)C#CC2CC2)CCN(C(c2ccc(C(F)(F)F)nc2)=O)C12CC2 C1(C(c2n(CCOCCOC)nnn2)NC2CC2)OCCOC1(C)C Cc1cc(-c2ccncc2N(C)C)cc(C)c1C#N CCC(CC)CCCC(=O)N(C)CC1(CNC(=O)CC2CCCCC2O)CC1 c1(NC(N2CCCC(CC3CCCCC3)C2)=O)cccc(C2CC2)c1 N1(C(C(C)N(C(C)=O)C)=O)CCC2CN(C(=O)Cn3cccn3)C(C)C12 C1(CCNC(C(C)=C2CC2)=O)CN(C(c2cnc(C3CCOC3)s2)=O)CC1C C1(CC(=O)NC2C(CNC(C(C)(C)c3cnc[nH]3)=O)C2)CCCCCCC1 C1(C(=O)NC2C3CN(C(C(CC)=O)=O)C(C3)C2)CCc2nc[nH]c2C1 CC(C)CC(C(=O)NCC1(C)CCC(=O)N1)NC(=O)C(C)(F)F C12(C(N(CCOCCCNC(C(C)C3CCOC3)=O)C)=O)CCC(CC1)C2(C)C C(=O)(CC(C)N(C)C)NCCSCC(C)(C)C.c1(C)cccnc1.C1CCOCC(=O)N1 CCCCC(C(=O)NC1(c2nc(C)no2)CC1)NC(C1CC12CC2)=O Cc1ncc(C(N2CCSC(C(=O)Nc3cnc(I)cn3)C2)=O)cn1 C1(c2ccccc2)(CNC(COCCC)=O)CCN(C(C2CC(C)=NO2)=O)CC1 C=CC1(C(=O)NCC2(F)CN(C(=O)Cc3ccco3)C2)CCC1 c1(C(=O)NCC(CN(C)C(c2ccc(=N)[nH]c2Cl)=O)(C)C)cn(C)c(=O)cn1 N1(C(CN(CCC)C)=O)CCC2(CCC(NC(C3(O)CCC(C)CC3)=O)CC2)C1 C1(C)(C(=O)NC(C23CCCC2CCC3)C)CN(C(c2cccc(F)c2)=O)C(C)(C)C1 N1(C(COCCOCC)=O)CCCCC2(C1)CN(C(=O)C(S(C)(=O)=O)C1CC1)C2 C1(CNC(=O)C=Cc2cccnc2)CCCCCN1C(=O)CC1CCCOCC1 S(=O)(=O)(c1cccc(-c2cnnc(O)c2)c1)NCCc1ccc(C)cc1Cl C(C(CO)N=c1ccc2nnnn2[nH]1)NC(Cc1cc2c(cc1)N(C)CC2)=O c1(N(C)C)ccc(NC(c2cc(NCc3cnc(Cl)cn3)cn2C)=O)cn1 C1(c2n(C)ccn2)CN(C(C2CC=CC2)=O)CCN1C(=O)CNc1ccccc1 c1(CNC2C(C(=O)Nc3c(C)cc(COC(F)(F)F)cc3)C2)c(F)cc(F)cc1Br N1(C(c2c(F)cc(C(F)(F)F)cc2Br)=O)CCCC2(CCC(OCCCl)C2)C1 C1(CCC)CN(C(CC(C)C)C(=O)N(C)CCN2CCOCC2)CCC1O N1(C(c2cccc(OC)c2O)=O)CC2OCCN(C(=O)C(=O)C3CC3)C2C1 C1(NC(C(C)(C)NC(=O)NCC)=O)CN(C=C2CCC(C)C2)C2(CCCC2)C1 C(=O)(C(C)(F)C(C)(C)F)N1CCN(C(c2cc(OCC)no2)=O)CC1 c1(C(=O)NC2C(C(=O)NCc3c(C)cccc3)C2)nccn2c(Br)cnc12 c1cc2nc(N3CCCCCCC3)[nH]c(=NC3CCOC(CC4CC4)C3)c2[nH]1 CC1CC(NC(C2CN(CC(F)(F)F)C2)=O)CN1C(c1c[nH]c(C#N)c1)=O c1(CNC2(CC(=O)Nc3c(OC)nccc3)CCC2)ccc(Br)c2cccnc12 C1(NC(c2ccc(OC)o2)=O)CN(C(=O)CC2CN3CCC2CC3)CCC1CO c1(C(N2CC(Cn3cc(C4(CC)CC4)nn3)OCC2)=O)cc(C)c2[nH]cnc2c1 c1(C(=O)NC2CC(N(C(c3cc(C)cc(C)c3)=O)C)C2)ccc2cc[nH]c2c1F Cc1nc(C)c(-c2cn(CC(=O)N(CC)Cc3ncoc3C3CCCCC3)nn2)s1 Cn1ccc2cccc(C(=O)NC3CCCC3NC(c3csc(C(F)F)c3)=O)c12 C1(C(=O)NC2CC2F)CCCCN(C(C2CC2(F)F)=O)C1 C(=O)(CCCCC(F)(F)F)N1CCN(C(C(COC(C)C)(C)C)=O)C(C)C1 CC12CN(C(C3C=CCC3)=O)C(C(=O)NC(CO)CCO)(C1)C2 N1(C(CC=CCNC(c2c(C)oc(CO)c2)=O)=O)CC2CCC(C1)N2C c1(C(C)C)cc(Br)ccc1CCNC1(c2nnnn2C2CC2)CCCN(C)C1 C1(NC(C2C(C)CC(=O)NC2)=O)CC2(CCN(C(=O)C(C)(C)C3CCC3)CC2)C1 C(C)(C)(CC(F)C(=O)NCc1ccncc1)NC(CC1CCCC(C)O1)=O C1(CC(=O)NCC2COCCN2C(C2CC3CCCC23)=O)CCCCCCC1 c1(N(CCNCN)C)cc(C2CC2)n(C)c(=O)n1.n1(CC(=O)N)nnc(CCO)n1 Cc1c(C(=O)Nc2cccc3c(C)cccc23)[nH]c2c1C(=O)CCC2 C(=O)(CCCCCN(C)C)NCC1CCCC(NC(CSCC)=O)C1 Cn1cncc1CCC(=O)NC(C1CCCCC1)CNC(=O)COC1CCCC1 c1(-c2cccc(NC(CC)=O)c2Cl)cc(C(=O)Nc2cccs2)cc2[nH]ncc12 N#Cc1ccc(C(=O)NC2CCC(NC(c3nc(Cl)cs3)=O)CC2)c(O)n1 C1(C(=O)NCC(C(C)C)CO)C2CC3C(C2NC(=O)CC=CC(C)(C)C)C13 c1(C(=O)Nc2nc(C(=O)OC)c(Br)s2)ccc2cccc(Br)c2n1 C(=O)(C1=NOC(C)(C)C1)NCC12CC(NC(Cc3nc(CC)sc3)=O)(C1)C(C)O2 C1(CC)CCCN1C(c1sccc1CNC(c1ccn(C)n1)=O)=O c1(OC)cc(I)ccc1N(C)C(C)=O.c12ccnc(c1)-c1cccc(c1)NC2=O C1(C)(C(=O)NCC2(C)N(C(Cc3nnc(C)s3)=O)CCC2)COC(=O)OC1 c1(C(=O)OC)ccc(C(C)=Cc2cn(CC3CCCC3C(F)(F)F)nn2)cc1 C1(CC)(NC(C2CC(=O)N(C)C2)=O)CCCN(C(c2snnc2C)=O)C1 C1(CN(C(=O)COC2CN(C(=O)CC3(C)CC3)C2)C)CCCCCC1 CC(CC(=O)O)C(F)F.C1N(CC(C2CCC2)=O)CCCCC1 N1(C(c2cn(CC=C)nc2)=O)C2COCC1CC(NC(=O)Cc1csc(C)c1)C2 C1(CCNC(C=C(CC)CC)=O)CN(C(c2cnc(CC)[nH]2)=O)CC1C c1(C(N2CC(C(C)NC(C=Cc3cnc(C)s3)=O)C2)=O)ccc(N)c(F)c1 Cc1cccc(CCC(=O)NC2CC(O)(CNC(C34CC(C)(C3)C4)=O)C2)c1 C1(C(N2CCC(NC(Cc3c(C)ncs3)=O)(CO)C2)=O)CCc2nccn2C1 c1(CC)ccc(C(=O)NCC(C2CCOC2)NC(=O)CC2CCOCC2)cc1F N1(C(C2CCCCCN(C(=O)C3CC3)C2)=O)CC2CCCC(O)C2C1 CCC(CNC(=O)COCC(=O)N(C)C)(CC)C(=O)N(CC(c1ncc[nH]1)C)CC c1(C(=O)NCC(C)CNC(C23CCC(C)(CC2)CO3)=O)cc2ccccc2[nH]1 N#Cc1cccc2c(C(N3CC(C4CN(C(C5(F)CC5(F)F)=O)C4)C3)=O)c[nH]c12 N1(C(c2c(COC)cccc2)C(=O)NCCOC)CCNC(=O)C1(C)C.C1CS1 N1(C(C(n2c(C)cc(C)n2)C)=O)CC(NC(c2cc(O)ncc2Br)=O)CC(C)C1 c1(N2CC(OC)(CNC(C)=O)C2)ncc(SC)cn1 c1(C(N2CCC(n3cc(CN4CCCC4)nn3)C2)=O)cccc2[nH]ncc12 C1(SCC)CCCC1N=c1[nH]c(=NC2CCN(C)C2C)[nH]c2c1COC2 Cc1csc(CCCC(=O)NC(C2(O)CN(C(=O)CC3CC(C(F)F)C3)C2)C)n1 C1(NC(C(C)N(C)CC)=O)Cc2ccccc2N(C(=O)OC(C)(C)C)C1 c1(CC(N2C(C(C)NC(CC=CC=C)=O)CCC2)=O)csc2nccn12 C1(C(=O)NCc2c(OC)cccn2)CN(C(c2ccsc2C#N)=O)CC12CCC2 c1(C(c2n(CCSC)nnn2)NCCC2C(F)(F)C23CCC3)ccc2c(c1)CC2 c1(-c2nc(C(CC)CC)nn2C(C)C)cccc2sc(CCOC)cc12 N1(C(C23C(CN(C(Cn4c(C)nc(C)n4)=O)C2)C3)=O)CC(C)c2ncccc21 C(=O)(C(C(C)(C)C)c1cn(CCN2CCCC2)nn1)NC1(CCC)CCNC1=O C#CCC(CC(=O)N1CC(CSC)C1)NC(c1cc(O)ccc1F)=O C12(C(N3C(C(=O)NC)(CC)CCC3)=O)CC(C)(CCO1)C2.N12CCCC(C1)CC2=O N1(C(C(C2(O)CN(C(C(COC)C)=O)C2)F)=O)CC(CO)C(C)C1 C12(CNC(C(F)=C(C)C)=O)CCCCC1N(C(=O)CCc1ccccc1F)CC2 c1(C(=O)NCC2C(NC(Cc3c(C)occ3)=O)C2)ncnc2cc[nH]c12 Cc1ccsc1C(N1CCC(OCCC2CCCCC2)C1)C(=O)NC1CCC1 c1(C(C(=O)NCCCOC)N(C2CC3CC(C2)N3C)C2CC2)cc(F)cc(F)c1F C1(NC(C(N2CCC(C)CC2)=O)=O)CC2(CO1)CN(c1ncc(O)cn1)C2 c1(C(CN(C(C(=O)NCC#C)=O)CC)C)ccc(N(C)C)cc1 C1(NC(C2CC(N3CCCC3)C2)=O)CN(C(=O)CO)CCC12CCOCC2 c12cc(Cl)ccc1C(=O)N2.C1(NC(C2(NC(C)C)CC2)=O)CN(CC)C1 C1(COC)CN(C(C2CC2C(C)NC(c2sccc2C)=O)=O)CCO1 C1(C(=O)NCC(CC=C)NC(c2nccc(CO)n2)=O)CCC(=O)N(C(C)C)C1.CC CCCCCC(O)CNC(C1(CC)CCN(C(c2nnsc2N)=O)CC1)=O C1(OCc2c(C)nc(C)o2)CN(Cc2nn[nH]n2)CC1(C)C C(=O)(C1=C(Cl)CCCC1)N1CCC(NC(C2C(C#C)C2(C)C)=O)C1 C1(c2nc(NC(N3CCCC3Cc3cc[n+]([O-])cc3)=O)on2)CCCS1(=O)=O N1(C(=O)CN2CCCC2CO)CC2CCC(C1)N2C(c1csc(CO)n1)=O N1(C(CCC(C)NC(N)=O)=O)CCN(C(C2(OC(C)C)CC2)=O)CC1C(F)F C1(CNC(C(C2CC2)SCCOC)=O)C(CO)C1(F)F.C1(C(=O)NC2CC2)CC(OC)C1 C1(C(=O)OC)OC(C(N2CCC(NC(C3CN(C4CCC4)C3)=O)C2)=O)CC1C CCC(CCC(=O)NCc1cc(C(C)C)no1)NC(c1nc[nH]n1)=O C(=O)(C(C(C)C)N(C)C)NCC(C(C)C)NC(C1(Cc2cnn[nH]2)CCC1)=O C1(CNC(C2C=C(C)CS2)=O)C(C)CCCN1C(=O)Cc1c[nH]nc1C C1(C)(C(=O)N(c2ccccn2)C(C)C2CC2)CCCN(C(C2CC(F)(F)C2)=O)C1 N1(C(C(C)=C2CCCC2)=O)CCC2(CCC2)C(NC(=O)COCC(C)C)C1 CC1(C)CCCC(NC(c2cn(CCNC(=O)CN3CCC(F)CC3)cn2)=O)C1 CC(F)(F)C(F)C(=O)N1CCCCC1C1CCCN(C(=O)CC2CC=CC2)C1 CCCC(C(=O)NCC1(N(C)C)CCC1)NC(C12CCC(OC)C1C2)=O N1(C(C(C(C)(C)C)CO)=O)Cc2n[nH]cc2C1C(=O)NC1CCC(C)(O)CC1 C(CCCC(=O)N1CCC(n2cccc2)C1)N(C(=O)Cc1cccs1)C S(=O)(=O)(c1cccc2c1CCCC2)NC1CC(C)(CC)OCC1 N1(C(CCC(=O)c2ccc(C)s2)=O)CCCN(C(C23CC(CO2)C3)=O)C(C)C1 C(=O)(C(C)C(C)NC(c1snc(C)c1N)=O)NCC(COC)C c1(CCC(=O)NC2CCCN(Cc3cc(C)n(C)n3)C2C)nc2ccccc2[nH]1 C12(CNC(c3c(C)nn(C(C)C)c3)=O)CCC1CN(C(c1[nH]ncc1C#N)=O)C2 C1(NC(c2ncc(OC)cn2)=O)CC(F)CN(C(=O)C(O)Cc2ccccc2)C1 CC1(C(F)F)CC1C(=O)N(CCC(=O)N(C1CCC1)CC#N)CC1CC1 C1(CC(=O)NCC(CNC(c2n(C(C)C)ccc2)=O)O)CCCC1(F)F O=C1CCC(C(=O)NCC2COC(CNC(=O)C3=CCC3)C2)CN1 c1(NC(=O)NC(c2c(OC)cccc2)CO)cc(C)c(OC)c(C)c1 Cc1oc(C#N)cc1C(=O)NC1CCN(C(=O)Cc2ccc(F)cc2Cl)C(C)C1 C#CC(C)(C)C(=O)NCC1CCCCN1C(=O)C(C)NC(c1cnoc1C)=O N1(C(C(C)C(C)O)=O)CC2CCCC(C1)N2C(C1(c2ccccc2C#N)CC1)=O Cn1cc(C(=O)NC2CCCC2NC(=O)COCC(F)F)c(O)nc1=O c1(C(=O)NC(CN(C(=O)C(O)CN2CCCC2)CC)C)cncn(C)c1=O C12(NC(N(C3CC4CC3CN4)C(c3ncc(N)nc3)=O)=O)CC3CC(CC1C3)C2 c1(CC)ccc(C(=O)NCCc2nc(-c3ccccc3)cs2)cc1F C(C)(CCC(=O)NCC(C)NC(C1(c2ccccc2)CC1)=O)OC CS(=N)(=O)C1CCN(C(CCCCC2CC2)C(=O)NCCCOCC2CC2)C1 c1(C(N(CCCNC(C(CC)CC(F)(F)F)=O)C)=O)sc2cc(C)ccc2c1Cl C12(C(=O)NCC(CC)(C)CC)CCCC1CN(C(c1cncn1C)=O)C2 C(CC(C)CCNC(=O)C(O)CN1CCOCC1)NC(CC(=O)OC)=O C(=O)(C(C)C(C)(C)C)N1CC(CC(C(=O)N(CCC#C)CCO)F)C1 c1(CCC(=O)NCCCN(C)C(C2CCC23CCCO3)=O)ccc2c(c1)CCO2 C12(C(N3C(NC(c4ccnnc4)=O)CC4CC43)=O)CC3CC(CC(C3)C1)C2 CC1CCN(C(=O)CC2CC3(CCC3)C2)CC1CC(N1CCCC2(C1)N=N2)=O CCCCC(=O)C(=O)N1CCCC(O)(CN(C)C(c2coc(COCC)n2)=O)C1 C1(OC)CC12CCN(C(C1CC3CCC(C1)N3C)=O)CC2 c1(C(=O)NC2CCCC(C(=O)NCC=CCCOC)CC2)ccc2cncn2c1 C1(NC(=O)CCCn2cccn2)CCOCC1C(=O)NCCCCCCF C(=O)(C1CCCc2ccnn21)N(CCCCNC(c1n(CC)ccc1)=O)C c1(C(=O)NC(CC)CNC(=O)C(C)(C)CC2CC2(F)F)ccc(OC)c(N)n1 C1(C(=O)NCCC(C)NC(C2CC3(C2)CC3(F)F)=O)CC2(CCCC2)CO1 C1(NC(c2nn[nH]c2Cl)=O)CC1C1CCCN(C(=O)COc2ccccc2O)C1 c1(C(N=c2nc(COC)[nH]s2)=O)cc2c([nH]1)CCN(c1ccc(Cl)c(Cl)c1)C2 N1(C(c2cnn(CC)c2C)=O)CCC2(CC2C(=O)Nc2cccnc2)C1 C1(=O)CC(C)N1.C(=O)(C(C)(C)SC)NCCN(CCC)C(C)C C1(CC)CN(CC(=O)NCCCNC(c2cccnc2F)=O)CCO1 C1(NC(C(n2ncc(C)c2)C)=O)CCOC(CNC(=O)Cc2c(C)cnn2C)C1 c1(-c2n(-c3ccc(C)cc3C)nc(C3CC3C)n2)cc([N+](=O)[O-])ncc1Br N1(CC)CCCC(C)(Nc2ccnc(CNC(=O)CCCN(C)C)c2)C1 O=C(N=c1c(Cl)c[nH]cc1Cl)C(=O)N1CCOC(c2cn(-c3ccc(F)cc3Cl)nn2)C1 c1(C(C)=O)cc(-c2cn(CCN(c3ncccn3)C)nn2)oc1C c1(C(=O)NCCC(C)NC(C2CCS2(=O)=O)=O)c(N)cccc1[N+](=O)[O-] C(=O)(C(c1ccco1)NC(=O)CNC(=O)C1CC1)NC(C)Cc1cccs1 C(CS(=O)(=O)CC(=O)NC12CCCN(C(=O)CCc3ccncn3)CC1C2)OC C(C)(CCC(=O)NCCn1cc(C(N2CCCCC2C2(O)CC2)=O)nn1)SC N1(C(CC2(C=C)CCC2)=O)CC(NC(=O)CC2(C)OCCO2)C(C)C1 C(CC(C(=O)N1CCC(CN=[N+]=[N-])C1)NC(=O)COCC1CCCC1)N(C)C c1(C(N2CCN(C(C3(C#C)CC3)=O)CC2)=O)ncn2c1CCCC2 C1(C)(C(=O)NCC(CNC(c2cc(C(C)C)[nH]n2)=O)OC)CC(C2CC2)=NO1 O=C1C2CSCC1CC(C(=O)NC1CCCC1NC(=O)C(=O)NCC1CC1)C2 c1(C(=O)NCC2C(C)CN(C(C3CCCSC3)=O)C2)ccc(O)c(O)c1 c1(SC)cn(C)nc1C(=O)N(C)CC1CC1.C12CCN(CC1)C(=O)C(=O)NCC2 N1(CNC(=O)Cn2cc(-c3cn(C(C4CCC4)C4CC4)nn3)cn2)CCC(F)CC1 c1(C(N(C2CCS(=O)(=O)C2)CCN)=O)cc2c[nH]cnc-2n1 N1(C(C=COCC)=O)CC2C(CN(C(=O)CCCSc3scnc3C)C)C2C1 c1(CC(=O)NC(CN(C(=O)C(c2ccc(C)cc2)C)CC)C)cnn(C)c1C c1(CC(=O)NC2(C3CN(C(C4(C#C)CC4)=O)C3)CC2)ccc(S(=O)C2CC2)cc1 C1(CCNC(c2n(CCC)ccc2)=O)CN(C(=O)CC2(C)CCCCC2)CCO1 CC(F)(F)C(C)(C)CC(=O)NCC1COCCN1C(=O)CC12COC(C1)C2 N1(C(C2CCCC(C)C2)=O)CCN(C(=O)Cn2ccc(O)nc2=O)C(C)C1 C(N=c1[nH]c(=NCCC2CC2C(F)(F)F)[nH]c2c1CSC2)C1(C=C)CCC1 c1(C(N2CCCC(N(C)C(c3ccc(CO)o3)=O)C2)=O)cc(O)c(F)cc1N c1(C(=O)NCCCOCCC(=O)NCC2(CCC=C)CC2)nccc(C)c1F c1(C(=O)OC)coc(C=CC(N2CCN(C(C)=O)CC2)=O)c1 C1(NC(COCC(=O)NC)=O)CS(=O)(=O)CC1NC(c1ccc(O)cc1SC)=O CCC(F)(F)CC(=O)N(CCNC(C1(C(C)C)COC1)=O)Cc1ccc(Cl)nc1 Cc1cccc(OCCCNC(=O)C(=O)NC(C)CC2CCC2)c1 c1(C(=O)NCC2(C)CC(NC(=O)C(C#N)C(C)(C)C)C2)ccc2n[nH]cc2c1 C1(C(=O)NCCNC(C(CC)C)=O)Cc2cc(Br)ccc2O1 c1(N2Cc3n(cc(C(F)(F)F)n3)CC2)nccc(=NC2CC3(C2)CC3(F)F)[nH]1 C#Cc1cncc(C(N2CCCC(CNC(=O)CCCNC(N)=O)CC2)=O)c1 N1(Cc2cn(CC3N(C(c4n(CC)ccc4)=O)CCC3)nn2)CCSC(C)(C)C1 C(C(CC)(CC)C(=O)NCc1[nH]cnc1C)NC(CCCOCCC)=O N1(C(C2CC(OC)C2)=O)CCC2(CC1)CCN(C(C1(C)C=CCC1)=O)C2 C1(CNCC)CCN(C(C2CC(O)CN2C(c2cccnc2Cl)=O)=O)CC1 Cc1ccc2c(c1)C(C(=O)N1CC(OCCNC(c3ccccn3)=O)C1)C2 c1(CN)cnc2ccccc2c1O.O=C1CCC(C(=O)NCC2(C(=O)NC)CC2)O1 Cc1cccc(C2CC2C(N2CCC2CNC(c2ocnc2C2CC2)=O)=O)c1Cl CC(C)(C(=O)NCCCn1cc(CC(CO)C2CC2)nn1)c1ccccc1 CCC(CCC(=O)N1CC(N(C)C)C(C)(C)C1)NC(c1c[nH]c(C)cc1=O)=O CC1(C)CCC(=CC(N2CCN(C(c3n[nH]cc3Cl)=O)C(CF)C2)=O)CC1 CC(C)(C)C(CO)C(=O)NC1CC=C(C(=O)N2CCOC(CN=[N+]=[N-])C2)C1 N1(C(c2scc(CNC(C3CC(C)=C(C)CC3)=O)c2)=O)CC2CC3CC2C1C3O C12(C(=O)NCC34CC(NC(CNC(=O)OC)=O)(C3)C4)C3CC(CC13)C2(F)F c1(C(C)NC(C)CNC(=O)OC(C)(C)C)cn(CCc2ccc(C)s2)nn1 C(CCC(=O)N(CC(C)OC)C1CCC1)N(C(=O)OC)C c1(C(=O)NC(CCNC(CCc2ccc(OCC)cc2)=O)C)ncc(F)cc1F Cc1cnn(CCC(=O)NCC2CCN(C(C3(C)CC3(F)Cl)=O)C2)c1 CC(C)(C)S(=O)(=O)CC(=O)N(CC=CCN=c1[nH]nc(CC(F)(F)F)s1)C1CC1 C1(CNC(c2c(C)scc2)=O)CN(C(=O)CC2SC(=N)NC2=O)CCO1 N1(C(c2cc(CC)sn2)=O)CC2(CC(C(=O)Nc3cccc4c3CCC4)CO2)C1 C=CC(C)(C)CCCNC(c1cccc(CNC(=O)C(C)(C)C2CC2)n1)=O C12(C(=O)NCC=CCNC(C3CC(F)C(=O)N3)=O)CCC(CC1O)C2 N1(C(c2ccn(CC(=O)OCC)n2)=O)CC(NC(=O)Cc2cscn2)C(O)C1 OCC(CN=c1[nH]c(N2CCSCCC2)nc2c1COCC2)C(F)(F)F CCCC(C)CN=c1[nH]c(=NC)[nH]c(=NC(CCSC)c2ccc(C)o2)[nH]1 c1(C(N2CCC(CC=C)(NC(=O)Cn3ncnn3)C2)=O)cccc2nc(C)[nH]c12 c1(C(=O)OCC)ccc(Cl)cc1C(F)F.c12sc(nc1C)OCC2=O C1(C(=O)NCC2CN(C(=O)CC3CC3)CCC2(F)F)(COC)CCCNS1(=O)=O S(=O)(=O)(c1ccc(F)c(F)c1F)NC1CCCC(C(N2CCOC(O)C2)=O)C1 c1(C(=O)NCCC(CNC(C2(C)CC(F)C2)=O)OC)ccn2ccnc2c1 N1(C(C2C3CCCC23)=O)CCC2(CCCN2C(c2sccc2C(F)F)=O)C1 N1(C(COC(C)C)=O)CCCCCCC1C(=O)NCC1CCOC(C)(C)C1 S(=O)(=O)(c1ccc(NCc2cc(-c3ccc(F)cc3)on2)cc1)NC c1(-c2sc(NC(COc3c(OC)cccc3)=O)c(C)n2)c[nH]c(=N)nc1C C1(CC)CN(C(=O)C=CC(=O)N(C)C)CCC1NC(c1[nH]cc(OC)c1Cl)=O c1(NC(C2CCC(F)(F)CC2)C)nc(C)cc(=NCC(F)(C(F)(F)F)C(F)(F)F)[nH]1 c1(C(N2CC(NC(=O)C3=C(Cl)CC3)C(CO)CC2)=O)c[nH]c2cc(F)ccc12 CCC1=C(C(=O)NC(CNC(=O)CC2OCCCO2)CO)CCCO1 C=C1CC2(C1)CC(C(N1CCN(C(c3c[nH]c(=NCC)s3)=O)CC1CCC)=O)C2 c1(CCNC(c2c(C)cc(O)nn2)=O)nc2c(s1)CN(C(C)(C)C(=O)OC)CC2 c1(COC)cc(C(=O)NC2CC2CNC(=O)CCCC2CC2)no1 CC1SCCCC1C(=O)NCc1cn(CC(=O)NC2CON(CO)C2=O)nn1 c1(CN(C(CCC)=O)CCNC(=O)CCc2cnco2)cccc(OC)c1 c1(NC(=O)NNC(=O)C2CC2)ncc(Br)cc1C(F)(F)F c1(NC(COCC(C)C)=O)cncc(C(N2CCC(C)C2)=O)c1 N1(C(C(c2cccc(Cl)c2)CC)=O)CCN(C(C2(n3cnnn3)CC2)=O)CC(O)C1 c1(OC)ccc(-c2nccn2C2CC2(c2ccccc2Br)C)nc1O N1(C(c2ccc(SC)o2)=O)CC(NC(c2cnsc2)=O)C2(CC2)C1 N1(C(CN2CCC(OC)C2)=O)CCC2CCN(C(=O)CN(C)C(C)=O)CC2C1 N1(C(C(C)NC(C)=O)=O)CCCC(N(C)C(c2coc(Cl)c2)=O)C1 C12(NC(c3occc3F)=O)CCOCC1CN(C(c1scnc1Cl)=O)C2 N1(C(COCCC)=O)CCC2CC2(C(=O)N(C2CN(C3CC3)C2)C)CC1 c1(C(=O)NCC2C(NC(C(C3CCC3)OC)=O)C2)ccc(OCCF)cc1F c1(C(C)C)cc(CNC(=O)CCN(C2CCCCC2)C)no1.C1C(=O)O1 C1(C(=O)O)CC2(CCOCC2)CN1C(C1CC1c1ccccc1C(F)(F)F)=O n1(CC(=O)NC(CNC(C2(OC)CCCC2)=O)C)nc(O)ccc1=O CC(C)C(CC(=O)N1OC2CCC1CC2)NC(=O)CC1CCC(C)CO1 C1(C(=O)NCCCC2CCN(C(c3nnc(CC)s3)=O)CC2)Cc2nncn2C1 CN1CCCC(NC(c2cccc(OCc3ncccn3)c2)=O)C1 C(CCc1ccccc1)(C(C)NC(c1coc(C(C)C)n1)=O)NC(C)=O c1(C(=O)OC)nc(NC(C2CCCCN2C(=O)CCN2CCC(C)C2)=O)c(C)s1 C(=O)(C(C)(C)F)NCCCCN(C)C(C1CC(CF)C1)=O c1(OC)cccc(S(=O)CC(=O)NCC(C)NC(=O)Cc2cc(C)ccc2F)c1 c1(C(=O)NC2CC3(C(NC(C=Cc4ccc(C)s4)=O)C3)C2)ccn(C)c(=O)c1 c1(-n2cc(C3(O)CN(C(C4(C(=O)O)CCCOC4)=O)C3)nn2)cccc(F)c1F C(=O)(CC(C)C(=O)NCCCCCC(=O)NC(c1cccs1)(C)C)OC c1(C(=O)OC)cc(CC(=O)NCC(C)NC(C2CC=CCO2)=O)cs1 c1(OC)csc(C(N2CCCC2C2(O)CN(C(=O)C(C)SC(C)C)C2)=O)c1 C1(N2CCOCC2)(CC(=O)N(C(C2CCOC2)C)C(=O)OC(C)(C)C)CCOCC1 c1(C(=O)NC(C)CCNC(=O)CC2(CO)CC2)nccnc1N N1(C(CNC(C(CC)CC)=O)=O)CCC(NC(C2CCCOC2)=O)C(O)C1 C12(C(=O)NCC=CC)CC1CCN2C(=O)CN1CCC(C)C1 C12(NC(c3cnn(CC(C)C)c3Cl)=O)CCCCC1CN(C(=O)CO)C2 C1(C(=O)NCc2cn[nH]c2)CN(C(=O)C=CC2CCCCC2)CCO1 N1(C(c2c(C)occ2)=O)CCC(C)(NC(c2cc[nH]n2)=O)C1 C1(C(C)NC(COCCOCC)=O)CN(C(c2c[nH]nc2Br)=O)CCO1 C1(CN(C(=O)C=C(Cl)Cl)C)CN(C(=O)C=Cc2ccc(Cl)s2)CCO1 c1(NC(C2N(Cc3c(C(=O)OCC)ccs3)C3C(C2)C3)=O)cc(I)cnc1Cl C(C1=COc2ccccc2O1)(c1nnnn1C1(C)CC1)C(C1CCCC1)C Cc1ccc(C(N2CC3CC3(CNC(=O)CC3CCC(=O)NC3)C2)=O)c(N)n1 c1(N2C3CN(C(Cc4c(OC)ccc(Br)c4)=O)C(C3)C2)ncnc2[nH]c(C)nc12 c1(C(N(C2CCC(NC(c3cnc(C)[nH]3)=O)CC2)C)=O)cc2ccccn2n1 C(=O)(CS(=O)(=O)C1CC1)N1CCN(C(CCn2c(C)ccc2C)=O)CC1 CCCCC(F)C(=O)N1CCOC(Cc2cn(C3CC(O)C3)nn2)C1 C(=O)(CCCC(=O)N(C)C)N1CCC(CN(C(C2C(CC)C2)=O)C)CC1 C(C(N=[N+]=[N-])C(=O)NC(C(=O)N(CC(O)CO)C)C1CC1)OCC n12cnc3c(ncnc13)N1CCC(O)(CC1)C(C)C2.c1(SC)cnccc1CO C1(NC(C(CC)NC(=O)C(C)=CC2CC2)=O)CCCCCC1(C)C C=CCN=C(NCc1cccc(CN2CCCCCC2)c1)N1CCC(C)C1C C1(CS(C)(=N)=O)CCN(C(=O)NCC(=O)Nc2nccs2)C1 c1(C(c2ccccc2)NC(COC(CC2(C=C)CC2)=O)=O)ccc(F)c(F)c1 c1(CCC)c(C(=O)NC(C)CC(C)NC(c2cnnn2C)=O)[nH]c(C)c1C(C)=O c1(C(C)C(=O)NCC=CCNC(=O)CCC(=O)c2ccc[nH]2)c(Cl)cccc1Cl CC1CC2(C(N3CC(O)(CNC(=O)C=CC=C(Cl)Cl)C3)=O)CC12 C1(C(=O)NCC(C)CN(C(=O)CNC(N2CCCC2)=O)C)CCC=CO1 CC(C)C(F)(F)CCNC(=O)C(c1cn(C)nn1)NC(=O)CC1CCOC1C C1(C(=O)Nn2cccn2)CC12CCN(C(c1nc3ccccc3[nH]1)=O)CC2 CC(C)C(C)(CN=c1nc[nH]s1)NC(=O)CCOC1CC1 C1(C)(C(N(CCN(C(C2CCC(OCCC)CC2)=O)C)C)=O)CCCCCCC1 c1(C(C(N2CC(NC(CC(=C=C)C)=O)(CO)C2)=O)C)ccc(S(C)(=O)=O)cc1 C1(C(=O)NC2(COC)CCN(C(C3(CC(F)F)CCC3)=O)C2)CCC(C)(C)CC1 C1(C(=O)NCC2(C)CCN(C(=O)CSc3n[nH]c(O)n3)C2)C2CCC3C(C2)CC13 N1(C(c2c(CC)[nH]nc2Cl)=O)CC2(CCCC2Nc2nc(Cl)nc(C)c2Cl)C1 n1(CCCC)cc(C(=O)NC2CC(C)(NC(C3CC3OC)=O)C2)nn1 c1(C(=O)NCC2C(C)CN(C(=O)C(F)=CC3CC3)C2)ccc(N)c(Cl)n1 C12(C(=O)NC(c3cccc(C)n3)C)CC(C)(CN1C(=O)C(CN(C)C)N(C)C)C2 N1(C(C2N(C(C3(C)CC3(F)F)=O)C3(CC2)CC3)=O)CCn2ncc(O)c2C1 C(=O)(C1=CCC(F)(F)CC1)NC(CNC(c1c(C)ccc(OC)c1)=O)(C)C(C)C c1(OC)cc(C)c(S(=O)(=O)N2CCC(NC(=O)C(O)CSC)C2)c(C)c1C Cc1cc(C(N2CC(C(N)=O)(CNC(c3cc(C)c(C)nn3)=O)C2)=O)cc(O)c1 N1(C(c2c(C)ncs2)=O)CC2CCN(C(=O)C(C)(O)C3CC3)CC2C1 Cc1cc(C)c(NC(=O)C(N2CC(NC(C3(O)CCSC3)=O)C(C)C2)=O)c(C)c1 c1(C(C)=O)cc(C(=O)NCC=CCNC(C2CC(C(F)F)C2)=O)n(C)c1 Cc1cc(N2CCCN(CC(C)O)CC2)nc(=NCCC(=O)N2CCCC2)[nH]1 c1(C(=O)NCCC2N(C(COCCC)=O)CCCC2C)n[nH]c2ccc(O)cc12 c1(NC(C2N(C(C(C)Cn3cccn3)=O)CC3(CC3)C2)=O)cccc2c1CNC2 C1(NC(C=CC(C)C)=O)CCCN(C(=O)CC2CCCC23CC3)CC1 C=C=CC(C)C(=O)NC1C=CCN(C(c2ccc(C)cc2)=O)C1 c1(C(=O)NCCCN(C(=O)C(c2cscn2)N(C)C)CC)cncc(O)c1 c1(OC(C)C(=O)NCC2(CNC(=O)CC3CCC(=O)N3)CC2)ccccn1 C12CCCC3CN(CC13)C2=O.C1(NC(C(C)OCCOC)=O)CCCC(CO)C1 n1(C2C(F)(F)C2)cc(N(C2CC23CCC3)C(c2nnnn2C2CCC2)C2CC2)cn1 C1(CNC(C2CC=CCO2)=O)CCN(C(=O)CC2CSCCS2)C12CC2 N1(C(c2cc(CC)on2)=O)CC(CNC(c2nc(C)sc2C)=O)CC12CCC2 C1(C(=O)NC2CC(F)(CNC(c3ncncc3Cl)=O)C2)CCc2nc[nH]c2C1 c1(C(=O)NC(C(CO)NC(c2cn(C(C)C)nc2)=O)C)cnc2ccsc2c1 Cc1cc(C(=O)NCCC2CCCCN2C(c2cc(CO)c(C)o2)=O)cc(F)c1 C#CC(C(C)OC)NC(c1coc(CNC(C2CCC(C(N)=O)O2)=O)n1)=O C(=O)(C(CC(F)F)N(C)C(c1cncc(C#N)c1)=O)N(CCCCCC=C)C C1(O)(C(C)CNC(=O)CC2CCCSC2)CCN(C(C2CN(C(C)C)C2)=O)C1 C#Cc1cnc(C(=O)NCC(C2CCC2)NC(=O)C(C2(O)CCCC2)F)c(C)c1 C(=O)(CCS(N)(=O)=O)NC1CN(C(C2(CC#C)CCCCO2)=O)CC1C C=CCN=C(NCCC(C)CC(C)(C)C)N1CCC(NC(=O)N(C)C)C1 c1(C(N(C2CCC(Nc3ncc(Br)cc3C#N)C2)CC)=O)ccc(F)c(Cl)c1F c1(CC(=O)N(C(C)CCNC(=O)C(C2CCOCC2)O)C)cccc2sccc12 Cc1ccc(CNc2ncc(CCC3CCCCO3)s2)cc1F.C12CC(C1)NC2=O C=CCC(C)(CC)C(=O)NCC(C)(O)CNC(=O)COC1CC=CC1 C(CN=c1nc2c(cnn2C)c(N2CCC(=NO)CC2)[nH]1)(C1CCC1)OCC c1(C(N2CCC3CCC(NC(C(CCCC)C)=O)C32)=O)[nH]c2ccccc2c1Cl Cc1cccc(C(N2CCC(CCCNC(=O)C=Cc3cncs3)CC2)=O)n1 n1(CC(=O)NC(CNC(C(C(C)C)SC)=O)C)cc(C)c2ccccc12 c1(C(N2CCC(C(C)(C)C)(CNC(C(CC)CC)=O)C2)=O)ccc(CC)nc1C c1(-c2ccc(C)cc2)cncc2nc(SCc3ncccc3C#N)n(C)c12 C1(NC(CSCCOC)=O)C2CCN(C(C3(C#N)CCCOC3)=O)CC12 N1(C(CC(C)c2ccncc2)=O)CCN(C(c2cnn(C(F)F)c2)=O)CC(O)C1 N1(C(C(CC(=C)C)OC)=O)CCC2CCN(C(c3cc(C)n(CC)n3)=O)CC2C1 N1(C(c2c(CC)n(C)nc2)=O)CCN(C(c2coc(C(F)F)n2)=O)CC1CO N1(C(C=CC(C)C)=O)CC(C(=O)Nc2ccc(C3CCN(C)CC3)cc2)C(O)C1 C1(C(=O)NC(C#C)C)CC=CCN1C(c1ccc(F)s1)=O N1(C(CNC(C)=O)=O)CCC(O)(C2CCN(C(=O)CC(C)N(C)C)CC2)C1 c1(CC(=O)NC(CNC(c2cc(OC)n(C)n2)=O)(C)CO)cn2c(C)csc2n1 CCCC(Cc1ccccc1)NC(=O)CC1CC1(Cl)Cl.CCN CCC(C(=O)N1CC(NC(=O)Nc2nnc(C)o2)C1)n1cccn1 C1(C(=O)Nc2cc(C(N(C)C)=O)cc(Br)c2)CCS(=O)(=O)C1(C)C CC1CCCCCCN1C(=O)CC1CC(C)N(C(c2cc(Cl)cs2)=O)C1 N1(C(C(C(C)C)n2cnnc2)=O)CCCC(NC(C2(C)CC2)=O)CC1 c1(C(=O)NCC2N(C(COCCCCC)=O)CC(O)C2)cccn2nccc12 C1(C(N2CCCC(N(C(c3csc(C)c3)=O)CC)C2)=O)CCC(C)(C)OC1 c1(C(=O)NCC(CCOC)NC(C2CCS(=O)(=O)N2C)=O)nnc(O)cc1O Nc1sc2ccccc2c1C(N1CCN(C(C2C3COCC23)=O)C(CF)C1)=O C1(NC(C2N(C(C(C)=O)=O)CCOC2)=O)Cc2ccc(Cl)cc2NC1=O C1(CC)CN(C(=O)CCC(C)C)CCN1C(=O)CCN1CCCCC1=O c1(C(=O)OC)ccc(CNC(C2CCC(c3cn(-c4cccnc4)nn3)C2)=O)s1 N1(C(CNC(CCC(C)C)=O)=O)CCC2(CC2C(=O)NCc2ccc(CO)o2)C1 C(=O)(C1CCc2scnc21)NC1CC(NC(C(C(C)C)C(C)C)=O)C(O)C1 CC(C)CC(C(=O)N(C1CCCN(C(C2CCCOC2)=O)C1)C)N(C)C c1(CNC(C2(CC)CCC2)=O)cnn(C)c1C(=O)NCCC(F)F N1(C(C(C)OCCC=C)=O)CCC(CNC(C2CCC(C(N)=O)CC2)=O)C(C)C1 C1(C(=O)NCCn2cc(-c3ccc(CC(C)(C)O)cc3)nn2)CCCCNC1=O C1(C(=O)NCc2nc(CNC(C(CCC)NC(C)=O)=O)sc2)CC(=O)NC(C)C1 N1(C(CCCCC#C)=O)CCC(NC(c2nccc(N)c2Cl)=O)C(C)(C)C1 CC1CN(C(=O)C=CCF)CC2(CCN(C(C3CCCC(=O)N3C)=O)C2)O1 CCC(COC)C(=O)NC(CCNC)C(C)C.C(=O)(CCCCSC)N1CCCC1 c1(N(CC(=O)NCCCC(C)NC(CCCN(C(C)=O)C)=O)C)ccc(Cl)nn1 c1(OC)nn(C)cc1-c1cn(C2CCCN(C(c3cscc3Cl)=O)C2)nn1 C1(CN(C)C)CCCN(C(=O)C(C)(C)CNC(=O)COC2CCOC2)C1 CC1CN(Cc2ncn(C)n2)CCC1NC(C1CN2CCC1CC2)=O C(=O)(CC1=CCCCC1)N1CCC(O)(C(C)CNC(=O)C=CCO)C1 C(C(CCC(F)(F)F)N=c1nc2sccc2c(NCC(C)(C2CC2)OC)[nH]1)OC C(C(CC(=O)N1CCC2(CC1)CC2NC(C12CCN(CC1)C2)=O)C(F)F)N(C)C C(=O)(C1=CCCO1)N(CC=C)Cc1ncccn1 c1(C(=O)NCCCC2N(C(C(F)OC)=O)CCCC2)csc2ccc(F)cc12 C1(S(C)(=O)=O)(C(=O)NC(C(C(C)C)C)CNC(c2cnn(C)n2)=O)CCOCC1 N1(C(C(COC)O)=O)CCN(C(C2CCCC23CC3)=O)CC12CCC2 N1(C(C)=O)CC2CC(C1)C(CO)C2NC(=O)CC(C)COC N1(C(c2n[nH]c(C)c2N)=O)CCCC12CCN(C(C1CC3CCC(C1)S3)=O)C2 N1(C(C2C(C)CCS2)=O)CCC2(C1)CN(C(=O)COc1cc(F)cc(Cl)c1)C2 CC(C)(CNC(=O)CCC12CC(CCN1)C2)C1=CCCCC1 c1(C(=O)NC2(CNC(=O)CCC3(O)CCC3)CCOCC2)csc2nccn12 CCC(CC(=O)NCC1(C(=O)N(CC(=O)NC)CC)CC2(CC2)C1)C(C)C C1(C(=O)NCC2(CNC(c3c(COC)noc3)=O)CCC2)CN(C)CCO1 N1(C(CC(COC)C)=O)CCCC(F)(CNC(C2(O)CCSCC2)=O)C1 c1(C(=O)NCC2C(CNC(CNC(C(CC)CC)=O)=O)C2)cc2ccccc2s1 CC1CN(C(C23CC(F)(C2)C3)=O)CCC1NC(=O)Cc1ccc(F)cn1 C1(NC(COCCCCCC)=O)CCN(C(=O)Cc2cnn(C)c2)C12CCC2 c1(CC(=O)NCC(C)NC(CC2N(C(C)C)CCC2)=O)ccc(C(F)F)cc1 N1(C(C)C)CC(NC(N2CCOC(CC(=O)NCC3CC3)C2)=O)CC1=O C1(OC)CN(C(C2(C)CC=CCC2)=O)CC1C(N1CC(CO)C(O)C1)=O CC1CN(C(=O)CCC2(NC(=O)CO)CC2)CCO1 C12(NC(C(CC)N(CC)CC)=O)CCC(CN(C(c3n[nH]c(C)c3C)=O)C1)C2 C(=O)(C(C(=O)NCCOCCNC(c1cnc(C2CC2)cc1C)=O)C(C)C)OC C12(C(=O)NC3COCCN(C(CNC(CC(C)C)=O)=O)C3)CC1COC21CCC1 c1(C(N(CC(=O)Nc2csnn2)CC)=O)csc(CC(C)C)n1 N1(C(C(C)OCC=C)=O)CC(NC(C2CC3CC2C(O)C3O)=O)C2CCCC12 c1(CN2CC(C)N(C(c3ccc(Cl)cc3)=O)CC2)ccc2cncn2c1 N1(C(C(CC2CC2)NC(CC(C)CN(C)C)=O)=O)CC(O)C2(CCCC2)C1 C1(NC(=O)C=CI)(CF)CCN(C(=O)C(c2ccc(O)cc2)=O)C1 N1(C(CCCSC)=O)C2CCC1C1CC1(NC(=O)COc1ccccc1Cl)C2 Fc1ccc(F)c(C(c2nnnn2CC2CC2)NCc2csnc2C2CC2)c1 C#CC1CCCC(CNC(=O)CC2CN(C(=O)C(C)CC3CC3)C2)C1 c1(OC)ccccc1OCC(=O)NC1CCCC(CNC(c2ccns2)=O)C1 c1(CC(=O)NC(CCCC)CNC(c2nsnc2O)=O)cc(F)ccc1F c1(SC(C(=O)N(C(CN(C(c2[nH]cnc2C)=O)CC)C)CC)C)ccc(Cl)cc1 C1(CC)CN(C(=O)CCc2ccc(C)o2)CCN1C(=O)C(CCSC)NC(N)=O C1(CC(=O)NCC2CN(C(=O)Cc3ccc(F)cc3F)C2)COCC2(CCC2)O1 CCCC(C)(CC)C(=O)Nc1cccc(NC(=O)C(F)(F)CC)c1 C(=O)(CCCC(N)=O)NCCC1CCCN(C(c2c(C)oc(Cl)n2)=O)C1 C1(C)(C)CC(=O)N1.C1(CCCNC)CCCCN1C(=O)C(C)NC(=O)NC N1(C(C(n2cc(C3(O)CCC3)nn2)C)=O)CCC(C2CCNCC2)C1 CC(C)(C)CCCC(=O)N1CC2(CC2)CC1CNC(c1ccc(F)c(CO)c1)=O C1(CC#C)(C(=O)NCC2(NC(=O)C(C)c3ccsc3)CC2)CCCCO1 c1(C(N2CC(NC(C=CC(=O)OCC)=O)C(F)C2)=O)cc(Cl)c(F)cc1F C1(C2CCCN(c3ncnc(O)c3Br)C2)(NC(C2CC3CCC(C2)S3)=O)CC1 N1(C(C=CC(C)(C)NC(=O)CN2CCCNC2=O)=O)CCOCC(O)C1 N1(C(CC=C)=O)CCN(C)CC1CNC(C1(c2ccc(Cl)c(Br)c2)CC1)=O N1(C(C(CCC)O)=O)CCC(NC(c2ncc(C3CC3)cc2F)=O)C(O)C1 C1(NC(c2c(OC)cccc2)=O)CN(C(=O)C=C(C2CC2)C2CC2)CC12CCC2 C1(C(N(CCNC(COCCOCC)=O)C)=O)CCC(F)(F)CC1(C)C C(=O)(C(C)(CC(=O)NNC(=O)CN(C(=O)OC)C1CC1)CC)OC(C)(C)C C1(O)(C(N(CCCCOC)CC)=O)CCN(c2cncc(SC)n2)CC1 CC1(C)CC(NC(C2(F)CC=CCC2)=O)CN1C(=O)Cc1cc(C2CC2)no1 n1(CC(=O)NCCc2cc(C(N(C3CCCNC3=O)C)=O)no2)cccnc1=O Cc1cc(C(=O)NCC2CC(C)(C)CN2C(=O)COc2cccnc2)cc(C)n1 c1(C(=O)NC(C2CCCN2C(C2(CCO)CC2)=O)C)cc(O)nn1C C1(SC)CN(C(=O)CC2(C)CCCCC2)CC1NC(C12CC(C)C1C2)=O C1(NC(C2CCN(C(C)C)CC2)=O)CCCN(C(c2cn(C)nn2)=O)C1C N1(C(=O)CSc2ccc(Cl)cc2)CC2CC1(c1cn(Cc3ccc(Br)o3)nn1)C2 C1(C(N2CC(CCC)OCC2)=O)CC(C)CN(C(c2sc(C)cc2C)=O)C1 CC(CC(=O)N(CCCNC(C1CC(=C2CCC2)C1)=O)C1CC1)C1CCCCC1 C1(N(C)C(c2cnc(C(C)(C)C)nc2)=O)CCC(NC(=O)C2=CCOC2)CC1 N1(CC)CC(C(=O)NCCC2(O)CCN(C(c3sccc3OC)=O)C2)NC1=O N1(C(c2cn(C)nc2Cl)=O)CC2CC(NC(C3(CO)CC(F)(F)C3)=O)CC2C1 C1(N(C)C(=O)OCC)CCCC(NCc2cc(Cl)ncn2)C1 C1(NC(=O)CCc2cn[nH]c2)CCN(C(c2cccc(F)c2)=O)CC1F C1(O)(CN(C)C(C2(Br)CC2)=O)CN(C(=O)COCc2nc[nH]n2)C1 N1(C(C2(C)C=CCN2C(=O)CCN2CCCC2)=O)CCC2CCC(C1)S2 C(=O)(CCC(C)NC(=O)Cn1cc(C#N)cn1)N(C(CSC)C)C C1(CN(C(C(C)(C)OC)=O)C)CN(C(c2ccc(-c3cc[nH]n3)s2)=O)CCO1 N1(Cc2c(CC)non2)CCC(NC(c2ccc(OCC)cc2)=O)C(C)C1 N1(C(C(C(CC)C)N(C(=O)CCc2nc(C)no2)C)=O)CCC2CCNC(=O)C12 C1(C(=O)NCC(C(C)O)C)(NC(=O)COCC(F)F)CCC(C)(C)C1 c1(OC)c(C)cc(C(N2CCC(OCCNC(=O)C(O)C3CC3)C2)=O)cc1C c1(C(=O)NCC2(CNC(C3CCC(C)(CC)O3)=O)CCCC2)cnc(O)c(F)c1 CC(C(=O)NC(CNC(c1ccn(CC2CC2)n1)=O)C(C)(C)C)C(F)(F)C(F)F c1(C(=O)NC(C)CC2CN(C(=O)Cn3cnnc3)C2)cc2n(c1)CCSC2 C1(NC(CN2CC(C)(C)C2)=O)CC12CCN(C(c1nocc1Cl)=O)CC2 c1(SC)ncc(C(N2CCC(CN(C)C(C3(C)CCCS3)=O)C2)=O)n1C O=C(CS(=O)(=O)C12CC(C1)C2)NC1CN(C(=O)CO)CC1O C1(O)(CN(C)C(c2ccc(N(C)C)nc2)=O)CCN(C(=O)C(C)(C)CF)C1 CC(C)(C)CCCCCC(=O)N1CCC(NC(c2cc3sccc3[nH]2)=O)C1 CC(C)(C)C(C(=O)N1CC(O)C1)NC(c1sccc1Cl)=O c1(C(N2C(CN(C)C(C3(CO)CC3(F)F)=O)CCC2)=O)cccc(F)c1N C(=O)(C(CC1CCCO1)C(F)(F)F)N1CC(OCCNC(c2[nH]n(C)c(=O)n2)=O)C1 Cc1cc(F)ccc1N(C)CCNC(=O)CN(C(=O)CC1C=CS(=O)(=O)C1)C N1(C(C=CCC)=O)CC2CC(NC(c3cnoc3C)=O)C2C1 N1(C(c2c(C(C)(C)C)ncs2)=O)CCCC1(C)C(c1ccccc1)=O c1(C(=O)NC(CC)CNC(=O)CC2CC2)nc(C)ncc1Br C(=O)(CC(CC)C(F)F)N1CC(CNC(C2(OC)CCCC2)=O)C(N(C)C)C1 c1(C(=O)NC(C)CC2CC3CCC(C2)N3)cc(F)cc([N+](=O)[O-])c1 C1(C(=O)NCc2nc[nH]n2)(OC)CCN(C(=O)CC2CCCC(C)C2)C1 c1(C(=O)NCC(=C2CN(C(C(C(CC)C)C)=O)C2)F)cc(F)cc([N+](=O)[O-])c1 c1(C(=O)NCC(C2CCCC2)NC(CC2(C)CC2(F)Cl)=O)ncc(F)cc1F C=C(C)CC(C(=O)NCc1ccc(C#N)cn1)NC(c1cc(Cl)cn1C)=O c1(CC)[nH]c(=N)sc1C(=O)NCCN(C(c1cc(C)on1)=O)CC c1(CNC(c2ccc(OC)cc2)=O)c(NC(=O)C(C)S)sc2c1CCCC2 N(C(=S)NNC(=O)c1cccc(OC)c1CC)c1cccc(C(=O)OCC)c1 N1(C(C(CCC)C#N)=O)CC2(C(=O)NC(COC)CCOC)CCC1CC2 c1(C(N2C(CO)CC(NC(C(CC)CN(C)C)=O)C2)=O)snc2ccccc12 CC#CCC(C)N=c1[nH]c(=NCc2cccc(F)c2)c2cccc(F)c2[nH]1 c1(C(N2CCN(C(CC(C)SC)=O)CC(C)(F)C2)=O)ccc2c(c1)CCNC2=O c1(OCCNC(=O)C(F)(F)C2(O)CCC2)cccc(NC(C23CCCC2C3)=O)c1 Cc1cc(N2CC(C)OCC(C)(C)C2)ncc1S(=O)(=O)NC1CCC(=C(F)F)CC1 C12(C(N(CC(CC)NC(=O)CC3CCNC(=O)C3)C)=O)CC3CC1C2C3 N1(C(C(C)C)=O)CCCC(C(F)C(N2CCN(C(=O)C=CC(C)(C)C)CC2)=O)C1 c1(C(=O)NC2CCCC(N(C(C3=C(C)CCC3)=O)C)C2)ccnc2ccccc12 N(C(=NCc1snnc1C)NCCCCC(=O)Oc1ccccc1C)C(C=C)C C1(NC(CC2(C)CC2)=O)(CNC(=O)COC2(C=O)CC2C(C)C)CCOCC1.CO CC(C)CC(C)(C)C(=O)NC1CCCC1CNC(C1CCOCC1)=O c1(C(=O)NC(CC)CN(C(=O)Cc2cnnn2C)C)ccc([N+](=O)[O-])cc1Cl C=CC(C)(C)CC(=O)N1CCC(C(=O)NCCc2cnn(C)c2)C1CC CC(C)(C)CC(O)C(=O)NCC1C=CC(NC(=O)CCCn2cccn2)C1 c1(C(N2CCCC(CCNC(C(C(C)O)(C)C)=O)C2)=O)cn2cccnc2n1 C(C(C(C)(C)C)NC(c1onc(Cl)c1C)=O)NC(c1ccn(C(CC)CC)n1)=O C(CC1CC1)(CC(=O)N1CCCC1C(O)CO)NC(=O)CC1CC=CCC1 C12CN(CC(C)(C)C1)c1nccc(n1)C(=O)N2.c1(C(C)=O)cc(C(F)(F)F)no1 c1(CC)cc(=NCC2CCCCC2NC(c2cccc(NC(N)=O)c2)=O)[nH]cn1 c1(CNC(c2n(CC)ccn2)=O)ccccc1CNC(C1CC1(C)CC)=O N1(C(Cn2ncc(CC)c2)=O)CCC(NC(c2cccc(OC)c2C)=O)C(C)C1 C1(NC(c2c(C)n(CC(C)C)nc2)=O)C2CCN(C(=O)C3=CCCC3)CCC12 CC1CCN(C(=O)Cn2nccn2)CCN1C(c1ccc(C#N)cc1)=O c1(CC)cc(C)c(NC(c2nnnn2C2(C)CC2)C2C(CC3CC3)C2)[nH]1 C(N=c1[nH]nc(-c2ccon2)s1)C1CN(C(C(C)n2cccn2)=O)C1 Cn1cnnc1C(=O)NCC1CC1CNC(c1cc(-c2cccnc2)no1)=O C1(OC)CC2CC(C1)N(C(c1cc(-c3ccc(Cl)cc3F)on1)=O)C2 CC1=C(C(=O)N2CC(C)N(C(=O)Cc3cn(C)nc3C)CC2C)C(C)(C)CCC1 CCC(CO)(C(=O)OC(c1ccc(C(=O)OC)cc1)C)OC CN1CC2CN(C(c3ccc(-c4ccnn4C)cc3)C(=O)NC(C)(C)C)CC2C1 N1(C(c2c(COC)cc[nH]2)=O)C2CCC(C2)C1C(=O)NOCc1ncc(C)[nH]1 c1(C(c2nnnn2CC(F)F)NCC2(OCC)CC2)csc(C2CCCO2)n1 N1(C(CCN(C(=O)CC2C(=O)NN=C2C)CC=C)=O)CCCCC1CC(N)=O C12(C(=O)NC3(CNC(Cc4c(C)noc4Cl)=O)CC3)CCCCC(=O)N1CCC2 n1(CC)ccc(C(=O)N(CCC(=O)N2CC(N3CCCCC3)C2)CCOC)n1 N1(C(Cc2cnc(C)o2)=O)CC2CCCC1C2CNC(=O)CN1CCC(=O)NC1=O c1(N2CC3CN(C(=O)Cc4ccc(O)nc4)CC3C2)ncc2c(n1)CCOC2 C1(CC=C)(C(=O)NCc2cc(CC)no2)CCN(C(C2CCSC(C)C2)=O)C1 N1(C(CC(CC)SC)=O)CCN(C(c2cnc(C(C)C)[nH]2)=O)CC1C(C)C C1(Nc2cnc3cc(C)[nH]c3c2)CN(C(C2(OC)CC2)=O)C2(CCOCC2)C1 C1(C2C(NC(C(C)C#N)=O)CCO2)CCN(C(=O)CCCn2ccnc2)CC1 C1(NC(C(C=C)O)=O)Cc2ccccc2C1NC(c1cnn(C(C)(C)C)c1N)=O N1(C(c2n(CC#C)ccc2)=O)CC2CC1(CNC(c1cc(SC)c(C)o1)=O)C2 Cc1nc(-c2ccccc2)oc1C(=O)NCCCNC(=O)C(C(C)O)NC(N)=O c1(N2C(CNC(C=CC=CC)=O)CN(C)CC2)ncnc2c1nnn2CC N1(c2nc(OC)nc(C)c2)CC(CNC(=O)C(C)C2CCOC2)OC(C)(C)C1 N1(C(CC2CCN(C)C2=O)=O)C2CCC(C(N3CC=CC3(C)CO)=O)C1CC2 CN=c1ccc(C(=O)NC(c2cn(C)nn2)C(N2CCOC3CC23)=O)c[nH]1 Cc1cc(C(=O)NCC2CN(C(=O)C(C)(C)CF)C2)oc1C C(=O)(C#CC1(C)CCCO1)N1C(C)CCC(NC(c2c(C)cn(C)n2)=O)C1 C1(CC)CN(C(=O)Cc2cncnc2)CC1NC(c1cc(-c2ccco2)[nH]n1)=O C(=O)(C(F)CC(C)(C)NC(C1CCCC(=O)CC1)=O)NC(CC)C(N)=O CS(=O)(=O)CCCCCNC(C12CC(CC(F)F)(C1)C2)=O c1(C(N2CCC(O)(CCNC(c3cnc(OCC)s3)=O)C2)=O)ccc(Cl)c(F)c1 C(C1CCCN1C(=O)Cc1ccnc(O)c1)=CC(=O)NCC(CC)(C)O n1(CCCOCC)cc(C2CC(NC(C3CCC(SC)C3)=O)C2)nn1 C1(C(=O)NC(CO)CCC2CC2)(CC)CCCN1C(c1sncc1C)=O C12(C(N3CC(C)(NC(c4cc(C)sn4)=O)C3)=O)CCCC1C2(F)F N1(C(C(CCNC(=O)C2=CCCC2)O)=O)Cc2cncnc2C1 c1(N(CC(CN(C)C(=O)Nc2ccccc2C(C)(C)C)O)C)ncc(O)cn1 C(=O)(N=c1cc2n([nH]1)CC(C)(C)OC2)N(CC1(F)CCN(CC(C)C)CC1)CCO C(=O)(C(C(=O)OC)N(C)C)NCC1OCCC1C(=O)NC(COC)CO C(=O)(C(C(C)(F)F)c1ccccc1)NCC1(O)CN(C(CC(C)C)=O)C1 C1(CC)CN(C(=O)Cc2sc(S)nc2C)CCC1NC(=O)C1=CCOCC1 CC1CC(C(=O)NCCc2cc(C(=O)NCc3ccc(O)nc3)no2)CCS1 C1(C(=O)NC2(C)CN(C(c3coc(CS(C)(=O)=O)n3)=O)C2)CC2CCCCC2O1 c1(OC)cccc(F)c1C(=O)NCC12CCC(CN1C(=O)C(C)C(C)C)C2 C=CCC(CNC(C1CC2CC2N1C(C1CCCN1C(C)C)=O)=O)CC(C)C c1(SCCC(=O)NCCN(C(c2cnn(C3CC3)c2Cl)=O)CC)ccc(F)cc1 Cn1cc(NC(=O)CC2CCCCN2C(=O)Cn2cc(CO)nn2)c(Br)n1 c1(C(=O)NCC(C)NC(=O)C(C)(C)O)ccc(N2CCC(C)C2)cc1 C(=O)(C1=CC(C)C1)N(CCNC(C1(NC(C)=O)CCC1)=O)C1CC1 CC(C)CCCC(=O)N(CCNC(=O)C(C)NC(=O)NC(C)(C)C)C(C)C C1(CNC(C2(C)CC2(F)F)=O)CN(C(=O)Cc2ccc(F)cc2)CC1CC1CC1 c1(C(=O)NC2C(CNC(C3C(CCOC)C3)=O)C2)cnc2n1CCOC2 C=CC1CN(C(=O)CSc2nccn2C)CC1NC(=O)CN1CCN(C)C(=O)C1 c1(C(N(c2nccc(SC)n2)C2CNCC2F)=O)ncc(F)cc1C Cc1cc2sc(C(=O)NCC3(O)CN(C(=O)CSCCN(C)C)C3)cc2s1 N1(C(c2nn(CC)nc2Br)C(=O)NCCOC)CCOC(C)(CC)C1 N1(C(C2(F)CCN(C(C3CC(C)C3)=O)CC2)=O)CCC2(CNC(=O)N2)C1 c1(CC(C(=O)NCc2c(C)non2)NC(C2CC(O)(CO)C2)=O)cnn(C)c1O CC1OCCN(C(C23COC(C2)C(NC(c2cnn(C(F)F)c2)=O)C3)=O)C1CO c1(C(N(C2CCN(C(=O)C(F)(F)CC)C2)CCC)=O)c[nH]c2cccnc12 N#Cc1nc[nH]c1C(=O)NC1CN(C(=O)C=CC2CCC2)C1 Cc1ncc(Cl)cc1NC(=O)CC1CN(C(C2CC(C3CC3)C2)=O)C(C)(C)C1 c1(C(=O)NCC2CN(C(CC(C)OC)=O)CC2C)cc2nc(F)ccc2o1 C1(C2CCN(C(=O)CC(CC)c3ccc(C)cc3)C2)(NC(C(F)=CC)=O)CC1 CC(O)C(C(=O)NC)NC(=O)OC(C)(C)C.C1(O)CCN(C(C2CCCS2)=O)C1.C1CC1 C1(C(=O)Nc2ncc(OC)nc2)CC(F)CN(Cc2c(Cl)cncc2Cl)C1 C1(OCC)CN(C(=O)C(=O)NCCC(C)(C)C(=O)O)CC12CC2 C(=O)(C1=CCC(C(F)(F)F)OC1)NCC1N(C(CCC#C)=O)CCCCC1 CC(Cc1ccco1)C(=O)NC(CO)C(C)NC(C1(C2CCCO2)CCC1)=O C1(c2ccccc2)(C(=O)NCCC2CC(NC(c3cn[nH]c3)=O)C2)CCCC1 c1(C(CNC(=O)CC2CSC2)CNC(=O)CCC2CC2(F)F)ccccc1 c1(C(=O)NCCCN(C(CCC2CCC(C)O2)=O)C)n[nH]c2c1CS(=O)(=O)CC2 Cn1cc(NC(=O)NCc2ccnc(N3CCCCCC3)c2)nc1-c1ccccc1 c1(C(N2CCCCC(CN)C2)=O)cc(C(F)(F)F)ccc1Cl CC1C=C(C(=O)N2CCC(CC(C)NC(=O)CCn3cc(Cl)cn3)CC2)CC1 N1(CC#C)CCC(C(=O)NC(CNC(C2CC3CC3C2)=O)C2CCC2)CC1 C=C1CC(C(=O)N(CC(=O)NC(C)(C)C)CCC)N(C(=O)C(C=C)C2CCC2)C1 N1(C(CCC#C)=O)CC(CNC(c2cnn(C3CC3)c2)=O)CC1(C)C C1(C(=O)NC2C(CC)CN(C(c3ccc(OCOC)cc3)=O)C2)CCC(F)(F)CC1 c1(C(=O)NC2CCN(C(COCC)=O)C2)cccc(-c2nc(=O)o[nH]2)c1 c1(C(C(N2CCC(N(C(c3ccc(SC)o3)=O)C)C2)=O)C)ccc(Br)cc1 Cc1ccc(CNC(C2CCC(NC(=O)C=CCBr)CC2)=O)cc1 C1(CC(=O)NCC2CC2(F)F)CN(C(C2CCC(=O)O2)=O)CCO1 c1(N(C2CCCC23CCNCC3)C(=O)CC2CCCO2)c(Cl)ccc2c1OCO2 CCC(CC)(C(=O)NC1CCCC1NC(c1coc(C2CCC2)n1)=O)OC N1(C(C2OCCN(C(c3c(CC)ccs3)=O)C2)=O)CC2CCCC2C1 C(=O)(CCCCCCCC)N1CC(NC(CCCC=C)=O)C(C=C)C1 C#CCC(O)C(=O)NC(C1CCN(C(=O)Cc2csc(COC)n2)C1)(C)C N1(CC)CCOC(C(N2CCC(C)C2CNC(=O)C(C2CCCO2)C2CC2)=O)C1 CC(C)CC(C)(CNC(=O)CC1CCC(=O)N1C)NC(=O)CN1CCOCC1=O N1(C(c2cocn2)=O)CCC(C2CCCN2C(c2cnco2)=O)C1 N1(CC(=O)OCCc2nnc(NCCC3CCOCC3)s2)CCS(=O)(=O)CC1 c1(CN2CC3C(C(=O)Nc4cncc(Br)c4Cl)C3C2)ccc(Br)c([N+](=O)[O-])c1 Cc1ccc(C(=O)OC2(CNc3ccccn3)CC2)cn1 c1(C(=O)NC(c2cn(C)nn2)C(=O)NCc2c(C)ccs2)c[nH]ccc1=O c1(C(N(CC(CN(C)C(c2ncccc2Cl)=O)O)C)=O)snc2ccccc12 Cc1ccc2c(c1)C(C(=O)NC(C)CNC(=O)C(C)(C)C(C)O)OCC2[N+](=O)[O-] C(c1ccco1)=C(C)C(=O)N(CCC(=O)NCC1CC(CO)CO1)C1CC1 C1(C(=O)NC2CN(C3CCCCC3)C2)CCC(O)CN1C(c1ccc[n+]([O-])c1)=O C12(NC(c3cn(CCOC)nc3)=O)COCC1CN(CCC1CC1(Cl)Cl)C2 c1(C(N2CCC(C)(NC(=O)CC3CC4CCC3C4)C2)=O)ccc2c(c1)COC2 CC1(C)CC(NC(=O)CC2CCC2)CN(C(=O)C#CC2CCCC2)C1 C=CC(C)(CCOC)C(=O)NCC1(C2CC2)CCN(C(c2cc(CO)on2)=O)C1 C1(C(=O)NCCCOCCCC)C(O)CCN1C(=O)C(COC)OC CC(C)(C)CCCCC(=O)N1CC2COCC2(C(=O)NOC(C)(C)C=O)C1 C(=O)(CCS(N)(=O)=O)N1CC(OC)C(NC(=O)C=Cc2ccncn2)C1 c1(C(C(=O)NCC)N(CC(C)C)CC)cnn(CC)c1C CCCCS(=O)(=O)N1CCC(C(=O)NCC2CCCN2C(c2cn[nH]c2)=O)CC1 Cc1cc(=NCC(C)N(C)C(C2CCC3(C2)CC3(F)F)=O)[nH]cc1C#N c1(CN2CC(C)(C(N(CCC)CCC)=O)C2)nccnc1Cl C(C1CC1)(C1CC1)=CC(=O)NCC1C(NC(c2scc(C(N)=O)c2)=O)CCC1 C1(NC(C(CC)CO)=O)CN(C(c2ccc(Cl)c(OC)c2)=O)CCC1CO c1(CNC(c2c(-c3ccc(NC)cc3)nccc2)=O)nc(Cl)ccc1F c1(CNC2(CO)CC(F)(F)C2)ccc2ccc(Br)cc2c1 C(C)(C(=O)NCC(C1CCN(C(C2CC(OC)C2)=O)CC1)(C)O)(C(C)C)OC N1(C(C2(CC=C)CC=CC2)=O)CC2COCC(C1)C2NC(C1CCSCC1)=O c1(SC)cncc(C(=O)NCC2CC2CNC(c2cc(C)n(C3CC3)n2)=O)c1 c1(CC)cc(CO)ncn1.C1(=O)C(C2(C)CC2)OCCN1.C1(C(=O)C)CC(OC2CC2)C1 N1(C(c2ncn(C(C)C)c2)=O)CCC(NC(=O)COCC2CC2)C(F)C1 C(C1=NOC2COCC12)Nc1c(F)ccc(C)c1 C(=O)(C(C)CC(F)(F)F)NC(c1nc(C(N2CCC(O)C(O)C2)=O)co1)C C(C(F)(F)C(C)(C)O)NC(C(CCC)NC(c1ccnn1CCF)=O)=O c1(NC(CSC(c2ccc(OC)c(OC)c2)CC)=O)cc(Cl)ccc1CO N1(CC)CCCC(ONC(=O)C2CC2CNC(c2ccsc2)=O)C1 c1(NC(=O)C(c2cccc(Br)c2)N2CCOC(C3CC3)C2)cc(F)c(F)cc1F c1(-n2c(CC)nc(C(C)OCC)n2)ccc2nc(N3CCOCC3)[nH]c2c1 CC1CC(NC(c2ncn3c2CCC3)=O)CN(C(=O)Cn2ccc([N+](=O)[O-])n2)C1 N1(C(c2c(C(C)C)cccc2)=O)CCC(NC(=O)CSc2nc[nH]n2)C(C)C1 c1(OCC(=O)NC(C2N(C(c3ccc(CSC)o3)=O)CCC2)C)cnc(Cl)cn1 C(=O)(CC1CN(C)c2ccccc21)N1CCCN(C(c2c(C)nns2)=O)CCC1 C1(CNC(CP(C)(C)=O)=O)CC2(CO1)CN(C(c1ccccc1Br)=O)C2 c1(CC2(CNC(c3n(CCC)nnn3)C3CC3)CC2)ccc(Br)cc1F N1(C(=O)NC(C2CCC2)C2CC2)CCCC(C2CCCO2)C1 CCC(CC(=O)NCCCCCCN(C(=O)C(COC)CC(C)C)C)C(C)C C(CN=C(NCCF)NC1CCN(CC2CC2)CC1)c1ccc(C(N)=O)cc1 N1(C(c2c(OC)ccs2)=O)CC2(C(=O)NC3CC=CC3)CC1CCO2 C(=O)(CS(=O)(=O)CCO)N(CCN(C(=O)C(F)(Cl)c1ccccc1)CC)CC CS(=O)(=O)c1cnc(N2CCCC3CN(C(=O)C(N)=O)CCC23)c(Cl)c1 C1(C(=O)NCC2(CC)CCCC2)CC2CCC1N2C(c1cccc(OC)c1O)=O Cn1cnc2cc(C(=O)NC3CN(C(=O)CC4CCCC45CC5)C3)cnc12 c1(CNC(Cn2cc(CC(C)(C)CO)nn2)=O)ccc(F)cc1 c1(CC(C(C)OC)=O)ccc([N+](=O)[O-])cc1 c1(C(=O)NC2CN(C(c3occ(OC)c(=O)c3)=O)CC2C)ccc(O)c(Cl)n1 CCCC(C(=O)OC)C(=O)N1CCN(NC(c2ccc(OC)nc2)=O)C(C)C1 S(=O)(=O)(c1ccc(NCC(C)(C)C#N)cc1Br)N1CC(CO)CC(C)(C)C1 C1(C(N(C2CCN(C(C(n3cc(Cl)cn3)C)=O)CC2)C)=O)CCC2(CCCC2)C1 C12(CNC(c3cc[nH]c3)=O)CCC1CCN2C(c1ccc(-c2cccs2)cn1)=O C12(C(C)=O)COC(CNC(=O)NC3CCC(C)CC3)(C1)C2 c1(C(=O)NCC(CN(C)C(C2CC(F)C2)=O)O)cc(Cl)ccc1O N=c1nc(C2CC2)nc(N2CCC(F)(CNC(=O)CNC(c3ccco3)=O)CC2)[nH]1 CCCC(C(=O)OC)C(=O)NCC1CCN(C(=O)COCc2ccccc2C)C1 C=CC1(C(=O)N(CC(CC)NC(=O)C(C)OCC(C)C)C)CCC1 N1(C(CC2(C=C)CCC2)=O)CCCN(C(c2cccn2C2CCCC2)=O)C(C)C1 O=C(C1CCc2scnc21)NCC1CC2CC2N1C(c1cc(Cl)ncc1O)=O N1(C(CCC)=O)CCCCC1C(N1CC(NC(C2CCC2(C)C)=O)C(C)C1)=O N(C(=NCC1CCCO1)N)C1C(O)CCC1.c1(CN2CC=CC2)ccc(F)cc1 c1(OC)nccnc1C(=O)NC1CCCC(NC(=O)CCSc2ccccc2)C1 N1(C(C2CC=C(C)CC2)=O)CCC2(CC1)CC(Nc1ncnc(O)c1Br)CCO2 c1(C(COC(=O)CC2CCc3ccccc3C2=O)=O)cc2ccccc2oc1=O c1(C(=O)NC2CC(N(C)C(c3ccco3)=O)C2)cc(Cl)nc(Cl)c1 N1(C(CC(C)C)C)CCC2CC(C(=O)NCCN3CCCC3=O)C2C1 c1(SCC)conc1CC(=O)NC(CC1CC1)C(=O)NC1CC1c1ccco1 C12(NC(c3nc(CNC(c4cc(C)[nH]n4)=O)oc3C)=O)CCC(C1)C(O)C2O N1(C(C(C)(O)C2CC2)=O)CCOC(CNC(c2nocc2C2CCC2)=O)C1 c1(C(N2C(C)CCC(NC(c3occc3C3CC3)=O)C2)=O)ccn2nccc2n1 c1(CC)[nH]nc(C(N2CCC(NC(C34CCC(C3)C4)=O)C2C2CC2)=O)c1Cl C1(C(N2C(CNC(C)=O)CCC2)=O)CCCN1NC(=O)c1ccc(N)cn1 C(=O)(CCCC(F)(F)F)NCC1(C(N2C(C(=O)NC)CC(O)C2)=O)CC1(C)C c1(NCC(=O)NCc2cn(CC(=O)OCC)nn2)ccc(Cl)c(C)c1 c1(OC)c(F)ccc(C(=O)NC2CCCC2CNC(=O)CC2CSCCO2)c1F CC#CCCCC(=O)NCC(C1CCCCN1C(=O)C(C)=CC1CC1)(C)C C1(C(N(CC(C)OC)C(C)C)=O)CC2(CC(NC(=O)COC3CCCC3)C2)C1 C(=O)(C(C)(O)CCC)NCCN(CCCCCC)C(c1cnc(C(C)OC)s1)=O c1(C(N2CC3CN(C(c4scc(CC)n4)=O)C3C2)=O)cc(F)cc(Br)c1F c1(OC)ncc(C(=O)NC(c2ccccc2Br)CNC(C)=O)c(C)n1 c1(C(N(CC(C)(C)NC(c2c(OCC)nccc2)=O)C)=O)ccc(C)c(Cl)c1Cl Nc1cc(F)c(Br)cc1C(=O)NC1CCCN(C(=O)C=Cc2cnc[nH]2)C1 c1(C(N(CCC(=O)NC(C=C)(C)C)C)=O)cc(C)c(CC)o1 C1(C(N2C(CNC(c3ccc4c(n3)CCC4)=O)CC2)=O)CC2CC1CC2(F)F C(C(C)N=c1nc(C)cc(C)[nH]1)NC(C1CCC(C)(CC)O1)=O Cc1cccc(C(N2CC3(CC3C(=O)Nc3ncn(C)n3)C2)=O)c1F C1(CCC)(NC(c2cn(CCO)nn2)=O)CCCN(C(c2cc(Cl)cnn2)=O)C1 c1(CNC(C(C(=C)C)(C)O)=O)nc2ccccn2c1C c1(C(N2CC(C)(NC(C(C(C)C)SC)=O)C2)=O)cccc2c1CCCN2 C1(NC(C(c2ccc(F)cc2F)(C)C)=O)CN(C(c2nonc2N)=O)CC1(C)C S(=O)(=O)(c1ccccc1F)NC1C(C(N2CC3CCCCC3C2)=O)C1 N1(C(C=CC(C)(C)C)=O)CCC2(CC1)OCCC2NC(=O)CCC(F)F N1(C(C=Cc2cccc(C)c2)=O)CCC2(C=C(C(=O)NCC3(Cl)CC3)C2)C1 Cc1cn2c(n1)CCC(C(=O)NCC1(NC(c3cnoc3C)=O)CCCC1)C2 c1(C(C(=O)NCCC(C)(C)NC(=O)Cc2cnoc2)O)ccc(Cl)c(Cl)c1 C1(NC(Cc2c(C)nc(S)s2)=O)CC2CN(C(c3c[nH]ccc3=O)=O)CC2C1 Cc1cccc(F)c1CNC(C12COC(C1)C(NC(=O)COCCCN(C)C)C2)=O C123CCC1CN(C2)N3C(CS(C)(=O)=O)=O.C1(C(N2CCCC2)=O)CC12CCC2 c1(OCC)nc(C(=O)NC(C)(CNC(C2CC2(C)Br)=O)C2CC2)co1 N1(Cc2[nH]c(=NCC=C)sc2)CCS(=O)(=O)C(C)(C)C1.c12ccc(cc1)s2 c1(NC(N2CC(CC(=O)Nc3csc(O)n3)C2)=O)ccc(Cl)cc1[N+](=O)[O-] N1(C(CN(C(C)CN2CCCCC2)C(C)C)=O)CC(F)CC1CO C1(CC)C(NC(=O)CCN(C)C)CCCN1C(=O)C(=O)NCCC(C)(C)C C1(NC(CN(C(CC(CC)C#N)=O)CC2CC2)=O)CC(C)CC(C)(C)C1 c1(CN2CC3CC(NC(C4C(C)C4)=O)CC3C2)cccc(S(C)(=O)=O)c1 Cc1ncc(C(=O)NCCCCC(=O)NCC2CC[Si](C)(C)C2)n1C C(=O)(C(C)(C)CCC#N)N(C(=O)C(C)CNn1cc(C2CC2)cn1)CC c1(CC(=O)NCCCC(C)NC(=O)CCN(S(C)(=O)=O)C)nnc2n1CCOC2 C1(C(N2CCN(C(CCCC=C)=O)C(COC)C2)=O)Cc2ccncc2C1 C#Cc1ccc(C(=O)N(CC(C)NC(c2cnc(C)cn2)=O)C)c(C)c1 c1(C(N(CC(CC)NC(C2C3CC4C(C3=O)C24)=O)C)=O)cccc2cnsc12 C1(CCC)CN(C(=O)CC2CCC2)CCN1C(c1cn(CC2CCCO2)nn1)=O C1(C(=O)NCC(=C)F)CNC(=O)CN1C(C1CC(CC)C1)=O C1(N(C(c2c(C)c(-c3ccccc3)[nH]n2)=O)C)CCCCN(C(=O)CC(C)F)C1 CC(C)(C)C#CCCNC(=O)CC1CCCN(C(C2(C)CCCOC2)=O)C1 CC1(C)C2CCC(C2)C1C(=O)NC1(CNC(C2CC=CC2)=O)CCOC1 c1(C(=O)NCC2C(CNC(=O)Cc3ccno3)C2)nc2cccnc2s1 Cc1nocc1C(=O)NC1CC(NC(=O)C(c2ccccc2)C)C1 c1(C(N(CC(C)C(=O)N(CC(C)(C)C#N)C)C)=O)c[nH]nc1[N+](=O)[O-] c1(C(N2CCCC(CCNC(C(CC=C)C)=O)C2)=O)c(N)ccc(F)c1F C1(C(N(C2CCN(C(=O)CN3CCOC3=O)CC2)CC)=O)CC(=O)N(C2CC2)C1 N(C(=NCC1CNC(=O)C1)NCC1CCOC1)CC(C)(C)OC c1(C(=O)NCC(CNC(C(COC)(C)C)=O)(C)C)ccc(C)c(-n2cccc2)c1 C1(C(N(C)Cc2cccc(C#C)c2)=O)CCn2nccc2C1 c1(SC)cc(F)ccc1C(N1CC2CCCC12)=O C1(CNC(CCCOCC)=O)CCC(C)CN1C(=O)CSc1cc(Cl)ccc1Cl C(=O)(CC1CC(C)c2c(C)cccc21)N(CCN(C(CC(=C=C)C)=O)C(C)C)C c1(CNC(C(c2cncnc2)C)=O)cccc(C(=O)NC2(C)CCCO2)n1 c1(CC)cc(C(=O)NC(C)CN(C)C(c2cccc(CC)n2)=O)ccn1 N1(C(CC2(OC)CC2)=O)CC2CCC(CNC(C3CC34CC(C)(C)C4)=O)(C2)C1 c1(OC)ccc(F)cc1NN(C)CCCCc1ccc(O)cc1 N1(C(CCN(C(=O)CC2CCCCCC2)C)=O)CCCC(O)(C2CC2)C1 C(=O)(C1=CCCC1)N1CC(CC=C)(C(=O)NCCOC)C1 C1(COC)CN(C(c2csc(C3CC3)n2)=O)CCN1C(C1CCC2CCC1O2)=O c1(CC(=O)NC2CC(CNC(CCCSC)=O)C2(C)C)ccc(C#N)cc1 c1(CC(=O)N(C(C)C(=O)N2CCC2C2CCC2)CCC)cc(C)nn1C c1(C(=O)NC2CCN(C(c3c(C)cc(Br)o3)=O)C2)cc2c(F)cccc2[nH]1 Cc1nc(Cl)ccc1CC(=O)NC(C1(CNC(c2cn(C)c(=O)cn2)=O)CC1)C c1(CC(=O)NCC(C)(C)OCCNC(C(CC)(C)O)=O)ccc2scc(C)c2c1 CN1CCCC(CCn2c(N3CCC(CCN(C)C)C3)nnc2C2CC2)C1 CC1CSCCCN1C(C1(CNC(=O)Cn2nccn2)CCC1)=O N1(C(c2cnc(CC)s2)=O)C2CCC1C(C)C(NC(=O)CC1CC1(C)C)C2 CCCC(CC(C)C)C(=O)N(C1(C(N2CC3CC3C3CC23)=O)CC1)C N1(C(C(CCCC)O)=O)CCC(C)N(C(=O)CC2CC(C3CC3)C2)CC1 N1(C(c2noc(CC)c2C)=O)CCC(NC(=O)C(F)=CCCF)C(CC)C1 C=CCC(CC(F)F)C(=O)NC(C)(CNC(=O)C1CC1)Nc1cc(C)nc(C)n1 c1(C(N(c2ccc(OC)cc2)CCC#N)=O)nccc(Cl)c1Cl CC1CC2CN(C(c3cc(F)c[nH]3)=O)CC2N1C(C1COCCN1CC(F)F)=O c1(C(=O)NCCCN(C(C2C(CC)CCC2)=O)C(C)C)cnc2ncccn12 c1(C(C(=O)NCSc2ccccc2)N(CCC(=O)OC)C)ccc(NC2CC2)cc1 CN1CCC(NC(C2(C3CC3)CN(C(=O)COCCCN(C)C)C2)=O)C(C)(C)C1 Cc1ccn2cnc(C(=O)NCC3(C)CCN(C(C4(C5CC5)CCC4)=O)C3)c2c1 Cc1onc(C(F)(F)F)c1C(=O)NC(C)CNC(C1(O)CC1(C)C)=O Cc1cc(C(=O)NCC2CC2NC(=O)Cc2ccn(C)n2)cc2ccsc12 C1(C)(NC(C2OCC(C)(C)C2)=O)CCCN(C(C2(c3ccc(O)nc3)CC2)=O)C1 Cc1ccc(C(N2CCCC(c3ncc[nH]3)C2)C(=O)NC2CCC2)cc1F C1(NC(c2csc(-c3ccoc3)n2)=O)CN(C(c2cc[nH]c2)=O)C2(CCC2)C1 N1(C(c2c(C)nco2)=O)CCC(NC(=O)C(c2cc(F)ccc2F)(F)F)C(C)C1 CC1CN(C(=O)C=Cc2nccs2)CCC1NC(c1cncn1C)=O c1(NC(C(=O)NCC2CCNCC2)=O)cc2ccc(Br)cc2s1 N1(C(C(C)C)=O)CCN(C(C2CCC2c2cncn2C)=O)CC1 c1(C(N(C2CCN(Cc3c(Br)cc(Br)cc3Br)C2)C)=O)ccc(O)c([N+](=O)[O-])c1 Cc1nc2c(s1)CCCC2C(=O)NCC1CN(C(=O)C(n2ccc(C)n2)C)C1 C(c1ccccc1Cl)=CC(C)NC(CSC1CCCCCC1)=O CC1=CCN(C(C23CC2CCN3C(=O)CN2CC(=O)NC2=O)=O)CC1 c1(C(=O)NCCN(C(=O)C(N2CCOCC2)C)CCOC)ccc(C(C)(C)C)s1 CC1(C)COCCC1C(=O)NC1CCCC1CC(N1CCCC1)=O N1(C(c2ccc(C)nc2)=O)CCN(C(=O)CCCCNC(N)=O)CC1CC(F)F N1(C(c2cnc(C)o2)=O)CC(CC(=O)NC(C)Cc2cccnc2)C(C)C1 C1(C(C)C)CN(C(=O)Cc2cccc(F)c2Cl)CCN1Cc1ccc(I)cc1 C1(OC)CCCCC1C.c1(C(N2CC(=O)NCC2)=O)ccc(CSCC)cc1 C1(OC)CC(NC(=O)CCN2CCN(C)CC2)CN(C(=O)C(C)(C)CC2CC2)C1 N1(C(Cc2ncc(C)s2)=O)CCC(CN(C(=O)CCc2cccnc2C)C)CC1 C(=O)(C1=NOC(C)C1)N1CC(C)C(CNC(c2cc(Cl)ncc2N)=O)C1 C(=O)(CCC(=O)NC1CC(O)CN1C(c1cc(OCC)n[nH]1)=O)NCCC c1(C(N2CCN(C(C(C#N)C3CC3)=O)C(CCO)C2)=O)ccc2oc(S)nc2c1 CC1(C)CC=C(C(=O)N2CCOC(C(N3CCC(C4CC4)CC3)=O)CC2)CC1 C(=O)(C(C(C)C)c1ccccc1)NCCC(C)NC(c1c(CC)nc[nH]1)=O C1(NC(=O)CNC(c2ccccc2O)=O)CCCCN(C(c2cc(F)c[nH]2)=O)C1 c1(C(=O)NCC2(NC(=O)CC(F)(F)F)CCCCC2)cn2ncccc2n1 C1(C(N2C(CNC(C(CC)(O)c3cccc(Cl)c3)=O)CC2)=O)OC2CCC1CC2 c1(C(N2CC(O)(CNC(COC)=O)C2)=O)ccc(Br)cc1C#N CC1(C)CCOC1CC(=O)NC1CC(CCNC(=O)Cc2ccc(O)nc2)C1 C1(C(=O)NC2CC(CNC(C3(SC)CCC3)=O)C2)CCN(C)C1C C12(NC(CCCCC=C)=O)CCCC1N(C(=O)Cc1ccc3c(c1)COC3)CC2 N1(C(CCC(=C)C)=O)CCCC(F)(CNC(C2(OC)CCCSC2)=O)C1 C1(C)(C(N(CCOC)C)=O)CCN(Cc2cc(C)cs2)CC1 N1(C(c2c(C)n[nH]c2C)=O)CCN(C(=O)CSc2nncs2)CC2(CC2)C1 c1nc(Cl)sc1C.c1(OCC)cc(C(=O)Oc2ncc(CCCC(=O)N)s2)c[nH]1 c1(C(=O)NCCN2CCN(C(c3c(C)oc(Cl)n3)=O)CC2)cc(S(C)(=O)=O)cs1 c1(C(=O)NC(CS(C)=O)C(C)(C)C)ccc2c(c1)[nH]c1ccccc21 CC1OC2(CNC(=O)CNC(=O)NCC3CCNC3=O)CC1(C(N1CCCC1)=O)C2 C#CCCCOCC(=O)N(CC(=O)N(C)CCOc1cnsc1)CCOC C1(C(C)NC(=O)CSc2ccccc2)CN(C(=O)C2=NOCC2)CCO1 CCC(C#N)C(=O)NCCC1(C(=O)NCc2ncn(C)n2)CCC1 C(CC(=O)NCC1C=CCN1C(c1ocnc1C)=O)(C(F)(F)F)OC N1(C(c2cnc(OC)s2)=O)CC2CC1(C(=O)NCCN1CC(CF)C1)C2 N1(C(C2(CC)COC2)=O)CCC2CN(C(=O)C(C)(O)CC(C)C)CC2CC1 C1(N(C(C)=O)C)CN(C(=O)CCCOc2ccc(C)cc2C)CC1(C)C c1(C(N(C)CCNC(=O)CC2C=CCCC2)=O)ccccc1Cn1cccn1 Cc1csc(C(C)C(=O)NCCC2CN(C(c3csnc3Cl)=O)C2)n1 CCC(C)C(C)C(=O)N1CCOCC(CNC(c2cncc(F)c2Cl)=O)C1 Cc1cc(CC(N2CCCCC2CNC(=O)COC2CC2)=O)ccc1CO C1(NC(=O)CN2CCCC2=O)COC2(CNC(C3COC4(CCC4)C3)=O)CC1C2 N1(C(C(C(C)C)O)=O)CCC(CNC(=O)C(N2CCN(C)CC2)C)C(F)(F)C1 C1(C2CCN(C(C3CCCOC3)=O)CC2)(NC(c2cc(C#C)cc(F)c2)=O)CC1 C#CCCCC(C)C(=O)N1CC(O)(CNC(=O)C(O)CC)C1 Cn1ccc2cnc(N3CCCC3(C)C(=O)Nc3nc(C#N)cs3)nc12 c1(NCC2(NC(C3CCCCC3)=O)CC2)ncnc2sc(C(=O)O)cc12 CCCC(CC)CCC(=O)NCCOCCN(C(=O)C(C)(C)c1cc[nH]n1)C Cc1cc(C(N2CC(NC(=O)CCC(=O)c3ccc[nH]3)C(C)C2)=O)nc(C)n1 c1(C(=O)NC2CN(C(c3c(C)c[nH]c3CC(N)=O)=O)C2)cccc(C2CC2)c1C CCC(CC)(CCNC(c1ccc(C(F)F)cn1)=O)NC(C1CSCCS1)=O C1(NC(C(C)OCC#C)=O)CN(C(c2ccc(S(C)(=O)=O)[nH]2)=O)CCC12CCC2 C1(CNC(c2cc(C)oc2)=O)CCCCC1NC(=O)CCC1CC1 CN1CCC(C(=O)NCCC2(C(=O)NCC3(C(N)=O)CC3)CCC2)C1 c1(OC)cc(-c2ccccc2C)c(C(=O)OCc2cc(C(F)(F)F)no2)cn1 C1(CNC(c2occ(C)c2)=O)CC2(CCC2)CN1C(c1cc(N)c(C)cc1C)=O c1(NC(C2CCC(CNC(C(C)OCC)=O)CC2)=O)cc(Cl)cc(C(F)(F)F)n1 c1(OC)ccc(OCC(=O)NCC2CN(C(=O)CN(C)CCO)C2)c(Br)c1 c1(C2C(C(=O)OC)C2)ccc(=NCC2(C)CCC(=O)C2)[nH]n1 c1(CNCc2ccc(OCCCC)nc2)cc(OC)cc2cccnc12 C1(CN(C(CCSCC)=O)C)CCCN(C(c2cc(C3(C)COC3)no2)=O)C1 C1(C(=O)NCCN(CCC)C(c2oc(C3CC3)nc2C)=O)CC12CC(F)(F)C2 Cc1cnc2cc(C(N3CC(CNC(=O)CC4(C)CCC4)C(O)C3)=O)nn2c1 N1(C(=O)Cn2ccnn2)CC(F)(F)CC1C(=O)N(C1CC1)Cc1ncc[nH]1 N1(C(C2CCN(CC#C)CC2)=O)CCCC(C)C1CNC(C1(O)COC1)=O N1(C(C(COC)(C)C)=O)CCC(NC(C2CN(C)CCO2)=O)C(O)C1 C1(C(=O)NC(CNC(Cc2nnc(C)s2)=O)C(C)C)CCc2ncc(C)n2C1 CCC(CC(F)(F)F)C(=O)N1CC(NC(c2cc(Cl)ns2)=O)CCC1C c1(C(N2CCOCC(CNC(C(C=C=C)C)=O)C2)=O)ccc(Cl)c(C#N)n1 CC1OC(=O)NC1C(=O)NC1CC(NC(=O)CCSC(F)(F)F)C(O)C1 Cc1ccc(N)cc1C(=O)NCC=CCNC(=O)Cc1ccn(CC(C)C)n1 c1(C(N(C(C)CCNC(C2CCCCS2(=O)=O)=O)C)=O)ccc2c(c1)CCN2C c1(C(=O)NC(C(=O)N(C(CCO)C(F)F)CCO)C2CCCC2)ncn2c1CCC2 C(=O)(C(F)(CNC(c1cnccn1)=O)C(C)C)NC(CC)(C)CCO Cc1c(C(=O)NC2CC(C)N(C(c3ccc(C(C)(C)C)s3)=O)C2)sc2cncn12 c1(C(N2CC(NC(c3c(C)nc(O)[nH]3)=O)CC2(C)C)=O)ccn2nnnc2c1 c1(C(c2nnnn2CCCOC)NC(CC=C)C2CC2)csc(C(C)C)n1 CCCCCCC(=O)N1CCC(CO)C(NC(=O)C(C)OCC2CC2)C1.C N1(C(c2ccc(CC)o2)=O)CCN(N2CCC(C(=O)OC)CC2)CC1 C(=O)(C(F)(F)c1ccccn1)NCC(N(C(C(C)N(CC(F)(F)F)C)=O)C)C1CC1 C(c1ccccc1)=CC(C)C(=O)OCC1CC(N2CCCC2)CO1 c1(CC(N2CC(NC(=O)CC3CCC(C4CC4)O3)C2)=O)noc2ccc(O)cc12 C(CO)(CCCCNC(C1CCN(C)C1)=O)NC(c1c(C)[nH]nc1Br)=O CCC(C)(CO)C(=O)NCC1CCN(C(=O)CCNC(=O)OC(C)(C)C)C1C C=Cn1nccc1C(C(N1CCOCC1)=O)N(CC(=O)NCC1CCCO1)C c1(CNC(COCCCC)=O)cnn2c1CN(C(C1CCCN1C1CC1)=O)CC2 N1(C(C(C)NC(N)=O)=O)CCC2(CCCN2C(=O)CC2CCCO2)CC1 N1(CC(=O)NC2CN(C(=O)CCn3cccc3)C3CC23)CCCCS1(=O)=O C(=O)(C1=C(C)CCC1)NCc1cn(CC(C)NC(C23CCC(OC)C2C3)=O)nn1 CCCC(C)C(=O)NCC1CC(F)(CNC(C2(C(C)C)CC2)=O)C1 C1(=CC(=O)N(C2CCC(NC(C3CCS(=O)(=O)N3)=O)C2)C)CN2CCC1CC2 N1(C(C2CN(CC)C(=O)N2)=O)CC(NC(c2ccc(C(N)=O)o2)=O)CCC1C N(C1CC2(CN(C(=O)C(F)CC(C)C)C2)n2ccnc21)C(Cn1c(C)ncc1)=O c1(C(C(=O)NCC=CC2CC2)NC(CCOCC(C)C)=O)c(C)cccc1Br C1(NC(=O)CC2CCSCC2)CC2CCC1(CNC(=O)C(F)(F)C1CCCC1)C2 c1(OC)ccc2[nH]nc(C(=O)NCCCC(C)NC(C3CCOC(=O)N3)=O)c2n1 c1(COc2ccccc2)ccc(C(=O)NC2(C(=O)NCC(=O)NC)CC2)cc1F CC1=NS(=O)(=O)NC(C)=C1CC(=O)NCCNC(=O)C(C)Oc1cc(C)ccc1Cl C=CCC(CC=C)C(=O)N1CC=C(C(=O)NC(CC)C(C)COC)CC1 N1(C(C2N(C)CCC2)=O)CC2CC1(C(=O)NCC1(C)CCCO1)C2 c12cc(cc(F)c1)N2.CCCC(C)C(c1nnnn1SC)Nc1ccccc1C c1(NC(C2N(C(c3c(=N)cc[nH]c3)=O)C3C(C2)C3)=O)c(F)cc(Br)cc1[N+](=O)[O-] C1(C(=O)NCc2cc(C)no2)CC2CCCC2N1C(=O)C(C)(C)C C1(CC)CCCC(CN=C(NCC2(O)CCCCC2)NCC)C1 N1(C(c2c(C)ccnc2)=O)CCC2C(C(=O)NCC(F)(F)C(F)F)C2C1 C(=O)(CCC(=O)N1CCOCC1)NC(CNC(COC)=O)N(C)C(N)=O Cc1nnccc1C(=O)NC1CCC(CNC(=O)CCc2cccnc2Cl)CC1 c1(C(N2CCN(CCN(C(C)=O)C)CC2)=O)cc(C)c2ncccc2c1C c1(OC)ccc2c(c1)N(C(c1cnn3ccccc13)=O)CC2C Cc1cncc(C(=O)NC2CC(C(=O)NCCC3CCC(C)O3)CC2O)c1 CS(=O)(=O)C=CC(=O)NC1CCC(NC(=O)Cc2cnccc2C(F)(F)F)C1 C1(NC(CC2(C)CCCO2)=O)CCCN(C(c2cc(C3CC3)on2)=O)CC1 C(=O)(CCCCC1CC1)NC(C(=O)NCC1CCN(C)C1)C1CCOC1 c1(C(C)NCC(COC)C(C)C)ccc(OC)cc1C N1(C(c2c(C)scn2)=O)C2CCC1C(C)C(NC(=O)CCOc1ccccc1)C2 Cc1noc2ncc(C(N3CC(C(C)NC(c4cc(=O)cc(Cl)[nH]4)=O)C3)=O)cc12 N=c1nc(N2CCC(C(F)(F)F)C(F)(F)C2)[nH]c(=NC2CCCN(CCF)C2)[nH]1 N1(C(CS(CC)=O)=O)C2CCC1C(NC(c1ccoc1CC(N)=O)=O)C2 c1(C(=O)NCc2ccc(NC(C(C)n3cccc3)=O)cn2)cccnc1CO C1(NC(C2C=CC(NC(c3ccc(C#N)s3)=O)C2)=O)CC2(COCCO2)C1 C12(NC(c3scc(COC)c3)=O)CC(C1)N(C(c1ncsc1NC)=O)C2 C(C(C)(C)C(=O)Nc1ccc(-c2cncc(NC(C)=O)c2)cc1)NS(CC)(=O)=O c1(CNC(CN(C(=O)CC23CCCC2C3)CC)=O)csc(C)c1 c1(C(N2CC3CCN(C(C(CC)=CC)=O)C3C2)=O)cc2c(Br)cncc2s1 Cc1cc(C(=O)NCC2CCCCC2NC(c2nc(C3CC3)cs2)=O)cc(O)n1 C(C)(Cc1ccccc1)(C(=O)O)N(C(c1ccccc1F)C)Cc1ccco1 CNS(=O)(=O)N1CCC(C(=O)NCCN(C)C(C2CC3(C2)CC3F)=O)CC1 C1(CNC(CCSC)=O)CN(C(=O)CN(C)C(C)=O)CC(C)(C)C1 N1(CC(c2nnnn2C2CC(F)(F)C2)NC(C2CCCC2)C)CCCCC1 Cc1cnc(Cl)c(N(Cc2cn(C3CCCCNC3=O)nn2)CC2CCCO2)c1 C1(NC(C(C)C(=O)OC(C)(C)C)=O)CC2CCC(C1)N2C(=O)CCC(N)=O C1(CNC(CCC=C)=O)CN(C(=O)CC2CCOCC2(C)C)CC1C=C c1(C(=O)NCC(C)N(C(=O)Cc2ncc(Cl)s2)CC)ccc2ccnc(O)c2n1 c1(C(=O)NCCC2CN(C(=O)CCCF)CCO2)cnc(O)c2cncn12 Cc1c(C(=O)NC2CC(C)N(C(=O)Cn3cnc([N+](=O)[O-])n3)C2)cccc1N N1(C(c2n(CCC)ccc2)=O)CCN(C(C2C(C)(C)C2(C)C)=O)CC1CCO c1(C(N2CC(C)(CNC(c3ccccc3-c3ncc[nH]3)=O)C2)=O)cc2scnc2[nH]1 C1(NC(C(C)NC(CC)=O)=O)CCCOC12CCN(C(=O)C=CBr)CC2 N1(C(CNC(C(CC)O)=O)=O)CCc2nc(C(=O)NC(C)C)sc2C1 N1(C(=O)COC2CC2)CC(NC(C2(CC3CC3)CC2)=O)CC(O)C1.C1(O)CCC1 c1(SCC(=O)N(CC(C)NC(C2(C)CC2c2ccccc2)=O)C)cccc(F)c1 Cc1noc(C)c1C=CC(N1CC(C)(C)CC1CNC(C1CC(=O)N(C)C1)=O)=O C(=O)(C1CCCc2n[nH]cc21)NC(C1CN(C(C2CC(C)(C)C2)=O)C1)C C(=O)(C1=CCC(C)CC1)NC(CNC(c1c(C)occ1-c1ccccc1)=O)C [N-]=[N+]=Nc1cncc(C(N2CCC3(CNC(=O)CSC(F)(F)F)CCCC23)=O)c1 CC1CC(C(=O)N(CCCNC(=O)Cc2ccns2)C2CC2)CC(C)C1 C1(C(N2CC3C(NC(=O)CSCC4CCCCO4)(C3)C2)=O)CC12CCSCC2 CC1(C)C(O)CC1(N)C(=O)NCCCCc1nccs1 Cc1cccc(-c2cn(C3CC(C(=O)NCc4cc(Cl)c[nH]4)C3)nn2)c1 Cn1cc(C2=NOC(C(=O)NCCCCNC(=O)Cc3ncncc3Cl)C2)cn1 C1(C(=O)NCCCCNC(C2(C(=O)OCC)CC2C)=O)CN2CCN1CC2 C(=O)(CC1=NN(C)C(=O)C1)N(CC(CC)NC(c1cc(C)c(Cl)cn1)=O)C C1(NC(Cc2ccn(C)n2)=O)CCCCN(C(c2cc(N)c(Cl)c(O)c2)=O)CC1 C1(CNC(C(CC)OC)=O)CN(C(=O)CN(C)C(N)=O)CC12CCC2 Cc1nn2cc(C(=O)NC3CCC4CN(C(C5(C(C)(F)F)CC5)=O)CC34)nc2s1 C=CC1(C(=O)NC2CNC(=O)C2)CCN(C(c2cccc[n+]2[O-])=O)CC1 C1(NC(C)=O)CCN(C(=O)NCC(CCSC)(F)F)C(c2ccccc2)C1 c1(CC(=O)NCC2CCCN(C(C(CC)(C)O)=O)CC2)ccc([N+](=O)[O-])c(N)c1 C1(C(=O)NC2CCN(c3nc(C4CCOCC4)ns3)C2)CC12CCC(F)(F)CC2 c12nc3onc(-c4ccccc4Br)c3c(=O)n1C2.Cc1ncc(CO)n1C(F)F c1(C(N(C2CN(C(C(C)NC(N)=O)=O)CC2O)C)=O)cc(Cl)c(Cl)n1C c1(OC)ccc(C(=O)NC2(C)CCN(C(C3CCN3C3CCCC3)=O)C2)c(C)n1 C1(NC(CC(COC)COC)=O)CN(C(=O)Cc2cc(OC)no2)CC2(CC2)C1 C(=O)(CCCCCCS(N)(=O)=O)NC(C1CCN(C(C2CC2[N+](=O)[O-])=O)CC1)C c1(C(N(C)CCOc2ncccc2Cl)=O)cc2cccnc2s1 CCCCC(O)C(C)C(=O)NC1(COC)CN(C(c2c(C(C)C)cnn2C)=O)C1 N1(C(C2CC(C)(NC(CNC(CN(C)C)=O)=O)C2)=O)CC2(CSC2)C1 N1(C(C(CC)C)=O)CCC(C)C(CNC(C2CN(C)CCO2)=O)C1 N1(C(c2ncn(C)c2)=O)CC2CCC(C1)C2NCc1c[nH]c2ccccc12 C(=O)(C(F)CC(C)(C)NC(=O)C#CC(C)(C)O)NC1C=CC(C(=O)OC)C1 CCCCC(C(=O)NC)NC(=O)C=CC(C)NC(C1CCCC1)=O C(C)(C)(C(C)CC(=O)NCCCC(N)=O)NC(c1cc(C(C)=O)on1)=O CCCC(CNC(=O)CC1CC1)C(=O)Nc1c[nH]ccc1=O N1(C(CC=CC)=O)CCC2(C1)CN(C(=O)CC1(C)CCC1)C2 c1(C(N)=O)c[nH]c(C(=O)NCC(O)CNC(=O)C2CC2)c1 Cc1ncc(Cl)cc1C(N1CCOC(CCNC(C2CCCCC2(C)C)=O)C1)=O N1(C(CC=CC)=O)C2CCC1CN(C(=O)CCc1cccs1)C2 N1(C(CC(COC)C)=O)CCN(C(=O)C=Cc2cnccn2)C(C)C1 c1(C(N2CCC2CNC(C(=O)Nc2cccc(OC)c2)=O)=O)cccc(F)c1Cl Cc1csc(C)c1C(N1CCC(O)C1C(=O)NCc1cc(O)ns1)=O Cc1nc2ncccn2c1C(N1CC(CO)(NC(c2cc3ccnn3cn2)=O)C1)=O C(=O)(C(F)(F)C(O)C1CC1)NCC(CC=C)NC(c1conc1C1CC1)=O C(C)(CCC(=O)NCCCCCO)NC(C1(CCC)CCC1)=O N1(C(c2cnn(CC)n2)=O)CC(C)OC2(CCN(C(=O)CN3CCC3C)CC2)C1 C1(CCC(=O)OC)CCCN(C(C(C2CCC2)NC2CC2)C(=O)OC)C1 C(CC(C)C)(C(=O)N1CCC1(C)C(=O)NC(C)(C)CO)NC(C)=O N1(C(c2cncc(NC)c2)=O)CCC(C(=O)N2CCOCC(C)(O)C2)=C(F)C1 c1(C(=O)NCC(c2ccccc2)CNC(C(N)=O)=O)cccc2c[nH]nc12 Cc1ccc(Cl)cc1-n1cc(CCN(C)C(C2CCC2C(=O)O)=O)nn1 C1(CC(=O)NC2C3CN(C(C4(C)CCOCC4)=O)CC32)CC2(CCCC2)CO1 C1(CNC(COC)=O)(CO)CCN(C(C2CC(C(F)(F)F)(OC)C2)=O)CC1 c1(C(=O)NCC(CNC(c2csc(C(N)=O)n2)=O)OC)ccn(C)c(=O)c1 c1(-c2ccc(CN(C)C(=O)OC(C)(C)C)cc2)ccn2ncnc2c1 C=C(Cl)CCC(=O)NCCC1CCN(C(c2[nH]ccc2C2CC2)=O)CC1 c1(C(N2C(CN(C(c3cnco3)=O)CC)CCC2)=O)ncn2c1CCC2 c1(C(=O)NC2CN(CC)C2)sc(CNC(C2CCC23CCC3)=O)cc1N C1(C(=O)NC2(CF)CCN(C(C3(C#N)CCC3)=O)C2)Cc2cccnc2C1 c1(C(N2CCCCC(N(C(C(C)=CC)=O)C)C2)=O)nccc2c1NCCC2 C(=O)(CCCS(N)(=O)=O)N1CCN(C(c2c(CC)nc[nH]2)=O)C(CC(F)(F)F)C1 N1(C(Cc2c(OC)cccc2Cl)=O)CCCC12CCN(C(C1(C)CC1(C)C)=O)C2 c1(C(N(C)CC2CCCN2C(=O)CCN2CCC(F)C2)=O)nc(Cl)ccc1N C(=O)(C1=NOC2(CCC2)C1)N1CCCC(N(C(C(CCCC)CC)=O)C)C1 C(=O)(C1CCCn2nccc21)NC1CC(C)CN(C(C2CC(O)C2)=O)C1 N1(C(=O)Nc2c3n(nc2)CC(C)CO3)CCCCCC(S(C)(=O)=O)C1 c1(C(=O)NC2C(NC(c3cc(C)on3)=O)CCC2)cc(N(C)C)ccc1F c1(COC(C2CC2c2ccccc2)=O)ccnnc1O C1(CO)CN(C(=NCCN2CCOCC2)NCCc2ccc(Cl)c(F)c2)CCO1 c1(C(=O)NCC(C)(C(C)C)NC(C2CCC(C)CC2)=O)cc2ccoc2cc1F N1(C(C(CC(N)=O)O)=O)C2CCC1CN(C(c1cn(CC3CC3)nn1)=O)CC2 C1(CCCC)CN(C(=O)COCC)CCN1C(=O)CC(c1ccccc1F)C O=S(=O)(c1cnc(NCc2ccc(Br)s2)c(Cl)c1)NCCCc1ccsc1 c1(NCN(C(C2(NC(C)=O)CC2)=O)C)ccc(-n2cncn2)cc1 N1(CCNC(C2CC(CC)C2)=O)CCCN(C(c2cc(N)c(F)cn2)=O)CC1 Cn1nccc1C(=O)OCC(c1ccccc1)(C)C.C12COC(C1)CNC2 N1(CCNC(c2ccn(CC#N)n2)=O)CCN(C(c2cnc(Cl)s2)=O)CC1 N1(C(Cc2nc(C)sc2)=O)CCC(C2CN(C(c3c(F)cccc3Cl)=O)C2)C1 C1(C)CCC(=O)S1.C(Cc1ccccc1)(CCc1ccccc1)NC(=O)NCC C(=O)(C(=O)N)N(CC)CC.C(CC(F)F)CN(CC(C)NC(C)=O)C(C)=O C1(NC(c2c(C)cc(CC)o2)=O)CCN(C(c2ccc(N)c(Cl)n2)=O)CC1O Cc1ccc(-c2noc(CCC(=O)N(C3CCNCC3O)C)n2)cc1 C1(C(C)(C)C)CCC(N=c2[nH]c(=NCCC3SCCS3)[nH]c3c2CCC3)C1 c1(C(C)=O)cc(C(=O)NC2CN(C(C3(C)C=CCC3)=O)CC2CC(C)(C)C)c(C)o1 C(=O)(C(C(C)(C)C)N1CCCCC1=O)N1CN(C(C2N(C)CCCC2)=O)C1 C1(NC(CCOCC(C)(C)C)=O)CN(C(C2CCC(C)(C)CC2)=O)CC1(C)C C(=O)(C1OCCc2ccccc21)N(CCCNC(c1csc(Cl)c1)=O)C1CC1 N#Cc1cccc2[nH]cc(CN3CC4CN(C(c5cccnc5F)=O)CC34)c12 c1(C(C(=O)N(C2CCN(C(c3c(C)csc3)=O)C2)CCO)O)ccc(Cl)cc1F C(C1CCOCC1)=CC(N1CC(C(C(=O)NCCCc2cnc[nH]2)OC)C1)=O C1(C(=O)NCC(=O)NCC2CSCCN2C(=O)CC(F)(F)F)CCCC(F)(F)C1 Cc1nc2[nH]c(C(=O)N(CC(C)NC(c3cc(Cl)c(F)cc3F)=O)C)cc2s1 N1(C(CCN(CC(C)C)C(=O)CSCC(F)F)=O)CCC2(CNC(=O)C2)C1 C1(C(=O)NCCOCCCC)CN(C(C2CCC(C)(C)C2)=O)CC12CCC2 C(=O)(C(C)(C)CCCNC(C1C=CC=CC=C1)=O)N1CCCC(N(C)C)C1 C1(CNC(=O)CNS(=O)(=O)Cc2ccc(N)cc2)CN2CCCCC2CO1 c1(C(C)SC)nocc1C(N1CC(NC(C2(C(O)CO)CC2)=O)C1)=O C(=O)(C1=CCC(C)(C)CC1)N1C(CCNC(c2ncc(C)c(C)c2)=O)COCC1 N1(C(c2cc(C)c(N)cn2)=O)CC2CN(C(=O)COC(C)(C)C)CC2(C)C1 N1(C(c2c(OC)c(Br)ccc2)=O)CC=C(CCNC(C2CCCC2C)=O)CC1 C1(C(N(CCCNC(=O)Cn2cccc2)C(C)C)=O)OCCN(C)C1=O N#Cc1nc(C2CC2)oc1NC(CSc1ccccc1OC1CC1)=O c1(C(=O)NC(CC)CNC(=O)Cc2c(C)nn(C)c2C)cccn2ccnc12 Cn1c(Cl)cnc1C(=O)NC1CCC(N(C(=O)CC2CCC(=O)O2)C)CC1 C(=O)(C(CC)C(C)C)NC(CC)CNC(=O)CCC(=O)O C12(CNC(CCCNC(C)=O)=O)CCCC(CN(C(=O)C#CC3(C)COC3)C1)C2 c1(C(=O)NCC(CC(C)C)NC(CCCCC#C)=O)onc2c1CCCC2 c1(C(=O)NCC2CN(C(C3C(OC)C3)=O)CC2(C)C)c(Cl)cccc1S(C)(=O)=O c1(CSC)cc(NC(=O)CC2CC(NC(=O)OC(C)(C)C)C2)c(O)c(F)c1 N1(C(CCCN(C(C)C)C)=O)CCC=CC1C(=O)NC1CC1O c1(CC)cc(C(=O)NC2CCCCN(C(=O)CC(O)CN(C)C)C2)c(C)nn1 C1(NC(c2c(OC)cc(Cl)cc2)=O)C2CCC1CN(Cc1cc(I)c[nH]1)C2 N1(C(C(CCN(C)C)NC(=O)Cc2cccn2C)=O)CCC2(CCCN2C)C1 C12(C(=O)NC3CC(CCNC(c4ccn(CCC)n4)=O)C3)CCC(CC1)C2(C)C CC(C)CC(CNC(=O)C(C1CC1)NC(=O)CC1(O)CCCCC1)N(C)C CCC(C)C(C(=O)N1CC=CC1(C(N1CCC(O)(CC)C1)=O)COC)N(C)C C1(CC(=O)NC(C2(O)CN(C(C3CCCCS3)=O)C2)C)(COC)CCCC1 c1(CC(=O)NCC(CCC)NC(c2cccs2)=O)noc2ccccc12 N1(C(C2(C)CCC(C)CC2)=O)CCC(NC(=O)CC2CC(F)(F)C2)C(CO)CC1 C1(n2cccn2)(CNC(C2(OC)CCCC2)=O)CCN(C(=O)C(O)C(F)F)CC1 Cc1cncc(C=CC(N2CCCCCC2NC(=O)OC(C)(C)C)=O)c1 CCCCC(CNC(=O)C(C)Sc1cccc(Cl)c1)NC(=O)C(C)(C)CN(C)C c1(NC(C2(C)N(c3nc(SC)c(Br)cn3)CCC2)=O)cc(C#N)ccc1Br C1(NC(CCNC(N)=O)=O)CCCC(NC(=O)COC(F)(F)C(F)(F)F)C1 N(C1CCc2cc(Br)ccc21)C(N1CC(C)C(C(=O)O)C1)=O Cn1cnnc1CC(=O)N(C1CC(NC(=O)COCC2CCOCC2)C1)C NS(=O)(=O)c1cc(C(=O)NC(c2ccc3ccccc3c2)C(=O)O)c(Cl)c(F)c1 c1(C(=O)NC2COCCN(C(C3(C(F)F)CC3)=O)C2)ccc(Cl)c2c1OCCO2 C1(C(=O)NC(CC(C)NC(=O)C=Cc2ccc[nH]2)C)CC2CC1CC2O C(=O)(C(C(C)C)NC(C1CCC(NC(=O)CSC)CC1)=O)NCC c1(C(N(CCCCC(=O)NC(C2CN(C)CCO2)C)C)=O)cc2cccnn2c1 N1(C(C(COC)C)=O)CCC(CNC(c2ccc(C(N)=O)[nH]2)=O)(COC)CC1 C1(C(N(C)CC2CC(CF)C2)=O)CN(C(c2cn(C(F)F)cn2)=O)CC1F N1(C2(c3cn(CCC=C)nn3)CC2)CCN(C(=O)COCCF)CC1 C1(NC(c2scc(C)c2)=O)CN(C(=O)CC2OCCO2)CCC1C c1(NC(C2CC2C(=O)Nc2cc(O)c(O)c(O)c2)=O)nc2ccc(Br)cc2s1 CC(C)C(C)CC(=O)NC(C)(CNC(=O)Cc1ccnc(F)c1)C1CCC1 c1(C(C(=O)NCc2noc(C(C)C)n2)N(CCCC)CC2CC2)cnc(C)cn1 CC(C)C(F)C(=O)N1CCCCC1CCCNC(c1cnn(CC(F)F)c1)=O Cc1onc(-c2cccs2)c1C(=O)NCCC1CC(NC(C2(F)CCC2)=O)C1 c1(CCCNC(C2C(NC(=O)CNC(C3CCC3)=O)CC2)=O)ccccc1 Cc1cccc(C(N2CC(NC(c3csc4nnsc34)=O)CC2(C)C)=O)c1N N1(C(C2(NC(COCC(=C)C)=O)CC2C)=O)CCC(C)(O)C(O)C1 CC1CN2CCN1C(C(=O)NCC1CC3(CC(NC(C4(C(N)=O)CC4)=O)C3)C1)C2 C(=O)(C1CCCc2scnc21)N1C(C)C(NC(=O)CCc2ccc(Cl)s2)CC1 N1(C(C2(CNC(c3nc(C)oc3)=O)CC2)=O)CCCCC(F)(F)C1 C=CC1(C(N2CCC3(CC2)CC3)=O)CCN(C(=O)CNC(=O)C(C)(C)C)C1 C(C(C(=O)NCc1ccnc(Cl)c1)C(C)C)NC(c1c(CC)nccn1)=O C1(CCC(N2CCC(COC)CC2)=O)(NC(C2CC3CCC3C2)=O)CCCCC1 N1(C(C2C(C)C2)=O)CCN(C(=O)CN2CCN(CCO)CC2)CC1c1ncc[nH]1 CC1(CNC(c2cc(C(N)=O)co2)=O)CC(F)(F)CN1C(c1cncc(Cl)c1)=O Cc1ccc(C=CC(N2CC(F)CC2CNC(=O)CCC(F)(F)F)=O)c(C)c1 S(=O)(=O)(c1c[nH]c(C(F)(F)F)c1)C(N(CCCNC(CSCC(N)=O)=O)CCO)=O CCC(C)C(C)(c1nnnn1C1CC1)NCCNC1CCCC1(C)C Cc1n[nH]c(=NC2CC(O)(CNC(c3cc(C(F)(F)F)ncc3)=O)C2)s1 C1(NC(c2ccc(OCC)c(OC)c2)=O)CN(C(C2CC2)=O)Cc2ccnn2C1 c1(C(=O)NCCN(C(C(C)(CO)OC)=O)C)ccc(C)c2c1CCC2 C1(C(N2CCCC(CCO)C2)=O)CC2(CCC2)CN1C(C1CCCCC1)=O C(C)(C)(CCC(=O)NC1(CNC(C2CCCC(CF)C2)=O)CCOC1)N(C)C C(C(O)CN=c1[nH]ccnc1F)NC(=O)CN1Cc2ccccc2C1 Cc1nc(Cl)ccc1CC(N1CC(N(C)C(C2CCCO2)=O)C2(CC2)C1)=O C(C(CC(=O)OC)OC(C)(C)C)NC(CC)CN(C)NC(=O)OC Cc1ccc2c(c1)CC(C(N1CC(O)CC1CNC(=O)CN1CCOCC1)=O)O2 C(=O)(C(F)C(F)(F)C(F)(F)F)N1CCC(N(C(=O)C=Cc2cccc(O)c2)C)C1 C1(CNC(C(CCF)NC(C=Cc2cc(C)no2)=O)=O)CC2CC1CC2O c1(C(=O)NC2C(C)(CNC(c3nc(C)n(C)n3)=O)CCC2)cccc2sccc12 C(CO)(C(F)(F)F)N1C(=O)c2c[nH]nc2C1.C1(C(=O)NC2CC2)CCCCC1F c1(CC(N2C(CNC(C(C(C)C)OC)=O)C=CC2)=O)cn2ccsc2n1 C1(CC=C)(C(=O)NCc2cncc(C)c2)CCN(C(=O)CCC2CCCCO2)C1 c1(C(=O)NCC2C(C(=O)NCc3nccc(C)c3)C2)nccc(C)c1N N1(C(CS(=O)(=O)NC)=O)CC2CCC(C1)N(C(c1c[nH]nc1C)=O)C2 C1(C2(O)CCOC2)(CNC(N(C(c2cccc(OCC)c2)C)C)=O)CC1 CCCCCCCCC(=O)N1CC2(CCC2NC(C2CN(C)CCO2)=O)C1 C1(c2n(CC)ccn2)NC(=S)N(c2ccc([N+](=O)[O-])cn2)C2=C1C(=O)NC(CC)C2 C1(C(=O)NCC2(CNC(=O)Cc3ccco3)CC2)(OC)CCCC(C)(C)C1 C1(NC(CCCOC)=O)CC(NC(c2ccnn2C(F)F)=O)CC1O S(=O)(=O)(c1ccc(NCC2(SC)CCOCC2)c(F)c1)N(CC(C)O)C c1(NC(=O)NCCS(=O)(=O)NC2CCCCC2)cc(Cl)ccc1C(F)(F)F C1(C(=O)NC2C(n3cc(CCCC=C)nn3)CCCC2)CCn2nnnc2C1 C#CCC(CC(F)F)C(=O)N1CCCC(C(=O)NC(c2cscn2)C)C1 N1(C(c2c(CC)c[nH]c2)=O)CCOCC1CC(=O)NCCOCCC(C)C N1(C(C(c2ccc(Cl)cc2)(C)C)=O)CCC(NC(c2ccc(Cl)s2)=O)C(F)C1 c1(C(N2CCC(CN(C(C3CC(C)C3)=O)C)C2)=O)cc(C(F)(F)F)cnc1O C1(NC(C(C)(C)F)=O)CN(C(=O)CNC(c2ccccn2)=O)CC1C1CC1 C1(NC(=O)NCCCOCC#C)CC2(CC(C)=NO2)C1 C(=O)(C(C)C(O)C(C)C)N(C1CCN(C(=O)Cc2ccc(Cl)nc2)C1)CCC C1(C2CC2)(C(N2C(CC)CC2)=O)CN(C(c2cc[nH]c2C)=O)C1 c1(C(N2CCCN(C(C(C)OCC=C)=O)C(CO)C2)=O)cc2cc(Cl)cnc2[nH]1 N1(C(C#CC2(CC)CC2)=O)CCC2CCCC(C1)N2C(c1cncc2sccc12)=O N1(C(C(C=C)CC)=O)CCCC2(CCN(C(=O)C(C3CCCCCC3)OC)C2)C1 N1(C(C2CC3CCC2O3)=O)CCC2C(CCN2CCC2CCCO2)C1 C1(CNC(CC=C(C)C)=O)C(C)CCN1C(=O)C1=CCSC1 CCCC(C(=O)NCCCC1CN(C(=O)CS(=O)(=O)NCC)CCO1)C(C)C C(CC(C(=O)NC1CC2C=CC1C2)NC(=O)C=CC1CCCN1C)OC c1(C(=O)NC(CCN(C(C(C=C)(C)O)=O)C)C)cc2nccnc2cc1F C1(NC(c2cc(I)c[nH]2)=O)CN(Cc2ccc(C(F)(F)F)s2)CCC1(F)F Cc1cc(NC(c2ccc(F)cc2)C2CC(C)C2)cc(C)c1 C(=O)(CCCC(F)(F)F)NC(C(=O)NCC1N(CC)CCCC1)CN(C)C CCC(C)CC(=O)C(=O)NCC(C)(C)C#CC(=O)NCc1cc(C)ccc1C c1(C(=O)NC(CN(C(C(C=C=C)C)=O)C)CC)cc2ccc(C)cc2[nH]1 N1(C(C2=C(C)CCC2)=O)CC2CCCN(C(C3CCC4CC4CC3)=O)C2C1 N1(C(c2c(Cl)cn(C(C)(C)C)n2)=O)CCC2(CCCN(C(=O)C3=CCCC3)C2)C1 c1(OC)ccc2c(=NCC=CC3CC3)[nH]c(N3CCC(F)C3)nc2c1 N1(C(C(COC)O)=O)CCN(C(=O)CN(C)Cc2ccc(Cl)cc2)CC1 c1(OC)ccc(-c2ncc(C(=O)NC(c3cccc(F)c3)C)cc2OC)cc1O c1(C(N2C(CNC(c3c(Cl)ccc(OC)c3)=O)CC2)=O)cc2nc[nH]c2cc1N C1(C(N2C(CNC(=O)CN)CC(OC)C2)=O)CCc2ccccc2C1O c1(OC)cccc(CCC(=O)N(C2CCC(CO)CC2)C2CC3CC2CN3)n1 C(CC(=O)N1CC(C2=NOCC2)C1)(C(C)(C)C)NC(C=CC(=O)OCC)=O C1(C(C)NC(=O)CCc2nccn2C)CCCN(C(=O)CCCc2cnn[nH]2)C1 C12(CNC(CC(CCC)C)=O)CN(C(c3cc(CF)on3)=O)CC1CS(=O)(=O)C2 c1(CC)ocnc1C(=O)NCC(=C1CN(C(c2sccc2C)=O)C1)F c1(CC)ccc(NC(C2CCCC2CNC(=O)COCCF)=O)cc1C N1(c2snc(CCOC)n2)CC(CNC(=O)C(F)C(C)C)OC(C)(C)C1 C12(NC(c3ncc(CC)cn3)=O)CCC(C1)N(C(C1CC1(Cl)C(=O)OC)=O)C2 C1(C(=O)NS(C(CCC)C)(=O)=O)CC(S(C)(=O)=O)CN1C(=O)OC(C)(C)C C1(C(C2CCCCC2)N2CC(CNC(C(C3CCC3)OC)=O)C2)COC(=O)N1C C(CCC(C)(c1nnnn1-c1ccccc1OC)NCC1CC1(C)C)OCC c1(C(=O)NC2C3(CNC(C4C(=C)C4)=O)CCC(C2)C3)cccc(OC)c1[N+](=O)[O-] C1(C(=O)NC(C(CO)NC(C=CC)=O)C)CCN(c2cnccn2)CC1 CCC(C)C(CC(=O)N(C(C)CO)C)NC(=O)CN(c1ncccn1)C C1(NC(CCNS(CC)(=O)=O)=O)CCCN(C(c2cc(OC)nc(Cl)c2)=O)C1C N1(C(c2sc(C)c(O)n2)=O)CC(NC(C2CC(OC(C)(C)C)C2)=O)CC(C)C1 C12(C(=O)NCC)CCC(CC1)N(C(=O)CCCCC1CC1)C2.CCC(=O)OCC Cc1nn(C)c(Cl)c1CC(=O)NCC1CN(C(=O)Cc2cccc(O)c2)CC1C N1(C(C(F)=CC)=O)CCC2(CCC(NC(c3sccc3CC)=O)C2)C1 Cc1ccc(O)c(CC(=O)NC2CN(C(=O)C(C)OCC3CC3)CC2(C)C)c1 c1(C(=O)NC(CNC(c2c(C(F)(F)F)ncn2O)=O)CO)ccc2nn[nH]c2c1 C=C(C)CCCC(=O)N1CC(C(=O)N(CCC(C)O)C)CC(C)C1 c1(C(=O)NCC(C)CNC(C2(CO)CCCO2)=O)cccc2ccnn12 C(=O)(C#Cc1ccccc1Cl)N1C(C(Nn2c(CC)nnc2)=O)CC(O)CC1 N1(C(c2nc(OC)c(C)s2)=O)CCN(C(=O)C(C2CC2)SC)CC2(CC2)C1 c1(C(=O)NC(CCCC)CNC(C2(Cl)CC23CCC3)=O)ncc2[nH]ncc2n1 CC(C)S(=O)(=O)c1ccccc1C(N1CCCC1(C)CNC(=O)CSC1CC1)=O N1(C(C(C)NC(C(C=C)(C)C)=O)=O)CCC12CN(C)C2 C(C(=O)N1CCC(F)(CNC(=O)C(C)(C)c2cccs2)C1)(C(C)C)SC CC1(C2CCN(C(C3CC4CC3CN(C(C3CCNC3=O)=O)C4)=O)CC2)CC1 c1(C(c2n(CC(=O)OC)nnn2)NCc2cccc(F)c2)cnc2[nH]cnc2c1 CC1(C)CC(CNC(=O)Cc2cc(F)cc(F)c2)N(C(c2cc(CF)on2)=O)C1 CP(C)(=O)c1ccc(C(N2CC3C(NC(=O)C(c4ccc(F)cc4)F)C3C2)=O)o1 Cc1cc(Br)cc(C)c1C(=O)NC1CCCC1CNC(c1cc(CO)[nH]n1)=O c1(CCC(=O)NC(C(=O)NC(c2nc[nH]n2)CC)C2(O)CCC2)conc1C c1(C(=O)NCC(CNC(C(C)(C)c2ccno2)=O)CO)ccc2c(c1)CCN2 Cc1nc(Cl)c(Cl)cc1NC(=O)C=Cc1ccsc1 c1(C(N2CCC(O)(C(C)NC(CS(CC)=O)=O)CC2)=O)cc(C)c(C)cc1N Cc1c(Cl)ccnc1C(N1CCOCC1CNC(c1ccncc1C(F)F)=O)=O c1(CSCCC(=O)NCC2N(C(C3(C)CC(=C)C3)=O)CC2)ccc(F)cc1 C1(C(N2CCCC(N(C(c3c(C)occ3)=O)C)CC2)=O)CCOC2(CCCC2)C1 C1(OC)CCCC(CC(N2CCCC2CN(C)C(c2cncc(CO)c2)=O)=O)C1 N1(CCC(=O)NC(C)C(C)NC(=O)CN2CCCCC2=O)CCCCC1=O N1(C(CCOC)=O)CCC(C(=O)NCC(C)(F)C(C)C)C12CC2 C(=O)(CCN=c1ccc(C)c[nH]1)NC1CN(C(c2ccc(OC)nc2)=O)C(C)C1 c1(-n2cc(CNC(C3CCCS3(=O)=O)=O)nn2)cncc(C(=O)NCC2CC2)c1 c1(OC)ccc2c(C(=O)NCC3CCC(N(C)C(C4CC4Cl)=O)CC3)cnn2c1 Cn1cc(C(C2CC2)NC(c2cc(-c3ccccc3)n[nH]2)=O)cn1 c1(NC(N(CCOC)CCO)=O)cc(C)n(C)c1C.C1=[SH]C1(C)C N1(C(C(=O)NCCC)C)CC2(CCCCC2)C1c1ccccc1 c1(NC(C)=O)ccc(C(=O)NC(Cc2nc(C)no2)CO)c(Cl)c1 C(=O)(CCS(=O)(=O)Cc1ccccn1)N1CCN(C(CCC(=O)OC)=O)CC1C CCCCC(C(=O)NCc1ccc(Cl)s1)N(C)Cc1cccs1 c1(C(N2CCC(NC(=O)C=Cc3ncco3)C(F)C2)=O)nc2cnccc2s1 Cc1[nH][nH]c(=N)c1C(=O)NCc1cccc(NC(C2CC23CC3(F)F)=O)c1 c1(NCC=CC(N2C(NC(C(C3CC3)SC)=O)CC(F)C2)=O)cc(N)ccc1Cl C(=O)(C1SCCc2ccccc21)NC(CN(C(c1ccc(CC(C)C)s1)=O)C)C Cc1ccc2c(N3CCN(C(c4ccn(C)n4)=O)CC3)nc(OCCO)nc2c1 Cc1nc2ncccc2cc1C(N1CC2(CCN2C(=O)C2=CCCC2)C1)=O N1(Cc2ccc(C(=O)O)s2)CC2CCC(C1)C2N=c1ccnc(Br)[nH]1 N1(C(C23CC(CC)(C2)C3)=O)CCN(C(=O)CCc2nnc(O)nc2O)CCC1C C1(C(N2CC(CC=C)(NC(=O)C=CC3CCC3)C2)=O)CCC(=O)C(C)C1 C1(NC(c2cn(CC)nc2)=O)CN(C(c2occc2Cl)=O)CCC1C(F)(F)F N1(C(c2c(C)ccc(OC)n2)=O)CCCC12CCN(C(C1(C)CCNC1=O)=O)C2 C12(C(N3CC(NC(C(C)C)=O)CC3(C)C)=O)CCCC(CCC1)C2 C12CC(C)CN(C1)C2=O.c1(NC(Cc2c(C)noc2C)=O)ccc(CO)cc1F C1(NC(c2ccc(CF)cc2)=O)CCN(C(=O)CCc2ncc[nH]2)C12CC2 Cn1c(O)ncc(C(=O)NC2CC3CN(C(=O)CCSC(F)(F)F)CC3C2)c1=O c1(C(=O)OC)c(C)ccc(NCC2N(C(C3(C)CC(=C)C3)=O)CC2)c1N C1(NC(=O)CCn2cccn2)CC(CNC(C2(O)CCSCC2)=O)CC1O c1(C(=O)NCC2C(NC(C3(CCC)CCC3)=O)C2)nccc2[nH]nc(C(C)C)c12 c1(OC(C)C)ncccc1C(=O)NCC1(O)CN(C(c2c[nH]nc2C2CC2)=O)C1 c1(NCCN(C)C2CC2)ccc(S(=O)(=O)N2CCC(F)C(O)C2)cc1F C=C(C)CCC(=O)NCC1CCC(CNC(C2(C(C)(C)C)CCC2)=O)CC1 C=CC1COCCN1C(=O)C(C(C)OC)NC(C1C2CC(=O)CC12)=O c1(C(N(C2CCC(NC(c3ccc(C)cc3)=O)C2)C)=O)cnc(O)c(C)c1 C1(C(N2CCC(N(CCC)C(c3sccc3C)=O)C2)=O)CC(OC)C(OC)C1 CC(C)CCC(C(=O)NC1CCN(C)CC1)NC(c1cncc(Cl)c1)=O c1(C(=O)OCC)c(NC(C2CC(NCc3cccs3)C2)=O)ncn1C C1(NC(CN(C(C(C)C)=O)C)=O)CC2(C1)CC(NC(=O)COCP(C)(C)=O)C2 C1(C(N(c2ccsc2)C)=O)CC1C1CN(C(C2CCCCS2)=O)C1 c1(CC(=O)NC2C(C)(C)N(c3nnco3)CC2)c[nH]c2cccc(F)c12 N1(C(CCC2C(C)C2)=O)CC2(C(N3CC(CO)CC(C)(C)C3)=O)CC1CCO2 N1(C(C(C)c2cccs2)=O)CCOC2(CCN(C(C34CC(CO3)C4)=O)CC2)C1 C(CC1CCCC1)(C(=O)NC(c1nncs1)C)NC(C=CCN(CC)CC)=O C1(CNC(c2cc(C)on2)=O)CCCN(C(=O)CCc2ccsc2Br)C1 CCS(=O)(=O)CC(=O)N1CCN(C(C2SCCCS2)=O)C(c2ccncc2)C1 c1(CC)ccc(C(=O)NC2CC(CNC(=O)CC3CCCOC3)C2)cc1 N1(C(=O)C=CC(C)(C)C)CCC(F)(CN)CC1.CCC(C=O)N(C)C C(=O)(C(O)CC(N)=O)NCCN(C1CCCCC1)C(CC1C=NN(C)C1=O)=O C1(N2CCC(CNC(=O)NC(C)CCC3CC3)C2)CCN(C)CC1 N1(C(C2CN(C(CCc3n(C)ncc3)=O)C2)=O)CC2CCCC1C2CO N1(C(CCC=C)=O)CC2(CCC(CNC(=O)CC(C)=C(C)C)O2)C1 Cc1cc(C(=O)Nc2cccc(NC(=O)C3=CCOC3)c2)nc(O)c1 C(=O)(CC(CC)CC)NC(CC)CNC(c1[nH]ccc1-c1ccccc1)=O N1(C(c2c[nH]nc2Br)=O)CC2CN(C(C34CCCC3CCC4)=O)CC2C1 CC1(C)CC(NC(=O)Cc2c[nH]c3cnc(Cl)cc23)CCN(C(=O)CO)C1 C12(C(N3CCN(c4ncnc(Cl)c4Br)CC(O)C3)=O)CC=CCN1CCC2 C(=O)(C1CCCc2sc(C)nc21)N1C(CNC(C=CC=CC)=O)C(C)(C)CCC1 C1(=O)C(O)CN1.c1(OC)noc(C2CCC2N)n1 c1(C(=O)NCC2(C(C)NC(C(COC)OC)=O)CC2)cc2c(C)ccc(F)c2[nH]1 C(c1cccc(F)c1)=CC(N1CCC(CNC(c2c(Cl)nc(N(C)C)s2)=O)C1)=O C1(NC(CCOCCC)=O)CCC(C)N(C(c2cccc(F)c2CC)=O)C1 c1(CNC(C2N(C=O)CCC2)=O)ccc(CNC(C2CCSCC2)=O)c(F)c1 N1(C(C(C23CCC(CC2)CC3)N)=O)CCC(c2ccccc2)C(CO)C1 Cc1cccnc1C=CC(N1CC(N(C(=O)COCCN(C)C)C)C(F)C1)=O C1(C(=O)NCc2ncsn2)CC2CCC1N(C(=O)C(O)CC(=O)O)C2 n1(CC)c(CN2CCC(O)(C(N3CC(O)C(F)C3)=O)CC2)nc2ccccc12 C1(NC(C(COC)Cl)=O)CN(C(c2cccc(Cl)c2Cl)=O)CC12COC2 C1(CC)CN(C(c2ccn(C(C)C)n2)=O)CCC1NC(c1ncncc1F)=O N1(C(CN(C(C)C)C)=O)CC2(CCN(C(=O)CN3C(=O)NC(C)(C)C3=O)CC2)C1 c1(C(=O)NC2CCC(NC(C3CCN(C)C3=O)=O)CC2)ccnc2ncccc12 c1(C(N2C(C)CCC(C)C2)=O)cc([N+](=O)[O-])c(O)cc1Br C1(NC(c2cn(CCOC)nc2)=O)CC(N(C(=O)CNC=O)C)C12CCC2 c1(CNC(C2CC(C)(CC)C2)=O)cnn(C)c1C(=O)NC(C1CCCCC1)CO N1(C(C2CCCS2(=O)=O)=O)CCCN(C(C23CC(F)(C2)C3)=O)CC1 N1(C(CCC=C=C)=O)CCC(F)(CNC(c2ccc(OCCF)cc2)=O)CC1 N1(CCC(=O)NCC2CC(CNC(c3csc(CO)n3)=O)CO2)CCCS1(=O)=O c1(NC)cnc(C(=O)NC(Cc2cn[nH]c2)C(=O)N(C2CCC(F)(F)C2)C)cn1 C1(CNC(CCNC(COC)=O)=O)CN(C(=O)C(C2CCCCC2)C)CC1O c1(C(=O)NC2CCN(C(C(CCC(C)C)=O)=O)C2)cnn2c1S(=O)(=O)NCC2 S(=O)(=O)(c1ccccc1Cl)N1C(C)(C)CC(O)C1 Cc1ccc(CC(N2CC(N(C(=O)CCOC3CC3)C)C3(CC3)C2)=O)cc1C C1(C(=O)NCCC(=O)OC)COCCC1NC(C1(C#N)CC=CC1)=O CC1=C(C(=O)N2CCOCC2CC(=O)NC(C)CCC(F)(F)F)CCO1 N1(C(C23OC(C)C(C2)C3)=O)CCC(C)(c2nc(COC3C=CCCCC3)no2)C1 C(c1cccc(F)c1)=C(C(=O)NC(CC)CNC(C1(CC)CCNC1=O)=O)O C(C(=O)N(CCC(=O)NCC1OC2CCC1C2)OC)OCC C1(CC(=O)NCCOCCC(N2CCCC(CF)C2)=O)CC2CCC1O2 C#Cc1cnn(CC(=O)NC2CC(CNC(=O)CCc3cn(C)cn3)C2(C)C)c1 c1(C(=O)NCCCC(C)NC(C2CCN(C)C2=O)=O)ccnc(C(C)(F)F)c1 c1(C(=O)NCC2CCC2NC(c2ncsc2C(F)(F)F)=O)cc2n(n1)CCCC2 N12CC3CC3(C1)SCC2=O.c1(C(C)Sc2ccccc2)ccccc1-c1ccc(C)cc1 Cc1c(CN2CC3CN(C(c4cc(O)n(C)n4)=O)C3C2)cccc1O N1(C(C(CC#C)O)=O)CC2CCN(C(=O)CCN3CCN(C)CC3)CC12 N1(CC(CCC(O)C2CCC2)=O)CCc2c(C3CCCCC3)cccc21 c1(C(N(C(C)CNC(C2(CN(C)C)CC2)=O)C)=O)ccc2oncc2c1 C=CC1(C(=O)NCCC2(CNC(=O)Cc3nnc(O)s3)CC2)CCCCC1 n1(CC(N2C(CNC(c3ncc(Br)cn3)=O)CC(F)C2)=O)nc(Cl)ccc1=O C1(NC(=O)COC2CCCC2)CC(F)CN(C(=O)CC2(CO)CCCC2)C1 C1(C(N2CCCC(CNC(c3ccc(F)cc3F)=O)C2)=O)CC12CCCCCC2 C1(C(C)C)CN(C(C2(N(C)C)CC2)=O)CCN1C(=O)CC1CCS(=O)(=O)C1 c1(OCCC(=O)OC)ccc(C)cc1C.C1(C)C(=O)N1C(C)C(C)C CC1CN(C(=O)CC2(S(N)(=O)=O)CC2)C(C)CCO1 c1(C(=O)NCCC(C)NC(C(F)=C(C)C)=O)oc(-c2ccccc2)nc1C C1(C(=O)Nc2cnc(SC)s2)CCN(C(=O)CSc2ccc(C)cc2)C1C(C)C C1(C(=O)NC(CCO)C(F)(F)F)(CC)CCCN(C(=O)C2=NOCC2)C1 c1(C(N2C(C(N3CCC(NC(C)=O)C3(C)C)=O)CC2)=O)cccc2[nH]ncc12 N1(CC)CC(C(=O)N(C2CCN(C(=O)CC3CNC(=O)C3)CC2)CCO)CC1=O C(N=c1nc(C2CC2)[nH]s1)C1(F)CC(NC(CCOC)=O)C1 C1(C(=O)NC2C(C)(C)CN(C(=O)C(C3CCOCC3)O)C2)CCOC2(CCC2)C1 C1(CNC(C(C)CF)=O)CN(C(c2ccn(C)n2)=O)CC1C C(=O)(C(C(C)(F)F)c1ccccc1)NCC(C)NC(c1c(C)n(C(C)C)nc1)=O Cc1ccc2scc(CC(=O)NC34CC(CNC(=O)C(C)OC(C)C)(C3)C4)c2c1 c1(CC(=O)NCC(CN(C(CN2C(C)CCC2)=O)C)O)cc(Cl)ccc1[N+](=O)[O-] c1(CN=C(NC(=O)CSC2CCCC2)NCc2cncs2)nnc2cccnn12 Cc1ccc(N2CC(N3CCCC3c3ccccc3)CC2=O)cc1C N1(C(c2nccc(N(C)C)c2)=O)CCC2(CC1)CN(C(c1cncc(F)n1)=O)C2 N1(C(C(C)C)=O)CC2CC(NC(C3(NC(=O)OC(C)(C)C)CCCC3)=O)C1C2 c1(C(=O)NC2CN(C(CCSC)=O)C3C2C3)oc2ccccc2c1C c1(N2C3CC(NC(CSC)C)CC2CC3)ncnc(NC)c1[N+](=O)[O-] CC1C(C)N(C(=O)Cc2c[nH]ccc2=O)CCN1C(=O)CCc1cnc[nH]1 c1(C(N2CC(OC)(CNC(=O)CNC(c3ccco3)=O)C2)=O)c(C)cccc1N n1(CCC)ncnc1CN(C)CC1CCN(C(=O)NC2CC2)C1 C1(Sc2nc[nH]n2)CCC(C)N(C(=O)N(CC(C)C)CCC)C1 c1(OC)ncncc1NC(=O)CCC1CCN(C(c2n[nH]c(C)c2C)=O)CC1 N1(C(c2cnc(OCC)s2)=O)CCOCC1CNC(C1(C(F)(F)F)CC1)=O C1(C(=O)NCC(CC=C)NC(=O)C(C2(O)CCCCC2)(F)F)CC(C)OC(C)C1 C1(NC(=O)Cc2csc(S)n2)CN(C(C23CCC(C2)C3)=O)CC2(CCC2)C1 Cc1nc2ccnn2cc1C(=O)NC(C1CCCN1C(=O)C(C)CN(C)C)(C)C c1(CC2(C(=O)NC3CCC(NC(C(CCC)O)=O)C3)CC2)ccc(C)cc1Br c1(CC(C2CCCCC2)NC(=O)NCC2CCOC2)c[nH]c2ncccc12 c1(C(=O)NCC(CO)NC(C(c2nccc(C)c2)(C)C)=O)cc(Cl)c(N)cc1Cl c1(C(N2CCOCC2c2nc[nH]n2)C(=O)NCCCC)n[nH]c(C)c1C CC(O)CCCCCC(=O)NCC1CCCN(C(=O)CN(c2ccccc2)C)C1 O=C(CCCCc1cnn[nH]1)N1CCCC1Cc1cn(C2CCCC2O)nn1 C1(C)(C(N(C)CCn2cccn2)=O)CC(O)CN1C(C1CCCCCCC1)=O C(=O)(CC(C)C(F)(F)F)N(CCCCC(=O)NC1CC(C)(CC)OCC1)C N1(C(CCC=C)=O)CC(NC(c2cncc(CC)c2)=O)C(CO)C1 c1(C(=O)NC(CC)CSc2ccc(Cl)nc2C)ccc2c(c1)CC(=O)N2 C12(NC(C3CC(O)(CC#C)C3)=O)CCC(CNC(=O)Cc3ccsc3)(C1)OC2 N1(C(CSCC=C)=O)CCCC(CN(C)C(c2cc(C3CCCC3)n(C)n2)=O)C1 Cc1ccc(S(N)(=O)=O)c(C(=O)NCCC(C)NC(=O)C(O)C(C)C)c1 C1(C(N(CCCCN(C(=O)C(C)(C)F)C)C)=O)CCOC2(CCC2)C1 c1(OC(CNC(C2(COC)CCCNC2)=O)C)ccc(F)c(Cl)c1 C1(c2cn(C(C(=O)OCC)C)nn2)CN(C(c2cc(C)c[nH]2)=O)CCO1 CC(CC(F)F)C(=O)NC1CC1CNC(c1cnc(C2CCC2)nc1O)=O CN1Cc2ccc(C(=O)N(CCCCNC(C3(C#N)CC4(CC4)C3)=O)C)cc2C1 Cc1ccnc(CNC(=O)CCC2CCN(C(c3c[nH]nc3C3CC3)=O)CC2)n1 c1(CC)nc(Cl)nc(N2CC(NC(=O)CC3(O)CCCC3)CC(C)(C)C2)c1C#N N1(C(C2C(CCOC)C2)=O)CC2CN(C(=O)C=C3CCOCC3)CC2(C)C1 c1(C(c2nnnn2-c2ccc(F)cc2)NC2C(COC)C2)ccc(C(F)F)nc1 Cc1c(Cl)ccc2c1CN(C(c1nnn3c1CSCC3)=O)CC2 C1(C(=O)Nc2cnccc2C)(CC)CCN(C(=O)C(C)=C2CCC2)CC1 Cc1cc(C)c([N+](=O)[O-])cc1C(=O)NC(CO)C(C)NC(c1cc(CO)[nH]n1)=O c1(C(C)C)cccc(C(N2CCCC(CNC(=O)CNS(=O)(=O)C3CC3)C2)=O)n1 CC1COCCC1C(=O)NCCOC1CN(C(c2ccn(C)c2C2CCC2)=O)C1 c1(C(C(=O)NC(CCNC(CCC=C(C)C)=O)C)=O)cc(F)c(F)cc1F Cc1cccc(CC)c1.O=C(CC(CC1CC1)NC(=O)Cc1cccc(O)c1)N N1(C(c2ncc(OC)cn2)=O)CC2CCC1CC2NC(c1c[nH]nc1C)=O CC1(C)CCc2c1n[nH]c2C(=O)NCCC1(O)CCN(C(C2C=CCCC2)=O)C1 N1(C(=O)C(c2ccc(Cl)cc2)O)CCCN(C(C2CCC3(CCC3)O2)=O)CC1 C1(CNC(c2cc(C)no2)=O)CCN(C(c2cccnc2C)=O)CC1(F)F c1(C(=O)NCC2C3CN(C(CNC(CCC)=O)=O)CC32)cncc(Cl)c1Cl CCC(CC)(CO)C(=O)NCC(C1(O)CCN(C(c2sc(=N)[nH]c2C)=O)C1)C N1(C(c2c(Br)cnc(C)n2)=O)CCC2(CCCC2CNC(C2(F)CC2)=O)CC1 C(=O)(C1=NOCC1)NCC1(CC(=O)OCCc2ncon2)CC1 Cc1ccc(C)c(SCc2nnc(N(C)CCOC(C)C)n2CC2CCCO2)c1 Cc1cccc(-c2cn(C3CCCN(C(=O)C(C)CC(N)=O)C3)nn2)c1F c1(CNC(c2ncc(C)s2)CC)cc([N+](=O)[O-])ccc1Cl N1(C(C(C(C)N)C)=O)CCCc2cc(Cl)cnc21 N1(c2nnc(C)s2)CC2CC1CN(C(C1(C3CCCCO3)CCC1)=O)C2 C1(CNC(=O)C=CC(F)(F)F)CCCC1NC(c1ccnn1Cc1ccccc1)=O CC1CCC(C)(C(=O)OCc2c(F)cccc2Cl)C1(C)C N1(C(c2cc(N(C)C)ncc2)=O)CCC2CCC(C1)N2C(C1(C(C)(C)O)CC1)=O C(CCCC(=O)NCc1cccc(C(=O)NCCC(O)C2CC2)n1)OC C1(NC(C2CC(CF)C2)=O)CC2CCC1C2.CC1(C)C(=O)N2C1CCC2 N1(C(CC2CC(=O)C2)=O)CC(NC(=O)CC2CC=CCC2)Cc2ccccc21 C1(CNC(=O)C(N2CCCC2CCO)C2CCSC2)CCC(F)(F)CC1 N1(C(C2C(C(C)(C)C)CC2)=O)CCC(CNC(C2COCC2(C)C)=O)CC1 C(C(C(=O)NCC(O)C1(C)CC1)NC(N)=O)OC(C)(C)C C12(C(N3CCC(N(C(=O)CCOc4ccccc4)C)C3)=O)CCC(C)(C1)OC2 N1(C(=O)NC(c2ccccn2)CC)CCS(=O)(=O)CC(F)C1 O=C(CCCCN1CCC1)NCC1(O)CC(NC(=O)C(c2cccc(F)c2)O)C1 C1(O)(CCNC(c2c(C)cns2)=O)CCCN(C(c2cnn(CC(F)F)c2)=O)C1 C12(C(=O)NCc3cc(Cl)cc(C)c3)C3CC1C1C(C(=O)NC(C)CC#N)C3C21 N1(CC(=O)NC2C(NC(C(C3CCC3)OCC)=O)CC2)CCOCC1 N1(C(CCCC=C)=O)CCN(C(=O)C(c2ccc(F)cc2)C)CCC1C C1(CC)(NC(=O)CC2CCC2(C)C)CCCN(C(=O)CCCOC)C1 c1(CN(C(=O)NCc2c(C)ncnc2)C)cccc2ncccc12 C(=O)(C(O)C1=CCCCC1)N1CC(CC(=O)NCc2nncn2C2CC2)(OC)C1 N1(C(C2CC3(CC(C)C3)C2)=O)CCC(C)(C)CC1C(=O)NCCC(O)C(F)(F)F c1(OC)cc(C)ccc1OCCC(N1CCCC1CNC(=O)C1=CCCC1C)=O C(=O)(CC(CC1CC1)NC(=O)C1=CCSC1)NCc1cnc(C)s1 CCC(CC)C(C(=O)NCCN(C(=O)Cn1nccc1-c1ccccc1)C)OC C1(CCC(=O)NC2(C3(O)CN(C(c4n[nH]cc4Cl)=O)C3)CC2)CCC(C2CC2)O1 C=CC(CCC)CC(=O)NCCCCC(C)(C)NC(=O)Cc1coc(C(F)F)n1 C(=O)(C(CC(C)(C)C)NC(=O)C(=O)NOC)N(C1CCN(CC)CC1)C N(C(=NCc1ccco1)N1CCC(OCC)C1)Cc1cccc(CC)c1 c1(C(C(=O)NCC2CC2)N(c2c(C)cccc2)C)cccc2c1CCC2 C(=O)(C(CC(N)=O)NC(=O)C(C1(O)CCCC1)F)NCC1(CCO)CN(C)C1 CCCC(C(=O)N(C(C)CCNC(c1sccc1S(N)(=O)=O)=O)C)C(C)C CC1CCn2cc(C(N3CCC(NC(C4C=CCC4)=O)C34CCCC4)=O)nc2C1 C1(C(N2CCC(OCC=C)C2)=O)CCN(C(=O)Cn2cccn2)O1 Cc1cc(=NC(=O)c2cncc(NCc3cccnc3O)c2)[nH][nH]1 c1(C(=O)NCC2N(C(CCCCC=C)=O)CCOC2)cccc2nn(C)cc12 N1(C(COCCCC)=O)CCC(O)(CCNC(=O)CC2C=NN(C)C2=O)CC1 C=C1Cn2c(C(=O)NCC(CC(F)(F)F)NC(c3ccc(F)o3)=O)nnc2S1 S(=O)(=O)(c1c[nH]ccc1=NCCCCCF)N1CCCC(C(CC)=O)C1 CC1CCN(C(=O)C=CBr)CC1NC(c1ccc(OC(F)F)nc1)=O c1(CC)ccc(C(=O)NC2CC(C)(NC(c3ccn(CC)n3)=O)C2)cc1Br N1(C(C2=C(C)OCC2)=O)CCCN(C(=O)C2=NOCC2)C(C)C1 C1(C(C)NC(c2cc(OC)n[nH]2)=O)CN(C(c2cc(SC)c(C)o2)=O)CCO1 CCC1(C)CN(C)CCO1.C(C(=O)NC1CC1)(c1csnn1)N(C1CC1)CC1CC1.OC N1(C(C2(C)C(C)OCC2)=O)CC2(CCCN(C(=O)CC3(C)OCCO3)C2)C1 C1(C)(C(=O)NCCCCCCN(C(CCOCCOC)=O)C)COC(C)(C)CO1 Cc1c(O)ccc(CN2CCC(C(=O)NCCc3cccc(O)c3)C(O)C2)c1O C1(C(=O)NC2CC(C)N(C(c3ccccc3O)=O)C2)CC2CCC1CC2 C12(C(=O)NC3CC(NC(c4ccsc4Br)=O)C3)CCCC1CC2 C(=O)(C(O)CCc1ccccc1)N1CC(O)(CNC(C(C)OCC(C)C)=O)C1 C1(NC(C(F)=CCC)=O)(CO)CCN(C(c2cc(-c3ccco3)on2)=O)C1 c1(CC)ccsc1C(N1CCC(CNC(c2ccc(CNS(C)(=O)=O)o2)=O)C1)=O c1(C(CNC(=O)C=Cc2ccco2)NCc2c(C)noc2)ccc(F)cc1 n1(CCOCCOCC)cc(CNS(N)(=O)=O)nn1.C(C(=O)N1CC(C)C1)(CO)OC C(CCCCCC(=O)NC1COC2(CCCC2)C1)NC(C(c1ccc(C)o1)C)=O C1(NC(CC(=O)OC)=O)(CO)CCN(C(=O)C=Cc2sc(Cl)nc2Cl)CC1 c1(C(N2CC=CC(NC(C=CCCC)=O)C2)=O)nc2nc(C)cc(C)n2n1 c1(C(N2CCC(N(C(=O)CSC3CC3)CC)C2)=O)cc2c(nc1N)CCCC2 c1(C(=O)NC(CC(C)NC(C=CCC)=O)C)cccc(Br)c1OC c1(CN(C(C(F)OC)=O)C)cccc(CNC(c2cnn(C3COC3)c2)=O)c1 CC(C)C(CNC(=O)CC1CCCC1)C(=O)NC(c1ccccc1F)C CCC(C)C(C(=O)NC1CC(n2ccnc2)C1)NC(=O)Cn1cc(C)cn1 C12(C(=O)NCC(C)(C)SC)COC(C1)C(NC(c1ccc(O)nc1)=O)C2 c1(OC)c(C(=O)N(C2CCN(C(C3CCC3)=O)C2)C)cccc1-c1ccncc1 c1(C(N2CCN(c3nc(C(=O)OC)c(Cl)cn3)CC2)=O)cc(C)c(Cl)cc1Cl c1(CC(N2CC=CC2CNC(c2cncc(C(F)(F)F)c2)=O)=O)ccc(O)cc1 c1(NCCNC(CCSCC)=O)ccc(NC(=O)CC(C)F)nc1 c1(C(N2CC(Cc3cn(CCCF)nn3)C(O)C2)=O)ccc(Cl)cn1 Cc1nc(CCC(=O)NCC2CN(C(C3CC(N=[N+]=[N-])C3)=O)C2)[nH]c1C CCC(C)C(CC(=O)NC1CN(CC)CC1C)NC(c1ccns1)=O C(=O)(C(F)(CNC(C1CC(=O)NC(C)C1)=O)C(C)C)N(C)Cc1onc(C)n1 N1(C(c2c(CC)onc2C)=O)CC(CNC(c2c[nH]nc2OC)=O)OC(CC)C1 N1(C(C2(CCC=C)CC2)=O)CC2(C)CN(C3CCCCCCC3=O)CC2(C)C1 c1(CC)cccc(C(=O)NC2CCC(CC(=O)NCC(O)C(C)O)C2)c1 C1(SC)CN(C(C)(C)C)CC1NC(=O)NCCn1nc(C(F)(F)F)cc1Cl N1(c2nc(CC)cc(CC)n2)CCC2C(CCCN2C(C2CCCN2C=O)=O)C1 N1(C(C(C)(C)OC)=O)CC2CCC1CN2C(c1scnc1COC)=O CCCN=C(NCC1COCCN(C(=O)OC(C)(C)C)C1)NC1CCCC1C1CC1 N(C1CN(C(c2ns[nH]c2=O)=O)Cc2ccccc21)C(C(C)C(F)(F)F)=O N1(C(COCCC#C)=O)CC(CNC(=O)C(C)P(C)(C)=O)CC1(C)C c1(C(C(=O)NCC(CC(=O)OC)C)F)nc2ccccc2s1 N1(C(C2C(c3onc(COC)n3)C2)=O)CCC(C)C(NC(=O)C2=CCCC2)C1C c1(C(N2C(CNC(C3(COC)CCC(=O)N3)=O)CC2)=O)ccc2c(c1)CC(C)O2 c1(NC(C2(C)N(C(C#CC)=O)CCC2)=O)ccc2c(C)n(C)nc2c1 C(CCCCC(=O)NCCC1CN(C(=O)CSCC(C)C)CC1C)OC c1(C(=O)NC(CNC(C(C)OCC)=O)C(C)C)cc(C)ccc1Br c1(C(=O)NCC(C)N(C)C(c2cncn(C)c2=O)=O)noc2c1CC(C)(C)CC2 C1(O)(CNC(C(C)(O)C2CCC2)=O)CCCN(C(c2cc3[nH]ccc3s2)=O)C1 c1(OC)cc(Cl)c(C(N2CCN(C(C3CC(O)C3)=O)CC2CF)=O)cc1Cl C(=O)(CCC(=O)N1CCC(NC(=O)CC2(O)CCOC2)C1)NCCOCCC CC1=C(C(=O)NCC2C(C)CCCN2C(c2ccc3nn[nH]c3n2)=O)CCCC1 N1(C(C2CCC(=O)O2)=O)CCOCC1CCNC(C1(CO)CCOCC1)=O c1(OC)cc([N+](=O)[O-])c(NC(C2CC2NC(c2cc(O)ccc2F)=O)=O)cc1F C1(CCC)CN(C(C2CC2CC)=O)CCN1C(=O)CC(O)C1CCC1 C1(NC(C(C)NC(=O)NC)=O)CC2CC(NC(c3cc(F)ccc3Cl)=O)C2C1 O=C1CCC(C(=O)N2CCC3OCC(=O)NC3C2)n2cccc21 C1(NC(C(C)(O)C2CCC2)=O)CN(C(c2cccs2)=O)CC1n1ccnn1 N1(C(c2ncc(OC)nc2)=O)CCCC(NC(c2[nH]c(C)c(C)c2C)=O)C1CC Cc1nc2nc(=S)[nH]n2c(C)c1CCC(=O)NCC#CCNC(=O)C(O)C(C)C N1(C(CC=C)=O)CCC2CC12C(=O)NCCSCc1cccnc1 c1(OC)ccccc1C(C(=O)NCC(C1CCC1)NC(c1cc(Cl)no1)=O)OC N1(C(CNS(N)(=O)=O)=O)CC(NC(=O)C=CC2CCC2)CC(O)C1 c1(C(N2CCC(NS(CC(=O)OC)(=O)=O)C(C)(C)C2)=O)ccc2ccncc2c1 c1(C(=O)NCC2CC(OC)CN2C(c2ccon2)=O)cc(N)c(C)cc1Cl N1(C(CN2CCC(C)C2)=O)CC(N(C)C(C2CC(n3ccnn3)C2)=O)C2(CC2)C1 Cc1[nH]nc(C(=O)NC2CN(C(=O)C=Cc3cn[nH]c3)C3CC23)c1C N1(C(C(CC)OC)=O)CCC(C)(C)C(C(N2CCCCCCCC2)=O)C1 C(=O)(CCCC(F)(F)CO)NCC(n1cc(COCC(=O)OC(C)(C)C)nn1)C C(C(=O)NC(c1cscn1)CO)(C(C)CC)N(C(C(F)=CCC)=O)C N1(C(C2CCCN(C(C(C)OCOC)=O)CC2)=O)CCCNC(=O)C1C C1CCN(CC(O)CC2CCCC2)CC1C(F)(F)F C1(C(=O)NCCOCCOCCO)CCC2CCC1N2C(C1CCCS1)=O CCC(N=c1[nH]c(N2CCc3ccccc3C2)nc(=N)[nH]1)c1cccnc1 c1(C(=O)NCC2(C(N)=O)CN(C(CCC=CC)=O)C2)ccc(F)c2ccncc12 c1(C(N2CC(N(C(c3ccc(C)s3)=O)C)C(F)C2)=O)cc2cc(Cl)ccc2n1C c1(C(=O)NC(C2CCN(C(c3cc(C4CC4)cs3)=O)C2)C)ccnc(F)c1N c1(OC)cnc(C(=O)NC(C2(O)CN(C(C3(CC)CCNC3=O)=O)C2)C)c(F)c1 C1(N(C(c2ccccc2)=O)Cc2cncc(Cl)c2)CC2CC1CN2 C1(C(=O)NCC2CCCN(CC#C)C2)CC(F)(F)CN1C(=O)C(CC=C)OC N1(C(COCCOCC)=O)CC2CCC1C1CN(C(=O)C(C)OC(C)(C)C)CC21 N1(C(c2ncc(CN(C)C)s2)=O)CC(F)(F)CC1C(=O)OC(C)(C)C C1(C(N2C(C)C(NC(=O)Cc3cn[nH]c3)CCC2)=O)CC2C=CCC(C1)C2 c1(CSCCOCCC#C)cccc(OC(C2CCS(=O)(=O)C2)=O)c1 c1(C(=O)NC(C(CO)NC(c2cc(C(C)=O)sc2)=O)C)cnnc(O)c1 N1(C(CNS(N)(=O)=O)=O)CCC(C2CCCN(C(c3cccc(F)c3F)=O)C2)C1 c1(OC)ccc(CC(N2CCC(NC(=O)CCC3CC(F)(F)C3)CC2)=O)cc1 c1(OC)ccn2c(C(=O)NCCC(C)(C)NC(=O)CCNC(N)=O)cnc2c1 c1(SCC(=O)N(CC(C)NC(c2nc(C(C)(C)C)no2)=O)C)cnn(C)c1 C1(CC(=O)NC(CN(C(c2cc(C(=O)OC)nn2C)=O)C)C)CCOC(C)(C)C1 CCCC(C)C(=O)N1CCC(O)(CCNC(c2coc(Br)c2)=O)C1 N1(C(c2cnc(C)s2)=O)CCC(NCc2cc(C(=O)O)ccc2F)C(F)C1 c1(C(c2nnnn2C)NC(C(COC)C)=O)ccccc1Cl.C12CCCN1C2 C(=O)(C1=CC2C=CC(C1)C2)NC(C(=O)Nc1ccc(OC)c(C)c1)C(C)(C)C C(=O)(C(C(C)NC(c1cn(C2CC2)cn1)=O)C(C)C)NCc1cc(C)no1 C(=O)(CC(C)CC(C)C)N1C(Cn2cc(CCCOC)nn2)CCC1 Cc1c(Br)sc(-c2nc(C3CCCC3)no2)c1C Cc1cccn2c(CC(=O)NC(CNC(C34CC(CO3)C4)=O)CC(C)C)cnc12 C12(C(N3C(COC)C(C)(C)C3)=O)CCC(CC1)N(C(=O)Cn1cc(C#N)cn1)C2 C1(N(C(=O)C(C)C2CCCO2)CCCC)CCN(C(C2CCS(=O)(=O)N2)=O)CC1 C(=O)(C1=C(c2ccccc2)CCC1)NC1C(C)C2CC(C1)C2(C)C c1(C(N2CCC(C(=O)NCc3n(CCC)ncn3)C2)=O)cc(C)ccc1F O=C1NCCCCC1C(=O)NC1CN(C(c2cc(Br)no2)=O)CC1O O=C1CN(CC(=O)NC2CC(CCC(=O)NC3CNC(=O)OC3)C2)CCN1 C#CCCN=C(NCCC1CSCCO1)N1CCC(Cc2ccccc2)C1 C(CCCCCN=c1cc(C2CC2)nc[nH]1)N(C)C(c1ccc2c(c1)CC2)=O n1(COC)ncc(C(N2CCC(CCNC(=O)CC(CC)OC)C2)=O)c1C C=C(CNC(=O)CCN(CC(C)C(C)C)C)CCNC(=O)CC1CCCN1C C=C1CC(C(=O)Nc2cccc(CO)c2)N(Cc2csc(-c3ccccc3)n2)C1 C1(CNC(CNC(C(CC)C)=O)=O)C2CC1N(C(=O)COc1cccc(C)c1)C2 c1(CCNC(N2CCCC(C(C=CNC(C)=O)C)C2)=O)cc(C)ccc1F c1(C(N2C(C(=O)NCCOCCCC)C(C)(C)CC2)=O)ccc(C)nc1C c1(-c2c(NC(Cc3c(OC)ccc(F)c3)=O)ccnc2)ccc([N+](=O)[O-])cc1 CS(C)(=O)=NCC(=O)N1CCN(C(c2ccc(C(F)F)cc2F)=O)CC1 C=CCC(CC(C)C)C(=O)NCc1cc(C(N2CCOC(COC)C2)=O)co1 C1(C2CN(C(=O)CCCC3(C(=O)O)CCC3)C2)(NC(CC2CCCC(C)C2)=O)CC1 C1(CC)CN(C(C2(F)CC2)=O)CC1NC(C1CC(=O)N(C(C)C)C1)=O c1(C(=O)NCC(C)(C)OCC(N2CCC(C(C)O)CC2)=O)csc2nccn12 c1(C(N2CC(F)(CNC(C(C)OCCOCC)=O)C2)=O)cc(C)nn1C N1(C(C(C2CCCC2)NC(C2N(CC)CCOC2)=O)=O)CCCC(C)(C)CC1 C(CC(C(C)(C)C)NC(=O)CCCCC#N)N(C(C1C(CC)C1)=O)C N1(C(=O)OC(C)(C)C)CCCC2(CN3CCC(C#N)CC3)CC2C1 C1(C(=O)NC2CCC(NC(C3C(C=C(C)C)C3(C)C)=O)CC2)CCCS(=O)(=O)C1 N1(C(CC2CCC(C)(C)O2)=O)CC(C(N2CCC(C)(C)C2)=O)C2(CC2)C1 c1(C(=O)NC(C(C)NC(C2(CC)CCCC2)=O)C)ccc2occc2c1 c1(OC)ccc(C(=O)NCC2(NC(C3CCN(C4CC4)CC3)=O)CC2)cc1 C12(C(=O)OC)CCC(C(N3CCN(C(=O)CC4CC(C)=NO4)CC3C)=O)(CC1)C2 CC1=NOC(=O)C1CC(=O)NC1C=CC(CNC(=O)C(C)(C)c2cccnc2)C1 C1(C)(C(c2n(CCOCC)nnn2)NCC(C)(C)COC)CC=CCC1 C1(CNC(C2CCCC23CC3)=O)CCCCN1C(c1cnc(CC2CC2)s1)=O C(=O)(C#CC1CCOCC1)NC(CC#C)(C)C(=O)NCCN1CCNC1=O n1(CCNC(C(C)n2ccnc2)=O)ccc(C(=O)NCC2COC(=O)N2)c1 N1(CC(=O)N(CCNC(c2ccnnc2O)=O)CC)CC(=O)N(C)C1=O N1(C(c2ccc(C=C)cc2)=O)CCC2(C)CN(C(=O)C(c3ccnn3C)C)CC12 Cc1cccc(C(=O)NC2CC(CNC(=O)COCC3CCC3)C2)c1F n1(-c2c(OC)cccc2)cccc(NC(c2ccn(C)c2)C)c1=O C(c1ccc(Cl)s1)=CC(=O)NC1(CNC(CCc2nc(C)sc2)=O)CCC1 c1(C(=O)NCC(C)N(C)C(c2coc(Cl)n2)=O)c(Cl)c([N+](=O)[O-])nn1C C1(C(=O)NCC(C)(C)SC)CC2CC1CC2NC(=O)C(C)n1cccc1 C1(NC(C(=O)NCCOC(C)=O)=O)C2CCCOC2C1(C)C c1(C(=O)NC2(C)CCN(C(c3cc(C#N)ccc3O)=O)C2)cc(S(C)(=O)=O)co1 C1(C(N(CCNC(c2ccncc2Br)=O)CC)=O)CCOC2(CCC2)C1 C1(C)(CC(N2CC(COC)(CNC(C3CC(C)CO3)=O)C2)=O)CCOCC1 CCC(CC)CC(F)C(=O)NCC(C(=O)N1CCC(C)(CO)C1)C(C)(C)C CCCCC(C)(F)C(=O)NCC1CCCN(C(c2ccc(SC)o2)=O)C1 C(=O)(C(CO)NC(C1COCOC1)=O)N(CC(CC)O)C c1(C(=O)O)nccc(OC)c1C.C1(CNCCCC)COCCN1CC N1(C(CC(CC)(F)F)=O)CC(C(N2CC3CCC2C(O)C3)=O)C2(CCC2)C1 Cc1c(CC(=O)NCCCN(C)C(C2CCC(=O)N(C)C2)=O)cccc1[N+](=O)[O-] C1(O)(C(C)NC(c2cc(Cl)c[nH]2)=O)CCN(C(c2cnn(C)c2Cl)=O)C1 CCC(C(=O)N(c1ccccc1)C1CN(C(=O)CC2OCCO2)C1)OC c1(C(=O)NCC2C(C)CCN(C(=O)Cc3cnns3)C2)cc(S(N)(=O)=O)c(Cl)o1 C=C(C)CCC(=O)NCCCC1CN(C(C2(N3CCNC3=O)CC2)=O)CCO1 c1(CN(C(C2(C=C)CCC2)C(=O)NCCC#N)C)cc(F)c(Cl)cc1F n1(C2(CC(=O)N(CCCN(C(COCC(C)C)=O)C)C)CC2)cncn1 c1(C2(C(=O)O)CN(C(C(CC)OCC)=O)C2)cc(Cl)cc(Cl)c1 C1(CC(=O)OCC)(NC(C2(CCF)CC2)=O)CCCS(=O)(=O)C1 c1(Sc2cc(C)nc(C3CC3)n2)nc2ccccc2[nH]1 c1(C(N2CC(O)(CCNC(C3CCC(C)O3)=O)C2)=O)ccc(-c2cccs2)cn1 CCC(C)(C(=O)OC)Oc1ccc(SC)cc1.C1(c2cn(COC)nn2)CCCCC1F C(=O)(C1=NN(C)C(=O)CC1)NC(C(=O)N(C)CCC1CCCN1C)CC(F)F c1(C(C(=O)NCCCOCCCNC(C(CC)F)=O)(F)F)ccc(C)cc1 c1(C(N2CCN(C(COC(C)=O)=O)C(C)C2)=O)cn2nc(C)cc2[nH]c1=O CC1(C)CCCN(C(=O)CN2CC3CCC2C3)C1CNC(C1(C2CC2)CC1)=O Cn1ncc2cccc(C(=O)NCCC3CCN(C(=O)CCC(F)(F)F)C3)c12 c1(C(N2CC(NC(C3CCCC(C)C3)=O)C(C)CC2)=O)cn2c(n1)CCCC2 C1(C)(CNC(CNC(=O)OCC=C)=O)CCN(C(=O)C(c2ccccc2F)F)C1 c1(N2CC(C)(C)OCC2)nc2ccccc2nc1N1CCC(C)(F)C1 C1(C(=O)NCC(O)C2CCC2)CN(C(=O)C=Cc2cccnc2)CC1C1CC1 Cc1cc(Br)ccc1NC(C1CCCCN1C(=O)CCOC(C)C)=O C#CC1CC2CCC1N(C(=O)CSCCNC(C1COCCO1)=O)C2 C#Cc1ccccc1NCC(=O)N(C1CCN(C(=O)C(CC)CC=C)C1)C N1(C(C(CC)=CC)=O)CCCN(C(c2csc(C(C)(C)C)n2)=O)CC1CO C1(C(=O)NCC2C(C)CCN(C(=O)COC3CCOC3)C2)CC2CCCCN2C1 N1(C(C(C)OCCN(C)C)=O)CC(O)(CCC2N(CC(=O)NC)CCC2)C1 C12(C(=O)NCc3c(C4CN(C(CCS(N)(=O)=O)=O)C4)ocn3)CCC(=O)N1CCS2 C1(C(N2CC(CC=C)(NC(c3ccccc3OC)=O)C2)=O)CC2(CC2)CN1C C(=O)(C(C)(O)CC(C)C)N1CC(O)(CCNC(C(CC)C)=O)C1 CC1CCCN(C(c2cc(CN3CCCC(O)C3)nn2C)=O)C1 C=C1CC2(C1)CC(C(N1CCC(CNC(C3CCCCC3F)=O)C1)=O)C2 Cn1cc2ccc(C(N3CCC(CF)(NC(=O)CC4CNC(=O)C4)C3)=O)cc2n1 Cc1cc(C2CCN(S(=O)(=O)CCCOC(C)(C)C)CC2)c2c(n1)CCCC2 CC1CC(NC(=O)C=CC2CCN(C(=O)C(C3CCCCC3)C)CC2)CC(C)O1 c1(C(N2CCCC(NC(C3(C(=O)OC)CC3)=O)C2)=O)cc2c(OC)cccc2s1 c1(OC)nccc(NC(C2CCCN2C(=O)C(C)(C)F)=O)c1Br C1(C(=O)Nc2ccc(C)cc2)CC(F)(F)CN1C(c1sc(C)nc1C)=O c1(OC)cc(C=CC(=O)N(C)C(c2ccccn2)C2CC2)ccc1F c1(C(=O)NC2CN(C(CCCOC)=O)CC2C)ccc2c(c1)NC(=O)CCN2 N1(C(c2c(C(C)NC(=O)Cc3ccc(F)nc3)noc2)=O)CCCC(F)CC1 c1(C(N(C2CC(NC(=O)C(C)(C)c3cc[nH]n3)C2)C)=O)ccnc(F)c1O CCCC(C)(O)CC(=O)N1CCC(NC(C2CCC=CO2)=O)C(CO)CC1 C12(C(=O)NC(CC(C)NC(c3ccccc3Br)=O)C)CC3CC1C2C3 Cc1cc(CNCC2CCC(C(=O)N(CC(C)O)CCO)CC2)ccc1[N+](=O)[O-] C1(OC2(C(=O)NCCC3CC(NC(c4c(C)cno4)=O)C3)CC2)CCCCC1C c1(C(C)OC)nc(N2CCOCC(NC(=O)Cc3cc(C)nn3C)C2)cc(Cl)n1 CC1CC(NC(=O)CCN2CCCC2)CCN1C(=O)C(C(C)(C)C)c1cc[nH]n1 N1(C(C(n2ncc(C)c2)C)=O)CCC2(C1)CN(C(=O)CCC1CC1C)C2 CC(=O)CCCC(=O)N1CC(CNC(=O)CCCn2nc(C)nc2C)C(C)(C)C1 C1(CCNC(C(C)(C)OCC)=O)CCCN(C(=O)Cn2ncc(Br)n2)C1 C1(n2cc(-c3cnc(C)o3)nn2)CCCN(C(=O)CCC2CC2(Cl)Cl)C1 Cc1coc(C(N2CCCC2C2(O)CN(C(=O)CSCCOCCN(C)C)C2)=O)c1 Cc1c(C(=O)NC2CCC(CC(=O)NC3CC(C)OC3=O)C2)cncc1F c1(C(N2CC(N(C(CC3(OCC)CCC3)=O)C)C2)=O)cccnc1CC(C)C N1(C(CC(C(C)C)C)=O)CCCCC2(CCN(CCO)C2)C1.c1(CCC)ccccc1 CC(CO)(CO)C(=O)N1CC2C(C(=O)NC(C)(CO)C3CCCC3)C2C1 c1(C(CC)=O)cccc(S(=O)(=O)Nc2c(F)cnn2-c2ccc(Cl)cc2)c1 N1(C(c2cc(C)ncn2)=O)CC=C(CNC(c2ccc(N(C)C)cc2)=O)CC1 C1(NC(=O)C(C2CCOCC2)F)C2CC1N(C(c1nccnc1C(F)(F)F)=O)C2 c1(CC)cc(C)c(C(=O)NCC2C3CN(C(C4CCSC4)=O)CC23)o1 CN1CCC(C(N2CC=C(CNC(=O)CCCCNC(N)=O)CC2)=O)CC1=O c1(C(C=CC(=O)OC(C)(C)C)=O)c[nH]ccc1=NC(=O)CCc1cccc(F)c1 CCCC(C(=O)OC)C(=O)NCC(C)(C)CC1CN(C(C2CCCS2)=O)C1 c1(SC)cc(C(=O)NCC(CO)NC(=O)C(c2cccc(Cl)c2)C)c(C)o1 C1(COC)(CNC(c2cc(CNC(=O)CCOC3CC3)cs2)=O)CCOC1 CC(=O)CCN=C(NCc1nc(C(F)(F)F)n[nH]1)N1CCC(c2nncs2)C1 N1(CCCNC(=O)CCc2cnn(C)c2)CCN(Cc2n(CCC)nnn2)CC1 C1(C(C)NC(c2ccc(Cl)nn2)=O)CCN(C(=O)CN(C)CCO)CC1 c1(C(=O)NCCCCC(C)NC(C2(O)CC2)=O)cc[nH]c(=N)c1[N+](=O)[O-] N1(C(C2C3CC(=O)CC32)=O)CC(C2CC2)(C(=O)NC2CCC(CO)CC2)C1 N1(C(C(COCC)(C)C)=O)CC2(C1)C(NC(C13CC(C)C1C3)=O)CCS2(=O)=O N1(C(COCc2cc(C)on2)=O)CCN(C(c2cc(C(F)F)n(C)n2)=O)C(C)C1 n1(CCOCC)nc(-c2ccn(C)n2)nc1-c1sccc1CC1CC1 N1(C(c2ccc(C(C)=O)o2)=O)CCC2CCN(C(=O)C(O)C3CCC3)CC12 C1(NC(CC(=O)NCC)=O)CC2CC1N(C(c1sc(C(C)C)nc1C)=O)C2 c1(NC(c2cccc(COC)c2)=O)cc2sc(OCC(F)F)nc2s1 CCC(CC(=O)NC1CN(C(c2cc3oc(C)cc3[nH]2)=O)CC12CC2)C(F)F N1(C(COCCCC#C)=O)CCC(CNC(c2ncccc2CSC)=O)C(O)C1 C(=O)(C(=O)N=c1cc(C)o[nH]1)NCC1C2N(C(C(F)=CC)=O)CC(CC2)C1 CC(C)CC(C(=O)NC(C(=O)NCC(F)CC)C(C)O)C(C)C N1(C(C)=O)CCN(C(CCS(N)(=O)=O)=O)C2CCC12 N1(C(Cc2cc(C)sc2)=O)CCN(C)CC1C(=O)NC1CC(C#N)C1 CC1CN(Cc2cccc(C(N3CCC(C)(c4nn[nH]n4)C3)=O)c2)CC(C)O1 c1(CC(=O)NC2CC(CNC(C3(O)CC3)=O)C(O)C2)c[nH]c2cc(F)ccc12 C(=O)(C(O)CC(F)(F)F)NC1CC(NC(c2ccccc2-c2cncnc2)=O)C1 C1(NC(c2c(OC)scc2)=O)CC2(CCN(C(c3csc(C(F)F)n3)=O)C2)C1 CC(C(=O)NC1CC(NC(=O)CC2(n3ccnc3)CC2)CC1O)C(C)(C)C Cc1cc(C(N2C(C)(CC(=O)Nc3ccc(C)nn3)CCC2)=O)cc(O)c1 C1(CC)C(NC(=O)C(C)COC)CCCN1C(c1cncc(NC)c1)=O CC(C)C(F)C(=O)N(C)CCOCCCN(C)C(C1C2CCC1CC2)=O Cc1ccn2ncc(C(=O)NC3(CNC(=O)Cc4nn(C)cc4Br)CCC3)c2c1 CC1(C(=O)NC2CCCCC2NC(c2ccc(OCCO)nc2)=O)CCCS1(=O)=O c1(C(=O)NCCN(CCC)C(c2cccs2)=O)ccccc1S(=O)CC C1(CNC(C2C(OC)(OC)CC2)=O)CCN(C(=O)C(C)(C)C2CCCC2)CC1 C1(NC(COCCOCC)=O)COCCC1C(=O)N(C)CCF.C(=O)C(CC)CC C1(C(=O)NCc2c(C)cccc2)CCCCC1(C)NC(C1CC=CC1)=O c1(C(N2CCC(CCNC(=O)COC(F)(F)F)C2)=O)cnc2c(c1)CNC2=O c1(C(=O)NCC2(O)CCN(C(C3CC(CC)C3)=O)C2)cc2ccccc2cc1F C(=O)(C(C)C(O)C(C)C)NC1C(NC(c2c(C)oc(C(C)(C)C)c2)=O)CCOC1 Cc1cc(Cl)c(CNC2CCNCC2)cc1C C1(O)(C(=O)NCC(CC)NC(=O)C(n2cc(C)cn2)C)CN2CCC1CC2 C=CCC(C)(CC=C)NC(=O)C(CCF)NC(C1CC1=C)=O C=Cc1ccc(C(=O)NCC(CNC(C2(CO)CC=CC2)=O)CO)cc1 c1(CC(N2CCC(N(C(COCCOCC)=O)C)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 N1(C(CN(C)C(N)=O)=O)CCC(C)(NC(=O)CC2C=NN(C)C2=O)C1 C=CCC(C)C(=O)N1CC(NC(=O)C(c2ccc(C)cn2)(F)F)C(O)C1 C=CCCCC(C(=O)NC1CCCN(C)C1)NC(c1cnsc1C)=O N1(C(c2cn(C)nc2)=O)C2CCC1CN(C(c1cc(Cl)sc1Cl)=O)C2 c1(C(N2CC(CC)C(NC(C3CC(=O)NC(C)C3)=O)C2)=O)cc(C)c(F)c(C)c1 c1(C(N2CCC(C)(CC(=O)NCCC(CC)(F)F)C2)=O)ncn2ccccc12 S(=O)(=O)(c1cc(C=CC(=O)Nc2nc(Cl)c(NCCSC)s2)ccc1OC)OCC C(=O)(C1CCCc2nc(C)[nH]c21)NC1(CN(C(=O)Cc2nnc(O)s2)CC)CC1 c1(CC(C(=O)OC)NC(c2cc(C(C)=O)c[nH]2)=O)ccc(C(F)(F)F)cc1Cl c1(CCC(=O)NC(c2cn(CC(=O)OC)nn2)C2N(CC)CC2)ccc(C)cc1 C1(C(=O)NC(C)(C)C=CC)(NC(C)=O)CCC1.C1(O)(C(=O)NCCO)CCC1 CC1OC(C)C(C(=O)NC(C)(C)CNC(c2cnc(Cl)c(N)c2)=O)C1C C1(N(C(CC(=O)OCC)=O)C)CN(C(c2cnn(CC)c2Cl)=O)CC1F C(=O)(C#CC1(C)CCCO1)NCC(C(C)C)NC(C1(S(C)(=O)=O)CC1)=O C1(NC(=O)C(c2ccccc2)F)CC2C1CCN2C(=O)CCc1cccc(Cl)c1 C(N=c1[nH]c(C)cc(=NCCN2CCP(C)(=O)CC2)[nH]1)c1ccc(CC)s1 C1(C(C(=O)NCC(C)(C2CC2)NC(C2(CC#C)CC2)=O)=O)CCCCC1 c1(C(N2C(CCNC(=O)C3CC3)CC(F)(F)C2)=O)cccc2c1OCO2 C1(C(N2CC(C)(OCC(N3CC(C)C(C)C3)=O)C2)=O)CC(C)(C)CN1C C(CCCC(CO)NC(=O)CCOc1ccc(C)c(C)c1)NC(C(CC)C)=O c1(C(=O)NC(CNC(c2c(C)coc2)=O)C(C)C)cccc(CC(C)C)c1 c1(NC(c2c(C3CCN(C(CC=CCC)=O)C3)n[nH]c2)C)ccc(C)n1CC ClC(Cl)CN=c1[nH]c(=NCc2ccc(-c3ccccc3)cc2)[nH]c2c1CSC2 N1(C(c2cnc(CNC(C(CCCOC)C)=O)nc2)=O)CC(C)(C)C2COCC12 N1(c2c(C)c(NC(C)C)ncn2)CCOc2cc(F)ccc2C1.C12CCN(C1)C2 c1(C(=O)OC)c(C)cc(CNCCCCc2cccnc2)cc1Cl c1(CCCNC(C2CCC(C)O2)=O)ccc2c(c1)CNC2 CC(C(=O)NC1(CF)CCN(C(c2cc(Cl)cs2)=O)C1)C(F)F c1(COC(C)C)ccc(C(=O)NCC2CCC2NC(c2cc(O)cs2)=O)cc1 C12CCCC3CN(CC13)CC1(CC1)C(=O)N2.c1(C(N(C)C)=O)ncoc1C(F)F c1(CC)ccc(C(N2CCCC2C2(O)CN(C(C3(C4CCCO4)CC3)=O)C2)=O)s1 C1(NC(Cc2cc(OC)no2)=O)CN(C(=O)CNc2ccsn2)CCC12CCC2 C1(O)(CNC(c2c(C(N)=O)coc2)=O)CCCN(C(=O)COC2CCOCC2)C1 CC(C(=O)NCC1(C)CC(NC(c2cn(C)nc2Br)=O)C1)C(F)(F)F C1(NC(c2c(CC)onc2C)=O)COC2(CCN(C(c3cocn3)=O)C2)C1 c1(C(=O)OC(CNC(C(C(CC)C)=O)=O)=O)ccc2c(c1)OCCO2 N1(C(c2c(CC)nco2)=O)CC2(CC2)CC1CNC(=O)CSCCN(C)C c1(C(N2C(CNC(Cc3c(C)ccc(F)c3)=O)C=CC2)=O)cc(F)cc(N)c1F N1(C(C(CCCC)(C)F)=O)CCC(C2(NC(C3CCCC4CC34)=O)CC2)CC1 N1(C(C2CC2F)=O)CCN(C(=O)CCCF)CC1c1cccc(Cl)c1 C(=O)(CC(CC)CCCC)NCC(N(C(CCCCC=CC)=O)C)C1CC1 N1(CC(=O)Nc2c(C)c([N+](=O)[O-])c(F)cc2)C(C)c2ccccc2C1C c1(C(C)(C)C#N)cc(CO)cc(C(F)(F)F)c1.C12CCC(C1)CNC2=O c1(SCCCC)cccc(C(=O)NC(C)CC(C)NC(c2nn[nH]c2Cl)=O)c1 c1(OC)cccc(C(=O)NC(C)C(C)NC(=O)C(c2ccccc2F)C)c1F c1(OC)cc(NC(=O)CC2CCO2)cc(F)c1F c1(C(=O)NC2CC(C(N3CC(COC)C3(C)C)=O)C2(C)C)ncc(F)cc1C N1(C(C=CSC)=O)CCC(C(C)NC(C2CC(O)(C(F)F)C2)=O)CC1 C(=O)(C(F)(F)C(F)(F)C(F)F)NC(C1CN(C(C2CC(F)C2)=O)C1)C C1(NC(C(=O)NC)=O)CCN(C(=O)CCCOc2ccc(F)cc2Cl)C(C)C1 N12CCC(O)C(C1)CN(C)CCC2=O.c1(SC)cc(Cl)ccc1C(=O)OC(C)=O C1(CC)CCCC1C(=O)NC(C1CN(C(c2ccnn2C(CC)CC)=O)C1)C N1(C(C(C)OCC)=O)CCN(C(c2nc(C(C)C)ncc2Br)=O)CC1CC C(=O)(C1=C(C#N)CCC1)N1C(C)(C(=O)NCC2C(C)(C)CCCO2)CCC1 c1(C(=O)OCC)sc(N(C)Cc2cn(C)cn2)nc1Cl C1(NC(CN(CCC#C)C)=O)CC(C(=O)NCC=C)C1.C(=O)(COCC)N c1(C(N(CC(C)NC(c2c(COC)cc[nH]2)=O)CC)=O)sc(C)c(C)c1C c1(OC)ncc(Cl)cc1C(N1CC(CNC(=O)Cn2cc(C#N)cn2)(OC)C1)=O N1(C(CCCC#C)=O)C(C)C2CC1C2NC(C1CCCCO1)=O Cc1nc(C)c(C(=O)NCCC2CN(C(=O)CSc3ccncc3)C2)s1 C1(NC(C(F)OC)=O)CCOC2(CCN(C(c3coc(Cl)c3)=O)CC2)C1 O=C1C=CC(C(=O)NC2CCC(C(=O)Nc3ccccc3C(N)=O)CC2)N=N1 c1(C(N2CCC(CNc3n(C)ccn3)CC2)C(N)=O)ccc(F)c(F)c1 S(=O)(=O)(c1cnc(NC(CN(C)C)CO)c(Cl)c1)NC(C)Cc1ccc(F)cc1 CC1(C(=O)NC2CC(CNC(=O)C(=O)NCC(F)F)C2)CC2CC2C1 C1(NC(C2OCC(=C)C2)=O)CCCCC1c1nc[nH]n1 OCCCCC(Cc1ccccc1)c1nc(-c2cscc2C(F)(F)F)no1 C(C(C)(C)C(F)(F)F)NC(c1n(CCCC)nnn1)CC(C)OC(C)(C)C c1(SCC)cccc(CC(N2CC(NC(=O)CCN(C)C(C)=O)C(SC)C2)=O)c1 Cc1cc(CCC(=O)NC2CCC2NC(C2COCC(C)(C)O2)=O)ccc1Cl C1(CNC(C(=O)NC(CC(C)C)(C)C)=O)CCN(c2ccccc2)S1(=O)=O C(CC(=O)NC1CCN(C(=O)C=CC2CCCC2)C1)(C1=CCCC1)OCC c1(NC(C2SCCN(Cc3n(C)ccc3)C2)=O)c(F)cc(I)cc1[N+](=O)[O-] N1(C(c2c(OC)cnc(F)c2)=O)CCCN(C(C2CCC(N(C)C)C2)=O)C(C)C1 N1(C(c2cc(C)ncc2)=O)CC2(CCCN(C(c3oc(C)cc3C)=O)C2)C1 C(=O)(C(CCC(C)C)NC(c1ncc(N)cc1C)=O)N1C(C)(CCC)CC1 C1(C(N(CCNC(C=CC)=O)CCC)=O)CCCN1C(=O)C(F)(F)F c1(C(N2C(C)C(NC(=O)CNc3ncccn3)CC2)=O)n[nH]c2ccc(Cl)cc12 C(=O)(CCCCCC#N)N1C(C(=O)NCC(C(=O)OC)(C)C)CC2(CC2)C1 Cc1sc(C(F)(F)F)nc1C(=O)NC(C)CNC(C1C(C)C1(F)F)=O c1(CC(=O)NC2CC(NC(c3csnn3)=O)C(O)C2)nsc2ccccc12 c1(C(=O)NCC2(F)CCC(NC(c3cc(SC)oc3)=O)C2)cc(Cl)cc(F)c1F c1(C(C)C)ccc(C(N2CCOC(CNC(c3cn(C4CC4)nn3)=O)C2)=O)cn1 C1(CCC)CN(C(=O)CC2CCCCC2)CC1C(=O)NOCCOCC1(C)CC1 c1(N(CCCOC)C)cc(NCC(N2CCN(C)CC2)C)ncn1 c1(C(N2CCCCC2CNCc2cccc(Cl)c2F)=O)cnc2cccnn12 c1(C(=O)NC(C(C)NC(COC(C)C)=O)C)c[nH]c(=O)c2ccncc12 c1(OC)nccc(C(C(=O)NC2CCOC2)N(C(C)(C)CCO)C)c1F N1(C(c2ccc(=NC)[nH]c2)=O)CCCN(C(c2cnc(C)cc2Cl)=O)C(CO)C1 c1(CCC)cccc(NC(=O)CCN(C(=O)CC2CCCN(C)C2)CCO)c1 n1(CC(=O)NC(c2ccccc2)C(=O)NCC2CC23CCC3)ncccc1=O C(=O)(CCCCC(=O)N1CC2CC(NC(c3ccnc(C(F)F)c3)=O)C2C1)NC C1(NC(Cc2c(C)ncs2)=O)CCN(C(c2c(Br)noc2C)=O)CC1 N1(C(c2nc(C(C)C)sc2)=O)CCC(C)(CCNC(=O)C(C)N(C)C)C1 O=C1CCCC(CC(N2CC(C(O)C(=O)NCC3CC(n4cncn4)C3)C2)=O)C1 c1(OC)ccc2[nH]c(C(=O)N(CCCCNC(=O)C(F)C(C)C)C)cc(=O)c2c1 CC(C1=CCN(C)CC1)NC(=O)CC(CNC(C1CC2CCC1O2)=O)C1CCC1 CCC(C)C(O)C(=O)NC1CCC(N(C(=O)COC2CCCOC2)CC)CC1 CCCCC(C(=O)NC)NC(=O)Cc1ccc(O)cc1Cl.c1(C2CCN2)ccccn1 Cc1cc(C(=O)NCC2CCN(C(C3COCC(C)(C)O3)=O)C2)[nH]c1C#N C1(NC(C=CSC)=O)CC2(CCC(NC(C3Cc4ccccc4O3)=O)CC2)C1 C(=O)(NNC(=O)Cn1cc(C(N)C(c2ccccc2)O)nn1)C1C(C)C1 C(C)(CCC(F)(F)F)c1nc(C2N(Cc3cc(C)ncn3)CCCC2)sc1 C1(CCC)CN(C(c2cc(O)nn2C)=O)CCN1C(=O)C(O)Cn1cncn1 c1(C(N2CC(C(C)NC(CN(C(C(C)C)=O)C)=O)OCC2)=O)cc(Cl)ncc1O CCC1=C(C(=O)NCC2CCN2C(c2c[nH]c(Br)c2)=O)CCCO1 C1(CNC(C=CCC)=O)CN(C(=O)C(C2CC2)OC)CCC12CCC2 C(C(=O)N1CC(C(C)(C)O)(CNC(C2CCC2COC)=O)C1)(C(C)C)SCC N1(C(c2cnc(CN(C)C)s2)C(=O)NCCSC)CCCOCC1 N1(C(C(CC)N(C)C)=O)CC(NC(c2ccc(C(=O)C3CC3)cc2)=O)C(C)C1 C(C(C)(C)CN=[N+]=[N-])NC(c1cc(CNC(C(C(C)C)OC)=O)sc1)=O c1(SC)ccnc(-c2nc(-c3ccc[nH]3)n(C(c3ccccc3)C)n2)c1 C1(C(=O)NC2CC3C(NC(=O)OC(C)(C)C)C3C2)CNc2ccccc2C1 C=CCCC(C)(C)NC(=O)C(C)NC(=O)CCCC(=O)OC Cc1cccc(CN2CCCC(C(=O)N(C)CC3CC3(C)C)C2)c1C N1(C(C(CC=C)c2ccccc2)=O)CCOC(C)(CC(=O)NC2(CO)CCC2)C1 c1(C(N2C(C(N3CC(C)N(C)CC3)=O)CC(C)C2)=O)ccc2ccncc2c1 c1(C(=O)NC(CNC(C2N(CC)CC2)=O)CCCC)cc(S(C)(=O)=O)cs1 CC1CN(C(c2ccc3c(c2)CCO3)=O)CCN(C(C2(NC(N)=O)CC2)=O)C1 C(=O)(C1=CC(O)C(NC(=O)CSC(F)(F)F)C1)NCc1ccnc(OC)n1 N12CCC3(CC1)CC3C2=O.n1(C(C)C)cnnc1CNC(C)CN1CCCCC1 N1(C(C(c2ccn(C)n2)C)=O)CCCC(N(C(=O)Cc2cnccn2)C)CC1 CC(C)C(CNC(c1ccc(N)cn1)=O)C(=O)NCC(=O)N(C)C1CC1 C12(CNC(Cn3c(C)cc(C)n3)=O)CCC1CN(C(=O)C=Cc1cc(C)on1)C2 N1(C(CC=CCNC(CCCCCN(C)C)=O)=O)Cc2ccncc2C1 C1(CNC(Cn2c(C)c(Cl)cn2)=O)(CO)CCN(C(=O)C(C)OCC2CC2)CC1 C1(C(=O)NC(CC(C)NC(=O)CSc2ccncc2)C)CC2(C1)CC1(CC1)C2 c1(OC)cc(NC(=O)CNC(=O)CCCCBr)c(CN2CCCCC2)cc1OC c1(C(=O)NCC2(C)CN(Cc3cc(C(F)(F)F)cc(F)c3)C2)ccc(F)cc1F CN1C2CCC1CC(C(=O)NCC(C)(C)CNC(C1CCCCC1C1CC1)=O)C2 c1(CC(=O)N(CCOC)CCNC(c2cccs2)=O)cnc(C(F)(F)F)s1 c1(CC(=O)NC2(CN(C)C(C34CCCC3CC4)=O)CC2)ccc(Cl)cc1F c1(C(C)C)nnnn1CC(=O)NCC(C(C)C)NC(=O)CC1CC1NC1CCC1 c1(OC)cc(-c2ccc(C#N)cn2)ccc1S(=O)(=O)N1CCN(CCC#N)CC1 C#CCC(C)(C)C(=O)NCCC1C(C)CCCN1C(=O)C(CC)CC N=c1ccc(C(=O)NCC2CC2CNC(C2(CC(F)F)CCNC2=O)=O)c[nH]1 c1(CC)ccc(C(=O)NCC(C2CC2)NC(c2c(C(C)C)n[nH]c2C)=O)c(Cl)c1 N1(C(CN(CCOC)C)=O)CC=C(CNC(=O)C(O)C2CCCC2)CC1 CC1C(CNC(=O)Cn2cc(CCN(C)CCO)nn2)N(C)CCN1C c1(NCC(=O)NCCc2c3cccc(C)c3[nH]c2)c[nH]c2cccc(C#N)c12 Cc1cc(Cl)c(C(N2CCC(NC(=O)CCn3cncn3)C23CC3)=O)cc1C C(CN=c1[nH]c2ccccc2o1)C1CCN(C(C(c2ccccc2)C)=O)CC1 N1(C(CCCC2(C)N=N2)=O)CCCC(CCNC(C23CCCCC2C3)=O)CC1 Cc1cc(NC2CCN(CCO)CC2)n(C(C)C)n1.C12CCC(CC1)C(=O)N2 C12(COC)CCC(C(N3CCC(O)(CNC(=O)C(C)C4CC4)CC3)=O)(CC1)CO2 N1(C(C(CC)NC)=O)CCn2cc(C(N3CCC(O)C(O)C3)=O)nc2C1 C1(NC(C(C)SC)=O)CCCC1(C)CN(C(=O)CCCc1cccs1)C N1(C(C(C(=O)OC)(C)C)=O)CCCC1C1CCCCN1C(c1cccc(Cl)c1)=O c1(C(N2CCOC(C(N3Cc4ccncc4C3)=O)C2)=O)n[nH]c2ccc(Br)cc12 c1(C(N2C3(CN(C(C(n4cc(Cl)cn4)C)=O)C3)CC2)=O)cc2cccnn2c1 c1(C(N2CCC(NC(c3c(C)nc(C)[nH]3)=O)CC2C)=O)ccccc1N=[N+]=[N-] c1(OCCOC)ccccc1C(=O)NCC12CC1CN(C(=O)C(C1CC1)OC)C2 C(c1ccc(Cl)cc1F)=CC(N1C(CNC(C(CC(C)C)C)=O)CC2(CC2)C1)=O N1(C(C(C)SCC)=O)CCN(C(c2occc2CC)=O)CC1C(C)C C#CC1CC1C(=O)NCCCN(C(=O)CCNC(C1CC1F)=O)C c1(C(=O)NC2(CNC(COCCCCC)=O)CCC2)cnc(C)nc1O c1(C(N(C)CC2CCCCN2C(C2OCC2(C)C)=O)=O)cc(O)cc(O)n1 c1(C(=O)NCCC(C)N(C(C(C)Oc2ccccn2)=O)C)ccc(F)cc1 C1(C(=O)NCC(CN(C)Cc2cc(Cl)cs2)O)CCC2(CCC2)O1 c1(CNC2CCN(CC)CC2)c(C)sc(C)c1Br C(C(O)C(=O)NCCCN(C(c1ccn(C)n1)=O)CC1CCCC1)SC CC1CC=C(C(=O)NCCC2(O)CN(C(c3cc(C4CC4)nnc3O)=O)C2)CC1 CCC(C)CCC(=O)N1CCCC(N(C)C(c2cc(C(C)(C)C)c[nH]2)=O)CC1 N1(C(C2N(CCC)CCC2)=O)CC2CC(NC(C3(CCOC)CC3)=O)C(C2)C1 c1(OC)ccc(Br)cc1C(=O)NCC(O)CNC(=O)C(O)C(F)F CN1CC2(C)CN(C(c3cc(-c4cccc(F)c4)c4cn[nH]c4c3)=O)CC2(C)C1 N1(C(C(C)CCN)=O)CCOC2(CCCCC2NC(c2ncc(F)cc2F)=O)C1 C(=O)(CCCC1CCCC1NC(C1CC1[N+](=O)[O-])=O)OC C1(C(=O)NCCN(C(c2ncc(C)nc2)=O)CC2CC2)CC(C)CC(C)C1 CC(C)CC(C)C(=O)N1CC(N(C)C)C(C(=O)NC2C=CC(C)(C)CC2)C1 c1(C(=O)NC2CC(NC(c3ncn(C(C)C)n3)=O)C2)cc(Br)ccc1N n1(CC(=O)NC2CCN(C(CC=C=C)=O)C2)ncn2nccc2c1=O c1(C(=O)OCC)ccc([N+](=O)[O-])o1.C12CC(O)CN1C2 S(=O)(=O)(c1cccs1)N1CCCC(O)C1.Cc1cc(-c2nnc(S)o2)ccn1 CC(C)N=c1nc(N2CCOCC2)[nH]c(=NCCC2=CCOCC2)[nH]1 C1(c2ccccc2Cl)(CNC(C2CCC(NC(C)=O)C2)=O)CCOCC1 c1(CC)ncc(C(C(=O)NC(C)C)N(CCF)C2CC2)o1 N1(C(CC2(N(C)C)CCCC2)=O)CCSCC1CCNC(=O)CCCCN(C)C CON(CCC(=O)NC1CCCC1CCO)C(=O)c1c[nH][nH]c1=N N1(Cc2nc(C)on2)CCC2(CC1)CC(C)N(C(=O)C(C)OCCC(C)C)C2 C1(NC(CN(C)CCO)=O)CCN(C(c2ncccc2CO)=O)C12CC2 CC(=Cn1ccnn1)C(=O)Nc1cccc(NC(c2ncc(Cl)cc2Cl)=O)c1 N1(C(CCCN(C(C)C)C)=O)CCCCC1CCNC(c1ccc(Cl)s1)=O C(CC(O)CC(=O)NC1CC(C)N(C(=O)C(O)Cc2cnc[nH]2)C1)SC C(CCCCC(=O)N1CCC=C(F)C1)N(C)C(C1(C)CCC2CC2C1)=O N1(C(CC2CC(=C)C2)=O)CCCC(C(=O)NC2CC2C2CC2C)C1C c1(C(=O)NCC2CCN(C(c3cc(C)[nH]n3)=O)C2)ccnc2c(Br)cccc12 C1(CNC(c2c(C)n(C)nc2)=O)CN(C(c2cc(Cl)no2)=O)CC12CC2 c1(C(=O)NCC(=O)NCC(C)NC(c2cn(C3CC3)cn2)=O)cocc1C(N)=O N1(C(c2c(CC)scn2)=O)CC2(CC(NC(c3ccc(C)cc3F)=O)CO2)C1 N1(C(C2C(CCOC)C2)=O)C2CCC1CN(C(c1ccc(C#N)n1C)=O)C2 CC1=CCSC1C(=O)N(C1CN(C(c2nnn(C(C)(C)C)n2)=O)C1)C C1(C(N(CC(C)(C)CN2CCC(C(=O)N(C)C)CC2)C(C)C)=O)CCCC(=O)C1 c1(OC(C(=O)NCC(CC)(C)NC(=O)C(F)F)C)ccccc1C1(C)CC1.C(C=C)O c1(-c2ccc(C(=O)NCCCCNC(c3cnc(C)s3)=O)o2)cccc(O)c1 CC(C)(C)CCC(F)C(=O)NC(CC(=O)Nc1cccc(N=[N+]=[N-])c1)C(C)(C)C C(=O)(C(O)CCC(C)C)NCC(CN(C(c1cnn(CCCC)c1C)=O)C)C C(CC(=O)NC(C)CC(C)(C)O)(C(F)(F)F)NC(CC1(OCC)CCC1)=O C(=O)(C(C)C(C)C)N1CC(CC(N2CCC(CCCC)C2)=O)(OC)C1 c1(OC)cccc2c(C(=O)N(C)CCNC(c3cn(C)c(C)cc3=O)=O)n[nH]c12 N1(Cc2ccc(OC)nc2Cl)CCC2(CC1)CCN2C(=O)Cc1ccccc1 C(CC(C)(C)CNC(c1cc[nH]c(=N)c1)=O)NC(c1c(C(C)C)n[nH]c1)=O N1(C(c2ccc(C#N)cn2)=O)CC2CCC1CC2NC(=O)CC1CCOC1 N1(C(CN2C(=O)CCCC2)=O)CCC12CN(C(=O)CC1COCCOC1)C2 C1(CCC)CN(C(c2ccc(F)cc2Cl)=O)CCN1C(=O)C(C)C(C)C CCCCCCCCC(=O)NCCC(=O)NC(c1ncc(Br)cn1)C c1(C(=O)NC2CCCN(Cc3cc(OC)c(Br)cc3)C2)cn2cc(Cl)ccc2n1 C(CCCCCNCCN(C(=O)COC(C)C)C)NC(C(C)SC(C)C)=O C12(CN(C(=O)COCc3cccnc3)C1)C(=O)NC2.C1(C(C)(C)C)CC1[N+](=O)[O-] C(=O)(CC(C(C)OC)NC(=O)CCSC)NC(c1ncc[nH]1)CC N1(C(CCCN(C)C)=O)CCC2CCCN(C(c3ccc4c(n3)CCC4)=O)C2C1 C1(C(=O)NC(C(C)(C)NC(CSCC=C)=O)C)CCCCN(C)C1=O Cc1cccc(C(N2CCCC2C2(O)CN(C(c3ccn(C)n3)=O)C2)=O)c1Cl c1(OC)c(NC(C2C(O)CCN2C(c2ccc(OC)s2)=O)=O)cccc1Br C1(C(N2CCN(CCNC(=O)Cc3csc(C)n3)CC2)=O)(OC)CS(=O)(=O)C1 c1(CCC(=O)NCCNC(C2(C(C)C)CC2)=O)ccc2cnn(C)c2c1 c1(C(N2CCN(C(C(CC=C)CC)=O)C(CCC)C2)=O)c(C)ccc2nonc12 C1(C(N2C(C#C)CCCCC2)=O)CCc2cnccc2N1 c1(C(=O)OC)ccc(S(=O)(=O)NC(c2cc(C(F)(F)F)nn2C2CC2)=O)cc1Cl C=CC1(C(=O)NCc2ncc(CO)[nH]2)CCN(C(C2CCCO2)=O)C1 c1(Cn2cc(C(C)NC(=O)Cc3cocc3Br)nn2)c(Cl)cccc1Cl c1(C(C)(C)C)cc(C(N2CC(CO)(NC(=O)CC3CC(F)(F)C3)C2)=O)no1 N1(C(C(C)=CC)=O)CCN(C(c2ccn(O)c(=O)c2)=O)CC1c1cccc(Cl)c1 c1(C(=O)NC2CC3CC2CC3(F)F)cn2cccc(Br)c2n1 c1(C(N2CCC(F)(CNC(C(CC=C)C(C)C)=O)C2)=O)ccc([N+](=O)[O-])c(C)n1 CC1=CCC(NC(=O)C(c2cnn(C)c2)NC(=O)CCC2CC2)CC1 C1(C(N2C(CNC(C3CC(=O)N(O)C3)=O)CC(OC)C2)=O)CCCCCCC1 CC1(C)C2CCC1(CC(=O)NCCC1CN(C(C3CC(F)(F)C3)=O)CCO1)CC2 C1(CC)C=CC(N=c2[nH]c(N3CCC(CN(C)C)C3)nc3ccccc23)C1 c1(C(=O)NC2(CO)CN(C(CCC(=O)OCC)=O)C2)cc2nc(Cl)ccc2s1 N1(C(c2ccc(COC)o2)=O)C2CCC1CN(C(=O)Cn1cncn1)C2 C=C(C)c1cccc(NC(C2CC2C2CN(C(c3ncncc3Cl)=O)C2)=O)c1 C1(NC(C)=O)CCC2(CC1)CC(NC(c1cc(C)no1)=O)C2 Cc1nnc(=NCCCCC(C)NC(=O)COc2cccc(F)c2)[nH]c1C N1(C(C2CCC2)=O)CCC12CCN(Cc1ccccc1CO)CC2 C1(C(N2CCC3(C(NC(c4cn(C5CC5)cn4)=O)C3)C2)=O)CCCN2CCCC12 C(CC(C)C(=O)N1CCC(N(C)C(C2(F)CCCC2)=O)C1)=CC Cc1nc(CCC(=O)NC(C)(CNC(c2cc[nH]c(=N)c2)=O)CO)oc1C CCCC(C(=O)NCc1nc(C(=O)NC2C=CCC2)c(C)o1)OCC C1(C(N(CC(=O)N(C)Cc2cn(C)cn2)C)=O)CCCC(C#N)C1 N1(C(C(C)C(F)F)=O)CCC(NC(c2nnn(-c3ccccc3)n2)=O)C(O)C1 C1(CC)CC(=O)OC1(C)C.C12C(C(=O)NC3(C(=O)NC)CC3)CCN1C2=O N1(C(CCCC(C)C)=O)CCCN(C(c2ccn(C)c(=O)c2)=O)CC1C(C)C C(=O)(CCC(CF)CF)N1CCN(C(c2c(C(C)C)cco2)=O)C(C)C1 C1(CNC(CC(C(C)C)C)=O)CN(C(=O)CCc2ccoc2)C2(CCOCC2)C1 N1(C(C(c2cccc(C)c2)O)=O)CC(N(C(=O)CC2(C(F)F)CC2)C)C2(CC2)C1 N1(C(C(C)O)=O)CCOC2(CCN(C(c3ccc(S(N)(=O)=O)cc3F)=O)C2)C1 c1(C(N2CCC3(CCCOC3)C2)=O)ccc(Br)c(S(=O)(=O)N2CCCC2)c1 C1(CNC(C(C(C)C)OCC)=O)CC(C)CN(C(c2sc(F)cc2Cl)=O)C1 c1(NC2CC(NC(c3nc(COC)oc3)=O)C2)snc(C)c1C#N C1(NC(C(C)OC(C)C)=O)CN(C(=O)Cc2cnc[nH]2)CC12CCC2 Cc1ccc2c(C(=O)NCC3(C)CN(C(c4cncn4C)=O)CCO3)coc2c1 c1(OC(C(=O)NCC(CC)NC(c2cnc(O)s2)=O)C)ccc(C)cc1 c1(CC(=O)NC(C2CN(C(c3cc([N+](=O)[O-])n[nH]3)=O)C2)C)c[nH]c2ncccc12 N1(C(C(C)=O)=O)CCn2ncc(CNC(=O)CCC(C)(C)O)c2C1 c1(CN2CC(c3cccc(OC)c3)C(O)CC2)cnn2ccccc12 C1(C(N2CC(C)C(NC(=O)CC3OC(C)(C)OC3=O)C2)=O)CC2(CCCCC2)C1 c1(C(=O)NCC(CN(C(C2CC(OC)(OC)C2)=O)C)C)c[nH]cc(Cl)c1=O C(=O)(C=C1SCC(=O)N1CC(=O)OC(C)C)Oc1cccc(COC)c1 C(CC1CCC1)(C(=O)NC1(C(=O)N(C)CC2CCOC2C)CSC1)OC C(=O)(C1=CCC(C)(C)CC1)N1CCC(CNC(c2c(OC)ccs2)=O)C(C)C1 C1(NC(C(C(=O)OCC)F)=O)CC2CCC1(NC(C1CC=CCC1)=O)C2 C1(NC(C(CCC)(C)O)=O)CC2CC(C1)N(C(C1(C#N)CC3CCC1C3)=O)C2 CN=c1[nH]cc(C(N2CC(=O)CC2C(=O)NCc2cocn2)=O)s1 CC1CN(C(=O)CSc2ccccc2)CCC1NC(=O)CN(C)CCO CCC(C)C=C.C(=O)(C(F)=C(C)C#N)N.C1CSCC1 O=C(CS(=O)(=O)CCO)NCC1(O)CN(C(C2CCCCC2O)=O)C1 C(=O)(C=C1SCC(=O)N1C)NCCC1CN(C(C(=CC2CCCC2)C)=O)CC1C C1(C(=O)NCCOCCN(C)C(c2cccc(=O)n2C)=O)CCCCC(F)(F)C1 c1(CC)ccccc1OCCC(N1CCC(N(C(=O)Cc2ncoc2C)C)C1)=O C1(c2cn(CC)nn2)COCCN1CCS.c1(-c2ccccc2)cccnc1OC C12(N)CC3CC(C1)CC(O)(C3)C2.C(CCNC)N(C(=O)CN(C1CCC1)C)C N1(C(CC2CCC(=O)NC2)=O)CC(NC(=O)Cc2csnn2)C2(CCOCC2)C1 c1(NC(c2n(CCCOCC)nnn2)C(C)CC2CCC2)ccc2c(c1)OCC2 C(=O)(C1=C(C#N)CCC1)OC1C(CC)CCCC1 c1(C(C)NC(C(=O)NC2C(C)C(C(=O)O)C2(C)C)=O)ccc2c(c1)OCO2 N1(CCC)CCN(C(c2ccc(C(=O)N(CC)CCOC)cn2)=O)CC1 C1(NC(C(CNC(=O)CCc2cnccn2)OC)=O)CCC(C)(C)CC1C c1(N2CC3CCCC(=O)N(C)C3CC2)nc(=NC2CCSC2)[nH]c2cc[nH]c12 C1(CNC(C2C(C(C)NC(Cc3c(C)nn(C)c3)=O)C2)=O)OC(=O)CC1(C)C N1(C(Cn2c(C)nnn2)=O)CC(CC(=O)NC2CC2F)CC1(C)C S(=O)(=O)(CC(=O)N(C)CCOCCCNC(=O)C(C1CC1)SC)NC c1(NC(C2CCC(C)N2C(c2nc(Cl)ccc2F)=O)=O)ncc([N+](=O)[O-])cc1O N1(C(CC=C(C)C)=O)CC2CCC2(CC(=O)N(CCCN(C)C)C)C1 Cc1ccncc1CC(N1CCCC1CC(=O)NC1CCSC1C)=O CCC(C)C(CO)NC(C1(C)CCN(C(=O)C(O)CSC)C1)=O C(=O)(C1=CC(O)C(NC(c2cccc(CO)c2)=O)C1)N(C1C(C)CC1)C CC1(C)CN(C(C2CCSC2)=O)CC1C(=O)NCC(C)(C)C1(O)CCC1 C1(NC(C(=O)N(C(c2ccccc2Br)CO)C)=O)CC2COCC(C1)C2 N1(C(CCS(C)=O)=O)CCN(C(c2occc2CN)=O)CC1c1ccccc1Cl N1(C(c2cc(C(C)C)on2)=O)CCC(CO)(NC(c2cc(N)ccn2)=O)C1 c1(CNC(C2(CN)CC3CCC2CC3)=O)ccc2c(c1)NC(=O)C(C)O2 c1(NC(CC2CCN(C(c3n[nH]c(CC)c3Cl)=O)CC2)=O)cccc2c1OCO2 c1(OC)cc(C(=O)NCC2(CS(=O)(=O)NCC(C)=O)COC2)cc(C(C)C)c1O C1(CN(C(c2n[nH]c(C)c2Cl)=O)CC)CCCCN1C(=O)CC1(COC)CC1 N1(C(CCOC)=O)CCC2CN(C(c3cc(O)ccc3F)=O)C2C1 Cc1nc2ccc(C(=O)NCC(C)(O)CNC(C3CCC(=O)N3)=O)cc2n1C N1(C(CSCC(=O)OC)=O)CCCC(N(C)C(c2cc(Cl)c[nH]2)=O)CC1 N1(CCNC(C(=O)N(CC(C(C)C)OC)C)=O)C(=O)CN(C)C1=O c1(C(N2C(CSCC)CC2)C(=O)NC(C)CC)ccc(Br)cc1 c1(CC(N2CCN(C)C(=O)C2C)C(n2c(C)ncc2)C)ccc2c(c1)OCO2 c1(CC(C)C)n[nH]c(=NCC2CC(CNC(c3scnc3C(F)F)=O)CO2)s1 c1(C(=O)NCC2C=CCN2c2ncc(F)cn2)cnc2n1CCOC2 c1(C(N2CC(COC)N(C(=O)C(C)N(C)C)CC2)=O)cnc2ccnn2c1C Cc1sc(=O)n(CC(=O)NCC2CCCCC2NC(C23CCC2C3)=O)c1C N1(C(c2n[nH]c(C)c2C)=O)CCC(C2(O)CN(C(=O)Cc3cccs3)C2)CC1 C(=O)(C(CC#CC)NC(=O)CC1CC2C=CC1C2)N(CCC=C)CCOC c1(OC)cc(F)ccc1C(N1CCC(NC(c2sncc2C)=O)C1)=O C(=O)(C1CCCc2ncccc21)NCC1(NC(CC(=O)NCC)=O)CCOC1 N#Cc1cc(Br)ccc1C(N1CC2CCC(C1)N2Cc1ccn2ccnc2c1)=O C1(CC(=O)NC2CC(CNC(c3nc(OCC)oc3)=O)C2)CCC2(CCC2)O1 CC1=NOC(=O)C1CCC(=O)NCC1CN(C(=O)Cc2ccnc(O)c2)CC1O C1(C(N2CCCC2)=O)C2CCC1(C)C2(C)C.CC1CN2CC1NC(=O)NCC2=O CCC(CC(C)C)C(=O)N1CC(N2CCN(C(c3cc(C)ccn3)=O)CC2)C1 C(c1cccc(C)c1)=CC(=O)NC1(C(=O)NCC2(CCC=C)CC2)CCCC1 c1(C(N2CCC(O)(CNC(Cc3cnn(C)n3)=O)CC2)=O)c[nH]c2cccnc12 CC1=NS(=O)(=O)N(C)C=C1C(=O)NNC(=O)c1ccc(F)cc1Br c1(C(N2CC(C)N(C)C(C)C2)=O)cnn2cc(-c3cccs3)cnc12 C(=O)(C(C)(O)CNC(=O)CC1(C)CCN1C(=O)C(C1CCOCC1)C)OC C=CCN=c1[nH]cc(C(N2CCC(N(C(=O)C(n3cc(Cl)cn3)C)CC)C2)=O)s1 c1(CC)cc(F)ccc1CC(=O)NCCOCCN(C)C(C1(C)CCOC1)=O N1(C(c2c(C(=O)OC)scc2C)=O)CCc2n[nH]cc2C1 c1(NC2(CSC)CCOCC2)ncc(C)c(=NCC(=O)NC2CC2(F)F)[nH]1 C1(C2CCN(C(C3CCC=CO3)=O)CC2)(NC(C2CSCC(=O)N2)=O)CC1 c1(NC(=O)OC(C)(C)C)ccc(Br)cc1C(=O)NC1CC(c2ncc[nH]2)C1 c1(CNC(C(CC)(C)C)=O)cn(CC2CCN(CC)C2)c2ccccc12 C12(NC(CC(CC)(F)F)=O)CCCC1CN(C(=O)C(n1nc(C)cc1C)C)C2 c1(C(=O)NCC(C)CN(C)C(c2n[nH]cc2Cl)=O)cn(C)c2c(Cl)cccc12 C(CCCCCN=C(NCCC1CC12CC2)NCCC1(C(F)(F)F)CCC1)SC C=CC(C)(C)CC(=O)NCCN1CCN(C(c2cc(C3(CC)CC3)on2)=O)CC1 C(=O)(CCCCC(N)=O)NC1CN(C(c2cn(CCCC)nn2)=O)CCC1F CCC(C(=O)N(C1CCN(C(c2cc(C(c3ccco3)=O)c[nH]2)=O)C1)C)N(C)C c1(CC(=O)NC(CN(C(CCN(C(CCC)C)C)=O)C)C)cc(Cl)cs1 C1(CC(N2C(C)CC(NC(c3cccc(C(F)F)c3)=O)C2)=O)CN2CCN1CC2 C1(CNC(CCC2(OC)CCCC2)=O)(CO)CC2CC2C1.C12(CC(O)C1)C(=O)N2 N1(C(c2c(C)nn[nH]2)=O)CC2CCCN(C(=O)C(C)c3ccsc3)C2C1 n1(CC)nc(C(=O)NCC2CCN(C(=O)CC3(C4CC4)CC3)C2)c(Br)n1 NC(=O)CC(O)C(=O)N1CC(CCCCNC(=O)CCOC2CCCOC2)C1 N1(C(C2(OCc3ccccc3)CC2)=O)CC2c3ccccc3CCC12 N1(C(c2nnn(CC)c2C)=O)CCCCC12CN(C(=O)C(C)C(F)F)C2 C1(C)(C(=O)NCCCC(C)NC(c2cc(C)n(C(C)C)n2)=O)CCCCNC1=O Cc1cn2[nH]c(=NC(=O)c3ccc(-n4ccnc4)nc3)cc(C)c2n1 N1(C(C2C(OCC)C2C)=O)CC2(C1)SCCC2NC(c1cc(C)sc1C)=O N1(C(C2CC2c2ccco2)=O)CCC2CCCC12C(N1CC2CC=CC1C2)=O C1(NC(c2c(CC)cns2)=O)C=CCN(C(=O)C=CC2CCOC2)C1 C1(CC#N)CC(N=c2[nH]c3c(c(=NCc4cc5n(n4)CCCC5)[nH]2)COC3)C1 C1(CNC(C(C)SC)=O)CC2(CCC2)CN1C(=O)CN1CCCCS1(=O)=O C1(NC(c2ncc(C)nc2)=O)CCN(C(c2cc(C3(C)CC3)n[nH]2)=O)C1(C)C C1(NC(c2cnc(C(C)=O)s2)=O)CN(C(C2CCCCC2)=O)C2(CCCOC2)C1 C(CC(C)C(=O)NCC(C)(C1CC1)NC(=O)CC12COCC(C1)C2)=CC c1(C(=O)NCCC2N(C(CCS(C)=O)=O)CCC2)c[nH]c2ccc(F)cc12 C1(CC=C)(NC(c2cn3ccnc3s2)=O)CCCN(C(=O)C(C)CCCOC)C1 N1(C(CCSCC)=O)CCN(C(=O)CCc2cnn[nH]2)C(c2cccnc2)C1 CC(C)(C)CC(O)C(=O)NCC1(F)CN(C(c2csc(-c3cnc[nH]3)n2)=O)C1 c1(C(=O)OC)ccc2c(c1)C(Nc1ccc3cccnc3c1Br)CCO2 C(=O)(C(C1=NOCC1)N1CCC(C(c2ccccc2)O)CC1)NCCCSC c1(C(=O)NC(C2CN(C(=O)C(C)C3(O)CCC3)C2)C)ccc2ncccc2c1 c1(C(=O)NCC(CNC(c2c(CC)sc(=N)[nH]2)=O)(C)O)n[nH]c2c1CC(C)CC2 N1(C(c2ccn(C3CC3)n2)=O)CCCCC(CNC(C2(F)CC2)=O)CC1 CCCCCC(O)C(=O)NCC1CCN1C(c1cccc(NC(N)=O)c1)=O N1(C(c2cc(Cl)c(Br)c(Cl)c2)C(=O)NCCC)CCC2(CC1)OCCO2 C1(CNC(C(C(C)(C)C)F)=O)CN(C(c2ncoc2C2CCC2)=O)CC12CCC2 N1(C(C(CCSC)OC(C)(C)C)=O)CCCC(O)(NCC2CC2)C1 N1(C(c2cncc(C)n2)=O)CCN(C(=O)CCSc2ccccc2)C(C#N)C1 C1(NC(CNC(CN(C)C)=O)=O)CC(NC(=O)C(C)(C)N2CCOCC2)C(O)C1 C(=O)(CC1COc2cc(O)ccc21)NCC=CCNC(=O)C=CC1CCOCC1 N1(C(CC2CC(OC)C2)=O)CCOCC(NC(C2(n3nccn3)CC2)=O)C1 C1(C)(CNC(COCCCC)=O)CC(OC)CN1C(c1cn(CC)cn1)=O C(C(C)(C)CNC(C1CC1[N+](=O)[O-])=O)N(C(c1ccc(Br)o1)=O)CC c1(C(N(C(CNC(CCCOC)=O)C)C)=O)cnc2nccn2c1 CC(C)C(CCN(C(=O)C(C)(C)C1CC1)C)NC(C1(C)CC(=O)C1)=O Cc1noc(C)c1S(=O)(=O)NCC(=O)NC1CC1CNC(c1ccc(Cl)c(N)c1)=O C(=O)(C(N=[N+]=[N-])C(C)C)NCCC1CCC(NC(C(c2cccnc2)OC)=O)C1 C1(C)(C(=O)NCCN(CCC)C(c2cc(CC)n(C(C)(C)C)n2)=O)CCSCC1 C12(C(=O)NCC(C)NC(c3c(C)n(CCO)nc3)=O)CCC(CF)(C1)OC2 C1(C(C)NC(=O)Cn2cccc2)CN(Cc2cc(Br)cs2)CCCO1 N1(C(C(COC)C)=O)CCCC(CO)(NC(c2cc(C)nc(O)n2)=O)C1 CC(CC(=O)N(C)C(c1ccc(Br)cc1)c1cnn(C)c1)C(F)(F)F C(c1ccc(Cl)cc1)=CC(=O)NC(CNC(C12CC(OC)C1C2)=O)C(C)(C)C C1(C(=O)NCC2CCC(NC(CCC(=O)N(CC)CC)=O)C2)CC(=O)NC1(C)C c1(C(=O)NC(C2CCCCN2C(=O)CCc2cncn2C)C)cc(O)cc(F)c1 C1(C(=O)NC(C)CNC(C2CCC(C)(C)OC2)=O)CCc2nccn2C1 C=CC1(C(=O)NCC(C(=O)NC)N(C)C)CCOCC1.C12CCN(C1=O)C(=O)N2 N1(CCCNC(c2c(C)coc2)=O)CCN(C(=O)CCc2cncs2)CC1 C1(CC(=O)NC(C(C)C)c2ncc[nH]2)CN(C(=O)CNC=O)C(C)(C)C1 CC1CCCC=C1C(=O)N(CC(C)(C)C(=O)N1CCSCC1)C CC1CCCN(C(=O)C2=CCSC2)C1CNC(=O)Cc1ncc(F)cc1F C1(O)(CC(=O)NCC(CN(C(C(CC)N(CC)CC)=O)C)C)COC(C)(C)C1 CCC(C)C(=O)C(=O)N1CCC12CN(C(C1(C)CCCC1)=O)C2 C1(NC(=O)C2=CCCSC2)CS(=O)(=O)C2CN(C(=O)C=CC3CCOC3)CC12 Cc1nncc(CNC(C2CCCN(C(c3c(F)cncc3F)=O)CC2)=O)c1C C(=O)(NNc1ccc(S(C)(=O)=O)cc1[N+](=O)[O-])NCCNC1C(C)(C)SC1 C1(O)(CNC(CCNC(=O)C=CCl)=O)CCCN(C(c2ccc(CO)s2)=O)C1 c1(C(N(C)CC2OCCN(C(c3[nH]cc(C)c3)=O)C2)=O)ccc(C2CC2)nc1O c1(CC(C(=O)N2C(CNC(c3conc3C3CCC3)=O)CC2)=O)ccc(Cl)cc1 C(=O)(CC1CCOc2ccccc21)NCn1nc(C)n(CC)c1=O c1(C(=O)NCCCN(C(C)C)C(C2C(F)(F)C23CC3)=O)cnoc1-c1cccs1 C#CCCCCCCC(=O)NC(C)(C)C(C)NC(C1CC1c1nccn1C)=O c1(C(=O)NC2C(NC(c3c(C)cc(C)[nH]3)=O)CCC2)nc[nH]c2ncnc1-2 c1(CN(C)C(=O)NCC2CCCN(c3cccc(F)c3)C2)cc(Br)ccc1Cl C1(OCC)CN(C(=O)CS(=O)(=O)CC)CCN1C Cc1ccncc1C=CC(=O)NCC1CN(C(=O)CCOCC2CC2)CCN1C C(=O)(C1=NOC(C)(C)C1)NC1CCC(C)(NC(C2CC23CCCCC3)=O)CC1 CC1C=C(C(=O)NC2CN(C(=O)CC3CCC(C(=O)OC)CC3)C2)CC1 S(=O)(=O)(c1c(C)noc1C)c1nnc(-c2c(C#C)nc(Cl)cc2)o1 N1(C(C(=O)N(C)C(C2CCCCS2)c2ccccc2)=O)CC2CCC2(C)C1 C(=O)(C1=CC2CCCCCCC12)NCC1(CCNC(c2c(C)csc2)=O)CC1 Oc1cccc(CNCC2CC23CCOC3)c1 C(=O)(C1CCCc2c(Br)cccc21)OCc1c(CC)cccc1 c1(C(=O)NC2CCN(C(C3N(CC)CCCC3)=O)CC2)cccc(Cl)c1O c1(C(=O)NC(C(C)NC(C(C(=C)C)(C)C)=O)C)cc2c(Br)cccc2cn1 c1(C(N)=O)ccnc2[nH]cnc12.C12(OC)CCCN(C1)CC(=O)NC2 Cc1nc(C(C)C)ncc1C(=O)NCCNC(C1CCCCC(=O)C1)=O c1(COC(C2N(C(C)=O)CCCC2)=O)c(C)cc(Cl)cc1C C=Cc1cncc(C(=O)NC2CCOCC2C(N2CCC3(CCO3)C2)=O)c1 c1(C(=O)NCCn2cc(-c3cc(OC)ncc3)nn2)cc2cc(Cl)sc2[nH]1 C(C(C)(C)CO)(c1cccs1)NC(CCn1cc(C(C2CC2)OC)nn1)=O N1(C(C(CCC)C)=O)CCc2sc(-c3cccc(NC(C)=O)c3)nc2C1 c1(C(=O)NC2C(CNC(CC3(COCC)CC3)=O)CCC2)ccn2cccc2c1 Cc1ccc(CNC2CC2N2CCOCC2)cc1C(F)(F)F N1(C(Cn2ccc(C)n2)=O)CCOCC1CN(C)C(c1csc(C)c1)=O C1(OC)CN(C(=O)Cn2cc(C(F)(F)F)cn2)CC1NC(C1CC(C)(F)C1)=O c1(C(N2CCSCC2)=O)cc(=NC2CCn3c(O)nnc3C2)[nH]c(Cl)n1 N1(C(c2c(CCC)n[nH]c2)=O)CCN(C(C2CCCC(C)CC2)=O)CC(C)C1 c1(N2CC(C(=O)OCC)N3C(C2)CCC3)nc(O)n(C)c(=O)c1[N+](=O)[O-] c1(CN2CC3N(C(c4ccc(C)c(Br)c4)=O)C3C2)c(O)cc(Br)cc1F Cc1cccc2[nH]c(C(N3CCCN(C(=O)Cc4ccon4)CC3)=O)cc12 n1(CC)nc(C(F)(F)F)cc1C(=O)N(CCCNC(C1(O)CCC1)=O)C CCCCC(C)(F)C(=O)N1CCCCC1C(=O)N(CCC(=O)OC)C C1(C)(CNC(c2nnnn2CCCSCC)(COCC)C)CCC(=O)N1 C(CC(C)(C)C(=O)NCC(C1CCC1)NC(=O)CC1CCCC(C)(C)C1)SC N1(C(c2c(C)n[nH]c2)=O)CCC(C(C)CNC(=O)COC2CCCCCC2)CC1 c1(C(C(=O)NCC(C(C)C)NC(c2ccoc2)=O)OC)c(F)cccc1F C1(F)(CNC(C2N(C)CCC2)=O)CCC(CNC(C23CSCC2C3)=O)C1 N1(C(C2CC(NC(C3(COC(C)C)CC3)=O)C2)=O)CCOCC(C)(C)C1 Nc1ccnc(C(=O)NC2CC2NC(c2cc(Cl)c(Cl)s2)=O)c1Cl c1(CNC(c2n(CC=C)nnn2)C(C)CCCC)ccc(SCC(=O)OC)cc1 c1(OC)cccc(C(=O)NCC2CCCC2C(=O)NOCN2CCCOC2=O)n1 c1(C(=O)NC2C(CC)CN(C(=O)CCCCF)CC2)ccc2nccn2c1 Cc1ccccc1C(=O)NC12CC(CNC(c3nocc3C(C)C)=O)(C1)C2 Cc1ccc(C)c(CCS(=O)(=O)CC2CCCCO2)c1.C1(=O)CO1 CC1(C)CC2(CC(C(=O)NC3CC(C(=O)NCCOC(C)(C)CO)=NO3)C2)C1 C1(C(=O)NC(C)(CNC(c2n[nH]cc2Br)=O)Cn2cccn2)CCC2CC2CC1 N1(c2nccc(C)n2)CC2(COC(CNC(c3cnc(N(C)C)cn3)=O)C2)C1 c1(C(C)=O)cccc(C(=O)NCC2CCC(NC(c3nscc3C)=O)C2)n1 c1(C(=O)NC2CC(CNC(CC3(C=C)CC3)=O)C2(C)C)c[nH]c2cc(F)ccc12 c1(C(=O)NC(C(C)NC(c2cccc(CN(C)C)n2)=O)CO)cccc(Cl)c1F Cc1[nH]nc(C(=O)NC(C)C(=O)NC2CCCC2(C)CO)c1O c1(CC(=O)OCC)cc(CNC=O)on1.C1(C2C(C(=O)NCC)C2)CC(C)(OC)C1 c1(CC(=O)N(C)CCNC(C2CC2Br)=O)c[nH]c2cc(Cl)ccc12 c1(C(=O)NC2C(C)CCN(C(C3CCC4CC34)=O)C2C)ccc2ccccc2n1 c1(CC)ncccc1NC(C1C=CCCN1C(=O)C=CC(C)C)=O C1(CSC2CCN(CN(c3ccccc3)C)C2=O)CC2(CC2)C(=O)O1 C=C(F)C1(CC(N2CCC=CC2C(=O)NCC2(C)COCCO2)=O)CCC1 c1(CC(C(=O)O)NC(=O)C=Cc2ccsc2)ccc2[nH]ccc2c1 c1(C(=O)NC(CCNC(C#CC(C)C)=O)C)ccc2c(n1)NCC(=O)N2 N1(C(CC2N(CC(C)C)CCC2)=O)CCN(CC(C)NC(=O)C(C)(C)C)CC1 Cc1ccc(C)n1C1CC(C(=O)NC2CC(CC(N3CC(O)CC3C)=O)C2)C1 CC1=C(C(=O)NC2(CNC(c3c[nH]nc3C)=O)CCOC2)Cn2nnnc2N1C N1(C(C2CC(CC)OCC2)=O)CCC(C2(NC(C3(F)CCOC3)=O)CC2)CC1 C1(NC(c2c(C)noc2)=O)CC(NC(=O)C(=O)NCCC(N)=O)CC1O c1(C(=O)NC2(COC)CN(C(c3ccc(CC)[nH]3)=O)C2)c(C)ccc(C)c1O c1(C(=O)OC)cnc(N(CC(C)CNC(c2ccc(F)cn2)=O)C)cn1 c1(NC(=O)NC(c2cccnc2)C)cc(F)c(NC(=O)C2CC2)c(Br)c1 C1(C(CNC(C(C)NC(CC)=O)=O)C)CCN(C(c2nc(Cl)sc2C)=O)CC1 C1(CNC(C2ON=C(C(C)C)C2)=O)(NC(c2cncs2)=O)Cc2ccccc2C1 c1(NC(c2c(C)ocn2)=O)nc(Cl)ccc1C(=O)NC(C)CCO C(=O)(C1=CC2(CCOC2)C1)NC1(CC=C)CCN(C(c2ncc(F)cc2C)=O)C1 Cn1cnc(C(=O)Nc2[nH]nc(-c3ccccc3)c2Br)cc1=O C1(NC(C2N(C)C(=O)CCC2)=O)CN(C(=O)C=CCO)CC2(CCC2)C1 C1(NC(c2c(CC)nc[nH]2)=O)CCN(C(C2CCSC2)=O)C1(C)C c1(CC)cccc(C(=O)NC2CC(O)CN(C(=O)C3=CCOC3)C2)c1F O=C1C2CCC3(CCC3)CN2C(=O)N1C1CCCN(c2ccncc2)C1 C1(CNC(CCCC)c2nnnn2-c2cccc(OCC)c2)CC2CCC(C1)C2 C1(OC2C(C)CC2)CCN(CC(=O)NCc2cn(-c3cc[nH]c(=N)c3)nn2)CC1 N1(CCOC)CCCN(CCC2CCCCN2C)CC1 C#CC1(F)CN(C(C2CCOC2CNC(=O)CC2CC2)=O)C1 c1(OC)ccc(OC)c([N+](=O)[O-])c1C(=O)NCCN(C(=O)CC1CCC2CC12)C C(=O)(C(CNC(C1(C(=O)OCC)C=CCC1)=O)CC(C)C)NC(CCC)CC CC(CC(=O)N(c1ccnc(N2CCCCC2C)c1)C1CCC1)C(F)(F)F.C1CO1 N1(Cc2c(C(C)C)noc2)CCC2(CC1)CN(C(=O)C(F)(F)C(F)(F)F)CCO2 c1(NC(=O)Cn2nccn2)cccc(CO)c1.N12CCCC(C1)NC(=O)C2.C(=O)(C1CC1)N S(=O)(=O)(c1cc(Br)c(Br)s1)N1CC2N(C(c3ccc(F)cc3Br)=O)C2C1 N1(C(c2cc(CC)n(C)n2)=O)CCCC(CC)(NC(=O)C=Cc2ccccc2)C1 CC1CCN(C(C2CCC(C)CC2)=O)CC1CC(N1CC(CN=[N+]=[N-])C1)=O Cc1nn(C)cc1CCC(=O)NCCCC1CCCN1C(C1(C)CC2CC2C1)=O Cc1nnnn1CC(=O)NCCC(C)N(C(=O)C(N1CCCC1)C1CC1)C c1(C(N(C)CCNC(=O)C(F)C2CCOC2)=O)cncc(C(F)(F)F)n1 c1(CC)cc(C(=O)NCC2CCCCCN2C(C2CC=CC(O)C2)=O)cc(F)c1 CCC(Cc1ccccc1)C(=O)NCCOC1CN(C(c2cc(OC)no2)=O)C1 c1(C(=O)NC2CCCC(C(=O)NCC3CC(CC)C3)CC2)ccc2c(c1)CCC2 CC1CN(C(=O)CCCN(C)C(N)=O)CCN1C(C1CNC(=O)O1)=O C1(NC(C(CC)N(C)C)=O)(NC(=O)CCOC2CCCC2)CC2CCC1C2 c1(OC)ccc(SC)c2cc(C)oc12.C1(C(CN(CC(=O)N)C)=O)CCCCC1 c1(C(=O)NCCC2N(C(CCC)=O)CCC2)ccnc2[nH]ncc12 N1(c2nnc(C(C)(C)C)o2)CC(C)(C)CCC1CNC(=O)C(C1(O)CCCC1)F C(CC(F)F)(C(=O)N1CCN(CCO)C(C)C1)NC(c1c(OC)ccs1)=O N1(C(c2[nH]cc(CC)c2)=O)CCOCC(NC(C2CCCCN2C(C)=O)=O)C1 C=CC(CCC)CC(=O)N1CCN(C(c2ccc(C)c(C(C)=O)c2)=O)CC(O)C1 C(C)(C)(C=CC(=O)NC1(C)CC1)NC(COCCC)=O CC1CCN(C(=O)CCc2cnc[nH]2)CC1CNC(c1ccc[nH]1)=O Cc1cnc(C(=O)NCC2(C)CCN(C(=O)C(C)(C)c3ccccc3)C2)nc1 Cc1nn(-c2cn(CC3N(C(C4(Br)CC4(F)F)=O)CC3(C)C)nn2)c(C)c1C C1(CC)CC(C(=O)NC2C3CC2N(C(C2CCCOC2)=O)C3)CCO1 C(C(COC)CC(=O)N1CC(CC(F)C(=O)NC)C1)OC C(=O)(CCS(N)(=O)=O)NC(C1CN(C(=O)CC2(O)CCOC2)CCO1)C Cc1cc(C(N2CC(F)(F)CC2C(N2CC(C)C2)=O)=O)c(Br)cc1F C12(CNC(c3cn(CC=C)nc3)=O)CC1CN(C(=O)C(=Cc1cccnc1)F)C2 C1(C(=O)NC23CC(C(=O)NC(C4(O)CCCCC4)CC)(C2)C3)CC2(CCCO2)C1 c1(CC(=O)N(C)CCNC(=O)C(C)(Cl)Cl)c(F)cc(F)cc1F c1(SC)cc(C)nc(N2CCC(O)CC2C(=O)Nc2ncccc2C)n1 n1(CC)cnnc1C1CCN(CC(=O)NC(c2cncs2)CSC)C1 N1(C(C2(C=C)CCN(C(=O)C(C)OC(C)=O)C2)=O)CC2CC(C1)C2(C)C c1(C(N2CC(C3(NC(c4c(C)cns4)=O)CC3)C2)=O)cccc2ncc(C)n12 C1(CC(N2CCCC(NC(c3ccc(CO)nc3)=O)C2)=O)CCCC(F)(F)C1 C(=O)(C=C1SCC(=O)N1C)N1CC(NC(C(C)P(C)(C)=O)=O)C(F)C1 N1(C(CC=C(C)C)=O)CCOCC1CC(=O)NCc1cnco1 n1(CC)c(CNC(c2c(Br)cnn2C2CCC2)=O)nc2ccccc12 C(=O)(C1=C(C)CCC1)N1C(C(N2C(C(CC)O)CCC2)=O)CCC1 Cc1[nH]nc(C(=O)NC2CCC(C)(CNC(=O)CNS(=O)(=O)N(C)C)C2)c1O CC1CC(NC(C2CC2c2cnccn2)=O)CCN1C(=O)CCNC(=O)C1CC1 CCCCCC(CC)C(=O)N.c1(CC(=O)N(CCN)CC)csc(COC)n1 CCCCCC(C)CC(=O)NC1CCCCC1CC(=O)NCC(O)CCOC C1(CCNC(c2nocc2C2CC2)=O)CN(C(C2(CO)CC2(F)F)=O)CCO1 C(=O)(N1CCCO1)NC(C1CC(NC)(OC)C1)=O.c12csc(c1)C2 c1(C(=O)NCCC(C)NC(=O)CCNC(c2ccccc2)=O)nc(Cl)sc1Cl CC(C)(C)C#CC(=O)NC12CCC(C1)N(C(=O)CC1(N(C)C)CCCC1)C2 N1(C(c2c(OC)noc2C)=O)CC(C)(C)CC1CNC(=O)C(C)CC(C)C CC(C)(CC(=O)N1CC(NC(=O)CC2CCCCCO2)CC(F)C1)C(F)(F)F N1(C(CC(C)(F)F)=O)CCCN(C(C2CCC(=O)O2)=O)CC1 C1(C(N2CCC(CCNC(CN(C)C)=O)C2)=O)CC(=O)N(C(=O)OC(C)(C)C)C1 c1(C(=O)NCCC(C)(C)NC(=O)CC=Cc2cccc(F)c2)cc(N)c(F)cn1 C1(C(=O)NCCN(CCOC)C(C2CCC(=O)O2)=O)CCC(=O)N(C(C)C)C1 CCC(CCCC(=O)N(C)Cc1ccn(C)c1)NC(c1oc(C)cc1C)=O N1(C(c2cc(C3CCCNC3)[nH]n2)=O)CCOc2cc(F)c(F)cc21 n1(CCC)ccc(C(=O)N(C2CCC(NC(c3ncsc3C)=O)C2)C)n1 C1(CC)CC(C)CN(C(C2CC(C)(NC(=O)C(O)CCCSC)C2)=O)C1 C(=O)(C1=CCCCC1C)N1CC(CNC(c2c(C)noc2)=O)OCCC1 Cc1cc2cc(C(=O)N=c3cc(CO)[nH][nH]3)ccc2[nH]1.N1(C=O)C2CCC1COC2 C(=O)(C(F)(CNC(C1CCC(CO)CC1)=O)C(C)C)N1CC(C=C)OCC1 C1(N(C)C(C2C3CCCC23)=O)CCCC(NC(=O)CC(F)(F)Cl)C1 C1(CNC(CCCC)=O)CC(C(=O)O)CN(C(=O)OC(C)(C)C)C1 C1(C(=O)NC2CC(c3ccccc3)(NC(COCC=C)=O)C2)CCC(C#N)CC1 c1(CCC(=O)N(C2CCN(C(CCCC3(C)CC3)=O)CC2)C2CC2)ccc(N)c(F)c1 C1(C(=O)NCCN(CC(C)O)C(=O)C=C2CCOCC2)CC12CCOC(C)C2 c1(C(=O)OC)cc(F)c(NCCC2CCC2=O)c(I)c1 C(CCNC(C1CCC2(CC2)C1)=O)(C(=O)N1CC(OCCO)C1)OC C(C(O)C(C)(C)C)N(C(c1c(CNC(C(C)NC=O)=O)occ1)=O)C Cc1ccsc1C=CC(=O)N(C(C)CN(C)C(C1(NC(C)C)CC1)=O)C C1(NC(C2C(C)(C)OCC2)=O)CC2CCC1N2C(c1ccn(CCF)n1)=O c1(C(=O)NCC(C)(CO)NC(C(COC)N(C)C)=O)cncn(C)c1=O c1(C(N(CCCN(C)C(C2(c3ccn(C)n3)CC2)=O)C)=O)ccc(F)nc1 C(C)(N=c1[nH]c(Cl)nc(CC)c1Cl)C1CN(C(C(CC)Oc2ccccc2)=O)C1 C1(NC(CC2(C(=C)F)CCC2)=O)CC(NC(C2CCS(=O)(=O)CC2)=O)C12CCC2 C(=O)(CC(O)CNC(=O)Cn1nc(C)cc1C)NC(CCCC)C C1(C)(C(=O)NC(CCCC)CC)CN(C(c2ncn(C)c2C)=O)C(C)(C)C1 Cc1ccc2c(C(N3CCCC(CCNC(=O)C=C4CC4)C3)=O)cnn2c1C c1(NC(C2CCCC(NC(C(CC)C)=O)C2)=O)cc(Cl)ccc1I c1(OCC(N2CCC(CN(C(C3C(=C)C3)=O)C)C2)=O)ccccc1Cl CC1CN(C)CC(C(N2CCN(CCN(C)C(c3cn[nH]c3)=O)CC2)=O)O1 C12(C(=O)NC3CN(C(CCCc4[nH]c(=N)sc4)=O)CC3O)CCCN(CCC1)C2 c1(SC)nc2nc(C)c(CC(=O)NC3CCC3(C(C)C)OC)c(C)n2n1 C12(NC(N3C(C)CC4(CC4)C3)=O)C3C4C1C1C2C3C41CO.c1(N)ccccc1 C1(CN(C(CCNC(=O)NC)=O)C)CN(C(c2ccc(C(N)=O)[nH]2)=O)CCO1 C(C(=O)C1CCCC(CCC)C(C)(N)C(=O)N1)(C(C)C)SC c1(C(=O)OC)cc(CC(C)C)c(C)s1.C12CC(C(O)C1)NC(=O)C1C(C1)C(=O)N2 O=C(C1=CCN(C(=O)CC2CSCCO2)CC1)NC1CCC2(CC2)C1 CS(=O)(=O)c1ccccc1CC(=O)NCCNC(c1cccc2cnsc12)=O CN1C(=O)NCC1C(=O)NC(CNC(c1cnc(CC2CC2)s1)=O)C1CCC1 C1(C(=O)NCC2CN(C(c3c(CC)cccc3F)=O)C2)CC(=O)N(C)C(=O)N1 C1(=O)CC(C)(O)N1.C(COCCN(C)CCC1CC1)OC CCCC(C)(O)C(=O)N1CCC(NC(c2cc(Cl)sc2Cl)=O)C(O)C1 c1(-c2c(C(=O)NCC)csc2)ccc2oc(CC(C)C=O)cc(=O)c2c1 c1(-c2nc(CS(C)(=O)=O)n(CCc3cccs3)n2)cc2ccccc2cn1 c1(C(N(C2CN(C(C(C=C)O)=O)C2)C)=O)sc(OC)nc1Cl C1(CNC(C2(CC#C)CC=CCC2)=O)C(O)C(O)CN1C(c1cc(O)nn1C)=O Cc1nc(CO)oc1C(=O)NCc1cccc(CNC(=O)CCC2CC2(F)F)c1 C(=O)(CCCC(F)(F)F)NC(C)C=CC(=O)NC1(C(O)CO)CC1 Cc1cc(C(=O)NC(C)C(C)NC(c2ncoc2C(C)C)=O)co1 N1(C(COCC#C)=O)CC(NC(c2ccn(C(C)C)n2)=O)C2CCCCC12 CCCCCCCC(=O)NCCC1C(C)CCCN1C(c1ccn(CCF)n1)=O C1(C)(NC(C(CCCNC(c2c(COC)ccs2)=O)O)=O)CN2CCC1CC2 c1(C(N2CCC(N(C(c3cc4occc4s3)=O)CC)C2)=O)ccc2ccoc2c1 N1(C(=O)CCC2CCOC2)CCC(C2CN(C(=O)CC3CC=CCC3)C2)CC1 N1(C(C2CC(C)OC2)=O)CCN(c2nc(CN3CCCCCC3)ns2)CC1 c1(C(=O)NCC2(C)N(C(CCC(=O)OC(C)C)=O)CCC2)cn2c(n1)COCC2 Cc1noc(CC(=O)NC2C=CC(CNC(C3(CC(F)F)CCC3)=O)C2)n1 c1(CNC(C2(N(C)C)CCC2)=O)ncccc1CNC(=O)CSc1ccccn1 Cc1nc(NCC2CCCCS2)cc(N2CCOC(c3ccc(F)cc3)C2)n1 c1(CN2CC(C)(CC(=O)NCC#C)C2)ccc([N+](=O)[O-])cc1C C1(NC(C2N(C)CCC2)=O)CC2(CCC(NC(c3cnc(C4CC4)s3)=O)CC2)C1 C1(NC(C(C(C)(F)F)F)=O)CC2CC(NC(=O)C=Cc3ccoc3)CC2C1 C1(C(=O)Nc2cccc(-c3c(C)cccc3)c2)CS(=O)(=O)CC1N C(=O)(C1CCCc2n[nH]cc21)N1CCC(n2cc(SCCC(=O)O)nn2)C(O)C1 c1(NC(=O)NCC)cc(Br)c(-c2nn[nH]n2)cc1F.c12nn(C)cc1NC2=O C1(C(=O)OC)CC(CC)CN(C(=O)Nc2cccc(Br)n2)C1.c12cccc(c1)S2 c1(-c2occ(C(=O)NC(C)CNC(C3(C)CCCCC3)=O)n2)c(F)cccc1F c1(CC)cnccc1NC(=O)NC1CCN(c2cccc(COC)n2)C1 C1(NC(COCCC)=O)CN(C(c2cc(S(C)(=O)=O)oc2C)=O)CC2(CCC2)C1 C(=O)(C1=C(Cl)CCCC1)NCC(C)(C(C)C)NC(C(CCC)C)=O N(C1CCCc2ncccc21)C(C(N1CCC(C(F)(F)F)(C(=O)OC)C1)=O)=O C(c1ccccn1)=CC(=O)NC(C1CCN(C(C2C3CC4C(C3)C24)=O)C1)C N1(C(C2N(C(C)=O)CCC2)=O)CCN(C(C2COC(C)(C)C2)=O)CC(O)C1 C1(CC(C)NC(c2cnc(S)[nH]2)=O)CCN(C(C2CC(C)(O)C2)=O)CC1 CCCCC(CC)C(=O)N(CCC(=O)NCC1COCCN1C)CC1CC1 c1(C(=O)NC(C2CCCN2C(c2ccncc2F)=O)(C)C)cc2n(c1)CCSC2 C(=O)(C(C)(C)CCCF)N1C(C(=O)Nc2cnc(OCC)nc2)CC(OCC)C1 c1(C(=O)NCC(C)N(C(c2ccc(CC)[nH]2)=O)CC)cc2c(C)n[nH]c2nc1O CCCCC(CC)CC(=O)N(C)CC1COCCN1C(=O)CCSC C1(NC(C(=O)NC2CCC(CCC(=O)NCC(F)(F)F)OC2)=O)CC2(CCC2=O)C1 c1(OC2(C(=O)NC(C)C(C)NC(=O)CCn3cccc3)CC2)ccccc1 c1(CC)cc(C(=O)N(CC(C)C#N)CC(C)C)c(C)o1 C1(NC(C(CC)N(C)C)=O)CCCC2CN(C(=O)CCCCC3CC3)CC12 C(=O)(CCC(C)OC1CCOC1)NCc1ncc(CC)o1.C1(=O)CN1 C(=O)(C(C(C)C)SC)NC1C(CC(=O)N(CCOC)CC2CC2)CCC1 CC1(C)CC(O)C(O)CN1C(N1CC2(CCC2)C1c1ccccc1)=O C12(NC(C34CC(C)(OCC3)C4)=O)CCCC1N(C(c1ccncc1Cl)=O)CCC2 CCC(CC(=O)N(CCCC(=O)N1CCC(c2nc[nH]n2)C1)C)C(F)F N1(C(C2(CC)CC2)=O)CC[Si](C)(C)C1.N12CC(C)(C1)OC(OCC)C2=O c1(C(=O)NCC(CN(C(=O)Cc2nn(C)cc2Cl)C)(C)C)ncccc1O CC1(C)CCCC12NC(=O)N(CO)C2=O.c1(C(=O)OCCCC=O)ccc(Cl)cc1 c1(N(CC(C)C)C)nc2ccc(S(=O)(=O)NCC3CC(O)CCO3)cc2s1 c1(OC)cc(CC(N2CCC3(NC(=O)C(C4CCC4)OC)CC23)=O)c(F)cc1O c1(C(N2C(CNC(Cn3c(C)nnn3)=O)CC(O)C2)=O)cccc2c1nnn2C N1(C(C2CSCN2C(=O)CCOCC2CC2)=O)CCOC(CC2CC2)C1 C(C(C)C(C)C(=O)NC1CCCCC1CNC(C1CC2(CSC2)C1)=O)OC C(C(=O)N(C)Cc1cc(C)on1)(C(C)CC)N(C(c1c(NC)scn1)=O)C C1(NC(Cc2c(C)cnn2C)=O)CCCCC12CCN(C(c1ccc[nH]1)=O)C2 C(=O)(CC(CC(C)C)NC(=O)CC1CCC(=O)N1)N(CC(=O)OCC)C C1(NC(C2(C(C)C)COC2)=O)CCCC1CNC(c1cnc(CN(C)C)s1)=O c1(C(N2CCC(O)(CN(C(C=CCC)=O)C)C2)=O)ccc(Cl)c(C)c1OC C1(NC(c2c(CCC)occ2)=O)CCN(C(=O)C=C2CCC(C)CC2)C(C)C1 Cc1ncncc1C(N1CCOC(Cn2cc(COC3CCC3)nn2)C1)=O N1(C(c2ccn(COC)n2)=O)CCC2CN(C(=O)Cc3ncoc3C)CC2C1 C(=O)(CCC(F)(F)C(F)(F)F)N1CC(CNC(C2N(C)CCC2)=O)OC(C)(C)C1 Cc1ccc(C(=O)NCCOCCNC(=O)C(N2CCC(C)C2)=O)nn1 Cc1cc(C(=O)NCC(O)CNC(c2cn(C)cn2)=O)cn(C)c1=O CCC(CC(=O)NCCC1CCCN(c2cc(O)ncn2)C1)C1CC1 N1(C(Cc2c(C)nc(C)s2)=O)CCC(NC(=O)CNC(=O)CN(C)C)CC(O)C1 CC(C)C(C(=O)NCC1(F)CN(C(=O)CC2CCC(C)(C)O2)C1)c1ccccc1 c1(C(=O)NC(CCC)CNC(c2n[nH]cc2C(C)C)=O)ccc2oc(O)nc2c1 C#CC1(CNC(C2C(CC)CCN2C(=O)C(C)S(N)(=O)=O)=O)CCOCC1 CC1(C(=O)NCC(O)CNC(=O)CC2(N(C)C)COC2)CCC2(CC1)CC2 c1(C(N2CC(C)OC(C(F)(F)F)C2)=O)ccc(Br)c(S(N)(=O)=O)c1 CC1CCN(C(=O)CCc2ccoc2)C1CNC(=O)C(c1cccc(F)c1)F C12(NC(=O)COC3CC3)CCCC1N(C(=O)C(O)c1cnc[nH]1)CC2 c1(C(N2CCN(C(CCOCCC)=O)C(CC)C2)=O)cccc2[nH]c(=N)oc12 N1(C(C(CNC(CN(CCC#C)C)=O)F)=O)CCN(C(C)=O)CC1CCC#C C(C)(CCC(=O)NCC(C)(C)CN(C)C(c1cccc(F)c1)=O)OC N1(C(C2(CF)CCN(C(=O)CC34CCC(CC3)CC4)C2)=O)CCN2C(=O)OCC2C1 N1(C(C2N(C)C(=O)CC2)=O)CC2OCC(NC(c3cnccn3)=O)C2C1 O=C1CSCC(C(=O)NC2(CC(=O)NCC(F)(F)Cl)CCCCC2)N1 CC1CC(C(N2CCCC2CC(C)(C)C)=O)CS1 CC(CN(C)C)CCC(=O)NCC1CCN(C(c2c[nH]nc2[N+](=O)[O-])=O)C12CC2 c1(C(=O)OCC)cccnc1N1CCC(C(C)NC(C2CCOC2)=O)C1 C(=O)(C1=CC2CCCCCC12)NCC1C2CN(C(C(CCSC)O)=O)CC21 C(C)(CCC(=O)NC1(C(=O)NCCCCSC)CC(O)C1)OC C(=O)(CC(C)(C)C)N1C(CCc2cn(CC(CC)O)nn2)CCC1 C=C(C)CC(=O)NC1CCCC1NC(c1ccnn1CC(F)F)=O C#CC1N(C(C2CN(C(=O)COCC(=O)OC)CCO2)=O)CC1(C)C N1(C(C(c2cncn2C)NC(C)=O)=O)CC2OCC(NC(=O)C#CC3CC3)C2C1 C=CC(C)(CCOC)C(=O)N1CC2COCC2(C(=O)Nc2cc(F)ccc2O)C1 C1(C(=O)Nc2c(O)ccc(C)c2)CCN(C(=O)CC2CC=CCC2)O1 C=CC(C)CC(=O)NCC1(O)CCN(C(c2cc(Cl)c(Cl)[nH]2)=O)C1 C(C(CO)CC(C)(C)C)SC1CC1.C12(CCCN(C(=O)OCC)C1)n1nnnc12 c1(C(=O)NCC(CN(C(c2cn(CC=C)nc2)=O)C)O)ccc(OC)nn1 N1(C(C(CC)CC(F)(F)F)=O)CCCC2(CCN(C(C3(O)CCOC3)=O)CC2)C1 C(=O)(C(O)C(F)F)NC1(COC)CN(C(=O)Cc2ccc(CC(C)C)cc2)C1 C1(C(=O)NCC2N(C(C(CC)C#N)=O)CC(O)C2)CC12CCOCC2 c1(OC)ccnc(C(N2CCCC(N(C)CCC3(O)CCOC3)C2)=O)c1 c1(C(N2CC(OCC)(CNC(=O)C(C)CCO)C2)=O)ccc(F)c(F)c1 N1(C(=O)CC2CC2c2ccccc2)CC2CCN(C(C34CC(CO3)C4)=O)CC12 C(=O)(C(F)(F)c1nccn1C)N(CCNC(C1CC(F)C1)=O)CC CC1(C(=O)NCC2CC(NC(=O)CCSC3CCCC3)CC2O)CC=CCO1 C1(NC(c2ccnc(Cl)n2)=O)CC2CCC(C1)N2C(=O)Cc1ccccc1F c1(C(=O)NCC2CC3(CN(C(C4(C=C)CCC4)=O)C3)C2)cccn2cc(C)nc12 C1(C(=O)NCC(N2CCCC2)C)CC(=O)CN1C(=O)C=Cc1cnccn1 Cc1cc(C(N2CCCC2C2CCN(C(=O)C(C)(C)c3cc[nH]n3)C2)=O)c(C)o1 C12(C(N(CC(CNC(Cc3nc(CC)sc3)=O)O)C)=O)COCC1C2(F)F C1(CC(N2C3(CNC(C=C(CCC)C)=O)CCC2CC3)=O)CC2(CCCC2)CO1 CC1CCC(C(=O)N(CCCNC(=O)CCCc2nc(C(C)C)no2)CCO)S1 N1(C(c2nncc(CCC)c2)=O)CC2CN(C(c3ccnc(C)c3Cl)=O)CC2C1 N1(C(CCC)=O)CC2(C1)C(NC(=O)CC1CCC3CC13)CCS2(=O)=O c1(NCC2(NC(=O)OC(C)(C)C)CC2(F)F)cc2ccncc2o1 C1(NC(c2c(CC)[nH]cc2)=O)CN(C(c2cc(Cl)cnc2O)=O)C2CCCC12 N1(C(CC)=O)CCC(NC(C2CCCCN2CC(F)F)=O)C(F)C1 c1(C(C(=O)N(CC(CN(C(CN(C2CC2)CC)=O)C)O)C)C)cc(C)cc(F)c1 N1(C(CCC(COC)C)=O)CC2CCC(C1)N2C(=O)C(O)C(F)(F)F C(=O)(C(C)C(C)(F)F)NCCOC1CCN(C(c2ccc(NC)cn2)=O)C1 N1(C(c2c(C)n[nH]c2)=O)CCCN(C(=O)CCC(C)C)CC1CO Cn1cnc(S(N)(=O)=O)c1C(=O)NC12CCCC1N(C(=O)CCCCO)CC2 C(=O)(C(CC(C)C(C)(C)C)N1CCN2C(=O)NCC2C1)NCCCC c1(SC)ccc2c(c1)NC(=O)C1N(C3C(C1)C3)C(=O)CO2.C(C(F)(F)F)OC N1(C(CCOC)=O)CCCC(N2CCN(C(c3cscn3)=O)CC2)C1 Cc1cc(Cc2cn(CC3CCN(C(=O)C(C)OCC4CCC4)C3)nn2)n(C)n1 N1(C(C(C)C(C)(C)C)=O)CCCC2(CNC(c3cc(N)cc(O)c3)=O)CCCC12 c1(CC(=O)OC(c2cc(Br)sn2)C)ccc(F)c(F)c1F c1(C(N(CC(C)NC(=O)C(C)(C)c2cscn2)C)=O)nn(C(F)F)cc1Cl C1(CNC(=O)CC2CC(F)(F)C2)C2CC2CN1C(=O)Cc1ccco1 c1(-c2ccc(N(C=O)CC3CCC(C)(C)C3)cc2)ccc(S(N)(=O)=O)s1 N1(C(c2c(OC)nsc2)=O)CCC2(COC(CNC(=O)CC3(C)CC3(F)Cl)C2)C1 c1(C(C)=O)cc(-c2nc(-c3ccc(I)cc3)no2)nn1-c1ccccc1 C(=O)(C(F)(F)CC1CCCO1)NCCC1(OC)CN(C(CSCC=C)=O)C1 N1(C(CCN(C2CCC2)C(C)=O)=O)CC(NC=O)C(C)C1 c1(C(N2CCCCC(NC(C(CC)SC)=O)C2)=O)c(O)cc(F)cc1F c1(C(=O)N)cccc2cnccc12.N1(C(C)C)CC2CC(N(C)CCO)CC1C2 c1(C(=O)NC(C2CCCN(C(CS(=O)(=O)NC)=O)C2)C)cccc2nnn(C)c12 N(C1CCc2c(Br)cccc21)C(C1C(C(=O)Nc2c(O)ccc(C)n2)C1)=O CCC(C)(CNC(=O)C(C)OC)NC(=O)C(C)NC(C1(CO)CCCC1)=O Cc1cccc(N(c2nnnn2C2CCOC2)CCCCCOC(F)F)c1 N1(C(CC2(C=C)CC2)=O)CCC2(C1)CN(C(=O)CN(CC)CC)CC(C)O2 N1(C(C2C(CNC(CCC(C)OCC)=O)CCC2)=O)CC2CC1C1CC21 c1(CN2C(C)(C(=O)NCc3cccc(-c4cnoc4)c3)CC2)cccc(Cl)c1Br c1(C(N(CCNC(c2c[nH]cc(C)c2=O)=O)CC)=O)ccn2cncc2c1 C1(NC(C(C)OCCN(C)C)=O)(CO)CCC(C)(C)CC1.C1(=O)CCN1 C1(NC(C2(Cl)C(C(C)=O)C2)=O)CCCC(C(=O)NCC(O)CCC2CC2)C1 N1(C(C2C(=C)C2)=O)CC2CCC1C(CN=c1cc(C(=O)OCC)nc[nH]1)C2 C(=O)(C1=CC2(CCOC2)C1)NCC1N(C(C2(CF)CC2)=O)CCN(C)C1 C(CC(C)(C)C(=O)N1CCC(CNC(=O)C(C)n2cnnn2)C(C)C1)OC C1(C(=O)NCC(C)(CO)CO)CC2CN(C(C3COCC3C(N)=O)=O)CC2C1 N1(C(c2c(NC)c(F)ccc2)=O)CC2CCC1C(CNC(=O)C(C)(O)C(C)C)C2 C1(NC(C(C)OCC2CC2)=O)CN(C(=O)CCC=CBr)CC12CCCC2 c1(OC)ccc([N+](=O)[O-])cc1-c1nc(CCCOC)nn1C(C)COC Cc1nnn(CC(=O)NC(C)C(=O)NC(C(C)(C)O)C2CC2)n1 Cc1nc(C(=O)NC2CCCN(C(c3ccc(C4CC4)s3)=O)CC2F)c(=O)[nH]c1C c1(CC(=O)NCC2CN(C(c3onc(CC)c3C)=O)C2)ccc(Cl)c(Cl)c1C C1(CNC(c2ccc(C3CC3)o2)=O)CCC(C)CN1C(C(N1CCCCC1)C)=O N1(C(C2N(C)C(=O)CC2)=O)CCC(F)C(NC(C2CCCC23CC3)=O)C1 C#Cc1ccc(NC(c2cccc(F)c2)(C)C(=O)OCC(=O)OC)nc1 Cn1cc(C(=O)NC2CNCC2(C)C)c(-c2cnn(C)c2)n1 C1(c2ccc(C(=O)OC)o2)CCN(C(c2n[nH]cc2Br)C(=O)NC(C)(C)C)CC1 C1(CNC(C2C=CCC2)=O)CC12CCN(C(C1CC1c1ccccc1)=O)CC2 CCCC(C(=O)N(CC(C)NC(=O)CNC(C1CCOC1)=O)C)NC(N)=O C1(CC)CN(C(C)=O)CCN1C(=O)C(C(C)C)N1CCCC1=O C12(CNC(Cc3cnc(C)[nH]3)=O)CCC1CN(C(c1cc(C(C)C)n(C)n1)=O)C2 c1(C(=O)NCCCCN(C)C(C2CCCCC23CC3)=O)cccc2ccsc12 N(C(=NCCC(CN(C)C)N1CCCS1(=O)=O)NC1CCOCC1)C(CC)C.CCCC N1(C(C2CC(=O)NC2)=O)CC2(CCOCC2C(N2CCC3COCC3C2)=O)C1 CN1C2CCC1CC(=CC(N1CCN(C(C3CC(F)(F)C3)=O)CC1CF)=O)C2 c1(C(N2CCC3(CC2)CC(O)C3)=O)cc(Br)cc2[nH]ncc12 C=C(F)CN=c1[nH]c2c(c(=NCc3nc[nH]n3)[nH]1)CSC2 N1(C(C(c2cccs2)SC)=O)CC2(CCC2NC(c2ccn(C(C)C)c2C)=O)C1 C1(C(=O)NCC(c2cccc(F)c2)OCC)CCc2nnc(C)n2C1 C1(CNC(C=CC(CC)C)=O)CC(F)CN1C(c1cc(CN(C)C)c[nH]1)=O c1(COC)cccc(NC(=O)C(C2CCN(C(C3CC34CC4)=O)C2)(F)F)c1 c1(-c2n(CC(C)C3CC3)nc(Cn3cccn3)n2)cc(C2CC2)cnc1O C1(OCC(=O)Nc2cn(C)nc2)CC2CC(OCCCC3CCCC3)CC12 C1(=CC(=O)NC(CC=C)CNC(C2(C)CCOC2)=O)CCN(C)CC1 N#Cc1ccc(-c2cn(CC3CC34CCSCC4)nn2)nc1 CCCC(C(=O)NCC1(CN(C)C(c2sc(C(C)(C)C)nc2C)=O)CC1)OC C(=O)(C1OCCc2cc(C)ccc21)OC(c1ccc(F)cc1F)CCC c1(C(N2CCC(C=C)(O)C2)C(=O)NC2CCC2)cc2ccccc2cn1 C1(C(CC)(C)C)CCC(C(N2CCC(O)(CNC(C3(C)CC=CC3)=O)C2)=O)CC1 C(C(C)CC(=O)NC1(C(=O)NCCC2CC(C)=NO2)CSC1)NC(C)=O c1(N(C(=O)CCCNC(N)=O)C)ccc(NC(=O)CCN2CCOCC2)cn1 C1(CNS(C)(=O)=O)CN(CC(=O)NC(c2ccccc2)CO)CCC1(F)F N1(c2snc(C(N)=O)n2)CCC2CC(CNC(C3CS(=O)(=O)C3)=O)CCC2C1 C(CC(C)(C)C(=O)N1CC2CC(CNC(=O)C=C3CCC(C)CC3)C2C1)OC N1(C(C(F)OC)=O)CCOC2(CCC(NC(C3C=CCCC3)=O)CC2)C1 c1(C(N2CCCCC(NC(C3C(C)C3)=O)C2)=O)cc(Cl)c(Br)cc1N Cc1ccc(F)cc1C(=O)NC1CC(CNC(=O)COC2CC=CC2)C1 C1(CNC(CC(COC)(C)O)=O)CN(C(c2sccc2C#N)=O)CC(C)(C)C1 c1(N2C(CNC(CC3(C)CC3)=O)CCCC2)cc(Cl)nc(-c2nccs2)n1 O=C(C1CCCc2ncccc21)NCCC1CCCN(c2cc(Cl)c(O)nn2)C1 Cc1c(C(N2CCC(NC(c3csnc3Cl)=O)C(CO)C2)=O)sc2ccccc12 C#CC1(C)CCN(C(C2C=CC(NC(c3ccn(C)c3C)=O)C2)=O)CC1 c1(C(C)(O)C(=O)NCCC2CCN(C(=O)CCC3CC3)C2)ccc(Cl)cc1 C1(c2cn(CC)nn2)CCN(C(C2(COC)COC2)=O)C(C)C1 c1(C(N2CC(NC(C3(C)CC(C)OCC3)=O)C2)=O)cnn2ncccc12 C(=O)(C1=NNC(=O)CC1)NC1(C2N(c3c(Br)cnc(C(C)C)n3)CCC2)CC1 c1(C(N2CC3N(C(c4c(C)nn(CC)c4C)=O)C3C2)=O)cccc2occc12 Cc1noc(Cl)c1CCC(=O)NCCCCn1cc(-c2cccnc2F)nn1 C(=O)(CC(O)CNC(c1ccc(Cl)cn1)=O)NCCN(CCC)C(C)C C1(C(=O)NCCCCN(C(C(CC)(C)O)=O)C)OCC2COCCC12 N1(C(c2c(CNC(C=C(COC)C)=O)c[nH]n2)=O)CCC(OC(C)=O)CC1 CCC(CCC(=O)NC(COC)C(=O)N1CCC(C(F)(F)F)C1)OC C(=O)(CCCC(C)(C)C#N)N1CC(Cc2ccccc2)CC(CC)C1 c1(NC(C2CCC(NC(=O)CCc3cccs3)CC2)=O)ccc(Cl)cc1F c1(C(=O)NC2C(NC(C(CCC)OC)=O)C2)cnn(C)c(=O)c1 c1(OC(C)C(N2CC3(COC3)C2)=O)ccc(Cl)c(Cl)c1 c1(OC(C2CCCN(C(=O)OC(C)(C)C)C2)=O)ccc(NC(=O)COC(F)F)cc1 CC(CC(=O)NC12CC(CNC(=O)CCn3cncn3)(C1)OC2C)C(C)(C)C C1(OC)CC(CCNC(=O)Cc2ccnn2C)N(C(C2CCC(C(N)=O)O2)=O)C1 N1(c2c(S(=O)(=O)NC(C)(C3CC3)C3CC3)cncc2)CCCC2(CCCNC2=O)C1 C12(NC(C(C)OC)=O)CC1CN(C(C13CC(C1)C(C)O3)=O)C2 C1(CC(=O)NCC2(C(=O)NC3(CO)CC(C)C3)CCCO2)CCOC1(C)C c1(N2CCOCC(C(=O)NCC(COC)(O)CO)C2)ccnc2ncnn12 c1(OC(C(=O)NC(c2cccs2)CC)(C)C)ccc(COC)cc1 c1(CN(C(c2cc(F)ccc2OC(F)F)CC)C=O)ccc(C)cc1Br C1(C(=O)NC(C2N(C(c3c(C)con3)=O)CCC2)C)CCCCN1C1CCCC1 C(COC(C)C)(C(=O)N(C)CCN(C)C(c1ccoc1C)=O)NC(C)=O.C(C)(C)O Cc1c(C(=O)N(C)CC2CCN(C(C3(C)CCCCC3)=O)CC2)c(Cl)nn1C C1(C(=O)NCCNC(=O)OCC)CCN(C(c2n[nH]cc2Cl)=O)C1(C)C C(=O)(C(O)CCC(F)(F)F)NCC1(F)CCCN(C(CCC2CC(OC)C2)=O)C1 c1(C(=O)NCCCN(C(C(CCC)=CCC)=O)C(C)C)cc(N)ccc1F C(c1c(C)nn(C)c1Cl)=CC(N1CC2C(NC(c3ncc(OC)nc3)=O)(C2)C1)=O CC1Nc2ccnn2C(C)C1CCC(=O)N1CCC1C1CCCC1 N1(C(CCCC)=O)CC2ON=C(CNC(c3cn(CC)nc3C3CC3)=O)C2C1 C#Cc1ccc(C(N2CC3CCC3(NC(=O)CC=C(C)C)C2)=O)cc1C c1(OCC=C)ccccc1C(=O)NC(C)(CNC(=O)CCCF)Cn1cccn1 CCC(C)(C)CCCC(=O)NC1(CCO)CCN(C(=O)CC2CC2C)CC1 C1(NC(C(C)(C)C2CCC2)=O)(CO)CCN(C(C2(c3cc[nH]n3)CC2)=O)C1 N1(C(CCCC(=C)C)=O)Cc2ccccc2C(CNC(=O)CC2CCCCC2)C1 C1(C(=O)OC(C)(C)C)CCN(C(=O)N(C(c2ccc(C)cc2F)C)C2CC2)CC1(F)F C1(NC(c2c(CC)nco2)=O)CC2CN(C(c3ccc(Cl)nn3)=O)CC12 c1(C(N2CC3C(NC(CCNS(CC)(=O)=O)=O)C3C2)=O)ccnc2c1CCO2 CC(C)(C#CC(=O)NCC1CC(O)C12CCC2)CNC(c1cc(C#N)cs1)=O C1(C(C)(C)CNC(=O)COC2CCOC2)CCN(C(C2CCCCO2)=O)CC1 C(=O)(C1=CCCC1)NCC1N(C(C2(C#C)CC2)=O)CC1 c1(OC)cc(C)c(C(=O)N(C(C)CCNC(C2(C(F)F)CCCC2)=O)C)c(C)c1 N1(C(C=CCNC(C2CC(C)OC2)=O)=O)CCCC2(CCC2)C1 Cc1cccc(C(N2CCCC2CNC(c2cn(C(C)C)nc2C)=O)=O)n1 N1(C(COC)=O)CCC2CCN(C(=O)CCCCc3cc(OC)cc(Cl)c3)C2C1 C#CCCCCC(=O)NC12CC(C1)N(C(c1cc(CN(C)C)c[nH]1)=O)C2 N1(C(C(CCC)C)=O)CCOC2CCN(C(=O)C=C(CC)CC)CC12 c1(C(N(CCCCNC(=O)C(C)NC(=O)NC)CC)=O)cc(C(C)C)no1 CCC(CC)C(C)C(=O)NC(CO)C(=O)N1CC(C#N)C1 c1(C(=O)NC2C(C)N(C(=O)C=CCN3CCCCC3)CC2)nnn2ccccc12 C(=O)(C(O)C(C)C(=O)N(C)OCc1ccccc1)N1CC(CNC)C1 c1(CC(N2CCC(C(C)NC(=O)C(C)NS(C)(=O)=O)CC2)=O)cccc(Cl)c1F C1(C(=O)NC(c2cnn(C)c2)C(=O)NCC(C#C)CC)CC(=O)C12CCC2 C(CN=C(NCc1ocnc1C(F)(F)F)NCC1CCCC(C)(C)O1)OCC C1(NC(c2noc3c2COCC3)=O)CN(C(C2CCCC2)=O)C2(CCCOC2)C1 c1(CC(=O)NC(C(C(C)C)Nc2ccncn2)C)nc2c([nH]1)CCCC2 Cc1nc2ccc(C(=O)NCC3(C)CC(NC(C4(Cl)CC4(C)C)=O)C3)cc2[nH]1 N1(c2nccc(N3CCCC(Sc4ccnc(C)n4)C3)n2)CC2CCC(CC2)C1 CC(C)C(CNC(c1cc(C(F)(F)F)ns1)=O)NC(=O)Cc1cncn1C CCCC(O)CC(=O)NC1CC(CCNC(C2CCN(CC)C2)=O)C1 Cc1c(C(N2CC3(CCCN3C(=O)CCc3cnc[nH]3)C2)=O)ccc(Br)c1F c1(C(=O)NCCCN(C(=O)CC2CSCCS2)C2CC2)cc(C(F)F)cc(CO)c1 N1(C(c2cnc(C)s2)=O)CCC2C1CCCN2C(=O)CSCCN(C)C C1(C(=O)NC2CC(CCNC(=O)COCC3CCCOC3)C2)CCC2(C1)N=N2 c1(C(N(c2ccc(CC)cc2)C)=O)ccn2c1CS(=O)(=O)CC2 C1(C(=O)NCC2(C(N)=O)CN(C(c3ccncc3F)=O)C2)CCCC2CCCN12 c1(C(C(=O)NCCCN(C)CCO)NC(C2CCSC2)=O)cnn(C)c1 c1(CN(C(C2(OC)CCC2)=O)C)cccc(CNC(=O)CC2CCC(=O)N2)c1 C1(CCC)(NC(=O)Cc2n[nH]c(C)n2)CCCN(C(c2[nH]c(C)nc2C)=O)C1 c1(OC)ccc(-c2cc(C(=O)NCC(C)(C)CNC(=O)C(C)OC)nn2C)cc1 C1(C2(NC(c3nsnc3O)=O)CC2)CCCCN1C(=O)Cc1ccnc(Cl)c1 Cc1ncncc1C(N1CCCC1C(C)C(N1CCC(OCCO)C1)=O)=O c1(C(N2CC(CNC(c3ccc(C(C)(C)C)[nH]3)=O)C2)=O)c(N)cccc1[N+](=O)[O-] N1(C(C(CCC)S(N)(=O)=O)=O)CCCC2(CCCN2C(=O)CC2=CCOCC2)C1 N1(C(C2=CCCC2C)=O)CC(C(=O)N(CCCCO)C2CC2)C2(CCC2)C1 C1(CNC(C2(C)CC(=C)C2)=O)CC2CCC(C1)N2C(c1ncnc2sccc12)=O C1(CC=C)(NC(c2cnc(CC)s2)=O)CCN(C(C2(c3cc[nH]n3)CC2)=O)C1 c1(C(N2CC(OCCNC(c3c(CC)occ3)=O)C2)=O)cccc(F)c1 n1(CC)cc(CC(=O)NCc2cc(C(N3CC(OCC(N)=O)C3)=O)no2)cn1 c1(C(N2C(C)CC(CNC(=O)Cc3ccno3)C2)=O)cc(F)cc(N)c1N CC(CCCNC(C1C=CCCC1)=O)NC(C1(OCc2ccccc2)CC1)=O c1(NC(C(c2ccccc2)OC)=O)c(F)cc(C(F)(F)F)cc1F C#CCCC(C(=O)OC)NC(=O)C(CNC(C1CCCN1C(C)=O)=O)CC1CC1 N1(C(C(N(C(Cc2nc(C)sc2)=O)C)C2CC2)=O)CC2C(N(C)C)C2C1 n1(CC)cc(C(=O)NC(C)CN(C(=O)CN(C)C)CC)c(C)n1.C1(=O)CN1 C12(C(=O)NCC3OCCN(C(CSC(C)C)=O)C3)COCC1CN(C(N)=O)C2 c1(C(C(=O)NCCC2CC2)N(CC(=C)C)C)nc(C)sc1C Cc1cc(C(N2CC(C)(C)CC2CNC(c2[nH]cnc2C)=O)=O)c2occc2c1 c1(C(=O)NC(CC)CN(C(=O)Cc2cc[nH]n2)C)ccnn1C(C)CC c1(C(N(C)CC2CCCN2C(C2(Br)CC2)=O)=O)ccccc1C1CC1 c1(NC(C2(C)COC2)=O)cc(Br)cc2[nH]ncc12 N1(C(C2CN(CC(C)C)C2)=O)CCC2(NC(=O)CC3(N(C)C)CCC3)CC2C1 CCC(CCCC(=O)NC1CCN(C)C(=O)C1)NC(C1C2CC(=O)CC12)=O Cn1cnc(C=CC(=O)NCC2(F)CC(NC(=O)Cc3sccc3Cl)C2)c1 N1(C(CC(C)=CCC)=O)CCCC(C)(CNC(=O)CCCOC(C)=O)C1 C12(CNC(Cc3cc(C)[nH]n3)=O)CCCC1CN(C(c1c(C)cnnc1O)=O)C2 Oc1c(C)cc(F)c2c1CN(N1CCC(N3CCOCC3)CC1)CC2 N1(C(c2nc(OC)oc2)=O)C2CCC1CC(C(N1CCOC(C)CC1)=O)C2 Cc1ccc(CC(N2CC(C)CCC2CNC(C2C3CCCCC23)=O)=O)cc1F c1(CCNC(N2CCC(CC(=O)OCC)C2)=O)ccc(F)c(Cl)c1F N1(C(CCN(C(=O)COC(C)=O)CC)=O)CCN(C(=O)CC)CC1 Cc1nc2c(s1)CCCC2C(=O)NCc1ccc(-n2c(C)cc(O)cc2=O)cc1 C(=O)(CCC(=O)NCCNC(c1nnc(C)s1)=O)NCCOC(COC)C.SC c1(CCC)cc(C(=O)N(CC(C)N(C(=O)CSc2n[nH]c(O)n2)C)C)no1 Cn1ccnc1C(=O)NC(C)(C(=O)NC1COCC1F)C1CC1 c1(NC(C2CCC(NCc3ccc4sccc4c3)CC2)=O)ccn2nccc2n1 c1(C(=O)NCCN(CCC)C2CC2)ccc(OCCO)cc1 Cn1ccc(C(F)=CC(=O)NC2CCCCC2NC(c2cc3c(s2)CCC3)=O)n1 c1(OC)cc(N2CCCC2C2(NC(=O)Cc3cncn3C)CC2)ncn1 N1(CCC(=O)NC2CC(NC(C(C)OCCOC)=O)C2)CCOCC1=O c1(OC)cc(Br)ccc1C(=O)NC12CC(C(=O)NCc3ccnc(Cl)c3F)(C1)C2 C1(C#N)(C(=O)NCCOC2CCN(C(c3cc(OC)no3)=O)C2)CCCO1 C=C(C)CC(C(=O)N1CCN(CC)CC1C)NC(c1ccc(C)cc1)=O C1(N(C(=O)Cn2ncnn2)CCNC(C2C(C=C)C2)=O)CCCCC1 c1(CC(=O)NC2C=CCN(C(c3cnc(C)[nH]3)=O)C2)cccc(S(C)(=O)=O)c1 c1(C(=O)NCC2C(NC(C(C)CC3CC3)=O)C2)c(F)cc(Br)c(F)c1F N1(C(c2c(CC)occ2C)=O)CCC(CNC(C2(C(F)(F)F)CCC2)=O)C(C)C1 c1(CN2CC(F)CC(C(=O)NC(c3nccs3)C)C2)cc2ccc(C#N)cc2[nH]1 C1(NC(C2(CC)CCC2)=O)CC2CCC(C1)N2C(c1cc(C2CCC2)[nH]n1)=O C=C(C)CC(C(=O)N1CC(NC(=O)CC2(C)CCC2)C(C)(C)C1)NC(C)=O N1(C(C(C)N=[N+]=[N-])=O)CC2CCCC2(NC(=O)C(C)n2cccn2)C1 C1(NC(=O)C=Cc2ccsc2)CN(C(c2ccc[nH]2)=O)CC1F C1(C2CCN(C(=O)CCC3CCCO3)CC2)(NC(C2(S(C)(=O)=O)CC2)=O)CCC1 c1(OC)cc(Cl)ccc1C(N1C(C(=O)Nc2cc(Cl)ccc2CO)CC2CC12)=O c1(C(=O)NC(CC)CNC(=O)CC2OCCCO2)ccc2nc(C)cn2c1 c1(CC(=O)N(C(C)C(=O)N(C(C)(C)C)C(=O)O)C)ccc(B(O)O)cc1.C1CC1 C1(C(N2CC3C(NC(c4c(CC)scc4)=O)(C3)C2)=O)CCC2(CCC2)CO1 C1(CCC)CN(C(=O)Cc2cccc(Cl)c2)CCN1C(=O)C(C)OC N1(C(CC=CCC)=O)CC(NC(=O)C(C(C)C)c2ccncc2)C(O)C1 c1(C(N2CCSCC2C)=O)cc(C(=O)OCC)c(C)o1 N1(C(c2c(C)nc(CCCC)s2)=O)CCN(C(=O)C=CC(F)(F)F)C2CC12 CC(C(=O)NC1CC(C)(NC(=O)CCCc2ccc(F)cc2)C1)C(C)(F)F N1(C(c2csc(Cl)c2Cl)C(=O)NCc2cccc(Br)c2)CCCC2OCCC12 CC1(C(=O)NC2(C3CN(C(=O)C(O)C4CC4)C3)CC2)CCC(F)(F)C1 CC(CC(C(F)F)c1ccccc1)NC(c1cncc(C)c1)=O c12ccccc1[nH]c(=O)o2.C1(C(C)(C)C)C2CN(C(=O)CN3CCOCC3)CC12 n1(CC)cc(C(=O)NCC2(O)CN(C(C3CCC(=O)C3)=O)C2)c(C(C)C)n1 C(CNC(=O)CN(C)CCO)(CCNC(=O)C(F)C1CCOC1)OC C(=O)(C1CCCn2nccc21)N1CC(CCNC(CN(CCOC)C)=O)C1 Cc1cc2[nH]c(C(=O)NCC3CCCN(C(C45CC(N(C)C)(C4)C5)=O)C3)cc2o1 CCCCCCCCCC(O)C(=O)N1CCSCC1CNC(=O)Cc1ccoc1 Cc1sc(S(N)(=O)=O)cc1C(=O)NC(CNC(=O)Cn1cnc(=N)[nH]1)C(C)(C)C C=Cc1ccc(C(=O)NCC(C)CC(=O)NC2CCCN(O)C2=O)cc1 c1(CN2C(C(=O)Nc3cn(CC)nc3)C=CC2)cnc2ccccc2c1 C1(CNC(COC2C(CC)CCCC2)=O)CCCN(C(=O)C2=CCSC2)CC1 C(CC(C)(C)C)(C(=O)NCC1CC1NC(c1ncoc1-c1ccco1)=O)OC C1(C(=O)NC2C(CNC(c3cc(CC)cc(F)c3)=O)C2)CCCC(C)(C)CC1 c1(C(N(C2CCN(C(c3c(CC)cncc3)=O)CC2)C)=O)cccc2c1CCN2 C(=O)(C1CCCc2ccnn21)NCC1N(C(Cc2cc(C)c(Cl)cc2)=O)CC1 C1(C)(CNC(C(CC)(C)O)=O)COCCN(C(c2cc(C)ncc2C)=O)C1 C1(CC)CN(C(c2cc(C)ccn2)C(=O)OC)CCC1N N1(C(C=C(C)C(C)(C)C)=O)CCC(O)(CN(C(=O)CC2COCC(C)O2)C)CC1 CC12CC(C(N3CC4(CCC4NC(c4csc(Cl)c4)=O)C3)=O)(C1)C1(CCC1)O2 Cc1cc(C(=O)NCC2CCCCN2CC(c2ccco2)O)cc(I)c1 CCC(CC(=O)NCC(C)CC(=O)N1CC(c2ccon2)C1)C(C)(C)C N1(C(C2CN(CC)C(=O)C2)=O)CC2(C1)CN(C(c1ccc(N)cn1)=O)C2 c1(C2(CNC(=O)NC(c3cnccn3)C)CC2)ccccc1Br C1(NC(Cc2cc(C)no2)=O)CC2CCC1N(C(c1cc(N)c(F)cc1C)=O)C2 c1(C(N2CC3C(CNC(c4cc(CCO)on4)=O)(C3)C2)=O)ccc2[nH]ccc2c1 c1(C(N2CC(C(C)(C)O)(CNC(=O)CC3CCC(O)C3)C2)=O)ccc(F)nc1 c1(CNC(=O)CC2CC3CN(C(c4ccncn4)=O)CC23)cc(Cl)ccc1[N+](=O)[O-] Cn1c([N+](=O)[O-])cnc1C(N1CC(NC(C2CC3OC2C2CC32)=O)CC1CO)=O C(C)(C(C(C)C)NC(c1c(CC)noc1C)=O)NC(C=CC=CC)=O N1(C(c2c(OC)csc2)=O)CC(OC)CC(NC(C2NC(=O)OC2C)=O)C1 N1(C(CCCC(C)=O)=O)CCC2CCCN(C(c3c[nH]cc(Cl)c3=O)=O)C2C1 N(C(=NCCC(C)C)N(C)Cc1cc(F)ccc1C)CC(COC)OC c1(C(c2ccncc2)NC(=O)NC(CC)C2CCC2)ccc(Br)cc1 n1(CC(=O)NC(c2cccnc2)CCC)ncc(Cl)c1C C(=O)(C(C(C)(C)C)c1ccc(F)c(C)c1)NC(CCNC(CCC=C=C)=O)C Cc1ccc(C=CC(=O)N(C2CCN(CCOc3ccc(OC)cc3)C2)C)o1 n1(CC(C)C)cc(C(=O)NCCC(C)N(C)C(c2cscc2Cl)=O)cn1 N1(C(C(CCC)C(=O)OC)=O)CC2CCC1C1CN(C(=O)CC(F)(F)CC)CC21 CC1CCC(C(=O)N(C)CC2(NC(=O)CC3CSC3)CC2)S1 c1(C(=O)NCC(CNC(c2on(C)c(=O)c2)=O)CO)cc2cc(Cl)ccc2o1 N1(C(c2ccc(C)o2)=O)CCCC(NC(c2nc[nH]c2C(F)(F)F)=O)C1 N1(C(C(=O)NCC)=O)CC(NC(c2nn(C)cc2N)=O)C(C)C1 c1(NC(c2cc(NC(CC)=O)c(C)cc2)=O)ccc(N(C)C(c2ccco2)=O)cc1 N1(CC)CCN(CC(=O)NCCCC(C)NC(c2ccon2)=O)CC1 Cc1ccc2cc(C(N3CC4CC(NC(C5(CO)CC5(F)F)=O)C3C4)=O)cn2c1 c1(CC)ccnc(C(=O)NCCC2CN(C(C3CC3C(=O)NC)=O)CCO2)n1 N1(C(CSCCCC)=O)CCCC(CN(C(=O)C(CC)n2cncn2)C)C1 C1(C(N2CC(CCNC(C3CCCN3C(C)C)=O)(OC)C2)=O)CC(F)(F)C1(C)C c1(C(=O)NC2C(CNC(C(C)C(F)F)=O)CCCC2)ccc2c(c1)CCOC2 C1(C)(C(=O)NC(COC)CNC(c2cc(CO)[nH]n2)=O)CC(C)(C)C1 CC1CN(C(c2cccc3ncnn23)=O)C(C)CN1C(=O)CN1CCC(=O)CC1 C1(CNC(C(C=C)O)=O)CCCN(C(=O)CCCOC(C)=O)CC1 C1(C)(C(N(C(C(=O)OC)C)C)=O)CN(C(=O)CCc2nc(=N)[nH][nH]2)C(C)(C)C1 CC1CC(NC(c2sccc2CN(C)C)=O)CN1C(=O)Cc1nnc(O)s1 C1(C(N2CCC(C=C)(O)C2)=O)CC2(CCN1C(c1ccc(C)c(C)c1)=O)CC2 C1(C(N2C(C)CCC2)=O)CCCC12CCN(C(c1ccc3ocnc3c1)=O)C2 C1(CC(=O)N(C2(C)CC2)C)CCCCN1C(=O)C=CCO C1(C(N2CC(n3nnnc3CO)C2)=O)(CC)CCN(C(C2CC(F)C(=O)N2)=O)C1 C=CC(C)(CC)C(=O)NCCC1(OC)CN(C(=O)CCc2ccc(Cl)s2)C1 N1(C(CC=CC)=O)CC(CC(=O)NC2CCCC3(C2)N=N3)C2(CC2)C1 N(C(=NCCCC(C)(C)C)NCc1ccc2c(c1)oc(=O)n2C)CCCSC NC(=O)CCCCC(=O)NC1CN(C(=O)Cc2cc(Cl)ccc2O)CCC1O C1(C(N2CCC(CCNC(c3c(OC)ccnc3)=O)C2)=O)CCn2cncc2C1 C=CCCCCCC(=O)N1CCC(CCNC(=O)CCCC(C)=O)C1 C1(NC(c2cccc3ccccc23)=O)CS(=O)(=O)CC1N=c1nc(CC2CC2)[nH]s1 C1(CCN(C(C(C)CN(C)C)=O)C)CCCCN1C(=O)C=Cc1ccnn1C C1(C)(CC)C=C(C(=O)N2CCC(C)(NC(=O)CNc3ccccc3C)C2)C1 c1(OC)ccc(C(=O)NCC2CCCN2C(=O)CC2CCC23CCC3)c(Cl)c1OC c1(C(=O)NC2CC3CC2N(C(=O)Cn2cccn2)C3)cc2cc(Cl)ccc2s1 C1(CC(=O)NC2CC(C(C)C)C2)CN(C(=O)CC2CCCN2C)CCO1 c1(C(N(CCCCN(C(C2CN(C)C2)=O)C)C)=O)nn(C)nc1Br N1(C(C(C=C)(C)O)=O)CCN(C(=O)C(CC)n2ccnc2)C(C(C)C)C1 C=CCC(CNC(c1nccn1CC)=O)C(=O)NCC12CC(CCO1)C2 C(=O)(CC(C)C(F)(F)F)NC(C)CNC(C1CCCN(c2ncccn2)C1)=O C(=O)(CCC(CF)CF)C(=O)C(F)CC1CNC1.c1(C(=O)N)cocc1C(N)=O C(C)(C(=O)N(C(C)C(=O)NCc1cccc(O)c1F)C1CC1)(C(C)C)OC C(c1ccc(=N)[nH]c1)=CC(N1CCC(O)(C(C)NC(c2cnns2)=O)C1)=O C(=O)(C(=O)C(C)(C)C)NC(CN(C(c1ccc(C)cc1)=O)C)C c1(OC)noc(C(N2CC(C)(NC(c3cnc[nH]3)=O)C2)=O)c1Br CC(O)C(F)(F)C(=O)NC1CC(N(C(=O)C(CC(F)F)C2CC2)C)C1 c1(CN2CC(F)(C(=O)Nc3c(C)cc(I)c(C)c3)C2)ccc2c(Cl)ccnc2c1 c1(N(CC(N2C(CC)CCCC2)=O)C)c(C)nc2ncnn2c1NC(=O)C(C)C C1(CN(C(c2ccns2)=O)CC)CCCCN1C(C1C=CCCC1)=O C12(CNC(CC(C=C)C)=O)CCC(CNC(C3CC(O)(C(F)F)C3)=O)(CC1)CO2 C1(C(N2CC3C(CNC(c4c(CC)n(CC)nc4)=O)C3C2)=O)CN2CCC1CC2 C1(C(N2C(C(=O)NCC(=O)NC3CCNC3=O)CSC2)=O)CC=CC(O)C1 C(c1ccc(F)cc1)=CCC(=O)NC(C)CNC(=O)CSc1c(O)cccc1F CC1CN(C(=O)C(=O)NCc2ccc(C(=O)N(C)C)nc2)CCS1=O C(=O)(CS(N)(=O)=O)N(CC(C)N(C(=O)CC1CCCO1)C)C C(=O)(CCCCCC#N)N(CC(CO)(CO)NC(CC1N(C(C)C)CCC1)=O)C C#CCC(CC(=O)N(CCCN(C(=O)CC1CCC1)CC)CCO)c1ccccc1 N1(CCCOCCOCCOC2CC2)CCCC2(CCC2)C1C Cn1c([N+](=O)[O-])cnc1C(=O)NC1CCCC1CNC(c1c[nH]cc1Br)=O C12(C(=O)NCC(C)NC(C3(N(C)C)CCC3)=O)C3CCC(CC13)C2(F)F N1(C(C(C)C)C(=O)N2CN(C)C(=O)C2C)C(=O)c2ccccc2C1=O c1(C(=O)NC2CCN(C(CC(CC)C3CCC3)=O)C2C)cc2n(n1)CCCC2 CC(C)(C(=O)N1CC2CC(C1)C2NC(=O)C=CC(F)(F)F)C(N)=O Cc1cccc(C(C)N(C)C(=O)NCC2(c3ccc(F)cn3)CC2)c1 C1(NC(c2n(CC)ncc2Cl)=O)CN(C(=O)CC2COC3CC2C3)C(C)(C)C1 C1(CC)CN(C(C2CCCC(CF)C2)=O)CC1C(=O)NCC=C(Cl)Cl C(=O)(C(C)(C)C(=O)N1CCC1C(=O)NC1CCC(F)(F)CC1)OCC C1(C(=O)NC2C(NC(c3[nH]cc(CC)c3)=O)CS(=O)(=O)C2)CCC2CC1C2(C)C C1(C(=O)Nc2cncc(OC)n2)CC(F)CN(Cc2cnc(F)c(C)c2)C1 C1(NC(C(C)OCCC=C)=O)CCCN(C(c2ccnc(C(C)(F)F)c2)=O)C1 c1(N2CCCC(CCNC(C=CCCC)=O)CC2)ncnc2c1cnn2C c1(NCC(CCCOC)O)ccc(Br)c(C#N)c1 C1(NC(CCSC)=O)CCN(C(c2cn(-c3ncccn3)cn2)=O)CC1C CC(=O)CCCC(C)C(=O)N1CC(F)CC1CNC(c1ccc(C)n(C)c1=O)=O C(c1c(Cl)cccc1Cl)=CC(=O)NC1(C)CC(NC(c2cc3sccc3[nH]2)=O)C1 CCC(C)C(C(=O)N(CCCCCC(=O)NCCN(CC)CC)C)OC CC1Cn2nccc2CN1CC(=O)N(c1nc(Br)cs1)c1ccccc1 c1(N(CC(=O)N(C(C)C)CCC)C(=O)CC2CCCCO2)ccc([N+](=O)[O-])cc1Br c1(C(=O)NCCNC(CCN2CCN(C)CC2)=O)c2c(nn1C)CCOC2 c1(S)ccc(S(=O)(=O)N)s1.Cc1nc(C)n(CCCC(=O)N(C)C)n1 n1(CC=C)c(N(C)CC2COC(=O)O2)nnc1-c1cncc(OC)n1 N1(C(C=C2CCC(C)C2)=O)CCCCC(NC(=O)CN2C(=O)CCC2=O)C1 C1(C(=O)NCC2C(CNC(c3cc4c([nH]3)CCCC4)=O)C2)Cc2cccnc2C1 c1(NC)cncc(C(=O)NC(C2CN(C(c3ccc(F)s3)=O)CCO2)C)c1 N1(C(C=CC2N(C(CCCNC(=O)OC)=O)CCC2)=O)CCOC(C#N)C1 C(=O)(C1Cc2ccc(C)cc21)N(c1ccccc1)C(c1cc(C)ccc1C)CC CC1(C)CC=C(C(=O)NC2CC3C(CNC(C45CC4COC5(C)C)=O)C3C2)CC1 C1(CNC(c2c(C)noc2C2CC2)=O)CC(F)(F)CN1C(=O)CSC(F)F c1(C(=O)NCC2C(NC(C(c3cc(C)cc(F)c3)C)=O)C2)cnc2c(Cl)cccn12 c1(COCCNC(c2n(CCC)nnn2)C2CC2)cccc(F)c1I CC(F)(F)CCCC(=O)NC1CN(C(=O)C(=Cc2cccnc2)F)C1 c1(C(N2C3CN(C(=O)C=CCO)C(CC3)C2)=O)ccoc1S(=O)(=O)c1ccccc1 Cc1ncc(CC(=O)NC(C2CN(C(C3(C)CC=CC3)=O)C2)C)s1 c1(C(N2CCN(C(C(CC)O)=O)C(CO)C2)=O)nc2cc(F)ccc2s1 CC1(C(N2CC(NC(c3cnsn3)=O)C(C)(C)C2)=O)CCC2(CC1)CC2 CCC(CS(C)=O)NCC(c1ccc(SC)cc1)=O C1(CCOC)(NC(c2cnn(C)c2Cl)=O)CCN(C(C2CCCC(F)C2)=O)CC1 c1(C(N2CCN(C(C=COCC)=O)CC2CF)=O)cccc2c1CC(C)(C)C2 Cc1ncsc1C=CC(=O)NCC1CN(C(c2ccc(CO)cc2)=O)C1 C1(NC(=O)NCC(=O)NCC=C2CN(C(=O)C=Cc3cccs3)C2)CCCCC1 CC(C)C(CC(=O)N1CCC(C)(O)CC1)NC(C1CCC(=O)N1)=O N1(C(C)=O)CC(O)CC1C(=O)NC1CCCC1CNC(C1CSC(C)=N1)=O C=C(CNC(=O)C(CC)NC(N)=O)CCNC(=O)CCNC(=O)CO c1(C(=O)NCC(CN(C(=O)CC2(C)CC2F)C)(C)C)ccn(C)c1C1CCC1 c1(C(N(c2ccc(NC(C3CCC4(CC3)CC4)=O)cn2)C)=O)c(F)cncc1F C12CN(CC3(CO)CC3)CC1CNC2=O.C(C=C(Cl)Cl)=S(C(C)(C)C)CC=O N1(C(C(C)=O)=O)CC(NC(c2cccc(C3CCOC3)c2)=O)C(C)C1 C1(CNC(C(c2ccc(F)cc2)(C)C)=O)CC2CCC1N2C(=O)Cn1ccnn1 c1(C(=O)NCCCC2CN(C(C3CC4CC4C3)=O)CCO2)cncc2c1CCC2 S(=O)(=O)(c1cnc(N(CCCOCCOC)C)c(Cl)c1)NC(C)CCO Cc1cnc(NC(C)CCC2CC2)c(S(=O)(=O)NC2(C)CC(C)(C)C2)c1 N1(C(C(CC)C)=O)CCC2(CC1)CC(NC(=O)Cc1nc(C)cs1)C2 c1(-c2cn(CCc3nnc(C(C)C)o3)nn2)cc(OC(C)C)ccn1 c1(OCC(=O)Nc2c(CCNC(CCC(C)OC)=O)n[nH]c2)ccc(C)cc1Cl c1(C(=O)NC23C(CN(C(c4cccc(OC)c4)=O)C2)C3)nn(C)cc1[N+](=O)[O-] N1(C(c2cccc(CC)n2)=O)CCN(C(=O)Cc2ccc(C#N)cc2F)CC1C C1(NC(CNC(CN(C)C)=O)=O)CCCN(C(=O)CCC2CCC2)CC1F c1(C(N2CCC(NC(c3cc4cccnn4c3)=O)C2)=O)cccc([N+](=O)[O-])c1Br Cc1ccncc1C(N1CCC(CCC(=O)NCCn2cnnn2)C1)=O N1(C(C(C)(C)F)=O)C(C(N2CC3CC2CS3)=O)CC2CCCC12 c1(C(=O)NC)ccc(OC2CN(C(c3ccc(OC)cn3)=O)CC2O)cc1 C(CCCCCNC(C1CCCN1S(C)(=O)=O)=O)NC(C(C)(C)N(C)C)=O CC1=C(C(=O)N2CC3CCC3(CCNC(c3ncc(F)cc3F)=O)C2)COCC1 C(CCN(CC(C)O)C)(C(=O)NCC(C)O)NC(C(CC)NC(C)=O)=O N1(C(C2NC(=O)OC2)=O)CCC2(CC1)CC(NC(c1cc3sccc3s1)=O)C2 C1(C)(CNC(C(c2scc(C)n2)C)=O)CCCN1C(=O)Cc1csc(Cl)c1 N1(C(C2CC(CC)C(=O)CC2)=O)CCC2(CC1)CN(C(=O)CC1CCCCO1)C2 C1(CNC(C2C(C)(CC)C2)=O)C(C)CCN1C(c1ccncn1)=O c1(C(N2CC(N(C)C(c3ccc(C(C)(C)C)cn3)=O)C2)=O)nc2ccccc2[nH]1 C(=O)(C1=NOC2(CCN(C(c3ccnn3C)=O)C2)C1)NC(C)Cc1ccccn1 C12CCCC(C1)C(=O)N2.c1(CN(C)C)cn(CCCCO)nn1.C1C(=O)N1C1CC1 C1(N(C(=O)C(=O)NC2CC2)CC)CCN(C(=O)CC2COC(=O)C2)C1 C(C)(C)(C(C)CC(=O)NCCCSCC)NC(CCC(CC)C)=O c1(OC)ccc(C(=O)NC23CCC2CN(C(c2cscn2)=O)C3)cc1Cl C1(C)(CNC(c2[nH]cc(C(C)(C)C)c2)=O)CCCN(C(=O)C(O)c2ccsc2)C1 c1(OC)cc(C#N)ccc1OCC(=O)N(C)Cc1ccc(-n2cccn2)c(F)c1 n1(CC(N2CC3C(NC(C4CC(=O)NC4)=O)(C3)C2)=O)nc2c(n1)CCCC2 C1(C(=O)NC(C)C(C)NC(c2ccc(C#N)cc2O)=O)CC2(CCOCC2)C1 CC1(C)CC=C(C(=O)NCC2CC(NC(=O)C(=O)Nc3ccccc3)C2)CC1 c1(N(C(C2N(C(C(CC)OC)=O)CC2)=O)CC)cccc(F)c1 Cc1cn(C)nc1C(N1CCC(C(=O)NCCC2(C)CCCO2)C1C(C)C)=O c1(C(=O)NCC2(F)CN(C(C34CCCC3C4)=O)C2)nnc(O)nc1O c1(C(N2CC3C(N(C(=O)Cc4ccnnc4O)C)C3C2)=O)ccc2nnnn2c1 N1(C(C(C)N(C)CC2CCCS2(=O)=O)=O)CCC(C2CC2)C1 C(CC(C(C)(C)C)NC(=O)Nc1cccc(O)c1)OC C1(CC)CC2(CC(C(=O)OC)C2)C1.N12CCCCC1NC(=O)NCC2 N1(C(CC2CC(=O)C2)=O)CCN2CCC1C2 N1(C(C(c2c(OC)cccc2)C)=O)CC2CCC2C1CNC(c1cc(C)cs1)=O c1(C(=O)NC2CCCC(N(C(=O)CCOC3CC3)C)C2)cc(Cl)nc(Cl)c1 N1(CC(=O)NCCC2CCCN(C(C(C3CC3)OC)=O)C2)CCCCCC1=O N1(C(C(CSC)C)=O)CC2CC(C1)CN(Cc1cc(O)ccc1F)C2 C1(NC(=O)C=Cc2ccoc2)C2CC1CN(C(c1cc(O)cs1)=O)C2 Cc1nnc2c(C(N3CCN(C(=O)Cc4c[nH]ccc4=O)C4CC34)=O)cccn12 N1(C(C=CC=CC)=O)CCCC(C)(NC(=O)Cn2ncc(Cl)c2C)C1 C1(C(C)(C)C)CC1N=c1nc(-c2ccccc2)[nH]c(=NC2CC3CCCC(C3)C2)[nH]1 C(N=c1ccc(C(F)(F)F)n[nH]1)=C1CCN(C(=O)Nc2ccn(C)n2)CC1 N1(C(C(C)(C)CCCO)=O)CCOC2(CCCN(C(=O)C3=CCCS3)C2)C1 C1(CCNC(C(C)OCC#C)=O)CC(F)(F)CN1C(=O)CCc1nccs1 CCC(CC(=O)NC1CCSC12CN(C(c1cccc(F)c1F)=O)C2)CC(C)C CCCC(C(=O)OC)C(=O)NCC1CCN(C(C2CCCC(O)C2)=O)CC1C C1(C(N2C(CNC(C(C#C)(C)C)=O)CCCC2)=O)CCCC2(C1)CC2(F)F c1(OCCC(=O)NC2CCOCC2NC(C23CC(F)(C2)C3)=O)ccc(Cl)cc1 c1(CC(C)C)ccc(C#N)c(N2CC3(C2)SCCC3NC(=O)C(C)C(C)O)n1 C(C1CCCN1C(=O)C(C)=C1CC1)=CC(=O)NCC(=C)C N(C(=NCCCF)NC1CC1(c1ccc(Br)c(OC)c1)C)CCOC N1(C(C2CN(C)C(=O)C2)=O)CC2CN(C(=O)Cc3ccsn3)CC(C1)O2 c1(C(=O)NCC23N(C(CC(=O)OC)=O)CC(C2)C3)cccc2c1NC(=O)CC2 C1(C(N(CCCNC(C2CNC(=O)N2C)=O)C)=O)Cc2ccncc2C1 c1(C(=O)NCCC(CNC(c2c(CC)cncc2)=O)O)c(F)cccc1F c1(NS(c2cccc(C)c2)(=O)=O)n[nH]c(=NC2CC3C(C2)C3(F)F)s1 N1(Cc2c(C)cc(Br)cc2)CCC2(CC1)CC(NC(C1CC3C=CC1C3)=O)C2 CC1CCC(NC(=O)NC2CC(c3ccon3)C2)C1 N1(c2cc(C)nc(N3CCCC(C(N)=O)C3)n2)CCC2(CC1)CC(C(N)=O)CO2 C1(COC)CCC(C)(C)N(C(C2CC(C)CC(C)C2)C(=O)NCCC#N)C1 N1(C(CN(C(=O)C(O)Cn2cncn2)C(C)C)=O)CC(F)(F)CCC1C C12(CCNC(c3c(C)cc(SC)o3)=O)CCC(C1)N(C(=O)CC1CCOC1)C2 n1(CC(=O)NCC2CCN2C(c2cc(CC3CC3)on2)=O)cnnc1O N1(CC(N2CCC(N(C(C(CC=CC)C)=O)CCO)C2)=O)C(=O)CC(C)(C)C1=O C1(NC(C2(C)CC2)=O)CN(C(=O)CC2C(C)(C)C2(C)C)CCC1C(F)(F)F CCCC(C(=O)N(C)Cc1ccccc1)NC(=O)CC(C)=C(C)C c1(C(=O)NC2C(CO)CCN(C(C(CC)NC(N)=O)=O)C2)cncc2nc[nH]c12 O=C1CC2(CC(=O)N2CN2CCCC(OCC3CC3)C2)CCO1 CCC(CCCC(=O)NOC1CC1)NC(=O)C(CC)CCOC c1(NC(=O)CSCc2nc(-c3cccs3)no2)cccc(Cl)c1Cl Cc1ccc(C)c(C(=O)NCc2cccc(NC(C3CCC(=O)NC3)=O)c2)n1 N1(C(C(=O)NCCOCC)C2CCOC2)CCCN(C(=O)CC)CC1 C1(C(N2C(CNC(COCC(=C)C)=O)CC3CC32)=O)COC2(CCC2)CO1 N1(C(Cc2c(C)n(C)nc2)=O)CCCC(F)(C(=O)NC2CCC3(CC3)C2)C1 c1(CC(=O)NC(CCC2CC2)C(=O)Nc2cnn(CCF)c2)ccc(F)nc1 C(=O)(C1=CC2C=CC(C1)C2)N1C(C(N(C(CC(C)C)C)C)=O)CC1C N1(C(CC=CC)=O)CC2(NC(=O)C(O)CCSC)CCC1C2 c1(C(=O)NC(C)CCNC(=O)C(C)(C)C2CC2)cc(F)c(F)c(F)c1F c1(C(=O)NCCN(CCOC)C(C2CC23CC3)=O)cncn1-c1ccccc1 c1(C(N(C2CCN(C(=O)Cc3cn[nH]c3)C2)CC)=O)cccn2cncc12 C=CC1OCCCC1C(=O)NC1CC1NC(=O)Cc1ccc(OC)c(F)c1 C1(NC(c2c(C)scn2)=O)CC2CC1CN(C(=O)CN1C(=O)CN(C)C1=O)C2 C1(CC(=O)NCC2OCC(CNC(COCCC=C)=O)C2)CCS(=O)(=O)CC1 N1(C(c2c(CC)scc2)=O)CCC(O)C(NC(C2CC3CCC2C3)=O)C1 C1(C(=O)NCC2N(C(c3c(C)ccs3)=O)CCC2)CC12CCOC2 C(=O)(CC(O)CN(C)C)NC1(CC(=O)NC2C(C(=O)OC)CC2)CC1 C1(C(=O)NCC2N(C(C3(C(C)C)CNC(=O)C3)=O)CC2)Cc2ccccc2C1 C12(CC=C)CCN(C1)C(=O)C1(CC1(C)C)C(=O)N2.c1(CC(=O)NC)csc(CC)n1 C1(C)(C(NOCC(N2CCC(C)(CCOCC)C2)=O)=O)CC2C=CC1C2.C(COC)S N1(C(C(C)Cn2cccn2)=O)CC2CC(C1)N2C(c1cc(C(=O)O)nn1C)=O c1(COC)ccc(NC(C2CCN2C(C2(OC)CCC(C)(C)C2)=O)=O)cc1 Cc1cc(C(=O)NC(C)CNC(=O)CCc2nc(-c3ccoc3)no2)ccc1F N1(CC)CCOCC1CC(=O)NC(C)CCCNC(c1cn(C(C)C)cn1)=O c1(C(=O)NC2CN(C(C(C)C3CCC3)=O)C2)ccc2nc(O)[nH]c2c1 c1(NC(C2CC(C)N2C(C2(CO)CC2)=O)=O)cnccc1CO c1(C(=O)NC2CCN(C(CC(CC)C3CCC3)=O)CC2)ccc(F)c(CO)c1 C(=O)(C(O)C1=CCCCC1)N1C(C)CC(CNC(c2ccc(C)c(C)c2N)=O)C1 N1(C(C2CCC(CC)CC2)=O)CC(N)C2(CCS(=O)(=O)CC2)C1 CCC(CCC(=O)N1CCCc2nccn21)NC(=O)CC(C)(C)COC Cc1ccc(SCC(=O)NCCC2CN(C(=O)CC34CCCC3C4)C2)c(C)c1 C1(NC(c2c(F)cc(CC)c(F)c2)=O)CC2CN(C(=O)C3=CSCS3)CC2C1 C1(N=c2cc(C)c(C#N)c(C)[nH]2)(CC)CCN(C(=O)C(C)NS(=O)(=O)CC)CC1 C1(F)(CNC(COc2c(C)cccc2)=O)CCN(C(=O)CCC(N)=O)CC1 N1(C(c2sc(C)c(O)n2)=O)CC2CCC(C1)C(NC(c1ncccc1Cl)=O)C2 Cc1oc(CNC(C2CCC2(F)F)=O)nc1C(=O)NC1CC(=O)N(O)C1 S(=O)(=O)(c1ccc(C(=O)OCC(=O)C(C)(F)F)cn1)N(C)C c1(C(N(C(C)CNC(c2nc(O)[nH]c(=O)n2)=O)C)=O)ccc(F)c2ccccc12 C1(CNC(=O)CCN2CCCC2)CC(F)(CNC(=O)CNS(N)(=O)=O)C1 c1(C(N(C(C)C)CCNC(=O)CCCC2CC2)=O)n[nH]c2c1CCOC2 C#CC1CN(C(C2CCCCC2F)=O)CCN1C(=O)C=Cc1ccc(C)o1 CC1CN(C(=O)CC2(C(F)F)CC2)CCC12CCN(C(C1CCCN1C)=O)CC2 C1(NC(c2c(C)ccc(C)c2)=O)CCC2CN(C(C3(Cl)CC34CCC4)=O)CC2C1 N1(C(Cc2ccc(CC)cn2)=O)CCc2sc(CO)cc2C1 C=Cn1nccc1C(=O)NC1CCN(C(=O)C(N2CCOCC2C)C)C1 c1(C(c2nnnn2CCOC)NCC(=O)OC(C)C)cccc(F)c1Cl CC(C)C(C)(CNC(c1cnc(O)s1)=O)NC(=O)CC1(C)CCC1 C1(NC(c2cc(C)no2)=O)CCN(C(c2cc(C(F)F)on2)=O)C(C2CC2)C1 c12cc(nc(Cl)c1)N(C)C2C(=O)NC1CC1.C(C)(C(=O)NC(C)C)NC.CS c1(C(=O)NCC2OCC(CNC(COCC)=O)C2)c[nH]c(=N)nc1C(F)(F)F C1(NC(c2c(C)noc2C(F)F)=O)CCN(C(=O)Cc2ccc(Cl)s2)CC1C N1(C(C2(C)CCSCC2)=O)CC2(CCCC2NC(=O)C(=O)C2CC2)C1 c1(C(=O)NCCC(C)S)ccnc(C(F)(F)F)c1[N+](=O)[O-] CCC1=C(C(=O)N2CCN(C(C3OCCN(C)C3=O)=O)C3CC23)CCCO1 C(C1CN(C(C2(CCC)CC(=O)C2)=O)Cc2ccccc21)NC(CC=C)=O c1(OC)ccccc1CC(=O)NC(CCNC(=O)Cc1ccccc1)C(C)C c1(NC(C2CN(C(c3cnon3)=O)CCC2O)=O)cn2c(Br)cccc2n1 C12(OC(C)C)CCCCCC1N(C(=O)OCc1cccc(C(C)C)c1)CC2 CCCC(C(=O)NC1CCCC12CN(C(=O)Cn1nccc1C)C2)C(C)C C(c1ccccc1C)=CC(=O)NCC(C1N(C(CCNC(C)=O)=O)CCC1)(C)C C1(C)(C(=O)NC(CC)CNC(C2CC3CC3C2)=O)CCCC1CC c1(OCC(=O)NC2(C3N(C(=O)C(F)(F)OC4CC4)CCC3)CC2)cccc(Cl)c1 c1(-c2cccc(C#N)c2)ccc(C(=O)NCC2CCC(F)(F)C2)c2c1OCO2 C1(NC(C2COCCO2)=O)CN(C(c2cc3sccc3s2)=O)CC12CCCC2 Cc1c([N+](=O)[O-])c(C(=O)NC(C)CN(C)C(C2CC3CCC3C2)=O)nn1C c1(-n2cc(C(C(OC)OC)C)nn2)ccc(C(=O)OCC)c(F)c1O CC1(C)CC(=O)NCC1C(N1CC(NC(C2CC(N(C)C)C2)=O)C1)=O C1(NC(=O)NC(c2ccc(C)o2)(C)C)CCC(=O)N(C)C1 N1(S(c2c(OC)ncc(Cl)c2)(=O)=O)CC(C2CC2)C(F)(CO)C1 O=C1CC2CCCC2(C(=O)NC2CN(C(=O)COCC3CCOC3)C2)C1 C12(CC3COC1C3)c1n(nnn1)C1(CC1)C(=O)N2.C1(CSC)CC(=C2CCC2)C1 c1(C(=O)OC)cccc2nc(C(=O)NC3CC(C)N(C(=O)C(C)C)C3)cn12 N1(C(c2ccn(C)n2)=O)CCC2(CC(C(=O)N(c3ccc(Br)cc3F)CC)=NO2)C1 c1(SC)nc2cc(n1)N1CCCC(C1)CC(CO)CNC(=O)N2.C(C)(C)(C)O C1(NC(C2(C=C)CCC2)=O)CC1C1CCCN(C(c2oncc2CC)=O)C1 C=CC1(CC(=O)NCc2cc[nH]n2)CN(C(C2CC3CC3C2)=O)C1 S(=O)(=O)(C(F)(F)F)N1CC(C(=O)NCCN(C(C=C(CC)C)=O)C2CC2)C1 C1(C(=O)NC(CC2CN(C(C(C)OCCCC)=O)C2)C)CC(=O)NC(=O)C1 CCC(C)(CO)C(=O)NCC1CCC(NC(=O)CC2CCC(=O)NC2=O)CC1 c1(N2CCN(CCOCCC=C)CC2)nc(F)nn2c(Br)cnc12 C(CNC(=O)CCCCN(C)C)(C(C)C)NC(C(C)OCCC#C)=O C(=O)(CS(=O)(=O)CCC(F)(F)F)N(CC(O)CNC(=O)C1=NN(C)C(=O)CC1)C N1(C(=O)Nc2c(N)n(CCO)nc2)CCc2ccccc2C(NC(=O)C(F)(F)F)C1 c1(OCCOC)cccc(C(=O)NC2CCCN(C(C3CC(N(C)C)C3)=O)C2)c1 N1(C(CCCN(C)C)=O)CC2(CCN(C(=O)C(C)(F)c3ccon3)CC2)C1 N1(C(C2C(C)(Br)C2)=O)CC2(CCN(C(C3CCCC(=O)CC3)=O)C2)C1 N1(C(C(CC=CCC)C)=O)CCC(C(=O)NCC2CC2COC)CC1C C(=O)(C(F)C(C)(C)O)NC1(C)CC(NC(C=C2CCN(C)C2)=O)C1 N1(C(c2cc(C)cc(C)c2)=O)CC2CCCN(C(=O)CCCS(N)(=O)=O)C2C1 C#CCCOCC(=O)N(C(CNC(C1CC1C)=O)C1CC1)C Cc1ccc2nc(C(N3C(CCn4cc(CNC)nn4)CCCC3C)=O)cn2c1 c1(CC(=O)N(C(C(=O)NCCCCC2C(C)C2)C2CC2)CC)coc2ccccc12 C1(CN(C(=O)CCC2CC2(Cl)Cl)C)CCN(C(c2cc(C#N)on2)=O)CC1 C1(C(=O)NC(C2CCN(C(=O)C(C)(C)N3CCCCC3)C2)C)CNC(=O)N1 C(=O)(CCC(O)C(C)(C)C)NC(C1CN(C(c2ccc(C(N)=O)o2)=O)CCO1)C N1(C(C(C)Oc2ccccc2Cl)=O)CC2CN(C(=O)Cc3cnc[nH]3)CC2(C)C1 CC1(C)CC(CO)CN(C(=O)C(CC2CCC2)NC(C2CCCC2O)=O)C1 CC(C)C(O)C(F)(F)C(=O)NCC1CN(C(=O)C(C)CC2CCCC2)C1 N1(CCNC(CSCC#C)=O)CCN(C(=O)CCc2nc[nH]n2)CC1 C(=O)(NNc1c(F)c(F)cc(F)c1F)C1CC(C(=O)OC)C12CCOCC2 c1(C(=O)NCc2cn(C3CN(C(C4C(C(C)C)C4)=O)C3)nn2)cnc2n1CCS2 c1(NC(c2cc(C)on2)C2CC2)nccc(CN2CCCO2)n1 CC1(C)CCC(C)(C(=O)NC2CC3CCC2C(NC(C2CCOC2)=O)C3)CC1 N1(C(=O)OC(C)(C)C)CCCC(O)(C(=O)NCC23COC(C2)C(O)C3)C1 c1(C(=O)NC2C(C(=O)NCC(c3ccccc3)CC)C2)cccnc1 C1(C)(NC(CCSc2n(C)ccn2)=O)CCN(C(=O)C(O)c2ccco2)CC1 N1(C(C2C(OC)CCC2)=O)CCC(=CCNC(C2(O)CCSCC2)=O)CC1 C1(NC(C2C(=C)C2)=O)CCCCC12CCN(C(=O)CC1C=CS(=O)(=O)C1)CC2 N1(C(C(C)SC)=O)CC2(CCC(NC(c3sccc3-n3ccnn3)=O)CC2)C1 C12(N(C=O)Cc3cn(CCOC)nc3)CCC(C1)OC2 N1(C(c2ccc(OC)o2)=O)CCC(C)(NC(=O)C=C2CCCCC2)C1 N1(C(c2cc(C)sc2)=O)CCOC(C(=O)N(C(C)C(N)=O)C)CC1 CCCC(C(=O)NC1CN(C(c2cnnn2C)=O)CC1CCC)C(C)C C1(CC(=O)NCC2OCCN(CC)C2)CC(C)(C)CN1C(c1[nH]c(C)cc1C)=O C1(NC(C2CC(SC)C2)=O)CN(C(c2nccnc2N)=O)CC2(CCC2)C1 CS(=O)(=O)c1cccc(NC(C2CN(C(=O)CC3(O)CCC3)CCC2O)=O)c1 C1(NC(C(C)NC(C)=O)=O)CCC(CNC(C2(S(N)(=O)=O)CC2)=O)CC1 c1(C(=O)NC2CC2NC(c2sccc2NCCOC)=O)ccc(OC)c(OC)c1.CC Cc1cc(C(=O)OC(C)COCc2ccccc2)nn1-c1ccccn1 c1(OC)ccc(C)c(C(N2CC(O)(CNC(c3cc(C#N)c[nH]3)=O)C2)=O)c1 C(Cc1ccoc1)(C(=O)N(CC)Cc1cnsc1)NC(C=CC=CCC)=O N1(C(c2scc(C)c2C)=O)CC2CN(C(=O)CCc3csnn3)CC(C1)O2 C(=O)(C(CO)C(C)(C)C)N1CC2(CC(CC(=O)NC(C)C(C)(C)CO)C2)C1 CN1CCN(CCNC(c2ccc(OCc3nc(C(C)(C)C)no3)cc2)=O)CC1 c1(C(N2CCCCC(NC(=O)CC3OCCO3)CC2)=O)nccc2ncccc12 c1(CNC(C2N(C(C=CC(C)(C)C)=O)CCC2)=O)cncc(F)c1 Cc1nc(C(=O)NC2(C(=O)N(C3CC(O)C3(C)C)C)CC2)sc1C C#CC1(CNC(c2nnnn2C(c2ccccc2)C)CC2CCCC2)CCCC1 C1(CC)COCCN1C(c1ccc(C2CCN(C(C)=O)C2)cc1)C(=O)NC(C)CC Cn1ncc2c1CC(C(=O)NCC(C)(C1CCC1)NC(c1cc(F)c[nH]1)=O)CC2 CCCCC(C(=O)NC(C)CCC1CCCC1)NC(C1C(C)C1C)=O C=CC(CC)C(=O)N1CC(F)(C(N2CCC(CN=[N+]=[N-])C2)=O)C1 C(CC(CC)C(=O)NC(CO)C(=O)NCC1(C)CCOC1)=CC c1(C(C(=O)NC)N(c2ccsc2C)C)nc(C)ccc1OC CC(C(=O)NCCC(=O)NNC(=O)CC1(C)CCO1)S(=O)(=O)c1ccccc1C#N C(=O)(C(CC)CC)NCC1C(NC(C(C)OCCC=C)=O)C1 N1(C(c2c(C)[nH]nc2Br)=O)CCCC2(CCN(C(c3cnc[nH]3)=O)CC2)C1 C1(C(=O)NC2C=CCN(C(C(Cc3ccc(C)cc3)C)=O)C2)CCCC(C)CC1 c1(NC(CN(C(C(c2cccnc2)OC)=O)C)C)ccc(C(C)(C)C)cc1 CCC(C)C(O)C(C)C(=O)N1CC=C(C(=O)NCCC(=O)NC)C1 c1(C(C)C)ccc(C(N2CCC(C(C)NC(c3nsnc3O)=O)C2)=O)s1 C(=O)(C#CC1CCOCC1)N1C(C)CC(NC(=O)COc2cccc(Cl)c2Cl)C1 C1(CNC(C(CC)n2ccc(Cl)n2)=O)CN(C(C2CC(O)C2)=O)CC12CC2 c1(C(=O)NC2CC(CCNC(C3(Cl)C(C)(C)C3)=O)C2)ccc(-c2cnc[nH]2)cc1 CC(C)C(O)C(=O)NC1(CCNC(C2CCCN2C(=O)OC2CCCC2)=O)CC1 C(=O)(CCC(=O)N1CCC(NC(c2cccnn2)=O)C1)OCC C1(CNC(COCCCC)=O)CC(C)N(C(c2cnccn2)=O)C1 N1(C(C2C(CC)CCC2)=O)CCCC1C1CCCN1C(c1nn(C)c(C)c1Cl)=O C1(C(N2CCC(C(C)C)C2)=O)CC=CCN1C(C1CN(C)C1)=O c1(C(=O)NCC2CCCC(NC(=O)C=Cc3ccsc3)C2)ccc2ncsc2c1 c1(C(=O)NC2C(C)CC23CC3)ccc2ncn(C)c2c1 N1(C(c2cc(C)ccn2)C(=O)NCCCSC)CC(C)Oc2ccccc21 c1(C(=O)NCC2N(C(CC3CC(=C)C3)=O)CCC2(C)C)c(C)cc(C)cc1C S(=O)(=O)(CCN=c1[nH]c(=NCC2(c3cccc(Cl)c3)CC2)[nH]c2c1SCC2)NC CC1CN(C(=O)C#CC2CC2)CC1CNC(c1cnccn1)=O C1(C(N(CCNC(c2c(C)nn(CC(F)F)c2)=O)C)=O)CCC12CCCO2 C1(CNC(C(C)CC2CCC2)=O)(CNC(c2cnccn2)=O)CC12CCC2 N1(C(=O)CC2CCCCO2)CCC2(C(=O)NCCCCC3CC3)CCCC12 C(=O)(C1CCc2nccn21)N1C2CC(NC(=O)C=Cc3ccc[nH]3)CC1CC2 C1(CC)CC(C(=O)NCC2CC(C)N(C(C3CCC(=O)CC3)=O)C2)CC(=O)N1 C(=O)(C(C)(CC)C(=O)NCC1COCCN1C(c1ccc2nncn2c1)=O)OC N1(C(c2cnccn2)=O)CCC2CC(C1)CN(C(c1ccc(C(N)=O)[nH]1)=O)C2 CCC(CC)C(C(=O)NCC(CC(=O)NCC1CC12CCC2)C1CCC1)OC C(CC(C)C)(C(=O)N1CCC(C(=O)NC2CSC(C)C2)C1)OC c1(O)cccc(C(c2nnnn2C(C)C)OCCOC)c1.C(C)(C(C)SCl)NC1CC1 c1(C(N(CCCNC(=O)CC2CCN(C)C2=O)CC)=O)ncc(F)cc1F C=C(C)C(C)(C)C(=O)N1CCC1C(=O)NCC1(O)CCN(C)C1 Cc1cc(C)c(C(N2CCCC(CO)(NC(=O)C(C)S(N)(=O)=O)C2)=O)c(S)n1 C(=O)(C(F)CC1CN(C(=O)CCc2nc[nH]n2)C1)NCC(C)N(C)C C(C)(C)(CC=CC(=O)NC(C)Cn1cncn1)NC(C(C)OCC)=O c1(Cn2cc(CNC(C)C(c3ccccc3)O)nn2)cccc(N)c1 CCC(CNC(=O)COCCN(C)C)(CC)C(=O)NCc1ccc(O)c(C)c1 N1(C(c2cc(COC)ns2)=O)CCC(NC(c2cn3ccnc3s2)=O)C(CO)C1 c1(CN(CC)Cc2cc[nH]c(=N)c2)c(I)ccnc1F C12(NC(Cc3nc(=N)[nH][nH]3)=O)CCCC1CN(C(c1cocn1)=O)C2 Cc1ccccc1OCC(=O)NCC1(O)CN(C(=O)CC2CCCNC2=O)C1 N1(C(C(C(=O)OCC)F)=O)CC2CC(CNC(=O)C(C)(C)CCCO)CC1C2 C1(C(=O)NCCNOC)CN(C(=O)Cn2cccc2)CC12CC2 CCCCC(O)C(=O)N1CCC(F)(C(=O)NCc2nc(C)ns2)CC1 c1(OC)ccccc1NC(C1(N(C(=O)CC(C)(C)OC(C)C)C)CC1)=O N1(C(c2cc(CCC)on2)=O)CC2CCC(CNC(=O)CC3CSCCO3)C2C1 c1(C(=O)OC)cc(SCCCN(C)C(c2cnc(O)[nH]2)=O)oc1C Cc1ccc(-n2cc(C(=O)NCCCCC3CCOC3=O)nn2)cc1C c1(CC(=O)NCC2CC(NC(C3CC(=O)N3)=O)C2)coc2cc(Cl)ccc12 N1(C(c2cnc(C3CC3)s2)C(=O)NCCOCC)CCOCC1C1CC1.CSC CC(C)C(CNC(C1CCN(C)C1=O)=O)C(=O)NCCCc1nncn1C c1(CN(C)C(c2cnc(CNC(c3ccccc3Cl)=O)nc2)=O)cccc(O)c1 CC1C(c2ccsc2)CCN1C(=O)CC12CC(C(=O)NC(C)(C)C)(C1)C2 Cc1ccc(C(N2CC(CC(N3CCC(OC4CC4)C3)=O)C3(CC3)C2)=O)cc1O N1(SC)CCCN(Cc2nc(NC(C3CC4CCCCC34)C)cc(O)n2)CC1 C=CCCCC(C(=O)N1CCOC(C2(C)CC2)C1)NC(c1cnc(C)c(C)c1)=O CCC(C)(CO)C(=O)OCc1ncc(C)c(NCC2CC2)n1.c1(O)ccccc1Cl c1(C(=O)NC2C(CC(=O)NCC(C#C)OC)CCC2)cccc2cncn12 N1(C(C2C(CC)CCO2)=O)CCN(C)CC1C(=O)NC(C)CN1CCCCC1 c1(NC(C(C)NC(c2ccc(OC)c(F)c2)=O)C(C)C)ncc(C#N)cc1F n1(COCCOC)cccc(C(N2CC(O)C2)=O)c1=O.C12CC1NC(=O)C2.CC c1(C(N2CCC(C(F)F)(CNC(CSC)=O)C2)=O)cc(C)cn2ccnc12 N1(C(CCOC)=O)CC(CNC(=O)CCCNC2CCCCC2)CC12CCC2 C(=O)(C(C)(C)CCC(=O)NC(CO)C(C)NC(c1sc(F)cc1C)=O)OC N1(C(c2cnc(C)s2)=O)CC2CCC2(CNC(c2cc(Cl)c(Cl)[nH]2)=O)C1 c1(-c2n(CCOCC)nc(C3CCC3)n2)cc2c(cc1C)OCO2 C1(OC(C)C)CCCCC1c1nc(S)n[nH]1.n12ccc(n1)COC(=O)C2 CCC(C)C(C(=O)NCC1(F)CN(C(=O)COCCN(C)C)C1)NC(C)=O N1(C(C(C=C)O)=O)CCN(C(c2cc(S(=O)(=O)NC(C)(C)C)c[nH]2)=O)CC12CC2 C=C(C)CC(C(=O)NC1COCC1C)NC(c1ccsc1C#N)=O C(=O)(C(C)(C)C(=O)NCCC1CN(C(=O)CCCOCc2scnc2C)C1)OC Cc1c(C)n(C)c2ccc(C(=O)NC(C)C(C)NC(C3CCCO3)=O)cc12 c1(CC)cc(C(=O)NCC2CC(NC(C3C4CCC3CC4)=O)C2)ncn1 c1(C(N2CCC(C#C)(CO)C2)C(=O)NC2(C)CC2)sc2ccc(F)cc2c1C CC1CCN(C(=O)C(c2ccccc2)NC(=O)CCC(=O)N(C)C)CC1(C)C C=CCCC(C)(c1nnnn1-c1ccccc1OC)NCC1CS(=O)(=O)C1 N1(C(C(C2CCOCC2)OCC)=O)CCOCC(F)(CNC(=O)CC(F)F)C1 n1(CC(=O)N(C(C)C(=O)N(CC(C(C)C)OC)C)CC)cnc(C#N)n1 C1(CNC(c2c[nH]nc2Cl)=O)CCCCN(C(=O)CCC2CC2(Cl)Cl)C1 c1(CC)cncc(C(=O)NC2CC(C)N(C(=O)Cc3cn(CC)nn3)C2)c1 C(=O)(C(CC1CC1(F)F)OC1CCCO1)N(CC(=O)OC)Cc1ccsc1 CC1CCC=C1C(=O)OCC1CCCCC1F S(=O)(=O)(c1c(Cl)cc(Br)cc1Cl)N(C(C)(C)C)Cc1ccc2c(c1)OCCO2 N1(C(c2cnc(SC)s2)=O)CC(C)N(C(=O)CCc2cc[nH]n2)CC1C CC(C)CC1C(=O)NC2CC(C2)COC(=O)N1.C(=O)(C(C)(C)C(F)F)NC1CC1 C(=O)(C1=CCCOC1)NC(C)CCNC(C1(C)CCN(C)C1)=O CN=c1ccc(C(N2CCC(C)(CC(=O)N(CC(C3CCC3)OC)C)C2)=O)c[nH]1 C1(NC(CC=CC)=O)CCCCC12CCCN(C(=O)Cn1nccc1C)C2 C1(C2CC2)(CNC(C2(CC(C)C)CCC2)=O)CCN(C(c2nncs2)=O)C1 CN1C(=O)CCCC1C(=O)NCCCC1CCCCN1C(c1cccnc1O)=O c1(OC)ccc(CC(=O)NCCCOCCN(C)C(c2ccc(CO)o2)=O)nc1 C1(C(=O)OC)CCN(CCn2cc(CO)nn2)CC1C N12CCC(CC1)C(=O)NC1CC(C1)C2=O.c1(C(N)=O)cc(C(N)=O)co1 CCCCC(F)C(=O)NC1CC(C(C)NC(c2[nH]nnc2CC)=O)C1 N1(C(c2cc(C)ncn2)=O)CCC(C)C(NC(=O)CC2CSC2)C1C CN1CCC(C)(C(N2CCC2C(=O)NCC2(CO)CC3CC3C2)=O)C1 c1(OCC(=O)NCC(C)(C)N2CCCC2)cccc2ccccc12 c1(NC(=O)C(N2CCC(c3nccs3)CC2)=O)ccc(F)c(Br)c1 CC1(C)COCC1CC(=O)NC1COCC1CNC(c1cnc(=N)[nH]c1)=O C(c1ccoc1)=CC(=O)NC(C1CCCC1)CNC(C(N(C)C)C1CC1)=O Cn1c(NC(=O)C(n2cc(Br)cn2)C2CC2)nc2ccc(Cl)cc12 C1(C(=O)NCC2(CNC(c3c(C)ncs3)=O)CCCC2)CCCN(CC)C1.C(C)C c1(SCC)ccc(CCCC(=O)N(CCNC(c2ncc[nH]c2=O)=O)CC)cc1 c1(OCC)ccc(CCN(C)C(=O)NCCc2cccc(OC)c2)cn1 c1(C(N(CC(CC)NC(=O)CCCCCF)CC)=O)cnc2[nH]nnc2c1 C1(CNC(C2OCCN(C)C2)=O)CC2CCC(C1)N2C(=O)CCCOC(C)(C)C C(=O)(C(C)(C)CC1CC1)N(CCCCN(C)C(c1cn(C)c(O)n1)=O)C c1(C(=O)NC2CC(C)CN(C(C3(C)CCC3)=O)C2)cc([N+](=O)[O-])ccc1Cl CC1(C)CC1(C#N)C(N1CCC(CCNC(c2cnc(S)n2C2CC2)=O)CC1)=O C(CC)(CCC(=O)NC(C)C#N)NC(C(CC)OCC)=O c1(CCNC(=O)Cc2cc(F)ccc2C(F)(F)F)ccc2c(c1)COC2 C1(CCC=C)(C(=O)NC2COCC2NC(=O)Cn2ccc(Br)n2)CCCC1 CC1CN(C(=O)COCC(F)(F)F)CCC1NC(=O)CNC(=O)CN(C)C N1(C(c2cncc(C)c2)=O)CCCC2CN(C(=O)CC3CCC3)CCCC12 CC(C)C(C(=O)NC(C)CNC(=O)CNC(=O)Nc1ccc(Br)cc1)NC(N)=O C=C1CCC(NC(C2(COC)CN(C(C3C4CC5C(C4)C35)=O)C2)=O)CC1 N1(C(C(=O)Nc2ccc(CN(C)C)c(Br)c2)=O)CC(F)(F)CC2(CCC2)C1 CCCCC(C)(F)C(=O)N1CC(CNC(=O)C=Cc2ccnn2C)C(C)C1 N1(CCOC)CCCN(C(=O)C(N)C(C)C2CC2)CC1 N1(C(C(C2CC2)OCC)=O)CC2CCN(C(=O)C=Cc3csc(C)n3)C2C1 c1(C(=O)NC(C2CCN(C(=O)Cc3cncs3)C2)C)cc(=O)n(C)c2ccccc12 CC1CN(C(=O)CC2CCC(=O)N2)CC1NC(c1cc(Br)c[nH]1)=O C(=O)(C(C)CCCc1ccccc1)NC(C)CCNC(C1(P(C)(C)=O)CC1)=O C1(NC(c2c(CC)nc(C)o2)=O)CC2(CCN(C(=O)CC(F)(F)F)C2)C1 N1(C(C(C)OCC)=O)CC(O)(C(C)NC(=O)C=CC2CCCO2)C1 N1(C(c2ccc(C(C)=O)[nH]2)=O)CCC(C2CCN(C(C3CC3(Cl)Cl)=O)C2)CC1 n1(CCOC)nnnc1C(c1ccnn1C)NCCCCO.C1(C)(CO)CC1 CCC(C)(CNC(=O)COC1CC(NC(c2occc2CN(C)C)=O)C1)C(C)O C1(OC)CN(C(c2scc(C)c2Cl)=O)CC1NC(=O)C(F)(F)C12CC(C1)C2 c1(CC)oc(C)cc1C(=O)NCCC1CCCN(C(=O)C(n2ccc(C)n2)C)C1 C1(C(C)C)CN(C(c2cnn(CCO)c2)=O)CCCN1C(C1CC=CCC1)=O N1(C(=O)CC2CCC3CC23)CC2(C(=O)NC3CC(OC4CC4)C3)CC1CO2 c1(C(=O)NC2CC(CNC(C3CC(CCC)C3)=O)C2)oc(Br)nc1C C(=O)(CC(C)(C)CN(C)C)N(C)CC1CCCN(C(=O)CCCC2CCCC2)C1 c1(C(C)C)ncncc1C(N1CCC(N(C(=O)C(C)Cc2ccco2)C)C1)=O N12CCSC(C1)C(=O)NOCC2=O.C(C(=O)OC)OCCC C1(CC(=O)NC2COC(C(F)F)C2)C2CCC(C2)N1C(=O)C=Cc1cc[nH]n1 CC(CS(C)(=O)=O)C(=O)NC(C)CNC=O.c1(N)csc(=NC)[nH]1 c1(C(NC(=S)NCC(F)(F)F)C)ccccc1Br.C1CC1 C1(C)(CNC(C2CCN(CC)C2)=O)CN(C(C2(C3CC3)CC=CC2)=O)CCO1 NS(=O)(=O)N1CC(C(N2CC3C(NC(=O)C(F)CC4CCC4)C3C2)=O)C1 C1(NC(C(C(CC)C)OC)=O)C2CCC1CN(C(=O)C#CC1(C)COC1)C2 C1(Nc2nc(C)nc(=N)[nH]2)CN(C(C2CC23CC(C)(C)C3)=O)CC(C)(C)C1 c1(NC(C2C(C=CC)CN(C(c3cc(C)oc3C)=O)C2)=O)cc(C)c(C)c(C)c1 N1(C(=O)CN(C)C2CC2)CCC(O)(CO)C1.C(C)(C(=O)NCCOC)NC(CC)=O c1(COC(=O)Cc2csc(Br)c2)nccc(N2CCCC2)n1 C1(N(C(C2N(C(c3ccc(OC)s3)=O)CC(F)C2)=O)C)CCCC(C)C1C c1(C(C)C)cccc(OC(C2CC3CC3N2Cc2ccc(F)cc2)=O)c1 Cc1c(CC(N2CCN(C(=O)Cc3nncn3C)CC2)=O)nc(Br)n1C c1(NC(C2(OC)CCS(=O)(=O)C2)=O)cnc2c(c1)NC(=O)CS2 N1(C(CC(=O)OCC)=O)CCC(NC(=O)CC2OCCCC2(C)C)C(C)(C)C1 C1(C(N2CC(N3CCN(C(CS(CC)=O)=O)CC3)C2)=O)CCN(CCO)C(=O)C1 Cc1ccc(C(=O)NC2COCCN(C(=O)CC3CC34CC4)C2)c(F)c1 c1(CCC=C=C)nc2nn1c1ccccc21.C(CCC)S N1(C(COc2ccc(CC)nc2)=O)CCCCCCC1CC O=S(=O)(c1cccnc1NCC1(F)CCC(CO)CC1)NC1CC2CCC1C2 c1(C(=O)NCCC2CN(C(CC(CC)(F)F)=O)CC2C)ccn2cccc2c1 c1(C(N2CC3C(CNC(c4ccc(C#C)cc4)=O)C3C2)=O)onc2ccccc12 c1(C(=O)NCCCN(C(C2(OC)CCC2)=O)C2CC2)nc(O)[nH]c1 c1(N(C23CCC(N)(CC2)C3)C(c2c(OC)ccs2)=O)ncnc2c1CCC2 C=C(C)CCCC(=O)NC1CCN(C(C2CN3CCC2CC3)=O)CC1F C1(N(C(COCc2cc(C)no2)=O)C)CCCC(NC(=O)CCC2CCCC2)C1 N1(C(=O)Nc2ccncc2Cl)CCOc2cc([N+](=O)[O-])ccc2C1 c1(C(C)=O)cc(CCC(=O)NCC2CC(O)CN2C(c2nnn(C)n2)=O)oc1C c1(CNC(C(=O)N(C2CCCN(CC#N)C2)CCO)=O)cn2ccccc2n1 C1(C(=O)NC2C=CCN(C(=O)C=CC3CCC3)C2)Cc2nccnc2C1 Cn1nc(CC(=O)NCCC2CCN(C(c3cnns3)=O)C2)c2ccccc12 C1(CC)CC(C(=O)NC2CCC(NC(=O)Cn3nc(C)cc3OC)CC2)CCO1 N1(CC)CC(C(=O)NCC(C)NC(=O)C(F)C2CCCC2)CCC1=O C1(C(N(CCC(=O)NCCCCC2CC2C)CC)=O)CCCOC1 c1(C(=O)NC2CCN(C(C3(SC)CCC3)=O)CC2O)ccnc2nc(C)nn12 C1(C(N2CC(NC(c3c[nH]cc(F)c3=O)=O)C2)=O)CC1C1CCOCC1 C(=O)(C(C)NC(=O)C(C)C1CCCO1)N1CC(CCC)C1 C1(COC(=O)Cc2ccc(N3CCCCCC3)cc2)CCCC(F)(F)C(=O)N1 C1(C(=O)NC2C(C)(C)CN(C(=O)OC(C)(C)C)C2)(CO)CCS(=O)(=O)CC1 N(C1CN(C(C2(CF)CC2)=O)Cc2ccccc21)C(C1CC(C(=O)OC)C1)=O C12(NC(C(C(=O)OC(C)(C)C)N(C)C)=O)CCC(CC1)N2C(=O)C(Cl)=CCl Cc1[nH][nH]c(=NC(=O)C2CC3CCCC(C2)N3C(c2ccsn2)=O)c1C c1(NC(=O)NC(C2CC(F)(F)C2)C2CC2)coc(C2CC2)n1 c1(C(=O)NC2C=CCN(C(COCc3cn(C)nc3)=O)C2)ccn(C)c(=O)c1 c1(N(C)CC2C(C)C2)nc(=NCCC2COCCO2)[nH]c2c1CCCCC2 c1(C(c2n(C(C)C)nnn2)NCCn2cnnc2)cccc(C(F)F)c1F C(=O)(C(C)=Cn1ccnn1)NC1C(CC)CN(C(c2cc(C)cc(C)n2)=O)CC1 C1(CNC(C2(SC)CC2)=O)CN(c2nc(Cl)c(C#N)s2)CC(C)(C)O1 N1(C(c2scc(C)n2)C(=O)NCC2CCCO2)CCCC12CCOCC2 N1(C(C2C(OCC)CC2)=O)CCCC(C)(C)C1CNC(C1(SC)CCC1)=O Cc1ccc(C)c(CN2CC3(CC3)CC2C(=O)Nc2cc(Br)ncc2F)c1 C1(C(=O)NCC(CC(C)C)NC(C(CC)F)=O)CC2CC(O)CC(C1)C2 CC1CC(C(=O)NC2(CO)CN(C(c3cc(Br)cnc3N)=O)C2)=NO1 C#CCC(C)C(=O)NCC1CN(C(=O)C(C)Cc2ccccc2)CC1C N1(C(C(C(C)C)OC)C(=O)NC(C)C)CCOC2COCC12 N1(C(CCCNC(C2(c3nc(=O)o[nH]3)CC2)=O)=O)C2CCCC1CC(O)C2 c1(C(=O)NCCCN(C(CCSC)=O)CCO)cc2cc(F)c(F)cc2[nH]1 N1(C(C(C=C)O)=O)CCN(C)C(CNC(c2nocc2C(C)(C)C)=O)C1 C(C(=O)N=c1cc(C)n(C)[nH]1)CC1(C)CN(C(C(CSC)OC)=O)C1 Cc1c(C(=O)NC2(C(=O)NC3CC(=O)N(C)C3)CCN(C)C2)cccc1F C1(NC(C(C)(C)C(F)F)=O)CN(c2ccncc2[N+](=O)[O-])CC2(CCOCC2)C1 c1(C(C(C)(C)C)NC(=O)NCC(C)OCC#C)cccc(Br)c1 C1(NC(=O)OCC)CCC2(CC1)CC2(F)F.C(C(CCOC(C)(C)C)CO)NC(C)=O C12(C(=O)NC3CC(NC(c4c(C(C)C)cccc4)=O)C3)CCCC(CO1)C2 C1(C2CCN(C(c3nocc3Cl)=O)C2)(NC(CCC#C)=O)CC1 C1(C(=O)NC(C(C)NC(C2(C(N(C(C)C)C)=O)CC2)=O)C)CCS(=O)(=O)C1 n1(C(C)C)ccc(C(N2CC(NC(=O)CC3CSC3)CC(F)C2)=O)cc1=O N1(C(C(CCC)O)=O)CC2CC(C1)N(C(c1ccc(OCF)cc1)=O)C2 C(CO)(C(C)NC(=O)CC1CCCN1C(=O)CC1(C)OCCO1)SC C1(CNC(C(C)(C)OCCC)=O)CCC2(CCC2)C1O c1(C(=O)NCCCC(C(=O)O)N(C)C)cnn2c(C3CC3)cc(C3CC3)nc12 C(=O)(C(CO)C(F)(F)F)NC(C(N1CC(C#C)C1)=O)CO C1(CC)CN(C(C2CCCN(C(=O)C=C(C)COC)CC2)=O)CC(=O)N1 C(=O)(C(C)(C)CN(CC)C)NS(=O)(=O)CCCCC(C)N N1(C(C2CC(C)N2C(C2CCC(C3CC3)C2)=O)=O)CCN2CCC1CC2 C=CCC(CC(=O)NC1CCCN(C)C1=O)NC(=O)Cc1cccc(F)c1 C1(CNC(CC(CC)OC)=O)CCCCCN1C(=O)Cc1cc(C)sc1C CC1CCC(c2cccc(F)c2)N(C(=O)C(=O)NC2COC(C(F)F)C2)C1 c1(C(Cn2cc(CC(=O)OC)nn2)=O)c(C)cc(C)cc1C.C12CCCCN1C2 C=CC(CC)C(=O)NCc1cc(C(=O)NC2CC=C(C)CC2)on1 CC1CN(C(=O)C(=O)NC2CC2)CCN1C(=O)CC(C)(C)c1cccc(Br)c1 N1(C(CC2ON=C(C)C2)=O)CC2(C)CC1(C(=O)N(C1(C)CCCC1)C)C2 c1(C(=O)NC2C=CC(C(=O)NCCC(C)C(F)F)C2)ccc(=O)n(C)n1 N1(C(c2c(C(C)C)ocn2)=O)CC2CCCC2(N=c2[nH]nc(O)s2)C1 CC(C)CC(C)(CO)NC(=O)CC1CCCN(C(=O)C(N)=O)C1 N1(C(CC(C)C2CCCCC2)=O)CCCC(N(C(C2CC(O)C2)=O)CC2CC2)C1 C1(CCNC(c2c[nH]nc2C2CCCO2)=O)CCCN(CC2CC=CC2)C1 C1(NC(C2CCCC(C)(C)O2)=O)CC12CCC(NC(C1C3COCC13)=O)CC2 c1(CC)cccc(C)c1C(N1CC2CC2(NC(=O)C(C2CCCCCC2)F)C1)=O N1(C(c2cn[nH]c2)=O)CC(C2CC2C(N2CC(O)(C(F)(F)F)C2)=O)C1 c1(NC(c2cc(-c3ccccc3C3CC3)cnc2Cl)=O)cccc(F)c1[N+](=O)[O-] C1(O)(CNC(C2CCOC2)=O)CN(C(c2ccoc2Br)=O)C1 c1(C(=O)NC(C(=O)NC(CC#C)C(N)=O)CCC=C)cccc(C)c1C#N N1(C(c2c(C(C)C)noc2)=O)CCOCC(F)(CNC(c2cc(O)no2)=O)C1 C1(COC)(NC(c2cn(C)c(C)n2)=O)CCN(C(c2ccc(C)nc2C)=O)CC1 C1(NC(C(C)N(C)C(C2CC3(CCC3)C2)=O)=O)COC2(CCCC2)C1 Cc1nc(C)c(C(N2CC2c2cn(Cc3ncon3)nn2)=O)o1 N1(C(CSC(C)(C)C)=O)CCC2(CCC(NC(=O)CCc3cnc[nH]3)CC2)C1 C1(NC(=O)OCC)CCC(C(N2CCC(c3ncccn3)CC2)=O)CC1 c1(C(CN(C)Cc2ccc(NC(c3ccc(C)s3)=O)cc2)O)ccc(F)c(F)c1 C1(CC)C(C(N2CC=CC2)=O)CCN1C(C1CS(=O)C1)=O C(=O)(C#CC(C)(C)O)N1CC(CNC(C(C)(C)C2CCCCO2)=O)OCC1 CC(C)CC(C(=O)NC(C)CCCNC(C1COCC(C)(C)O1)=O)N(C)C Cc1ccc(C(=O)NCC2CCN(C(c3oc(Br)nc3C)=O)CC2C)cc1O C1(NC(CCCOCC)=O)CN(C(c2ccc(O)c(Cl)c2)=O)CCC1CO CCCCCCCNC(=O)C(C1CCC1)NC(=O)Cc1ccsc1C N1(C(C2=NOC(CNC(C(C)=C3CCC3)=O)C2)=O)CCC2(CC=CCO2)C1 C(C(C)(CC(C)C)NC(=O)CC1C=CS(=O)(=O)C1)NC(Cc1nc(C)sc1C)=O c1(C(N(C2CCN(C(=O)C(O)Cc3ccc(F)cc3)C2)C)=O)ncccc1N C(N=c1ccc(C(N2CC(C(=O)OC)CC2C)=O)c[nH]1)c1ccc(OCC)cc1 N1(C(C(C)N(C(CCC=O)=O)CCC)=O)CC2CCC(C1)N2C.OC N1(c2ccnc(COC)n2)CC(NC(C2CCSC2)=O)CC(C)C1 c1(N)ccc(Cl)c(F)c1.C1(C(=O)NC(C)CNC(=O)CC2CC2)CCCN1C1CC1 c1(C(=O)NCCOCCN(C(c2ccc(C)cc2C)=O)C)cc2occc2n1C C12(NC(c3c(C)nc(CO)s3)=O)CCCC1CN(C(c1[nH]ncc1C#N)=O)C2 C(N=c1cc(C(=O)N(CC(N2CCCC2)=O)C)nc[nH]1)c1cc(C)cc(C)c1.N(C)C N1(C(C2(CC)CC2(F)F)=O)CCCN(C(c2cnns2)=O)C(C)C1 CCCC(C)CC(=O)NC1C2CC3C1C3C2C(=O)NC1CCC(N(C)C)C1 c1(C(=O)OC)cccc2oc(NC(CNC(=O)CCOCC3CC3)CO)nc12 c1(C(=O)OC)cc2sc(C(=O)NC3CC(NC(=O)CSC(F)F)C3)cc2[nH]1 C1(CNC(C2(C=C)CCC2)=O)CC2CCC1N2C(=O)COCCc1ccc(Cl)s1 C1(C(=O)NC(C)CCCNC(=O)CSc2nncs2)CC2(C1)CC(F)(F)C2 c1(C(N(C2C(C)CCN(C(C3(OC)CCC3)=O)C2)C)=O)cc(C#N)c(N)cc1O CN1C2CCC1CC(=CC(=O)NCC(CC(F)(F)F)NC(=O)CC1CCCC1)C2 CC(C)(CNC(=O)C(c1ccccc1)NC(N)=O)CCNC(c1n[nH]cc1Cl)=O CCC(O)C(C)C(=O)NC1CC(CNC(=O)C(C)Cc2c(C)n[nH]c2C)C1 c1(OCCC)ccc(NCC(c2cccc(C)c2)F)cc1 C(C(CC(C)C)C(=O)N(C)CCOCCNC(=O)C(C)C(C)(F)F)OC c1(NC(=O)NCCC(=O)NC(C2(CO)CC2)C)cc(F)cc(F)c1 C(=O)(C(C)(C)CNC(C1CN(C(c2oc(C)cc2C)=O)CC1C)=O)NC C12(C(=O)NCCOC3CCN(C(C(C)CF)=O)C3)CCCCCC1OCC2 N1(C(Cc2ccc(CC)cc2)=O)CCC(C)C(CNC(=O)C(CC)OC)C1 N1(C(C23CC(NC(c4c(C)cc(CC)o4)=O)(C2)C3)=O)CC2(COC(C)C2)C1 N1(C(CCC(=C)C)=O)CCC(CNC(c2cc(Cl)cnc2C)=O)C(C)C1 S(=O)(=O)(c1ccccc1)NC(C(=O)NC1CC(CNC(C2(CC=C)CC2)=O)C1)C CCCCCC(=O)NC1(C(=O)NC2C(C)CCC2C)CC1(C)C C1(c2cn(CCCNC(=O)Cc3cnoc3)nn2)CCC2(CCCC2)C1 CC(F)(F)C(F)(F)CC(=O)NCC1COC(CNC(=O)Cn2cnc(=N)[nH]2)C1 C1(CC(=O)N(CCCNC(c2c(C)nsc2C)=O)CC)CC2(CCO1)CC2 c1(C(=O)NC(CN(C)CC)C)ccc(OC(F)(F)F)cc1C C1(N(C(C2CCN(CC)C2)=O)C)CCN(C(=O)CCn2cccc2)CC1 N1(C(c2c(CNC(c3ncc(NC)nc3)=O)nnn2C)=O)CCCC1C1CCCO1 C1(C(N2CCN(CCN(C(=O)COC(F)F)C)CC2)=O)CCC2(CCC2)OC1 c1(OC)cccc(CN(C)C(=O)NC(C2CCN(CCCF)CC2)C)c1 N1(C(CC(C)(C)OC)=O)CCC2CN(C(=O)Cc3c(C)cccc3C)CCC2C1 c1(C(=O)NCc2ccc(C(=O)NCC3C(C)COC3)o2)ccc(N)c(F)n1 C1(CNC(c2ccsn2)=O)CCCN(C(=O)CCCC2CCCC2)C1 C12CCN(CC1)C(=O)N1CCCC21.n1(CC)nccc1OCCOC1C=CCC1 C(C(C(=O)N1CCCOCC1C)C(C)(C)C)NC(c1c[nH]c(=NC)o1)=O C1(CNC(CC2CC(C)(C)C2)=O)CC2(CCOCC2)CN1C(=O)C(=O)C(F)(F)F C=CCCCC(C(=O)N(C)Cc1csnn1)NC(c1ccoc1)=O C1(C(=O)NCCC2(O)CN(C(C=CC(CC)C)=O)C2)CCn2c(C)nnc2C1 c1(C(N(CC(O)CNC(c2ccnn2C(F)F)=O)C)=O)ccc(CC(N)=O)cc1 C#CC1CC2CCC1N(C(c1cc(I)ccc1Cl)C(=O)Nc1cccc(C)c1)C2.SCC c1(C(=O)OC)nc(NC(=O)NCCCc2cccn2C)ccc1Cl c1(OC)c(C)csc1C(=O)NC1CC(CNC(c2cc(C3CC3)[nH]n2)=O)C1 C1(C(=O)NC(CN(C(C(c2ccc(OC)cc2)C)=O)C)C)CCC2CC1CO2 C1(NC(C2CC(C#C)(O)C2)=O)CCCC(C(=O)Nc2ccc(CO)c(C)c2)CC1 CP(C)(=O)c1cc(Br)ccc1C(=O)NC1CCOC(C2CC2)C1 N1(C(c2c(CC)cc[nH]2)=O)CCC12CC(C(=O)NOCC(C)(C)O)C2 C1(NC(CCn2cc(COCC)nn2)=O)CCC(S(C)(=O)=O)C1 N(C1CC(C)Oc2ccccc21)C(c1c2ccc(C)cc2sc1)c1nnnn1C C(C(C)(C(C)C)NC(=O)Cc1ccccc1Cl)NC(C12CC(C(=O)OC)(C1)C2)=O C1(CNC(C2CCC(C)O2)=O)CCC(CNC(=O)Cc2cnc[nH]2)CC1 N1(S(CCCC)(=O)=O)CCC2CC1(C(=O)NCc1cc(C(=O)OC)n(C)n1)C2 Cc1cc(C)cc(S(=O)(=O)N2CCC(NS(=O)(=O)CCBr)C(F)(F)C2)c1 c1(C(N(C)CC2CCCN(C(C(C(C)O)N(C)C)=O)C2)=O)cnn2ncccc12 CCCCC(F)C(=O)NC1CN(C(C2OCC2(C)C)=O)CCC1O c1(C(N2CC(C(C)(C)O)(CNC(C3OCC(C)C3)=O)C2)=O)ccc(F)c(F)c1 C1(CNC(C(C)OCC2CCCCO2)=O)CC(C)(C)CN1C(=O)C(F)=C1CCCC1 C1(NC(CCC(C)N(C)C)=O)CN(C(C2CCCOCC2)=O)CCC1C(F)(F)F CCC(C)CC(C(=O)NCCN(C1CC1)CC)NC(c1ccc(CC)cc1)=O C1(NC(CC=C(C)C)=O)CCCC(CNC(c2ncncc2Cl)=O)C1 C1(C(=O)NC(C)CNC(c2nc(C(C)(F)F)cs2)=O)CNC(=O)C(C)(C)C1 N1(CCC(=O)NC(CC(C)C)C)CCC(O)C(C(N2CC(O)C2)=O)C1 C1(C(C)C)CN(C(=O)C(O)Cc2cnc[nH]2)CCN1C(=O)C=Cc1ncc[nH]1 Nc1ccc(C(N2CCSCC2CCNC(C2(C(F)F)CCCCC2)=O)=O)nc1 CCS(=O)(=O)CC(=O)NC12COC(C1)C(NC(=O)C(CC=CCl)c1ccccc1)C2 N1(C(C(CSCC)NC(CN(C(COC)=O)C)=O)=O)CCNC(=O)C1C C(=O)(C1=CCN(C)C1)NC(C(=O)N(CCCC)CC)(C)C1CC1 CCCC(O)CC(=O)N1CCCC(C)(CNC(C23CCC(CC2F)C3)=O)C1 C1(NC(C(n2cc(C(c3cnn(C)c3I)C)nn2)C)=O)CCC(CO)CC1.C1CCC1 N1(C(c2c(C)noc2)=O)CC(CC(=O)N(C2CN(C)CC2O)C)CC1C CCC(C(=O)N1CC(NC(=O)CCc2cccc(OC)n2)CCC1C)C(C)O c1(CNCCc2nnc(C)s2)cc2scnc2[nH]1 C1(C(=O)NCC2C(C)C2)CN(C(=O)CCSCC(N)=O)CC1(C)C c1(C(N2CC3CC3C2)=O)cc(-c2cscn2)c2cn[nH]c2c1 N1(C(C(C)CN(C(=O)C(O)C2CCCC2)C)=O)CC2CN(C)CCC2C1 Cc1cc2[nH]c(C(=O)NC3(CO)CN(C(C4(C(F)F)CCCCC4)=O)C3)cc2o1 C=CCC(CC(=O)N1CCC1CN(C)C)NC(c1cn(C(C)C)cn1)=O O=C(C1=COCCO1)NC1CCC1CNC(C1(c2cccc(Br)c2)CC1)=O C1(C(N(CC(CC)NC(c2ccnc(C(C)(C)C)n2)=O)C)=O)CCCS1(=O)=O c1(OC)cc(NC(C2CC(C)CN2C(=O)CSc2cn[nH]c2)=O)cc(O)c1 c1(C2C(C(=O)N(C(C)(CNC(c3csc(Cl)n3)=O)C3CC3)CC)C2)cccc(Cl)c1 n1(CC)nc(C(N2CCCC2(C)CNC(=O)CC23CCC(CC2)C3)=O)cc1O C1(C)(C(N(C)Cc2ncc(C)o2)=O)CCCN(C(c2nccnc2N)=O)C1 CC(C)C(O)C(C)(C)C(=O)N1CC2CCC(C1)C2NC(C1CCC1C)=O C(=O)(CCCCC(C)(C)C)N1CC(NC(C(CC(C)C)N(C)C)=O)N(C)CC1 c1(C(=O)NCC2CN(Cc3ccccc3Cl)CCO2)ccc2nc(O)[nH]c2c1 c1(C(=O)Nc2c(C(=O)NCc3ccc(C)cn3)cccn2)ccc(O)c(C)c1 c1(C(=O)NC2C(C)CCN(C(C3(O)CCCCC3)=O)C2)ccc2ncnn2c1 C(C(C)(C)C(=O)NCCc1n[nH]cc1C(=O)Nc1cccc(Cl)c1)OC c1(NC(c2c3cccc(C)n3nc2)=O)ccc(Br)c2cccnc12 c1(NC(c2c(NC(C3(C)CC3)=O)nc(Cl)cc2)=O)cc(F)c(F)c(F)c1Br C1(CC(=O)NCC(CN(C(CCCC)=O)C)O)CCN(OC)CC1 C1(NC(C2N(C)CCOC2)=O)CN(C(c2csc(C#N)c2)=O)CC12CCC2 c1(OC)ccc2c(c1)CN(Cc1cncs1)C2.C1(=O)CCCCCO1 c1(C(=O)NCC2N(C(CN3CCC(C)C3)=O)CC(C)(C)C2)ncnc2ccsc12 Cn1cc(C(=O)NC2CC2CNC(=O)CC2CC(F)C2)c(=O)n(C)c1=O N1(C(c2cc(C(C)=O)on2)=O)CCC2(CCCC2CNC(c2cccs2)=O)CC1 Cc1nccc(C(=O)NC(C2CCCC2)CNC(c2nc(Cl)cs2)=O)c1C c1(C(N2CCC(C)(CNC(C3CCCCNC3=O)=O)C2)=O)cccc2nn[nH]c12 C1(CC(=O)NC(CC)COC)CCC(NC(C2COCCO2)=O)CC1 c1(C(=O)NC2(CC(=O)O)CCCCC2)ccc2[nH]ccc2n1 c1(C(N2C(CN(C(C3C(C=C)C3)=O)C)CCCC2)=O)cccc2c1OCC2 c1(C(N2CC(CCNC(CC(C=C)(C)C)=O)C(C)C2)=O)c[nH]c2nc(F)ccc12 C(=O)(C(CN(C)C)C(C)C)N1C(C(=O)NC(CC=CC)C(=O)NC)CCC1 N1(NC(=O)C(F)(F)C2CC2)CC(C(=O)NC2C(OCCOC)CCC2)CC1=O CC1CCC(Cl)=C(C(=O)N2CCC3CCN(C(c4ccc(CO)nc4)=O)C3C2)C1 C1(NC(c2cccnc2)=O)CC2CN(C(c3ccco3)=O)CC12 CC(C)C(C(=O)N1CC(C(=O)NC(c2ccnn2C)CO)C(F)C1)n1ccnc1 C1(NC(C2C(=C)CC2)=O)CC2(CCC(NC(c3ncccc3OC)=O)CC2)C1 C1(c2c(C(=O)OC)c[nH]n2)CCN(N2CC3(CCCN3CC3CCC3)C2)CC1 n1(CC(=C)C)nnnc1C(c1ccc(Cl)s1)NC1CC(C(C)C)C1 C1(CC(=O)NC)CCCCC1N=c1[nH]c(=NC2CN(C)C2)[nH]c2cc(C)ccc12 N1(C(C2(SC)CC2)=O)CCN(C(=O)C(S(C)(=O)=O)C2CC2)C(CCO)C1 CCC(C)(C)C(C)CC(=O)N1CCC(CO)(NC(c2cc(C)n(C(F)F)n2)=O)C1 Cc1cc(C)c(OCCC(=O)Nc2c(Cl)cccc2I)c(C)c1 N1(C(C(CSC)C)=O)CC2(CCC(NC(C3(C)CCC(C)C3)=O)CC2)C1 c1(C(=O)NC(C)CNC(=O)C2=C(Cl)CCC2)nn2ccccc2c1Br C1(CNC(c2n(CC=C)ccc2)=O)N(C(=O)CC(C)O)CCC1(C)C CC1CC(C(N2CC(O)(C(F)F)C2)=O)N(C(=O)CCCC2CCC2)C1 c1(N2CCC(C)C2)ccc(C(N2CCCC(C(=O)NC3CCCC3)C2)=O)c(F)c1 N#Cc1cnn2cc(C(=O)NC3CN(C(=O)C(F)F)C4CCCCC34)cnc12 Cc1cccc(C(C)NCC2(NC(c3ccc(S)cc3)=O)COC2)c1 c1(C(=O)NC2C(CNC(c3cc(C)oc3C)=O)C2)cnc(O)c(Cl)c1 c1(NC(=O)Cn2cc(-c3cc(CO)c(CO)cc3Br)nn2)cc(F)c(Cl)c(Cl)c1 CC1(C(=O)N)CCCCC1.C1(C(=O)NOCCCF)CCCC1 CCC(CC(C)O)N=c1[nH]c(N(C)CC2CC(F)(F)C2)nc2ncn(C)c12 C12(C(N3CCC(C)(CO)CC3)=O)CCCC1CCN2C(=O)C=Cc1cnccn1 N1(Cc2c(C)ccc(SC)c2)CCC(c2ccccc2)C(c2ccccc2)C1 CC#CC1CCN(C(C2CC23CCN(C(=O)C(n2ccnc2C)C)C3)=O)C1 CC1(C)CN(C(C2CCCN2C2CC2)=O)CC1NC(C1CC2C=CC1O2)=O C1(N(C)C(C2CC3CCC(C2)O3)=O)CN(C(=O)COCCF)CC1N=[N+]=[N-] c1(CC(=O)NC2CC23CCN(C(=O)C(F)C(F)(F)F)C3)cccc2occc12 C1(O)(CC(=O)NC2CC(CNC(C3CC(C(N)=O)C3)=O)C2)CCCOC1 c1(C(N2CCC(NC(=O)CC3CCCC3)(CF)C2)=O)cccc(F)c1Cl Cc1nc2c(s1)CCCC2C(=O)NCC1CN(C(=O)C(C)O)CCC12CCC2 C(C(C(C)C(C)C)NC(=O)C=C1CCC1)NC(C(=Cc1ccncc1)C)=O C1(C(=O)NC(C)(CNC(=O)CCc2ccc(Cl)cc2)CO)CCOCC12CCC2 c12ccccc1CN(N1CCCC1)C(C1CC1)C(=O)N2.C(C)(C)(C)OCCN(C)C N1(C(C=CCCC)=O)CC(CNC(C2(C)CCNC(=O)C2)=O)CC(C)(C)C1 Cc1ccc2c(c1)C(C(=O)NCCCNC(c1ncn3c1COCC3)=O)OCC2 c1(C(N2CC3C(N(C(c4nc(COC)oc4)=O)C)C3C2)=O)cnc(Cl)cc1N c1(CN=C(NC(C#C)C)NCC)cc2ccccc2nc1O.C12CC(C1)OC2 C1(C(=O)NCCN(C(C(C=C)(F)F)=O)Cc2ccccc2)(CF)CCC(F)(F)CC1 C1(NC(C23C(CN(C(=O)CC4(N(C)C)CCC4)C2)C3)=O)CC2(CNC(=O)O2)C1 CC(C)CCCCCC(=O)N1C(C(=O)N(C)Cc2cn(C)nn2)CCC12CC2 Cc1cnccc1C(=O)N(CCCOCCN(C)C(c1ccncc1O)=O)C c1(OC)ccc(NC(=O)NCC2(C)CCCC2NC(=O)OC(C)(C)C)nn1 C12(C(=O)NC3(C4CN(C(CN(C(C)=O)C)=O)C4)CC3)OCCCC1C2(F)F CC1CCN(C(C2CC(C)(C)CO2)=O)CCN1C(C12CCCN(CC1)C2)=O N1(C(c2cc(Br)ccc2O)=O)C2CCC1CN(S(=O)(=O)CCCl)CC2 c1(C(N2CC3CCN(C(C4CCCO4)=O)CC3C2)=O)ccccc1C#CC1CC1 N1(C(C=CC=CC)=O)CC2CCC2(CCNC(=O)C#CC(C)(C)O)C1 C(C(CNC(=O)CCC=C(C)C)C(F)(F)F)NC(C(C(=O)OCC)C1CCC1)=O C1(CNC(C(C)n2cnnn2)=O)CN(C(C2OCCC2C(F)(F)F)=O)CCCO1 C(=O)(C1=NNC(=O)CC1)NCC1CC(NC(c2ccc(C)[nH]2)=O)C1 c1(C(=O)NCC(C)CNC(c2nccc(C(F)F)n2)=O)cnn2cc[nH]c(=O)c12 C1(NC(C(COC)O)=O)CN(C(C2CCS(=O)(=O)N2)=O)CC1(C)C C1(NC(=O)C2CC2)COC2CN(C(c3cc(F)cs3)=O)CC12.C(CN)O c1(OCC)cc(C(=O)NCC(CNC(=O)CCc2cccnc2F)CO)ccn1 c1(C(=O)NC2(CNC(C(c3n(C)ncc3)O)=O)CC2)cc2cc(F)cc(F)c2[nH]1 c1(C(=O)NC(CNC(=O)CCC2CC2)C2CC2)cnnn1-c1ccccc1 C1(NC(CC(CC)CN(C)C)=O)CCC2CCN(C(=O)CC(C)C(C)C)C1C2 c1(CNC(=O)NC(c2ccc(Br)cc2)CCc2ccccc2)ccc(I)cc1 N1(C(CCn2cc(C3CCOC(C)C3)nn2)=O)CCC(n2cccn2)(CC2CC(O)CN2)CC1 C1(NC(Cc2nc(C)[nH]n2)=O)CN(C(=O)Cn2cc(C)cn2)C2CCCC12 C1(O)(C(C)C)CCN(C(c2cc(C3CCCC3)[nH]n2)C(=O)NCCC2(C)CC2)C1 C1(CNC(COCC(=C)C)=O)CN(C(c2cc(C)nc(C)n2)=O)CC1(F)F N1(C(C(C)Sc2ccccn2)=O)CCC2CN(C(C3CCC3(F)F)=O)CC2C1 Cc1cccc(C)c1CC(=O)NC1C2CCN(C(=O)CNc3cnn(C)c3)C12 c1(CCC)ccccc1NC(C1CCN(C(=O)C(c2cccn2C)=O)C1)=O c1(C(=O)NC(CC)(CNC(C2CC2(C)CC)=O)CC)ccc2c(c1)COCC2 C1(C(=O)NCCCn2cc(-c3cccc(C(=O)OC)n3)nn2)CC1C1CCCC1 c1(C(N(CC(CNC(c2cc(CCC)n(C)n2)=O)O)C)=O)cc(C)cc(C)n1 c1(C(C)(C)C)cc(N)ccc1C(=O)NC1CCCCC1NC(c1ccc(Cl)o1)=O c1(C(=O)NC2C(NC(=O)C=Cc3cccc(CO)c3)C2)cc2cc(F)ccc2s1 C12(C(N3CCN(C(=O)CC4(CSC)CC4)CC3)=O)CCCCC1CS(=O)(=O)C2 N1(C(CCCNC(=O)NCC#C)=O)CCC(NC(C2CS(=O)(=O)C2)=O)CC(O)C1 C1(NC(=O)CC2CCCO2)CCCCC1N(C(=O)CCc1cncnc1)CCO N1(C(C=CCN(C)CC)=O)CCCC(C)C1CCNC(c1cccc(CC)n1)=O C=C(C)C1CN(C(c2cccc(CNC(=O)CCc3cccs3)n2)=O)CCO1 N1(C(CCN(CCC)C)=O)CCOC(CNC(=O)CCc2cnn(C)n2)C1 c1(CCCC(=O)OC2C(COc3ccc(CC)cn3)C3CCN23)ccccc1F CC(CCCCNC(c1ccc(C2(C)CC2)cc1)=O)NC(C1CC1CF)=O C1(NC(CCSCCCC)=O)CCCN(C(=O)C(n2cc(C)cn2)C)CC1 CC1=CCC(C)(C(N2CC(CNC(c3ccnc(N4CCCC4)c3)=O)C2)=O)CC1 c1(CNC(C(C)(C)C)CC(F)(F)F)cc([N+](=O)[O-])cc2c1OCOC2 N1(C(CC(CC)O)=O)CCC2(CC1)CCN(CCNC(c1ccccc1C)=O)CC2 N1(C(C2(C)CCCO2)=O)CCOCC(C(=O)NC2CCCC2CF)C1 C1(C2CCCOC2)(NC(C2(C(C)C)N(C(C3(OC)CCC(C)C3)=O)CC2)=O)CC1 C(CCS(C)(=O)=O)(C(=O)Nc1cn(CC(c2ccc(S(C)=O)cc2)O)nn1)NC N1(C(C(CC(C)C)CNC(=O)CC2CCC(O)C2)=O)CC2C(=O)NC(=O)C2C1 c1(C(=O)NCCCCC(C)NC(=O)C(F)=C2CCCC2)cc(Cl)c(F)cc1N C(=O)(C1Cc2ccc(F)cc21)NCC1(C)CCN(C(=O)CC2CC=CC2)C1 N1(C(C(CSC)O)=O)CCC(CNC(c2cccc3cncn23)=O)C(F)(F)CC1 CN1CCN(C(C2CCCC3(CC3)C2)=O)CC1CNC(=O)CCS(N)(=O)=O N1(CCC(=O)NC(C(C)C)CNC(C2(C(F)F)CCCO2)=O)C(C)CCCC1C Cc1nn(C)cc1C(=O)NCC1(C(=O)NCCN2CC(OC)CC2)CC12CCC2 c1(C(=O)OCCN(C(=O)Cn2nccc2C)CCC)cc(OC(C)C)cc(Br)c1 NC1(C(N2CC=CC(c3ccccc3)C2)=O)CCS(=O)(=O)C1 N1(C(C=CC=CCC)=O)CCC(COC(N2CCOCC2CCO)=O)CC1 c1(C(=O)NCC2CC(C)N(C(=O)Cc3ccco3)C2)ccc2cnnn2c1 c1(OC)csc(C(N2CC(=C(CNC(C(C3CC(SC)C3)F)=O)F)C2)=O)c1 CCCC(CCCNC(c1cc2scnc2[nH]1)=O)NC(=O)Cc1ccoc1C C1(C(=O)NC(C(CO)NC(c2c(C)ccc(O)c2)=O)C)CCOCC1(C)C c1(C(=O)NC(CNC(C2(C)CC(=C)C2)=O)CCOC)ccccc1OCCF C1(NC(C2=NOC(C)C2)=O)CC12CCC(NC(=O)Cc1ccsc1)CC2 c1(CC)c(NC(=O)CC(O)CCn2cc(C3CN(C(C)=O)C3)nn2)cnn1CC Cc1cc(C(N2CCC(CC(C)NC(c3ccoc3)=O)CC2)=O)c[nH]c1=N N1(C(Cc2c(C)occ2)=O)CCC2(CC1)CN(C(C1CCCC1F)=O)C2 N1(C(c2c(OC)cccc2)C(=O)Nc2ccccc2)CCCC(C2CNC(=O)C2)C1 N1(CC2(N(N(C)CCO)C(C3(C)CCC3)=O)CC2)CCN(C(C2CCCO2)=O)CC1 C1(C)(NC(c2c(C)noc2C(C)C)=O)CCCN(C(c2cnc(C3CC3)nc2)=O)C1 N1(C(C(CO)NC(CCCCNC(C)=O)=O)=O)C(C)CC2CCCC12 c1(NC(C(n2ncc(C)c2)C)=O)cccc(N2CCN(C(=O)CN(C)C)CC2)c1 C1(NC(c2cc(CCC)nc(O)c2)=O)CCN(C)C12CCCN(C(=O)CO)C2 C1(CNC(CSCC#C)=O)CCC2(CCN(C(c3cn(C)nc3O)=O)CC2)CO1 c1(COCC)nc(C)c(C(N2CC3C(NC(c4cnc(C(C)C)[nH]4)=O)C3C2)=O)s1 C1(NC(N2CCC(n3cccn3)C2)=O)CC(C(F)(F)F)CC(C(F)(F)F)C1 c1(CCC(=O)NCC(C(C)C)NC(c2nnc(C)s2)=O)n[nH]c2ccccc12 CCC(C)(C(=O)OCc1conc1C)NC(=O)NCc1ccc(F)cc1 C1(NC(CCN(CCCCC)CCC)=O)CCC12CN(C(=O)C#CC(C)C)C2 N1(C(CCN(C(=O)C(C)(F)F)C(C)C)=O)CCC(O)C(C)C1 C12(C(=O)NCCC3(O)CN(C(CC4CCCC(C)C4)=O)C3)CC3CC1C2C3O C(CN=c1nn[nH]n1-c1ccccc1)N(C(C(C)OCCC(C)C)=O)C1CC1 c1(OC)cc(N)c(Cl)cc1C(N1CCC(OCCNC(C2CC(OC)C2)=O)C1)=O Cc1ccsc1-c1cn(C2COCC2NC(=O)C=CCO)nn1 CC1CCN(C(=O)CC2(O)CCCOC2)C(C(=O)NCC2CCCCN(C)C2)C1 c1(C(=O)NC2CC(NC(=O)COCC(F)(F)F)C2)cc(F)c(Cl)cc1Cl CC1C(F)(F)CCN1C(C1CN(C)CCN1C(=O)CCCCC#N)=O c1(C(=O)NC)cccc(CCC(=O)N2CCC2CNC=O)c1.c12coc(c1)C2.NC c1(C(N(C)CC2CCCN(C(C=CSC)=O)C2)=O)cc(N)ccc1Cl C(=O)(C(C(C)C)Nc1sc(=O)n(C)c1N)Nc1scc(C(C)C)n1 C1(NC(C(c2cn(C)nn2)NC(CCCOCC)=O)=O)CCN(C2CC2)C1=O c1(C(N2CCC(N(C(C3C(CCC)C3)=O)CC3CC3)C2)=O)ncncc1Cl N1(C(c2cnc(C#N)s2)=O)Cc2ccccc2C(CNC(=O)C=CCF)C1 N1(C(C2CC(SC)C2)=O)CC2CC(NC(=O)CCCCN3CCOCC3)CC2C1 CCC(F)(F)C(C)(C)NC(=O)C(CC(N)=O)NC(=O)CCCOC(C)(C)C c1(OC)cc(C(=O)N(CC(C)NC(=O)C2=CCC(C)CC2)C)cc(N)c1N c1(C(N(C(C)CNC(=O)Cc2csc(S)n2)C)=O)ccc(F)c(CO)c1 C(CCCC(=O)N1CCC(CC(F)(F)F)C1)n1cc(CCN(C(C)(C)C)C)nn1 c1(C(=O)NCC(CN(C(Cc2c(C)nc(C)s2)=O)C)O)noc2ccc(Cl)cc12 C1(C(N(C)CC2CCCCN2C(C2CC(F)(CO)C2)=O)=O)CC(C)(C)CN1C C1(O)(CNC(c2cnc(CC(C)(C)C)s2)=O)CCN(C(=O)COCCN(C)C)C1 C1(C(=O)NCCNC(C(C)(C)C2CC2C(F)(F)F)=O)CCS(=O)(=O)C12CCC2 c1(CC(N2CCC(C)(CC(=O)N(CCCCCC)C)C2)=O)cc(F)ccc1C n1(CCC(=O)NCC(CC(C)C)NC(=O)CC2CC2C)ccc2ccccc12 N1(C(c2c(C)cnn2C)=O)CCCC2(NC(C3CC4COCC4C3)=O)CC2C1 C1(C(N(C(CCCC)C)C)=O)CN(C(=O)CC(O)C(C)CC)CCC1(C)C c1(C(C)N(C)C(C2(F)CC2)=O)ccc(Cl)cc1 C(=O)(CCC(O)C(C)(C)C)N1CC(c2cn(CCC=C)nn2)(C)C1 C1(CC(N2CCN(CCSc3n(C=C)ncc3)CC2=O)=O)CSC2CCCC2N1 c1(C(C)=O)cc(C(N2CCC(N(CC(C)C)C(C3CC=CC3)=O)C2)=O)n[nH]1 C1(COC)CC(CSC2(N3CCCC3)CCC2)C12CCC2 Cc1cc(NC2CCC3CN(C(=O)OC(C)(C)C)CC3C2)cn2ccnc12 C1(C)(C(=O)NCC2N(C(C3CCN(C)C3)=O)CCC2)CCC2CC2C1 C1(C(=O)N(c2ccc(F)c(Cl)c2)CC(F)(F)F)CC2(CCCCO2)C1 C1(NC(CC=C)=O)CC2CC1N(C(c1c(OC)cccc1COC)=O)C2 CCC(CCOC)C(=O)N1CCCCCC1C(=O)NC(c1[nH]c(C)nc1C)C c1(C(N2C(C3(NC(C=C(COC)C)=O)CC3)CCC2)=O)cccnc1C(N)=O N1(C(C2=CCC(C)CC2)=O)CC2CC(NC(=O)C3=CS(=O)(=O)CCC3)CC(C2)C1 N1(C(C2(F)CCN(C(C3(CC)CCCC3)=O)C2)=O)CCC12CCN(C)C2 C(=O)(CCCC(F)(F)CO)N1CC2(CCN(C(C3(CC=C)CCCC3)=O)C2)C1 Cc1ccc(NC(C2(C(C)C)CC2)=O)nc1Cl.c12nc(Cl)ccc1C(=O)N2 CCCCC(CC(=O)NC1CCC(C2CC2)C1)NC(=O)CCCC1CCC1 N1(C(CN(CCC)C)=O)CCCC(O)(CNC(=O)C(C)(C)CC2CC2)CC1 N1(C(C(CC=C)NC(C)=O)=O)CC2(CCC2NC(c2cc(OC)ccc2F)=O)C1 C(C1(CO)CCc2ccccc21)NC(C(C)(C)S(C)(=O)=O)=O c1(OC)ccc(C(=O)NC2CC2NC(=O)C(=Cc2c[nH]cn2)F)cc1Cl c1(C(=O)NC(C)CNC(C2CC(N(C)C)C2)=O)ccc(CO)c(F)c1 N1(C(CC(C)CC2CC2)=O)CC(NC(c2ccc(N(C)C)nc2)=O)C(C)(C)C1 c1(C(=O)NC(CC)C(F)(F)F)ccc(NC(c2occc2C)=O)c(C)c1 N1(C(c2ccc(CC)cc2)=O)CCC(CO)(CNC(=O)Cc2cn[nH]c2)CC1 CCCCCCCCCC(=O)NC1CCN(C(C23COCC2C3)=O)CC1F Cc1cc(Cl)cc(C(=O)NC(CO)C(C)NC(=O)C=Cc2cccnn2)c1O c1(C(N2CC3C(CNC(C4C(C)(C)NC(=O)C4)=O)(C3)C2)=O)cnc2cccnn12 N1(C(C(C=CC)O)=O)CC(OC)CC(NC(c2ccc(C3CC3)cc2C)=O)C1 N1(C(C2C(CC)CCN2C(c2sc(F)cc2C)=O)=O)CCCN2CCCC2C1 N1(C(C(c2cn(C)nc2)(F)F)=O)CCC(NC(=O)C=CC=C(Cl)Cl)C(CO)CC1 N1(C(=O)OCC)CCC2(CC1)CC2(C)C(=O)NCc1ccc(OC(F)F)cc1 C1(NC(C2=CCC(C)CC2)=O)CN(C(c2cnn(C)c2)=O)CCC12CCOCC2 C1(C(=O)NC(C)CCNC(c2cn(C)nc2Br)=O)CCCC2CCCCC12 c1(C(=O)NCC2CN(C(C(C)N3CCC3)=O)C2)cn(CC2CCCC2)nn1 N1(C(CC2(C=C)CN(C(=O)CCCCOC)C2)=O)CCC(O)CC1CC CC(C)(C)CCC(F)C(=O)NC(CNC(C1(C#N)CCCC1)=O)C1CC1 Cc1nnc(-c2ccsc2C(=O)NCC2CCCN2C(C2CNC(=O)N2)=O)n1C c1(C(N2CCC(C#N)C2)=O)noc2c1CN(C(=O)C(N)CN)CC2 c1(OCC(=O)NCC(C2CC2)NC(c2cnc(SC)s2)=O)cccc(F)c1 c1(NCC)cncc(C(=O)NCC2(O)CCN(C(=O)COC3CC=CC3)C2)n1 CCC(C)CC(C(=O)N(C)Cc1nc(=O)o[nH]1)NC(=O)C(O)CSC c1(C(=O)O)ccc(S(=O)(=O)N2CCC(c3cccc4ccccc34)CC2)cc1 N1(C(C(N2CCCC(F)(CO)C2)=O)=O)CCOc2c(C(F)(F)F)cccc2C1 C1(CN(C(=O)C=CC(C)(C)NC(=O)C=Cc2ccoc2)C)CCCC(C)(C)C1 Cc1ccc(F)c(C(=O)NC2CCCC2CNC(c2nc(C)c(C)[nH]2)=O)c1 CCC(C)C(C(=O)NCC1CC(O)C(O)C1)N(C)C(c1cc(O)nc(O)n1)=O N1(C(c2cc(C)c(Br)o2)=O)CCCC2(C1)CN(C(C1CCCN1C1CC1)=O)C2 N(C1COc2ccccc21)C(C(CCN(C)C)NC(C12CC1CNC2=O)=O)=O C#CCCCCCC(=O)NC1CCN(C(c2cnn(C(C)(C)C)c2C)=O)C(C)C1 c1(C(=O)OC)cccc(C(=O)NC2CCCC2NC(=O)CSc2ccccn2)n1 CC1CCN(C(C2(CO)CCCC2)=O)CC1NC(=O)COCc1nc[nH]n1 C1(C(N2CC(NC(C(CC)CC)=O)C(O)C2)=O)CCC2CC1CO2.C(C)(=O)O c1(NC(=O)CO)ccccc1C.C1(COCC(=O)NC2CC(OCC)C2)CCCOC1 c1(C(N(C2CCN(C(c3cc(C(F)F)nn3C)=O)CC2)CC)=O)ncccc1Cl C(=O)(CCC1CCc2ccccc21)NC(C)CCNC(C1CCC(=O)N(C)C1)=O C(=O)(CC(C)(C)C(C)=O)N1CCC(=CCNC(c2c(CC)[nH]cc2)=O)CC1 Cc1nn(C(F)F)c(C)c1S(=O)(=O)N1CCCC1C1(S(=O)(=O)N(C)C)CC1 C(=O)(C(C(F)(F)F)C(F)(F)F)NCCN(C(C1CC(CCC)OCC1)=O)CC C(=O)(C(CCOCCO)NC(c1nccnc1N)=O)NC(C(=O)OCC)C C=CC(F)(F)C(=O)N(CCCCN(C(=O)C(C)(C)OCC=C)C)C C1(CNC(c2n(C(C)C)nnc2)=O)CCCCN(C(c2ns[nH]c2=O)=O)C1 CC(C)CC(C(=O)NCCCS(C)=O)OCc1nccs1 c1(CC)nccnc1C(=O)NCC(F)(F)Cn1cc(COC(C)C)nn1 N1(C(C(C2CC2)OC)=O)CCCC12CCN(C(C1(C)CS(=O)(=O)C1)=O)C2 c1(C(c2n(CC=C)nnn2)NCC2CCOC2)ccc(SCC2(CF)CCC2)cc1 C(=O)(C(C(=O)NOCCCO)OCC(N1CC(CO)CC1CO)=O)OCC Cc1nc2c([nH]1)CC(C(N1CCC3(CCC3NC(=O)CC(C)(C)O)CC1)=O)CC2 Cc1cc(-n2cc(CNC(c3cccc(OCCC(C)C)c3)=O)nn2)ccc1F C(=O)(C1=COCCC1)N(CCCN(C(c1ccc(-n2ccc(C)n2)cc1)=O)C)C C1(CNC(C(COC)OC)=O)CN(C(c2ccc3c(c2)CC3)=O)CC12CC2 c1(CNC(N2C(c3cn(C)nc3)C(C)(C)C2)=O)ccc(F)c2[nH]ncc12 c1(CCC)cc(C(=O)NCC2CCCN2C(=O)C(N2CCOC2=O)C)no1 CN1CCCC(CC(C(=O)O)NC(=O)CC(O)N(C)C(=O)OC(C)(C)C)C1 N1(N2C(CN=c3scc(-c4c(OC)ccs4)[nH]3)CCC2)CCc2sccc2C1 N1(C(CC2C(NC(=O)CC3CCCC3)CC2O)=O)CCCC2(CCOC2)C1 c1(OC)ccc(C(F)(F)C(=O)NC(C)C(CO)NC(c2ccn(C)n2)=O)nc1 C(=O)(CC(C)CC(C)C)N1C(C)(COC)CC(NC(=O)CC2CC(C)(C)CO2)C1 C1(c2nc(COC)[nH]n2)CCCN(CC(c2cccc(Cl)c2)c2ccccc2)C1 c1(N(C2CN(C(c3coc(S(N)(=O)=O)c3)=O)C2)C)ncc2c(n1)CCCCC2 c1(C(C(=O)NC(CNC(C(=CC=C(Cl)Cl)C)=O)C(C)C)=O)ccc(F)c(F)c1 C(N=c1[nH]c(N2C3CCC2CC(=O)NC3)nc2c1SCC2)c1c(C)cn(C)n1 CC(C)C(O)C(c1cccs1)NCCCc1cncn1C CC1(C)CCCC(C(=O)NC2CC(NC(c3cccc(-c4cscn4)c3)=O)C2)C1 C1(C(=O)NCC(CNC(CCOCCCOC)=O)OC)CCCC(CF)C1 C1(NC(COCC(C)C)=O)CN(C(=O)CC2CCC(=O)N2C)CC2(CCC2)C1 C12(NC(C(C)NC(=O)NC)=O)CC(C1)N(C(=O)Cn1ncccc1=O)C2 C1(COC)(NC(C2CCCS2)=O)CCN(C(c2c[nH]c(=N)cc2C)=O)CC1 c1(OC)nc(N2CC(NC(=O)CCCN(C)C)CC(C)C2)ncc1F Cc1cccc(OC2CC2C(N2CC(C(=O)NCCO)C2)=O)c1.c12cccc(c1)O2 O=C1COc2c(C(=O)NCc3csc(CNC(c4ccno4)=O)n3)cccc2N1 c1(C(N2CCN(C(C(C(C)O)(F)F)=O)CC2)=O)cc(S(C)(=O)=O)cnc1O C=CCCCCCC(=O)NCCC1CCN(C(=O)COc2cn[nH]c2)C1 C(=O)(CCCCCCC(=O)NCC(C)NC(c1cscn1)=O)OC C1(C(=O)NC2CN(C(C34OCC(C)(C3)C4)=O)C2)CC(c2cccc(Cl)c2F)=NO1 N1(C(c2c(C)cc(C)o2)=O)CCN(C(=O)C(O)C2CC2)CC1c1cccc(F)c1 C(CCC(C)CC(=O)N(C1CCC(NC(=O)C2=CS(=O)CCC2)CC1)C)=C(C)C N1(C(=O)OC(C)(C)C)CC(C(=O)Oc2cccc(Cl)c2I)CCCC1C CCCC(C)(C)C(=O)NCCC1CC(F)(F)CN1C(c1ccc(Br)o1)=O CC(C)(C#CC(=O)NC1CN(C(N)=O)C1)CNC(C1CCCC1C1CC1)=O C1(C(=O)NCCCOC)CN(C(c2ccn(C)c2)=O)C2(CCC2)C1 C=CCC(CC=C)C(=O)N1CC(O)(CCNC(c2c[nH]cc2CC)=O)C1 c1(C(N2CC(CC=C)(C(=O)Nc3cnncc3O)C2)=O)cc(C)n(CC)n1 N1(C(CSc2ccc(C)cc2)=O)CCOCC(CNC(c2cn[nH]c2)=O)C1 c1(CCNC(=O)C(c2ccc(F)cc2)C2CC2)cc(Br)c(Cl)cc1[N+](=O)[O-] c1(OC)cccc(O)c1C(N1CCC(CNC(C2CCC(=O)N2C)=O)C1)=O C=CCC(CC(=O)NC(C)CCCCC)NC(c1cccc(F)c1F)=O C(=O)(C(CO)N(C)C(C)=O)NC(C)(C)C.C(=O)(CCNC(=O)C(C1CC1)S)NCC(C)C c1(C(N2C3(CNC(C(C)OCCCC)=O)CC(C2)C3)=O)cccc(C)c1CC C1(C(=O)OCCOCC(=O)OCC)(CO)CCCCC1.OCC C=CC(C)(C)CC(=O)NC(CNC(=O)CCC(=O)N(C)C)C(C)C(C)C C1(C(N2CCC(NC(c3c(SCC)cccc3)=O)C2)=O)CCc2ccccc2N1 C(=O)(CC(O)CN(C)C)NC(CNC(CC1CC(=C)C1)=O)C(C)C C1(C(N(C2CC(NC(=O)C(F)=CC3CC3)C2)C)=O)CC12CCCOC2 N1(C(c2scc(OC)c2)=O)C(C)CN(C(c2nn(C)c3c2CCC3)=O)CC1C C1(CC(=O)NCC(CC)NC(c2cnc(C)s2)=O)Cc2cc(F)ccc2O1 CCC(CC)CC(=O)NCC1CC(NC(c2cnn(CCO)c2N)=O)C1 C(=O)(CCCC(F)(F)F)NCC(CC)NC(=O)C(n1nccc1C)C C1(CC(=O)NC(CC(C)NC(c2cnc(C(C)C)[nH]2)=O)C)CCN(C)CC1 CCCCCCC(C)C(=O)N1CCOC(C(C)NC(c2cc(C)cnc2F)=O)C1 c1(-c2onc(C)n2)cccc2cccc(NC(=O)NC(CCN(C)C)C(C)C)c12 c1(CC)cc(C(=O)NCC(CNC(=O)C(C(C)C)NS(C)(=O)=O)CO)cc(Cl)c1 c1(OC)cc(C(=O)NC(C2CCCCN2C(=O)Cc2ccno2)C)c(Cl)cc1Cl C1(NC(C(F)OC)=O)CN(C(C2CCCN(C(=O)C3CC3)C2)=O)CCC1C c1(C(=O)NC2CC(OC)CN(C(C3(NC(N)=O)CC3)=O)C2)nc2cnccc2s1 N1(C(C2(C=C)CCC2)=O)CC(C2CN(C(=O)Cc3c[nH]nc3O)C2)C1 CC(CCCCNC(=O)CN(C)C)NC(=O)CCCN(C)C CCCCCS(=O)(=O)CC(=O)N(CC(C)N(C(=O)COCCOC)C)C c1(C(=O)NCC(CC)NC(=O)C(CC)CCOC)cc2c(cc1N)CCC2 C=CCCCCC(=O)NC12CCN(C(c3cc(Cl)ccc3Br)=O)CC1C2 N1(C(c2c(CC)nco2)=O)CCN(CCCNC(C2(c3cccs3)CC2)=O)CC1 C(=O)(C#CC1CCCCO1)NCCN(C)C(C1(C)C(C)(C)C1(C)C)=O C1(CCNC(=O)NCC(COC)OC)CCCC1C Cc1ccnnc1C(=O)NCC1COC(CNC(=O)CC2CC3(CC3)C2)C1 CC(C)(O)C(F)CNC(C1C=CCN(C(C2CC(N(C)C)C2)=O)C1)=O C1(N(C(C(CC)SC)=O)C)CC2CC1N(C(=O)Cc1cccnc1OC(F)F)C2 C1(C(N(CC2=CCSC2)C)=O)CCN(C(=O)C(C)(C)C2CCOC2)O1 c1(C(C)C)cccc(C(=O)NCCNC(C2CC2(C)C)=O)c1 c1(C(=O)NC2CN(C(c3c(C)nc(C)[nH]3)=O)CC23CC3)cc([N+](=O)[O-])ccc1N c1(C(=O)NC2CC3CN(C(CN(C(COC)=O)C)=O)CC32)cccc2[nH]ccc12 Cc1ccc2cc(Nc3cccc(S(=O)(=O)N(C)C)c3)ccc2c1 N1(C(C2(CC)COC2)=O)CCC(C)(CCNC(=O)C(C)Oc2ccc(Cl)cc2)C1 c1(CC)nc(C)c(C(=O)NCC(C)C(C)(C)C)o1.C12(O)CC(C1)C(=O)NC2 c1(C(N(C(C)CNC(=O)CCCCC#N)CC)=O)cnc2[nH]nnc2c1 C(CCCCCNC(C1(C(=O)N(C)C)CC1)=O)NC(C(C1CCOCC1)C)=O C1(NC(c2cc(C)cc(C)c2)=O)COC2(C1)CN(C(C1CC(C3CC3)=NO1)=O)C2 C1(n2cc(C3(NC4CC(SC)C4)CCCOC3)nn2)CC2CCCC2C1 CC(CCCCNC(=O)C(C1(C)CC1(Cl)Cl)C)NC(=O)CCC1CCCOC1 CCC(C(=O)NCC(N1CCOCC1)=O)NC(C)=O.C1(Cc2ccccc2)C(=O)N1 c1(Cc2cn(C(C(C)C)Cc3nccn3C)nn2)cc(Cl)cc(Br)c1 c1(NCCCC(C)(C)F)nc2ccccc2nc1NC1CC1 C1(CNC(c2cc(CC)no2)=O)CCN(C(c2ncc(Cl)cc2O)=O)CC1(F)F c1(OC)c(C=CC(=O)NC2CC(CNC(c3cn(C)c(O)n3)=O)C2)cnn1C N1(C(CCC=C(C)C)=O)CCN(C(C#N)C(N)=O)CC1.C1CC(=O)OCCO1.C(=O)C c1(C(=O)OC)cc(C)nc(NC2CCCC(NC(c3cnccc3OC)=O)C2)n1 C(=O)(C#CC1CCC1)N1CC2C(NC(c3cn(CC(CC)O)nn3)=O)(C2)C1 n1(CC(N2CCCC(CNC(C3(COC)CC3)=O)C2)=O)ccc2ccc(F)cc12 C1(NC(C2(C)CCN(Cc3cccc(Br)c3)C2)=O)CCCCC1(F)F Cc1nccc(C(=O)NC(C2CCCN2C(C2(C)CSC2)=O)C)c1C c1(C(N2CC=CC(NC(CC(CC)C)=O)C2)=O)ccc(C2CC2)cc1F CN1CC(C(N2CC(CO)(NC(c3scnc3Br)=O)C2)=O)CC1=O N1(C(C(CC=C)NC(C)=O)=O)CC2CN(C(=O)Cc3cc(Cl)n(C)n3)CCC12 c1(CN(CCNC(=O)Cn2nccn2)C(c2cc[n+]([O-])cc2)=O)cccc(Cl)c1 N1(C(C(C)(F)F)=O)CCCC(C)(NC(=O)CC2CC(Cc3ccccc3)C2)C1 CC(C)C(C(=O)NCCCC1CC1C)NC(C1CCN(C)C1=O)=O c1(C(N2CC(COC)(CNC(C3CC3F)=O)C2)=O)cccc(NC(C)=O)n1 c1(C(N2C(CNC(CCNS(CC)(=O)=O)=O)CC2)=O)cccnc1C(F)F C=CCCCCC(=O)NCC1(O)CCN(C(c2ccc(O)cc2Cl)=O)C1 Cn1c(O)nc2c(C(=O)NCCCNC(=O)Cc3cncn3C3CC3)cccc12 Cc1ccccc1C#CCNCC12CCOCC1CNC2 N1(C(c2ccc(Cl)c(Cl)c2)C(=O)NC2CCCC2)CCN2CCOCC2C1 c1(OC)cc(C(=O)NCCN(C(c2snnc2C)=O)C2CC2)cc(F)c1 C1(NC(C(COC)N(C)C)=O)CCC2(CC1)CN(C(=O)C(C)(C)C(C)(F)F)C2 c1(C(=O)OCC)c[nH]ccc1=NCC1(O)CCCN(C(=O)C(CC)OC)C1 C12(C(=O)NC3CC(N(C)C(c4cncc(N)n4)=O)C3)CCOC1CC(=O)NC2 CCC(CCC(=O)NCC1(NC(c2ccnc(-c3ncc[nH]3)c2)=O)CC1)OC C(=O)(C(O)CC(C)C)NCCC(=C)CNC(c1cccn(C)c1=O)=O C=C(C)CC(C(=O)NCC1CC1NC(=O)C(C(C)O)NC(=O)C(C)C)OC C1(C(N2CC(F)(CNC(c3cc4cccnc4s3)=O)C2)=O)Cc2ccccc2S1 N1(CC(=O)N(CC(C)NC(c2nccc(C(F)(F)F)n2)=O)C)CCCCCC1 C(CC(C)(C)CNC(c1ccccc1C1CC1)=O)NC(C(C1(O)CCCC1)C)=O O=C1NC(C(=O)NC2CCC2NC(c2csc(C(F)F)c2)=O)CO1 C1(CNC(C(C)(C)NC(=O)C2CC2)=O)CC2COCC2N1C(C1CCOCC1)=O N1(C(CC(=C)C)=O)CCC(CNC(c2cccc(COC(C)=O)c2)=O)C(O)C1 CCCC(C)CC(=O)NCC1C=CCN1C(c1cnc(N(C)C)s1)=O N1(C(=O)OC(C)(C)C)C(C(=O)NCc2n[nH]c3c2CCC3)CCCC1C(C)(C)C c1(C(N2C(C(=O)Nc3ncc(Cl)cc3F)CC(F)C2)=O)cc2ccccn2n1 c1(C(=O)NCC2(NC(C3CCC(OC)C3)=O)CCOC2)cccnc1C(F)(F)F C#Cc1ccc(C(=O)NC2(OC)CCOC2)nc1 CCC(CC(=O)N1CCC(C2CCCN2C(=O)CNC(=O)C(C)C)CC1)C(F)F c1(OC)cc(C(=O)NC2CCN(C(=O)C(N3C(=O)CCC3=O)C)C2)ccc1Br c1(C(=O)NC2CCC(CN(C(CCCCSC)=O)C)CC2)ccc(O)c(F)c1F C1(CNC(C2C(C)=C2)=O)COCCN(C(=O)COc2cc(C(C)C)on2)C1 N1(CC)CCN(C(=O)NCc2cc(OCC#N)ccc2F)C(C)C1 CC1CN(C(C2(C)CC3CCC2C3)=O)CCC1C(=O)Nc1ccc(C#N)nc1 CCC(O)C(C)(C)C(=O)N1CCOC(CNC(=O)CCCc2cnn[nH]2)C1 CC1OC2(CN)CC1(C(=O)N)C2.C(=O)(C(C)(C)C(N)=O)C(C1CCCC1)=O C1(C(=O)NC2(SCCN(C)CC3CC3)CC2)CCCCN1C(N)=O C1(O)(CC#C)CCN(C(C2CSCCN2C(=O)C=C=C(C)C)=O)CC1 C1(CC(N2CC(CN(C(C(C)OCCC=C)=O)C)C2)=O)CCC(=O)NC1=O C1(NC(C(C)OC(=O)C(=O)Nc2ccccc2)=O)CCS(=O)(=O)N1C O=C(C1=CCc2ccccc21)NC1CCCC1NC(c1ccc(C(F)F)s1)=O c1(OCCN2CCCC(C(CCCO)=O)C2)nc2ccccn2n1 C1(NC(c2csc(C3CC3)n2)=O)CCCC(N=c2[nH]nc(C(F)F)o2)C1 C1(C(=O)NCCC(C)F)CC12CC(NC(C1(C)CCC1)=O)C2 c1(C(=O)NC(C(=O)N(c2ccc(OC)cc2)CC)C)cn2cc(C)nc2s1 C1(NC(CN2CC(=O)NCC2)=O)CN(C(=O)CC(F)(F)F)C2CCCCC12 C1(NC(c2cc(F)ccc2Br)=O)CC2CCC1N(c1ncc(F)cn1)C2 C=C1CC2(C1)CC(C(=O)NC13CCN(C(c4cc(CC)on4)=O)CC1C3)C2 CC(CCCCCO)NC(C1C2CC1N(C(C1CCCSC1)=O)C2)=O C1(C#N)(C(=O)NCCCN(C(c2cc(C)sc2C)=O)C)CC2(CC2)C1 C(=O)(C(C)(F)C(C)(C)F)NCc1occ(C(N(CCCN=[N+]=[N-])CC)=O)c1 C(=O)(C(C)(C)C1=CCSCC1)NC(C)CNC(C1CCC2CC2CC1)=O N1(C(c2n(CC)nc(C(C)C)c2)=O)CCCC1C1CCCN1C(=O)CCCSC c1(C(N2CCCC(N(C)C(C3CC(F)C(=O)N3)=O)C2)=O)cc(Cl)c(F)c(Cl)c1 CS(=O)(=O)C1(C(N2CCC(O)(CNC(=O)CC3CCCO3)C2)=O)CCC1 c1(C(=O)NCC2CC(C)N(C(c3ccns3)=O)C2)coc2c1CSC2 N1(C(=O)NCC2CN(C(=O)OC(C)(C)C)CC(O)C2)CCCC2(CCCO2)C1 c1(NC(C2(c3nc(CC)on3)CC2)=O)cc(Br)cc(C(=O)OC)c1F C(=O)(CC(C)CC(C)C)N1CCC(c2cn(-c3c(Cl)ccc(C)c3)nn2)C(O)C1 C1(NC(c2c(CNC(C(C)(CO)OC)=O)cc[nH]2)=O)CCC2(CC1)COC2 C(=O)(C1=CCCC1C)N(CCCOCCN(C(CCC=CCC=C)=O)C)C C1(NC(c2ccn(CCN(C)C)n2)=O)CC2(C1)CC2N=c1[nH]ccn2nnnc12 c1(CC(=O)N(CC(C)(C)CNC(=O)CN2CCCC2CO)C)cc(Cl)ccc1Cl c1(CC(N2CC(C(C)NC(=O)C(C)(C)CF)OCC2)=O)c[nH]c2ccccc12 CCC(CN(C)C)CC(=O)N1CC(C2CN(C(=O)CCC(F)F)CCO2)C1 c1(C(C)=O)cc(N2CCC(C(C)NC(c3ccc(Cl)s3)=O)C2)ncn1 n1(CC2C(CNC(=O)NCc3ccc(OC(F)(F)F)o3)C2)cc(C(C)(C)C)nn1 c1(C(=O)NCC(C)N(C(COCCOCCOC)=O)C)c(C)noc1N C=CCCC(C)(C)C(=O)N(C1CCCN(C(C2(O)COC2)=O)C1)CC1CCCO1 C1(NC(c2ccn3cnnc3c2)=O)COC2(CCN(C(=O)C3=C(Cl)CC3)CC2)C1 C1(C(=O)NCC(c2cc(F)cc(Cl)c2)NC(CSCC#C)=O)CCC(C)(C)CO1 C1(C(N2CCN(C)CC2CNC(=O)C(C)(C)NS(C)(=O)=O)=O)CCCC1S(C)(=O)=O c1(SC)n[nH]c(=NCc2ccc(-c3ccc(C(=O)N(C)C)cc3)s2)s1 N1(C(CC2C(C)(C)OCC2)=O)CCC(CO)C(NC(c2ncncc2Cl)=O)C1 C(=O)(C(F)CC1CCCC1)N(CC(CC)NC(=O)C(C)(C)c1cncnc1)C CC1CCN(C(C2CC(O)CN2C)=O)CC1NC(c1cc(C#N)c[nH]1)=O c1(C(C)C(=O)NC(CNC(c2cnc(Br)s2)=O)CO)cccc(C#N)c1 CCC(C)(CNC(=O)C=CC1CCC1)C(=O)N1CCCC(NC(C)=O)C1 N1(C(c2cc(SCCCC)oc2C)=O)CCOc2ccc(F)cc2C1 c1(C(N(C)CC2CCCN2C(=O)Cc2nccn2C)=O)cccc(CCO)c1 C(CN=c1[nH]nc(C2CC2)s1)=CNC(=O)CC1CCC1 C1(NC(C(C)Cn2ccnc2)=O)CN(C(c2cnncc2O)=O)CC(C)(C)C1 c1(C(=O)NC(CNC(CC2(C)CCCO2)=O)CO)cccc2nonc12 c1(CCNC(C2CS(=O)(=O)CC2N2CCOCC2)=O)ncc(C(F)(F)F)cc1Cl N1(C(COC)=O)CCCC(NC(c2ccccc2OCc2ccccc2)=O)CC1 N1(C(C(c2cccc(C)c2)=O)=O)CCC(NC(=O)Cc2cc(C(C)C)no2)C12CC2 C1(N(C(=O)C=Cc2ccco2)C)CN(C(C2CC(F)(F)C2)=O)CC1F N1(CCC(=O)NC(CNC(CCCOC(C)=O)=O)C2CC2)CCC(O)CC1 C1(NC(C=CCC)=O)(CF)CCN(C(=O)C(c2cccc(OC(C)C)c2)(F)F)C1 c1(C(c2n(C)nnn2)NCCCSc2ccc(NC=O)cc2)cc(Br)n(C)c1 CC(CNC(=O)CCOC1COC1)CC(=O)OC(C)(C)C C(Cn1cccn1)(C(=O)N1CCC1C1(O)CCCC1)NC(C(C1CC1)SC)=O C(C(=O)N1CCCCCO1)(C1CCCO1)NC(CCCC(CC)CC)=O N1(C(c2c(C#C)c[nH]n2)=O)CC2CC1CC2NC(c1ccc(=O)n(C)c1)=O c1(C(=O)NCCC2(O)CCN(C(c3csnn3)=O)C2)cc(O)cc(F)c1 CC(C)(C)C(O)C(=O)N1CCSC(C(=O)NCC=Cc2cccc(CO)c2)C1 N1(C(CC(C)OC)=O)CC2CC1CN2C(c1ccccc1CC(C)(C)C)=O C1(C(=O)NC(C(=O)NCC(=C)Br)CC2CC2)CC(=O)NC(C)C1 C1(NC(c2cnc(CCC)s2)=O)CN(C(=O)CN2CCCC(CC)C2)CCC1F C12(C(=O)NC(c3c(C(N4CCC(C(=O)OCC)C4)=O)con3)C)CCN(CC1)C2 C(=O)(C1=CS(=O)(=O)c2ccccc21)N1CCN(C(C=CC(C)C)=O)C2C1CCC2 c1(OC)cnccc1C(=O)NCC(c1ccc(C)cc1)NC(=O)C(C)C(C)C c1(OC)cc(CC(=O)N(CC(C)N(C)C(C2CCC3CC2CO3)=O)C)ccc1C Cc1cnc(C(=O)NC2CCC(CCNC(=O)Cn3ncnn3)C2)nc1 C(=O)(C=CS(C)=O)NCC(C)CNC(=O)C=CCO N1(C(C#CCNC(=O)CCOC2CCOCC2)=O)CC2CC3CC2C1C3 C(=O)(C#CC(C)(C)C)NCCC1N(C(c2ccc(C(C)(F)F)nc2)=O)CCSC1 N1(C(C)=O)CCC2CCC(NC(C3CN4CCN3CC4C)=O)C1C2 C(C(C(=O)NC(C(=O)OC)C1CCC1)C(C)C)NC(c1cnn(CC)c1C)=O c1(C(N2CCC(C)(C)CC2)C(=O)NCc2nnn(C)n2)csc([N+](=O)[O-])c1 N1(C(CCC(C)SC)=O)CCCC(NC(c2cnccc2C)=O)C1C n1(CC)nc(C(=O)N(C2CCN(C(=O)C(C3CCOCC3)C)C2)C)c(Br)n1 N1(C(c2c(OC)c[nH]n2)=O)CC2(CCC2NC(=O)CC2CCCOC2)C1 C1(NC(c2cn(CC)nc2)=O)C(C)CN(C(C2(Cl)CC2)=O)CC1C C1(CC(=O)NCCOC2CCN(C(c3ccc(CC(F)(F)F)s3)=O)C2)CCC(=O)N1 Cc1c[nH]c(C(=O)NCC(c2ccc(-c3nn[nH]n3)cc2)N2CCOCC2)cc1=O C(=O)(C1c2ccccc2C2CC1C2)NCC(CC)NC(c1nc(CC)sc1N)=O c1(C(N2C(CNC(c3n(CCC)ncc3)=O)CC(F)C2)=O)cc(F)cc(C)c1C C(=O)(C(C)C(O)C(C)C)N1CCC(CN(C(COC)=O)C2CC2)CC1 n12cc(nn1)C(=O)N1CC2C1.c1(OCC)sncc1C(=O)OC(C)(C)C Cc1[nH]nc2c1CCC(C(=O)NC1CCCC1NC(=O)CSCCC#N)C2 c1(C(=O)NC2CC(NC(=O)CCc3nc[nH]n3)C2)cc(=O)c2ccc(Cl)cc2o1 N1(C(C2CCC(C)N2C(c2scc3c2OCCO3)=O)=O)CCC(F)C(N(C)C)C1 C(CNC(=O)CC1CCCO1)(CC(=O)NCCOCCN(C)C)OC CC1CN(C(C2CC3OC2C2CC32)=O)CCC1NC(c1ccc(C(F)F)cc1)=O N1(C(C2CC3(CCCC3)CO2)=O)CCCC2(CC=CCO2)CC1 C1(C(=O)NCC2CNC(=O)O2)CC(O)CN1C(=O)CC1CC2CCC1O2 c1(OC)ccc(NS(=O)(=O)CCNC(CO)CF)cc1 Cc1cc(Cl)c(C(=O)NC2CC(C)N(c3ncnc(O)c3Br)C2)cc1C Cc1cc(C(=O)NC2C3CCN(C(=O)CCc4cn[nH]c4)C23)c(F)c(Br)c1 CCCCS(=O)(=O)CC(=O)NCC1CCCN1C(c1ccc(C#N)cc1OC)=O N1(C(C2(C(=O)N)CC2)=O)CC(n2cc(C3(OC(C)(C)C)COC3)nn2)C(O)C1.NC=O N1(C(C2CCCCC2)C(=O)NCCN(C(c2cnc(C)s2)=O)C)CCCC(O)C1 CC1(c2cn(CCC3CC3)nn2)COCCN1C(c1cc(C2CCC2)n[nH]1)=O N1(C(C(CC(C)(C)C)(C)C)=O)CCC(C2CCN(C(=O)Cn3cnnc3)C2)C1 C1(C(=O)NCC2CCN(C(c3cccnn3)=O)CC2)CCC2CCCCC2C1 c1(C(N2C(CNC(c3c(SC)snn3)=O)CC(OC)C2)=O)cnc(O)cc1C c1(C(C)OC)ccc(S(=O)(=O)NC(c2ccccc2Cl)C)cc1 C(CCCC(=O)N(CC(C)NC(c1ncccc1Br)=O)C)OC c1(N(CCC(=O)OC)C(C2(C#N)CC2C(F)(F)F)=O)ccc2ccccc2c1 c1(C(CC(=O)N(CC(C)C)Cc2nc(C)[nH]n2)C)ccc(O)cc1 c1(SC)nc(N2CC(NC(=O)CCOCC(F)F)CC2C)cc(C)n1 N1(C(C(C)NC(C2C(OC)(OC)CC2)=O)=O)CC2CC1CN2C(=O)C(C)C C1(NC(c2cccc(SCC)c2)=O)COCCN(C(c2cc(O)no2)=O)C1 CCC(CC)C(C(=O)NC(CNC(c1ccc(C(C)C)cc1)=O)C1CC1)OC C1(NC(C(CC(C)C)C)=O)CCOC2(CCN(C(=O)COC(F)(F)F)CC2)C1 c1(NC2CC(NC(c3cc(OC)n(C)n3)=O)C2)c(Br)cccc1[N+](=O)[O-] N1(C(=O)C(O)Cc2ccccc2)CC(C2CN(C(c3c(F)cccc3Cl)=O)C2)C1 CCC(CNC(c1cn(C(C)C)nn1)=O)(CC)NC(C1CC2CC1C2)=O Cc1cccc(Cl)c1OCC(N1CC2(CCC2NC(=O)CCC2CC2(C)C)C1)=O C(=O)(CC(CC)CC(C)C)N1CC(CC=C)(NC(c2nncn2CC)=O)C1 N1(C(C(=O)Nc2c(C(=O)OC)scc2C)=O)CCCC2(C1)OCCO2 N1(C(C(C=C)OC)=O)CC(NC(c2ccc(Cl)c(F)c2)=O)C(C)(C)C1 Cc1c(C(=O)NC2CCCC(NC(=O)CCC(N)=O)C2)[nH]c2ccccc12 N1(C(c2c(C)onc2)=O)CCCCC2(CCN(C(c3cnc(CO)cn3)=O)C2)C1 c1(C(=O)NC(C(C)NC(C=C(CC)CC)=O)(C)C)cnnc2ccccc12 c1(C(=O)NCC(C)(C)NC(=O)CSC2CCCCO2)ccccc1N1CCCC1 C1(C(=O)OCC)(C(=O)NCCOCCNC(c2nsc(N)c2C)=O)CCCC1C C1(CNC(c2nc(NC(C)=O)sc2)=O)CCCC(N=c2[nH]nc(C3CC3)s2)C1 C(CCC(C)CC(=O)NC1CC12CC(NC(=O)C=C1SCC(=O)N1C)C2)=C(C)C c1(CC(N2CCC(O)(CC3(C(N(C)C4CC4)=O)CC3)C2)=O)ccc2c(c1)COC2 N1(C(C(COCC)C)=O)CCC2(CCN(C(=O)CCc3cncs3)C2)C1 N#Cc1ccc(C(=O)NC(C2CCOC2)CNC(c2sccc2F)=O)c(O)c1 N1(C(=O)CSCC2CCCCO2)CC2CC1CN(C(C1(n3nccn3)CC1)=O)C2 N1(C(c2c(C)cccc2)=O)CCC2C(CCN2Cc2cocn2)C1 C(C(C)C(C)(C)C)N(C(CC1(NC(Cc2nc(C)oc2)=O)CCC1)=O)C N1(C2N3CCC(CC3)NC2=O)CC(OCCOC)C2(CC2)C1.C(CC1CC1)O.SC C(C(=O)N(CCCCNC(=O)CN1CC(C)(C)C1)C)(C(C)C)SC C1(NC(c2cccc(C3CC3)c2)=O)CCCN(C(=O)C(F)(F)c2ccccc2)C1 C1(C)(CCC(=O)NCCCN(C(=O)C(Cl)=CCl)CCOC)CCC(=O)N1.CC N1(C(C(C(C)NC(c2cc(F)ccc2F)=O)C)=O)CCN2CCCC2C1 N1(C(CNC(CC)=O)=O)CCCCC(C(C)C(=O)NC2CC2CC(C)C)C1 CCC(C)(C(=O)NCCCN(C(=O)CCC1CC(C)(C)CO1)C)OC c1(C(N(CCCCNC(=O)CC(C)(C)C)C)=O)cc(S(N)(=O)=O)c[nH]1 C1(C(=O)NCCN(C(C)C)C(N)=O)CCC(NC(C2(O)CC2(C)C)=O)CC1 Cc1ncccc1C(N1CCOC(C2CN(Cc3ccccc3)C2)C1)=O C=C1CCN(C(C2CCOC2(C)C)=O)C(C(=O)NCC(C)C(C)C)C1 C1(NC(=O)CN2CC3CC3C2)CC2CCC(C1)N2C(c1cccc(F)c1O)=O C12(CC)CCN(CC1)C(=O)c1ccc(nc1)NC2.n1(CCC)cc(COC)nn1 N1(C(c2c(C)nn(C)c2)=O)CC(C)OC2(CCN(C(c3ccns3)=O)C2)C1 C1(C(C)C)CN(C(C2CCNC(=O)C2)=O)CC1C(=O)NCCC(O)C(F)F c1(N(CC(CC(=O)NC)C)C)nc(N2CCC(F)CC2)c2c(n1)CCC2 c1(CC)ccc(C(N2CCOC(CNC(=O)CC3SC(=N)NC3=O)C2)=O)c(F)c1 C1(N(C)C(=O)C2CC2)CCCN(C(=O)C(C)(C)NC(C2CCCCS2)=O)C1 c1(C(N2CC3(CC(NC(C=CC=CC)=O)C3)C2)=O)ccc(Br)c(Cl)c1Cl C(=O)(C1=CCCOCC1)NC1C=CC(C(N2CCC(O)(COC)C2)=O)C1 c1(C(N2CC(NC(C(CC)(C)O)=O)C2)=O)cc(Br)c2ccccc2c1F N1(C(C(CC)OC)=O)CCC(CCNC(=O)C=CCF)CC1.C1C(=O)N1 C1(C(=O)NCC(C(C)C)OC)C=CCN(C(=O)C(C)CC2CCC2)C1 c1(C(N2CCCC(N(C(c3cnn(CC)c3Cl)=O)C)C2)=O)cc(OC)ccc1O C1(CC)CN(C(=O)CC2(C(F)(F)F)SCCS2)CCC1NC(=O)CNC=O c1(C(=O)OCc2nc(COC)sc2)cc2cc(Br)ccc2c(=O)[nH]1 Cc1c[nH]cc(C(N2CCN(C(=O)C=CCCC(C)C)C(CC3CC3)C2)=O)c1=O N1(C(CCC=C(C)C)=O)CC(=O)CC1C(=O)NCCSC(F)F CCC(C(=O)OCC=C(C)C)S.C1(O)CC(C(F)(F)F)C1 C1(NC(c2ncc(NC)nc2)=O)CCCCCC1NC(=O)C(C)OCC(F)(F)F N1(C(C(C=C=C)C)=O)CCCN(C(=O)Cc2cc(C(C)C)no2)CC1CO N1(C(CCCSC)=O)CCCC(C)C1CNC(=O)CCc1cccc(O)n1 C(C(C)C)(C(O)C(=O)NCC(=O)N1CCCO1)OC.c12nocc1C(=O)NC2 N1(C(c2c(C)scc2)=O)CCOC2(CCN(C(=O)C3CCCn4nccc43)C2)C1 N1(C(CCc2n(C)cnc2)=O)CCC(F)(CNC(C2CCCN2N=O)=O)C1 N1(C(CCCOC)=O)CCCCC1C1CCCN1C(c1cc(C(F)F)nn1C)=O c1(C(=O)NCC(CNC(c2nc(C)sc2C)=O)O)c(C)sc2ccccc12 CCS(=O)(=O)CC(=O)NCC1CCN1C(c1cccnn1)=O Cc1nc(CC(=O)NCC(C2CCCN2C(c2cc(Cl)cnn2)=O)(C)C)c(C)s1 C1(CCC)(NC(=O)CCS(C)(=O)=O)CCN(C(C2(N3CCOC3)CCC2)=O)CC1 c1(C(=O)NC(C(N2CC(=CC)C2)=O)C2CCOC2)ccc(O)nn1 N1(C(C(C)OC2CCCC2)=O)CC(NC(c2cnsc2)=O)C2CCCCC12 N1(C(c2c[nH]ccc2=O)=O)CCN(C(c2cc3n(n2)CCO3)=O)C(CF)C1 N1(C(c2c(C)c[nH]c2)=O)CCCC(NC(c2csnn2)=O)C(F)C1 N1(C(CCSCCCC)=O)CCC2CCC12CNC(c1cc(O)cc(=O)o1)=O C12(CNC(CC(C)n3cccn3)=O)CCCCC1N(C(=O)C1=CCCCC1)CC2 c1(C(=O)NC2CN(C(c3n(CC)nc(C)c3)=O)CC2C)cccc(O)c1C C1(OC)CCCCN(C(=O)C(N)CCN)C1 C1(CNC(C2(C)CC2)=O)CC12CCN(C(=O)CCN1C(=O)NC(C)(C)C1=O)CC2 C1(C)(NC(C2(C(=O)OCC)CC2)=O)CCN(C(=O)CCC2(C)CC2)C1 c1(C(N(CC(C)NC(C23CCC2CC3)=O)C)=O)cccc(N)c1O N1(C(c2c(CNC(CCc3cnc(C)o3)=O)ccs2)=O)CCC(C)(C2CC2)C1 N1(C(CC(C(C)C)O)=O)CCCC2(C1)CN(C(c1cc3ncccn3n1)=O)C2 C1(NC(C2CC(C)(CC)C2)=O)CCCC(N(C(=O)CS)C)C1.N1(C=O)CCCC1 c1(OCC=C)ccc(Cl)nc1C(=O)NCC1CN(C(c2nncs2)=O)C(C)(C)C1 C1(CCC)CC(C(=O)NCC(C)(C)CN(C(c2coc(Cl)n2)=O)CC)CCO1 C1(NC(CN(C)C2CC2)=O)CCN(C(=O)C(C)(CO)NC(=O)OC(C)(C)C)CC1 C1(C(=O)NCCCOCCCNC(=O)Cc2ccsn2)CC2(CCO1)CC2 c1(C(N2CCC3C(NC(c4c(C)cn(C)c4)=O)C32)=O)ccc(F)c(F)c1 N1(C(c2ccc(CNC(C3CCC(C)C3)=O)o2)=O)CCC(CN=[N+]=[N-])CC1 C1(NC(CCc2onc(CC)n2)=O)CN(C(C2CC(O)C2)=O)CCC1(C)C n1(C(C)C)cc(C(=O)NC2(CCCNC(C3(C)CC3(F)Cl)=O)CC2)cn1 COn1cnc(C)c1C(=O)NC(C)CCC(=O)NC(CO)C1CCC1 CC1CCc2[nH]nc(C(N3CCC4(CC3)CN(C(C3COC(=O)O3)=O)C4)=O)c2C1 C12(C(=O)NC34CC(CNC(c5cc(CC)on5)=O)(C3)C4)CCCC1C2(F)F N1(C(C(CCC)C(C)C)=O)CC(CO)C2(C1)CN(C(c1occ(C)c1C)=O)C2 C1(NC(c2sc(CC)c(C)c2)=O)(COC)CCN(C(=O)C(C)OCCC(C)C)CC1 c1(C(c2nnnn2C2CCOCC2)NCC2CC(OCC)C2)nccnc1C N(C(=NCCc1ccccc1Cl)NCc1ccc(C)cc1)C(C=C)C C(C)(C(=O)NCC(C1CC1)NC(=O)CCSC1CCCC1)(C1CCOCC1)OC C1(C(=O)Nc2c(OC)nccc2)CN(C(=O)CSC(F)F)C(C)(C)C1 C1(C(N(C(C(C)C)C)C)=O)COCCN(C(c2ncc(F)cn2)=O)C1 N1(C(C=Cc2cn(C)nn2)=O)CC(NC(C2CCCOCC2)=O)C(C)(C)C1 C1(CC)OCCC1C(=O)NCCC1CC(NC(=O)C=CC2CCC2)C1 C1(C#N)(C(N2CCC(CCNC(C(C)OCCC=C)=O)CC2)=O)CC12CCCC2 C(C(C(=O)N1CCCC(NC(C2CCCC(C)(C)CC2)=O)CC1)C(F)(F)F)OC C(=O)(C(CCC(N)=O)N(C)C)N1CCN(C(CC(C)(C)C#N)=O)CC1c1cccs1 c1(C(C)C)cnc(NC2CCC(NC(C3(c4ccccc4)CCOC3)=O)C2)s1 C12(C(=O)NC(C3CCN(C(C4(COC)CC=CC4)=O)CC3)C)CC(C)(C1)OC2C C(=O)(C1CCc2cccnc21)N1CC2(CN(C(c3cc(C)c(Cl)cc3)=O)C2)C1 c1(C(N2CC3(CCN(C(c4cc(C)[nH]n4)=O)C3)C2)=O)ccc(S(N)(=O)=O)c(C)c1 C1(C(NOC(C)C2CC2)=O)CCCC(NC(c2ccn(C)c2)=O)C1 N1(C(CNC(C2=C(C)OCCC2)=O)=O)CCN2CCCCC2C1 C(=O)(CC(F)(F)C(F)F)N(C1CN(C(c2c(C)nsc2)=O)CC1F)C c1(CC(N2CC(C)(NC(C(CCC)C)=O)C2)=O)c(C)nc(C)nc1O C1(CNC(C(CC)N(C)C)=O)CN(C(c2ccc(OC)o2)=O)CC2(CCC2)O1 C(=O)(C(F)C(C)(F)F)NCCC(=C)CNC(=O)CCc1ncc(C)[nH]1 C12(CNC(Cn3ccc(C)n3)=O)CCCC1CCN2C(=O)C1=CCN(C)C1 C1(C(N2CC3C(NC(c4cc5scnc5[nH]4)=O)(C3)C2)=O)CC2(CCC2)CCO1 N(C(=NCCOc1ccc(Cl)cc1)NC(C)C1CC1)CC(C)OC c1(C(=O)NCC(C2CCCC2)NC(CCC(C)OC)=O)ccc(C#N)n1C C1(C)(CNC(c2n(CCCOC)nnn2)c2cocn2)C2CCC1CC2 C1(C(=O)NCCC2CN(C(C(C)N3CCC3)=O)C2)CCC(C(N)=O)CC1 N1(C(C(COC)O)=O)CCC(C2(NC(C3CCC(C(F)(F)F)CC3)=O)CC2)CC1 C1(CCNC(C(C)SCC)=O)CN(C(=O)C=CBr)CCO1 c1(NC(C)=O)ccc2c(C(=O)N(c3cccc(Br)c3)C3(C#N)CCOC3)c[nH]c2c1 C1(N(C)C)CCC(C(N2CC3C(NC(C4CCCSS4)=O)C3C2)=O)CC1 N1(C(c2cccc(OCC)c2)=O)CCN(C(=O)CCCC(=O)NC)C(C)C1C N1(C(CS(=O)(=O)NC)=O)CCC(C)N(C(c2nccc(OC)c2OC)=O)CC1 CCC(C)(C)CC(=O)NCC1CC1CNC(C1(c2c(F)cccc2F)CC1)=O c1(C(=O)NCCCN(C(=O)CCc2ccc(C)s2)CC)cc(Cl)nnc1O C1(C(=O)OCC(=O)OCC)CCC2(CCC2)C1.c1(NC(=O)CCCOC)ccccc1 n1(CC)cc(CC(N2CC3CC2(CNC(C2CC=CCC2)=O)C3)=O)c(C)n1 CCC(C)(C)C(O)C(=O)N1CC(C(F)C(=O)NOCCO)(O)C1 c1(OC(C)C(N2CCC(NC(=O)C(c3cnn(C)c3)O)C2)=O)ccccn1 C1(C(=O)NC(CCC)C2CCC2)CCCCC1NC(C1CC=CC(O)C1)=O N1(C(Cc2cn(CC)nc2)=O)CC(C)(C)CC1C(=O)NCC(C(C)C)OC C1(C)(C(N(C(CC)C2CC2)C)=O)CC(O)CN1C(c1cn(C)c(C)n1)=O C#CCCC(O)C(=O)N1CCCC(N(CCO)C(c2cc(Cl)c(Cl)s2)=O)C1 N1(C(C2N(Cc3c(C)ccs3)CCC2)=O)CCN2CCC1C2 C(=O)(C(F)C(C)C)N(C(CNC(c1nc(CC(C)C)sc1)=O)C)C(C)C C1(CC(=O)NCC(N(OCC)C)=O)CN(C(C2(CC)COC2)=O)CC12CC2 N1(C(C(C)NC(=O)Cc2cn[nH]c2)=O)CCC2(COC(=O)N2)C1 C1(NC(C(CC)C)=O)CC(OC)C12CCN(C(c1nn[nH]c1Cl)=O)CC2 C1(NC(C=C(C)C)=O)CCS(=O)(=O)C12CN(C(=O)CSCC(F)F)C2 C1(CNC(C(C)C2CCCC2)=O)(CO)CCN(C(=O)C(C2CCCCC2)F)C1 S(=O)(=O)(c1cccc(F)c1C)N1CCCC(C(N(C(CC)CO)C)=O)CC1 Cc1nccc(Cl)c1C(=O)NCC1(CO)CCN(C(C2CC=CC2)=O)C1 C=CC1(NC(=O)C(Cn2cccn2)NC(=O)C=C(C)COC)CCCC1 C12CC3CCC1N3C(=O)COC2=O.N1(C(CN(CCOC)C)=O)CCCC1 CC1(C(=O)N(CCOCC(N)=O)C2CC2)CCN1C(=O)CN1CCCC1=O C=CCCCC(=O)NC1CN(C(=O)C(C)N(c2ccc(C(F)(F)F)cn2)C)C1 CCCCC(C)CCC(=O)NC(CNC(C1(c2ccsc2)CC1)=O)CO C1(C(F)(F)F)(C(=O)NC2C(NC(c3c(C)cno3)=O)CC2)CC2C=CC1CC2 C12(C(=O)NCC(O)C(=O)OC)CCCN1C2=O.C12(CC)CCC(CC1)C2 Cc1nnc2n1CCN(c1ccnc(-c3cccc(Br)c3)n1)C2 CCC(CCCC(=O)NC1COCCC1(F)F)NC(=O)Cc1c[nH]nc1C CC1CC(NC(=O)Cc2c(Br)cnn2C)CN1C(=O)Cc1c(Cl)cnn1C C1(CC#C)(NC(C2(CF)CCN(C(C3C(Cl)(Cl)C34CC4)=O)C2)=O)CCOCC1 N1(C(C(CC#C)C)=O)CCC(C)N(C(c2cnn(CCOC)c2C)=O)CC1 C1(C(N2C(C)CC(CNC(=O)Cn3cc(C#N)cn3)C2)=O)CCC(C)(C)CC1 O=C(C1=Cc2ccccc2C1)NCC1CCC(NC(=O)C2=COCC2)C1 CCCC(C)(CC)C(=O)N1CCC(N(C(C2(C)CC(C)(C)C2)=O)CC)C1 C1(CCOC)(C(N2CC(C)C(C)C2C)=O)CCN(C(=O)C2=CCCSC2)CC1 CC1CN(C(c2ccc(C#N)n2C)=O)CCCN1C(=O)CN1C(=O)CN(C)C1=O C1(NC(C2C(CC)C2)=O)CN(C(=O)C(C)(O)Cc2ccccc2)CCC1O Cc1ncc(Cl)cc1NC(C1OCCC1NC(C1CC(=O)C1(C)C)=O)=O CCC(C)(C)CCCC(=O)NC(C)C=CC(=O)NCC1CC(F)(F)CO1 N1(C2(C(N)=O)CC2)CCC(NC(=O)Cn2cc(C(F)(F)F)nn2)C1=O C(CCC(=O)N1C2CCC1CC(F)C2)(C(C)C)NC(c1cccc(C)n1)=O c1(CC)onc(C)c1C(=O)NCC1CCC1NC(=O)CCSC N1(C(CC=C)=O)CC2CCC2(CC(=O)NCC2(C(=O)N(C)C)CC2)C1 C1(NC(c2c(SC)cccn2)=O)CN(C(C2CC2(Cl)Cl)=O)CCC12CCC2 N1(C(CCCc2c(C)ccs2)=O)CCN(C(C2CCCCC2(C)C)=O)C(CO)C1 C1(C(N(C2CC(NC(CCC)=O)C2)C)=O)CC(C)(C)OC(C)(C)C1 N1(C(=O)CC2CCCOCC2)CCCC2(C1)CN(CC(O)CC(F)(F)F)CCO2 c1(CCC(N2CCC(CN(C(=O)C(C)CF)CC)C2)=O)ccc(Cl)nc1 N1(C(c2ccc(SC)nc2)=O)CCCOC(COc2ccccc2)C1 C(c1cccc(C)c1)=CC(=O)NCC1(CC(=O)NCC(CCC)O)CC1 C1(NC(C2CCN(C(C)=O)CC2)=O)CCN(Cc2ccc(O)cc2C)CC1F Cc1coc(C2CC2)c1C(=O)NCC(C1CCCC1)NC(c1ncn(C)n1)=O N1(C(c2c(CC)n(C)nc2)=O)CCCC(C)(CNC(c2ncnn2C(C)C)=O)C1 c1(C(N2CC(CC=C)(NC(c3cc(Br)no3)=O)C2)=O)c(C)ncn1O c1(NC(C)=O)cc(F)ccc1C(=O)NCC1(F)CN(C(=O)C(C)S(N)(=O)=O)C1 C(=O)(C(C)(C)c1cccs1)N(CCCOCCNC(=O)C=CBr)C C12(C(N(CCC)CCN(C)C)=O)COCC1CN(C(c1cc(C)c(N)cn1)=O)C2 C1(CN(C(c2ccc(C(C)C)s2)=O)C)CN(C(=O)C(F)C2CC2)CCO1 C1(NCc2n[nH]c(=N)s2)CC(NC(C23CCC(CC2)CC3)=O)C12CCOCC2 C(CC(=O)NCC1CN(C)CCN1C)(C(C)(C)C)NC(CC1(CC)CC1)=O CC1CN(C)CC(C(N2CCC(C(=O)NCC3CCCC34CCC4)C2(C)C)=O)O1 N1(C(C(CC#C)NC(C2CCN(C)C2)=O)=O)CCCCC(C)(F)C1 c1(C(=O)NC2C(CNC(C=C(C)c3ccsc3)=O)C2)cc(F)c(F)cc1N N1(C(C(CCC)NC(N)=O)=O)CC2CCCC2(NC(=O)C(C2CCOCC2)O)C1 C(=O)(CC1OCCc2ccsc21)NC(C)CNC(=O)CCS(C)=O Cn1cnc2ncnc(N3CC4(CN(Cc5cc(F)ccc5Br)CCO4)C3)c12 c1(C(=O)NCC(CC)NC(C2(C#N)CC3(CC3)C2)=O)cccc2c1CCC(=O)N2 C1(C(=O)NCC(c2cnc(C)[nH]2)=O)CCC(C2CC2)N1CC1N(C(C)=O)CCC1 C(=O)(CCCCCF)NC1CC(CCC(=O)NCCS(=O)(=O)NC)C1 c1(C(N(CCCNC(=O)CCOCC(F)F)C)=O)cn(CC2CCCO2)nn1 C1(NC(c2[nH]c(=NC)sc2)=O)CN(C(=O)Cc2occc2C)C2(CCCOC2)C1 C(=O)(CC(C)(C)CNC(=O)CC1CC(C)(C)C1)NCCC(C)N(C)C C1(CNC(COCC)=O)CN(C(=O)C(c2ccccc2)O)CC12CC2.C12CC(C1)O2 N1(C(c2nc(C(C)=O)sc2)=O)CC2CC(N(C)C(C3CC(=C4CCC4)C3)=O)C1C2 C12(C(=O)Nc3cccc(-c4on(C)c(=O)c4)c3)CCC(CC(=O)C1)S2(=O)=O C(=O)(CC(C)(C)CN1CCC(CN2CCC(c3nc(C)cs3)C2)C1)NC C(=O)(C(CO)OCC=C)NC(=O)CC1(C)OCCO1 CCCC(C)(C)C(=O)NCC(C1CCOC1)NC(c1cncc(C(F)F)c1)=O C(=O)(CCC(F)(F)Cc1ccccc1)NC1CCN(C(CNC(C)=O)=O)CC1 N1(C(CCCC)=O)CCC2(CC1)CCN(C(=O)CCOc1cc(F)ccc1F)C2 C12(CCN(C(=O)C(F)OC(F)(F)F)CC1)C(=O)N2.C1(N)CCC(=O)NC1C.CC n1(CC(=O)NCC2CN(C(CCC=C(C)C)=O)C(C)C2)ccc2c(C)cccc12 C12CCCCN1C(=O)C=CCCC=CC(=O)NCCC2.C1(C(C)=O)CC1Cl C(=O)(CS(=O)CCC(F)(F)F)N1CCN(C2CCCC(N)C2)CC1 C1(NC(C(C=C)(F)F)=O)CC12CCN(C(=O)COc1c(Cl)cccc1Cl)CC2 c1(OC)cc(C(=O)NCCC(C)NC(c2cc(SC)ccc2C)=O)ccc1C#N N1(C(CC=CC=C)=O)CCN(C(=O)C(C2CC2)Sc2ccccc2)CC1COC Cc1cccc(OCC(N2CCCC2C2CCN(C(=O)C=CC3CC3)CC2)=O)c1 c1(C(=O)NC2CN(C(C#CC(C)C)=O)CC2(C)C)ccc2nc[nH]c2c1 c1(C(=O)NCCC(C)N(C(C(C=CCCC)O)=O)C)cc2c(F)c(Cl)ccc2[nH]1 Cc1noc(C)c1C(C)C(=O)NCCOC1CCN(C(C2CCC=CO2)=O)C1 N1(C(C2(C(C)C)CC2)=O)CC2(C1)C(NC(=O)Cc1cccnc1)CCS2(=O)=O c1(N2CC(C(C)NC(C(C)C3CCOC3)=O)OCC2)nc2ccc(F)cc2s1 c1(C(=O)NC2CCCCN(C(C3(C)CCCCO3)=O)C2)cnc(S(C)(=O)=O)s1 c1(C(N2CC3C(NC(CCc4n(C)ccn4)=O)(C3)C2)=O)c[nH]ccc1=O C1(C(=O)NC(C(C)O)CO)COCCN(c2cc(C3CC3)ncn2)C1 C1(NC(c2ccc(OC)nc2OC)=O)CC1C1CCCN(C(C2(Br)CC2)=O)C1 C1(CNC(c2cnc(C)s2)=O)CCCCN1C(c1cncc(C(N)=O)n1)=O Cc1ncc(Br)c(C(=O)NC2CC3CC2CN3C(c2cccc(C#N)c2)=O)n1 c1(C(=O)NC(C2CCCN(C(=O)C(F)OC(F)(F)F)C2)C)cnc(Cl)n1C N1(C(C)=O)CCOCC(C)(CNC(c2c(C)coc2C(C)(C)C)=O)C1 c1(CNC(c2c(C)ccc(NC(=O)N(C)C)c2)=O)cc2cnccc2n1C c1(CNC(C2CCC3C2C3(F)F)=O)nc2c(s1)CN(C(C1CC1F)=O)CC2 C=CCC(C(=O)N1CCCC(CNC(c2cscc2Cl)=O)C1)C(C)(C)C N1(CC(C(=O)NCC(=C)C)SCCC)CCCC(C2CC2C)C1 c1(C(=O)NC2CCCN(C(Cc3nn(C)c(Cl)c3)=O)C2)cccc(Br)c1Cl N1(CC)C(=O)CCC1CC(N1CC(NC(=O)CC2CCCC2)C(C(F)F)C1)=O c1(C(=O)NC(C(C)NC(c2cc(OC)nn2C)=O)C)cc2nccnc2cc1F CC1CC(NC(c2cc(CCCO)on2)=O)CN1C(c1cnn(CC(F)F)c1)=O c1(OC)ccc(O)c(NC(c2ccc(COc3c(O)cccc3O)nc2)=O)c1 C1(C(=O)NCC(CNC(Cc2cccc(C(N)=O)c2)=O)O)CC12CCSCC2 N1(C(C(C)OCCC#C)=O)CCC(C(C)NC(=O)C(C(C)C)n2cnnc2)CC1 c1(CN2CCC(C(C)NC(=O)C(N3CCNC3=O)C)C2)c(F)cccc1Cl c1(C(CCCCl)=O)c[nH]nc1C1CCCNC1.C12CCCN1C2=O c1(NC(CN2CCC(OC)CC2)=O)ccc(NC(=O)CC)cc1C c1(C(=O)NCCCNC(=O)CC2CCS(=O)(=O)C2)c[nH]c2c(F)cccc2c1=O Cc1ccc(C(=O)NCC2CC(NC(=O)CC3CC3C)C2)s1 CC1CC(NC(C2(O)CCOCC2)=O)CN1C(=O)CCN1CCOCC1 N1(C(C(C)OCC#C)=O)CCN(C(=O)C(CC)CC)CC1CC1CCCC1 N1(C(C(C)Oc2ccc(F)cc2)=O)CCC(NC(=O)CCP(C)(C)=O)C(C)C1 C1(C(=O)NC(c2ccc(C(C)C)cc2)CNC(CSC)=O)CN=C2N=CNN2C1 N1(C(c2n(CC)ccn2)C(=O)NC2CCOC2)C2C=C(c3cccs3)CC1CC2 c1(CCC)c(C(=O)NCC(C)(CC)NC(=O)CO)cnn1C N1(C(C(C(C)C)C(C)C)=O)CCC2CCN(C(=O)COc3ccccc3C#N)C2C1 C(C)(C(C(C)C)NC(=O)CN(C)C(C)C)NC(C1(SC)CC1)=O N1(C(C(CCCC)CC)=O)CCCC2(CCC2NC(c2coc(CO)c2)=O)C1 C1(C(=O)NC(C)Cc2ncn(C)n2)CC(C)CN1C(C1CCCCS1)=O C1(C(N(C)CC2CCSC2)=O)C2CCC(C2)C1NC(c1cnn(C)c1Cl)=O c1(OC)ccc(C(=O)NC2CC(C(=O)Nc3cnccn3)C2)c(OC)n1 c1(OC)cc(CNC2(CO)CCC2)cc(Br)c1OC(c1cccs1)=O C1(C2CC2)(C(=O)NC(CNC(=O)CSCC2CCCO2)C2(OC)CC2)CC1 CC1(C)CC(NC(=O)CCOCC2CCC2)CN1C(C1CC=CCC1)=O c1(C(=O)NC(C2CN(C(C3COC(=O)C3)=O)C2)C)cc2ccc(F)cc2o1 CCC(CC)(CCNC(c1ccc(Cl)cc1C)=O)NC(c1ccn(C)c1C)=O Cc1cc(C(N2CCC(C3OCCC3NC(=O)CC=CC(=O)O)CC2)=O)ccn1 c1(C(=O)NCC2CN(C(C(C)O)=O)C(C)CC2)cc2ncccc2s1 c1(OC)cc(C)cc(C(=O)NC2CN(C(C3OCC3(C)C)=O)CC2(C)C)c1C c1(N2C(CN(C)C(c3cnn(C)c3N)=O)COCC2)ncc2scc(Br)c2n1 C1(C(=O)NC2CCCCC2CNC(C2CC2(F)F)=O)CCCC12CCOCC2 CN1CCN(c2nc(N3CCC(CO)(CO)C3)c3ncsc3n2)CC12COC2 N1(C(C(C)SCC2CCCO2)=O)CCN(C(=O)CC2(C#N)CCC2)CC1C1CC1 CC1CCC(C)(NC(c2cc(CNC(=O)C(F)=CC3CC3)no2)=O)C1 C1(CNC(C(C)OCC2CCCO2)=O)CN(C(C2CC2(Cl)Cl)=O)C2CC12 c1(OC)cncc(-c2ccc(C3CCN(C(=O)CN(C)C(C)C)CC3)cc2)n1 N1(C(C(CCC)CCC)=O)CC(NC(=O)C=Cc2ccccn2)CC2(CCC2)C1 N1(C(c2conc2OC(F)F)C(=O)NCC(C)C)CCCC(CO)C1 c1(NC(CCC=C)C)ccc(S(=O)(=O)NCC(CC)OC)cc1Br Cc1cc(Cl)nc(N)c1C(=O)NCC1CCC(NC(C2CCC3(CCC3)C2)=O)C1 N1(C(C(CC#C)(C)C)=O)CCC2(CC1)CC2NC(=O)Cn1cccn1 C1(CNC(C=CC(C)C)=O)CC2CN(C(C3(C(=O)N(C)C)CC3)=O)CC12 C12(C(=O)NC3CC(CNC(c4cccc(O)c4F)=O)C3)CCCCC1C2(F)F C1(NC(c2ccc(F)cc2)=O)CC2C=CCC(C1)C2.C1(=O)CCC2(CC2)N1C N1(C(=O)OC(C)(C)C)CCC2CC12C(=O)NC1CCC(OCC2CC2)CC1 c1(OC)cc(C)cnc1C(=O)NCC1(O)CCCN(C(C2CC2CF)=O)C1 C#CCCCCC(=O)N(CC(C)N(C)C(C1CC(N(C)C)CCO1)=O)C C1(C(=O)NC2CCCC(CNC(c3cnc[nH]3)=O)C2)CCc2ccccc2O1 c1(C(=O)NCC2N(C(COCC#C)=O)CC(F)C2)ccc(F)cc1Cl N1(C(c2cnc(C)nc2C(C)C)=O)CCC(NC(=O)C2=CCCC2)CC(O)C1 C(=O)(C(C)S(=O)(=O)C1CCOCC1)NC(CN(C(C1(CC=C)CCC1)=O)C)C C1(NC(=O)CN2CCC(Cc3nn[nH]n3)C2)CCCCC12CC2 c1(OC)cc(Br)ccc1C(N1CCN(C)CC1CNC(=O)C(C)(C)C)=O C1(NC(C2C(C)OC(=O)N2)=O)CC2CCC(C1)N2C(C1CC(C)(C)C1)=O [N-]=[N+]=NCCCCC(=O)N1CCC(CNC(C2CC3CCCC3C2)=O)C1 n1(CC)cc(NC(=O)CC2CCCN2C(=O)C(C(C)C)N(C)C)c(C)n1 CN1CC(N=c2[nH]c(NC3CCN4CCCCC34)nc3ccsc23)CC1=O C(=O)(CCC(C)NC(=O)C(c1ccccn1)O)NC1CCN(CC)C1 C=CCC(C(=O)N1CCC(CNC(=O)CCn2c(C)csc2=O)CC1)OC c1(C(CNS(CC)(=O)=O)=O)cc(C(=O)O)c([N+](=O)[O-])c(C)c1 C(=O)(C1CSc2ccccc21)N1CC(SC)C(NC(=O)Cc2ccns2)C1 c1(OCC)ccc(CNC(=O)C(CO)C(C)C)cc1OC.C1(=O)CCO1 Cc1ccc(O)c(C(=O)NCC(C)N(C(=O)CN2C(=O)CNC2=O)C)c1 N1(C(=O)C=CCN2CCCC2)CC(CN(C(=O)Cn2cn[nH]c2=N)C)C2(CC2)C1 C1(CNC(CC=C)=O)CCCCCN1C(=O)C=Cc1ccc(C(N)=O)o1 N1(C(CNC(=O)OCC=C)=O)CCCC(NC(=O)Cc2ccc(C)nc2Cl)CC1 N1(C(c2c(CCC)n(C)nn2)=O)CC(O)C(O)C1CNC(=O)C(C)C(C)(C)C CON(CC1CCCCC1)C(=O)C(CC(F)F)NC(=O)CC1COCC1O C(CCCC(CO)NC(C1C2CCC(F)(F)C12)=O)NC(c1c(C)cnn1C(C)C)=O Cc1cccc(OCCC(=O)NC2CN(C(C3(F)CCC3)=O)CC2C)c1 C1(C)(C(N(C(C(=O)NCC(C)Cn2cccn2)C)C2CC2)=O)COCCO1 C12(C(=O)NC3(CNC(=O)Cc4cccc(N)c4)CCCCC3)CC(C1)S(=O)(=O)C2 N1(C(C2C(C(C(C(CC=C)OC)=O)=O)C2)=O)CCC(F)(F)C(N)C1.NC c1(SC)c(C(=O)NC23CC(NC(=O)C=Cc4ccccc4C)(C2)C3)cccc1F c1(C(=O)NC2CCCN(C(C3N(CCC)CCC3)=O)C2C)c[nH]c2ccncc12 C(C)(C(=O)N=S(C)(=O)CC(C)CC)O.C(CCNC)CC#C C1(CNC(C(CC)N(C)C)=O)CN(C(c2cnns2)=O)CCCO1 c1(C(=O)NC(CCNC(C2C(C)CCO2)=O)C)cc(F)cc2nccnc12 c1(N2CC(CC=C)(NC(c3cc(C(C)=O)c(C)o3)=O)C2)ncc([N+](=O)[O-])cn1 CC(C)CC(C)(C)CNC(c1ccnc(CNC(C2CCN2C)=O)c1)=O C(CC(O)C(=O)NC1CCCC1CNC(=O)CSc1ccc(F)cc1)SC c1(CNC(CCCOCC=C)=O)cccc(CNC(C2(S(N)(=O)=O)CC2)=O)c1 Cc1cccc(C)c1C(N1CCCC(NC(C2CCOCC2(C)C)=O)C1)=O C1(C(N2CC(CO)(NC(C3CCOCC3)=O)C2)=O)(COC)CC(F)(F)C1 C1(NC(CN(CCCCCC)C)=O)(CF)CCN(C(C2CCCCCC2)=O)C1 C1(F)(CNC(c2c[nH]ccc2=O)=O)COCCN(C(C2CCCOCC2)=O)C1 C1(C(=O)NCCC2(NC(CCOCC(C)C)=O)CC2)CC2(CCC2O)C1 c1(N(C)Cc2cccc(Cl)c2)nc(=NCC23CCC(CC2)C3)[nH]c2ccsc12 c1(C(=O)NCC2C(NC(C(F)=CCC)=O)CCC2)nn(C)cc1C c1(C(=O)OCC(=O)N(C2CCN(C)C2)C)c(Br)ccc2ccncc12 c1(CC)cccc(C(=O)N(C)CC2(O)CN(C(=O)CCOC3CCOC3)C2)c1F C1(CNC(C(CC)(CC)CC)=O)CC2(CCN(C(=O)C(O)C(C)C)C2)CO1 Cc1ccc(N)c(C(N2CCC3(NC(c4[nH]ncc4C#N)=O)CC3C2)=O)c1 CN1CCC(NC(c2cncc(OCCF)c2)=O)C12CCCNC2 C1(C(=O)NCC(C2CCOC2)NC(c2c(CC)con2)=O)(CO)CCOCC1 C1(CNC(=O)CCOCC(F)F)CC2CCC(C1)N2C(=O)CSc1ccccc1 C(C1CN(C(c2cc(Cl)ncc2N)=O)Cc2ccccc21)NC(C1C(=C)CC1)=O n1(CC(=O)NCCC(C)NC(=O)CNC(=O)Cc2ccccc2)ncn(C)c1=O c1(C(=O)NC2C(CNC(c3c(CC)ccs3)=O)C2)c(N)ccc2nccnc12 CCC(C(=O)NC1CCN(C(c2ncoc2-c2ccco2)=O)C1)n1cccn1 C(=O)(CP(C)(C)=O)N1CCC(C(C)(C)NC(c2nc(N(C)C)sc2)=O)C1 C1(CNC(CC=C(C)C)=O)CC2(CCN(C(C3CC(n4ccnn4)C3)=O)C2)CO1 C(N=c1[nH]cnc2c1COC2)C1CN(C(C2N3C(C)CN(CC3)C2)=O)CC1C C(=O)(C(CC(C)C)C(N)=O)N(CC1C(OCC)CN(C(=O)C2=COCC2)C1)CC CC(C)CC(C)(CNC(=O)CNC(N)=O)NC(=O)NC1CC1 CCC1=C(C(=O)NCC2CCCN(C(=O)Cc3cc(C)on3)CC2)SCCO1 Cc1cc(Cl)c(C(=O)N(C)CCOCCCN(C(=O)CCCC(C)C)C)cc1C c1(C(N(C(CSCC)C)C(=O)NCC(O)C(F)F)C)ccccc1 c1(C(=O)NC(COC)CCO)c(CNC(=O)C(C(C)OC)OC)cnn1C c1(C(=O)NC2CC(CNC(C=CC)=O)C2)cnc(-c2ccoc2)s1 C1(NC(CNC(CC)=O)=O)CC(CNC(=O)CCC(C)C)C(O)C1 c1(CC)[nH]ccc1C(=O)NCC1CCC(NC(=O)C(CC)n2cncn2)C1 N1(C(Cc2ccc(C#N)nc2)=O)CCN(C(C2C3CCCOC23)=O)CC(O)C1 C(=O)(C(CO)C(C)(C)C)NC12CCC(CNC(CCCCCC)=O)(OC1)C2 Nc1ccc(Cl)cc1C(=O)NCC1CCCN(C(C2CCCC3CC23)=O)C1 c1(C(=O)NC(CNC(C2C(C=C)OCCC2)=O)C)coc2c1N(C)C(=O)CCC2 S(=O)(=O)(c1ccc(N2CCC(F)(F)C2)cc1Br)NCC1(OC)CC2CCC1CC2 N1(C(Cc2nc(=N)[nH][nH]2)=O)CCN(C(=O)C=CC2CC2)CC1C(F)F c1(N2CC(C)(NC(=O)C=Cc3cnccn3)C2)cc(C2CC2)nc(S(C)(=O)=O)n1 C#CCC(C)(C(=O)NCC1CN2CCC1C2)NC(C1CNC(=O)CC1C)=O c1(SC)ccc(N)cc1NC(=O)CCC1CCCN1C(=O)CNC(=O)C(C)C C(=O)(C(C)CC)N(CCC)CCNC(=O)CCNC(=O)C(C)NC(N)=O c1(C(=O)NC(CC2CC2)C2CC2)cccnc1O.C12(CC1)C(=O)N(C)C2 N1(C(c2ccc(C(C)=O)o2)=O)CCOCC(F)(CNC(=O)CCCS(C)(=O)=O)C1 Cc1c(C(N2CC(N(C)C(c3c[nH]c(C(N)=O)c3)=O)C(O)C2)=O)noc1C1CC1 CC(C(F)C(=O)NCC12CCC(C1)N(C(c1ccc(C#N)o1)=O)C2)C(F)(F)F C1(N2CCN(c3n(CC=C)c(-c4ccccn4)nn3)CC2)C(C)CCCC1(C)C N1(C(Cc2cc(OC)c(F)cc2)=O)CC2CC(NC(=O)C=C3CCCC3)C(C2)C1 C1(F)(C(N(C(CNC(COCC)=O)C)CC)=O)CCS(=O)(=O)C1 C=CC(C)(O)CC(=O)NC(C)(CNC(=O)C=Cc1ccccc1Cl)CC c1(C(N2CCCC(NC(CNC(C)=O)=O)C2)=O)ccc(Cl)c(F)c1 N1(C(c2cc(C)nnc2)=O)CCN2C(=O)C(NC(c3ccc(O)cc3)=O)CC2C1 c1(C(C)C)ccc(C(N2CCC(C(C)NC(c3c[nH]c(C#N)c3)=O)C2)=O)nc1 C(=O)(C(C)(C)CS(N)(=O)=O)NC(C1CCN(C(=O)CCC(F)F)C1)C n1(CC(N2CC(C)(NC(C3C=CCCC3)=O)C2)=O)cnc2ccc(F)cc2c1=O C12(C(=O)NC3(CNC(c4ccc(CC)[nH]4)=O)CCC3)CSCC1C2(F)F C1(C(=O)OCC)CCCCC1CC(=O)OCCC(=O)Nc1cccnc1Cl C(=O)(CCCCC(N)=O)NC(C(C)C)CCC(=O)Nc1ccc(CO)cc1 c1(SC)cc(C)c(C(=O)NCC(C)(F)CNC(=O)C=CC(F)F)o1 c1(C(=O)NCC(C)N(C(=O)Cc2cnoc2)CC)cn(C)c(=O)cn1 C(=O)(CCCC(=O)N1CCCC(CN(C)C(C2CC(C)(C)C2)=O)C1)OCC c1(CC)ccc(CN(C)C(C2CCN2C(c2ccc(Br)cn2)=O)=O)cc1 N1(C(=O)COc2ccccc2F)CCCN(C(n2nnc(C3CC3)n2)=O)CCC1 c1(NC(=O)NC(c2ccc(S(N)(=O)=O)cc2)CO)ccc(C#CCCO)cc1 C(C1CN(C(=O)CNC(C)=O)CC1C(=O)NCC(F)Cl)=CC C#Cc1cccc(C(N2CC(OCC)C(NC(=O)CC(=O)OC)C2)=O)c1 N1(C(CCCC(=O)OC)=O)CCCCC(N(C)C(C2CC(C3CC3)C2)=O)C1 N#Cc1ccc(C(N2CC(N(CCO)C(c3ccn(C(C)(C)C)c3)=O)C2)=O)c(O)c1 C#CC1(C(=O)NC(C(=O)OCC)C(C)O)CCN(C(C2CC3(C2)CC(O)C3)=O)C1 n1(COCC)nnc(C(=O)NCC2CCCN(C(=O)C(CCSC)OC)C2)c1N CC(CNC(=O)CCC1CCC(=O)N1)(CO)NC(C1(F)CC1)=O c1(C(CNC(COCCOC)=O)Oc2ccccc2OC)ccc(OC)cc1 Cc1nn(C)c2c(NC3CCCN(C(C)C)C3)nc(=NC3COC(C)(C)C3)[nH]c12 C#CCC(C(=O)NCC1CC12CC2(F)F)NC(=O)C=Cc1nccs1 c1(C(=O)NCC(C)NC(=O)CCS(C)(=O)=O)cncc(P(C)(C)=O)c1 C(=O)(C(C)(C)C(C)(C)C)N(CCNC(C1CCCCC1c1nncn1C)=O)CC N1(C(C2(F)CCCN(C)C2)=O)CCC(NC(=O)CC2=CCCC2)C(C)(C)C1 N1(C(CN(C(=O)OC)C)=O)CC(NC(c2[nH]cc(C)c2C)=O)CC1C C(=O)(CC(C)(C)C#N)NCC1(COC)CCN(C(=O)COCC2CCC2)C1 CCCCC(CC(=O)NCc1nnn(C)n1)NC(C1(CCOC)CC1)=O N1(C(CCC#N)=O)CCC2(CCC2)C(CNC(=O)CC2CC2(Cl)Cl)C1 C(=O)(CCCCCCS(N)(=O)=O)NC1(C)CC(NC(C2ON=C(C(C)(C)C)C2)=O)C1 C1(NC(c2ccccn2)=O)CC(C(=O)NCc2cnccc2Cl)C12CCC2 Cc1cc(O)nnc1C(=O)NC1CCCN(C(=O)C(c2ccc(Cl)s2)C)CC1 N1(C(C2C(C)C2)=O)CCCCC1C1(O)CN(C(=O)CCc2cccc(Br)c2)C1 N1(C(C(COCC)NC(c2ncccc2O)=O)=O)CC(CC)CC(C)C1 N1(C(C=CCOC)=O)CCC(CNC(C2CC2c2cccc(C#N)c2)=O)C1(C)C C1(CNC(CC=C=C)=O)CC2(CCN(C(c3ncc(Br)cn3)=O)CC2)CO1 c1(C(=O)N(C(CNC(C2C(C)C2)=O)CO)C2CC2)cccnc1S(=O)(=O)C(F)(F)F c1(C(N2CC(C)(NC(=O)Cc3cccnc3)C2)=O)csc(=NC2CCOCC2)[nH]1 N1(C(C2C(CC)C2)=O)CC(C2CN(C(=O)CCc3cc(Br)ccc3C)C2)C1 C=CCC(C(=O)NC1(O)CCN(C(=O)COCC(c2ccccc2)C)C1)N(C)C N1(C(C(C)(C)OC)=O)CC(OCC2CCOCC2)CC(F)(F)C1 C1(N(C(c2c(C)oc(CNC(C3(C)CC4CC4C3)=O)n2)=O)C)CCN(C)CC1C C1(C#N)(NC(c2c(C)nccc2)=O)CCN(C(c2cnn(CCO)c2)=O)C1 C(=O)(C(CO)C(C)(C)C)N1CCCC(C(C)(C)CNC(C2CCCCCC2)=O)C1 C12(NC(CNC=O)=O)CCOC(NC(c3ccnc(N4CCCC4)n3)=O)(C1)C2 CCC(CC)CC(=O)N1CCC(C2CCCN2C(=O)COC2CCOCC2)CC1 N1(C(C)=O)CCCCC1C(N1CCC1CNC(C1NC(=O)OC1C)=O)=O CC1(C)CC(C(=O)NC(CO)C2CC2)CCN1C(C1CCC=CCC1)=O c1(NC(C(=O)NC2CC3(C(NC(COC)=O)C3)C2)=O)cncc(C#N)c1 c1(OC)c(C(F)(F)F)nc(C)nc1C.C12(CCCCCC1)C(=O)N2 N1(C(c2[nH]cc(CC)c2)=O)CCN(C(=O)CC2(CO)CC2)CC1CCOC CC1Cn2nc(C(=O)NCCCNC(C3CC=CCC3)=O)cc2C(=O)N1 n1(CCNC(CNC(C(C)SCC)=O)=O)cc(C(C)O)nn1 NS(=O)(=O)c1sccc1C(N1CCC(NC(C2CN3CCCC3CO2)=O)C1)=O CC(CN=c1nc2c(ncn2C)c(NCc2ccc(C#N)cc2)[nH]1)C(C)(C)C Cc1c(NCCOC2CCCOC2)cnn1CCO C1(NC(=O)Cc2ccsn2)CC2CC1N(C(=O)C(c1ccc(F)cc1)(F)F)C2 N1(C(CC2CC(OC)C2)=O)CCCCCC1C(=O)N(C)CC1CC1C CCCC(CC)CC(=O)N(C)CC1(CNC(=O)CN2CCC(C)CC2)CC1 C(=O)(C1CCCc2c(O)cccc21)NCC1N(C(c2c(C)oc(C#N)c2)=O)CC1 C(CC)(CCCO)NC(C(C)N(C(=O)COCC(=O)OC)CCC)=O c1(OCCC(N2CCC(CCNC(C34CCCC3C4)=O)C2)=O)ccccc1Cl CC(CC(F)(F)F)C(=O)NCC1CC2(CCC2)C1 C(C(=O)NCC=CCNC(=O)CN1CCCCC1=O)(C(C)C)NC(CC(C)C)=O C1(C(=O)NC2CN(C(c3c(C)c(C)n(C)n3)=O)CC2F)CCCC(F)(F)CC1 c1(C(=O)NCCCCN(S(C)(=O)=O)C)ccc(CCNC(=O)CN(C)C)s1 N(C1CCc2cccnc21)CC(c1cc(Cl)ccc1Cl)O CC1CCN(CC2CCCO2)CCC1(F)F.S(=O)(=O)(c1ccc(OCC)cc1)N N1(C(C(C(CC)C)OC)=O)CC2(C(N3CC(=O)NC(=O)C3C)=O)CC1CCO2 N1(C(c2cc(C(=O)OC)n(C)n2)C(=O)NC)C2CCCC1CC(N=[N+]=[N-])C2 c1(C(N2C(CCC)CN(C(C3C=CCS3)=O)CC2)=O)cnc2c(c1)COC2 C12(C(=O)NCC3(O)CCN(C(c4nc(Br)c[nH]4)=O)CC3)CCCC1C2(F)F C(=O)(C1=NOC(CNC(c2cncc(O)c2)=O)C1)NC(C)CCc1cn[nH]c1 C1(CNC(CCOC(CC(C)C)C)=O)CCN(C(=O)CN(C)CCO)C12CC2 c1(C(N2CC(C)C(CNC(C3CC3C3CC3)=O)C2)=O)ccc(O)c2ccccc12 FC(F)(F)CCCCNCc1ccc(C2CC2)cc1F C(=O)(C1=CCCCCC1)NC1(CO)CCN(C(C2C(C)(C(F)F)C2)=O)CC1 c1(C(N2C(CNC(CC3CC(C(=O)OC)C3)=O)CC2)=O)cc(C)c(N)cc1Cl c1(C(=O)NC(C(C)NC(c2cccc(SCCC)c2)=O)C)cc2sccc2cn1 C12CCN(C1CNC(=O)C(C)OC)C(=O)CCN(C)C2.C1(OCC)CCCC1 C1(NC(C2(CC)CCOC2)=O)CCCCC1NC(C1C=CCS1)=O c1(C(=O)NC2CC(NCc3c(F)cc(I)cc3F)C2)ccc(Cl)c2ccccc12 C1(NC(C2CCC(C)C2)=O)CCN(CCNC(=O)C(C#N)=CC(F)(F)F)CC1 Cc1cc(F)c(CC(=O)NC2CCN(C(C3CC3C)=O)C2)cc1F c1(CC(N2C3CN(C(C(C(=O)OC)C)=O)C(CC3)C2)=O)ccc2c(c1)COCC2 c1(C(=O)NCC2C(NCCNC(CN(C)C)=O)CCCC2)ncc(C#N)cc1Cl O(NC(=O)C(CCP(C)(C)=O)N(C)C)C(C)CNC c1(NC(C2CCCN(C(Cc3ccc(C)cc3)=O)C2)=O)ccc(Br)c(C)n1 C(=O)(C1CCCc2ccnn21)N1C(C2CCN(C(C(C)O)=O)CC2)C(C)(C)C1 N1(C(CC(C)F)=O)CCCCC(N(C(=O)CNC(N2CCCC2)=O)C)C1 N(C1CCc2c(Cl)cc(F)cc21)C(c1cc(CO)on1)=O C(=O)(CCCCCC(C)C)NCC1CCC(CN(C(C2C(COC)C2)=O)C)CC1 C1(CS(N2CC(C(C)(C)O)OCC2)(=O)=O)CC2(CCOCC2)CO1 C(CCN(C(=O)CSc1ccccc1C)C)(C(C)C)NC(C1(CC)CCC1)=O N1(C(C(CC=C)(C)O)=O)CC2CN(C(c3ccn(C4CC4)n3)=O)CCC12 c1(COC)nc(C(=O)NCCN(C(c2c[nH]nc2C2CCC2)=O)C2CC2)co1 n1(CC(=O)NC2CCN(C(C3(NC(C)C)CC3)=O)C2)ccc2ccccc2c1=O C(CC1CC1)(CC(=O)NC(C)COCCOC)NC(CCCCC)=O c1(OCCC)c(-c2ccc(CC(=O)NCc3cccnc3)cc2F)c(C)nn1C N1(C(CCCNC(=O)OC)=O)CCC(C)(C)C1C(=O)NCCN1CC2CC2C1 c1(SC)cn(C)nc1C(=O)NCC1(O)CC(CNC(=O)C=Cc2cnn(C)c2)C1 C1(CC(=O)N(CC(C)NC(C(CN(CC)CC)F)=O)CC)OC(C)(C)OC1=O N1(C(N(c2nc(C)sc2)C(C)C)=O)CC(F)C(F)C1 c1(CN(CCOC)Cc2nccs2)cccc(-c2ccsc2)c1 CCCCC(O)C(=O)NC1(c2cn(-c3cccc(SC)c3)nn2)CC(F)(F)C1 c1(OC)cc(CC(N2CC3CC2C3NC(C2CCCC(C)CC2)=O)=O)ccc1Cl c1(C(=O)Nc2ccsc2CNc2cccc(C(=O)OCC)c2)ccc(Cl)cc1F N1(C(C(CC)N(C)C)=O)CCN(C(=O)CN(c2ccccc2Cl)C)CCC1C Cc1ccc(COCC(=O)N(C2CCC(NC(c3csnn3)=O)CC2)C)cc1 c1(OC)cccc(Cl)c1C1CC1NC(=O)CNC1CCOCC1 C1(NC(CCC(=O)N(C)C)=O)CCCN(C(C2(C)CCCS2(=O)=O)=O)CC1 c1(OC)cc(C(CC(=O)NS(=O)(=O)C(C)C)SC)ccc1C C(=O)(CCCCCN1CCSC(C)(C)C1)NCCC(C)N(C(=O)C(Cl)=CCl)C C1(SC(C)C)CN(C(=O)C=CC(c2ccsc2)=O)CCC12CCC2 N1(CC2CCCOC2)CCCC(C2CC2)CC1.c1(C(C(=O)NCCC)N)ccc(CO)cn1 c1(C(=O)NCC(CC(C)C)NC(C2(C(F)F)CCCC2)=O)ccc(CO)c(Cl)c1 N1(C2C(C(=O)OCc3nc(Br)ccc3F)CCC(C)C2)CCc2ccccc21 c1(OC)cncc(C(N2CCCCC2CCN(C(=O)C(C)SC)C)=O)c1 c1(SC(C)C(=O)NCC2CN(C(=O)C(C3CCOCC3)F)C2)ccc(C#N)cc1 C1(NC(CCOC)=O)CC(NC(=O)COCC2(c3ccncc3)CC2)C12CCC2 C12(NC(CCSc3n(C)ncn3)=O)CCC1CN(C(C1CC3CC3C1)=O)C2 c1(C(=O)NCC2(CNC(C3(C)CCC3)=O)CCCC2)cc2cccnc2cn1 CN1N=C(CC(=O)NCC2CC3(C2)CN(C(c2ccc(F)cc2F)=O)C3)CC1=O N1(C(c2cc(C)[nH]c2C)=O)CCC2CCN(C(=O)C#CC3CCCCC3)C2C1 C(C(C)C(=O)NCC(C)(C1CC1)NC(C1CCC(F)C1)=O)OC c1(C(=O)NC23CC(NC(C(c4cncnc4)C)=O)(C2)C3)nn(C)c2ccccc12 C(=O)(C(CC(C)C)C(C)C)N1C(CC)(CC)CC(NC(c2cc(N)ccn2)=O)C1 c1(C(=O)NCC2CCN(C(C(C)(F)F)=O)C23CC3)cnc2c(F)ccc(F)c2c1 O=C(CSCc1ccccc1Br)NNC(=O)OC1CCCCC1 Cc1cnc(C(=O)NCc2cncc(C(=O)NCC(C3CCCO3)O)c2)cc1C c1(CN2CC(CNC(c3cc(COC)[nH]n3)=O)C2)nc2ccccc2o1 c1(C(N(C)C(C2CC2(C)C)=O)=O)cccc(CO)c1.C12(CC1)C(=O)NCCN2C C(=O)(C1=CC2(CCOC2)C1)NC(CNC(c1cc(-c2n(C)ccc2)[nH]n1)=O)CO Cc1cc([N+](=O)[O-])ccc1NC(=O)CCOC(=O)CC1CC(O)C1(C)C N1(C(c2c(C)noc2)=O)CCC2(CNC(=O)CCC3CC3(F)F)CCCCC12 c1(CC)ncoc1C(=O)NC1COCC1CNC(=O)COCCc1ccccn1 Cc1cnc(C(=O)NCCC2COCCN2C(=O)CCCCCF)c(C)c1 C1(CNC(C2C(C)N(C)CC2)=O)CN(C(=O)CC2CC=CC2)C2(CCOCC2)C1 C1(CC)CN(C(=O)COCCCOC)CCC2(CN(C(=O)CCSC)C2)O1 N1(C(c2c(C)nc(O)cc2)=O)C(C(=O)NCCn2cnnn2)C2CC(O)C1C2 c1(C(=O)NCC(CNC(c2cc(CCOC)on2)=O)C)cccc(C(F)(F)F)n1 C1(C(=O)OC(CCCCC)CC)CN(C(=O)OC(C)(C)C)CC(F)(F)C1 C(CN=c1cc(NCCc2csc(C)n2)nc[nH]1)n1c(C)nc(C)n1 CCC(C)CC(=O)NCCC1(NC(=O)COCC2CC2)CCC1 C(C1=CCCN(C(c2cnc(Cl)s2)=O)C1)NC(c1cc2sccc2[nH]1)=O CC(C)C(C(=O)N1CCC(CN(C)C(C23CC(CO)(C2)C3)=O)C1)N1CCCC1=O C(=O)(CC1=Cc2ccccc2C1)NCCCC(C)NC(=O)CN(c1ccsc1)C C1(C(N2CCC(N(C)CC)C2)=O)CN(C(=O)C(O)CN(C)C)C2(CCC2)C1 C(=O)(C1=CCCN(C(=O)C(CC)(CO)OC)C1)NC(CC=C)C1CC1 C(CC(CNC(=O)CSc1ccncc1)NC(=O)C(C)C1CCCC1)OC c1(C(N(CCNC(c2c(C)nc(Br)o2)=O)C(C)C)=O)cnc2c[nH]nc2c1 C(CNC(c1sccc1Br)c1nnnn1Cc1ccccc1)(C(C)C)OC C=CCCCCCCCC(=O)N1CC(NC(c2cccc(CO)n2)=O)C1 CC1(C)CCC(CCNC(C2(NC(=O)C=CC(=O)NC3CC3)CC2(C)C)=O)C1 C(C(=O)N=c1cco[nH]1)N1CCC(N(C)C(c2cccc(Br)c2O)=O)C1 C1(C(=O)NC2CC=C(C)CC2)CC(C)(C)CCN1C(=O)CCCC(=O)N(C)C c1(C(=O)NC2(C)CC(NC(c3nc(C#C)sc3)=O)C2)ccc2ccccc2c1F N1(C(C2(OCC)CCOC2)=O)CC2CC1(C(=O)NCC=Cc1ccco1)C2 Cc1ccc(C(=O)NCC2CC2CNC(=O)C=CC2C(C)C2(Cl)Cl)nn1 C(=O)(C(CC1CC1)NC(c1ccsc1)=O)N(C1CCOC1=O)C C1(C(=O)NCc2nc(C)oc2)CCC2(CC2)N1C(c1sccc1C#N)=O C1(OC)CC2CC1CC2CNC(C1(c2ccc(C(F)(F)F)cn2)CCC1)=O N1(C(CC(C=C)CCC)=O)CCC2CCN(C(C3CCC(CC)O3)=O)CC12 C1(C(=O)NCCN(CCO)CC)CC(C)N1C(=O)C(C1CCCCC1)O C1(CNC(C(COC)(C)C)=O)CN(C(c2cc(C)nc(C)n2)=O)CCCO1 C12(C(=O)NCC3(O)C(C)CCC3)CCC(CN(C(C34CCC(CC3)O4)=O)C1)C2 C12(CNC(C=CC)=O)CC(COC)(CN1C(=O)C(c1ccc(Cl)nc1)(C)C)C2 C(=O)(CC(O)C(C)C)N(C)CC1CCC(NC(c2c(C)nc(C)s2)=O)CC1 CC#CCC(C(=O)N(CC)OCC)NC(c1cc(O)nn1C)=O CC(N=c1[nH]c(=NC(C)c2ncn(C)n2)[nH]c2c1COCC2)c1ccc(Br)s1 N1(C(c2n(C=C)nnc2)=O)CCC(NC(=O)CCc2ccc(C#N)cc2)CC1C c1(CNC(CN(CC(=O)NC(C(F)(F)F)C2CCCO2)C)=O)ccc(C#N)cc1 C1(C(=O)N(CCC(C)NC(=O)C=Cc2ccccc2)C)(OC)CCCCCCC1 c1(C(=O)NCCCN(C(c2cc(C(C)C)sn2)=O)CC)occc1Br C1(C(=O)NC2CC(N(C(C(CNC(C)=O)(C)C)=O)C)C2)CN2CCCN1CC2 c1ccc(-n2cc(CCNCCCC3CCOCC3)nn2)cc1-n1cccn1 C1(C(N2CCN(CC#C)CC2)=O)CN(C(=O)CCOCC(C)(C)C)CCC1(C)C C=CCC(CCCCC)C(=O)NC1CCN(C(=O)C(F)(F)CCC)CC1F Cc1ccc(C(=O)NC2CCN(C(=O)C(O)Cc3cn(C)cn3)C2)cc1 N1(C(C23CCCCC2C3)=O)C2CCC1CC(CNC(C13CCC(F)(CC1)C3)=O)C2 C1(CNC(c2c(NC)cncc2)=O)CCN(C(c2cnn(C(F)F)c2)=O)CC1C C(C)(CCC(=O)NCC(C1CCCN1C(=O)Cc1ccc(N)cc1)(C)C)OCC C1(CNC(c2ccc(C3CC3)c(F)c2)=O)CSC2(c3ccccc3)CCC(=O)N12 c1(CNC(NC(C)C)=NCCN2CCCOCC2)cccc2c1CCCC2 N1(C(C2(C)CNC(=O)C2)=O)CC(C2CN(C(C3CCCN3C=O)=O)C2)C1 c1(C(N(CCNC(=O)C(C)(CO)OC)CC)=O)cc2cccn2cn1 Cc1sc(N)c(C(N2CCCCC(NC(=O)C(O)C(F)F)C2)=O)c1C c1(C(N2C(CNC(COCCSC)=O)CC2)=O)cccc2nnn(C)c12 c1(C(N(C(CNC(C2COC(C)(C)C2)=O)C2CC2)C)=O)nc2ccccc2s1 C(=O)(C1=CCCCCC1)NCCCNC(C1(c2c(OC)cccc2)CCOCC1)=O N1(C(COC2CN(C(C)=O)C2)=O)CC2CCN(C(c3cc(F)cc(F)c3)=O)C2C1 C1(C(=O)NCC2CCCN(C(c3n(C(C)C)nnc3)=O)C2)COC2(CCC2)C1 N1(C(C(c2ccccc2)C)=O)CC2CN(Cc3ccsc3)CC2C1 C1(C)(C(N2CC(NC(Cc3c(C)con3)=O)(CF)C2)=O)CCNC1=O C1(NCC2CC(OCC)C2)(NC(=O)CCC=CC(C)C)CC(O)C1 C1(N(C(CCSC)=O)C)CCN(C(c2cc(C#N)cs2)=O)CC12CC2 C(=O)(C1=NNC(=O)CC1)NCC(CNC(C1C(C)N(C)CC1)=O)C(F)(F)F C12(C(=O)NCc3cccc(CSC)c3)CC3CC(CC(C3)C1NC(=O)C(C)C)C2 C1(C(=O)NCCCn2cc(CCS(C)(=O)=O)nn2)CCCN(C(=O)NC2CC2)C1 c1(C(C(=O)OC)NC2CN(c3ccccc3)C2=O)ccc(C2CC2)c(C)c1 C(CCC)(C(=O)N(C(C)CN(C)C(C1CC(c2ccccc2)C1)=O)C)=CCC CC1CN(C(C2CC(=O)C23CCC3)=O)CC(C)CN1C(C1OCC2CCCC12)=O C(N=c1[nH]c(=NCc2cnn[nH]2)[nH]c2cccnc12)c1c(N)cncc1 c1(NC(C(=O)NCC(C2CC=CCC2)N)=O)cc(Cl)cc(N2CCC2)n1 c1(C(=O)NC2C(NC(c3ccc(C(=O)OC)[nH]3)=O)CCC2)ccc(Cl)cc1C C1(CNC(C2C(N(CCOC)C(=O)OC(C)(C)C)CC2)=O)C(C)(C)C1(C)C CC1OC2CCC1(C(=O)N(CCn1cc(C(C3(C)CC4CCC3O4)=O)nn1)CC)C2 c1(C(C)C)cc(C(=O)NC2CCC2NC(C2(C#N)CC23CCC3)=O)ccc1F C1(C(=O)NCC(CC)O)CN(C(c2cncnc2CC)=O)CC(C)(C)C1 C1(N(C(c2occ(C)c2)=O)CCc2cnn(C)c2)C2CCC1CNC2 c1(C(CC)C)ccc(NC(N2CCN(c3cccc(O)c3)CC2)=O)cc1 Cc1cc(Cl)ccc1-n1cc(C2CCN(C(=O)C(C3CCC(=O)CC3)F)C2)nn1 N(C1CCCn2ncnc21)C(C1N(C(CNC(C(CC)SC)=O)=O)CCC1)=O N1(C(C(C(C)C)SC)=O)CC(N(C(=O)CCOC2CCC2)C)C2(CC2)C1 C12(C(=O)OC)CCC(C(=O)N(C3CCN(C(=O)C=CC=C(Cl)Cl)C3)CCO)(C1)C2 CC1(NC(=O)CC2CCCC2)CC(NC(c2cc(C(F)(F)F)n[nH]2)=O)C1 c1(C(=O)NC2C(CNC(C(CC)N(C)C)=O)COC2)ccc(OC)c(Cl)c1 C1(CC(=O)NC2CCC(CNC(c3c(C)c[nH]c3)=O)CC2)CC2(CCC2)CO1 c1(-c2n(CC)c(N3CCC(c4ccc(F)cc4Cl)C3)nn2)ccc2c(c1)OCO2 C1(COC)(NC(=O)CCc2ncc[nH]2)CCN(C(c2ncccc2F)=O)C1 C(=O)(CC(C)C(=O)c1ccc(OC)cc1)N1C(CCC)CCC1 C1(OC)CCCN(C(C2CN(C(C3C=CCS3)=O)CC2(C)C)=O)CC1 c1(C(=O)NCCOCCN(C(=O)CC2(O)CCC2)C)onc2ccccc12 c1(C(N(CCNC(CC(=O)NCCC)=O)CC2CC2)=O)ccc(Cl)nc1OC c1(C(C(=O)NC(COC)CO)C)cn(C)nc1C CC(CN=c1nc(N2CC(C)(C)OC(C)(C)C2)c2cc(Cl)ccc2[nH]1)N(C)C C1(C)(C(N(CCCC)CCO)=O)CCCN(C(=O)C(C2CCOCC2)O)C1 c1(CC)ccccc1OCCC(N1CC2CC1C2CNC(=O)CCSC)=O c1(C(N2CCOC(O)C2)C(=O)NCCCCCC)cncc(OC)c1 CC1CC=C(C(=O)N2CC(C(N3CCC(SC(F)F)C3)=O)(CF)C2)CC1 CCC(C)N=c1nc2c(ncn2C)c(NCCC(c2ccccc2)C)[nH]1 C1(CC(=O)OC)Cn2cnc(OC(CCCC(=C)Br)=O)c2NC1=O CC(CC1CC1)N=c1c(C#N)c[nH]c2c(F)ccc(Cl)c12.C12CC(C)(C)CCN1C2 Cc1ccccc1Cn1cc(CN2CCC(N(C)C)CC2)cn1 c1(CNC(C2(c3cn(CCN(CC)CC)nn3)CCC2)=O)nc(C2CCCC2)n[nH]1 c1(C(N2CCCC(N(C(=O)CCCCCF)CC)C2)=O)cc(C(F)F)ccc1F N1(C(c2cnc(CC)o2)=O)CC2COCC2(C(=O)NCC2CCCC2C)C1 Cn1nc(C(=O)NC2CC3CC2N(C(c2cnc(C4CC4)o2)=O)C3)c(Br)c1Cl C1(NC(C2CC(=C)C2)=O)CC(C(=O)NCC(c2ccccc2F)O)CC1O CC(C)C(C)(O)C(=O)NCC(=C1CN(C(C2CC(C3CC3)=NO2)=O)C1)F C1(C(N2CC(NC(c3cnc(COC)s3)=O)C(O)C2)=O)CCCCC12CC2 Cc1nn(CC(F)F)cc1C(=O)NC(C)CNC(c1csc(-c2ccoc2)n1)=O Cc1nc(O)ccc1C(=O)NC1(C(=O)NC2CC3CCCC3C2)CCN(C)C1 CC(C)C(C(=O)NC(C1C(C(N2CCC(F)CC2)=O)C1)=O)OC1CCCC1 c1(C(N2CCC(N(C(C3(C)CC4CC4C3)=O)CC)C2)=O)cc(Cl)c(OC)cc1C N1(C(C(C)(C)SC)=O)CCCN(C(c2ncnc3c2OCCO3)=O)C(C)C1 Cn1c(O)nc(C(=O)NCC2CCN2C(=O)C=Cc2cccc(O)c2)cc1=O Cc1ncc(F)c(=NCC(C)(C)CNC(c2occc2C2CC2)=O)[nH]1 N1(C(=O)CC2CC2(F)F)CCN(CCNC(C2(C3CC3)CCCO2)=O)CC1 Cc1ccc(C(=O)NC2CC(C)(NC(=O)C(c3ccccn3)C)C2)[nH]1 C1(CCC)(C(=O)N(CCCn2cc(CCC3CCOC3)nn2)C2CC2)CCOC1 N1(C(C(C(C)C)SC)=O)CC(O)(C2(CNC(c3c[nH]c4cccnc34)=O)CC2)C1 C1(CCCNC(CC#N)=O)CCN(C(=O)CC2CCOC2)CC1 Cc1cc(C)c(C(=O)NC(C)CC(C)NC(C2CCC(=C3CCC3)CC2)=O)[nH]1 N1(C(c2c(C)cncc2)=O)CCCOC(CNC(=O)CCc2cnoc2)C1 c1(NC(C2CCC(NC(c3ccc(CC)cc3)=O)CC2)=O)cc(Br)ccc1Cl CC1CCN(C(=O)CC2CCC(C)C2)C1CNC(=O)CCc1ccccc1 C1(C(=O)NCC(N(C)C(c2ccccn2)=O)C2CC2)CCc2nncn2C1 N1(c2ccnc(COC)n2)CC2CCC1C(NC(=O)Cc1sc(O)nc1O)C2 CCC(C)CC(C(=O)NCC(=O)OCCOC)NC(C1OCCC1C)=O N1(C(c2cc(C)cc(C)c2)=O)CCN(C(=O)CN2CCS(=O)(=O)CC2)C(C#N)C1 O=C(C(CNC(C1(CO)CCCC1)=O)CC1CC1)N1CCC(F)(CO)C1 c1(C(=O)NC(CN(C(=O)CC2CCCOCC2)CC)C)ccc2ccsc2c1 CC(=O)C(C)CC(C)C(=O)N1CCCC1C(=O)NCC(O)CC(C)(C)C CC1CN(C(C2(C)SCCCS2)=O)CCN1C(=O)CCS(N)(=O)=O C#CCC(C(=O)NCC(C)(COCC)CO)NC(=O)C=CC(=O)NC1CC1 C1(C(=O)NCC2CC2c2cccc(OC(F)(F)F)c2)(OC)CCOC(C)(C)C1 CC1CN(C(=O)Nc2ncc(C(F)F)s2)CC1(F)F C12(CNC(C3(CC(C)C)CCC3)=O)CC(CO)(CN1C(=O)C(C)n1cncn1)C2 c1(NC(C(N(C(C(CC)O)=O)C)C2CC2)=O)cn(C)nc1C#N CC(O)(CNC(=O)NC(c1ccc(C#N)cc1)CF)C(F)(F)F C1(C)(C(N(CCCCN(C(=O)COc2ccccc2Cl)C)C)=O)CCCS1(=O)=O N1(C(C2CC(C(C)C)C2)=O)CCC(F)(CNC(c2cc3cscc3s2)=O)CC1 CC1CC(C)(C)CC1(c1nnnn1C1CC1)NCc1ccc(NC(N)=O)cc1 C(=O)(CC(CC)C(C)C)NC1(C)CCCN(C(C2(OCC)CCCCC2)=O)C1 N1(C(CCC2(C)CC2)=O)CC(C(=O)NCCSC2(C)CCC2)CC1(C)C C1(C(=O)NC2C(NC(=O)CN3CC4CC4C3)CC2)CN2CCC1CC2 c1(CC(=O)NC2(CC=C)CN(C(=O)CC3(C#N)CC3)C2)ccc2c(cnn2C)c1 C12(CNC(c3c(C)n(CC4CC4)cc3)=O)CCCCC1N(C(=O)C(C)C)CC2 c1(OC(C)=O)cc(-n2cc(C(=O)NC3C(=O)OCC3CO)nn2)ccc1Br C(CCC(C)C(=O)N1CC2CC(C(N3CC(O)CC3CN(C)C)=O)(C2)C1)OC c1(CN2CC3(C(C(=O)NCC(C)C)C3)C2)ccnc(F)c1Cl c1(CCCC)nc(CN2C(C(=O)Nc3cccc(Br)n3)CC3CC23)c(Cl)[nH]1 C(=O)(C(O)C(C)C)NCC1C(NC(C(CSC)c2ccccc2)=O)CC1 CCCCNC(=O)N(CCNC(=O)NCC)C.C(=O)(COCC=O)NC C1(NC(C(C)(F)F)=O)CCOC2(CCN(C(c3ccc(F)cc3CO)=O)CC2)C1 c1(CC(C(=O)NCC2(NC(c3cc(C)on3)=O)CCOC2)O)cccc(Cl)c1 N1(C(c2cc(OC)n(C)n2)=O)CC2CCCC(N(C)C(c3ccnnc3)=O)C2C1 N1(C(COCCC)=O)CC2CCC(N(C)C(C3CCCN3N=O)=O)C2C1 CC1(C)CCCOC1CNC(=O)C(c1ccoc1)NC(C1(O)CCCCC1)=O c1(C(C)C(=O)NC2CC(O)(CNC(=O)CCS(C)=O)C2)ccc(F)cc1Br CCCC(C(=O)NCCC1(CNC(C2(c3cc[nH]n3)CCC2)=O)CCCC1)OC c1(C(N2C(CO)CC(NC(C3CC3CF)=O)C2)=O)ccc2c(O)nnc(O)c2c1 C1(NC(NNC(=O)C2(OCC)CCOC2)=O)CCn2ccnc2C1 C(=O)(C1=NOC2(CCC2)C1)N(CCCCCNC(C1CCOC1C(F)(F)F)=O)C c1(NCc2c(OC)c(C)cc(C)c2)[nH]c(=NCc2cnc(C)s2)nc2scnc12 c1(CCC(=O)N(CCCNC(=O)C(F)(F)C(F)F)CCO)ccc([N+](=O)[O-])cc1 N1(C(=O)NC(c2ccc(C(N3CCOCC3)=O)o2)C)CCC(C)(C(F)F)CC1 C1(CC(N2CCC(=CCC)C2)=O)CC(NC(=O)CCn2cccn2)C1(C)C C(=O)(CCS(C)(=O)=O)N1CCCC(CN(C(C(c2cccc(Cl)c2)OC)=O)C)C1 N1(C(C2(C)CC(C)C2)=O)CCC(=CCNC(c2cc(CN(C)C)cn2C)=O)CC1 N1(C(C=C(C)Cl)=O)CCCC(NC(=O)Cc2nonc2C)CC1 c1(CC(C)C(=O)NCC(C)(O)CNC(=O)CC2(C)CC2)ccc(N)cc1 C1(NC(COCc2cc(C)on2)=O)C2CC1N(C(c1cn(C)nc1C(C)C)=O)C2 C(CCC(=O)N1CCCC1C1(C(=O)NCC(C)OCCO)CC1)OCC c1(C(N2C(CNC(CC(c3ccc(CC)cc3)C)=O)CC2)=O)c(C#N)cnn1C N1(Cc2cccc(OC(C)(C)C)c2)CCN(C(C2CCCC2)=O)C(CC#N)C1 C1(C(=O)NCCCN(C(C2COCC2C)=O)CC)OCC2CCCC12 c1(C(N(C(CN(CCCOC)C)=O)C(c2ccc(F)cc2)=O)C)ccc(F)cc1 c1(C(C)O)ccc(C(=O)NC2CC(CNC(=O)C(c3cncn3C)O)C2)cc1 C(=O)(CC1=NNC(=O)C1)NC1CCCN(C(C(C(C)C)c2cc(O)no2)=O)C1 C1(NC(c2n(CC)ncc2)=O)CC2CCC1N(C(c1cc3cnccc3o1)=O)C2 C(=O)(CCCCN(C)C(c1cncnc1C)=O)N1C(CNC(C)=O)CCC1 C(=O)(N=c1cc[nH]cc1)C1CC(NCC(CC(C)C)OC)C1(C)C Cc1oc(C(C)(C)C)cc1C(=O)NC(C)C(CO)NC(C1CC2C=CC1O2)=O C1(CC=C)CCCCC1(c1nnnn1CC=C)NCCSCCC.S(=O)(=O)(CC)N c1(N(C(=O)C=C2CCCCC2)CC)ccnc2[nH]nnc12.N12CCN(CC1)C(=O)C2 CCCCCC(O)C(=O)N(C(C)CCNC(c1cccc(CC)c1C)=O)C c1(C(C(=O)NCC(C)NC(=O)CCn2ncn(C)c2=O)O)ccccc1C(F)(F)F c1(-n2c(C(C)CC(F)F)nc(-c3ccncc3)n2)ccc(S(N)(=O)=O)cc1 c1(N(CCC)C(c2cccn2Cc2ccncc2)=O)ccc(F)cc1Br S(=O)(=O)(c1ccc(NCC2CC(n3cccn3)C2)cc1Cl)N(C)Cc1ccco1 c1(COCC(CN(C)C)(C)C)cccc(-c2ccsc2C#N)c1 C1(NC(c2ccn(C)n2)=O)CC2CC1CN2C(c1cc(C(F)F)cs1)=O c1(C2(C(N(CC=C)CCOC)=O)CC2)ccc(Br)cn1 C1(NC(N(C(C)CC(N)=O)C)=O)CCCOC1c1ccncc1 c1(N2C3CC(C(N)=O)CC2CCC3)nc2ccccc2c(=NCC2COC(=O)O2)[nH]1 c1(C(=O)OC)ccc2c(c1)CN(CC(C1CCOC1)NC(=O)OC(C)(C)C)C2 C(=O)(CC(C)(C)CN(C)C)N1CCC(C)(C(N(C(CC#C)C)C)=O)C1 n1(CCC)ncc(C(c2ccccc2)NC2CC23CCCC3)c1C c1(C(C)C)cc(C(=O)N(C2CCCN(C(C3CC=CCO3)=O)C2)CCF)n(C)n1 C1(CC(=O)NCC2(NC(c3cc(CC)on3)=O)CCOC2)CCCCCC1 c1(C(=O)NCCOCC(=O)NCC(CC)n2cccn2)ccc(Cl)o1 O=C1CCC(NC(C2COCCC2NC(=O)CC(F)(F)F)=O)C(=O)N1 N1(C(C(=O)N(C)C)=O)CCCC(NC(=O)Cc2ccc(Br)c(F)c2)CC1 CC(C)(CCC(=O)N1CC(NC(C2CC(O)(c3ccccc3)C2)=O)C1)[N+](=O)[O-] C1(CC(N)=O)(CO)CCN(C(=O)Nc2ccc(OC(F)F)cc2)CC1 c1(C(N2C(CNC(Cc3n(C)cnc3)=O)COCC2)=O)c[nH]cc(Br)c1=O C1(C)(CNC(CC2CC(CC)C2)=O)CCN(C(=O)CC2CC=CCC2)C1 c1(C(=O)NCCCN(C(=O)CCc2cnc[nH]2)C(C)C)cc(S(N)(=O)=O)c[nH]1 C#CC1(C(=O)NCc2cnnc(C)c2C)CCN(C(C2OCCC2C)=O)CC1 C(CCCCNC(c1cnn(C(F)F)c1)=O)N(C)CC.C1(=O)C(C2CC2)N1 N1(C(C2N(CCCC)CCOC2)=O)CC(NC(c2cccc(N)c2)=O)C2(CC2)C1 C1(C(=O)NC(C2(C(=O)NOC3CC3)CC2)C)CCOC1C c1(C2(NC(C3(n4nccc4-c4nn[nH]n4)CC3)=O)COC2)ccc(C(F)(F)F)cc1 c1(CNC(N2CC(c3ccccc3)C(O)C2)=O)ccc(N2CCCOC2=O)cc1 C1(SC)CN(C(c2cc(C(F)F)no2)=O)CC1NC(C1C2CCCCC12)=O Nc1c(F)c(F)cc(C(=O)NC2CC3CCC(C2)N3C(=O)C2=CCCOC2)c1Cl c12ccc([N+](=O)[O-])c(c1)CN(C(C)(C)C)C(=O)OCCCO2.CC(C)(C)C c1(C(=O)NCCCN(CCCCNC(c2cc[nH]c2)=O)C)ccnnc1 Cc1coc2c(NC(=O)C=CCNC(C3CCC4CC34)=O)cccc12 Cc1cc([N+](=O)[O-])ccc1C(=O)NC1CC1NC(c1cnn(C)c1F)=O Cc1ccc2c(c1)CCC2NC(N1CC(C)(C#N)C1)=O c1(-c2cccc(OC)c2)cccc2[nH]cc(CC(=O)NCc3ccncc3Cl)c12 Cc1ccc(CCC(=O)NC2CCN(C(=O)CCn3ccnn3)CC2C)c(C)c1 C(=O)(C(O)C1=CCCCC1)N1CCC(NC(c2ccc(C(F)F)s2)=O)C(F)C1 N1(C(C(CC(C)C)N(C)C)=O)CC2(C=C(C(=O)NC(C)C(F)(F)F)CO2)C1 C(CCCCC(=O)NC1CCCC1CC(=O)NC1(CO)CC=CC1)NC(N)=O C(C(COC)CC(=O)NCC1CCN1C(c1scnc1C(F)(F)F)=O)OC CCCCC(=O)C(=O)NCCOCCN(C(=O)C(C(C)C)n1cnnn1)C N(C(=NCCCF)NCC1C(c2ccccc2)C1(C)C)CC(CCN(C)C)OC c1(CNCC(CCC(C)C)O)ccc(F)c2ccccc12 N1(C(CC2CC(NC(=O)C=CCN3CCCCC3)C2)=O)CCCC2OCCC2C1 c1(-c2cn(C)nn2)cnn2c1NCC2.Cc1nc(CC(C)C)no1 c1(N(CC(C)C)C(c2c(OC)ccs2)=O)ncc(O)cc1Cl.C123CC(C1)(C2)CNC3=O C(=O)(C1CCCc2nc[nH]c21)NC(CN(C)C(C1CC12CCOCC2)=O)(C)C CC1=C(C(=O)N(CC(C)CNC(C2(CC(F)(F)F)CC2)=O)C)CCC1 c1(-n2cc(C3N(C(C4CC5(CC(C)C5)C4)=O)CCC3)nn2)ccc(F)c(F)c1F C(=O)(C(CC(F)F)NC(=O)CC1CCOC1C)NC1CCC(COC)CC1 C(C)(C)(C(C)CC(=O)NCC(C)(C)C#N)NC(C(CCC)N(C)C)=O N1(C(C(=C)C(F)(F)F)=O)CCC2(CC1)CC(C(=O)NCc1cc(C)no1)=NO2 CC(C)CC(CNC(C1CCC1C)=O)C(=O)NCC1CCO1 n1(CC)cnnc1CNC(c1sccc1CNC(C12CSCC1C2)=O)=O C1(NC(CCCN(C)C)=O)CN(C(=O)CC2CCCC3(CC3)C2)C(C)(C)C1 C1(C(N(CCNC(c2cnc(C)nc2)=O)C2CC2)=O)CC2COCC(C1)C2 CON(C)C1CCN(C(=O)CC2CCCN(C(=O)CN3CSCC3=O)C2)CC1 C1(C(N2CCCC2CCNC(C23CCCC2CCC3)=O)=O)CCn2nccc2C1 C#Cc1ccc(CC(N2CC(CCNC(=O)Cn3cnc(=N)[nH]3)(OC)C2)=O)cc1 Cc1cc(C(=O)NC2CCC2CNC(=O)C(C)(C)CC(C)C)c2n[nH]cc2c1 c1(C(N2CCCC3(CC(O)C3)C2)C(=O)NC(CC)(C)C)cc(Cl)c2c(c1)OCO2 N1(C(c2c(C)nns2)=O)CC2CC1CN2C(c1cncnc1)=O c1(CC(N2CCC(n3cc(C(C=C)(C)O)nn3)CC2)=O)cc(Br)c(F)cc1C C1(C(=O)NCC2N(C(C=CC(CC)=CC)=O)CCC2)CCc2cc(F)ccc2O1 C1(C(N(CC(=O)N(CCOCC#C)C)CC(C)C)=O)SCC=C1C C1(CCNC(c2c(C)nns2)=O)CCCCN1C(=O)COC(C)(C)C(F)(F)F CCC(C)(C)C(O)C(=O)NCC1CCCCN(C(c2c(Cl)cnn2C)=O)CC1 C1(C(=O)NC(CC=C)CO)CCN(C(C)=O)CC1CSc1ccccc1 Cc1c(Br)cnn1CC(=O)NC1CC(C)N(C(C2CC3CC2C3)=O)C1 Cc1ccc2c(c1)CC(C(N1CCC(CNC(c3cncc(O)c3Cl)=O)C1)=O)S2 N1(C(CC(C)C2CC2)=O)CC2CC(C1)C2NC(c1ccc(Cl)c(Cl)c1)=O N1(C(C(CC)N(C)C)=O)CCC(C(=O)NCCCCCC2CC2)(CC)C1 CN1C(=O)c2ccc(C(=O)NC3CC3NC(c3c[nH]ccc3=N)=O)cc2C1=O C(C1=NOC2CN(C(=O)C=CC3CCC3)CC12)NC(c1cc(C)n(C(C)C)n1)=O CCCC(O)CC(=O)NCC1CC(F)(F)CN1C(c1cnn2c1CCC2)=O n1(C(C(=O)NCC2CN(C(C(CCC)C#N)=O)C2)C)nc(C)c([N+](=O)[O-])c1C Cc1ccc(CNc2ccc(-c3ccc(OCCC(C)C)cc3)cc2O)c(O)c1 c1(C(N2CCCC(C(=O)NC)C2)=O)ccc2c(c1)C(CC=O)C(=O)N2 c1(C(=O)OC)cc2c(N(CC(CO)CO)C)nccn2c1 CC(CCCCNC(=O)COC1CCCC1)NC(=O)C(C)OCOC C1(CNC(C2(Br)CCC2)=O)CC2(CCN(Cc3cnc(O)nc3O)CC2)CO1 N1(CC(=O)OC)CCN(CCCN(C)NC(c2nc(C(N)=O)sc2C)=O)CC1 C1(NC(C2CN3CCN2CC3)=O)CCCCN(C(=O)C(c2ccccc2)O)C1 N1(C(CNc2c(NC(N)=O)cccc2)=O)CCC2C(NC(C3CC3CF)=O)CC12 c1(C(N2CC(CNC(c3cccc[n+]3[O-])=O)C2)=O)cc([N+](=O)[O-])sn1 C(=O)(C#CC(C)(C)C)N1CCC(C(C(=O)N(CCN(CC)CC)C)C)CC1 c1(OC)ccc(OC(C)C(N2CCC(N(C(=O)Cc3nccn3C)C)C2)=O)cc1 c1(COCC=CC(=O)OC2CC3CCC2C3)ccc(F)cc1 c1(C(=O)NCC2CCC(NC(=O)Cc3ccoc3)CC2)ccc(F)cc1C1CC1 C1(F)(CNC(c2nc(OC)oc2)=O)CCCN(C(C2(C)CCC(=O)N2)=O)C1 Cc1cnc(N(C)CCN(C)C2CC2)c(S(=O)(=O)NCc2ccc(F)c(O)c2)c1 Cc1cc(CNC(=O)CC2CCN(C)C2=O)oc1C(=O)NC(C)(C)CN(C)C c1(NC(c2n(CCOCC)nnn2)C2C3COCC23)cnc2sccc2c1 Cc1cc(C(CSC2CCCCCC2)Oc2ccccc2)ccc1[N+](=O)[O-] c1(C(=O)OC)cc(SC)nc(Cl)c1.N12CC=CC(C1)NC(=O)C2=O C(=O)(C(CO)C(F)(F)F)N(C(C)C)CCN(C)C(C1CCCC(=O)CC1)=O C12(CC(N3CC(N(C(C(CC)O)=O)C)C(O)C3)=O)CCCN1CCC2 C1(C)(CNC(C2(CNC(C=CC(C)(C)SC)=O)CCCO2)=O)COCCO1 C1(C2CCCO2)(C(N(CCC(C)NC(c2ccc(C#N)s2)=O)C)=O)CCCCC1 C1(CCN(C(C(=O)N(CC(F)F)CC2CCCCC2)=O)C2CC2)CC1C1CC1 c1(C(=O)NC(C(C)NC(CCN(CCCCC)C)=O)C(C)C)cc(C)nc(O)n1 N1(C(C(=O)NC(=O)CC(C(c2ccccc2F)C)C)=O)CCCC2CCCCC12 S(=O)(=O)(c1ccccc1C(N1CCN(C(=O)COC2CC=CC2)CC1C)=O)OCC N1(C(C(=O)NCc2ccc(C(=O)NCCC)cc2)=O)CCC(C)(C)C1C C(CNC(C1C(C)C1C)=O)(CC(F)(F)F)NC(c1nccc(C(=O)OCC)c1)=O c1(NC(C(=O)N(C(c2cccc(C)c2)CC)CC=CCN)=O)ccccc1Cl C(=O)(C(C)CC(C)C)N1CCC(C(=O)NCCCc2ncco2)(OC)C1 C1(NC(CC(C)CN(C)C)=O)COCCN(C(=O)CC2(C#N)CCOCC2)C1 N1(C(C)C)N=C(C(=O)N2CCc3nn(C)cc3C2)CCC1=O CCCC(CNC(=O)C(C)(C)Cl)C(=O)NCCCCN1CCC1 c1(-c2ncc(C(=O)NCC(CCNC(CCSC)=O)O)s2)ccc(OC)cc1 C=C(C)c1ccccc1NC(=O)C(O)CCCNC(c1ccsc1C)=O C1(NC(C(N2CCNC2=O)C)=O)CCCCCN(C(=O)CCS(=O)(=O)N(C)C)C1 O=C(C1=CCOCC1)NCC(c1ccccc1)CNC(c1cscc1Cl)=O c1(NC(C2CC3CC3N2Cc2cnccn2)=O)cccc(-c2nc(O)n[nH]2)c1 C1(C(N2C(C)(CNC(C3CC4(C3)CC43CC3)=O)CCC2)=O)CCc2nncn2C1 C(CS(=O)(=O)CCN=c1ccc(Br)c(S(=O)(=O)N2CCC(C)C(F)(F)C2)[nH]1)OC c1(C(N(CC(CNC(CCCOC(C)C)=O)O)C)=O)cncc(C(C)(F)F)c1 C12(NC(c3c(COC)cccc3)=O)CCC(CN(C(c3ncc[nH]c3=O)=O)C1)C2 C(=O)(C1=C(C)CC(C)(C)CC1)N(C1CCN(C(=O)Cc2c(C)noc2C)C1)CC c1(C(N2CCC(O)(CNC(C3(CO)CCCO3)=O)C2)=O)cncc(C(F)F)c1 C1(O)(CNC(C2CC(CNC(c3n[nH]c(C)c3O)=O)C2)=O)CCCC(C)C1 Cc1cnc(C(=O)NCCCOCCNC(C(=O)C2CC2)C)c(C)c1.C(CN)O.CO C1(CC(=O)NC(C=CC(=O)N(CCCOC)CCO)C)CCC(C)CO1 C=C(C)CCCC(=O)NCC(CC)NC(c1occc1CN1CCOC1=O)=O C1(NC(C(C)N(C)C)=O)CN(C(c2nnn3c2COCC3)=O)Cc2nccn2C1 c1(CNCC2CCN(C(C3CC3c3ccc(Cl)cc3)=O)C2)cc(O)ncc1F CC(CC(C)(C)C)C(=O)NC1CC2CC(NC(C3(CF)CC4(CCC4)C3)=O)C2C1 c1(C(C)=O)cc(NC(=O)C(=O)NC(C2CCCO2)C)ccc1C C1(CC)CN(C(c2ncn(C)n2)=O)CC1NC(=O)C(C)(C)Cc1cnn[nH]1 c1(SCC(=O)NC(CCCCNC(C2(C#C)CCC2)=O)C)ccc(F)cc1F C1(F)(C(=O)NCC(C)CC2CCCC2)CCCN(C(c2ccccc2CO)=O)C1 c1(C2(C(N(CCOC)CC)=O)CCC2)ccc(F)c(F)c1.C(=O)(C#CC1CC1)OC C1(CCOC)CN(C(=O)C(C2CC2)SC)CCN1C(=O)CCc1ccsc1 C1(C(C)(C)C)CC(C(=O)N2CCC(CNC(=O)Cc3ccsc3)C2)=NO1 C1(CC(=O)NC2CCC(NC(C(CC=C)(C)C)=O)C2)CSc2ccccc2O1 Cc1nc(CC(C)C)sc1C(N1CC(C(C)NC(=O)C(O)c2ccco2)C1)=O c1(NC(c2n(CCC)nnn2)(C)CC2CCCO2)ccc(CO)c(Cl)c1 c1(C(N2CC=CC(NC(CSCC(N)=O)=O)C2)=O)nnn2c1CCCC2 C1(C(=O)OC)CC2(C1)CC1(CC(NC(C3CNC(=O)C34CC4)=O)C1)C2 C1(C(=O)O)N(C(c2ccccc2C2CC2(F)F)=O)CC12CCOCC2 c1(C(N(C2CCCN(C(C3(C=C)CCC3)=O)C2)CCF)=O)ccc(C)nc1OC c1(C(=O)NCC2CCCN(C(C(OC)OC)=O)C2)cnc(OC)c(F)c1 N1(C(C2CCC(CCCC)CC2)=O)CCC2(CC2C(N2CCn3nccc32)=O)C1 N1(C(c2c(C)nncc2)=O)CC(NC(c2csnc2C)=O)CC(F)(F)C1 c1(CCN=C(NC(C=C)C)NCC(C2CC2)OC)ccc2c(c1)CCN2C CC1CCNC(=O)C1CNC(C12CC(C)(CN1C(=O)COC(F)F)C2)=O C=CCCC(C)C(c1nnnn1CCCC)NCC1(c2cccc(OC)c2)CC1 CC1(C)C(NC(c2nc(F)ccc2Cl)=O)CCN1C(=O)CC1CCCOC1 CC(C)(C)CC(O)C(=O)NCC(C)(O)CNC(C1CCOC1C(F)(F)F)=O N1(C(C(C)=C(CC)C)=O)CCN(C(C2CCS(=O)(=O)C2)=O)C(c2cccnc2)C1 C(CC1=CCCCC1)Sc1nc(NC(=O)NCCOc2cccc(C)c2)sc1 c1(C(=O)NCC2OCC(C(N)=O)C2)cc(Br)cc(C(F)(F)F)c1N CS(=O)(=O)c1cccc(S(=O)(=O)N2CCOC(CNC(c3cccnn3)=O)C2)c1 C1(C(F)(F)F)(C(=O)NCCN(CC(C)O)C(C2CC2[N+](=O)[O-])=O)CC(C)(C)C1 c1(C(N2C(CNC(C(c3c(C)noc3C)C)=O)CC2)=O)cc(N)nc(Cl)c1 Cc1cc(C)c(C)c(C(N2CC(CC(C)NC(c3cnncc3C)=O)C2)=O)c1C N1(Cc2cnc(C(C)C)s2)CCC(C(=O)Nc2nccc(Cl)c2I)C(O)C1 c1(C2CCN(C(C3CCN(C(C(=O)NCC)C)C3)=O)CC2)nc2ccccc2o1 CC(F)(F)C(C)(C)CNC(c1conc1CNC(=O)Cc1cnsc1)=O N1(C(c2c(F)ccc(C)c2)=O)CCC2(CCCC2C(=O)Nc2ccccc2Cl)C1 c1(NC(C2(CNC(C(c3cn(C)nc3)O)=O)CC2)=O)ccc(=O)n(C)c1 C1(C(N)=O)(NC(=O)CC2(CN(C(CC)C(=O)OCC)C)CC2)CCCC1C Cc1nc(N2CCC(C(C)(C)C)(CNC(C3CC3F)=O)C2)c2scc(C)c2n1 C=CC1CN(C(=O)CC2CCCCC2(C)C)CC1NC(c1ncccc1N)=O c1(CC(=O)NC)cccc(NC(c2cn(-c3cccc(COC)c3)nn2)=O)c1 C1(NC(c2ccc(F)cc2C)=O)CC(C(F)(F)F)CN(CC(=O)OC)C1 CC1CN(C(=O)OC(C)(C)C)CCC1CC(=O)NCc1nc(N(C)C)n[nH]1 Cc1sc(C)c2sc(C(=O)NC3CC3NC(=O)Cc3cncn3C)cc12 c1(C(=O)NC2(CC=C)CCN(C(C=CCC)=O)C2)oc2c(OC)cccc2c1C C1(=O)C(CC2CCCC2)N1.C1(C(=O)OC)CC1C(=O)N(C)CCN(C)C1CC1 C1(COC)CN(C(=O)CCOCc2cccnc2)CCN1C(=O)C(F)OC C1(NC(C2CC(=O)NC2)=O)CCN(C(c2csc(C3CC3)n2)=O)C12CCCC2 n1(CC(=O)NCCCNC(=O)C=CCC23CCC(CC2)C3)ccccc1=O N1(C(CC)=O)CCN(C)C(CNC(=O)COc2c(F)cccc2F)C1 C1(C(=O)NCC2CCC(C)CN2C(=O)Cc2cncnc2)CCCCC1N=[N+]=[N-] O(C1CCCc2cccnc21)C(Cc1c(C)n(Cc2ccccc2)nn1)=O N1(C(C2C(NC(CNC(=O)OC(C)(C)C)=O)COC2)=O)CC2CCCC12 CC1(C)CCC(C(c2nnnn2C2CCC2)NCCc2cc[nH]n2)CC1 c1(C(N2CCC(N(C)Cc3c(C)noc3)C2)=O)ccc(-c2cnn(C)c2)nc1 C1(C(=O)OC)CC(CN)N(C(c2nnc(SC)s2)=O)C1 c1(C(=O)NC(C)CNC(=O)CC2CCOC2)cc2cnccc2o1 c1(OC)ccc(C)cc1C(=O)NC1CCCC1NC(c1cc[nH]c1C1CCC1)=O c1(C(N(CC(CN(C(c2c(C)c[nH]c2)=O)C)O)C)=O)ccc(F)c2occc12 CC1(F)CCCN(C(C2CC23CC(NC(C2COCC2C(N)=O)=O)C3)=O)C1 C(=O)(C(C)(C)C(C)O)NC1CCC(CNC(c2cc(C(=O)OC)[nH]c2)=O)CC1 C12(C(N3CC(C)(CNC(CCOC(C)C)=O)C(C)C3)=O)CC3CC(CC(C3)C1)C2 C#Cc1cncc(C(N2CCC(CO)C(NC(c3ccnc(CC)c3)=O)C2)=O)c1 c1(C(CC)NC(C2(NC(=O)CCCC3CC3C)CCC2)=O)ncc(C)[nH]1 C(=O)(CCCc1cnn[nH]1)N(C(C(=O)N(CCC)CCO)C1CC1)C c1(C(=O)OCC)nocc1CC.c1(C(=O)NCC2CC(CO)C2)coc(C(=O)N(C)C)c1 C1(NC(CCN(C(c2n(CC)ncc2)=O)C(C)C)=O)CCCC(C(C)C)C1 C1(NC(c2coc(Cl)n2)=O)CC2CN(C(=O)CC3CCCCCC3)CC2C1 C(C(F)(F)C(F)F)OCCNC(N1CCN(c2ccc(I)cc2)CC1)=O C(=O)(C(CC)CCCCC)NC(C(NOCC=C)=O)CC=C C1(NC(C2CN(C)C2)=O)CC2CCCC(C1)N2C(C1CCCS(=O)(=O)N1)=O CCCCC(=O)C(=O)NOC.C=CCN(C)CCO.C1CO1 N1(C(CNC(CC(C)C)=O)=O)CCC(CNC(=O)C(C2CCOCC2)C)C1C Cc1ccccc1CC(C)(C)NC(=O)C(N1CC(F)CC1C)C CC1CC(NC(=O)C(F)C(C)(F)F)CCN1C(C1CC2(CSC2)C1)=O C(=O)(C1=CC2CCC1C2)NC1(C)CN(C(c2csc(CSCC(F)(F)F)n2)=O)C1 c1(C(=O)NC2(CNC(CCC=C)=O)CCOCC2)n[nH]c2c1CC1CC21 N1(C(Cc2cc(OC)c(F)cc2)=O)CC(C2CN(C(C3(CF)CC3(F)F)=O)C2)C1 C(C)(C)(CCC(=O)NC(Cc1cn[nH]c1)C(=O)NCc1cc(F)cc(F)c1)OC C1(O)(CNC(CC)=O)CCN(C(C2CCCO2)=O)C1 C(N=c1[nH]c(N2CCc3cccc(N)c3C2)nc2ccsc12)C1CC(=C)C1 C=C(C)c1cn(C2CCN(C(C34CCC(C)(C3)OC4)=O)CC2)nn1 Cc1ncc(Cl)c(C(N2CCC(C(C)NC(=O)C=Cc3cocn3)C2)=O)n1 c1(C(=O)NCCCC(C)NC(C(=C(C)C2CC2)F)=O)cnc2sccn12 C1(CC(=O)N(C2CCN(C(=O)CC3(C)CC3)C2)CC#C)CC2CCC1C2 O=S(=O)(c1cccnc1NCC1(CF)CC1)NCc1cn2cccc(F)c2n1 N1(CCF)CCCCC12CN(CC1(c3ccccc3)COC1)C2 CCC(C(C)CCN(C)C)NC(=O)CCN(C(C1CC1(C)C)=O)C1CC1 c1(C(N2C(CNC(CC(C)SC)=O)CC2)=O)ccc(-n2ccnc2)c(F)c1 C1(N(C)C(C23CSCC2C3)=O)CN(C(=O)C(O)C(F)(F)F)CCC1O Cc1ccc(C#N)cc1C(N1CCOCC1CNS(=O)(=O)CCC(F)(F)F)=O C1(C(=O)NCC2CC[Si](C)(C)C2)N(C(C2CCCCC2)=O)CC12CCCC2 c1(C(N(C)C)=O)cccc(CN2CCC(C3CCCN3)C2)c1 CC(=O)CC(C)(C)CC(=O)N1CCC(NC(C2CCCCN2C)=O)C1 c1(NC(C)=O)c[nH]c(C)c1C(=O)NCC1(C)CCN(C(C2CC(C(F)F)C2)=O)C1 C=CC(C)(C)CC(=O)NCc1ncoc1CCNC(=O)CC(CCC)N(C)C N1(C(C(C)C2CC2)=O)CCN(C(=O)C(C)C2CCOC2)C(CCC2CCCC2)C1 c1(CN(C(C(C)C2CCOC2)=O)C)nc(Br)c(C2CCCCC2)s1 C1(NC(CC(C)(C)N(C(=O)C2=C(Cl)CC2)C)=O)CCn2nccc2C1 c1(CCC)cc(C(=O)NC2(C)CC(NC(=O)Cn3cccn3)C2)ccn1 C1(NC(CCC(C)SC)=O)CC(O)(C2CCN(C(=O)C(C)(C)C)CC2)C1 N(C(=NCCC(C)F)N1CCC(OC)C1)CC(COC)Oc1ccccc1 Cc1cc(C(N2CCN(C(=O)NCc3cc(C)n(C)c3)CC2)=O)n(C)n1 CC(C)(C)C(O)CC(=O)N1CC(Cc2cn(C3CCCNC3=O)nn2)C1 CC(CC(N)=O)C(=O)N1CCC(n2cc(CC3(O)CCSC3)nn2)C(O)C1 C1(NC(c2ccc[n+]([O-])c2)=O)CCCC(C(=O)Nc2cnn(CCF)c2)CC1 c1(C(=O)NC(CNC(c2n(CC)ncn2)=O)CO)cc(Br)c2c(c1)OCO2 C12(NC(=O)COCC(c3ccccc3)F)CCCC1N(C(=O)C(F)=C1CC1)CC2 C1(CNC(C(C(CC)C)OC)=O)CC2CCC1N(C(C1(C#N)CC1(C)C)=O)C2 CCC(C(=O)NCCC(C)N(C)C(C1(c2ncc(C)o2)CC1)=O)C(C)(F)F C1(C(=O)NCC2(C(=O)NC(C)C)CC2)CCN(C(C2CC(C)(CC3CC3)C2)=O)C1 C1(C(NOC(=O)CN2CCCCC2)=O)(C(C2CC(Cl)(Cl)C2)=O)CCCCC1 C(=O)(CC(C)(C)CC(=O)N1CC2(CCN(C(=O)Cn3ccnn3)CC2)C1)OC Cn1ncc2c1CCCN(c1nnc(-c3cnnc(O)c3)n1CCCCO)C2 C1(CNC(C2CCN(C)C2=O)=O)CN(C(=O)CCn2cccnc2=O)CCCO1 CN1CCN(C)C(CNC(=O)CC(CC2CC2)NC(c2cnn(C(F)F)c2)=O)C1 c1(C(=O)NC2CN(C(CCC(C)(C)F)=O)CC23CC3)ccc2cccnc2n1 N(C1CSc2ccc(Br)cc21)C(C(=O)NC(C1CC1c1ccccc1Br)C)=O c1(C(N2C(C(=O)OC)CCC(CC)C2)=O)cc2c(cc1[N+](=O)[O-])OCCCO2 c1(C(=O)NC2C(CC)CN(C(=O)CN(C)C(C)=O)CC2)c(C)nc(C)nc1C C(=O)(C(F)(F)C(F)(F)F)N(CCC(C(C)C)NC(C1CC(C)(C)OC1(C)C)=O)C N1(C(=O)C(c2ncc(Cl)n2C)(F)F)CCC(C)NCC1.C(C=O)=CCC c1(C(=O)NCC2CC(O)(CNC(=O)CCc3ccccc3)C2)cccc[n+]1[O-] N1(C(C(C)=C2CCCC2)=O)CC2CC2(CNC(=O)Cc2cnn(C)c2)C1 C(=O)(CS(=O)(=O)CCO)N1CCCC(NC(=O)C=Cc2cncc(F)c2)(CO)C1 c1(OCC)ccc(C(=O)NC(C)CC(C)NC(c2cnc(Cl)[nH]2)=O)cc1C c1(C(N2CCC(C)(NC(C(CCC)O)=O)C2)=O)cc(N)ccc1O c1(C(=O)Nc2ccc(OCCCC)c(Cl)c2)c(C(C)(C)C)nc2n1CCCC2 C1(C)(C(=O)NC(C2CCN(c3nnc(C)s3)CC2)C)CCCNS1(=O)=O.CN C1(NC(CCCSC)=O)CN(C(=O)CCc2ccccc2Br)CC1CO C(=O)(C1=Cc2ccccc2OC1C(N)=O)N1CCC(Oc2ccc(C)cn2)C1 N1(C(C(C(COC)C)C)=O)CC(C)(C)OC2(C1)CN(C(c1ns[nH]c1=O)=O)C2 N1(C(COCC(C)(C)C)=O)CC2CCC1CN2C(=O)C#CC1CC1 c1(C(=O)NC(CC(C)NC(c2cc(SCC)ncc2)=O)C)cc(OC)ccc1Cl c1(CC(N2C(C(=O)NCC3CC3CO)CC(OC)C2)=O)ccc(C)cc1Cl c1(OCC(=O)NC(CC=C)CNC(=O)CN(C2CCC2)C)ccccc1[N+](=O)[O-] N1(C(C=C(C)C(C)(C)C)=O)CC2(C(N3CC4(CC4)CC3C)=O)CC1CO2 C1(C)(C(N2CC(CNC(c3c(C)nc[nH]3)=O)C(O)C2)=O)Cc2ccccc2C1 C(=O)(CCCCCCNC(=O)CCS(N)(=O)=O)N(C1CS(=O)(=O)C1(C)C)C C1(NC(C2(COCC)CC2)=O)CC(NC(=O)Cc2cnn(C)c2C)C12CCC2 C1(CN(C(COCCOCCOC)=O)C)CCN(C(C2CC2[N+](=O)[O-])=O)CC1 c1(C(=O)Nc2ccc(-c3ccc(NC(C)=O)cc3)cn2)nc2ccc(N)cc2s1 c1(CC(=O)NC2C(NC(CCC(C)SC)=O)C2)cc(Cl)ccc1Br c1(OC)ccc(C(c2nnnn2C2COC2)NCC2CC(=O)NC2=O)c(F)c1 C1(NC(N2CCC(CCC(=O)N(CC(C)(C)CO)C)CC2)=O)CCC2(CC1)CC2 C#Cc1ccccc1CC(=O)NCC1CC(C)N(C(=O)Cc2cc(C)sc2C)C1 C1(C(N(C2CCN(C(=O)C(O)C(C)(C)C)CC2)C)=O)CC2CCCCN2C1 C1(NC(C(CC)SC)=O)CCC(NC(=O)Cc2csc(C(C)C)n2)CC1 C1(NC(C23OCC(CC)(C2)C3)=O)CCC12CN(C(=O)CCC(C)C)C2 C(CCN=C(NCCC1CCOC1(C)C)NCC1(C)CCC(=O)N1)SC CC(CCCCNC(=O)CCC(F)F)NC(c1coc(C2CCC2)n1)=O C1(NC(C2CCCOC2)=O)CN(C(=O)CC2CCCCC2O)C2CCCCC12 CC1C2CCCCC2CN1C(=O)C(CC1CCC1)NC(=O)CC1CCCC(=O)C1 Cc1cc(C(N)=O)c(NC(C2CCN(Cc3ccccn3)CC2)=O)s1 CCC(CC(F)(F)F)NC(C1(CCNC(=O)CCCOC(C)(C)C)CCC1)=O N1(C(c2n[nH]c(=N)[nH]2)=O)C2CCC1CC(CNC(C1CCc3ccnn3C1)=O)C2 N1(C(c2c(C)cc[nH]2)=O)CC(F)(F)CC1C(=O)NCc1cncs1 c1(C(=O)NC(CC(C)NC(c2cccc(C)c2F)=O)C)cccn2c(O)nnc12 c1(OCC(=O)NCCCOC(C2(C)C(C(=O)OC)C2)=O)ccccc1.C1CCO1 N1(C(C(C(CC)C)=O)=O)CCC(C)(C)CC1C(=O)Nc1c[nH]ccc1=O CCCCCC(CC)C(=O)NC1CC(CC(=O)NCc2ccc(C3CC3)cc2)C1 C=C1CCC(C(=O)N(C(C)C(=O)NCc2cc(OC)n[nH]2)CCC)CC1 C1(C(N(CC(C)CNC(c2cccc(SC3CC3)c2)=O)C)=O)CCCCC(=O)N1 c1(N2C(C)CCC(NC(=O)CC3(CO)CCCCC3)C2)ncnc2c1nnn2C C(C(CC(C)C)C(=O)N(C1CC2CC2C1)C)Nc1c(C(=O)OC)con1 c1(CC(=O)NCC(C)(C2CCC2)NC(c2cccc(=O)o2)=O)cc(F)cc(Cl)c1 C=CCC(CC)C(=O)NCC1CCN(C(=O)Cc2nc(=N)[nH][nH]2)C1(C)C CC1CCC(CNC(C2CN3CCN2CC3)=O)N(C(c2nsnc2O)=O)C1 Cc1cncn1CC(=O)NC(C)CC1CN(C(C2CCCN2C)=O)C1 C1(C)CS(=O)(=O)CC12CC2.c1(NC)cnccc1C(N1CCC(C2NCCC2)C1)=O c1(C(N2CCC(=CC(N3CC(C)C(O)C3)=O)CC2)=O)ccc(I)c(F)c1F CCCCC(CC(=O)NC1CC12CCCC2)NC(c1nccc(C)c1N)=O CC1CC(CC(=O)NC2CC(CNC(=O)C(F)n3cccn3)C2)C(C)O1 N1(CCCNC(C)CF)CCC(c2nnnn2CC)(NS(CC)(=O)=O)CC1 N1(C(CC(C=C)(C)C)=O)CC2CC(Nc3ncc4ncnc-4[nH]3)CC1C2 C=C(C)C(CC(=O)OC1CC(OC)C1)OCC.C12CCN(CC1)CC(=O)N(C)C2 C=C(Cl)CC(C(=O)N1CC(CCCC)C1)NC(C1CCC1N(C)C)=O N1(C(CNC(=O)CNC(c2conc2C2CC2)=O)=O)CCC(O)(CO)C1.C(CO)S c1(C(=O)NC2CC2NC(C2CC(F)(F)C2)=O)ccn2ccccc12 c1(OC)cccc(C(=O)NCC(C)(C)NC(=O)CC(O)C2CCCC2)c1OC C1(NC(C(C)OCC=C)=O)CCC(C)(C)N(C(=O)Nc2ccc(OC)cc2Cl)C1 C1(NC(CCN(C(CCCCC#C)=O)CC2CC2)=O)CCC2(CCCC2)C1 CC(CCCC(=O)O)NC(=O)C(=O)NCCC=CC(=O)O CC1(C)CC(=O)OC1CNC(=O)CC1CN(C(c2cccc[n+]2[O-])=O)C1 N1(C(CCCC#CC)=O)CCC2CCCC12C(=O)NCCCSCCCO Cc1cncc(C)c1C(N1C(C(N2CC(F)(F)CC2CO)=O)CC1C)=O c1(NC(C(=O)Nc2ncc(CC3COCCO3)s2)=O)ncc(Cl)cc1F n1(C(C)C2CC2)cnc(C(=O)NCCN(C)C(c2cc(C(F)(F)F)[nH]n2)=O)c1 N1(C(Cc2ccc(OC)cc2C)=O)CC2(CCC(CNC(=O)C(=O)N(C)C)O2)C1 C(=O)(C(CSCC)NC(=O)CCc1nc(O)n[nH]1)NC(c1cccnc1)CC C1(C)(CC)CCN(C(C2C=CCN2C(=O)C2=C(C)CC2)=O)CC1 Cc1nc(CC(=O)NC(C2CCCC2)CNC(C2(CC3CC3)CCCO2)=O)n[nH]1 C(=O)(CC(C(F)F)C(C)(C)C)NC12CC(NC(C(C)OCCC(C)C)=O)(C1)C2 c1(C(=O)NC2COCCN(C(C3CC(C#C)(O)C3)=O)C2)ccc2ccnn2c1 C1(CN(C(C(C)Sc2cc(-c3ccccn3)nn2C)=O)C)CCS(=O)(=O)CC1 N1(C(CC(C)=C(C)C)=O)CCC2(CC1)CN(C(c1ccc(-n3cnnn3)cc1)=O)C2 C1(C(=O)NCCCNC(c2coc(Br)n2)=O)CCC2(CCC2)OC1 N1(C(Cc2cc(C)on2)=O)CCCC(N(C(=O)C(N2CCC(C)CC2)=O)C2CC2)C1 C(=O)(CCCC(=O)N(C)C)N1CCCC(CN(C(C(C=C)C)=O)C)C1 C(C)(C)(CC(=O)NCc1cn(CC2CCCN2C(=O)CC2(C)CC2)nn1)OC n1(CC(=O)NC(CC=C)CNC(=O)CC(C)C2CC2)nc(C(F)F)cc1C N1(C(C(C)=CC2CC2)=O)CC2CC1CN(C(C1CC1(C)C(F)F)=O)C2 N1(C(C(=O)NCC)=O)CC2(CC(NC(C3CCN(C)C3CC)=O)CO2)C1 Cc1cncc(C=CC(=O)NC(C)CC(C)NC(C2CN3CCN2CC3)=O)c1 Cc1cc(=O)ccn1CC(N1CCN(C)CC1CNC(c1cnn(C)c1)=O)=O n1(CCC)nccc1C(N1CC(C)(CCC(=O)NC(C)CCCO)C1)=O C1(CCCC)(NC(=O)Cn2cc(CNC(C3CC3Cl)=O)nn2)CCCC1 O=C(CC(O)c1ccccc1)NC1(CCNC(=O)CC23CCCC2C3)CCC1 C1(C(=O)NC2C(C)CN(C(C3(CF)CC3)=O)CC2)CCCC2(CCC2)C1 c1(C(C)C)cc(C(N2CCC(NC(=O)Cc3ccccc3)C2)=O)on1 c1(CCC(=O)NCC(C)(C)CNC(=O)CC(C)(C)C)ccc(Cl)c(Cl)c1 CCCCC(CNC(C1CCC(C)CC1)=O)OC(F)F.c12cccnc1OC2=O c1(CN2CCOCC(NC(c3c(C)cc(F)nc3)=O)C2)c[nH]c2ccc(O)cc12 N1(C(COCC)=O)CCOCC1CNC(c1c(-c2ccc(C)cc2)noc1C)=O C(=O)(CCCCCCC(=O)N1CCC(NC(c2ccc(F)c(Cl)c2F)=O)C1)OC N1(CCc2ccc(OC)cc2)CC(NC(C2CC2(C)C)=O)CC2(CCOCC2)C1 C(=O)(CS(=O)(=O)C(C)(C)C)NC(CNC(C1(COC)CCCO1)=O)C(C)(C)C c1(OC)cc(Br)c(N(C(=O)COc2nc3ccccc3s2)C)cc1OC C(C(O)C(=O)NCCCc1nccs1)NC(C1(CC)CCCO1)=O N1(C(c2c(CC)non2)=O)CCC(C(=O)NC2CCCC(C)(C)C2)C1(C)C N1(C(c2cc(C)c(F)c(C)c2)=O)CCn2c(cc3ccccc23)C1 C(=O)(C1=COCCO1)N1CCC(C(C)(C)C)(CNC(C(c2ccccc2)C)=O)C1 c1(N(CC(C)C(C)(C)C)C)nc(NCC2Cc3ccccc32)nc2c1cnn2C C1(NC(c2c(C)noc2)=O)CN(C(=O)COc2cc(F)cc(F)c2)CC2(CC2)C1 CN(C(=NCc1ccc(Cl)c(Cl)c1)NC1CCCC1)Cc1nnnn1C CCC(CC)C(C(=O)N1CC(C)(OCC(=O)NCCS(N)(=O)=O)C1)OC CCC(CCCC(=O)Nc1cccc(Cl)c1C)NC(c1sccc1C)=O C1(C(=O)NCC2(CNC(COCCC#C)=O)CC2)NC(=O)CC1c1ccccc1 c1(C(=O)NC(CC(C)NC(CN(S(CC)(=O)=O)C)=O)C)cn2ncccc2n1 C(CCC(=O)NC(Cc1cnc[nH]1)CO)(C(C)C)NC(C(CCCC)=O)=O CNS(=O)(=O)NCC(=O)NCC(C(C)C)NC(=O)COCC(c1ccccc1)C N1(C(c2ccc(Br)c(O)n2)=O)CCCCC2(C1)CN(C(C1CC(C)(O)C1)=O)C2 S(=O)(=O)(c1ccc(Br)cc1NCC=C(Cl)Cl)NC1C(C)C2CCC1C2 c1ccc2c(-n3cc(-c4ccc(Cl)c(Cl)c4)nn3)cccc2c1 N1(C(C2CCCCC(O)C2)C(=O)Nc2ccc(Cl)cc2F)CCC(C2(O)CC2)C1 C1(C(=O)NCC2(NC(COCCCCC)=O)CC2)CC2CCCC(C1)C2=O Cc1nn(CC(F)(F)F)cc1C(=O)NCCCN(C(C1(O)CC1(C)C)=O)C1CC1 C(=O)(C1=COCC1)NCCC1(NC(C2C(C)(c3cccs3)C2)=O)CCC1 c1(NC(CCC)C2CC2)cc(N(C)Cc2n[nH]c(=N)s2)nc(CC)n1 C1(NC(CC(COC)(C)C)=O)CCC2(CC1)CC(NC(c1cn(C)c(O)n1)=O)C2 N1(C(CC(CC)CC)=O)CC2COCCC2(NC(=O)C=CC2CCCCC2)C1 c1(C(=O)OC)ccc(CCC(=O)NC(C)CCCNC(=O)C(C)(C)F)cc1 c1(CSCC(CC(=O)OC)N)cc(C)c(Br)c(C)c1 CC(C)(O)C(F)(F)CNC(N1CCCC(Nc2ccccc2)C1)=O C(=O)(C1CCc2cccc(F)c21)N(CCCCN(C(=O)CC1CCC(=O)N1)C)C N1(C(C2CN(C(c3ccc(C)cc3F)=O)CC(F)C2)=O)CCC(C(N)=S)CC1 CC1C(NC(c2cc3ccccc3s2)=O)C(C)CCN1C(=O)CCCCO C1(NC(c2cc(CCCCC)[nH]n2)=O)CC(O)CN(C(=O)CC2CCCCO2)C1 c1(C(=O)NCC2CN(C(C(c3cn(C)nc3)O)=O)C2)nc2ccccn2n1 CC(C)(C)C(O)C(=O)NC1CC2CC2C1.N12CCOC(C1)c1cn(nn1)C2 N1(C(C(C)(C)C(F)(F)F)=O)CCCC2CN(C(c3ccc([N+](=O)[O-])o3)=O)CCC12 CC1CN=C2NNC(C(=O)N3CCCC3CCO)=C2C1 c1(C(=O)NCC23C(CN(C(C4(CC)CCC4)=O)C2)C3)csc2ncnc(O)c12 C1(NC(c2cncc(F)n2)=O)(CO)CCCN(C(=O)Cn2ccnn2)C1 C(=O)(CC(=O)NCC1C(C(=O)NC2CC(O)C2O)C1(C)C)OC(C)(C)C c1(C(N2CC(N(C(c3ccc(SC)cc3)=O)C)C2)=O)cc(C(F)(F)F)cc(F)c1 C=CCC(CC=C)C(=O)N(C1CCN(C(C2COCCO2)=O)C1)CCC C1(C(N(CC(=O)OC)CC(C)C)=O)COCCC1NC(c1ncsc1C)=O CC1=C(C)CC(C)(NC(C2CC3(CC3)CN2C(C2CC3(CC3)C2)=O)=O)CC1 c1(CNC(C)C2=NOCC2)nnc2n1CCN(c1nccs1)C2 C=C1C(NC(=O)N(C2CCN(c3ncc(Cl)cn3)C2)C)CC2CC1C2(C)C N1(C(C2CS(=O)(=O)C2)=O)CC2CCC(C1)N2C(c1ccnc(OCC(F)F)c1)=O N1(C(COCCOC)=O)CC2(CCN(C(=O)Cc3c[nH]ccc3=O)CC2)CC1C n1(CC(=O)NC(C(C)C)CNC(=O)Cc2nc(C3CC3)cs2)ccc([N+](=O)[O-])n1 c1(-c2nc(CCC(C)C)nn2C(C2CCCC2)C)cccc2c1CCOC2 C1(C(=O)NC2CN(C(C)C)C2)CC12CCN(C(=O)C(N)=O)CC2 C(Cc1ccccc1)(C(=O)NCC1(C(N)=O)CN(C(C2C=CCCC2)=O)C1)C(N)=O c1(OCC)cc(Cl)ccc1C(=O)NCc1cn(CCNC(=O)CC(C)OC)nn1 C1(NC(CCC2(C)CC2)=O)CCC2(CC1)CC(NC(=O)C1=NOC(C(C)(C)C)C1)C2 N1(C(c2c(C)nc[nH]2)=O)CCC2CN(C(C3(c4cccc(F)c4)CC3)=O)CC2C1 C(=O)(C(F)CC(C)(C)NC(C1CC=CCC1)=O)NCCC(C(C)C)CO CCC(CC(=O)NCCC(O)C(=O)N1CC(C2CCCO2)C1)CC(C)C C1(NC(c2cncc(COC)c2)=O)CC(F)CN(C(=O)C(O)CC2CC2)C1 Cc1c(C2(C#N)C(=O)CCC2)ccc2ccccc12 C(=O)(C(C)CC1CC1)N(CC(C)CNC(=O)CN1CC2CC2C1)C c1(C(=O)NC(CC=C)CNC(=O)CCOc2ccccc2)cnc2nccn2c1 C1(COC)C(CC(=O)NC2CCC2NC(c2ccn(C(C)(C)C)c2)=O)C1(F)F N1(C(C(CC)O)=O)CC(CNC(=O)CC2OCCO2)C2(CC2)C1 C1(NC(C(CC)O)=O)CCC2(CC1)CN(C(c1cncc(C)c1Cl)=O)C2 N1(C(c2ncc(OC)nc2)=O)CCCC(C)(CNC(C2CC2C)=O)C1 C1(C(N2CCN(C(CSCc3ccc(C)cc3)=O)CC2)=O)OCC2CCCCC12 c1(C(=O)NC(C)CC2CN(c3cc(Cl)nc(C4CC4)n3)C2)cn2cccnc2n1 c1(CC)conc1CC(=O)N(CCNC(c1cscc1Cl)=O)C(C)C c1(C(N2CCC(C(=O)OC)C2)C(=O)NCC)cnn(C2CC2)c1CC.C(COC)CC C12(COC)CN(C(c3csc(Cl)n3)=O)C(CNC(C3(C)CCNC3=O)=O)(C1)C2 N#Cc1cccc(OCC(N2CC3C(C2)N3C(c2cc(F)cc(F)c2)=O)=O)c1 N1(C(CN(C(C)C)C)=O)CC2(CCN(C(c3cnc(S)nc3)=O)CC2)C1 N1(C(=O)COC2CC2)CCCC(n2cc(-c3ccc(Br)cc3)nn2)CC1 N1(C(C(CC=C)C)=O)CC(CNC(=O)CSc2cccc(OC)c2)CC12CCC2 c1(C(N2CCC3(C(NC(CC4CCC(C)CO4)=O)C3)C2)=O)nc[nH]c2ncnc1-2 C(C)(C1OCCc2sccc21)NC(c1c(NC(=O)OC)cccc1)=O C1(CCNC(C23CC(C)C2C3)=O)CN(C(c2cc(CO)[nH]n2)=O)CCCO1 c1(C(N)=O)cnc(Cl)nc1N1CCC(NS(=O)(=O)C(F)(F)F)CC1.C1(=O)CCN1 Cn1cc(CCNC(=O)C(C2CCCC2)NC(C2CC2C(C)(C)C)=O)cn1 c1(C(=O)NC2CC(C)(NC(c3c(C)ccs3)=O)C2)cnc(O)c2c1NCCC2 Cc1sc(C)c2sc(C(N3CC(O)(CNC(=O)C=Cc4cncn4C)C3)=O)cc12 C1(C(=O)NC2CC(C)(NC(=O)C(c3ccnn3C)C)C2)(CC)CC(C)(C)C1 N1(Cc2nnc(-c3ccc(N(CC)CC)cc3)n2CC)CCOC(C#N)C1 c1(C(=O)NC2(CC=C)CN(C(=O)CCN3CCC3)C2)ccc2c(Br)cccc2c1 CS(=O)(=O)c1ccc(Cl)c(C(N2CCC3CC3(NC(c3cnco3)=O)CC2)=O)c1 c1(CC)c(C(=O)NC23CC2CN(C(=O)CC2CCN(C)C2)C3)cnc2ncnn12 c1(C(=O)NC(CC(C)NC(c2c(OC)cc(C)s2)=O)C)ccc(F)cc1SC c1(CN(C(=O)NC(Cc2cn(C)nc2)CO)CCO)cscc1S(C)(=O)=O c1(CCCCC)cc(C(=O)NCC23CC(NC(=O)CC4CCCO4)(C2)C3)no1 C1(C(N2CCOC(C3CC(F)(F)C3)C2)=O)CCCOCC1 C(=O)(C(CN=[N+]=[N-])NC(=O)CCNC(=O)OC)NC1CCC(CCC)CC1 N1(C(CC(=O)NCC(C)NC(c2c(C)ncs2)=O)C)CCCCC1=O c1(C(=O)NCC2C(NC(c3cc[nH]c3)=O)CC2)nc(C2CC2)ncc1Br C1(CNC(C2N(C(C3C(CC(C)C)C3)=O)CCCC2)=O)CC2CCC1CC2 c1(C(=O)NC2CC(n3cc(-c4c(COC)cccc4)nn3)C2)cncc(C)c1Cl C(CCCCCC(=O)N(C1CCN(C(=O)Cc2cncn2C2CC2)C1)C)SC C1(NC(CCC=CCC=C)=O)CC(C)CN(C(C2(c3n[nH]cc3C)CC2)=O)C1 c1(C(C(=O)NC(C)C)N(CCCO)CC)[nH]nc(C(F)(F)F)c1C CCC(CCCC(=O)NC1CNC(=O)C12CC2)NC(=O)C(C1CCCCC1)F C1(CNC(C2CN(C(C)=O)C2)=O)CCC(C)(C)CN1C(C1C=CCC1)=O C1(NC(C2C(CC)C2)=O)CN(C(C2CCn3cc(C)nc3C2)=O)CC2(CCC2)C1 C#CC(CC(C)C)NC(=O)Cc1ccc(Nc2ccc(C(=O)O)cc2)cc1 Cc1ccc(C(=O)OCCNC(=O)Cc2ccccc2Sc2ccccc2F)n1C N1(C(C(C)Cn2cccn2)=O)CC(C2CC2)(C(=O)NCCCc2cccnc2)C1 C(=O)(C(C(C)C)n1cncn1)N1CC(C(Cn2cc(CCCC=C)nn2)F)C1 C(CC(C(=O)NOCC(N)=O)NC(C1CCN(C)C1)=O)OCC N12CC(C)CCC1C2=O.C(C)(C(=O)N1CC(OCCSC)C1)OCC=C c1(C(=O)NC2C(OC)CN(C(C3(C)CC(C)=NO3)=O)C2)cccc2nc[nH]c12 Cc1nc(NCC2(NC(=O)C(=O)N=S(C)(C)=O)CC23CCC3)ccc1[N+](=O)[O-] c1(C(N2C(CN(C(c3cn(C)nn3)=O)CC)CCC2)=O)ccc(C)cc1 c1(C(N2C(C)(CNC(CCC(C)SC)=O)CCC2)=O)ccc(N)c(F)c1 N1(C(c2ccc(=NC)[nH]c2)=O)CCC2(C=C(C(=O)NC3(COC)CCCC3)C2)C1 CC(C)C(F)(CNC(=O)CCC1CCCO1)C(=O)NCCOCC1CCC1 C1(Oc2cc(C(c3nnnn3CC3CC3)NCCOC)sn2)CCC(=O)NC1 CC(C)C(C)C(=O)N(C)CCOCCCNC(C1CC12CCCC2)=O Cc1cncc(C(=O)NCCC(C)(C)CNC(=O)CCC2C(=O)NN=C2C)c1C C1(CN(C)C(C2(N3CCOCC3)CC2)=O)CCCN(C(C2CC(C)(C)CO2)=O)C1 C(C)(C(C(C)C)NC(CCC)=O)NC(c1cn(C(F)(F)CO)nn1)=O C1(C(=O)NCCCN(C(CCCOC)=O)C)CC(O)CN1C(C)=O CCCC(C)C(=O)NCC1CCC1NC(C1CC(C)(C)C1)=O Cc1cccc(NC(c2cccn2C(c2ccccn2)C2CC(OC)C2)=O)c1C N1(c2n(CCC=C)c(-c3[nH]nc(Br)c3C)nn2)C2CCCC(O)C1CC2 c1(CN(C)CCOC)cc(F)ccc1C.C1(C(=O)NC(C2CCOC2)C#C)CC(C)C1 Cc1cn(C)nc1C(=O)NCC1CCN1C(=O)CCNC(=O)C=Cc1ccco1 c1(C(=O)NCC2N(C(C(C)SC)=O)CCCC2C)c(C)[nH]c2ccccc12 C1(C(=O)NCC2CCC(C(=O)NC3(CC(N)=O)CC3)CC2)CCC2CC1CO2 N1(C(COCCC)=O)CCCC1C(C)(C)CNC(c1ncc(C(F)F)s1)=O C(=O)(C1=CCCC1(C)C)NC(C1CCCC1)CNC(CC1CCCC(C)O1)=O N1(C(=O)CC2CCCC2)CCC2(COCCO)CN(C(C34CC3C4)=O)CC2C1 C1(C(=O)NC(C2CCCC2)C#C)CCCCN(C(C2CCC(N(C)C)C2)=O)C1 C(=O)(CCCC(=O)NCC1(C)CCCN(c2ccnc(C)n2)C1)NCCC N1(C(c2n(C)c(Cl)nc2)=O)CC2CC(C1)CN(C(c1ccc3c(c1)NCC3)=O)C2 Cc1ccn(C)c1C(=O)NC1C=CC(CNC(C2(C)CCCCC2)=O)C1 Cc1c(C(=O)NCCC(C)N(C)C(c2cc([N+](=O)[O-])n[nH]2)=O)oc2ccccc12 C1(NC(C2(CNC(C3N(C)CCOC3)=O)CCCC2)=O)CCn2nccc2C1 N1(C(CC(CN(C)C)O)=O)CC=C(CNC(c2cnn3c2CCC3)=O)CC1 C(=O)(C(C)C(C)CC)NCc1ccc(CN(C(C2(SCC)CC2)=O)C)cc1 C1(OCCN(C(=O)C=CCF)C2CC2)CCN(C(=O)C(O)c2ccsc2)C1 c1(N2CCC(CNC(CC)=O)C23CC3)ncnc2scnc12 C(=O)(CC(O)CNC(=O)C=CCF)NC(C)CCN(C)C C(=O)(CCCC(=O)NC1CC2(C1)CC2C(=O)NCCS(C)(=O)=O)OCC O=C(N1OC2CCC1CC2)C1CCC(C2CC2)N1C(c1coc(N(C)C)n1)=O C#CC(C)(C)C(=O)NC1CC(NC(C2(C)CCCN2C)=O)C(O)C1 C1(C(=O)OC)CN(Cc2occ(CNC)n2)CCO1 N1(C(c2n[nH]c(C)c2C)=O)C(C)CN(C(c2cc3scnc3[nH]2)=O)CC1C C1(C)(OC)C(OC(=O)C(c2cc(F)cc(F)c2)(F)F)CC1(F)F N1(C(C(CCC)OCC)=O)CCC(C2CCN(C(=O)CNC(=O)COC)C2)CC1 c1(C(=O)NCCC2CCN(C(C3N(C)C(C(N)=O)CC3)=O)C2)ccc(F)c(F)c1 CCC(C)C(O)C(C)C(=O)N1CCC(C(=O)NCC2CN(C3CC3)C2)C1 C1(NC(c2ccnc(O)c2)=O)CCN(C(c2cc(CC3CC3)on2)=O)CC1CO c1(C(=O)N)cncc(C(=O)NCC(C)(C)OCCOCC2CC2)n1.CN S(=O)(=O)(c1cc(C)cc(Br)c1)NC(C#C)(C)C1CC1 C1(C(N(CCNC(=O)C(C)n2cncn2)CC)=O)CCCCC1(F)F N1(C(c2c(CC)oc(C)c2)=O)CCN(C(c2cc(F)cnc2Cl)=O)CCC1C C1(C(N(C2CC2)CC)=O)CC(O)CN1C(=O)CC1CCOCC1 N1(C(CNC(CC)=O)=O)CC2CC(N(C(=O)CC34CCC(CC3)C4)CC)CC1C2 O=C(CCS(=O)(=O)C(F)(F)F)N1CC2CC(O)CC1C2 c1(C(C)=O)cccc(NC(=O)CCc2scnc2C)c1.c12ccc(cc1)[nH]c2=O N=c1cc(CC(=O)NC2CC(CNC(C3(CC4CCC4)CC3)=O)C(O)C2)cc[nH]1 c1(NC(C(CC2CN(C(C=C(CCC)C)=O)C2)F)=O)cnn(C)c1COC c1(C(=O)NC2(C)CC(NC(C(C)OCCC(C)C)=O)C2)ccc(F)c(N)c1 N1(C(c2ccc(C)cc2)=O)CCC(C2CCCN(C(c3cnccc3C)=O)C2)C1 c1(C(=O)NC(CNC(c2cnc(OC)nc2)=O)C)cc(Cl)c(OC)c(Cl)c1 C1(CNC(=O)CCC2CCCCO2)CCCN1Cc1ncnn1-c1ccccc1 c1(NCC(c2nccs2)C)cc(Br)ccc1S(=O)(=O)N1CCC(C)(C)CC1 N1(C(C(C)OC2COC2)=O)CC2(CCN(C(c3cnc[nH]3)=O)C2)C1 C12CCC(CC1)C=CC(=O)C2=O.C1(NC(C=CC(=O)OC(C)(C)C)=O)CC(NNC)C1.N c1(NC(=O)C(n2cc(-c3ccc(C(F)(F)F)cc3)nn2)C)cccc(OC)c1.CO c1(C(N2CCCC(NC(CCC(=O)NCC)=O)C2C)=O)c[nH]c2c(Cl)cccc12 C1(C(N(CC(=O)N(C)C)C)=O)CC12CCN(CC1OCCC1(C)C)CC2 C1(C(C)C)CN(C(=O)CN(C2CCC2)C)CCN1C(=O)C(C)Cc1ccncc1 C(=O)(CC(c1ccccc1)N(C)C)NC1C(NC(C2(OC)CC2)=O)CC1 c1(C(N2C(Cn3cc(COC)nn3)CCCC2)=O)cc2oc(C)c(C)c2[nH]1 Nc1c(F)ccc(Cl)c1C(=O)NCC1(F)CCCN(C(c2ccc(Cl)s2)=O)C1 N1C(=NCC#Cc2cnn(C)c2)NCC2CC1(CCOCC(C=C)C)C2 C1(NC(c2c(COC)n(C)nc2)=O)CCCCN(C(c2csc3cncn23)=O)C1 CC(C)CC(C)C(=O)NCC(C(N1CCC(N(C)C)C(C)C1)=O)C1CC1 Cc1cc(F)c(C(N2CC(C(=O)NCCCC(F)(F)F)CC(F)C2)=O)cc1F c1(C(=O)NCC2CN(C(C3CCC(CC)CC3)=O)C2)ncc(C(F)(F)F)cc1Cl c1(C(N2C(C)CC(NC(C3(CCF)CC3)=O)CC2)=O)ccn2c1CCCC2 C(=O)(CC(C)(C)O)N(C1CCN(C(=O)CCCc2nncn2C)C1)CCC Cc1oc(Br)cc1NC1(c2nnnn2C2CCC(C)C2)CCCCC1 N=c1[nH]c(CC(=O)NCCCNC(c2ccc(-c3ccccn3)o2)=O)cs1 c1(C(N2CC3CN(C(c4c(O)cccc4Br)=O)C3C2)=O)nc2ccccc2[nH]1 c1(C(N2C(CNC(COC)=O)CCC2)=O)cccc(N2CCN(C)CC2)n1 CCCC(C)CC(C)NC(=O)NCC#CC1CCCCO1 c1(SC)nc(C)c(CC(=O)NCC2C=CCN2C(C2CCCOC2C(C)C)=O)s1 c1(OC)c(C(=O)NCC2CN(C(=O)Cc3ccccc3O)CCO2)csc1Cl N1(C(C2ON=C(C)C2)=O)CCC(O)(CN(C(=O)CCOC2CCCOC2)C)CC1 n12nnnc1C2.C12COCC1NC(=O)N2.CC(C)(C)OC(=O)NC1(C(F)F)CC1 c1(NCC(C)N(C(=O)C(O)C2CCC2)C)ncnc2sc3c(c12)CCCC3 Cc1cc(O)cc(C)c1CS(=O)(=O)NCC1CCN(c2ccc(C(N)=O)nn2)CC1 c1(C(=O)NCCC2(NC(c3cc(C)c(Cl)cc3)=O)CCC2)cccn2nncc12 c1(NCCc2ccc(SCCC)cc2)cc(C)cc2c[nH]nc12 c1(OC)ccc(C(=O)NC(C)CCCNC(c2snnc2C2CCC2)=O)c(Cl)n1 c1(C(N2CCC(NC(C(CO)NC(N)=O)=O)C2)=O)cc2ccc(Cl)cc2[nH]1 C(CC(C(C)C)Nc1ccc(I)c(C)c1)(OC)OC C(CN=c1[nH]c(N2CCCC(N3CCCC3)C2)nc2c1CCC2)N(C(=O)OC)C CC1=NNC(=O)C1CC(=O)NC(C1CCN(C(c2nnc(S)n2C)=O)CC1)CO n1(CC(=C)C)nnnc1C(c1ccnn1COC)NCCCC1CCCO1 c1(CC(=O)NCCC2CN(C(=O)C=C3CCC3)CCO2)ccc2c(c1)OCCO2 Cc1cc(F)c(C(N2CC(C(C)NC(c3cccc(=O)n3C)=O)C2)=O)c(F)c1 c1(C(N2CCCC(NC(C3CC(n4cccn4)C3)=O)C2)=O)cncc(Cl)c1Cl CCCC(C)CC(=O)N1CCCCC1CNC(c1cc2scnc2[nH]1)=O Cc1ccc(N)c(C(N2CC(C)(NC(=O)C(N3CCSCC3)C)C2)=O)c1 CCCCC(CC(=O)N(C1CC2CC2C1)C)NC(=O)CCn1cnnn1 c1(NC(N2C(C)(C)COCC2)=O)ccnc(S(C)(=O)=O)c1 C(CC(C(=O)N1CCC(N(C(=O)Cc2nnc(C)o2)CCO)CC1)NC=O)SC C1(C(=O)NCc2ccc(CNC(C)=O)c(F)c2)CCCC2(C1)CC2(F)F c1(C(=O)NC2C(C)CN(C(c3cc4ncsc4[nH]3)=O)C2)ccc(O)c(O)c1 C1(C(c2ccc(F)cc2)C)CC2CCC1CC2.c12cc(nc(C)n1)C(=O)NC2NC c1(C(=O)NC(CC(=O)OCC)C)n[nH]c2c1CN(Cc1cnc(CC3CC3)s1)C2 CC1CCc2n[nH]cc2C1C(=O)NCC1CN(C(c2ccc(F)c(F)c2)=O)C1 c1(CC)nn(C)cc1C(=O)NC(C)C(C)C(=O)NCC1CC1Cl CC(C)CC(C(=O)N1CCC2(C1)CN(C(C13CC1COC3(C)C)=O)C2)C(C)C N1(c2nc(C)nc(=N)[nH]2)CCC2(CC1)CN(C(C1(O)CC1)=O)CC2CO Cc1nccn1CC(=O)NCc1ccoc1C(=O)NC(C)CC(C)O c1(C(C)C)ccc(C(=O)NCCC2CCN(C(c3cnc(O)o3)=O)C2)s1 c1(CC(=O)NCC2(O)CC(CNC(CC(C(C)C)C)=O)C2)ccc2n[nH]cc2c1 c1(OC)ccc2[nH]c(CN3CCC4OCCN(CCOC(C)=O)C4C3)c(C)c2c1 C1(C(=O)NCC(O)CN(C)C2CC2)(CNC(CCC=C)=O)CC2(CC2)C1 Cc1coc(C)c1C(=O)NCC12CC1CN(C(=O)C(C)CSC(F)(F)F)C2 Cc1c(C(N2CCCC(C(C)NC(c3cnoc3)=O)C2)=O)cccc1[N+](=O)[O-] c1(C(N(C)CC2(O)CCN(C(C(C)CN(C)C)=O)CC2)=O)cnc([N+](=O)[O-])n1C CC(C(CCc1ccccc1)NC(c1cccc(Cl)c1)=O)NC(=O)CC1(O)CC1 C1(CNC(C2C(=C)C2)=O)C(C)CCCN1C(C1CCN(S(C)(=O)=O)CC1)=O C(CN=c1cc[nH]cc1S(=O)(=O)N(CC(C)CCO)CCC#N)SC CCC(C(=O)NCC(C)NC(=O)C=Cc1cn(C)nn1)C(C)(F)F c1(C(=O)NC(CN(C(c2nn(C)c(C)c2Cl)=O)CC)C)ccc(C)nc1N CC1CCN(C(=O)CC2CCC(C)C2)C1CNC(c1ccc(N(C)C)cc1)=O c1(C(=O)NCC(C)N(C(CCOC(C)C)=O)C)cccc(N(C)C)c1.C1(COC)CC1 C(=O)(C(C)CC(C)(F)F)NC(C1CN(C(=O)CCc2cc(F)cc(F)c2)C1)C c1(C(=O)NC(C)C(C)NC(=O)C#CC2CC2)c(C(F)F)nc2ccccn12 N1(C(CC2C(C)C2)=O)CCC(C)(CNC(c2cc(Br)no2)=O)C1 C1(NC(CC(C)NC(N)=O)=O)CN(C(=O)CN(C)C)C(C)(C)C1 c1(C(=O)NCC(C)NC(CC2(C=C)CCOCC2)=O)cc(Cl)c(Cl)cc1O CCC(C(=O)NCC1CN(CC(=O)NC2CC2CC)C1)n1cncn1 C1(C(=O)NC2CC(N(C)C(c3ccc(Cl)o3)=O)C2)COCC2(CCC2)O1 C1(CC)C(NC(c2cc(C(C)(F)F)on2)=O)CCN1C(=O)C(C)COCC C(CCC(CO)NC(C1CN(C)CCO1)=O)NC(C(C)SC(F)(F)F)=O N1(C(CCC(CC)OC)=O)CCC2(CCC(NC(c3cc(C)sn3)=O)C2)C1 C1(CNC(C2CCC2)=O)CC2(CO1)CN(C(=O)C(c1ccc(Br)cc1)O)C2 C1(NC(c2ccnc(N(C)C)n2)=O)CCCN(C(=O)CCC(=O)C2CC2)CC1 COC=CC(=O)NCCC(=O)NC1CC(CNC(=O)CSCC(N)=O)C1 CC1=C(C(=O)NCC2CC3(CCC3)CN2C(=O)C(O)C(C)C)CCCC1 C1(NC(c2ccc(C)nc2O)=O)CN(C(=O)CC(C)P(C)(C)=O)CC(C)(C)C1 C1(NC(c2n(CC)cc(Br)c2)=O)CC(O)CN(C(=O)Cc2cnccn2)C1 C(=O)(C(C(C)(C)C)n1ccnn1)N1CCC(C(C(C)C)NC(c2ccc[nH]2)=O)CC1 C(=O)(C1Cc2ccccc21)N1CC(C(=O)N(N2CCCOCC2)C)C(O)CC1 N1(C(CCCC(CC)CC)=O)CC2CN(C(c3cc(CC)[nH]n3)=O)CC(C1)O2 C(=O)(CCC(C)(C)NC(C1CCCCS1)=O)N1CC(CC)C(F)C1 N1(C(C(CC)C)=O)CC(CNC(c2cccc(F)c2)=O)OC2(CCC2)C1 C1(CNC(C(C2CCN(C(C(COC)C)=O)C2)C)=O)CC1C1CCC1 C=C1CC2(C1)CC(C(=O)NCC1(O)CCCN(C(=O)CCN(C)C(C)=O)C1)C2 N1(C(Cc2c(C)ccnc2)=O)CC2CCN(C(c3cc(C#N)c[nH]3)=O)CC2C1 C1(P(C)(C)=O)(C(=O)NCCCNC(C2C(C)(COC)C2)=O)CC1 S(=O)(=O)(c1cccc(-c2cc[nH]n2)c1)N(C1CCCC1)C1C(C)C1 C1(NC(C(C)(CO)NC(c2cccc(C#C)c2)=O)=O)CCCC2(CC1)CC2 c1(NC(C(c2ccc(Cl)cc2)NC(C(C=C)O)=O)C)nccc(SC)n1 c1(CC(=O)NCC2N(C(CC(=O)OC)=O)CCC2C2CC2)ccc2c(c1)NC(=O)C2 c1(C(N2CCC(NC(CN(C(C)=O)C)=O)C(O)C2)=O)cc(Cl)c2ccncc2n1 C(=O)(CC(C)(C)C(=O)NC(CO)C(=O)NCCCc1ccncc1)OC c1(C(=O)NC(CC=CC)C(=O)NCCC#CCC)cc(C)c(C)cn1 C1(NC(CNC(=O)NC)=O)CC=C(C(=O)NCC(C)C2CCC2)C1 C1(C)(NCc2cccc(-c3nc(NC(C)=O)sc3)c2)CCC(=O)NC1=O CC1=C(C(=O)NC2CCC(NC(c3coc(O)n3)=O)C2)CCO1 c1(OC)ncc(Cl)c(C)c1C(N1CCCC(N(C)C(c2cc(C)n(C)n2)=O)C1)=O C1(NC(CCOCCOC)=O)CN(C(=O)CSCC2CCCO2)CC2(CC2)C1 N1(C(CNC(C)=O)=O)CCCC1CC(=O)NCc1[nH]cnc1C CSC=CC(=O)NC(C)CC1CN(C(=O)CCSCC(C)C)C1 c1(OCCOC)cc(OC)ccc1C(N1CCC(CCNC(=O)C(C)O)C1)=O C(=O)(C(C)(C)CF)NC(C)CCNC(C1CC1c1cnn(C)c1)=O C1(CNC(C(C)(F)F)=O)CN(C(c2cnc3n2CCOC3)=O)C2CCCCC12 C1(CC#C)(C(=O)NCC2(C)CC(C)(C)C2)CCN(C(=O)C(C2CCC2)OC)C1 N(C1c2ccccc2CC1NC(C1CCCCC1)=O)C(C1(C=C)CCCCC1)=O N1(C(C(CCOC)C)=O)CCCC(C2CN(C(c3c[nH]nc3C(F)(F)F)=O)C2)C1 N1(CCCC(=O)NCC2CN(C(C(COC)C)=O)CC2O)CCc2ccccc21 c1(CC)ccc(C(N2CCN(C)C(CNC(=O)C(F)=C(C)C)C2)=O)c(Cl)c1 C(=O)(CC(C)C(F)F)N(C1N(C(C(=O)N(CC)CC)C)CCC1)CC C1(C(=O)NC(CCN(CC)CC)C)CCN(C(c2csc(C)n2)=O)C12CCC2 N1(C(C2C(NC(C3C(C=C)OCC3)=O)CCO2)=O)CCC(C)C(C)(C)C1 C1(NC(=O)C=CC2CC2)CCC12CN(C(c1cc(O)nc(O)c1)=O)C2 Cc1nc(CO)sc1C(=O)NCCc1ocnc1CNC(C1CCC1C)=O N1(C(C2(CC#C)CCCC2)=O)C(C(=O)NC2CCCCC2(F)F)C2CC(O)C1C2 C12(C(N3CC(COC)OCC3)=O)CCC(NC(C3COCOC3)=O)(CC1)C2 C(=O)(CC1=CCN(C(c2cc(C)cc(F)c2)=O)CC1)NC(CC(CC)C)CO CN1CCC(C(=O)NCCC2(O)CCN(C(c3ncn(C)n3)=O)C2)S1(=O)=O N1(C(c2ccc(OC)nn2)=O)CC(NC(C2CCC2)=O)CC(C)(C)C1 C=CC(O)C(=O)N1CCCC1CC(c1ccccc1)O.n12cc(nn1)C2(C)C CCC(C#N)(CC)C(=O)NC1CC12CCC(O)CC2 c1(NC(c2occ(C)c2)=O)ccc(NC(=O)CC2CCCN(C)C2)cc1C c1(C(=O)NC2CN(C(c3c(C)nc(=N)[nH]c3)=O)C2)cc2c(F)cc(Br)cc2[nH]1 Cc1ccnc(O)c1C(N1CCN(C(=O)CNC(C2CC3(CC3)CO2)=O)CC1)=O N1(C(CC2(OC)CCCC2)=O)CCN(C(=O)C=C2CCN(C)CC2)C(COC)C1 N1(C(C2C(C)C2(F)F)=O)CCCC2(C1)CN(C(=O)CC(O)Cc1ccccc1)C2 N1(C(C(COC)C)=O)CCC(NC(=O)CN2CC(=O)N(C)C2=O)C12CC2 CC(C)CC(C)CC(=O)NC1CN(C(C2CC(=O)N(C3CC3)C2)=O)C1 N#Cc1ccc(C(N2CCCCC2CCNC(=O)CC2CCOCC2)=O)[nH]1 N1(C(C2=CCCC2(C)C)=O)CCC2C(C1)CN2C(C1CCC(C)(F)CC1)=O C1(N(C(N(C)CCO)=O)C)CCN(C)C1 c1(C(=O)NCCN(C(c2cc(OC)ccn2)=O)CC)ccc2c(c1)C(C)CO2 Cc1nn(CC(N2CCCCC(NC(c3cnc(C4CC4)s3)=O)C2)=O)c(=O)n1C c1(SC)nc(NC)cc(C)n1.C12CN(CC1C#C)c1cc(ncn1)OCCOC2.OCC C1(NC(Cc2c(C)scc2)=O)CN(C(C2(O)CCCCCC2)=O)CC2CCCC12 CN(O)C(=O)CNC(c1c[nH]nc1CCNC(c1c[nH]nc1C(F)F)=O)=O CC1(C#CC(=O)NCC2(F)CN(C(C3CN(CC(F)(F)F)C3)=O)C2)CCCO1 Cc1nccc(=NC(C)C2CN(C(=O)CCc3ccccc3Cl)CCO2)[nH]1 Cc1ccc(SCC(N2CCC(NC(C34COCC(C3)C4)=O)CC2)=O)cc1 c1(OC)cc(C)sc1C(=O)NC(C1CCCC1)CNC(C1CC(C)(C)O1)=O c1(C(=O)NCC(CC=C)NC(c2cc(Br)oc2C)=O)cccc(CCO)c1 c1(CCC(=O)N(C)CC2N(C(C(C)=CC)=O)CCC2)cc(C)sc1C C1(NC(C(=O)N(C)C)=O)CC2(C(=O)NCCC(O)CO)COC1C2 N1(C(c2cnc(C)[nH]2)=O)CCN(C(=O)CC(C)(C)CN(C)C)CC1C CC1OC(C)CC1C(=O)NC1CN(C(c2cccc(N3C(=O)CCC3=O)c2)=O)C1 c1(C(=O)NCC(C)NC(=O)CN2OC(C)(C)CC2=O)csc([N+](=O)[O-])c1 C1(C(N2CCC(OC)(CNC(c3cc[n+]([O-])cc3)=O)C2)=O)CCS(=O)(=O)C1(C)C n1(C(C)(C)C)ncc(C(=O)NCC2CC(NC(C3(C)CC3F)=O)C2)c1N N1(C(c2ccc(OC)cn2)=O)CCOC2(C1)CN(C(C1CC(F)(CO)C1)=O)C2 C(C(C)(C)C(=O)NC1CCN(C(=O)CC2COCCO2)CC1)NC(CC(C)C)=O c1(C(=O)NCCCCCNC(C2CCC(CC)O2)=O)cc(F)ccc1C1CC1 C(=O)(CC(F)F)NC(COCCCNC(C(C)N(C)C)=O)(C)C c1(OC)ccc(Cl)c(C(=O)NCC(CNC(c2c[nH]cc2Br)=O)OC)c1F N1(C(Cc2cnc(C)s2)=O)CCN(C)CC1CNC(c1c[nH]nc1Cl)=O CC(C)(C#N)CC(=O)NCC(C)(C)CNC(C1CC(CCF)C1)=O c1(C(=O)NCC(CN(C(c2c(C)c[nH]c2)=O)C)C)cncc(C(F)(F)F)n1 CCCC(C)(O)C(=O)N1CCC(C(=O)NCCN2CCC3CC23)C1 CCCCCC(O)CC(=O)NCCNC(=O)CCc1ccc(C#N)cc1 c1(CC(C)N2C3(CCNCC3)C2=O)ccccc1C.N(C)C.CCO N1(C(C2C(C(N)=O)C2)=O)CCC(NC(C2CC(N3CCCC3)C2)=O)C12CC2 c1(CC(=O)NCC(CC=C)NC(=O)CN2CC=CC2)cccc(C(C)C)c1 c1(C2(C)CC2C(N2CCC(NC(=O)Cn3nnc(=O)[nH]3)C2)=O)ccc(Cl)cc1 C(=O)(CCCCCC(C)C)NC(CCCCNC(C(CC)n1ccnc1)=O)CO C1(NC(C(C)N(C)C)=O)CN(C(C2CCCC2(C)C)=O)CC1CO N1(C(C2C(=C)C2)=O)CCC2(CC1)CN(C(=O)CC1CC3(CC3)CO1)C2 c1(C(=O)NC(CCNC(C(C(=O)OCC)F)=O)C)sc2cc(C)ccc2c1Cl c1(C(=O)NC2C(CNC(CC=C(C)C)=O)CCCC2)c(F)ccc(O)c1F C(C)(C(CO)NC(=O)C(C)n1ccnn1)NC(CNS(CC)(=O)=O)=O c1(C(=O)NCC2C(NC(Cc3c(C)cco3)=O)C2)nnc(S)n1C c1(N(C)C)ccc(NCCNC(=O)CCC2(C)N=N2)nn1 c1(N2CC(F)CC(C(=O)NCc3c(OC)nccc3)C2)ncnc2ccsc12 C12(C(=O)NCC3C(CCC)C3)CC(CO1)N(C(c1cocc1C)=O)C2 Cc1cc(=NC2CCCC3CN(C(C4CC(F)(CO)C4)=O)CC23)[nH]c(Cl)n1 CC1(C)C(C)(C)C1(F)C(N1CCC2(NC(c3ccc(Cl)c(F)c3)=O)CC2C1)=O C1(C(=O)Nc2c(CC)csc2)CN(C(=O)CCCC(=O)N(C)C)CCN1C C1(NC(C(c2cccnc2)OC)=O)CCN(C(=O)C=Cc2ccsc2)C(C)C1 c1(C(N)=O)cc(F)ccc1C(=O)NC1CCCN(C(=O)CCc2ccco2)C1 C(CC(=O)N(CCC(C)O)C)(C(F)F)NC(C1=CC(C)(CC)C1)=O c1(OCCC(=O)NCC(C)N(C(C(C)SCCCC)=O)C)cccc(F)c1 c1(C(N2CCCC(C#C)(O)C2)=O)cc2ccc(COC(=O)C(F)(F)F)cc2o1 C(CO)(CO)(C(=O)O)NC(c1ccc(NCc2ccccc2I)cc1)=O N1(C(C(C)C)=O)CCC(CCNC(=O)Cc2nc(-c3ccccc3)n[nH]2)CC1C N1(C(C(C)(C)NC(c2ccc[nH]2)=O)=O)CCN2C(=O)NCC2C1 c1(C(=O)OC)nc(N2CCCC2CNC(=O)Cc2cccnc2)[nH]c2ncnc1-2 CCCCC(F)C(=O)NC(C)(C(=O)NC1(CCCC)CC1)C1CCC1 N1(C(C2CCC(C)C2)=O)CC2(CCC2)CC1CNC(=O)C=C1CN2CCC1CC2 c1(C(=O)NCCO)nccc(Cl)c1O.c1(S)cc(C(=O)N(C)CCOCC)ccn1 C=CCC(CC)C(=O)NC1CC(NC(c2ccc(=O)n(C)n2)=O)C1 N1(CC)CCOC(CNC(=O)Nc2ccc(OCC)cc2)C1.C(C)(C)O c1(C(CC(=O)NCCC(C)N(C)C(C2CC2C(N)=O)=O)C)ccccc1Cl c1(N2CC=C(C)CC2)cc(N2CCC(OC(C)C)C2)nc(C(C)COC(C)(C)C)n1 C1(CNC(c2ccc(C)cc2)=O)CCN(C(=O)C(F)(F)c2csc(=N)[nH]2)CC1C C1(OC)CCN(C(=O)CCC2CCC(NC(c3cnc(O)cc3C)=O)C2)C(C)C1 C1(CCNC(C2N(C(N)=O)CCC2)=O)CCCN(C(=O)CCC2OCCO2)C1 CC(C)(C)CCCCC(=O)NCCCNC(c1cc(Cl)c(Cl)s1)=O C(C(C)C)(C(O)C(=O)NCc1cc(C(N2C3COCC2C3)=O)ccn1)OC Cc1cc(C(=O)NCCC(C)N(C(=O)C=CS(C)=O)C)n(C(F)F)n1 N1(C(c2nc(CC)oc2)=O)CCCC12CCN(C(c1cc(C(N)=O)co1)=O)CC2 C1(C(=O)NCCN2CC3CC3C2)CCC2(CC2)N1C(C1CCCCO1)=O CCC(C)(C(=O)N1CCC(O)(CCNC(=O)CC2CCCC23CC3)CC1)C(N)=O c1(OC)ccc(CN2CCC(CNC(=O)C(C)n3cccn3)C2)cc1Cl N1(C(C(c2ccc(C)o2)C)=O)CCC2CCN(C(=O)C(O)CC3CC3)C2C1 CCC(CC(C)C)C(=O)N(CC(CC)NC(c1ncc(F)cc1C)=O)C Cc1ncc(C(=O)NC2CN(C(=O)CC3CC=CCC3)CC2(C)C)cc1N C1(OC)(CNC(=O)CCC#N)CN(C(C2CN(C(N)=O)C2)=O)C1 C(CC(C)CC(C)(C)C)NC(C(=O)Nc1ncc(CCC=C)cn1)=O CN(C(=NCCNS(C)(=O)=O)NCc1ncc(Br)s1)Cc1ccsc1 C12CCN(CC1)C(=O)N2C.c1(C(=O)OC)ncc(OC(C)=O)s1 C1(CC=C)(C(=O)OCC)CN(c2cc(C)nc(SC(C)(C)C)n2)CCO1 C(CC(N)=O)(C(=O)NCCC(=O)NC1COC(C(C)C)C1)NC(C)=O C1(C)(CNC(CCCC#C)=O)CN(C(C2CC3(CCCO3)C2)=O)CC1C O=C(CS(=O)c1ccc([N+](=O)[O-])cc1)N(C1CC1)C1CC1.C12COCCN1C(=O)C2 C1(C)(C(=O)Nc2c(CC)cccc2)CCCN(C(c2ncccn2)=O)C1 C12(NC(C3(OC)CCN(C(c4nc(CC)oc4C)=O)C3)=O)COCC1C2(F)F c1(CNC(C2CCC(O)(C(F)(F)F)C2)=O)cccnc1N1CCCCC1 Cc1nsc(N)c1C(=O)N(CCCCCNC(=O)C(C(C)C)n1cnnc1)C N1(C(C(C2CCN(C(COCCOC)=O)C2)(C)C)=O)CC(CO)C(C)(C)C1 N1(C(=O)NCC=CCCCC)CCC2CCCN(C(=O)OC(C)(C)C)C2C1 C=C=CC(C)C(=O)N1CC(O)CC1C(=O)NC(C)C(=O)NC(C)C C1(CN(C(=O)Cc2cc(C)[nH]n2)CC)CCCN(C(=O)CSC(C)(C)C)C1 C(=O)(CC(O)CNC(=O)CCC(=O)N(C)C)NC(c1ccccc1)CC c1(C(=O)NC2C(SC)CN(C(c3c[nH]ccc3=O)=O)C2)snc2ccccc12 N1(C(COC(C(c2ccc(Br)cn2)(C)C)=O)=O)Cc2ccccc2C1 c1(C(=O)NC2C(OC)CN(C(c3cnc(SC)s3)=O)C2)cccc(SC)c1Cl Cc1cc(C(=O)NC(C2CCCN2C(c2cc(F)cc(F)c2)=O)C)cc(F)c1 c1(OC)cc(NC(c2c(NC(=O)CC(C)C)sc(C)c2C)=O)cc(OC)n1 N1(C(C2CC(OC)C2)=O)CCSCC1CCNC(=O)CSCC1CCCCO1 c1(NCC2C(NC(c3nc(OC)oc3)=O)CCCC2)ncc2scc(Br)c2n1 C1(NC(c2nc(C)[nH]c2C(F)(F)F)=O)CCN(C(=O)CC2CCCC2)CC1C n1(CC)cnc2[nH]c(=NC3CCOC(C4CC4)C3)nc(N3CCC4(CC4)C3)c12 N(C1CCc2ccc(C)c(C)c21)C(=O)N(c1ccc(S(C)(=O)=O)c(C)c1)C(CC)=O c1(C(N2C(CNC(CNC(c3ccccc3Cl)=O)=O)CC2)=O)cc(CO)ccc1F c1(C(=O)NC2COCC2NC(C2CC2(F)F)=O)snc2ccccc12 C(=O)(C(C)(C)CCNC(c1cnn(CCO)c1)=O)NC(CC)CN(C)C c1(C(=O)NC(CN(C(c2cc(C(=O)OCC)ccn2)=O)CC)C)ccncc1Cl C1(CNC(C2CN(C(CCCOCCOC)=O)CC2CC)=O)OC(=O)NC1(C)C N1(C(Cc2c(Br)cn(CC)n2)=O)CCN(C(C2CCO2)=O)C(C(C)(C)C)C1 C=CCCC(C(=O)N1CC(C)(C(=O)NC)C1)NC(c1cnc(CC)o1)=O c1(CC)cnnc(NC(CN(C(c2c(OC(C)=O)cccc2)=O)C)CC)c1 C1(C(C(=O)NC2(CCOCC)CCC2)SC2(CNC(=O)CF)CC2)CCCCC1 c1(CN(C)C)ccc(CNC(c2ccccc2OC(F)(F)F)=O)cn1 C12(COC)CN(C(C3CCNC(=O)C3)=O)C(CNC(C3(C)CCC(=O)N3)=O)(C1)C2 N1(C(c2nn(C)c3c2CCC3)=O)CC2CCN(C(C3CCS3(=O)=O)=O)CCC2C1 C1(NC(CCOCCOC)=O)CC(C2CCN(C(C3COC(=O)N3)=O)CC2)C1 c1(C(N(C)CC2(O)CCCN(C(C3CCCS3)=O)C2)=O)nn2cccnc2c1Cl C1(CC)CN(C(=O)Cn2cnnn2)CCN1Cc1cccc(C(F)(F)F)c1 C(CCCN=c1[nH]c(N2CCC(O)CC2)nc(=N)[nH]1)NC Cc1ccn2cc(C(=O)N(C)CCNC(c3sncc3C)=O)nc2c1 Cc1c(NC(CNC2CC2)C(C)C)ncnc1NS(C)(=O)=O.C12CC(C1)N2 N1(C(CCC)=O)CC2CC(C1)CN(C(C1CC(C)(F)C1)=O)C2 c1(OCC(=O)N(CC(C)NC(c2cscc2C(F)F)=O)C2CC2)ccc(F)cc1 C(=O)(CC(O)CNC(=O)OC(C)(C)C)N1C(Cn2cc(-c3c(C)ccs3)nn2)CC1 N1(C(C(C)N(C(C)=O)C)=O)CCC2C1CCN2C(c1cc(I)ccc1Cl)=O c1(CC)cc(NC(c2cccc(-c3noc(C)n3)c2)=O)cc(C)c1 N1(C(CC2(C)CC2(F)Cl)=O)CC2CCC(C1)N2C(c1cncc(N)c1)=O c1(C(=O)NC2CC(O)(CNC(C3CC(N4CCCC4)C3)=O)C2)ccc2c(c1)CC2 C1(NC(c2c(CNC(c3ccsc3)=O)occ2)=O)CC1C1CCCC1 Cc1nc(CCC(=O)NCCC(C)NC(=O)C(C)NS(C)(=O)=O)[nH]c1C Cc1nocc1CNC(c1occc1CNC(=O)COC1CCOCC1)=O C=C(C)C(C)(O)C(=O)NC(CNC(=O)Cn1nnc(C)n1)CCOC C1(CN2CCN(c3c(C#N)cc(F)cc3)CC2)CC2(CCOCC2)C(=O)O1 N1(C(CCc2cc(OC)c(Cl)cc2)=O)C2CCC1c1cncnc1C2 Cc1cncc(C(C(=O)NC2CCC2C)N(C)Cc2cccc(Br)c2)c1 Cc1c(C(F)(F)F)cnn1-c1ccc(C(=O)OCC2CC2)cc1.C1(C)C(=O)N1 N1(C(Cn2cc(CCCC)nn2)=O)CCOC(C(=O)OC)C1 C12(CNC(CCCCC#C)=O)CN(C(=O)CC3CCCO3)CC1CS(=O)(=O)C2 C(=O)(C(O)C1=CCCCC1)NCCC1OCCN(C(C(CCC)O)=O)C1 c1(NC(C(CCC=C)NC(=O)C(CC2CCCC2)CC)=O)cc(C)c(O)cc1C c1(NC(C(c2cnn(C)c2)NC(C)=O)=O)c(C(C)(C)C)nsc1-c1nn[nH]n1 N1(C(C(CCC)CC)=O)CCC(NC(=O)CC2(C)CC2(Cl)Cl)C(CO)CC1 c1(C(N2C(C)CC(NC(c3cc(COC)[nH]n3)=O)C2)=O)cc2n(c1)CCOC2 CC(CC(F)(F)F)C(=O)N(C(C)C(N1CCCC(F)(F)CC1)=O)C1CC1 Cn1ncc(Cl)c1C(=O)NCCOCCNc1nccc(CO)n1 C1(OC)CC(C(=O)NC2C3CC(NC(C4CCCN4C(C)C)=O)CC23)C12CCC2 C1(CC)CCN(C(c2cnn(C)c2N)=O)C1CNC(=O)CCc1ccc(C)s1 C1(C(N(CCCCN(C)C(C2(O)CCC2)=O)C)=O)CCCC(C)(C)CC1 C12(C)CN(C(C)(C)C1)N(C1OCCC1C)C2.C1(C(=O)OC)C=CCN1SC12CC(C1)C2 C1(C(=O)NC(c2cccs2)(C)C)CN(C(=O)C=C(C2CC2)C2CC2)CC12CC2 S(=O)(=O)(c1ccc(N(CCCS(N)(=O)=O)C)c(Br)c1)NC(CC)CO c1(OC)ccc(F)c(C(N2CCC(C(C)(C)NC(=O)CS(N)(=O)=O)C2)=O)n1 Cc1ccc(COCC(=O)NCC2COCCN2C(=O)C(F)C(C)C)cc1 c1(CCNC(C2N(S(CC=C)(=O)=O)CCC2)=O)cc(I)ccc1F c1(C(N2C(CNC(COCCC#C)=O)C=CC2)=O)ccc(F)c(Cl)c1N c1(N)nc(Cl)nc(Cl)n1.c1(C(=O)OC)ccc(CNC(CC2N(C=O)CCC2)=O)[nH]1 CN1CC2(CCN(c3ncn(C)c3Br)C2)CC1=O C1(C(=O)NCCC(C)N(C)C(c2cc3ccsc3n2C)=O)Cc2nccnc2C1 n1(CCC(=O)NCCC2CCC(NC(c3c(OC)csc3)=O)C2)c(C)ccc1C c1(CNC(C(COC)(C)C)=O)ccc2c(c1)CN(C(=O)Cc1c(C)noc1Cl)C2 C1(NC(c2cncnc2)=O)CC2CC(NC(C3(n4cccc4)CCCC3)=O)C2C1 c1(C(=O)NC(C2CCN(C(=O)CCc3nc[nH]n3)C2)C)c(N)cc(Cl)nc1Cl Cc1cccc(CN2CC(NCc3ccccc3O)C2)c1Cl N1(C(c2c(C)[nH]cc2)=O)CCN(C(=O)CC2SC(=N)NC2=O)CC(O)C1 c1(C(N(CCCNC(CC(CC)CN(C)C)=O)C2CC2)=O)ccn2c(C)cnc2c1 C1(N2CCCN(Cc3cc(C)[nH]n3)CC2)CC2CC3CC(C2)CC1C3 C(C1=CCN(C(c2cnn(C3CC3)c2C)=O)CC1)NC(Cn1c(C)csc1=O)=O N1(C(c2c(OC)ccs2)C(=O)NCCCC2CC2)CCC2CCCC2C1 N1(CCC(=O)NC2C(NC(C3C(COC)CC3)=O)CC2)CCCC1=O C(=O)(C1CCc2ccccc21)NC1(C)CCN(C(c2ccc(N(C)C)cc2)=O)C1 C(CC(C(C)(C)C)NC(C1C(C)(C)C1(C)C)=O)N(C(Cc1c(C)ocn1)=O)C c1(C(=O)NCC(CN(C(C(C)OCC)=O)C)(C)C)cc(C)nn1CC(F)(F)F c1(CC(N2CC(C(C)NC(C(C(C)C)N(C)C)=O)(CO)C2)=O)coc2ccccc12 Cc1ccc(SCc2cn(CCCC(=O)NC3CC(=O)NC3=O)nn2)n1C Cc1csc(C(=O)N(C(C)CNC(c2ccc(C(F)(F)F)nn2)=O)C)c1C N1(C(c2occ(C)c2)=O)CCC(C(O)CNC(C2CCCC(=O)C2)=O)CC1 N1(C(=O)NC(C)C(C)(C)C)CCC(CSc2ccc(Cl)cc2)CC1 C=CCCC(C)(C)C(=O)NCCC1(O)CN(C(C2OC3CCC2C3)=O)C1 CN1CCC2CCN(C(C3CCN(C(=O)C4=CC(C)(C)C4)C3(C)C)=O)C2C1 C(CC(=O)NCCC(=O)OCCC)(C(F)(F)F)NC(C(C=C)OC)=O c1(C(C)C(=O)N(CCCNC(=O)CN(C)C(N)=O)CCO)ccc(Cl)cc1 c1(C(=O)OC)ccc(C(C(C)(C)C)Nc2cc(C(C)C)sn2)cc1 Cc1cc(C)c(OCC(=O)NC(c2c(C)cccc2F)C)c(Br)c1 c1(C(=O)NCC2CCN(C(C(CC(C)C)F)=O)C2)ccc2c(c1)C(=O)N(C)C2=O CCCC(C(=O)N1CCC(OC2CC2)C1)NC(=O)Cc1cn(C)cn1 C1(C(N(c2ccsc2)C)=O)CC2CN(C(=O)CCC3(O)CCC3)CC2C1 c1(NC(CC2OCCN(C(CC(C)(C)O)=O)C2)=O)cccc(Cl)c1Cl CC(C)CC(C)(O)C(=O)N1CCCC(O)(CCNC(C2CC2C)=O)C1 C(CN=C(NCC1CC1[N+](=O)[O-])N1CCC(CSc2ccccc2)C1)SC c1(C(N2CC3C(N(C(c4cc(C)on4)=O)C)C3C2)=O)c(C)ccc(C)c1O N1(C(=O)CCc2cnn[nH]2)CC2(C1)CN(C(C1CC3CCC1O3)=O)C2 Cc1nc(NC(C(C)NC(C2(C)CC=CCC2)=O)C(C)C)cc(SC(C)C)n1 C(=O)(CC1OCCc2ccsc21)NC1C(C)(C)C(CNC(c2nsnc2O)=O)C1 C1(NC(C(CCCC)=O)=O)CC2COCC(C1)C2NC(c1[nH]c(O)nc1C)=O CCCC(C)(CC)C(=O)N(CCC(=O)NCc1cc(C)cc(C)c1O)CCCO Cc1cc(CCC(=O)NCCCC(C)NC(c2ncc(C(F)(F)F)s2)=O)c(C)s1 CCC(CCOC)C(=O)NCc1ccc(C(=O)NC2CC=C(C)CC2)o1 c1(C(=O)NCCCC(C)NC(C2C(C)=C2)=O)c(C)oc(C)c1Br C1(C(N)=O)C(O)CCN1C(=O)CNC(C1CCC1)=O.c12conc1CNC2=O C(N=c1[nH]cc2ncnc-2[nH]1)C1N(C(c2cc(C)n(CC3CC3)c2C)=O)CCC1 CC1(C)CN(C(=O)CC2CCCCN2C(c2ccncc2F)=O)CC(C)(C)O1 N(C(=NCc1ccsc1C)NC1CCCCC1)CC1CCN(CCC)C1 Cc1cccc(-c2nnc(CC(=O)NC3CCN(C(=O)Nc4ccccc4)C3)o2)c1 C1(CC=C)(NC(=O)CC2NC(=O)NC2=O)CCN(C(c2cccc(Cl)c2)=O)C1 O(NC(=O)CN(C(=O)CO)CCOCC)CCCC#C.C1(CN)CC1 c1(C(N2CC(NC(=O)CC34CC(C3)C4)CC(OC)C2)=O)cc(Cl)cc(Cl)c1Cl c1(C(=O)NC2C(CNC(=O)C#CC3CCC3)COC2)ccn2nccc2c1 C1(F)(CNC(c2cn(CC=C)nn2)=O)CCN(C(C2CS(=O)(=O)CCO2)=O)CC1 C1(NC(c2c(C)ccc(C)c2)=O)CC2CCC1C(NC(=O)C(C)CC(N)=O)C2 N1(C(c2cc(CC)[nH]n2)=O)CCC(C(=O)N(C)Cc2ccsc2)(CC)C1 c1(C(=O)NCC(C)(O)CNC(=O)C=CC2CC2)ncc(Br)cn1 CC1C2CCCCC2CN1C(=O)C(C)(C)NC(C1C2CC(=O)CC12)=O c1(OC)ccc2c(c1)nc(NCCN(C)C1CCCc3ccccc31)n2C N1(c2ncc(C)cn2)CCOCC12COCCN(C(c1coc(Cl)n1)=O)C2 c1(NCC2C3CN(C(Cn4c(C)cc(C)n4)=O)C2C3)ncnc2cccnc12 N1(C(C2CCN(C)CC2)=O)CCOC2CCN(C(=O)Cn3cc(C#N)cn3)CC12 Cc1ccc(=O)n(CC(=O)NC2CCN(C(c3cc(N)cnc3Cl)=O)C23CC3)n1 C1CC12CCCC2.C12(COC)CN(C1)C2=O.C1(CC(=O)N(C)C)(C(=O)OC)CCC1 c1(CN2C(C(=O)Nc3cc(OC)nnc3)CCC2)ccc(O)c(C)c1O C1(C(N2CC(C(C(=O)NCCN(C)OC)OC)C2)=O)CC2(CCC2O)C1 c1(C(=O)NC(CNC(C2(C(F)(F)F)CCCC2)=O)C2CCC2)c(Cl)csc1Cl N1(C(C(CC#C)C2CC2)=O)CCC2(CC1)CCN(C(C1(COC)CC1)=O)CC2C C1(C(=O)NC2C3CN(C(CC4CCN(C)C4=O)=O)C2C3)CC12CCC(C)(C)CC2 CCCC(C)CCN=c1nc2c(cnn2C)c(NCC2CC2CC)[nH]1 c1(CC)nc(C(=O)NC(C)C(=O)NCC2(CC)CCCO2)cs1 C1(CNC(C2(CCNC(C(CC)C)=O)CCC2)=O)CCCOCC1 C12(CNC(C3(SC)CCC3)=O)CCCC1CN(C(C1(C)CCC(C)C1)=O)C2 C=C(C)CCCC(=O)N1CC2CC2(CNC(=O)CCCC(=O)NCCC)C1 CN1N=C(CC(=O)N(C)CC2(O)CN(C(C3CS(=O)(=O)C3)=O)C2)CC1=O C1(CN(C(=O)CN(C)C)CC)CCCN1C(c1ccc(CN2CCOCC2)s1)=O C1(C(N(C)CCNC(=O)CCOCC(F)F)=O)OCCC1(C)C C1(CC)CCN(C(c2cccnc2OC)=O)C(C(=O)NOCCCOC)C1 c1(CCC(=O)N(CC(F)F)CCOCCNC(c2cc[nH]c2)=O)nc(C2CC2)no1 C1(C(=O)NCC2C3CN(C(C(=O)NCCOC)=O)C2C3)C2C3CCC(C3)C12 c1(OCCC)c(OC)cc(C(N2CCOC(CNC(=O)C(C)C)C2)=O)cc1Cl S(=O)(=O)(c1ccc(S(F)(F)(F)(F)F)cc1)N1CC(C)N(C2CC2)CC1 Nc1c(F)c(F)cc(C(N2CCC(CNC(C34CCCC3C4)=O)CC2)=O)c1Cl Cc1nn(C)c(C(=O)NC2CCN(C(=O)CC3CCCOCC3)C2)c1Br C1(C(=O)OCC(C)CC2CC2)CCCC(C(F)(F)F)C1 C12(CC(=O)NCC3C(NC(CCc4c(OC)cccc4)=O)C3)CCC(CC1)OC2 C1(CNC(C2CCN(C(=O)CSC3CC3)C2)=O)CCC2(CC1)CC2 C1(CC=C)(NC(c2cn(-c3ccccc3)nc2C)=O)CCN(C(c2cnn[nH]2)=O)C1 Cc1nc2ccccc2nc1C(N1CC(O)(C(C)NC(=O)Cc2cnoc2)C1)=O N1(C(c2cc(C(C)=O)c(F)cc2)=O)Cc2ccc(C(N3CCC(C)C3)=O)cc2C1 N1(C(C2C(=C)C2C(=O)OC)=O)CCOCCC1C(=O)N(CCOC)CC CC(COC(=N)O)N=c1[nH]c(N2CCC(c3cccnc3)CC2)nc2c1SCC2 N1(C(C2CC(OC)C2)=O)CCCC(C(=O)NCC2CC23CCOCC3)CC1 CCCCC(CNC(c1cc(-c2ccccc2)co1)=O)NC(=O)CSc1nccs1 CCC(CC(=O)OC(C)(C)C)SCC1CC1.c12n[nH]cc1-c1nc-2no1 N1(C(Cc2cc(C)ns2)=O)CC(F)(F)CC1CNC(c1nnn(C(C)(C)C)n1)=O c1(N(CCOCCOCC)C)nc(N2CCOC(C)(C(F)F)C2)c2sccc2n1 C(=O)(CCCCn1ccnn1)N(C)CCNC(c1cc(C2CCC2)on1)=O O=C1CC2CCC(CN1)N2C(=O)C=Cc1cocn1 N1(C(=O)OC(C)(C)C)CCOCC(C(N2CCCC2(C)Oc2ccc(Cl)cn2)=O)C1 Cc1ccc(Cl)c(NC(=O)CN2CCOCC2CC(F)(F)F)c1 C1(CNC(C(C)n2cccn2)=O)CCCN(C(=O)CCc2nncn2C)C1 c1(C(=O)NCC2CCCN2Cc2c(F)cccc2Br)cccc2ccccc12 C(=O)(CCCCC(C)(C)OC)N1CC2C(N(C(C(CCCCCC)F)=O)C)C2C1 CC(C)(C)C(CO)C(=O)NCC(CN=[N+]=[N-])C(=O)N1CCC(N2CCCC2)C1 c1(OC)ccccc1CC(=O)NC1CCC(NC(C2CC3C=CC2C3)=O)C1 C(CC(C)CCNC(c1nc(O)sc1C)=O)NC(c1ccc(C)o1)=O c1(CN(C(C(CCC)C)=O)CC)ccc(OCC)c(OC)c1.C12CCN(C1)C2=O c1(C(=O)NC2(CNC(C3(CO)CC3)=O)CCC2)cncc2cc(Cl)ccc12 C1(OC)CC(NC(c2cc3n(n2)CCO3)=O)CN(C(C2CCCCC2)=O)C1 Cc1ccc(-n2nc(-c3ccc(Cl)cc3)nc2C(C)C(O)C(F)F)c(C)c1 CC(C)CCC(F)C(=O)N1CC2CCCC2(NC(c2cccc(=O)o2)=O)C1 c1(CC)ccc(C(C)C(=O)NC(C)CC2CN(C(c3cc(C4CC4)[nH]n3)=O)C2)cc1 C1(C(=O)OCC)(C(=O)NC2CC(NC(C3(CO)CCC3)=O)C2)CC12CC2 N1(C(CCCC(=O)OCC)=O)CCCC2(CNC(c3ccc(Cl)s3)=O)CCCC12 Cc1ccc(C(=O)NC(CCC2CCC2)C(=O)NC(CF)C(F)(F)F)cc1 c1(CCC(=O)NCC(CNC(CC(CN(C)C)(C)C)=O)O)ccc2c(c1)CCO2 c1(C(=O)NCC(C)CN(C(=O)CC(C)(C)C2CC2)C)nccc2cccnc12 CCC(C)(CNc1ncc(C)c(SC)n1)C(=O)NCc1occ2c1CCC2 Cn1ccnc1S(=O)(=O)NC1(NC(=O)C(O)CCCc2ccccc2)CCCCCC1 O=C(CC(CC1CC1)N(C(C1CC(=O)N1)=O)CCO)N=c1cc[nH]cc1F CN1CCCCC1CCC(=O)NC(C)(CNC(=O)CSCc1ccccc1)CO c1(C(=O)NCC=CCNC(C2N(C(C)=O)CCCC2)=O)ccc2n[nH]cc2c1 c1(SC2CCN(C(=O)OCc3nnnn3C3CC3)C2)cc(Cl)cc2ccccc12 c1(C(N(C)CCNC(=O)COC2CCCC2)=O)cnn(C2COC2)c1 N1(C(COC(C)=O)=O)CC2(CO)CC1(CNC(=O)C(c1ccc(F)cn1)(F)F)C2 c1(NC(CCC2N(C(c3c(CC)ccs3)=O)CCC2)=O)cc(O)ccc1OC N1(C(c2nnnn2Cc2nnn(C)n2)C)CCSCC1 C(=O)(C(=O)N=S(C)(C)=O)NC1C(OC)CN(C(=O)Cc2ccc(F)cc2F)C1 C1(CNC(C(C=C)O)=O)CCC2CN(C(c3ccc(CC)cc3F)=O)CCC2C1 c1(NC(=O)CSCC2CCCO2)ccc(Cl)cc1.c1(C(=O)N)coc(C)n1 N1(C(c2nnn(CC)c2C)=O)CC2CC(NC(c3ccncc3F)=O)C(C2)C1 c1(CNC(C(n2cc(C3C4COCC34)nn2)C)=O)cc2ccccn2n1 Cc1nscc1CC(=O)NCC=CC(N1CCC(c2cc[nH]n2)C1)=O Cc1nn2cc(C(=O)NCC3CCC4(CN(C(C5(C)CCOC5)=O)C4)O3)nc2s1 Cn1cc(C(N2CCCC(C)(CNC(C3CC3C(F)F)=O)C2)=O)cc1S(N)(=O)=O N1(Cc2nc(CC)on2)CCN(C(c2sc(C3CC3)nc2C)=O)CC1=O c1(OC)cc(C(=O)NC2CC3CC2N(C(=O)CCC2CC2CC2CC2)C3)cc(C)n1 CCC(C(=O)NC(C(=O)NC1CCCC1)C(C)C)C(C)C c1(C(N2C3CN(C(c4c(C)snn4)=O)CC2CC3)=O)cc2cncn2c(O)n1 CCCC(C)CN(C)C(C1CC(CNC(=O)C(CO)N(C)C)C1)=O Cc1ccc2n[nH]cc2c1C(N1CCCN(C(=O)Cc2cn(C)cn2)C(C)C1)=O C(=O)(CCCC(C)NC(=O)NCCCC(N1CCC(OC)CC1)=O)OC CC1(C)CC(C(N2CC(CNC(=O)CNC(c3ccccn3)=O)C2)=O)O1 c12ccc(cc1OC)CC(=O)NCC(C)NC2=O.c1(OCC)cccc(SC)c1 Cc1c(CNC(=O)CC2CC(NC(=O)CC3CC(=O)NC3=O)C2)cnn1C C1(NC(C2CC(O)CN2C(c2cccc(=O)o2)=O)=O)C2CCCC1CC2 c1(C(=O)OC)ccc(NC(C2CCC(C)N2c2ccnc(SC)n2)=O)c(C#N)c1 C(C)(C(C(=O)NCCC1COCCO1)C(C)C)NC(C1C(C(C)C)CCO1)=O Cc1cc(C(=O)NC2CN(C(c3sccc3OC(F)F)=O)CC23CC3)nc(O)c1 c1(C(=O)OC)cc2n(n1)CCCC2NC(=O)Cc1cnc(C)o1 C(C(C)(C)C(=O)N1CCOC(C2(NC(C3CN(C(C)=O)C3)=O)CC2)C1)OC C1(NC(COCCN(C)C)=O)CC2CCC1N(c1ccncc1C#N)C2 CC1(c2cn(CC(F)(F)CO)nn2)CCN(C(=O)C(C2CCCOC2)N(C)C)C1 C=C1CCC(C(=O)N(CC(C)NC(c2c[nH]nc2C)=O)CC)CC1 CC1CCN(C(=O)CCC(=O)N(c2ccc(F)c(Cl)c2)CC#N)CC1C(F)(F)F N1(C(CN(CCOC)C)=O)CC2CC(NC(=O)C(n3nc(C)cc3C)C)C1C2 c1(C(=O)NC2CN(C(C(C)=CC)=O)CC(C)(C)C2)cc(C)c(F)c(S(C)(=O)=O)c1 c1(C(=O)NCC(C)N(C)C(c2coc(C(F)F)n2)=O)ccc(=O)n(CCO)c1 c1(C(N2CCC(CNC(c3c[nH]c(=NC)o3)=O)CC2)=O)cccc2c1CCO2 N1(C(CC(=O)NCC)=O)CCN(C)CC1C(=O)NC(CC)C(C)O C1(NC(c2cc(Cl)c(Cl)[nH]2)=O)CCCN(C(C2CC2[N+](=O)[O-])=O)C1 CC(=O)CCCC(C)C(=O)NCc1csc(C(=O)NCc2ccc(C)nn2)c1 N1(C(=O)C(=O)N2CC(F)C2)CCCC1c1ccccc1 CCCCC(O)CC(=O)N1CCN(C(c2sccc2CC)=O)C(CC(C)(C)C)C1 N1(C(c2ccc(CNC(COC(CC)CC)=O)o2)=O)CC(C)C(C)C1C CC(C)CCCOCC(=O)NC(CCCNC(=O)C(C)O)c1ccccc1 N1(C(CN(C(C)C)C)=O)CC(NC(=O)CCCOc2cccnc2)C2(CC2)C1 C1(NC(c2cc(Cc3ccccc3)[nH]n2)=O)CN(C(C2CC2F)=O)CCC1F CC(CS(C)(=O)=O)C(=O)NCC1(C)CCCN1C(c1cccc2ccnn12)=O c1(C(=O)NC2C(NC(CC3(C=C)CCC3)=O)CC2)c(C2CC2)nn2ccccc12 C(CCC(C)(C)C(=O)NC1CN(C(C)C)CC1C)NC(CC(C=C)(C)O)=O C#CC1CN(C(C2CC2[N+](=O)[O-])=O)CCN1C(c1cc(O)cc(=O)o1)=O O=C(Cn1nccc1C1CCCN1)N=c1c2ccccc2[nH]n1-c1cccs1 CC1CN(C(c2cnnn2C)=O)CC1(C)CNC(=O)CC1(C(F)(F)F)CCC1 c1(C(=O)NC(C2OCCN(C(c3ccn(CC)n3)=O)C2)C)ccc(O)cc1Cl N1(C(C=C(CC)C)=O)CCCN(C(c2nc(-c3ccccc3)oc2C)=O)CC1C c1(CCCC(=O)N2CC(NC(CC3C(C)(C)C3)=O)C2)ccc(C#N)cc1 N1(C(c2cc3nc(C)sc3[nH]2)=O)CC2(C1)CN(C(=O)C(C)C(C)(C)C)CC2CO C12(CNC(C(C)N(C(=O)CC3CCCCO3)CC)=O)CC=CC(C1)OC2 CC(CC(=O)NC1C2CC1N(C(c1c(N)cc(Cl)nc1Cl)=O)C2)CC(C)(C)C C1(C(C)(C)C)CCC(C(=O)NCC=CCNC(=O)C(C)(O)C2CC2)O1 C1(CNC(c2c(OC)ccs2)=O)CC2CC2N1Cc1cc(Br)co1 C1(NC(C=C2CCC(C)CC2)=O)CC2(C1)CC(C(N1CCCC(C)(F)C1)=O)C2 C1(NC(c2ccc(COC)[nH]2)=O)CN(c2nc(O)nc(O)n2)CC2(CC2)C1 C1(CCOC)CN(C(=O)COC(C)C)CCN1C(=O)C=Cc1ccc(C)s1 N1(C(c2c(C(C)C)scn2)=O)CC(NC(=O)C2=COCCO2)C(C)(C)C1 C1(C)(CNC(C2CCN(C(Cn3c(C)nnn3)=O)C2)=O)COCCO1 C(=O)(C(C)CCCC(C)=O)Nc1cncc(OCCOC)c1.C12CN(C1)C2=O C12(NC(C3CN(C(C)=O)C3)=O)CCC(CN(C(C3CCCN3C=O)=O)C1)C2 C(=O)(C1=CS(=O)(=O)c2ccccc21)N1CCC(CNC(C(C#C)(C)C)=O)C1 C1(C)(C(c2n(CCCSC)nnn2)NCCCOCC(C)C)CCC(C)C1(C)C CCCC(C(O)C(=O)NCC1C2CCCCCC12)NC(=O)C(C)(C)C(N)=O CCC(CC(=O)NCCC1CC(NC(=O)C(c2cccc(C)c2)C)C1)C(C)C c1(C(=O)NC(C(C)NC(=O)CN2CCOCC2)CO)c(Cl)ccc2c1OCO2 C=CCCCCCC(=O)N1CC(=C(F)CNC(c2nc(C)sc2C)=O)C1 c1(COC(c2ccc(Cl)c(F)c2)=O)csc2ccccc2c1=O Nc1cc(C(=O)NCC(CNC(c2cc(O)ncn2)=O)C(F)(F)F)ncc1F c1(C(N2CC(NC(c3[nH]cc(CC)c3)=O)C(C)C2)=O)cccc(C)c1OC CC(C)C(C)C(=O)N1CC(O)(CNC(C2CC(F)CN2C)=O)C1 C1(C2CN(C(Cc3n(C(C)(C)C)ccn3)=O)C2)CN(C(=O)C(C)(C)Br)CCO1 C(=O)(CC(C(C)OC)NC(C1C2CCC(F)C12)=O)N(C(C)C1CC1)CC CC1CCC=C1C(=O)N1CCN(C(c2cc(-c3ccns3)on2)=O)C(CO)C1 C1(C(=O)OC)CCN(C(=O)NCc2ccn(C(F)F)n2)C12CCC2 c1(OCC(=O)NCCCN2CCCCC2)cc(Br)cnc1F c1(C(=O)NCC(C)NC(c2sc(C(=O)OC)c(C)c2)=O)cccc2c(C)[nH]nc12 N1(C(=O)CC23CCCC2C3)CCN(CCNC(c2csnc2C2CC2)=O)CC1 c1(NC(c2nnnn2C2CC2)CCOC)ncnc2c(F)c(Br)ccc12 n1(CCC(=O)NCCOC(CNC(CC(C)(F)F)=O)(C)C)cc[nH]c(=O)c1=O C1(NC(c2ccnn(C)c2=O)=O)CC2CN(C(=O)CN3CCC(C)(C)C3)CC2C1 c1(C(=O)NCCC(C)NC(=O)C=CCO)csc2ncnc(O)c12 CCC(CCCC(=O)NC(c1cn(C)nn1)C)NC(c1cc(C)co1)=O N1(C(CNC=O)=O)CCC(CNC(=O)Cc2ccc(-n3cccn3)cc2)C(O)C1 C(C(C(=O)OC)OC)NC(C=CCCC#C)=O.C1C(=O)N1CCOC C(=O)(C(CC1CCCC1)NC(C1(N(C)C)CC1)=O)NC(CC)CN1CCCC1 N1(C(CCC#C)=O)CCC(NC(c2noc(CC)c2C)=O)C2(CCC2)C1 O=C(N=c1ncc(F)c[nH]1)N1CCOCC(Sc2nc3ccccc3[nH]2)C1 C(c1ccc(F)cc1)=C(C)C(=O)NCC(C(C)C)NC(=O)C(c1ccccc1)O c1(OC)cc(CC(N2CCN(C(=O)C3=CCCCC3)C(C)C2)=O)ccc1C C1(COC)(CNC(c2cn[nH]c2)=O)CCCN1C(C1CCCC1SC)=O C1(C(=O)NCCOCCNC(COCC(C)C)=O)CC(F)(C(=O)NCC(C)O)C1 c1(OCC)nc(C(=O)NC2CCC2NC(=O)CNC(c2cccnn2)=O)ns1 N1(C(C2COCCN(C(C3CCCN(CC)C3)=O)C2)=O)CC2(CCN(C)CC2)C1 c1(C(=O)NCC(CN(C(CSC)=O)C)O)ccc(OCC(F)(F)F)cn1 N1(C(c2ccc(C(C)C)o2)=O)CC(NC(=O)CS(=O)(=O)CCO)CC(C)(C)C1 N1(C(C)C)CCC(C(=O)NCC2(O)CN(C(c3ncoc3-c3ccon3)=O)C2)C1 N1(C(c2c(C)cc(CC)o2)=O)CC(C(=O)NCCCOC(F)(F)F)CCC1C c1(NC(c2ccc(-n3cnnn3)cc2)=O)cc(Cl)cc([N+](=O)[O-])c1O c1(OC)ccc(CNC2CC(C(=O)Nc3cc(O)cc(Cl)c3)C2)cc1CC(=O)O c1(CC(=O)NC2CCCC2NC(c2cnc(S)n2C2CC2)=O)cn2ccsc2n1 Cc1nc(C(=O)NC(CC(=O)NCC2(O)CC(C)(C)C2)C2CC2)sc1C CCCC(C(=O)OC)C(=O)NC(C)(C)C(=O)NC1CN(C)C(C)(C)C1 n1(CC(=O)NC(C(=O)N(C2CCC(CO)CC2)C)CC2CC2)ncccc1=O c1(C(N(CC(C)NC(CCC#C)=O)C)=O)nn(-c2ccc(F)cc2)cc1C c1(C(=O)NC(CC(=O)NCC(C2CCC2)OCC)C)ncccc1N N1(C(C(c2ccccc2)C2C(C)C2)=O)CC2(NC(=O)CCN3CCCC3)CC1C2 N1(C(c2c(C)oc(C(C)C)n2)=O)CC2CC1CN(C(c1ccoc1C1CC1)=O)C2 c1(OC(C(=O)NCC2(NC(C(CC)C)=O)CCCC2)(C)C)c(F)cccc1F Cc1nc(-c2cc(C(N3CCC(CNC(C4CC(OC(F)F)C4)=O)C3)=O)cs2)cs1 c1(C(=O)NCCN(C(C(CC)OCC)=O)C)ccc2c(c1Cl)OCCO2 n1(CC)nnnc1C(c1cnsc1)NCc1nnc(CO)s1.C(C)(C)(C)NC(=O)O C(=O)(C(CC(F)F)N(C(C1CCC(=O)N(C)C1)=O)C)NC(CC#C)(C)C c1(C(=O)NC(C)CCNC(=O)C2(C)C3CC3CCC2CC)coc2c(F)cccc12 Cc1cccc(C(C)NC(=O)C(CCF)NC(=O)C#CC2CC2)n1 CP(C)(=O)c1cncc(C(=O)NCC2CC2NC(c2ccoc2Br)=O)c1 c1(C(N(CCNC(CC2CC(N(C)C)C2)=O)C2CC2)=O)ccc(C(C)(F)F)nc1 N1(C(C(C=CC)O)=O)CC(CNC(=O)CCNc2ccc(Cl)cc2)OC(C)(C)C1 CCC(CC(=O)NC1CCC(C(C(C2(O)CC2)=O)=O)CC1)C(C)C.C(C1CC1)(C1CC1)N N1(C(c2cc(OC)nc(Cl)c2)=O)CCC2CN(C(=O)C(C)S)CC2C1 C12CCC(C(=O)NC3CC(NC(=O)C(C)(C)C)C34CCC4)(CC1)CO2.CC C1(C)(CNC(CC2N(C(c3n(CC)ncc3)=O)CCOC2)=O)CCCC(=O)N1 C1(C(=O)NCC(C)(C)OCCNC(C2(F)CCCC2)=O)CCC2(C1)CC2(F)F C=CCC(C)(C)CC(=O)NCC1CCCC1NC(c1cnc(C)cn1)=O C1(CNC(CCCC#C)=O)N(C(c2ccnc(OCC)c2)=O)CCC1(C)C c1(OC)ccc(C(=O)NCC2(C(=O)Nc3c(Cl)c(C)nn3C)CC2)c(F)c1 N1(Cc2ccc(OCCC)cc2)CCC(=O)N(Cc2ccc(CC)c(C)c2)C1=O N1(C(=O)C=Cc2cncs2)CCC2(CCCN(C(C3CCC3(F)F)=O)C2)C1 c1(C(=O)OCC)c(C)csc1NC(C1(C)CN(Cc2cccc(OC)c2)C1)=O C(c1ccccc1Br)=CC(=O)NC1CC(CCNC(c2nn(C)c(O)c2)=O)C1 c1(C(=O)NC2(CCC)CCN(C(=O)C=C(C)Cl)CC2)cc2c(CC)cccc2[nH]1 N1(C(c2c(C)nc(=N)[nH]c2)=O)CC(NC(C2CCCCS2(=O)=O)=O)CC2(CC2)C1 c1(OC(C)C(=O)NCC2(NC(c3cc(C(F)F)[nH]n3)=O)CC2)ccc(Cl)cc1 N1(C(c2cc(SC)oc2)=O)CCC(C)C(NC(c2cccc(F)c2Br)=O)C1 c1(C(=O)NC2CCC(CNC(c3c(C)nccc3)=O)C2)cc2cc(F)ccc2s1 c1(C(N(C2CCN(C(C3(C)CC(C)C3)=O)C2)CC)=O)cn(CC(F)F)cn1 C(C(C)C(=O)N1CCCC1C(C)NC(c1ocnc1C1CCC1)=O)OC c1(C(=O)NCc2ccc(CSCC)cc2)cccc(C#N)c1O Cc1ccc(C(=O)Nc2cc(N3CCC(O)CC3)ccn2)c(F)c1Br C(=O)(CC(C)(O)C1CC1)N1C(C(C)NC(C(C)(C)OC(C)=O)=O)CCC1 CC(C)C(C)CN(C(=O)C(O)C1CN(C(=O)C(C)(C)F)C1)C Nc1ccc([N+](=O)[O-])cc1C(=O)NC(C1CCOC1)CNC(C1CCCC1)=O Cc1cnc(C(N2CCC(C(N3CCC(CN(C)C)CC3)=O)C(O)C2)=O)c(F)c1 N1(c2cc(NCCC#N)nc(C)n2)CC(C)C(CO)C(C)C1 c1(NC(CC)C)ncc(S(=O)(=O)N2CCN(C(C)C)CC2)cc1Cl c1(C(C)C)cc(C(N2CCC(O)(CNC(c3ccsc3)=O)C2)=O)ccc1F c1(C(=O)Nc2n(C)cnn2)cc2c(cn1)CCCC2 CCCC(C)(C)CC(=O)NCC12CC1CN(C(c1cc(F)c(C3CC3)c(F)c1)=O)C2 c1(NC(=O)NCC2C3CCC23)ccn2nccc2c1 C=C(C)CC(C)C(=O)N1CC(NC(c2ccc(-c3csc(C)n3)s2)=O)C(C)(C)C1 c1(-n2cc(C(CCC)NC(c3cc(Br)cn3C)=O)nn2)cccc(Cl)c1F C=C(C)C1CC(=O)N(C(C)C)CCCO1.C(=O)(CC(C)C)OCCC(=O)N C(C1c2ccccc2CN1C)NC(=O)NC.C12CCCCCN1C(=O)NC2 C1(N(C(C2C(OC)C2)=O)C)CCN(C(=O)NC(c2ccsc2)C)C1 c1(C(=O)NC(C2CCN(C(c3ccc(F)s3)=O)CC2)C)cccc2oc(O)nc12 C1(NC(CNS(N)(=O)=O)=O)CCN(C(=O)CC2CCCCO2)C12CCC2 N1(C(C(C)CN2CCOCC2)=O)CCOC(CNC(c2cccc(F)n2)=O)C1 c1(C(=O)NC2CC(CNC(C3CC4CCC3O4)=O)C2)cnc2cc(Br)ccn12 CCCCC(O)CCC(=O)NCC1CCCN(C(C2(CO)CCCO2)=O)C1 C1(COC)(NC(c2ccn(C(C)C)n2)=O)CCN(C(c2cn(C)c(=O)s2)=O)C1 CC1Cc2cccc(C(=O)NC3CN(C(c4sccc4C(F)F)=O)C3)c2O1 c1(C(N2C(C)CC(NC(=O)C(C3CCCCC3)O)CC2)=O)onc2c1CCCC2 C1(O)(CN(C)NC(=O)CC(C)(C)O)CCN(C(c2cnn(CCO)c2)=O)C1 C12(SCC(=O)NCc3nc[nH]n3)CC(CNC(CC3(C)CC3)=O)(C1)OC2(C)C.CN CC(C)CC(C(=O)N(C)C)NC(=O)C(n1cc(C2CCC=CO2)nn1)C c1(CC)nc(C)c(CNC(=O)NC2(C)CC(Cn3ccnn3)C2)s1 c1(C(=O)NCC(C)NC(c2cscc2C(F)F)=O)ccc(-n2cnnc2)cc1 C1(NC(CSCC)=O)CC(F)CN(C(c2cnc(C)nc2)=O)C1 CC1=C(C(=O)NC2CCC(CNC(=O)C(C)(O)C3CCOC3)CC2)CCC1 CCCC(C)C(C(=O)NCc1ccco1)N1CCCC(CC2CCOC2)C1 N1(C(C=C(C)C)=O)CCC2CCN(C(=O)Cn3cc(-c4ccccc4)cn3)C2C1 c1(CCNC(C2C3(CCC3)N2C)=O)cccc(O)n1.n1(C)ccccc1=O.CO C1(C(N(CCCNC(=O)C(C)(C)CCF)C(C)C)=O)CCn2nnnc2C1 C(=O)(CS(=O)(=O)C1CCCC1)NCCC1(O)CN(C(CC(COC)(C)C)=O)C1 c1(Cn2cc(CCC(C)=O)nn2)ccc(C(=O)N(CC(C)O)C)c(Cl)c1 C1(CC2CC(n3cc(CNC(C4C(OCC)C4C)=O)nn3)C2)CCCCC1O C#Cc1ccc(C(=O)NC2(CF)CCN(C(=O)CCN(C)CC)C2)cc1F C=CCC(C(=O)NCC(CC)N(C(=O)C=Cc1ccc(OC)cc1)C)C(C)C Cc1cc(=NCCN2CCC(C)CC2)[nH]c(=NCCC(=O)NC(C)C)[nH]1 C(C)(C(=O)NC1CN(C(=O)COc2ccc(F)cc2Cl)C1)(C(C)C)NC(C)=O O=C1CC(C(F)F)N1.C(CCN)C(C1CC1Cl)=O.C(C)(C)(C)OC(=O)NCCO C1(NC(CCSC)=O)CCC2(CC1)CN(C(C1CCSC(C)C1)=O)CCO2 Cn1c(C(N2CCC(NC(C3CNC(=O)C3)=O)C(O)C2)=O)cc2ccsc12 C1(NC(c2cc(OC)no2)=O)CN(C(c2oc(C)nc2C)=O)C2(CCCCC2)C1 N1(C(CSCCCC)=O)CCC(NC(c2c(CC)cccc2CC)=O)C(OC)C1 c1(C(N(CCC)CCNC(=O)C(n2cc(Cl)cn2)C)=O)cc(Cl)c(F)c(Cl)c1 C(=O)(C=C1SCC(=O)N1C)NC(C1N(C(Cc2c(C)noc2C)=O)CCCC1)C Cc1c(C(=O)NC(C2(O)CN(C(=O)C(F)C(C)(C)O)C2)C)cc(C2CCC2)n1C Cc1cc(C(=O)N(CCNC(=O)CS(=O)(=O)N(C)C)C(C)C)c2cnccc2c1 N1(C(c2cnn(CCO)c2)=O)CC2(CNC(C3(O)CCC3)=O)CCC1CC2 CCC(C)C(CNC(=O)CC1(C)CCN(C(c2cc(C)n(C)c2)=O)C1)CO C1(C(=O)NC(C)Cc2nc[nH]n2)CC(F)CN(C(=O)CC(C)c2ccco2)C1 C1(C(=O)NCCC2CC(NC(c3cnc(C(C)=O)s3)=O)C2)CCC(C)(F)CC1 C(=O)(CCCC(F)(F)CO)NCC(C)(C(C)C)NC(CC(C=C)(C)C)=O N1(C(C2(OC)CCSC2)=O)CCCC2(CCN(C(=O)C3=CS(=O)CCC3)CC2)C1 C1(C(N(C2(C(=O)N(CC(O)CN)C)CC2)C)=O)COCCC1C.CO Cc1c(C(=O)NC2(CNC(=O)C(C3CCCCC3)=O)CCOC2)cnn1CCO c12ccc([N+](=O)[O-])c(c1)NC2.C1(C(N)=O)CCCC1NCC(F)(F)F C(=O)(C1Cc2ccccc21)OC(c1ccc(Cl)c(C)c1)CC N1(S(C)(=O)=O)CCC(NC(=O)NC(c2n[nH]c(=N)s2)C2CC2)C1 Cc1ccc(C(=O)NCC2CC(C(=O)N3CC4CCCC4C3)=NO2)c(F)c1 c1(CC)cc(F)ccc1C(C(=O)OC)NCCCC(=O)OC c1(C(=O)NC(CNC(C(c2ccc(F)cc2)OC)=O)C2CC2)cc(Br)n(C)n1 N1(C(c2ccc(CC)c(C)c2)=O)CC2CCC1CN(C(c1cc(F)n(C)n1)=O)C2 CC1N(C(=O)CN(C(=O)C2=C(Cl)CCC2)CC(C)(C)C)CCC1(C)C C(=O)(CCN=C(NCC=Cc1ccccc1)NC1CN(CC2CC2)CCC1C)NC C1(O)(CNC(C(C)Oc2cccnc2)=O)CCCN(C(=O)COC(C)(C)C)C1 C#CCCCC(=O)NC1CCN(C(=O)CCCC#N)C1C c1(C2(NCCC)CC2)cc(Sc2nnnn2CC2CC2)ccc1Br c1(C(CC)=O)cc(C(=O)NCC2CCN(C(=O)C3=CCCOC3)C2)ccc1Cl N1(CC)CC2(C1)CN(Cc1ccc(OC)cc1)C2.c12cnc([nH]1)C(=O)N1CC2C1 C1(NC(c2ccc3c(c2)CC3)=O)CN(C(=O)Cc2cnc[nH]2)C2(CCCCC2)C1 N1(C(C2OCCN(C(C3(F)C(C)(C)C3(C)C)=O)CC2)=O)CC2(COC(=O)C2)C1 c1(N(CC(=O)NCC(c2nn[nH]n2)(F)F)Cc2ccccc2)ccc(Cl)cc1 CC(C)CCCC(=O)N1CCC(C(=O)N(C)Cc2cnn[nH]2)(CF)C1 C1(C(=O)NC2CC(NC(c3c(NC)nccc3)=O)C2)Cc2nccn2C1 C1(NC(c2ccc(C(C)CC(=O)O)cc2)=O)(CO)COCC12CCC2 C1(COCC)COCC1C(=O)NCCC(CC)OC.C12(CC1C)C(=O)N2 c1(C(=O)NCC(CC)(CC)NC(C2(C)CCOCC2)=O)c(C)[nH]c2ccccc12 C1(OCC)CN(C(=O)C(=Cc2ccccc2)C)CC1CNC(c1cccn1C)=O c1(C(N2CC(COC)N(C(c3nc(=O)n(C)[nH]3)=O)CC2)=O)ccsc1S(N)(=O)=O c1(C(=O)NCc2cncc(-c3cccc(CO)c3)c2)ccc([N+](=O)[O-])cc1 CC1CC(NC(C2(O)CCOCC2)=O)CN1C(=O)Cc1cccnc1Cl c1(OCC(=O)NC2CC(NC(c3c(CC)cc[nH]3)=O)C2)ccc(C)cc1F C1(CC(C)C)CCCN1C(=O)CN(C)C(C1CCCC1n1cccc1)=O c1(C(N2CC(CN(C)C(C3(C)CCC(=O)C3)=O)C2)=O)nc2cnccc2s1 c1(OC)ccc(C(C)C(N2CC3CC2CN3C(=O)CCCC2CCC2)=O)cc1F C(CCC(C(=O)NC(c1cncnc1)C)NC(=O)Cc1ccc(O)nc1)OC c1(COC)c(C)nc2ccc(NC(C3N(C(C(CC#C)(C)CC)=O)CC3)=O)nn12 C1(CCNC(C2CC(N(C)C)C2)=O)CCN(C(C2CCNC2=O)=O)CC1 CCCC(C(=O)N(C1CC(C(=O)NC(C)C(C)(C)c2cccs2)C1)C)OCC C1(C(=O)NC(c2nccn2C)C)COCCN(C(=O)C(C)NC(C)(C)C)C1 O=C(C1CCCc2nccn21)N1CCCC2CCN(C(=O)C(F)(F)C(F)F)CC12 c1(C(N(C(CNC(CCC(C)C)=O)CN2CCCC2)C)C)ccc(F)c(F)c1 c1(C(=O)NC2CCCC(NC(CN(C(C)C)C)=O)C2)ccc(Cl)c(O)c1N c1(C(=O)NC2CCN(C(C(C=CCCC)O)=O)C2)c(C)nc2ccccn12 c1(C(=O)NCCCC(C)NC(CCCC=C)=O)cn(CCO)c(=O)nc1O C(=O)(N=S(=O)(c1ccccc1)C(F)(F)F)Nc1cc2c(nc1)N(C)C2 N1(C(C(CC)C#N)=O)CCN(C(c2cc(C(C)(C)C)nn2C)=O)CC(O)C1 CC1(C(=O)NCC(C2CCOC2)NC(=O)Cc2cccc(F)c2)CCNC1=O N1(C(C2C(C=C)CC2)=O)CCC2(CCCN(C(=O)CC(C)(C)O)C2)C1 c1(OCCC(=O)NCC(CCOC)NC(c2cc(Cl)ns2)=O)ccc(C)c(C)c1 CCCCC(O)C(=O)NC12CCC(CC1NC(=O)CCNC(C1CCC1)=O)C2 C1(CC(=O)NCC2(O)CC(C(NOCC(=O)OCC)=O)C2)CC(C)(C)CO1 c1(C(=O)NCCn2cc(CCO)nn2)cccc(Cc2cccc(F)n2)c1 C(=O)(C1CCCc2n[nH]cc21)NC1C2CN(C(CCc3onc(C)n3)=O)CC21 C(=O)(C1=CCCN(C(C2CC2(F)Cl)=O)C1)N(C)CC1(N(C)C)CCCC1 C(CCC(C)(C)C(=O)N1CCOC(CF)C1)NC(C(C(C)C)CN(C)C)=O c1(C(=O)Nc2cc(O)ncn2)ccc2ccccn12 n1(CC(N2CC(NC(Cc3n(C)cnc3)=O)C3C2C3)=O)nc(C2CC2)n(C)c1=O c1(C(=O)NCC2(O)CN(C(C3(CC#C)CCOC3)=O)C2)cnc(SC)n1C c1(C(=O)NC2CN(C(C(C)NC(COC)=O)=O)C2)ccc(S(C)(=O)=O)cc1 C1(C(N2C(C(C)NC(Cc3c(C)ccs3)=O)CCC2)=O)CN2CCN1CC2C c1(OC)c(CN(c2nc(O)ns2)CC(=O)O)cccc1F c1(C(=O)NCC(CN(C)C(c2nn(C)cc2C(F)F)=O)O)cc([N+](=O)[O-])cn1C c1(CC)cnc(C(c2nnnn2CSc2ccccc2)NCc2cccnn2)s1 c1(CC(CC)NCC(C)(C2CC2)OCC)ccc(O)cc1 CC1CN(C(c2ncncc2Cl)=O)CCCN1C(=O)Cc1ccc(Cl)cc1Cl C1(C(=O)NCC2C3CN(C(c4c(C)cn(C)n4)=O)CC32)CNc2ccccc2O1 c1(C(=O)OC)ccnc(C(=O)NC(CNC(c2cn[nH]c2)=O)C(C)C(C)C)c1 CC(C(C)C(=O)NCC1CN2CCC1C2)NC(=O)Cn1cc(C#N)cn1 C1(c2nnnn2-c2ccccc2)(NCC2(SCC)CC2)CCOC(C)C1 N1(C(CC(CCC)(C)O)=O)CCN(C(c2cn(C)c(=O)n2C)=O)C2(CCC2)C1 c1(CC(=O)NCC2C(NC(C3(c4cc(C)no4)CC3)=O)C2)cc(Cl)n(C)n1 N1(C(Cc2nc(C)oc2)=O)CCOC(C)(CNC(c2nccn2C(C)C)=O)C1 C1(C(N(C2CCN(C(=O)CC3CCCCN3)CC2)CCC)=O)CC(CC)=NO1 C(C)(C(=O)N1CC2CC1C2CNC(=O)CC1CC(=O)NC(=O)C1)(C(C)C)OC N1(C(c2cc(C)sc2N)=O)CCC2(NC(c3cc(C(N)=O)c[nH]3)=O)CC2C1 c1(C(N2CC(NC(c3cnc(CC)s3)=O)C2)=O)nc(OC)c(C)s1 O=C(NN1CCCC1C(=O)NCC1CC2(CC2)CO1)C1C2CCCC12 C(=O)(C1CNC(=O)c2ccnn21)N(C1CCCN(C(c2cn[nH]c2)=O)CC1)CC C12(C(N3CCCCC3)=O)CCC(N=[N+]=[N-])C1C2.CCCC(=O)OCC.N12CCC1C2=O c1(C(=O)NC2CN(c3ccc(OC)cc3)C2)cc2n(c1)CCCC2 c1(C(=O)NCCN(C)C(c2ncoc2C2CCC2)=O)cn2cccc(Cl)c2n1 N1(C(=O)CC2(C(F)F)CC2)CCCC2(CCN(C(=O)CN3CCSCC3)CC2)C1 N1(C(CC(C)(C)O)=O)C2CCC1CC(NC(c1cc3ncccc3[nH]1)=O)C2 N1(C(COC(C)C)=O)CC2CC1CN(C(C1(C(C)(F)F)CCOCC1)=O)C2 C1(CNC(C2(C#C)CC2)=O)OCCC1C(=O)NCCOCCF Cc1ncc2n1CCC(C(N1CCC1CNC(c1ccc(CO)c(Cl)c1)=O)=O)C2 c1(OCC=C)c(C(=O)NC2CCC(CNC(=O)C(C)=CC)C2)cccc1C C1(O)(CNC(C2(CSC)CC2)=O)CCCN(C(C2CCCC(CF)C2)=O)C1 C1(N(C(C2CC(OC)C2)=O)CCO)CCN(C(C2CC(n3cnnc3)C2)=O)CC1 CCCCCC(C)(C)C(=O)NC1CN(C(c2cc(OC)no2)=O)C2(CCOC2)C1 C1(NC(C(CC=C)OC)=O)CC=C(C(=O)N2CC(O)CC2(C)C)C1 C1(NC(CC2(N(C)C)CC2)=O)C2CN(C(=O)C(F)(F)c3cncs3)CC12 CC1(C)CCN(C(C2CN3CCCC3CO2)=O)CC1CNC(c1cc(Cl)no1)=O C(=O)(C(CCC)C1CCCCC1)N1CC(N(C(CCOC(C)=O)=O)C)C1 c1(C(=O)NCCC2CN(C(c3c(C)ncn3O)=O)C2)nc(O)nc(O)c1N CCCCC(CC)CC(=O)NCC#CCNC(C1(O)CCCC(C)(C)C1)=O c1(CNC(C(=O)NCCc2ncn(C)c2)=O)ccc(-c2cncn2C)cc1 c1(OCC)cc(C(=O)NC2CC2CNC(c2cncc(C)c2)=O)ccn1 N1(C(c2cc(CNC(C(CC)C)=O)oc2)=O)CCC(C)(O)CC1 c1(OC)cc(CNC2CC(NC(c3ccc(F)cc3C(F)(F)F)=O)C2)ccc1I C1(F)(C(N(CCCC)CCOC)=O)CCN(C(=O)NC)CC1 c1(C(C)(C)OC)ccc(C(=O)N(CCNC(C2OCC2(C)C)=O)CC)cc1OC N(C(=NCCNS(C)(=O)=O)NC1CC(C)N(c2ccccc2)C1)CC(=C)C C12(NC(Cc3nnc(C)o3)=O)CC1CN(C(=O)CC1CCC(C)CC1)C2 c1(C(=O)NCC2(NC(=O)C3=COCC3)CC2)ccc2cc(N(C)C)ccc2c1 C(C(C(=O)NC(C1(O)CCCCC1)C)C(C)C)NC(c1cc(C)nn1C)=O N1(C(Cc2c(C)ccc(C)c2)=O)CCC(C)(C)C(NC(c2nc(=O)n(C)[nH]2)=O)C1 C(C(=O)N1C2CCC(C2)C1C(=O)NCCCc1ccncc1)(C(C)(C)C)OC c1(NC(C(CC2CC2)NC(Cc2ccn(CC)n2)=O)=O)cnc(F)cc1C C(C)(CC(=O)Nc1cnc[nH]1)NC1(CNC(C=CCOC)=O)CCC1 C1(CC(=O)NCc2ncc[nH]2)CCCCN1C(=O)CCC1CCCC1 N1(C(C(C(C)C)O)=O)CC2(C1)SCCC2NC(=O)CCCc1cnn[nH]1 Cc1nc2nccc(C(N3CC(N(C(=O)C(O)CC4CC4)C)C4(CC4)C3)=O)n2n1 c1(C(=O)NCC(=C)CCNC(C2(CSC)CCCC2O)=O)n[nH]c2c1CCC2 C1(NC(C(C(C)C)N2CCCC2=O)=O)CCCCN(C(=O)Cc2ccns2)C1 c1(C(=O)NC(CCCC)CNC(=O)Cc2ccc(F)nc2)c(F)cc(F)cc1F c1(C(C)C)nocc1C(=O)N(C1CN(C(C2CC2c2ccnn2C)=O)C1)C C(CN=c1[nH]nc(C(N)=O)s1)N(C(c1c(OC)ccc(OC)n1)=O)CC NS(=O)(=O)c1ccnc(C(N2CC(CNC(C34CCCC3CC(=O)C4)=O)C2)=O)c1 C1(OC)CN(C(=O)COc2ccc(Cl)cc2)CC1NC(=O)C=CSC N1(C(C(n2cc(CCC(CC)O)nn2)C)=O)CC(CN(C)C)CC1C Cc1nn(CC(F)F)c(C)c1C(=O)NCC1CC(NC(C2CCC(=O)N2)=O)C1 C1CCC2(CCCN(CCCSC)C2)OC1.C1CCCN(N2CCCCC2)CC1 CC1NCCCC1C(=O)NCCc1ccc(OC(F)(F)F)cc1 c1(C(=O)NCC(CC=C)NC(C2(CCOC)CCC2)=O)cc(C)c(C#N)c(C)c1 N1(C(c2cc(C)oc2)=O)CC(CC(=O)NC(C(C)C)C(C)C)C2(CC2)C1 c1(C(=O)NC2CC(NC(=O)CCC3CCC3)C2)cccc2c1OCC2 c1(NC(=O)CC2CC(OC)CN2C(=O)C(O)CSC)cc2cccn2cn1 Cc1nn(C)c(C)c1CC(N1CC2CC2(CNC(=O)Cn2nnc(=N)[nH]2)C1)=O N1(C(CNC(CN(C)C)=O)=O)CCCC2C1CCN2C(C1CCCS(=O)(=O)C1)=O c1(CC(=O)NC(CNC(CCC(C)SC)=O)(C)C2CC2)cccc(Cl)c1F Cc1nc(C)c(C(=O)NC2(CO)CN(C(c3c[nH]cc3-c3cnn(C)c3)=O)C2)o1 c1(NCC(CC)N(C)C)ncnc(NCC2CC2(C)C)c1C CC1COC2(CCN(Cc3cn(-c4ncccc4Cl)nn3)CC2)O1 Cc1cc(C2C(COC(=O)CCNC(c3cc(C)nn3C)=O)C2)cc(Br)c1 c1(C(=O)NC(C)C(C)NC(c2ccc(C(C)(C)C)s2)=O)c(Cl)ccc2ccoc12 Cc1c(C(=O)NC(c2cn(Cc3cccs3)nn2)C)sc2ccc([N+](=O)[O-])cc12 C1(C(=O)NCC2(C(N)=O)CN(C(c3c(CC)nc[nH]3)=O)C2)CC2C=CCC(C1)C2 C1(C(=O)NCCCOCCNC(CC(C)(C)C2CC2)=O)CC2(CCC2)CO1 C1(C)(NC(Cc2cn(C)nn2)=O)CCN(Cc2cc(F)ccc2F)CC1 C(=O)(C1=C(Cl)CCCC1)NCC(C(C)C)C(=O)NC(CC1CC1)C1CC1 c1(C(N(CC)CC2CCC(C)CC2)=O)nn(C)c(CC)c1Br CCCC(CNC(c1nc(CC)oc1C)=O)C(=O)NC.C(=O)(C(C)(C)OC)NC C1(C(=O)NC2CCC(CNC(CCOC(C)C)=O)C2)CCC(C(F)(F)F)CC1 c1(C(=O)NC2C(NC(C3C(C)C3)=O)CCC2)cc2ccccn2c1 N1(C(Cc2cc(COC)on2)=O)CC2CC2(NC(=O)CC(C)(C)C)C1 C=C(C)CCC(=O)NC(C1CCN(C(c2cc(C3(C)CC3)on2)=O)CC1)(C)C c1(NC(=O)NC)ccc(C(N2CCOC(COC(C)=O)C2)=O)c(F)c1 C1(C2(NC(C3(OC(C)C)CCC3)=O)CC2)CCCN1C(=O)Cn1cc(Cl)cn1 C1(C(=O)NC23CN(C(CCNC(N)=O)=O)C(CC2)CC3)CCc2nnc(O)n2C1 c1(OC)cc(CO)ccc1C(=O)NCCCCCNC(c1ccc(Cl)c(C)c1)=O C1(C)(C(=O)NCC(C2CCCC2)NC(C2C(COC)(CC)C2)=O)CCCN1C N1(C(CC2(C=C)CN(C(=O)CCc3cn[nH]c3)C2)=O)CCc2ccccc2C1 c1(CCC(=O)NC2(C(N)=O)C(C)CCCC2)ccc2ocnc2c1 N1(C(C(CC=C)OC)=O)CC2CC1CC2NC(c1ccc(OC)s1)=O Cc1nc2n(n1)CC(C(=O)NCC(C)(CO)NC(c1ccc3c(c1)CC3)=O)CC2 C(=O)(C(CC(C)C)NC(=O)C(N1CC(O)C(C)(C)C1)c1cccnc1)OC C1(NC(C2(C)CCN2C(=O)COC2CCCOC2)=O)CCCC12CC2 N1(C(CCCN=[N+]=[N-])=O)CC2CC(NC(C3COC(=O)C3)=O)C(C2)C1 C1(NC(c2c(CC)cc[nH]2)=O)CC2CCC(C1)N2C(c1cc[nH]c(=NC)c1)=O C=CCN=C(NCc1cc(Br)cs1)NC(C)(C)CCC CC(N=c1nc(N2CCCOC(C)C2)c2sccc2[nH]1)c1ncc(Cl)cc1Cl C=C=CC(C)C(=O)NC1(C(=O)NCc2nnn(C)n2)CCSC1 c1(OCCCC(=O)NCC(CNC(C(F)=CC)=O)O)ccccc1Br CC(CF)CC(=O)NCCCCN1CCC(NC(C2(CF)COC2)=O)CC1 c1(C(=O)NC2CC(NC(c3n(CCCC)ncc3)=O)C2)cc2c(C)nn(C)c2s1 CON1CC(C(N2CCOC(CC(=O)NCC(C)CN(C)C)C2)=O)CC1=O CC1(C)C=CC(NC(=O)C(O)C2CN(C(C3CCC4(CCC4)C3)=O)C2)CC1 Cc1cc(C(N2CCCC2CN(C(=O)C2=CCCOC2)C)=O)cc2ccoc12 N1(C(C(C)CF)=O)CCCCC1CCCNC(=O)CCCc1cccs1 c1(C(=O)NCC(=O)NCCCNC(CN2CC(C)C2)=O)ccc(O)cc1C(C)C C12(C(N3CC(O)(C(=O)OC)C3)=O)CC1CCN2C(=O)CC1COC(=O)C1 c1(-n2c(-c3n(CC=C)nnn3)nc(-c3cccc(C)c3)n2)cc(CSC)ccc1Cl c1(C(=O)NCC(C)N(C)C(c2cnc(Cl)c(N)c2)=O)cc2ccncc2c(O)n1 c1(N(C)CC2CCCS2)ccc(S(=O)(=O)NC2CCC3(CCCC3)C2)c(Cl)c1 N1(C(=O)NCCCC(C)c2ccccc2)CC(C)(C)CCC1CO CC(N=c1ccnc(NC2CCN(C3CCCCC3)CC2)[nH]1)c1nnc(CO)s1 C(=O)(C(C)C(=O)NCC1CN(C(C2(CO)CC(F)(F)C2)=O)CC1C)OC C1(NC(c2c(C)nc[nH]2)=O)CCN(C(c2ncnc3c2CCC3)=O)CCC1(F)F CC12CC1CCN2C(c1ccc(C(Cl)Cl)cc1)C(=O)NCc1cccs1 c1(SC)ccc(NC(=O)C(N)CCc2cn[nH]c2)c(C)c1.C12CCCCN1C2 C1(C(=O)NCC#CC(N2CC(F)(C(=O)OC)C2)=O)CC(O)C(F)C1 C=C1CCN(C(=O)CC2CCOC2=O)C(C(=O)Nc2ccc(CO)nc2)C1 C=CC1CN(C(c2nncn2C(C)C)=O)CCO1 CC(C)(C)CCCCC(=O)N1CC(NC(=O)C(F)C2CCOC2)C2(CCCC2)C1 N1(C(CC(C)C)=O)CCC(CN(C)C(c2ccncc2Br)=O)CC1 c12cccc(c1)C(=O)NC1CC2C1.c1(COC)ccc(C(F)(F)F)[nH]1 c1(C(=O)NCC2CC3CN(C(Cc4cc(C)no4)=O)CC32)cc2c(s1)CCSC2 C1(C(N2CCC2CNC(C2(Br)CC2)=O)=O)CC(O)(c2cccnc2)C1 N1(C(C2C(=C)C2)=O)CCC2(CCCN(C(c3onc4ccccc34)=O)C2)CC1 CC(C(=O)NC1(CNC(=O)CCN2CCCCCC2)CCC1)C(F)(F)C(F)F N1(C(=O)OC(C)(C)C)CC2CC(C1)C(F)(C(=O)NCCCc1cn[nH]c1)C2 c1(C(N2C(CS(C)(=O)=O)CC2)=O)c(F)cc(C(F)(F)F)cc1F N1(C(=O)Nc2nc(NC(c3coc(Cl)n3)=O)sc2)CCC(F)(F)CC1 C1(NC(c2c(N)cccn2)=O)CC2CCC(C1)N2C(c1cocn1)=O c1(C(=O)NC2CCC2NC(=O)C(O)C(F)(F)F)cncc2ccccc12 C=Cc1ccc(C(=O)NOCC(=O)NCCc2cnoc2)cc1 c1(C(N2CCCC(NC(C34CC(F)(C3)C4)=O)CC2)=O)cccc2cc(O)ncc12 C1(CNC(c2cn(C3CC3)cn2)=O)CC(C(=O)NCC2CC23CCCCC3)=NO1 C1(NC(C2C(C)CCC2)=O)CC2(C1)CN(C(c1ccc(=O)oc1)=O)C2 C1(NC(C2CCC(CC)O2)=O)CC2CC(C1)N(C(c1c(C)noc1Cl)=O)C2 N1(C(c2cc(CNC(CCOC)=O)ncc2)=O)Cc2ccc(C)cc2C1 CC1(C)CCC(C(=O)NC2CCCC2CNC(C2CC2C2CCCO2)=O)CC1 C1(C(N(CCCN(C)C(c2cc(O)n(C)n2)=O)C)=O)CCC2(C1)N=N2 C1(C(=O)NC(C(=O)NCC(C#C)(C)C)CC2CCCC2)CCCN1C=O N1(C(=O)NC2C(OC)(OC)CC2)CCCC(C)(C(=O)N(c2ccccc2)CCF)C1 CCC(CCOC)C(=O)NCCC1CCCCN1C(c1nn(CC)cc1Cl)=O c1(C(C(=O)NCC2(O)CCN(C(C(C=C)O)=O)CC2)(F)F)ccc([N+](=O)[O-])cc1 C1(NC(C(CC)C)=O)CN(C(c2cc(CO)n(C)n2)=O)CC1(C)C CC1CCN(C(=O)CN2CCCCCC2)C(C)C1NC(c1c[nH]c(C(N)=O)c1)=O N1(C(c2nc(C)sc2)=O)CCN(C(=O)CCc2cccn2C)CC(CO)C1 C(=O)(CCCCCC(C)(C)C)N1CC(CNC(C(C)C2CC2)=O)C(C(F)(F)F)C1 c1(C(N2CCC(NC(C(CCCCC)O)=O)C(C)C2)=O)cc(C)cn2ccnc12 N1(C(c2scc(CCC)n2)C(=O)NC(C)C)CC(C(=O)OC)OCC12CCC2 C1(C(N(C2CCCCCC2)C)=O)COCCN1C(c1cocn1)=O CC(C)(CCNC(C1(C)CC1(F)Cl)=O)NC(=O)Cc1cccnc1 C(=O)(NNc1ccc(Cl)cc1Cl)C1C2(CCN(C(=O)OC(C)(C)C)CC2)CC1 N1(C(c2c(C)occ2)=O)CC2CC(CNC(=O)COCCOCCO)CC1C2 C1(CNC(CC(COC)C)=O)CC2(CO1)CN(c1cc(C)nc3ncnn13)C2 CC(C)CC(CNC(C1CC(C)CCO1)=O)C(=O)N(C1CCC(CO)CC1)C C1(OC(C)(C)C)CC2(C1)CC2C(=O)Nc1cccc(C(=O)NCc2ccoc2)c1 C1(C(N2CC(C)(NC(=O)CC3CC3(C)C)C2)=O)Cc2ccccc2S1 Cc1cc(F)c(F)cc1C(N1CCC(F)(F)C(NC(=O)Cc2ncccn2)C1)=O C1(C(=O)NC2CCC2C(=O)NC(C2CCN(C)C2)C)(COC)CC=CC1 C(C1(C)CCOCC1)=CC(N1CCC(COC)(NC(C2CCSC2)=O)C1)=O N1(C(c2nc(C)sc2)=O)CC(CNC(=O)CCc2cc(Cl)cs2)CC(C)C1 CC1=CC(NC(c2cncc(CNC(=O)Cc3cccnc3)c2)=O)CCC1 C(C)(c1ccccc1)=CCONC(C1N(C(CC(C)SC)=O)CCC(O)C1)=O C1(C)(OCCOC)CCCN(C(=O)CC(C)(O)CN)C1 C1(NC(c2n(CC)c(O)nc2)=O)CC2CC(NC(C3CCC3(C)C)=O)C2C1 Cc1ccc(C=CC(=O)NC2CCC(CCNC(=O)Cn3cnnc3)C2)cc1Cl c1(-c2cc(C)c(F)cc2F)ccc2[nH]c(C(=O)NC(c3ncccn3)C)nc2c1 N1(C(C(CC(C)(C)NC(c2c(OC)nn(C)c2)=O)F)=O)CCC(C2(C)CC2)CC1 C1(CC(=O)NC(C2CN(C(Cn3ccc(C)n3)=O)C2)C)CCS(=O)(=O)CC1 C1(CC(N2CC(CNC(N)=O)C2)=O)CN(C(c2ccc(F)cn2)=O)CC12CC2 C1(CNC(c2nc(COC)sc2)=O)CC2CCC1C2 C1(CC(=O)N(C2CN(C(=O)Cc3nc[nH]n3)CC2F)C)CCC2(CC2)CO1 Cc1ccc2c(c1)CN(C(C1CSCCN1C(C1CC1(F)F)=O)=O)C2 N1(C(C2CN(C(N)=O)C2)=O)CCCC2(CCN(C(=O)CCC3CCCOC3)C2)C1 N1(C(C2CC(CNC(C3(C)CCC(=O)CC3)=O)OC2)=O)CCCC2(C=CCO2)C1 c1(C(N2CCC(COC)(NC(C3CC(n4cnnc4)C3)=O)C2)=O)ccc(F)cc1O c1(C(=O)NC2C(NC(CC(C)n3cccc3)=O)CC2)cnn2ccccc12 Cc1cccc(OC(C)C(=O)NCC#CCNC(C2(COCC)CCOC2)=O)c1 c1(NC)ccc(CN(C)CCNC(C2CCCN2C2CCCC2)=O)s1 c1(C(=O)NC(CC=C)CNC(=O)Cc2csc(C)c2)cc(Br)n(C)c1 C(C(C)N=c1[nH]c(=NCC2CC2(Cl)Cl)c2ccc(C(F)(F)F)cc2[nH]1)OC C1(C(N(C(CC)CO)C)=O)(CNC(=O)CCN2CCCCC2)CC(C)(C)C1 c1(CCC(=O)N2c3cc(n(C)c3)C2)ccc(F)cc1Cl.Cc1cncc(N)n1 c1(N(CC(F)(F)F)C)ccncc1S(=O)(=O)NCCSCC1(CC)CC1 C1(NC(CS(=O)(=O)NCC)=O)CCC12CN(C(c1sc(COC)nc1C)=O)C2 c1(NC(C(=O)Nc2c(CC(=O)OCC)cccc2)=O)c(C)cc(C#N)cc1C c1(CC(=O)NCC(C)(C2CCC2)NC(c2[nH]cc(C(C)=O)c2)=O)cnccc1Cl c1(CCC=C)ccc(NC(CC2CCN(C(c3ccccc3)=O)C2)=O)cc1.C1COC1 C1(C(=O)NC2C(NC(c3ccn(C)c3)=O)COC2)CCC12CCC2 C=CC1(C(=O)NC2CC2CNC(C2CC2c2cccc(OC)n2)=O)CCOCC1 c1(CCCOC)cc(Cl)c(C(=O)NC2(CC(C(=O)NCSC)C3CC3)CC2)cc1Cl CC(C)CC(F)C(=O)Nc1cnn(C2CCN(Cc3cc(Cl)ccc3O)CC2)c1 C1(C(=O)NC2CC(C(=O)OC)C2)CN(C(=O)CCc2ncnn2C)C2(CCC2)C1 C1(NC(c2n(CC)ncc2)=O)CCC(NC(=O)COC2CCC2)CC1 N1(C(C=CC)=O)CCCC(CNCc2cc(O)ccc2F)C1c1ccccc1 CCC(CNC(c1cc(F)ccc1C)=O)(CC)C(=O)NC1(CO)CC2CCCC12 C(C(O)(CNC(C1CC(C)(NC(=O)CC(C2CC2)C2CC2)C1)=O)CO)OC C12(CNC(C=C(C)C(C)(C)C)=O)CC(CO1)N(C(c1cnn(C(F)F)c1)=O)C2 N#CC1(C(=O)N(C2CCN(CC(F)(F)F)C2)CC)CCC1.N1CCC1CN1CCCC1 Cc1nn(C)c(C)c1CC(N1CC(CC(C)N(C(=O)CCc2cnoc2)CC)C1)=O N1(C(CCCc2cn(CCCCSc3cn(C)nc3)nn2)=O)CCNC(=O)CC1 C1(C(N2CCCCC2CNC(c2cnsc2C)=O)=O)(CC)CCOCC1 N1(C(c2c(C)snn2)=O)CC(NC(=O)C(F)C2CCC2)C(C(F)F)C1 C1(CNC(C=CC(CC)=CC)=O)CC2CCC1N(C(=O)Nc1ccc(N)cc1)C2 CCC(CC(=O)N(C)CCC1CCN(C)CC1)C1CCC1 c1(C(C(=O)NCCC2OCCN(C(COCC(=C)C)=O)C2)C)c(F)cccc1F C1(C2CC2)(CNC(C(C)OC)=O)CCN(C(C2(OC)CCS(=O)(=O)C2)=O)C1 N1(C(c2ncn(CC)c2)=O)CCN(C(c2cccc(CSC)c2)=O)C(CCO)C1 C1(C)(CNC2(COC)CCC2)CCCN(C(=O)Cc2nn(C)cc2Br)C1 c1(C(=O)NC2CCN(C(CC3(C#N)CCC3)=O)C2)csc2nnsc12 CCCCS(=O)(=O)NC(C)C(=O)NCC1(NC(C2CCC3CC23)=O)CCCCC1 C1(C(=O)NCCN(C(=O)C#CC2CCOC2)CC)CCc2cncn2C1 c1(C(=O)NC(C2CCN(C(c3ccncc3)=O)C2)(C)C)ccc2c(c1)OCCO2 c1(SC)cccc(N2CCC(C)(NC(=O)CC3CC4CCC3C4)C2)c1[N+](=O)[O-] c1(CC(=O)N(CCNC(c2ccc(O)nc2Cl)=O)C2CC2)nnc2n1CCOC2 C12(CNC(CSCC=C)=O)CCC(C1)N(C(c1ncc[nH]c1=O)=O)C2 N1(C(C(CNC(c2ccsc2)=O)N(C)C)=O)CC2(COCC(=O)N2)C1 c1(C(N2C(C(C)NC(=O)C=Cc3cocn3)CCC2)=O)cc(Br)c(F)cc1N C1(NC(CC2(OC)CC2)=O)CCC(NC(=O)COCC2CCOC2)C1 C(=O)(C1=CCCCCC1)N1CCCC(C(N(C)Cc2snc(C)n2)=O)C1C C#CC1CN(C(c2ncn(C)n2)=O)CCN1C(c1nnsc1N)=O c1(OCC)cc(C(=O)NC2(CCNC(C3CC(C#N)C3)=O)CCC2)cc(F)c1 N1(C(C(C)c2ccsc2)=O)CCC(O)(Cn2cc(CC3CCN(C)CC3)nn2)C1 Cc1ccc2c(c1)CN(C(=O)N(C1CCCCC1)C1CCC1)C2 C1(c2n(CCOC)nnn2)(NCCOCCNC2(C)CSC2)CCCC1C CCC(CC)C(F)C(=O)N(C1CCN(C(=O)C(C)(C)C(C)O)C1)CCO c1(C(=O)NC2CN(C(=O)C(c3cccc(F)c3)C3CC3)C2)cc2n(n1)CCCC2 Cc1cc(C(N2CCC2CNC(c2c[nH]nc2C)=O)=O)c(N)c(Cl)c1 N1(C(C=CC(=O)NC2CC2)=O)CCN(C(=O)CCC2CCCCO2)C(CCO)C1 C1(NC(c2c(CC)ncs2)=O)CCN(C(c2cc(S(N)(=O)=O)cs2)=O)CC(O)C1 c1(C(C)Nc2c(C(=O)OC)cc(C)cn2)nccc2ccccc12 C1(NC(=O)CC2CC(O)C23CCC3)CC2CC(C1)CN(CC=Cc1ccoc1)C2 Cc1cc(CN(C(=O)C(N2CCCC(c3ncc(F)cn3)C2)=O)C)ccc1Br c1(C(N2CCCC(C#N)C2)C(=O)NC)ccc2c(c1)OCC2(C)C C12(CNC(c3cccc(NCC(N)=O)c3)=O)CCC1CCN2C(=O)C1=COCC1 N1(C(C(Cc2ccc(OC)cc2)=O)=O)CCC(C)(C)C(NC(c2cnco2)=O)C1 C1(CNC(c2cc(CC)ncn2)=O)CN(C(=O)C2=CCCC2C)C2CCCC2O1 C1(NC(C2C(OCC)CC2)=O)CCCC(NC(c2nnn(C)c2CC)=O)C1 Cn1ccc2nc(N3CCCC3CN(C)C(c3cn(C4CC4)cn3)=O)ncc12 c1(C(C)(C)C)ccc(NC(N2CCC(c3ccncn3)CC2)=O)c(Cl)c1 c1(C(=O)NCCC(CNC(C2CCN(OC)CC2)=O)O)cccc2sncc12 C1(CC(=O)N(C(C(C)SC)C)C)C2CCCC2N1C(=O)C(C1CCCCC1)F N1(C(C(C)N(C)C)=O)CCCC2(C1)CN(C(c1cc(N)ccc1Cl)=O)CCO2 c1(NC(C2(CO)COC2)=O)cc(Oc2ccccc2)ccc1CO c1(C(=O)NCC2CCC2NC(c2c(F)cccc2Cl)=O)ccc2c(n1)CCC2 C(N=c1ccnc(N(CCCC(C)O)C)[nH]1)c1n(C)nc(OC)c1CO C(CC(C)N=c1cc(C(C)C)nc(C)[nH]1)NC(n1ncc2cc(CC)cnc12)=O C1(C)(CC)CC(NC(=O)C(c2ccco2)NC(=O)CC2CCCC2O)C1 C1(C(=O)OCC2CC3CN(C(C(C(C)C)C)=O)CC32)COc2ccccc2O1 C12(NC(CCN(C)CC)=O)CCC(CNC(=O)C(F)n3cccn3)(C1)OC2 N1(C(C2C(=C)C2)=O)CC(O)CC1(C)C(=O)NOCCCC n1(CCCC)cc(NC(C2CCCN2C(=O)C(Br)NC(C)=O)=O)cn1 N1(C(C2CCC(C)(C)CC2)=O)CC2CC1CCC2NC(=O)CN1CCCNC1=O c1(C(N2CC(O)(CNC(C(C)(C)F)=O)C2)=O)nccc2c(Cl)cccc12 C1(CC#N)(NC(=O)CCc2ccc(O)cc2)CCN(c2nccc(C#N)n2)CC1 C1(CC(C)(C)C)CN2CCN2C1.C1(CC(=O)NC2COC2)CCCCS1 C1(NC(C2CCC(=C)CC2)=O)COC2CN(C(C3(CF)CC3(F)F)=O)CC12 n1(CCNC(=O)NC(C)C)cnc(C(=O)NC(C2CCCC2)CO)c1 C1(F)(CNC(CN(CC(C)C)C(C2CCOCC2C)=O)=O)CCCCC1 CCS(=O)c1ccc(-c2ccc(C3(NC(=O)C4=NNC(=O)CC4)CCC3)s2)cc1 c1(C(=O)NC2(C)CN(C(c3cnc(C(C)(C)C)o3)=O)C2)csc2nccn12 CC1(CNC(=O)CCOc2ccccc2F)CCN(c2nnc(C3CC3)s2)C1 N1(C(COC(CC)C)=O)C2CCC1C1CC1(NC(=O)Cc1c[nH]nc1O)C2 C1(O)(CNC(=O)CC2CCC2)CCCN(C(=O)CCOCC(F)(F)C(F)F)CC1 C(=O)(CC(F)(F)CS(C)(=O)=O)N(CCCNC(=O)CCn1ccnn1)C N1(C(c2cc(O)no2)=O)CCC(c2ccccc2)C(NC(=O)C2=COCC2)C1 CCC(C)(CNC(=O)C(C)C1CCCC1)C(=O)N1CCN(CCF)CC1 c1(C(=O)NCC2(C)C(C)CN(C(COCCC=C)=O)C2)c[nH]c2cc(Cl)ccc12 c1(N(C)Cc2n(CC)ncc2)ccc2c(c1)nc(C(=O)O)n2C C1(NC(C2N(CC)CCOC2)=O)C2CC(O)C1N(C(=O)CCP(C)(C)=O)C2 C1(CNC2(C)CC2)CC2CCC(C1)N2c1cc(NC(=O)OC(C)(C)C)ncn1 C1(C(=O)NCC2(C(N)=O)CN(C(c3c(F)cccc3F)=O)C2)CCC2C1C2(F)F C1(NC(c2nc(C)[nH]n2)=O)CN(C(c2ccc(O)c(Cl)n2)=O)CC2(CC2)C1 Cn1cc(NC(=O)NCC23CC=CCN2CCC3)cc(Br)c1=O C(=O)(CC(COC)COC)NC1(CCNC(C2C(CC)OCC2)=O)CCCC1 c1(C(=O)NCCN(CCOC)C(c2cnc(Cl)cn2)=O)cnc2c(c1)CCOC2 C=Cc1ccc(C(N2CCCCC2CC(N2CC(C(C)(C)O)C2)=O)=O)cc1 N1(C(CN(CCC)C(C2CC(C)CO2)=O)=O)CCC2CN(C)CC12 CC1CC(C)N(C(C23CC(C)(C2)C3)=O)CCN1C(=O)CCCc1cnn[nH]1 c1(CC)cc(CNC(=O)CCCN(C)C)on1.C12(CSC1)C(=O)N2 N12CCC(CC1)NC(=O)C2.C(C(C(=O)NC(CN(C)C)CC)NC(C)=O)OCC c1(C(N2CC(C(C)NC(C(CC)C#N)=O)OCC2)=O)cnc2sccn2c1=O N1(C(C=C(C)C)=O)CCC(N(C)C(c2cc(C(F)(F)F)ccn2)=O)C(C)C1 C12(CNC(CCC#C)=O)CCC(CC1)N(C(C1OCCCC1(C)C)=O)C2 N1(C(COCCCC(C)C)=O)CC(NC(=O)CC2CSCCS2)CC1(C)C C1(NC(C(C)CO)=O)CCN(C(=O)NC2CCCC2C#N)CC1 C(=O)(C(C)C(C)CC)NC(CC)CNC(C12CC(CC(F)F)(C1)C2)=O N1(C(c2ncc(C)c(C)c2)=O)CCC(NC(c2c(Cl)nsc2Cl)=O)C(CO)CC1 Fc1ccc(CCC(Cl)Cl)cc1.c1(C(CC2CCC2)NCC)nnnn1CC(F)F C1(NC(=O)CCC2CCOCC2)CC2CC(NC(c3cnc(C(F)F)s3)=O)CC12 C(=O)(CC(C)(O)COC)N(C(C)CNC(c1csc(-c2cn[nH]c2)n1)=O)CC CCC(COC)C(=O)NC(CNC(c1ccc(OC)s1)=O)CCOC C(C(C)(O)C(C)(C)C)NC(C(C)OC)=O.C(=O)CC=C(Cl)Cl N1(C(c2c(C)nn(C)c2)=O)CC2(CCC(NC(C3OCC4CCCC34)=O)CC2)C1 c1(CC)c(C(=O)N(C)CCOCCN(C(=O)C(C)COC(C)=O)C)cnn1C C1(O)(C(=O)NCC(C)CNC(c2c[nH]nc2-c2ccoc2)=O)CCSC1 c1(OC)cc(F)c(C(=O)NCC2CCC(NC(=O)CCS(C)(=O)=O)C2)cc1OC c1(C(C)(C)C)cn(CC(N2CCC(OCCOCCOCCNC(N)=O)C2)=O)nn1 c1(CC(=O)N(C(C)CNC(=O)CC2(N3CCCC3)CC2)C)ccnn1C1CCC1 C1(CNC(C2N(CCCC)CCCC2)=O)CC(F)(F)CN1C(=O)CC1CN(C)C1 C#CC1CC2CCC1N(C(c1conc1C(C)NC(=O)CCCN=[N+]=[N-])=O)C2 C1(CNC(C(C2CCOCC2)OC)=O)CC2(CCN(c3nc(CO)ns3)C2)CO1 C1(N(C(CC2N(C)CCC2)=O)C)C2CN(C(=O)CCCCN3CCCC3)CC12 C=CC(C)CC(=O)NCCC1CC(NC(c2c(C)noc2CC)=O)C1 N1(C(C(C)OC(C)(C)C)=O)CCC2(NC(=O)CSc3ccc(CO)cn3)CC2C1 N1(C(C23CCC(OC)C2C3)=O)CC(C(=O)NCc2ccc(Cl)nc2)C(C2CC2)C1 c1(C(N(C)C)=O)cc(C(=O)NCC2(NC(=O)CCCC3CC3)CCOC2)ccn1 c1(C(=O)NCC2OCCN(C(CC(C)CF)=O)C2)n[nH]c2c1NCCC2 C1(C(=O)NCC(C)(O)CNC(=O)CC2CCSC2)CCC(=O)N(C2CC2)C1 C1(C(N2CC(C)(N(C(C3(C(=O)OCC)CC3)=O)CC)C2)=O)CCS(=O)(=O)N1 CC(C)(CO)C(=O)NCC(C)(O)CNC(C1(Cc2cccc(Cl)c2)CCC1)=O c1(C2N(C(C(C)NC(C=C(COC)C)=O)=O)CC2)ccccc1 N1(C(c2nn(C)c(CO)c2)=O)CCN(C(c2csc(Cl)c2)=O)CC2CCCCC12 C(c1ccc2cc(F)ccc2n1)=CCNC(=O)NC(c1c(C)ccc(Cl)c1)=O C1(CNC(c2cc3ccccc3cn2)=O)CC2(CCN(C(=O)CCF)CC2)CO1 C(=O)(C(C(C)CC1CC1)N(C)Cc1sccc1C)NC(CC)(C)C C1(C(N(CCNC(C(CC)Oc2ccccc2)=O)C2CC2)=O)CCCC(=O)O1 c1(OCC(=O)N(CC(=O)N(CC(COC)O)C)CCOC)cccc(F)c1F Cc1cc(C(N2CC3C(CNC(=O)C=Cc4ccncn4)C3C2)=O)c(C)nc1C c1(C(=O)NC2CCC2CNC(=O)C(C2CC2)C2CC2)ccc(Br)cc1 c1(CN2CCN(Cc3c(C(=O)OC)cccc3)CC2)coc2c(Cl)cc(F)cc12 c1(C(=O)NC2C(NC(C(C(C)(C)C)OC)=O)COC2)c(Cl)ccc2c1OCO2 N1(C(CC2(OC)CCC2)=O)CC(CNC(=O)OC(C)(C)C)CC2COCCC12 Cc1nn(CCO)cc1C(=O)NCC1CC1.c1(C(=O)NCC2(C)CC2)cnc(CO)o1 CC1CN(C(=O)Cn2cnc(Br)c2)CC1NC(c1cc(CF)on1)=O CC(c1ccsc1)=CCNC(C1N(C(=O)OC(C)(C)C)CC1(C)C)=O C(=O)(CS(=O)(=O)C1CCCC1)NC(CC)CNC(=O)CC12COC(COC)(C1)C2 C1(N(CCC)C(C2CC2n2nccn2)=O)CCN(C(=O)C=CCOC)CC1 C1(NC(CCCC(C)C)=O)CN(C(=O)CCC(C)O)CC12CCS(=O)(=O)CC2 c1(C(=O)NC2CCC(C)N(C(=O)C=CC(=O)N(C)C)C2)cnc2sccc2c1 C=C(C)CCC(=O)NC(CNC(c1ncc[nH]c1=O)=O)CCCC N1(C(C=C(CC)C)=O)CCC(CCNC(=O)C=C2CCC2)C(F)(F)C1 Cc1cc2nccnc2cc1C(=O)NCCC(C)(C)NC(c1ccccc1O)=O CCC(CC)C(F)C(=O)N1CCOCC1C(=O)NCc1cncn1C(C)C c1(C(=O)NCC(c2ccccc2)NC(CC(=O)NCC#C)=O)cc[nH]c(=N)c1 c1(C2(NC(C=CCN(C)C(C3CCC(C(N)=O)C3)=O)=O)CC2)ccc(F)cn1 c1(C(=O)NCCCNC(c2c(C)nc(=N)[nH]c2)=O)nc(Br)c2ccccn12 C(C(=O)NCC(C1CCCC1)NC(=O)CC1NC(=O)NC1=O)(C(C)(C)C)OC C1(C(=O)NCC(C)NC(C2CN(S(CC)(=O)=O)C2)=O)CCCC1CC(F)(F)F Cc1sc2nc(SCc3ccc4c(c3)CCNC4)nc(N(C)C)c2c1C c1(C(N2C(C3CCN(c4nnc(C)s4)C3)CCC2)=O)ccnc(F)c1Cl C1(CNC(c2cn(C)nc2Cl)=O)(NC(c2ccncn2)=O)CC2CCC1CC2 C12(NC(C(COC)(C)OC)=O)CCC(CN(C(=O)CCc3cnc[nH]3)C1)C2 CC(C)(CO)C(=O)NCCCNC(=O)Cc1ccnn1C1CCOCC1 C1(NC(C2C3CN(Cc4ccc(S(N)(=O)=O)o4)CC32)=O)CCCC2CCCCC12 C(=O)(CCCCC(F)(F)F)NCC1(C)CC(NC(c2c[nH]cc2Br)=O)C1 c1(C(=O)NCCN(C(CCC#CC)=O)CC2CC2)ccc2c(c1)CC(=O)NC2 c1(C(=O)NCC(CC)NC(c2cnc(O)c(C)c2)=O)ccc(O)nc1Cl c1(C(=O)NC2C(CNC(C3CC(=C)C3)=O)CCCC2)cc(C(N)=O)ccc1O CC1(C)CC(N=c2[nH]c3c(c(=NCc4ncc(C(C)(C)C)s4)[nH]2)CCCCC3)C1 c1(OC)ccc(-n2nc(-c3ccccn3)nc2-c2cnc(C)[nH]2)cc1 S(=O)(=O)(c1cccnc1Cl)N1C2C(C(=O)Nc3ccnc(Br)c3F)C(C2)C1 CCCCC(C(=O)NCC=CCC(N1CCCC1C1CC1)=O)C(C)C.C(C)(C)C C1(N(C(c2cc(CSC)on2)=O)CC)CCCN(C(C2(C)CC2)=O)CC1 CCCCC(C(=O)NCC1(C)CCCO1)NC(c1cn(C)nc1C)=O C1(NC(C=NOC)=O)CCCC(NC(=O)C(c2cscc2Br)C)C1 C=CCC(C)(C)CNC(=O)C(C)=CCNC(=O)Cc1sccc1C CC(C(=O)N1OC2CCC1C(O)C2O)C1CC(NC(=O)OC(C)(C)C)C1 CS(=O)(=O)c1cccc(C(N2CCOC3(C2)CN(C(=O)C2=COCC2)C3)=O)c1F C1(C(=O)OC)CCN(CCn2nnnc2COCC(F)(F)F)c2ccccc2C1 c1(C(N2CCC(CCC)C2)C(=O)NC)cnc(C)n1CCOCC C1(NC(C2C(CC)OCC2)=O)CCCCC1NC(C1(COC)CC=CC1)=O C(=O)(C1=CCC(C)(C)CC1)NCC1C(NC(c2c(C)nn(C)c2N)=O)C1 CC(C)(O)CC(=O)N1CCC(CC(=O)NC2COC(C(F)F)C2)CC1 C(=O)(CC1=NN(C)C(=O)C1)NCC(CNC(COc1c(CC)cccc1)=O)OC C1(NC(c2ccc(C(F)(F)F)o2)=O)CCCCC1NC(C1CC12CCC2)=O c1(C(F)(F)F)ccc(N2CC(c3ccc(F)nc3)C2)nc1 N(C)(C1CCOc2cc(F)ccc21)C(C1OCC(=O)N(CC)C1c1nccn1C)=O CC12CC(C(=O)NC3CCCCC3NC(=O)C(F)C3CC3)(C1)C1(CCC1)O2 c1(CC(N2CC(CNC(C(c3n(C)ncc3)(C)C)=O)C2)=O)ccccc1S(C)=O C1(CC(=O)NCc2ccnc(C(F)(F)F)c2)CN(Cc2ccno2)CCO1 Cc1nc(CC(N2Cc3ccccc32)=O)sc1SC(F)(F)F N1(C(CC(C)N(C)C)=O)CC2C(CC(=O)NC3CCCCCC3)C2C1 N1(C(c2c(OCC)cc(Cl)cc2)=O)CCC2C1CCCN2C(=O)C1=CCCS1 C1(CC(=O)NC)CN(CC(c2cccc(OCC(Cl)(Cl)Cl)c2)=O)CCO1 c1(C(=O)NCC2CCCC(CNC(=O)CCF)C2)cncc2sccc12 N1(C(CCCSC)=O)CCn2ncc(S(C)(=O)=NC(=O)C(O)CSC)c2C1 C1(NC(c2cnc(CCC)s2)=O)CCCC(NC(=O)Cn2cc(C3CC3)cn2)C1 N1(C(C(C)C2CCC2)=O)CCC(NC(c2cc(C(C)(C)C)no2)=O)C(O)C1 N1(C(C2C(C(=O)OCC)C2)=O)CCC(n2cc(-c3cnn(CC)c3)nn2)CC1 C1(N(C(C(CC(C)C)O)=O)C)CC2CCC(C1)N2C(C12CC(C)(CO1)C2)=O C=CCC(CNC(C1(CCN(C)C)CC1)=O)NC(=O)C(C)CC1CC1 C1(NC(C(C2CCOCC2)C)=O)CCN(C(=O)CCS(N)(=O)=O)CC1(C)C N1(C(C(C2CC2)OC)=O)CC2CC(C(=O)N(C)CC3CCN(C)C3)(C2)C1 c1(C(N(C2CCCN(C(=O)C=CC(C)(C)C)C2)CC)=O)cc(F)c(Cl)cc1Cl C#CCCC(C(=O)Nc1cccc(Cn2cc(C3CC3)nn2)c1)OC c1(C(=O)NCC2(O)CCCN(C(C3CC3F)=O)C2)cccc2scnc12 N1(C(C2C(CC)OCC2)=O)CCCC(N(C(=O)C=C(C)c2ccco2)C)CC1 C1(C(=O)NC2CCC(OC)C2)CC2(CCN(C(=O)C3Cc4ccccc43)CC2)C1 C1(C(=O)NCC2CC(NC(CC(C)(C)O)=O)C2)CCC2C(C1)C2(F)F c1(-n2c3ccc(cn3)c2=O)ncnc2c1CCC2.C1(CCOC)CCCNC1 CC(C)(CC(F)C(=O)NCCCc1nncs1)NC(=O)C(O)CC(F)(F)F C=CC1(CC(=O)NCc2nc(C3CC3)no2)CN(C(=O)CC(C)F)C1 C(CC)(CC(F)(F)F)NC(CCC1CCN(C(CN(C(COC)=O)C)=O)C1)=O CC1(C(=O)N(CCNC(=O)COCCF)CC2CC2)NC(=O)NC1=O N1(C(CNC(C(CC)CC)=O)=O)CC(C2CN(C(c3ccccc3Cl)=O)C2)C1 N1(C(c2c(C)scn2)=O)CCC2(CC1)CC(NC(C1(F)CCCOC1)=O)CO2 C12(C(N3C(CCNC(c4cc(CC)on4)=O)CCCC3)=O)CCCC(C1)OC2 c1(NC(N2CCC(c3ccccc3Br)C2)=O)ccc2cc(CO)oc2c1 C(=O)(C(F)(F)C(C)(C)O)NCC1(C)CCCN(C(c2nccc(C(N)=O)c2)=O)C1 c1(CC)nnc(C)cc1NC(C1CC(n2cnnc2)C1)=O C1(CNC(C2CCCC(C)C2)=O)CCC(C)(C)CN1c1ncnc2[nH]cnc12 c1(C(N(C2CCN(C(CC(C)SC)=O)C2)CCO)=O)nccc2n[nH]cc12 c1(C(C)C)ccc(C(=O)NCCOCCCNC(C2CC(O)C(F)C2)=O)cn1 Cc1ccc(C(=O)NCC2(O)CCN(C(=O)C3=NOCC3)C2)nc1C Cc1cc(C(N2CCC(C(C)CNC(=O)C(N)=O)CC2)=O)oc1C CC1=C(C)CC(C(=O)NC2CC3CC2N(C(C2CC(Cl)(Cl)C2)=O)C3)CC1 C(=O)(C1=CC2(CN(C(C3CN(C(N)=O)C3)=O)C2)OC1)NC(C)(C)CCCO C(=O)(CS(=O)(=O)C1CC1)NC1(CC=C)CCN(C(=O)C=C(C)c2cccnc2)C1 N1(C(c2c(Cl)c(CC)n(C)n2)=O)CC2CCN(C(c3ccn(C)n3)=O)CCC2C1 C=Cc1cncc(C(=O)NCC(O)CCNC(=O)C(C)C(C)C)c1 Cc1nn(C)c(C)c1C(=O)C(=O)N(C1CC2(C1)CN(C(C1CCOC1CN)=O)C2)C c1(NC(c2n[nH]c3c2CN(Cc2csc(Br)n2)CC3)=O)cc(Cl)cnc1[N+](=O)[O-] C(=O)(C(O)CCC(C)C)NC(C(C)C)CCN(C)C(C1CCC(=O)N(C)C1)=O N1(C(c2c(SC)nn(C)c2)=O)CCCC12CCN(C(=O)C1=CC3CC=CCC13)C2 C1(CCC(=O)N(CCCNC(c2cnc(C(C)(C)C)s2)=O)C2CC2)CCCC(O)C1 S(=O)(=O)(CCC(=O)Nc1cccc(NCCSC(F)(F)F)c1)NC C(=O)(C1=CC2(CCOC2)C1)N(C)CC1(O)CN(C(C2C(C(=O)OC)C2)=O)C1 c1(CC)ccc(N)c(C(=O)NCCCCC(C)NC(c2cn(C)cn2)=O)c1 c1(OC)ccc(NCCC2CCCC23CC3)c2cnccc12 O=C(C1=CCC(NC(C2CCSC2)=O)C1)Nc1ccc(F)cc1 CC1(C)C(C)(C)C1(F)C(=O)NCC1CC(C(=O)N2CCC(F)(F)C2)=NO1 N1(C(CCOCCC)=O)CCCC(C2CN(C(C3(C4CC4)CCOC3)=O)C2)C1 C1(C(N2CCN(C(CCC=CC)=O)C(CC(F)F)C2)=O)CCCN(S(N)(=O)=O)C1 C=CCC(CC(F)F)NC(=O)CN(C(=O)C(C)C(F)F)C CCC(C)(C#N)C(=O)N1CCOC(CC(=O)N(C)CC2CCCS2)C1 c1(C(N(C)CC2(O)CN(C(CCCC(=O)N(C)C)=O)C2)=O)ccc2snnc2c1 C(=O)(C(C(C)(C)C)NC(N)=O)N1CCCC(C(=O)NC2N(C(C)C)CCCC2)C1 C(=O)(C1c2ccccc2C2CC1C2)N1CC(CN(C(CSC)=O)C)OCC1 C1(NC(=O)CCc2cncnc2)C2CCC(C2)C1C(=O)Nc1ccc(Cl)c(F)c1 N1(C(Cc2nc(COC)sc2)=O)CCCN(C(=O)CCC2CCCOC2)CC1 c1(C(N2C(CNC(C3C4CCCOC34)=O)CCCC2)=O)cc2n(c(=O)c1)CCS2 C1(F)(CNC(c2c(OC)cncn2)=O)CCCN(C(c2nccnc2C)=O)C1 CC1OCCN(C(=O)CCCn2cccc2)C1C(=O)NCCC(C)(C)O N1(C(c2sc(C)c(Br)c2)=O)CCN(C(=O)C=CC2CC2)C(CC(C)(C)C)C1 [N-]=[N+]=NC1CCN(C(=O)CC2CN(C(=O)CC3CCOC3=O)CCO2)CC1 c1(CNC(=O)CC2CN(C(C3CC4CCC4C3)=O)CC23CC3)cnc2ccccn12 CC1=C(C(=O)N2CCOC(C(C)NC(=O)COCc3cc(C)on3)C2)SCCO1 c1(C(N(C(CNC(C(CC)F)=O)C)C)=O)cccc(C(C)C)c1N N1(C2CCCN(C(C(C)N(C)C)=O)C2)CCN(C(C2(C)COC2)=O)CC1=O CCC(N=c1[nH]c(=NCC(F)(F)Cl)c2sccc2[nH]1)c1ccc(OC)cc1 c1(CC(=O)NC2CC(CNC(C3(COC)CCC3)=O)C2)nc2c([nH]1)CCCC2 C1(NC(C)=O)CCCC12CCN(C(c1cc(Cl)c(Cl)c([N+](=O)[O-])c1)=O)CC2 CCC(CC(C)C)C(=O)N(CCNC(c1ccnc(N2CCC(C)C2)c1)=O)CC c1(C(=O)NCCCN(C(C(CCC)CC)=O)C2CC2)ccc2nnc(O)n2c1 c1(CNC2C(C(=O)Oc3ccc(CC)cc3)C2)ccc(F)c(OC)c1.CC1CC1.CO CC(C)(C(=O)NCCCCNC(=O)Cc1nc2ncccn2n1)C1=CCSCC1 C1(CNC(CCCC#C)=O)(CO)CCN(C(=O)CCOC2CC2)CC1 C1(C)(C(=O)NCc2ncccc2C(=O)NCC2CC2)CCCC(F)(F)C1 c1(C(N(C2CCN(C(c3cc(SC)oc3C)=O)C2)C)=O)ccnc2[nH]c(C)nc12 C(CC(C)C(=O)NCC#CC(=O)NCC1COCCN1C)=CCC C1(C(=O)NCCNC(c2cc(NC)ccc2Cl)=O)COc2ccc(Cl)cc2O1 S(=O)(=O)(c1ccc2ccccc2c1)N(c1ccc(Br)cc1)CC(NOC(C)C)=O C1(NC(N2CC(CC(N)=O)C2)=O)CCCC(CC2CC2)C1 C(c1cccs1)=C(C)C(=O)NC1CCC(CNC(C2CC(=C3CC3)C2)=O)C1 N1(C(c2c(CC)onc2C)=O)CCC(O)C(NC(C2CC3C=CC2C3)=O)C1 c1(C(=O)NC2CCC(NC(c3n[nH]cc3Cl)=O)CC2)cc(C(F)(F)F)ccc1O c1(C(N2CCCC(CC=C)(NC(=O)C(F)OC)C2)=O)csc2ncnc(O)c12 N1(C(C=Cc2ccc(C)cc2Cl)=O)CCCC2C1CCN2C(=O)CS(C)(=O)=O CCCCCCCCCCS(=O)(=O)N1CC2CCCC2N1C(c1n[nH]cc1I)=O C#Cc1ccc(C(=O)NC2(C)CCN(C(C3CCN(C)C3C)=O)CC2)cc1F C(CCCC(=O)N1CCC1CCC(=O)N(C)Cc1ccc(F)cc1)NC(C)=O N1(C(C=CC)=O)CCC(NC(C2CC(CC3CC3)C2)=O)CC(O)C1 C1(C(=O)NCC(C)C)CC12CCN(C(=O)C(C)CC1CCC1)C2 CC1(C)COC(CN(c2cc(F)ccc2Oc2ccccc2)CCSCC(N)=O)CO1 CC1=C(C(=O)NC(C(=O)NC(CC2CCCC2)CO)C2CCC2)CCCO1 Cc1nn(C)c(Cl)c1C(=O)NC1CC12CC(NC(C1(C3CCCO3)CC1)=O)C2 c1(CCC)ncoc1C(=O)NC1COCC1NC(C1CC1c1ccsc1)=O C(CC(C(=O)NC1(CC(=O)NC(CO)C2CC2)CCCCC1)OC)OC c1(C(=O)NCC2CC(NC(COCCOCC#C)=O)C2)cc(CC#C)n(C)n1 C1(NC(C2CC(O)(C(F)F)C2)=O)CC(F)CN(C(c2ccccc2)=O)C1 c1(N(C)C(C2CCC(F)(F)C2)=O)cc(Cl)c(Br)cc1N C1(NC(=O)CC2CC2)CN(C(=O)CCc2ccc(F)cc2Cl)CCC12CCC2 c1(OC)cc(OC)c(S(=O)(=O)NC(c2ccc3nnnn3c2)=O)c(OC)c1 c1(C(=O)NCC(C)NC(c2cc(C)nn2C)=O)ccc2[nH]c(=N)oc2c1 N1(C(C2(C)CCCC2)=O)CC2CCCCC2(NC(=O)CCc2ccc[nH]2)C1 N1(C(CCNC(N)=O)=O)CCCC(O)(CNC(=O)C(O)C2CCC2)CC1 N1(C(C=CCCC(C)C)=O)CCN(C)CC1C(=O)NCC1CNC(=O)CO1 CCCCC(O)CNC(=O)CCCNC(c1c(C)noc1N)=O C1(C(N2C(COC)CCCC2)=O)CCCN(C(c2ccc(I)c(F)c2)=O)CC1 C(=O)(C(F)CC(C)C)N1CCC(OCCNC(CC(CC)SC)=O)CC1 CCC(F)(F)C(=O)N(C)CCN1CCN(C(C2CCC(F)(F)C2)=O)CC1 c1(OC)cccc(CC(=O)NC2COCCN(C(c3ncccc3O)=O)C2)c1C C12(CCC(=O)NC(C(=O)OC)(C)Cc3ccccc3)CCC(CC1)NC2 c1(C(N(CC(C)NC(c2cc(C)sc2)=O)C)=O)sc(-c2ccccc2F)nc1C N1(C(COCCCOC)=O)CC(CNC(c2csc(C(C)=O)c2)=O)OC(C)(C)C1 C1(C(=O)NCCCCCNC(Cc2cn(CC(C)C)nc2)=O)CCCC(O)C1 N1(C(c2c(C)nns2)=O)C(C)CC2CN(C(C3(C(F)F)CCCO3)=O)CC12 c1(OCc2nc(CCCC)on2)nc2cc3c(cc2[nH]1)OCO3 c1(C(N2CC(CCC)N(C(=O)CC3CCCCO3)CC2)=O)c(N)cc(Cl)cc1Cl Cc1nc(C)n(O)c1C(N1CCCC(F)(CNC(=O)C2=CCCOC2)C1)=O C#Cc1ccc(C(=O)N(CC(CC)NC(=O)CCNCC(CC)CC)CC)cc1C N1(C(c2cc(CC)nn2C)=O)CCN(C(=O)Nc2ccccc2)C2CC12.OCC C(C(C(=O)NC1CC(C)(C(=O)N(CCC(F)(F)F)CC)C1)N(C)C)OC c1(C(N2C(C(C)NC(c3ccc(CC)cc3)=O)CCC2)=O)cnc2nccn2c1 N1(C(c2on(C)c(=O)c2)=O)CC2CCC1C1CN(c3ncc(Br)c(O)n3)CC21 C1(C(=O)NC(c2ccccc2)CO)CCCCN1C(C1CC2CCC1O2)=O N1(C(C2CCCC(C)C2)=O)CCN(C(c2cnc(S)[nH]2)=O)C(CC(F)F)C1 C1(F)(C(N2CC(O)CC(NC(=O)CN3CCCOCC3)C2)=O)CCC(F)(F)CC1 c1(C(N2CCC(C(=O)NC(C(C)C)CO)C2)=O)ccc(I)c(F)c1F CC1CCN(C(c2cnc(C3CC3)nc2)=O)CC1NC(=O)C=CC=C(Cl)Cl c1(NCCc2ccc(OC)c(F)c2)ncccc1S(=O)(=O)NC1CCC(F)CC1 c1(OC)cccc2[nH]c(C(=O)NCCCN(C)C(C3(C)CC3F)=O)cc12 c1(NC(C(N2CC(C)SCC2)=O)=O)ccc(Oc2ccc(F)cc2)cc1F c1(C(N(CCCNC(=O)C2=NOCC2)CC)=O)cc2c(O)ncnc2cn1 C(CCC(CO)NC(c1cnc(CC2CC2)s1)=O)NC(C1(C)CCCC1)=O N1(C(C(C(C)C)C2CCC2)=O)Cc2n[nH]cc2C1C(=O)NC1CC(O)C1O c1(C(N2C(C(N3CC(C#N)(F)C3)=O)CCC2C2CC2)=O)ccc2cc[nH]c2c1 C#CC1(CN(C2CCCC2C#N)C)CCOCC1 N1(c2c([N+](=O)[O-])ccc(C)c2)CCC2(CC1)COC(CNC(c1ncc[nH]1)=O)C2 c1(C(N(C(C)C2CC2)CC)=O)ccnc(CNC(=O)CCC(=O)OC(C)=O)c1 c1(C(=O)NCCCCCN(C(C2CC2(C)C)=O)CC)ccn2cncc2c1 CC1(C(=O)NCCC2CCN(C(C3(CCF)CCOCC3)=O)C2)CC2CC2C1 c1(CC(N2CCC(NC(C(CCC)(C)C)=O)C(C)C2)=O)cn2c(n1)CCCC2 C1(C(C)C)C(C(=O)NCC(C)(C)C2CC2)CCN1C(=O)CCNC1CCC1 N1(c2nc(=NC)[nH]c(=NCC3CC4(CC4)C3)[nH]2)CCS(=O)(=O)N2CCCCCC12 CCC(CC)CC(C(=O)NCCCF)N(C)Cc1cnc(OC)cn1 CC(=NO)c1cc(C(N2CC(NC(C3CC34CC4)=O)CCC2C)=O)cnc1O c1(N2CC(NC(c3c(C)[nH]c(C(F)(F)F)c3)=O)C(C)CC2)ncnc2scnc12 Cc1nc2cc(C(=O)NC(C)(CNC(C34COCC3C4)=O)CO)ccc2s1 C(=O)(C(C#N)C(C)(C)C)OC(c1nnc(-c2nc(C)oc2C)n1C(C)(C)C)C CC1CCN(C(c2cccc(F)c2)=O)CCN1C(C1CN(C2COC2)C1)=O C(N=c1cc(NCC2(C)CSC2)nc(C)[nH]1)c1ccc(C)cc1C CC1CC=C(C(=O)N2CC3(CCC(CNC(=O)C(C)(C)CC4CC4)O3)C2)CC1 c1(C(N2C(CNC(Cc3c(C)cc(F)cc3)=O)CCC2)=O)[nH]cc2c1CCCC2 CCS(=O)(=O)c1ccc(-c2csc(C(N)=O)c2)cc1 C12(CNC(c3cncs3)=O)CN(C(c3cnc4scnc4c3)=O)CC1CCO2 C(=O)(CC(C)(C)NC(c1ncsc1C)=O)N(C1CCN(C(C)=O)C1)C c1(N(C(=O)NCCN(C(CC)C)C)C(C)C)cccc(C#N)c1 c1(C(=O)NCC2CCN(C(=O)C=C3CC3)C2)cc2c(cc1Cl)OCCO2 c1(C(N2CC3C(NC(c4c(C)nc(C)s4)=O)C3C2)=O)ccn2nnnc2c1 C1(F)(CNC(C2CC(F)(F)CS2)=O)CC2CCC(C1)N2C(c1ccccn1)=O c1(OC)cc2c(cc1OC)NC(C(=O)NCc1ccn3ccnc3c1)C2 C(=O)(CC(C)P(C)(C)=O)N(CCCCN(C(C=CC(CC)C)=O)C)C C1(O)(CNC(C(F)=CC)=O)CCN(C(c2cnoc2Cc2ccccc2)=O)CC1 C(=O)(CC(C)C(C)(C)NC(=O)CC1OCCO1)NCCC(C(C)C)N(C)C N1(C(Cc2nc(CC)sc2)=O)CCC2CCN(C(c3cnc(Cl)s3)=O)CC12 C1(C(N(CCNC(C2C=CCC2)=O)CC)=O)CN(C(C)=O)CCN1C C1(C(=O)NCCNC(c2ccsn2)=O)CC2CC12 c1(OC)cc(NC(=O)CCNC(c2ccco2)=O)cc(C)n1 CCC(C)(CO)C(=O)N1CCC1CNC(=O)C(C)c1cncs1 C(c1ccccc1CCC(C)O)=CCCOC.c1(OC)ccccc1C c1(C(N2CCC(C)(CNC(=O)CC3CC3)CC2)=O)cccc2c1C1CCC2CC1 C1(OC)CN(C(=O)C(C)CSC)CC1C(=O)NC(C1CCCCO1)(C)C CCC(F)(F)CC(=O)NCC1CCN(C(c2nc(C)ncc2Cl)=O)C1(C)C C1(NC(C(C)SCC)=O)CN(C(c2cccnc2C2CC2)=O)CC2(CCC2)C1 N1(C(c2c(CC)cno2)=O)CCC(C(N2CCCOCC2C)=O)C(O)C1 c1(C(=O)NC2CCCC(CNC(c3c(C)ncn3C)=O)C2)c(C)cc(=O)oc1C C(=O)(C1CCc2ccccc21)N1CCC(C(=O)NCCn2ccnn2)C12CCC2 c1(C(N2CC(CNC(C(F)=CC)=O)C2)=O)cnn(-c2ccccc2)c1I c1(CC(=O)Nc2cscc2C(=O)O)ccc(F)cc1F c1(C(=O)OCc2cc(C)c(F)cc2)cc(S(=O)(=O)NC2CC2)ccc1O c1(CC)ccc(Cl)c(C(=O)N(C(CNC(=O)CC2CNC(=O)C2)CC)C)c1 c1(CC)cc(C(=O)NC2CCCCC2NC(c2cc(OC)ccn2)=O)ccc1F CCCC(CNC(C1CCCCO1)=O)C(=O)NC1(C)CCCCCC1 CCN(OC)C(=O)C1=C(F)CN(C(c2cn(C)nc2OC)=O)CC1 S(=O)(=O)(c1ccc(Cl)cc1)N1C(CNC(=O)CN2C(=O)CSC2=S)CCC1 c1(CC(N2CC(O)(C(C)NC(C3CC4C=CC3O4)=O)C2)=O)nc(F)c(F)cc1F C(c1ccccc1)=CC(=O)NC(C1CN(C(=O)CN(C)C)CCO1)C.C(C)(C)(CC)O C1(n2cc(CC3CN(C(CC(C)O)=O)C3)nn2)CC2CCC1(C(=O)O)C2 CCN=C(NCc1ccc(C(N)=O)o1)N1Cc2ccc(F)cc2C(C)(C)C1 Cc1ccc(O)c(C(=O)NC(CCN(C)C(c2ccnc(F)c2)=O)C(C)C)c1 C1(C(N(CCNC(CCCCOCCC=C)=O)C)=O)CC(C)(C)CCO1 C1(NC(c2c(C)ccc(C)n2)=O)(CNC(c2cnsc2)=O)CCC(F)(F)CC1 c1(COC)cnc(=NCc2cccnc2NC(=O)Nc2ccc(OC)cc2)[nH]c1 c1(C(=O)NC(CNC(c2ccc(C)cc2)=O)C2CC2)c(Cl)ccc2c1OCO2 N1(C(=O)CSc2ncccn2)CCN(C(C2CCCN2C2CC2)=O)CC(O)C1 c1(N2CCN(C(COC)C)CC2)nc(=NCC2CCCC23CC3)[nH]c2c1CCC2 N12CCCC(C1C)NC(=O)C(C)c1ccc(o1)C2=O.C(=O)CCCCF c1(C(=O)NC2CCN(C(C34CC(O)C3C4)=O)C2)cc(CCCO)on1 C1(NC(C2=C(C)CCC2)=O)C(C)CN(C(=O)CCCNC(=O)C2CC2)CC1C N1(CC(C)C)CCC(C(=O)NCC#CC(=O)O)CC1 CCCCC(C)C(=O)NCC1CC(NC(c2cc(C)cc(F)c2)=O)C1 N1(C(c2scc(C(=O)OC)c2)=O)CCN(C)CC1CNC(=O)C(CO)N(C)C CS(C)(=O)=NC(=O)C(=O)NCC1CN(C(c2cncs2)=O)CC12CCC2 N1(C(CCCC#C)=O)CCC2(CC(NC(c3sccc3CC#C)=O)CO2)C1 C1(N(CCC)C)CCN(C(c2cnn(C)c2Br)C(=O)NC2CCOC2)CC1 C(CCC(=O)NCC1CCCN1C(=O)C(O)C1CCC1)=CC(C)C C1(CCOC)(NC(C2CCCCC2)=O)CCN(C(=O)Cc2occc2C)C1 C1(NC(C(C(C)(C)C)O)=O)CC1C1CCCN(C(c2cc3ncccc3[nH]2)=O)C1 C1(C(=O)NCC2(OC)CCCC2)CC2CC1CN(C(C13CCC(CC1F)C3)=O)C2 Cc1cc(F)c(N)cc1C(=O)NCC(O)CNC(c1cnc(C2CCCO2)s1)=O C1(C(=O)NCC)CN(S(=O)(=O)CC(C)(C)OC)CC1C1CC1 Cc1ccc(F)c(C(C(=O)NC2CCOC2)N(C)C(c2ccccc2Br)C)n1 C1(C(C)NC(C(C)NC(C)=O)=O)CCCN(C(=O)C(O)CCN(C)C)C1 C(=O)(C(F)CCCCC)NC(=O)NCc1nccc(C)c1F.C12CCN(C1=O)O2 CN1CCC(NC(N2CCC2C2CCC2)=O)C(C#N)C1 N1(CC(=O)N(C2CCN(C(c3c(C)onc3)=O)CC2)CCO)CC(=O)N(C)C1=O CC1CCN(C(=O)CC2CCNC23CCC3)CC1(C)C N1(C(N2c3cc(C)nn3CC2)=O)C(C)CC2CCCCC12 c1(C(=O)NC2C(CNC(c3[nH]cc(CC)c3)=O)CC2)ccc2ccc(O)nc2n1 CCCCC(C)C(=O)NC1CCN(C(C2CCOC(=O)N2)=O)C1 C(=O)(C(C(C)C)NC(=O)Cc1ccc(O)cn1)NCCCCCOC c1(CNC(=O)CC2CCCC2NC(C2(C3CC3)CC2)=O)nc(C2CC2)no1 c1(C(=O)Nc2cc(OC3CC(C(C)C)C3)cc(Cl)n2)c[nH]c2cccnc12 Cc1cn2c(n1)CC(C(N1CCOC(CN(C(=O)Cc3cc[nH]n3)C)C1)=O)CC2 C1(C(N2CCCC(NC(c3ccn(C(C)C)c3)=O)C2)=O)CNC(=O)CC12CCC2 N1(S(C)(=O)=O)CC2CC(NC(=O)CCNC3CC3)CC(C2)C1 c1(C(=O)NCC2C3CN(C(c4c(C#N)scc4)=O)CC32)nccc2cc[nH]c12 C12(C(=O)OC)CCCC1(C(=O)NC1CC(N(C(=O)CCC=CBr)C)C1)C2 C1(NC(c2c(C)coc2)=O)CCCCCN(C(c2[nH]c(O)nc2C)=O)C1 c12ncccc1S(=O)(=O)N(C)C1CCN2C1.C1(CSC)OCCCC1(C)C C1(NC(C(c2cccn2C)C)=O)CCOC1c1ccnn1C C1(C(N2C(C)(COC)CC2)=O)CC(F)(F)CN1C(C1CCSC1)=O c1(NC(C(C)N(CCC)C(C2CCCC2C#N)=O)=O)cccc(CCO)c1 c1(C(=O)NC2CC(N(C(CSCCC)=O)C)C2)ccc2c(c1)CCC(=O)N2C Cc1sc(C)c(C(=O)N(C)CCOCCNC(C2CCCCC2F)=O)c1C C1(C#N)(C(=O)NCCCN(C(CCCn2ncc(C)c2)=O)C)CC12CCCC2 c1(C(=O)NC2CC3CN(C(Cc4c(C)noc4)=O)C2C3)cc2cccc(Cl)c2o1 C(=O)(C(C(=O)OC)C(=O)CC)N(C(CCC)CC)c1ccccc1 C(C1=NOC2CN(C(=O)Cc3ccc(CC)cc3)CC12)NC(CCC=CC)=O C1(OC)CC2CC(C1)N(C(=O)CCCN(C)C(C1CC(C(C)C)C1)=O)C2 C=CCCC(CC(C)C)C(=O)N1CC2CCC1CN2C(C1(C)COCCO1)=O C1(C(N(CC)CC2CC2)=O)CCCCN1C(C1CC(O)CN1C)=O CC1(CNC(c2sccc2Cl)=O)CC(NC(C2CC2CF)=O)C1 CC1CC(CC(=O)NCC=Cc2cccnc2)CN1C(=O)Cc1nc[nH]n1 N#CC1(CC(=O)NCC2(NC(=O)Cn3nnnc3C3CC3)CCC2)CCOCC1 N1(C(CNC(C2CCCN(C(CC)=O)CC2)=O)C(=O)NC)CCN(C)C(=O)C1C N1(C(C2C=CC(NC(c3cc(Cl)ncc3Br)=O)C2)=O)CCc2c(O)noc2C1 C1(C(=O)NC2(CNC(C(C)(C)N3CCOCC3)=O)CCCC2)CC2CCC(C1)O2 c1(C(=O)O)ccnc(COC(=O)C(CC2CCOCC2)SC(F)(F)F)c1 C1(OC)(OC)CC(NC(N2CC(C(C)(C)CF)C2)=O)C1 CC1(C)CC(NC(c2ccc(C(C)(C)C)nc2)=O)CCN(C(C23CCC2C3)=O)C1 c1(C(=O)NC2CN(C(C3CCC(C)(CC)O3)=O)C2)ccc(Cl)nc1O CC1CCCC(C)N1CCC(N1CC(O)(CCNC(=O)CSC(F)(F)F)C1)=O N1(C(c2cc(COC)on2)=O)CCN(C(c2cccc(C(N)=O)c2N)=O)C(C)C1 N1(CC(=O)NC(CN(C(C2C(C(=O)OC)CCCC2)=O)C)C)CCCCCC1=O N1(C(c2cc(C)[nH]n2)=O)CCCC12CCN(C(c1ccc(B(O)O)cc1)=O)CC2 N(C)(C1CCc2ccc(Br)cc21)C(C(=O)NCCCC)C(C)CCC C(=O)(C=NOC)N(C1CCN(c2nnc(C(N)=O)s2)C1)CCC CC1CN(C(C2(C(F)F)CCC2)=O)CC1CCNC(=O)Cn1ncnn1 C=CC1(C2(C(=O)NCCCCNC(=O)CN3CC4C=CC3C4)CCC2)CCC1 c1(C(N2CCC3C(NC(CC(C)(C)OC)=O)C32)=O)ccc(C(C)C)c(Br)c1 C(CC(=C)C)(C(=O)Nc1ccc(O)cc1)NC(COCCC=C)=O n1(CCC(N2CCC(C)(NC(c3ccsn3)=O)C2)=O)ccc(O)nc1=O CC1CN(C(=O)CNC=O)CC1CCNC(=O)CCCC1CC1 C1(NC(c2cc(F)c(F)c(F)c2Br)=O)CN(C(=O)C(F)(F)F)CC12CCOCC2 C(=O)(C1=C(C)OCCC1)N1C(CCC(=O)NC2CCCC2N=[N+]=[N-])CCCC1 N1(C(C2C(CC)N(C)CC2)=O)CCC(NC(c2ccnc(SCC)c2)=O)C1(C)C N1(C(C=C(C)C)=O)CC2CC1C2CNC(c1ccc(C2CCCOC2)cc1)=O C1(C(=O)NCC#CCNC(C(c2ccccc2)N(C)CC)=O)CCN(C(C)C)C1 c1(NC(=O)NC(c2n[nH]c(CC3CC3)n2)C)cccc(-n2cnnc2)c1 c1(OC)ccnc(N(C)CCN(C(=O)CC(C)SC)C(C)C)n1.C1CC1 c1(C(=O)NCC2(OC)CCN(C(C3CCCS3)=O)CC2)ccc2nc(C)[nH]c2c1 c1(C(N(C2CCCN(C(C3(OC)CCC3)=O)C2)C)=O)ccc(C#CC2CC2)cc1 C1(C(=O)NC(C(CC)NC(c2cccn3ccnc23)=O)C)CCC([N+](=O)[O-])CC1 C1(NC(c2cc(C(=O)OC)no2)=O)CC(NC(C2CCC(O)C2)=O)C12CCC2 N#Cc1ccc(C(N2CCCC(CNC(C3CCCC3O)=O)CC2)=O)cc1O C(C1=NOC2CCCC12)NC(C1(C2N(C(CN=[N+]=[N-])=O)CCC2)CC1)=O c1(OCCCC)cc(-c2c[nH]nc2C(=O)NCC(=O)NCC)ccc1F c1(C(=O)NCC(CCNC(C(CC(=C)C)C)=O)=C)cn2c(n1)CC(OC)CC2 C1(NC(C2CC(F)C(=O)N2)=O)CC2CCC(C1)N2C(c1cc(Cl)c[nH]1)=O N1(C(C(N2CCCCC2=O)C)=O)CCCN(C(c2ccc(Cl)nc2)=O)C(C)C1 CCCC(CC)C(=O)N1CCC(C(=O)NCCC(C)(C)N(C)C)C1 c1(C(N2CC(CC(C)NC(C(CSC)O)=O)C2)=O)cccn2nccc12 c1(C(N2C(CNC(C3=C(C)CCC3)=O)CC(F)C2)=O)ccc2c(n1)COCC2 N1(C(c2cc(C(N)=O)c[nH]2)=O)CCC(F)C(NC(=O)C(c2ccc(Cl)cc2)O)C1 O=C(CCCN=c1ncc(I)c[nH]1)N1CCN(CC2CCOC2)CC1 C(CCC1CC1)(C(=O)N1CC(c2cscn2)C1)NC(C(C)SC(C)C)=O c1(SC)cc(C(=O)NCC2(C(F)(F)F)CC2)c(Cl)cc1Cl.c12cc(ccc1O)SC2 c1(N(C(C)C)C(C2CCC2C)=O)cn2cc[nH]c(=O)c2n1 C1(NC(C2C(C)=C2)=O)CCN(C(c2c[nH]nc2C2CC2)=O)CC1C c1(CC(=O)NC2CCC(N(C(C=CSC)=O)C)C2)cn(C)c(=O)c2ccccc12 C1(CNC(c2c(C)cc(C(F)(F)F)s2)=O)CC2CCC1N(C(C1CC(=O)N1)=O)C2 O=C(CCCCc1cnn[nH]1)NC1CCN(C(=O)CSC2CCCC2O)CC1 CCCN=C(NCC1CCN(S(C)(=O)=O)CC1)N1CCC2CCCCC2C1 c1(C(N2C3C(NC(COC(CC)C)=O)C(CC3)C2)=O)ncc2n1CCCC2 N1(C(C#CC(C)(C)C)=O)CCC(CNC(c2ccc(Cl)s2)=O)C(F)(F)C1 C1(NC(c2nc(C)on2)c2ccccc2)CC2CCC1CN2C(=O)C(C)CCO CN1CCC(=CC(=O)NC2CC2CNC(C2CC2c2ccccc2)=O)C1 C(=O)(C(F)(CNC(=O)CC1CC=CC1)C(C)C)NCCn1c(C)ncc1 N1(C(c2c(C)sc(Cl)n2)=O)CCC(C2CC2)(CNC(C2CCCC2C)=O)C1 c1(C(=O)NCC(CC)NC(C2(CC=C)COC2)=O)cc(F)c2ncccc2c1 CCCCC(F)(F)C(=O)NC(CNC(c1cccc(C2CC2)n1)=O)CC(C)C c1(C(N(C2CC(c3ccc(F)cc3)C2)C)=O)cc(F)ccc1Cl C(=O)(C1COc2ccc(Cl)cc21)C12CC(c3c(=NC(CSC)=O)[nH][nH]c3)(C1)C2 c1(-c2scc(CC)n2)cccc(NC(=O)C(CC2CCCCC2)OC)c1 Cn1[nH]c(=N)cc1C(=O)NCC1CCC(NC(c2cccc(C(N)=O)c2)=O)C1 O(N=c1ncn(-c2ccccc2C(F)(F)F)[nH]1)CC(F)(F)Cl N1(C(C2C(NC(C(C(CC)C)N(C)C)=O)CCCC2)=O)CCCC2(C=CCO2)C1 N1(C(c2c(CNC(CC(CC)C3CC3)=O)noc2)=O)CCCC(O)(CO)C1 N1(C(C(c2cn(C)nn2)N(C)C)=O)CCC(CC(=O)NCCC2CCCN2C)C1 c1(OC)cc(OC)cc(N2CCN(CC(O)CO)CC2)c1.C1(=O)C(C)CN1 C1(NC(=O)COCC2CC2)CCOC(CNC(c2cccc(CCF)c2)=O)C1 C(=O)(C(F)C(C)CNC(=O)Cn1cccnc1=O)NC1(CCOC)CCC1 NS(=O)(=O)c1ccc(C=CC(N2CCCN(C(=O)CO)C(CO)C2)=O)cc1 N1(C(c2c(CCC)n[nH]c2)=O)CC(NC(C2COC2)=O)C(C2CC2)C1 C1(NC(=O)OC(C)(C)C)CCCC(C(=O)NCC2CCCCC2O)C1 N1(C(Cc2ccc(OC)cc2)=O)CC2CN(C(c3cc(C)n(C)n3)=O)CCC12 c1(OC)ccc(N2CCC(NC(c3cncc(C)n3)=O)C2)cc1 CC1CN(C(c2ccc(N)c(Cl)n2)=O)CCN1C(=O)CCc1cc(F)ccc1F C1(C(=O)NC(C)CN(C)C(C2SCCCS2)=O)COC2(CCC2)CO1 CCCC(CCC)C(=O)N1CCCC(N(C(c2cc(CSCOC)on2)=O)CC)C1 C1(C(N2CC(C)(NC(=O)C(F)C3CCC3)C2)=O)CCc2nnc(O)cc2C1 c1(C(=O)NC(C)CN(C(=O)Cc2cc(C3CC3)on2)C)cc2ccoc2cc1F N1(c2n3c(nn2)C2CC2C3)CCC2(CCC2)C1.c1(COCCOC)ccccc1 c1(CC(=O)NC2C(Nc3snc(C)n3)CCC2)ccc(OC(F)F)cn1 N1(C(c2n(C)c(S)nc2)=O)CC2CCC1CN2C(C1CC=CCO1)=O c1(C2C(C(N3CCOCC3)C(=O)NCC3CCOC3)C2)cccc(O)c1 C1(CC)C(C(=O)Nc2cccc(C)c2)CCN1C(=O)Nc1cncc(C)n1 C(C)(CNC(c1cccnc1S)=O)(C(C)C)NC(C(CSC)OC)=O C1(C(N2C(C(N(C(CO)C3CC3)C)=O)C=CC2)=O)CC2C=CC1CC2 N1(C(c2cn(C)nn2)=O)CCCCC1CNC(c1nnc(C(C)(C)C)s1)=O C1(C(=O)NC2CC(F)(CNC(CCC)=O)C2)CC2CCC1CC21OCCO1 C(=O)(CCCCC#N)N1CCCC(NC(C(c2ccc(C)cc2)C)=O)C1 C1(CCNC(c2ncn(C(C)(C)C)n2)=O)CN(C(C2CC2(F)F)=O)CCS1(=O)=O c1(CNC(C(=O)N(C(CC)CO)Cc2ccccc2)=O)ccccc1C Cc1ccc2cc(C(=O)NC(CNC(c3ccns3)=O)C(C)C)[nH]c2c1 CCCCCCC(C)C(=O)NCC1CCCN1C(=O)CC1CCC(F)(F)C1 c1(C(N(CC(C)N(C(=O)C=C(F)c2ccccc2)C)C)=O)ccn(C)c(=O)c1 c1(CC)cccc2ccc(C(=O)NC(C)CCNC(c3ncccc3F)=O)nc12 Cc1ccc(C(N2CC(NC(=O)CCc3ccc(C)nc3)CCC2C)=O)c(O)n1 N1(C(c2nc(C)oc2)=O)CCN(C(=O)CNC(=O)NC(c2ccco2)C)C2CC12 CC1CN(C(c2cccc(Cl)c2N)=O)CCC1CNC(=O)C#CC1CC1 C1(C)(C(N2CCC(C#C)C2)=O)CN(C(c2cc(OCC)no2)=O)C(C)(C)C1 CC(C)C(N)CCOC(c1cc(-c2ccco2)on1)=O c1(C(CNC(C(C)NC(=O)NC)=O)NC(=O)CN2CCC2C)ccccc1F C#CCC(C)(C)C(=O)N1CCC(N(C(=O)C(c2cnccn2)C)CC)CC1 C1(CC)CCCC1(C)C(=O)Nc1ccc(CN(C)C(=O)OC(C)(C)C)cc1 CC(C)C(CNC(=O)C(C)n1cccn1)NC(c1cnc(C(C)(C)C)s1)=O c1(N(C2CCC(F)(F)C2)C(C(C)NC2CCNC2)=O)nc(Cl)c2c(ccn2C)n1 c1(C(C)=O)ccc(C(=O)NC(C)C(C2CCCCC2)O)cc1F c1(CNC(C2(S(N)(=O)=O)CC2)=O)cc2n(n1)CCN(C(=O)C1=NOCC1)C2 N1(C(CCSCCC)=O)CCC2CCN(C(=O)CCc3cnn(C)c3C)C2C1 N1(C(C(CC)C)=O)CCC2(CC1)CN(C(=O)C(C)n1cccn1)C2 c1(OC)cc(C(N2CC(n3cc(-c4cscn4)nn3)C(C)C2)=O)ccc1Br N1(C(C2(CNC(c3noc(CC)c3C)=O)CCC2)=O)CCn2ncnc2C1 N1(c2ncc(C)cn2)CCC(O)(CCNC(c2ccc3c(c2)CC3)=O)CC1 C(=O)(CCC(=O)NN(C)C)NC1CN(C(C(C)(C)OC(C)C)=O)CC1CC1CC1 c1(C(N(C)CC2(CNC(C3(C)CC3(Cl)Cl)=O)CC2)=O)cccc([N+](=O)[O-])c1F N1(C(c2c(C)cccn2)=O)CC(NC(=O)COCC(C)C)C(C2CC2)C1 C1(C(=O)NC(C2(O)CN(C(c3ccc(C)nc3O)=O)C2)C)CCn2nnnc2C1 c1(C(C)C)nc2c(F)cccc2c(=NCC23CCCCC2CN(CCC#N)C3)[nH]1 N1(C(CNS(=O)(=O)NCC(F)(F)F)=O)CCC(NC(c2cc(C)ns2)=O)C(C)C1 c1(C(=O)NCC2N(C(C(C)N(C)C)=O)CCC2)cnnc(C(F)F)c1 N1(C(C(CC)Br)=O)C2CCC1CN(C(c1cc(C)[nH]n1)=O)CC2 CC1(C#N)CCN(C(C2(N=[N+]=[N-])CCN(C(=O)CCCC(F)(F)F)C2)=O)C1 N1(C(C(CO)N(C)C)=O)CCN(C(c2ccc(F)c(O)c2)=O)CC1C1CCC1 N1(C(c2cc(CC)oc2C)=O)CCC(NC(C23CC(CC(F)F)(C2)C3)=O)C(C)C1 c1(-c2cn(CCC(=O)NCCSC3(O)CCOCC3)nn2)cccc(F)c1Cl Cc1nn(C)c2c(Nc3nc(CC4CC4)n[nH]3)nc(=NC(C)c3cnsc3)[nH]c12 c1(C(N2CCOCC2c2cn(C3CCC(F)(F)CO3)nn2)=O)cc2n(n1)CC(F)C2 c1(CCC)ccc(C(=O)NC(C)(C)C(=O)OC(CC2CC2)C(=O)OC)cc1 CCCC(C)(CC)C(=O)N1CC(NC(C23CC(C2)N(C(C)=O)C3)=O)C(SC)C1 C1(C(N2CCC(C)(CNC(c3c(F)ccnc3Cl)=O)C2)=O)CC2CCCCN2C1 N1(C(C2(c3cc(C)no3)CC2)=O)CCOCC1CNC(C1CCC=CCC1)=O C=CC1(CC(=O)N(CC(=O)NCc2cccc(C)c2)C)CN(C(=O)OC)C1 Cn1cc(S(N)(=O)=O)cc1C(=O)NC1CCSC12CN(C(=O)C(F)CC1CC1)C2 CC1CN(C(=O)C(=O)Nc2cnc(C3CC3)nc2)CC1CNC(=O)C1CC1 O=C(CCn1cc(CC(C(=O)O)C2CC2)nn1)NO.O1CP(=O)(O)OCCOCC1 C(=O)(CC1=NN(C)C(=O)C1)N1CCCC(CC(N2CC(C)OCC2C)=O)C1 C1(CC)CCN(C(=O)CCc2ccn(C)c2)C1C(=O)NC(C)(C)CC c1(C(N2CC(NC(C3(C)C=CCC3)=O)C(O)C2)=O)cccc2[nH]nc(O)c12 C12(CNC(C(=O)NC(C)C)=O)CCCCC1N(C(C13CCC1C3)=O)CC2 c1(CNC(C2C=CCN2C(=O)Cc2ccon2)=O)ncccc1F c1(C(N(CCCCNC(C2(F)C(C)OCC2)=O)C)=O)c(Cl)ccc(F)c1F C12(CNC(=O)Cc3csc(Cl)c3)CCC(CN(C(C3CC4(C3)CC4(F)F)=O)C1)C2 N1(C(C(C)N(C(C)=O)C)=O)CCC(C)CC1CC(=O)Nc1cccc(CO)c1 N1(C(C)C)N=C(C(=O)N2CCC(O)(CNC(C3CC3F)=O)CC2)CCC1=O c1(C(=O)NCC2N(C(C(CC)OC)=O)CC2)ccc(C(C)=O)cc1 c1(C(=O)NCCCC2N(C(C(C)C3CCC3)=O)CCCC2)cc(O)c(F)cc1N Cc1ccc(C(=O)NCCN(C(=O)CCn2cc(Cl)cn2)CC(C)O)s1 C1(CCNC(C(c2cncn2C)N(C)C)=O)COCCN1C(=O)Cc1cc[nH]n1 C1(C(N2CCC(CC(C)(C)CO)C2)=O)C2CC(F)C1N(C(=O)OC(C)(C)C)C2 C#CC1(C(=O)NCC2CSCCO2)CCN(C(=O)CCC(=O)CC)C1 CC1=NS(=O)(=O)N(C)C=C1C(=O)NC1CN(C(c2ocnc2C)=O)C2CC12 C1(C(N2CCCC(NC(C34C(C(N)=O)(CCC3)C4)=O)C2)=O)C2CC3C(C2=O)C13 Cc1cccc([N+](=O)[O-])c1C(N1CCC(C2CCCN2C(=O)C(=O)N(C)C)C1)=O c1(-c2cn(CC(CC)O)nn2)ccc2c(c1)N(C(=O)CCNC(=O)C1CC1)CC2 Cc1[nH]cc(C(N2CCC(NC(c3c(F)cccc3F)=O)CC2C)=O)c(=O)c1Cl c1(CC)nn(C)cc1C(N1CC(OC)C(NC(c2ccccc2NC)=O)C1)=O c1(CC(=O)NCC2CC(CO)N(C(=O)CCOC3CCC3)C2)cnccc1Cl C1(C(=O)NCC(C(C)C)NC(=O)CCc2ccc(C3CC3C)o2)CCC(C)(F)CC1 CC1CCC(C)(C(=O)NCC(C)NC(=O)C(C)(C)c2cscn2)C1 C1(Nc2nc(C)nc(C#N)c2)CC2CCCC(C1)N2C(=O)C(F)(F)C(O)C1CC1 C12(CNC(=O)C3=CCCSC3)CCC(CN(C(c3ccc(Cl)s3)=O)C1)C2 N1(C(c2cc(OC)c(C)nc2)=O)CC2CC(C)N(C(=O)CC3CCC3(C)C)C2C1 N1(C(C(C)N(C)C)=O)CCC2(CC1)CC(C)N(C(c1cc3n(c1)CCSC3)=O)C2 c1(C(=O)NC2CCCN(C(C3NC(=O)OCC3)=O)CC2)cc2cc(Cl)ccn2n1 N1(C(C2CCCN(CC)C2)=O)CCC(NC(c2cnccc2C)=O)CC(O)C1 c1(C(=O)NCC(CC)NC(CCNC(=O)OCC)=O)[nH]c(=N)ccc1C c1(C(N2C(C(=O)N(C)CCOCC)CC(=C)C2)=O)c(C)cc(O)cc1C C(C(COC)CC(=O)NCC(C)(F)CNC(=O)Cc1cc(C)cc(C)c1)OC C1(C(=O)NOCCc2cn(CCc3ccccc3)nn2)CCn2c(O)nnc2C1 c1(C(=O)NCCN(C(=O)CCC2CCC2)CC)ccc(C(N)=O)nc1 C1(C(=O)NCC(C)(CO)NC(c2cc(Cl)ccc2F)=O)CCCCC12CCC2 N1(C(C2(C#C)CCN(C(=O)CC3CCCC3)C2)=O)CC(C2CCCCC2)C1 CON=CC(=O)NC1CC1CNC(=O)C=Cc1cocn1 c1(CNC(C(C)C2CCCO2)=O)c[nH]nc1C(=O)N(C)Cc1nncn1C C1(NC(CCCC#C)=O)CN(C(=O)CCCCC)CCC12CCC2 C1(O)(CNC(C2C(CC)C2)=O)CCCN(C(C)=O)C1 C=C(C)C(C)(C)C(=O)N1CCC(NC(=O)Cc2cc(F)ccc2C)C(CO)C1 C1(C)(C(=O)NCC2CC(NC(C(C)Cc3cnn(C)c3)=O)C2)CCCNS1(=O)=O c1(CC(=O)NCC(C)(C2CCC2)NC(=O)C(F)F)ccnc(O)c1Br N1(C(C2(c3ccc(Cl)cc3)CC2)=O)CC2CN(Cc3ncc(Cl)cc3F)C2C1 c1(CC)cc(NC(=O)C2=NOC(CNC(=O)C(CC)CCOC)C2)cc(O)c1 CC1CCCC(CC(=O)NC2CC(CC(=O)Nc3cccc(Cl)c3)C2)C1 C(CCC(C)C)(C(=O)NC(c1cn(C(C)(C)C)nn1)C1CCCO1)OC N1(C(CCCC#C)=O)CCCOC(CNC(c2cn(CC)cn2)=O)C1 C(=O)(C(C)(C)CCOC)N1CCC(CNC(c2ccnc(OC)n2)=O)(OC)C1 Cc1nc(CC(N2CC3C(N(C(=O)C(C4CCCCC4)F)C)C3C2)=O)c(Cl)s1 C1(NC(CCCCCCC)=O)CCC12CCN(C(C1(C)CC(=O)N(C)C1)=O)CC2 C(=O)(CCC[N+](=O)[O-])N(C)CC1(O)CN(C(CCC=CCC=C)=O)C1 N1(C(C(F)OC)=O)CCc2ccccc2C1CNC(c1occc1C1CC1)=O C1(C(N2C(CNC(C(C)(C)O)=O)CC(F)C2)=O)CC2OC1C1CC21 CC1(C)CCCN(C(c2cnn3ncccc23)=O)C1CNC(=O)CSC(F)(F)F c1(C(=O)NC(C(C)NC(C2(COC)CC2)=O)C)ccc(S(=O)(=O)C(F)F)cc1 Cc1ncsc1C(=O)NCC1CCC1C(=O)N(C1CC1)Cc1ccoc1C c1(NC(CCCCC=C)=O)ccc2nc(NC(=O)CC(=O)OC)sc2c1 C1(NC(C2(CC)CNC(=O)C2)=O)CN(C(c2csnc2C)=O)C2(CCC2)C1 C1(CN(C(C(N2CCN(C)CC2)C)=O)C)CN(C(=O)Cc2ccncc2)CCO1 N1(C(C23CC(COC)(OC2)C3)=O)CCOCC(CNC(=O)CC2C=CCC2)C1 N1(C(c2c(C)cc(I)cc2)=O)CCC2CN(C(c3cc([N+](=O)[O-])cs3)=O)CC2C1 C(=O)(C1CCC(=O)c2cccn21)NC1C(CNC(c2c(SC)cccc2)=O)CC1 c1(C(C)=O)cccc(C(=O)NCC=CCNC(C2CCCCO2)=O)c1 N1(C(C2N(CCC)CCC2)=O)CC2CCN(C(=O)C(C)(C)CC(C)C)CC2C1 N1(C(C(CC)SC)=O)CC2CC(O)C1C2NC(=O)Cc1ccco1 CC1COCCCN1C(C1(NC(C2CCCCC2O)=O)CCN(C)C1)=O N1(C(C2CC(C(C)C)C2)=O)CC2(CCC(CNC(C3CC3C3CC3C)=O)O2)C1 c1(CC)cncc(C(N2CCC(F)(CNC(C3(CN(C)C)CC3)=O)C2)=O)c1 c1(C(=O)NC(CNC(=O)C=C2CCCC2)CO)c(Cl)oc2ccccc12 CC(C)(C(=O)NCCCN)C(N)=O.c1(C=O)ccc(-n2cc(C3CC3)nn2)cn1 c1(NC(=O)NC2C(C(=O)OC)C2C2CCC(CC)C2)cccc(SC)c1 N1(C(CNC(=O)OC)=O)CCC(NC(c2cc(C)n(C3CC3)c2C)=O)CC1C1CC1 C1(NC(c2cc(C(C)=O)on2)=O)C2CCC(C2)C1C(N1CCC(C)C1(C)C)=O N1(C(CN(C)CC)=O)CCC2(CCOCC2)C(NC(=O)C(=Cc2c[nH]cn2)F)C1 Cc1c(C(N2CC(O)(C(C)(C)CNC(=O)C=Cc3ccco3)C2)=O)cccc1N c1(C(=O)NC2CC3(C(NC(C(C)OCCCC)=O)C3)C2)cc2c(s1)CCOC2 c1(C(=O)NCC2(CNC(c3cncn3C(F)(F)F)=O)CC2)cc(Cl)c[nH]1 C(C(C)C(C)C(=O)NC1CN(C(=O)C(C)(C)C(C)C)CC1O)OC Cc1ccc(-c2ccc(C(=O)OCC(=O)NC(N)=O)s2)cc1 C=CCC(F)(F)C(=O)N1CCN(C(C2(c3ccncc3)CC2)=O)C(COC)C1 Cc1ccc(CN2CCCC2C(C)(C)C(=O)NCCNC(=O)C(C)C)s1 C1(NC(C=CC)=O)CCCCC12CCN(C(c1nccc3n[nH]cc13)=O)C2 N1(CC)N=C(C(=O)N2CCC(CN(c3nccc(C)n3)C)CC2)CCC1=O C(C(=O)N1CC(NC(C2CN(C3COC3)C2)=O)C(C(F)F)C1)(C(C)O)NC(C)=O c1(C(=O)NC(C)CC2CN(C(=O)C=CCO)C2)ccc2c(c1)COC2 c1(C(=O)NCCCCN(C(=O)Cn2nccn2)C)cn(CC2CC=CCC2)nn1 C(=O)(CN=c1cc[nH]cc1)NC1(C(=O)NCC2CCC(C)C2)CSC1 C#Cc1ccc(C(N2CCC(CCC)(NC(=O)CC(=O)OCC)CC2)=O)c(F)c1 C1(F)(C(=O)NCC2(NC(c3c(OC)ncc(Cl)c3)=O)CCC2)C2CCCCC12 C1(NC(C=NOC)=O)CN(C(=O)C(C)(C)CC(F)F)CC12CCOCC2 CCC(C)(CNC(c1cc(C)nn1C)=O)C(=O)N(C1CCOC(C)(C)C1)C N1(C(C2CC(C#N)(OC)C2)=O)CCC(C)CC1C(=O)NCc1csnc1OC c1(CCC(=O)NCC2CC(F)CN2C(=O)CCOC2CC2)cc(F)cc(F)c1 Cc1cc(C)c([N+](=O)[O-])c(C)c1C(N1CCC2(CC1)CN(C(=O)C(C)C#N)C2)=O Cc1cccn2cc(C(=O)NCC3CC3CNC(=O)C(=O)Nc3ncc[nH]3)nc12 c1(C(N2CCC(CNC(C3C4CC5C(C4)C35)=O)(CO)C2)=O)ccc2cccnn12 c1(CNC(c2nc(CNC(c3cc(CCC)[nH]n3)=O)oc2)=O)ccc(C)c(F)c1 C1(NC(=O)CC2CSCCS2)CCS(=O)(=O)C12CN(C(=O)C=C1CCCC1)C2 N1(C(c2cc(C)c(C)nc2O)=O)CCC2(CC1)OCCCC2NC(=O)C=C(Cl)Cl CC(N=c1nc2scnc2c(NC2(C(N)=O)CC2)[nH]1)c1ccc(S(N)(=O)=O)cc1 c1(OCCC(=O)NCCC(C(C)C)NC(C(C)SCC)=O)cccc(CC)c1 c1(C(=O)NCC(CC)NC(C2CNC(=O)C2)=O)ccc(-c2ccccc2)n1C C12(C(=O)OC)CC3CC(C)C(=O)N(C(=O)Nc4nc[nH]c4Br)C3(C1)C2 Cc1cc(CC(=O)NCCCC2CN(C(=O)C(O)C3CCC3)CCO2)c(C)s1 CC(=O)C(C)CC(C)C(=O)NCC1(O)CC(C(=O)N(CC(C)C(C)C)C)C1 c1(C(=O)NC(CC(=O)NCCC)Cc2cccs2)ccc(Br)c(Cl)c1F C1(NCC(Cn2cc(CCOC)nn2)(F)F)CC(NC(=O)CSC)C12CCC2 C(=O)(CCNC(=O)C=CCCOC)NCCOCCC#C C1(C(=O)NCC(C2CCC2)OC)CNC(=O)CN1C(=O)Cc1cnn(C(C)C)c1 CC1CN(C(=O)CCCN(C)C)CC1NC(C1(Br)CC1(C)C)=O C1(C(N(CCCC)Cc2cccc(F)c2)=O)CC2(CCC(F)(F)CC2)C1 N1(C(c2cc(CC)n(C)n2)=O)CC2COCC(C1)C2NC(c1cocn1)=O C=CCC(CC(C)C)C(=O)N1CCN(C(c2ccn(CCO)c2C)=O)C(CC)C1 C1(NC(C(C)c2ccco2)=O)CN(C(C2CC3(CSC3)C2)=O)CCC1(C)C c1(C(=O)NCCCc2cocn2)ccc2c(c1)CCCO2 N1(C(CCOCC#C)=O)CC(C(N2CCn3nccc3C2)=O)CC(F)(F)C1 N1(C(C(C)P(C)(C)=O)=O)CCC2(CC1)CC2NC(=O)CCCC(=O)N(C)C C(=O)(C#CC1CCC1)NCCN(C1CCCCC1)C(c1ccn(CC)n1)=O c1(C(=O)NCC(C)N(C(C2CCC(=C)CC2)=O)C)cc(Br)c(C)cc1OC c1(CC#N)ccc(C(=O)NCCC2CN(C(C3(C#N)CC3(C)C)=O)CCO2)cc1 C1(=CC(=O)NCCC(C(C)C)NC(=O)C2=NNC(=O)C2)CCCCC1(C)C C1(C)(CNC(c2c(C)onc2CO)=O)CN(C(=O)C(C)n2ccnc2)CC1C Cn1c([N+](=O)[O-])cnc1C(=O)NC1COCC1NC(=O)CCC(=O)c1ccc[nH]1 C1(C2CCN(C(=O)C(C)CCO)C2)(NC(C2CCN(C(C)C)CC2)=O)CC1 CC1CN(C(=O)C(C)(C)C2CC2)CCC1CNC(=O)COc1ccc(F)cc1O c1(Cc2cccc(C(Cc3n(CC)cnn3)=O)c2)ccc(F)cc1Cl C1(NC(c2cccc(CC)c2)=O)CC=C(C(=O)NC2CC(O)C2OC)C1 N1(C(c2c(C)n(CC(F)F)nc2)=O)CC2(CCN2C(C2OCCOC2(C)C)=O)C1 C(=O)(C1CCCc2occc21)N1C(C)(CNC(C2(CCCC)CC2)=O)CCC1 CCCC(C(O)C(=O)NC(C)C(N)=O)NC(=O)CCC(C)N(C)C c1(C(=O)NCC(CC)NC(C2CCC(SCC)CC2)=O)cn2c(C)cccc2n1 c1(OC)ccc(Cc2nc(C3CCC(F)(F)C3)n(C3CC(OC)C3)n2)cc1OC CCS(=O)(=O)CCC(N)C(=O)Nc1nc(C#N)c(C)n1-c1ccccc1 C=CCC(C(=O)NC1CC(CCNC(C2CCOC(=O)CC2)=O)C1)C(C)C C1(NC(COCc2onc(CC)n2)=O)CCN(C(C2CCC3CC3C2)=O)C(C)C1 c1(C(N2CC(F)(CNC(C3CC3F)=O)C2)=O)cc2n(n1)CCOC2 CCC1=C(C(=O)N2CCCC2(C)CNC(C2CCC([N+](=O)[O-])CC2)=O)CCCO1 c1(C(=O)NCC(C)(C2CC2)NC(CCCOCCC)=O)cc2n(n1)CCN(C)C2 c1(C(N2CC3C(CNC(=O)Cc4cncc(F)c4)C3C2)=O)cc(Cl)cc(Cl)c1O c1(OC)ccc(CSCC(=O)NC2CC2NC(=O)C=Cc2ccoc2)cc1OC C(=O)(Nn1nnc(C)c1C)C1CCN(C(c2nc(CC)oc2C)=O)C1 C1(NC(=O)Cn2ncc(O)nc2=O)CCC2(CC1)CC2NC(C1CC1F)=O c1(OCC)ccc(N2CCN(CC3COC(C)CO3)CC2)cc1F Cc1c(C(=O)N(C2CCCN(C(c3conc3C(C)C)=O)CC2)C)cccc1F N1(C(c2ccc(CC3CC3)s2)=O)CCCC2(C1)CN(c1nnco1)CCO2 c1(C(N(C)CC2CCN(C(c3ccc(F)cc3N)=O)C2)=O)ccc2c(n1)CCO2 c1(NC(C(=O)NCC2CCN(CC)CC2)=O)ccc2c(c1)C(O)CC2 c1(OC)cnc(C(N2CC3(CNC(C4CC(F)(CF)C4)=O)CC2CO3)=O)c(F)c1 C(C(=O)NCCC(C(C)C)NC(C1SC2C=CC1CC2)=O)(C(C)(C)C)NC(C)=O N1(C(c2c(C)scn2)=O)CC2(C1)C(NC(C1CCCC(O)C1)=O)CCS2(=O)=O C1(O)(C(C)NC(CS(CC)=O)=O)CCN(C(c2c(C(F)(F)F)noc2C)=O)CC1 C1(C(N2CCC(O)(n3cc(COCC)nn3)CC2)=O)CNc2cnn(C)c2C1 CC(C)(C)C(C)(C)C(=O)NCC(C1(C2CCC2)CC1)NC(=O)C(F)C1CCC1 c1(NCC2N(CC)CCC2)cc(C)c(S(=O)(=O)N2CCC(c3nccs3)C2)cn1 O=C1CCC(C(=O)NCC(N2CC(C3CCCO3)C2)=O)O1 Cc1cc[nH]c(=N)c1C(=O)NCC1CC2CCC1N2C(C1CC2(CCCC2)C1)=O Cc1cc(CNC(=O)CCCN(C(=O)CCc2ccc[nH]2)C)nc(C)c1 C(=O)(CC(CC#N)c1ccccc1)NC(CCNC(C(COC)C)=O)C N1(C(C(C)NC(C2CNC(=O)O2)=O)=O)CC2NC(=O)OC2C1 C1(C(=O)NCCC2CN(C(=O)COC(C)C)C2)(CC)CCC1 c1(C(=O)NC(CC)CNC(=O)CC2C=CCC2)ccc(OCC(F)(F)F)nc1 C1(C(N2CCC(OCCNC(C3=CCCC3C)=O)CC2)=O)COC2(CCC2)CO1 C1(CC=C)(C(=O)OC(C)(C)C)CCCN1C(=O)Oc1cc(C(N)=O)ncn1 N1(C(c2cc(C)c(Br)cc2)=O)CCC2CCN(C(c3nc[nH]n3)=O)C2C1 C1(NC(c2c(C)scc2)=O)CC2CC(NC(c3cccnc3N)=O)CC2C1 C(=O)(C(CC)C(F)(F)F)NCC(CCNC(CCCCC=C)=O)=C CC#CCCCC(=O)OCc1ccc(-n2cncn2)cc1 N1(C(Cc2ccn(C)n2)=O)C(CC(=O)NN2CCOCC2CCO)C2CCCC12 N1(C(C(C)(C)C2CCOC2)=O)CCC(N=[N+]=[N-])(C(=O)NCc2cncc(F)c2)C1 c1(C(N(CCOC)CCNC(=O)CC2(C(F)(F)F)CC2)=O)ccc2n[nH]cc2c1C C1(NC(c2c(NC)snc2C)=O)CC2(C1)CC(CNC(=O)C(C)(C)C(=O)NC)C2 C(c1ccc(Br)cc1Cl)=CC(N1C(CC(N2CCC3(CC2)COC3)=O)CCC1)=O c1(CNC(C(C)C)C(F)F)cc(Br)ccc1Cl c1(C2C(C(=O)Nc3cccc(C#N)n3)C2)ccc2c(c1)OCO2 c1(C(N2CCC3(C(=O)NC4CCC(F)(F)C4)CC3C2)=O)ccc2c(c1)CCO2 N1(C(c2c(C)snc2)=O)CC(NC(=O)C2=CCCOC2)CC(C)C1 c1(C(=O)NC(c2ccccn2)C)nc2ccc(-c3ccc(F)c(F)c3)cc2o1 C1(n2cccn2)(C(=O)NCC(CC)(CC)OC)CCN(C(c2occc2C)=O)CC1 C(=O)(C1=CCCCCC1)N1CC(C)C(NC(C2(C(=O)N(C)C)CC2)=O)C1 C(C)(C)(CCC(=O)NC(CO)C(C)NC(C1CC1c1ccccc1Cl)=O)OC C1(C(=O)NCCCCCO)CC12CN(C(c1cccc(-n3cncn3)c1)=O)C2 Cc1ccc(C)n1CCCC(=O)NC(CNC(c1csc(C(C)C)n1)=O)C1CC1 c1(C2C(C(=O)OC)C2)ccsc1NC(=O)Nn1cc(C(C)(O)CCO)nn1 c1(OC)cc(N)c(C(=O)NCC2(NC(=O)C3CC3)CCCCC2)cc1F C1(C(N2CCC(CN(C)C(c3cncc(Cl)c3)=O)C2)=O)Cc2c(F)cccc2O1 c1(C(=O)NC(C)C(C)(C)NC(c2ccc(C(O)CF)cc2)=O)ccc(O)nc1 CC(CN(C)C)C(=O)NCCN(C1CC(C(N2CCC2)=O)C1)C=O c1(C(=O)NCC2(F)CC(CNC(C3C(C(C)C)C3)=O)C2)ccc(F)c(O)c1 c1(C(=O)NCC2(C)C(C)CN(C(CSCC=C)=O)C2)cc2cccn2cn1 C1(C)(CNC)CC2CC2C1.c1(N(C)C)scnc1C(N1CC2(C1)C(=O)N2)=O CC1(CNC(c2cnc(Cl)c(Cl)c2)=O)CCCN(C(c2n[nH]cc2Cl)=O)C1 c1(OC)ccc(C2CC2)c(C(N2CCC(NC(=O)C=C3CC3)C(F)C2)=O)c1 CCC(CC)C(C)C(=O)Nc1cccc(NC(=O)Cn2cc(Br)cn2)c1 C12(CCNC(CCCNC(C)=O)=O)CCC(C1)N(C(c1cnc(N)cn1)=O)C2 C(=O)(CC(O)CC(C)C)NC(C(=O)NC(CCCCC)C)C(C)(C)C C1(CC)(CC)CC(NC(c2ccoc2CNC(=O)CC2(C)CCOC2)=O)C1 c1(C(N(CCCNC(c2cnc(-c3ccccc3)o2)=O)CC)=O)cc(C)n(C)c1 c1(C(=O)N(C(C#C)CC2CCCC2)C2(c3ccncc3)CC2)cccc(Cl)c1C C1(CN(C(=O)CCCc2ccsc2)C)CCCCN1C(=O)CC1CSCCS1 c1(C(C(=O)NCC)N(C)CC2CCC(C)C2)cc(Cl)cc(Br)c1OC N1(C(C2(OC)CCC2)=O)CCC(O)C(NC(=O)CSc2ccc(C)cc2C)C1 c1(C(=O)OC)cc(N2CC(CNC(C34CC(SC)(CO3)C4)=O)CC2C)ncn1 c1(CN(C(=O)C(C)C)C)cccc2[nH]ncc12.c12nnc(n1CCC#N)C2C N1(C(c2cncc(CC)c2)=O)CC(CNC(c2ccc(F)cc2)=O)N2CCC1C2 c1(C(=O)NC(C2N(C(c3c(C)c[nH]c3)=O)CCCC2)C)nnc2ccccn12 C1(NC(CCCSC)=O)C2CN(C(c3ccc(CC#N)cc3)=O)CC12 CCCS(=O)(=O)CC(=O)N(C1CCN(C(C2CC2Cl)=O)CC1)C CCCC(CC)NC(=O)C(O)CNC(c1csc(C)c1)=O CC1CN(C)CC(C(N2CC(O)(C(C)NC(c3nccs3)=O)C2)=O)O1 C1(NC(c2c(C)ncs2)=O)CC(C(=O)N(C)CCF)C1(C)C N1(C(c2cc(OC)no2)=O)CC(C)CN(C(c2ccc(S(C)(=O)=O)o2)=O)CC1C c1(C(=O)NCCOCCNC(C2ON=C(CC)C2)=O)cc(C)ccc1Br C(=O)(CCCCCF)NCCc1c(CNC(C2(C)CCC(C)C2)=O)nco1 C(=O)(C1CCCn2ccnc21)N1C(Cn2cc(-c3cncc(C)c3)nn2)C=CC1 c1(C(N2C(CNC(C3C(C)(C)C3(F)F)=O)CC(F)C2)=O)cc(C(F)F)ccc1F C=CCC(C)(CC=C)NC(=O)C(C)N(C(C1CC(O)C(F)C1)=O)CC c1(CC)cc(CC(N2CCC(O)(CNC(c3cocn3)=O)C2)=O)n(C)n1 C(=O)(C(=O)CCC(C)(C)C)N(C(C)CNC(=O)COc1cccnc1Cl)C c1(SC(CN2C(=O)N(CCC)C(C(C)C)C2=O)=O)cccc2ccnn12.C1CO1 C(C(C)(C)C(=O)NCc1nc(C)c(-c2cccc(C)c2)s1)N(CC)CC c1(C(=O)NCCC2N(C(c3nc(C)oc3)=O)CCSC2)n[nH]c2c1COCC2 CC1c2ccccc2OC1CC(N1CCCC(CNC(C2(O)CCCC2)=O)C1)=O O(N1CCC(NC(C2CC(O)(Cn3cc(CCC4CC4)nn3)C2)=O)CC1)CC C1(NC(C=Cc2ccc(C(N)=O)o2)=O)CCC2(CC1)CN(C(C1CC1(Cl)Cl)=O)C2 C(CN=c1cc(C)c(S(=O)(=O)NC2CSCC2C)c[nH]1)N(CCO)CC N1(C(c2[nH]c3cc(C)oc3c2)=O)CCC2CN(C(=O)Cc3ccoc3)CCC2C1 CCCCCN(CCN(C)C)C(=O)NCC1CCC1C(C)(C)C CS(=O)(=O)c1ccc(C(=O)NCCC2CC(NC(c3cc[nH]c3C3CC3)=O)C2)o1 C=CC(C)CC(=O)N1CC=CC1C(=O)NCc1nnc(O)n1CC C1(C(N2C(CNC(C(C=C=C)C)=O)CC3(CC3)C2)=O)CCC2(CC1)CC2(F)F c1(OC)ccc(C(C)NC(=O)NCCc2cc(C(N)=O)no2)c(C)n1 C(CC(C)CC(C)(C)C)NC(C(C(C)OC)NC(C1CCC(C=C)CC1)=O)=O N#Cc1ccncc1C(=O)NCC(O)CNC(=O)C=Cc1ccccc1F c1(N2CC3CC(NC(c4ncc(OC)cn4)=O)C3C2)c(Cl)cccc1[N+](=O)[O-] N1(C(c2c(COC)cc[nH]2)=O)CCC(C)C(CNC(c2ccc(C)cc2C)=O)C1 Cn1cc(-c2cc(C(=O)NC3CCC(NC(=O)Cc4cc[nH]c4)C3)n[nH]2)cn1 N1(C(c2[nH]c(=N)sc2)=O)CC2CC1CCN2C(C1C2CCCCCC12)=O CC(CCC(C)(C)C)C(=O)NC1CC(NC(=O)C(=O)NCCC(N)=O)C1 N1(C(c2n(C)ncc2[N+](=O)[O-])=O)CCCC2(C1)CN(C(C1CC3CCC1C3)=O)C2 c1(C(N(CCC(=O)NCC(CCC)(C)C)C2CC2)=O)c(C#N)cnn1C c12cn(nn1)CCN(C)C(=O)CC2.C1(N(C)C)CC(C(=O)O)C1 N1(C(C)C)CCCC(NC(=O)NCCNC(=O)CC2CC2C)C1 N1(c2nccc(CC#N)n2)CCC(NC(c2cccn(O)c2=O)=O)C(CO)CC1 CCC(C)(C)CC(=O)NC(CC(=O)N(C12CC(C1)C2)C)C(F)F c1(C(=O)NCC2C(C(=O)NC(C3(CO)CC3)C)C2)noc2ccccc12 C(CC(=O)NCC1CCCS1)(C(C)OC)NC(c1c(OC)n(C)nc1)=O N1(C(C2CC(CC)C(=O)CC2)=O)CC2(CCN(C(=O)CC(CC)OC)C2)C1 CCC(CC)C(F)C(=O)NCC1CCN(C(C2CC3(CCC3)C2)=O)C1 C(=O)(CC(O)CC(C)(C)C)N1CCC(C(C)NC(C2CC(C#N)C2)=O)CC1 C1(C(=O)NC2CCS(=O)CC2)CC12CCN(C(C1CC3CC1CC3=O)=O)C2 c1(-c2cc(OC)c(O)cc2)ccc2[nH]c(C(=O)Nc3ccno3)nc2c1 c1(CNC(C(=O)NC2C(C#N)(C(=O)OCC)CC2)=O)cc(N)cc(N)c1 C1(C(=O)NC2CC3(CN(C(CC4(C)CC4)=O)C3)OC2)CCCC12CCOCC2 Cn1cc(NC(C2(c3cccc(N)c3)CC(=O)C2)=O)c(OCC(F)F)n1 CN1CCC(NC(c2sccc2CNC(C2(C)CCC2)=O)=O)C(C#N)C1 N1(C(C2CCC(CNC(CSCC)=O)C2)=O)CC2CCC1CC2 c1(C(N(C)CC2CCCN(C(C(C)NC(N)=O)=O)C2)=O)ccc(S(C)=O)cc1 C1(C(N2CC3CC(NC(C(N)=O)=O)C3C2)=O)CC2COCC(C1)C2=O C1(CC(=O)NC23CC(CNC(c4c(OCC)scc4)=O)(C2)C3)C(=O)NN=C1C CC1(C)CCN(C(C2C3CCC(F)(F)C23)=O)C(C(N2CCC(C3(C)N=N3)C2)=O)C1 c1(NC(C2CCCN(C(C3(CC)CC3)=O)C2)=O)ccc(C(F)(F)F)c(I)c1 c1(C(N2CC3CC2CS3=O)C(=O)NCC)cc(C)nnc1C C(=O)(CCCC(F)(F)Br)N1CCCC(C(N2CCCCCC2CO)=O)C1 C(=O)(CC(C)(C)C(F)(F)F)N1C(c2ccc(C)o2)COCC1 N1(C(c2cc(C(N)=O)[nH]c2)=O)CC(NC(=O)CC2CSCCS2)CCC(O)C1 Cc1cc(CN2CCOCC2C(=O)Nc2cccc(C#N)c2)cc(O)c1 n1(CC)cnc2c(NCCCN(SC(F)F)C)[nH]c(=NCC3(CCO)CC3)nc12 c1(CC)cc(F)ccc1C(=O)NC1CC(NC(=O)CN(S(C)(=O)=O)C)C12CCC2 C(CCC(=O)N(C)C(C)C1CC1)NC(C=C(C)C(C)C)=O C1(C(=O)NC(c2cn(C)nn2)C(=O)NCCc2ncc(C)o2)COCCC1C C1(NC(c2cccc(OC)c2)=O)CN(C(c2ccc(O)c(Cl)n2)=O)CCC1C c1(-c2cc(CO)no2)nnc(N2CCC(Cl)CC2)n1CC1CCCO1 N1(C(C(c2c(C)cccc2Br)NC(c2nc(C)oc2C)=O)=O)CCS(=O)C(C)C1 C1(CCNC(C(CC)OC)=O)CC2CCC(C1)N2C(c1nc(O)c(C)s1)=O c1(C(=O)NC(C)CCN(C)C(c2ccc(F)o2)=O)ccc(OCC(F)F)cc1 N1(C(C(C)=CC)=O)CCCC2(CCN2S(=O)(=O)Cc2cccc(C)c2)C1 c1(C(=O)NC(CNC(C2CC(=O)OC2)=O)CC(F)(F)F)cccn2ccnc12 CN1C(=O)CSC1=CC(=O)NCC1CC(O)(CNC(=O)Cc2cocn2)C1 Fc1cc(CNC2CCCC2(Cl)Cl)ccc1OC(F)(F)F C1(C(N2CC(NC(CC(=C)C)=O)C2)=O)CCCCN1C(c1nn(C)cc1SC)=O c1(C(=O)NC2CC(C)(NC(C(C3CCC(C)C3)=O)=O)C2)ccc(CCF)cc1 c1(C(N2CC(NC(CC3(COC)CC3)=O)(COC)C2)=O)ccc(C(N)=O)cc1 C(=O)(C1=C(Cl)CCCC1)NCC1OCC(C(N(CCCOC(C)C)C)=O)C1 Cc1nocc1C(=O)NCCN(C(C1CS(=O)(=O)C1)=O)C(C)C Cc1ccc(SCC(=O)NC2CCC2CNC(=O)CCC(C)(C)C)cc1C C1(N(C)C(C2CC23CCCC3)=O)CCCN(C(=O)CCN2C(=O)CCC2=O)CC1 c1(C(c2n(C(CC)(C)C)nnn2)NCC2(C)CCCS2)ccccc1N(C)C CC(N=c1ccnc(NC(C)COCC2CC2)[nH]1)c1ccns1 C1(CCC2N(C(C3CC(=C)C3)=O)CCC2)CCCCN1C(=O)C(C1CC1)C1CC1 C1(CNC(C(CCC)C)=O)CCC2CN(C(c3cscc3C(N)=O)=O)CC12 N1(C(C2C(OC)CCC2)=O)CCC(NC(=O)CCCF)C1C C1(NC)(CO)CCOCC1.C1(CCn2c(CCC(=O)NC)nnn2)CCC(C)(C)C1 c1(CC(=O)N(C2CCCN(C(=O)CC3CC3)C2)CC)ccc(F)c(Cl)c1 C1(C(=O)NC2C(CNC(c3cncc(C4CC4)c3)=O)C2)Cc2ccc(F)cc2C1 N1(CC(=O)NCCCCCCNC(C2(C)CC3CC3C2)=O)CCn2ccnc2C1 c1(C(N(CC(C)NC(=O)CC2SC(=N)NC2=O)CC)=O)cccn2[nH]c(=N)nc12 c1(CC(=O)OC)cc(SC2CCN(C)C2=O)c2c(c1)CCO2 c1(C(=O)NCCCNC(c2cc(=O)cc[nH]2)=O)cncc2nc(O)[nH]c12 CS(=O)(=O)c1coc(C(N2CCC(O)(CNC(=O)C(O)CF)CC2)=O)c1 N1(C(C2N=C(C)SC2)=O)CCCC(N(C(=O)CN2CCCNC2=O)C)CC1 N12CCCC3C1CCCN3CCSCCC2=O.C1(C(N)=O)CC1C(F)F C1(C(N2CC(C)OC(C(N3CC(C)(C)C3)=O)C2)=O)COc2ccccc2O1 N1(C(CC=CC)=O)CCC(CCNC(=O)C(C)C(O)C(C)CC)C(F)(F)CC1 C1(C(=O)NC2(C3N(C(C=C(C)Cl)=O)CCC3)CC2)CC(C)(C)OC1(C)C C1(C(=O)NC2(CO)CN(C(=O)C(O)Cc3ccccc3)C2)CC2CC1CC2O Cc1ccc(CN2CCCC(NC(C3(n4cccn4)CCC3)=O)C2)cn1 c1(CC(N2CC(SC)C(NC(=O)CSC3CCCC3)C2)=O)csc2nccn12 N1(C(CCCCCC)=O)CCN(C(c2c(F)cc(F)cc2Cl)=O)CC(C)(F)C1 C(=O)(C(F)C(C)C)N(CC(CC)NC(=O)CCc1ccsc1Br)CC N1(C(C2C(NC(C3CCCC(=O)N3)=O)CCOC2)=O)CCCC12CCNC2=O O=C(C#CC1CCCOC1)NCC1C=CCN1C(c1ccc(N2CCC2)nc1)=O C(c1cc2ccccc2o1)=CC(=O)N(CCNC(C1CC(=O)C1(C)C)=O)CC c1(OCC)nc(C)ccc1C(=O)NCC1(C)CCN(C(c2cccnc2O)=O)C1 C1(CCC)(C(=O)NC(C)C(CO)NC(=O)Cc2cc(C3CC3)no2)CCNC1=O C(=O)(C1CCCc2nncn21)N1C2CN(C(c3cnc(OC)s3)=O)C(CC2)C1 c1(C(=O)NCC2(C(C)NC(=O)CP(C)(C)=O)CC2)ccc(F)cc1C#N c1(C(N2C(C3(CNC(CCC(=O)NCC)=O)CC3)CCC2)=O)cc(C#N)[nH]c1C C(CCO)(C(C)(C)O)NC(CCN(C(C1CCCN1C=O)=O)CC)=O N1(C(=O)OC)CCC12CC(COCC)C2.N12CCN(C)CC1C2C(=O)NCC C(C(CC(F)(F)F)NC(c1cccnc1)=O)NC(C(c1ccnn1C)C)=O c1(C(=O)NC2C(NC(c3c(C)n[nH]c3)=O)CS(=O)(=O)C2)ccc(F)c(F)c1F c1(C(=O)OC)cc(C(=O)NC(C)CCNC(=O)C(n2ccc(C)n2)C)c(C)s1 N1(C(CC2(O)CC(C)(C)OC2)=O)CCCC2(C=CCO2)CC1 N1(C(CC=C=C)=O)CC(CNC(c2cc(C)nn2-c2ccccn2)=O)C2(CC2)C1 C1(NC(c2cc(C)cc(C)c2)=O)CCN(C(=O)C2=CC(O)CCC2)CCC1(F)F C1(NC(c2n(CC)ccc2)=O)CCN(C(c2cccc(=S)n2O)=O)C(C)C1 C1(C(N(C(C=C)C)C)=O)CC2CC1CC2NC(=O)C(COC)COC c1(C(N2CCOCC(NC(c3ccc(Cl)cc3)=O)C2)=O)cccc2c1OCO2 CC1C(C)N(C(c2cccc3nccn23)=O)CCN1C(=O)C=Cc1sccc1Br C12(CC(=O)NC3C4CC(NC(c5cnc6n5CCC6)=O)CC34)CCCN1CCC2 C(=O)(C(C)(F)C(F)(F)F)N1CCC(NC(C=CC(=O)OCCCC)=O)C1 Cc1nn(CC(=O)NC(CNC(c2cc(Cl)ccc2Cl)=O)CO)c(C)c1C c1(C(=O)NC2C(CNC(CCCSC)=O)C2)ccc(C(C)(C)C(F)(F)F)cc1 C(CC(C)(C)C(=O)NCCCCn1cc(CCC(=O)N(C)C)nn1)OC c1(C(N2CC(C(C)NC(CN(C(COC)=O)C)=O)C2)=O)cc(C2(Cl)CC2)n(C)n1 c1(C(=O)NCC(C)(C)CC2CC2)cccc(NC(=O)CC2CSC2)n1 Cc1ccc(C(C)CNCCCNC(c2cccs2)=O)cc1 CC1(C)CCC(CNC(C2CCCC2n2cccn2)=O)OC1 N#Cc1ccc(=NCC2CN(C(c3cnc(C4CC4)s3)=O)CC2C(F)(F)F)[nH]c1 C1(COC)(NC(C2CCCCS2)=O)CCCN(C(c2nocc2C(C)(C)C)=O)C1 C1(C(N2CCCC2Cn2cc(COC3CCOC3)nn2)=O)CCc2ncncc2C1 c1(C(=O)NCCC2CCN(C(CNC(C)=O)=O)CC2)ccc(S(=O)(=O)N(C)C)o1 c1(OC2(C(=O)NC3CC(N(C)C(c4ccncn4)=O)C3)CC2)cccc(Cl)c1 N1(C(c2cn(CC)nc2)=O)CC(NC(C2(C(N)=O)CC(O)C2)=O)CC1COC C1(NC(C2C(C)(C)CC2)=O)C2CCC1CN(C(C1(Cl)CC1)=O)C2 c1(C(=O)C(c2noc(C)n2)C)cccc(C2CC(O)CN2c2cncc(Cl)n2)c1.CO Cc1ccn(CC(N2CCC23CN(C(=O)C(c2cccc(F)c2)C)C3)=O)c(=O)c1 N1(C(CCCN(C(C)=O)C)=O)CC2C(CN(C(=O)CNC(=O)C(F)(F)F)C)C2C1 C1(NC(Cn2ccc(C)n2)=O)CC(C)CN(C(=O)NC2CC2c2ccno2)C1 c1(C(=O)NCC(CNC(c2cncc(C)n2)=O)CO)c(C(F)F)cccc1N c1(C(=O)NC2CC(C(C(=O)NC(CCOC)CO)F)C2)cc(O)ncc1F CC1(C)CC(NC(=O)C(O)CCCc2ccccc2)CN(C(c2cncs2)=O)C1 N1(C(c2c(CC)con2)=O)CCC(NC(c2cc(-c3ccco3)c[nH]2)=O)C(O)C1 C(C)(C(=O)NC1CCC(CNC(C2(C)CCOCC2)=O)C1)(C(C)C)NC(C)=O CC(CCC(=O)NCC12CCC(CC1)C2)NC(C1CC(C2CC2)C1)=O CC1CCN(C(=O)CCc2ncc[nH]2)C1CNC(=O)C(C1CC(F)(F)C1)O C(CC(=O)N1CCC(C(F)F)C1)(C(F)(F)F)NC(C1(C(C)C)CCC1)=O N1(C(C(c2nc(C)sc2CC#N)=O)=O)CCC(c2ccccc2C)C1(C)C C(=O)(C1=NN(C(C)C)C(=O)CC1)NCC(CN(C(C(CC(C)C)(C)C)=O)C)(C)C c1(C(=O)NCCCC(C)NC(c2c(C(F)(F)F)nc(C)o2)=O)cccc(C)c1F CCCCCCC(=O)NCCC12CCC1CN(C(c1cc(C)oc1C)=O)C2 O=S1(=O)CCC2(CC1)CN(c1cncc(OCCOCC(F)(F)F)n1)CCN2 CC(C)(CC(=O)NC1CCCC(CC(=O)O)C1)c1ccccc1 C1(CC)CN(C(=O)CCC(C)OC)CCC1NC(c1cc(OC)ccn1)=O c1(C(=O)NC2(C)CC(NC(C(C)C(C)O)=O)C2)nc(N(C)C)ccc1Br C(=O)(C(O)CC(N)=O)N1CC(CC(C(=O)N(c2ccsc2)C)F)C1 Cc1nsc(CN(C)C(C2(CNC(=O)CC3CCSC3)CCC2)=O)n1 C1(OC)(CNC(=O)CCCSC)CN(C(C2CC(=O)N2)=O)C1 CC(C)CC(=O)N1CCCC1CC(N1CCCC1CC1CC1)=O Cn1nc(CNC(C2(O)CCCC2)=O)cc1C(=O)NCc1cscn1 N1(C(C2CC(C#N)C2)=O)CCN(C(C2CC=CCO2)=O)CC1CS(C)(=O)=O c1(NC(CCC2N(C(C(C)OCOC)=O)CCC2)=O)cnc(F)cc1C N#Cc1nc(Cl)ccc1NC(c1ccncc1-c1[nH]cc2c1CCC2)=O C1(NC(c2cc3sccc3[nH]2)=O)CN(C(=O)Cc2ccc(F)cc2Br)CCC1O CC(CC(C)(C)C)C(=O)OCc1ccc(Cl)cc1 CC(C)CCC(=O)NC1C=CC(CNC(C2CCN(CC(C)C)C2)=O)C1 C(=O)(CCC(C)(F)F)NCC1N(C(CCNC(=O)OC)=O)CCCC1 n1(C(C)C)cnc(C(=O)NCCC(O)CNC(=O)C=Cc2nccs2)n1 C1(NC(Cc2c(OC)cccc2)=O)CN(C(C2CC3CCC2O3)=O)CC1(F)F c1(NC(CC2CCN(Cc3cc(C)sc3)C2)=O)cc2cnccc2o1 c1(CC)ncnc(CC)c1C(N1CC(NC(C2CCCSC2)=O)C(O)C1)=O C12(C(=O)NCCC3CCN(C(c4c(C)n(C)nc4)=O)C3)CCN(C1)S(=O)(=O)C2 c1(C(N2CC(NCc3ncc(OC)nc3)C(C)C2)=O)nc(C)c(C)nc1C C1(CC)(CC)CN(C(=O)C(=O)NCc2nnc(CO)s2)CCO1 Cn1nc(C(=O)NNc2nc(-c3ccccc3)cs2)c2c(c1=O)CCCN2 C12CCC(CC1)C(=O)OC2.c1(C(CC(=O)NC)C)ccc(CO)cc1 O=C1CC(C(N2CC(CCNC(c3cncc(Cl)c3)=O)C2)=O)CCN1 N1(C(c2c(C)nc(=N)[nH]c2)=O)CCC2CC2(NC(=O)C(F)=CCCF)CC1 N1(C(C2CC(C)C2)=O)CCC2CN(C(c3ccc(C(C)C)s3)=O)CC12 C(=O)(CCCN(C)N=O)NC1CC(O)C1CCO.C1(C2(C)CC2)C(=O)N1 c1(C(N2CCC(NC(C(N3CCOCC3)C)=O)C2C)=O)cccc(Cl)c1F c1(NC(N(CC)CC2(CC)CCCC2)=O)nccnc1F Cc1cccc(CN2CCC(CC(=O)NCc3ccc(F)cc3Cl)C2)c1O c1(C(=O)NC(C2CCCCN2C(=O)C2=CCC2)C)cnc(O)n(C2CC2)c1=O N1(C(c2c(OC)csc2)=O)CC(NC(=O)Cn2cnnc2)CC(O)C1 Cc1cnc2c(C(=O)NC3CC(NC(C4CC5(CC5)C4)=O)C(O)C3)cccc2n1 c1(C(=O)NCC(C)(C2CC2)NC(=O)Cn2cnnn2)cnn(CC2CC2)c1 N1(C(CC(CC=C)NC(=O)C(C)(C)CCF)=O)C(CO)CCC12CCC2 CN1N=C(CC(=O)N2CC(C)(OCC(N3CCOCC3C(F)F)=O)C2)CC1=O N1(C(c2c(F)ccc(C)n2)=O)CCN(C(=O)CSc2cccs2)CC(C)(F)C1 c1(C(=O)NC2CC(C)(CNC(c3cc(COC)on3)=O)C2)cnn2ccn(C)c12 CC1(C)CCCC1(C)NC(=O)CC1CC1CNC(C12CCCC1C2(F)F)=O N1(C(C2CCCC(C#N)C2)=O)CCC2(CCC2)C(CNC(=O)CC2CCC2)C1 Cc1cccc(C(N2CC3CC2C3NC(C2CC(NS(C)(=O)=O)C2)=O)=O)c1 C1(CNC(CCN(C(C)C)C(C2CC(C)(C)CO2)=O)=O)OCCC1(C)C CCCC(C)(C)C(=O)NCC1CC(NC(c2cc(=N)[nH]n2C)=O)C1 c1(CC(=O)N(CC(C)(C)N(C(C=CC=CC)=O)CC)C)ccc(C)c(C)c1 N1(C(C(COC)OC)=O)CCC(C(C)(C)NC(c2csc(C)c2)=O)CC1 c1(C(N(C(CC(=O)N(C)Cc2cc(C)n(C)n2)C)C)=O)nnc(O)nc1O CC1(CC(=O)NCC2(C)CC(NC(c3cnc(C(F)(F)F)s3)=O)C2)CCCO1 C1(OC)CC(CNC(=O)CCC(F)F)N(C(=O)CCC2(C)CC2(F)F)C1 Cc1nn(C)c2sc(C(=O)NCC3CCC3NC(=O)C(C)(C)CC3CC3)cc12 C(=O)(C(C(C)C)Oc1cccc(Cl)c1)NC1CC(NS(CCC)(=O)=O)C1 c1(O)cc(C)ccc1Cl.c12ccccc1COC(=O)COC=CC(=O)OC2.CO C1(NC(CCCCC=CC)=O)CC1C1CCN(C(C2CCC(C)O2)=O)CC1 C1(C(=O)NC2CN(C(C3CCN3C(C)(C)C)=O)C2)(CC)CCCCC1 C1(C(=O)NCc2ccc(-c3cccc(Cl)c3)o2)CCC2C1C2(F)F C1(OC)CC(C(=O)N(C)Cc2ccc(SC)o2)N(C(c2coc(C)n2)=O)C1 C1(NC(C2CSC2)=O)(CO)CCCN(C(=O)CCc2cnoc2)C1 CC1CC(NC(C2CCCC2(C)C)=O)CN1C(c1cc(-c2ccn(C)n2)on1)=O c1(NC)ccc(CNC(=O)C(=O)NCCC(=O)NC2CCC(CC(C)C)C2)cc1 C=CCC(C(=O)NC(C)C(C)NC(=O)CCN1CCOCC1)C(C)C c1(C(N(C(C(=O)N(C(C)C)Cc2ccccn2)=O)C)C)cccc(F)c1I N1(C(CCOCCC)=O)CCC2CCC(NC(C34COC(CSC)(C3)C4)=O)C12 C1(CNC(COC(CNC(c2c(CC)non2)=O)(C)C)=O)COCC1(C)C Cc1sc(C)c(C(N2CC3CC2C3NC(C2CC(=O)NC2=O)=O)=O)c1C#N N1(C(c2cc(CNC(c3cc(C(C)=O)[nH]n3)=O)[nH]n2)=O)CCCC(CF)C1 C12(CN(C)Cc3c(CC)noc3)CC(CCO1)C2 c1(C(N2CC(CC)N(C(C3C4CCCCCC34)=O)CC2)=O)cc(C)nc(C)c1O N1(C(Cc2c(C)nn(C)c2)=O)CC2(CCC2)CC1C(N1CCOCCC1C)=O N1(C(CC)CC)CCC(N=c2[nH]c(=N)[nH]c(=NCCc3nc(O)n[nH]3)[nH]2)C1 c1(C(=O)NC2CN(C(c3n(CC)nc(C)c3)=O)C2)cc(C)cc(C)c1 C1(C)(CNC(CN(C)C)=O)CN(C(=O)C(F)(F)c2cscc2C(F)(F)F)CCO1 c1(CC(=O)NC2C(CNC(c3ccc(SC)o3)=O)C2)c(F)cc(F)cc1F c1(NC)cc(Cl)ccc1C(N1CCN(C(=O)Cc2ccc(F)cc2C)CC1)=O C1(C(=O)NC2C(C)N(C(c3csc4nnsc34)=O)CC2)Cc2cccc(F)c2O1 CC1CN(C(=O)CSCCN(C)C)CC(C)N(CCN2CCC(C)(C)C2)C1 N1(C(c2n(C)ccc2)=O)CCC(C2CC(NC(c3ncccc3Br)=O)C2)C1 N1(C(C(C2CCCOC2)OC)=O)CCC(CNC(=O)CC(F)(F)F)C(F)(F)C1 N1(C(=O)Cc2ccon2)CC(NC(C2(n3ccnc3)CC2)=O)C(CO)C1 c1(C(=O)NC(C(=O)NCC(C)S(N)(=O)=O)Cn2cccn2)cn2c(n1)CCC2 N1(CC(=O)N(CC(CN(C(c2c(CC)csc2)=O)C)O)C)CCCNS1(=O)=O Cc1cn2cc(C(=O)N(C3CC4CC3N(C(=O)C=CBr)C4)C)ccc2n1 C(=O)(CC(C)C(C)C)N1CCCC(CN(C(c2c(C)nc(CO)o2)=O)C2CC2)C1 c1(C(=O)NCC(C)NC(C2CC(=C)C2)=O)ccc(CC=C(C)C)cc1 CC(C)C(C)(CNC(c1ccc(-c2ccsc2)nc1)=O)NC(C12CC(F)C1C2)=O C#CC(C)(C)C(=O)NC1C=CC(C(N2C(C)CC2(C)C)=O)C1 CN1CCCC(F)(C(=O)NC2CCCC(CN(C(=O)CCOCC(F)F)C)C2)C1 CCC(CN(C)C)C(=O)NCC1(F)CC(NC(=O)CCC(C)OC)C1 c1(C(=O)NCCCCc2ccccc2Br)cc([N+](=O)[O-])c[nH]1 C#Cc1cc(N(C(=O)C=CC(=O)NCC2COCC(=O)N2C)CC)ccc1C Cc1oc(C(C)(C)C)cc1C(=O)NC(C1(O)CCN(C(c2ncn(C)n2)=O)C1)C N1(C(CCC2CCC(=O)NC2)=O)CC(NC(=O)Cn2cccn2)C2CC2C1 C1(C(=O)NCC2(CCC)CC2)CC(NC(c2coc(C)c2)=O)CCO1 C(=O)(CCC(C)S(C)(=O)=O)NCC1CN(C(C(CCC)C#N)=O)C1 N1(C(C2(c3ccccc3)CC(F)(F)C2)=O)CC2(CCN2C(C2COC(=O)C2)=O)C1 c1(N2CCCC(C(C)NC(=O)CC3=CCCC3)C2)nc2cccc(F)c2o1 C1(C(N2CC(C(C)NC(C3(CN(C)C)CCC3)=O)C2)=O)CCCC12CCC2 C1(C(N(CC(CN(C(C2CC(C(C)C)C2)=O)C)O)C)=O)CN(S(N)(=O)=O)C1 C(=O)(C1=CN=C2N=CNN2C1)NC1C(C)CN(C(C2CC(N(C)C)C2)=O)CC1 C(CC(O)C(=O)NC(CNC(c1ccnc(-n2ccnc2C)c1)=O)C1CC1)SC C(CNC(=O)C(=C1CCCCC1)F)(C(=O)NC(C(N)=O)C1CCCC1)N(C)C O=C(CC(F)(F)C(F)F)NCCC1(O)CCCN(C(C2CC2(F)Cl)=O)C1 c1(C(=O)NC2C(NC(CCOC(C)C)=O)CCC2)noc2c1COCC2 C1(CN(C(CCOC(C)=O)=O)C)CCCCN1C(C1CCC1(C)C)=O C1(CC(=O)NC2C(O)CCN(C(c3c(CC)c[nH]n3)=O)C2)CC(C)CC(C)(C)C1 c1(CC(=O)NC(CC)CNC(c2nn(C)cc2C)=O)cccc2c(C)csc12 c1(C(=O)NCC(CNC(CC(C)F)=O)F)ccc(-c2ccncc2)cc1 c1(C(CC)NC(C2CCC2NC(=O)CSCC(F)F)=O)nc(C)no1 C1(N(C)C)CCN(C(C2CC2NC(c2c[nH]c(C(C)(C)C)c2)=O)=O)CC1 CCC(C#N)(CC)C(=O)N1CC2CN(C(=O)C(c3ccc(CC)cc3)C)CC2C1 c1(C(N2CCC(CC(C)NC(C3CCCCO3)=O)CC2)=O)cc(N)cc(F)c1 C1(C(C)(C)NC(CCCC2(C)N=N2)=O)CCN(C(=O)C(C2CCCCC2)F)CC1 C1(NC(c2cc(OC)nc(OC)c2)=O)CN(C(=O)C(C)SC)C2(CCC2)C1 c1(CCCC(N2CCCC2)=O)cc(C)sc1C.N1(C(CC)=O)CCC1(CO)CO c1(C(c2n(CC)nnn2)(CC)NCCN2C(=O)CCC2=O)ccc(Cl)cc1C c1(CNC(c2nnnn2C2CCCCC2)(CC)C2CC2)cnn(C(C)C)n1 N(C(=NCCOC)N1CCCC(C(F)(F)F)(C(=O)OC)C1)C1CC(CCOC)C1 C(=O)(CC(C(C)(C)C)NC(=O)C(O)c1ccsc1)NCCC(C)P(C)(C)=O C(C)(C)N(C(C)=O)CCO.C1C=CC(=O)N1C N1(C(C2CCCOC2)C(=O)OCC)CCC(N(C(=O)COC)C)CC1 CCC(C)(C)C(O)C(=O)N(C(C)(C(=O)N(CC(C(C)C)OC)C)C1CC1)C c1(C(N2CC(CN(C(C3CN(CC)C(=O)C3)=O)C)C2)=O)cccc2c1OC(C)C2 C1(O)(CNC(C(C)OCCN(C)C)=O)CCN(C(=O)CN2CCCOC2=O)CC1 C1(C(NOC(C=C)C)=O)CCC(C)(C)N(C(c2nnc(O)nc2O)=O)C1 C(=O)(C(C)(C)C(O)C(C)C)NCc1cccc(C(N2C(C)(C(=O)NC)CC2)=O)n1 c1(C(=O)NC2(CCCNC(C3(N(C)C)CCC3)=O)CC2)ccc(N)c([N+](=O)[O-])c1 C1(C(=O)Nc2cncs2)CC(O)CCN1Cc1cccc(Br)c1Cl c1(C(N2CCC(N(C(=O)CCC3CC3(Cl)Cl)CCO)C2)=O)ccc2c(c1)OCC2 Cc1n[nH]c(Cl)c1CC(=O)NC1CCCC(NC(=O)C=CCN2CCCCC2)C1 C(=O)(C(C)(O)CC(F)(F)F)NC1(CNC(C(C)N(C)C)=O)CCOC1 c1(C(=O)NCC2(F)CCN(C(Cc3cc(OC)no3)=O)C2)cnc(C)nc1C N(C(=NCc1noc(C(C)C)n1)NC1CC1C(C)(F)F)C(CC)C CC1=NOC(C)(C(=O)NC2CC(C(C)NC(=O)Cn3cnnc3O)C2)C1 C(=O)(C(Cc1cn[nH]c1)NC(=O)CN1CC(C)(C)C1)N(C1CC(CO)C1)C c1(COC)nocc1CNC(C1CC(CNC(=O)CCc2nc(=N)[nH][nH]2)C1)=O C1(C)(CNC(c2c(C)[nH]cc2)=O)CCN(C(=O)C=CCNC(=O)OC(C)(C)C)C1 c1(C(=O)NCC(C2CCCCC2)NC(CNC(CC(C)C)=O)=O)cn(C)nc1O CCC(C)(CNC(=O)C(C1CCCC1)N(C)C)NC(=O)CSCc1ccccn1 C(C(O)(CNC(c1cc(CNC2CC3(CC3)CO2)[nH]n1)=O)CO)OC CCCCC(C(=O)N(CC(F)CO)CC)NC(=O)C=CCN(CC)CC c1(CCC)ncncc1C(N1CC(CNC(c2cc(C)n(C)n2)=O)(COC)C1)=O N1(C(C2(O)CC2)=O)C2CCC1CN(C(=O)OC(C)(C)C)C2.c12ccc(nn1)n2C C(=O)(C#Cc1ccccc1)N1CC(CNC(=O)Cc2ccccc2)OCC1 Cc1cccc(COCC(=O)N(CC(C)(C)NC(=O)C(C)C(F)F)C)c1 C=CCC(C(=O)N1CCCC1c1cn(C(c2cccnc2F)C)nn1)C(C)C N#Cc1ccsc1C(=O)NCC1CCN(C(c2ccnc(-n3cccn3)c2)=O)C1 CCCCC(c1nnnn1C1COC1)NCC1(C2CCCCC2)CC1 C(=O)(C(CC1CC1)NC(C1CCCN1C)=O)N1C(C(=O)NC)CC1 C1(NC(C2C=CC(NC(CCc3cn(C)nc3)=O)C2)=O)COC(C)(C)C1 C1(NC(C=C(C)C(C)(C)C)=O)CC2CC1N(C(C1(C)CC(C)(C)C1)=O)C2 C=C=CC(C)C(=O)NC1CCCCC1NC(C1(CS(N)(=O)=O)COC1)=O c1(COC2CCN(C(NC(CC)C)=NCC(C)C)C2)ccc(S(C)(=O)=O)c(Cl)c1 C(C(CNC(=O)C(CC)c1cccnc1)CO)NC(C(=O)NCCOC)=O C(=O)(CCCC(=O)NC)NC1CC(CNC(C2C(C(=O)NCC#C)C2)=O)C(O)C1 Cn1nc([N+](=O)[O-])cc1C(=O)NC1CCCCC1NC(c1csc(=N)[nH]1)=O c1(O)ccccc1Cl.CCS(=O)(=O)N(C)NC(CCC=CC(=O)NCC(C)SC)=O N1(C(C=CCOC)=O)CCC(CNC(=O)COc2ccc(F)cn2)C(O)C1 CC1CC(C)CC(c2nnnn2CC(F)F)(NCCOC)C1.c1(C)nncs1 C1(CNC(C2(CC)CCCC2)=O)CC(F)(F)CN1C(c1ccncc1Br)=O C(=O)(CCC(F)(F)C(F)F)NCCC(C)N(C(C(CC(C)C)NC(=O)OC)=O)C C(c1ccc(C)cc1)=CCC(=O)NCC1(C)N(C(C)=O)CCC1 C(=O)(C1=CCCCO1)NC(COC)CNC(=O)Cc1cccn1C O=C(CCCCCCn1cc(C2(CCF)CC2)nn1)N1CCCCC1 CCCC(C)(C(=O)OC)NC(c1occ2c1CCC2)=O c1(-c2ccc(SCCCC)s2)cc(C(=O)NC(c2ccc(Br)s2)C)c(F)cc1C C(N=c1[nH]c(Cl)ncc1C(F)F)C1CC(NC(C2CCOC2)=O)C1 c1(C(N(C(CNC(C2N(C(CC)=O)CSC2)=O)C)C)=O)ccnc2nc(C)nn12 CC1CCN(C(=O)C(C)(F)F)CCN1C(=O)COCc1cccc(C(C)(C)C)c1 N1(C(c2c(C)ncn2C)=O)CC2(CC2)CC1CNC(=O)C(C)Cn1ccnc1 c1(C(N2CCC(CN=[N+]=[N-])C2)C(=O)NCC(=C)C)cc2ccnc(Cl)c2s1 C1(C(=O)NC2C(CCC)C2)CCCN(C(=O)Nc2csc(Br)c2)CC1 c1(C(=O)NC(C)CC(C)NC(=O)COC2CCC2)cc(O)cc(=O)o1 C1(C(=O)NC(c2ccnn2C)C)C2CCN(C(C3COCCC3C)=O)CC12 N1(C(C(C)=CC2CC2)=O)CC(C2CC2C(N2CC(C(C)C)C2)=O)C1 Cc1c(C(=O)NCC(C)CNC(C2COC(=O)O2)=O)ccc2ccccc12 CCC(C(=O)NC1CC(NC(=O)CN(C)C2CC2)C1)C(F)(F)F Cc1sc(O)nc1C(=O)N(C1CCN(C(=O)C2=CSCS2)CC1)CC1CC1 C1(CC(=O)NC2(C(=O)NCC(c3cccs3)C)CC2(C)C)CC2CCC2C1 CCC(CCOC)C(=O)NCC1CC(NC(C23CC4CC2C3C4)=O)CCO1 C1(C(=O)NC)CCCNC1=O.CC1C(=O)N(CCO)CCCS1.n1(C2CC2)ccnn1 c1(C(=O)NCC(CN(C(c2csc(O)n2)=O)CC)(C)C)cc2n(n1)CCCC2=O c1(SC)ccc(NCC(=O)N(C)CCOCCN(C)C)nc1 N1(C(c2c(CC)sc(=N)[nH]2)=O)CCC2CCCN(C(=O)C=C3CCCC3)C2C1 C1(C)(CC)CCCN(C(=O)CC2CCCCC2NC(=O)Cn2cc(Cl)cn2)CC1 CC(C(=O)N(CCCN(c1ncnc2c1CCO2)C)C)C(C)S(C)(=O)=O c1(C(=O)NC)cccc(C(=O)NCc2[nH]nc(NC(C(C)C)=O)n2)c1.C1(C)(CCN)CC1 Cc1c(C(N2CCCC(C(C)NC(c3ncc(Cl)n3C)=O)C2)=O)cccc1Cl C=CCC(CC)N=c1[nH]c(N2CCOC(CC)C2)nc2ccc(OC)cc12 c1(OC)c(C(=O)N(CCC(C)NC(=O)C2=CCOC2)C)cccc1Br N1(C(c2ccc(COC)o2)=O)CCSCC1C(=O)NC(c1ccc(C)s1)C C12(O)CCCN(C1)C2=O.C(=O)(C1=NOCC1)NC(=O)NC1(c2ccncc2)CC1 c1(CC(=O)OCc2nnc(C(=O)OCC)s2)csc2cccc(F)c12 C=CC1CN(C(=O)CCn2ncn(C)c2=O)CC1NC(C12CC(C(C)C)(C1)C2)=O C1(C)(C(=O)NC(COC)CCO)CCCN(C(=O)CN=[N+]=[N-])C1 CN1CCC2CC(NS(=O)(=O)c3ccn(C4CCCC4)n3)CCC12 c1(NC(CCNC(=O)CC2(O)CCC2)C)ncnc2[nH]c3ccccc3c12 C(=O)(CCC(N)=O)NC(CNC(CC=CC(C)(C)C)=O)C1CC1 c1(C(N2C(CNC(C3(C)CCSCC3)=O)CC2)=O)cc(C2CC2)cc(F)c1 C1(C(N(CC(CNC(c2cc(SC)oc2)=O)O)C)=O)CC(=O)N(C)C1 CCC(F)(F)C(C)(C)C(=O)NCC1CC(F)(CNC(=O)Cc2sc(C)nc2C)C1 CCCCC(CCCC)C(=O)NC1CN(C(c2cccc(F)c2Cl)=O)CC1C C1(C(C)(C)N(C)C)CCN(C(=O)Cn2cc(CO)nn2)C1.C12CCC(C1)CN2 C1(C(=O)NCC(C)N(C(c2cnco2)=O)CC)CCOCC12CCC2 Cc1cc(C)c(C(N2C(C(=O)NC(c3cnc[nH]3)C)CCC23CC3)=O)cn1 CCC(CC)C(C)C(=O)NC1CN(C(=O)CC2(C3CC3)CC2)CC1OC Cc1nnc(N2CCC(NC(=O)C3=NNC(C(F)(F)F)C3)C(C)C2)nc1C c1(NC(C(C)C)=O)ccc(Cl)c(C(=O)N(C)CCN(C(=O)C(C)CF)C)c1 C1(NC(=O)NC(COC)C)C2C=CC(C2)C1c1ccccc1 c1(CCC(=O)NC2CN(C(=O)C(O)C3CC3)C2)cccc(Br)c1 CC(C)CCC(=O)NCC(N1CCCC1CCNC(=O)CC1CC2(CC2)C1)=O C1(NCc2ccc(SC)o2)CCCCC1N(C)C c1(CC)nn(C)cc1C(=O)N(C1CCN(C(=O)Cc2cncn2C)C1)CCO N1(C(CCN(C(=O)CCC2CCCOC2)C2CC2)=O)CC2(CCC1CO)CC2 c1(C(N2C(CN(C(COC)=O)C)CCC2)=O)cccc(-n2c(C)cnc2O)c1 C(=O)(CCC(=O)NCC1C(C)CCN1C(c1cnc(C(C)C)nc1C)=O)NCC C12(C(N(C3CCN(C(C4(F)CCCC4)=O)CC3O)C)=O)C3C4C1C1C2C3C41CO c1(NC(C2C(NC(c3scc(COC)n3)=O)C2)=O)cc(C(N)=O)cc(C)c1 Cc1cc(F)c(CC(=O)N(CCC(C)NC(C2CCC23CCC3)=O)C)cc1F C(=O)(C(C)(CNC(C1CCCCO1)=O)CC)NCCC=CC=C C(=O)(CCC(=O)NC1CC1)NC(C1CCN(C(c2n(CC)ccc2)=O)C1)C C#Cc1ccccc1CC(N1CCOC(C)(CNC(=O)Cc2ccsc2C)C1)=O Cc1cc(C(=O)NCC(C2CC2)NC(=O)CCSCC(C)C)ncc1C#N C1(NC(C2(Cl)CC2)=O)CCCCC12CCN(C(C1CC1(F)F)=O)C2 C(C(C(=O)NCc1ccc(OCC)cc1)NCCC1CC1)(C1CC1)OC N1(C(CCOCCC)=O)CCCC1CNC(=O)C=CCOC C1(NC(c2cc(CC)on2)=O)CCN(C(C2COC2)=O)CCC1c1ccccc1 C=C(C)CC(C)C(=O)N1CC(CC)(NC(=O)CCN2C(=O)CCC2=O)C1 N1(NC(C23N(C(C4CN(C(N)=O)C4)=O)CCC2C3)=O)CCOC2(CCCC2)C1 C1(CCC(N2CC(C)(CC(C)C)C2)=O)(NC(=O)COCC2CC2)CCCCC1 N1(C(c2ccc(OC)o2)=O)CCC2(C=C(C(=O)N(C)CCOC(C)=O)C2)C1 N1(C(CCc2cnn(C)n2)=O)CC2CC(C1)N(C(c1cc(Cl)nnc1O)=O)C2 c1(C(N2CCC(N(C(C3CCC(COC)C3)=O)C)C2)=O)cc(Cl)ccc1O C1(C)(C(=O)NCCN(C(=O)CCNC(C)=O)CC)CCOC1 C1(CNC(c2ccc(SC)s2)=O)CC2(CCN(C(=O)CC3(C)CCCCC3)C2)CO1 C(CC(C)C(=O)N(C1CCC(NC(=O)CCCc2ccc(C)s2)CC1)C)OC c1(OC)ccccc1C(N1CCC(C(=O)N(C)CCF)(CO)C1)=O Cc1nccc(Cl)c1C(=O)NC(CO)CCCNC(c1ccc(Cl)c(N)c1)=O c1(CC)ccc(Cl)c(C(=O)N(C)CCNC(c2ccc(C(C)(C)C)cc2N)=O)c1 c1(C(=O)NC(CCNC(CC2(C)CC2)=O)(C)C)cc(Br)cc([N+](=O)[O-])c1 C1(NC(c2ccccn2)=O)CCN(C(=O)Cc2ccsc2)C1 c1(C(N2CC(COC)N(C(c3cnns3)=O)CC2)=O)c[nH]c2ccc(O)cc12 N1(C(CNC(C(C)=C(C)C)=O)=O)CCC(N(C(=O)C(C)CF)CCCCO)CC1 C(=O)(CCCC(=O)NCCC1CCC(NC(=O)COC2CC2(F)F)C1)OC c1(CN2CCC(c3cccc(C(=O)OC)c3)(F)C2)cccc2cn(C(C)C)nc12 Cc1ccc(NC(=O)C(O)CNC(=O)C(C)(C)F)c(F)c1 Cn1cc(Br)c2c(CNCCc3c[nH]c4cc(F)c(Cl)cc34)ncnc12 N1(C(CCCN(C(=O)C(C2CCCCC2)O)C)=O)CCC2C(=O)NCC2C1 C=CCN=C(NCC1CCN1C1CCCC1)N1CCC(NC(=O)C(C)C)C1 N1(C(C(C)(F)F)=O)CC(NC(C2(Cc3ccc(F)cc3)CC2)=O)C2CC2C1 C1(NC(C2(C)CCSCC2)=O)CN(C(=O)C=Cc2cscn2)CCC1F C#CC1(O)CC(C(=O)NC(C)CC2CCN(C(=O)CSC)CC2)C1 C=CCCCCCC(=O)N1CCC(NC(=O)COC(F)(F)F)C(CO)CC1 C1(NC(C2C(C)OCCC2)=O)CN(C(c2ccc(=O)oc2)=O)CC2CCCC12 C1(CCC(=O)NCC(CN(C(=O)C(F)(F)c2ccncc2)C)O)CCCCC1 c1(NC(C2SCCN(C(C(C)(C)c3ccccc3)=O)C2)=O)ccc(C#N)c(O)c1 N1(C(C2C(C)=CCS2)=O)CCCC(C(C)C(=O)Nc2cnn(C(C)C)c2C)C1 N1(C(c2cn(C(CC)C)nc2)C(=O)NCc2ccco2)CCC(C)C(F)(F)C1 C1(CC(=O)N(C(CNC(COCCC=C)=O)C)C)COCCO1 N1(C(C2(C)N(C(C=C3CCC(C)CC3)=O)CC(O)C2)=O)CCn2c(O)nnc2C1 C(=O)(C1CCc2cccnc21)N1CC(NC(c2c(C)ccnc2C)=O)CC1(C)C c1(C(N2CCC(NC(=O)C=CC3CCC3)(CF)C2)=O)ccnn(C2CC2)c1=O c1(C(=O)OCCCOCCCC)nc(C2(C)CC2)n[nH]1 Cc1cocc1C(=O)N(CCC(=O)NCCC12CCCC1C2)CCO c1(NC(c2c(OC)ccc(F)c2)C)nccc(=NCCCS(C)(=O)=O)[nH]1 N1(C(C(CC)C#N)=O)CCCC(CO)(CNC(c2coc(C)n2)=O)C1 c1(CC)ccc(C(=O)N(C2CN(C(C3(N(C)C)CCC3)=O)CC2F)C)c(CC)c1 C=C1CC2(C1)CC(C(N1CCC(NC(c3ncoc3C(C)C)=O)C(C)C1)=O)C2 c1(N2CCN(C(=O)NC3CCC(C#C)CC3)CC2)[nH]cc(C)c(=O)c1C C(=O)(C(CC)C(F)(F)F)NC(CC)CNC(c1ccc(C(N)=O)c(Cl)c1)=O C(=O)(CC(C)(O)C(F)(F)F)NCCCCNC(C(CC)n1cncn1)=O N1(C(Cc2nc(C)on2)=O)CCC(O)C(C(=O)Nc2ccc(Br)c(Br)c2)C1 C1(CC(=O)NC(C(C)NC(C2(N3CCOCC3)CCC2)=O)C)CCC2(CCC2)O1 N1(C(C2C(=C)C2)=O)CCC2(C(=O)Nc3c(C)ccc(O)c3C)CCCC12 c1(CCC(=O)NCC2CCCCC2NC(c2cnco2)=O)ccc2[nH]ccc2c1 N1(C(CCOCCCOC)=O)CCN(C(=O)C(O)C(C)c2cccs2)C(C)C1 N(C1COc2ccc(F)cc21)C(c1ccc(Cl)cc1-n1cccc1)=O Cc1cc(C(=O)NNC(=O)c2cccc(C(F)F)c2)sc1C Cc1c(C(N2CCC3C(NC(=O)CCOc4ccccc4)C3C2)=O)cccc1F c1(C(=O)OCC)ncc(NC(=O)C(N2CCOC(C3CC3)C2)=O)cn1 CC1(C(N2C3CCC2CC3)C(=O)NCc2cnn3c2CCC3)CC2(CCC2)C1 Cc1nc(N2CCCC(CCNC(C3CC(C4CC4)=NO3)=O)C2)c2ccsc2n1 CC1CCCC(CC(N2CCC(C)(CCNC(c3cc(O)cs3)=O)C2)=O)O1 c1(NC(C2CCCC3(CCCCC3)O2)=O)ccc2nc(Cl)cnc2c1 CC(CC(C)(F)F)C(=O)N1CC(CNC(c2csc(C(C)(F)F)n2)=O)C1 O=C1CC(NC(=O)CC2CCCCC2NC(=O)C(F)F)CC(=O)N1 c1(C(N2C(CNC(c3cc(C)sc3)=O)CCC(C)C2)=O)cccc2oc(C)cc12 N1(C(C(CC)OC2CCCC2)=O)CC2CC2(NC(c2cnc(C)nc2)=O)C1 C1(CNC(=O)C(F)C2CCC2)CC2(CC2)CN1C(=O)C(C1CCCCC1)F C1(CCNC(c2c(C)cc[nH]2)=O)CCN(C(c2cc(Br)co2)=O)C(C)C1 CC(C)(C(=O)N(CCC(=O)Nc1cccc(C2CC2CO)c1)CCCO)C(N)=O N1(C(c2cnns2)=O)CCC2CC12C(N1CC(CC(F)F)C1)=O C1(C(=O)NC(CSC)C)(CNC(=O)Cn2nc(C)oc2=O)CC2(CC2)C1 C1(C(=O)NC2(CCNC(=O)CSc3ccccc3)CC2)CCC(C2CC2)O1 C(=O)(CCCCC(=O)N1CC(NC(=O)C(F)CC2CCCC2)C(O)C1)OC c1(C2(CNC(=O)OC(C)(C)C)CCC2)ccc(Br)cc1.C12CC1CN2C c1ccc(SC(F)F)cc1.C(CC(CNC(=O)CC)NC(=O)CN1CC=CC1)OC C1(N(C(C(CC)C)=O)C)CCN(C(c2cccc(F)c2)=O)CC1 N1(CCCC)CCCCC1C(=O)NC1CC(CNC(=O)Cc2nc(C)cs2)C1 N1(C(C(N(C(=O)CN2CCCCCC2)C)C2CC2)=O)CC2CCC(O)C2C1 c1(C(=O)NCC(CC)(CC)NC(c2cncc(OC)n2)=O)scc2c1CCCC2 C1(NC(c2c(C(C)C)ocn2)=O)CCCCC1N(C(=O)CCc1n[nH]c(=N)s1)C C1(O)(C(=O)NC2CN(C(c3cc(CC)sn3)=O)C(C)C2)CCC(C)(C)CC1 O(N=C1CCCCCC1)Cc1cn(C(C(C)C)NC(C2CC2C(N)=O)=O)nn1 CN1C(=O)OC2CN(C(C3CCCC3NC(C3(C#N)CCCO3)=O)=O)CC12 C1(NC(c2c(C)c[nH]c2)=O)C2CC1N(C(C1(C)CCCCO1)=O)C2C N1(C(CN2CC(C)C2)=O)C2CCC1C(NC(=O)CCF)C2 c1(OCCOC)ccc2cc(NCC(N3CCCCCC3=O)C)ccc2c1 C(c1cc(C)no1)=CC(N1CC(C(=O)NC(CC)C)(SC)C1)=O C1(CC(=O)NCCn2ncc(Br)n2)COCCN1C(C1CC=CCO1)=O C1(C(=O)NCC2(CO)CC2)CCC(c2cn(Cc3ncoc3C3CCC3)nn2)CC1 c1(C(=O)NC2CC(CCNC(c3c(=N)cc[nH]c3)=O)C2)cc(C(F)F)ccc1F N1(C(c2nccc(N(C)C)c2)=O)CC2CCC2(CNC(c2ccccc2Cl)=O)C1 N1(C(c2cn(CC)nc2)=O)CC2CN(C(c3n[nH]cc3Br)=O)CC(F)(F)C2C1 C1(OC)(CNC(c2ocnc2C2CC2)=O)CCN(C(=O)C(F)C2CCOC2)CC1 C#Cc1ccc(C(=O)N(CC(C)CNC(c2cnn(C)c2)=O)C)nc1 N1(C(=O)NCc2n[nH]c3c2COC3)CCc2nnnn2CC1 C1(C(=O)OCC)CC(C)N(C(=O)Nc2ncc(N(C)C(C)=O)s2)C1 CC1C2CC(CO)(C2)N1C(C1(c2ccccc2)COCCO1)=O C(CCCCC(=O)N1CC(O)(CCNC(=O)CCCNS(C)(=O)=O)C1)SC CP1(=O)CC(NC(=O)COCCOCc2ccccc2)C(O)C1 Cc1c(C(=O)NC2CCC2NC(C2(C#N)CC(C)C2)=O)sc2cncn12 c1(C(=O)NCC2(CN(C)C(C3CCC(=O)N3)=O)CC2)cscc1C#N c1(C(N2CC(O)(C(C)NC(=O)Cn3cccc3)C2)=O)cc2ccccc2o1 C(=O)(C(O)CC(F)(F)F)NCCOCCN(C)C(c1ccc(N2CCC2)cc1)=O C(=O)(C1CCC(=O)c2cccn21)N1CCC(F)(CNC(=O)Cc2csnn2)C1 c1(NC(C2C3N(C(CC(C=C)(C)O)=O)C(CC3)C2)=O)ccc2nn[nH]c2c1 c1(C(=O)NCC2C(CC(=O)N(CCOC(C)=O)C)C2)cc(=O)n(C)cn1 N1(C(C(C)OCc2ccc(C)cc2)=O)CCCCC(NC(=O)CS(N)(=O)=O)C1 C1(C(=O)NC(C)CCCNC(=O)CSc2nc[nH]n2)Oc2ccccc2C1C CC1CCC(CC(=O)NC(C)C(CO)NC(=O)Cc2ccon2)CC1 CC1NC(=O)C2=C1N(c1cccc(F)c1F)C(=S)NC2c1cc(I)n(C)n1 N1(C(c2cc(C(=O)OC)oc2C)=O)C2CC3C4CC(C3C2O)C1C4O C1(NC(c2nc(C(C)OC)sc2)=O)CC(NC(C2CCCC(=O)C2)=O)C(O)C1 C1(=CC(=O)N(C2CC(C(=O)NCCOCC#C)C2)C)CCCCC1 C(C1=NOC2COCC12)NC(N(C1OCCC1(C)C)CC(C)C)=O c1(OC)ccc(CC(=O)N(CCNC(C2COCCOC2)=O)C(C)C)c(C)c1 c1(C(N(CC(C)(C)C)CC)=O)cc(CNC(=O)C(O)C2CCCC2)nn1C c1(CC(=O)NCC(CC)(C)NC(C2CCCCCN2C)=O)cccc(F)c1F c1(C(N2CC(C)C(NC(c3cc(O)cc(O)n3)=O)C2)=O)cccc(Cl)c1Cl c1(OC)cccc(C(=O)NCC2(C)N(C(C3C(C(C)OC)C3)=O)CC=C2)n1 c1(C(=O)NC(C(C)C)CO)ccc(OCCN(C)C)cc1 CC1(C)COC(CC(=O)NCC2CCN(C(=O)CC3(C)CC(F)(F)C3)C2)C1 CCCC(C(N)=O)NC(=O)C(C)(C)CNC(=O)C(C)CN(C)C C1(C(=O)NOCC(O)CO)CC(O)CN1C(=O)Cn1ccnc1 C1(C)(C(=O)Nc2ccc(Cn3cc(C4(C(=O)NC)CC4)nn3)o2)CCCN1C.COC C1(NC(c2cn(CC)nc2)=O)CCOCC1C(=O)NCC(F)(F)C(C)C N1(C(c2nc(OC)c(C)s2)=O)CC(C)CN(C(C2CC(OC)C2)=O)CC1C c1(C(=O)NC2C=CCN(C(C=C(C)C(C)C)=O)C2)cc(C)c(C)nc1C c1(C(=O)NCC#N)ccc2c(c1)CCN(C(c1cnc(O)c(Cl)c1)=O)C2 N1(C(C2CCCN(CC)C2)=O)CC(C(=O)NCC2(C)CC3CC3C2)C(C2CC2)C1 N1(C(C(=Cc2cn(C)nc2)F)=O)CCCC2(CCN(C(c3nocc3Cl)=O)C2)C1 C(=O)(C1CCOc2ccccc21)N1C(NC(CCN(CC)CC)=O)CCC1 CN1CCC(C(=O)NCC2CCN(C(c3ccc(O)c(Cl)n3)=O)CC2)CC1=O C(C)(C)(CCC(=O)NCC(CO)NC(C1C2CCC1CC2)=O)N(C)C Cc1nc(O)nc(O)c1CC(=O)NCCOCCN(c1ccco1)C C=CC(C)(CC)C(=O)N1CC(CNC(=O)CCC(=O)N(C)C)C2(CC2)C1 CCCN=C(NCC1CSCCS1)N1CCC(c2nc3ccccc3[nH]2)CC1 C1(NC(C2CCC(C)CC2)=O)C2CC1N(C(=O)CN1CCSCC1)C2C c1(CC)ccc(C(=O)NC(C2CN(C(=O)CCN3CCCC3=O)CCO2)C)nc1 C(=O)(C(C)(C)NC(=O)Cc1cnsc1)NC(CC=CC)C c1(C(=O)NCC2N(C(Cc3cncc(C)c3)=O)CC2)cc(C)ncc1C C1(S(C)(=O)=O)(C(=O)NCC2CCN(C(CCCOCC=C)=O)CC2C)CCCC1 C1(NC(C2(CC=C)CCOC2)=O)COCCN(C(C2(CC3CCC3)CC2)=O)C1 C1(C(N(C(CN(C(COCCSC)=O)C)C)C)=O)CCCC(F)(F)C1 C(=O)(C1=CCC(C)(C)CC1)NC1(C)CC(NC(c2ccc(C)cc2C2CC2)=O)C1 N1(c2nnc(C(=O)OC)s2)CCC(C2(NC(=O)CCC(F)F)CC2)CC1 Cc1cn2c(n1)CC(C(N1CC(N(C(=O)CCC(C)(F)F)C)C(C)(C)C1)=O)CC2 C=Cn1nncc1C(=O)NCCNC(c1ncc(OC)cn1)=O C#CCC(CC(F)F)C(=O)N1CC2(CCC(CNC(C3CC34CCC4)=O)O2)C1 N1(C(c2cccnc2O)=O)CC2OCCN(C(=O)CCC3CCOC3)C2C1 CC(C1CC1)=CC(=O)NC1(CNC(=O)CNC=O)CC1 c1(OCC)nc(N2CCC(CNC(c3cc(Cl)n(C)n3)=O)C(C)C2)ncc1Cl c1(NC(c2ccc([Si](C)(C)C)cc2)=O)ncc2c(n1)CCCC2=NO C1(O)(CN(C(c2ncn(CC)c2)=O)C)CCCN(C(=O)C(C)NS(C)(=O)=O)C1 Cc1[nH]nc(C(N2CC3CC3(CNC(=O)CC3CCC3)C2)=O)c1[N+](=O)[O-] N1(C(c2ccc3cc(C)sc3c2)=O)CCCC2(CC(NC(=O)CSN)CO2)C1.CC=C(C)C N1(CCCC)CCN(C(C2CC=CCN2C(C2CCN2CC)=O)=O)CC1 c1(C(=O)NCC2(CNC(=O)C(C3CCOCC3)O)CC2)c(O)ccc(Cl)c1F CCC(O)C(C)(C)C(=O)N1CCC(CO)C(NC(=O)Cc2c(F)cccc2F)C1 N1(C(c2cnc(CC)nc2)=O)CC2COCC2(C(=O)NCCc2ccccc2)C1 C1(F)(C(=O)NCCC(C)(O)C2CC2)CCCN(C(=O)CCc2cnoc2)C1 C1(CNC(c2cncc(CNC(C(CCC)O)=O)c2)=O)CC2(CCO1)CC2 n1(CC)nc(C(=O)NC2CCC2NC(=O)Cn2nnc(=N)[nH]2)cc1O N1(C(CSCC#C)=O)CCC2(CC1)CN(C(C1(c3cccc(F)c3)CCC1)=O)C2 c1(OCC)cc(C(F)(F)F)ccc1-c1nc(C(=O)NCc2ccc(Cl)cc2F)cs1 c1(C(C(=O)NCC(C)NC(CC(c2ccc(C)cc2)C)=O)O)ccc(F)cc1F CCCC(CNC(c1ncccc1F)=O)C(=O)NCC1(n2nccn2)CC1 c1(C(=O)NC2CCC(NC(C(C3CCN(C)CC3)C)=O)CC2)ccc(N)cc1Cl c1(C(N2CC(NS(=O)(=O)C(F)(F)F)C(F)C2)=O)c(F)ccc2[nH]ccc12 C1(N(C(c2ccc(CCC)s2)C(=O)NCC(C)C)C)CCN(C2CC2)CC1 CC1=CCC(C)(C(=O)NCCC2CCN(C(c3cn4ccnc4s3)=O)C2)CC1 C1(N(C(=O)Cc2cn(C)nn2)C)CCCCN(C(=O)C(c2cnn(C)c2)O)C1 C#Cc1cc(C(=O)NCC2CCCN2C(C2CCCCCC2)=O)ccc1C c1(NC(C(C2CCN(C(C(C=C)OC)=O)C2)F)=O)ccc(O)c(Cl)c1 C1(CNC(Cc2cnn(C)n2)=O)CCC2(CN(C(c3cc4sccc4[nH]3)=O)C2)O1 N1(C(C(C(CC)O)C)=O)CCC2CN(C(c3ccc(C(C)C)s3)=O)CC2CC1 c1(C(N(CCNC(=O)Cc2ccc(Cl)cn2)CC)=O)cc(Br)cnc1N c1(C(N(C)CCN(C)C(c2ccncn2)=O)=O)cc2ccnc(Cl)c2s1 N1(C(c2nccc(OC)c2)=O)C2CCC(C2)C1CC(=O)NCC1COCC1O C(=O)(CCC(=O)N1CCC(NC2CCC(NC(c3ccns3)=O)CC2)C1)NCC Cc1cc(C(N2CCCCC2CCNC(=O)C=Cc2cnc[nH]2)=O)ccc1Cl C1(C(N2CCC(OCCNC(C3CC(O)C3)=O)C2)=O)CCc2ccc(F)cc2O1 Cc1nn(CC(C)C)c(Cl)c1C1CCCN1C(c1ncnn1C)=O c1(C(N2CC(NC(CC3C(C)(C)C(O)C3)=O)(CO)C2)=O)ccc2nc(S)oc2c1 C1(NC(c2c(O)ncc(CC)c2)=O)CCN(C(=O)CC2(O)CCOC2)CC1(C)C c1(C(=O)NCC(C)(C)NC(Cc2c(C)nc(Cl)cc2)=O)cc2cccnn2c1 N1(C(C(CC)C(C)O)=O)CC2CCC1C(NC(=O)COCC(F)F)C2 C1(CCOC)(NC(=O)COCC(C)C)CCN(C(=O)C(CC)OC)CC1 C1(NC(c2noc(CC)c2C)=O)(CNC(=O)C(C)(C)CO)CCCCC1C c1(C(=O)NC(C)CC(=O)NCCC2CCOC2)nccnc1N c1(C(N2CCCC(NC(c3cc(C(C)=O)c(C)o3)=O)C2)=O)cnc2ccccn12 C(C(=O)NCC)(n1ccnn1)NC(C1CC1C(=O)OC(=O)COC1CC1(F)F)=O C1(CC(=O)NC(CC#C)(C)C)CN(C(C2(C)CCOCC2)=O)CCO1 C(CCCN=c1ccn2ncc(S(=O)(=O)NC3CCC=CCC3)c2[nH]1)OCC N1(Cc2ccccc2)CCNCC12CCOC2.C(c1ccccc1)=CCCC(=O)N c1(CC(=O)NC(CN(C(CC=C=C)=O)C)C)ccc(-c2nnco2)cc1 N1(C(c2c(C)ccn2C)=O)CC2CC(C1)CN(C(=O)CCCCCCN=[N+]=[N-])C2 C1(C)(CNC(C(c2cnn(C)c2)C)=O)CCCN(C(C2CC=CC2)=O)C1 C1(CCC(N2C(COC)CC2)=O)CCC(NC(c2scnc2C)=O)C1 N1(CC)CCOCC1C(=O)NCCCCC(=O)NC(C(C)(C)O)C1CC1 N1(C(C)C)CC(C(=O)NC2CCC(C)N(C(c3c(Cl)nsc3Cl)=O)C2)CCC1=O c1(CNC2(C(CC)=O)CC2)c(F)cccc1Br.C12(CCCC1)CC(=O)N2 CCCCCCn1nnnc1C(C)(CCNCC1CC1(C)CC)OC c1(C(N(C2CCCN(C(C3CCN(CC)C3)=O)C2)C)=O)cccc2nc(O)oc12 N1(C(C(=O)NC(C)C)=O)CC2CC2(C(=O)NCC(C)(C)C2CCOC2)C1 C(CC(=O)NCC1CCN1C(=O)Cc1sccc1C(C)=O)(C1=CCCC1)OCC c1(C(=O)NCC#CCNC(C2(C=C)CCC2)=O)cc2cnccc2cc1F N1(C(COCCC#C)=O)CC(C)(C(N2CC(F)(CF)C2)=O)C1 C(=O)(C(O)C(C)(C)C)NCC1N(C(c2cnc(C(C)(C)C)[nH]2)=O)CC1 Cc1ccc(F)cc1C(N1CC(NC(=O)C(C)CC(N)=O)CC1(C)C)=O C(=O)(C#Cc1ccc(Cl)cc1)N1C(CN(C(c2ccc(Cl)cc2)C)C)CCC1 C1(C(N(C2CCN(C)CC2)C)=O)CC2(C1)CN(C(C1CCOC1C1CC1)=O)C2 c1(C(C)C)c[nH]nc1C(=O)NCC1CCCC1NC(=O)CNC(c1cscn1)=O c1(C(=O)NCC2C(C(=O)NC(C=C)COC)C2)ccc(COC)cc1 CC(C(CCc1ccccc1)NC(=O)C(F)F)NC(=O)CS(N)(=O)=O N1(C(c2nn(CC)c(C)c2)=O)CCC(F)(C(=O)N(C)CC2(O)CCCCC2)CC1 C(=O)(C1=CCN(C(C23CCCCC2C3)=O)C1)NC(c1ccncc1F)C C#Cc1cnc(C(N2CCSCC2C2CCC2)=O)c(C)c1.C(CO)(N)C1CC1 C#Cc1ccc(C(=O)NC2(CO)CN(C(c3ccc(CN(C)CC)cc3)=O)C2)o1 c1(CNC(C(CC)NC(=O)C(C(=O)OC)OC)=O)cccc(C#N)n1 C(=O)(CC(C(C)OC)NC(C1CC(=C2CC2)C1)=O)N1CCCC(CC)C1 C=CCC(CCC=C)NC(=O)CC12CCC1CN(C(=O)C=C1CCCCC1)C2 C(=O)(C1CCCc2ccnn21)NCC1=CCN(C(C(COCC)C)=O)CC1 CCCC(C(=O)NC1(CCO)CN(C(c2cc(SC)n(C)n2)=O)C1)NC(N)=O C(C(C(=O)Nc1ccc(O)c(CO)c1)C(C)(C)C)NC(CCNC(COC)=O)=O C1(NC(=O)CN2CCCNC2=O)(CNC(=O)COCCF)CC2CCC1C2 C(=O)(CCC(C)(C)C#N)N1CCC(OCCNC(CN(C)C(N)=O)=O)C1 c1(C(C(=O)NCC(C)C)N(C)Cc2nnc(C)n2C)cnc2ccnn2c1 CCC(CC(=O)NCC=CCNC(c1cnn2c1N(C)CC2)=O)CC(F)(F)F C1(CC(=O)NC(CNC(Cn2c(C)ccn2)=O)C(C)C)CCCCN1C c1(C(N(C(C)CCNC(C2CC(=O)CC(=O)N2)=O)C)=O)cc2cccnc2s1 C1(C(=O)NCC23CC(CNC(C4CC5CCC4O5)=O)(OC2)C3)CCC2(CCC2)C1 CC1(C(N2CCC(C(F)C(=O)NCc3ncccc3F)C2)=O)CC(F)(F)C1 c1(CCC)nsc(N(C)CCOC2CN(C(c3cnc(C)[nH]3)=O)C2)n1 N1(C(c2cccc(C#C)c2F)C(=O)NCCC)CCc2ccc(C#N)cc21 c1(C(=O)NCCCCCN(C(=O)COCCF)C)cccc(C=C(F)F)c1 N1(C(C(C)c2ccco2)=O)CCC(C2CC2)(CNC(c2cc(Br)co2)=O)C1 c1(C(N(C)CN(C(C(=O)C2C(CCC)C2)C)C(c2ccoc2)=O)=O)n[nH]cc1Br Cc1ccc(NC(c2ccc(CNC(=O)CCC(C)(F)F)nc2)=O)cc1O C=C1CC(C(=O)NCC(c2ccsc2)C)(CNC(c2cc[nH]n2)=O)C1 Brc1cccc(COc2nnc(N3CCCC(CO)C3)s2)c1.C1(C)CCC1 C1(NC(c2nc(OCC)oc2)=O)CCCN(C(c2conc2C(C)(C)C)=O)C1C c1(OC(C(=O)NCCCCn2cc(CC(=O)NCC)nn2)C)ccc(F)cc1 C1(C(N(C)C2CC2)=O)CCN(C(=O)Cc2cnsc2)CCO1 C(=O)(C(C)CCNC(c1ccccc1)C1CCCCC1)OC C1(NC(=O)CSc2nnc(S)s2)CN(C(c2cccnc2O)=O)CC1O N1(C(CC(C(C)C)(F)F)=O)CCCC(C2CCN(C(=O)CC3CCC(=O)C3)C2)C1 c12oc(cc1C)C(=O)Nc1cn(C)c(n1)C(=O)NC1(CC1)C(=O)C2=O.CCO.CC C(=O)(C(C(F)(F)F)(C1CC1)NC(=O)C(C)=C1CCC1)OCC c1(C(C)N(C(C)CCNC(c2c[nH]nc2C(F)F)=O)C)ccc(F)cc1F C(=O)(Nn1cnc2ccccc12)C1(C)CC(NC(=O)CC2CC3CC3C2)C1 CC(C)(CNC(=O)Cc1cccnc1F)CCNC(=O)Cn1nccn1 c1(C(N(C2CCN(C(CC(C)(C)SC)=O)CC2)C)=O)cc2sccc2cn1 N1(C(CC=C(C)C)=O)CCC2(CCOC2)C(CNC(=O)CCc2ccsc2Cl)C1 c1(C(N2C(CNC(C(C)Oc3c(C)cccc3)=O)CCC2)=O)cnc(Cl)cc1Cl c1(N2CCC(N(C(c3ccc(CC)cn3)=O)CC)C2)nc(C#N)c(Cl)s1 c1(CC(=O)NCC(C)NC(C2CCCC(=O)O2)=O)cc(C2CC2)nn1C C=C(C)CC(C(=O)N1CCC(CCO)C1)NC(=O)CN=[N+]=[N-] Cc1nccc(COC(C2(NC(=O)OC(C)(C)C)CCN(C)C2)=O)n1 CCCC(C)(O)CC(=O)NC(CNC(c1cnc(O)cc1C)=O)C(C)C C12(CNC(C(CC)COC)=O)CN(C(=O)CC3(NC(C)=O)CC3)C(CO)(C1)C2 C1(N(C(=O)C=C2CC2)CC)CCCN(C(c2cnc(C(C)C)n2C)=O)CC1 c1(C(N(C)CC2(O)CCN(C(=O)CNC(N)=O)C2)=O)cc([N+](=O)[O-])c[nH]1 CC1CC(C(=O)NCC2(CCOC(c3ccc(OC(C)C)nc3)=O)CC2)=NO1 C(C(C)(C)CC(=O)N1CCC(CN(C(c2csc(O)n2)=O)C2CC2)CC1)N(C)C c1(CC)nc(C)c(C(=O)NCCCN(C(c2cncn2C)=O)CC)s1 C1(NC(C2CC(OC)(OC)C2)=O)CC2(NC(=O)C=CBr)COC1C2 N1(C(=O)NCCCN(c2n[nH]c(C)c2Cl)CC)CCCC(C)C1 C(CCCCC(=O)NCC(O)CO)N(C(C(C)c1cncs1)=O)C1CC1 c1(OC)cc(C(=O)NCC(C(C)C)NC(C2(C)CCCCCC2)=O)ccc1C C1(C(=O)NCC2C(C)CN(C(=O)CC3CCC(C)C3)CC2)CCC2CCCCN12 C1(NC(C2CC(N(C)CC)C2)=O)CCCCCN(C(=O)CC2CC3C=CC2C3)C1 C1(C(N2CC(NC(C=Cc3c(C)ccnc3)=O)C2)=O)CCC2C(CC1)C2(F)F C1(C(C)C)CCC(C(=O)NC2CCC2CNC(=O)C=C2CCN(C)C2)C(=O)N1 C1(O)(CNC(=O)CSc2cccc(Cl)c2)CCN(C(=O)CCc2ccc[nH]2)CC1 c1(OCC)ccc2c(c1)CCC(NC(=O)NCc1cc(O)ccn1)C(=O)N2.OCC Cc1ccc(-n2cc(C3CCC(NC(C4COC(=O)C4C)=O)CC3)nn2)cc1 c1(C(=O)NC2C(NC(=O)Cc3ccc(Cl)s3)CC2)ccc(F)c(Cl)c1F C(=O)(C1=CCCC1)NCC(C1CCC1)NC(c1c(C(C)C)[nH]nc1)=O C1(C(N(C2CCOC(C)(C)C2)C)=O)CCC2(CC2)N1C(C12CCCC1C2)=O C1(C)(CNC(c2c(NC)nn(C)c2)=O)CCCN(Cc2cc(C(=O)OC)sc2)C1 c1(CCOCC2CC(CNC(COC(c3nnc(C)s3)=O)=O)C2)nc2ccccc2o1 c1(C(N2CCC(NC(C(C)OCCOC)=O)C2C(C)C)=O)cc(C)ccc1F c1(OC)ccc(C(=O)O)cc1CNCC1(Br)CCC(C(F)F)CC1 C(CNC(C1CC(N2CCCC2)C1)=O)(CC(F)(F)F)NC(COC(CC)C)=O c1(OCC)cc(C(=O)NC2CC(CNC(C3CC3(C)C(C)C)=O)C2)ccn1 Cc1c(C(=O)NCCCN(C)C(c2nn(C)cc2N)=O)nnn1-c1ccn(C)n1 C=CCC(CC(C)C)C(=O)N1CCC2(CC1)CC(NC(c1ccn(CC)n1)=O)C2 C12(NC(CCCn3c(C)ncc3)=O)CCC(NC(=O)C(F)C3CCOC3)(CC1)C2 C1(O)(CN(C(C(C)N(C(C)=O)C)=O)C)CCN(C(c2cc(C#N)c[nH]2)=O)C1 C(=O)(C(C)CC(C)C(C)=O)NC(CC#CC)C(=O)NC1CC(O)C1OC CCCCC(O)C(C)C(=O)NCC1(O)CCCN(C(c2cncc(C)c2C)=O)C1 C(c1cnc(O)nc1O)=CC(=O)Nc1ccc(N2CCN(CC)CC2)nc1 C12(CNC(C(CC)NC(C)=O)=O)CN(C(=O)CC(F)(F)Cl)CC1(C(F)(F)F)C2 N1(C(CC2CC(OC)C2)=O)CC2CCC(C1)N2C(C1(C2CCCCO2)CC1)=O c1(C2CCN(C(c3ccc(C(C)C)s3)C(=O)NC)C2)ccccc1C C1(C(=O)NC(C2(O)CCN(C(=O)CC3CCOCC3)CC2)C)CC2CCCCC12 C1(F)(CNC(C2C(=C)C2)=O)CCN(C(=O)CCc2ccccc2C)CC1 CN1CCN(C(c2cc[nH]c2C2CC2)=O)C(CNC(c2ccc(Cl)c(Cl)c2)=O)C1 O=C1CC(C(N2CCC2C(=O)NCC2CC23CC3)=O)NC1 N1(C(C(C)OCC=C)=O)CCN(C(=O)Cc2cccnc2)CC1CCC C1(O)(C(=O)NC2CC(C)(CNC(C3CC3F)=O)C2)CCCCCC1 c1(-c2cccc(OCC)c2C)cccc2[nH]nc(C(=O)NCC(N)=O)c12 CC1CN2CCC1CCCCC2=O.C(=O)(CC(C)(C)CBr)N(C)C C1(C(N2CC3N(C(C(CC(=O)OC)C)=O)C(CC3)C2)=O)CCc2ccccc2O1 c1(CC)ccccc1CC(=O)NC1CC1CNC(=O)C(c1ccc(F)cc1)C c1(NC)ncccc1C(=O)NC(CNC(=O)C(C1CCCCC1)C)CCOC C12(NC(C(C)NC(=O)NC)=O)CC(C1)N(C(c1c(C)n[nH]c1C)=O)C2 c1(CNC(=O)NC(CC#C)(C)C)cc(N(C)CC)ccn1 C(=O)(C(C(=O)NC1(CN(C(=O)CCC(N)=O)C2CCCC2)CC1)C1CC1)OCC c1(CO)cc(C(N2CC(CC(C)NC(c3c[nH]nc3Br)=O)C2)=O)no1 Cc1cc(C(N2CCC(NC(c3c(C)cncc3C)=O)C2)=O)cc(C)n1 c1(CC)ccccc1C(CNC(c1ccn(C2CC2)n1)=O)NC(c1[nH]cnc1C)=O N1(Cc2c(O)ccc(SCC)c2)CCN(C(C2(CC(C)C)CC2)=O)C(C#N)C1 C12(COC)CC(NC(C3CCCC3C)=O)(CN1C(=O)CCCC(=O)OC(C)(C)C)C2 N1(C(C2CN(C3COC3)C2)=O)CCCC(N(CCO)C(c2c[nH]nc2F)=O)C1 c1(CC(N2C(CNC(C3=C(C)OCC3)=O)CC(F)C2)=O)ccc2c(c1)COCC2 N1(C(C23CC(C)(C2)C3)=O)CCCC(CCNC(c2ccncc2F)=O)C1 c1(CC)cc(NC(C2CC2C2CN(C(c3cnsc3)=O)C2)=O)cc(O)c1 C(=O)(CCCNC(C1CSCCS1)=O)NC(c1cn[nH]c1)C N1(C(COCc2n(C)ccn2)=O)CC2CC(N(C)C(c3cnccc3Cl)=O)C1C2 N1(C(c2cccc(C(C)C)c2)=O)CCN(C(C2CCC2(C)C)=O)CC1CCO Cc1ccnc(O)c1C(=O)NCC1(O)CCN(C(C2CCCN(C)C2)=O)C1 CCCC(CC)CC(=O)NC1CN(C(c2ccc(CC)nc2)=O)CC1O c1(C(=O)NCC2(F)CCN(C(C3C=CCC3)=O)C2)cc(F)c(O)cc1Br c1(C(=O)NC(C(=O)NC(CC)CO)(C)C)cn(C)c(=O)n1C CCCCCCCC(=O)N1CCCC(CNC(=O)COc2ccsc2)C1 C#CC1CN(C(=O)C(F)C(C)(F)F)CCN1C(=O)CCCC(C)=O N1(C(Cc2nn(C)c(NC(C3CCC34CCCC4)=O)c2)=O)CC(CO)CC1(C)C c1(C(=O)NC2CN(C(C3N(C(C)=O)CCCCC3)=O)C2)cc2n(n1)CC1(CC1)C2 CCCC(COCc1nc(-c2ccccc2)no1)OCC C1(CC=C)(NC(c2sc(CC)nc2C)=O)CCN(C(=O)CC2CCN(C)C2)C1 N#CC1(C(=O)NC2CC(CNC(c3cn(CC4CC4)nn3)=O)C2)CCC1 C1(NC(C(CC)C)=O)CCN(C(c2csnc2C2CC2)=O)CC1CC CC1(C)CN(C(=O)CC2CCCOC2)CC1NC(c1csc(-c2ccsc2)n1)=O C(CCCCC(=O)NCCCSCC(=O)N1CCCO1)OC C1(N(C(Cc2c(OC)cccc2)=O)C)CCN(C(C2CC3CC3C2)=O)CC12CC2 C1(C(=O)NC(CC)CNC(=O)C(F)F)CCCCC1C(=O)OC(C)(C)C C(=O)(C(CNC(=O)CC1C=CCCC1)C(C)C)NCCc1cnc(C)s1 N1(C(C(CCC)CCC)=O)CCC2CCCC(C1)N2C(=O)Cc1cc(C)oc1C c1(NCc2ncc(-c3cn(COC)nc3C3CC3)[nH]2)ccc(Cl)c(F)c1 CCC(CC(=O)NC1COCCN(C(=O)Cc2ccccc2COC)C1)C(C)C Cc1nn(C2CC2)cc1C(=O)N(C)Cc1cccc(NC(C2CCO2)=O)c1 C(=O)(CCCCCC(C)O)NCC1N(C(Cc2c(CC)cccc2)=O)CC1 C(=O)(C(O)(CN(C)C)C(F)(F)F)NCC(C)NC(c1ccc(C(F)F)cc1F)=O c1(C(=O)NCC(CNC(C2C(COC)CC2)=O)F)c[nH]c(=O)c2ccnn12 N1(C(CC2CCC(OC(C(CC)OC3CCCCC3)=O)C2)=O)CCC(OC)CC1 c1(N(C)CC2N(C(CC(CCC)C)=O)CCC2)nc2cccc(C)c2o1 CC1(CNC(=O)Cc2cnns2)CCN(C(c2nccnc2C(N)=O)=O)C1 C1(NC(C(Cc2c(C)cccc2)C)=O)CCC(C)N(c2nccc(CC#N)n2)C1 N1(C(C=Cc2ccc(C)o2)=O)CC=C(C(=O)NCCC2C(=O)NN=C2C)C1 C(N=c1[nH]c(=NCCC(N)=O)c2cccc(F)c2[nH]1)c1ccc(=N)[nH]c1 c1(C(C)NC(C(=O)NC)C)ccc(OCCC(C)C)cc1 C#CCCCCCC(=O)N1CCC2CC2(NC(=O)COc2ccnc(Cl)n2)CC1 C1(C)(C(N(C2CCN(C(C3CC3c3ccccc3)=O)C2)C)=O)CC2(CCC2)C1 C(C(C(=O)N1CC(Cc2nnn(C)c2C(N)=O)C1)C(C)C)NC(CC1CC(=C)C1)=O C1(C(F)(F)F)(C(=O)NC(C)CN(C(=O)CC2CCOC2)C)CCCC1 c1(CC)ccccc1C(=O)NCc1cccc(CNC(c2cc(O)n(C)n2)=O)c1 N(C(=S)N1CCCC1)c1n(C)c(C2CCCN2CS(=O)(=O)c2cccs2)nn1 CC1(C)CC(C(=O)NCC2CN(C(c3cnn4c3CCC4)=O)CCO2)=NO1 c1(C(C(=O)NCC(CCOC)NC(=O)Cc2cscn2)C)cccc(C)c1 CC1CCN(C(=O)COc2ccsc2Cl)CCN1C(=O)C=Cc1ccoc1 C1(NC(CCCC#N)=O)CN(C(c2cncc(N)n2)=O)CCC1C(F)(F)F C1(NC(c2ccc3cnnn3c2)=O)CN(C(=O)C=CC2CC2)Cc2nccn2C1 c1(C(=O)NC(C(C)C)CNC(C2CC23CCOCC3)=O)cnc2ccoc2c1 c1(C(N2CC(C)C(NC(=O)CN3CCCC3=O)CC2)=O)cc(F)c(Br)cc1F C1(OC)(CNC(c2ccnnc2)=O)CCN(C(C2CC2(Br)Br)=O)C1 c1(OC)n[nH]cc1C(=O)NC1CC(C(=O)NCCCCF)C1 Cc1nc(N2CCCC2)ccc1NC(=O)NC(Cc1ccccc1)CCO CN1N=CC(CC(=O)NCCCC2CCCCN2C(c2ccsc2C#N)=O)C1=O Cc1noc(Cl)c1CCC(=O)NC(CNC(C1COCCO1)=O)C1CC1 C(=O)(CCCC(=O)N1CCN(C(=O)C(C)N2CCC2)C(CC)C1)NCC Cc1cc2c(C(N3CC=CC(NC(C4(C)CCCN4C)=O)C3)=O)ccc(C)c2[nH]1 N1(C(=O)CCOc2ccccc2)CCCC(C(=O)O)C1 C1(CNC(c2onc(OC)c2Br)=O)C2CN(C(=O)C(C)NC(C)=O)CC12 c1(C(=O)NC2C(CNC(COC(CC)(C)C)=O)CC2)cc(-c2cccnc2)no1 C1(NC(CCSC)=O)CN(C(c2cc(Cl)ncc2O)=O)CCC12CCC2 C12(C(=O)NCCC(C)N(C(CCC(=C)C)=O)C)CCCN1CC(OC)C2 c1(C(C2N(C(c3on(C)c(=O)c3)=O)CCC2)=O)ccc2c(c1)CCC2 Cc1oc(CNCCN(C)C)cc1C(=O)NC(C)Cc1csnn1 N1(CCC(=O)NCC2(CNC)CC2)CCOCC1.c1(C=O)csc(-c2ncc[nH]2)n1 C(=O)(C(C)C(O)C(C)CC)NC1C2CCN(C(c3ccc(C#C)cc3)=O)C21 C(=O)(C(C)CC(N)=O)NCC1C2CN(C(C3C(c4c(C)cccc4)C3)=O)C1C2 Cn1nc(C(F)(F)F)c(C(N)=O)c1C(=O)NC1CC(NC(=O)C2=CCCCO2)C1 C(CCCN=c1[nH]c(Cl)c(C#N)s1)NC(C(C)n1cncn1)=O O=C(C1Cc2ccccc21)NCC1CCCC(CNC(=O)CCc2ccc[nH]2)C1 C1(NC(c2ccc(CC)s2)=O)CC(O)CN(C(=O)C=C2CCC(C)CC2)C1 CCC(C(=O)N1CC2CC1C2NC(c1cnc(C)nc1)=O)C(C)C c1(C(C(=O)NC(C)CCNC(C2CC=CCC2)=O)CO)ccc(F)cc1 c1(C(N(C2CCCN(C(c3ccoc3)=O)CC2)C)=O)nc2c(Br)cccn2n1 CCCC(C)(O)CC(=O)NC(CC(N1CCCOC(C)(C)C1)=O)C(F)F N1(C(Cc2c(C)cnn2C)=O)CCC2(COC(CNC(=O)C(N)=O)C2)C1 N1(C(CC2(CNC(C)=O)CC2)=O)CCCC(NC(=O)CCCC(C)=O)C1C C1(CC=C)(C(=O)NCc2nc(CC)cs2)CN(C(=O)C(C)SCC)C1 C1(C(N2C(CNC(CN(CC)CC)=O)CC2)=O)CCc2c[nH]nc2C1 C1(COC)CN(C(c2cnsc2)=O)CCN1C(c1cc(N)ccc1O)=O Cc1c(CC(=O)NC(C)CNC(C2CC2c2ccccc2)=O)ccc(Cl)c1Cl Cc1cc2c(N(c3ncncc3C#N)C3CCCNCC3)ncnc2[nH]1 c1(CC)ccc(CN2CCC(O)C2C(=O)Nc2cc(C)c(Cl)cn2)c(F)c1 c1(OCc2cn(C(CNC(C3(CC(CC)C)CC3)=O)C)nn2)ccc(F)cc1 c1(NCC)cc(Cl)ccc1C(=O)NCC1CCN(C(=O)C(CC(C)C)N(C)C)C1 N1(C(CCSC)=O)CCN(C2CCCN(C(=O)C=C3CCC(C)C3)C2)C(=O)C1 C1(C)(OC)CC(NC(c2cc(CNC(=O)CCC3(C)N=N3)cs2)=O)C1(C)C N1(c2nnc(C(=O)Nc3cncc(OCC)c3)s2)CCC2(CCCCC2)C1 N1(C(C2(C=C)CC2)=O)CC2COCC(C1)C2NC(c1ccccc1OC(F)F)=O c1(CC)oc(C(=O)N(CC)CC2CCN(C(C3CC3CCOC)=O)CC2)cc1C C1(n2cccc2)(C(=O)NCC2C(NC(c3nc(CC)sc3)=O)C2)CCCCC1 C1(C(=O)NCC(CN(C(C(CC)CN(C)C)=O)C)O)CC2(C1)CC(O)C2 n1(CC#C)ccc2cc(NC(c3ccc(SCCCC)cc3)=O)ccc12 c1(-c2cncc(C)c2)nc2c(s1)CCN(Cc1cc(O)nc(Cl)c1)C2 c1(C(N2CC3(CC(NC(c4c(CC)scn4)=O)C3)C2)=O)ccc2ocnc2n1 C(=O)(C#CC(C)(C)CNC(=O)C(O)C(F)(F)F)N(CC(O)CF)CC Cc1[nH]nc(Cl)c1C(N1CCCC1CNC(=O)CC1COCCO1)=O Cc1c(F)ccc(N)c1C(=O)NC1CC(CCNC(c2ccccc2F)=O)C1 c1(NC(C2(C)CCN2C(c2ccc(F)nc2F)=O)=O)nc(O)c2nc[nH]c2n1 C(=O)(C#CC1(CC)COC1)N(C1CCN(C(C2CCC2(C)C)=O)C1)CC c1(C(N(CCNC(C(C2CCCO2)OC)=O)C)=O)ccoc1Br NS(=O)(=O)c1ccc(NC(C2CC(F)CN(C(C3CCCO3)=O)C2)=O)cc1 CC1(C)CCCC(O)(C(=O)NCC2CN(C(c3ccc[nH]3)=O)CCCO2)C1 N12CCC(CC1)C2.c1(C(=O)O)ncc(NC(c2n(C)ccn2)=O)n1C N1(C(CC(CC)C2CC2)=O)CCC2CN(C(c3c(C)ccnc3O)=O)CC2C1 C1(NC(C2C(COC)CC2)=O)COCC1CNC(C12CC(F)(C1)C2)=O c1(C(=O)NCC2OCCN(C(C=CC(C)C)=O)C2)c(F)c(F)c(F)c(F)c1F N1(C(C2COCCO2)=O)CCC2CC2(C(=O)NCCC#CCO)CC1 Cc1cc(F)c(C(=O)NC2CCCC(CNC(C34CC(C)C3C4)=O)C2)c(Br)c1 c1(C(=O)NCCC(C)NC(C(C)OCC#C)=O)cc(O)ccc1OC(F)F C(=O)(C(F)C(=O)NC(C1CC(NC(=O)C=C(C)C(C)(C)C)C1)C)OCC C1(NC(CC(CC)(F)F)=O)CCCC12CN(C(=O)C(C)CC(=O)N(C)C)C2 C1(NC(C2(OCCCCCCSCC)CCC2)=O)CC(O)(CNC(N)=O)C1.CO CCCC(O)C(=O)N1CCC(C2CCCN2C(c2ocnc2CC)=O)C1 N1(C(CC(=O)NC2CC2)=O)CC2(CC(NC(c3cc(Cl)c[nH]3)=O)CO2)C1 c1(NC2CCN(C(C#CC)=O)C2)ncc(C(=O)OC)cc1[N+](=O)[O-] C1(NC(CCS(C)=O)=O)CCC2(CC1)CC2NC(=O)Cc1coc(C(F)F)n1 C1(C(=O)NCC2CC(NC(CCNC(=O)OCC)=O)C2)C2CCOCC12 C(CCC(N)=O)(C(=O)OC(C1C(C23CC(CO2)C3)CCC1)=O)COC(C)(C)C Cc1cc(=NC(=O)C(C)N2CCn3ncc(C(=O)O)c3C2C)[nH]o1 c1(CCC(N2C(CNC(C(COC)O)=O)CC(OC)C2)=O)nc2ncccn2n1 c1(CC)nc(C)cc(=NC2CC(F)(CNC(=O)Cc3[nH]cnc3C)C2)[nH]1 N1(C(c2n[nH]c(CC)c2F)=O)CC2(C1)CN(C(c1ccc(CO)c(C)c1)=O)C2 C1(F)(CSC)CCN(c2c(S)cccc2F)CC1.C1(C(NC)=O)CCCC(C)CC1 C(=O)(CCCCCc1ccccc1)NC(CNC(Cc1c(C)ccnc1)=O)CO C1(NC(=O)C=C)CC2(C(N3CC(C)CC3CO)=O)COC1C2.C(C)(C(C)(C)C)=C(CC)C C1(CC)CN(C(=O)C(C)(C)CCSC)CCC1NC(=O)CCc1ccc[nH]1 C1(CNC(=O)C(F)n2ccnc2)CC2(C1)CN(C(c1cccc(Cl)c1O)=O)C2 N1(C(c2c(CC)c[nH]c2)=O)CC(CC(=O)NCCC2CC2C(=O)OC)CC1C N1(C(CC(CC)C)=O)CCCC2(CC(NC(=O)CCc3ccccc3F)C2)C1 C12(NC(CCC)=O)CCOCC1CN(C(=O)Cc1scnc1C)C2 C(c1ccc(F)nc1)=CC(=O)N(CCC(C(C)C)NC(C1CC12CCCC2)=O)C C(=O)(C#CC1CCCO1)N1CCC(CCN(C(=O)CSc2cccs2)C)CC1 N1(C(C2C(OC)C2)=O)CCOCC1CNC(C1(CO)CCOCC1)=O CCCC(C)(O)CC(=O)NCC1CC(NC(C2(P(C)(C)=O)CC2)=O)CCO1 c1(C(=O)NC2(C)CCCN(C(C3CC(F)(CO)C3)=O)C2)ncn2cccnc12 c1(C(=O)NC(C)C(C)(C)NC(C2CC2C(F)(F)F)=O)ccc2c(c1)[nH]c(=N)n2C Cc1cc2c(cc1C)C(C(=O)OCCOc1cccc(Cl)c1)CO2 C(=O)(C(C(CC)C(C)C)N(c1cc(OC)c(O)cc1)C)NCCCC(C)C c1(C(N2CCCC(O)(CNC(c3n(C)c(S)nn3)=O)C2)=O)cccn2cncc12 C1(CNC(C(C)OCC2CC2)=O)CN(C)CCN1C(=O)CN1CC(=O)N(C)C1=O C(=O)(CN=c1cc[nH]cc1)N1CC(CNC(C(CCOC)C)=O)OCC1 C(C)(C1CCCCC1)=CC(=O)N(C)Cc1c(OC(C(=O)OC)C)cccc1 c1(CC)c(C(N2CCCC(CNC(c3cc(Br)n[nH]3)=O)C2)=O)cnn1CC c12ccn(n1)C(CCCC)C(CCCS)C(=O)N(C)CCCCN(C)C2=O C1(F)(CNC(c2c(C)nco2)=O)CCCN(C(C23CCCC(CO2)C3)=O)C1 C1(NC(CC2CC(OCC)C2)=O)CCN(C(=O)C(c2ccc(Cl)cc2)C)C12CC2 c1(C(N2C3(CN(C(C4C(=C)CC4)=O)C3)CC2)=O)cc(OC)c(F)c(F)c1 N1(C(N2CC3CCN(C)C3C2)=O)CCN(Cc2ccccc2)CC12CCC2 C1(CC)CN(C(=O)CC2CCCCC2NC(C2CC(F)(CF)C2)=O)CCS1 C12(C(=O)NCC3N(C(CC(COC)COC)=O)CC3)C3C4C1C1C2C3C41C(N)=O N1(C(c2c(C)c([N+](=O)[O-])c(Cl)c(Cl)c2)=O)CCc2cc(Br)c(S(N)(=O)=O)cc21 C1(NC(C(N2CCC(C)C2)=O)=O)COc2ccc(Cl)cc2C1.C12(O)CN(C1)C2=O c1(N2CC3N(C)C(CC3)C2)nc(=NCc2cc(Cl)n(C)n2)[nH]c2c1CSC2 CC(C(=O)N(CC(=O)N(C)CCOCCNc1ccon1)C)C1CCCO1 CC1CN(C(c2ccc(-c3ccco3)nc2)=O)CC1NC(=O)C(C)n1ccnn1 Cc1cccc(CNC(C2CCN(C(=O)C=CC(C)(C)N)C2(C)C)=O)c1O C1(OC)CCCCC1C(=O)NCc1occc1C(=O)NC(CO)CCOC c1(C(N(CC(C)O)C(C)C)=O)cc(S(=O)(=O)N2CCC23CCCOC3)c[nH]1 C(C)(C)(CCC(=O)NC(c1ccccc1)C(N1CC2CCCC2C1)=O)N(C)C C(c1csc2ccccc12)=CC(=O)NCCCCNC(c1nnc(C)s1)=O N1(C(CCOCC#C)=O)CC(CC(N2CCC(=C)C2)=O)CC1(C)C Nc1ccc(Cl)cc1C(=O)NC1CC2(C1)CN(C(=O)CCCC1CCOCC1)C2 C1(CC(=O)NCC(=O)NCCC)CN(C(C2(CC)CCOC2)=O)CC12CC2 c1(C(=O)NC(CNC(C(C(C)C)SCC)=O)CC(F)(F)F)coc(S(C)(=O)=O)c1 C(=O)(C#CC1CCCO1)N1CC2C(CNC(c3n(CCOC)ncc3)=O)(C2)C1 C(CNC(c1occc1Cl)=O)(CC(F)(F)F)NC(CCn1c(C)ncc1)=O c1(OC)cc(O)ncc1C(=O)NCC(C(C)C)NC(c1cnn(C)c1)=O C1(NC(N2CC(C)(OC(C)(C)C)C2)=O)CC(C)(NC(COC(C)(C)C)=O)C1 Cc1nc(Cl)c(Cl)cc1NC(C1CN(C2CCC2)C1=O)=O N1(C(CCOCCCOC)=O)CCC(C)(CNC(=O)C(C(C)C)N(C)C)C1 n1(CC)nc(C)cc1C(=O)N(N1CCOCC1CO)C1C(C(=O)NC)C1(C)C C=CCC(CC)C(=O)NCC1CCCCN1C(=O)COCCCOC CCC(C)CC(c1nnnn1-c1ccccc1Br)NCC1CCC(F)(F)C1 Cc1csc(CCC(=O)NC(C)(C)C(C)N(C(=O)CC2CC3CC3C2)C2CC2)n1 Cc1cc2ccc(C(N3CCN(c4cc(C#N)n[nH]4)CC3)=O)cc2[nH]1 CC1CCc2[nH]c(=NCC(CC(=O)N(C)C)C(F)(F)F)[nH]c(=NCC3CC3)c2C1 C(=O)(C(C)(CNC(c1ccc(C)n1C)=O)CC)NCCCOCC=C C(CC1=CCCCCC1)N(C(C1C(C)(C)C1NC(c1nccnc1N)=O)=O)CC C1(C(N(CCOC)Cc2ccnn2C)=O)CC(O)C(F)C1 Cc1[nH]nc2c1CC(C(N1CC(C(C)NC(C3CCC3(C)C)=O)C1)=O)CC2 CC(C)(C)CCCCC(=O)NCC1C2CCN(CC(F)(F)F)C12 C(=O)(C(C#N)C(C)(C)C)NCc1ccc(C(N(CC(C)O)CCF)=O)nc1 c1(C(=O)OC)cncc(C(N2CCCC2CNC(C2CCCOC2)=O)=O)c1 CCCCC(O)CNC(=O)CC(O)CNC(=O)CC(C)(C)C C12(C(N3C(CN(C(COCCCC#C)=O)C)CC(F)C3)=O)CCC(C1)C2(C)C C1CCS(=O)(=O)CC1.C1(C#N)(COC)CCCO1 N1(C(Cn2c(C)ncc2)=O)CC2(CCN(C(c3ccc(N(C)C)cc3Cl)=O)C2)C1 C(C(CC(=O)NC12CC(NC(=O)CC3CCCN3C)(C1)C2)C(F)F)N(C)C CC(C)(C)CCC(=O)C(=O)NCC1CN(C(C2CCCC3C2C3(F)F)=O)CCO1 C1(C(=O)NCCC(C)N(C)C(c2cccc(F)c2F)=O)CCC(=O)N(C)C1 CC1CCCC=C1c1cccc(CNc2ccc3c[nH]nc3c2)c1 C1(CCCCCC)CCCN(C(c2cn(C)nn2)C(=O)Nc2ccc(F)cc2)C1 C1(C(=O)NCCOCC(=O)NCC2CCC=CO2)CCCN1C=O Cn1ncc2c(=O)n(CC(=O)NCC3COCCN3C(C3CC3CF)=O)cnc12 Cc1cnc2c(C(=O)NCC(CO)NC(=O)C=Cc3cccn3C)cnn2c1 c1(C(N2CC(CC=C)(NC(C3CCS(=O)(=O)N3)=O)C2)=O)nccc(C)c1O C1(NC(c2c(C)cc(CC)o2)=O)C2CC3CN(C(=O)Cc4cccn4C)C1C3C2 N1(C(c2cnc(C(C)(C)C)nc2)C(=O)NCC)CCC(P(C)(C)=O)CC1 C1(C(N2C(C3(NC(c4c(C)onc4)=O)CC3)CCCC2)=O)CCOCC1(C)C C1(NC(C(C(=O)OC)C)=O)CC=C(C(=O)N(C)CC2(CO)CC2)C1 c1(C(N2CCC(C)(NC(C)=O)C2)=O)cc(S(=O)(=O)NCC2CCCO2)ccc1C O=C1CCCC2CN(C(=O)C(NC3CCc4ccc(F)cc43)=O)CC2N1 C1(OC)CN(C(=O)CC2(OC)CCC2)C(C)(CN(C(=O)C(F)(F)CO)C2CC2)C1 C1(C(=O)N(C)CC2CCCCN2C(c2cccnc2Cl)=O)(CC)CCNC1=O CCC(C#N)(CC)C(=O)N(C)CCNC(=O)CC1CCCC1(F)F O=C(C(O)CC(F)(F)F)N1CCCCC1Cc1cn(C2CCCCCC2)nn1 N1(C(C(c2cnccn2)C)=O)CCN(C(C2CC(F)(CO)C2)=O)CC1C(F)F c1(C(=O)NCC2CCC(NC(C3(C)CC(C)C3)=O)C2)cccc(C(N)=O)c1 C1(CC=C)(NC(=O)Cn2cnnc2O)CCCN(C(c2sccc2C2CC2)=O)C1 C(=O)(CC(O)CC(C)C)NCC1(CNC(C=CSC)=O)CC1(F)F c1(CC)cc(NC(C2(C(=O)N(C)CCOCCCOC)CC2C)=O)n(C)n1 Cc1ccc(C(N2CC3CC3(NC(=O)CC3CCCOC3)C2)=O)cc1C(C)(C)C N1(C(Cc2c(C)non2)=O)CC(C(N2CCOC(C)CC2)=O)CC1(C)C CC1CCN(C(=O)C(C)NC(N)=O)C1C(=O)N(C1(C)CCCC1)C C1(C(=O)NC(C2CCN(C(C)=O)C2)C)CC2C(C1)C2(F)F C(C)(N=c1[nH]c(N2CCCC(C(F)F)C2)nc2cc[nH]c12)c1c(C)ccnc1 CCCCCCCCC(=O)N1CCCC(N(C(=O)C(C)CN(C)C)CCO)C1 N1(C(C(C)=CCC)=O)CCC(C(=O)N(C2CSC2)C)(CC)C1 c1(CC)cccnc1C(=O)NCCOC1CCN(C(C2C(C)C2C)=O)C1 CCCC(C(=O)OC)C(=O)N(C1CN(C(=O)C=Cc2ccc(SC)cc2)C1)C C1(CNC(=O)C=CC2CCCO2)CC2(CC2)CN1C(=O)CSC1CCC(=O)N1 c1(C(N(C)CC2CCCN(C(c3c(C)nsc3N)=O)C2)=O)nn(C)c2c1CCC2 C1(C)(CC)C=C(C(=O)N(C2CCCCC2N(C)C(c2cc(C#N)cn2C)=O)C)C1 c1(C(=O)NC2C=CC(C(=O)NCC(C)(C)C#N)C2)ccc(Cl)cc1 C(C)(C(=O)N=c1[nH]oc2ccccc12)c1cccc(NC(C)=O)c1 c1(C(=O)NCC2C(NC(c3ncn(CC)c3)=O)C2)cccc(F)c1F c1(CSCCC(=O)NCC(C)(C)NC(=O)CO)csc(C(F)F)n1 CC1CC(C)N(C(=O)CN2CC(C)(C)C2)CCN1C(=O)CSCC(N)=O c1(CCC(=O)NC2CN(C(C(C)=CC)=O)CC3(C2)CC3)ccc2c(c1)CCCO2 c1(C(N2CC(O)(CNC(=O)CC3CSCCS3)C2)=O)ccc2ccccc2c1O N1(C(CNC(C2C(OCC)C2)=O)C)CCN(C(C2(CC3CCC3)CC2)=O)CC1 N1(C(C(CC)C)=O)CC(CO)C2(C1)CN(C(c1ccnc(C(F)(F)F)n1)=O)C2 C1(C(N(CCCNC(c2ncc[nH]c2=O)=O)CC)=O)CC2CCC(C1)C2O S(=O)(=O)(c1ccc(NC(c2cc(C)no2)C)c(F)c1)N1CCC(OC)C(C)(C)C1 C(CC(C)(C)CNC(c1ccc(C2(O)COC2)cc1)=O)NC(C(C1CC1)OC)=O C(=O)(C1=CCC(C)CC1)N1CCC(CC=C)(NC(=O)CC2CCC=CCC2)C1 c1(CNc2cnc(N(CCNC)C)nc2)csc2c1CCCC2 C12(C(N(CC(C)O)C)=O)CCC(CC1)N(C(C1(C)CCOC1)=O)C2 N1(C(c2ccn(CCC)n2)=O)CCCC(NC(C2(C)CCC3CC3C2)=O)CC1 C1(C(=O)NC2CC(CCC)C2)(CNC(CC)=O)CCC1 CN=c1[nH]cc(C(=O)NCC(CNC(c2cc(N(C)C)ccn2)=O)OC)s1 c1(C(C)NC(=O)NCCC2CC(O)C2)cc(Br)cc(F)c1O N1(C(c2ncc(N(C)C)nc2)=O)CC2CCN(C(c3cc(O)n(C)n3)=O)CC2C1 Cc1cc(Br)ccc1CC(=O)NCC1CCN(C(c2ccc[nH]2)=O)C1 CC1(C)CC2(CC2C(=O)NCC2(C)CCN(C(=O)CNS(=O)(=O)C3CC3)C2)C1 c1(CC(N2CCC(C)C2CNC(=O)C2=NOCC2)=O)c(Cl)cccc1Cl c1(C(N2C(C(N(CC)CC3CCC3)=O)CCC(O)C2)=O)ccnc2cc[nH]c12 N#Cc1ccc(O)c(C(N2CC(OCCNC(C34CC(O)C3C4)=O)C2)=O)c1 C(=O)(C1Cc2ccc(F)cc21)N1C(C)CN(C(c2cc(F)cc(F)c2)=O)CCC1 c1(C(N(CC(CN(C(=O)C=Cc2nccs2)C)O)C)=O)occc1Br CN1CCC2CCN(C(C3CCCC(NC(=O)CC4CC(=O)C4)CC3)=O)C2C1 C(CCC(=O)N(C)CC1CCCO1)=CCC=C.C12CCCN1C(=O)CNC2=O C1(C(N(CC(=O)NCCCNC(COCC(=O)OC)=O)C)=O)CCC1(C)C C1(C(=O)NCC(C)(C)CNC(C2CCC(C)(C)OC2)=O)OCCOC12CCC2 c1(CC(=O)NCC2(OC)CN(C(c3ncccc3C(F)F)=O)C2)c(C)n[nH]c1C C1(CC(=O)N(CCOCCN(C(C2C(C)C2C)=O)C)C)NC(=O)CNC1=O CCC1CCC(=O)N2CC=CC2(C)C(=O)N1.c1(COC)coc(C)n1 C1(N(C(C(COC)C)=O)C)CCN(C(C2(F)CC3(CCC3)C2)=O)CC12CC2 Cc1c(C(=O)NC2CCC(CNC(c3coc(C4CC4)n3)=O)C2)ccn1C1CC1 CCCC(F)(F)C(=O)NC1OCCC1C(=O)NCCOc1cccnc1 C1(CC(=O)NC(c2ccc(F)cn2)C)CCCCN1C(=O)CCC1CCCCC1 CC(C(C)(C)C(=O)NCCOc1ccsc1)NC(=O)Cc1ccon1 CCC(C(C)CN(C)C)NC(C1C=CCN(C(=O)CC2CC2)C1)=O c1(C(=O)NCC2N(C(CC3CN(C(C)=O)C3)=O)CCC2C)cc(N)c(F)cc1C C1(C(N2CC(NCC(F)F)C2)=O)(NC(c2cn[nH]c2)=O)CCSC1 C1(NC(C(c2cccc(C)c2)O)=O)CCN(C(=O)CN2CC(F)(F)C2)C(C)C1 N1(C(=O)NCC2CCCC(CF)C2)CCOc2ccncc21 C1(C)(C(=O)NCC2(C)CCN(C(CN(C)C(N)=O)=O)C2)CCCNC1=O N1(C(C=Cc2occ(C)n2)=O)CCN(C(C2COC3(CCC3)C2)=O)CC(C)(F)C1 CC(O)(CNC(c1ccc(C(N)=O)cc1)=O)CCCO.C12(C)CCCN(C1)C2=O Cc1nn(C)c(N)c1C(=O)NC1CCCC1NC(=O)CCN(C)C CC(C)(C)CCCC(=O)NCC1CCN(C(c2cncc(Cl)c2)=O)C1 c1(-c2cn(C(CNC(CCc3c(OC)cccn3)=O)C)nn2)cc(F)ccc1F C1(CNC(=O)Cc2cnn(C(F)F)c2)CC2(CCC2)CN1C(C1SCCCS1)=O CCCCC(O)CCC(=O)NCCC1(Nc2nccc(CO)n2)CCC1 C(C)(C)(CC(=O)NCC(=O)NC(C)C)OC.C12CCCC1(C)N2 CCCC(CCC)CC(=O)NC12CC(C(=O)NC(C)C(C)C(=O)OC)(C1)C2 C1(CC)CCCC1C(=O)NC(CNC(=O)C(F)(F)c1cnn(C)c1)C(C)C c1(SC)ncc(NC(=O)CC2(C)CCN2C(=O)C(=O)N(C)C)cn1 C#CCC(C)C(=O)NC(C)CNC(c1cccc(-n2c(C)cnc2O)c1)=O C=C=C(C)CC(=O)NCC1(C(C)(C)C)CCN(C(=O)CN2CCOCC2)C1 c1(OCC)ccc(C(=O)NC(C(=O)OCC)C(C)C)cc1Br n1(CC)nc(C)c(C(=O)NC(C)CC2CN(C(c3[nH]c(O)nc3C)=O)C2)c1C C(=O)(C(=O)NNc1ccc(Br)c(C)c1)NC1CCN(C(=O)OCC)C(C)(C)C1 Cc1c(C(=O)NC2CCN(C(=O)Cc3cccnc3)CC2F)cnc2ncnn12 N(S(=O)(=O)N1CCOC(C)C1)Cc1cccc(NC(=O)NC)c1 C(C1OCCc2sc(-c3nn[nH]n3)cc21)NC(C(c1ccc(Br)cc1)(C)C)=O Cc1ccc(SCC(=O)NC2CN(C(=O)CCN(C)CCO)C3CC23)cc1 N1(C(C)=O)CCOC(C(=O)NCC2(CO)CC23CCC3)C1.n1(CC(=O)N)cncn1 c1(C(=O)NC2C(C)N(C(=O)CCc3cccnc3F)CC2)cc(Cl)ccc1F N1(C(C=C(C)Cl)=O)CCC2(CCCN(C(=O)C=Cc3cccc(Cl)c3)C2)CC1 C1(C(=O)NCCOCCNC(=O)CCc2cccc(O)n2)(CC)CCC(O)CC1 c1(NC(c2nnnn2CC2CCOC2)(CC)C2CCCO2)ccc2sncc2c1 C1(CNC(c2ncccn2)=O)CCN(C(=O)Cn2cccc2)CCC1(F)F c1(C(=O)NC(C)(CNC(=O)CCc2nccs2)C2CCC2)ccc(O)c(Cl)n1 Cc1nsc2ncc(C(=O)NC3(CNC(=O)C(C)CS(C)=O)CCOCC3)cc12 c1(C(=O)NCC(C)CNC(C2CCCC(CF)C2)=O)c(F)cc(Cl)cc1F c1(CC)cc(C(=O)N(CC(CC)NC(c2cnsc2C)=O)C)cn(C)c1=O C1(NC(C2(CC#C)CCCO2)=O)CN(C(=O)C(C)(C)OC(C)=O)CC1CCC C(C)(C(C(=O)NCC1C2CN(C(c3csc(C(C)=O)c3)=O)CC12)N(C)C)OC N1(C(C2CC3CC3N2C(=O)CCc2ccco2)=O)C2CCC1(CO)CC2 C1(C(=O)NCC2N(C(C(CC)C)=O)CCCC2C)CC2(CCOCC2)CO1 C(=O)(C1=CCN(C(C2CC(C)CCO2)=O)C1)NC(CC)CC(C)O c1(CNC(C(N2C(C#C)CCC2)c2ccsc2)=O)c(C)cccc1C C=CC1(CC(=O)NCC2(C(F)(F)F)CC2)CN(C(c2cc(OC)ncn2)=O)C1 CC1CCCC(C(=O)NC(C(=O)NCCn2ccnn2)C2CCCC2)C1 C1(C(=O)NC(C)CN(C(=O)Cc2ncc[nH]2)C)CCCN1C(=O)C(C)(C)C C(=O)(C(O)(C(C)C)C(F)(F)F)NC(CC)CNC(c1cc2sccc2[nH]1)=O N1(C(C(CC)F)=O)CC(C)OC2(CCN(Cc3c(C)cccc3C)C2)C1 Cn1c(C(=O)NCC2(F)CCN(C(c3n[nH]cc3Cl)=O)C2)cc2sccc12 Cc1cc(Cl)ccc1CNCC1COCCN1C(=O)Cc1c(F)cccc1F Nc1cncc(-c2noc(C3CC3(c3ccc(Br)cc3)F)n2)n1 N1(CC(=O)NCCC)CCN(C(c2ncn(CCN(C3CC3)NC)c2)=O)CC1 O=C(C(CCc1ccc(F)cc1)N1CCC(CC2CCC2)C1)NCc1cccs1 C1(CNC(c2cc(C)oc2C)=O)CC(C)CCN1C(c1[nH]nnc1C)=O N1(NC(C2C3(CC(NC(c4ccc(CC)cn4)=O)C3)C2)=O)CC2CSCC(C2)C1 S(=O)(=O)(C(F)(F)F)N(CCC(=O)NCC1CC1CNC(=O)CCNC(N)=O)C C(=O)(C(CC(F)F)N(C)C(c1ccc(C(C)=O)o1)=O)N(CCC)CCC C1(NC(=O)Cc2cnsc2)CCN(C(c2ccc(Br)o2)=O)C1c1ccccc1 c1(OC)ccc(C(=O)NC2(C)CCN(C(c3ccsn3)=O)C2)cc1 Cc1nc2c(s1)CCCC2C(=O)NC1CCC1NC(=O)C=CC(=O)N(C)C c1(-n2ccc(C(C(=O)NCC(=C)C)N(CCOC)CC)n2)ccccc1Cl c1(OCC(=O)N(C)CC2N(C(C=CCOC)=O)CCOC2)ccc(Cl)cc1Cl CC1=NOC2(C1)CC(C(N1CCN(C(=O)C(C)C(C)(F)F)CC1C)=O)C2 N1(C(Cc2c(C)noc2Cl)=O)CC(NC(=O)C(F)C(F)(F)F)C(N=[N+]=[N-])C1 N1(C(C=Cc2n(CC)ncc2)=O)CCC(NC(c2n[nH]c(O)n2)=O)C1(C)C Cc1cccn2cc(C(=O)NCC3(F)CCC(CNC(=O)CNC=O)C3)nc12 C(=O)(CN=S(C)(C)=O)N1CCC(C)(NC(c2c(CC)n(C)nc2)=O)C1 N1(C(C2N(C(C(CCCC)F)=O)CC3(CC3)C2)=O)CCCN(C)C(=O)C1 N1(C(C2(CF)CC2(F)F)=O)CCCC(NC(c2cnn(C3CCC3)c2)C)C1C c1(C(N(C(C)CNC(=O)Cc2cocn2)C)=O)nc(C(C)C)ncc1Cl CCCC(C)CCCC(=O)N1CCC2(CC2NC(=O)CC2CCCN2C)C1 C1(O)(N(C(CC(OCC)OCC)=O)C)CCN(C(=O)C(C)(C)c2cscn2)CC1 N1(C(C(CCCC)NC(c2nc(C)oc2C)=O)=O)CCC2CN(C)CC2C1 C(=O)(CC(C)CC(C)C)NCCC(CNC(c1c(C)coc1C)=O)(C)C C[Si](C)(C)C1(C(=O)NCC2(NC(=O)C3=CCOC3)CCCCC2)CC1 CCCCCCCCCCCCNC(=O)C(N1CCCc2c(O)cccc21)=O C1(C(N2CCOCC(NC(=O)CCF)C2)=O)Cc2cc(F)ccc2O1 c1(C(=O)NC2CC(NC(c3c(CC)con3)=O)C2)ccc2c(c1)nnn2C C(=O)(C(O)C(F)(F)F)N1CCCC(OC(c2cn(CCO)nn2)C)C1 C(=O)(CC(F)(F)C(F)F)NCC(CN(C(c1cc(C(C)C)no1)=O)CC)(C)C C(=O)(C1CCCc2scnc21)NCC1(OC)CN(C(C2(Cl)CC2(C)C)=O)C1 Cc1cn2c(n1)C(C(=O)N1CC(NC(=O)CN3CCOCC3)CC(C)C1)CCC2 c1(C(C(=O)NC2CCC2)N(C(C#C)C)C)snc(OC)c1Cl C(C(C)CNC(=O)CC1CC12CC2)N(C(C1(CC)CC1)=O)C c1(COC)cc(OC)ccc1-c1ncccc1NCC1CCOCO1 N1(C(C)=O)CCC2(CCN(C)C2)C1.C12(CC=C)CCCN1C(=O)CONC2=O N1(C(c2ncc(CC)nc2)=O)CC(NC(c2csc(CC)n2)=O)CCC1C c1(C(=O)NC2(C)CC(NC(C(CCOC)C)=O)C2)ccc2c(c1)CCCS2(=O)=O c1(C(=O)NC23C(CN(C(CCC(=O)NC)=O)C2)CCC3)cc2n[nH]cc2cc1C C1(NC(C2C(C)(C(F)F)C2)=O)CCCC1CNC(=O)CC(=O)NCC(F)(F)F c1(C(=O)OC)cc(-c2cn(CC3CCCN3C(=O)C(C3CC3)SC)nn2)c[nH]1 N1(C(C(C(C)C)NS(N)(=O)=O)=O)CCN(C(=O)CC(C)(C)CN(C)C)C2CC12 CC1CCC(CN(C(=O)CC2C=NN(C)C2=O)C)CC1 Cc1nc2ccc(NC(C3COC4CN(S(=O)(=O)CCCCl)CC34)=O)cc2o1 CN1CCC(C(=O)NC2(C)CCN(C(=O)CC3CCOC(C)(C)C3)C2)S1(=O)=O N1(C(C2(C)C(C)(C)CCC2)=O)CC2(C(=O)NCC(N)=O)CCC1CC2 C1(CNC(CCNC(CC(C)C)=O)=O)CC(C)N(C(=O)CN2CCCCCC2)C1 Cc1cc(C(N2CC3(C2)CN(C(c2cnc(C(C)C)nc2C)=O)C3)=O)cc(F)c1 N1(C(C2CC(NC(CC(=O)OC)=O)C2)=O)CCC(N(C)C)CC1 CCC(C)C(C(=O)N1CC(C)(C(F)(F)F)C1)NC(c1cc(OC)cnn1)=O C(=O)(CCC(C)C)N(CCOCCN(C(C(CC)OC)=O)C)C.C1CN1 c1(CNC(=O)NC(c2ccco2)C)ccc2c(c1)CCC2NC(=O)CN=S(C)(C)=O Cn1nccc1Cn1cc(C2CCCC2O)nn1.N12CCC1SCC2=O N1(C(C2(CNC(CC=CCC)=O)CC=CC2)=O)CCC(N=[N+]=[N-])C(O)C1 N1(C(C(CC)(C)CNC(c2nn(C)cc2Cl)=O)=O)CCC(N(C)OC)CC1 C(=O)(C(O)C(O)C(F)(F)F)N1C(C(N2CCC(C#N)CC2)=O)CCCC1 N1(C(c2c(NCC=C)cccn2)=O)CCCC(C)(CNC(c2coc(Cl)n2)=O)C1 N12CCN(CC1)C2.CCS(=O)(=O)NCCCC1(NC(=O)COCC(=O)OC)CC1 C(CC(C(=O)NCC(=C)CC)NC(c1ccc(C)s1)=O)=CC C1(CNC(COC2CCN(C(C3C(CCOC)C3)=O)C2)=O)CC2(CCC2)CO1 C(=O)(C(O)C(N)COC)N1C(c2cccc(C(=O)OC)c2)CCCC1 c1(C(N(CC=CC(=O)N(CCCC)C)C)=O)nonc1N N#Cc1ccc(=NCC2CC(NC(c3n[nH]cc3[N+](=O)[O-])=O)C2)[nH]c1C(F)(F)F C1(NC(Cn2ccc(C(=O)OC)n2)=O)CN(C(=O)CC2(C)CC2)CC1C S(=O)(=O)(c1ccc(NCCC2CCOCC2)c(Cl)c1)NC(C)CC1CCCCO1 C1(CNC(C2C(C)(Br)C2)=O)CC(F)(F)CN1C(=O)CN1CC2C=CC1C2 N1(C(C2CC2[N+](=O)[O-])=O)CC2OCCN(C(c3cc(C(F)F)[nH]n3)=O)C2C1 C1(C)(CC(=O)NCC(COC)OC)CCN(C(C2OCCC2C)=O)C1 C1(NC(C(CC)CC)=O)CCN(C(c2cc(C(F)(F)F)n(C)n2)=O)C12CCC2 c1(C(N2C(CNC(=O)CC(F)(F)F)CCC(C)C2)=O)cc2c(cc1N)CCC2 CN1CCN(C(=O)C=C(Cl)Cl)C(CNC(C2CCCC2(F)F)=O)C1 N1(CCC(=O)Nc2c(OCC)cccc2)CCC(P(C)(C)=O)CC1 C(CN=C(NCC1CCC12CCC2)NCC1(C2CC2)CCCO1)OC c1(NC2CC(NC(C3(CCC)CC3)=O)C2)c(F)cc(F)c(OCC)c1[N+](=O)[O-] CCCC(C)NC(=O)C=CCNC(=O)CN(C)CCOC c1(N(C2CCS(=O)(=O)C2)C(c2cnn[nH]2)C)nnc(C2CC2)n1C C=CCCC(C)(C)C(=O)N1CCN(C(=O)CN(C)C(C2CC(CCO)C2)=O)CC1 C1(NC(c2cnc(S)[nH]2)=O)CCCN(C(c2csc(F)c2)=O)CC1 C1(C(=O)NC2CC(C)N(C(c3c[nH]cc(F)c3=O)=O)C2)Cc2ccccc2N1 c1(NC(c2cccn(CC)c2=O)=O)ncn2ccccc12 c1(CN(C(=O)C#CCNC(=O)CCOCC2CCC2)C)cncn1C1CC1 N1(C(C23N(C(CN(C(C)C)C)=O)CC(C2)C3)=O)CCC12CCCOCC2 N1(C(c2ccnc(CO)c2)=O)CC2(CCCN(C(C3SC4C=CC3CC4)=O)C2)C1 C12(CC(=O)NC(CCC)C(=O)NC)CCC1CN(C(c1nc(C)ccc1F)=O)C2 C1(CNC(=O)CCF)CC2(CO1)CN(C(c1cc(F)c(F)cc1F)=O)C2 Cc1ccccc1NC(C1CCOC1CNC(=O)CC1(CO)CCC1)=O N1(C(=O)C(O)C(F)(F)F)CCCC(C2CN(C(C3(Cl)CC3(F)F)=O)C2)C1 C1(O)(CN(C(C=CC(C)C)=O)C)CCCN(C(c2cnn(C)c2Br)=O)C1 C(C)(CN=C(NCC1CNC(=O)C1)N(C)CC(=O)OC(C)(C)C)OCC=C c1(C(=O)NC(CC(=O)N(C2CC(SC)C2)C)C(C)OC)ccc2nccn2c1 C(=O)(C(CN=[N+]=[N-])NC(=O)CCc1ncnn1C)Nc1c(C)nn(C)c1 CN1C(=O)C(=O)N(CC(N2CCC(CO)(NC(C3CCOC3)=O)C2)=O)C1=O c1(CNC(NCc2c(Br)c(C)n(C)n2)=NCC2CCC2)ccc(C#N)cc1F Cc1cnc(C)c(C(N2CC(NC(=O)C3=CC(C)(C)C3)CCC2C)=O)c1 C1(C(N(C2CCCCCN(C(=O)CSCC(N)=O)C2)C)=O)CC(C(C)(C)C)=NO1 C1(CNC(C2C(F)(C(=O)OC)C2)=O)CC12CCN(C(C1CC(O)C1)=O)CC2 n1(CCOC)cc(C(=O)OC(C(=O)NCC(C)(C)NC(=O)C(C)(C)C)C)ccc1=O N1(C(c2ccc(C(=O)OCC)cc2)=O)CC2CCC(C1)N2C(=O)C1=CCSC1 C123CN(CC(CO)(C1)C2)NC3=O.c1(CC)nc(-c2ccco2)n[nH]1 N1(C(c2ccn(CCC)n2)=O)CCC(C)(CNC(=O)CCc2cccn2C)C1 c1(C(=O)NC23CC(C(N(C(C4CCOC4)CO)C)=O)(C2)C3)cc2ccccc2n1C N1(C(c2ccc(F)c(Cl)c2)=O)CCC2CCN(C(=O)CCCCO)C2C1 CC(C)C(F)(CNC(=O)CC1CCOC1C)C(=O)NC1CCN(CCO)CC1 S(=O)(=O)(c1ccc2c(c1)CCO2)N1CC2C(C(N3C(C)C(=O)N(C)C3)=O)(C2)C1 c1(C(N2CC(NC(CC=CC=C)=O)C(NC3CC3)C2)=O)cc2c(ccn2C)[nH]1 c1(C(=O)OCC(=Cc2cccnc2)C)cc2cc(N)ccc2[nH]1 c1(CNC(CC(CC)C)=O)ccc2c(c1)CN(C(c1c(C)nsc1NC)=O)C2 n1(CC)ccnc1C(=O)NC(CC1CCC1)C(=O)NC1CCCC1F C(=O)(C1Cc2ccccc21)NCCCN(C(=O)Cc1cccc(F)c1)CCC c1(C(C)C)cncc(C(=O)NCC2CC(CNC(C3(N=[N+]=[N-])CC3)=O)CO2)c1 c1(NC)ccccc1C(N1CCCC(N(C(=O)C(c2ccc(O)cc2)=O)C)C1)=O C(CCCCC(=O)NCC1CCC(F)(CNC(=O)C(=O)C(C)C)CC1)SC c1(C(=O)NC)cccc(C(=O)NCCCCN(C(=O)CCOCC(F)(F)F)C)c1 N1(C(c2ccc(C)s2)=O)CCC(C)(NC(=O)C(C)Cn2ccnc2)C1 c1(CC(=O)N(C2CN(C(=O)CCF)CC2F)C)nc2cc(Cl)ccc2s1 CC(C)CC(C(=O)NCCOCCNC(c1nonc1N)=O)C(C)C C(=O)(CS(=O)(=O)C(C)C)N(C(C)C)CCNC(=O)CS(=O)(=O)NCC1CCCO1 CC1ON=C(C(=O)NCCC23CCC(C2)N(C(=O)CCCS(N)(=O)=O)C3)C1C N1(C(CN2CCN(C(C(C)OCOC)=O)CC2)=O)CCOCC(C)(O)C1 S(=O)(=O)(c1cccnc1NCC1(n2ccnn2)CC1)N(C)Cc1cnn(C)c1 C(=O)(CC(C)CC(C)C)N(CCC(c1cccs1)NC(CC)=O)C CCCCC(O)CC(=O)N1CC(N(C(=O)CN2CC3(CC3)C2)C)C2(CC2)C1 C(=O)(C1=NOC2(CCCN(CC(C)(C)C)C2)C1)NC(c1nccn1C)C(=O)NC C1(C(C(=O)N(CCNC(c2nc(CC)oc2)=O)CC)F)CCC(=O)CC1 N1(C(C(CCCC)O)=O)CCC2(CC1)CN(C(c1snnc1C1CCC1)=O)C2 Cc1cc(C(=O)NCC2CN(C(=O)C=CC3CC3)CC(C)(C)O2)cc(C)c1F C(=O)(C(C#N)C(C)(C)C)N1C2(CN(C(C(=C(C)C3CC3)F)=O)C2)CC1 c1(C(=O)NCC(C(C)C)NC(C23CSC(C2)C3)=O)cc(C(N)=O)cc(F)c1 Cc1cccc2sc(C(N3CCC(F)(c4cn(C5CC(O)C5)nn4)C3)=O)c(Cl)c12 C12(C(N3C(CNC(C4N(CC)C(=O)CC4)=O)CCCC3)=O)C3C4C5C3C1C5C24 c1(C(=O)NC(C2OCCN(C(c3ccc(C)nn3)=O)C2)C)cc(Cl)c(F)cc1Cl N1(C(Cc2c(C)noc2C)=O)CCCC(C)(NC(C2CC3(CCC3O)C2)=O)C1 C1(O)(C(C)C)CCN(C(=O)C(O)CN(C(=O)OC(C)(C)C)C(C)C)C1 c1(CC)ccnc(CNC(=O)CN(C(=O)Cc2ccns2)CCOC)c1 c1(NC(Cn2ncc(C(N)=O)c2)=O)cccc(NC(C2CC(F)C2)=O)c1 C1(C(=O)OCc2cccc(Br)c2)Cc2ccc(Cl)cc2C1 N1(C(CC(=C)C)=O)CCN(C2CCCC2NC(=O)CC(CC)SC)CC1 N1(C(C=C(C)C2CC2)=O)CCC(C2N(C(=O)CS(=O)(=O)N(C)C)CC2(C)C)CC1 Cc1cc(CN(C(=O)CNC2(F)CCN(C(=O)OC(C)(C)C)C2)C)cc(C)c1 C(=O)(CC(C)NC(=O)C(O)C1CN(C(C2CC=CCO2)=O)C1)OCC C1(N(C(C2(C(C)C)COC2)=O)CC)CCCN(C(=O)C=CC2CCC2)C1 N1(CC(=O)N(C2CCN(C(c3n[nH]cc3Cl)=O)C2)CCO)C(=O)CNC1=O C(CCC=CC(=O)NC(C)CN(C(=O)CN(CC(=O)N(C)C)C)C)=C(C)C c1(NC(N2CC(N3C(=O)CC(N(C)C)C3)C2)=O)cc2ccnc(Cl)c2s1 C12(c3ccsc3)C3C4C1C1C2C3C41C.C1(OC)CC2N(C1)C(=O)c1cc(ccn1)C2 N1(C(CS(N)(=O)=O)=O)CCN(C(c2csc(Br)n2)=O)CC(O)C1 C1(CNC(C2(CC)CC2)=O)CCC2CN(C(c3nccc(Cl)c3F)=O)CC12 Cc1cc(C(N2CCCCC2CNC(=O)Cc2ccco2)=O)nn1C N1(C(c2c(CC)[nH]nc2Cl)=O)CCOCC(CNC(C2CCSC2)=O)C1 Cc1nc(Cl)ccc1C(=O)NC1C=CCN(C(=O)C(C)(O)C(C)C)C1 Cc1[nH]nc2c(C(=O)NCC3(F)CC(NC(c4csc(=N)[nH]4)=O)C3)cccc12 c1(C(N(CC2CCCN(C(C3(C#C)CC3)=O)C2)CC)=O)csc2nnsc12 c1(C(=O)NC(CNC(C2C(=C)CC2)=O)(C)Cn2cccn2)cc(C)ccc1Cl C1(NC(c2cnc(C)o2)=O)CCSC12CN(C(c1c[nH]cc1Br)=O)C2 C12(CNC(=O)CCOCCNC=O)CCC(CC1O)C2.C1(N)CCCO1 N1(C(c2ccc(N(C)C(=O)OC(C)(C)C)cc2Cl)=O)Cc2ccccc2C1CO N1(C(C(C)O)=O)CC2(CO)CC1(C(=O)Nc1cncc(C(F)F)c1)C2 N1(C(C(c2c(OC)cccc2)=O)=O)CCC2CN(C(c3ccc[n+]([O-])c3)=O)C2C1 Cc1cncc(C)c1C(=O)N(CC(C)NC(c1ccncc1-n1cccn1)=O)C c1(C(=O)NC(COC)C(=O)NC(c2noc(C)n2)C)ncc(C)cc1F C1(CNC(c2c(CC)nco2)=O)CCCN(C(c2c(C)noc2C)=O)CC1 N1(C(COC2CC(SC)C2)=O)CC(N(C(=O)C=CBr)C)C(F)C1 N1(C(CCCOCC=C)=O)CC(C)(C)CC1C(=O)N(C1CCC(F)(F)C1)C C1(C(=O)NCC(C)CNC(=O)CC(C)c2ccccc2)CCCC1(C)C C1(C2CCC2)(C(=O)NCC(C)(C)NC(c2ccc(CCC)s2)=O)CCC1 C1(C(=O)NCCc2c(C)ccnc2)CN(C(C2SCCS2)=O)C2(CCC2)C1 Cc1ccccc1CSCC(N1CCC(C)C1CNC(=O)CCC1CC1)=O Cc1cc(C)nc(SCC(=O)NCC2(C)CCN(C(C3CC34CCCC4)=O)C2)n1 c1(C(=O)NC2C(NC(C=C(C)C(C)(C)C)=O)CCC2)cccc(Br)c1 N1(C(CN2CCN(C)CC2)=O)CCCC(CC(=O)N(C2CCCC2(C)O)C)CC1 CC1(C)CC(CO)CN1C(c1ccnc(CNC(c2cc(Cl)no2)=O)c1)=O C#Cc1ccc(C(N2CC(CCNC(=O)C(O)C(F)F)C(C)C2)=O)c(C)c1 N1(C(C(c2ccccc2)NC(C)=O)=O)CCC(C=CC(=O)NCC(C)C#N)CC1 N1(C(C)=O)CCCC1C(=O)NCCC(C)N(C(=O)CC1CCCCC1)C N1(C(=O)CCSC(F)(F)F)CCOC2(CCN(C(C3(CCF)CC3)=O)CC2)C1 c1(C(N2CC(C(C)NC(C3=C(C)CCC3)=O)C2)=O)cccc2nsnc12 N1(C(c2cc(C)ns2)=O)CCCC2(C1)CN(C(c1ccccc1OCCF)=O)C2 c1(N2CCC(CCC)(NC(C3CC3OC)=O)CC2)nc(OCC)c(F)c(C)n1 N1(C(CC(C)SC)=O)CCC2(CC1)CCN(C(=O)CCN(S(C)(=O)=O)C)CC2 O=C(C#CC1CCCC1)NCC1CCCN(C(C2CC23CCOCC3)=O)CC1 c1(C(N(CC(CC)NC(=O)Cc2cncnc2)C)=O)ccc2oc(O)nc2n1 CCCC(C)(C)C(=O)NC1CN(C(c2cccc(CS(C)(=O)=O)c2)=O)CC1C Cc1oc(C(=O)NC2C3CC2N(C(=O)CC2OCCCO2)C3)cc1CO C1(NC(=O)CCC2CC(F)(F)C2)CN(C(c2cncc(CO)c2)=O)CCC1O c1(CN(C(c2cc(Cl)sc2Cl)C(=O)OC)C)nc(O)c2ccc(Cl)cc2n1 N1(C(C2C(CCC)C2)=O)CCC(NC(=O)Cc2coc(C)n2)C(F)(F)CC1 c1(C(=O)NC2C3CN(C(CC(CC)C4CC4)=O)CC32)cc(N)cc(N)c1 N1(CCC(=O)OCC)CCN(C(c2cccc(F)c2)=O)CC1 C(=O)(C#CCNC(C1CSC1)=O)NC(C1CCC1)C c1(OC)cc(CN2CCC(O)(C(=O)NCc3cccc(CO)c3)CC2)ccc1C#N C1(C2CN(C(C3N(C(c4[nH]cc(C(C)=O)c4)=O)CC3)=O)C2)NC(=O)NC1=O C(=O)(CCCCCSC)NCCOCCNC(=O)CC1C=CCC1.C(=O)NCC C1(CNC(c2nc(C)nn2C)=O)CN(C)CCN1C(=O)CCc1cnco1 C#Cc1ccc(F)c(C(=O)NCC2(C(C)NC(=O)C=CCCC)CC2)c1 N1(C(C=CCCC)=O)CC2CC(NC(c3ccn4c(C)ncc4c3)=O)CC(C2)C1 C1(CNC(C(COCC)NC(C2(C)CSC(C)=N2)=O)=O)CN2CCC1CC2 N1(C(C2NC(=O)OC2)=O)CC=C(CNC(C2CC3(CCCO3)C2)=O)CC1 c1(NC2(CNC(C(C=C)(C)O)=O)COC(C)(C)C2)nn2cc(C)nc2s1 Cn1cc(-c2c[nH]nc2C(=O)NC2(c3ccsc3)CC2)c2cccnc12 N(C1CCCc2c(Br)cccc21)S(=O)(=O)c1ccc(-n2nccn2)cc1 c1(N2CCC(NC(CC(C)C)=O)CC2)nccc(N2CCCCCC2)n1 c1(C(=O)NCC=CCC(N2CCC(C(C)C)C2)=O)cnc2n1CCC2 C1(CNC(CCCOC(C)C)=O)C(C)CCCN1C(c1ccco1)=O c1(C(=O)NCC(O)CNC(c2ccoc2Cl)=O)ccc(OCC2CCCO2)cc1 c1(C(=O)NCC(C)(C(C)C)NC(Cc2ccc(C)o2)=O)ncc(C(F)(F)F)cc1Cl c1(C(=O)NCCCN(C(C2CC(CC(C)(C)C)C2)=O)CC)c(C)cnn1C N1(C(C23N(C(C(CC)n4ccnc4)=O)CC(CO)(C2)C3)=O)C2CCC1CN(C)CC2 CN1CCC=C(CNC(=O)CCC2CCCN(C(C3(C)CC(C)(C)C3)=O)C2)C1 n1(CCC)nnnc1C(C1(COCc2ccccc2)CC1)NCC1CC(C)C1 c1(OC)ccc2occ(C(N3CCN(Cc4ccc(Cl)s4)CC3)=O)c2c1 C(=O)(CCC(=O)NN(C)C)N1CCN(C(Cc2c(C)noc2)=O)C2C1CC2 c1(C(N(C(=O)CN2CCCCC2)CC)=O)cccc(C=C(F)F)c1 NC1CCCc2ccc(C(=O)Nc3cc(Br)cc(C(F)(F)F)n3)cc2C1 c1(C(N2C(CNC(CCCSC)=O)C(C)(C)CCC2)=O)c(C)c(C)nn(C)c1=O C12(C(=O)NC(C(CSCC)O)=O)CCC(CC1OCCNC(=O)NC)C2 C1(NC(C2C(CC)CCC2)=O)CCCC12CN(C(=O)CC(=O)OC)C2 C1(NC(C2C(C(=O)NC)C2)=O)CCCC12CCN(C(C1(CC)CC1)=O)CC2 n1(C(C(=O)Nc2c(OCC)nccc2)C)cnc2ccccc12 c1(C(N2C(CNC(Cc3scc(C)c3)=O)CC(O)C2)=O)cc2ccccn2c1 C1(C(=O)NCC(CC)NC(=O)C=CCN2CCOCC2)CCCC(C)(C)O1 C1(C(=O)NC(C(=O)N(CC(Cl)Cl)C)(C)C2CCC2)CC1C1CCC1 N1(S(=O)(=O)Cc2cccc(-c3csc(C(F)(F)F)c3)c2)CCC12CN(C1CC1)C2 CCC(C)CCCC(=O)NCC(C)(C1CCC1)NC(=O)Cc1n[nH]c(C)n1 N1(C(C2NCC(O)C2)=O)CCC2(CC1)COC2.c1(OC)c(C=O)cccc1Cl c1(CN2CC3C(C(=O)Nc4ccc(Br)nc4Cl)(C3)C2)c(O)ccc(Cl)c1Cl Cn1nc2ccccc2c1C(=O)NC1CCC(C)(CNC(c2cnccn2)=O)C1 N1(c2nnn(C)n2)CCCC(S(=O)(=O)N2CCCC2OCc2cc(Cl)cnc2O)C1 N1(C(CC2CCC(=O)NC2)=O)CC2(C1)CN(C(C1COC(=O)N1)=O)CC2CO CC1(CNC(C2CN3CCN2CC3)=O)CN(C(C2OCCO2)=O)CCO1 S(=O)(=O)(c1cccnc1NC(C1CCCCC1)Cc1nccs1)NC(COC)C C1(CNC(CCCCOC)=O)CN(C(=O)CS(=O)(=O)NC(C)C)CCC12CCC2 N1(C(CCC(=O)OCC)=O)Cc2n[nH]cc2C1C(=O)NC1(CC(=O)OC)CC1 C(CC(C)(C)C(=O)N1CCC(C)(NC(C2CCCC(C)CC2)=O)C1)SC c1(C(=O)NC(CC=CC(=O)NC2C(CN(C)C)C2)(C)C)ncc(N)cc1C C1(NC(C2(C)CC3CC3C2)=O)COC2(C1)CN(C(=O)C(F)(F)c1csc(Cl)c1)C2 C(=O)(CCCCCCCCC1CC1)NC(C)CCCNC(=O)CCc1nc(O)n[nH]1 CCC(CCCC(=O)NCc1c[nH]ccc1=O)NC(c1cc(OC)cnn1)=O N1(C(c2c(C)cccn2)=O)CC(CNC(=O)CC2(CO)CC2)CC12CCOCC2 Cc1nc2cc(OCC(N3CCCC(C4CNC4)C3)=O)cnc2[nH]1 Cc1cccc(CC(=O)N(C)CCN(C)C)c1I.C12CCC(CC1)N2 c1(C(N2CCC(N(C(=O)CCC3CCC3)CC#C)C2)=O)cc(Cl)cn1C c1(CC)cc(C)c(C(=O)NC(CCN(C(=O)Cc2c(Cl)cnn2C)C)C(C)C)o1 c1(C(=O)NC2C(NC(c3cnc(O)o3)=O)CCC2)cccc2ccoc12 c1(C(=O)NC2CCN(C(c3ncc(C)c(C)c3)=O)CC2C)cc(F)c(F)c(F)c1 O=C1CC2(CCC2)C(C(N2CC3CCN(C(C4CC(OCCO)C4)=O)CC23)=O)CN1 C1(C(=O)NC(C)Cc2ccns2)(N(CCC(=O)OC(C)(C)C)C)CCO1 Cc1c(CN2CCN(C(c3cc4sccc4s3)=O)CC2C)[nH]c2ccccc12 c1(OC)ccc(Cc2nnc(N3CCC(CO)C3)n2CC2CCCCO2)cc1 CN1CCOC(C(=O)NC2CC(C)(NC(=O)CS(N)(=O)=O)C2)C1 C1(CCNC(C2C(NC(c3n(CC)ccc3)=O)CCO2)=O)CCOC1(C)C CCC(F)(F)CC(=O)N1CCC2C(NC(C3C(C4CC4)C3(F)F)=O)C12 C(=O)(C1CCc2nccn21)NCC1N(C(CCC=CC)=O)C2C(C1)C2 CCC(CC(=O)N1CCC(NC(c2cc(F)c(C#N)c(F)c2)=O)C1C)C(C)(C)C c1(NC(=O)NCC23CCC(OC)(CC2)C3)cccc(Cl)c1[N+](=O)[O-] CON(CCC(=O)N(CC(Cl)Cl)C)C(=O)c1ncn2c1CCC2 c1(C(N2CC(N(C(C(C(C)C)O)=O)C)C(O)CC2)=O)cc2c(cc1N)CCCC2 C(=O)(C(F)(F)C(C)O)NCCC(Cn1cc(C(C2CCOCC2)C)nn1)F C12(C(=O)NC3C(CNC(C(COCCOC)(C)C)=O)CC3)CC3CC1C2C3O c12ccc(C)c(c1)OC2=O.n1(CC)cc(CCCON)nn1.OC N1(C(=O)CC2CC2C(F)(F)F)CCCN(C(=O)CCOCC(F)(F)F)C(CO)C1 C12(C(=O)NCC3CC(C(=O)NCC4OCC(C)(C)C4)C3)CCCC1C2(F)F CC1OC2CCC1(NC(C1(C)CC3CCC1O3)=O)C2.N12CCCN(CC1)C(=O)C2 C#CCCCC(=O)NCC1CC(NC(c2cn(C)c(C(F)F)n2)=O)C(O)C1 C(=O)(C(O)CC(F)(F)F)N1CCNCC1.C1(CC(=O)NCCSC)CC2(CC2)CO1 C(=O)(CCC(=O)NC(C1CCCC1)CNC(=O)Cn1c(C)ccc1C)NC c1(CC(N2C(CNC(C(C(C)C)SC)=O)CC2)=O)cc(C(F)(F)F)ccc1C C1(CNC(CCCCc2ccc(C)cc2)=O)CN(C(C2COC2)=O)CC(C)(C)O1 Cc1nc(F)ccc1CN(C)CC1CN(C(C2CC(C)C2)=O)C1 C(=O)(C1CCc2cccc(O)c21)NC(c1cc[n+]([O-])cc1)C.c12cccc(c1)OO2 CCC(C(=O)N(CC)CC1CCCN1C(c1cnc(NC(C)=O)o1)=O)SC c1(NC(=O)NCCC2CN(C(=O)OC)C2)csnc1C(C)C c1(CC(=O)N(CCC)CCNC(=O)CC2(O)CCCC2)coc2cc(Cl)ccc12 N1(C(C(CCCC)(C)F)=O)CC(NC(c2cc(Cl)ns2)=O)C2(CCOCC2)C1 C12(NC(C3(F)CCCN(C(C4CC(C#N)C4)=O)C3)=O)CCC(C1)C(O)C2O C(C(CNC(C1N(C(C)=O)CC(O)C1)=O)S(C)(=O)=O)NC(=O)Cc1cc[nH]n1 C1(N(C(C(=O)NCC)=O)C2CC2)CN(C(C2(CC#N)COC2)=O)CC1C(F)(F)F C#CCCCCCCC(=O)NC1CN(C(=O)COCC2CCCC2)CCC1C N1(C(C=CC)=O)CCCC(N(CCO)C(c2ccc(C3CCCOC3)cc2)=O)C1 C#CC(C)(C)C(=O)N1CC(O)(C2CCCN2C(=O)C(C)OC2CCCC2)C1 N#CC1(C(=O)NC2CCC(NC(c3ccc[nH]3)=O)CC2)CCSCC1 c1(C(N2CC(OC)C(NC(c3cc(C)[nH]n3)=O)C2)=O)cc(Br)c(F)cc1F c1(CC(=O)NC2CCCN(C(C(CC)C(C)C)=O)CC2)nn(C)cc1[N+](=O)[O-] c1(C(=O)OCC)cnc(NNC(=O)C2CCC2C(F)(F)F)nc1C CC1CN(C(C2(CCNC(=O)Cc3cn(C)cn3)CCC2)=O)CCS1=O Cc1cc(C(=O)N(C)CC2COCCN2C(C2CCC2CF)=O)c2nccn2c1 C(=O)(C(C)(C)CCC)NCCC1N(C(CCC=CC)=O)CCC1 CC1CC(C)CCN(C(=O)C(C(C)O)NC(C2CCCO2)=O)C1 C(c1ccccc1C)=CC(N1CCCC(NC(CC=C)=O)C1)=O C1(C(=O)NCC(N2CCN(C)CC2)C(C)C)C2CCC(C2)C1N c1(OC)ccc2c(c1)CCC(CNC(c1c(F)ccc(Cl)c1C)=O)O2 Cc1ccc(C(=O)NCC(C)N(C)C(C2CC3CC3C2)=O)c(Br)c1 C(=O)(C(C)(C)CC(=O)N1CCC(NC(=O)Cc2ccnc(F)c2F)C1)OC c1(C(N=c2cc(C)n(C)[nH]2)=O)n[nH]c2c1CCN(Cc1cnc(N(C)C)nc1)C2 C1(NC(C(C(=O)OC)OC)=O)CC=C(C(=O)Nc2c[nH]c(=O)cn2)C1 C(N=c1[nH]c2cccc(Br)c2o1)C1CN(C(C2(COC)CCCCC2)=O)C(C)C1 N1(C(c2c(CC)cno2)=O)CC(C(=O)NCC(c2ccncc2)C)C(C)(C)C1 N1(C(C)C)CC(NC(=O)CC2CN(C(C3CC(=C4CC4)C3)=O)CC2C)CC1=O C(N=c1cc(C)[nH]c(=NCCc2ncoc2C)[nH]1)C1CC(=C)C1 C1(NC(C2N(C(C(C)C)=O)CCC2)=O)CC2(CCN(C(=O)CC3CC=CC3)C2)C1 Cc1ccc(C(N2CCC(CNC(=O)CC3CCC3(C)C)CC2)=O)c(C)n1 N1(C(CN(CCC)C)=O)CCCC1CCNC(=O)C(C)NC(=O)NC C1(NC(CC(C)F)=O)CCN(C(=O)COc2cc(Cl)cc(Cl)c2)CC1C(N)=O C1(C(N(C)CCN2CCCC2)=O)CC12CC(NC(=O)CC1CSCCO1)C2 c1(C(N2CCC(NC(CCc3ccc(C#C)cc3)=O)C2)=O)cc(O)c(F)cc1N C1(CC(=O)NCCC(C)N(C(=O)Cc2cccnc2)C)C=CCCC1 c1(C(=O)NC2C(C)N(C(C3CCC3)=O)CC2)cc(O)nc(O)n1 CN1CCN(C(C2(C)CCCN(C(=O)CCCn3cccn3)C2)=O)CC1=O c1(CNC(c2cnc(COC)s2)=O)ccc2c(c1)COC2 C#Cc1ccc(F)cc1C(N1CCCC(C)(NC(=O)CN(CC=C)CCOC)C1)=O c1(CNC(C)=O)ccc2nnc(S)n2c1.N12CCCN(CC1)C(=O)C1CC1C2 c1(C(=O)NCC2(COC)CCCN2C(C2CCC2)=O)cc(S(N)(=O)=O)co1 c1(C(=O)NC2(CC=C)CCN(C(=O)CC(C)C(C)C)CC2)nccc2ccsc12 c1(NC(C2N(C(C(CC)(C)O)=O)C3C(C2)C3)=O)cc(Br)cc(C#N)c1 C1(C(=O)NCCC(C)(C)O)COCCN(C(c2cc(Br)ncc2Br)=O)C1 c1(C(=O)OCC)ccccc1C(C)NCc1nc(CO)n[nH]1 Cc1csc2c(N(C34CCC(N)(CC3)C4)C(c3ncnn3C)=O)ncnc12 C123CCC1CN(C2)C(=O)C3.C1(N(C(C=C(C)CN(C)C)=O)C)CCC1C CCCCCCCCS(=O)(=O)NC1CC(NC(c2cnco2)=O)C1 Cc1cnc(C(=O)NCCN2N=C(C)CC2=O)cc1C c1(N2CCC(CNS(NC)(=O)=O)CC2)cc(N2CCCC(C(N)=O)C2)nc(C(C)C)n1 C1(C(=O)OC)CCC2(CC1)CCN2C(c1sccc1NC(C)=O)=O C(=O)(C1CCc2c(Cl)cccc21)NCC(CC)NC(=O)C(N)=O Cc1ccnc(C)c1CNC(=O)CC(C)CNC(=O)C(C)(C)Cl C1(CCNC(Cc2cn(CC)nn2)=O)CCN(C(=O)CCC2CCC2)C(C)C1 C1(C(N(CC(C)NC(=O)C(C)C2CCOC2)C)=O)CCCSC1C N1(C(c2cc(OC)ncc2)=O)CC2CCN(C(=O)CCOCCN(C)C)CC2C1 C(=O)(C1=CCCCO1)N1CC(CCCCNC(c2c(CSC)ocn2)=O)C1 N1(C(C2CCN(C(c3c(C)cccn3)=O)C2C(C)C)=O)CC(C#N)C2(CCC2)C1 C=C(F)C1(N=c2[nH]nc(Br)s2)CCOC1C C1(NC(=O)C=Cc2ccoc2)CN(C(=O)CCc2cnc[nH]2)CC12COC2 c1(CNC(C(N2CCC(CC)C2)c2ccc(-c3cc[nH]n3)o2)=O)ccc(Cl)cc1 C#CC1(C(=O)NC(CO)C(C)C)CN(C(C2CCN(C)C2)=O)C1 N1(C(CCOCC)=O)C2CC1CN(C(C1CCCC(O)CC1)=O)C2 N1(C(C)=O)CC(C2CCCN(CCC3CC3)C2)C1 c1(C(=O)NC2(CNC(C(COC)N(C)C)=O)CC2)ccc(C)c(C)c1O CC1CCCN(C(=O)CC(C)(C)N(C)C(c2ccc(O)cc2F)=O)C1CO C(C)(C)(C(F)(F)F)OC1CN(C(C(=O)NCC(CC)(C)Cl)=O)C1 Cc1ccc(C(F)(F)F)cc1CCNC(C1(C(=O)O)C(C)C1C)=O N1(C(Cc2c(C)n(C)nc2)=O)CCC2CC(C(=O)NCC(C)(C)CN(C)C)C2C1 CCC(Cc1ccccc1C)C(=O)NC1CC(O)(CNC(C2(C(C)C)CC2)=O)C1 Cc1nc2cc(C(N3CCC(NC(=O)Cc4conc4C)C(F)C3)=O)cnc2s1 N1(C(C2C(C)=CCS2)=O)CC(CNC(C2CC(=O)N2)=O)OC(C(F)(F)F)C1 N1(C(c2nc(C)nc(O)c2)=O)CC2CCC1CN2C(c1cc(O)nc(Cl)c1)=O c1(C(=O)NCC#CCNC(C2C(C(=O)OC)CC2)=O)cc2c(s1)CCSC2 c1(OCCN(C(c2ccc(Cl)cc2Cl)CO)C)ccc2c(c1)OCO2 C1(c2n(CCOC)nnn2)(Nc2ccc(CC#N)cc2)CCC(CC2CC2)C1 C1(N(C(=O)C(CC2CC2)NC(c2sccc2F)=O)C)CCCC(O)C1 C(=O)(C(=O)CCC(C)C)NC(CNC(c1c(Cl)cc(C)s1)=O)CO CC1C2C(CCN2C(=O)Cn2cnnc2)CN1C(=O)C1CCc2c[nH]nc21 c1(N(CC(=O)NC)CC)ccnc(C(C)Cc2cnn(C)c2)n1 N1(C(CN(CCOC)C)=O)CC(NC(c2cnc(CC(C)C)s2)=O)CC(O)C1 N1(C(CCC=C)=O)CCC2(CCC(CNC(c3cc(F)cc(F)c3)=O)CC2)CC1 N1(C(C2N(C)CCCC2)=O)CCC(C2CCN(C(C34CCC(CC3)CC4)=O)C2)C1 c1(C(N2CC(NC(c3ccc(C#C)cc3F)=O)C2)=O)ccc2c(n1)OCCO2 N1(C(CNC(=O)C=CC2CCCC2)=O)CCC2CCCC2CC1 C1(CNC(c2cc(OC)n[nH]2)=O)CC(C)(C)CN1C(=O)CC1CCN(C)CC1 C1(NC(c2ncc(C)nc2)=O)CCCN(C(c2cnc(C)o2)=O)CC1 C(=O)(C1=COCC1)N(C(C)CC(N1CCN(C(=O)CC(=O)N(C)C)CC1)=O)CC N1(C(c2cc(C(=O)OC)c(N)cc2)=O)CCC2(CC1)OCCc1cc(Cl)sc12 C(CC(CC)C(=O)NCc1cc(C(=O)NC2CCCC2C(C)C)n[nH]1)=CC C(=O)(CCCCCC(C)C)NC1CC(CNC(CCC(=O)OCC)=O)C1 C1(NC(C(CCC=C)(F)F)=O)CCC2(CCCN(C(C3(CN(C)C)CC3)=O)C2)C1 c1(SCC)cccnc1C(=O)NCCC1CC(NC(C2NC(=O)OC2C)=O)C1 C1(C(=O)NC(C(C)NC(c2ccccc2N(C)C)=O)C)CCC2CC2CC1 c1(C(=O)NC2(COC)CCN(C(COC)=O)CC2)nsc2ccccc12 Cc1c(CC(=O)NC2CCC(NC(C34CC(CC(F)F)(C3)C4)=O)CC2)cnn1C C(=O)(C(C(C)(C)C)c1cn[nH]c1)N(CCC)CCNC(C1COC(=O)N1)=O C1(NC(c2cn(C(C)C)nn2)=O)CN(C(c2cc(Cl)c(Cl)[nH]2)=O)CC12CC2 C1(C)(CNC(C2N(CC)CCC2)=O)CCN(C(c2cc[nH]c2C(C)C)=O)CC1 CC1CN(C(=O)COCC(F)F)CCC1NC(=O)CC1(N2CCCC2)COC1 C1(O)(C(=O)NC2CC(NC(c3n(C)nnc3)=O)C2)CCCC(C)(C)C1 Cc1cc(F)c(C(N2CCC(C(C(C)C)NC(=O)CN(C)C)CC2)=O)c(Cl)c1 N1(C(CC2(C=C)CC2)=O)CCN(C(c2cocn2)=O)CC(CO)C1 Cc1cc(Cl)ccc1CNC(c1cncc(CNC(C2CC2(F)Cl)=O)c1)=O Cc1cccc(CCC(=O)NCCN(C(=O)CSCc2ncc[nH]2)C)c1 N1(C(=O)NC(c2ccc(C)o2)c2ccccc2)CCC2NC(=O)OCC2C1 C1(C(N(CCC)CC2(Cl)CC2(F)F)=O)CCN(C(=O)CSCC(F)(F)F)CC1 N1(C(c2c(SC)cccn2)=O)CCCC12CN(C(C1CCCC1)=O)C2 N1(C(CC2C(C)(C)C2)=O)CCC2(C=C(C(=O)N3CC4(CC(O)C4)C3)C2)C1 c1(C(C)NCC(C)C(=O)N2CCCC2)cc([N+](=O)[O-])cc2c1OCOC2 c1(CNC(CC(C)C(C)(C)C)=O)nn(C)c2c1CN(C(=O)C1=CCOC1)CC2 N1(C(CC(CNC(c2c(C)nco2)=O)C)=O)CCC2C(C(N)=O)C2C1 C1(C(=O)NC(C)C(C)NC(=O)CN(C)CCO)CN(S(=O)(=O)N(C)C)C1 C1(C(=O)NC(CCN(C(CCN(CC)CC)=O)C)C(C)C)OC(C)(C)OC1(C)C C(=O)(C(F)C(C)(C)O)NCC(c1c(OC)cccc1)NC(=O)C=C(C)C N1(C(C(C(=O)OC)C)=O)CC2CCN(C(c3c[nH]nc3C(F)(F)F)=O)CCC2C1 C(C(C)(CO)CO)N(C(C)(C)C)CC.C12(Br)CC1C(=O)OC2=O c1(C(N2CCCC(CNC(C3C(C#N)C3)=O)C2)=O)csc([N+](=O)[O-])c1 c1(C(=O)NC(CNC(c2c(CCC)cccc2)=O)(C)CO)ccc(N)c(F)c1F c1(C(=O)NCC2OCCN(C(C(Cn3ccc(C)n3)C)=O)C2)c[nH]cc(C)c1=O N1(C(c2ccc3c(c2)CC(C(=O)O)C3)=O)CCOc2ccc(Cl)cc21 N1(C(c2ccc(CC3CC3)cc2C(F)(F)F)=O)CC2(OC)CCC2(C(=O)O)C1 N1(C(CC23CC(C)(OC2)C3)=O)CC2CCN(C(c3cc4n(c3)CCCC4)=O)CC2C1 Cc1cc(C)c(C(=O)NC(c2ccccc2)CNC(C2CCCO2)=O)[nH]1 Cc1ccc(C(=O)NCC2CC3CC2CN3C(C2CCCC(C)(C)C2)=O)nc1C C1(NC(C(C)NS(CCC)(=O)=O)=O)COCCN(C(=O)CNC=O)C1 N1(C(C(C)NC(C)(C)C)=O)CCC(CO)(NC(C2CCCCC2)=O)CC1 C1(CNC(C(CC=C)C)=O)CC2COCC2N1C(=O)CNc1cccc(F)c1 Cn1cnn(CC(N2CCC(NC(C3CC(C(C)(C)O)C3)=O)C2)=O)c1=O C1(NC(C(CC2CC2)NC(=O)CCCC2CCC2)=O)CC2(C1)CC21CCC1 c1(CC(N2CCCC(COCCOCC)C2)=O)cccc2cnccc12 c1(C(=O)NCCCOCCNC(COCCC)=O)cc2ccc(C)cc2[nH]1 N1(C(C2(C(=O)OCC)CC2)=O)CC(NC(c2ccn(C)c2)=O)CC2(CCC2)C1 CS(=O)CCC(=O)NCC(C1CCC1)NC(=O)CCc1cccnc1Br Cn1nc(C(=O)NCc2ccc(C(=O)NC3C=CCC3)cc2)cc1O c1(CC)[nH]nc(C(=O)NC23CC(CNC(c4ccc(OC)cc4)=O)(C2)C3)c1Cl c1(OCC(N2CC(CN(C)C(C3(C)CC(F)C3)=O)OCC2)=O)ccc(C#N)cc1 c1(C(=O)NCc2c(CCNC(=O)Cn3cncn3)ocn2)scc2c1OCCO2 c1(N2Cc3c(ccc(C)c3)C2)ccc(S(=O)(=O)N2CCC2)cc1F.C12CN(CCO1)C2 Cc1cc(NC(=O)CN2CCN(C(=O)CCN(C)C)CC2)cn2ccnc12 C1(S(C)(=O)=O)(C(=O)NC(C)CCNC(c2cc(C(C)(C)C)c[nH]2)=O)CCC1 Cc1oc(CO)cc1C(=O)N(CCC(C)(C)NC(c1ccncc1N)=O)C C(C(C)(C)C(=O)NC1CCN(C(=O)CCC2CCCCCC2)C1)SC c1(OC)cc(-c2c[nH]nc2NC(c2cc(O)ccc2Br)=O)cnc1F c1(C(N2C(C)CC(NC(COCC#C)=O)C2)=O)cc(N)cc(O)n1 Nc1c(C(N2CCCC(O)(CNC(=O)C(O)CC(N)=O)C2)=O)cccc1[N+](=O)[O-] C(=O)(C(C)(C)S(C)(=O)=O)N1C(C)C(NC(C2CC2C(=O)NCCO)=O)CCC1 C1(CNC(C(C)Sc2c(C)ncs2)=O)(CNC(=O)CCNC(N)=O)CC12CCC2 c1(C(N2CC3CCN(C(C=CCCC)=O)CC3C2)=O)ccc([N+](=O)[O-])c(C#N)c1 Cc1cc(C(=O)NC2CCCC2CNC(=O)CCc2cccs2)c(C)n1C c1(C(N2CC(C3(NC(C4CC4Cl)=O)CC3)C2)=O)cc(Cl)c2ccccc2n1 C(=O)(C#CC1CCCOC1)NCC1C(C)CCCN1C(C1CC1F)=O Cc1cncc(C(=O)NCC2CC(C)N(C(=O)COCC3CC3)C2)n1 C1(C(=O)NC(C)(C)CCNC(=O)CC2CC3CC3C2)CCC(F)(F)C1 C(c1cccc(CO)c1)=CC(=O)NCC1N(C(C(C)OCC)=O)CC=C1 C(=O)(CC(O)CCC(C)CC)NC(CN1CCN(C(CCC#C)=O)CC1)C Cc1nn2cc(C(N3CCCC(c4noc(C5CC5)n4)C3)=O)nc2s1 CC(CC(=O)N1CC(CN(C(=O)C(C)CSC(F)(F)F)C)C1)CC(C)(C)C c1(C(N2CC(NC(=O)CNS(=O)(=O)C3CC3)C(F)C2)=O)ccc2cccnc2c1 CC(C)C(O)CC(=O)NCc1cn(-c2ccc(Oc3ccccc3)cc2)nn1 c1(C(CC)C(=O)N(CC(C)NC(C2(F)CN(C)C2)=O)CC)ccc(OC)cc1 C1(NC(=O)Cc2csc(Cl)c2)C2CCN(C(=O)C(=C3CCCCC3)F)C12 c1(C(=O)NCCNC(C(CCCOC)C)=O)cc2ccncc2o1 CC1COC2(C1)CN(C(C13CCCC1(F)CN(C(=O)OC(C)(C)C)C3)=O)C2 n1(CCN(C)C)cc(C(N2CC(O)(C(C)NC(=O)CC3CCC(O)C3)C2)=O)cn1 C12(C(N(C3CCN(C(C(C)CN(C)C)=O)C3)C)=O)C3C4C1C1C2C3C41C c1(OC)ccc(Cl)c(C(=O)N(C)CC2CCN(C(C3(C#N)CC3)=O)C2)n1 C1(OC)CC(C(=O)NCc2ncccc2Br)N(Cc2ccccc2Cl)C1 N1(C(c2nc(CCCCC)sc2)=O)CC(C(F)F)C(N)C1 c1(C(C)=O)cc(C(=O)NCCOC2CCN(C(C3(C)CSC3)=O)C2)ccc1O CC1CN(C(C2C3CN(C(=O)CN4CCCC4)CC23)=O)CC1NC(=O)C1CC1 c1(C(=O)NCC2=CCN(C(C(C)C(C)(F)F)=O)CC2)cc(Cl)c2n[nH]cc2c1 C(C1CCCCC1)=CC(N1C(C)CC1C(=O)NCCC(Cl)Cl)=O C1(CC(N)=O)(NC(c2scnc2Cl)=O)CCN(C(C2CC2[N+](=O)[O-])=O)CC1 C(=O)(CCCC(=O)N(C)C)NC1CCCC(CNC(C2CC(COC)C2)=O)C1 C(c1ccccc1)=C(C(=O)NCC(CCOC)NC(C1C(COC)C1)=O)C N1(C(c2cn[nH]c2)=O)CCC2CCN(C(c3cc4n(n3)CC3(CC3)C4)=O)C2C1 c1(C(=O)NCCN(CCC)C(C2(C)CC=CCO2)=O)cc(C)[nH]c(=NC)n1 N1(C(CS(=O)(=O)NC)=O)CCN(C(=O)COCC(=O)NN(C)C)C(C)CC1C C(C(COC)CC(=O)NC(C1CCCCN1C(c1cscc1F)=O)C)OC CCC(C)C(C(=O)N1CC(NC(=O)CCc2cnccc2C)C1)NC(C)=O C1(CN(C(C(C)NC(CC)=O)=O)C)CCCCN1C(=O)CC(C)(C)O CCC(CCC(=O)NC1(COC)CC1)NC(C1CC(=O)N(C)C1)=O N1(C(c2c(COC)ncs2)=O)CC(CNC(=O)CCC2CC2(C)C)CC1(C)C CC1(C)OCCOC1CC(=O)NC1(CF)CN(C(c2ccon2)=O)C1 Cc1nc(N2CCC(CC(C)(C)C)CC2)nc(N(C)C)c1N C1(CNC(C=CCOC)=O)CC2CCC1N2C(C1CN(CC(C)C)C1)=O C1(NC(c2cc(C(F)(F)F)n[nH]2)=O)CCCN(C(c2ccc(F)o2)=O)C1 c1(CC)ccc(C(=O)NCC2CCN2C(C2CN(C(=O)N(C)C)C2)=O)nc1 c1(CS(=O)(=O)NCC2CCC(NC(CCOC)=O)CC2)ccc2ccsc2c1 Cc1ccc2c(CC(N3CCC(N(C(=O)C=CC4CC4)C)C3)=O)coc2c1C C(=O)(C(O)CC(C)(C)C)NCCC(C)NC(c1cc(N)cc(O)c1F)=O c1(C(N2C(C(=O)NCCn3ncccc3=O)CCC2)=O)ccnc(Cl)c1O C1(CNC(c2cc(OC)c(Cl)s2)=O)CCCCCN1C(=O)Cc1nocc1C Cc1nc2ccccc2c(C)c1C(=O)N(CC(O)CNC(=O)C(C)(C)N(C)C)C N1(C(Cc2cccc(C)c2F)=O)C(C)CN(C(=O)CC(O)CN(C)C)CC1C c1(CC)cccc(Br)c1NC(=O)NC1(C(=O)OCC)CCCCC1 C1(NCc2ccc(NC(CC3CCN(OC)C3)=O)nc2)COc2ccccc2O1 c1(OCC)cc(-c2nc(-c3ccccc3)nn2CC(F)F)oc(=O)c1 n12ncc(c1C)C(=O)NC21CC1.C(O)(C(F)(F)F)C1(C(N2CC(OC)C2)=O)CCC1 c1(C(=O)NCCN(C(=O)C(C)(C)c2ccccc2)CC)cnnn1C1CCCC1 C1(N(C(c2cn(CCCC)nn2)=O)C)CN(C(C2(C(N)=O)CCC2)=O)CC1O c1(C(=O)NC2C(CNC(C3CCC(NC(N)=O)CC3)=O)CC2)cc(F)ccc1F c1(C(=O)NCCN(C(=O)COc2ccc(F)c(F)c2)C)ccc2ccoc2c1 N1(C(c2c(CC)scn2)=O)CC(CNC(c2oc(C(C)C)nc2C)=O)C2(CC2)C1 C(=O)(C1=C(C)OCC1)NC(C(=O)N(C1CCOCC1)CC#C)CC1CC1 N1(C(Cc2ncc(C)s2)=O)CC2(CCN(C(c3ccc(C(F)F)cn3)=O)CC2)C1 C12(NC(CCC)=O)CCCC(CN(C(=O)Cc3c(C)cccc3F)C1)C2 C1(CCNC(CN(C(C)=O)C)=O)CN(C(c2cscc2F)=O)CCO1 C(CCC(=O)NC(C)CNC(c1ccn(COC)n1)=O)=CCC=C C(CC(=O)Nc1cccc2nsnc12)(C(C)(C)C)N(CC)CC c1(C(C(=O)NCCSC)N(C)CC2CC2)ccc(C2CCC2)nc1.c1cnc(Cl)s1 C(=O)(C1=CC2CCC(C1)C2)N1CCCC(CN(C(=O)CC2(C)CCC2)C)CC1 c1(CC(=O)NC(C(C)C)C(C)NC(=O)CCCc2cccs2)ncn2c1CCC2 N1(C(c2c(C)nsc2)=O)CCC(NC(=O)CCSCC(C)C)C(CO)C1 C=CC1CCN(C(=O)CCCCNC(C2CCCN2CC)=O)C1 N1(C(CCN(c2ccccc2)C)=O)CC2CC1C2C(=O)NCc1ccnnc1O Cc1cc(C)[nH]c(=NCC2CCN(C(c3c[nH]nc3C(C)C)=O)CC2C)n1 c1(CCCCC)cc(CN2CC(C)C(F)(F)C2)c([N+](=O)[O-])o1 c1(CC(=O)NC2C(NC(CCC(CC)C)=O)CCCC2)ccc2ncccc2c1 N1(C(c2ccc(CC)o2)=O)CC2CN(C(=O)CCc3ncc[nH]3)CC2(C)C1 N1(C(C2(C)C(C)OCC2)=O)CCC(C)(C(N2CC=CC(O)C2)=O)CC1 C(=O)(C#CC(C)(C)CNC(c1csc(O)n1)=O)NCc1c(C)cccc1C c1(C(=O)NC(CNC(C(CCC)O)=O)C(C)C)cc(Cl)c(Cl)[nH]c1=N C(=O)(C1CN(CC)c2ccccc21)NCC1(F)CCN(C(CCCCC=C)=O)C1 c1(C(CCO)NCCCN(C(C(=O)NC2C(C)C2N)=O)C)ccccc1 C1(NC(C(c2ccn(C)n2)(C)C)=O)CC(NC(c2cc(C(F)F)[nH]n2)=O)C(O)C1 N1(C(CCOC)=O)CCC2CCN(C(c3ccnc(O)c3)=O)C2C1 CCC(C(=O)NC1(CF)CN(C(c2cncc(C3CC3)c2)=O)C1)C(C)C c1(OCC)ccc(NC(=O)NC2CC(C(=O)OC(C)(C)C)(OCC)C2)cc1 N1(CC)CCOCC1CC(N1CC(C(N)=O)(CNC(C2CCC(=O)N2C)=O)C1)=O C1(C(=O)NC(CN(C(COC(CC)C)=O)C)C)Cc2cc(Cl)ccc2O1 N1(Cc2ccc(OC(C)C)nc2)CCC(NC(c2ocnc2C(F)F)=O)C(C)C1 C1(NC(CC(CN(C)C)C(F)F)=O)CC1C1CCN(C(=O)CC2CC2)CC1 C12(NC(c3cc(N(C)C)ncc3)=O)CN(C(C3(O)CCC3)=O)CC1CS(=O)(=O)C2 CC1=NOC2(C1)CC(C(N1CCC(CF)(NC(C3CC4CCC3O4)=O)C1)=O)C2 C#CCCC(O)C(=O)N=C(C)C.C1CCOCCO1.C(=O)C=CC C(=O)(C1=NN(C)C(=O)CC1)N1CC(NC(c2cc(C)sc2C)=O)C2(C1)CC2 C1(C(N(C2CN(C(C3(C#N)CCCOC3)=O)C2)C)=O)CC2(CCO1)CC2 c1(C(N(CCNC(C(C(C)O)C)=O)CC2CC2)=O)cccc2c1ccn2C C1(COC)CC(CNC(C2CCC(=O)N2C)=O)N(C(=O)CCCCC2CC2)C1 c1(OC)cnc(C(N2C(C)CCC2C)=O)c(F)c1.c12ccc(cn1)c(=O)[nH]2 CC(C)CC(C(=O)NC(C)C(=O)Nn1cnnc1)C(N)=O CC1OCCCC1C(=O)N(CC(O)CNC(c1ccnc(C(F)F)c1)=O)C C1(CNC(=O)CN2CCCCC2)CC2CCC(C1)N2C(C1(c2ncco2)CC1)=O c1(C(N2C(CC)CN(C(c3ccc(OC)o3)=O)CC2)=O)cc(OC)c(O)c(Cl)c1 C(=O)(C1Cc2ccc(F)cc21)NC(C)CN(C(=O)Cn1cc(Cl)c(O)nc1=O)C CC1CN(C(=O)C(CCN(C)C)NC(c2ccccc2F)=O)CC(=O)N1 N1(C(C(C)(C)n2cccn2)=O)CCC(c2nc[nH]n2)CC1.C1(=O)C=CS1 C1(C(=O)NCC(CCOC)NC(=O)Cc2cc[nH]n2)CCCC(=O)N1 C(=O)(CCCS(N)(=O)=O)N(C1CCCCN(C(C2CN(CC)C(=O)CC2)=O)C1)C C(=O)(CCCC(C)(C)CC)N(C)CC1N(c2nnc(C)s2)CC(F)C1 c1(CC)cnc(O)c(C(N2CC(NC(=O)CC3CCCC3O)C(O)C2)=O)c1 C1(C(=O)NC2CCN(CC)CC2)(NC(c2[nH]ccc2COC)=O)CCC(C)(C)C1 N(C)(C(=NCCn1cccc1)NCC1CCCO1)C(c1cn(CC)nc1)C C(=O)(C(C(C)NC(=O)CN1CCCCC1)C(C)C)NCC1CCC(OC)C1 C(C(N=c1ccnc(CC2CCCC2)[nH]1)C1CC1)NC(CCC(CCC)CC)=O N1(C(c2cc(Cl)cc(Cl)c2Br)=O)CCn2cc(O)c(=O)cc2C1 C#CCC(CN=c1[nH]c(=NCC2CCOCC2(C)C)[nH]c2cccc(F)c12)OC C1(CNC(CCN(C)CCO)=O)(CNC(c2ccnn2CC#N)=O)CCOCC1 N1(C(C(CC)COC)=O)CCC(C(=O)NCC=CBr)C1(C)C c1(C(=O)NCC(CNC(C2(C(F)F)CC(=C)C2)=O)O)nn(C)cc1CC CC1(CNC(c2c(Cl)csc2Cl)=O)CCN(C(=O)C=CC2CCOC2)CC1 CC1CCCc2cc(C(=O)N(CCCCNC(C3CCCCCCC3)=O)C)nn21 C(=O)(C1CCc2nccn21)N1CCC(C(N(C(C)C2CC2)C)=O)CC1 c12ccc(cc1)CC(=O)N2CCC#N.C1(COCCN)CCCO1 CC1CCC(C(N2CC(O)(CN(C(=O)Cc3nncn3C)C)C2)=O)O1 CN1CCC(C(N2CC(O)CC2C(=O)NC2(C3CC3)CCC2)=O)C1=O CN1CC(C(N2CCC(OCCN(C)C)C2)C(=O)NCc2ccco2)CC1=O C(C)(CCC(=O)NCC1(CC2CC2)CCCO1)SC.N12CCC(CC1)NC(=O)C2 C1(C(=O)NCC(CC)(CC)Nc2cc(C)c(C(=O)OC)cn2)CCCC(C)(C)C1 N#Cc1cc(S(=O)(=O)NCC2CCCCO2)ccc1NCc1cnn(CCF)c1 C1(C(=O)NC2C3(NC(=O)C4=NOCC4)CCC(C2)C3)CCc2nc[nH]c2C1 CC1CCN(C(=O)CCC(=O)N(C)C)CC1CC(=O)NC1CCCCC(=O)N1 N1(C(C(=O)NCC(N2CCC(O)CC2)=O)=O)Cc2ccnn2CC(C(=O)O)C1 c1(OCC=C)cc(Cl)ccc1C(=O)NCC(CC)NC(=O)CCN1CCC(F)C1 Cc1ccc(C)c(C(=O)NC2CCCC(C(=O)NC3CC(=C4CC4)C3)CC2)c1 c1(CC)ccnc(C(=O)NCCC(O)C(=O)NC2CCCC2(F)F)c1 C1(n2cc(-c3cc(C)oc3)nn2)(NC(C(=O)NC2CC2)=O)CC(C)(C)C1 Cc1ccc(F)c(NC(=O)C(C(C)O)NC(=O)C(C)n2cccn2)c1 C=CCC(CNC(=O)C(=O)N(C)C)C(=O)NCC(c1ccccn1)C C12(NC(C(C(C)C)C)=O)CCC(CC1)N(C(=O)CCCC1CCC1)C2 c1(OC)cc(OC)cc(CC2CCCN2C(c2nc(=O)n(C)[nH]2)=O)c1 c1(C(N2CCC(NC(=O)Cc3cnc[nH]3)C(F)C2)=O)cnc2scnc2c1 CC1CCNC(=O)C1NC(=O)NCc1ccc(Sc2c(F)cccc2F)cc1 N1(C(c2cnc(C)[nH]2)=O)CC2CN(C(C3(C4CCCO4)CC3)=O)CCC12 N1(C(c2c(N)cc(F)cc2)=O)C2CCC1CN(C(=O)C(F)CC1CCCC1)CC2 C1(O)(C(CNC(c2ccc(C)o2)=O)C)CCN(C(=O)C=Cc2scnc2C)C1 c1(C(=O)NC(c2nocc2NC(c2csnn2)C)C)cc(C2CCC2)no1 C1(C(=O)NCC2(F)CC(NC(c3c(CC)occ3C)=O)C2)CCC2C1C2(F)F C(=O)(CCCC(F)F)N(CCCCN(C)C(c1cnc(CN)[nH]1)=O)C c1(SC)cc(CNC(c2cn(-c3ccccc3)nn2)C)ccn1 C=CC(CC)C(=O)NC1C=CC(CNC(c2cn(C(C)C)cn2)=O)C1 c1(C(N2CC(C)OC(CO)C2)=O)cnn2ccnc(N)c12 c1(NC(c2ncc(-c3ccccc3F)cc2C(F)(F)F)=O)nccc2[nH]ccc12 CN1CC2CC2(NC(=O)C(C2CCC2)NC(=O)CC2CCCOC2)C1 C(C)(C)(CCC(=O)N1CCCC(N)CC1)CCn1cc(CCOC)nn1 CCC(CC(=O)NCC12CCCC1N(C(=O)COCC(C)C)CC2)C(F)F N1(C(c2ccc(C)cc2)=O)CC2CN(C(c3onc(C)c3C)=O)C2C1 N1(CC(=O)NC2CCC(NC(=O)Cc3ccoc3)C2)Cc2ccccc2C1=O c1(C(N2CC(COC)(CNC(=O)C(C)N(C)C)C2)=O)cc(C(C)C)n(C)n1 c1(OCC(N2CCC(F)(C(=O)NCC3CN(C(C)=O)C3)C2)=O)c(C)occc1=O C(C(CC(C)C)c1nc(-c2ccccc2)nn1CC1CCCOC1)NC(C)=O CCCC(C(=O)NCC(C)(F)CNC(C1OCC2CCCC12)=O)C(C)C N1(Cc2ccc(C(=O)NC(C)(C)CN3CCOCC3)nc2)CCN2CCCC2C1 N#Cc1cncc(C(=O)NCCCCCCNC(=O)Cc2nc[nH]n2)c1 c1(SC)cc(C)ccc1-c1cc(C(N2CCCC(C)CC2)=O)ccn1 Cc1cc(C(=O)N(CC(C)CNC(=O)C(CC(F)F)C2CCC2)C)ncc1N c1(C(N(C)CC2CCCCN2C(C2C3COCC23)=O)=O)c(Cl)ccc(O)c1N C(N=c1[nH]c(=NCCC2CCC(=O)N2)[nH]c2ccc(Cl)cc12)C1(C)CSC1 c1(C(=O)OCC)cnc(NC2CCCN(C(c3cc(C)c(Cl)s3)=O)C2)nc1 C1(CNC(C2(C)C(C)C2)=O)CCN(C(C2(CN(C)C)CCCCC2)=O)CC1 C(C1=CCN(c2cc(C(N)=O)nc(Cl)n2)CC1)NC(CCN(C)C)=O CCCC(C)(C)C(=O)NC1CCOCC1NC(c1csc(Cl)c1Cl)=O CN1CC(NC(C2CC3CCC2N3C(=O)C(C)(C)C(F)F)=O)C(C)(C)C1 c1(C(=O)NC2CCCC(NC(C(C)(C)OC)=O)CC2)cc(F)c(F)c(F)c1 c1(N2CC3C(CNC(C4CC(C(C)C)OCC4)=O)C3C2)[nH]cnc2nc(Cl)cc1-2 n1(CCC)ccnc1C(F)(F)C(=O)N(C)CCN(C)C(C1(F)CCOC1)=O c1(CCNC(=O)NC(C(=O)NC)Cc2ccccc2)ccc([N+](=O)[O-])cc1 C12(C(N(CC(=O)NCC(C)(CC)CO)CC#C)=O)CCCC1C2(F)F c1(CC)oc(C(=O)NCC2C3CN(C(C4(Br)CC4(C)C)=O)CC23)cc1C c1(NC(C(=O)N(C2CCC(CNC3CC3)CC2)C)=O)ccc(S(N)(=O)=O)cc1 C1(C(N2CCC(C)(NC(c3ccc(N=[N+]=[N-])cc3)=O)C2)=O)CC2(COCCO2)C1 CC1CC(C)N(C(=O)Cn2cc3ncccc3n2)CCN1C(C1CCCC1)=O c1(C(C)NCc2c(OC)n(C)nc2)cc(OC)cc(C(C)C)c1 C1(NC(COc2c(C)cc(Cl)cc2)=O)CCCC12CCN(C(=O)CCF)CC2 C1(NC(COCC=C)=O)(COC)CCN(C(c2ccnc(C(C)C)n2)=O)C1 N1(CC)CCOC(C(N2CCC(CCN(C(=O)CSc3cccs3)C)CC2)=O)C1 O=C(CCC(=O)NCC(F)CNC(C1CC=CCC1)=O)c1ccc(Cl)cc1 C1(CC=C)(C(=O)OC)CN(C(=O)Nc2nc(C(F)(F)F)cs2)CCO1 c1(C(=O)NCCC2(OC)CN(C(C(CCOC)C)=O)C2)cc(S(N)(=O)=O)cn1C C1(NC(CCc2n(CC)ccn2)=O)CC(CO)N(C(C2CC(C)(CC)C2)=O)C1 C(=O)(CCCCC(C)(C)C)NCC(C)C(N1CC2COCC(C2)C1)=O Cc1cc(C)c(C(N2CC(CNC(=O)C(O)C(F)(F)F)C3(CC3)C2)=O)c(O)c1 c1(C(N2CCN(C(C=C(C)C)=O)CC2)=O)ccc(Cl)cc1Nc1ccccc1 n1(C2(C)CC2)cc(NC(=O)COC(=O)CCN(C)C(=O)OCC#C)cn1.CC.OCC C(CN=c1nc2scnc2c(NCC2CCOC(CF)C2)[nH]1)c1n(C)nnc1Br O=C(C1=CCCCC1)N1CCCCC1C1CCN(c2ncnc(=N)[nH]2)C1.CC=O C1(O)(CCNC(c2ccc[nH]2)=O)CCCN(C(=O)CCCCNC(N)=O)C1 c1(NC(CNC(C2(C)CC(=C)C2)=O)C2CCC2)ccnc(C(=O)OC)n1 C1(CCCNC(CCSCCCC)=O)CCCN1C(=O)CCCc1csc(C)n1 C(=O)(C1OCCc2c(O)cccc21)N1CCC(C)N(C)C(C)C1 c1(C(N2C(C)CCN(C(=O)Cc3cnns3)CC2)=O)ccc2c(c1)B(O)OC2 c1(C(=O)NCC2(C)N(C(C(CCC)OCC)=O)CCC2)cc2n(n1)CCOC2 c1(C(=O)NC2(C)CCCN(C(C=C(C)C3CC3)=O)C2)nc2nc(C)cc(C)n2n1 CC(CCCC(=O)NCCC1CCOC1(C)C)NC(=O)CCCN(C)C1CC1 Cc1nnc2c(NC(c3ccncc3-c3cccc4nccn34)=O)cc(Cl)nn12 C(=O)(C(F)(F)C(F)F)NCC(C)(C)NC(C(C)OCCC(C)C)=O C(=O)(CC=CCC(C1CSC1)C)NC(=O)CCC1(C)CC1 N1(Cc2n(C)cnn2)CCC2(CC1)CC2NC(=O)CCc1cn[nH]c1 Cc1onc(CO)c1C(=O)NCC1CN(C(=O)Cc2cscn2)CCO1 C1(N(C(C(N2CCOC2=O)C)=O)C)CCCCC1N(C)C(c1ccncc1)=O c1(C(N2CCC(F)(CNC(c3cn[nH]c3)=O)C2)=O)c[nH]c(=O)c2ccncc12 C1(NC(c2c[nH]nn2)=O)CC2CC(C1)N(C(=O)CN1CCc3sccc3C1)C2 c1(CC)nc(C)n(C)c1C(=O)N(C(C)CCNC(c1coc(C)n1)=O)C C=C(C)CCCC(=O)N1CCC(O)(CC(=O)NCCCn2ccnc2)C1 Cn1c(=O)n(C2CC2)c2ccccc12.C12(CCNC1)c1ccc(cc1)-c1noc2n1 C1(C=C)(C(N(CC=C)CCC)=O)CN(C(=O)C(C)n2ccnc2)C1 c1(C(N2CCC(CN(C(C(C)C(C)(C)O)=O)C)CC2)=O)cc2cnc(Cl)cc2s1 n1(CC(C)C)cc(C(=O)NCC)cn1.C1(CC(=O)NCC2(N)CCC2)OCCC1C C1(CCC(=O)NC2CCS(=O)CC2)CCN(C(=O)C(C2CCOCC2)F)CC1 N1(C(CCCC#C)=O)CC2ON=C(CNC(=O)C=Cc3cocn3)C2C1 Cc1cccnc1CCNC(C1(NC(C2CN(C)CCO2)=O)CC(CO)C1)=O c1(C(=O)NC2CCCC(NC(C(CC)(C)F)=O)C2)cccc(Br)c1Cl c1(C(=O)NC(C2CN(C(C(CCC)NC(C)=O)=O)C2)C)ccc(S(N)(=O)=O)s1 O=C(CC1=CCCC1)NCC1OCCC1C(=O)NCC(O)C1CC1 c1(CC(CN(C(CCSCCC)=O)C)NC(=O)CC2CC=CCC2)ccccc1 c1(CNC2C(C(=O)Nc3onc(C)c3Br)C2)cccc(Cl)c1[N+](=O)[O-] C1(CC(=O)NCC2N(C(C(C)OC)=O)CC2)CCCS1(=O)=O N1(CC(C2CCC(C(=O)OC)C2)=O)CC=CC1(C)C c1(OC)ccnc(N2CCOCC2CC(=O)Nc2nc(C)c(I)s2)n1 CC(C)CCCC(C)C(=O)NC1(C(=O)NCc2ccn(C)c(=O)c2)CC(F)C1 c1(C(N2C(C3CCN(C(C(CC)C)=O)CC3)CCCC2)=O)c[nH]nc1[N+](=O)[O-] C1(NC(CN(C)S(N)(=O)=O)=O)CCC(NC(=O)CC2(C(F)(F)F)CC2)CC1 Cn1ccc(C(=O)NCC2CN(C(=O)C=C(C3CC3)C3CC3)C3CC23)cc1=O C1(NC(C2CCC(NC(CNC(=O)NC)=O)C2)=O)(CO)CC2(CCC2)C1 Cc1cc(C(=O)NCC(O)CNC(=O)C(C)c2ccsc2)c(C)n1C(C)C N1(C(C(=O)N(C)C)=O)CC(CNC(c2cc(Cl)ccc2C(F)(F)F)=O)CC1(C)C C(=O)(CCNC(C)C(=O)NCC(N1CCCC1)=O)OC c1(C(=O)NCC(CN(C(c2c(C)nc(C)[nH]2)=O)C)O)cc2c(C)ccc(F)c2[nH]1 CC(C)CC(C(=O)N1CCOCC1CCNC(C1(C(N)=O)CCC1)=O)N(C)C1CC1 C1(CN(C(=O)C=CCN2CCCC2)C)CCN(C(C2CC2c2cnc[nH]2)=O)CC1 Cc1cc(NC(=O)C(c2cccc(C#N)c2)C)ccc1NC(=O)C#CC(C)(C)C c1(NCCCNC(c2ncc(C)cc2C)=O)ncnc2c1nnn2C1CC1 S(=O)(=O)(c1cnc(NC23CCCC2C3(F)F)c(Cl)c1)NCC1CCCN(CC)C1 C1(CNC(c2c(C)ncs2)=O)CCCCCN1C(=O)CC1CCSC1 C1(NC(=O)CCn2cnnn2)CCC2CN(C(c3cnnc(Cl)c3)=O)CCC2C1 N1(CC=C)CCC(N2CC(NC(C3CC3(F)F)=O)C2)C1=O.c12ccccc1CO2 C(c1ccc(OC(C)C)c(C)c1)=CC(=O)NC(CCNC(C(C(C)C)SC)=O)C C(C(O)CN=c1[nH]c2cccc(F)c2o1)NC(C1(O)CCOC1)=O N1(C(c2c(C#C)c[nH]n2)=O)CCN(C(=O)CSc2nncn2C)C2CCCCC12 C1(CNC(CNC(C(C)CCN(C)C)=O)=O)CCC2(CC2)CO1 C1(CC)CN(C(=O)CN(C)CC)CCC1NC(c1ccc(OC)nc1)=O Cc1cccnc1C=CC(=O)NC1CCCCN(C(C23CCC(CC2)CC3)=O)C1 c1(C(N2CC3N(C(COc4ccc(OC)cc4)=O)C3C2)=O)cnc(Cl)c(Cl)c1 C12(C(=O)NCCCOCCCNC(c3cc(OC)n[nH]3)=O)CC1COC2C C1(N(C(=O)CC2OCCCO2)CC)CCN(C(c2cccnc2)=O)CC1 c1(C(=O)NC2CCCN(C(C3CC(CCC)C3)=O)C2C)sc([N+](=O)[O-])cc1Cl C#Cc1cnc(N(CCCNC(=O)C=CC(=O)NC2CC2)C)nc1 C(C(CC(C)C)C(=O)NCC(C)CC1CC1)NC(c1c(CC)n(C)nc1)=O CC1CC2(CC(C(=O)NC3(CNC(=O)CC4CCCCCO4)CCC3)C2)C1 CS(=O)(=O)CCCC(=O)N1CC(C(=O)O)C(Cc2nc3ccccc3s2)CC1O C1(OC)CCCN(N2CC(c3cccnc3)(Nc3ccccc3)C2)C1 N1(C(=O)OCC)CC2CC2(C(=O)Nc2nccc(C(C)(C)O)n2)C1 N1(c2snc(C(C)(C)C)n2)CCC2(CCCN(C(=O)CC3CCCCO3)C2)C1 C(c1ccc(F)cc1)=CC(=O)NC1CN(C(c2c(C(F)(F)F)ncn2O)=O)C1 O(C1CCCc2ccccc21)S(CCNC(N1CCC(CO)C(F)(F)C1)=O)(=O)=O c1(C(=O)NC(CCOC)CNC(=O)CCC(C)SC)cc(F)cc(N)c1F N#Cc1ccccc1CC(N1CCCC(NC(=O)C(C2CCCCCC2)O)C1)=O N(C(=NCCCCl)NCC(C)CO)CC(C)CC1CCCCC1.C1C(=O)N1 N1(CC(=O)N(C2C(NC(CCCCOCC)=O)CCCC2)C)CCCCCC1=O C1(C(=O)NCC2CCN(Cc3c[nH]c(Br)c3)C2)CC2CCNCC2C1 N1(C(c2onc(C(C)(C)C)n2)=O)CCOCC(CNC(c2coc(O)n2)=O)C1 c1(OC)ccc(-n2nnnc2C(C(C)(C2CC2)OC)Nc2cc(C)nn2C)cc1 c1(C(=O)NCCC(C)NC(c2cc(C(CC)CC)no2)=O)nccnc1C c1(OC(CC)C(=O)NCCN(C(c2cncs2)=O)C(C)C)ccccc1F Cc1nn(C)c(Br)c1C(=O)NC1CC(CNC(C2(C)CC(C)C2)=O)C1 c1(C(=O)NC2(CNC(C3CC(C#N)C3)=O)CC2)cc2cc(Cl)ccc2[nH]1 c1(COCC)noc(CONC(=O)Cc2nc(-c3ccccc3)no2)n1 N1(C(CCNS(C)(=O)=O)=O)CCN(C(=O)C(c2ccccn2)O)CCC1C C(C(=O)NCC1CCCCN1C(=O)CCOCC1CC1)(C(C)(C)C)OC c1(C(=O)NC2(CNC(C(CC=C)(C)O)=O)CCC2)cc2c(ccn2C)[nH]1 C(=O)NNC1CCCC1.N1(CN=[N+]=[N-])CCC(C(C)O)CC1 C#Cc1cn(C)nc1C(=O)NC1CC2CCC1(NC(c1cccc(C)c1C)=O)C2 C=CC1(C(N2CC(C)(NC(=O)C(c3ccnn3C)C)C2)=O)CCC1 C(=O)(CC(C)(O)C1CC1)NCCCN(C)C(c1ccn(C(C)(C)C)n1)=O c1(-c2cn(CSc3nc(C)sc3)nn2)cnn2c1CCC2.C12CCCC(C1)C(=O)N2 C(=O)(N=c1cc(C2CCCO2)[nH][nH]1)OC(=O)CNC(c1cc(B(O)O)co1)=O C1(C)(CN(C)C(c2cnco2)=O)CCCC1NC(c1coc(-c2cccs2)n1)=O CCC(CC)C(C(=O)NCc1nc(C(N2CC3C=CC3C2)=O)co1)OC C1(C(N2CC(NC(COCCC#C)=O)C(C)(C)CC2)=O)CN2CCCCC2CO1 N1(C(C(CC)NC(N)=O)=O)CCC(NC(=O)Cc2ccc(F)cn2)C12CC2 C1(NC(Cc2n(C(C)C)ncc2)=O)CC12CCN(C(=O)C(F)OC(F)(F)F)CC2 c1(OC)cccc(C2CCN(c3nnc(C(F)F)s3)C2)c1.N12CC(C1)NCC2=O CC(C)C(CO)C(=O)NCC1CN(C(=O)CSc2n[nH]c(O)n2)CCO1 C1(COC(=O)Cn2cc(NC(=O)OC(C)(C)C)cn2)CCS(=O)(=O)N1 c1(CN2C(CNc3cc(OC)c(Br)cn3)CCC2)c(Cl)cc(O)cc1Cl CC1CC(CNC(=O)CCNS(C)(=O)=O)CN1c1nnc(C2CC(F)(F)C2)s1 C1(OC)CN(C(c2ccc(O)nc2)=O)CC1NC(=O)CCCNC(=O)C(C)(C)C C(=O)(C#CC1(C)CC1)NCC1CC(OC)CN1C(=O)CC1CCCCCO1 c1(CC(=O)NCC2CC(CNC(C3(C(C)=O)CCC3)=O)OC2)cccc(F)c1 N1(Cc2c(OCCC)cc(OC)c(Br)c2)Cc2nn(C)c(C(=O)O)c2C1 c1(C(=O)OC)ccnc(C(=O)NCC2CCC(NC(C3CCSCC3)=O)C2)c1 C(CN=C(NCC(F)F)NCC1NC(=O)CC1(C)C)C1(N(C)C)CCCCC1 C1(NC(CCSC)=O)Cc2ccccc2C1NC(C1CCN(CCO)C(=O)C1)=O CC(C)C(CNC(C1CC2(CCC2)C1)=O)C(=O)NCC1C(C)(C)C1(C)C c1(NC(CC)CC)[nH]c(=NCC2(CF)CCC2)nc2scnc12 CCCC(C)(O)CNC(=O)CCC1CCN(C(=O)CCOCCOC)C1 C1(CNC(c2cc[n+]([O-])cc2)=O)CN(C(c2snnc2C2CC2)=O)CCC1(F)F c1(C(C)C(=O)N2CCC2CNC(=O)CC2(C)CCC2)cccnc1 C1(C(=O)NC2CC3CC(NC(C4CC(=O)NC4)=O)C3C2)CCC2(CCC2)CC1 c1(C(N2CCC(O)(CN(C(=O)CSc3nccn3C)C)C2)=O)ccc(F)c(O)c1 O=C1CCCC2CN(C(=O)Cc3csc(C(=O)O)c3)CC2N1 c1(C2(C(=O)NC3C(OC)CN(C(=O)C(C)C(C)C)C3)CC2)cc(F)cc(C#N)c1 N1(C(C(=CC2N(C(COC)=O)CCC2)C)=O)CC(OC)C2(CC2)C1 c1(OC)ccc2c(C(N3CCCC(CNC(=O)C(O)C(F)(F)F)C3)=O)cnn2c1 N1(C(C2(CC=C)CCCN2C(C2C(C)C2C)=O)=O)CCc2cccnc2C1 CC(C)C(CC(=O)NC1CC(NC(C2CC23CCCC3)=O)C1)c1ccccc1 c1(C(N2CCC(C(C)(C)C)(CNC(C(C)CO)=O)C2)=O)coc2ccc(F)cc12 N12CCOC3(CCN(CC3)CC1=O)C2.Cc1nccc(=NC(=O)C2CC2(F)F)[nH]1 c1(C(=O)NCC2C(NC(c3ccnc(OC)n3)=O)COC2)ccnc2[nH]nnc12 C(C1=NOC2CN(C(C3CC4CCC(C3)C4)=O)CC12)NC(c1nc(C)c(C)s1)=O C1(NC(CCc2c(C)noc2C)=O)CCN(C(=O)C2=C(Cl)CC2)CC1F N#Cc1ccc(NCC(C2CC2)NC(=O)Cc2cccc(OC(F)F)c2)cn1 n1(C(C)C)ccc(C(=O)NC2CCC(CNC(=O)Cc3nncn3C(C)C)C2)c1 CCC(O)C(F)(F)C(=O)N1C2CCC1CN(C(c1ccc(C)nn1)=O)C2 C1(CNC(=O)NCC(CC#C)(C)C)CCC12CCCO2 N1(C(c2c(C)[nH]cc2)=O)CC2(CC2)CC1CNC(=O)CCOC1CCOC1 C(=O)(CCCC(=O)N(CCNC(C1CCCNC1=O)=O)CCOC)NCC C1(C(=O)NCC)CC12CCCN(C(c1csnc1OC)=O)C2 N1(C(c2c(C)csc2Cl)=O)CCCOC(CNC(=O)Cn2cnc(C(F)F)c2)C1 Cc1cc(C(N2CCCC2C2(O)CN(C(C3CCC3C)=O)C2)=O)ncn1 C(=O)(CCC(C(C)C)NC(c1ccncc1)=O)NCC1(OC)CCCCC1 C(C(F)(F)C(=O)N(C)CC1CN(C(=O)C(c2cncn2C)N(C)C)C1)NC(C)=O c1(NC(C)=O)ccc(CNC(CC2CCN(Cc3ccccc3Cl)CC2)=O)cc1 c1(CNC(C23CC(NCc4ccc[nH]4)(C2)C3)=O)ccc(Cl)cc1 C1(CNC(C(N2CC(C)C2)C)=O)(NC(=O)CSc2cccs2)CCCCCC1 Cn1c(C(=O)NC2CN(C(=O)Cc3cccs3)C3(CCC3)C2)cc2sccc12 N1(C(C(C(=O)OCC)(C)C)=O)CCC(C)N(C(=O)Cc2cc(C)on2)CC1 n1(CC(=O)NCCC2(NC(C3CCC(OC)C3)=O)CC2)ncc(Cl)c1C N1(C(C(Cc2ccccc2)N(C)C)=O)Cc2cc(Br)cnc2C1 c1(-c2nnc(OCCOCC)n2CCSC2CCOCC2)cccn2ccnc12 C1(C(=O)NCC(CCOC)OC)CCC(Cc2ncc(C(=O)NC(C)=O)o2)CC1 C1(CNC(C(C(C)C)CN(C)C)=O)CCC(C)(C)CN1C(=O)CCCC#N c1(C(=O)OC)c(C(=O)N(C)CC2CCCCN2C(c2nocc2C)=O)n[nH]c1C C12(NC(C3(C)CN(C(CC4CCCC(C(C)(C)C)C4)=O)C3)=O)COCC(C1)OC2 c1(SC)ccc(CC(=O)NCC2(O)CN(C(=O)CC3CC(=O)C3)C2)cc1 C(=O)(C1Cc2ccc(F)cc21)NCC1CCCN(C(c2c(OC)cccn2)=O)C1 Cn1cc(S(=O)(=O)N2CCOCC2CC(=O)Nc2cc(Br)ccc2I)cn1 N1(C(c2ccccc2N2CCOCC2)=O)CC(NS(=O)(=O)C2CC2)C(F)C1 C1(C(=O)NCC2C(NC(c3ccc(C)o3)=O)COC2)CCCN1N=O OC1(CNC(=NCc2csnn2)NCc2ccco2)CC2C=CC1C2 C(=O)(C(CCC)N(C)C)NCCn1ccc(C(N(CCCC)C(C)CC)=O)c1 C1(C(N2CC(C(=O)OC)C2)=O)COC2CN(C(c3coc(C)n3)=O)CC12 c1(C(=O)NC(C)CNC(=O)C(F)(F)CC(F)F)cc(S(C)(=O)=O)ccc1F N1(C(C2(Cn3cc(CC(COC)O)nn3)CC2)=O)CCC(C2CC2(F)F)C1 Cc1c(N2CCC(N3CCCC3=O)C2)ncnc1N1CCOC(c2nccs2)C1 Cc1cc(C(=O)NCc2cccc(NC(C34CC(O)C3C4)=O)c2)n(C)n1 CCC(F)(F)CC(=O)NC1CN(C(=O)CCc2cncc(C)c2)CCC1CO c1(C(=O)NC(CNC(C(C)OCC(C)C)=O)CO)cc(S(=O)(=O)N(C)C)c[nH]1 C1(C(C)CNC(=O)Cc2ccsc2)CCN(C(=O)CC2(C)CC2)C1 n1(CCC(=O)NC(C2CN(C(c3c(C)noc3C)=O)C2)C)ccc(O)nc1=O C12(CNC(Cc3c(C)non3)=O)CCCC1CCN2C(=O)CC12COC(C)(C1)C2 C1(NC(C(CC)C)=O)CN(C(=O)Cc2ccc(C(C)(C)C)cc2)CCC1F c1(C2(C)CC2C(=O)NCC2CCN(C(c3cnc(O)o3)=O)C2)ccc(F)cc1 N1(C(C2CC(C)(F)C2)=O)CCC(F)(CNC(=O)COc2ccc(F)cc2F)CC1 C1(NC(CCC2CC(OC)C2)=O)(CNC(c2cnccn2)=O)CC2CCC1CC2 c1(N2CCN(C(Cc3ccc(C#N)cc3)=O)C3C2C3)ncnc2occc12 C(=O)(CC1CCc2ccc(O)cc21)N(CCCNC(c1cc(C2CC2)[nH]n1)=O)C N1(C(=O)NCc2cc(S(N)(=O)=O)oc2)CCOc2cccc(Br)c2C1 N1(C(c2[nH]cc(C)c2)=O)C2CCC1CC(NC(c1c[nH]nc1C(F)F)=O)C2 CC1=NS(=O)(=O)NC=C1C(=O)NC(C)CNC(C1CCN1C1CCCC1)=O N1(C(c2n(CC)ccc2)=O)CCC(NC(c2ccc(F)cn2)=O)C(C)(C)C1 N1(C(CC(C)N2CCCC2=O)=O)CCN(C(c2ccc(N)cn2)=O)CC1CCO C(CCC(C)CC(=O)N1CCN(C)C(CNC(c2cccc(C)n2)=O)C1)=C(C)C O=S(=O)(c1ccc(Br)c(Cl)c1)NC1CCN(Cc2ncccc2Br)CC1 C1(n2cc(C(=O)Oc3ccccc3)nn2)CCCN(C(C2CC(C)(F)C2)=O)C1 C(C(=O)N(CC(C)O)CCNC(c1cn(CCO)nc1C)=O)(C(C)C)SCC C1(C(=O)NCC(CCOC)NC(c2ccccc2N(C)C)=O)CCC(F)(F)CC1 c1(NC(C2CC(O)CN2C(c2ccc(F)c(F)c2O)=O)=O)nccc(Cl)c1Cl Cc1c(Br)c(C(=O)NC2CN(C(c3ccc(C(F)(F)F)[nH]3)=O)CC2O)nn1C N12CCOCC1C2C(=O)NCCC#N.C(COC(C)C)(CCC)SC c1(C(=O)OC(C)C)ccc(S(=O)(=O)NCC2CC23CCS(=O)(=O)CC3)cc1 N1(C(c2cnc(C(C)O)s2)=O)C2CCC1C(CNC(C13CCC(C)(CO1)C3)=O)C2 c1(CC)cn2c(n1)CC(C(N1CC(C3(NC(=O)C=CSC)CC3)C1)=O)CC2 c1(C(N2CCCC(NC(C(C=C)(C)C)=O)C(F)C2)=O)cc2c(F)cccc2s1 N1(C(=O)OC)CCCN(C(=O)Nc2ccc(NC(C34CC(C3)C4)=O)cc2)CC1C C(C)(C1CCCCC1)=CC(=O)NCCN(C(C1(C)CC=CCO1)=O)CC C=CCC(C)(C)CC(=O)NC(Cn1cccn1)C(=O)NCC(C1CCCC1)C N1(C(c2nc(CC)sc2N)=O)CC2CCC(C1)C(NC(=O)C(C)C(C)C)C2 CN1CCN(C)CC(C(=O)N(C2CN(C(=O)Cc3n[nH]c4c3CCCC4)C2)C)C1 C1(C(C)C)CN(C(=O)Cc2c(Cl)cnn2C)CCN1C(=O)C(O)C1CC1 CC1(C)CCC(CCNC(c2nnn[nH]2)CCc2nccs2)C1.C1(C)CCOC1 c1(NC(C(CN(C)C)NC(COC2(C#C)COC2)=O)=O)ccc(C(C)C)cn1 CC(C)(CC(=O)NCC1CCN1C(c1ccc(C(F)F)nc1)=O)c1ccccc1 C(=O)(CCCCCCn1cc(-c2ccn(C)n2)nn1)NC(C)CC(F)(F)F CN1CC(C(N2CC(CNC(C3CC(C)(c4ccccc4)C3)=O)C2)=O)CC1=O c1(C(N2C(C(N(CC(C)C)CCOC)=O)CC2C)=O)ccnc2cc[nH]c12 c1(C(=O)NCC(CO)NC(c2cc3ccccn3n2)=O)n[nH]c2ccccc12 c1(C(N2C3C(CNC(CSCC=C)=O)C(C3)C2)=O)cn(C)c(=O)cn1 N1(C(C2(F)CCN(C(C(CSC)(C)C)=O)CC2)=O)CCC2(CC1)CC2(F)F c1(CN2CCN(C(CC(C)c3ccccc3)=O)CC2C)ncccc1[N+](=O)[O-] C1(C(N(CC(C)CNC(c2coc(C3CCC3)n2)=O)C)=O)CC2CCCCC12 c1(C(=O)NC(C2CN(C(C3CC=CC3)=O)C2)C)cnc2c(cnn2C)c1N C(=O)(C1=CC2CCCC12)NCC1(C(C)(C)O)CN(C(COC(C)=O)=O)C1 c1(CC(=O)NC(CN(C(C2CC(F)C2)=O)CC)C)occc1C(=O)NC c1(CC)nc2sc(C)cn2c1C(=O)NC1COCCN(C(=O)C(C)COC)C1 C1(C(N2CC(OC)(CNC(=O)CN(C)C(=O)C3CC3)C2)=O)C2C3CCC(C3)C12 C1(CNC(C2CC(CCO)C2)=O)CCN(C(=O)C(F)(F)CO)CC1C1CC1 C(=O)(C1=CNC2=NCCC2=C1)N(CC(CN(C(C1C(C)N(C)CC1)=O)C)O)C N1(C(c2c(C)noc2)=O)CCC(C)(CNC(=O)C(N2CCOCC2)C)C1 c12cc(CNc3ccccc3C)ccc1OC2.C1(CC)CCCCN1CC1CC1 CN1CC(C(=O)N(C)CC2(NC(c3ccncc3N)=O)CC2)NC1=O CCC(C(=O)N1CCC(NC(c2ccccc2COC)=O)C1C)NC(N)=O C(=O)(C(CC(F)F)NC(C1CC=CCO1)=O)NCC(C(C)(C)C)O CCC(O)C(C)C(=O)N1CCN(C(C2(Br)CC2(C)C)=O)CC1 C1(OC)(OC)CCCCC1NC(C1CCC2CNCC12)=O CS(=O)(=O)CCC(=O)NCCC1CN(C(=O)CCOCCF)CCO1 c1(C(=O)NC2CCN(c3nc(OC)nc(C)c3)CC2O)cc(C)c(=O)n(C)c1 C1(C(=O)NC(CC(C)NC(c2n(C(C)C)ncc2Br)=O)C)CCC(=O)CC1C c1(N(C23CC(CC)(C2)C3)C(N2CC(C)OC(C)C2)=O)cc(F)c(C)cc1[N+](=O)[O-] CCC(C)C(C(=O)NC(CNC(c1ncc(Cl)nc1Cl)=O)C(C)C)NC(N)=O C1(C(N2CC(N(C(CCc3c(C)n[nH]c3C)=O)C)C2)=O)Cc2ccccc2C1 c1(C(=O)NC(CNC(C(C2CCC2)OC)=O)C)cccc(C(C)=O)c1 c1(N(CC(C)NC(=O)CCc2ccccc2F)C)nc2cc(Cl)ccc2s1 C1(NC(C(C)C(C)O)=O)CCCN(C(c2ccc(C3(O)COC3)cc2)=O)CC1 c1(CN(C)CCN(C)C(c2ccc(-n3cncn3)nc2)=O)ccc(Cl)cc1 c1(OC(C)C)cccnc1C(=O)OCc1csc(CCN)n1 n1(CCC(=O)NC(C2CCN(C(C3CC(CC)(CC)C3)=O)C2)C)cnccc1=O CC1CCC(CO)N(C(C2CCN(C(c3nccn3C(C)C)=O)CC2O)=O)C1 c1(C(=O)NCCN(C(c2c(C)nns2)=O)C2CC2)cc2n(n1)CCNS2(=O)=O CC1CN(C)CC(C(N2CCC(NC(C3(C(=O)NCC4CC4)CC3)=O)CC2)=O)O1 c1(C(=O)NC(CC(C)NC(c2ocnc2C2CC2)=O)C)ccc2c(c1)CCC2=O Cc1cc(CC(=O)NC(C)(C)CCCNC(=O)C(C)N2CCC2)ccc1Cl N#CCCCC(=O)NCC1CC1CNC(=O)CC1CCC12CCC2 N1(C(CC=CCNC(C2(CC)CCCC2O)=O)=O)CC2CC(C1)N(C)C2 C1(CNC(C2CCC(OC)CC2)=O)CN(C(C2COC(=O)N2)=O)CC(C)(C)O1 N1(CCC#C)CCN(C(C2C(NC(=O)C(C)OCC3CC3)C2(C)C)=O)CC1 c1(NC(CC2(C=C)CN(C(=O)Cc3cncnc3)C2)=O)cnc2ncnn2c1 c1(SC)ccc(C=CC(N2CCCC(CNC(=O)C(CN(C)C)N(C)C)C2)=O)s1 c1(C(N2CC(C3N(C(C4(C)COC4)=O)CCC3)(O)C2)=O)cc2scnc2[nH]1 N1(C(C(COCCOCC)c2ccccc2)=O)CCC2(CC1)CC2NC(=O)OC N(C(=NCC1CC1(C)C)NCC1CCC(C2CC2)O1)C(CC)CC CCC(CC)(CC(=O)OC)C(=O)N1CC2CC(NC(c3snnc3C)=O)CC2C1 N1(C(c2c(C)nc(CO)nc2)=O)CC(NC(=O)CC2CSCCS2)CC12CCC2 CC1CN(C(C2(C)CC(F)C2)=O)CC2(CCN(C(=O)CCF)C2)O1 N1(C(CC=C)=O)CC2CC(NC(C3(C4CCCO4)CCCC3)=O)C1C2 c1(C(=O)NC23CCN(C(C4C(C#C)C4)=O)C2CCC3)csc2cc(C)ccc12 c1(C(=O)NC2C(NC(C3CCC(N(C)C)C3)=O)CCC2)ccc(CCC#N)cc1 CC1(NC(c2coc(CNC(C3CC3C3CC3)=O)c2)=O)CCC(O)CC1 N1(C(c2c(C)cn(C)c2)=O)C2CCCC1CN(C(=O)CCc1scnc1C)CC2 CC(CC1CC1)C(=O)NC(Cn1cncn1)C(=O)N1CCC(c2nn[nH]n2)C1 C1(C2CCN(C(c3coc(Cl)c3)=O)CC2)(NC(C2CC3CCCCN3C2)=O)CC1 c1(OC)ccc2ccccc2c1C(=O)NC1CC1NC(=O)C(C)(C)N(C)C C(=O)(CCC(F)F)NC1CCC(NC(CCCNC(=O)OC)=O)C1 c1(CC)nccn1C(C)CC(=O)N(CC(C)(C)NC(C1CC1C(N)=O)=O)C C(=O)(C(CN(C)C)CC)NC1(C(N(C(C(=O)OCC)C)C)=O)CC(CO)C1 N1(C(C(F)=CC)=O)CCC(CCNC(c2cc(C)sn2)=O)CC1 N1(C(=O)Cc2cscn2)CCC2(CC1)CC(C(N1CC3CC3C1)=O)CO2 c1(NC(c2nc(Br)cn2C)c2n(CCCC)nnn2)ccc2nc(C)[nH]c2c1 N1(C(COCC)=O)CCN(C)C(CNC(=O)C(C)Oc2cc(F)cc(Cl)c2)C1 c1(C(N(CCNC(CN2CCC(C)CC2)=O)C2CC2)=O)cnn2c1OCC2 C1(CNC(c2cc3ccsc3s2)=O)CC2COCC2N1C(=O)CCC[N+](=O)[O-] Cc1cc(=NCCOCc2ccccc2)[nH]c(=NCCCn2cccn2)[nH]1 c1cc(Br)c(Br)o1.C1(NC(c2nnnn2CC(F)F)C)C=CCCC1 C1(CCNC(C2(COC)CCC2)Cc2nnnn2CCC2(C)CC2)CCCOC1 C1(C(=O)NCCC(=C)C)CC(F)(F)CN1C(=O)CC1CCCCN1C C1(OC2C(C(=O)OCC)CCC2)CCN(C(c2nn(CCOC)nc2C)=O)CC1 Cc1cnn(C)c1C(=O)NC(c1ccccc1)CNC(=O)CC1CC(C)C1 C1(NC(CC=C)=O)CN(C(c2sc(CCC)nc2C)=O)CC1(C)C c1(C(C(=O)NCC(CNC(c2cc(C)on2)=O)F)=O)ccc(F)cc1.C(C)(C)(C)N S(=O)(=O)(c1ccc(NCC2CCC=CCC2)c(Br)c1)NC1CCS(=O)C1 c12ccccc1CCCO2.N1(CCCNC(C)C)CCCOCC1 N1(CCNC(CC2(C)CCN(Cc3cn[nH]c3)C2)=O)C(=O)CCCC1=O c1(C(N(CCN(C(C(CCC)=CCC)=O)C(C)C)C)=O)cc(C)c(F)cc1Cl CCS(=O)(=O)CC(=O)NC(c1ccccc1F)CNC(c1ccc(F)cc1F)=O c1(C(=O)NCC2OCCN(C(C=C(CC)C)=O)C2)c(S(C)(=O)=O)cnn1C N1(C(COCCC(C)C)=O)CCC(CNC(c2ccc(Br)o2)=O)C1(C)C N1(C(c2c(C)ncs2)=O)CCCC(C)(C(N2CCC(c3ccccc3)C2)=O)C1 C1(NC(COCCCOC)=O)CCC2CN(C(=O)CSCc3ccncc3)CC12 CCC(C(=O)OC)C(=O)Nc1cccc(NC(=O)C=CC(C)(C)SC)c1 C1(C(=O)NCCC(C)SC)CC(NC(C2CCCN2C(C)C)=O)C(O)C1 N1(C(c2n(CCC)ccc2)=O)CC(O)CCC1C(=O)NCCC(C)O C1(N(C(c2n(C)nnc2)=O)C)CCC2CN(C(=O)CCCC3CCCO3)CC12 C1(C(N2CC3CCC2C3)=O)CC(O)CN1Cc1cncc(C(F)(F)F)c1 CCC(C)C(CN(C)C)NC(=O)CN(C(C1(C)COC1)=O)C(C)C c1(CC)cccc(C(=O)NC(C)(C(=O)NC2CCC(O)C2)C2CCC2)n1 OC1CCC(O)C1n1cncn1.c12ccc(cc1)SCC2O CC(C)(CC(=O)N1CCC(C(F)CNC(=O)CCF)CC1)C(F)(F)F N1(C(C(F)=C(C)C)=O)CC2CCCC2(CNC(=O)CN2CCC(C)C2)C1 C#Cc1cccc(C(=O)NC2C=CCN(C(C3(C)CC4CC4C3)=O)C2)c1C C=CC1(C(=O)NCC(CNC(=O)CCc2cncc(F)c2)CO)CCOCC1 c1(C(N2CC(N(C(Cc3cc(C)[nH]n3)=O)C)C(C)CC2)=O)cnc2ncccn12 N1(C(C(C)NC=O)=O)CC2CN(C(=O)CC(C(F)(F)F)c3ccon3)CC2C1 c1(NC(C2C3CNC2C3)=O)cccc2[nH]cc(Cl)c12 c1(C(N2CC(NC(C(CC=CCC)C)=O)C2)=O)cc2cc(Cl)sc2[nH]1 Cc1ccc(Br)c(F)c1C(=O)Oc1csc(=N)[nH]1.c12nc(cs1)CC(=O)N2 C=C(C)CC(C(=O)Nc1ccc(O)c(CO)c1)NC(C1CC=C(C)CC1)=O c1(C(N2CC3C(NC(c4c(Cl)ccc(F)c4F)=O)(C3)C2)=O)ccc2snnc2c1 C(=O)(C(F)(F)C(O)C(C)C)NC1CCN(C(c2c(CC)cno2)=O)C(C2CC2)C1 CC1=NC(C)(CNC2CCC(N)C2)CS1 c1(NC(c2cc(F)ncc2NCc2cccc(Cl)c2Br)=O)c(Cl)cc(Br)nc1Br c1(C(N(C2CCN(CCOC)CC2)CCC)=O)noc2c1COCC2.C1(=O)CN1 C(=O)(C(CCC1CC1)NC(=O)COCCCC1CC1)N1C(COC)CCC1 C(CC(C(C)C)NC(C12CC1CCN2C(=O)CC=C(Cl)Cl)=O)OC Cc1cccc(C(N2CCC(C(C)(C)C)(CNC(C3COC(C)C3)=O)C2)=O)n1 c1(C(=O)NC2CC(C(=O)NC(c3nn[nH]n3)CC)C2)cccnc1O c1(C(=O)NCC2(O)CCN(Cc3ccccc3)C2)cc2c(nc1O)CCCCC2 C1(C(=O)NCC2(O)CCN(C(=O)CCc3ccncn3)C2)CS(=O)(=O)CCO1 CCC(CC(=O)NCC(C)NC(c1cocc1C)=O)OC CCCCC(CNC(=O)CCC1(C)CC1)NC(=O)C(c1ccc(CC)cc1)CC C1(NC(Cc2ncc(CC)[nH]2)=O)CC2CC(C1)N(C(c1c[nH]nc1F)=O)C2 C1(CNC(CN(CCC)C)=O)CC2CCC(C1)N2C(C1CC1c1ccsc1)=O N1(C(c2c(C)nc(CO)o2)=O)CC(NC(c2[nH]nnc2C)=O)C(C)(C)C1 N1(C(CN(C(=O)OC)C)=O)CCC2CC2(NC(c2cn(CCO)nn2)=O)CC1 c1(CC)ccccc1OCC(=O)N(CC(CC)NC(c1[nH]nnc1C1CC1)=O)C c1(N2CCN(C(CC(CCC=C(C)C)C)=O)CC2)nc(C2CC2)nc2c(C)csc12 c1(C(N2CCC(CC(=O)Nc3ccc(O)cc3F)CC2)=O)cc(Cl)c(Cl)cc1Cl C1(CNC(C(C)CF)=O)CC2(C1)CN(C(c1cc(O)ccc1Br)=O)C2 c1(C(=O)NC23C(n4cc(CC(C)O)nn4)CC(CC2)C3)ccc2c(n1)OCO2 C1(C(=O)NC(C(C)C)CNC(=O)C=Cc2cnn(C)c2)CCC2(CCC2)CC1 n1(CC)cc(C(=O)NCC2(C)CCCN2C(c2cnc(Cl)nc2)=O)c(C)n1 C1(CNC(c2ccc(CO)o2)=O)CCCN1C(c1coc(C2CC2)n1)=O C1(CNC(c2cc(CCOC)on2)=O)C(C)CCCN1C(=O)C1=CSCS1 C1(NC(=O)C(O)C2CC2)(CO)CN(C(=O)COc2ccccc2)C1.C1(C)CCC1 Cc1ccc(-c2nccc(C(=O)NC3CN(C(=O)CNC=O)CC3C)n2)cc1 C(=O)(C(C)S(=O)(=O)C(C)C)NC1CC(C)(NC(C(C)Oc2ccccc2)=O)C1 C#CCCCCC(=O)N1CC2CC2(NC(C2CN(C3CCOC3)C2)=O)C1 Cc1cccc(NC(CC2C=CC(C(=O)NOCCCCF)C2)=O)n1 C(C)(C(=O)NOCC1CCC1)(C1CCC1)NC(C(C)NC(CC)=O)=O c1(CNC(CN(C(C=C(C)C(C)(C)C)=O)C2CC2)=O)c(C)cnn1C c1(C(=O)NC2CC(CNC(CCCC)=O)C2)cc(OC)nc(C)c1 C1(C(=O)NCCC(C)NC(C=Cc2c(C)cncc2)=O)Cc2cncn2C(=O)N1 C1(=CNC(C2CC(SC)C2)=O)CCN(C(c2cc(C(N)=O)co2)=O)CC1 N1(C(C(C)OC(C)(C)C)=O)CCC(C(=O)NCC=CBr)C(C)C1 c1(CNC(C(F)=CC)=O)cccc(CNC(c2cccc(CC)c2)=O)c1 Cc1ccc(OCCCC(=O)NC2CCCN(C(C3CC3F)=O)C2)c(Cl)c1 CCCCC(CC(=O)NC1CC2(CCOC2)C1)NC(=O)CSCCC(C)C c1(CC)cccc(F)c1-c1cccc(-c2ccc(C)cn2)c1 C1(NC(C(C)C)=O)C2CC1CN(C(=O)NC1(F)C3CCCC13)C2 CC(C)C(O)CC(=O)NCC(O)CC(=O)N(C1CCCCC1)C C=CCC(CC(=O)NC1CCOCC1(C)C)NC(c1cc(C)cc(O)n1)=O C1(CNC(C(=O)NCCOC)=O)CCCN(C(c2ccc(C#N)[nH]2)=O)CC1 c1(OC)cncc(NC(=O)C(CCSC)NC(=O)CC(C)COC)c1 S(=O)(=O)(c1ccc(N2CCOC3(CCCC3)C2)c2cnccc12)NC(C(C)O)C CC(C)C(C)(F)CNC(=O)CCC1(C)CCCN1C(c1ccc(CF)cc1)=O c1(C(=O)NC2CCN(C(=O)CCc3ccncc3)C2)cnc2c(c1)CCC2 CC(=O)CCCC(=O)NC1CCN(C(=O)C(c2ccc(Cl)cc2)CO)C1(C)C CCCC(C(O)C(=O)NCC(F)CO)NC(c1snnc1CC)=O CC1OC2(CNC(=O)COCC3CCOCC3)CC1(NC(=O)Cc1cnsc1)C2 c1(OC)nc(C(=O)NC2CCC(CCNC(=O)Cc3ncc(Cl)s3)C2)cc(O)n1 N1(C(C(C)N(C)C)=O)CCN(C(=O)CC2(NC(=O)CC3(C)CC3)CCCC2)CC1 C1(C)(C(N(CCNC(=O)Cn2cc(C#N)cn2)CC)=O)CCC(C)(C)CC1 CC1CN(C(c2csc(F)c2)=O)CCN(C(c2nn(C)cc2Cl)=O)C1 N#Cc1cc(N2CCCCC2CNC(=O)CCOCCN(C)C)ccc1[N+](=O)[O-] c1(C(=O)NCCN(C(C(C2CCCO2)OC)=O)C)ncc([N+](=O)[O-])n1C N1(C(C2N(CC(C)C)CCC2)=O)CC=C(CNC(=O)C2=CSCCO2)CC1 C(=O)(C1=C(F)CN(C(C2(C#N)CCOC2)=O)CC1)N1C2CC(C)CC1CC2 N#Cc1cncc(C(=O)NC(CC(=O)NCCCSC(F)F)C(F)F)c1 c1(CC(N2C3CCC2C(NC(=O)C2=C(Cl)CCC2)C3)=O)ccc([N+](=O)[O-])cc1F CCC(C)C(O)C(=O)NCC1CCCCN(C(=O)C(C)C2CCC2)C1 C1(NC(CN(C2CCC2)C)=O)CCC2CCN(C(=O)CC3CCCC3)C1C2 CCCCC(CNC(=O)Cc1ccccn1)NC(=O)CC1C=CCC1 c1(CC(=O)NCCCN(C(c2nccn2C)=O)CC)n[nH]c2ccccc12 Fc1cc(-n2nc(C3CC34CC4)nc2-c2ccon2)c(F)cc1F CCCCC(O)C(=O)NCc1ccccc1CN(C(=O)CN1CC2CC2C1)C CC(C)(C(=O)NC1C2CCC(F)(F)C12)C1=CCN(C(c2ccoc2)=O)C1 C(CCC)(CCCNC(C1(CO)CCOC1)=O)OCC.c1(CC(=O)N)cccc(C)c1 O=C1CCN(CC(=O)NC2CC3CN(C(C45CCCC(C4)OC5)=O)CC23)C(=O)N1 c1(C(=O)NCC(C(C)C)NC(C2CCN2S(C)(=O)=O)=O)c(F)ccc(Cl)c1F c1(OC)ccc(Cl)c(C(N2CC(OC)C(NC(=O)CC(C)(C)C)C2)=O)n1 Cc1ccc(CNC(=NCCCC(C)O)NCCNC2CCOC2)c([N+](=O)[O-])c1 N1(C(=O)Cc2ccns2)CCC2CCCC12C(N1CC(F)C(F)C1)=O C(=O)(CCS(C)(=O)=O)NC(C1(O)CCN(C(c2cc(F)ccc2Cl)=O)C1)C C1(C)(C(=O)NCC2(C(N3CC(CO)C3(C)C)=O)CC(=C)C2)C(C)(C)C1(C)C C(C(=O)NC(CC(F)F)C(=O)N(C)C(C)C)(C(C)(C)C)OC c1(N(CC=C)C)nc2c(c(=NCc3cc4c(cc3F)NC(=O)CC4)[nH]1)CCCC2 c1(CC(=O)NCC(CN(C(C23CCC(OC)C2C3)=O)C)C)cn2c(C)csc2n1 c1(-c2nc(CC)nn2CC)sc(C=O)c(Br)c1Br C(=O)(CC(C)(C)N(C)C(c1cncnc1)=O)N(C)Cc1scc(C)n1 C(=O)(CC(O)C(C)CC)N1CC2C(N(C(C3(C=C)CCCCC3)=O)C)C2C1 S(=O)(=O)(c1ccc(=NCC(O)COC2CC2)[nH]c1)N1CCC(c2c(C)cccc2)C1 O(NC(=O)C#CC1CC1)C(CCOC(=O)NC(C)(C)C)=O.CC(C)CC1C(=O)N1 C1(C(=O)NC2(CN(C)C(c3cccc(F)c3F)=O)CC2)CCC2(CCCCC2)C1 CCC(CC(=O)N1CC(NC(c2cncc(C)n2)=O)CC12CCCC2)C(C)(C)C Cc1ccc(SCC(=O)NC2CCN(C(=O)C3=NNC(C(F)(F)F)C3)C2)c(C)c1 c1(CC)ncccc1NC(=O)C(CN(C)C)NC(=O)CN1CC(C)(C)C1 C(C(C(=O)NOC)N(C)C)NC(C1CC(O)(CC#C)C1)=O.O=C(C)N CCC(C)C(=O)NCCCOCCOCCNC(C1CC1Cc1ccccc1)=O c1(C(=O)NCCCN(C(=O)C(=O)Nc2ccc(Cl)cc2)C)ccc2c(c1)CCO2 Cc1ccc(C)c(C(=O)N(C)CCOCCNC(c2cc(C)n(C(C)C)n2)=O)c1 N1(C(c2ccc(CC)nc2C)=O)CCN(C(c2ccsc2Cl)=O)CC(C)(F)C1 c1(N(C)C)ccc(C(N2CCN(CCNC(=O)CCCC3CCC3)CC2)=O)cn1 C1(NC(CCc2cc(C)[nH]n2)=O)CN(C(C2CCC2(F)F)=O)C2(CCCC2)C1 CCCC(CC)C(=O)N1CCC(COC)C(O)C1 CC1(C)CN2CC1CC2=O.C1(O)(C(=O)NC2(c3ccno3)CC2)CC2CCC1O2 Cc1nc(NC(=O)C(c2cnn(C)c2)C)cc(NC(CN(C)C)CCO)n1 C1(=CC(=O)NC(C2CCN(C(C(CC)(C)OC)=O)CC2)C)CN2CCC1CC2 c1(C(N2CCC(N(C)C(c3ccc(C(C)(C)C)[nH]3)=O)C2)=O)cc2c(ccn2C)s1 C#Cc1cccc(C(N2CC(c3ocnc3CNC(=O)C(C)OC)C2)=O)c1F c1(CC)cccc(C(N2CCC(C(=O)NCC(F)CC)C2)=O)c1 c1(OC)ccc(NC(C)=O)c(OC)c1.c12nc(ncc1Cl)N2C1CC2(CNC2)C1 C1(CC(=O)NC2CCC(NC(C3(CC)CCCC3)=O)CC2)COC2(CCC2)CO1 c1(C(=O)NC2C(OC)CN(C(C3CC3(C)C)=O)C2)cc(F)c(Br)c(Cl)c1 c1(OC)cc(C(=O)NC(C)(C)CNC(C2CSCCS2)=O)ccc1Cl S(=O)(=O)(c1ccc(N(C2CC3CC2CN3)C(=O)CC)cc1)N(CCCC)CC C(=O)(CS(C)(=O)=O)N(C)CC1(NC(c2cnc(C(N)=O)cn2)=O)CC1 c1(C(=O)NCCN(C)C(c2ncn3c2CCC3)=O)ccc(C2CC2)cc1Cl O=C1NCc2ccc(C(=O)NC3CCCC34CN(C(=O)C3=CCSC3)C4)cc2N1 C(=O)(CCS(=O)(=O)N(C)C)NC(C(C)NC(c1cnn(C)c1C(F)(F)F)=O)C C1(C(=O)NCCCCn2cc(CSCC)nn2)CCN(C(C)C)CC1 C1(C2CCN(C(=O)CCCCO)CC2)(NC(=O)CCC(F)(F)F)CC1 O=S(=O)(c1ccc(NC2COC3(CCC3)C2)c(F)c1)N1C2CCCC1COC2 c1(C(N2CCCC(F)(CNC(=O)CC(F)(F)F)C2)=O)cc(F)c(Cl)c(Br)c1 C(=O)(C(CC)C(=O)NCC1COCC1C(=O)NCC1CC2CC1CC2O)OC N1(C(CC2ON=C(C)C2)=O)CC(NC(=O)Cc2csnn2)C(CC(C)(C)C)C1 C(C(C)(O)CC(=O)N(CCC(N1CC(O)CC1CO)=O)CCCO)OC N1(C(c2cccc(OC)c2)=O)CCC2CC1CN2C(c1ccc(C(N)=O)cc1)=O C(=O)(C1=CCS(=O)(=O)C1)NC1C(NC(c2oc(CC)c(C)c2)=O)CC1 CCCC(C)(O)CC(=O)NCC1CCC1C(=O)Nc1cccc(C)c1CC C(=O)(C(CCC1CC1)NC(=O)C=Cc1ccc[nH]1)NC(C)C(F)F C(=O)(C(CC)C(=O)NCC(N1CC=CC1)=O)OCC.C1(Cc2cnc[nH]2)C(=O)N1 C(=O)(CC(C)CN(C)C)NC(CC1CN(C(c2ccc(COC)s2)=O)C1)C c1(C(=O)OC(C(C=C)C)C(=O)OC)cccc2sncc12 Cc1ccc(CCC(=O)Nc2cccc(C(=O)NCc3ccccc3Cl)c2)cc1 N1(C(Cc2cccc(SC)c2)=O)CC(NC(=O)CC2CCCC2C)C(N=[N+]=[N-])C1 c1(C(=O)NC2CC(C)N(C(=O)C=CCN3CCCC3)C2)cc(Cl)cnc1O c1(C(=O)NCC2(F)CC(NC(CC(=C=C)C)=O)C2)cccc2c1ncn2C c1(CC(=O)NCCNC(COCCOCC)=O)cccc2c1CCC2 CC1(C)CN(C(C2CC(C3CC3)=NO2)=O)CC1C(=O)NC1CCNC1=O Cc1cnc(C(=O)N(C2CN(C(c3nnn(C)c3N)=O)CCC2C)C)cc1Cl C1(O)(C(C)CNC(c2cn(CCO)nn2)=O)CCN(C(C2(CF)COC2)=O)C1 c1(NC(=O)OC(C)(C)C)ccccc1O.c1(CC(C(=O)OCC)OC)ccc(F)nc1 C1(CNC(C(c2ccc(Cl)cc2)CC)=O)CN(C(=O)C2CC2)CC12CCOCC2 C(=O)(C(O)C(C)CC)NCC(N(C(C(Cc1cccc(OC)c1)=O)=O)C)C1CC1 CN1C(C(=O)NC2CN(C(c3c(C(F)F)nn(C)c3Cl)=O)C2)CCS1(=O)=O C1(C(=O)NCCNC(c2c(CC)csc2)=O)Cc2ccc(F)cc2O1 C1(S(N)(=O)=O)(C(=O)NCC2N(C(CCCN(C(C)C)C)=O)CCC2C)CCC1 c1(C(=O)NCC2CCCN2C(=O)CSc2ccccc2)ncc2c(F)cccn12 Cc1cc(NC2CCn3ncnc3C2)ncc1S(=O)(=O)N1CCC=C(Cl)C1 C1(CN(C)C(c2cn(CCO)nn2)=O)CCCN(C(=O)C(O)CC2CCCC2)C1 CCC(CC(=O)NC(c1cccnc1)C(=O)NC1(C)CS(=O)(=O)C1)SC N1(C(c2n(C(C)C)ccn2)=O)CC(C)C(NC(c2c[nH]c(=N)s2)=O)C(C)C1 C(=O)(C1=CN2CCS(=O)(=O)N=C2C=C1)NCCOC1CC(NC(C2C(C)(C)C2)=O)C1 Cc1ccccc1-c1noc(C)c1C(=O)NC1CCC(NC(C2C(C)C2C)=O)C1 c1(C(c2n(CC)nnn2)NCCC2CCCCO2)cccc2ccc(Cl)cc12 N1(CC2C(C(N3C(C)CCCC3)=O)C2)CCc2cc(C(C)(C)C)ccc2C1 C1(C(=O)NC2(CCNC(C(C)=C(C)C)=O)CC2)CCC1(C)C C1(C)(C(N(CCNC(c2ncccc2F)=O)CC)=O)CCC(C)(C#N)CC1 C1(NC(C(=Cc2cccs2)C)=O)CC(C)CN(C(C2CC2C(NCC)OC)=O)C1 C1(CCN(C(Cc2cn(C(C)C)nc2)=O)C)CCCCN1C(=O)C(O)CN(C)C c1(C(N2CC(NC(C(CCOC)C)=O)C(F)C2)=O)c(F)ccc(C)c1Br N1(CC(=O)NC(C(C)C(C)(C)C)=O)CCc2c(nnn2-c2ccccc2)C1 C(=O)(C(CCC(C)C)NC(c1cnco1)=O)NCc1nc(C)oc1 CC(C)CCC(=O)C(=O)NC(Cc1cn[nH]c1)C(=O)NCCN1CCNC1=O C(=O)(C1=CCN(C(=O)CC=Cc2ccccc2)C1)N1C(C(C)O)CC1 Cc1ccc(S(=O)(=O)N2CCC(CC(N3CCC4(C3)CC4(F)F)=O)C2)cn1 c1(C(N(c2c(C)nsc2)C)=O)ccc2c(c1)nc(O)n2C#N C1(CC(=O)NC)CN(C(C2CC2(C)C)=O)CCN1C(=O)CCCNS(C)(=O)=O N1(C(CCCN(C(C)=O)C)=O)C(CC(=O)N(C(C)CO)CCO)C2CCCC12 C1(NC(c2c(OC)cc(C)s2)=O)CN(c2cc(C)nc(CSC)n2)CC(C)(C)C1 CC1(C)CCOC(C(=O)NC2CC3C2CCN3C(=O)CCC2OCCO2)C1 C(CC(C)(C)C)(C(=O)NCc1nc(C(N2CCOCC2CC2CC2)=O)c(C)o1)OC N1(C(CC2C(C)(C)C2)=O)CCN(C(c2cccc(C(F)F)n2)=O)CC1 N1(C(c2scc(C)c2)=O)CCC(C)(C)C1C(N1CCC12CCC2)=O C1(C(=O)NCc2cnc(C(F)F)o2)CCCCN1C(=O)C=Cc1ccncn1 C(CCF)(C(=O)N(C1CCSC1)C)NC(C(C)OCC=C)=O N1(C(C(CC)C(=O)OC)=O)CCC(NC(=O)CCOc2ccccc2)CC(F)C1 C1(NC(c2c(C)sc(O)n2)=O)CC2(CCN(C(=O)C3=CCCCCC3)CC2)C1 N1(C(=O)Nc2nc(CC)c(C(=O)O)s2)CCOC2(CCSC2)C1 c1(C(=O)NC(C(C)C)(C)CNC(=O)C(CO)N(C)C)ccnc2ccc(Cl)cc12 c1(CC(N2C(C)CC(NC(CCCC#C)=O)C2)=O)cccc2ccoc12 c1(CCC(=O)NC(C)C(C)NC(=O)COc2ccon2)cn(C)nn1 C=CCC(CC=C)C(=O)NCC1CCC(C)CN1C(C1CC2C=CC1CC2)=O N1(C(C)C)CCC(CC(N2CCC2CNC(C2(F)CCOC2)=O)=O)C1 N1(C(c2c(C(C)C)c[nH]n2)=O)CCC2(CCCC2NC(=O)C(F)=C2CCCC2)C1 c1(CC)n[nH]c(=NC2CCCN(C(=O)C(C)(O)Cc3ccccc3)CC2)o1 c1(C(N2C(C)(CNC(c3c(C)ncn3O)=O)CCC2)=O)cc2c(nn1)CCCC2 CCC(C)CCCCC(=O)NC(C)CC1CN(c2nnc(C#N)s2)C1 c1(C(=O)NC2C(C)N(c3ncc(F)cn3)CCC2)ccc(S(C)(=O)=O)o1 CC(C)C(C)(O)C(=O)NC1CN(C(=O)CCNC(c2ccsc2)=O)CC1(C)C c1(CNCc2ncc(OC)cn2)cccc2c1sc1ccccc21 C(=O)(C1CCSc2ccccc21)NCCN(C(=O)C(C(C)C)NC(N)=O)CC CC(CN=c1[nH]c2ccc(S(=O)(=O)N3CCC(SCC(N)=O)C3)cc2s1)N(C)C CC(F)(C(=O)NCC(C1CCCC1)NC(=O)CSc1cccc(F)c1)C(F)(F)F c1(C(N)=O)ccc(C(=O)NCCCN2CCCCC2)o1.c12ncc(o1)c(=O)[nH]2 C(=O)(CCC(=O)N1CC(CNC(c2n[nH]c(C)n2)=O)CC1C)OC C12(C(=O)N)CCCC1CCC2.Cc1cccc(C(O)C2n3cc2nn3)c1.C1CC1 N1(C(C(C)O)=O)CCCC(C2CCN(C(c3c[nH]c(=N)nc3O)=O)C2)C1 c1(C(N2CCC3(C(C(=O)OC)C3)CC2)=O)c(F)ccc(OC(F)F)c1F Cc1ncc(N)cc1C(N1CCCOC(CNC(C2C3CCCC23)=O)C1)=O N12C3CCC1C(C3)COC(=O)C=CC2=O.CCCCNC(C1CC1C(N)=O)=O C1(OC)(CNC(=O)CC(C2CC2)C2CC2)CCN(C(c2ccnn2C(C)C)=O)C1 N1(C(c2c(C(C)NC(=O)CCC3CC3)noc2)=O)CCCC(C2CC2)CC1 C(CC(CC)C(=O)NCC(C(=O)N1CC2CC1CC2CF)C(C)C)=CC N1(C(C2CCN(CC(C)C)C2)=O)CCC2(C1)CN(C(=O)CC1CC(CF)C1)C2 c12ccc(OC)c(c1)C(=O)N1CCOC(C1)NC2CC.C1(C(=O)OC)CCN1.OCC CC(C)CC(C)(C)CNC(C1CCC(C)CN1C(=O)CCN(C)CCO)=O C1(N(C(=O)OC(C)(C)C)C)CCCCN(C(=O)C(C)C(=O)N2CCC(C)C2)C1 N1(C(C(CC)(C)O)=O)CC(NC(=O)CCC2OCCO2)CC(C)(C)C1 CC(C(=O)NC1(CNC(c2cc(-c3ccc(Cl)s3)on2)=O)CC1)C(C)(F)F C=C(C)CC(C(=O)N(C)CC1CCN(C(=O)CN2CCOCC2)C1)NC(C)=O Cc1nnc2n1CC(C(N1CCCCCC1CNC(=O)CC(C)(C)O)=O)CC2 CC1OCCC1C(=O)NCCNC(C1(n2cc(CCS(C)(=O)=O)nn2)CC1)=O CN1CCN(C(c2cnns2)=O)CC1CNC(c1cnc(C(C)(C)CF)o1)=O c1(C(C(=O)NC2CCC(NC(=O)COCC(F)F)C2)OC)ccc(Cl)cc1 N1(CC(=O)NCC(C(C)C)NC(C2(n3cnnn3)CC2)=O)CCC(C)(C)C1 c1(C(=O)NCC2C(CNC(CCCCCOCC)=O)C2)coc2c(Cl)cccc12 N1(C(Cc2c(C)cccc2)=O)CCN(C(c2ccn3c2CCC3)=O)CC(C)(C)C1 CC1CC(NC(C2CCN(C)CC2)=O)CN(C(=O)CCN2CCCS2(=O)=O)C1 C1(C(=O)NC)(CNC(COC(CC)CC)=O)CC=CCC1.N12CCCC1CC2=O N1(C(C2(CC=C)CC=CC2)=O)CC2CC(C1)N2C(=O)C(C)(C)n1cncn1 c1(OC)cc(OC)cc(C(N2CCC(n3cc(C)cn3)C2)C(=O)NC2(C)CC2)c1 Cn1cc(CC(N2CC(C)(C(=O)NC3CC(=C4CCC4)C3)C2)=O)cn1 c1(C(=O)NC2CN(C(C(CCC)O)=O)CC(O)C2)cccc2ccc(Br)nc12 O=C1CN(CC(N2CCN(c3ccc(-c4ccco4)s3)CC2)=O)C2CNCC2CN1 CC1(C)CN(C(=O)CCN(C(C2CC(C(F)(F)F)C2)=O)CCO)CC(CO)O1 c1(C(=O)NC(CC=C)CNC(c2cccc(O)c2Cl)=O)cnn2c1C(=O)NCC2 c1(NC(CC(C)N(C(c2cn(CC)nn2)=O)C)=O)cnc(C)c(C)c1 C1(C)(CNC(CCN(CCCCC)C)=O)CCN(C(c2ncccn2)=O)C1 N1(C(C2(NC(CC(C)n3cccn3)=O)CC2)=O)CCCC2COCC12 N1(C(=O)OC(C)(C)C)CCCCC1CN1CCN(C2(C=C)CCC2)CC1.C1(C)CC1 C(=O)(N=S(C)(=O)c1ccccc1OC)C(CCC(F)(F)F)CCOC N1(C(C(=O)OC)(C)C)CCCN(C(=O)Nc2oc(C(N)=O)cc2C)CC1 c1(C(c2n(CC)nnn2)NC2COCC2C2CC2)cc(OC)ccc1OC C1(NC(C=CCN(CC)CC)=O)CCCN(C(=O)Cc2csc(C(C)C)n2)CC1 C1(CC(=O)NCC2CCN(CC)C2)CCCCN1C(c1ccn(C)n1)=O C(=O)(CC(C)CC(C)(C)C)N(CCCNC(=O)C1=NOC(C)(C)C1)CC c1(C(=O)NC2CCN(C(=O)C(F)n3ccnc3)CC2F)cc(Cl)cc(Cl)c1F C(Cn1cccn1)(C(=O)NCCCCN1CCCC1)NC(=O)CCC1OCCO1 n1(CCOC(C2(C)ON=C(C)C2)=O)c(=O)cc(C)c2ccccc12 CCCCC(C(=O)N1CC(F)(CO)C1)NC(C1CC=CC1)=O N1(C(c2c(CC)occ2)=O)CCCC1(C)CNC(C1CCC(C(C)C)CC1)=O N(C(=NCCCCl)NCC(=O)Nc1ccccc1)Cc1c(CC)onc1C N1(C(C(CC)(C)COC)=O)CCC2C(CCCN2C(c2cncn(C)c2=O)=O)C1 C=CC1(C(=O)NCCC2COCC2O)CCN(C(c2nnsc2N)=O)C1 CCC(CC(=O)N1CCN(C(=O)CC2(CSC)CC2)CC1CC)CC(C)C C1(C)(CNC(c2c(C)onc2C(F)(F)F)=O)CCN(C(C2CNC(=O)C2)=O)CC1 N1(C(c2c(CC)c[nH]c2)=O)CC2CCC(CNC(c3c(C)nsc3C)=O)C2C1 CC1C(NC(=O)CCn2cc(Cl)cn2)CC2CCC1N2c1ccnc(CO)n1 c1(C(C(=O)NCC)N(CC(=O)NC2CC2)C)cccc(Br)c1 N1(C(CNC(=O)OC)=O)CCN(C(=O)CN2CCOCC2)CC1C.C(C)(C)(C)O CN1Cc2ccccc2C(Nc2cccc(C(N3CCCC(O)C3)=O)c2)C1=O N1(C(CCC2N(C(c3c(C)n(C)nc3)=O)CCC2)=O)CC2CC(N(C)C)CC1C2 c1(C(=O)NCCCN(C(C2(C)CCN(C(C)=O)C2)=O)CC)scc(C)c1OC CCCC(C)(C)C(=O)N1CC(CCCCNC(c2cc(Cl)ncc2F)=O)C1 C(C)(C(C(=O)N1CCOC2C(c3cn(CC(=O)O)nn3)CC12)C(C)C)OC C1(C(=O)NC2CN(C(C)C)C(=O)C2)(CO)CCc2ccccc2O1 Cc1ccc(C(=O)NCC2CCCN(C(c3sccc3C(F)F)=O)C2)cc1C CCC(CC)(CO)C(=O)N1CC(NC(c2ccn(CC(F)F)n2)=O)CC2(CC2)C1 c1(C(N(C2CCN(C(C(C)(CO)NC(C)=O)=O)C2)C)=O)cccc(Cl)c1Cl N12CCC(C(F)(F)CC1)CC2=O.c1(OC)cc([N+](=O)[O-])cnc1O Cc1ncnc2c1CC(C(N1CC3CC1C3NC(C1CC3CC3C1)=O)=O)CC2 c1(C(=O)NC2(CNC(C(C)OCC(F)(F)F)=O)CC2)cnc2ncccc2c1 C1(C(=O)NC2CC3CN(C(CCCCC)=O)CC2C3)CCc2nnc(C)n2C1 N1(C(CC2(C#N)CCC2)=O)CC(NC(C2CCCCS2(=O)=O)=O)C2CCCC2C1 C(CCN=C(NCC(N1CCOCC1)C)NC1CCCC(F)(F)C1)OC c1(OC)c(O)cc(CN2CCC(C(N3CC4CCCCC4C3)=O)C2)cc1Br c1(C(N(CCC(C)NC(c2c(CC)nccc2)=O)C)=O)ncc2ccccn12 Cc1cc(C(=O)NCCC2(NC(=O)CC3OCCO3)CCC2)nnc1O CCCC(C)(CC)C(=O)N1CC(n2cc(C3C4COCC34)nn2)C(C)C1 CC1CN(C(=O)CC2COCC(C)(C)O2)CCN1C(=O)CCC1(C)CC1 c1(CC(=O)N(CC(C)O)CCNC(=O)CC2CN(C)C2)ccc(Cl)cc1Cl C1(OC)CC(NC(C2CN(C)C2)=O)CN(C(=O)CN2C(=O)CCC2=O)C1 C1(C)(C(N(C(C2CCCC2)CNC(c2ccnn2CCF)=O)C)=O)CC1(F)F CC(C)CCCC(C)C(=O)NCC1CC1NC(c1cccnc1N(C)C)=O n1(CCCC(=O)N(C)CC2(O)CN(C(C3(C(C)C)CC3)=O)C2)ccccc1=O c1(C(=O)NCCN(CCC)C(C2(C3CCCO3)CC2)=O)ccn(CC)c1C C(CC(C)C)(C(=O)N(C)C)NCc1nnc(COC)o1 c1(-c2n(CC(=C)C)c(N(C)Cc3ccc(Br)o3)nn2)ccc(C)nc1Cl c1(SCCNC(=O)C(N2CCCC2C2CC2)=O)noc2cc(F)ccc12 C1(N(C(c2nc(OC)oc2)=O)CCO)CCCN(C(C2(CC(C)C)CC2)=O)C1 c1(CC)cc([N+](=O)[O-])ccc1NC1(CNC(c2cncnc2CC)=O)CCC1 C1(C#N)(SC)CN(C(=O)C(C2CC2)N(C(=O)CNC(=O)C2CC2)C)C1 C=CCCN=C(NCC(=O)NC)NC(c1nnnn1C)c1ccc(F)s1 c1(C(=O)NCC(C2CCC2)NC(CC2C(CC)C2)=O)cscc1SC S(=O)(=O)(CC(C)C)N1CCC(C(=O)Nc2ccc(C(=O)OCC)[nH]2)C1 C12(C(=O)NC(C(N3C(C)CCCC3)=O)Cc3cnc[nH]3)CCCCC1OCC2 N1(C(CC)=O)CC(NC(=O)C(C)(C)C2CCOCC2)C(CC)C1 CCC(C)(C)C(=O)N1CCOCC1C(=O)NCC1CCOC1 CC1=NOC(C(=O)NCC2CC2CC(=O)N(C)OCc2ccccc2)C1 C(C1CCN(C(=O)CC2CC2)CC1)=CC(=O)NCc1ccc(O)c(F)c1 c1(S)ccc(C(N)=O)cc1.C1(N(S(C)(=O)=O)Cc2ccc(OC)o2)CCN(CC)C1 C(CC(C)(C)C(=O)N1CCC1C1CCC1)NC(CCc1onc(C)n1)=O c1(OC)cccnc1C(=O)N(CCCNC(C1(O)CCC1)=O)Cc1ccccc1 N(C(=NCCCF)NC1CCC1n1ccnc1CN1CCc2ccccc21)CC N1(C(CCC(C)=O)=O)CC=C(C(C)(C)C(=O)N2CCCC2C(C)(C)C)C1 N1(C(C2CC(OCC)(OC)C2)=O)CCC2CN(C(c3cc(O)nn3C)=O)CC2C1 CC1C(NC(c2cc(Br)c[nH]2)=O)CCCN1C(c1cc2n(c1)CCC2)=O CC1CCC(CNC(c2cscc2Cl)=O)CN1C(=O)CN1CCNC(=O)C1 c1(OC)c(C(N2CCC(=CCNC(=O)CC3COC(=O)C3)CC2)=O)ccnc1Cl c1(CCC)cc(C(=O)NC(C)C(C)NC(=O)CNC=O)no1 C1(CNCC(c2ccccc2C)OC)CCc2c[nH]nc2C1 c1(C2CCN(C)C2)cc(C(N2CCC3CC23C)=O)cnn1 c1(CC(=O)N(CC(C)NC(C2(CCC)CC2)=O)C)cc2ccccc2cc1O S(=O)(=O)(c1ccc(NC2CC(OC)C2)c(Br)c1)N1CCC(CC)(CC)C1 c1(C(N(C2CCN(C(=O)C(CSC)c3ccccc3)C2)CC)=O)sccc1F CC(C)C(CNC(c1ccc(C#N)n1C)=O)C(=O)NCCCC1(C)CC1 N1(c2c(OC)cncn2)C(CNC(c2ccc(C3CC3)o2)=O)CC2COCC12 C(=O)(CCS(C)(=O)=O)N1CC=CC(NC2C(C(=O)NC(C)(C)C)C2)C1 N1(C(c2c(C(=O)N(C)C)csc2)=O)CC2CCN(C(C3COCCO3)=O)CCC2C1 c1(OC)cc(NC(C2(NC(C3CC(SC)C3)=O)CCCC2C)=O)ccc1O C1(CSCCNC(CCCCC=C)=O)CN(C(=O)CCC(=O)NC)C2CCN1C2 C1(C(=O)NCC(CC)C)CCN(C(=O)c2ccc(CO)cn2)O1 CC(CC1CCC1)C(C(=O)NCC1CC1)N1CCC(n2cc(Cl)cn2)C1 Brc1ccc(C2CC(C(F)(F)F)(Nc3ccccc3F)C2)nc1 c1(C(=O)NCC(C2CCCCC2)NC(=O)CN2CC3CC3C2)ccc(O)cc1F c1(C(=O)OCC)c(C)sc(NC(C2CC2N2CC(NC(=O)NCC)C2)=O)c1C.OC c1(C(=O)NC(CC=C)CNC(=O)C=CC(=O)OCCCC)cnc2n1CCC(C)C2 C(=O)(C1=C(Cl)CCOC1)NC(C1C(C(N2CCC(C)(C(=O)OC)C2)=O)C1)C O=CS(=O)CCc1cn(CCCNC(=O)C(c2ccccc2)O)nn1 C(=O)(C(C)(C)C(N)=O)N(CCN(c1snc(SC)n1)C)C N1(C(C(CC=C)CC)=O)CC(CNC(c2cc(Cl)cn2CC)=O)OC2(CCC2)C1 c1(C(N2CC(CNC(C(C(=O)OC)C)=O)C2)=O)cc(N(C)C)ccc1Br C(CNC(c1ccc(CN2CCCC2)cc1)=O)(C(C)(C)C)NC(C=COCC)=O c1(C(=O)NCC2C=CCN2C(=O)C=CC=C(Cl)Cl)c(F)cc(F)cc1Cl C1(NC(CONC(Cc2cnc(C)s2)=O)=O)CCCN(C)C1C C1(OC)(CNC(=O)CCCN(C)C(C)=O)CCCN(C(=O)C(C(=O)OC)OC)C1 N1(C(C(C(C2C(CC)C2)CC)OCC)=O)CC(COC)C(O)C1.C12(CCOCC1)C(=O)NC2 C1(c2cc(C)no2)C(NC(=O)CC2CC2)CCCN1C(=O)CCCN1CCCC1.N1(CS)CCCC1 C1(NC(c2cc(C)[nH]n2)=O)CN(C(=O)C=Cc2ccc(C(F)F)o2)CC1C C=C(CNC(c1conc1C)=O)CCNC(c1c[nH]cc1-c1cnn(C)c1)=O O=C(C1=COCCO1)NCC1CCCCN1C(=O)Cn1cnc(C(F)(F)F)c1 c1(CC)ccc(C(=O)NC(C(=O)N(CC(C)O)C)C2CCCC2)nc1 C1(CCC2N(C(C(C)CC3CC3)=O)CCC2)CCCCN1C(=O)CN(C)C1CC1 Cc1ccc(C)c(C(N2CCC(NC(=O)CNc3nccs3)C(C)C2)=O)c1N C(=O)(CCCCCc1cccs1)N(C1(CNC(C2CCC3CC3C2)=O)CC1)C N1(C(C(C)OC)=O)CC(CNC(=O)CCCN=[N+]=[N-])C2(CC2)C1 CCC(C)(C)C(C)CC(=O)NC(C)CNC(c1cc(C(C)(C)C)ccc1O)=O N1(C(c2c(C)sc(Cl)n2)=O)CCCCC(NC(C2(C)CCCOC2)=O)C1 C1(C(=O)NCCC2C(C)C2)CC2(CC(NC(=O)C(c3ccc(F)cc3)(C)O)C2)C1 CC(C)(O)C(F)C(=O)N1CCCC1C(=O)N(C(C)(C)C1CC1)Cc1ccc(Cl)nc1 N1(C(CCc2cc(OC)no2)=O)CCC(NC(c2ccn(C)n2)=O)C1(C)C C1(C(=O)NC(C)(C)CNC(=O)Cn2cnnn2)CCn2cnnc2C1 C1(C2CC2)(CNC(C(CC)SC)=O)CCN(C(=O)CCCN(C)C(C)C)C1 Cc1cc(F)ccc1C(O)C(N1CCC(F)C(NC(=O)Cn2cncn2)C1)=O C=C1CCC(C(=O)NCCCN2CCC(NC(c3ccc(OC)cn3)=O)C2)CC1 c1(C(N2CC(F)CC(NC(C3CC(C#N)(OC)C3)=O)C2)=O)c(C)cc(Cl)cc1C C(=O)(C(F)C(F)(F)C(F)(F)F)NCC(CNC(C1(C(=O)OCC)CC1)=O)(C)C C1(CNC(C=CCCC)=O)CC2(CCN(C(=O)C(CC)C3CCOCC3)C2)CO1 C(C)(C(C(=O)NCCC1CCSC1)NC(=O)C(F)C(C)C)OC C(=O)(C1OC(=O)c2ccccc21)N1C2CC(CC(CNC(C)=O)C2)C1 c1(NC(CC(c2ccc(C)cc2)C)=O)cc2c(C)noc2cc1C C1(CCCCNC(C=C(C)C(C)C)=O)CCN(C(=O)Cn2cc[n+](C)c2)CC1 c1(N2CC(OC)(CNC(C3CC3(C)C(F)F)=O)C2)cc(C(C)C)nc(C(C)C)n1 C=C(Cl)CC(C(=O)NC(c1cccnc1O)C)NC(=O)CC(O)CN(C)C C1(C(C(=O)NC2CC(N)C2)F)CCCCC1 C(C(C)C)(CC(C)C)NC(C(CN(C(=O)CC1(O)CCCOC1)C)C)=O CCC(C)(COC)CNC(=O)CCC1CC(NC(C2COCCN2C)=O)C1 c1(C(C)=O)ccc(C(=O)NCC(C)(C2CC2)NC(=O)C(O)C(F)F)c(F)c1 C1(C(=O)NCC(CC(=O)NC(CCOCC)C)OC)CC(=O)N(OC)C1 CC1=C(C(=O)N2CC(O)CC2CC(N2CCC3CCCC23)=O)CCCO1 c1(C(N2CC(CNC(c3nc(CCCC)sc3)=O)C2)=O)ccc2nc(O)[nH]c2n1 CC(C)C(F)(CN(C(=O)CCc1ccn(C)n1)C1CC1)C(=O)NCC(F)F Cc1nc2c([nH]1)CC(C(=O)NCC1C3CN(C(=O)Cn4cccn4)CC13)CC2 C(=O)(CS(=O)(=O)CCO)NCCC1CN(C(=O)C2=NOCC2)CC(C)O1 C1(C(=O)N(C2(CNC(=O)CN3CCOCC3)CC2)C)(OC)CC(C)CC(C)C1 C12(CNC(CCSC)=O)CCCN(C(=O)Cn3cnnc3O)C1C2 CC1CN(C(C2(O)CCOCC2)=O)CCC1N(C)Cc1ccc(OCF)cn1 C1(NC(Cn2ncc(C)c2)=O)CC2CN(C(C3CCCSC3C)=O)CC12 C1(C(=O)NCC2CC2Cc2ccoc2)(CNC(C(C)=C(C)C)=O)CC(C)(C)C1 c1(CC(=O)NC(C2CCN(C(=O)C(c3ccccc3)C)C2)C#C)ccc(Cl)cc1 C(CCN=C(NN1CCOCC1)N1CCC(C)(CN(C)C)C1)OCCOCC C1(O)(C(C)NC(CCCSC)=O)CCN(C(=O)CN(C)C(=O)C2CC2)C1 C(=O)(CC(C)(C)CC(=O)NC1CC1CNC(c1cc(Br)c[nH]1)=O)OC CCC(C)(CC)C(=O)N(C)CC1CCC(CNC(c2ccc(C#N)s2)=O)CC1 C1(NC(CC(COC)C)=O)CN(C(C2(OC)CS(=O)(=O)C2)=O)CC(C)(C)C1 N1(C(CCCOC(CCC)=O)=O)C2CCC1CN(C(=O)CC1CC3(CC3)C1)CC2 C1(NC(CS(CC)(=O)=O)=O)CCN(C)C12CCCN(C(=O)C(C)C)C2 C1(C(N2CCC(N(C(=O)Cn3ncccc3=O)CCC)C2)=O)CCC(O)CN1C N1(C(C=COc2ccc(OC)cc2)=O)CC2CC1CN2Cc1csc(C)n1 C1(C(=O)NC(CCNC(C2CCC(NC(C)=O)CC2)=O)C)CNC(=O)C(C)(C)C1 N1(C(CNS(N)(=O)=O)=O)CCC(Cn2cc(-c3ccc(C(=O)O)o3)nn2)C1 c1(C(=O)NC2C3C(C)N(C(=O)CCC4CCCCC4)C2C3)ccc2nccn2n1 Cc1cc(CNC(=O)C(Cn2cncn2)NC(=O)CCC2CCCO2)c(C)s1 N1(C(COC2(C)CCC2)=O)CC=C(CNC(C2CCCC(N(C)C)C2)=O)CC1 C1(NC(C(C)OCC#C)=O)CCCCC1NC(=O)C=C(C)CN1CCOCC1 c1(C(=O)NC2C(NC(c3scc(C)c3)=O)CC2)cccc(Cn2ccnn2)c1 N1(C(C(C2CCCCC2)C)=O)CC(O)(CNC(c2c[nH]c(=N)s2)=O)C1 C1(C)(CC)CC(NC(=O)C2=CCC(NC(=O)CC3(C)CCCCC3)C2)CCO1 c1(OC)cc(C(=O)OCC2CCCC3CCCN23)c(F)cc1Br N1(c2cccc(C(=O)OC)c2)C(=O)NC(C(c2ccccc2)C)C1=O N1(C(C=C(CC)C)=O)CCC(NC(c2ccc(C)nn2)=O)C1(C)C c1(SCCC(=O)NC2(CN(C(=O)Cc3cncs3)C)CC2)ccc(Cl)cc1 Cc1nn2c(NC(=O)CC(C(F)F)n3cccn3)c(N(C)C)nc2s1 c1(COC)nc(OC)cc(N(CCCNC(=O)C(c2cc(F)cc(F)c2)O)C)n1 C1(NC(CC(=O)OC)=O)CCOC2(CCN(C(c3ccc(Br)cc3Br)=O)CC2)C1 c1(OC)cccc2c(O)nc(=NCC(c3ccc(Cl)cc3)C3CC3)[nH]c12 C=Cc1cnn(C)c1C(N1CCN(C(C2CCN2S(C)(=O)=O)=O)C(C2CC2)C1)=O c1(C(N2CCC(O)(CNC(CC(C)OC)=O)C2)=O)cc(O)ccc1C(C)C C1(C(=O)NCCn2cc(C(=O)Nc3ccc(O)cc3)nn2)C2C3CCC(C3)C12 CC1CC2CCN1C2=O.c1(NC(=O)COCC(F)F)cnn(-c2nccs2)c1 N1(C(=O)OC(C)(C)C)CC=C(CCC(N2CC(CC3(C)COCCO3)C2)=O)CC1 Cc1nn(C)c(=O)c(C(=O)NC2CC2CNC(=O)CCCCC(F)F)c1C C1(C(=O)NCC(C(=O)N(CC(N2CCCC2)C)C)O)CCCN1C=O c1(C(=O)NC(CNC(C2CC(C)(CC)OCC2)=O)CO)ccc2nc(O)[nH]c2n1 C(CN(C(c1[nH]cnc1C)C(=O)NCCCF)C)(CC(C)(C)C)OC c1(OC)cccc2c1OCC(NC(c1ccc(C)cc1)C1CC1)C2.c1(S)n[nH]cc1Br CC1CC(CNC(c2ncccc2Cl)=O)CN1C(=O)CCc1ccnc(Cl)c1 c1(NC(=O)NC(c2ccncc2)CC)ncccc1OCC1CC1.c1(NS)cscn1 C1(NC(=O)Oc2ccccc2)CCC2CN(C(=O)CCc3nc(O)n[nH]3)CC2C1 c1(C2(C(=O)NC3(CC)CN(C(CCC=CCC=C)=O)C3)CC2)cc(F)ccc1C Cc1cccc(C(=O)NCCC(C)(C)NC(C2CC2c2ccccc2F)=O)c1C C(=O)(CCCC(C)O)NC(C1CN(C(C2(C3CCC3)CC2)=O)CCO1)C C12(CC(=O)O)CCOCC1CN(CCc1ccc(CCO)cc1)C2 C1(NC(C=Cc2ccc(CC)o2)=O)CN(C(=O)CCC(C)(C)F)CC1(C)C N1(C(C2(C(=O)OC)CC2)=O)CC2(C1)CN(C(=O)C(C)CC(F)F)C2 c1(C(=O)NC(C)CCCCNC(=O)CCc2cnoc2)ncn2c1COCC2 c1(C(C)N(C=O)C)ccccc1S(C)(=O)=O.C12CN1CCC2(C)C c1(CC(N2C3CC(CNC(C(C)NC(=O)NC)=O)(C3)C2)=O)ccc2c(c1)COC2 C1(CNC(C2CCCOC2)=O)CCCC2(CN(C(=O)CCCC3CCC3)C2)O1 C(=O)(C(C)(O)CC(C)C)NCC1CC2(CN(C(C3N(C(=O)NC)CCC3)=O)C2)C1 c1(C(=O)NCC2CCC(F)(CNC(CNC(CC)=O)=O)C2)cnc2ccccn12 N1(C(C(CCCOC)C)=O)CCC2CN(C(C3(C)C=CCS3)=O)CC2CC1 C(=O)(C1=CSCCO1)N1C(CN(C(C=CC=CC)=O)CC)CCC1 CCCCC(CCCC)C(=O)N(C)CCOCCCNC(=O)CCP(C)(C)=O c1(OC)ccc(C)c(NC(=O)C(c2cnn(C)c2)NC(c2nnccc2C)=O)c1 C1(NC(c2occ(C)c2)=O)C2CC3C(C2)C13C(N1CC2C(C1)C2(F)F)=O c1(C(=O)NC(CCCCNC(c2c(C)csn2)=O)C)scc2c1CCCC2 c1(NC(CNC(C=C(C)C2CC2)=O)=O)ccc(Oc2cccs2)cc1 Cc1ccc(F)c(OCC(=O)N(C)CCNC(=O)C=CCN2CCCC2)c1 C#Cc1ccc(F)cc1C(=O)N(CCCNC(=O)C(C)CC(N)=O)C1CC1 C1(CNC(Cn2cc(C(C)=O)nn2)=O)CC2CC1CN2C(=O)C(C1CCCCC1)C c1(C(N(CC(C)C)CC(=O)NCC2CCC(F)C2)=O)nc(O)nc(O)c1F C12(NC(C(F)OC)=O)COC(CNC(C3CCN(C)C3=O)=O)(C1)C2 N#Cc1cccc(C2CCCN2C(c2ccc(CO)o2)=O)c1 CC1C=C(C(=O)N(CCCCN(C(=O)C(C)N(C)C)C)C)CC1 N1(CC)CC(C(N2CC(OC)C(C(=O)N(CCCC(C)O)C)C2)=O)CC1=O c1(C(=O)NC(c2c(OC)cccc2)c2nccn2C)c[nH]c(C)cc1=O C12(CNC(c3c(C)c(CO)ccc3)=O)CN(C(=O)Cc3ccon3)CC(F)(C1)C2 C(=O)(CCCCCC(C)C)N1CC(CNC(c2n(CC)ncc2)=O)CC12CCC2 C(=O)(C(C)CS(C)(=O)=O)NC1CCN(C(COCc2cc(C)on2)=O)C1C C(=O)(C(CNC(=O)CCC(C)CC)C(C)(C)C)N(CCOCC)CC Cc1cccc(C(N2CC3(C2)CN(Cc2cccc4nccn24)C3)=O)c1[N+](=O)[O-] C=C=CC(C)C(=O)N1CCCC1CN(C(c1cnc(CC)s1)=O)CC c1(C(=O)NC(C2CCN(C(C3(C)CC(C)OCC3)=O)C2)C)ccn2ccnc2c1 c1(C(=O)NC(CN(C(c2ccc(OC)cc2)=O)CC)C)ccncc1NC N1(C(c2ccc(CC)s2)=O)CCCCC(NC(=O)CCCC(C)C)C1 c1(C(=O)OC)ccc(O)c(C(N2CCC(NCc3cscn3)C(F)C2)=O)c1 C1(NC(c2cnn(Cc3nc[nH]n3)n2)=O)(CF)CCN(CC(=O)NCC2CC2)C1 CC(C)C(COCc1ccccc1)N(CCCN(C(=O)C)C)C.C(=O)(C1CC1)N [N-]=[N+]=NCC(C(=O)NCC12CCC(CC1)C2)NC(=O)CSc1nc[nH]n1 C1(OC)CC(C(=O)NCCC2CSCCN2C(=O)CC23CC(C2)C3)CC1OC n1(C(N2CCN(CC(c3ccccc3)O)CC2)C)cnc2cccnc12 C(=O)(C(C)CCC(C)(C)C)NC1CN(C(c2c(F)ccc(CC)c2F)=O)C2C1C2 C1(NC(c2cccs2)=O)CC1C1CCCN(C(C2CC23CCC3)=O)C1 C(=O)(N=c1cc(C)c(C)n[nH]1)N1C(Cn2c(C)cc(C)n2)CCCC1 c1(CC)cc(C)c(C(=O)NCC(O)CNC(c2c(C(F)(F)F)noc2C)=O)o1 c1(C(C)OC(c2cccc(CNC(=O)OC(C)(C)C)n2)=O)c(F)cc(Br)cc1F C#Cc1cc(C(=O)NC2CCCCC2NC(c2ccc(C)cc2N)=O)ccc1C CC(C)(C)C(O)C(=O)NCC1(C(C)(C)C)CCN(C(c2cncc(F)c2Cl)=O)C1 CCC(C)(C(=O)NCC1CC(O)CN1C(c1sc(C2CC2)nc1C)=O)C(N)=O c1(NC(=O)NC2CN(C(=O)C(F)OC(F)(F)F)CC2F)ccc(Br)cc1F c1(C(=O)NCC(CNC(C(C)NC(COC)=O)=O)(C)C)ccccc1OCCF C1(NC(C(C=C)O)=O)CC2CC1CN(C(c1cnc[nH]1)=O)C2 C1(NC(C2C(C)C2C)=O)CCCC(NC(=O)CN2CCOCC2=O)CC1 C1(N2CCC(C(=O)OCC)C2)CCS(=O)(=O)CC1 C(C(=O)COC(C1CC1F)=O)SC(C)(F)F Cc1cc2nc(C(=O)NCC3CC3NC(=O)Cc3cscn3)ccc2c(=O)n1C C1(c2n(C)ccn2)CN(C(=O)C=C2CC2)CCN1C(C1CCCCC1(C)C)=O C(=O)(C(CC(F)F)NCCCO)N(C(CC(=O)OC)C=O)CCO C12(CNC(NOC(c3ccc(O)nc3)C)=O)CCC(C)(C1)C(=O)N2 C1(OC)CC(CNC(=O)C(C)(C)CN(C)C)N(C(C2OCCC2C(F)(F)F)=O)C1 c1(C(C)CNC(c2cccc(NCC3CC4C=CC3C4)c2)C)cc(Cl)cc(Cl)c1 c1(C(=O)NC2C=CCN(C(C(C=C)(C)O)=O)C2)cnc2ccnn2c1 C1(CC(N2CC(NC(c3ccc(C(N(C)C)=O)cc3)=O)C2)=O)COCC(C)(C)O1 c1(C(=O)NCC2C(NC(C(C3CC3)OCC)=O)CCC2)ccc2oc(S)nc2c1 N1(C(C(CC(C)=O)(C)C)=O)CCC2(CCN(C(=O)Cn3cncn3)CC2)C(C)C1 C1(C(N(C(=O)CCOCCCSC)N2CCCC2)=O)CC(=O)N(OC)C1.CC c1(-c2c(C(=O)Nc3c(OC)nc(Cl)nc3)nccc2)cc(Cl)c(O)cc1F N1(C(Cc2nccc(OCC)n2)=O)CCCN(C(C2(OC)CC2)=O)CC1C c1(C(N2CC(NC(CN(C)C(c3ccoc3)=O)=O)C(F)C2)=O)ccc(F)cc1Cl C(C)(C)(C(C)CC(=O)NCCN(C1CCCC1)C)NC(CCC(C)OCC)=O C#Cc1ccc(C(N2CCC(C)(C)C(NC(=O)C(O)CCC)C2)=O)c(F)c1 C1(C(=O)NC2C3CN(C(C(C)=C4CC4)=O)CC32)CCC(C)(O)CC1 c1(OC)c(C(N2CC3CC2CN3Cc2cc(F)nc(F)c2)=O)cc(Cl)cc1Cl N12CC3(CC(CO3)C1=O)C2.N1(C(c2c(CC)cc[nH]2)=O)CCC(CC)CC1CC c1(COC(C(C2CCN(CC)CC2)C)=O)ccc(Cl)c(Cc2cc(F)cc(Br)c2)n1 N1(C(C2N(C)CCC2)=O)CC2CC2(C(=O)NC2C=CCCC2)C1 C1(CNC(=O)Cc2cccs2)CN(C(c2csc(-c3ccncc3)n2)=O)C2CC12 C1(CN(C(=O)CCC2CC2(C)C)C)CCN(C(=O)CCCc2n[nH]c(=N)s2)CC1 c1(OCCC(=O)NCC(CO)NC(C2(C)CC2)=O)ccccc1 C(N=c1[nH]cnc2c1CCCC2)c1c(C(=O)OC)cncc1 c1(C(N2CCCC2C2CCCN(C(=O)C(F)(F)C3CC3)C2)=O)cc[n+]([O-])cc1 CCC(CCCC(=O)N(CC(C)(C)N(C)C)C)NC(c1cc(CCO)on1)=O c1(N2C(=O)CN(C(N3CCC(CC#N)CC3)=O)C2)ccnc(C(=O)O)c1 c1(C(=O)Nc2ccnnc2)cc2nc(-c3c[nH]c4ncccc34)ccc2[nH]1 N1(C(C(CC=C)OC)=O)CC2(CNC(c3occ(C)c3C)=O)CC1CCO2 C(c1ccc(CN2C(C(=O)Nc3cccc(I)n3)CC3CC23)cc1)=CC(=O)O N1(CC(=O)NCC2CC(F)(CNC(C3CC3(Cl)Cl)=O)C2)CCCCCC1 c1(C2(CNC(=O)NC(C(CC)O)c3ccccc3)CC2)ccccc1OCCO N1(C(c2ccn(C)n2)=O)CCC(C)(C)C1CC(=O)NCC1CNC(=O)C1 c1(C(=O)NC2C(NC(c3nc(C)nc(O)c3)=O)C2)ccc2c(n1)CCC2 CC(C)(C)C(CN=c1[nH]cnc(Cl)c1Br)NC(=O)Cc1ccccn1 C1(C(N2CC(C3CC3)(OC)C2)=O)CC2C=CC1N(C(=O)CCC(C)(C)F)C2 C=C(C)CCCC(=O)N(C1CCN(C(c2cc(C)cc(F)c2)=O)C1)C CCC(F)(CNC(C1(F)CCN(C(=O)CC2CC(C)(C)CO2)C1)=O)CC CC(C)C(O)C(C)C(=O)NC(C1CN(C(c2coc(CN(C)C)n2)=O)C1)C N1(C(C(C)OCCOC)=O)CCCC(N(C(c2csc(CC(F)F)n2)=O)CC)C1 c1(C(=O)NC2CCC(NC(C3N(CC)CC3)=O)C2)ccc(OC(F)(F)F)cc1C N1(C(C(C=C=C)C)=O)CC(C(=O)NCC2CCCC(C)(C)O2)C2(CCC2)C1 C(=O)(CC(C)F)NCCN(C(=O)CCNC(=O)OC(C)(C)C)CC(C)O c1(C(N(C)Cc2c(Cl)csc2Cl)=O)cc(NS(C)(=O)=O)ccc1F C1(CN(C)C(C2CC(C)(O)C2)=O)CN(C(=O)C(Cl)=CCl)CCO1 c1(C(=O)NC2C(CNC(CC(COC)(C)O)=O)CCC2)csc2c1CCCC2 C12CCC(CC1)C(C(=O)NC)N2C1CCCCC1.C1(COC)CC(CO)C1 CCC(C(=O)NCC1(F)CCCN(C(c2conc2C)=O)C1)C(C)C C1(C(C(=O)NC(C)C)N(C)CC2(OC)CCC2)Cc2ccccc2C1 c1(C(=O)NCC2CC(CNC(c3cc(C)oc3C)=O)OC2)ccn2cncc2c1 C(=O)(CCCC(=O)NCC)NCC(COCC)NC(=O)C(CC)C(C)O.C(C)(C)(C)O N1(C(CCC(C)C)=O)CCC(NC(c2ncc[nH]c2=O)=O)C(c2ccccc2)CC1 c1(NC(C)=O)ccc(C(=O)NCC2(NC(C34CC(F)(C3)C4)=O)CC2)cc1F C=CCC(C)(C(=O)NC(C)CC(C)NC(c1cccc(CC#N)c1)=O)N(C)C N(C)(C1CCOc2c(C)cccc21)C(c1scc(C)n1)C(=O)NC1COC1 C1(CNC(COCCCC)=O)CN(C(=O)Cc2nccn2C)CCCO1 C(=O)(C(C)C(C)C)NCCC1CC(NC(CSCCN(CC)CC)=O)C1 c1(CNCC(C(F)C2CCCN2)F)ccccc1-n1ccnn1 C1(NC(C(C)OC)=O)CN(C(c2cc(Cl)c(F)cc2Cl)=O)CCC1(C)C N1(C(COCC(C)C)=O)CC2CN(C(=O)Cc3ccc(C#N)cc3)CCC12 C(CCCCC(=O)N1CC(C)(C(=O)N(C2CCCC2C)C)C1)OC c1(C(=O)NC(C(CO)NC(c2c(SC(C)C)nccc2)=O)C)cccc(O)c1F N1(C(C2N(C(C)C)CCC2)=O)CCC(C)C(CNC(=O)C2=C(Cl)CCC2)C1 N1(C(c2c(C)nc(Cl)s2)C(=O)NC2COC2)CCC2CCC2C1 N1(C(CC)=O)CCCCC1C(N1CCC(CNC(c2cc(C)c(C)o2)=O)CC1)=O C(=O)(CC(CC1CC1)NC(c1ccc(C)cn1)=O)N(CC)Cc1noc(C)n1 c1(C(=O)NCCCN2CCN(C(c3c(C)nn[nH]3)=O)CC2)cccc(F)c1F N1(C(=O)CN(C(C23CCC(CC2)C3)=O)C2CC2)Cc2n[nH]cc2C1CO N1(C(C2C(C)(C)CCO2)=O)CC(NC(C2CC3(CCO2)CC3)=O)C(C2CC2)C1 C1(NC(C(c2c(C)cc(F)cc2)O)=O)C2CC3CN(C(c4ccc[nH]4)=O)C1C3C2 C(=O)(CC(C1CC1)C1CC1)NCCOC1CC(N(C(=O)CCC2CCCO2)C)C1 C1(NC(c2n(CC#N)ncc2)=O)CC2(CCCCN2Cc2cccs2)C1 c1(C(C(=O)O)N(C(C(F)(F)F)c2ccccc2)C)ccc(F)c(F)c1.C(C)(C)(C)OCCl c1(CCC)n[nH]c(=NCCCCC(C)NC(=O)C(=Cc2ccncc2)C)s1 N1(C(COCCCC(C)C)=O)CC2CC1C2NC(C1CCC1)=O n1(CCC)ncc(C(=O)NC2CC3(C2)CC3NC(c2ccc(CC)[nH]2)=O)c1C N1(C(C(c2ccccc2)OC)=O)CCCC(C(N2CCCC2CN=[N+]=[N-])=O)C1 C1(N(C2CCCN(CCC)C2)CC=CC)CCC2(CCCC2)C1 C1(C(=O)OCC)CCN(Cc2ccccc2)CC1N(c1cc(N)ccc1F)C c1(C2N(C(c3sccc3CCCSCC)C(=O)OC)CC2)ccc(F)cc1 c1(CNC(=O)NC2(c3ccc(C)cc3)CCC2)cnn2c1OCCCC2 C1(CN(C(=O)COc2cccc(F)n2)CC)CCCCN1C(=O)C=CCF C1(C)(NC(C(CC)COC)=O)CCN(C(c2sc(Cl)c(Cl)c2C)=O)CC1 Cc1cc(C(C)C(=O)NC2CC(CNC(c3ccnc(C)c3C)=O)C2)cc(F)c1 N1(CC(=O)NCC(C)N(C(C(C)=CC)=O)CC)CCC(CC)CC1 Cn1cnc2c1CCC(C(N1CC(NC(c3ccc4scnc4c3)=O)C1)=O)C2 N1(C(C(N)=O)=O)CC2(NC(=O)Cn3cnc(Br)n3)CCC1C2 CCCCC(F)C(=O)N1CC(CNC(c2cc(C)cc(C)n2)=O)CC1(C)C C1(C(=O)NC(C(=O)OCC)CC)CC(C)(C)CCN1C(c1ccnc(C)n1)=O N1(CC)CCCC(CNC(=O)CCOc2ccc(Cl)cc2)C1.C12CC(C1)C(=O)N2 c1(C(=O)NC2CCOC2)ccc(CNC(C(C)CC2CC2)=O)cn1 c1(OC)ccc(Cl)nc1C(=O)NCc1cc(N2CC3C(NC(C)=O)C3C2)ncn1 C(=O)(C(C)(C)C(=O)OCC)N1CCC(O)(CN(C(CC=C)=O)C)C1 O=C(CC1(CN(C(C2CCC2)=O)C2CC2)CC1)NOCCc1ccccc1 N(C(=NCCCCl)NCC(N1CCOCC1)C1CNC(=O)O1)C(CC)C c1(C(=O)NC(C)CCN(C)C(C2CCC2)=O)ccc(Br)c2c1OCCC2 c1(C(C(=O)NCCCOC)N(C2CCCCC2C)C)cc(Cl)c(Br)cc1F C(=O)(C(C)CC(C)CC)N1CCC(C(CNC(c2n(CCC)ncc2)=O)C)CC1 C1(CNC(C2N(CC)CCC2)=O)CCN(C(=O)Cc2ccc(F)cn2)C12CC2 N1(C(C2CC(OCCOC)C2)=O)CCC(CCNC(=O)CC2CCC(C#N)C2)CC1 c1(CN(C(C2(CNC(C(N3CCCCC3)C)=O)CC2)=O)C)cccc(O)n1 c1(NC(C2(C)CCN(C(CC(C)(C)C)=O)C2)=O)ccn2nccc2c1 N1(C(C2(C)CC(C)OCC2)=O)CCCC2(CCCCC2NC(=O)CO)C1 c1(C(=O)NC(C)C(C)NC(=O)CCC(C)CN(C)C)ncc(F)cc1F N1(C(CCOCCC)=O)CCC(C(=O)N(CC(C)C(=O)OC)C)C1 c1(C(=O)NC(CC)CNC(=O)CC2(C)CC2)csc(CC2CCCC2)n1 n1(CCC=C)cc(C(=O)NCC2(O)CN(C(=O)C(F)(F)c3ncccn3)C2)nn1 N1(C(CNC(c2ccccc2)=O)=O)CCOCC1CNc1ccc(C(F)(F)F)s1 C=CCCCC(C(=O)NCC1CCC(CC)CC1)NC(=O)C=NOC C1(C)(C(=O)NC(C)CCNC(=O)CSc2nncn2C)CCC(=O)N(C)C1 C(=O)(C(C)C(=O)NCC1CN(c2cc(N3CCCCC3)ncn2)CCO1)OC Cc1ccc2ncc(C(=O)NC3(CNC(=O)CCC4CCCC4)CC3)c(=O)n2c1 N1(C(c2ccc(C)nc2)=O)CCN(C(=O)C(c2cccc(C)c2)C)CC12CCC2 C1(NC(c2cc(C)ns2)=O)CC12CCN(C(=O)CC1COCC1O)C2 C=C1COCCN(C(C(=O)NCCN2CCOCC2)C2CC2(C)Br)C1 C(=O)(CCCCC(=O)NC)NCC(CC)(C)NC(=O)CC(C)(C)C1CC1 C1(N(C(CCN(C(C)=O)C)=O)CC2CC2)CCN(C(C2(C)CC2(F)F)=O)C1 n1(CC)nnc2c1CCC(C(=O)NCCn1cc(C3CC4(CC4)C(O)C3)nn1)C2 C1(C)(C(N2C(CNC(c3c(CCCC)ocn3)=O)CCC2)=O)CCOC1C C12(C(=O)NCC3(NC(CC(CC)C4CC4)=O)CC(F)(F)C3)CCC(F)(CC1)C2 c1(CNCc2c(NC(c3ccc(I)c(Cl)c3)=O)cccn2)csc2ccccc12 N1(C(c2scc(CC)c2)C(=O)NC2CC2)CCn2c(-c3cccs3)nnc2C1 c1(OC)ncc(F)cc1-c1cn(CCC(=O)NC2CCCN(C)C2)nn1 C1(NC(C2(C)CC3C=CC2C3)=O)CC2COCC(C1)N2C(=O)CC1CCSC1 c1(NC2C(C)OC(C)C2)nccc2c1c(Br)cn2C C12(CNC(CCN(C)CC)=O)CCCC1N(C(C1CCC1(C)C)=O)CCC2 c1(CN2CC(C#N)C(NC(c3ccccc3)=O)C2)cccc2ccoc12 N1(C(c2cc(CCC)[nH]n2)=O)CCC(O)(CNC(=O)C(C)CCOC)C1 C1(C(N(CC(=O)NCC(CO)C2CCC2)CC#C)=O)CC(C2CC2)=NO1 C1(NC(CC(C)c2ccncc2)=O)CN(c2nccc(C#N)n2)CCC12CCC2 Cc1cccc(CC(=O)NC2CC23CCN(C(c2cc([N+](=O)[O-])sn2)=O)C3)c1F N1(C(c2ccc(C(C)C)o2)=O)CCCC2(CCN(C(=O)Cc3ccsn3)CC2)C1 C(CC(C)C)(C(=O)NC(C)CCF)ONC(c1occ(C(C)=O)c1)=O C(C1=CCN(C(C2CCC(Cc3ccccc3)O2)=O)CC1)NC(=O)C=CC1CC1 c1(CC)cnc(CC(=O)NCC=CCNC(C23CCCC2C3)=O)[nH]1 C1(C(=O)NC(C)CCCO)CCC2(CC2)N1C(c1ccon1)=O C1(C)(N(C)C)CCCN(C(=O)C(C(C)(C)C)ONC(=O)CC2(C)CC2)C1 c1(SC)ccnc(N2CCN(C(C)CNC(=O)COc3ccc(O)cc3)CC2)n1 C#CCCCCC(=O)NCC1CC1CNC(c1ccc(C)c(-n2cccc2)c1)=O Cc1cc(C(N2CC(NC(=O)CCCn3ccnc3C)C(C)C2)=O)cc(C)c1 c1(SCC(=O)NC2C(NC(C(C=C)(C)O)=O)CC2)ccc(C#N)cc1 C1(NC(C2CC3CCC2O3)=O)CN(C(=O)CS(=O)(=O)CC2CCCO2)CC12CC2 C(N=c1ccc(C#N)c[nH]1)C1N(C(C2CCN(OC)CC2)=O)CCCC1 C(=O)(CC1COCc2ccccc21)NC(CNC(C(C)(C)CC#N)=O)(C)C c1(CCC)cc(C(N2CCC(N(CCC)C(c3ocnc3C)=O)CC2)=O)nn1C Cc1nc(C(N2CCC(CO)(NC(c3ccn(C)n3)=O)C2)=O)c(C)n1C c1(C(=O)NCC(C)N(C(=O)Cc2nonc2C)CC)ccccc1Br c1(C(=O)NC2C(NC(C(=Cc3cccs3)C)=O)C2)cnn(C(C)C)c1F c1(N2CCOCC(CNC(C3CCCSC3)=O)C2)nc2ccc([N+](=O)[O-])cc2s1 C1(NC(C2(COC)CCCCO2)=O)CN(C(=O)Cc2cc[nH]n2)CC1(C)C Cc1cccc(F)c1C(=O)NC(=O)CCN1C(=O)CN(C)C1=O Cc1ccc(CC2C(=O)O2)cc1.c1(OCC2CN(CCO)C2)ccccc1 c1(C(=O)NCC2C(NC(c3c(COC)onc3)=O)CCC2)nc(C(C)C)oc1C CC1=C(C(=O)NC23CCC(CC2)N(C(C2(C)CC2(F)Cl)=O)C3)CCS1(=O)=O C1(CCC(=O)NCCN(CC(C)O)C(=O)C=CC=C(Cl)Cl)CCCC(=O)N1 c1(OCC(n2cc(CNC(C(c3ccccn3)C)=O)nn2)C)ccc(F)cc1Br C(CC(N)=O)(C(=O)NCC(C)(C)N1CCCC1)NC(C1CCC(CC)O1)=O N1(C(C(C2CC2)OC)=O)CCOC(CNC(=O)C=CC2CC2)C1 N1(C(C)C(=O)NCC(O)CNC(c2ccsn2)=O)CCCCCC1 c1(C(=O)NC2CC(NC(=O)C(CO)c3ccccc3)C2)cccc[n+]1[O-] c1(C(N2CCC(n3cc(CC(=O)OC)nn3)C2)=O)cc2cc(C)ccc2nc1C N1(C(c2c(C)n[nH]c2)=O)CCC(OC2CN(C(C3(S(N)(=O)=O)CC3)=O)C2)CC1 c1(C(=O)NC2(C)CN(C(=O)COC(F)F)C2)cccc(=O)n1O N1(C(c2cc(N)c(N)nc2)=O)CC2COCC(C1)C2NC(c1cnsn1)=O CC1(C)C(NC(=O)Cn2nccn2)C2CCCN(c3ccnc(C4CC4)n3)C12 C12(C(C)=O)CC3CC(C1)CC(N=c1ccnc(C(=O)NCCC4CC4)[nH]1)(C3)C2 c1(NC(c2nnnn2C)C)ccc(C(F)(F)F)cc1I C(=O)(CC(C)(C)C(F)F)NC(CNC(CCC(C)CN(C)C)=O)(C)Cn1cccn1 C12(NC(CC(n3c(CC)ncc3)C)=O)CCC(C1)N(C(C1(C)CSC1)=O)C2 C1(C(N(CCCOCC)CCO)=O)CCC(C(C)C)N1C(=O)C(O)CC Cc1ccc(C)c(-n2nc(-c3cccc(C)c3)nc2-c2cc(C3(C)CC3)on2)c1 c1(CCC(N2C3C(NC(C=CCC)=O)C(C3)C2C)=O)c[nH]c2ccc(C)cc12 C1(C(N2CCN(C)CC2CNC(C2CSCCS2)=O)=O)CCC2(CCCC2)CC1 N1(C(C(C)(C)O)=O)C2CCC1(Cn1cc(CCC3CCCCO3)nn1)CC2 C(C)(C(C(C)C)NC(c1ccc(-c2ccco2)o1)=O)NC(C(C)=CC(C)(C)C)=O C(=O)(C(C)(C)C(C)(F)F)NCC(C(=O)N(C)Cc1cnc[nH]1)O C1(C)(COC)CC(NC(=O)CNC(=O)CC(C)(F)F)CN1C(c1nncs1)=O N1(C(COCCC)=O)CCC2(CC1)CN(C(=O)C(=O)C(C)(C)C)CCO2 CC1CC(=O)NC(C(N2CCN(C(c3cc(C4(C)CC4)on3)=O)CC2C)=O)C1 N1(C(=O)NCCC=C)CC2CCC1C(Nc1cc(Cl)c(OC)cc1Cl)C2 C1(C(=O)NC2CCNC2=O)(OC)CCN(CC(=O)N2CCC2)CC1 c1(C(=O)OC)cc(NC(C2(C)CC3CCC2C3)SC2CCC2)cc2c1OCCO2 c1(C(=O)NCCC(CNC(C(CCC)C)=O)O)ccc2c(c1)C(=O)CCN2 CC(C(=O)N(CCCC(=O)NCC1CC1C)C)C(F)(F)F c1(OC)ncc(C(=O)Nc2cc(Cl)ccc2Cl)cc1-c1ccccc1NC(C)C C1(C)(C(N(CCOCCNC(c2c(NCC)scn2)=O)C)=O)CCOCC1 C(CC(C(=O)NCc1coc(C)n1)NC(C1CCC(C)(C)C1)=O)SC C1(NC(CN2CC(C)C2)=O)CC12CC(NC(C1CC3CC3C1)=O)C2 c1(CNCc2c(C)c(N)ccc2)c(Cl)ccc(F)c1C c1(CC(=O)N(C2CN(C(C(C)n3ccnc3)=O)C2)C)nnc(S)n1C CN=c1[nH]c(=NC(C)c2csc(C)n2)[nH]c(=NC(C)C)[nH]1 N1(C(C(=O)NC)C2(C)CC2)CCC(SC(F)(F)F)C(C)(C)C1 CC1CN(C(c2cccn2C)=O)CC(C)CN1C(=O)CCc1c(F)cccc1Cl c1(NC(CC2(C)CCN(C(C(CC)CC)=O)C2)=O)cnc(C)c(C)c1C CCCC(C(=O)NC1CC2CCC1C(NC(=O)CN(C)C(=O)C1CC1)C2)C(C)C N1(C(Cc2nc(C)sc2Cl)=O)CCC(C)CC1CNC(c1cncc(F)c1)=O C(C)(CCCCNC(c1nonc1N)=O)NC(CN(C(C(C)C)=O)C)=O c1(C(=O)NC2CC(C)(CNC(CCOC(C)C)=O)C2)[nH]c2ccc(F)cc2c1Cl C(c1ccc(Br)cc1)=CCC(N1CC2(C1)CNC2)=O N=c1nc(N2CCC(CN3CCOCC3)C2)[nH]c(N2CCCC(CC(N)=O)C2)n1 CC(CNC(=O)CCN1CCOC1=O)(CO)NC(=O)C(O)CN1CCCC1 CC(C(=O)N1CCC(F)(CNC(c2c[nH]nc2[N+](=O)[O-])=O)CC1)C(C)S(C)(=O)=O C=C1CCCN(C(=O)C(CN(C)C)NC(=O)CC2CCC(=O)N2C)C1 C1(C(=O)NCc2cn(CC(C)NC(CCCNC(C)=O)=O)nn2)CCCC(O)C1 CC1(C)CCCCC1NC(C1CC1C1CN(C(=O)CC2CCCC2)C1)=O c1(CS(N2CCCCC2C2(O)CC2)(=O)=O)ccc2ccccc2c1 c1(C(N2CCCC(CNC(C(C)C3CCC3)=O)C2)=O)cc2n(n1)CCCC2 C12(CNC(CCCc3nc(C)sc3)=O)CC(NC(=O)C=CC(C)C)(CO1)C2 c1(C(CC2CN(C(=O)OC(C)(C)C)C2)O)ccccc1F.C12CCN(C1)C2 c1(C(=O)NC2C(NC(c3cncc(OC)c3)=O)CC2)ccc(Cl)c(F)c1O c1(CC)cc(C(N2CCC(N(C(=O)CCC(C)N(C)C)C)C2)=O)c2c(c1)CCO2 CC1=NN(C)C(=O)C1CC(=O)NC(C)(C)CNC(=O)C=C1CCC(C)(C)CC1 C1(C(=O)NC2(C(=O)NC3CCCC(CC)C3)CC2(C)C)CCC(C)(O)CC1 N1(C(CCC)=O)CCC(C)C1CNC(c1cc(C2(Cl)CC2)n(C)n1)=O C1(CNC(=O)C=Cc2cccs2)C2CCC1CN(C(c1ncoc1C1CC1)=O)C2 CC(CC(C)NC(=O)CC1(N2CCOCC2)CC1)NC(=O)Cc1ccns1.C1CS1 c1(CC(=O)N(CC(NOCCOC)=O)C2CC2)csc2ccccc12 N1(C(CC2(O)CCCN(C)C2)=O)CC2=C(C1)CN(C(C1CCC=CCC1)=O)C2 S(=O)(=O)(c1cccnc1Cl)N1CC2N(C(c3c(F)cc(C)c(Br)c3)=O)C(CC2)C1 Cc1coc2ccc(C(N3CCC(CNC(C4CC(O)C4)=O)C(F)(F)C3)=O)cc12 CC1CCCC(O)(C(=O)NC2CC(C)N(C(c3cc(F)ccc3F)=O)C2)CC1 C1(C(=O)NCC(C2CN(C(C3(SC)CC3)=O)C2)O)C2CCC1C2 C1(N(C(Cn2ccc(C(=O)OC)n2)=O)C)CCCN(C(=O)Cc2csc(C)n2)C1 c1(CNC(CC2(C)CCN2C(=O)CCC(=O)C2CCCC2)=O)ncccc1F n1(CC(=O)NC(C2CCOC2)CNC(COCCC)=O)cccc(C)c1=O C(=O)(C1=CC(C)(C)C1)N1C(CNC(C(c2ccccc2)N(C)CC)=O)CCCC1 N1(C(COC)=O)C2CCCC1CN(C(c1cn(CC3CC3)nn1)=O)CC2 CC1CN(C(c2occc2C2CC2)=O)CC(CCNC(c2ccc(O)nn2)=O)O1 Cc1c(C(N2CC(F)(C(=O)N(C)CC3CCC(=O)N3)C2)=O)cnn1C C1(NC(C2CCCCS2)=O)CC1C1CCCN(c2ncc3cccnc3n2)C1 C1(C(N2C(C(=O)NCc3ccc(O)cc3F)CCC2)=O)CC2OC1C1CC21 CN1CCC(C(=O)NC23CCC(CC2)C3)(NC(c2cnn(C)c2N)=O)C1 O=C1OCc2c(CN3CC4CC4(C(N4CCCCC(O)C4)=O)C3)cccc21 N1(C(c2nc(C)n(C)c2)=O)CC(C(=O)NC2CCC3(CC2)N=N3)CC12CCC2 C1(NC(C2(C)CC2(Cl)Cl)=O)CCN(C(=O)C(c2ccc(F)cc2)=O)C12CCC2 C1(C(=O)NCc2nc(OCC)c(C)s2)CCN(C)C(=O)C1 c1(C(=O)NCC(CNC(c2cccc(C#C)c2)=O)O)cc2cc(C)ccc2[nH]1 c1(CC(N2C(CNC(C=C(COC)C)=O)C=CC2)=O)c(C)cc(O)cc1C C1(NC(c2c(C)nc(O)[nH]2)=O)CN(C(c2cncc(Cl)c2)=O)C(C)(C)C1 C(C)(C(=O)N1CC(CNC(=O)C(c2ccccc2)C)C1)(C1(C)CC1)OC c1(CC(=O)NC2(CO)CCN(C(CC(C)F)=O)C2)nc2ncccn2n1 N1(Cc2ncc(C)s2)C2CCCC1CC(O)C2.N12CCC(O)C(C)(C1)C2=O c1(C(=O)NC2(CNC(C3C(C(=O)OCC)C3)=O)CC2)ccc2nc(O)[nH]c2c1 Cc1cc(C(N2CCC(CNC(C3CC34CC4)=O)C2)=O)cc(F)c1C#N N1(C(C=C(COC)C)=O)CCC(NC(c2cc(Br)ccc2C2CC2)=O)C(C)C1 Cn1ncc(CNC(=O)CC2(C)CCC2)c1C(=O)NCCC1CCOC1(C)C c1(C(=O)NC2CCC(NC(C(C)OC)=O)CC2)cc(Cl)cc2c1CCC2 CN1CC=C(CCNC(C2CC3C=CC2N(C(=O)C(F)OC(F)(F)F)C3)=O)CC1 N1(C(CCc2cc(C)on2)=O)CC(C(=O)NCCCN2CCC2)C2(CCC2)C1 c1(C(N2C(C)CCC(NC(c3ccc(=N)[nH]c3)=O)C2)=O)ccnc2[nH]nnc12 C1(NC(C(C2CC2)OC)=O)CC2CCC1CN(C(c1c(C)cnn1C(C)C)=O)C2 c1(C(N2CCC(O)(C(C)NC(C(C)=C3CC3)=O)C2)=O)nccc2cccnc12 N1(C(C2(CC#C)CC2)=O)CC=C(C(=O)NCC(F)(F)Cl)C1 C1(NC(C2C(C)CN(C(c3nc[nH]n3)=O)C2)=O)CN(C)C(=O)C12CC2 c1(C(N2CC(NC(C3CC3(F)Cl)=O)C2)=O)ncc(F)c2ccccc12 CN=c1nc(N2CCC3(COC(C)(C)C3)C2)[nH]c(=NC(C)CF)[nH]1 CC(C)(C(F)(F)F)c1cccc(CN(C)CC2CN(C(=O)C(N)=O)C2)c1 CCC(C)CCC(=O)N1CC2CC1(c1cn(C(C)C(C)O)nn1)C2 c1(C(N2CC(O)(C(C)NC(C3CCCCC3C)=O)C2)=O)cc(Cl)c(F)cc1O CC(C(C)C(=O)N1CC(N2CCCC2)C1)NC(=O)CC1CCOC1 c1(CC)nocc1C(=O)N(CC(=O)N(CCN=[N+]=[N-])C)C1CCC1 c1(CNC2CC3CC(N)C3C2)ccc2cccnc2c1 C1(NC(C(C)OC)=O)CCC(N(C)C(C2CC23CCCOC3)=O)CC1 c1(CC(=O)NC(CN(C(C2C(F)(C(=O)OCC)C2)=O)C)C)ccc(OC)cc1Cl N1(C(CSCC#C)=O)CC2ON=C(CNC(c3cccc(F)c3C)=O)C2C1 c1(OC)cc(C(N2CCC(N(CCO)C(C3CC(C#N)C3)=O)CC2)=O)ccc1C C1(N(C(C=C(C)Cl)=O)C)CCCC2CN(C(C3CCCCCC3)=O)CC12 C(=O)(CS(=O)(=O)CCOC)NCC(CCC)NC(=O)C(C)NC(C)=O c1(C(=O)NC(=O)C(F)NC2(Cn3cccn3)CC2)ccnc(C(F)(F)F)c1F c1(C(=O)NCCC(C)NC(C(CCOC)C)=O)cn2ccc(C)cc2n1 C(=O)(C1CCc2ccc(Cl)nc21)N1CCC(OCCNC(C2(CC)CC2)=O)CC1 C1(C(N2CC(C)(COC)C2)=O)CN(C(=O)C=Cc2cnn(C)c2)C2(CCC2)C1 Cc1[nH]nc2c(C(=O)NC3CCC(N(C)C(c4cn[nH]c4)=O)C3)cccc12 C(=O)(CCS(=O)(=O)NC)N1CCCC(NC(C2N(CCC)C(=O)CC2)=O)C1 c1(SC)ccc(N)cc1C(=O)NCCCC(C)NC(=O)Cc1cscn1 c1(C(=O)NCC2CN(C(c3cc(C(C)=O)c(C)o3)=O)C2)[nH]nc2c1COC2(C)C Cc1cn2nc(C(N3CC(C4CN(C(C5CCCCC5)=O)C4)C3)=O)cc(C)c2n1 C1(C(=O)NCC(C(=O)OC)O)CCCN(C(=O)Cc2csnn2)C1 Cc1ccc2nc(C)c(CNN(C3(CO)CCC(F)(F)CC3)C)nc2c1 C1(C(=O)NCCC2CC(NC(Cc3c(CC)con3)=O)C2)CC2CCC(C1)O2 C1(=O)CC(CC2CC2)N1.C1(CN(C)C)(NC(=O)CN2CCOC2=O)CCCC1 C(C(C(=O)NC(C)CC(C)NC(=O)Cc1cc(Br)cs1)OC)OC C1(C(N(CC(C)C(F)(F)F)C)=O)CC2CCC(C1)N2C(=O)C=CC1CCCN1C Cc1[nH]c2ccccc2c1CC(N1CC(NC(=O)CC2CCCCC2C)C1)=O Cn1nc(CNC(C2CCCN2C=O)=O)c2c1CCN(c1nnc(C#N)s1)C2 c1(OC)cccc([N+](=O)[O-])c1C(N1CCC(O)C1C(=O)NC(C)(C)CC)=O N1(C(c2ccc(SC)cc2)=O)CC2CC1CN2C(C12CCC(C1)C2)=O N1(C(c2ncc(C(=O)OC)cn2)=O)CC2(CCCCN(C(C3(F)CC3)=O)C2)C1 C1(NC(C=CC(C)(C)SC)=O)CCCCCC1NC(C1CCCC12CC2)=O Cc1[nH]cc(C(=O)N(C2CCCCC2NC(=O)CC2(C)CCCC2)C)c(=O)c1Cl c1(OCC(CNc2cn(-c3ccc(OC)cc3)nn2)O)ccc2ccccc2c1 CCC(C)(C)CC(=O)N1CCCCC1CN(C)C(c1cc(CSC)c(C)s1)=O Cc1ccc(SCC(=O)NC2(C)CC(NC(C3CSCC(=O)N3)=O)C2)cc1 C1(NC(CCCC(=O)NCC)=O)CCN(C(=O)CN(S(C)(=O)=O)C)CCC1CO c1(C(=O)NCCCN(C(=O)C(O)Cc2cnc[nH]2)CC)cccc2c[nH]nc12 c1(C(N2CCCCC2CCCc2cccs2)=O)ccc(-c2cn(CO)nn2)cn1 Cc1ncc(F)c(NC(CCNC(=O)Cn2cnnc2)C(C)C)n1 C1(CNC(CC2(C=C)CCC2)=O)CC(F)CN1C(C1CN(S(=O)(=O)C(F)F)C1)=O Cc1ccc(F)c(OCC(=O)NCCCCCCNC(C2(F)CC=CCC2)=O)c1 C1(C(=O)NCCN(C(CCSCCCC)=O)CC)CCCC1c1nc(S)n[nH]1 c1(C(=O)NC2C(NC(=O)CC3CCCCO3)CCC2)cc(F)cc([N+](=O)[O-])c1 c1(C(=O)NCCNC(CNC(C2CN(C(CC=C)=O)C2)=O)=O)ccc(O)cc1F C=CC(C)(C)CC(=O)N1CC(N(C)C(c2c(Cl)cnn2C(C)C)=O)C(F)C1 N1(C(CC2OCC(C)(C)C2)=O)CC2(C(N3CC(O)(CO)C3)=O)CC1CO2 C(=O)(C1COc2ccc(Br)cc21)NCC(CNC(c1c[nH]c(=NC)o1)=O)C C1(C(=O)Sc2c(NC3CN(C(=O)C4CC4)C3)nccc2)CCCC2(C1)CC2(F)F C(=O)(C1CCCn2cc(C)nc21)NCC1C(NC(CC(C)(C)SC)=O)CCOC1 CC(CN(C)C)CC(=O)NC1CCC(NC(c2c[nH]c(=N)o2)=O)CC1 C1(NC(=NCc2cc(COC)on2)Nc2ccccc2)C2Cc3ccccc3C12 N1(CC(N2CC(NC(c3ccn(CCC)n3)=O)C(C)C2)=O)CCS(=O)(=O)CC1 CCC(CC(=O)N1CCC(NC(=O)CN(C)C)C1C1CC1)SC N1(C(=O)NCC(N2CCN(C(C=CS(C)=O)=O)CC2)=O)CCSC(C)(C)C1 Cc1cc(C)n(C(C)C(=O)NCC2(NC(c3cnc(NC4CC4)s3)=O)CC2)n1.OC Cc1c(CNC(C2CC2c2cn[nH]c2)C)cccc1Br CN=c1[nH]nc(CC(N2CC(NC(C3(C(C)=O)CC3)=O)CC2C)=O)s1 c1(C(C)NC(N2CCCC2=CCNC(C)=O)=O)ccc(F)cc1 C(=O)(C1=CC(C)(CC)C1)N(CC(CNC(C1C(C#C)C1(C)C)=O)(C)C)C CCC(CC)(C(=O)NC1C=CCN(C(=O)CC2CCC(C)(C)C2)C1)C(C)C CCCCN=C(NCCN1CCOC(C)(C)C1)NC1CCOCC1F Cc1cc(N2CCC(C)C(NC(=O)CCCC(N)=O)C2)n2nc(C)nc2n1 N1(C(C=CCN(CC=CCCCCC)C)=O)CC2(CC(NC(=O)C3=CC(C)(C)C3)C2)C1 C(=O)(CCC[N+](=O)[O-])NC(C1CCN(C(C2(C#N)C(C#N)C2Br)=O)CC1)(C)C C1(NC(COCCCC)=O)CC2CC(NC(c3nocc3Cl)=O)CC2C1 C1(N(C(CNC(=O)OCC)=O)C)CCN(C(C2(F)CCOC2)=O)C1 C(=O)(C(C)(F)C(F)(F)F)N(C1CCC(NC(c2coc(C(C)C)n2)=O)CC1)CC c1(C(=O)NC(C(C)(C)NC(C(CCSC)NC(N)=O)=O)C)ccc(S(C)(=O)=O)o1 C(=O)(CC(N)c1nccn1C)N(C1CCCC1Cn1cccn1)C c1(C(C)NC(C2N(CC)CC2)=O)ccc2c(c1)CN(C(C1C(C)(C)C1(C)C)=O)C2 c1(C(c2nnnn2C)NCc2scc(CC)n2)cccc(S(F)(F)(F)(F)F)c1 c1(OC)cc(C#N)ccc1CN1CCC1C(=O)NCc1ccccc1SC Cc1cc(C(N2CCCC(CCCCNC(C3(Cl)CC3(C)C)=O)C2)=O)oc1C C#Cc1ccc(C(=O)NCC2C=CC(NC(=O)C(F)CC3CCOC3)C2)cc1C c1(OCC)cc(C(=O)NCCN(C(=O)C(O)CC2CC2)C)ccn1.C1CCO1 N1(CC(CCC(N2C(C(C)(C)CO)CC2)=O)O)CCCCC1 C1(C(=O)NCC(CC)(CC)NC(c2cc(C)n(C3CC3)n2)=O)CC(=O)NC(=O)C1 Cc1ccc2c(C(=O)NC3CC(C)N(C(=O)C(=O)NCC4CC4)C3)csc2c1 C1(C(N2C(C)(CCC(=O)NCC(=C)Cl)CCC2)=O)CCN(C)C(=O)C1 N1(C(CC)=O)CCC(CNC(=NC)NC2CC3(CC3)C2)C(C)C1 c1(C(=O)OC)cc(NC(=O)OC(C)C)cc(C(F)(F)F)c1.N12CC(CC1=O)C2 c1(CC(=O)NCCN(C(=O)C(C)P(C)(C)=O)CC)cc(F)ccc1OC CC12CN(C(=O)CCN3CCCC3=O)C(C(N3CCCCC(CO)C3)=O)(C1)C2 CC1CCOC1CC(=O)NC1CC(CCNC(c2ccnn2C(F)F)=O)C1 C1(N(C(C(c2ccoc2)N(CCC(=O)OC)C)=O)C)CCOC(C)C1 N1(C(c2cc(OC)ccc2Br)C(=O)NC)CCCCC1C1(C)CCCO1 CCCC(C)(O)C(=O)NC(CNC(C1CC(OC(C)=O)C1)=O)CCOC C1(NC(C=C(C)Cl)=O)(CNC(c2cnc(C3CCCO3)s2)=O)CCOC1 N1(C(C(C=C)c2ccccc2)=O)CCN(C(=O)C=CCOC)C(CCOC)C1 C(=O)(C(C)(C)CS(N)(=O)=O)N1CC(C)N(C(c2coc(CO)c2)=O)CC1C N1(C(C(=Cc2n(C)ccc2)F)=O)CCN(C(C2(C)CC(C#N)C2)=O)CC1CCO c1(NC(CN(CC)CC)=O)cc(-c2ccccc2OC)cc2cc[nH]c12 CON(CCC(=O)N(CCC(C(C)C)N(C)C)C1CC1)C(=O)C(C)C1OCCO1 N1(C(CC(CC)C2CC2)=O)CC2CC(C1)C2NC(=O)CC1CCCNC(=O)C1 CC1CCN(C(=O)C(C)(C)CN(C(=O)C=Cc2ccccc2)C)CC1O C=CCC(C(=O)NCC1(NC(=O)CNC(=O)CN(C)C)CCOC1)NC(C)=O c1(C(N2CCC(C(C)(C)NC(C(CC)OCC)=O)CC2)=O)ccnc2[nH]cnc12 C(=O)(C(O)CC(F)(F)F)NCCOCCCN(C)C(c1cccc(O)n1)=O CC1(C)COCCN(C(=O)C(CC2CC2)NC(=O)Cc2cncnc2)C1 C1(C(N2CCCC(CNC(c3c(N)nccn3)=O)C2)=O)CCC2(CCCC2)CC1 C=CCC(CNC(c1csc(CO)n1)=O)C(=O)N1CC2(CCCC2)C1 c1(CCC)onc(C)c1C(=O)NCC=CCNC(c1nccn1C)=O C1(NC(C2(COC)CCCN2C(=O)C(C)(C)CN(C)C)=O)CN(CC)CC1OC c1(C(N2C3CC(CNC(=O)CC4CCC4)C2CC3)=O)cc2ccccc2o1 C12(C(=O)NC3CCC(N(C(CCC4(C)CC4)=O)C4CC4)CC3)CCC(C)(C1)OC2 N1(C(C2(OCC)CCOC2)=O)CC2CC1CN2C(=O)CCN1CCCCC1 c1(C(N2CCC(CN(C)C(=O)OC(C)(C)C)C2)=O)cc(F)c(F)c(Cl)c1F N1(C(CC(C=C)C)=O)CCCC(CNC(=O)C=CC(=O)N(C)C)CC1 c1(C(N(C2(C(=O)NCC(C)N(C)C)CC2)C)=O)ccnc(O)c1 Cn1ncc(C(N2CCC2CNC(=O)CSc2cccc(F)c2)=O)c1N N1(C(=O)OCC)CCC(c2nnnn2C2CC2)(NC(CCO)C(C)C)CC1 CC(C)(C)C(CNC(c1cc(O)ncn1)=O)NC(=O)C(F)=CC1CC1 C1(NC(C(C)SCC)=O)CCC(O)CN(C(C2CCCN2CC(C)C)=O)C1 C1(NCc2cc(O)c(Br)cc2)CCN(N2CC3CC2(CC)C3O)CC1 C1(NC(C=C(COC)C)=O)COC2(CCN(C(c3[nH]cnc3C#N)=O)C2)C1 C(=O)(CC(C)CC(=O)N1CC(O)CC1C(N1CCC(CO)C12CCC2)=O)OC Cc1nc(C2CC2)sc1C(=O)NCCC(C)NC(=O)C(C)(C)C1CCCC1 C1(NC(C(CSC)(C)C)=O)CN(C(c2ccc(=O)n(CCF)n2)=O)CC2(CC2)C1 Cn1cccc1CCC(N1CCCC1C1CCN(C(=O)Cn2ccsc2=N)C1)=O C1(NC(c2c(C)cco2)=O)CC2(CCCN(C(c3cc(C)c(C)cc3N)=O)C2)C1 C1(CNC(=O)COCCCF)CC2(CCN(C(c3cccc(Br)c3)=O)CC2)CO1 c1(NCC2(C)CCCN2)ncncc1Br.C123CC(C1)(C2)NC3=O C(c1cc(Cl)c2c(c1)OCO2)=CC(=O)N(CCC(C)NC(C=C(C)C(F)F)=O)C C1(NC(C2CCCN(C(C)C)C2)=O)CN(C(=O)COC2(C)CCC2)CCC1(C)C N1(C(c2c(OCC)ccc(C)c2)=O)CCC(N=c2nc(C#N)[nH]cc2Cl)C1 c1(CC(=O)N(c2c(C)noc2C)CC)ccc(N2CCNC(=O)C2)cc1 S(=O)(=O)(N=c1ccn(C(C)(C)C)[nH]1)NC(c1cc(-n2cc(CC)nn2)nn1C)=O C(=O)(C1Cc2ccc(F)cc21)N(C)CC1CCN(C(c2ccn(CC)n2)=O)CC1 CCC(C)C(C)C(=O)N1CC(F)CC1CC(N1CCN(CC)C(=O)C1)=O N1(CC(O)COc2ccccc2I)CC2CC(C1)C2O C1(C(F)(F)F)(C(N(CCC(C)NC(C2CCC(=O)C2)=O)C)=O)CC(C)(C)C1 C1(CCNC(=O)Nc2cncc(N(C)C)n2)CCC(F)(F)CC1 c1(-c2nc(CC)[nH]n2)cccc(C(=O)N(C)CCNC(C2CCO2)=O)c1 N1(C(CC(C)CF)=O)CC(O)(C2(CNC(=O)CCc3cnco3)CC2)C1 CS(=O)(=O)C1CC(C(N2CCC(CCCCNC(=O)C3=CCOC3)CC2)=O)C1 C=CCC(C)(C)CC(=O)N1CCC(F)(F)C(CNC(=O)C2=CC(C)CC2)C1 N1(C(C2(CCC)CC(=O)C2)=O)CC(COC)CC1CNC(=O)CC(C)C C1(N(C)C(c2cnsn2)=O)CCCN(C(c2cnc(O)c(Cl)c2)=O)CC1 C1(CNC(=O)CCSC(F)(F)F)C=CCN1C(C1CC1c1ccccn1)=O Cc1cc(C)c(C(=O)NCCC2(CNC(C3CC4CCC3O4)=O)CC2)c(S)n1 C1(C(=O)NC2CCC(NC(c3ccc(C#N)[nH]3)=O)CC2)CCn2c(O)nnc2C1 C(C(=O)NN1CC(CC2CCOCC2)C(C(F)(F)F)C1)(C(C)C)n1cc(CC)nn1 Cc1cc(CC(=O)NCC2C3CC2N(C(c2cnns2)=O)C3)c(C)s1 CS(=O)(=O)C1CCCN(C(=O)CC2COCCN2Cc2cc(Br)cc(F)c2O)C1 C1(C(N2CC(C)(CCO)C2)=O)CCCCCCN1C(C1C2CCC(F)C12)=O C#Cc1ccc(C(N2CCN(C(=O)CSCCOC)CC2COC)=O)c(C)c1 c1(C(N2C(C)CCC(NC(C)=O)C2)=O)cc(F)cc(Cl)c1O N1(C(C(CC)OC)=O)CC2CCN(C(c3cnc4c(F)cccn34)=O)C(C2)C1 c1(C(=O)NCCC2(OC)CN(C(=O)C(C)OC(C)(C)C)C2)cc2n(n1)CCCO2 C1(NC(CCN(CC)CC)=O)CCN(C(c2ccoc2)=O)CC1F C1(C(N2C(C(=O)NC34CCC(CC3)C4)CC(C)C2)=O)CCCCCCC1 N1(C(C2N(C(N)=O)CCC2)=O)CCC(CO)(NC(=O)Cn2cccn2)C1 CCC(C(=O)NC12CC(C(=O)NC3CC(OCC)C3)(C1)C2)OC c1(C(=O)NC2CCC(C(=O)Nc3c(C)[nH]nc3Cl)C2)ccc(Cl)nc1Cl N1(C(C(C)(C)C2CCOC2)=O)CCC2C(C(=O)NCC3(CO)CC=CC3)C2C1 c1(CC(N2CCOCC(NC(c3nc(C)nn3C)=O)C2)=O)c[nH]c2ncccc12 Cc1nc2c(C(=O)NCC(C)(C)NC(C3CCCNC3=O)=O)ccnc2[nH]1 N1(C(CN(C)Cc2ccccn2)=O)CC(NC2(C)CCC2)CC(O)C1.C1(=O)CO1 CC(=O)CCCC(=O)NC(C1CC=CCC1)C(=O)NCCCCN(C)C1CC1 C(=O)(C1c2ccccc2C2CC1C2)N1CCC(C)(CNC(=O)C=CCF)C1 c1(C(N2C3CN(C(C(C)N(C(C)=O)C)=O)C(C3)C2)=O)ccc2c(n1)NCCO2 c1(CC)cc(NC(C2CC(NC(C3CCC4(CCC4)C3)=O)C2(C)C)=O)cc(O)c1 N1(C(CCOCC#C)=O)CCOC2CCN(C(=O)Cn3ncc(Br)n3)CC12 Cc1nc(C(=O)NCCC2CN(C(c3cc(F)cnc3O)=O)C2)c(C)n1C C(=O)(C1=CC2CCC(C1)C2)N(CC(C)(C)CNC(C1CCCS1)=O)CC c1(C(=O)NC(CN(C(CC(=O)NCC)=O)C)C)sc(Cc2ccccn2)nc1C N1(C(CCCOCC=C)=O)CCOCCC1C(=O)NCCCC(O)CO C#CC1(C(=O)NCC(C2CCCN2C(C2CC3CCCC23)=O)(C)C)CCCC1 C(CCCC(=O)NCC1CCCN(Cc2ccc(CCBr)cc2)C1)N(C)C C1(CC(=O)NC(CNC(C(C2CCCCC2)N(C)C)=O)CO)CCCOCC1 N1(Cc2n(CC)ccn2)CC(C(=O)N(C)CC2(C)CCCC2)C(C)C1 C1(C(N(C2C(OC)COC2)C)=O)CN(C(=O)Cc2ccsc2)CC12CC2 CCCCCC(CC)C(=O)NC(C)CC(C)NC(=O)C(c1ccccc1C)C N1(C(c2c(OC)noc2C)=O)CCCN(C(=O)CC2OCCOC2(C)C)C(C)C1 CCC(C)C(=O)C(=O)NCC(C)(C)C(=O)NCC1(C)CCC1 S(=O)(=O)(c1cccc(-c2ccccn2)c1)NCC1CC(CC)C1 C1(C(N2C(CN(C)C(c3cccn3C3CC3)=O)CCCC2)=O)CC2COCC2C1 C1(CC)(CNC(=O)C(c2ccoc2)NC(=O)COc2cccs2)CCCO1 C1(=CC(=O)NC(CC)C)CCN(C(=O)Nc2cccc(SC)c2)CC1 C=CC(C)(C)CC(=O)NC(C)CCCNC(C1(n2cccn2)CCC1)=O C=C(C)c1cnccc1C(c1nnnn1C(C)C)NC(c1ccccc1OC)CF N1(C(c2c(OC)scc2)=O)CCOCC1CN(C)C(c1ccc(CO)o1)=O C1(CCCc2onc(C)n2)CCCN(C(=O)C(N2CCC(C(F)(F)F)CC2)=O)C1 c1(C(=O)NC(CC)CO)cc(C2=CCNCC2)c(C)cc1F C(=O)(C(O)CC(C)(C)C)N1CCC(N(C(c2cc(C(N)=O)c[nH]2)=O)CC)C1 N1(C(COCCCC#C)=O)CCN(C(c2ccc(F)s2)=O)C(CO)C1 N1(C(c2c(OC)c(Cl)ncc2)=O)CCC2(CCCCN(C(=O)C(O)C(C)C)C2)C1 C1(CNC(C=CCC)=O)CN(C(c2c(C)noc2C2CC2)=O)CC12CC2 c1(C(=O)NC2(CC=C)CN(C(c3c(SC)cccc3F)=O)C2)c[nH]cc(C)c1=O Cc1cc(C(=O)NCC2(C(C)(C)C)CCN(C(C3(O)CCCC3)=O)C2)ncn1 c1(C(N(C2CCCN(C(C3(OC)CC3)=O)C2)CCF)=O)ccc2c(c1)OCCC2 N1(C(=O)NC2(CO)CC2)CCc2ccccc2C(NC(=O)C=C2CCC2)C1.CO N1(C(c2ccc(C)nc2O)=O)CCn2c(C(N3CCCC(CO)C3)=O)cnc2C1 N1(C(CCc2c(C)ncs2)=O)CCC2C(CCCN2C(c2ccc(O)nn2)=O)C1 Cc1c(C(NC2CCc3c(Cl)ccc(Br)c32)=O)oc(S(N)(=O)=O)c1C C1(C(=O)NCC(CCNC(C(C)(Cl)Cl)=O)O)CC2(C1)CC1(CC1)C2 c1(-n2cc(CONC(c3cc(C)[nH]c3)=O)nn2)cccc2c1CCCC2 Cn1ncc(S(=O)(=O)N(C)C)c1CNCC(C)(C)NC(=O)OC(C)(C)C c1(CC)cc(C)ccc1NC(=O)C(C(C)O)NC(C1CCC(F)(F)C1)=O C#CC12CCC(C(=O)NC3CN(C(=O)CN4C(=O)Cc5ccccc54)C3)(CC1)CC2 C(=O)(CCC(C)CC(=O)OC)N(CCN(C(CCN(CC)CC)=O)C)C C1(n2c(=O)c2=O)CCc2ccccc2C1.c1(OC)cc(C)nn1CC(F)(F)F c1(C(=O)NC(CC(C)NC(c2c(C)nc(C)[nH]2)=O)C)cnn2c1CCCN2 N1(C(C(C)=CC)=O)CC2CC1CCN2C(C1(CO)CCCCC1)=O.C(=O)(C(C)C)N N1(C(c2c(CC)noc2)=O)CC2CC(C1)CN(C(=O)Cc1ccc(C#N)cc1)C2 C(CC(C)C)(C(=O)NCCNC(C)=O)N(C(C1(OC)CCOC1)=O)C c1(NC(COC)=O)ccc(Nc2cc(C#N)ncn2)c(F)c1 n1(CCC)nc(C)cc1C(=O)N(CCNC(C1CCCN1CC)=O)C(C)C C1(C(=O)NCC(c2ccccc2F)(C)C)CC2CCC1N(CCn1cnnc1)C2 c1(N(CCC(C)O)C)nc(N2CCCC(F)(F)CC2)nc2c1ncn2C c1(OC)ccc2c(C(N3CCC(NC(C4CCC4(C)C)=O)C(C)C3)=O)coc2c1 N1(C(C=CSC)=O)CCC2CCN(C(c3cnc(CCC(F)(F)F)s3)=O)C2C1 Cn1cc(C(=O)NCC2(CNC(=O)CCC3(C#N)CCC3)CC2)n(C)c1=O c1(C(=O)NC2C(CNC(CCC=C=C)=O)CCCC2)ccc2nc(O)oc2c1 C1(NCC(O)CC2CCC2)CCCCC1c1ccccc1 C1(C(C(=O)NC2(CC#C)CC2)C)CCN(C(c2csnn2)=O)C1 c1(C(=O)OC)ccc(C(=O)OC2CCC2C2CC2)cc1F c1(C(N(CC)CC2CCN(C(c3cc(Cl)c[nH]3)=O)CC2)=O)cnn2ccncc12 c1(C(=O)NCCCCC(C)NC(C(CCCC)O)=O)cc(O)c2[nH]c(C)nc2c1 n1(CC)cc(C(=O)NCC(C2CCCC2)NC(=O)CC(C)(F)F)c(C)n1 c1(CC(=O)O)cn(CCCC2CCN2C(=O)COc2ccsc2)nn1 c1(C(N(C)CC2CCCN(C(CCC#C)=O)C2)=O)cc2ccoc2cc1F C1(C(=O)NCC(CNC(C(C=C)(C)C)=O)O)CCN(C2CC2)S1(=O)=O c1(C(CC(=O)NCCN(C(=O)C=CC2CCC2)C(C)C)O)cccc(F)c1 C1(C(=O)NC2C(CNC(c3conc3C3CC3)=O)C2)CCSCC1 C1(NC(c2nn(CC)c(C3CC3)c2)=O)CC2(C1)CC(NC(=O)CC1CC1)C2 C(C(C)(O)C(=O)NCCN(C(C1(C(N)=O)CC1)=O)Cc1cccc(Cl)c1)OC CCC(CC(=O)NCC12CC(C1)C(NC(c1ncn(C)c1C)=O)CO2)C(C)(C)C C(c1cccc(Cl)c1)=C(C)C(N1CCC(NCc2ncccc2C)C(F)C1)=O c1(CNC2C3CN(C(C(C)n4cccc4)=O)CC32)cccc2ccccc12 C1(CNC(C2C(C)CCCC2)=O)CCN(C(=O)CCC2CC2(C)C)CCC1(F)F CCCC(O)CC(=O)N1CCN(C(=O)CCOC2CCC2)CC1c1ccnn1C C=CCC(CC)N=c1[nH]c2c(c(=NCC3(CC(C)C)CCC3)[nH]1)COC2 C1(CNC(=O)CN2CCCCC2)CC2(CO1)CN(C(C1CC(=C3CC3)C1)=O)C2 C1(CC=C)(NC(=O)C=CI)CC2CCC(C1)N2c1cncc(Cl)n1 C1(CNC(C(C)CSC(F)(F)F)=O)COCCN(C(C23CCC(C)(CO2)C3)=O)C1 C1(OC(=O)CCc2nc(-c3ccncc3)no2)CCC(F)(F)c2ccccc2C1 CCC(C)CCCCC(=O)NC1(CNC(c2cnn3ccccc23)=O)CCCC1 C1(N(C)C)CCN(CC(N2CC3CC3(CNC(=O)CC3CCCCC3)C2)=O)CC1 c1(C(=O)NC(C)CCN(C)C(c2coc(Cl)n2)=O)ccc(F)c(Cl)c1 C1(CNC(c2cc(C3CC3)on2)=O)CC2(CO1)CN(C(c1n[nH]cc1Cl)=O)C2 N1(C(c2ccn(C)c(=O)c2)=O)CC2(C1)CN(C(c1nc(Cl)sc1Cl)=O)CC2CO c1(NC(N(C)Cc2ccc(NS(C)(=O)=O)cc2)=O)ccc(S(=O)(=O)F)s1 c1(CC)ccc(C(=O)NC2CCCC2CNC(=O)CCCNC(=O)C(C)(C)C)[nH]1 C1(N(c2ccon2)C(CC2(C)CCC2)=O)CCC2(CCN(C(=O)CN(C)C3CC3)C2)C1 C(C1CCC(C)(C)c2ccccc21)NC(c1cc(NC(CCC)=O)ncc1)=O C(=O)(C1=NNC(=O)CC1)NCCC1N(C(CCN(C(CC)CC)C)=O)CCCC1 C1(CNC(=O)NCC2CCC=CCCC2)OCC2CCCC12 CC(C)(C)C(CNC(C1(CO)CCOC1)=O)C(=O)NCC(F)(F)Cl C1(NC(=O)NCC(=O)NCCCN(C(c2ccoc2)=O)CC)CCCCC1 N1(C(c2cnnc(O)c2)=O)CCN(C(C2(CO)CC2)=O)CC(O)C1 N1(C(C(C)Cc2cnc[nH]2)=O)CCCCC1CNC(=O)C=CC=C(Cl)Cl C(CNC(C1CN(C2COC2)C1)=O)(CC(=O)NCCC1CCCC(C)C1)OC c1(C(N(C)Cc2cccc(CNC(C3(C4CC4)CC3)=O)c2)=O)cc(O)ccc1F C(=O)(CC(O)Cc1ccccc1)NC1C(CNC(CSCC(C)C)=O)CC1 c1(C(N2CCC(CNC(c3c(=N)cc[nH]c3)=O)C2)=O)cc(O)ccc1Br C1(C)(CNC(C(C)N2CCC2)=O)CCN(C(c2cncc(N)c2)=O)C1 C1(C(=O)NCCC2C(C)(C)CCO2)CCC(C)(C)N(C(=O)CN2CCOC2=O)C1 C1(CCC=C)(C(=O)NC(C(F)(F)F)C2CC2)CN(C(=O)C(Cl)Cl)C1 N1(C(c2c(C)oc(CO)c2)=O)C(CNC(C2(C(C)C)COC2)=O)CC2COCC12 C1(O)(CNC(C2CC23CC3)=O)CC2CCC(C1)N2C(c1cccc(C2CC2)n1)=O c1(C(C(=O)N(CCC)CCNC(C2CN(C)CC2C)=O)(F)F)ccc(F)c(F)c1 n1(CC(=O)N(C2CCN(c3ccnc(Cl)n3)CC2)CC#C)nc(C)c(Cl)c1C C1(CNC(c2c(C)scn2)=O)CN(C(=O)CCc2ccccc2)CC1C CC1(C=CC(N2CCCOC(CNC(C3CC(F)C3)=O)C2)=O)CCOCC1 N1(C(c2ccccc2)=O)CCN(C(C2CC3(C2)CC3(F)F)=O)C(CCO)C1 c1(C(=O)NC2CC(C)(CNC(CCc3cc(C)on3)=O)C2)cnn2c1OCCC2 CC(C)C(CC(=O)N1CC(O)(CN(C)C(c2cc(Br)ccn2)=O)C1)C(C)C O=C1OCc2ccc(C(=O)NC3CC4CC3N(C(=O)CCC(F)(F)F)C4)cc21 c1(OC)c(C(=O)NCCNC(c2ccc(C(C)=O)o2)=O)nc(O)nc1O N1(C(CN(C2CCC2)C)=O)CCC(O)(C(C)CNC(=O)Cc2ncc(Cl)s2)C1 C1(C(C)(F)F)(C(=O)NC2CCN(C(c3ccns3)=O)C2C2CC2)CCOCC1 Cc1sc(C(F)(F)F)nc1C(N1CCC(C)(CNC(C2CC(O)C2)=O)C1)=O N1(C(COCCCOC)=O)CC(NC(c2cc(C(F)(F)F)cn2C)=O)CCC1C N1(C(=O)CC2CCCOCC2)CC2CCC(C1)N2C(c1csc(Cl)c1Cl)=O c1(NC(CCCNC(CN(CC)CC)=O)=O)cc(N2CCCC2)ncn1 C12(C(N3CC(C(C)NC(=O)C(C)S(N)(=O)=O)C3)=O)CCC(C1)C2(C)C C1(COC(C(C)NC(CSC)C)=O)CCN(Cc2ccccc2)CC1 CC1CCN(C(C2C=CCCC2)=O)CC1CC(=O)N(C)CC1CCOC1C C(=O)(C(F)CC(C)(C)C)NCC1CN(C(C(C)(C2CC2)OC)=O)C1 CC1(C)CN(C(c2ncc(N)cc2Cl)=O)CC1NC(=O)Cc1ccnc(O)c1 N1(C(Cc2n(CC)ncc2)=O)CCC(C(C)C)CC1.C12CC1C2 c1(OC)cc(C(N2CCN(C(C3(F)CC3)=O)C(C(C)C)C2)=O)ccc1Br C1(C(F)(F)F)(C(=O)NC(C)CCCNC(=O)CCC2CCCO2)CCCCC1 N1(C(C(C)CF)=O)CCC(O)(CNC(=O)CC=Cc2ccc(Br)cc2)CC1 N1(C(c2cncc(C#C)c2)=O)CCC(C2(NC(=O)CNS(=O)(=O)N(C)C)CC2)C1 C(=O)(CS(=O)(=O)C(C)(C)C)NC12CC(NC(C3CC(C)OC3C)=O)(C1)C2 C#Cc1cnn(C)c1C(=O)NC(C)CC1CCN(C(C2(C#N)CC(C)C2)=O)CC1 c1(C(N2CC(NC(c3c(CC)nc(C)[nH]3)=O)C3(C2)CC3)=O)cc2n(n1)CCCN2 C(CS(=O)(=O)CC(=O)N1CCCC(c2cn(C(C3COCCC3O)=O)nn2)C1)OCOC C#Cc1cnc(C(=O)NCc2ccccc2CNC(=O)C2=CS(=O)CCC2)c(C)c1 C=C(C)CN=C(NCC1CC(C)CO1)NC1CN(C(=O)OC(C)(C)C)C1 n1(CC)nccc1C(=O)NC(Cc1cn[nH]c1)C(=O)NCC1CC1c1ccoc1 N1(CCC2(CS(C)(=O)=O)CC2)CCC(OCC2CNC2)CC1 c1(OC)n[nH]c(C(N2CCCC2CN(C(=O)CC2CC(C)(C)C2)C)=O)c1Cl C12(CNC(c3c(C)cno3)=O)CCC(CN(C(C3CC(=O)OC3(C)C)=O)C1)C2 N1(C(CC=CCC)=O)CC2CCN(C(=O)Cc3ccc(Cl)c(OC)c3)CC2C1 C12(C(=O)NC3C4CN(C(c5csc(C6CC6)n5)=O)C3C4)CCCN1CCC2 CC1CCC(C)(C)CN1C(C1CC2CCC(C1)N2C(=O)C1=C(Cl)CCC1)=O c1(NC(c2ccc(C(C)C(F)(F)F)cc2)=O)ccccc1S(N)(=O)=O N1(C(CSc2c(C)cccc2C)=O)CCCC2(C1)CN(C(=O)C(C)C#N)CCO2 O=C1COC2(CN1)CN(C(c1ccc(=O)n(Cc3ccc(Cl)cc3)n1)=O)C2 C1(NC(=O)CC2CCC3(CC2)CC3)CN(C(=O)C2=CCCOC2)CC2(CCC2)C1 c1(CC(=O)NC2CCC(NC(C(c3ccccc3)OC)=O)C2)cncc(Br)c1 c1(C(N(CCN(C(C(C=C)(C)C)=O)C)C)=O)ccc(F)cc1NCC=C(C)C N1(C(CCCOCC)=O)CCC(O)(CNC(=O)CCCc2ncc(C(C)C)o2)C1 c1(C(=O)NCC2C3CN(C(CCCC(C)C)=O)CC32)cc2c([nH]1)CCC(C)C2 N1(C(c2c(C)nco2)=O)CCCC2CN(C(=O)CS(=O)(=O)NC(C)(C)C)CCC12 N1(C(Cc2ccc(C#N)cc2)=O)CC2(C1)SCCC2NC(=O)Cc1cnns1 c1(C(=O)NC2C(CNC(C)=O)C2)cc(Cl)c(F)c(Cl)c1 N1(C(c2cc(CC)sn2)=O)CCCCC1C(C)N(C)C.c12ccc(o1)CNC2=O C1(CNC(C(C)OCCOCC)=O)CCN(C(=O)C(C)(C)C2CCOC2)CC1 C1(NC(CCOc2c(C(N)=O)cccc2)=O)CC2CC1N(C(C1CC1Br)=O)C2 N1(CC)CC(C(=O)NC2CCCCC2NC(c2ccc(O)cc2Cl)=O)CCC1=O N1(C(c2c(CC)nc(C)nc2)=O)CC2CCC(C1)N2C(=O)CCc1nccs1 Cc1nnccc1C(=O)NCCCOCCC(=O)NCc1cnnn1C c1(C(N2C(COC(C(=O)OC)C3CCC3)CCC2)=O)cncc(CNC(C)=O)c1 c1(C(N(C2CCN(C(C3(C(F)F)CC(F)(F)C3)=O)C2)C)=O)occ2c1CCC2 Cc1c(Cl)cnn1CC(=O)NC1CCC(CNC(=O)C=CCN2CCCCC2)C1 c1(C(=O)NCC2OCCCN(C(C(C)O)=O)C2)cccc2c1OCCO2 C1(C(=O)Nc2cc(OC)c(C)cc2)CCC2CCC1N2C(=O)CC1CC(F)(F)C1 N1(CC)C(=O)CCC1C(=O)NCCOCCCNC(=O)CCc1c(C)n[nH]c1C c1(C(=O)NCC(C2CC2)NC(c2n(CC)ccn2)=O)ccnc(-c2ccco2)c1 C1(CNC(C(CN(C)C)O)=O)CC2(CCN(C(=O)C(C3CC3)C3CC3)CC2)C1 Cc1ccc(=O)n(CC(=O)NCCC2(NC(c3ccoc3)=O)CC2)n1 C1(CC(C)NC(CSCC(=O)OC)=O)CCN(C(c2cn(C3CC3)nn2)=O)CC1 C1(NC(C2(OC)CC2)=O)CC12CC(NC(=O)CC1CNC(=O)C1)C2 CC(C)CCC=CC(N1CC(O)(C(F)C(=O)NCCCn2ccnn2)C1)=O C1(NC(c2ccn(C(C)(C)C)n2)=O)CCCC(NC(c2cncc(Cl)c2)=O)CC1 c1(C(C2CC=CCC2)OC)cn(CC(=O)NCc2nc(C(F)(F)F)n[nH]2)nn1 C1(CC(=O)N(c2cc[nH]n2)C)CCN(C(=O)COCC2CC2)C1(C)C C1(C(=O)NC(C(=O)NCCC2(C)CC2)C2CCC2)CCOCC1 N1(C(C(C#N)=CC2CC2)=O)CC2C(CNC(=O)Cc3cccc(Cl)c3)C2C1 Cc1cccc(COC(C)C(N2CCC(N(C(=O)CSC3CC3)C)CC2)=O)c1 C1(C(N(CC(C)NC(c2cc(C(C)=O)c(C)o2)=O)C)=O)CCc2nc(O)[nH]c2C1 c1(C(=O)NCc2c(C(N(C3CCC(F)(F)C3)C)=O)n[nH]c2)cc(C#N)ccc1N c1(N2CCCC(C)(CNC(=O)CCCN3CCOCC3)C2)ncnn2cccc12 C(C(=O)NCc1ccc(C)c(F)c1)(C(C)CC)N(C(C(CCC)F)=O)C C(=O)(C1(C)COc2ccccc21)N1CCC(NC(C2C(C(C)(C)C)C2)=O)CC1 N1(C(c2cnn(CC)c2C)=O)CCC2CCN(C(C3(F)CCS(=O)(=O)C3)=O)CC12 C12(C(N(C)CC3C(C)OCC3)=O)COCC1CN(C(C1CCCC13CCC3)=O)C2 c1(OC(CC)C)ccc(C(=O)NCC(O)CNC(c2cocn2)=O)cc1 N1(C(c2cc(OCC)no2)=O)CCC(NC(C2(N(C)C)CC2)=O)CC1 c1(C(N2CC(C)(NC(C3(C(=O)OC)CC3)=O)C2)=O)cn2cccc(Br)c2n1 C1(CC(=O)NC2(CC)CN(C(=O)CC3CCCCC3)C2)CCCCC1O C1(NC(CN(C2CCC2)C)=O)CC1C1CCCN(C(C2CCCO2)=O)C1 C1(C(N(C)Cc2c(C)noc2C)=O)CCN(C(=O)CCC2CC2(F)F)C12CC2 N1(C(C2C=CC(NC(=O)C(C3CCCCC3)O)C2)=O)CCC12CCC(O)CC2 CCCC(CCC)C(=O)N1CCCC(CN(C)C(C2CCCS2)=O)C1 c1(C(N2C3(CN(C(c4c(C)nsc4)=O)C3)CC2)=O)ccc2c(c1)NC(=O)CN2C C(=O)(C(C)(C)C#N)NC1C(NC(c2cc(OC)no2)=O)CC1 Cc1nc(C(N2CCCC2CC2CCC2)C(=O)NCc2ccco2)nn1C c1(C(N)=O)c(-c2cccc(OC(F)F)c2F)ccnc1O C1(NC(CC(C)CN(C)C)=O)CC2(CCN(C(C3(C#N)CC34CCC4)=O)CC2)C1 CCC(C)(C)C(O)C(=O)NC1CCN(C(=O)CCC2CC2(Cl)Cl)CC1(C)C C1(C(=O)N)Cc2nccn2C1.N1(C(C)=O)CC(O)CC1C(=O)NC1CC(CO)C(O)C1 CC(C)CC(CNC(c1cncc(C(C)(F)F)c1)=O)NC(C1CCCO1)=O c1(CC(=O)NC2CCN(C(c3cc(CCC)n(C)n3)=O)C2C)cc(C)ccc1C C(=O)(CC(C(F)(F)F)c1c(Cl)cccc1Cl)NCCCCNC(C(CC)O)=O Cc1ccc(C(CO)NC(=O)NCc2ccccc2N2CCCCC2)c(F)c1F N1(C(c2c(C)ncnc2O)=O)CCC2(C1)CN(C(=O)CC1(O)CCCCC1)C2 C1(CN(C(CC(=O)NCC)=O)C)CCCCN1C(C1OC(C)CC1C)=O c1(CC(=O)NCC(C)N(C(CCC(=O)NC)=O)C)ccccc1S(C)=O N1(C(c2cncc(OC)c2)=O)CC2CCC1C(NC(=O)CCCC(=O)N(C)C)C2 C(CCCCCNC(c1cc[n+]([O-])cc1)=O)N(C(=O)CCCCNC(N)=O)C C12(C(=O)NC(C)CCNC(C3(C)CCCOC3)=O)C3C4C1C1C2C3C41C(N)=O c1(C(C)=O)ccc2nc(N3CC(O)(C(C)NC(C4CC4(C)Br)=O)C3)sc2c1 Cc1cc(C(=O)Nc2cnc(F)cc2C(=O)Nc2cncs2)ncc1CO C(C)(CCC(F)(F)F)(c1nnnn1CCC1CC1)NC(c1cncn1C1CC1)C C(=O)(C(C)(CC)C(=O)NC(C)CCCCNC(c1ccc(F)c(C)c1)=O)OCC C12(CCNC(c3cn4ccnc4s3)=O)CCC(C1)N(C(=O)C1=COCCC1)C2 C(=O)(C(C)(C)C(=O)NCC(CNC(C1(Cc2ccccc2F)CC1)=O)CO)OC N1(C(C(C)N(C(C(CC)C(=O)OC)=O)CC)=O)CCC2(CCSC2)C1 C(=O)(CCC(C)(C)C)OCC.C1(=O)NNC(=O)NC2COCC12 C(C)(C)(CCCC(=O)NC1CCC(O)C(O)C1)NC(c1ccc(C#C)o1)=O C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CC(C)N(C(c2cnn[nH]2)=O)CCC1 C1(n2cccn2)(C(=O)NCCNC(CC(C)C2CC2)=O)CCOCC1 CC1CN(c2c(Cl)cccc2Cl)Cc2ccccc2O1.C(F)(F)F C12(C(N(OC)CCO)=O)CCC(CC1)N(C(c1c(C)nsc1C)=O)C2 c1(C(C)=O)ccc(C(=O)NCC(C)(C)NC(=O)CC=CCc2ccccc2)nc1 C1(C(=O)NC2COCC2O)C2CCC(CC2(F)F)N1C(=O)Cn1nccn1 Cc1c(C(=O)NCCNC(C2CCCC23CCOCC3)=O)sc2ccc(F)cc12 C1(C)(NC(C(COC)OC)=O)CCCN(C(c2ccc(C(C)(C)C)o2)=O)C1 N1(C(c2ncn(CC)c2)=O)CCCC(F)(CNC(=O)CC2CCCC23CC3)C1 CCCC(C(O)C(=O)N1CCOCC1C)NC(=O)CC1CCC(C)CC1 N1(C(c2ccc(COC)[nH]2)=O)CCC(CCNC(=O)CN2CCSCC2)CC1 C1(CNC(C2CC(n3cc(CO)nn3)C2)=O)CCCCS1 CCC(C)(C)C(=O)N1CC(N2CC(NC(=O)CNS(=O)(=O)C3CC3)CC2=O)C1 C1(CCNC(COCCCCCC)=O)CCN(C(=O)C=CCF)CC1 C1(C(N2C(CNC(C(C)=C3CCCC3)=O)CCCC2)=O)CC2CC(O)C(C1)C2 CC(C)(C)CC(=O)NCC(CO)NC(=O)CC1CCSCC1 c1(C(N2CC3C(CNC(c4cncc(O)c4)=O)(C3)C2)=O)nc2ncccn2n1 C1(NC(C(C)OC)=O)CC2CC1CC2C(=O)NCc1ncoc1C.C(C)(C)(C)O Cc1nc(C(F)(F)F)ccc1C(=O)NC1CCC(NC(=O)CC2CC(F)C2)CC1 N1(C(C(CC=CC)C)=O)CC2(C(N3CC(CO)C4(CC4)C3)=O)CCC1CC2 C12(NC(CC=CC=C)=O)CCCC1CN(C(c1sc(Br)nc1C)=O)C2 C1(NC(C(CC(C)C)O)=O)CN(C(=O)CCc2ccc(Cl)nc2)CCC1(C)C C(=O)(C(C)CC(C)(F)F)NCC1CCN(C(c2cc(C)cc(N)c2)=O)CC1 c1(CNC(C(C)C2CC2)=O)ccc(CNC(C2CC2C)=O)c(F)c1 c1(C(=O)NCC23OCC(NC(C4(CC=C)CC4)=O)(C2)C3)nc2ncccn2n1 N1(C(C(C)C(F)F)=O)CCCN(C(C2CN(C3CCOC3)C2)=O)CCC1 N1(C(C(CNC(c2cc(C#C)c(C)cc2)=O)CC2CC2)=O)CCCC2CN(C)CC12 N1(Cc2c(C(=O)O)ocn2)CC(CC2COCC(=O)N2)c2ccccc21 Cc1ccc([N+](=O)[O-])c(C)c1C(=O)NCC1CCCC1NC(=O)Cc1nccs1 c1(CC(CNC(c2cn(-c3ccc(F)c(F)c3)nn2)=O)C(=O)O)cc(Cl)cc(Cl)c1 N1(C(C2C(CCC)CCC2)=O)CCN(C(=O)CC(Cl)Cl)C2(CC2)C1 Cc1ccc(-n2cnnc2)c(C(=O)NCC2CCN2C(c2cccnc2C)=O)c1 c1(C(N2CCC(N(C(=O)C(C)SC)CCC)C2)=O)ccc(SC)cc1OC C12(CNC(CC(C)c3ccco3)=O)CCCCC1N(C(c1cc(Br)co1)=O)CC2 c1(C(=O)NC2CN(C(c3ccn(C(C)C)n3)=O)C(C)CC2)cccc2nccn12 N1(C(C(CCC)NC(=O)CN(C)CCOC)=O)CC(C)OC(C)(C)C1C c1(CC)cccc(CNCC2(CCCO)CCCC2)c1F c1(C(C)C)ccc(NC(=O)CN2CCN(C(=O)C(C)CN(C)C3CC3)CC2)cc1O CCCCCCC(C)SCc1ncccn1 c1(C(=O)NC(C)CC2CN(C(=O)CS(=O)(=O)N(C)C)C2)c[nH]c2cccnc12 CC1CC(C)CCN(C(c2coc(CNC(C34CCC(CC3)CC4)=O)n2)=O)C1 C1(NC(CCc2n(C)cnn2)=O)CS(=O)(=O)CC1NC(c1ccc(N)cc1F)=O n1(CC)ccnc1C(=O)NCC1CCC1NC(=O)C(C)COC c1(C(c2n(CC)nnn2)NCC(c2ccc(F)cc2Cl)(C)C)cc(Cl)ccc1Br N1(C(CC(C)=C(C)C)=O)CCCC12CCN(C(=O)Cc1cccc(C(F)F)c1)C2 Cc1ccc2[nH]c3c(c2c1)CN(C(=O)C(=O)Nc1cccc(F)c1)CC3 CCS(=O)CC(=O)NCCCC(C)NC(c1nccc(N2CCCCC2)n1)=O Cc1c(C(N2CCc3ccccc3C2)=O)[nH]c2c1CCCC2 c1(OCC)nc(Cl)ccc1C(N1CC(NC(=O)COC(C)=O)CC(C)C1)=O N1(CC(C)(C)C2CC2)C(=O)CC(COCC2CC2)C1=O N1(c2cc(C)ncc2C#N)Cc2nccn2CC(NC(c2c(Cl)cnn2C)=O)C1 c1(C(C)C(N2CCCC(C(N3CCC4CC34)=O)C2C)=O)ccc(F)cc1F c1(C(=O)NCC2OCCN(C(C3CC4(CC(=O)C4)C3)=O)C2)cccc2cc[nH]c12 C1(F)(CNC(c2ccc(NC)nc2)=O)COCCN(C(=O)CN(C)C2CC2)C1 c1(N(C(=O)N)C)cccc(-n2ccnc2)c1.c1(CC(c2cncnc2)C)ccccc1 c1(C(=O)NC2C(C#N)CN(c3ccnc4ccnn34)C2)ccc2ccnn2c1 N1(C(C(CC)SC)=O)CC23CCCC2(C1)CN(C(=O)CC1CC=CC1)C3 C1(NC(c2cc(C(F)(F)F)no2)=O)C2CCN(C(c3ccsc3)=O)CCC12 N1(C(CN(C)C(c2cscn2)=O)=O)CC2CC2(CNc2ccnc(Br)c2)C1 C1(C(=O)NC2CC(CCC(=O)NC(CC#C)C)C2)(CC)CCC(=O)N1 CC1CCN(C(c2cc(CCNC(=O)CC3C=CCC3)on2)=O)CC1O N1(C(=O)CC2CN(C(c3ccc[n+]([O-])c3)=O)CCO2)CCCC12CCOCC2 OC1CCCCC1Cc1cc(NC2CCC(C3CC3)C2)ncn1 N1(C(c2nccc(C#C)c2)=O)CCC2(CC1)CC(C)N(C(=O)C(O)C1CC1)C2 C1(OC)CCN(C(=O)C=Cc2ccc(Cl)s2)CC1c1cn(C2CCOC2)nn1 c1(OC)cc(CCC(=O)NCCCCNC(C2(n3cnnn3)CC2)=O)ccc1Cl N1(C(CS(N)(=O)=O)=O)CCC2(NC(C3COC4(CCC4)C3)=O)CC2C1 N1(C(C2C(C)C2)=O)CCC1(C)CNCc1ncc(Br)s1 C(C(=O)N1CC(C)(O)CO1)(c1cccnc1)NC(C(C)OCCOC)=O Cc1ccc(F)c(C(C(=O)O)N(C(=O)CCF)C)c1 C1(SCC)CCC(c2cn(CC3CC4CC4C3)nn2)CC1.C1(C(=O)OC)CN(C)CCO1 N1(C(C(C(C)C)OC)=O)CCC2(CC1)CC2C(=O)NCc1cnn(C)c1 N1(C(C2CC(C(=O)OC)C2)=O)CCCN(C(C2CCCC2OC)=O)CC1 O=C1NC(=O)C2(CCCC2C(OCPc2ccc(Oc3ccccc3)cc2)=O)N1 CC1(C)C(NC(C2CCCC2O)=O)CC1CC(=O)NC1(CC2CCC2)CC1 Cc1cc(C)c(C(N2CCC2CNC(c2nc(C3CC3)cs2)=O)=O)c(=O)o1 C1(C2CC2)(CC(=O)NCC(CNC(c2cc[nH]n2)=O)OC)CC1 N1(C(c2cncc(-c3cccc(C)c3)c2)=O)CC2CN(c3ccccc3)CC2C1 C=CCC(CNC(C1CC1(C)C)=O)C(=O)NCC1CN(C(C)C)C1 c1(C(=O)NC2C(NC(C3CCC(=C)CC3)=O)CCCC2)cc(C(C)C)ccc1O C12(CNC(CCCC#CC)=O)CN(C(C34CC(C)C3C4)=O)CC1CCO2 C12(CNC(Cn3cc(CNC(c4[nH]cc(C)c4)=O)nn3)=O)CC(CCO1)C2 N#CCCCCCC(=O)NCC1CC1C(=O)NCCN1CCCC1=O C12(C(=O)OC)CNCCC1CN(Cc1sc3ncccc3c1Cl)C2 c1(OC)c(C(N2CC3CC2C3C(=O)NC2CC3(C2)CC3(F)F)=O)nc(O)nc1O O=C1c2ccsc2CCC1CC(=O)Nc1cc([N+](=O)[O-])ccc1O c1(C(=O)NCC(CC2CN(C(CC(C=C)C)=O)C2)(C)C)nnc(Cl)cc1N N1(C(C(COC)CNC(C(CC)NC(C)=O)=O)=O)CC2CC1CC2CF C1(C(N2C(CC(=O)NC)CC2)=O)CCCN1NC(=O)COc1ccc(F)cn1 C=CCCCC(=O)NC1CCCC(c2cn(CC3CCCO3)nn2)C1 N1(C(C2=C(C)OCCC2)=O)CC2CCC1C1CN(C(=O)C=Cc3ccco3)CC21 C1(OC)CC2(C(=O)NCCC(O)CNC(C3CC(C(=O)NC4CC4)C3)=O)CC12 CC(C)(C#CC(=O)N1CC(C#N)(CCF)C1)CNC(=O)CCc1nccs1 N1(C(CCOCC(C)C)=O)CCC(NC(=O)CCn2ccccc2=O)CC1C1CC1 N1(C(C2C(OC3CC4CC(C(=O)NC)CC43)C2)=O)CCC(CC)(CO)CC1.C1CC1 c1(C2C(C(=O)NCc3c(C)scc3)C2)ccc(F)cc1.C1(CCN)CCCN1CC Cn1c(C(=O)NCCNC(C23COCC2CS(=O)(=O)C3)=O)c2n(c1=O)CCCC2 C1(NC(c2c(CC(C)(C)C)c[nH]c2)=O)CN(C(=O)CNC(=O)C2CC2)CC1F N1(C(CCSCC)=O)CCCC2(CCCN2C(C2CCC(C)CC2)=O)C1 Cc1c(Br)ccc(C(=O)NCC2CCC3COCC3O2)c1C c1(C(=O)On2cc(C3CCN(C(=O)C(F)(Cl)c4ccccc4)C3)nn2)ccc(CC)cc1O c1(C(N2CCC(NC(Cc3cc(C)no3)=O)C2C)=O)ccc2c(c1)CCC(O)C2 c1(CN(C)C(c2cc3ncsc3[nH]2)=O)ccccc1[N+](=O)[O-] c1(CN2C(C(=O)NCc3ccc(OC)c(Br)c3)CC(O)C2)cc(I)cc(I)c1O C(CCCCn1cc(CCO)nn1)NC(CCOCC(C)C)=O Cc1c(Cl)ccc(C(=O)NCC2CCC(NC(=O)Cc3cnco3)C2)c1N C1(CNC(Cc2cnc(C)o2)=O)C2CCCC1N(C(C1(C)CCN(C)C1=O)=O)C2 n1(CC(N2CCC(NC(C(C=C)(C)CC)=O)C2C)=O)c(=O)n(C)c2ccccc12 C(=O)(CCCCC(C)(C)C)NC1COCCN(C(C(C(CC)CC)F)=O)C1 Nc1cc(F)cc(C(=O)NC2CC(NC(C3CCCC(C(F)(F)F)C3)=O)C2)c1F C(=O)(C(O)CCNC(C1(CO)CCCO1)=O)NCCNC(COC)=O CC1CCC=C1C(=O)NCC1C2CN(C(c3ccc(C(F)F)o3)=O)CC12 C(=O)(CC1OCc2ncccc21)NCC(CC)NC(=O)CSc1ccccc1O Cc1nn(C)c(Cl)c1C(=O)NC1CCC(F)(CNC(c2ccn(CCF)n2)=O)C1 c1(C(=O)NC2CCCCN(C(=O)CC3CC(C4CC4)C3)C2)cc(O)ccc1Br C(=O)(C(N)C1CCc2ccccc21)NCC(=O)Nc1cc(OC)nc(OC)c1 c12cc(F)ccc1S2.C=CC1(C(=O)N(O)Cc2cn(C)nn2)CCC1 Cc1ccc2c(c1)CN(C(=O)CC1Cc3ccccc3C1)CC2(C)C N#CC1CN(C(c2c(Br)ccnc2Cl)=O)CC1NC(=O)C1CC1 C(CCCC(=O)NCCc1nc[nH]n1)N(C)C(C1(C#N)CC(=O)C1)=O C1(C(=O)NCC2C(C)(C)CN(C(C3(n4ccnn4)CC3)=O)C2)CC2CCCC(C1)C2 C(C(=O)NCC1CC1Cl)(C1CN(C(C2(CO)CCC2)=O)C1)OC c1(C(=O)NC(C(=O)NC2C(C)OCC2)CC2CCOCC2)cc(O)cc(=O)o1 c1(C(N2CCC(NC(=O)NC3CCC(O)C3)C2=O)C)ccccc1Cl c1(C(=O)NCCC(C)NC(C2(C=C)CC2)=O)cccc2c1ncn2C c1(C(=O)NC(C)(CNC(c2cc3scnc3[nH]2)=O)CO)nc(O)nc(O)c1F CC(C)CCCCC(=O)N1CCCC1C1(NC(C2CC3(CC3)CO2)=O)CC1 N1(C(C(=O)Nc2ccc(C)cc2)=O)CCCC(C)(NC(=O)CC2CCCOC2)C1 Cc1ccc(C#N)cc1C(N1CC(C)(C)C1C1CCN(C(=O)C=CI)CC1)=O CCC(CO)C(=O)NCC1(CNC(c2csc(C(=O)OC)n2)=O)CC1 C#Cc1ccc(CNC(=O)Nc2ccc(NC(C3CCOCC3)=O)cc2CC)cc1 C(=O)(C1=NN2CCCN=C2N1)N1CC(CNC(c2c(CCC)occ2)=O)C2C1C2 c1(OC)ncc(C(N2CC(NC(C3(O)CCC3)=O)C(C)C2)=O)cc1Br N1(C(C2(C)CCCCC2)=O)CCCC2(CCN(C(C3CNC(=O)C3)=O)CC2)C1 C1(NC(c2cccc(O)n2)=O)C2CC3CN(C(=O)CCc4cncs4)C1C3C2 C(=O)(C(C)CC#N)N(CC=CC(=O)NC(COC)CCO)C CC(C)CCCCCC(=O)N1CC2(CCCC2)C1C(N1CCCC(CCF)C1)=O C1(CNC(C2C(COC)C2)=O)CN(C(C2(CN(C)C)CCCC2)=O)CC(C)(C)O1 c1(C(=O)NCC2C(C)CCN(C(c3cnc(Cl)s3)=O)C2)cc(F)c(F)c(F)c1N N1(Cc2cnc(OC)c(C)c2)CCC(NC(C2CC2C)=O)C(C)(C)C1 c1(CC)oc(C(=O)Nc2ccc(-c3nnn(C)n3)cc2)cc1COC C=C(C)CCC(C)N=c1nc(N2CCCCC(S(C)(=O)=O)C2)c2c([nH]1)CCS2 CC(C)(O)C(=O)N1CCCC1C(C)(C)C(=O)NCCCc1nc[nH]n1 C(C(C)(C)CS(C)(=O)=O)N(C(C(C)OCC1CC1)=O)C.C(=O)(CCc1nncs1)N N1(C(CNS(N)(=O)=O)=O)CCC(CCNC(C2C3COCC23)=O)C(F)(F)C1 c1(C(N2CC(CNC(CCC=C=C)=O)CC23CCC3)=O)cn2ccc(F)cc2n1 C#Cc1cccc(C(N2CC(CNC(=O)CC3CCCO3)C(C)(C)C2)=O)c1 C1(CC(=O)NCc2cccc3c2OCO3)COCCN(C(c2csc(O)n2)=O)C1 N1(CC)CCOC(CC(N2CC(CNC(C3CC3C3CC3)=O)(OC)C2)=O)C1 c1(OC)c(F)ccc(C(=O)NC2CCCN(Cc3cccc(O)c3Cl)C2)c1F c1(NC(c2cc(-c3ccc(-c4cncs4)cc3)on2)=O)cnc(I)cn1 C1(NC(c2cnc(S)nc2)=O)CC2CC(NC(=O)C(F)CC3CC3)C1C2 C#Cc1cc(C(=O)NCCN(C(C2C3COCC23)=O)Cc2ccccc2)cc(F)c1 c1(C(N2CC3C(C(N4CCC(C)C4)=O)(C3)C2)=O)c(F)cccc1Br.C(C)(C)(C)O CCC(C(=O)NCCC1CC(N(C)C)C1)N(C)C(c1nonc1C)=O Cc1nn(C)c(C)c1CC(N1CC(CO)(NC(=O)CCCC(=O)N(C)C)C1)=O c1(C2ON=C(C)C2)nc(-c2cccc(Cl)n2)nn1C(c1cccc(C)n1)n1cncn1 N1(C(C(C(C)O)(F)F)=O)CCC2CCN(C(C3CC=CC(O)C3)=O)C2C1 c1(C(C(=O)NC(c2cccnc2)c2nn[nH]n2)O)cc(F)c(F)cc1F C#CC1CCC(C(=O)N(CC(C)O)CCNC(=O)CCC=C(C)C)CC1 N1(C(CCSCC)=O)C(C(=O)NOCCC(C)O)C2CC(O)C1C2 c1(C(N2CC(NC(CC(C)(C)C3CC3)=O)C(F)C2)=O)cc2n(n1)CCCCO2 Cc1csc2cc(C(N3CCCC(CN(C(=O)CCS(C)=O)C)C3)=O)[nH]c12 C1(NC(CCCNC(=O)CO)=O)CCN(C(=O)C2=CCCCO2)CC1O CC(O)(CC(=O)NCCCCNC(C12CCCCC1CCC2)=O)C(F)(F)F CC1CN(C(C2CC(C)(C)C2)=O)CC1CC(=O)Nc1cn(C)nc1C1CC1 N1(CC(=O)N(C)C)CCN(CC2CC3(CCC3)CN2)C(c2ccoc2)C1 C1(O)(CNC(C2N(S(CCC)(=O)=O)CCC2)=O)CCCN(C(c2csnn2)=O)C1 C#Cc1ccc(C(=O)NC(C(=O)NCCCOC2CCCC2)C2CCC2)o1 C1(C(N2CC(CC)C(C(N3CC4C(N(C)C)C4C3)=O)C2)=O)CN2CCC1CC2 Cc1c(C(N2CC=CC2CNC(=O)CC2CSCCO2)=O)[nH]ccc1=O c1(N2CCC(C)(NC(CC(CCC)O)=O)CC2)ncnc2c1CCO2 c1(C(=O)NC2CC(C(C)NC(c3n[nH]cc3C3CC3)=O)C2)ccc2occc2c1 C(=O)(C1=NOC2(CCN(C(=O)C(C)NC(=O)NC)C2)C1)OCC N1(C(C2(COC)CC=CCC2)=O)C2CC1CN(C(C1CCC(C)=C(C)C1)=O)C2 C(C)(CC(=O)N(C1(C)CCN(C(=O)Cn2ccnn2)C1)C1CC1)(C(F)(F)F)N(C)C N1(C(=O)CC(F)(F)F)CCC(C2CN(Cc3c(F)cccc3Cl)C2)CC1 c1(N2CC(C)(CC(=O)NCC(C)(C)O)C2)ccc([N+](=O)[O-])cc1 c1(C(N(C)CC2OCCN(C(C(C)C#N)=O)C2)=O)cc2c(ncn2C)[nH]1 C1(C(=O)NCCCC2CC(C)C2)(CNC(C2CCO2)=O)CC12CCC2 C1(C=O)CSCC(=O)N1.C1(C)(N(C)C)CN(N(CC(=O)N)CCOC)C1 O=C(C1CCCc2ccnn21)NC12CC(CNC(=O)CC3CC4CCC3O4)(C1)C2 C1(CCC(=O)NCC(=C)Cl)CCCN(C(C2(CC3CC3)CC2)=O)C1 N1(C(CCOCCNC(CN(CCC#C)C)=O)=O)CC(CSCC)CCC1C.OCC c1(C(=O)NCC(C)N(C(C2C(C(C)C)OCCC2)=O)C)c(Br)cccc1[N+](=O)[O-] C1(C(=O)NC(C)(C)C(F)(F)F)CCCCN(C(=O)CCCNC(=O)C2CC2)C1 c1(SCC)cccc(F)c1-c1cc(C(=O)NC2CN(C)C2)n[nH]1 c1(CC)c(NC(=O)CCC2(NC(c3sccc3F)=O)CCC2)cnn1CC CN1C(=O)C(CC(=O)NC23CC(C2)N(C(C2(CO)CCC2)=O)C3)c2ccccc21 N#Cc1cc(NC(c2nc3ccccc3s2)=O)ccc1Br Cc1cnc2n1CCN(C(=O)CCCN(C(=O)Cc1csnn1)C)C2 CCC(C)(CO)C(=O)N(CC(C)(C)CC1CN(C(c2cccc(=O)n2C)=O)C1)CC N1(C(C=CCN(CC#C)C)=O)CCCC(NC(C2CN(CC)CCO2)=O)CCC1 N1(C(CC2CC(OC(C)(C)C)C2)=O)CC2C(CNC(=O)CS(C)(=O)=O)C2C1 c1(C(CC(=O)NC2(CNC(C3(C=C)CCC3)=O)CCOC2)C)cccc(F)c1 c1(C(=O)NCCNC(=O)C2CCOc3ccccc32)ccc2c(c1O)CCCC2 CC(C)(CC(=O)N1CC2CC2(NC(c2cnn3c2CC(F)(F)C3)=O)C1)C(F)(F)F C#Cc1cccc(CNC(N2CCCC(c3ccc(NC(C)=O)cc3)C2)=O)c1 N1(C(c2scc(C)c2C)=O)CCC(NC(=O)C(C)CSC(F)(F)F)C(F)(F)CC1 C=CCCN=C(NCCc1c(C)n[nH]c1C)NCc1ncccc1OC C(=O)(C(C)(C)CC(F)F)NCC(C1CCC1)NC(C(CC)(C)CC)=O C1(C(N(C2CCN(C(CN(C(C(C)C)=O)C)=O)CC2)C(C)C)=O)CC12CCCOC2 C1(S(=O)(=O)N2CCCC2CCC(C)C)(COC)CCC1 C(=O)(C(C(C)O)C(C)C)NCCOCC.C1(OCCCSCC)CCCC1 c1(C(N(C2CCN(C(C3(CF)CC(F)(F)C3)=O)CC2)CC)=O)nc(O)sc1C C=CCCN=C(NCC1CCCN(C2CC2)C1)NC1CCOC2(CCCC2)C1 C(CN=c1[nH]c(=NCC2CC2OC(C)(C)C)c2[nH]ccc2[nH]1)N1C(C)CCCC1 C1(OCC)CCC(N=c2cc(N(C)CCC3CCCCCC3)nc(C(C)C)[nH]2)C1 C1(NC(c2c(C(C)(C)C)cccc2)=O)CCN(C(=O)Cc2cocn2)C1(C)C c1(C(=O)NC(C)CCCCNC(=O)C=CC2CCOCC2)ccc2nsnc2c1 Cc1n[nH]c2cnc(C(=O)NC3CCCCC3NC(c3cc(O)cs3)=O)cc12 c1(OC)cc(C(=O)NC(C)C(CO)NC(c2ccccn2)=O)cc2c1OC(C)C2 C12(C(=O)NC3CCN(C(=O)COCC(F)F)CC3F)CCC(CO)(CC1)CC2 N1(C(CC(C)SC)=O)CCC(C2CCCN2C(=O)CCF)CC1 C12(N(C3CCSC3)C(C)=O)CCCCCC1N(C(c1coc3c1CSC3)=O)CC2 CN=c1[nH]c(=NCC(C(C)(C)C)OC(C)(C)C)[nH]c(=NC2COC(C(C)C)C2)[nH]1 c1(C(=O)OCc2cc(C(=O)OC)n(C)c2)cc(Oc2ccccc2)ccc1Cl CC(F)(CNC(c1cc(C2CC2)no1)=O)CNC(C1CC1C1CCCO1)=O N1(C(CCCc2cc(C)no2)=O)C2CCC1CN(C(c1cc(F)oc1C)=O)CC2 N1(C(Cc2c(C)nc(C)s2)=O)CC(CO)C2(C1)CN(C(C1(C)CCC(=O)O1)=O)C2 N1(C(C(COC)(F)F)=O)CCCC2(CCN(C(c3cnc(S)[nH]3)=O)CC2)C1 c1(C(N(C(C)CNC(c2occ(C)c2C)=O)CC)=O)cnccc1C C(N=c1cc(Cl)nc(C)[nH]1)C1C(NC(CN(CC)CC)=O)C2(CC1)CCC2 N1(C(C)=O)CCCc2cc(C(=O)NCCN(C(=O)CC(F)F)CC3CC3)ccc21 c1(C(N2CC(C(C)C)C(N3CCCC3)C2)=O)cc2nc(=O)ccn2[nH]1 CN1CC2OCCN(C(=O)C(C(C)(C)C)NC(c3ccco3)=O)C2C1 CC1CNC(=O)N1C(=NC1CC1C1CCOCC1)NCc1cn2ccsc2n1 CCCS(=O)(=O)CC(=O)NCCn1cc(CNC(C2CN(C)C(=O)N2)=O)nn1 N1(C(C2(CCNC(C(COC)N(C)C)=O)CC2)=O)CCC(C)CC1 c1(NC(C2(NC(=O)CC(F)F)CC2)=O)ccc(CO)cc1 C(=O)(C(C)CCO)N1CCC(C(C)NC(c2c(-c3cn(CC)nc3)n[nH]c2)=O)C1 N1(C(C(C)(C)N(C)C)=O)CC23CCCCC2(C1)CN(C(c1cccnc1O)=O)C3 c1(OC)ccc(N2CCNC2=O)cc1C(=O)C(=O)NC1(CO)CC1(C)C CCC(C)CCCC(=O)NC(CO)C(C)NC(C1CC1c1cccc(F)c1F)=O C1(C(=O)NCCCC2(NC(c3c(C)coc3)=O)CC2)Cc2ccccc2S1 c1(C(N2C3CN(C(C4(C=C)CC4)=O)C(CC3)C2)=O)ccnc2cc(OC)ccc12 N1(C(c2c(COC)nn[nH]2)=O)CCC(O)(CCNC(=O)COCC(C)C)C1 C1(CNC(Cc2c(Br)ccc(OC)c2)=O)CC2CCC(C1)N2C(=O)C(C)(C)CF Cc1ccc(C2C(C)CN2C(c2sccc2C(=O)NS(C)(=O)=O)=O)cc1 C(CCCN=c1[nH]c(=NCc2ccncc2Cl)[nH]c2cccnc12)(C(C)C)OC N1(C(C(CC)(C)F)=O)CC2(C1)CN(C(=O)CC(C)N(C)C)CCO2 C1(CCC)CN(C(=O)C(C)CO)CC1C(=O)N(C1CCCCCC1)C O=C(C1CCCc2ncnn21)OCc1nc[nH]n1 N1(C(CC=C=C)=O)CC2(CCCN(C(c3ccc(CC)cn3)=O)C2)C1 C1(NC(c2cc(C(C)C)[nH]n2)=O)CCN(C(c2cccc(O)n2)=O)CC1F c1(C(N(C(C)CCNC(=O)CN2CCOCC2)C)=O)cccc(CC#N)c1 c1(C(=O)NCCOCCNC(c2c(CC)occ2)=O)sc(C)c(Br)c1C c1(NC(C2N(C(c3nccc(OC)c3)=O)CC(C)C2)=O)ccc2[nH]nc(I)c2c1 C1(N(C(CCc2cc(C)[nH]n2)=O)C)C2CN(C(C3CC=CCC3)=O)CC12 N1(Cc2c(OC)cc(C)cc2)CCC(NC(=O)Nc2ccc(C)nc2)C(C)(C)C1 C1(C(=O)NCCCC(C)(C)OC)CCC(C)N(C(=O)C=C(C)C)C1 C(=O)(CC(C(C)C)c1ccccc1)NCC(CNC(c1cc(Cl)c[nH]1)=O)OC c1(C(N2CCCN(C(=O)CC3CC4CC4C3)CC2)=O)cc2cccnc2o1 C1(CNC(c2cccc(C3CCC3)c2)=O)CN(C(OC(F)(F)F)=O)CC1(F)F Cc1ccc(C(=O)NCC2COC(CNC(c3ccncc3Br)=O)C2)nc1 N1(C(CC(COC)C)=O)CCCN(C(=O)C(C)CC(N)=O)CC1 c1(C(N2CC(CCNC(c3c(CC)scc3)=O)(OC)C2)=O)ccc([N+](=O)[O-])[nH]1 c1(NC(C(N2CCCCC(CSC)C2)c2cc(C)[nH]n2)=O)ccc2c(c1)CCC2 c1(CC(=O)N(C2C3CN(C(C4CCC5(CC5)C4)=O)CC23)CC)cc(Cl)ccc1F N1(C(C2CS(=O)C2)=O)CC2CCCN(C(=O)CC3CCCCC3O)C2C1 CCCC(CCC)CC(=O)N1CCC(OCC(N2CCC(C3(C)N=N3)C2)=O)C1 C1(CNC(=NC)NCCCC(C)C)CCOC(CC)C1 C1(C(N(CCNC(c2scnc2C2CC2)=O)CC2CC2)=O)CC2(CO1)CC(F)(F)C2 c1(C(N2CCOCC2)C)nc(C2CCCO2)n(CCC2CC2)n1 c1(C(N2CCCC2c2ccco2)=O)cnc2c(C3=CCC(O)CC3)cnn2c1 CC1CN(C(c2ocnc2C(F)F)=O)CC(C)C1NC(=O)CSCCC(F)(F)F C1(CNC(C(N2CCNC2=O)C)=O)CCC2(CO1)CC(NC(=O)CC1CCC1)C2 Cc1cnc(C(C)NC(c2cc(CNC(C3(C)CC=CC3)=O)[nH]n2)=O)o1 N(C(=NCC(C)c1nccs1)NC1CCCS(=O)(=O)C1)C(COC)C Cn1c(=O)c(CSCCOc2ncco2)c(O)c2ccccc12 CC1(C)CC(CNC(c2ccnc(C3CC3)n2)=O)N(C(=O)CCCN=[N+]=[N-])C1 c1(C2C(C(=O)CN3CC(C4CCCN4)C3)C2)ccc2c(c1)CCCC2 c1(OC)ccc(C(C)C(=O)N2CCC2CNC(C2CC2F)=O)cc1F N1(C(COCCCC)=O)CCN(C(=O)C(C)(C)C)CC1CS(C)(=O)=O C1(C(N2CC3N(C(CC(CC)C)=O)CC(C3)C2)=O)CC1C1CC(N=[N+]=[N-])C1 C1(NC(c2cnc(N3CCOCC3)s2)=O)CCCC(NC(c2cncs2)=O)C1 Cc1nc(Br)oc1C(=O)NCc1cn(C2CCN(C(=O)C(C)CF)C2)nn1 N1(C(C2CCN(CC3(C=C)CCC3)C2)=O)CCC2(CCOCC2)C1 C1(CCC2N(C(CN(C)C3CC3)=O)CCC2)CCN(C(C2CC2C(F)(F)F)=O)CC1 CC1NC(=O)CCC1CNC(=O)CCN(C(=O)CCCNC(N)=O)C C=CCC(CC=C)C(=O)N(C1CCC2CN(C(C3CCCOCC3)=O)CC12)C C1(NC(C(C(=O)OCC)F)=O)CC2(C(=O)NCCC(C)C(C)C)COC1C2 C1(NC(c2scc(C)c2)=O)CN(C(c2ccnc(C)c2N)=O)CCC1C C(=O)(CC(O)C(C)C)N1CCC(CNC(COc2cc(C)on2)=O)(CO)C1 c1(C(N(CCCNC(c2cn(CC)nc2C)=O)CC)=O)cccn2nccc12 N1(C(C2CCC(n3cc(CCc4cnccn4)nn3)C2)=O)CCCOCC1 CCC(CC)CC(=O)NC1CC2CC(C(=O)NCC(CC)(CC)CO)CC12 C1(NC(N2CC(c3ccn(C)n3)OCC2)=O)CCC(F)(F)CC1 C1(CNC(C(C)NS(C)(=O)=O)=O)CCC(C(=O)NCCCCc2ncc[nH]2)O1 N1(C(c2cnccc2C)=O)CCC(N(C(C(C)OCC=C)=O)CC(C)C)CC1 C1(NC(=O)NC2CC(NC(C3CC(C(N)=O)C3)=O)C2)CCCCCC1 C(=O)(CC(CCC)CCC)N1CCC(NC(c2c(C#C)cnn2C)=O)C1 c1(C(N(C(C(=O)N(CC#CC)CC#C)C2CC2)C)=O)cccnn1 CC(CCC(=O)NC1CC2(CC2)C1)NC(c1ccc(Cl)s1)=O c1(N2C(CNC(C3(CC=C)CC3)=O)CN(C)CC2)cc(OC)c([N+](=O)[O-])cc1F S(=O)(=O)(c1ccccc1Cl)N1CC(NC(c2c(C)scn2)=O)C(F)C1 [N-]=[N+]=NC1CCCN(C(C2CC23CCN(C(C2(O)CC2)=O)C3)=O)CC1 C1(CC(=O)NC2CC2c2cncs2)C2CN(C(C3CC3F)=O)CC12 CC(O)C(C)(C)C(=O)NCc1ccc(CCNC(=O)CC2CN(C)C2)cc1 C12(NC(CN3CCC(=O)NC3=O)=O)CC3CC1CN(C3)CC2 CCCCCCCC=CC(N1CCCC1CNC(c1ccnc(O)c1)=O)=O C(C)(CN=c1cccc(S(=O)(=O)NC2CC=CCC2)[nH]1)N(CCCOC)C c1(C(=O)OCCOCC#C)ccc(OCC)cc1Cl.C12CC(C1)NC2=O Cc1ncccc1CN(C=O)C(C1(O)COC1)C c1(N(C)Cc2cccc(CNC(COCC)=O)c2)cc(Cl)c(C)nn1 C1(C(N(CCNC(C2CN(C(C)C)C2)=O)C)=O)CCOCC12CCCC2 c1(CNC(CN(C(=O)Cn2cc(-c3cccs3)nn2)C)C(=O)O)c(F)cccc1F C1(C(=O)NCC2CCCC2NC(C2(C)CC2)=O)(OCC)CCCCCC1 CC1=NOC(C)(CNC(=O)C(C2(O)CN(C(C3C4CC(=O)CC34)=O)C2)F)C1 c1(C(=O)OC)sc(C(=O)N(C2CCN(C(c3cc(Cl)no3)=O)C2)C)cc1C c1(CC(=O)NCCN(C)C(c2cnoc2-c2ccco2)=O)cn(C)nn1 N#CC1CN(C(c2cn(C3CCCNCC3)nn2)=O)CCC1(F)F N1(C(CC)C(=O)NCC(CO)NC(C2(CF)CC2)=O)C(=O)CCC1=O c1(C(=O)NC2C(CNC(c3n[nH]c(C)c3Br)=O)C2)cnc(O)n(C)c1=O C#Cc1ccc(C(=O)N(CC(C)O)CCNC(c2cnc(O)n2C)=O)cc1C c1(NC(C2CCCCN2C(=O)CCc2ccco2)=O)ccc2nc[nH]c2c1 C(c1ccc(C)c(C)c1)=CC(N1CCN(C(C(CCC)CC)=O)C2C1C2)=O c1(C(=O)NCCC(O)CNC(c2ccncn2)=O)scnc1CCC(F)(F)F c1(C(C(=O)NC2CC(F)(CNC(c3ccc(F)cn3)=O)C2)O)ccc(O)cc1 C(C1OCCc2sc(I)cc21)NC(c1ccc(C#N)cc1)C1CC1 N1(C(CCCCCOC)=O)CCN(C(=O)C(N2CCOCC2=O)C)CCC1C C1(N(C(CSC(C)C)=O)C)CN(C(=O)CN2CCCCS2(=O)=O)CC12CC2 c1(NC(CCN(C(c2cc(C)ns2)=O)CCO)=O)cnc(C(C)C)nc1 C(=O)(C#CC(C)(C)CNC(=O)C(COCC)(CC)CC)N(C(CC#C)C)C N12CCCC(CC1)C(=O)NC(C)C(=O)NC(COCC)C2=O.C#CCNC(C)=O c1(CCC(=O)NCCCOCCN(C(=O)C(O)C2CC2)C)nccn1C CN(C)S(C)(=O)=NS(=O)(=O)NC1CC(C)(C)C1 C(=O)(C1COCc2ccccc21)N1CCC(CNC(c2cc(C)n(C)c2)=O)CC1 c1(C(=O)NC2CC(CNC(C(C)CC(N)=O)=O)CC2O)cc(F)cc2nc[nH]c12 c1(C(N2CCOCC(C)C2)C(=O)NC(C(=O)OC)C)ccc(SC)cc1Br C1(C(N2CCCC(NC(=O)CCSC(F)(F)F)C2)=O)Cc2nncn2C1 N1CCC=C(C=O)C1.Cc1ccnnc1C(=O)NOCCCN(C)C c1(NC(C=CCC)=O)ccc(NC(=O)CCc2ccccn2)c(C)c1 C1(CNC(C(C)=C2CCCC2)=O)CCCN1c1nnc(CN(C)C)s1 C1(F)(C(=O)NCCN(CCCC)C)CCN(C(C2SCCS2)=O)C1 c1(C(N(C2C(NC(C(F)=CC)=O)CCCC2)C)=O)cc2cc(C)ccc2nc1C C=CC1(C2(C(=O)NC3CC4CC3N(C(=O)Cc3cc[nH]n3)C4)CCC2)CCC1 N1(C(c2cc(CC)[nH]n2)=O)C2CCC1CC(CNC(C1CC1CCN(C)C)=O)C2 C(=O)(C(C)(C)CCCO)N(C)CCNS(N)(=O)=O.C1C(=O)N1 C1(CCOC)CN(C(=O)C2=CCCCC2)CCN1C(C1CC1C#N)=O C=CC(C)(C)CC(=O)NC(CCN(C)C)C(=O)NC1CNC(=O)C1(C)C c1(C(=O)NCC2(C)CCC(NC(C3(C4CC4)CC3)=O)C2)c[nH]c2c(Cl)cccc12 c1(CC)cc(C(N2CCC(CO)(NC(c3ccnc(C(F)F)c3)=O)C2)=O)ncn1 N1(C(c2ccc(C)nc2)=O)CCc2sccc2C1CNC(=O)CC1CN(C)C1 C1(NC(c2c(CC)non2)=O)CCCCC1NC(c1cscc1Cl)=O n1(CC)nnc(C)c1C(=O)NC(C)C(C)NC(=O)Cc1nc(C2CC2)nn1C C(=O)(CC(C)(C)CN(C)C)N1CCC(N(C(Cc2cc(C)sc2C)=O)CCO)C1 S(=O)(=O)(c1ccc(C)c(C)c1)N1CCC(NC(c2c(OC)nccc2)=O)C(C)C1 Cc1cc(Br)cnc1C(=O)NC1CC(CNC(=O)CNC(C2CC2C)=O)C1 C1(NC(C)=O)CC(S(C)(=O)=NC(=O)c2ccc(OCC(F)(F)F)nc2)C1 c1(NC(C2CC(F)CN2C(c2cc(Cl)c(Br)cn2)=O)=O)ncc(Br)cc1[N+](=O)[O-] c1(CNC(CC)=O)ccccc1CNC(=O)CC1CCCC1.CC(C)(C)OC(N)=O c1(C(N(C)CCNC(C2CCCN2C2CCCC2)=O)=O)ccc2sc(O)nc2c1 CCN=c1[nH]cc(C(N2CCN(C(=O)Cn3ccc(C)cc3=O)C(C)C2)=O)s1 N1(C(CCCCC)=O)CCC2(CCN(C(=O)CC3CCCC(=O)C3)C2)C1 c1(C(N(CC(C)O)CCNC(=O)Cc2sccc2Cl)=O)ccc(CN(C)C)cc1 c1(CC)cnc(O)c(C(=O)N(C(C)CNC(c2c(O)noc2C)=O)C)c1 C1(NC(CCCC=C)=O)CN(C(C2(COCC)CCCC2)=O)CCC1O Cc1[nH]c(=N)nc(-c2ccc(C(=O)NC(c3cccs3)C)cc2)c1C c1(C(N2C(CNC(=O)CCCC(=O)N(C)C)CC(OC)C2)=O)ccc(N)c(O)c1 CCC(C)C(C)C(=O)NC1(n2cccn2)CCN(C(c2ccnc(C3CC3)c2)=O)C1 C(c1ccc2ccc(Cl)cc2n1)=CC(=O)NCC1CC1NC(c1n[nH]cc1Cl)=O c1(CC)c[nH]cc1C(=O)NCc1n[nH]cc1C(=O)N(C(C)C(C)SC)C C12(C(N3C(CCNC(CN(CC)CC)=O)CSCC3)=O)CCC(CC1)C(C)O2 n1(CCCNC(C2N(C(c3ccc(C)c(C)c3)=O)CC2)=O)cc(S(N)(=O)=O)cn1 C123CC1CN(C2)C(=O)CN3C1CC1.c1(C(=O)NC(CC2(C=C)CC2)=O)ccc(C)s1 N1(C(C2CC3(C)OCC2C3)=O)CCCC(C2CN(C(=O)C(O)c3ccsc3)C2)C1 C1(C(=O)NC(CN(C)CC2(CN)CC2)=O)CCCO1.C1(C(=O)NC2CC2)CC1 c1(NS(CC(=O)OCC2CC2)(=O)=O)ccc(OC(F)F)cc1F Cc1cc(S(=O)(=O)NC(c2ccccc2)CN2CCCC(C)C2)cc([N+](=O)[O-])c1C N1(C(c2c(COC)ccs2)=O)CC(CNC(=O)CCc2cnn[nH]2)OC(C)(C)C1 C1(NC(C(CCC)N(C)C)=O)CC2CN(C(c3nnccc3C)=O)CC2C1 c1(OC)cc(C(N2CCC(F)(C(=O)NCC(C3CCCCC3)OC)C2)=O)nn1C c1(OC)ccc(NC(C2CCCN(C(C3CC4CCC3CC4)=O)C2)=O)cc1C Cc1c(-c2cn(C3CC(C(=O)NCCC(C)(C)O)C3)nn2)cccc1F C1(C(N(CC(CO)(CO)NC(c2onc(C)c2C)=O)C)=O)COC2(CCC2)C1 C(=O)(C(C)(O)C1CC1)NCCCNC(=O)CCOCC(C)(C)SC1CC1 C(=O)(C1=C(C)CCC1)NC(COCC)C(=O)N1CCCC1CN=[N+]=[N-] c1(OC)ccc(NC(=O)CN2CCCC(C(O)C(F)(F)F)C2)cc1 C=C(C)CN=C(NCCCN(C)C)NCC(c1ccc(F)cc1C)C c1(C(=O)NCC2N(C(c3c(C)[nH]nc3Cl)=O)CCCC2C)cccc2oncc12 C#CCC(C)(C)C(=O)NC1CCOCC1NC(C1CCC(=O)N(C2CC2)C1)=O C(=O)(C1Cc2c(Cl)cccc21)NC(C(C)C)(C)CNC(=O)Cc1cccc(F)c1 N1(C(C(CCC)C)=O)CCN(C(c2c(C)cnc(OC)c2Cl)=O)CC(C)(F)C1 C1(NC(C(c2ccn(C)n2)C)=O)CC2CN(C(=O)Cc3ccsc3)CC12 C1(NC(CC(C)n2ccnc2)=O)CCOC12CCN(C(=O)C1=CCCCC1)CC2 CC1=CCSC1C(=O)NC1(CC2CCC2C(=O)NCCc2nccn2C)CC1 N1(Cc2c(OCC)c(Cl)ccc2)CCC(F)(F)C(C(=O)Nc2ncc(Br)s2)C1 CC(=O)CCC(=O)NCCC(=O)NCC1CC(F)C1 c1(CC)ncc2c(n1)CCC(C(=O)NCCc1ccc(O)c(F)c1)C2 c1(C(N(CCC)CCNC(C2CC2C(C)C)=O)=O)c(F)cc(N)cc1F C1(CC)CCCCC1OCC(=O)N(CCCN(C(=O)C1=CCCC1)C)C Cc1cn(C2CCOCC2)nc1C(=O)NC1CC1CNC(=O)C=CBr C(=O)(CC(C(F)(F)F)c1nccn1C)NCCCN(C(=O)C(O)CF)C C1(=O)CC(=O)N(C(=O)CC2CCOC2C)C(C)N1.C1(N(C)CC)(C=O)CC1.C(C)(C)(C)O N1(C(C(C(C)C)(F)CNC(c2cc[n+]([O-])cc2)=O)=O)CC2CCCC2C12CC2 S(=O)(=O)(CC(C1CC1)NC(=O)CCCc1ccccc1Cl)NC N1(C(c2oc3ccc(C)cc3c2)=O)CC2(C1)CN(C)CCO2 c1(CC(=O)NCC2C(C)CCN(C(C3CCOC3)=O)C2)ccc2c(c1)OCO2 c1(C(=O)NCCC2N(C(CC(C)(C)C)=O)CCCC2)cc(O)nc(O)n1 c1(C(=O)NCC2CCN(C(C(C(CC)C)OC)=O)C2)cccc2nsnc12 C1(CC)CCCCC1C(=O)NCC(C)CNC(c1nn[nH]c1Cl)=O c1(OCC)cncc(C(=O)NC2CC(C(=O)NC(c3nc[nH]n3)C)C2(C)C)c1 C1(=CC(=O)NC(C(=O)OCC)C(O)c2ccc(F)cc2)CCCCCC1(F)F c1(C)ccc(Cl)c(F)c1.n1(C2CC2)nnc(CC)c1C.C12C3CN(CC13)NC(=O)C2 c1(C(=O)NC2CCN(C3CN(C(=O)OC)C3)C2=O)cc2sc3ccccc3c2s1 N1(C(C)=O)CCC(C)(C(N2CC(NC(=O)Cn3cnnn3)C2)=O)C1 Cc1ccc(C(C)C)cc1C(=O)NCCc1noc(=O)n1C1CCOC1 Cc1cc(C(=O)NCCC2COCCN2C(C2CC2F)=O)cc2ccsc12 N1(C(C(=O)NC(c2c(C)cccc2)C(F)(F)F)=O)CC(C)C12CCOCC2 N1(C(COC)=O)CCCC2C(CCCN2C(=O)CCCC2CCCO2)C1 CCCCC(F)C(=O)N1CCOCC(CNC(=O)C=CC2CCCN2C)C1 c1(C(=O)NC(CC=C)CNC(c2ncn(C)n2)=O)ccc2ncsc2c1 c1(C(=O)NCC2(CNC(=O)CCc3ccc(F)cc3)CC2)cc2cccnc2s1 CC1CN(C(C2(CO)COC2)=O)Cc2nncn21 N1(C(c2c(C)[nH]cc2)=O)CCC2(CC(NC(C3(O)CCC3)=O)CO2)C1 C1(C(C)NC(C2CSC2)=O)CCN(C(C2(C3CC3)CC2)=O)C1 c1(C(=O)OC)nc(CNC(C2CCCC2NC(c2ccc(CF)cc2)=O)=O)oc1C N1(C(c2c(C(=O)OC)csc2)=O)C2CCC1C1CC1(NC(=O)C(O)CC(C)C)C2 C(=O)(N=c1cc(-c2ccc(C)cc2)o[nH]1)NC1C(CCC)CCC1 C(C(O)C(=O)NC(C)CC1CN(C(c2cnc(Cc3ccccc3)s2)=O)C1)OC N1(C(C)C)CCCC(CC(N2CCCC2C2(NC(C3CCS(=O)(=O)N3)=O)CC2)=O)C1 Cc1ccc(C)c(C(=O)NCC2CC2NC(=O)CCCCCc2ccccc2)n1 N(C(=NCC1CCC(=O)N1)N1CCSC(C)CC1)C(C)Cc1ccccc1 C1(C(=O)NC(c2cccs2)CC)CCN(C(c2oc(C)nc2C)=O)CC1(C)C C1(C(=O)NC2CCN(C(CCc3cc(C)[nH]n3)=O)C23CC3)CCn2nncc2C1 C=CC1(CC(=O)N(CC(N2CC3(C2)CN(C)C3)=O)CC(C)C)CCCCC1 c1(OC(C)C(=O)NCC(C)CNC(=O)CSc2ccccc2)ccc(O)cc1 C(CC(C(=O)N1CC(N2CCOCC2)C1)OC)N(C(Cn1cc(SC)nn1)=O)C c1(CCC(=O)NC2C=CCN(C(c3coc(CO)c3)=O)C2)cncc(Br)c1 N1(C(C=Cc2cn(C)nc2)=O)CCN(C(=O)CNC=O)C2CCCCC12 C#Cc1cccc(CC(=O)NC2CC3(C2)CN(C(=O)C(CC)CCOCC)C3)c1 C(=O)(C(C)CC(C)(C)C)NC1C(CNC(c2cncc(CC)c2)=O)CCC1 CCCCCC(O)C(=O)NC1CCN(C(=O)CN(c2ncccn2)C)C1C1CC1 N1(C(CC(CNC(C(CCCC)F)=O)C)=O)CCn2cc(C)nc2C1 Cc1cnc(N)c(C(N2CCC(NC(C3CC(F)CN3C)=O)CC2)=O)c1 C(C)(C)(CCCNC(c1cnc(O)s1)=O)NC(Cc1nnc(C)o1)=O C(CCCCC(=O)NCCC1CCCCN1C(c1cc(Cl)ccn1)=O)OC N1(C(c2cc(SC)oc2)=O)CC2CC2(C(=O)NC2CCCC(O)C2)C1 C1(O)(CNC(=O)CC(F)(F)F)CCCN(C(=O)Cc2cccnc2Br)C1 C1(C(C)C)CN(C(=O)CSC2CC2)CCC1NC(=O)C=Cc1nnn(C)n1 C(=O)(CC(CNCC(c1ccc(Cl)c(C)c1)=O)C(F)(F)F)OC N1(C2CCC(=O)N(CCF)CCCCC2)CC1.Cc1cscc1CO N1(C(N2C(C(C3(C(F)(F)F)CC3)C)CC(O)CC2)=O)CCC2(CC1)CC2(C)C c1(C(=O)NCC(CC)NC(c2c[nH]c(Br)c2)=O)cc(C)nc(O)n1 c1(C(C(=O)OCC(=O)CC2CCCC2)NC(C)=O)ccccc1 C1(CC)(CC)CCCN(c2cc(N3CCSC(N4CCCC4)C3)nc(C)n2)C1 c1(OC)ccnc(CNC(=O)CC2CCCCN2C(=O)Cn2nc(C)nc2C)n1 N1(C(c2ccc(I)s2)C(=O)NC)CC(CC2CCOC2)C(C(F)(F)F)C1 CCCCC(C)C(=O)NCC1CCCC1NC(C1CCCC(C)(C)C1)=O c1(NC(c2cccc(OC)c2O)=O)ccc2c(c1)CN(Cc1ccc(Cl)nc1)C2 C1(NC(CC2CC(C)C2)=O)CN(C(c2cccnc2N(C)C)=O)CC1C c1(C(=O)NCC(CNC(C(CCC)CC)=O)(C)C)c(S(N)(=O)=O)ncn1C c1(C(N2C(CNC(C3(COC)CCCC3)=O)CCC2)=O)c(C)ccc2nsnc12 C1(C(=O)NCC2CCCCN2C(C2(C(=O)N(C)C)CC2)=O)(CC)CCCCO1 c1(CC(=O)NCC2CN(C(c3cc[nH]c3)=O)CC2O)ccc2ncccc2c1 C1(NC(CCCCOC)=O)CCN(C(c2ccc(OC)c(Cl)c2)=O)CC12CCC2 N1(C(c2cncc(C)n2)=O)CCCC1C1CCCCN1C(=O)CCCF C1(NC(COCCOC)=O)CCC(C)(C)CC1CNC(=O)C(CC)C(=O)OC.OC N1(C(Cn2c(C)nnn2)=O)C2CCC1C(CNC(=O)CC1CCOC1)C2 c1(CCOCC(=O)O)cnc2c(C#N)cnn2c1.c1(CC(C)NC)ccc(O)cc1 C1(CC(C)NC(COC(CC)(C)C)=O)CC2CCC(C1)N2C(c1cccnc1)=O N1(C(=O)NCC2(c3ccc(C)cc3)CCCCC2)CCSC2CCC12 C#Cc1ccc(C(N2CCCC2C(=O)NCC(N2CC3(CCC3)C2)=O)=O)c(C)c1 C1(CNC(C(=O)NCC(CCOC)NC(=O)C(C(C)C)SC)=O)CCOC(=O)CC1 N1(C(c2[nH]cc(CC)n2)=O)CCC2(CC1)CN(C(C1(C)CCN(C)C1)=O)C2 N1(C(c2c(C)cc(C)[nH]2)=O)CCC(NC(=O)CN(C)C(c2ccoc2)=O)CC1C C1(NC(CC23CC(C)(OC2)C3)=O)CN(C(c2ccn(C3CC3)n2)=O)CC2(CC2)C1 CC1(CNC(=O)COCC2CCCO2)COCCN(C(=O)Cn2nccn2)C1 Cc1cc(C(=O)NCC2CC3CC(C2)N(C(C2(CO)CCC2)=O)C3)cc(=O)n1C N1(C(CS(CCOC)(=O)=O)=O)CCC(CC(=O)NCC2CC2C#N)C(F)(F)CC1 C#CCCCC(C)C(=O)N1CCC1CNC(c1ccncc1)=O c1(CN(CCO)Cc2cn(C3CCN(C)C3=O)nn2)ccc(Cl)cc1Cl C(=O)(CC(C(F)F)NC(c1cccc(O)c1)=O)N(C1CC(F)(F)C1)C c1(CCC(=O)N(CCNC(C(COC)O)=O)Cc2cccc(Cl)c2)ccc(=N)[nH]c1 C1(C(=O)NCCC2(O)CN(C(C(COCC)C)=O)C2)CCN(C)CC1 c1(C(=O)NCCN(CCOC)C(c2cc(OC)cc[n+]2[O-])=O)cnc(O)cc1C C1(CNC(c2ccc(F)c(F)c2)=O)CC(C(=O)NCc2ccnc(Cl)c2)=NO1 c1(NC(=O)CC2(c3ccncc3)CCC2)ccc(NC2CCCC2)nc1 C1(C(C(C)C)NCC(c2ccc(Cl)cc2)(F)F)CCN(C(=O)C=CCO)CC1 C(=O)(C(F)C(F)(F)C(F)(F)F)NC1CCC(C)(NC(=O)CC2OCCO2)CC1 N1(C(C(C)=C(C)C)=O)CCC(C2CC(NC(c3cc(Cl)cnn3)=O)C2)C1 S(=O)(=O)(c1cnn(C)c1)NCC(=O)NC1C(C)N(C(=O)CCCC(N)=O)CCC1 O(NC(=O)C(c1cnn(C)c1)NC(=O)CC1CCCN(C)C1)CC(=O)OC N1(C(C(CCC)c2ccccc2)=O)CCCC12CCN(C(C1(F)CC1)=O)C2 C1(OC)CCN(C(=O)C(CC2CC2)NC(C2CCCCC2F)=O)C1C N1(C(C=CCCC)=O)CCCC2CCN(C(C3CC(n4ccnn4)C3)=O)CC12 c1(NC(CNCCC(COC)O)=O)cccc(C)c1O C(=O)(C1CCCc2cncn21)N1C(CNC(C2(C)CC(C#N)C2)=O)CCCC1 N(C(=NCCCCl)NCC1CC(=O)N(C2CC2)C1)CC(=C)CC N1(C(C(N2CCCCC2=O)CC)=O)CC(NC(c2c(C)cnn2C)=O)C(C)(C)C1 C1(OC)CC2(C1)CC2C(N1CC2(NC(=O)C=Cc3ccc(C)o3)CC1C2)=O C1(C(=O)NCC2(c3nccc(OC)c3)CCCC2)CC(=O)NC(=O)C1 CC1(C)CC(C(N2CCC3C(NC(c4cc(C(N)=O)co4)=O)C23)=O)CCO1 CC(C)(C)CCCCC(=O)N1CC2C(NC(c3nccc4ccsc34)=O)C2C1 CC1OCCN(C(c2cc(F)n(C)n2)=O)C1C(=O)NCCC(F)(F)Cl c1(CC)cc(C(=O)NCC2CCCN2C(C2(CO)CCS(=O)(=O)C2)=O)cc(O)n1 c1(OC(C)C)ccccc1C(=O)NC(C1CN(C(C2CC2C(C)O)=O)C1)C c1(C(=O)NC2C(C)CCN(C(C(CC)(CC)CO)=O)C2)cc2cccc(Cl)c2s1 CCCC(C)(O)CC(=O)N1CCN(C(c2c[nH]nc2Cl)=O)C(c2ncc[nH]2)C1 c1(C(C(=O)Nc2ccccc2)N(C(CC#C)C)C)sc(=O)n(C)c1Cl c1(CC)[nH]nc(Cl)c1C(=O)NC1CCCC(NC(C2CCCCS2)=O)C1 C12(C(N3CCC4(NC(CC(CC)(F)F)=O)C(C3)C4)=O)CC1COC21CCC1 C(=O)(C(CCCC(C)C)N1CCOC(c2ccc(C(F)(F)F)cc2)C1)OC C1(OC)CC(NC(=O)CC2CCCCCC2)C12CCN(C(=O)C(N)=O)CC2 C12(CNC(CCN(C(Cn3ncc(C)c3)=O)CCCO)=O)CCCCC1C2 N(C(=NCCF)NC1CC(C)N(CC(C)C)C1)Cc1cc(C(C)(C)C)on1 CC(C(=O)N(C)CCN(C)C(C1CC(=O)N(c2cn[nH]c2)C1)=O)C(C)(C)O N1(C(c2c(CC)cno2)=O)CCCCC1C1CCN(C(=O)C(C)CSC)C1 CCCCCC(O)CC(=O)NCC12CC1CN(C(c1n[nH]cc1C(F)(F)F)=O)C2 N1(C(CC=C)=O)CCC2(COCC(CNC(=O)CC3CN4CCC3CC4)O2)C1 C1(CC(N2C(c3cn(CCC=C=C)nn3)C(C)CC2)=O)CCCN2CCCC12 C(C)(CCN=c1[nH]ccc(C)c1[N+](=O)[O-])NC(CCCc1ccc(CC)cc1)=O C1(NC(C2CN(C(N(C)C)=O)C2)=O)CC2CC1N(C(=O)C(F)n1ccnc1)C2 N1(C(c2csc(C(F)F)n2)=O)CCC2CCN(C(=O)C=C3CCCCC3)C2C1 CC(C)CN=C(NC1CC12CC(OC(C)(C)C)C2)N1CCC(C)(F)C1 Cc1ccc(C(N2CCOC(CC(N3CC4(CC=CC4)C3)=O)C2)=O)cc1C#N C1(C(=O)NCC2CC(C(N(CC(C)O)CC)=O)C2)COCC1N(C)C N1(C(c2ccc(C)cc2Br)=O)CC2CN(C(c3nocc3C)=O)CCC12 N1(C(Cn2c(CCC)ncc2)=O)CCC2CC2(NC(=O)CS(=O)(=O)C2CC2)CC1 Cc1cc(OCC(=O)NCC2(CNC(=O)CNC(N)=O)CCCC2)cc(C)c1 C12(CNC(=O)CCC3(NC(c4ccoc4Cl)=O)CCC3)CCCC1OCC2 N1(C(c2n(CCC)ncc2)=O)CCN(N2CCC(NC(C)=O)C2)CC1.C(=O)C(C)SC N1(C(c2n[nH]cc2F)=O)CC2CC(C1)N(C(c1ccnc(OC(F)F)c1)=O)C2 c1(NC(c2cc(F)c(F)c(F)c2)C)ccc(S(=O)(=O)NCc2cn(C)cn2)cn1 Cc1nn(C)c(Cl)c1C(N1CCN(C2CCC(NC(=O)C3CC3)C2)CC1)=O C1(NC(CSCC=C)=O)CN(C(=O)Cc2ccc(OC)nc2)C2(CCOC2)C1 Cc1ncn(C)c1C(=O)NCC12CC(NC(=O)C(F)(F)c3nc(CPNC)cs3)(C1)C2 N1(C(CC(C)(C)N(C(C2C(C(=O)OC)CC2)=O)C)=O)CCCC2(CC2)C1 C1(C(=O)NCC(CC(=O)NCC2(CO)CC3CC3C2)OC)CN2CCN1CC2 N1(C(c2cnc(CCC)s2)=O)CCOCC1CNC(=O)CCc1cc(C)on1 c1(C(N(C2CCCN(C(C3C(C)C3)=O)C2)CC2CC2)=O)ncn2c1CCC2 c1(C(N2CCC(C(C)NC(=O)CS(=O)(=O)C3CC3)C2)=O)cccc2oc(O)nc12 C1(CNC(=O)Cc2c[nH]ccc2=O)CC2(CC2)CN1C(=O)CC1COCCO1 CC1CN(C(C2(C)CC2)=O)CC(C)CN1C(=O)CN1C(C)CCC1C c1(OC)ccc([N+](=O)[O-])c(N(CCCN(C(=O)CN2CCCS2(=O)=O)C)C)n1 N1(C(C(C)OCC)=O)CCN(C(c2nccc(Cl)c2F)=O)C(CF)C1 Cc1nnc2n1CC(N(CCO)C(C1CC3CC3C1)=O)CC2 Cc1ccc(C(F)C(N2CC(NC(c3snnc3C(C)C)=O)C3CC23)=O)cc1 CC1CC(NC(=O)CSc2nnnn2C2CC2)CCN1C(=O)C(C#N)C(C)C c1(SCCCC(=O)NC(C(=O)OC)CC2CCC(=O)N2)nc2ccccc2[nH]1 CC1CCNCCC1N(C1CC1O)C(c1c(Cl)ccnc1Cl)=O C(C)(CC1CCC1)(C(=O)NCC1CCN(C(=O)C=C2CCN(C)C2)C1)OC c1(C(=O)NC2(COCC(=O)NC3CC(CO)C3)COC2)ccsc1-n1cnnn1 C1(C(=O)NCC(C)NC(C2(c3ccc(O)cc3)CC2)=O)(OC)CCCCOC1 c1(C(=O)NCC2CC(NC(C(CCCC)N(C)C)=O)C2)cc(F)c(C)cc1N c1(C(N2CCC(C)C2)C(=O)NCCN(CCC)CCC)ccccc1F c1(C(=O)NC(CNC(CSCCC)=O)CC(C)C)c(C)ncn(C)c1=O N1(C(CCCCC)=O)CCCC(C2CCCN(C(c3nc(Cl)sc3Cl)=O)C2)C1 N1(C(CC=CC=C)=O)CCC(O)(C(C)CNC(=O)C=C2CCC2)C1 C12(NC(CCC#N)=O)CCN(C(c3cc(Cl)cc(Cl)c3)=O)CC1C2 c1(C(N2CC(CCO)(NC(c3ncc(C)cc3C)=O)C2)=O)cccc2c[nH]nc12 C1(C(=O)NC(C)CNC(=O)CNC(=O)C(C)(C)C)(CC)CCNC1=O c1(N(C)C)ncccc1C(=O)NC1CCN(C(c2ccn(C3CC3)n2)=O)C1 C(N=c1[nH]c(=NCC2COCCN2C)[nH]c2c1COCC2)c1c(C)sc(C)c1 N1(C(c2cnc(COC)nc2O)=O)CCC2(CC1)CCN(C(=O)CNC=O)CC2 c1(C(N2CC(C(C)NC(=O)C=C(Cl)Cl)OCC2)=O)cc([N+](=O)[O-])cc([N+](=O)[O-])c1 Cc1ccc2cc(C(=O)N(c3ncc4[nH]cc(I)c4n3)C3CC(N)C3)[nH]c2c1 C#CC1(O)CCN(C(=O)CN(C(c2cnnn2CC)=O)C2CC2)C1 C(C)(C(=O)NCC12CC(NC(C3CCN(C)C(=O)N3)=O)(C1)C2)(C(C)C)OCC N1(C(CC#N)=O)CCC2(CCCC2NC(c2cc(Br)ccn2)=O)C1 CN1CCC(C(N2CCCC2CCNC(=O)CCOc2ccccc2Cl)=O)C1=O C1(C(N2C(CC)COCC2)=O)C2CCN(C(c3coc(OC)n3)=O)CC12 Cc1ccc(C(=O)NCC(CNC(=O)Cc2sc(C3CC3)nc2C)CO)cc1F c1(C(N(C)CCNC(C2(C)CC2F)=O)=O)ccc2cc(O)ccc2c1 c1(C(N2CC(O)(CCNC(c3c(CC)nc(C)s3)=O)C2)=O)cnc(O)c(OC)c1 C1(CNC(C(C)OCCOC)=O)CCC(N(C(=O)C=CBr)C)CC1 O=C1CCC(C(=O)N2CC3CC2CN(C(c2cc4n(n2)CCCN4)=O)C3)=NN1 C1(OC)CC(NC(=O)CC2(C)CC2)CN(C(=O)COc2cccc(C(C)=O)c2)C1 C1(C(=O)NCC(=O)OCC)CC12CCN(Cc1cc(OCC)c(C#N)cc1)CC2 c1(CNC(NCc2cccc(COC)c2)=NCCOCC)cc(Cl)c(Cl)cc1Cl c1(OC)cccc(C(=O)NC(C)(C)CN(C(=O)C(C)OCC(F)(F)F)C)c1C Cc1c(C(N2CC3CC2CC3NC(C2CCOC(C)(C)C2)=O)=O)ccc(F)c1F C1(CC(=O)NC2C3CN(C(Cc4n(C)ncc4)=O)C2C3)CCn2cncc2C1 CCC(C)C(C(=O)N(C)CC1CCCN1C(=O)C=C1CCC1)N(C)C c1(C(=O)NC2CCCC(NC(C3CC(N(C)C)C3)=O)C2)cnc(Cl)cc1N N1(C(Cn2c(C)cc(C)n2)=O)CC(CC(N2CCC(N3CCCC3)C2)=O)C2(CC2)C1 Cc1ccc(CCC(N2CCC3CCC23CNC(=O)CCC(C)(C)C)=O)cc1C c1(CC2C(OC(c3nc(CO)no3)C)C2)ccc(Br)cc1 N1(C(c2c(C)[nH]cc2)=O)CCCCC12CC(NC(C1CC(C(C)C)C1(C)C)=O)C2 CC1CC(C(=O)NC2CC3CC2N(C(c2cnc(O)n2C)=O)C3)=NO1 Cc1cc(C(=O)NC2CC(O)CN(C(=O)CCS(C)(=O)=O)C2)c2ncccc2c1 N1(Cc2c(N(C)C)cncc2)CC2(COC(CS)C2)C1.Cc1nc[nH]c1CCN C1(N(C(=O)CC2(OC)CCC2)CC)CCN(C(=O)CN(c2nccn2C)C(N)=O)C1 N1(C(c2nc(CNC(C(CC)N(C)C)=O)oc2)=O)CCC(NC)CC1 N1(C(C(c2c(C)cccc2)C)=O)CC(NC(=O)CN2CCCCCC2)CCC1C Cc1ccc2nc(C(=O)NCC3CCN3C(C3COCCN3C)=O)c(N)n2c1 C12(C(N3CC(CC(C)NC(c4c(C)n[nH]c4)=O)C3)=O)CCC(O)(CC1)CC2 C1(NS(CC)(=O)=O)CCCC1(C)O.C1CS(=O)(=O)N1.CC c1(OC)cnc(F)cc1C(=O)NCC1COCCN1C(c1csc(Cl)n1)=O N#Cc1ccc(NC2CCCC2CCF)cc1 c1(OC)cccc2cc(C(=O)NC(C)CCCNC(c3cnco3)=O)oc12 c1(CN2CCC(C)(C(=O)NC(c3ccc(Br)cn3)C)C2)cccc(Br)c1F C(N=c1[nH]c(Cl)ncc1Cl)C1OCCCN(C(C2(C)CCC(=O)NC2)=O)C1 c1(C(=O)NCC23C(CN(C(C4ON=C(C)C4)=O)C2)C3)nc(O)nc(O)c1N N1(C(CCN(CCCO)C(c2cnn(C=C)c2N)=O)=O)CC2(COC(=O)N2C)C1 C(CC(=O)N(C(C)C(C)SC(C)C)C)N(C(=O)C(C)c1cc[nH]n1)CC(C)C CC1CC(C(=O)NCC2(C(N)=O)CN(C(C3(N4CCCC4)CC3)=O)C2)=NO1 Cc1cc(C(N2CC(NC(C3CCC4CC3C4(C)C)=O)C2)=O)c(N)c(C)c1 CC(C)CC(O)C(=O)N1CCC(C(N2CCC(c3cnco3)C2)=O)C1(C)C O=C(C1=CCS(=O)(=O)C1)NC1C2CC1N(C(=O)CC1CCC(=O)N1)C2 C(=O)(C(C)CC#N)N1CC(OCC#C)C1.C12(C)CN(C1)C(=O)CC2 C(=O)(C(C)CC(C)(F)F)N1CC(CCOC)N(C(c2nnc(S)n2C)=O)CC1 C1(NC(C2N(C)CCC2)=O)CCC12CN(C(=O)C(F)(F)c1ccccn1)C2 C1(OC)CC(C(=O)NC(C)(C)CNC(c2csc(C(N)=O)n2)=O)CC1OC c1(C2CCN(C(c3c(OCC)c(Cl)ccc3)=O)CC2)nc2c([nH]1)CCCC2 C#CCCCCCCCC(=O)NC1CCCN(C(=O)CC(C)(C)COC(C)=O)C1 N1(CC)CCCC1CNC(=O)NCC(C)(O)Cn1cc(Br)cn1 C=CC1OCCC1C(=O)NCC1(C(N)=O)CN(C(=O)C(c2cnn(C)c2)C)C1 C(=O)(C(CN=[N+]=[N-])NC(=O)CCNC(=O)CNC(C)=O)NCC#C C=CC(CC)CC(=O)NCCC1CN(C(c2ccc(C3CC3)c(F)c2)=O)CCO1 N1(Cc2ccc(C3(C)OCCO3)cc2)CC2CC1CN2CC(F)F N1(C(c2cccc(OC)n2)=O)CC(NC(C2CC2(Cl)Cl)=O)CCC1C C=CCN(OC)C(=O)C1c2c[nH]nc2CN1C(c1cccc(O)c1F)=O c1(C(=O)NCC2CCN(C(C3C(CC)C3)=O)C2(C)C)cc(OC)c(F)cc1N C12(C(=O)NC3CCC(N(C(CC(C)(C)OC)=O)C)CC3)CC3CC1C2C3(F)F c1(CNC(=O)CN(C2(SC)CC2)CC(=O)C2CC2)ccc(NC(C2CC2)=O)cc1 Cn1cc(C(=O)NC2(c3ccccc3)CN(Cc3ccc(N)cc3F)C2)ncc1=O c1(C(=O)NC2(CNC(C(C)CC3CC3)=O)CCOC2)ccc(P(C)(C)=O)o1 c1(N(C2CC3CNC2C3)C(Cc2scc(C)c2)=O)ccc2[nH]c(C)c(C)c2c1 c1(C(N2C(CNC(CCC3N(C)CCC3)=O)CCC2)=O)c(F)ccc2ccoc12 C1(C(=O)NCC(CC(=O)NC(CC=C)CO)OC)CC(=O)N(OC)C1 c1(OCC)cc(C=CC(N2CCN(C(C3CC34CC4(F)F)=O)CC2)=O)ccc1O c1(C(=O)NCC(CNC(C(C)(O)c2ccccn2)=O)O)ccn(O)c(=O)c1 c1(C(=O)NC(C2N(C(C3OCCC(C)C3)=O)CCC2)C)n[nH]c2c1COC2 CC(F)(F)C(F)C(=O)NC(CC1CCCC1)C(=O)NC1COC(=O)C1 C1(N(C(c2cnc(CC)nc2)=O)C)CN(C(=O)Cc2sc(C)nc2C)CC1(C)C N1(C(C(CCC)OCC)=O)CC(NC(=O)CC2CC(N(C)C)C2)CCC(O)C1 C(=O)(CCCCCN=[N+]=[N-])N(C(C)C(N1CCC(CN(C)C)C1)=O)CC C#CC1(NC(=O)C(F)C(C)CNC(=O)CCc2nccs2)CCCCC1 C1(CC(=O)NCC(C)CNC(=O)C(C)(Cl)Cl)CCCC(=O)N1 c1(OC)cc(C)ccc1C(=O)NCc1ccccc1CNC(=O)C(C)CF C(=O)(C1=CCCOCC1)CCNC(C12OC(C)C(C1)C2)=O.C12CN(C1)O2 Cc1cc(C(=O)NC(CO)C(C)NC(c2ccnc(C(F)(F)F)c2)=O)cc(C)n1 CC1(C)CC(C(N2CC(C)(C)C2C2CC2)=O)CN(C(C2CCOCC2)=O)C1 Cn1nc(Cl)cc1C(=O)NC1(CO)CCN(C(c2ccnn2C(C)(C)C)=O)C1 c1(C(N2C(Cn3cc(C(COC)(C)O)nn3)CC2)=O)ccc2ccn(CC)c2c1 N1(C(C(C)N(C(c2c(C)c(C#N)[nH]c2)=O)C)=O)CCC2(CC1)CC2C#N c1(C(=O)NCC2C(C)CCN2C(c2ccccc2Cl)=O)ccc2c(n1)CCC2 c1(C(=O)NC2CCCC(NC(c3cncc(SC)c3)=O)C2)cc2c[nH]cnc-2n1 N1(C(C(C)C)=O)CC(C)C(NC(=O)COC2(C)CCCC2)C(C)C1 C1(CNC(c2n(CC)ncc2Br)=O)CC2(CC2)CN1C(=O)CSC(C)C c1(C(C)C)n[nH]c(=NC(CNC(=O)C2CSc3ncccc32)C2CC2)o1 C1(NC(C2CC3C=CC2CC3)=O)CN(C(C2C=CCC2)=O)CCC12CCOCC2 C1(NC(CC=CC=C)=O)CCCN(C(c2ccnc3ccsc23)=O)CC1F n1(C(CC=C)CC)cnc2c(N3CCOC4CCCCC34)ncnc12 C1(NC(C(CC)NC(C)=O)=O)CCC(NC(=O)C(C)(C)C)C(O)C1 c1(C(=O)NC2(C3CCN(C(C4C(C(=O)OC)C4)=O)CC3)COC2)cc2c(s1)CCC2 N1(C(c2c(N)cc(Cl)cc2)=O)CCCC2(NC(C3CC(O)C3)=O)CCCC12 C#Cc1cnn(CC(=O)NCC2(F)CCN(C(=O)CN3CCC(C)CC3)C2)c1 c1(CC)ncnc(N2CCCC(NC(c3cnn[nH]3)=O)C2C)c1F N(C1CN(C(c2cc[nH]n2)=O)Cc2ccccc21)C(C(c1cc(C)sc1)(C)C)=O C12(C(N3CCN(CC=CC)CC3)=O)CC(CO)(CN1C(=O)C(C)(O)C(C)C)C2 N1(C(CC(C)(C)C)=O)CC2CN(C(c3ccccc3Cl)=O)C2C1 c1(C(N2CCC(CNC(c3ncc(C)c(Cl)c3)=O)C2)=O)cnc2c(C)cccn12 C1(C(=O)NCCc2cnc[nH]2)CN(C(c2ccoc2)=O)CC1O c1(N(c2ccc(C)cn2)C2C(C(=O)OC)CC2)c(N(C(C)(C)C)CC)cnn1C CN1CC(NC(C2(F)CCCN(C(c3cccnc3S)=O)C2)=O)C2(CC2)C1=O C1(C(N(c2ccsc2)C)=O)CCN(C(=O)C=CC(C)(C)C)C(C)(C)C1 c1(C(=O)NC(CCN(C(C(CC)NC(N)=O)=O)C)C(C)C)nccc2cc[nH]c12 C1(NC(C(N2CCN(C)CC2)C)=O)CN(C(c2cc[nH]c(=N)c2)=O)CCC1C c1(OC)ccc(Br)c(CC(N2CC(O)CC2C(=O)NCC2(OC)CCCC2)=O)c1 C(=O)(CC(CC)CCCC)N1CCC(C=C)(C(=O)NCC2(C)CC(C)(C)C2)C1 CCC(C)(C)CCCC(=O)NC(C)(C)CCNC(=O)C=CS(C)=O N1(C(CC2(CC)CCC2)=O)CCCC1CN(C1CC1)CC1CC=CC1 CCN=C(NCc1ccccc1CN1CCOCC1)NC1CCN(S(C)(=O)=O)C1 N1(C(N2CCN(C(c3c(C)cccc3)=O)CC2)=O)CCCC2(CCC(O)C2)C1 C1(C(=O)OC(C)(C)C)CCC(C(C)(C)C)C1.C(=O)(C(=O)N)N(C)CCNC C1(C)(C(N2CC3(CN(C(c4cc(SC)c(C)o4)=O)C3)C2)=O)C2CCC(C2)C1(C)C CCC(CC)C(F)C(=O)NC1CCCC1(C)CN(C)C(c1csc(F)c1)=O N1(C(c2cccc(C)c2O)=O)CC2COCC(C1)C2NC(C1CCCN1N=O)=O c1(OC)cccc(I)c1C(N1CCC12CN(C(c1cccn1C)=O)C2)=O N1(C(c2ncn(C)c2)=O)CCOCC(F)(CNC(=O)Cc2cc(C3CC3)no2)C1 Cc1nn(C)cc1C(C)C(=O)NC(C)C(CO)NC(=O)CC1(O)CCOCC1 C1(C(=O)NC2CC(CNC(=O)C(c3ccccc3Cl)C)C2)(CC)CCNC1=O S(=O)(=O)(c1nc(N2CCCC(C(C)C)C2)ccc1Br)N1CCCC(SC)C1 C1(NC(C(C#C)(C)C)=O)CCN(C(c2ccc(=O)oc2)=O)CC1O N1(C(COc2c(C)cccc2)C)CCC(NC(C2CCC3CC3C2)=O)CC1C CCC(CC)C(C(=O)NCC12COC(CNC(=O)C(C(O)CC)OC)(C1)C2)OC N1(C(CCC=CC)=O)CCCCC1CCN(C(=O)COCC(N1CCCC1)C)C CCC(C)(C#N)C(=O)NCC1CCN(C(c2ccc(=O)n(CCOC)c2)=O)C1 c1(C(C(=O)NC2CC(NC(C3(O)CC3)=O)C2)OC)ccc(O)cc1 CCC(F)(F)C(=O)NC1CCCC(N(C)C(c2cnc(C)cn2)=O)C1 N1(C(C2CN(C(C3CCC(OC(F)(F)F)C3)=O)C2)=O)CCN(C2CCCC2)CC1 C(CC(F)F)(C(=O)NCC(CC1CC1)OC)N(C(c1cnc(C(C)C)o1)=O)C Cn1[nH]nnc1=NC1CCCC(NC(C2CCC3(CCC3)O2)=O)C1 CC(C)(C)C(CO)C(=O)NCC1(O)CCN(C(c2ccc(S(N)(=O)=O)s2)=O)C1 N1(C(CC(C)SC)=O)CC2(CO)CC1(C(=O)NCC1(C)CCCC1O)C2 C(=O)(C1OCCc2ccccc21)NC(C)CCNC(C1CC2(C1)CC2(F)F)=O N1(C(=O)OC(C)(C)C)CCC2CC(NC(c3nc4ccccn4n3)=O)CCC2C1 Cc1cc(C)nc(SCC(N2CC=C(CNC(=O)CC(=O)NC(C)C)CC2)=O)n1 C1(CNC(C2CCN(CC)C2)=O)CCN(C(=O)Cc2cc[nH]n2)C(C)C1 C#Cc1ccc(F)cc1C(=O)NC1CCN(C(=O)Cc2cncn2C)CC1 c1(C(N2CC(C)CC(NC(C3(CC=C)CCC3)=O)C2)=O)cc2ccccc2nn1 CCCCCC(CC)C(=O)N1CCC(OCCNC(C23CC(F)(C2)C3)=O)CC1 c1(C(N(C2CN(C(C3(CCC)CCC3)=O)C2)C)=O)cc[nH]c(=N)c1[N+](=O)[O-] c1(NCC2CC(NC(CC)=O)C2(C)C)nc(C)ccc1C#N.N12CCC(C1)C2=O c1(C(=O)NCC(CCCC)NC(=O)C=C(Cl)Cl)c(F)ccc(OCC)c1F c1(C(=O)NC(CN(C(=O)CC2(C#N)CCC2)CC)C)ncc(N)cc1C C1(CC(=O)NCC2ON=C(C)C2)CN(C(c2oc(C)nc2C)=O)C(C)(C)C1 N1(C(C(F)=CC)=O)C(C)CC2CN(C(c3ccnn3C3CC3(F)F)=O)CC12 c1(CCC(=O)NC(CC)(C)CNC(c2cc(C)cnc2C)=O)nccc(OC)c1C Cc1cccc(C(CNC(=O)C(O)C2CC2)NC(=O)CCCc2cnn[nH]2)c1 C(C)(C(=O)N(CCC)CC1CC1)N(C(C=CCOC)=O)C(C)C.C1CC1 C1(C(N2CC(C(C)C)N(C(C3CC(C)(C)C3)=O)CC2)=O)CCOCC12CCCC2 Cc1cc(C(C)C(=O)NCC2(O)CN(C(C3C(C(=O)N(C)C)C3)=O)C2)c(C)o1 Cc1noc2ncnc(NCC3CN(C(=O)Cc4cnn(C)c4)CCC3C)c12 c1(C(N2CCC(NC(c3c(CC)noc3)=O)C(CO)C2)=O)ccc2nonc2c1 CC1(C(=O)NCC2CC3(CO2)CN(C(=O)Cn2cnnn2)C3)CCCNS1(=O)=O c1(C(=O)NC2CC(C)(C)CN(c3nnc(O)s3)C2)coc2c1C(O)CCC2 CC(C(F)(F)F)NC(=O)C(Cc1cn[nH]c1)NC(=O)CC1CCCOC1 N1(C(c2c(C)nn(C(C)C)c2C)=O)CC2COCCC2(NC(=O)C(O)C(F)F)C1 c1(C(C)=O)ccc(C(=O)NC(C(C)NC(C2(CC(F)F)CCC2)=O)C(C)C)nc1 C(=O)(C#CC(C)(C)CNC(c1ccc(F)c(F)c1)=O)NCC(CC(C)C)O c1(C(N2C(CNC(c3c(C)c(Br)cnc3)=O)CCC2)=O)nc2cccnc2s1 C1(CNC(CC(CC)OC)=O)CCCN(C(=O)C(F)(F)C2(O)CCCC2)CC1 N1(C(c2nc(C)sc2)=O)C2CCC1C(NC(c1cn(C)nc1C(F)F)=O)C2 C1(CNC(CC2(C(=C)F)CCC2)=O)CCN(C(C2CC=CC2)=O)CC1(F)F c1(SC(C)C(=O)N(CCN(C(c2cscn2)=O)C2CC2)C(C)C)ccccc1 C1(NC(CC(=C=C)C)=O)C2CC1N(C(=O)C=CCN1CCCC1)C2C c1(C(N2CCC(C)(NC(C(C)Sc3nncn3C)=O)C2)=O)ccnc2c1CCO2 C1(NC(c2cncs2)=O)CN(Cc2cccc(-c3ccsc3)c2)CC1F C1(NC(=O)OC(C)(C)C)CCc2nc(C(=O)NCC34CCCC3CCC4)cn2C1 C1(C(N(C2(C(=O)OC)CC2)C)=O)COCCN(C(=O)C(O)C2CC2)C1 C(CNC(c1cc(C)c(Cl)s1)=O)(CC(C)C)NC(COCCCC#C)=O C(=O)(CCCC(C)(C)C)NC(CCC)CC(=O)N(CC(O)CO)CC n1(CCOCC)nnnc1C(CCC1CCOC1)NCCc1ccccn1 CC1(F)CN(C(=O)C(F)(F)C(O)C2CC2)CCN(c2ncnc3c2COC3)C1 Cc1nc(C(=O)NCC2CCC(NC(c3ccc(CO)o3)=O)C2)ccc1C#N c1(CC(=O)NC(c2nccn2-c2ccccc2)CC)cc(OC)cc(Cl)c1 c1(C(=O)NC2C(C)CN(C(=O)CC(C)(F)F)CC2)ccc2ccccc2c1O n1(CC(CC)CC)nc(-c2ccn(C)n2)nc1-c1cnc(C(C)(C)C)o1 CN1CC2CC1CN2C(C1CC(O)CN1C(c1ccc[n+]([O-])c1)=O)=O CCCC(C)(CCC)C(=O)NCC(O)CCNC(=O)C(C(C)C)OCC(C)C C(=O)(C#CC1CCCN1C(=O)OC(C)(C)C)NC(c1cnc(C)c(CCO)c1)C C1(CC(=O)Nc2cccc(CO)n2)CN(C(c2csc(Cl)c2)=O)CCO1 C1(C(N(CC(C)NC(c2ncc(F)cc2F)=O)CC)=O)CCCCN(C)C1=O Cc1ccc(O)c(C(=O)NCc2cc[nH]c2C(N2CCOCC2CC(C)C)=O)c1 N1(C(C2(c3ccc(NC)cc3)CC2)=O)C2CCC1CC(NCCN1CC=CC1)C2 CCCCCCCCCC(=O)N1CCCN(C(c2c(Cl)nsc2Cl)=O)CCC1 C(=O)(CCCCC(=O)N1CCC(C(=O)NC(c2nccs2)C)C(O)C1)OC Cn1nnc2c1C(C(=O)NC(CNC(=O)C(F)(F)C1CC1)C1CC1)CCC2 C(C1COc2ccccc21)n1cc(CCCN(C(=O)C(C(C)(C)C)N(C)C)C)nn1 O=S(=O)(c1cnc2ccsc2c1)N1CC(n2cnnc2)C1 N1(C(C(CSC)OC)=O)CCOCC(CNC(=O)C=Cc2sccc2C)C1 C(CC(C(C)(C)C)NC(=O)CC1CCCCC1)N(C(CC(C)C1CCCO1)=O)C C(=O)(N1CCCCCO1)C1CC2(CC(NC(Cc3ccc(C)nc3)=O)C2)C1 N1(OC(N2CC(C3CC(CNC(C(C)(C)C)=O)C3)C2)=O)CC(S(N)(=O)=O)CC1(C)C c1(C(N2C(CNC(C3C(c4ccc(C)o4)C3)=O)CC2)=O)ccc2c(n1)CCOC2 C1(NC(Cn2ccc(C)n2)=O)CCC(CNCc2nccc(C(F)(F)F)n2)CC1 c1(CC)cnn2c(NC(C)C)cc(Cl)nc12.c1(C(C)SC)cccc(C#N)c1 C(=O)(C1CCc2cc(Cl)ccc21)NC1C(NC(CCC(=C)C)=O)COC1 c1(C(=O)NCC(CC(C)C)(C)NC(c2cnsc2)=O)ccc2cc[nH]c2c1F Cc1nc(C(N2CC=CC(NC(c3ncn4c3CCC4)=O)C2)=O)ccc1[N+](=O)[O-] c1(NCC)ccc(C(=O)NC(C)(C)C(C)NC(=O)CCCOCC)cc1[N+](=O)[O-] C1(C(=O)NCCCCC)CCCCN1C(=O)C(C)NC(c1ccc(C#N)s1)=O c1(C(=O)NC2CC(F)(CNC(c3cnc[nH]3)=O)C2)cnc(O)o1 C(=O)(C(S(C)(=O)=O)C1CC1)N1CC2C(N(C(CC(=C)C)=O)C)C2C1 c1(C(N2CCC(CN(C)C(C3CCO3)=O)C2)=O)cc2oc(Br)cc2[nH]1 C1(C(=O)NC2(CC)CCCCC2)CN(C(=O)C(C)CCOC)CC12CCC2 c1(C(N2CCCC(CNC(CC=CC=C)=O)C2)=O)ccc(O)c(Br)c1 c1(N(CCC)C(=O)NCc2nc(Br)cs2)ccnc(Cl)c1OC N1(C(C2C(C)C3CCC2C3)=O)CCC2(CCN(C(C3CCC(F)(F)C3)=O)C2)C1 C1(N(C(CC2(COC)CC2)=O)Cc2ccc(Cl)s2)CCC2(CCNCC2)CC1 c1(CCN(CC(F)F)C(=O)NC(CC=C)C)ccccc1 N1(C(C2(N(C)C)CCCOC2)=O)CC2OCC(NC(C3CCC(O)C3)=O)C2C1 N1(C(c2cc(OC)c(C)cc2)=O)CCOCC(F)(CNC(c2occc2C)=O)C1 C1(c2onc(-c3ccc(SC(C)(C)C)cc3)n2)CC2CCC1N2NC(=O)OC c1(CCC)nc(-c2ccc(OCc3ncccn3)cc2)n(C2CCOC2C)n1 C(=O)(C1COc2ccc(Cl)cc21)NC(C1CCCN1C(C1CCCC1)=O)C C1(C(N2C(CC(N3CC4CC(CO)(C4)C3)=O)CC(O)C2)=O)Cc2nccn2C1 C1(C(=O)OC)(NC(CCc2cccc(CC)c2)=O)CC(O)C1(C)C C(CC(CC)C(=O)NC(C(=O)NCC1CC1c1ccccc1)C1(C)CC1)=CC c1(NC(=O)NCCC(CS(C)(=O)=O)O)ccc2c(c1)CCN2Cc1ccccc1 c1(OC)ccc(Cl)c(C(=O)N(C2CCC(NC(c3n[nH]cc3OC)=O)CC2)C)c1 O=C(C1CCCc2nc[nH]c21)N1CC2(CCCN(C(c3cnc(C4CC4)[nH]3)=O)C2)C1 N1(C(C2C(CNC(C(c3ccn(C)n3)C)=O)CCC2)=O)CCC12CC(C)(CO)C2 c1(OCC)cc(CNC(=O)C(c2ccc(Cl)cc2)Cc2ccccn2)cc(O)c1 CC1(NC(=O)CSCCCCl)CCCCC1C(=O)NCCC12CCCC1C2 C(=O)(C(F)CCC(C)C)N1CC(NC(C(CC)(C)OC)=O)C2(C1)CC2 C(CC(O)C(=O)NCC1C(CO)C1(F)F)NC(=O)CCc1cscn1 NC1CCN(Cc2ccc(C(=O)NCCc3n[nH]c(O)n3)cc2)CC1 N1(C(C2N=C(C)SC2)=O)CCC(NC(c2ccc(C)c(CO)c2)=O)CC1C c1(CNC(C(CC)C(C)C)=O)n[nH]c2c1CN(C(C1CCCCC(=O)N1)=O)CC2 n1(CCC(=O)NC(C(C)(C)NC(c2cc(CC)on2)=O)C)ncn(C)c1=O c1(C(N2C3CN(Cc4c(C)nn(C)c4C)CC32)=O)ccc(C#N)cc1F C1(C(=O)NCC2N(C(C3C(C)C3)=O)CCC2)Cc2ccccc2C1 C(C(F)(F)C(=O)NCC(C1CCCN1C(c1ncc[nH]c1=O)=O)(C)C)N(C)C C1(CC(=O)N(C2CCN(C(c3c(COC)ccs3)=O)C2)C)CC(O)C1(C)C c1(NC(C2COCCC2N)=O)cccc2c(-c3cn(CC(O)CO)nn3)n[nH]c12 N1(C(CC(CC)C(F)F)=O)CCC2(CCC2)C(NC(c2cc(CO)oc2C)=O)C1 N1(C(CSC(C)C)=O)CCCN(C(=O)COc2ccc(C(C)(C)C)cc2)CC1C c1(CC(=O)NCCCN(C(c2ccc(C(F)F)s2)=O)CC)ccnc(Cl)c1 N1(C(CCN(CC#C)C)=O)CCC(C)C(NC(=O)C(C)OCC(C)C)C1C N1(C(c2c(C(C)=O)nccc2)=O)CC2(C)CN(CCn3ncnn3)CC2(C)C1 C12(O)CCN(CC1)C(=O)OC1CCN(C1)C2C(=O)NC.C(C)(C)(C)OC(=O)NC N1(C(C2CC3(CCOC3)C2)=O)CCN(CC2CC2)CC1CC(F)(F)F c1(C(N(CC(CNC(C2(C=C)CCC2)=O)O)C)=O)cc2n(n1)CCCO2 C1(C(=O)NCC#CCOC)CC2CCC1N(C(C1CC(C)C1)=O)C2 C1N=C2C=C(N=CN2)N2CCC(CC2)C2COC(=O)N12.O=C1NC(=O)C(CO)N1 c1(C(=O)NC2C(NC(Cc3ncc(CC)[nH]3)=O)CCC2)ccc(OC2CC2)nc1 c1(C(N(CCCNC(C2CCN(C)C2)=O)CC)=O)cc([N+](=O)[O-])c(C)cc1Cl c1(NCC(=O)NC2Cc3c(nc(C)s3)CC2)[nH]c(=NCC(C)(C)F)nc2sccc12 Cc1ccn(C)c1C(N1CCC1Cn1cc(C2CCCC2)nn1)=O CC1(NC(C2CCC(C(F)(F)F)CC2)=O)CCN(C(c2cnc(F)cn2)=O)C1 N1(C(C2(COC)CCC2)=O)CCC(C(F)F)(CNC(=O)Cn2ncc(Cl)c2C)C1 N1(C(c2n(CCC)nc(C)c2)=O)CC=C(CNC(=O)C(O)C2CC2)CC1 C(=O)(C(C(C)CC)NC(C1CCC(C)(C)CC1)=O)N(C1CCCCC1)CCC N1(C(C(CN(C)C)O)=O)CCOC2(C1)CN(C(C1CCN1S(C)(=O)=O)=O)C2 C#CCC(CC(F)F)C(=O)NC(CC)C(=O)N(CC(C1CCC1)OC)C C1(CN(C(=O)C=CC2CCCC2)C)CN(C(=O)CC2CC(C)(C)C2)CCO1 C=CC(CCC)CC(=O)NC(C)CCN(C)C(c1n[nH]c2c1CCOC2)=O c1(CCSC(C)C(N2CCSCC2)=O)c(F)cc(Br)cc1F N1(C(C2(c3c(C)cccc3)CC2)=O)CC(CNC(=O)C(C)(C)CO)C(F)(F)C1 C1(NC(Cc2n(C)nnc2)=O)CC(NC(=O)C=Cc2ccc(Cl)cc2)C12CCC2 C(CCC(c1ccccc1)NC(=O)C(C)(C)SC)NC(C(C)OC)=O n1(CC)nccc1C=CC(N1CC(NC(=O)CO)CC1C)=O C#CCCC(C(=O)Nc1ccc(F)c(C)c1)NC(=O)CC1(OC)CCC1 C=CC(C)(CCOC)C(=O)N(CC(C)CNC(c1csc([N+](=O)[O-])c1)=O)C c1(OCC)cc(CNc2cc(C(N3CCC(C)(CC)C3)=O)ccn2)cc(Cl)c1 C(CC(=O)NC(c1cncn1C)CO)(C(F)(F)F)NC(C1(COC)CC=CC1)=O CC#CCC(C(=O)N(CCSC)CC)NC(=O)COC1(C)CCC1 C(C)(C(=O)N(CCCNC(=O)C=C(C)C(C)(C)C)CCO)(C(C)C)OCC.CC C(=O)(C(O)CC[S+](C)C)N1CC2C(NC(C3N(C)C(=O)NC3)=O)C2C1 C1(CCNC(=O)C=C(Cl)Cl)CCCN(C(=O)Cc2ccc(O)c(F)c2)CC1 C(=O)(C1=CC2(CN(C(c3ccc(F)s3)=O)C2)OC1)NC(CCC)CCC c1(-c2nc(NC(=O)NC3CC(OCC)C3)sc2)cc(C)ccc1C CCCCCCCC(F)C(=O)N(C)CCNC(c1ccc(OC)nc1)=O c1(C(=O)NCCC(CNC(C(CC=C)C)=O)O)ccc(C(F)F)nc1O N1(C(C(C)SC)=O)CCC2(CCN(C(c3ccccc3CN(C)C)=O)C2)C1 CON(CC1CCCC1)C(=O)C1CCC12c1nnnn1CCN2.S(C)C1CC1 n1(C(C)C)nnc(C(N2CC3CC2C3NC(=O)CCCF)=O)c1C(F)(F)F C1(C(=O)NCC(CC2CC2)C(=O)NC2CC2)CC12CCCC2 C(CCC(O)C(=O)NC1(CN(C)C)CCCC1)NC(CCC=C)=O C1(CNC(Cc2ccn(CC)n2)=O)CCCCN(C(c2cc(N)cc(F)c2)=O)C1 C1(CCC(=O)N(CC(COC)O)C)CCCCN(C(C2CCCC2F)=O)C1 CN1CC(C)(C)CC1C(=O)NCC1C(O)C(O)CN1C(c1ccnn1CCF)=O c1(CC(N2C(C)CC(NC(c3cccc(C)c3Cl)=O)C2)=O)c(F)cccc1C#N CCC(C)CC(CO)NC(=O)CC(C)(C)CNC(=O)C(C)(C)C(=O)N(C)C C12(C(=O)NC(C3N(C(C4OCC(C)C4)=O)CCOC3)C)C3CC(CC13)C2(F)F C=CCCCC(C(=O)NCc1cnc(O)c(F)c1)NC(c1cncn1C(C)C)=O C1(CCC)(NC(=O)CC2CCCOCC2)CCCN(C(=O)CCc2cnc[nH]2)C1 C1(C(=O)NCC2CC(NC(Cc3cccc(C)c3)=O)C2)Cc2nncn2C1 C(=O)(C=C1SCC(=O)N1C)N(CC(C)NC(c1cnnc(Cl)c1)=O)C N1(C(C2C(C#C)C2)=O)CCN(C(c2cc(C)on2)=O)C(CO)C1 C1(C2N(C(c3nc(C(C)=O)sc3)=O)CCC2)CCN(C(=O)COC2CCC2)CC1 N1(C(C2(COC)CCC2)=O)CC2CC1CN2C(c1nc(Br)c(C)s1)=O C12(C(=O)NC3(C(=O)OC)CCCC3)CC(CNCCCC(=O)NCC)(CO1)C2 CN1C(=O)OCC1C(N1CC(n2cc(CNC(=O)C=CC(=O)N(C)C)nn2)C1)=O C1(NC(CN2C(C)CCC2)=O)CN(C(=O)CSCc2csc(=N)[nH]2)C2(CCC2)C1 C1(N)CCCC1NC(CC(=O)N)=O.N1(C(=O)OC(C)(C)C)CCC1CNC=O Cc1nn(C)c(C)c1CCC(N1CCCC(NC(=O)CCOCCN(C)C)C1)=O C(N=c1nc(NC)c2c([nH]1)c(C)nn2C)C1CC(NC(C=C(CCC)CCC)=O)C1 CCC(C(=O)OC)C(=O)NC1(CF)CCN(C(C2(C)CCC(=O)N2)=O)C1 Cc1cc(C(N2CCC(C3CCCN3C(c3cnc(C)n3C)=O)C2)=O)c2[nH]cnc2c1 C1(CCCC(=O)NCC(C)(C)OCC(N2C(CC)CCC2)=O)CCCC(=O)N1 N1(C(C2(C(C)C)CCCC2)=O)CCCC2(CC(NC(=O)C=C3CCC3)C2)C1 C1(NC(c2c(N)cc(Cl)cc2)=O)COC2(C1)CN(C(=O)CCCCC(F)F)C2 CCCCC(CO)NC(=O)C(CCN(C)C)NC(=O)CC1CC(=O)C1 C1(NC(C2(N(C)C)CCCC2)=O)CC2CC1CN(C(=O)CCC(F)(F)F)C2 C1(C(C(=O)NCc2nnc(CC)o2)C)CCN(C(=O)C=CCF)CC1 c1(C(N(CC(O)CNC(=O)CC(C)(C)C#N)C)=O)sc2ncccc2c1Cl C(CC(CC)C(=O)NC(Cn1ccnn1)C(=O)NCC(=O)OCC)=CC C=Cc1cncc(C(N2CC(C(O)C(N3CC(F)(C(=O)OC)C3)=O)C2)=O)c1 C#Cc1ccc(CC(N2CC(CNC(C3CC4(CC4)C3)=O)C3(CC3)C2)=O)cc1 c1(CSc2cc(N3CCOCC3)nc(C)n2)ccc2c(c1)CCC2(C)C C(c1cocn1)=CC(=O)NCC(CNC(C(C)NC(C1CCC1)=O)=O)F n1(CC)nccc1C=CC(=O)NCC1CC(NC(=O)Cn2nnc(C)n2)CC1O N1(C(C(CC)SCC)=O)CCC(C)(C(=O)NC(C)Cc2ccccc2)CC1 C=CCC(C)(CNC(c1cc(CCNC(=O)CCC2CCCCO2)on1)=O)CO c1(C(N2CCC(C(N(C)CC)=O)C2)=O)ccc2c(c1)ncn2C(C)C N1(C(CCC(=O)NC)=O)CCCC(CNC(=O)CC2CCC2)C1C c1(C(C2CCCN2CC2CC2)C)cn(C2CN(C(=O)Cc3ccc(Cl)s3)C2)nn1 Cc1cn[nH]c(=NC(=O)C2=NOC3(CCN(Cc4c(C)nn(C)c4C)C3)C2)c1 C1(C(=O)NCCCN(C(=O)CCSc2ccccc2)CC)CC(=O)NC(C)C1 c1(NC(CN(C(c2ccco2)CC2CCCC2)CC)=O)cccc2nc(O)oc12 c1(C(=O)NCCC(C(C)C)NC(c2ccnc(O)c2)=O)cn2ccc(F)cc2n1 Cc1ccc(C(=O)NCC2(C)CCN(C(C3CC(=O)N(C)C3)=O)C2)c(Cl)c1 C1(C(N2CCC(CC3CCC3)C2)=O)(OC)CC(F)(F)C1.C12CC1CC(=O)N2 C(=O)(CCCC(F)(F)CO)N1CCC(NC(CCCC(=C)C)=O)C(CC)C1 N1(C(C)=O)CCC(CNC(c2nnc3n2CCCC3)=O)C(F)(F)CC1 c1(OC)cccc2cc(CNCC3CCOC(=O)N3)[nH]c12.C(C)(C)(C)OC(C)=O C(CCCCC(=O)N1CCC(CCNC(=O)CSCCC)(OC)CC1)=CCC=C CC1=NN(C)C(=O)C1CC(N1CCCC(O)(CCNC(=O)CC2CC2)C1)=O C1(CCC)CCOCC1(c1nnnn1C1COC1)NCC(C)(C)C1CC1 C#CCC(C(=O)NCC=CCCCCC)NC(=O)CC(O)C1CC1 C1(NC(CC(=O)NCC)=O)CN(C(=O)COc2cccc(Cl)c2)CCC1C C1(CNC(C(CC)Sc2ccccc2)=O)C2CN(C(C3OCCO3)=O)CC12 Cc1sccc1C(=O)NCC1CC1CC(=O)NCC1CCC1(F)F C1(NC(C(=Cc2cn[nH]c2)C)=O)CC(NC(c2nccn2C)=O)CC1O c1(COC)cc(N2CCC(CNC(C3(N4CCCC4)CCCC3)=O)C2)ncn1 c1(C(=O)NC(CCOC)CNC(=O)Cc2cnccc2Cl)cccc(N)c1C C1(NC(CSC(CC)C)=O)CCC(C)N(C(=O)CCNC(N)=O)C1 CC1(C)CN(CC(=O)N(c2ccccc2F)C(=O)Cc2ccccc2)C1=O c1(C(=O)NCC(CC)NC(c2ccc(CO)o2)=O)cccnc1C CCCC(C(O)C(=O)NCC1CCN(C(C)=O)C1)NC(=O)C1=CCCC1 CCCCC(C(=O)N(C)CCNC(c1cccnc1C1CC1)=O)N(C)C [N-]=[N+]=NC1(C(N2CCC2C(N)=O)=O)CCN(C(C2C3COCC23)=O)C1 CC1CC2(CCO1)CC2C(N1CCN(C)CC1CNC(c1ccc(Cl)cc1)=O)=O CCC(F)C(=O)N(C(c1ccccc1)CNC(=O)C=CC(=O)N(CC)CC)C C1(CNC(=O)OC(C)(C)C)CC(n2cccn2)C12CCC2.c1(CNC(=O)N)ccccc1 CN1CCOc2cc(CNC3CCC(C(=O)NCC(O)CO)C3)ccc21 C1(C(=O)NCCC(C)SC)CCN(C(C2CC(CF)C2)=O)C1C C(=O)(C#CC1CCOCC1)NCC(CN(C(C(COC)(C)OC)=O)C)O C1(C(N2CCC(C(C)C(=O)NC(C3CCCOC3)C)CC2)=O)OCCCC1(C)C C1(C(=O)NC(CNC(c2ccc(C)cc2F)=O)(C)C(C)C)CN2CCCC2CO1 C1(C(=O)NCC(C(C)C)C)CC(=O)CN1C(c1c[nH]c(=O)cn1)=O c1(C(=O)Nc2cccc(NC(CC(CCSC)O)=O)c2)cnc(C)c(C#N)c1 C1(C(N2C(C(N)=O)CCC2)=O)CC(=O)NC1(C)C.C1=CC(=O)NC1(C)C N1(C(C(CC)C#N)=O)CCN(C(c2cc(CO)[nH]n2)=O)CC1CCO C(=O)(CCCCCCSC)NC1(CC=C)CCN(C(=O)C(C)CC(=C)C)C1 C(=O)(CC(C)(C)C(C)(F)F)NC1CN(C(COCC(C)C)=O)CC12CC2 N1(C(COCCCCCC)=O)CC(NC(=O)COCCc2cccs2)CC(O)C1 N1(C(C(c2cccs2)NC(=O)CCn2ccnc2)=O)C2CCCC1CC2 c1(OC)ccc(C2(CNC(N3CCOC(CS(N)(=O)=O)C3)=O)CC2)cc1 C1(CNOCCCNC(CNC(C2C(C)C2)=O)=O)CC2CCC(C1)C2 c1(C(CNC(C(C)OC)=O)NC(=O)CN(CC(=O)NC(C)C)C)cccnc1 N1(C(C(CC)C(C)C)=O)CC2(CCC(CNC(C3CC(C)OC(C)C3)=O)O2)C1 C(c1c(C)nn(C)c1Cl)=CC(=O)NCC1CN(C(C(C(CC)C)NC(N)=O)=O)C1 CC1(C)CC(CC2CN(C(c3cc(CO)on3)=O)C2)C1.C1(=O)C(C)(C2(C)CC2)N1 C1(CC(=O)NOC(C2CCC(CC)O2)=O)CCC2(CCN(C(=O)CCC)CC2)O1 c1(C(N2C3CC(NC(C(C(CC)C)O)=O)C2CC3)=O)cccc2c1CCO2 C1(CNC(C2CCN(C)CC2)=O)COCCN(C(=O)CC2CCCO2)C1 c1(C(N2CCC3C(NC(C(C)n4cnnn4)=O)C32)=O)ccc(Cl)c(N)c1Cl C1(NC(N2CCC3(C2)NC(=O)NC3=O)=O)CCNC2(CCS(=O)(=O)CC2)C1 N1(C(C2(NC(c3c(C)c[nH]n3)=O)CCCC2C)=O)CC(C#N)C2(CCC2)C1 C(=O)(C(C)CC(N)=O)N1CC(CNC(C2N(CC)CCC2)=O)C(N(C)C)C1 c1(OC)c(C(N2CCC(O)(C(C)NC(c3c(Cl)cnn3C)=O)C2)=O)ccnc1F CCCC(C)(O)C(=O)NC(C)CC(C)NC(=O)CSc1cnn(C)c1 N=c1[nH]c2ccc(C(N3CCCC(NC(=O)CC4(C(F)F)CC4)C3)=O)cc2s1 c1(CNCC=CC(N)=O)ccccc1.c1(C(=O)NCCC(=O)NCO)ncoc1C1CC1 CC(O)C(C)C(=O)NC1CC(NC(C2(c3ccc(Br)cc3)CCC2)=O)C1 C1(NC(CCc2ncc(C)[nH]2)=O)CN(C(C2CNC(=O)N2)=O)CC12CC2 c12cnc(O)c(c1)N2.C1(C(=O)NCC(=O)OC)CCCN1C(=O)NCCC(C)C C(=O)(C(C(C)(C)C)C1CC1)NCC(c1ccc(F)cc1)NC(C1(COC)CC1)=O S(=O)(=O)(CC(=O)NC1CC(NC(=O)C=CC2CCOC2)CC1O)N(C)C S(=O)(=O)(c1cc(C(=O)O)cc(F)c1F)Nc1c(C)cc(C)nc1C Cc1cc(Br)cc(CN2CCCCC2c2nc(-c3cc(F)cc(F)c3)no2)c1F c1(C(N2CC3(CC(NC(c4ccc(F)nc4)=O)C3)C2)=O)c(F)ccc(Cl)c1Cl c1(-c2nc(C(C)NC3C(C=C)C3)on2)ccc(OC)cc1 C1(NC(C(CCCC)C)=O)CC2CC(C1)N(C(C1CCC(F)C1)=O)C2 C12(C(N(C3CCN(C(c4cc(OC)n[nH]4)=O)C3)CCC)=O)CCCC1(C(N)=O)C2 n1(CC)nnc(C(=O)NCC#CCNC(c2cccc(CCO)c2)=O)c1C C(=O)(C1CCCc2nc[nH]c21)N1CCN(C(c2ccc(C(N)=O)o2)=O)CC1CF Cc1ncc(N)cc1C(=O)NC(CNC(c1cc(C(F)F)no1)=O)C(C)C(C)C N1(C(COCCC)=O)C2CCC1CC(C(=O)NC(c1ncc(C)s1)C)C2 CC1CCCN1CC(=O)NC1CCCC1C(=O)NC(c1ncccn1)(C)C N1(C(c2c(CC)scn2)=O)CCCC2CN(C(C3CC(C)(O)C3)=O)CC12 c1(C(=O)NC(C(C)NC(CCc2cc(C)[nH]n2)=O)(C)C)nc(N(C)C)nc(=N)[nH]1 c1(C(=O)NCC2CC(NC(CC=CC)=O)C(O)C2)cc(C)c(F)cc1Cl C(=O)(C1CCCc2nc[nH]c21)OCC(=O)NC(CO)C(C)NCc1c(C)ncs1 c1(CCOC)ccc(C(=O)NC2CCC(C(=O)NC3(CO)CCCCC3)C2)cc1 N1(C(CCc2n(C)cnc2)=O)C(C(N2CCOC(CC3CC3)C2)=O)CC2CC12 C1(NC(C2CCC(C)O2)=O)CN(C(c2c(Br)cnn2C)=O)CC12CC2 Cc1cc(CC(N2CC(NC(c3c(Cl)csc3Cl)=O)C(C)(C)C2)=O)cc(C)c1 Cc1sc(C)c(C(=O)NC2CCN(C(c3cnn(C)n3)=O)CC2)c1Br N1(C(CC(COC)C)=O)CCC2(CCC2NC(c2cc3n(c2)CCCC3)=O)CC1 N1(C(CCN(C)C(C)C2CC2)=O)CCC2(CCCC2C(=O)O)C1.C1(O)CC2CCC1C2 N1(C(C2CC(C)CN(C(C3C4CC5C(C4)C35)=O)C2)=O)CCCCC(F)(F)C1 CC1CC(C)(C(N2CCN(C)C(CNC(=O)C(C3CCOCC3)O)C2)=O)CCO1 C1(C(N(CCNC(C(CSC)C)=O)CCc2ccccc2)=O)CC12CCOCC2 C1(C(C2CN(C3CCCC3)C2)=O)CC(O)(c2cc[nH]n2)CN1C(c1cccs1)=O C1(NC(c2cn(CC)nc2)=O)CCN(C(C2(C3CCC3)CC2)=O)CC1CO N1(S(c2ccc(C)cc2)(=O)=O)CCC2(CC(=O)NC2=O)C1 c1(C(=O)NC(CC=C)CNC(=O)C=Cc2sccc2C)cnn2ccccc12 C#CCCCCC(=O)NC1CC2CC(NC(=O)CCC(F)(F)F)C2C1 c1(C(=O)NCCc2cc(C(=O)NCCS(CC)=O)no2)ncc(F)cc1C c12cccc3nc([nH]c13)C(C1CC1)CC(=O)N1C(C)C2CCC1.C(=O)(CO)N(C)C C1(C2C(=O)N2)CCN(CCOCCN(CCC(=O)N(C)C)C)C1.CO.SC CCC(C#N)C(=O)NCC1(C)CC(NC(C2CN(CC(F)(F)F)C2)=O)C1 CN1CCN(CC(C)(C)C(=O)N2CCCCC2C(=O)NCCC2CCCC2)CC1 N1(C(CN2C(C)CCC2C)=O)CCCC(O)(CNC(=O)CCC(C)(C)N(C)C)C1 C1(C(=O)NCC2(O)CN(C(C(CC)C)=O)C2)C2CCC1CC2 C12(C(=O)NCC3CC(NC(CN4C(C)CC4)=O)C3)CCC(CC1)OC2 C1(NC(c2cn3cccnc3n2)=O)CCC(N=c2[nH]ccn3ncc(Br)c23)C1 c1(N2C(=O)CC(C(=O)NC(c3ccc(OC)cc3)C(C)O)C2)cccc(C#N)c1 c1(CN2CC(N3CCN(C(=O)NC4(F)CCOCC4)CC3)C2)cccc(Cl)c1Br C1(NC(CCN(C)C)=O)CCCN(C(=O)C(F)(F)Cc2ccc(Br)cc2)C1 c1(C(=O)OC)cc(OC)c(Cl)cc1[N+](=O)[O-].c12cc(cc(OC)c1OC)C(=O)C2 N(C(=NCCF)NCC=CC1CCOCC1)CC(COC)(C)OCCO C1(C(=O)NC(C(C2CC2)OC)C)(N(C(=O)Cc2cc(C)on2)CCO)CC(F)C1 N1(C(CCC2CCN(C)C2)=O)C2CCCC1CC(NC(=O)CCCC1CC1)C2 N1(C(CC=CC=C)=O)CCC12CN(C(c1ccc(-n3nc(C)cc3C)cc1)=O)C2 N1(C(c2cccc(CC)n2)=O)CC(C)CN(C(c2cc(C)ccc2C)=O)CC1C N1(C(Cc2c(C)ncs2)=O)CCC(C)(NC(=O)CCc2cc[nH]n2)CC1 C(CC(CNC(=O)C=Cc1cn[nH]c1)NC(=O)CCCc1nc(C)no1)OC C1(NC(c2c(CCC)n[nH]c2)=O)(CO)CCN(C(=O)Cc2coc(CC3CC3)n2)C1 C1(CNC(CC(=O)OCC)=O)COCCN1C(c1ccccc1O)=O C(CCC(CCC)NC(=O)C(c1cccc(Cl)c1)O)NC(COCCC=C)=O N1(C(C2CCS(=O)(=O)N2)=O)CCCCC(NC(C2(CO)CCCO2)=O)C1 C1(N(C(CCCSC)=O)C)CN(C(=O)C(C)Oc2ccccc2Cl)CC1(C)C C1(N(C(=O)COC2CCCOC2)C)CN(C(c2c[nH]ccc2=O)=O)CCC1(C)C C1(NC(Cc2cccc(SCC)c2)=O)CCN(C(c2nnn(C)c2N)=O)CC1C Cc1ccc(C)c(CNC(C2CN(C(c3ccns3)=O)C2)=O)c1 Cc1cncc(CCNC2CCC(CC(=O)O)C2)c1 C1(NC(=O)Cc2cncnc2)C2CCC(C2)C1C(=O)N(CC(O)CC1CCC1)CC CCCC(C)CC(=O)N(C(c1ccccc1)CNC(c1ncnc(O)c1Cl)=O)C C1(C(=O)NC2(C(=O)NC(C)Cc3ncon3)CSC2)CCC(C)O1 C1(CNC(c2ccc(C#N)cn2)=O)CCC2CN(C(c3nc(Cl)cs3)=O)CC12 N1(C(c2ccc(COC)o2)=O)CCC(CC(=O)NCC2CC(CF)C2)CC1 C(c1ccc(F)cc1)=CC(=O)NC1C2CC(NC(c3cc(Cl)n[nH]3)=O)CC12 Cc1c(NC(C2CCCO2)C2CC2)ncnc1N(C)CCc1ccoc1 CC1CN(C(c2cnc(Cl)s2)=O)CCCN1C(C1CCCCC12CCC2)=O c1(C(=O)NCC2N(C(C(C)OC)=O)CCC(C)C2)cn(C)c(=O)c2ccccc12 c1(C(=O)NC(CNC(c2nc(Br)c[nH]2)=O)CO)cc(O)cc(=O)o1 c1(C(=O)NC(C(C)NC(C(C)(C)OC(C)C)=O)C)cc2cc(Cl)cc(Cl)c2[nH]1 CC(C)(C)C(CNC(C12CCCC1C2(F)F)=O)C(=O)NCc1cc(Cl)no1 c1(C(=O)NCCC2(O)CCN(C(C3N(CC)CC3)=O)C2)ccc(Br)nc1N C(=O)(C(F)CNC(=O)OC(C)(C)C)NC1C(CNC(CCOC)=O)CC1 C(CC(C(=O)NCCCN=[N+]=[N-])NC(=O)C=CC(C)CC)=CC C1(CC(N2CCCC(C(C)NC(c3ccsn3)=O)C2)=O)CCC2(CC1)CC2 C(=O)(CC(C)C(C)C(C)C)NCC(CC(C)C)NC(=O)CC1CCC(O)CC1 c1(NC(C(CCOCCO)NC(C(C)OCC(C)C)=O)=O)ccc(F)nc1F c1(C(=O)NCC(N(C)C(C2(CO)CCCO2)=O)C2CC2)cccnc1N N1(C(CCCCOC)=O)CCCCC2(CCN(C(=O)C(CC(C)C)OC)C2)C1 c1(SNC2CC(NC(C3CC3c3cccc(CSC)c3)=O)C2)cccc2[nH]ccc12 CCC(C)CC(C)C(=O)N1CC(O)(C(C)(C)CNC(c2cncc(N)n2)=O)C1 c1(CCC(=O)NCCN(C(=O)C(n2ccnc2C)C)CCC)c(C)noc1C CC1(C)CCOCCN1Cc1nc(C2CCCCC2)no1 C(=O)(CC(C)CC(C)C)NC1CCC(CC(=O)NC)CC1.C1(CC)(CC)CCCN1 C(CCCNC(=O)COC1CC(NC(C2CC2(F)Cl)=O)C1)C1(C)CC1 C(=O)(C(F)(F)CC1CC1)NC1CC(CNC(C(=C(C)C2CC2)F)=O)C1 c1(C(C(=O)NC2CC(=C3CC3)C2)NC(C=C)=O)cnn(C)c1 CCC(CC)(CCC(=O)NCC(C)(O)CNC(=O)CC(C)CC1CCC1)[N+](=O)[O-] N1(C(c2cccc(CC)n2)=O)CC2(CCNC(=O)C(F)(F)CC)CCC1CC2 N1(Cc2nc(C)sc2)CCC(O)C(C(=O)NCc2noc(C(C)C)n2)C1 c1(C(N2C3C(N(C(CCCSC)=O)C)CC(C3)C2)=O)ccc(F)c2ccncc12 c1(C(=O)NCCC2(NC(C3CSCC(=O)N3)=O)CC2)c(Cl)ccc(F)c1F c1(OC)ncc(C)c(C(=O)NC2CCCN(C(c3cc(Cl)cnc3O)=O)C2)c1Cl C1(NC(c2nc(CC(C)C)oc2)=O)CN(C(=O)Cn2ccc(C3CC3)n2)CC1O N1(C(c2ncc(CC)s2)=O)CCCCC(CNC(=O)CSC(F)(F)F)C1 c1(CCC(=O)N(CC)CC)ccc(OCC)cc1.c1(C=O)ccoc1C(C)(C)C C12(C(N3CCC(C(C)NC(c4cccn4C)=O)CC3)=O)CC=CC(C1)OC2 N1(C(C)C2CC2)C(=O)NC(C)(c2ccc(OCCc3nn[nH]n3)cc2)C1=O N1(C(CN(C2CCCC2)C)=O)CCCCC1C1CCN(C(c2ncoc2)=O)CC1 C#CCC(C)C(=O)N1CCC(CC2(Nc3ncccn3)CC2)C1.n12cc(nn1)C2 Cc1cc(F)c(F)cc1NC(C1CC(F)CN1Cc1cccc(Br)n1)=O C1(C(=O)NCCC(CC)(F)F)CC2(CC(NC(=O)C3=NOC(C)C3)C2)C1 CC#CCC(C(=O)N1CCC(CN(C)CC)C1)NC(=O)C(N1CCNC1=O)C C1(NC(CC(C)C2CC2)=O)CCC12CCN(C(c1ccc(C3CC3)cc1)=O)CC2 N1(C(C=CC)=O)CCC2CCCN(C(c3cc(C)c(F)c(C(=O)OC)c3F)=O)C2C1 c1(C(=O)NC2C(NC(c3nc(C(C)(F)F)sc3)=O)CC2)nccnc1N N1C(N2CCC(c3ccccn3)C2)=NCCNC1=O.CCCCSC(C)(C)C C(=O)(C(C(=O)N1CCC(N(C)C(c2ccc(C(C)(C)C)nc2)=O)C1)OC)OCC c1(C(=O)NC(CC)CNC(=O)C(O)Cc2cnc[nH]2)cc(OC)cc2c1OCC2 c1(C(=O)NC(c2ccoc2)C)coc2c1CN(C(=O)CCc1ccc[nH]1)C2 c1(OC)cc[n+]([O-])c(C(=O)NC(C)(C)C(C)NC(c2coc(C(F)F)n2)=O)c1 c1(N(C(=O)C(C)=CC(C)(C)C)CC)cccc(C#N)c1 C1(C(=O)NC2C=CCC(C(N(C3CCCCC3)CC)=O)C2)CCCC12CCC2 c1(C(=O)NCCC(C(=O)NCCOCCC#C)O)nccc2cc[nH]c12 N1(CC)CCN(CC(N2CCN(CCF)CC2)=O)CC1.N12CC(O)(C1)C2=O CC1(CNCc2cc(F)c(C(F)(F)F)cc2F)CC2(C1)CC2(F)F C(=O)(C(O)C(C)(C)C)N1C(CC(=O)Nc2c(C)n[nH]c2C)COCC1 C(CC(=O)N(CCCO)OC)N(C(C1CC(C)(CC)C1)=O)C c1(C(=O)N(C2(C)CN(C(c3c(C)n(C4CC4)nc3)=O)C2)C2CC2)cc(Cl)nnc1O c1(NC(C(C2CC2)OC)C)cc(C)c(S(=O)(=O)NCCc2ccccc2F)cn1 C12(CNC(C(C)c3cccs3)=O)CCC(CC1)N(C(C1CCN1C)=O)C2 N1(C(CCCOCCOCC)=O)CCN(C(=O)CN2CCC2)CC1CC N1(C(CCOCCOC)=O)CCCN(C(c2ccsc2)=O)C(C)C1 CC1(C)CC(C(=O)NC2CCC(=O)NC2=O)CN1C(c1csc(Cl)c1)=O C(=O)(C1CC=Cc2ccccc21)N1CC(C)(NC(c2ccc(C)c(C)n2)=O)C1 N1(CC)CCN(CC(=O)NCC2CC2NC(C2(C(F)F)CC2)=O)C(=O)C1=O C12(CC(=O)NCC(C(=O)NC34CC(F)(C3)C4)N(C)C)CCC(CC1)C2 n1(CC(N2CC(C(=O)OC(C)(C)C)CC(C)C2)=O)ncc(S(C)(=O)=O)n1 C1(CC#C)(C(N2CCN(C(c3ccnc(C4CC4)n3)=O)CC2)=O)CCCCO1 CC(C)CC(C)(O)C(=O)N1CC2CC(N(C)C(c3ccn(C(F)F)n3)=O)C1C2 CC1(C)CCCCC1N(S(=O)(=O)Cc1cccc(Cl)c1)C c1(CNC(C2(C)CCCN2C(c2ccnc(CO)c2)=O)=O)nc(Cl)ccc1Cl C1(O)(C(C)NC(c2ccc[nH]2)=O)CCN(C(=O)COCC2(F)CC2)C1 Cc1cccc(Cl)c1C(=O)NC1CC(C(C)NC(c2cccn(C)c2=O)=O)C1 C12(C(N(C)CCNC(=O)C(F)CC3CC3)=O)COC(CCO1)C2 c1(C(c2ccc(NC(=O)Nc3ccc(OC)cc3)cc2)=O)cccc2c1OCO2 C#CC1(C(=O)NCC2(CO)CC=CC2)CCN(C(=O)C(N2CCCCC2)C)C1 CCCC(C(=O)NCCC1CCN(C(c2sc(OCC)nc2Cl)=O)C1)OC C(CCC(C)C)(C(=O)N(C)CC1CC(O)C1)NC(c1c(CC)nn(C)c1)=O c1(CC(=O)N(CCCOCCNC(c2c(C)ncs2)=O)C)cncnc1O C1(CNC(CCn2c(C)cc(C)n2)=O)CN(C)CCN1C(c1[nH]cnc1C)=O C(C(C)(C)CNC(=O)CCC1CC1(C)C(F)F)NC(C1CC(C(=O)OC)C1)=O C1(C(=O)N)CCCCC1C1CC1.c1(C(=O)NC)ccc(C(=O)NC2CC(C)C2)cc1 Cc1nn(C)c(C)c1C(=O)NC1CCC(C)(CNC(=O)CC2CCCCCC2)C1 c1(C(N2CC(NC(=O)Cc3ccnc(Br)c3)C(F)C2)=O)cc(F)cc(Br)c1Cl c1(C(=O)NC2CCN(C(C3C(C)CC3)=O)CC2)ccc2nc(O)n(C3CC3)c2c1 CCCC(CCO)NC(C1CCN1C(c1ncsc1NC)=O)=O C1(C(=O)NCC2(O)CCN(C(c3c(C)n(CCO)cc3)=O)C2)CCCC(C)(C)C1 C1(NC(C2C(=C)CC2)=O)CCC(CCNC(=O)COCCC)C1 C12(CCCN(C(=O)Cn3cnnc3)C1)C(=O)N(CC)C2.C1(O)(C)CCC1.OC CC1(C)OCC(N)(Cc2nccc(I)n2)CO1 c1(C(=O)NCCCC(C)NC(c2ccc(CCF)cc2)=O)cc(F)cc(Cl)c1O c1(C=O)sccc1OC(F)F.C1=CCN(C)N(C)C(C2CC2)CNC1=O C(N=c1nc(N2CCC(OC(C)(C)C)CC2)c2c([nH]1)CCC2)c1c(C)occ1 c1(NC(=O)C(C2CCNCC2)O)ccnc(-c2nccs2)n1 N12CC(=O)NC1=CC=CC=C2.CC(C)C(C)CN(C)CCN(C(C)C)CCN(C)C N1(C(C(CCOC)OC)=O)CCC(F)C(NC(=O)Cn2cc(F)ccc2=O)C1 N1(C(=O)NCCSCc2c(NC)cccc2)CC2OCCN(C)C2C1 c1(C(=O)NC(CCC(=O)NC(CC)(C)CNC(C)=O)=O)ccc(F)cc1C C1(CC=C)CCCCC1C(=O)OC.C1(=O)C(C)=CCNC(=O)C2(CC2)N1 O=C(CCCCC1CC1)NCC1CCN1C(C1CC1CF)=O c1(OC)ccc(CN(C)CC2COCC2O)c(C)c1OC c1(C(=O)NCC(C2CC2)NC(c2n(C(C)C)ncc2)=O)ccc(S(C)(=O)=O)cc1 Cc1nc(-c2ccc(Br)cc2)sc1C(=O)NCC(C)NC(=O)C1CC1 n12cnc-1c2.C1(C(=O)NC)(CNC(=O)C(C)OCC2CC2)CCCC1.COC c1(OC)cccc(CN2CC(CO)CC2C(=O)Nc2nc(-c3cccnc3)cs2)n1 c1(OC)cc(NC(=O)CC2CN(C(=O)Cn3cc(Br)ccc3=O)C2)ccc1C c1(N2CC(C)OC(C)C2)ncc(S(=O)(=O)NCC23CC(CN2C)C3)cc1Cl C1(C(=O)NCC2(O)CCN(C(C3CCSC(C)C3)=O)CC2)(CC)CCC(O)CC1 C1(CNC(C(CC)C(=O)OC)=O)CC2CCC1N(C(=O)C1=CCCSC1)C2 C1(NC(C2C(OC)CC2)=O)CC2CN(C(=O)CC3(O)CCCCCC3)CC2C1 c1(C(=O)NC(CCCNC(c2c(SC)snn2)=O)C)cnc2c(F)cccn12 C1(C(N(C(CC)COC)C)=O)CCCN(C(c2cnncc2C)=O)C1 c1(OC)cc(NC(C2CCN(C(=O)C(C)O)CCO2)=O)ccc1F C12(CNC(C3CC(CNC(COCC(=O)NC)=O)C3)=O)CC1COC2(C)C Cc1cc(=O)ccn1CC(=O)NCC(CO)NC(=O)CC(C)c1ccccc1 Cc1cnc(C(=O)NCCC(=O)NC(CO)C(=O)OC2CCCC2)c[n+]1[O-] C(c1ccc(C=O)cc1)=CC(=O)N(CC(=O)OC)C(=O)C=C(C)C C(=O)(CC(O)C(C)CC)N(C(C(=O)NCCOCC(=C)C)C1CC1)C CC(CCCNC(=O)COC(F)(F)F)NC(C1CCCN1C1CC1)=O Cc1nn(C)c(C)c1C(=O)NC1CCC1CNC(=O)C(C)Sc1ccccc1 C(C(O)CC(=O)NC1CC(NC(c2ccc(F)cn2)=O)CC1O)N(C)C N#Cc1ccc(F)c(C(N2CCC(OCC(N3CCC(CCF)C3)=O)C2)=O)c1 c1(C(N(CCNC(C(C)(C)NC(=O)NCC)=O)CC)=O)cc2cccn2cn1 c1(N2CCC(NC(c3cc(OC)cc(Cl)c3)=O)C2)cc(OC)nc(S(C)(=O)=O)n1 C(=O)(C(C(C)C)Sc1ccccc1)N1CC(N(C(COCCCCC)=O)C)C1 C=CCCCC(C(=O)NCCC(C)C(C)C)NC(=O)CC1(OCC)CCC1 C(C(=O)NCC1CCN(C(C2(C3CCCO3)CCC2)=O)C1)(C(C)C)OCC c1(OC)cc([N+](=O)[O-])ccc1NC(=O)COC(=O)C(c1ccncc1C)C C(=O)(C(CNC(=O)C(CC)OC)N(C)C)N(C1CCCCC1)CC#C C(CC(F)F)(C(=O)NC1CCC1)NC(C=CC(=O)NC1CC1c1ccccc1)=O S(=O)(=O)(c1ccc(Cl)c(Cl)c1)N1CC2(CCC(C(=O)Nc3ccccc3O)O2)C1 C(CN(C)C)(CC(C)C)NC(C1C(NC(C2(CC#C)CCCC2)=O)CCC1)=O N1(C(COCC(=O)OC)=O)CC2(CCCC(CNC(c3cc(Br)n[nH]3)=O)O2)C1 c1(OC)nc(Cl)c(C(N2CC(NC(=O)C(c3ccc(Cl)s3)=O)C(C)C2)=O)s1 C1(F)(CNC(C(C)OC(C)(C)C)=O)CCC(NC(=O)C(c2ccc(F)cc2)O)C1 C(=O)(C1CCCn2nccc21)NC1CCC(CNC(C2(C#N)CCOC2)=O)C1 N1(C(C(n2ccc(C)n2)C)=O)CCCC(NC(=O)CCC2CC2(C)C)C1 C(CCC)(C(=O)NC1CC(NC(C2(CN3CCCCC3)CC2)=O)CC1O)=CCC c1(C(=O)NC2C(CNC(C3(CC(C)C)CC3)=O)CCCC2)ccc(Br)c(O)n1 Cc1csc(=O)n1CCNC1CCC1NC(C1(c2ccc(F)cn2)CC1)=O C1(CNC(C2(C)CCCCC2)=O)CN(C(=O)CSc2cccc[n+]2[O-])CC12CC2 c1(CCC(=O)NCC(C2CCC2)NC(CSCCCC)=O)ccnc(C)n1 C1(C(=O)NC(C)CCCNC(=O)CN2CCCC2)COCCOC1 C1(CN2CC(F)(C(=O)NCCC)C2)CCC(C(N)=O)O1 C(=O)(C1CCc2cc(OC)ccc21)N(CCCNC(c1conc1CC)=O)CC C#Cc1ccc(Cl)c(C(N2CCC(O)(C(C)NC(=O)CC=CC(C)(C)C)C2)=O)c1 c1(C(=O)NCC2N(C(c3snc(C)c3N)=O)CC2)cnn2c1CCCC2C c1(OC)cc(CC(=O)NC2CCC(NC(c3ccc(C(C)(C)C)s3)=O)C2)on1 C1(N(C)C)CC2CCC(C1)N2C(C1(NC(=O)CC2CCOC2(C)C)CC1(C)C)=O CC1CCCCC1(CNC(c1cc(C2CCC2)[nH]n1)=O)NC(c1nnn(C)n1)=O c1(C(N(CCCN(C(=O)C=CCN2CCCCC2)C)C)=O)cnc(Cl)s1 c1(C(N(CC(CN(C(=O)C=Cc2cocn2)C)O)C)=O)ccc(F)nc1 C1(NCc2cccc(C)c2)CN(C(C2CC2C2CC2)=O)CC(F)(F)C1 C1(CCC)CN(C(=O)CC2CC(NC(=O)CCSC)C2)CCO1 N1(C(c2n(C)nc(Br)c2)=O)CC2CC1C1CC21 N1(C(c2c(Cl)cc(C)nc2)=O)CC2=C(C1)CN(C(c1sncc1C)=O)C2 Cc1nsc(N(C2CN(C(=O)C=Cc3ccnn3C)C2)CC)c1C(=O)NC1CC1 Cc1ccccc1CCNC(=O)C(CCF)NC(C1CCCSC1)=O CCC(CC)CCC(=O)NCC1(C)CCCCC1C(N1CC(=O)NC2(CC2)C1)=O Cc1cc(-n2cc(CC(C(=O)O)NC(C3CC(C(C)C)NC3=O)=O)nn2)ccn1 CON1CCC2=C(C1=O)C(c1cc3c(cn1)COCC3)NC(=S)N2c1cccnc1 C1(NC(C(C)=Cc2ccccc2)=O)(CNC(c2ccc(C)s2)=O)CCCCC1 c1(C(N2CCC(NC(COCCCC)=O)C2C)=O)cc(F)c(OC)cc1N NS(=O)(=O)c1csc(C(=O)NC(CNC(C2CC(n3cccn3)C2)=O)CO)c1 CCCC(C(=O)Nc1ccc(SC)cc1)NC(c1ccc(CO)cn1)=O N1(C(CCC(C)SC)=O)CCCCC(C(=O)N(CCCC(C)C)C)C1 c1(SCC(=O)NCC2C(NC(Cc3nc(C)[nH]n3)=O)COC2)ccccc1F CCCCC(O)C(=O)NCC12CCC(NC(=O)Cc3coc(C(F)F)n3)(CO1)C2 C1(C(=O)NCc2c(OC(C)C)nsc2)C2CN(C(=O)C=CCOC)CC12 C=Cn1nncc1C(=O)NC1CCC(CNC(=O)CCOCCC)C1 CN1CC2(CC2)CC1C(N1CCC(N2CCC(NC(c3ccon3)=O)C2)CC1)=O c1(OC)nc(C(=O)NCC2CCN(C(c3cc(C)cnn3)=O)C(C)C2)cc(O)n1 CC(C)C(C)CCNC(C1(NC(c2cc[nH]c2)=O)CCOCC1)=O c1(C(N2CCN(C(CS(CC)(=O)=O)=O)CC2C2CC2)=O)c(C)cc(Cl)cc1Cl c1(C(=O)NCCC(CNC(C2CCOC2)=O)OC)cccc(C(N)=O)n1 CN=c1nc(N2CCCc3c(cnn3C)C2)[nH]c(=NC(C)c2scnc2C)[nH]1 Cc1cc(C(F)F)n(CC(=O)N(C(C)CN(C)C(c2nsnc2O)=O)C)n1 N1(C(CC(C)OC)=O)CCC(NC(=O)CCc2cc(C)on2)C12CC2 c1(OC)cc(F)ccc1C(=O)NC(c1ccccc1)C(C)NC(=O)CC(C)(C)O C1(C(N2CCC(CCCNC(CSCCCC)=O)CC2)=O)CC2CCC(C1)N2C C1(C(=O)NC2CC(C)(CNC(C3CCCC3C(N)=O)=O)C2)(OC)CC(C)(C)C1 C1(C)(NC(c2c(C)n(C3CC3)nc2)=O)CCN(C(=O)CC23CCCC2C3)CC1 N1(C(C(c2c(C)n[nH]c2C)C)=O)CCN(C(=O)CCC#N)CC1C(C)C Cc1nn(C)c2ncc(C(=O)NCCC3CC(NC(C45CC(C)C4C5)=O)C3)cc12 N1(C(COCCCN=[N+]=[N-])=O)CCOCC(NC(c2cnn3c2SCC3)=O)C1 C#Cc1ccc(Br)c(C(=O)NCC2CC2NC(c2cnc3cc[nH]c3c2)=O)c1 C1(C)(CNC(C(CC)OC)=O)CN(C(=O)Cc2cc(Cl)cc(Cl)c2)CC1C n1(CC)cc(NC(=O)C(C)(C)CN(C)C(C2CC2CC(C)C)=O)c(C#N)n1 C(c1cccc(Cl)c1Cl)=CC(=O)NC(C1CN(C(C2CCCN2N=O)=O)C1)C c1(C(=O)NC(C(=O)NCc2onc(C)n2)CC2CCC2)cnn(C)c1C N1(C(C(c2cncc(F)c2)C)=O)CCC2(C1)CN(C(c1cnn(C3CC3)c1)=O)C2 N1(C(COCP(C)(C)=O)=O)CC(NC(C2CCC(C)(C)O2)=O)CCC(O)C1 N1(C(c2n(C)ncc2)=O)CC2CCC1CN2C(c1cc(F)cn1C)=O C1(C)(C(=O)NC2C(NC(COCCC(C)C)=O)CCCC2)CCC(F)(F)C1 c1(C(=O)NC(c2ncc(C)o2)C)ccc(OC(C)C)cc1C C1(O)(CNC(C2(CC#C)CCCC2)=O)CCN(C(C2CCN2CC)=O)C1 C1(NC(C2(OCC)CCC2)=O)CN(C(=O)CC2CN(C)CC2O)CC2(CC2)C1 C(=O)(C1CCCc2cncn21)NC1CC2(C(NC(c3cccc[n+]3[O-])=O)C2)C1 Cc1cc(C(=O)NCCCCC(CO)NC(C23CC=CC(C2)OC3)=O)cc(C)n1 N1(C(C)COC(C)(C)C)CCN(C(=O)OCC2CC=CCC2)CC1 CC(C(C)C(=O)N1CCC(CNC(=O)C(C)S(C)(=O)=O)C12CC2)S(C)(=O)=O C1(C2CCN(C(C3CSC3)=O)C2)(NC(c2nc(C)[nH]n2)=O)CC1 C1(C)(C(N(CCCCN(C)C(C2CC3(CC3)C2)=O)C)=O)CCC(O)CC1 C#CCC(CC(=O)NCC(c1cn(C)cn1)O)NC(=O)CC1CCC1COC C1(NC(C(CC)N(CC)CC)=O)CN(C(c2cc(Cl)ccn2)=O)CC1C(F)F C1(C2CCN(C(c3csc4cncn34)=O)C2)(NC(C2CC3CCC2CC3)=O)CC1 C1(CNC(c2cnc(NC(C)=O)o2)=O)CC12CCN(C(C1(CO)COC1)=O)CC2 C1(C)(C(=O)NCC2=CCN(C(C#CC(C)(C)O)=O)CC2)CC(C2CC2)=NO1 C1(NC(C23CC(COC)(OC2)C3)=O)CC2CC(C1)N(C(=O)C(C)CC(F)(F)F)C2 C1(NC(C(CCC)OC)=O)CC2CCC1N(C(=O)C=C1CCN(C)C1)C2 S(=O)(=O)(c1cnccc1N1CCC(C#N)C1)NCCCCCCOCC C#Cc1ccc(C(=O)NC(Cn2cccn2)C(=O)NC(CC)(CC)CC)nc1 c1(C(=O)Nc2scc(CC(=O)Nc3c(Cl)ccnc3Cl)n2)cc(I)ccc1Cl c1(NS(C)(=O)=O)cccc(C(N2CC=CC2CNC(c2cc(CF)on2)=O)=O)c1 c1(CC(=O)CN2CCC(O)(c3cccc(F)c3)CC2)nc2cccnc2[nH]1 Cc1ccc(OCc2nc(C3CC3C)nn2CC(C)(C)C)cc1C C1(C(=O)NC(CC)CNC(c2cccs2)=O)CC(C)CC(=O)N1 c1(N2CCN(CC)CC2)ccc(Cc2cn(CCCC(=O)O)nn2)c(C)c1 C1(CNC(C(C(C)OC)NC(=O)C(C)SC(C)C)=O)NC(=O)OC1(C)C c1(C(=O)NCC(CN(C(=O)COCCCF)C)(C)C)cccc(-n2ccnn2)c1 C#CCC(CC(F)F)C(=O)N1CCCC1C(C)NC(=O)CC1(C=C)CCCC1 c1(OC)c(Cl)cccc1Cl.C12CN(CCO1)CCN(CCCc1ccnc(Cl)c1)C2=O n1(CC)nnc(C)c1C(=O)NCC(c1ccccc1)NC(c1cc(F)n[nH]1)=O C1(C(=O)NC2CC3CN(C(C4(CC(=O)OC)CC4)=O)CC32)CCc2ccnn2C1 C(=O)(C1CCc2cccnc21)N1CC2C(CNC(C(C)(C)c3ccsc3)=O)(C2)C1 CC1CN(C(=O)OC(C)(C)C)C1CNC(=O)NCCC1CC1(C)C c1(C(=O)NCC2C(CC(=O)N(CCOC)CC3CCC3)C2)ccc(C)o1 CC(C(=O)N1CC(O)(CNC(C2CCCCN2C)=O)C1)C(C)(C)C C(=O)(CCS(=O)(=O)C(F)(F)F)N1C(CNC(=O)CSc2ccc[nH]2)CC(OC)C1 C1(C(=O)NCC(C)NC(C2(O)CC(C)(C)C2)=O)CCc2nc(C3CC3)ncc2C1 c1(C(=O)Nc2c(C)c(CO)ccc2)cc(C#N)ccc1O.C12CC(C1)CC(=O)N2 C(C1c2ccsc2CCN1C(=O)COC(F)F)NC(CC(C)(C)CC(F)F)=O C=CCC(C(=O)NC1CCCN1CCC)NC(C1CCCC1O)=O C1(N(C)C(=O)NC2(SCC(F)F)CCC2)CCN(C(=O)C(C)(C)C)CC1 Cc1cc(F)ccc1CC(=O)N(CCC(C(C)C)NC(C1CSCCS1)=O)C c1(CN(CC(CC=C)(C)C)C)ccc([N+](=O)[O-])cc1Cl CCCC#CC(C)(C)NC(C1CC(CCNC(C2C3CCCCCC23)=O)C1)=O Cc1cnc2c(cnn2CC(N2CCCCC(NC(=O)C=C3CCC3)C2)=O)c1 n1(CC(=O)NC(CNC(C(c2cccnc2)OC)=O)C)ccc(=O)n(C)c1=O C(C)(C(=O)NCC1(CC(N)=O)CC1)N(CC)CC.C12CC1CCOC2=O N1(C(CC(C)(C)OC)=O)CCC2CCN(C(=O)C(O)CCCOC)CC2C1 c1(C(=O)NC(CNC(C(CC)C)=O)C2CC2)c(-c2ccccc2)nsc1N c1(OC)cnc(C(=O)NC(CCF)C(=O)NCC(O)CCC2CC2)cn1 C(C1CCCN(C(=O)OC(C)(C)C)CC1)=CCNCN1CC(C)(F)C1 c1(C(C)OC(=O)CCc2cn[nH]c2)ccc(S)cc1.C12(CCC1)CC(=O)N2.C(CO)N C(=O)(C1=NNC(=O)CC1)NC1C(CNC(c2noc(CC)c2C)=O)CCC1 N1(C(CSCCC)=O)CCC2C1CCCN2C(c1ccc2c(c1)CCCC2C)=O n1(CC)nc2c(c1CNC(N1CC3(C1)CN(C)C(=O)N3)=O)COCC2 Cc1nsc2ncc(C(N3CCCC4CN(C(C5CCS5(=O)=O)=O)CC34)=O)cc12 C1(C(N(CC(O)CF)C(=O)OC(C)(C)C)=O)COCCC1C1CCC1 c1(Cc2nnc(N(CC#C)C)n2CC2CC2)nc2cc(C)c(C)cc2s1 C(=O)(CS(=O)(=O)CCc1ccccc1)NCc1ccc(OC)c(N2CCOC2=O)c1 N1(C(=O)Cn2cnnn2)CCOC2(CCN(C(C3CC3c3cccs3)=O)CC2)C1 c1(C(=O)NC2CC(C)CN(C(=O)C#CC3CCCO3)C2)csc2c(F)cccc12 C1(C(=O)NC2C(CNC(c3cc(C)[nH]c3C)=O)CCC2)CC12CCC(F)(F)CC2 c1(OC)ccc(CO)cc1C(N1CCCC(N(C(=O)C(C)(C)F)CCO)CC1)=O NS(=O)(=O)c1cnn(CC(N2CC3CCC2C(NC(=O)Cc2cscn2)C3)=O)c1 C1(CC)CN(C)CCCN1c1ncnc(NCC(C)(OC)OC)c1C CN1CCN(CCC(N2CC(C(C)(C)O)(CNC(=O)CC3C=CCC3)C2)=O)CC1 c1(OCCCC)cnc(F)c(-c2csc(C(=O)NCc3sc(CC)nc3C)n2)c1 c1(C(=O)NC2C(NC(c3ccc(C)o3)=O)COC2)ccn(C)c1C c1(CNC(C(=O)NCC)=O)ccc(C)cc1.c12ncc([nH]1)NC2C CC1CCN2N=C(C(=O)NC3CC(NC(=O)C(C)CC4CCCC4)C3)NC2=N1 c1(C(=O)NCCCCC2CN(C(C3(C)COCCO3)=O)C2)cnc2ccnn2c1 N1(C(C2(n3cc(-c4ccc(Cl)cc4)nn3)CCC2)=O)CCC2CCCCC2C1 C(=O)(CCCC1(NC(C2CCS2(=O)=O)=O)CCC1)N(C1CC1)CC C1(OC)CC(C(=O)NC(c2ncc(F)cn2)C)N(C(=O)CC2CCCC(C)C2)C1 Cc1cc(Br)c(NC(C2CCCN2C(=O)CSc2ccncc2)=O)c(Br)c1 C1(N(C(COCCC)=O)CCC)CCN(C(C2(C(F)(F)F)CC2)=O)CC1 Cc1cc(Cl)ccc1CC(N1CCC(NC(c2nocc2Cl)=O)CC1C1CC1)=O C1(C(N(CCC(C)NC(c2nc3cnccc3s2)=O)C)=O)Cc2ccccc2C1 c1(C(=O)Nc2nc(-c3ccc(OC)nc3)sc2)cn(C)c2cc(Cl)ccc12 c1(C(=O)NCCC(CCNC(C(CC)CCOC)=O)C)cnn2c1CCCC2 c1(C(=O)NC(C2CCCCC2)C(=O)N(CC(c2nn[nH]n2)C)C)cncc(Cl)c1 N1(C(C(CC(=O)OCC)CC)=O)CCC2CCC(C1)N2C(=O)C(F)(F)C(O)CC c1(NC(N2CCOCC2C(F)(F)F)=O)ccnc(Cl)c1Cl C1(C)(NC(C2CC(CCC)C2)=O)CCCN(C(=O)COc2nc(O)nc(O)n2)C1 N1(C(C(C=C)O)=O)CCC2(CCCCN(C(c3ccc4c(n3)CCCC4)=O)C2)C1 c1(CC)c(N2CC(NC(=O)C=C3CN4CCC3CC4)CC2C)ncnc1Cl C(CCC(C)C(=O)NC1CCN(C(=O)C(C)(C)CNC(C)=O)CC1C(N)=O)OC C#CCC(CC(=O)OC)NC(C1(NC(=O)COC(C)C#C)CCSC1)=O C1(NC(CN(C(=O)OCC)C)=O)CC2CC1CN2C(c1ccncc1)=O c1(C(N2CCSC(C)C2)C(=O)NC(CC)C)ccc(Br)cc1C C1(CC)CC(C(N2CCN(C(=O)CC3COCCO3)CC2)=O)CC(=O)N1 Cc1ccnc(C(=O)NCCN(C2CCCC2)C(C2CCNC(=O)C2)=O)c1F N1(C(c2cc(CC)c(C)s2)=O)CC(NC(c2csnc2OC)=O)CCC(O)C1 c1(C(N2CC3CN(c4ncc5ccsc5n4)CC23)=O)cccc2cccc(Br)c12 c1(NC(Cc2nc(NCc3n(C)ccc3)sc2)=O)c(F)cc(Br)cc1Cl c1(C(=O)NCCCN(C(CC2CC(C)C2)=O)CCO)c[nH]nc1C1CCCO1 N1(C(C(C)n2ccnn2)=O)CC2(CCN(C(C3(N(C)C)CCCC3)=O)CC2)C1 C1(C(=O)NC2CC(N(C(C3(C=C)CCC3)=O)C)C2)CCc2cn(C)nc2C1 N1(C(CCCC=C)=O)CCN(C(C2CCN(C)C2)=O)CC1CC(=O)NC c1(C(N2CC(NC(CN(C3CC3)CC)=O)C(O)C2)=O)nn(C)c(C)c1Cl N1(C(C2(NC(N)=O)CC2)=O)CCOC(CNC(c2csc(Cl)c2Cl)=O)C1 C1(C(=O)NC2(CCC(=O)NCC(=O)NC3CC3)CCCC2)CC1C1CC=CCC1 CC(C)(C)C(C)(O)CNC(C1(COC)CN(C(C23CCCC2C3(F)F)=O)C1)=O CCS(=O)CC(=O)N1CCCC(C(C)C(=O)N(C(CN(C)C)CO)C)C1 c1(C(N2CCC(C)C(CNC(C3CCS3(=O)=O)=O)C2)=O)cc(F)cc([N+](=O)[O-])c1 CC(C)CC(C)C(=O)NC(CO)C(=O)NC1CC(CCC(N)=O)C1 C1(NC(c2ccc(Cl)c(Cl)c2F)=O)COC2(CCN(C(c3ccoc3)=O)C2)C1 C(=O)(C(C)CCCC(C)=O)N1CCCCC(CNC(c2cc(SC)oc2)=O)C1 c1(C(N2CC(CN(C(=O)CSCC(N)=O)C)OCC2)=O)cccc2[nH]nc(O)c12 c1(C(N2CC3CCC2C3C(=O)O)=O)ccc(C2=CCCC2)cc1 C1(CNC(C(C)CC2CC2)=O)CC2CCC(C1)N2C(=O)C(=CC1CCCCC1)F N1(C(C2(C(=O)NC)CCC2)=O)CC(C(=O)N(C)CC2CCCOC2)C2(CC2)C1 N1(C(CC(=O)OCCC(C)C)=O)CCCC(NC(=O)CC2CCSCC2)C1 c1(CC(N2C(CCC(=O)NCC(CC(=O)NC)C)CCCC2)=O)ccc(C#N)cc1 C1(C(C)NC(=O)C=Cc2cn[nH]c2)CCCN1C(=O)CCOC(CC)=O Cc1ccc(Br)c(NCc2ccc(-c3ccc(C(F)(F)F)[nH]3)s2)n1 C(=O)(CCCCC(N)=O)NCCC1CN(C(=O)C(C)(C)O)CC(C)O1 C1(NC(C(C=C)O)=O)CCC2CN(C(c3ccc(CO)nc3)=O)CC2C1 CC1CCC(NC(=O)CN(C)C(c2ccccn2)=O)CN1Cc1cccs1 N1(C(C(CCC)C)=O)CCCC2C1CCN2C(c1cc(Br)c(C)o1)=O N1(C(C(C)=C2CC2)=O)CCN(C(c2cc(O)cc(C#N)c2)=O)CC2CCCCC12 N1(C(=O)Cc2ccccc2F)CC2(CCCN(C(C3CCCO3)=O)C2)C1 N1(C(c2[nH]nc(OC)c2Cl)=O)CCN(C)C(CNC(c2cnc(C3CC3)s2)=O)C1 c1(C(=O)NCC2(C)N(C(C(CCCC)C)=O)CCC2)ccc2nc(C)nn2c1 c1(C(=O)NC2(CO)CN(C(c3cc(C(C)(F)F)n[nH]3)=O)C2)ncncc1F C=C(CNC(C1CN(C(c2ccc(SC)o2)=O)CC1F)=O)C1CCOCC1 C12(CNC(C3C(C)CC3)=O)CCC(CC1)N2C(=O)Cc1csc(C(C)(C)C)n1 c1(C(C)=O)c(C)[nH]c(C(=O)CN(C)CC2CC2c2ccco2)c1C C1(C(N(C2CCN(C(C(C)CO)=O)CC2)CCO)=O)CCn2nnnc2C1 CC(CC(=O)N(C1(NC(=O)CNS(=O)(=O)C2CC2)CC1)C)c1ccccc1 N1(C(C=CC)=O)CC(NC(C2(NC(C)=O)CCC2)=O)CCC1C N1(CCNC(c2cccc(N3CC=CC3)c2)=O)CC(NC(=O)C=CCO)CC1=O CN=c1ccc(C(=O)NC2(CCC(=O)NC(C)C(=O)NCCOC)CCC2)c[nH]1 C1(CC)(NC(C2CCC=CO2)=O)CCN(C(=O)CC2(N3CCCC3)COC2)CC1 c1(OC)ccc(C(=O)NC2CCCN(C(C3CC3(Cl)Cl)=O)CC2)c(OC)c1OC C1(CC)CCCC1NC(=O)CC(C)NC(=O)COCC(C)(C)C N1(C(C2(CNC(=O)CC3CC4CC4C3)CCC2)=O)CC2(CCC2)C1 CCCC(F)C(=O)NC1CCOCC1NC(=O)CCCc1ncco1 c1(CC(=O)NCC2(C(C)(C)O)CN(C(C(C=CC)O)=O)C2)cccnc1C C1(OCC)CC1C(=O)OC(C)(C)C.C12CC1OC(=O)N2 c1(CCC)ccc(N)c(C(=O)OCCC(c2cnc(Cl)s2)=O)c1 c1(-c2cn(C3C(OC)CN(C(C4C(C)(C)CCO4)=O)C3)nn2)ccc(N)c(F)n1 c1(C(=O)NC2C(NC(C(CC(=C)C)C)=O)C2)cccc2oncc12 CC(C)CS(=O)(=O)CC(=O)NCC1C2CC1N(C(=O)CC(C)O)C2 N1(C(=O)Cc2cccs2)C2CC1CN(C(c1cnccn1)=O)C2 c1(CC(=O)N(CC(C)CNC(=O)C=C(Cl)Cl)C)ccc(O)cc1Cl O=CN1CCCN(C(C2CN(C(C3C=CC=CC=C3)=O)CC23CC3)=O)CC1 c1(C(=O)NCc2cccc(C(C)C)c2)cc(F)c(C(=O)O)c(F)c1 N1(C(C2N(C(C)=O)CCCC2)=O)CCC(NC(=O)CC2(C)CCCC2)CC1C c1(C(C(=O)NCC(=C)C)N(C(C)C(=O)OC(C)(C)C)C)oc(CC)cc1Br.N(C)CC Cn1[nH]c(=N)cc1NC(N1CCCC(c2cccc(C(F)(F)F)c2)C1)=O N1(C(C(C2CCC2)OC)=O)CCC(C(F)CNC(c2nc(C)sc2C)=O)CC1 Cc1ccc(C(F)F)cc1C(=O)NC1CC(C)CN(C(=O)C=CC=C(Cl)Cl)C1 c1(C(N(CCC(=O)NC2CCSC2C)CC)=O)snc(C)c1N N1(C(C(C(C)(C)C)O)=O)CCC2CCN(C(=O)CC3CCC=CCC3)CC2C1 c1(C(N2C(C(=O)NCCCCCC)CC3CC32)=O)nc(C)ccc1C c1(C(=O)NCC2CC(NC(c3cc(C4CC4)no3)=O)C2)ccc(O)cc1Cl C1(C(=O)NC(CNC(CS(N2CCN(C)CC2)(=O)=O)=O)(C)C)CC(S(N)(=O)=O)C1 c1(C(N2CCCC(NC(=O)Cc3ccc(Cl)s3)CC2)=O)nccc2ccncc12 c1(C(=O)NCC2CC(C)(C)CN2C(=O)CC2(CO)CC2)cccn2cnnc12 Cc1ccc([N+](=O)[O-])c(NC(c2n[nH]cc2NC(c2ccc(Br)c(C)c2)=O)=O)c1 C(=O)(CC(C)CC(C)C)N1CC(N(C(c2c(SC)cn(C)n2)=O)C)C1 C(=O)(C(C)(F)C(=O)NC1CCCN(C(=O)Cn2ncc(O)nc2=O)C1)OC S(=O)(=O)(c1ccc(Br)s1)N1CC(C(=O)Nc2cc(Br)cnc2O)C1 N1(C(c2ccc(CC)cc2Cl)=O)CCC(C2CCCN(C(=O)C(N)=O)CC2)CC1 c1(C(N(C)CC2N(C(C3C(C)CC3)=O)CCCC2)=O)ccc(Br)c(N)n1 C1(CC(=O)NCC2C=CC(NC(c3c(CC)n[nH]c3)=O)C2)CCC(OC)CC1 C=CCCCCC(=O)OC(c1cc(-c2ccsc2)[nH]n1)=O N1(C(c2scc(C)c2Cl)=O)CCCCC2(CCN(C(=O)CC3(O)CCOC3)C2)C1 c1(C(N2C(CCNC(C(C)OCCC#C)=O)CCC2)=O)cc2nnn(C)c2s1 N1(C(C(N2C(c3onc(N(C)C)n3)CCC2)=O)=O)CCSCC1C1CC1 CCC(C(=O)N1CC(C(=O)NC2(C)CN(C(=O)C3CC3)C2)C(C(C)C)C1)C(C)C C1(NC(Cc2scc(C)n2)=O)CN(C(=O)Cc2ncc(C)s2)CC1O c1(C(N2CCC(OCCCNC(CSC)=O)CC2)=O)c(C)[nH]c2ccc(O)cc12 S(=O)(=O)(c1c[nH]c2ccc(Br)cc12)NC1CCCN(N(C)C)C1.C(=O)O C12(NC(c3c(C)ccc(Br)c3)=O)CCC(CC1)N(C(C1CC1(C)C(F)F)=O)C2 c1(-c2c(CN3CC4(C(C(=O)OC)COCC4)C3)n[nH]c2)coc2cc(O)ccc12 C1(C(=O)NC(C2CCCN(C(=O)CN3CC(C)(C)C3)C2)C)CCCN2CCCC12 N1(C(c2cc(Cl)c(Br)cn2)C(=O)NCCCSC)CCCc2sccc2C1 C(CCCCC(=O)N1CC2CC1CC2O)c1cn(C(C23CCC(C2)C3(C)C)C)nn1 C1(C(C)(C)C)CN(C(=O)C2=CCSC2)CCN1C(=O)CC1CCOC1(C)C Cc1cc2ccccc2nc1C(N1CCCC(CNC(=O)CC#N)C1)=O C1(NC(C2CC(=O)NC(=O)C2)=O)C2CCC1CN(C(C1CCCCO1)=O)C2 C(=O)(C1=CC2C=CC1C2)N(C1CCN(C(C2CC2C2(C)COC2)=O)CC1)CC#C C(CN=c1nc2sccc2c(N(CCCN2CCCC2)C)[nH]1)C1CCC(C)CC1 c1(OCC(=O)NC2(C3N(C(CC(C)OC)=O)CCC3)CC2)ccccc1C C(=O)(CCCC(=O)NCC(C)CNC(C1(OC(C)C)CCC1)=O)NCCC C1(=CC(N2CCC(NC(C(C3CCCC3)OCC)=O)C2)=O)CN2CCC1CC2 c1(C(=O)NC2CCCN(C(CSCC=C)=O)C2)c(C)nc(C2CC2)nc1S Cc1ccc(C(=O)NCc2ccc(CNC(=O)C(C)n3ccnn3)cc2)cc1F C1(CCNC(C2C(c3n(C)cnc3)C2)=O)COCCN1C(=O)Cn1nnc(=O)[nH]1 CC(C)(CNC(C1CCCN1C(=O)CNc1ccccn1)=O)CC(F)F C1(C(=O)NCc2ccc(C(=O)NCC(CC)SCC)o2)CCCC12CCC2 c1(C(N2CC(C)CC(C(=O)NCCCOC=C)C2)=O)cnc2cc[nH]c2c1 c1(C(N2CCC(N(C)C)C2C)C(=O)NCC(=C)C)cc(Cl)c(Br)cn1 CC1CC(C(=O)NCCC2CCCN2C(c2csc(-c3cn[nH]c3)c2)=O)C(C)O1 N1(C(C2(C)COC(=O)N2)=O)CCC2(CC1)CC2C(=O)NCc1ccnc(O)c1F N1(C(C(C(C)C)NC=O)=O)CCC(F)(CNC(=O)CN2CCNC(=O)C2)CC1 C(=O)(CCCC(=O)N(CCCOCCNC(=O)CCc1cc(C)n(C)n1)C)NC c1(CNC(C2CCCC2NCc2ccnc(Br)c2)=O)noc2ccc(Br)cc12 CC1COCCN(C(C2(NC(=O)C=Cc3cn(C)cn3)CCSC2)=O)C1 c1(C(N2CC3C(NC(c4scc(C)c4Cl)=O)C3C2)=O)ccc(N=[N+]=[N-])cc1 c1(C(C(=O)NCCCC)N(C)CC2CCCCCC2)ncc(F)cc1F C1(C)(C(=O)N(C(C)(C)C)C(C2C(NC(COCCCOC)=O)C2)=O)CC1(C)C N1(C(C(CCC)OC)=O)CCCC(CO)(NC(=O)C(C)=C2CCCC2)C1 N1(C(CCCCOCC)=O)CCCC(C(=O)NCC2CC(=O)N(C)C2)CC1 C(=O)(C(CC(F)F)c1ccccc1)NCC1N(C(CSCCCC)=O)CC=CC1 C1(C(C(N2CC(CNC(=O)Cc3ccno3)C2)=O)F)CCCCC1 c1(OC)ccc(C)c(NC(C2CC(C)(C)CN2C(=O)C(O)CC(N)=O)=O)c1 C1(C(N2C(C(C)(C)C)CCCC2)=O)CCCCC1N=c1[nH]cnc2cnccc12 c1(CC2CCN(C(c3nc(CC)sc3)=O)CC2)nc2ccc(C)cc2[nH]1 N1(c2ccc(C#C)nn2)CCC2(CC1)COC(CO)C2.C12COCCC1N2 N1(C(C2(C)COC2)=O)CCCC2(C1)CN(C(c1snc(O)c1Cl)=O)CCO2 S(=O)(=O)(c1ccc(Br)cc1NCCCn1cncn1)N(C1CCCC(OC)C1)C c1(CC)cccc(C)c1NC(=O)C(N1CCOC(C)CC1)CC1CC(F)(F)C1 C(=O)(CCS(N)(=O)=O)N(CC(C)CNC(c1ncc(F)cn1)=O)C c1(C(=O)NC2CC(C(N(CC(C)C#N)CC)=O)OC2)cc(OC)ccn1 N1(C(c2cc([N+](=O)[O-])cs2)=O)CCOC2(CCC(F)(F)CC2)C1 c1(C(N2C(c3cc(C)ncc3)CCC2)C(=O)NC(C)C)c(Cl)nc(Cl)n1C CC1CN(C(=O)CC2(n3ccnc3)CC2)CCCN1C(C1CC(O)CN1C)=O CC1(C)C(NC(=O)C(F)n2cccn2)CCN1C(c1ccccc1)=O c1(C(=O)NCC2CC(NC(CCc3cn(C)nc3)=O)C2)ccc(Cl)c(Cl)c1 c1(NC(C)=O)cccnc1C(=O)NC1CCC(NC(C2(c3cccs3)CC2)=O)C1 CC(C)(C)S(=O)(=O)CC(=O)N1CCOCC(CNC(=O)C(C2CCOCC2)=O)C1 N1(C(C2CCN(C(=O)NCC=C)C2)=O)CCN(C(=O)CC=C(Cl)Cl)C(COC)C1 n1(CC(=O)NC(CC)CN(C)C(c2csc(C#N)c2)=O)ccc2ccccc12 C1(NC(c2c(CC)c[nH]n2)=O)CCC(C)(CNC(c2cccc(N)c2)=O)C1 C1(CN(C(C)(CCBr)c2nnnn2-c2ccc(F)cc2)C)CCCC1(C)C C1(C(N2CC(CC)C2)=O)CCCC2(CCC2)O1 C1(NC(CCC(=O)NC)=O)CC(CC(=O)NC2(c3cn[nH]c3)CC2)C12CCC2 C12(C(N3CCCC(C(=O)NC4CC5(CCC5)C4)C3)=O)CCN(CC1)CC2 C1(NC(c2ncn(C)c2)=O)CCCC(CN(C(=O)Cn2cnc(=N)[nH]2)C)C1 C(CNC(=O)CNc1nccs1)(C(C)(C)C)NC(C1(OC)CCCC1)=O C1(NC(C2CC23CCCC3)=O)CN(C(c2[nH]nnc2C2CC2)=O)C2(CCOCC2)C1 CC(C)C(O)CC(=O)NCC1CC2(CC(NC(C3COC4(CCC4)C3)=O)C2)C1 n1(C(C(=O)Nc2ccc(C(=O)NCC(=O)OC)cn2)C)nc([N+](=O)[O-])cc1C C(=O)(C(C)C(F)F)N1CC2(C1)C(=O)N2.C1(C(C)SC)CCCCC1 c1(CSCC(=O)Nc2ccc(CCCCCC)cc2)nnc2n1CCN(C)C2=O CC(C)CC(CNC(c1cc(CCO)on1)=O)C(=O)N1CCC(N(C)C)C(C)C1 CC(C)(C)C#CC(=O)NC1CCN(CCNC(=O)C(F)Cc2ccccc2)CC1 CC1CCc2c(sc(NC(c3nnc(-c4cc(Cl)ncc4F)s3)=O)c2C(N)=O)C1 c1(C(C(=O)NCCN(C(c2ccc(=N)[nH]n2)=O)CC)=O)ccc(F)cc1 N1(C(CCc2c(C)ncs2)=O)CCC(NC(=O)C=CCOC(C)(C)C)CC(O)C1 c1(C(=O)NCC(C)NC(=O)C(c2ccccc2F)(C)C)ncc(Br)cc1N Nc1c(F)cc(C(=O)NC(CCCNC(C2CSC2)=O)c2ccccc2)cc1F O=C1CCC(CC(=O)NCCCN(CCO)C(C2C3COCC23)=O)C1 C(=O)(Nn1nnc(C)c1C)C1CCN(C(c2c(NC)nccc2)=O)CC1O C(=O)(C1Cc2ccc(F)cc21)N1CC(CC)(NC(c2sc(C)nc2C)=O)C1 c1(C(=O)NCC2(NC(C3C(=C)C3)=O)CCC2)ccc(F)nc1F c1(C(C(=O)NCCCC)N(C)C(c2ccncc2)C)cc(OC)ncc1Cl N1(C(C(C)CF)=O)CC2CCC1CN2C(=O)Cc1cc(O)nnc1O C1(NCc2[nH]nc(COC)n2)CCCC2OCCC12 N1(C(CC2C(C)(C)C(NC(c3scnc3Cl)=O)C2)=O)CC2CCC1CC2 Cc1onc(C(=O)NCC2(NC(c3cn(C)cn3)=O)CCOC2)c1[N+](=O)[O-] N1(c2occ(C(C)SC)n2)C(=O)NC(Cc2ccccc2)C1=O C#Cc1ccc(C(N2CC(O)CC2CNC(C2CC2F)=O)=O)o1 Cc1cc(CN2CCC(O)CC2C(=O)Nc2cnc(C3CC3)cn2)ccc1Br C1(NC(C(C)CC(F)F)=O)CC12CCC(NC(c1ccc(F)c(Cl)c1F)=O)CC2 C#CCCCCC(=O)NC(COCC)C(N1CC2C=CC1CC2)=O Cc1ccc(=N)[nH]c1C(=O)NCC(C(C)(C)C)NC(C1CCCNC1=O)=O c1(OC)ccc(NC(=S)NNC(=O)C2(N3CCOCC3)CC2)cc1Br C(=O)(N1CCCc2nncn21)c1c(CNC(C2CC2C2CCC2)=O)ocn1 c1(NC(C23CC(n4cc(COC)nn4)C2C3)=O)cccc(C(=O)NCCN=[N+]=[N-])c1 Cc1ccc(C(=O)N(CC(=O)NCc2n[nH]cc2C)C2CCC2)s1 c1(CNC(=O)C(N2CCC(Br)CC2)=O)cccc2c1OCO2 c1(NC(=O)NC2(CC)CC2)cnc(N(C)C)cc1C C(=O)(C(C)CC(C)C(C)=O)NC(CCCNC(CC(CCC)(C)O)=O)C C(N=c1[nH]n(C)cc1Br)c1c(C(=O)OCC)cno1 N1(C(c2c(C)nsc2C)=O)CCC2(CC1)CN(C(c1nocc1Cl)=O)CC(C)O2 C1(C(=O)NCCCn2cccn2)CCN(C(C2CC(F)C(=O)N2)=O)C12CC2 C12CCC(CC1)C(=O)NC2.N1(C(C2(CC)CCCO2)=O)CC(N(C)C)C(F)C1 N1(C(C2C(CNC(c3ccc(C#C)cc3)=O)OCC2)=O)CCC(=C(F)F)CC1 N1(C(C(COCC)NC(=O)C(C)N2CC(C)C2)=O)CCC(NC=O)CC1 c1(C(N(C2(C)CCC2)C2CC2)=O)ccc(CO)o1.n1(CC)cc(COCCOC)nn1 c1(CCC(=O)NC2CN(C(c3n(CC)ncc3)=O)C2)cc2ccccc2o1 C#Cc1ccc(CC(=O)NC2CCC(C)N(C(C3CCOCC3)=O)C2)cc1 Cc1c(C(N2CC(C(=O)N(C)Cc3ccc(Br)cc3)C2)=O)ccnc1Cl N1(C(C(C)=O)=O)CC2(CC(NC(=O)C(c3nocc3C)C3CCCCC3)CO2)C1 c1(C=O)oc2ccc(C)cc2c1C.C1C(=O)NCC(C2CCC2)N1C1CC1.CO c1(C(=O)NC2C(CO)CCN(C(C(C)CO)=O)C2)cnc2c(c1)COC2 C(=O)(CCC(C)(C)C)N1CC=CC(C(N(CCO)CC)=O)C1 Cc1cnc(C(=O)NC2CCCC(CC(=O)NC(C)CCCCCO)C2)c(F)c1 c1(C(=O)NC(CC)CNC(C2CCCS2)=O)ccc(Br)nc1O C(=O)(CC(O)C(C)C)NCCC(C(=O)N(C(C)C)CC)OC C(=O)(C1=CCCN(C(C2CCCOC2)=O)C1)NCCSCCC=C C1(Cn2cc(C(C=C)(C)O)nn2)CC(C(F)(F)F)CN1C(C1C=NN(C)C1=O)=O C1(C(=O)NC2(c3ccsc3)CC2)C2CCCC2CN1C(=O)CC1COCCO1 c1(SC)ncc(C(=O)NC(C)CCCNC(c2cn(C)c(=O)cn2)=O)c(O)n1 N1(C(C(CC#C)O)=O)CC2CC(C)N(C(c3c(C)cc(C)nc3C)=O)C2C1 c1(CC)ccccc1C(CNC(=O)C(C1CC1)SCC)NC(C1CCOCC1)=O c1(OC)cncc(C(=O)NC(CC2CCCC2)C(=O)NCC(C)OC(F)F)c1 C1(NC(C(CNC(CC(CC)OC)=O)(C)C)=O)CCC2CC2CC1 CC1(C)CC(C(N2CCOC3C(O)CC23)=O)CN(C(C2C=CC=CC=C2)=O)C1 C(=O)(CCCCC(C)(C)C)N1C(SCC)CCC1.C12CCCCC1NC2=O C=CCC(CC=C)C(=O)NC1CCC(CNC(C2CC(C(C)C)=NO2)=O)CC1 C(=O)(N1CC(O)C(O)CO1)C1N(C(c2cc3scc(C)c3[nH]2)=O)CCC1(C)C C1(n2c(C)n[nH]c2=N)CCCN(N2CCCC3(CCCO3)C2)C1 c1(N2CCC(NC(COCc3ccc(C)s3)=O)C(F)C2)c[n+]([O-])ccc1[N+](=O)[O-] C(=O)(C#CC1CCCO1)NCCC(C)N(C)C(c1ccc(S(C)(=O)=O)o1)=O C1(C(=O)NC(CN(C(c2nc(Br)c(C)s2)=O)CC)C)CCC=CCC1 c1(C(C(=O)NCCCC)N(CCC(F)(F)F)C)cc(Br)c(F)cc1F C1(C(=O)NC(C)CCCNC(=O)CCc2nc[nH]n2)CC1C1CCC1 C(=O)(C1=NN2CCCN=C2N1)NCC(C(C)C)NC(C1(C)CCC(F)(F)CC1)=O c1(CNC(C2C(NC(=O)CNc3cccnc3)CC2)=O)ccccc1Cl c1(C(=O)NCCC2(O)CN(C(C(CCC)=CCC)=O)C2)cn2nc(C)sc2n1 N1(C(C(=O)Nc2cc(CNC)c(Cl)cc2)=O)CC2CNCCCC2(CO)C1 c1(C(N(C(c2cn(-c3ccccc3)nn2)C)C)=O)sc(F)cc1Br c1(C(=O)NCC(=O)NC2CCCC(C(N)=O)C2)cc(Br)ccc1[N+](=O)[O-] CC1c2cccc(Br)c2CCN1C(=O)C(=O)NCCn1cnc(CO)n1 Cc1ccc(CC(=O)NC(C2(O)CN(C(c3ccn(CC#N)n3)=O)C2)C)c(Cl)c1 C1(NC(=O)C2=NOC(c3ccc(F)cc3)C2)Cc2ccccc2C1O c1(C(=O)NCC2C(OCC)CN(C(C(C=C)O)=O)C2)cccn2cnnc12 N1(C(COCC#C)=O)CCC(OCC(C)O)C1.c12coc(n1)OC(C)CNC2=O CCCCC(O)C(=O)NCC(CNC(=O)C=Cc1cnn(C)c1)CO C(=O)(C1CCCn2ccnc21)NC1C(OC)CN(C(c2ccc(C)cc2C)=O)C1 c1(SCC(C(C)C)(c2nnnn2-c2ccccc2)NCCO)cnn(C)c1C#N C(=O)(C#CC1CCCCC1)NC(CNC(C1=CCC(C)CC1)=O)C(C)(C)C C1(CCC)CCCN1N1CC(C2C(=O)N2)C1.C(c1ccco1)=C(C=O)C Cc1cc(C(F)F)n(CC(=O)NCCN(C)C(c2ccc(C3CC3C)o2)=O)n1 n1(CCOC)cc(NC(=O)CC2CC(F)CN2C(=O)C(=O)C2CC2)c(C)n1 c1(C(=O)NC2CN(C(C=Cc3n(C)ccc3)=O)CC2O)ccc2sccc2c1 C1(C(=O)NCC23C(CN(C(CC4(C#N)CCC4)=O)C2)C3)Cc2cccnc2C1 CC(=O)CCCCC(=O)N1CCCC1C(=O)NC(CO)C(C)(C)CO S(=O)(=O)(c1ccc(Br)s1)N1CCCC(C(=O)NC(CC)CCO)C1 N1(C(C2(OC)CCC2)=O)CCC(C2CCN(Cc3cnc(Cl)cc3C)C2)CC1 c1(CNC(c2[nH]cc(C(N)=O)c2)=O)cccc2c1CCN(C(C1CC13CC3)=O)C2 C(C(C)(C(=O)NCC(CC1CCCC1)C(=O)NCCCCC(C)C)OC)OC N1(C(C2CC(O)(CC#C)C2)=O)CCN(C(=O)CCOC)C(CCC)C1 Cc1cc(O)c(C(=O)NC(C)CN(C)CCCOc2ccccc2)cc1Br c1(C(N(CC(CC)NC(=O)CN(S(=O)(=O)CC)C)C)=O)nocc1C N1(C(COC(C)=O)=O)CCOC(CCNC(=O)CCCc2cccs2)C1 c1(C(=O)NC2C(C(C)C)N(C(=O)CNc3cccnc3)CC2)ccc(Cl)c(F)c1 C(CO)(C(=O)N1CCCC1C(C)(C)CNC(c1csc(Cl)c1)=O)N(C)C N1(C(C2(NC(C(C)OCCN(C)C)=O)CC(F)(F)C2)=O)CCOCC(O)C1 CCCCCC(C)CC(=O)NC1CN(C(=O)CNc2ccccn2)CC2(CC2)C1 c1(C)cccc(CO)c1.N1(CC(=O)NC2C(NC(=O)C=C3CC3)CC2)CCOC1=O C(=O)(C(O)P(C)(C)=O)N1CC(OC)C(NC(=O)CCCc2ccc(Cl)cc2)C1 CCCC(CC)C(=O)NC1COCC1NC(=O)C(C)(C)NC(c1ccccc1)=O C(=O)(CS(=O)c1ccc(Cl)cc1)NC1C(NC(C23CC(C)(C2)C3)=O)CCCC1 C1(CC#C)(C(=O)N(C)Cc2cn(C)cn2)CCN(C(=O)C(C)C2CCCC2)C1 S(=O)(=O)(c1cc2c(cc1Cl)NC(=O)CO2)NCC(c1scc(C)n1)(C)C C1(NC(C(CCC)NC(C)=O)=O)CC2(C1)CN(c1cc(OC)ncn1)C2 c1(-c2scc(C)n2)cc(NC(=O)Nc2ccc(CO)c(Cl)c2)cc(Br)c1 c1(C(C)C)ncccc1NC(C1CCN(C(=O)C(F)n2ccnc2)C1)=O c1(OC)ccnc(NCC2CC2NC(=O)OC(C)(C)C)c1OC S(=O)(=O)(c1cnc(Cl)nc1)N1C2(CNC(=O)C2)CC1 c1(SC)ccc(OC(c2ccccc2F)CNC=O)cc1.C(C)(C)O c1(C(N2C3CN(Cc4cccc(C=C)c4)CC2CC3)=O)cnn2cc(C)cnc12 C=C(C)C(C)(C)C(=O)NC1CCC1NC(c1cc(-c2ccn(C)n2)on1)=O C(=O)(CC1=CCN(C(=O)C2=CCCCC2)CC1)NCC(CC)CO CC1(NC(=O)CN)CN(C(C23CCCC2C3)=O)C1.c1(N)ccc(F)o1.C1(=O)CN1 c1(C2CCN(C(C=C(C=CC(C)(C)C)C#N)=O)C2)cc(F)cc(F)c1 c1(OC)ccnc(C(=O)NC2CCN(C(c3ccnnc3S)=O)C2)c1 Cc1cccc(C(O)C(=O)NCCCN2CCN(C(C3CC3C#N)=O)CC2)c1F c1(NC2(C(F)F)CC(CCOC)C2)ccc(N2CCC(O)CC2)cc1 c1(NCCC2CCC(NC(Cn3nnc(C)n3)=O)C2)ncc(Br)cc1[N+](=O)[O-] C1(C(=O)NC2CN(C3CCC3)C2)(CNC(=O)Cc2cncs2)CCC1 Cc1nc(CC(=O)N(C(C2CCN(CC(F)(F)F)C2)=O)CC2CCC(=O)N2)n[nH]1 c1(C(=O)NC2(C3CCCN3C(C34CC(F)C3C4)=O)CC2)ccc(NCCO)cc1 C1(Cl)(C(=O)NCC(CNC(CCCOC)=O)C)CC12CCC2 c1(C(N2CC(C(=O)OC)OC(C)(C)C2)=O)cccc2occ(Br)c12 N1(CC)CCN(C(c2coc(C(C)NC(=O)CCc3cncs3)n2)=O)CC1C CC1CN(C(=O)C(O)CNC(=O)C2=NN(C)C(=O)CC2)Cc2c[nH]nc21 c1(C(N2CCCC(NC(CC3(CSC)CC3)=O)C2C)=O)ccc2n[nH]cc2c1Cl C12(NC(CC3CC(=C)C3)=O)CC(C1)N(C(c1ccc(C)o1)c1ccccc1)C2 c1(NC)ccc(C(=O)NCCC2CCCN(C(C3(C)COC(=O)C3)=O)C2)nc1 c1(NC(=O)NCC2COC(CNC(=O)C3CC3)C2)nc2ccccc2s1 c1(C(=O)NCC(=O)OC)ccncc1Br.c1(C(C)=O)ccc(SC)cc1 Cn1ccnc1CCC(=O)NCC1(C(=O)NCC2(F)CC2)CCC1 C=CC1OCCC1C(=O)NCCCC1N(N2CC(C=O)C2)CCCC1.C(C)=O N1(C(CC(C)C2CCCCC2)=O)CC2CC1CCC2NC(=O)CCCC1CCC1 C(=O)(C#CC1(C)CC1)N1C(CC)C(NC(=O)C(c2cnn(C)c2)=O)CC1 c1(NC)cc(C(=O)NCC2COC(CNC(C)=O)C2)c2ccccc2n1 c1cc(NCc2ccc(C3CCC3)nc2)ccc1-n1cncn1 c1(C(=O)NCCCC2OCCN(C(C3CC(OC)C3)=O)C2)cnn2c1CCCC2 Cn1nccc1C1=CCN(C(=O)C(N2CCCCOC(C)(C)C2)=O)CC1 CC1=C(C(=O)NCCCC(C)NC(=O)Cc2csc(C(C)C)n2)CC1 C1(C(N(CCCN(C(C(N2CC(C)C2)C)=O)C)C)=O)CC2(C1)CC21CC1 N1(C(c2c(N)ccc(Cl)n2)=O)CCC2CCN(C(c3ccc(CO)cn3)=O)C2C1 c1(C(=O)NCC2(C)CN(C(c3ccc(Br)c(CO)c3)=O)C2)cccc(F)c1O C1(C(C)C)(CO)CCN(C(=O)C(C)CF)CC1.C(=O)(CCn1cccn1)OCCN N1(C(CCC#C)=O)C2CCC(C(=O)Nc3ccccc3COC)C1CC2 C12(NC(c3ccnc(OC)n3)=O)CCC(C1)N(C(=O)CCCC(F)F)C2 N1(C(=O)C(C2CCOCC2)O)CCC(F)(CNC(C23CCCC2CCC3)=O)CC1 C1(NC(CCCCSC)=O)CN(C(c2csc(C(C)=O)n2)=O)Cc2nccn2C1 C(=O)(C#Cc1ccc(F)c(F)c1)N(C)CC1CC(C(F)(F)F)C1 c1(C(=O)Nc2ccc(C(=O)Nc3n(C)ccc3I)cn2)cc(F)c(Cl)cc1F CCC(CC(=O)NC1CCN(C(=O)COc2ccc(C)cc2)CC1(C)C)C(C)C C1(C(=O)NC(CC2(CNC3CC(=O)NC3)CC2)=O)C2CCC3C(C2)CC13 c1(C(N2CC(OCCNC(=O)COC(F)F)C2)=O)cnc2c(c1)COC2 c1(NCC=CC)cc(N(C)Cc2ccc(C(F)(F)F)c(F)c2)nc(C)n1 N1(C(C(CCCC)F)=O)CC2CC1CN(C(=O)C(C1CCCC1)OC)C2 CCC(CC(=O)NC1CC(C(=O)N(c2cnn(C(C)C)c2)C)C1)OC C#Cc1cc(C(N2CC(CNC(=O)C(C)(O)C(C)C)C2)=O)cc(C(F)(F)F)c1 C1(CCNC)CCN(C(=O)NCCCC2CCC(=O)N2C)CC1 C(=O)(CCCC(=O)N(C)C)NCC(c1nc(C)cs1)N(C(C=C(C)C)=O)C c1(C(N(C2CCCC(NC(c3cnn(C)c3Cl)=O)C2)C)=O)cncc2c1CCC2 C1(CC)(NC(=O)CCCSc2ccccc2)CCN(C(=O)CNC(=O)OC)CC1 C1(NC(C)=O)CCC(C(=O)NCC(F)CNC(c2ccc(Cl)cc2)=O)CC1 CC1(C)CCOC(CNC(C2C3CCC(C3)C2NC(=O)C(O)c2ccsc2)=O)C1 C1(CCNC(C2CCC(C)CC2)=O)CCN(C(=O)CNc2ccccc2)C(C)C1 C1(NC(C2(C)CC3(CC3)C2)=O)CCCCN(C(c2ccc([N+](=O)[O-])o2)=O)CC1 CC1CN(C(=O)CCc2ccn(C)c2)CC1C(=O)N(CCCc1ccco1)C c1(C(=O)NCCOCCNC(C2(CC)CC2(F)F)=O)c(O)cccc1Cl C12(C(CO)NC(CN(C(CNC(C(CC)C)=O)=O)C(C)C)=O)CCC(CC1)C2 CC1CCOC1C(N1CC(N(C(=O)CNC(c2ccc(Br)o2)=O)C)C1)=O C(CN=C(NCC1CCCO1)NCC12CCC(CC1)OC2)c1c(C)ncs1 C(=O)(C1=C(SC)CCCC1)N(CCN(C(C(C)OCC=C)=O)C)C C1(NC(C)=O)CCN(c2cnc(C#N)cn2)CC12CCC2.c1ccc2cnsc2c1 C(=O)(C(C(C)(C)C)C1CCC1)NC1C(C)N(C(c2cc3sccc3[nH]2)=O)CC1 c1(ONC(C2N(C(C(C)C3C(C)C3)=O)CC2)=O)cccc(F)c1 N1(C(C2C(C(=O)OC)CCO2)=O)CC(NC(C2C=CC=CC=C2)=O)C(C)(C)C1 C1(NC(c2n(C(C)C)cnc2)=O)CC2CCC(C1)N2C(=O)CNC(C1CCC1)=O c1(NC(c2c(Cl)ccc(SC(C)C)c2)=O)ccc2c(c1)CN(CN)C2.C(N)(=O)N Cc1nc(N2CC(CC(=O)N3CCC3N3CCOC3=O)C2)ncc1F C1(C#N)(CCC=C)CCN(C(=O)Nc2nc(C(F)(F)F)ccc2Br)CC1 c1(C(=O)NC2CCC(CCNC(C(C)S(N)(=O)=O)=O)C2)ncc2cc(Cl)ccn12 N1(C(c2c(CC)cccn2)=O)CCCC2(CCN(C(=O)CC3C(C)C3(F)F)C2)C1 CC1=C(C(=O)N(C2CCCCN(C(C3(C)CNC(=O)C3)=O)C2)C)CCO1 N#Cc1nccnc1NC1CCC1NC(c1cnc(-c2ccoc2)s1)=O Cc1nn(CC(C)C)c(Cl)c1C(=O)OCCCC1CC1 C(C(N=[N+]=[N-])C(=O)N1CC(CCCCNC(c2c(CO)n[nH]c2C)=O)C1)OCC N1(CCC(=O)NC2(C(=O)NCC(=O)NCCC)CCC2)CCOCC1 C1(C(N2CC(O)(C(C)NC(C3CCCO3)=O)C2)=O)CCCC1(C)C Cc1cnc(CNC(=O)C(C2CCCC2)NC(C2(C#N)CCC2)=O)c(C)c1 CC(C(=O)NC1CN(C(=O)COCc2ncnn2C)CC1F)C(C)(C)C c1(C(C(=O)N2CC(C3CCCO3)C2)N(C)CC2CC2)ccccn1 c1(C(=O)NCC2N(C(CC=C(C)C)=O)CCC2)ccc(NS(C)(=O)=O)c(Cl)c1 CC1CN(C(=O)COC(F)(F)C(F)(F)F)CCC1NC(N)=O.C1(=O)CCCN1 C1(CC)(NC(c2cnn(CC)c2C)=O)CCN(C(C2C3CCC(=O)C23)=O)CC1 CC1CN(C(=O)C2=CCC2)C(C)CN1C(c1n[nH]c2c1COC2)=O n1(CC)nc(CNC(=O)N(CC(C)(C)O)CCc2ccccc2)cc1C CC(F)CCN=C(NCC1CCN1C(=O)OC(C)(C)C)NC1CCN1C(C)(C)C C1(c2nc(CNCC(=O)N(CCCC)CC(C)C)sc2)CCC(F)(F)CC1 c1(C(=O)NCC(C)(O)CNC(=O)CCn2cc(Cl)cn2)cnc2ccc(F)cn12 C12(CNC(Cc3scc(C)c3)=O)CCC(C1)N(C(c1cc(Cl)ccc1N)=O)C2 C1(C(=O)NCCNC(=O)CSc2ccc(Cl)cc2)COCC2(CCC2)O1 CC(C(=O)N1CC(OCCC(=O)NCC2CC23CC3)C1)n1ccnc1 c1(C(=O)NCCC2(C)CCN(C(C(C)C#N)=O)C2)ccn2cncc2c1 N1(C(c2c(COC)ncs2)=O)CCCC1(C)CNc1cc(C(F)(F)F)ncn1 CCC(C(=O)NC)NC(=O)CC1(NC(C2CCCSC2)=O)CC1 c1(CC(C(=O)NC2CC(N(C(CC=C(C)C)=O)C)C2)O)c(F)cccc1Cl C1(C(=O)N(C)CCNC(N)=O)(NC(C(c2ccn(C)c2)C)=O)CCCC1 c1(N2CCC(NCc3cc(OC)nc(C)c3)C(C)C2)ncc(C#N)cc1C N1(C(CC(c2ccc(C)cc2)C)=O)CCC(NC(=O)CCc2cccs2)CC1C c1(C(=O)NCC2(NC(C34CCCC3CC4)=O)CC2)ccc2ncncc2c1 Cc1ccc(S(C)(=O)=O)cc1CN1CCN(C)CC1c1cccc(C(F)(F)F)c1 CCC(CC(=O)NCC1(C)CCCN1C(C1CC(=O)NC1(C)C)=O)C(F)F c1(SCC(C)C)nc(Cc2ccccc2)nn1-c1ccc(Cl)nc1 c1(CCC)nc(Cc2cc(C(F)(F)F)co2)n(-c2ccccc2)n1 Cc1nc(CC2CC2)oc1C(=O)NCC=C1CCN(C(c2cccnn2)=O)CC1 N1(C(COCCOC)=O)CCC(CC)CC1.C1C(=O)N1.C(N)(=O)NCN c1(C(=O)NC2(C(C)NC(C(CSC)OCC)=O)CC2)ccc(C2CC2)cc1F c1(C(=O)NC2CCC(N(C(Cc3c(C)n[nH]c3C)=O)C)C2)c(C)oc(C)c1C c1(C(C)C(=O)NC2COCCC2NC(C2CSCCS2)=O)ccc(Cl)c(F)c1 C(=O)(C(CN(C(=O)C(=Cc1ccco1)C)C1CC1)C(C)C)N1CC(C=C)(O)C1 c1(OC)cccc(C(N2CCN(C(c3ccc(Cl)s3)=O)C(C(C)C)C2)=O)c1N c1(C(=O)NC(CNC(c2cc(C(C)=O)on2)=O)(C)C2CC2)cc2cccnc2s1 C(C1COC1=O)OC.C=C1CC(N(C2CCC2)C(C)=O)C1 C(=O)(CC1CCNc2ccccc21)N1C2N(C(CCCCC)=O)C(CC2)CC1 c1(C(=O)NC2CCN(C(c3n(C)ncc3)=O)CC2)cccc(Cl)c1[N+](=O)[O-] C(=O)(CCCC(=O)N(C)CC1CCCN(C(=O)Cc2cnns2)C1)NC(C)C N1(C(CCOCCC)=O)CCN(C(c2c[nH]cc2CC)=O)CCC1C C1(NC(c2ccc(CC)o2)=O)CCN(C(c2sc(SC(F)F)nc2C)=O)CC1F c1(-c2ccc(NC(c3cc(C)n(C)c3C)=O)cc2F)c[nH]c2cccc(F)c12 c1(O)ccccc1-c1nc(Cn2nccn2)n(-c2nc(C)nn2C)n1.C1(SCC)CC1 c1(OC)cccc(CC(=O)C(N2CCCCC2C)C2CCCOC2)c1.C1CCNO1 C(=O)(C(C)C(=O)OC)N(CCCNC(c1ccsc1OC)=O)CC C#CCC(CC#C)C(=O)N1CC2CC2(NC(=O)CCn2cncn2)C1 C1(C(N2C(CSC)CCC2)=O)CCN(C(=O)C=Cc2cscn2)C1C C1(C#N)(C(N2CC(CCNC(CCCSC)=O)OCCC2)=O)CC2CCC1CC2 c1(C(=O)NCCN(CCC)C(C2(N)CCC2)=O)cc(C)n(C(CC)CC)n1.C1(C)CC1 c1(NC(C2C(CNC(C3C(CC)CCO3)=O)C2)=O)cc(C)cnc1O CCCCCCCN(C(=O)CC1CCCN(C(c2c(C)noc2C)=O)C1)C N1(C(CSCC#C)=O)C2CCC1(CNC(=O)C(CN(C)C)N(C)C)CC2 C1(CNC(CCC(=C)Br)=O)CN(C(C2CCC(=O)C2)=O)CCC1(F)F Cc1cc(C)cc(C=CC(=O)NC(C(C)NC(c2ncsc2C)=O)C(C)C)c1 N1(C(C=CSC)=O)CCN(C(C2CC2OC(C)(C)C)=O)CC(C)C1 N1(C(Cc2c(C)nsc2)=O)CC2CCC(C(=O)O)(C1)C2(F)F c1(C(=O)NC(C2(O)CCN(c3cc(CC)ncn3)CC2)C)ccc2[nH]ccc2c1 CCCC(C(=O)NCCC(=O)NCCn1cnnc1)OCC C1(CC)CCN(C(=O)CC(C2CC2)NC(=O)CCn2ccnn2)CCO1 CCS(=O)c1ccccc1C(=O)N(CC(CC)NC(C1CC(OC)C1)=O)C c1(C(=O)NC2CC(F)(CNC(C3CC(C)C3)=O)C2)ccc(C(F)F)cn1 c1(C(C(C)C)NC(=O)NCc2ccc(CC)o2)ccc(F)cc1 c1(C(N(C(C)CCNC(=O)CC2(C)CCOCC2)C)=O)ccc(O)cc1[N+](=O)[O-] C1(C(=O)NC(C=C)COC)(CC)CCN(C(C2CCN(CC)C2)=O)C1 C1(NC(c2nc(CCC)oc2)=O)CCCCN(C(c2cc(OC)ccn2)=O)C1 C1(C(=O)NC2(CC(N3CCC3c3ccccc3)=O)CC2)CC1C1CC1 CCS(=O)(=O)CC(=O)N1CC(c2ccccc2)(NC(=O)Cc2nccn2C)C1 Cn1cc(C(N2CCC(N(C(=O)CC(F)F)CCO)CC2)=O)c(C2CCCO2)n1 C(=O)(NNC(=O)CCOC1CCOC1)NC(C1(CO)CC1)C.c1(O)ncco1 C1(NC(C2N(C(C)C)CCC2)=O)CCC2CCCC1O2.N12CC(OC(C)C1)C2=O C=CCN=C(NCC1C=CC2CC1CO2)N1CCC(OC(C)C)C1 N(C(=NCCCc1cccc(C2CC2)c1)NCC1CC1(C)C)Cc1cn(C)nn1 N1(c2cc(C)[nH]c(=NCC3CCCSC3)n2)CC(C2CCCN(S(C)(=O)=O)C2)C1 C1(CC)CN(C(=O)CC2(C)CCN2C(C2CCN2C)=O)CCO1 C1(C(=O)NCC(CC)NC(C2COC(=O)C2)=O)CCC(=O)NC1 c1(C(=O)NC2(CNC(C34N(CC(C)C3)CCC4)=O)CC2)cc2c(n1C)CCOC2 N1(C(C(C)c2ccsn2)=O)CC(NC(=O)Cc2cnn(C(F)F)c2)C(C)C1 c1(CCC(=O)N(C(C)CCNC(=O)COCCF)C)ccc(N(C)C)cc1 C(=O)(C(O)C(C)(C)C)N(C)CC1(NC(c2c(C)n[nH]c2)=O)CC1 CC1Cc2cc(Br)ccc2CN1Cc1cccn1C N(C(=NCCCC1CC2C=CC1C2)NC1CCOCC1)C(c1ncccn1)C CC(CC(F)(F)F)C(=O)NC1CN(C(=O)C(C2CCCCCC2)C)CC1C N1(CC(C)C)CC(N(c2ccc(F)cc2)C(=O)C(N2CC(C)(CF)C2)=O)CC1=O C12(NC(=O)COCC3CCCCO3)CCC1CN(C(=O)CCC1CCOCC1)C2 CC(C)(C)CCCC(=O)N1CC(F)(F)CC1C(=O)NCC1CC2(CCC2)CO1 c1(C(=O)NC(C(C)NC(C(CCC)CC2CCCC2)=O)C)cc2ccccc2o1 c1(OC)nc(Cl)ccc1C(=O)NCCC1CCCN1C(c1ccc(O)cc1F)=O N1(C(C(C)N(C)C)=O)CCN(C(=O)C=CC2(C)COC2)C(C)C1 c1(C(=O)NC(CN(C(CCCC)=O)CC)C)ccc2c(c1)OC(F)(F)O2 C1N=C2NC(=NC(C)=C2F)S1.N1(C(C2(COC)CC2)=O)CC(CN(C)C)C(C)C1 N=c1nc(O)c(CC(=O)NC2CC2CNC(C2(C(N)=O)CC2)=O)c[nH]1 C1(CC(=O)NC(CCC=C)C2CC2)C2CCCC2N1C(C1CC2CCCC2C1)=O C12CN(CCO1)C(c1ccc(Cl)o1)C(=O)N2.C1(NS(C)(=O)=O)CCCCC1 N1(C(CC(C)SC)=O)CCC(C)C1CNC(C1CC=CCC1)=O N1(C(CCCCC)=O)CCOC(C)(CNC(C2CCCC(F)(F)C2)=O)C1 C1(C(=O)NCCC2(CNC(=O)C3=C(Cl)CCC3)CC2)CCCC2(CCCCC2)C1 N1(C(C=C(C)CNC(c2ccn(C)c2)=O)=O)CCc2cc(CO)ccc2C1 C1(NC(CCC2CC(C)C2)=O)CC(O)C1CC(=O)NC1CCSCC1 c1(C(=O)NC2CC(N(C(c3ncc(CC)cn3)=O)C)C2)cc(Cl)c(N)c(Cl)c1 N(C(=NCCn1ccnc1)N(C)CC(c1ccccc1)OC)CC1(N(C)C)CC1 C1(CN(C(Cn2c(C(C)C)ncc2)=O)C)CCCN(C(=O)C(F)C2CCC2)C1 c1(CC)ccc(NC(C2CCC(C)N(C(=O)C(c3ccn(C)n3)C)C2)=O)cc1O CN1CCC(C)(C(N2CCOC(C(=O)NCCn3cnc(CO)c3)C2)=O)C1 N1(C(C(OC)OC)=O)CC(CC(=O)NCc2cccnc2C2CC2)C2(CC2)C1 N1(C(CS(CCOC)(=O)=O)=O)CCN(C(C23CC(C)(C2)OC3(C)C)=O)CC(O)C1 c1(C(=O)NCCN(C(C)C)C(C2CC3C=CC2CC3)=O)cncc2nc[nH]c12 Cc1ccc(Br)cc1CCC(=O)NC1CCN(C(=O)C=CCF)CC1CO CCC(C)C(O)CC(=O)N1CCC2C(NC(=O)COC(F)F)C2C1 CCC(C)C(C)CNC(=O)NCC1(N2CCCC2)CCCCC1 C(=O)(C(C)(O)CCc1ccccc1)NC1C(CNC(c2c(C)ocn2)=O)C1 N1(C(COC)=O)CCC(NC(=O)Cc2sccc2C)C(O)C1 C1(C)(C(=O)NCC2CC(NC(C=C(C)Cl)=O)C2)Cc2ccccc2N1 c1(OC)cc(CN2CCSC(CNC(=O)OC(C)(C)C)C2)ccc1S(C)(=O)=O c1(-c2ncc(C(=O)NC(COC)C)nc2)cnc(F)c(OC)c1 CC(C)CS(=O)(=O)CCC(=O)NC1(C)CCN(C(=O)CCCc2cnn[nH]2)C1 CC(C)C(C(=O)NC(C)CCN(C)C(C1C2CCC1CC2)=O)Nc1ccccc1 CCC(C)(CO)C(=O)NCCOCCN(C(=O)C(C)(C)c1cnn(C)c1)C Cc1sc(C)c2sc(C(=O)NC(CNC(C3(CC4CC4)CC3)=O)C3CC3)cc12 c1(N2C(C)CCC(NC(=O)CSCCN(C)C)C2)ccc(S(C)(=O)=O)cn1 CC(C)S(=O)(=O)CC(=O)NC1CC(NC(c2ccc(F)o2)=O)C12CCC2 C1(CCC=C)CCCN(C(=O)CCC2CCN(C(=O)Cc3nonc3C)C2)C1 N1(C(COC(C2C(C(=O)OCC)C2)=O)=O)CC(NCC)CC1c1ccccc1.OCC CC1(C)CN(C(C2CC3CCC2C3)=O)C1C1CCN(C(C2CSC2)=O)CC1 C(=O)(C(F)CC(C)(C)C)NC(CC#CC)C(=O)NCc1snnc1C c1(CC(N2CC(CC=C)(NC(C3COC(=O)N3)=O)C2)=O)cc(F)cc(Cl)c1 C1(=O)CCC(F)(F)Cn2cc(nn2)C(C)N1C.N1(CCC(C)CO)CCCCC1=O c1(C(=O)NCCC(C)(C)NC(CCC(C)OCC)=O)cccc(O)c1Cl CC12CC(C(N3CCCC(N4CCOCC4)C3)=O)(C1)OC2CO C(=O)(C(O)CC(C)(C)C)N1CC(CNC(C(c2ccccc2F)OC)=O)OCC1 N1(C(c2[nH]cc(C)c2)=O)CCC2CCN(C(c3cc(CN(C)C)c[nH]3)=O)CC12 CC1(C)CCC(C(=O)NCc2ccncc2)CN1C(C1CC2(CCC2=O)C1)=O c1(CNC2CC(NC(CNC(CCC)=O)=O)C2)cc(OC)cc(Cl)c1O c1(CC(=O)NCC(CCC)NC(c2cnn(C)c2C#N)=O)cccc(C)c1C c1(C(=O)NC(C(C)NC(C2(C)CCN(C(C)=O)C2)=O)CO)ccc(C)c(Cl)c1N C1(C(=O)NC2CN(CC)C2)CC(F)(F)CN1C(=O)CCN=[N+]=[N-] c1(OC)cc(CN2CCN(CCOC3CCOC3)CC2)ccc1OC N1(C(c2c(C)cco2)=O)CCC2CCCC(C1)N2c1c[n+]([O-])ccc1[N+](=O)[O-] O=S(=O)(c1ccc(O)cc1)NC1CN(Cc2cccn3nccc23)CC1F C(=O)(C1=CCOCC1)NC(C)Cn1cc(CN(S(=O)(=O)C2CC2)CC2CC2)nn1 C(CCC(c1nnnn1CCOC)NC1CC1(C)C)OCC C12CCN(C3(CCCC3)C1)C2.N1(S(C)(=O)=O)CCCN(C2CCC2)CC1=O C(C(=O)NC1CCCO1)(C1=CCCCCCC1)N1CCCC(COC)(CO)C1 CC1CCN(C(=O)Cc2nc(C(C)(C)C)cs2)CC1CNC(=O)C(F)C(F)(F)F N1(C(C(C)C)=O)CCOCC12COCCN(C(=O)CC1CC3CC3C1)C2 c1(C(N2C(C)CC(NC(c3cccc(CC)n3)=O)C2)=O)ccc2ccn(C)c2c1 c1(CN2CC3N(C(c4c(OC)ccc(F)c4)=O)C3C2)cc2cccnn2c1 C1(CC(=O)NCCCN(CCC)C(c2cc(C)cc(O)n2)=O)OCCCC1(C)C Fc1ccc(-n2nc(C3CCCCC3)nc2-c2c[nH]nn2)cc1 N1(C(CSC)=O)CC(C(=O)NC(CCO)C2CCC2)CC1(C)C C1(CC)CC(C(=O)NC2CCN(C(=O)C(c3ncccc3C)(F)F)CC2)CCO1 c1(NCC(CNC(C=Cc2c(C#N)cccc2)=O)O)ccc(F)cc1[N+](=O)[O-] C(=O)(C(=O)NNC(=O)CC1CCCCC12CC2)NC(C)CCSc1ccccc1 C1(NC(c2cnc(S)nc2)=O)CCN(C(=O)Cn2cncn2)CC1O C1(C(=O)NCCN(C2CCCC2)C(c2c(C)cc(CO)o2)=O)CCCNS1(=O)=O c1(C(=O)OCC)ccc2c(c1)C(NC(=O)C(N1CC3CCC1C(CO)C3)=O)CC2 CC1CN(C(c2cnsc2)=O)CC(CCNC(=O)COC2CCC2)O1 N1(C(c2c(NC)cnnc2)=O)CCC2(CCC(NC(=O)C(C)CO)C2)CC1 C1(NC(CN(CC)CC)=O)CCC(C)(CNC(c2coc(C)c2)=O)C1 N1(C(C(CC(C)(C)C)O)=O)CCN(C(=O)CCC(=O)N(C)C)CC2(C)CCCC12 C1(c2nnnn2C2COC2)(NCC23C(C)(C)C(CC2)CC3)CCOC2(CCC2)C1 Cc1cc(O)nnc1C(=O)NC(C1CN(C(c2cccc(CO)c2)=O)CCO1)C c1(CN(C)C(=O)NCc2cc(CC3CC3)on2)ccc(N2CCCCC2)cc1 C1(CNC(c2cc(CO)[nH]n2)=O)COCCN(C(c2ccc(Cl)s2)=O)C1 N1(C(C(CC#C)C2CC2)=O)CC(NC(c2sc(OC)nc2Cl)=O)C(S(C)(=O)=O)C1 N1(C(COCCN(C)C)=O)CCC(C2CCN(C(c3coc(C(F)F)c3)=O)C2)C1 c1(C(=O)NCC(CC=C)NC(=O)C2CC2)ccc(S(=O)(=O)Nn2nccn2)cc1 c1(CNC(=O)CNCC2(C)CCCN(C(C(C)C)=O)C2)nnc2n1CCCCC2 C1(NC(c2cc(CC)co2)=O)COC2CN(C(=O)C(C)OCC3CC3)CC12.CC C1(NC(CC(C)C2CC2)=O)CCCCC1n1ccnc1.C12CC(C1)NC(=O)CO2 c12cc(n(C)n1)NC2=O.CCC(C)C(=O)Nc1cnn(C2CN(C(C)=O)C2)c1 C1(C(N2C3(CN(C)C3)CC2)=O)CCN(C(c2c[nH]ccc2=O)=O)C12CCC2 C(=O)(CCC(C)CC)NC(CC=CC)C(=O)NCCCC1CC(C)C1 C1(CNC(C2(CC)CC2)=O)CN(C(c2csc(C3CCCCC3)n2)=O)CCC1C Cc1cc(-c2nc(NC(=O)C(c3ccccc3)C)cs2)c(C)cc1Br c1(C(=O)OC2COC3CCCCC23NC(=O)OC(C)(C)C)cc2c(cc1N)CCC2 C=CCCCCCC(=O)NC1CC(C(F)F)(NC(c2ccc(O)cc2F)=O)C1 C1(C(C)C)C(NC(c2cc(O)n(C)n2)=O)CCN1C(c1coc(C2CCC2)n1)=O NC1CC2(CCN(C(=O)NC3(O)CCC3)CC2)Oc2ccccc21 CCC(C)C(O)C(=O)N1CC(O)(CCNC(C2CC2c2ccccc2)=O)C1 c1(C(CNC2(C#C)CCOC2)=O)ccc2cc(Br)ccc2c1 C1(NC(C2(F)CCN(C(c3ccc([N+](=O)[O-])[nH]3)=O)C2)=O)CCCOC12CCC2 N1(C(CCC(=O)OC)=O)C2CC=C(C(=O)NCC34CCCC3OCC4)C1CC2 n1(C(C(=O)OC(C)C)C)c(CCNC(=O)CC2CCC(=O)N2)nc2ccccc12 C1(C(=O)NCCC2(NC(c3nsnc3O)=O)CC2)CC2CC1CC2(F)F C(=O)(CCCN=C(NCCNC(=O)C1CC1)NCC12CCCC1CC(=O)N2)NC N1(C(C2CC(=C3CC3)C2)=O)CCN(C(C23CCCC2C3(F)F)=O)C(C2CC2)C1 C12(CCNC(c3c(C)cnnc3)=O)CCC1CN(C(=O)C#CC1CC1)C2 N1(C(C(COC)OC)=O)CC(O)(C2(CNC(C3(C)SCCCS3)=O)CC2)C1 N1(C(=O)CCSC(F)(F)F)CC2CC(C1)N2C(c1ccc(F)cc1F)=O C1(C(N2CC(OC3CCN(C(CCCC#C)=O)CC3)C2)=O)CC2CC1CC2(F)F c1(CCOC)nc(=NC2(CO)CCCN(C(=O)C(C)CC3CCC3)C2)s[nH]1 N1(C(C(CCSC)O)=O)CCCC2(NC(c3cn4ccnc4s3)=O)CC2C1 c1(C(=O)NC(C2CCCCN2C(=O)CSC(F)(F)F)C)cc(F)cnn1 C1(C(=O)NCC2CCCN(C(c3cc(Br)sc3)=O)C2)CCC2CC1CO2 Cc1ccc2ncc(C(=O)NCCC3CC(NC(=O)C(C)(C)CF)C3)c(=O)n2c1 N1(C(=O)OC(C)(C)C)CC2(CNC(C3(C)CCNC3=O)=O)CC2(C)C1 c1(C(N2CCC3(C2)CN(C(C24C(=O)C5CCC2C45)=O)C3)=O)cc2cccnc2[nH]1 C1(CNC(c2cncc(C)c2)=O)C(C2CC2)CCN1C(=O)C1=CCC1 C(=O)(CCCCC(=O)OC)NC(C(CC)C)C(=O)NCC12CCCC1C2 Cc1nc2c(CCCNC(=O)NCC34CCCNC3C4)cccc2o1 C1(CC(=O)NCCC2CC(NC(C3C(C(C)=O)CC3)=O)C2)CCN(C)C1=O C1(NC(C(C)C2CCC2)=O)CN(C(=O)CC=Cc2cccc(F)c2)C2(CCC2)C1 S(=O)(=O)(c1cnn(CC2CCC2)c1)N1C(CC(C2CCCCCC2)C)CCC1 C1(OC)CC(CNC(=O)CC2C=NN(C)C2=O)N(C(c2n[nH]c(C3CC3)n2)=O)C1 C1(C(=O)NCCC2CC(N3CCOCC3)C2)CCCN(C(C2CCCN2)=O)C1 N1(C(CC(C)(C)O)=O)CCCCC(NC(=O)C(F)(F)C2CC2)C1 C(=O)(C(C(F)(F)F)C(F)(F)F)NCc1ccc(-n2c(C)cnn2)cc1 N1(C(C2C(CC)C2)=O)CCN(C(c2cnn(-c3ccc(F)cc3F)c2)=O)CC1C C12(CNC(c3c(CC)csc3)=O)CCCC1CN(C(c1cc(O)nc(Cl)c1)=O)C2 C(C(=O)N1CC(O)CCO1)CCC1CCN(C(c2c[nH]ccc2=O)=O)CC1 C#Cc1ccc(Cl)c(C(=O)NCC2CN(C(=O)C=Cc3ccccn3)CC2O)c1 C1(C(=O)NCCN(C(CN(CCOC)C)=O)C2CC2)CC(NC(C)C)C12CCC2 c1(C(=O)NCC2(F)CN(C(c3c(C)nc(C4CC4)s3)=O)C2)cnc2sccc2c1 C=C(C)CC(C)C(=O)NCC(O)CNC(c1cnc(-c2ccccc2F)nc1)=O c1(C(CC)NC(=O)Cc2ccc(Cl)s2)ccc(CCC2CCCNC2)cc1 Cc1ccc(C=CC(=O)NCC2CCC(C(=O)NCc3cc[nH]n3)CC2)cc1 N1(C(c2cccc(CS(N)(=O)=O)c2)=O)CC(C2(NC(C3CCCSC3)=O)CC2)C1 C(CCC(=O)NCC1(CO)CC=CC1)(C(C)C)NC(CC=CC)=O c1(C(N2CCC(CCOC)(NC(C34CC(C3)C4)=O)C2)=O)cc(C(C)C)ccc1C C(=O)(CCCCCCCC(=O)NCC1CCN1C(C1CC2CCC(C1)S2)=O)OC C1(C(N2CCOC(CC(N3CCCC(CC(N)=O)C3)=O)C2)=O)(OC)CCOCC1 C1(C(N2C3(CN(C(c4c(C)snc4)=O)C3)CC2)=O)Cc2ccccc2O1 CC1=NS(=O)(=O)NC=C1C(=O)NCc1cccc(NC(c2occc2C)=O)c1 c1(-c2c(OC)cc(OC)nc2)cccc2c(C(=O)NC3CNC(=O)C3)[nH]nc12 N1(C(c2nc(C)c(C)s2)=O)CC2(CCOCC2C(=O)NC2COC(=O)C2)C1 N1(C(C(C)NC=O)=O)CCSCC1C(=O)NCC(=O)N(C)Cc1ccco1 c1(C(N2CC(NC(=O)C3=CSCS3)(CO)C2)=O)cnc2ccsc2c1 CC1CCCN(CCC(=O)Nc2cc(C(C)(C)C)cc(C(C)(C)C)c2)CC1 O=C(CCCCF)NCC1C2CN(c3nncs3)CC12.c1(C)ccc(CO)o1 Cc1nn(CC(=O)N(C)CCn2cc(-c3ccc(Cl)c(Cl)c3)nn2)c(=O)n1C c1(CC)c(C(N2CCCCC2CCNC(=O)CCSCC(C)C)=O)csc1C N1(C(CC(CC)NC(c2csnc2OC)=O)=O)CCN(CC)C(C)C1 c1(OC)cc(F)c(CC(N2CC(F)(CNC(=O)C(O)CC(N)=O)C2)=O)c(F)c1 Cc1c[nH]c2cc(C(N3CCN(C(C4CCC(C)O4)=O)CC3C(C)C)=O)ccc12 c1(CCC)nc(=NCC2CC2CNC(=O)CCC2CCCC2)s[nH]1 Cn1cncc1S(=O)(=O)NCC1C2COCC12.N12CCCC(C)(C1)C2 C1(NC(COC)=O)CN(C(=O)CCC2CC(F)(F)C2)CCC12CCOCC2 C1(C)(NC(C(CC)C)=O)CCN(C(=O)COCCN2CCCS2(=O)=O)CC1 C1(CC(=O)NC23C(CN(C(COCC#C)=O)C2)C3)Sc2ccc(Cl)cc2NC1=O c1(OCCC)ccc(NC(C2CC=CCC2)c2nnnn2C2CCCC2)cc1C n1(CC)ccc(C(=O)NC(C)CCN(C)C(c2cnc(CO)nc2C)=O)cc1=O N1(CC(=O)NC(C)CCCNC(=O)CC(=O)NCC(F)(F)F)CSCCSC1 c1(CC(=O)NCC2(C)CCN(C(C3(CCC)CC3)=O)C2)ccc(OC)cc1OC C1(C(=O)NCCCCC2C(C)C2)CCN(C)C1=O.C1(O)(CNC(CN)=O)CC(CO)C1 C1(NC(c2c(OCC)ccs2)=O)CCN(C(C2(O)CCCC2)=O)CC1C C1(N(C(=O)Cc2[nH]cnc2C)CCOC)CCN(C(=O)CSC(C)(C)C)CC1 Fc1ccc(CNC2CN(Cc3ncc(C4CC4)s3)CCO2)cc1F c1(CC)oc2ccccc2c1C(=O)NCCN(C)C(c1ncccc1O)=O c1(C(N(CC(C)NC(c2c(C(F)F)cccc2F)=O)C)=O)cnc2ccnn2c1 CC1CC2(CCN(C(=O)CSC3CC3)CC2)CN1C(=O)C(C)S(N)(=O)=O N1(c2nnn(C)n2)CC2(C)CN(C(=O)C(c3cccnc3)O)CC2(C)C1 c1(C(C)C)cc(C(=O)NCC=CCNC(c2ccc(F)cn2)=O)c(C(C)C)[nH]1 C=CCC(CC(=O)NCCC(O)C(F)F)NC(=O)C1=C(C)OCC1 N1(C(C(C)SC(C)C)=O)CCCCC1CN(C)C(c1cnn(C(C)C)n1)=O CCC(CC(=O)N1CCC(N(C(C2CC3C=CC2C3)=O)CC2CC2)CC1)OC c1(-c2cn(CC(N3CCN(C(C(C)C)=O)CC3)C)nn2)cc(Cl)ccc1Cl C1(NC(CC2C(CC)C2)=O)CCC(NC(=O)Cc2conc2C)C1 C1(c2n(C)cnc2)CN(C(c2cc[nH]n2)=O)CC1CNC(=O)CO CC1(C(N2CC=CC(NC(=O)CCCn3cccn3)C2)=O)CCC(F)(F)CC1 Cc1cc(Br)cnc1CN1CCC(F)(C(=O)NCc2nn[nH]n2)C1 N1(C(c2cn(CC)nc2C)=O)CCC(NC(c2cnc(C(F)F)s2)=O)C(CO)C1 C(=O)(C1CCC(=O)c2ccccc21)N1C2CC(CNC(C(C(C)C)O)=O)(OC2)C1 N1(C(C(N)=O)=O)CCc2ccccc2C(N)C1 c1(C(=O)NCC2C(CNC(=O)CC3CCOC3)C2)cccnc1S CCCCCCCCC(=O)NC1CC(CNC(c2cncc(NC)c2)=O)C1 c1(C(=O)NCC2CN(CC(=O)NC3CC(C#N)C3)C2)c[nH]ccc1=O Cn1nc(CNC(=O)CSCCC#N)cc1C(=O)NCC1CCCOCC1 Cc1cc(C(=O)N(C2CCC(NC(c3scnc3C)=O)CC2)C)c(C)s1 c1(C(=O)NCC(CC(C)C)NC(C(CC)(C)C)=O)cc(C)cc2c1NCCC2 N1(C(C2CCC(=C)CC2)=O)CC2CC1CN(C(C1CC(C)CC(=O)N1)=O)C2 Cc1c(NC(c2nc(C)c(C)s2)C)ncnc1N1CCOCC(CO)C1 c1(C(=O)NCCOCCNC(C2NS(=O)(=O)N=C(C)C2)=O)cccc2c1COC2 N1(C(C(C)C)=O)CCOC(CCNC(C2CC2C(C)C)=O)C1 c1(NC(c2c(C)cccc2Cl)c2nnnn2C(C)C)ccc2ccccc2c1 N1(C(C2(COC)CN(C(c3cc[nH]c3C)=O)C2)=O)CCC(O)CC(C)C1 C1(CNC(C2(C)CC(F)(F)C2)=O)CC2(CCN(C(C3COC3)=O)CC2)CO1 C(=O)(C1CCCc2ccccc21)NCC(CNC(c1oc(C)c(CO)c1)=O)CO C12(NC(=O)Cc3ccsc3)CC(C(=O)NC3CC(F)C3)(C1)C2 N(C1CC2(CCCC2)Oc2ccc(Cl)cc21)C(c1ccc2c(c1)OCCNC2)=O Cc1ccnc2c(C(=O)NC(C3CCN(C(=O)C(C)(C)CC4CC4)C3)C)cnn12 C1(CNC(C2(NC(c3c(C)nc(CC)o3)=O)CCCCC2)=O)CC2CCC1CC2 C(CCC(C)C(=O)NCC1CC1CNC(c1ccoc1S(C)(=O)=O)=O)OC c1(C(=O)NCCCCNC(C)=O)ccccc1-n1cc(-c2ncccc2F)nn1 C(=O)(C1COc2ccc(Cl)cc21)N1CC2CN(C(COCCOC)=O)CC2C1 C1(C(N2CC(C(=O)O)C2)=O)(NC(C2(COC)CCC2)=O)CCC1.C1(COC)CCCC1 CN1CCC(NC(C2CNC(=O)CN2C(c2ccc(F)cn2)=O)=O)C(C#N)C1 c1(OCC)cccc2[nH]cc(CC(=O)NCC(C)CNC(=O)CSCC)c12 Cc1ccc(OCC(=O)NC(C)CCNC(c2cn(CCF)nn2)=O)cc1 C1(C(N2C(CC(=O)OCC)CCC2)=O)CCCC(Nc2ccnn2CCO)C1 C1(C(N2CCC(C(N3C(C(=O)OC)CC(O)C3)=O)O2)=O)Cc2ccccc2C1 C(=O)(C1CCCc2cccnc21)NCC(C)(C)NC(CS(C(C)C)(=O)=O)=O C(=O)(C1=CC(C)(C)C1)NCC1CC(OC)CN1C(c1cn(C2CC2)nn1)=O C1(OC)CC(C(N2CCC(C(C)(C)C)C2)=O)N(C(=O)C(C)=CC(C)(C)C)C1 O=C(CCC(=O)C1CC1)NC1CCN(C(C2(c3cccc(F)c3F)CC2)=O)C1 C1(C(=O)NCC=CCNC(C(P(C)(C)=O)O)=O)CCc2ncnn2C1 C=C1COc2c(C(=O)NCC3CN(C(=O)Cc4cccnc4)C4CC34)cnn2C1 CCC(CC)CCC(=O)NC(CCN(C)C(c1cnc(C2CC2)s1)=O)C(C)(C)C N1(C(C=CCOCCOC)=O)CCC(C(=O)NC2CC(C)(CO)C2)C1 C=Cc1cnn(C)c1C(N1CC(CNC(=O)C(C#N)C(C)C)C(C(F)(F)F)C1)=O N1(C(c2c[nH]c(=N)o2)=O)CCCC(CN2CCN(C(C3CC(O)C3)=O)CC2)C1 N1(C(=O)OC(C)(C)C)CCC2(CO)CN(CC3(C(F)(F)F)CC3)CC2C1 Cc1c(Br)noc1C(=O)N(C)CC1(CNC(c2ccc(O)nc2)=O)CC1 N1(c2nc(C)nc(Cl)c2)C2CCC1CC(NC(=O)C(C)CN1CCOCC1)C2 C1(NC(CSC(C)(C)C)=O)CN(C(=O)NC2CC(n3cccn3)C2)CC1C1CC1 C=CC(CC)CC(=O)N1C(=O)CN(Cc2ccc(Cl)cc2F)C1=O c1(C(=O)NCCCN(C(c2c(CC)con2)=O)CC)ccc(C)c(S(N)(=O)=O)c1 c1(C(N(C)CC2CCN(C(CN(C3CCCC3)C(C)=O)=O)C2)=O)ccnc(C)n1 CC1(NC(=O)NC2CCC(C(F)(F)F)C2)CCCC2(CC2)C1 C(=O)(CCCC(=O)OCC)NC1(CCC(=O)N(CC(=C)C)C)CCCCC1 Cc1oc([N+](=O)[O-])cc1C(=O)NC1CCC1NC(=O)C=CC(C)C C1(CC(=O)NCCC(C)CO)OCCCC1(C)C N1(C(c2c(C)onc2)=O)CCC(CCCNC(=O)C=CCN(C)C)CC1 C1(NC(C(C(C)(C)C)O)=O)CCC2(CC1)CC(NC(C1(C)CC(=O)N(C)C1)=O)C2 C1(C(C)(C)C)CN(CCSCCCNC(=O)C)CC12CC2.c1ccc(N)cn1 N1(CC=C)CCCN(C(=O)C(C2(C)CC2)NC(=O)CN(C)NC(=O)C(C)C)CC1 c1(OC)ccc(C=CC(N2CC(NC(=O)CCCOC(C)=O)CCC2C)=O)cc1 CC(N=c1cccc(S(=O)(=O)N(C)Cc2ccncc2)[nH]1)c1ccnc(Cl)c1 c1(OCCC)ccc(C(=O)NC(CNC(c2csc(C)c2)=O)CC)c(OC)c1 c1(C(=O)NC2CC2Cc2ccccc2)nc2cc(Cl)cc(Cl)c2[nH]1 c1(CNC(CC=C)=O)cnn2c1CN(C(c1nc(C)ncc1Cl)=O)CC2 c1(C(=O)N(CC2C(NC(C(C)NC(=O)NC)=O)C2)C2CC2)cnccc1C#N Cc1ccc2c(C(=O)NC3CC(CCNC(=O)CC4CCC(C)O4)C3)coc2c1 C1(CCC)CN(C(c2cc(OC)nn2C2CC2)=O)CC1C(=O)NC1(NC2CC2)CC1 CN1CCN(CC(N2CCCC(CNC(C3C(C)(C)C3(C)C)=O)C2)=O)CC1 c1(NCC23CC(C(=O)NC4CCCC(C5CC5)C4)(C2)C3)ncnc2cnccc12 N1(C(c2ncc(C)nc2)=O)CCC2CCCC(C1)N2C(c1cc(C#N)c[nH]1)=O c1(C(CC)C)nc(C2CCCC(CS(C)(=O)=O)C2)n(-c2cccnc2C)n1 O=S(=O)(c1[nH]c(=NC2CN(CCC(F)(F)F)C2)ccc1Br)NCCc1cncs1 N1(C(c2c(C)ncs2)=O)CC2ON=C(CNC(=O)C(C)(C)N(C)C)C2C1 c1(C(=O)NCC2N(C(C(C)(C)SC)=O)CCC2)cnc2c(c1)CS(=O)(=O)CC2 Cc1nn(C)c2nc(C(N3CC(NC(=O)CCc4ccsc4)C3)=O)ccc12 c1(NC(COC)CNC(N2CC(c3ncn(C)n3)C2)=O)cc(F)ccc1O C1(C(N(C(CC)C)CCO)=O)N(C(=O)C=CCOC)CC12CCCC2 N1(CC2CCN(CC(=O)NCc3cc(C)on3)CC2)CCCCCC1=O N1(C(c2cnc(COCC)s2)=O)CC23CCCC2(C1)CN(Cc1ccccc1)C3 N1(C(c2ccc(C)c(C)n2)=O)CCCC2C1CCN2Cc1scnc1Cl N1(C(=O)NC(C)(C)C)CCC(NC(Cn2c(C)c(Br)cn2)=O)C(O)C1 N1(C(C)=O)CSCC1C(=O)NC(CC1CC1)C(=O)NCc1cnn[nH]1 N1(C(C(=O)N(C2(C#C)CC2)CC)=O)CCC(c2cccc(O)c2)CC1 c1(-n2cc(C3(C)N(C(C4C(=C)CC4)=O)CCC3)nn2)ccc([N+](=O)[O-])cc1F CCCCCC(C)(C)CNC(N1CCC(c2ccnc(OC)c2)C1)=O N1(C(C(COC)COC)=O)CC(C2CC2)(C(N2CCC23CCC3)=O)C1 C(=O)(CC(C)C(F)F)NC(CC)CN(C(=O)C(C1CCCCCC1)C)CC C1(NC(c2ccccn2)=O)CC1C1CCCN(C(c2csnn2)=O)C1 c1(N(C)CC2CCCN2C(=O)CCC2CCCCO2)cc(=O)n(C)cn1 C1(c2noc(C3CNCCO3)n2)(NC(=O)OC(C)(C)C)CC2(CCOCC2)C1 c1(NC(C(C)N(CCCNC(C(CC)=CC)=O)C)=O)ccc(Br)cn1 CC1C(N=c2[nH]c(=NCc3c(Br)cnn3CC(F)F)[nH]c3c2CSC3)CCCN1C C1(NC(C2CN(C(=O)C(O)C(F)(F)F)CC2(F)F)=O)CCC2(CC1)CC2 N1(C(C(C2CCC2)OCC)=O)CC2(CCOCC2)C1CC N1(C(c2ccc(OC)s2)=O)CC2CCN(C(=O)C(=O)NC3CC3)CC12 c1(CC(=O)NC(C)(C)C)cc(C)n(C)n1.C(CC(=O)NCCCN)=CC.C(CO)OC=O c1(CN2CC(C)(CC(=O)NC(CCCC)CO)C2)cnc(O)nc1O C12(CNC(=O)CCc3cocn3)CCC(CC1NC(c1ccc(Cl)o1)=O)C2 Cc1nc(C)c(C(=O)NC2CN(C(=O)Cc3nnn(C(C)(C)C)n3)C3CC23)s1 C(=O)(CC(C)C(=O)NCC1CC(F)(CNC(=O)C(CC)C(C)C)C1)OC N1(C(CC(=O)OC)=O)CC2(C1)SCCC2NC(C1CCCC(F)(F)CC1)=O C1(NC(c2c(O)ccc(C)c2)=O)CC(C(=O)N2CC=CC(O)C2)=CC1O Cc1oc(C(F)(F)F)nc1CNC(C1CC1C(=O)NCCC1CCCCCC1)=O c1(C(N2C(CNC(=O)CC3C=CS(=O)(=O)C3)CC2)=O)nn2cccnc2c1Cl C1(C(=O)NCCCC)CC(C)(C)CCN1C(=O)CC12CCC(CC1)C2 C1(NC(Cn2c(C)ccn2)=O)CCCN(C(c2ccc3c[nH]nc3n2)=O)CCC1 Cc1ncc(Cl)cc1C(=O)NCC(C)NC(=O)C1=NNC(=O)C1 O=C(N=c1cc2c(n[nH]1)CCC2)C1CCC2(CCOCC2)O1 C1(C(=O)NCC2C=CC(NC(=O)CCc3cnccn3)C2)CC2(C1)CS(=O)(=O)C2 c1(NCC(C)(C)CC2CCCCC2)nccc(=NCCS(=O)(=O)CCC2CC2)[nH]1 C1(NC(CN(C(C)C)C)=O)CN(C(=O)Cc2ncsc2Cl)CCC1O C1(C(N2CC3(CC(NC(=O)C4=CCSC4)C3)C2)=O)CCCC2(CCC2)O1 N1(C(Cn2c(C)cc(C)n2)=O)CCC2(CCC2NC(=O)CN2CCC(C)C2)CC1 c1(C(N(CC(CN(C(CCc2nc(C)c(C)o2)=O)C)O)C)=O)cn(C)ccc1=O N1(C(C(C)(C)C)=O)CC(NC(c2cscc2C(F)F)=O)CC12CCCC2 C=C(C)CCCC(=O)NCC1CCCCN1C(=O)CC1COCC1(C)C C1(C(=O)NCCN(CC)CC)CC(NC(c2cnc(O)o2)=O)C1(C)C C12(C(=O)NCC(CN(C)C(c3csnn3)=O)(C)C)CCCC(=O)N1CCC2 N1(C(c2c(C)ncn2C)=O)CC(F)(F)CC1(C)CNC(=O)Cc1cccs1 c1(C(=O)NC(C=CC(=O)N(C(COC)C)C)(C)C)cnn(C)c(=O)c1 Cc1cc(C(CNC(c2ccnn2C2CCCCC2)=O)N(C)C)cc(F)c1 N1(C(c2c(C)nns2)=O)CC(C(=O)NCCc2cccnc2O)CC(C)(C)C1 N1(C(CCOCC#C)=O)CC(NC(C23CC(COC)(CO2)C3)=O)CC(O)C1 CC(CC(C)NC(C1CC(C)(C)C1)=O)NC(=O)CSCCC#N C1(CC)C(C(=O)NCC2(F)CN(C)C2)CCN1C(=O)C=Cc1nccs1 c1(C(C)N(C(c2cnc(C3CC3)nc2)C(=O)NCC2CC2)C)ccccc1F N1(C(=O)NCCC=CCCC)CCC(O)(C(=O)OC)C1 c1(NC(C2(C#C)CN(C(C3COCCO3)=O)C2)=O)ccc2c(c1)COC2 C1(C(N(CCC)CCC(=O)NC2(C)CCN(C)C2=O)=O)COCCC1(F)F c1(-c2cn(CC3C(NC(=O)Nc4ccc(Cl)cc4)CCC3)nn2)cncc(F)c1 c1(N(C(c2ccnc(Cl)c2)C(=O)NC2CCOC2)CC)ccc(O)cc1C C(=O)(CCC(O)Cc1ccccc1)NCCOC1CN(C(CS(=O)(=O)NC)=O)C1 N1(C(C2CCC(n3cc(CC(=O)OC)nn3)C2)=O)CCc2nc(C)ncc2C1 C1(C)(NC(COC(c2ncc(C)[nH]2)CC)=O)CCN(C(=O)CCCC(C)=O)CC1 Cc1c(N2CCOC(c3cccnc3)C2)ncn2ccnc12 c1(CNC(C2(C)CC3CC3C2)=O)nc(CNC(=O)Cc2ccncc2)cc(O)n1 c1(C(=O)NCC2(O)CN(C(CC(C)(C)OC)=O)C2)c(C)c(C)nc2ccccc12 CCCCC(O)C(=O)NC1(C)CCCN(C(=O)C(O)Cc2ccccc2)C1 c1(C(=O)NCCCCC(CO)NC(C(CCN(C)C)O)=O)cc2ccncc2[nH]1 O=S(=O)(c1c[nH]ccc1=NCC1CCCS1)NCCc1nnc2n1CCCCC2 C1(C(N2CC(F)(C(=O)Nc3ccc(CC)cc3)C2)=O)OCCCC1(C)C N1(C(C(C)SCCCC)=O)CCC(NC(c2cc(OC)n[nH]2)=O)C2(CCC2)C1 c1(C(=O)NC2(NC(C(COC)NC(C)=O)=O)CCCCC2)nn(C)c2c1CCC2 N(C(=NCCc1ccccc1)NC1CCCCCCC1)CC(F)F c1(C)ccc(C(F)(F)F)cn1.N1(NCC(O)CO)CCC(C)C1 CCCCC(C)C(=O)N(CC(C)(C)CNC(C1(C)CCN(C(C)=O)C1)=O)C C(=O)(N=c1cc(Cl)n(C)[nH]1)c1c(Nc2nc(SC)nc(C(F)(F)F)c2)cccn1 N1(C(COCC)=O)CCN(C(C2CCC2)=O)C(c2cn[nH]c2)C1 C1(C(NOCC(=O)NCCCS(=O)(=O)C2CC2)=O)CC(=O)NC(=O)C1 C1(C(=O)NC2N(C(c3ccc(OC4(C)CC4)cc3)=O)CCC2)CCCCC12CC2 C12(CCCC1C)C(=O)N2C1CC1.Cc1ncsc1CCNC12CSCC1C2 c1(C(C)C)ncc[nH]c1=NCC1(C)CCC(NC(=O)C(C)OC2CCCC2)CC1 CS(=O)(=O)c1ccc(C(=O)NC2C3CN(C(C4CC=CCC4)=O)CC23)s1 C(=O)(C#CC(C)(C)C)NC(C1CCCN1C(=O)CCc1cnoc1)C Cc1ccc2c(=NCC3CCSC3(C)C)[nH]c(N(CCC(C)(C)C)C)nc2c1 C1(C(N(C)CCNC(C2(C(F)(F)F)CC2)=O)=O)CC(=O)N(C2CC2)C1 N(C(=NCC1CCOC1)NC1C=CCCC1)C(C)CF C1(C(=O)NCC(CCC)NC(c2cn(CC)nc2C)=O)CCCOCC1 C1(NC(C2(O)CCC2)=O)CC(NC(C2(CO)CCCC2)=O)C12CCC2 C#Cc1cccc(NC(CC2CC(CC(=O)NCC3(O)CC4CCC3C4)C2)=O)c1 c1(C(=O)NC(C)CN(C(C)C(=O)NC)C)cc(F)cc(Cl)c1.Cc1nnn(C)n1 CCC(C)C(C(=O)NCC1CC(F)(F)C1)N1CCCCC1CC CC1CCc2nc(C(=O)NCC34CC(CN3C(=O)CC(C)N(C)C)C4)cn2C1 C(=O)(C(O)CC(C)(C)C)N1CC(CCOC)N(C(=O)C=CCO)CC1 CC1ON=C(C(=O)N2CCC(C3CC3)C2CNC(=O)C2=NOCC2)C1C N#Cc1c[nH]c2ccccc2c1=NCC1CN(C(c2scnc2Cl)=O)CCO1 C12(OC)CN(C(c3cccc4c3OC(C)(C)C4)=O)CC1CS(=O)(=O)C2 c1(C(=O)OCC2CCC(C(F)(F)F)CC2)cnc(N2CCOCC2)cn1 C(=O)(C1CCCc2ccnn21)NCC12CC(NC(C(CC)N(C)C)=O)(C1)C2 CC1=C(C)CC(C)(C(N2CCC3CN(C(c4ccc5c(c4)CC5)=O)CC23)=O)CC1 C1(C(C)(C)NC(=O)CSC(=N)N)CCN(C(=O)CO)C1 c1(C(N2CCN(S(CCC)(=O)=O)C3C2C3)=O)c(C)ccc(Br)c1C C(=O)(CCCCC#N)N1C(C(C)NC(C2CCCCC2O)=O)CCC1 Cc1cn(C)cc1C(=O)NC1(C(N2CC(C(C)C)C2)=O)CCSC1 CC1(C(N2CC3(NC(=O)C4=CCCC4)CCC2C3)=O)CC(c2ccccc2)=NO1 C(CC)(CC)(CCNC(=O)CS(=O)(=O)NC1CC1)NC(C(CC)C)=O c1(CC)cncc(C(N2CC3CC2(C(=O)Nc2cccc(N(C)C)c2)C3)=O)c1 C1(C(C)CNC(c2ccc[nH]2)=O)CCN(C(C2CC2C(F)F)=O)CC1 c1(NC(C2COCCN2C(=O)CCC2CC2)=O)cc(Br)cc2cn[nH]c12 c1(C(=O)NC(C(C)NC(=O)CCc2ccncc2)(C)C)c[nH]c2cc(O)ccc12 c1(OC)ccc(C(=O)NCC2CC2CNC(c2ccc(N(C)C)nc2)=O)c(C)n1 C1(NC(c2c(C)nncc2)=O)CN(C(c2cnc(Cl)c(F)c2N)=O)CC2(CC2)C1 n1(CC)nnc(C(N2CCCC2(CO)CNC(=O)C=Cc2cc[nH]n2)=O)c1C C12(C(=O)NCC3N(C(COC(CC)CC)=O)CCCC3)CCC(CC1F)C2 C1(CC(N2CCN(C(c3cc(COC)on3)=O)C(C)C2)=O)COc2ccccc2O1 C(C(C(F)(F)F)N1CCN(C(=O)CNC=O)CC1)NC(C1(Cl)C(C)(C)C1)=O CON=C(C(=O)N1CCCC12CCN(C(c1cccc[n+]1[O-])=O)C2)c1ccco1 C1(C(=O)NC(C(=O)OC)C)CCCN(C(=O)C(C)(CC)CO)CC1 c1(CC(=O)NCC(C(C)C)NC(C2CC(C)(F)C2)=O)ccc(N(C)C)cn1 Cc1ncsc1CCC(=O)NC(C)C(C)NC(=O)CC(O)C1CC1 C(=O)(C(O)CC(C)(C)C)NCC(C(=O)Nc1cn(C)c(=O)nc1O)N(C)C C(=O)(C1=CC2CCC=CCCC12)N1CCN(C(Cn2c(=N)scc2)=O)CC(O)C1 C1(NC(c2cn(CCC)nn2)=O)CC2CN(C(c3cc(C)c[nH]3)=O)CCN2C1=O C1(CNC(CCSc2n(C)ccn2)=O)COCCN(C(C2CC(C)(C)C2)=O)C1 N1(c2c3[nH]cc(CC)c3ncn2)CCC2(CC1)CC(C)=NO2 C12(CNC(C=C(C)Cl)=O)CC1CN(C(c1ccc(CC(C)(C)C)cc1)=O)C2 CC1CCC(NC(c2cc(O)n(C)n2)=O)CN1c1cc(=O)n(C)cn1 C(=O)(C1(C)CCc2ccccc21)NCC1CCCCN(C(CC(C)C)=O)C1 C1(NC(CCCSC)=O)CCC(C)(C)CC1CNC(c1nc(=O)n(C)[nH]1)=O C(=O)(CCCCCCCCC(=O)Nc1cc(C#N)ccc1C)OC C1(NC(C(CC)N(C)C)=O)COC2(CNC(c3scnc3C)=O)CC1C2 c1(C(N2CCC(C)C(O)C2)=O)cc2cc(Br)cc(Cl)c2[nH]1 c1(NC(C2OCCC(NC(CCCC(C)C)=O)C2)=O)cccc([N+](=O)[O-])c1 c1(C(=O)NCC(CCNC(C2N(C)CCOC2)=O)(C)C)cc2c(nn1)CCC2 c1(C(=O)NC2CC(NCc3ccsn3)C2)cccc([N+](=O)[O-])c1 C(=O)(C=CSc1nc[nH]n1)N(C)CCOCCCNC(=O)CC#N C12(C(N(CC(C)C)CC(C)C)=O)CCN(C(c3ccncc3Cl)=O)CCC1C2 C(N=c1[nH]c(=NCc2ccc(Cl)cc2F)c2ccccc2[nH]1)c1[nH]ccc(=N)n1 N1(C(C=CC2N(C(c3c(C)nn[nH]3)=O)CCC2)=O)CCN(CC(C)O)CC1C N1(C(c2c(CC)nco2)=O)CCC(NC(=O)CCC2CCCC2)CC1 C#CC1(O)CC(C(=O)NC(CCSC)C(=O)N2CC(CC)C(C)C2)C1 N1(C(C(CC=C)C)=O)CCCC12CCN(C(=O)CNc1nccs1)C2 C(N=c1[nH]c(=NCCCNS(C)(=O)=O)[nH]c2c1CCC2)C1CC(OC)C1 c1(C(=O)NC2CN(C(C(Cn3ccc(C)n3)C)=O)C(C)C2)cc(C)c(F)cc1N N(C(=NCc1ccsn1)NC(CN(C)C)Cc1ccccc1)C(C)C1CC1 c1(C(CC(=O)NC(C(CO)NC(c2c(CC)noc2)=O)C)O)ccc(F)cc1 C1(CC(=O)NCCCN(C(c2cccs2)=O)Cc2ccccc2)CCCC1(F)F C(=O)(C(C)CS(C)(=O)=O)NCCC1CC(NC(c2cc(C)on2)=O)C1 c1(C(N(CC(C)C(=O)O)C2CC2)=O)cccc(N(C)C)c1 Cc1ccc(C(=O)NCC(C2COC(C)(C)O2)CO)cc1S(C)(=O)=O c1(C(=O)NC(C2CN(C(c3nc(CC)sc3)=O)C2)C)cccnc1-n1cccn1 N1(C(CCCC=C)=O)C2CC=C(C(=O)NC(Cn3ccnc3)CO)C1CC2 c1(C(C)C)nc(NC(C2(C)CCCO2)C)cc(N(C)CCNC(C)=O)n1 c1(C(=O)NC2CC(NC(c3cc(N)c(F)cc3)=O)C2)ccc2oc(O)nc2n1 Cc1cc(C#N)cnc1C(=O)NC(C1CCN(C(=O)OC(C)(C)C)C1)c1cncs1 CC(C)C(O)CC(=O)N1CCC(CCC(=O)NC(C)COC(F)(F)F)C1 N(C1c2ccccc2CC1NC(c1nnn2c1COCC2)=O)C(C(CC)OC)=O C1(CN(C)C(c2cncn2C)=O)CCCC(NC(c2cn(C3CCC3)nn2)=O)C1 Cc1c(Cl)ccnc1C(=O)NCC1(NC(c2cnn(C)n2)=O)CCCCCC1 N1(C(C(C)(C)c2cccs2)=O)CC2(C1)CN(C(C1(Cl)CC1)=O)CC2CO C12(C(=O)NC3CC(N(C)C)C3)COCC1CN(C(c1ccc(Cl)o1)=O)C2 c1(C(N2CCC(N(C(c3nnn(C)c3C)=O)CC)C2)=O)cc2c(cn1)COCC2 C1(NC(C(CCF)NC(c2ccc(C#C)o2)=O)=O)CCOCC12CCC2 N#CC1=C(C(=O)NCC2CCCC2NC(C2CCc3n[nH]cc3C2)=O)CCC1 Cc1c(Br)ccc2c1CCN(C(=O)CN(CCCCN(C)C)C)C2 Cc1sc2ncc(C(=O)NCCOC3CN(C(C4C=CCC4)=O)C3)n2c1C CC(C(=O)N1CCC(C2CCCN2C(c2ccc(C(N)=O)o2)=O)CC1)C(C)(F)F N1(C(c2ccn(CCC)n2)=O)CC(CNC(=O)CC(C)(C)C(F)F)CC12CCC2 C12(NC(c3ccc(=NCC)[nH]c3)=O)CN(C(=O)C(C)(C)CO)CC1CS(=O)(=O)C2 c12nccc(n1)CO2.c1(CN(C(CCOC)=O)CCN(C)C)cccc(Cl)c1 C1(C(=O)NCCC(CC)(F)F)CN(C(=O)CCC(C)CN(C)C)CC1(C)C C(=O)(C(C#N)=CN(C)C)N1CC(C(=O)NC(CCSCC)C(=O)OC)(SC)C1 C=CC(C)(CC)C(=O)NCc1ccc(CN(C(=O)CCc2ccco2)C2CC2)cc1 c1(C2C(C)C2)ccc(F)cc1Cl.C12CCN(CC1)C(=O)C(C)N(C)CC2.CC(C)O Cc1cn(C)cc1C(=O)NC(C)(CO)C(=O)NCC1(O)CCC(C)C1 c1(C(=O)NCC2N(C(C3C(C)(C)OC(=O)C3)=O)CC(O)C2)cc(Cl)cc(Cl)c1N C=CCC(CC(C)C)C(=O)N1CCC(NC(=O)C2=C(Cl)CCC2)C1 C1(NC(CCC(C)C)=O)CC2CCC1CC2NC(=O)CCCCCF N#Cc1ccc2c(c1)N(C(=O)CC1(NC(=O)C(c3ccccc3)F)CC1)CC2 c1(OC)cccc(CC(O)C(=O)NCCCCCNC(=O)CCCNC(N)=O)c1 C(=O)(CCP(C)(C)=O)NC1(C)CC(C(N2CCC(C(C#C)C)CC2)=O)C1 N1(Cc2nc(CCC)sc2)CC2CCCN(C(c3cnc(OC)c(C)c3)=O)C2C1 c1(C(C(=O)N(CCC)CCNC(=O)COCc2ncc(C)o2)C)c(C)n[nH]c1C C1(C(C)(C)C)CN(C(=O)Nc2ccc(C3CC3)o2)CC1F N1(C(CCN(CCC)C)=O)CCC(NC(=O)CC2(CO)CCOCC2)C12CCC2 c1(C(=O)NC2C(C)CCN(C(C3(C)CC(C)(C)C3)=O)C2)cc(O)c2sccc2c1 C(=O)(C(C(C)NC(c1nc(C)ccc1C)=O)C(C)C)NCC(CC)(CC)OC c1(C(N2CCC(C)(CNC(C(C)CF)=O)C2)=O)ccc2c(c1)CCN2C C1(C(C(=O)N(C(CNC(C(C)OCc2ccccc2)=O)C)C)O)COC(C)(C)O1 N1(C(c2c(C)nc(CO)s2)=O)CCN(C(c2ccc(O)cc2Cl)=O)C(C)C1C CC1CCCC(CNC(C2C(C)CN2C(C2CCCN2C2CC2)=O)=O)O1 CC(C)CCC(=O)NCCC1CCCCN1C(=O)C(=Cc1c[nH]cn1)F Cc1cc(-c2cn(C(C)C(=O)NCC3CCC(O)C3)nn2)cc(C)c1 c1(C(=O)NC2C(C(=O)NCC(C)CC3CCCC3)C(O)C2)cc2ncccc2o1 CP(C)(=O)CCC(=O)N1CCC(C(CO)NC(=O)C=Cc2cnc[nH]2)CC1 C1(N(C(C2CCN(CC)C2)=O)C2CC2)CN(C(=O)C=C2CCC2)CC12CC2 C1(CNC(=O)C2=NOCC2)CN2CCCCC2CN1C(=O)CCC1CCOCC1 N1(C(C=C(CCC)C)=O)CCC(CCNC(c2ccc(OC)cn2)=O)(OC)C1 c1(C(=O)NC2C3CN(C(C(C)=C4CC4)=O)C2CC3)ccc2c(c1)CCN2 C1(CNC(C2=C(C)OCC2)=O)C(C2CC2)CCN1C(c1cc(N)ccn1)=O c1(C(N(C(c2cn(CC)nn2)C)C)=O)cc(Cl)ccc1C(F)F c1(CC(=O)NCCCC(C)NC(C(C2CCOCC2)OCC)=O)ccc(Cl)c(F)c1 C=CCC(CC=C)C(=O)N1CCN(C(C23CC2COC3(C)C)=O)CC1C1CC1 Cc1cccc(Cl)c1CC(=O)NCC1CN(C(=O)CCN2CCN(C)CC2)C1 N1(C(c2cc(C)cc(Cl)c2)=O)CCCC(C)(C)C1CNC(=O)COC1CCCC1 C1(CN(C(CCC=CC)=O)C)CN(C(c2noc(CC)c2C)=O)CC12CC2 C1(C(=O)NCc2cc(=O)cc[nH]2)CC2CC2N1C(=O)CCC1CCOC1 N1(C(c2c(O)cn(-c3ccc(C)c(C)c3)n2)=O)CCc2c(nc(Br)n2C)C1 c1(C(C)NC2CC(CC(=O)NC3(C(=O)OC)CC3)C2)c[nH]ccc1=O c1(C(=O)NC(C2CCN(C(c3ccncc3Cl)=O)C2)(C)C)cc2ncccc2o1 N1(C(c2n(CC)ncn2)=O)CCN(C(=O)C=Cc2ccccc2C)C2(CC2)C1 C1(C(N(CC(CN(C)C)O)C)=O)CCCN(CCCc2ccccc2)C1 c1(CNC(=O)NCC(c2cc(C)cc(C)c2)C)ccn2ccnc2c1 c1(C(=O)NC2(C(=O)NC3CC(SC)C3)CCC2)cnoc1C1CC1 c1(CN2CCC(N(C)C(C3CC3F)=O)C2)ccc2n[nH]cc2c1 c1(CC)cc(C(N2CC(NC(C3C4CCCCC34)=O)C(CO)C2)=O)c(C)o1 CCCCCCC(=O)NC1CC(CNC(=O)Cc2csc(COC)n2)C12CCC2 N1(C(CC2(CSC)CC2)=O)CCCC1C1(NC(=O)Cc2cnc(C)s2)CC1 C1(NC(CS(CC)(=O)=O)=O)CN(C(C2CN(C(C)=O)C2)=O)CC2(CCC2)C1 C1(C(=O)NC2C=CC(CNC(=O)CCF)C2)CCN(c2cc(O)ncn2)CC1 C(=O)(C(C)(C)CC(C)=O)NCc1c(C(=O)NCC(COC)(C)O)nccc1 c1(CC=C)ccccc1SC(C)C(=O)NCC1CCC(NC(=NC)N)CC1 C1(C)(CCC)CCN1C(=O)COC1CCN(C(=O)C(C)OCCOC)C1 c1(C(C)C)nc(NCC(C)NC(c2ccccn2)=O)cc(=NCC2CCCC2O)[nH]1 Cc1nn(C)c(=O)c(C(=O)NC(C)C(C)NC(=O)CC(C)N2CCCC2=O)c1C N1(CC(=O)NC(CC)CNC(c2ccc(SC(C)(C)C)cc2)=O)C(=O)CNC1=O CCN=c1[nH]c(C)c(C(N2CCC(N(C(=O)C=C3CC3)CC3CC3)CC2)=O)s1 N(C1COc2c(Cl)cccc21)S(CC1(C)CCOC1)(=O)=O C(CC(C(=O)NC1CC(C(F)F)(NC(C2CC(=O)N(C)C2)=O)C1)OC)OC C1(CNC(=O)CCC(F)(F)F)CC2(CCN(C(=O)CCCCC3CC3)C2)CO1 CC(C)C(C)CC(=O)NCCNC(C1(F)CC1(F)F)=O c1(C(=O)NCC2N(C(CCC=C(C)C)=O)CCC2C)ccc2c(c1)COC2 c1(OC)nsc(OC)c1C(=O)NCC1CCC(NC(c2cnc(C)n2C)=O)C1 C(=O)(CC(C)N(C(C1CC1C(C)NC(=O)Cc1cnc(C)s1)=O)C1CC1)OC N1(C(C2(OC)CCCOC2)=O)CCC(O)(C(C)NC(c2ccsc2C#N)=O)CC1 N1(C(C2CCN(C(CCC(=C)Cl)=O)C(CC)C2)=O)CCN2CC(C)CC2C1 N1(C(C2C(C)C(=O)C2)=O)CCC2CN(C(C3CC=CCO3)=O)CCC12 c1(OC)cnc(C(N2CCC(O)(C(C)NC(C3(CF)CCOCC3)=O)C2)=O)cn1 c1(CNC(C2CC(NC(=O)CC(O)c3ccccc3)C2)=O)ccc(O)c(F)c1 C(=O)(C(F)(F)C(F)(F)C(F)F)N1CC(CNC(C2(C)CC(F)C2)=O)C2(C1)CC2 c1(C(N2CCN(C(C3CN(C)C3)=O)CC23CCC3)=O)cc2ccccc2cc1O N1(C(c2ccc(CNC(=O)CCC3CCCO3)nc2)=O)CCc2ncccc2C1 N1(C(CC)C(=O)NCCCN(c2ncc(Br)c(O)n2)C)CCc2ccccc21 c1(NC)nccc(C(N2CC(OC)C(F)C2)C(=O)NCC2CC2)c1F.c1ccccc1 c1(C(=O)NCC2(NC(CC3C(C)C(=O)CC3)=O)CCCC2)cc[nH]c2nccc1-2 c1(CC(=O)NC2(CCNC(Cc3c(C)ncs3)=O)CCC2)ccnnc1O C1(CNC(C2(C(C)N(C)C)CC2)=O)CCCCC1NC(=O)CN1CCSCC1 N1(C(CCCNC(C)=O)=O)CCN(C(=O)CN2CCC(C)C2)CC2(CC2)C1 N1(C(c2ccc(CNC(c3nn(C)c(Cl)c3)=O)cc2)=O)CCC2(CCO2)C1 Cc1nn2cc[nH]c(=O)c2c1C(=O)NC(CNC(=O)Cc1cncc(O)c1)CO c1(OCC(=O)NCCCN(CC(CNC(C)=O)O)C)ncc(C(F)(F)F)cc1Cl S(=O)(=O)(C1CC2CCC1C1OC21)Nc1n(C)ncc1-c1ccc(Cl)c(F)c1 Cn1ncc2c(O)nc(=NCC(CNC(C3CCCC3O)=O)C(F)(F)F)[nH]c12 CC1C(NC(C2CN(C)CCN2C)=O)CCCN1c1nnccc1C#N c1(-c2nc(NC(=O)CNC(C3CC(F)(F)C3)=O)sc2)cc(O)cc(F)c1 c1(C(=O)NCC(C)=CC(=O)NCC2CC2Cl)c[nH]c(=S)cn1 C1(NC(CN(CC)CC)=O)CC2(CCCN(C(c3ccnc(S)c3)=O)C2)C1 c1(C(N(C)CC2N(C(c3cncc(C)n3)=O)CCOC2)=O)ccc(C)c(Cl)c1Cl c1(NC(c2c(C)noc2C)C=C)ccc(S(=O)(=O)NC(CO)CCC)cc1C#N c1(C(N2CCC(NC(c3nc(OCC)oc3)=O)C(F)C2)=O)ccc2scnc2c1 C1(C(=O)NC2(CNC(c3cc(CO)[nH]n3)=O)CCC2)CCCc2ccccc2C1 N1(C(C2C3CC2N(Cc2ccc4c(c2)CNC4=O)C3)=O)CCc2c(O)n[nH]c2C1 c1(C(=O)NCC2(O)CCCN(C(C=C(C)Cl)=O)CC2)[nH]c2ccc(Cl)cc2c1Cl CC1CC(C(=O)NCc2cn(CC(=O)NC3(C)CSC3)nn2)CC(=O)N1 c1(-n2cc(COC(C)C(=O)O)nn2)ccccc1C(N1CCCC1C(N)=O)=O C1(NC(c2cnns2)=O)CN(C(=O)CSc2cccc[n+]2[O-])C2(CCCC2)C1 c1(C(CC(=O)NC2C(NC(c3nnn(C(C)(C)C)n3)=O)C2)O)ccc(F)cc1 Cc1cccc(OCC(=O)NC(C)C(C)NC(C2(F)CC2Br)=O)c1C c1(C(=O)NC2C3CN(C(c4ccc(OC)o4)=O)C2C3)cc2cc(Cl)ccc2[nH]1 c1(C(N2C(CNC(c3ncc(OC)cn3)=O)CC2)=O)cc(OC)ncc1F c1(C(=O)NC(C2(O)CN(C(CN3C(C)CC3)=O)C2)(C)CC2CC2)cc(Cl)c(Cl)s1 c1(C(=O)NCCC(C)N(C(=O)CCC2CC2(F)F)C)cncc(-n2ccnn2)c1 Cc1ccnn1C(C)C(=O)NC(C1(O)CN(C(=O)C(O)Cc2[nH]cnc2C)C1)C N1(C(c2ccc(CNC(c3c(C)c(C#N)[nH]c3)=O)cn2)=O)CCC(O)CC12CC2 C(CC(C)(C)C(=O)NCC12CC(C1)C(NC(C1(CCOC)CCC1)=O)CO2)OC c1(CCN(C(=O)C=CCBr)CCO)c(F)ccc(C(F)(F)F)c1F.N1CC=CC1 CN1CCN(C(C2CCSC2)=O)CC1C(=O)NCC1(O)CC(CO)C1 c1(C(N(C2CCC(NC(C(C)(C)SC)=O)C2)C)=O)cccnc1O C(C1c2ccccc2CN1C(C1COCCC1(F)F)=O)NC(c1cc(Cl)n[nH]1)=O Cn1ncc2c(C(N3CC4CCN(C(C5CCNC5=O)=O)CC4C3)=O)ncnc12 C1(CC=C)(C(=O)NCCCN(C(=O)Cn2cccn2)C)CCC1 C(CS(=O)(=O)c1ccc(F)cc1)NCC(=O)NCCc1ccccc1 C1(CCNC(c2cnc(C(C)O)s2)=O)CCN(C(C2CC3CCCC23)=O)CC1 c1(C(N(CCCNC(C2CN(C)CCO2)=O)CC)=O)ccc2ncc(C)n2c1 CC#CCCC(=O)NCC(C)CN(C(=O)C(F)C1CCOC1)C C(=O)(C=CS(=O)(=O)CC)NCCCNC(C1CN(CCOC)C(=O)C1)=O N1(C(CC2(C)CN(C(c3n[nH]c4ccccc34)=O)C2)=O)CCc2c(O)noc2C1 Cc1noc(CC)n1.C1(NCC(=O)O)(CNC(=O)OC(C)(C)C)CNC1 C(=O)(C1=C(CCl)N(CCC2CC2)C(=O)NC1c1cc(Cl)cnc1F)OCC N1(C(c2c(C)[nH]cc2)=O)CCC(NC(c2csc(C(F)F)n2)=O)C12CC2 C(=O)(C(C)S(=O)(=O)CCC)NCC1CC(NC(C2CC(CCC)OCC2)=O)C1 CCCCCCC(=O)N1CCN(C(C2CC=CCO2)=O)C(CS(C)(=O)=O)C1 c1(C(c2n(CCCC)nnn2)NC(c2cccc(OC)c2)C)cc(OC)ncc1Cl CC(CC(=O)NC1CCCC1CN(C(=O)CC1CCC(=O)N1)C)C1CCCO1 N1(C(C2N(C)CC2)=O)CCC(C(C)(C)NC(=O)COC2CCCC2)C1 CC(C)CC(C(=O)N1CC(=O)CC1C(=O)NCC1(CC(C)C)CC1)N(C)C c1(C(C(=O)NCC2CC2)N(CC(C)(C)C)C(C)C)cc(C(F)F)no1 CC(CC(=O)NC1CC1CNC(c1cccc(N2CCOCC2)n1)=O)CC(C)(C)C C1(CNC(Cc2ccc(NC)cn2)=O)CC2CCC(C1)N2C(C1(C)CC1(F)Cl)=O N1(C(c2c(CC)noc2)=O)C2CCC1CC(CNC(=O)C(C)(C)c1nccs1)C2 N1(C(C(C(C)C)O)=O)CC(NC(c2cc(F)n(C)n2)=O)CC1(C)C CC1(C)CN(C(=O)CC#N)CC1NC(c1cn(-c2ccccc2CO)nn1)=O c1(N(C)C)nc(N2CCC(N3CCC3)C2)nc(=NCc2cnns2)[nH]1 C(CC(C)(C)C(=O)NCC1(F)CN(C(c2cc(C)c[nH]2)=O)C1)SC CC(C)(CC(F)F)C(=O)N1CCCC(CCC(=O)NCC2(C)CCCS2)C1 c1(NCCN(C)C)ccc(S(=O)(=O)NC2CCSC3(CCCC3)C2)cc1C#N c1(C(=O)NC(C2CCCO2)(C)C)cccc(CNC(C23CCCC2C3)=O)n1 C1(NC(c2c(N)c(C)n(C)n2)=O)CC(NC(C2CCS2(=O)=O)=O)C12CCOCC2 Cc1nc(O)nc(C)c1CC(=O)NCC1COCC1NC(C1(C2CCC2)CC1)=O c1(C(=O)OC)ncn2c(C)cc(=NC3=NC3CC3OCC3C)sc12 c1(C(C)(F)F)cccc(C(N2CC(N(C)C(C3(C(F)F)CCC3)=O)C2)=O)n1 c1(C(=O)NC(CNC(CC2(COC)CC2)=O)C)cnc(SC)s1 c1(C(N2CC(CNC(C(C)C(F)F)=O)C3(C2)CC3)=O)cc2c(F)c(F)ccc2[nH]1 c1(C(=O)NC2(C)CC(C(=O)NCC(CCC)c3ccccc3)C2)nnccc1C C(c1ccc(C)cc1)=CC(=O)N(CC(C)NC(c1c(CC)nc[nH]1)=O)C c1(C(N2CC(NC(c3c(CC)nc(C)o3)=O)C2)=O)c2c(nn1C)CCCC2 c1(C(N)=O)cc(F)c(NC(=O)C(O)Cc2ccccc2Cl)cc1F C1(C(=O)NCc2cnc(OC)c(F)c2)C2C(CN1S(=O)(=O)C(F)(F)F)C2(C)C Cc1ccc(CN(C(=O)CONC(=O)COCC(C)C)C)s1 C1(CNC(CN(C)C(=O)C2CC2)=O)CN(C(C2COC(=O)N2C)=O)CC(C)(C)C1 CC(C)CC(C)(O)C(=O)Nc1cccc(CNC(C2Cc3ccccc3O2)=O)c1 C1(NC(C=COCC)=O)CCN(CCNC(=O)Cc2ccccc2OC(C)=O)CC1 C12(CC)CN(C(c3ccc(C4CC4(F)F)cc3)=O)C(CNC(C3CC3C)=O)(C1)C2 S(=O)(=O)(c1ccc(C#N)cc1)NCCNC(=O)Nc1c(OC)ncnc1 Cc1ccc(C)c(OCCC(=O)NC2CCN(C(C3(O)COC3)=O)CC2F)c1 CC1CN(C(C2CC(O)(CNC(C3CCCOCC3)=O)C2)=O)CCO1 N1(C(C(C)(C)n2ccnn2)=O)CCCC(C(=O)NCc2nnc(C3CC3)o2)C1 c1(C(=O)NCCC2CCN(C(c3cc(C(N)=O)no3)=O)C2)ncccc1O Cc1nc(NC(c2ccoc2)C)cc(NC2CC(NCCN(C)C)C2)n1 C(=O)(CC(C)C(C)(C)CC)NC(CCCNC(C1(CC=C)CC1)=O)CCC N1(C(C2CCCO2)=O)CC(F)(F)CC1CNC(C1(c2c(Cl)cccc2Cl)CC1)=O CCC1=NOC(CC(N2CC(CC(C)NC(c3nc(=O)n(C)[nH]3)=O)C2)=O)C1 CCCCC(C(=O)N1CC(c2nncs2)C1)NC(=O)CCOCC(C)C CCCC(CNC(C1(OC)CCOC1)=O)C(=O)NCCC(C)O c1(C(N(CC(CC)NC(C2(C)CC2(Cl)Cl)=O)C)=O)cccc(C(F)F)c1F c1(-c2c(C(=O)OC)n[nH]c2)ccc2[nH]cc(CNCc3cnc(C)cn3)c2c1 CC(O)(C(=O)N1CCCC(C(N2CCC(C3(C)N=N3)C2)=O)C1)C(F)(F)F c1(C(C(=C)C)NC(c2csc(-c3cnn(CCCCO)c3)n2)=O)ccccc1C C1(C(N2CC(O)(C(=O)OC)C2)=O)CC=CCN1C(=O)CN1CCNC(=O)C1 n1(CC)ccc(C(=O)NCC2CCN(C(=O)Cn3nccc3C)C2)n1 c1(N2CCCC(N(CC(N3CCCCC3)=O)CC)C2)nc2ccc(O)cc2s1 N=c1ccc(CC(=O)NC2CCCC2NC(c2ccnn2CCF)=O)c[nH]1 N1(C(C(CC)CN(C)C)=O)CC2CCCC2(C(=O)NCC(c2ccncc2)C)C1 C1(C(=O)NCCOc2cccc(OC)c2)(CNC(=O)OC2CC2)CC12CCOCC2 C1(C(=O)NCC2(O)CCN(C(C(CC=C)C)=O)C2)(OC)CCCCCC1 n1(CCSCC(N2CCC(O[Si](C)(C)C(C)(C)C)C2)C)ccc2cc(Br)cc(F)c12 N1(C(COCCCC)=O)CC(O)CC1C(=O)N(C)Cc1cc(C)no1 C(=O)(C(C)(C)CCCF)NC1CCC(C(N2CCC(C(C)C#N)CC2)=O)C1 N1(C(=O)C=Cc2cn[nH]c2)CCN(C(c2c(F)cccc2F)=O)CC(CO)C1 c1(CC)nnc(O)c(C(=O)NCC(C)(CO)NC(=O)CCCSC)c1CC C1(C(C)C)CCC(C(=O)NCCOCCF)N1C(=O)CC1COC(=O)C1 C1(C(N2CC(CCC)OCC2)=O)C2CCN(C(=O)CC3CC(OC)C3)CC12 N(C1CCOc2ccc(Cl)cc21)C1(Nc2ccc(OC)cc2)CCCCC1C c1(C(=O)NC(C(C)NC(CC(CC)CC)=O)C)cc2ccccn2n1 c1(C(N2CC3C(NC(C(COC)O)=O)CC(C3)C2)=O)cccc([N+](=O)[O-])c1N C12CN(CC1C)C2=O.C(=O)(CCC(C)C)N(C(C1C(C(=O)OC)CC1)=O)C1CC1 N1(C(Cn2c(C)ccn2)=O)CCC(C)(C)CC1C(N1CCCCCCC1)=O C1(CNC(=O)CSCCc2c[nH]c3ncccc23)CCC2(CC1)OCCO2 CCCCC(C(=O)N(CC)CC)NC(c1cn[nH]c1)=O c1(NCCC(CNC(CCN(C(C)=O)C)=O)O)nccc(C(N)=O)c1[N+](=O)[O-] N1(C(c2cc(=O)c(Br)c[nH]2)=O)CCC2(CC1)CN(C(C1CCC3CC13)=O)C2 N1(C(C2CC(O)(CC#C)C2)=O)CC(CC(=O)NC(C)CCC=C)C(C)C1 C(C(=O)N1CCC(C)(CC(=O)Nc2cnsc2)C1)(C(C)C)SC c1(N(CCOCCOC)C)nc(N2CCC(F)(C#N)C2)c2c(n1)CCCCCC2 C1(NC(C(C)(F)F)=O)CC12CC(NC(=O)CN1CC3CC3C1)C2 N1(c2c(C)c(NCC34COC(CO)(C3)C4)ncn2)CCC2CCCC2CC1 C1(C(C)C)COCCN(C(=O)COC(C)(C)CNC(=O)COC(C)(C)C)C1 C1(CNC(COCP(C)(C)=O)=O)CC2(C1)CN(C(=O)CC1CC=CCC1)C2 N(C(=NCc1ccccc1)NC1CCC(C(F)(F)F)CC1)CC1CCN(CC)C1 S(=O)(=O)(c1ccc(NC2CC3CCC(C2)O3)c(C#N)c1)NC(c1csc(Cl)c1)C CC1=C(C(=O)N(C)CCN(C(=O)C(c2cccc(O)c2)(C)C)C)CCCC1 N1(C(c2cn(CCC)nn2)=O)CCC(C)(C)C(CNC(=O)C(Br)=C(C)C)C1 C12(NC(C=C(CCC)C)=O)CCC1CN(C(=O)CCNS(C)(=O)=O)C2 C1(CCC)CN(C(=O)C(C)CN(C)C)CC1NC(c1oc(C2CC2)nc1CC)=O C1(NC(C(C)=C2CCC2)=O)C2CC3C1C3C2C(=O)Nc1cnn(C)c1 CCCC(C)(O)C(=O)NCC1CC(O)CN1C(c1csc(C(=O)OC)c1)=O c1(CC(N2CCCC(NC(C3CC3C(F)F)=O)C2)=O)ccc(Br)cc1F C(c1ccncn1)=CC(=O)NCCOC1CN(C(C)=O)C1 N1(C(C(CC)OCC)=O)CCOC(CNc2ccnc(Cl)n2)C1 c1(NC)ccc(Cl)c(C(=O)NCC2CCCN2C(c2cccn2C(C)C)=O)c1 C1(c2c(C)n[nH]c2)COCCN1C(c1c[nH]nc1Cl)=O C1(C(=O)NCC2(C(=O)NC(C(=O)OCC)C)CCCO2)CC(=O)C1(C)C C=CCCCCC(=O)NCc1cccc(CNC(=O)C(C)C#N)c1 c1(C(=O)NCC2CCN2C(C23CC2COC32CCC2)=O)cc2c(Cl)cccc2s1 Cc1cc(C(N2CC3CC2CC3NC(=O)C(F)(F)C2(O)CCC2)=O)cc(O)c1 C1(NC(C(CC)OC2CCCCC2)=O)CC2CCC1(NC(=O)C1=CSCS1)C2 C1(O)(CCSc2n(C)nnn2)CCN(C(=O)N(C(C)(C)C)CCO)C1 c1(NC(CNCC(c2ccncc2)C)=O)sccc1OC(F)(F)F c1(CCNC(Cc2c(C)n[nH]c2)=O)nc2cc(F)ccc2n1Cc1ccccc1 C1(NC(CC2(CC)CC2)=O)CCC(C)(CNC(c2ccc(C#N)s2)=O)C1 C(=O)(C1CCc2c[nH]nc21)NCC1(CNC(=O)CN2CCS(=O)CC2)CCCC1 N1(C(c2ncc(C)c(OC)c2C)C(=O)NC)CCC(C2(C)CC2)C1 C(C(C)(CO)CO)N(C(C1C(NC(C(C)N(CC)CC)=O)COC1)=O)C C1(C(=O)NC2CN(C(c3cn(CC)nn3)=O)CC2C)COc2ccccc2O1 CC(C)(CNC(=O)OC(C)(C)C)C(=O)NCC(F)CNC(C1CNC(=O)C1)=O CCC(C)C(C(=O)NOC(CO)C(C)C)N(C)C(C12CC(C#N)(C1)C2)=O c1(COC)n[nH]c(=NC2CCCC3CN(C(=O)C(C)(C)CC(F)F)CC23)s1 C1(CNC(CC2CCN(C)C2=O)=O)CN(C(=O)Cn2cnc(=N)[nH]2)CCC1(C)C C1(CC=C)(C(=O)N(C(C)C(F)F)C)CCN(C(c2ccnc(O)c2)=O)C1 N1(C(CN(S(CC)(=O)=O)C)=O)CCCN(C(=O)C(C)O)CC1 C1(CNC(C=CC)=O)CCCCN(C(=O)C(C)Cc2ccc(OCC)cc2)C1 c1(CCCNc2c(C(N)=O)cn(C)n2)nc2cnccc2[nH]1 c1(C(N(C2CCCN(C(C(C=C)OC)=O)C2)CCF)=O)ccc2n[nH]cc2n1 C(c1ccc(Cl)cc1F)=CC(=O)NC1(CNC(C(CC)OCC)=O)CCC1 C1(CCC)CCC(C(=O)NCC#CCNC(c2cn(CC)nn2)=O)CC1 c1(CC#N)ccnc(NCC2(C(C)(C)C)CCN(C(C3SCCS3)=O)C2)n1 C1(NC(CCCN(C(c2cnc(CC)o2)=O)C)=O)CCN(C)C1(C)C C(C(C)(C)C(=O)N(CCCC(=O)N1CCC2CC12)C)SC C1(CCC(=O)N(C(C(=O)NCC(C)CC2CC2)CC2CC2)C)CCCC(O)C1 N1(C(=O)Cn2ncccc2=O)CC2CN(C(C3CCCC(O)C3)=O)CC2C1 c1(C(N(CC(C)(C)NC(CC(=C=C)C)=O)C)=O)ccc(F)c(N2CCCC2)c1 CCC(CC)CC(F)C(=O)NC(CC)CCC(=O)NCCCC1CCOC1 C1(C(=O)NCCCN(CCCNC(CC2CC(=C)C2)=O)C)CCC(=O)O1 C(=O)(CS(O)(=O)=O)N(C)CC1N(C(C2CC(C)OC2)=O)CCC1 c1(C(=O)NC2C3CCN(C(c4cccc(OC)c4)=O)C32)cc2ccc(C)cc2[nH]1 Cc1cccc(S(=O)(=O)N2CCC(O)(CC(N3CC(F)C3)=O)CC2)c1 C1(CNC(C(=O)NCC)=O)(NC(=O)CCC2CCCCO2)CCCC1 c1(CC=O)nc(C)c2c(n1)CCCC2.c1(CNC(CSCCC)=O)cn(CC)nn1 c1(C(N(C2CCN(C(c3ccccn3)=O)CC2)C)=O)cnn2c(Br)cccc12 CCC(C(=O)NCCCOCCNC(c1n[nH]cc1F)=O)NC(N)=O O=S(=O)(c1ccc(NCC2C3COCC23)c(Cl)c1)NC1CC(CCO)C1 C(C(C(C)C(C)C)NC(C1(CN(C)C)CC1)=O)NC(CC=C=C)=O c1(C(=O)NCCOCCC(=O)NCCC2CCC(C)O2)ccncc1F C1(C(N2CCC(NC(C(C)SCCCC)=O)C2)=O)(NC(C)=O)CCC(F)(F)CC1 C(=O)(C(C)(F)C(C)(C)F)N1CC(C)C(NC(=O)CC2CCOCC2)C1 CCCC(C)(CCC)C(=O)NC1CCCCC1NC(=O)CC1CCOC1 N1(C(C2N(C(C)=O)CC(O)C2)=O)CCC(NC(c2cnc(S)n2C)=O)C(F)C1 c1(CC(N2CCC(C)(NC(C(COC)O)=O)C2)=O)cc(F)c(F)cc1F n1(CC)ncnc1CNC(=O)CCN(C(C1CCSC1)=O)C1CC1 C(=O)(C1CCc2c[nH]nc21)N1CCC(N(C(C(CC2C(C)C2)O)=O)C)CC1 C#Cc1cncc(C(=O)OC2CCN(C(=O)OC(C)(C)C)C2)c1 C1(C(=O)NC2CC(F)(CNC(C(CC)CC)=O)C2)CCc2ncsc2C1 n1(CCC)cc(C(=O)NCC(F)CNC(=O)C(F)(F)C2(O)CCC2)nn1 Cc1cc(N)cnc1C(N1CCC(N(CCO)C(C2CC3(C2)CC32CC2)=O)C1)=O C(=O)(C(C)(C)CCCNC(c1ccccn1)=O)Nc1cn(C)nc1 Nc1c(C(N2CCN(C(C3CC3C(F)(F)F)=O)C(CF)C2)=O)cccc1Cl c1(NC(=O)C=CCNC(=O)CN2CCCC2=O)cc[nH]c1C1CC1 C1(C(=O)NC2CCCN(C(CCCC#N)=O)CC2)CCOCC12CCCCC2 N1(C(CNC(=O)OCC)=O)CCCN(C(=O)COC(C)CC)C(C(C)C)C1 C1(CC(=O)NCC2N(C(c3c(C)coc3C)=O)CCCC2)CC(C)(C)C(=O)N1 C12(NC(C3NC(=O)CC(C)C3)=O)CCCCC1CN(C(c1ncncc1F)=O)C2 C1(C(N)=O)COCC1NC(C1CC(O)(C(F)F)C1)=O C(=O)(CCC(C(F)(F)F)NC(C1CCC1)=O)OCC(n1c(C)cc(C)n1)C N1(C(C2N(C)C(=O)NC2)=O)CCN(C(c2ccc(C#N)cc2)=O)C(C(F)F)C1 CC(C)C(O)C(C)(C)C(=O)N(CC(C)NC(c1ccc2cccnc2c1)=O)C Cc1ccc(C)c(C(N2CC(CNC(=O)CCCCCF)C2)=O)c1N c1(CC(=O)NC2C(NC(c3c(OC)cncc3)=O)CCC2)n[nH]c2ccccc12 N(C1c2ccccc2CC1O)C(c1ccc(Cl)cc1)=O c1(CC(=O)N(CC(C)(C)CNC(C2CC2C(F)(F)F)=O)C)ccc(O)nc1 c1(C(=O)NC2(CNC(=O)Cn3cnnc3)CCCC2)noc2cc(Cl)ccc12 C12(CNC(C3CC4(CCNC4)CO3)=O)CCCCC1OCC2 CC(=O)CCCC(=O)NCC1(C(=O)Nc2cccc(CO)c2C)CCCO1 N1(C(C2(CNC(C(C)c3ccsc3)=O)CC3(CC3)C2)=O)Cc2cncnc2C1 O=C1CCC(C(=O)N2CCCCC2CNC(=O)C(O)C2CCC2)c2ccccc21 C1(CCNC(C2(C)CC2)=O)CN(C(=O)C(O)CCc2ccccc2)CCS1(=O)=O C1(C(=O)NCC2CC(NC(C3C(C(C)C)C3)=O)C2)CC2C=CCC(C1)C2 c1(C(N2CCCC(N(C(=O)Cc3cnsc3)C)CC2)=O)ccnc2c1CCO2 Cc1cc(C(F)(F)F)ncc1C(=O)NC1(C)CCCN(C(C2CCCCS2)=O)C1 CC(C(F)(F)F)NC(C1CC1c1ccco1)=O C(=O)(C1=CC2(CCN(C(=O)C(C(C)(C)C)OC(C)C)C2)C1)NCCCCOC C(C(C)(C(=O)NCC(c1cccs1)O)NC(=O)Cn1ccnc1)SC c1(CC)cnc(O)c(C(=O)NCCC2CC(NC(=O)CC(C)CC)C2)c1 C1(NC(c2cc(O)nc(O)c2)=O)CC2CC1N(C(c1cc(CO)on1)=O)C2 N#Cc1cc(F)c(C(=O)NC2COCCC2NC(c2cc(Cl)cnn2)=O)c(F)c1 C1(C(=O)NC(C#C)C)CC12CCN(C(=O)CNC(N)=O)CC2 c1(CC)ccc(C)c(C(=O)NC2CCCN(C(=O)C(C)N3CC(C)C3)C2)c1 C1(OC)CC(CNC(c2n[nH]cc2Cl)=O)N(C(c2ccc(C(F)(F)F)n2C)=O)C1 C1(C(N2CCC(O)(CN(C)C)C2)=O)COCCN(C(=O)CC2CCC(C)CC2)C1 C(=O)(C1=CCCC1C)N(C1CCN(C(c2c(C)nns2)=O)C1)CCO c1(C(=O)NCC23C(CN(C(C=C(C)C)=O)C2)C3)cccc2cnccc12 c1(C(N2C(CN(C(=O)C(C)CSC)CC)CCC2)=O)cc(C)c(C)c(F)c1 C1(NC(C(C)SC)=O)C2CC3C1C3C2C(=O)NC1(C)CCSCC1 C1(O)(CNC(c2nc(C(C)C)oc2)=O)CCC(C)(C)CC1 C1(NC(c2nc(C(C)C)oc2)=O)CC2CN(C(C3(N=[N+]=[N-])CC3)=O)CC2C1 S(=O)(=O)(c1cccnc1NCC(CCC1CC1)OC)N1CC(CC)OCC1 CC1(C)OC2CCN(C(C3CCCN(S(=O)(=O)c4ccc(Br)s4)C3)=O)CC2O1 C1(COC)CN(C(c2ccc(SC)cc2O)=O)CCN1C(C12CC(C1)C2)=O N1(c2c(OC)c(C)ncn2)CCCC2(NC(=O)C(O)Cc3ccccc3)CC2C1 c1(C(=O)NCC(CC)NC(c2cnn(C)c2Cl)=O)cccc(-n2ccnc2O)c1 C1(CC=C)(NC(c2ncccn2)=O)CCN(C(c2cn(C)nc2C2CCC2)=O)C1 C(C)(C(=O)OC(C)(C)C)(C(F)F)NC(C(=O)NC(c1ncc(C)s1)C)=O C(=O)(C(F)(F)C(C)O)NC1C(C2CCN(C(C=CC=CC)=O)CC2)OCC1 c1(C(=O)NCC(C)(C)CNC(=O)C(C)(O)c2ccccc2)ccc2ncsc2c1 C(=O)(C1=CC(C)(C)C1)N1C(CN(C(=O)CS(=O)(=O)CC)CC)CCC1 c1(NC(N(C(C)(C)C)CC)=O)nn(C)c(C)c1Cl.C1(=O)C(C)N1 N1(CCN2C(=CC(=O)N3CCC(C)C3C)SCC2=O)CC2CCCS(=O)(=O)C2C1 C1(CCC=C)(C(=O)NC(C)C(C)O)CN(C(=O)COC2CC=CC2)C1 c1(CC)ccc(C(=O)N(CC(N2CCC2(CO)CO)=O)C)s1 N1(C(C2CC(N(C)C)C2)=O)CC(NC(=O)Cc2cccc(O)c2)C(C)(C)C1 C1(COC)CCC2(C(C)C)CC12.C1(C)(OC)CNC(=O)N1 C1(NC(c2ccc(C(C)=O)c(F)c2)=O)C2CC(O)C1N(C(C13CC(F)(C1)C3)=O)C2 c1(C(=O)NC(C(C)C)CCN(C(=O)C(C)CC2CC2)C)cnn2c1C(=O)NCC2 c1(C(=O)NCCOCCN(C)C(C2CNC(=O)N2)=O)cc(=O)n2nccc2[nH]1 C1(=CC(=O)NCC(CC)(C)NC(c2cccnc2S)=O)CCN(C)CC1 c1(C(=O)NC2CCC(F)(CNC(C(C(C)C)C)=O)C2)cc2n(n1)CCNC2=O C1(CNC(C2(N(C)C)CC2)=O)CCC(C(=O)N(c2ccccn2)C2CCOC2)O1 Cc1nc2ccccc2nc1C(N1CCC(CCNC(=O)CCN(C)C)C1)=O N1(C(C2(C)COCC2(F)F)=O)CCOC2(CCCN(C(C34CC(F)(C3)C4)=O)C2)C1 C(=O)(C(CCc1ccccc1)C(C)C)NCC(CNC(CCSC)=O)F S(=O)(=O)(c1ccc(Br)c(Cl)c1)N1C(C(N2CCC(C)(O)CC2)=O)CCC1 C(CC(CO)NC(=O)CCCNC(=O)C(C)NC(=O)NC)=CC C1(O)(CNC(C2N(C=O)CCC2)=O)CCCN(C(c2cnn[nH]2)=O)C1 N1(C(CCCCCC)=O)CCC2(CC1)COC(CNC(=O)CC1(O)CCCC1)C2 C(=O)(C1c2ccccc2C2CC1C2)NCCCN(C(=O)C(C)=CC(C)(C)C)CC C(=O)(C#CC(C)(C)O)NC1(CC=C)CCN(C(c2ncc(C)cn2)=O)C1 O=C(CCC(CF)CF)NC1COCCC1NC(C1CC12CCCC2)=O CCS(=O)(=O)CCCN=c1[nH]c(=NCc2ccoc2)[nH]c2ccsc12 CCC(CC)(C(=O)N1CCCC1C(N1CCN(C2CC2)CC(C)C1)=O)C(=O)O C#CC1(C(=O)NCC(O)(CO)CO)CCN(C(c2cc(Cl)n[nH]2)=O)C1 N1(C(c2c(C)cncc2)=O)CC(NC(C2(N3CCCC3)CC2)=O)CC2(CC2)C1 Cc1cc(Br)c(NC(C2C3CN(C(c4ccn(C(F)F)n4)=O)CC23)=O)cc1F c1(OC)cc2nc(N3CCCC(c4ccccn4)C3)c(=O)n(C)c2cc1OC C1(NC(c2oc(C)c(CO)c2)=O)CN(C(=O)Cc2cncnc2O)CC(F)(F)C1 N1(C(c2nc(C)oc2C)=O)CC(O)C(O)C1CNC(=O)CC(C)F c1(C(=O)NCC2CCC(CNC(c3c(C)ccs3)=O)CC2)c(C)nn(C)c1F c1(N2CC(F)C2)nnc(C(F)(F)F)s1 c1(C(N2CC(C(C)NC(CNC(CC)=O)=O)OCC2)=O)cnc2ccncc2c1 N1(C(c2ccc(OC)c(OC)n2)=O)CC(F)(F)CC1C(=O)Nc1ncc(C)s1 CN=c1nc(C(=O)NC2(CO)CCCN(C(c3cc(C)c[nH]3)=O)C2)cc(C)[nH]1 C1(CNC(C2(CC)CCCCO2)=O)COCCN(C(c2c[nH]cc2C)=O)C1 Cc1cnn(C(C)C(=O)NCC2(C(=O)N(c3cn[nH]c3)CC(C)C)CC2)c1 N1(C(C2C(C)(C(C)C)C2)=O)C(C(=O)NC2CC(CO)C3CC23)CC2CCCC12 n1(CC)ncc(C(=O)NCCC2CCCN(C(=O)Cc3cn(C)nc3C)C2)c1C C(C)(C(=O)NC1CC(NC(=O)C(=O)NC)C1)OCCCC c1(C(N(CCCN(C(C(CC#C)C)=O)C)C)=O)cc(OC)cc2c1OCC2 c1(OCCC(=O)N(C2CCN(C(c3ccsc3C(F)F)=O)C2)CC)ccccc1 C#CCC(CC#C)C(=O)NCCCCCCN(C)C(c1ccc(C)cc1)=O CC1CC(NC(=O)C(F)F)CCN1C(C1CC1C(F)(F)F)=O c1(NC(=O)NCC2(C3CCCO3)CCOCC2)nc2cc(F)ccn2n1 Cc1cc(O)nnc1C(N1CC(=C(F)CNC(=O)Cn2cnnc2O)C1)=O N1(C(c2c(COC)ccs2)=O)CC(C)C(C)(CNC(C2C3CCC2CC3)=O)C1 N1(C(=O)OC)CCCC(C(C)OCC)C1.C12CCN(C1)C(=O)CNC(=O)CN2 C(=O)(CCN=c1[nH]ccs1)N1C2CC(NC(CCn3c(C)csc3=O)=O)C2CC1 c1(C(=O)NC(C)CCN(C(=O)C(C)C2CCCC2)C)cc(Cl)c(F)cc1O c1(NC(N2CCC(NCCCC)C2C)=O)sc(C)c(C)c1C(N)=O C(C)(CNC(=O)C=CCN(C(=O)C(F)C1CC1)C)(C1CC1)OC C(C)(CN=c1[nH]c(=N)[nH]c(=NCC2CCCN2C)[nH]1)OCCOCC C1(C(N(C2CCN(C(c3ncn(CC)c3)=O)CC2)C)=O)Cc2c(F)cccc2O1 C1(NC(c2cn(C(C)C)nn2)=O)CC2CCC1CC2NC(C1C(F)(F)C12CC2)=O C(=O)(C(C)(C)COCC(F)F)NC1CC(NC(C2(C(F)(F)F)CC(=C)C2)=O)C1 c1(C(=O)OCC)cnc(SC)[nH]c1=NC(C)CC(C)NC(c1nc(Cl)oc1C)=O c1(C(=O)NCCC(=C)CNC(C2CC2c2cccnc2)=O)cc(OC)cc(F)c1 CC1CN(C(=O)C=CCN(CC(F)(F)F)C)CCC1N(C)C(C1CC=CC1)=O c1(NCCCNC(=O)NCCC(COC)(C)C)ccc(Cl)cc1Cl.OCCCN C1(C(=O)NC2C(CNC(Cc3cn(C)nc3)=O)CCCC2)CCn2ncnc2C1 C(=O)(CCCN=[N+]=[N-])NC1(CCOC)CCN(C(=O)C2=CC(C)CC2)C1 c1(OC)c(C(=O)NC2(CNC(=O)C=C(C3CC3)C3CC3)CCOCC2)csc1C c1(CNC(=O)CNC(C2(CO)CC2)=O)cn(CC2C3CCCC23)nn1 c1(CC(N2C(CCCNC(C(CO)OC)=O)CCCC2)=O)cnn2ccccc12 C1(n2cccn2)(CNC(C)=O)CCN(C(=O)COC(F)(F)F)CC1 C1(C)(C(N2CCC(C)(NC(C3C(C)CC3C)=O)CC2)=O)CCC(C)(C)CC1 C(=O)(CCC1(C)CC1)NCCN(CCCN(C)C)C(C1CC(n2cnnc2)C1)=O C(CCN=c1cc[nH]cc1S(=O)(=O)N1CCCCC1C1CCOC1)NC1(C)CC1 CON1CCC(CC(=O)NCC2CCN(C(c3ccc(Cl)s3)=O)C23CC3)CC1 c1(CC(=O)NCCC2C(NC(C3(C)CC3)=O)CC2)csc(Cc2ccccc2)n1 C(CC(N)=O)(C(=O)N1CCNC(=O)C1C)NC(COCC(C)C)=O CC1CCN(C(C)C)CC1NC(C1CCN(Cc2nc(C3CC3)cs2)CC1)=O N1(C(C(C)=O)=O)CC(NC(=O)C(F)(F)CC2CC2)CCC1C C1(CNC(c2c(SCC)cccn2)=O)CC2(C1)CN(C(=O)COCCF)C2 c1(C(=O)NCC2CCN(C(=O)CC3CC4(CC4)CO3)C2)cc(Cl)c([N+](=O)[O-])[nH]1 C(CN=C(NCc1ccc(O)c(OC(F)F)c1)N1CCCC(S(C)(=O)=O)C1)SC C1(CNC(C(C)OC2CCSC2)=O)CC2CCC1N(C(c1cc(N)cc(O)n1)=O)C2 CC(=O)CCCC(C)(C)C(=O)NCC1OCCC1C(=O)NCCCC(O)CO C1(C)(C(=O)NC(C)CCO)CC12CCN(C(=O)C(Br)Cc1ccccc1)CC2 C1(C(=O)NCCCN(C(c2ccccc2)=O)CC)CC(C)CC(C)C1 c1(CC(N2CC3(C(C(=O)NCCCCCO)C3)C2)=O)cccc(Br)c1F O=C(C(O)CC(F)F)NCc1ccccc1-n1cc(C2(O)COC2)nn1 c1(C(N2CCC(O)(C(C)NC(=O)COC3(C)CCC3)C2)=O)cnc2ccoc2c1 C1(NC(CC2C(C)=NNC2=O)=O)CC2(CCN(C(=O)Cn3ccc(C)c3C)C2)C1 c1(CC(=O)NC2CCN(Cc3cn(CCCCOC)nn3)C2)ncn(C)c1Br c1(CCC)cc(C(=O)N(CCN(C)C(C2CSCN2C)=O)C(C)C)no1 C12(C(=O)N(CC3CCN(C(C)C)C3)CCO)CNCC(F)(C1)C2 N1(C(c2c(C)oc(C(C)C)n2)=O)CCC(NC(C2C(C)C2C)=O)CC1C c1(CC(=O)NC(C(=O)NCC(C)(C)F)c2ccco2)ccccc1C#N C1(C(N(CCN(C(C(CSC)OC)=O)C)C(C)C)=O)CC2CC1CC2(F)F c1(CC(=O)NCC2CC(NC(C3(O)CC(C)(C)C3)=O)C2)ccccc1[N+](=O)[O-] c1(C(=O)NCCCN(C(c2nc(C)ccc2C)=O)CC)cccc2oc(O)nc12 C1(C)(COC)CC(NC(=O)CC(F)F)CN1C(=O)CC1(C)OCCO1 C(=O)(C(C)CS(C)(=O)=O)N1CC(F)(CNC(C(C)CCc2ccccc2F)=O)C1 C12(C(=O)NCCCN(C(C(CCCOC)C)=O)C3CC3)CCC(O)(CC1)CC2 C12(NC(CS(=O)(=O)NCC)=O)CCC(CN(C(C3CCCS3(=O)=O)=O)C1)C2 N1(C(c2ccn(C)n2)=O)CCN(C(C2CCCS2)=O)C(c2nccn2C)C1 N1(C(CCCn2cc(-c3ccc(C)s3)nn2)=O)CCC2C(C(F)(F)F)C2C1 c1(C(N2CC(N(C)C(c3cnncc3O)=O)C(O)C2)=O)cccc(F)c1F C1(O)(CNC(C(C(C)C)c2ccccc2)=O)CCN(C(=O)Cc2ccsc2)CC1 c1(OC)ccc(C(=O)N(C2CCC(NC(c3ccn(C(F)F)n3)=O)C2)C)c(C)c1 C1(COC)(NC(=O)COC2CC2)CCN(C(c2ccc(OC(F)F)nc2)=O)C1 C(C(=O)N(CCNC(=O)COC1CC1)C1CC1)=CCN(C)CC C1(NC(C(C)NC(=O)C(C)(C)C)=O)CC2COCC(C1)N2C(=O)Cn1cnnn1 N(C1CCc2cc(C#N)ccc21)Cc1cc(C)c(OC(F)(F)F)cc1 C1(NC(C(CC)C(C)C)=O)CCN(C(=O)C(=Cc2ccccc2Cl)C)C12CCC2 c1(CNC(=NCC=C)NCC(=O)NC2CC2)cn2cc(Cl)cc(C)c2n1 C1(NC(C(CC)CC2CCCC2)=O)CN(C(c2ccco2)=O)CC(C)(C)C1 c1(NC(C2CCN(Cc3ccc(F)cc3[N+](=O)[O-])C2)=O)cc(F)cc2[nH]ncc12 C(CC(C)C)(C(=O)NCC1(F)CC(CNC(=O)CC2CC3CC3C2)C1)OC CC1=CC(C)CN(C(C2(NC(C3COCC3(C)C)=O)CCC(C)(C)C2)=O)C1 CC1(CNC(c2nnnn2Cc2ccco2)c2ncco2)CCCCO1 C(=O)(C1CCCn2nccc21)N(C)CCN(c1nc2ccccc2s1)C N1(C(CC=C(C)C)=O)CC(NC(=O)C(C)CC(F)(F)F)CC(C)(C)C1 C(=O)(CCCC(=O)NCC)NC(C1CCCC1)CNC(CC1(C(=C)F)CCC1)=O c1(C(N(C)CC2(O)CCC2)=O)occc1CNC(=O)COc1ccccc1 c1(C(N(CCc2cccc(OC)c2)C)=O)c(C)oc2ncn(C)c(=O)c12 N1(C(C(C)O)=O)CC2(CCOCC2)CC1CNC(c1cc2ccsc2[nH]1)=O c1(COC)nc(N2CC=C(CNC(c3cnc(C)nc3O)=O)CC2)cc(C)n1 C=C1CC(C)(C(N2CCCC2CCC(=O)NCCCOC)=O)C1 N1(C(c2c(C(=O)O)scc2)=O)CCn2nccc2C1CO N1(C(C(C2CCC2)OC)=O)CC2C(CNC(=O)CN3CCC(F)(F)C3)C2C1 C1(CNC(C(C)SCC)=O)CC(O)CN1C(=O)CC1(O)CCOC1 c1(CC(N2CCC(CN(C(C3CC3(Cl)Cl)=O)C3CC3)CC2)=O)ccc(CO)cc1 c1(C(=O)NCC(C)(C2CCC2)NC(c2c(C)ccnn2)=O)ccc2nncn2c1 N1(c2c(C)c(NN3CC(O)C4CCCCC34)ncn2)CCC2(CCC(=O)NC2)CC1 Cc1cc(C)n(C(C)C(=O)NCC(O)CNC(c2ncc(C(F)F)s2)=O)n1 C1(NC(c2c[nH]c(=N)o2)=O)CN(C(c2cc3scnc3[nH]2)=O)CCC1C(F)(F)F Cc1cnc(C(C)NC(=O)C(C)(C)CN(C(=O)CN2CC=CC2)C)nc1 c1(C(=O)NC2CN(C(c3c(OC)scc3)=O)C(C)C2)cnn2ccn(C)c12 c1(CC)nn(C)cc1CNC(=O)C(CCN(C)C)NC(=O)CC1CCOC1 C(=O)(C1=C(C)OCCS1(=O)=O)NCC(CNC(C=Cc1ccc(CC)cc1)=O)O C1(NC(COC)=O)CCOC(CNC(c2ncccc2OC(F)F)=O)C1 C(C)(CC(=O)NCC1(O)CCN(C(C2CCSCC2)=O)CC1)(C(F)(F)F)N(C)C N1(C(CSc2c(C)n[nH]c2C)=O)CCC(C2(O)CCN(C(=O)C(C)(C)F)C2)CC1 N#Cc1ncn(CC(=O)NCC2CCN(C(C3CC(O)C3)=O)CC2)n1 c1(C(N(C2CCCN(C(C3CC(C#N)C3)=O)C2)C)=O)ccnc(C(F)(F)F)c1 c1(C(N2CC(N(C(C(C)=C3CC3)=O)C)C(O)C2)=O)cc2c(O)ncnc2cn1 C12(CNC(C(CC)(C)OC)=O)CCC1CN(C(c1ccc(C(=O)OC)s1)=O)C2 C(=O)(C1=NOC2(CCN(C(=O)OC(C)(C)C)C2)C1)N1CC(CC)CC(F)(F)C1 N1(C(C(CCCC)C)=O)CCC2(CCCC2NC(c2ccc(F)cn2)=O)CC1 C1=CC(=O)OCC(=O)N2C1CCC2.C(CC=CC)OC.C(CO)OCC C(C)(c1ccccc1)=CC(=O)NC(CC=C)CNC(=O)CC=CC(C)(C)C N1(C(c2cc(OC)n(C)n2)=O)CCC2(NC(c3cnccn3)=O)CC2C1 N1(CC(C)NC(C(c2c(C)noc2C)CC)=O)CCN(C(C2(C)CC2)=O)CC1 CC(CC(=O)NC1CC(CC(=O)N(C2CC3(CCC3)C2)C)C1)C(F)F c1(OC)ccc(F)cc1CC(=O)NCCC(C)(C)CNC(c1c[nH]ccc1=N)=O N1(CC)CCC(C)(OC)CC1.c1(NCCC=Cc2ccccc2)ncc(CN)cn1 c1(OC)ccc(Br)c(OC)c1C(N1CCCC1C(=O)NCCC1CCCOC1)=O c1(Cn2cc(-c3cn(CC)nc3)nn2)ccc(F)c(F)c1.C1(C(C)O)C(=O)N1 Cc1cc(C(=O)NCC2CCCCC2NC(=O)CN2CCOC2=O)c(C)[nH]1 c1(C(=O)NC2CC2C(=O)Nc2ccnnc2O)cc(O)cc2ccccc12 N1(C(COC(CC)C)=O)CC(F)(F)CC1CNC(=O)Cc1cnc(C)[nH]1 Cc1nn(C)c(Br)c1C(=O)NCCN(C(c1ccccn1)=O)C1CC1 C1(C(=O)NCC(CNC(c2c(C)snc2)=O)C)CN2CCN1C(C)C2 c1(SCC(=O)NC(CN(C(=O)CCSC)CC)C)cc(F)c(F)c(F)c1 N1(C(c2c(C)nn(CCO)c2)=O)CCC2CN(C(C3CC(F)CN3C)=O)CC12 C1(F)(CNC(C2CCCCC2F)=O)CCCN(C(=O)COC(F)(F)F)CC1 c1(CC(=O)NCCCC(C)(C)NC(C2CC(=C)C2)=O)ccc(OC)c(Cl)c1 C1(C)(CC)C=C(C(=O)N2CCC(C(=O)NC3C(O)C4CCOC34)(OC)C2)C1 C1(C(=O)NCC(O)CC2CCCC2)(NC(C=C)=O)CCC(C)(C)C1 C=CC1(C(N2CCC(C(C)C(=O)N(CCOCC)CC)CC2)=O)CCOCC1 C1(C(=O)NCC(C)NC(c2ccc3n[nH]cc3c2F)=O)Cc2cc(F)ccc2O1 CC1CC(NC(=O)CC(C)(F)F)CCN1C(=O)CC1CCC(O)C1 C1(C(=O)NC2(CNC(C(CO)OC)=O)CCCCC2)CCn2c(O)nnc2C1 N(C(=NCc1cccc(C(=O)NC(C)C)c1)N1CCCC(CC2CC2)C1)C(C)C CC1CN(C(c2cocc2Br)=O)CCC1C(=O)NCC1(CO)CCOCC1 CCCCC(C)CCC(=O)N1C2CCC1CC(NC(C1(CC(F)F)CC1)=O)C2 c1(C(=O)OC)[nH]c(C)c(C(=O)NC2CC(NC(c3nn(C)cc3Cl)=O)C2)c1C C=CC(C)C(C)C(=O)NCC1(NC(c2nc(=N)cc[nH]2)=O)CCCCC1 C1(NC(C(F)OC)=O)CN(C(=O)CSc2nc3ccccc3o2)C2(CCC2)C1 c1(C(=O)NCC(CCOC)NC(C2OCC2(C)C)=O)csc(S(N)(=O)=O)c1 c1(CCC(N2CCCC(N(C(CC=C=C)=O)CCO)C2)=O)ccc(OC)c(Cl)c1 N1(C(c2ccn(CC)c2C)=O)CCN(C(=O)C#CC(C)(C)O)C(C)C1 c1(CC(=O)N(C)Cc2cccc3occc23)cccc2ccncc12 N1(C(C(C)N(C(C)=O)C)=O)Cc2ccnn2CC(NC(c2cc(Cl)cs2)=O)C1 Cn1cc(CNCC2(c3cccs3)CCCC2)c(Br)n1 C(=O)(C(C)(CCC1CCC1)SC)NC(c1ncc(CC)[nH]1)c1nnnn1CCOC N1(C(C2N(C(CC(CCC)C)=O)C(C)C2)=O)CCc2ccc(C)cc21 c1(CC(=O)N(CCCN(C(c2cc(C)nn2C)=O)C)C)cccc(F)c1F N1(C(c2cc(C)c(C(N)=O)cn2)=O)CCN(C(=O)CC2(C)CC2F)C2(CCC2)C1 C1(NC(C(=O)NCc2cc(OCC)c(C)cc2)=O)CN(C)CC12CCCC2 CC(C)C(O)CC(=O)N1CCOC(C)(CNC(=O)C(F)(F)C2CC2)C1 C(=O)(C1=NNC(C(F)(F)F)C1)NCCN(C(C)C)C(C1CC=CCC1C)=O C1(NC(c2cn(CCC)nc2)=O)CCN(C(C2CC(=O)N(C)C2)=O)C1CC CC(C)CN=C(NCc1sccc1Cl)N1CCC2(O)CCOCC2C1 C#CC(C)(C)C(=O)NCC(CC(C)C)NC(c1cc(Br)c(OC)s1)=O C1(C(=O)NCC(C)N(C(=O)CSCC(=O)OC)CC)C2CCCCCCC12 Cc1ccc2snc(C(N3CCCC3CCCNC(C3COCCO3)=O)=O)c2c1 CC1=C(C(=O)NC2CC(F)CN(C(C3CC3(C)C(C)C)=O)C2)S(=O)(=O)CCO1 CCCCCCC(C)C(=O)NC1CCC(NC(=O)C(C)CC(F)(F)F)CC1 CN1CCS(=O)(=O)CCC1CCNC(=O)CCCc1ccc(Br)s1 c1(N2CCN(C(C3CC3CCS(N)(=O)=O)=O)C2)cncc(NC(C)=O)c1 N1(CC(C)C2CC2)CCc2cc(C#N)ccc21 N1(C(c2c(C)nc[nH]2)=O)CCCC(CN2CCN(C(c3cc(O)cs3)=O)CC2)C1 c1(CN(C(C2CCN(Cc3cccc(C(C)C#N)c3)C2)=O)CC)ccc(OC)cc1 c1(C(=O)NCCNC(C2(CF)CC2)=O)cncc(C2CCOCC2)c1 N1(C(C(C(C)C)C)=O)CCC2CCN(C(=O)CSc3ccccc3)C2C1 Cn1nc(C2CC2)c(Br)c1C(N1CCCC1Cn1cc(CCCCCO)nn1)=O N1(C(C23CCC(OC)C2C3)=O)CC(NC(=O)C(F)=CCCF)CC(O)C1 C1(C(=O)NCCCCNC(c2cc(-c3ccco3)no2)=O)CCC2(CC1)CC2 C=CCC(C(=O)N1CC2CN(C(=O)Cn3ncc(O)nc3=O)CC2C1)C(C)C c1(CC(=O)Nc2onc(C(=O)OCC)c2C)ccc2n[nH]cc2c1 c1(CNC(c2n[nH]c(C)c2C)=O)cccc2c1CCN(C(C1(C)CC1Br)=O)C2 c1(C(=O)NC(CC=C)CNC(C2(CCN(C)C)CC2)=O)cc(CSC)c(C)s1 N1(C(c2c(C)ncc(Cl)c2)=O)CCCN(C(=O)Cc2cccc(F)c2)C(CO)C1 n1(CC)nnc(C)c1C(=O)N(CCC(C)NC(=O)COCCOCCO)C C1(NC(C2(C)CN(C)C(=O)C2)=O)CC2CCCC(C1)N2C(C12CCC(C1)C2)=O C1CCCCCC(=O)N1.C1(C2CCN(c3nc(C=CC(N)=O)nc(=N)[nH]3)C2)(SC)CC1 N1(C(C(C)Sc2cccnc2)=O)CCC2CCC(C1)N2C(=O)CC(F)(F)F N1(C(Cc2ccc(CC)cc2)=O)CCCCC2(C1)CN(C(C1CCC1(F)F)=O)C2 C(=O)(CC(C(F)F)NC(c1cccs1)=O)NCC(N(OCC)C)=O c1(C(N2CCN(CC(=O)Nc3ccc(C)nc3)C(=O)C2)=O)cc(Cl)c(Cl)nc1Cl C(C(CNC(=O)COC(=O)CO)S(C)(=O)=O)NC(CCc1ncn(C)c1)=O c1(OCC)cc(C(=O)NCC2CCCN2Cc2cnc(Cl)nc2)ccn1 CC(C)CC(C(=O)NC(C(=O)N(C)C)C(C)c1ccccc1)C(N)=O c1(OC)cc(Br)c(CN2CCC(C(=O)Nc3cccc(C(C)=O)c3)C2)cc1O C(CCCC(=O)N1CCC(N(C)C(c2cccc(Br)c2)=O)C1)N(C)C N1(C(CCc2c(C)noc2C)=O)C2CCC1CC(C(N1CCC(C#N)C1)=O)C2 c1(CC)cccc2[nH]c(C(=O)NCC(C(C)C)NC(C3CC(F)C(=O)N3)=O)cc12 CC1CN(C(=O)Cc2ccccc2)CCN1C(=O)Cc1cnc[nH]1 N1(C(=O)COC2CCCOC2)CC2CCN(C(c3cc4c([nH]3)CCCC4)=O)C2C1 CCC(C)(C)CC(=O)N1CCOCCC1C(=O)NC1CC(=O)N(CC)C1 C1(C(=O)NC(C)CNC(c2cc(F)ccc2Cl)=O)CCc2ccccc2O1 C12(C(=O)NC3C(NC(=O)CC4CC=CC4)CCCC3)CCC(=O)N1CCS2 C#Cc1ccc(OCC(=O)NC2CN(Cc3ccn(C)n3)CCCO2)cc1 c1(C(N2CC3(CN(C(=O)CCc4nc[nH]n4)C3)C2)=O)cc2ncccc2o1 c1(CCC(=O)NCCN(C(C2CC2CC(C)C)=O)CC)cncc(O)c1.C1(C)CCC1 CCC(C(=O)OCc1nc(=N)[nH][nH]1)SC.C1(O)CCCC1 N1(C(C2CC(C)(C)C2)=O)CC(F)CC1C(=O)NC1CCCN(CCO)C1 CC12CN(C(=O)CC3CCC(C)(C)C3)C(C(=O)NC3C(C)(C)C3(C)C)(C1)C2 C1(C(=O)NCCCCNC(=O)CCNC(c2ccco2)=O)CCCC(C)(C)O1 c1(C(=O)NC(CNC(C(CCC#C)O)=O)(C)CO)ccc2oc(O)nc2c1 C1(CN(C(CSC(C)C)=O)C)CCCC(NC(c2conc2C(C)C)=O)C1 N1(C(C2N(C(CC3CCCN(C)C3)=O)CCC2O)=O)CCCC2(C1)N=N2 C1(C)(C(=O)NCC(C(C)C)NC(C2(CO)CCCO2)=O)CCC(=O)NC1 C=CCC(C)C(=O)N1CC(NC(=O)Cc2ccc(C)cc2)C(O)C1 c1(C(N2C(CNC(CCC=C)=O)COCC2)=O)ccnc(Cl)c1F c1(C(=O)NC2C(SC)CN(C(=O)CC3(O)CCOC3)C2)cc(Cl)cc(Cl)c1 c1(C(=O)NC2CCC(NC(c3cnc(C)[nH]3)=O)C2)ccc(Cl)c(Cl)c1Cl c1(C(=O)NC2C(NC(CC(C)n3cccc3)=O)COC2)cnc2cccnc2c1 CCCCC(CC)CC(=O)N1CCC(F)(C(=O)NC2CC(=O)N(C(C)C)C2)CC1 Cc1ncc(C(N2CC3CC3(NC(=O)CCCc3ccc(C)s3)C2)=O)c(=N)[nH]1 CN=S1(=O)CCCC2(CCCN2C(=O)C(=O)Nc2ccccc2P(C)(C)=O)C1 N1(C(CCCNC(c2nc(C(F)(F)F)cn2C)=O)=O)CCC(OCC2CC2)CC1 C1(NC(C2CC(CC)C2)=O)CC2CCC1N2C(c1cc(Br)cn1C)=O N1(C(Cn2ncc(C)c2)=O)CCCC(CO)(NC(c2cc(=O)cc[nH]2)=O)C1 O=C1CCN(CCn2cccnc2=O)C(=O)N1CC(c1ccccc1Cl)O N1(C(C(n2ncc(C)c2)C)=O)CCCC(F)(CNC(=O)C(C)CC(C)C)CC1 C(=O)(C1COc2cc(C)c(C)cc21)NCCCn1cc(CC=C)nn1 CC1CC(C)(C)N1C(=O)CN1CC(NC(c2ccncc2)=O)CC1=O C1(C(N2CCCC(CN(C(=O)CNS(N)(=O)=O)C)C2)=O)CC(=O)NC(C)C1 c1(C(=O)NCCC2N(C(CCCCC#C)=O)CCSC2)cn2cc(C)sc2n1 S(=O)(=O)(CC(CC(F)F)C(C)(C)C)Nc1ccc(CNCC)s1 Cc1cc(C)c2[nH]c(C(N3CCCC(NC(c4occc4F)=O)C3C)=O)cc2c1 C1(C)(CNC(c2c(C)c[nH]n2)=O)CCCN(C(=O)CC2CCSC2)C1 c1(C(=O)OC)cc(C(=O)NCC=CCNC(c2cc(OC)cnn2)=O)ccc1O N1(C(CCc2ccc(C)s2)=O)CCC(CCNC(c2cnnn2C2CC2)=O)CC1 N1(C(C(CCCCC)O)=O)CCCCC2(CCN(C(=O)CC3COC(=O)C3)C2)C1 c1(OCC(=O)NC2(c3onc(C)n3)CCC2)ccc(Br)c(F)c1F C1(NC(CCN2CCC(C)CC2)=O)CN(C(c2cncn2C)=O)CC2CCCC12 C1(CN(C)Cc2onc(CC)n2)CCC2(CCCOC2)O1 Cc1cn2c(C)c(C(N3CC(NC(c4cccc(OCCF)c4)=O)C3)=O)nc2s1 C12(C(=O)NCCCC#C)CC(CO1)N(C(=O)C(O)C1CCC1)C2 C1(OC)(CNC(=O)Cc2ccno2)CN(C(c2sccc2C)=O)C1 N1(C(CC=C)=O)CCC(C(C)NC(C2CNC(=O)N2)=O)CC1 C1(NC(C2CCSCC2)=O)CCCCC1CNC(C1CC2CCC1C2)=O C1(NC(C(=O)NCCCOCCCC)=O)CCCN(C(C2CC3CCC2C3)=O)C1 c12cccc(c1)CC(=O)NCC(C)CNC(=O)C(C)C2.C1(CC)CC1COC c1(CCC(=O)OC(c2cccs2)C)nc(-c2ccoc2)no1 C#CCCCCCC(C(=O)OC)N1CC(N(C)C(=O)OC(C)(C)C)CC1C.OCC N1(C(C2C(OC)CCCC2)=O)CC2(CCCN(C(=O)C(C)(C)n3cnnn3)C2)C1 c1(C(=O)NC2CN(C(C3(COC)CCC3)=O)CC2C)cc(S(C)(=O)=O)ccc1Cl c1(CC(N2CCC(CNC(c3cc(C(N)=O)no3)=O)C2)=O)cc(Cl)ccc1Cl c1(CCC(=O)N(CCCCCNC(C(C)C#N)=O)C)nc(O)c2cnn(C)c2n1 C1(CCCNC(CC(C)OC)=O)CCN(C(C2CC2c2ccncc2)=O)CC1 Cc1cn2c(C(N3CC(NC(=O)CCC(C)(F)F)C3)=O)c(Cl)nc2s1 c1(COC)ccc(C(=O)NC2CN(C(=O)Cc3cc[nH]c3)CC23CC3)cc1OC C1(C(=O)NCCCN(C(C(C=C)(C)C)=O)Cc2ccccc2)CC12CCCCC2 N1(C(C2(CC=C)CN(C(c3cc(OC)ns3)=O)C2)=O)CCC(O)C(O)C1 c1(C(=O)NC(C2CCCC2)CNC(c2cn(C)nc2)=O)cc2cccnc2s1 N1(CC)CCN(C(=NCCC(=O)N(C)C)NC2CCCN(C(CSC)C)C2)CC1=O CN1CCC(CCNC(=O)C(C)(C)NC(=O)CC2NC(=O)NC2=O)CC1 C(=O)(CC1=CCCCC1)N(C)CC1(C)CCCC1NC(=O)Cc1cnc[nH]1 c1(C(=O)NCCCC(C)NC(=O)C(C)OCC(C)C)cc(C2CC2)oc1C1CC1 C1(NC(c2ccnc(C(F)F)c2)=O)CCC(NC(=O)C(C2CCCCC2)F)CC1 N1(C(C2C(CC)CCC2)=O)Cc2ccccc2C1CNC(c1cc(CO)on1)=O c1(C(N(CCCNC(c2cnnn2C)=O)CC)=O)ccnc(-n2ccnc2)c1 Cc1ncc(S(N)(=O)=O)cc1C(=O)N(CC(C)O)CCO C(N=c1ccnc(Cl)[nH]1)C1C(C)CN(C(c2ccc(CN(C)C)cc2)=O)C1 N1(C(C(C)N(C(C2(C(CC)=O)CC2)=O)C2CC2)=O)CCC(C#N)CC1 CCCC(C)CC(=O)N1CC=CC1CNC(c1ccc(N(CCO)CC)cc1)=O c1(C(=O)NCCCN(C)C(c2c(O)cc(O)cc2O)=O)cc(F)cc(F)c1O CC1OCC2C(=O)N(CC3CCCN3)C(=O)N2C1=O CC1OC(C)Cc2c(C(N3CCN(C)C(CF)C3)=O)n[nH]c21 c1(-n2c(C(c3cc(C)on3)NCC(C)(C)C3CCC3)nnn2)ccccc1C CCC(CC(=O)N1CCC(CCCNC(c2c(C)nsc2NC)=O)CC1)C(C)C C1(C(N2CCC(N(C(c3cc(C)nnc3)=O)C)C(C)C2)=O)CCCCC(F)(F)C1 N1(C(C)C)CCCC(NC(=O)C#CCNC(=O)C(N2CC(C)(C)C2CN)=O)C1C C(=O)(C(CP(C)(C)=O)NC(c1c(Cl)cnn1CCN1CCC(C)CC1)=O)OC c1(N(CC(F)F)C)nc(=NCc2cc(N)ccc2Cl)[nH]c2ncn(C)c12 c1(C(N(C(C2CCC(C(=O)OC)CC2)C(=O)NCC)C)C)nc2ccccc2s1 C1(C)(C(=O)NCC(C2CCC2)OCC)CC(O)CN1C(c1ccc(CC)s1)=O N1(C(C(C(=O)OC)C)=O)CC2CC1CN2C(=O)CC1CCCN1C(=O)OC(C)C N1(C(CC2(C(=O)OC)CC2)=O)CC2(C)CC1C2NC(=O)C(c1cccc(Cl)c1)C c1(CCC)c(C(=O)NC(CO)CCCNC(=O)CC(C)COC)nnn1CC c1(CNC(=O)NC2(CC3C(OC)C4C3CCC4)CC2)ncc2nccnc2n1 N1(C(C2(C)CC(F)(F)C2)=O)CC(C(=O)NCC(O)C2CC2)CCC1(C)C N1(C(C2(NC(C)=O)CCCC2)=O)CCN(CCC(N2CC(O)(CO)C2)=O)CC1 Cc1c(C(N2CCC(O)(CNC(C3C4CNC(=O)C34)=O)C2)=O)[nH]c2ccccc12 C1(NC(c2c(SC)nn(C)c2)=O)CN(C(C2(F)CCOC2)=O)CC1(C)C N1(C(c2ccc(CC)cn2)=O)CCN(C(=O)CC(C)(C)O)C(CCOC)C1 C(=O)(CCCC(C)(C)C#N)N1CCC(NC(C#CC2(CC)CC2)=O)C(F)C1 c1(C(N2CCN(C(C3N(C)C(=O)OC3)=O)CC2CO)=O)cc2ccccc2s1 C1(C(C)C)CCC(C(=O)NC2(COC)CCN(C(=O)CC3CSC3)C2)C(=O)N1 C1(C(=O)OC)CCC12CN(CC1NC(=O)CC1(C)C)C2 C(C)(CNC(=O)CSc1ccc(Cl)cc1)(CC(C)C)NC(c1sc(C)c(O)n1)=O C1(CC(=O)NC(C(=O)N(C2CC(OCC)C2)C)Cc2cnc[nH]2)COCC(C)O1 N1(C(C(C(C)C)O)=O)CC(NC(=O)COCc2cccnc2)CC(C)(C)C1 N1(C(C2CCCC(NC(c3cncc(C)c3)=O)C2)=O)CC2(CNC(=O)C2)C1 N1(C(c2cn3c(n2)SCC3)=O)CCC2CN(C(=O)CC(F)F)CCC2C1 n1(C2CC(C)(F)C2)nc(-c2cccnc2)nc1C1CC1C1CC1.C1CC1 CC1(C#CC(=O)NCC2COCCN(C(c3cccs3)=O)C2)CC1 O=CN1CCOCC1C(N1CCC(O)(CNC(=O)Cc2ccncc2Cl)C1)=O CC1(C)OCCC1C(=O)NCC1CCN1C(c1ccccc1C(N)=O)=O N1(C(c2cccc(NC(=O)NC(C)C)c2)=O)CCOC2(CCOCC2)CC1 CC1(C)CCN(C(=O)C2=C(Cl)CCCC2)C(C(N2CC(C34CCC(CO3)C4)C2)=O)C1 c1(CN2CCC(c3ccccc3)(C(=O)O)CC2)cc(F)c(Cl)cc1C Cc1ccc(C(N2CC(O)C(O)C2CNC(=O)CCc2ncc[nH]2)=O)c(C)c1 c1(C(=O)NC2CC(NC(C=C(COC)C)=O)C23CCC3)ccc(Cl)c(F)c1F C#Cc1ccc(C(N2CCOC(C(=O)NC3CCN(C(C)C)C3)C2)=O)cc1C c1(OC)cc(CNC(C2CC(OC)CN2C(=O)C(C)NC=O)=O)cc(C)n1 C1(C(=O)NCc2ccnc(F)c2)(COC)C=CCN1C(=O)Cc1cc(C)oc1C N#Cc1ccnc(NC2C3CN(C(=O)C(O)CC4CCCCC4)CC23)n1 c1(C(c2nnnn2C2COC2)NC2(CCCCC)CC2)ccc(Cl)c(Br)c1 c1(C(N2CCCC(CCNC(CS(CC)=O)=O)C2)=O)ccc(C(C)C)c(N)c1 C1(C(=O)OC(C)(C)C)(NC(=O)CCCn2cc(C3(O)CSC3)nn2)CCN(C)C1 CS(=O)c1ccc(C(=O)OCCn2nc(Cl)ccc2=O)cc1 c1(CN2CC(C)(CC(=O)NCCCC3COC(=O)C3)C2)c[nH]c2nccc-2c1 c1(OC)cnncc1C(N1CC2CC2(CNC(c2cc(Cl)cn2C)=O)C1)=O c1(C2C(C(=O)NC(C3CN(C(=O)C(F)(F)C4CC4)C3)C)CC2)ccccc1F N1(C(C2CC(C#C)(O)C2)=O)CCC(CNC(=O)CSC)C1(C)C N1(C(CCC=CC)=O)CC2CN(C(c3c(C)[nH]c(C)c3C)=O)CC2C1 N1(C=O)CCC(C(F)Cc2c(C(C)(C)OC)ocn2)CC1.C(=O)(C(Cl)=CCl)N C1(NC(c2c(CCC)n[nH]c2)=O)CCN(C(=O)CCc2csc(CC)n2)CC1O n12ncc(c1C(F)(F)F)C2.C1(C(=O)OCC)C=CCN1C(=O)CC(C)C N1(C(c2cccc(NC(C)=O)c2)=O)CC2CN(C(=O)CC3=NNC(=O)C3)CC2C1 C1(COC(=O)CCc2cocn2)COc2ccccc2C1 c1(C(N2C(CO)CC(NC(CSC(C)C)=O)C2)=O)cnc2n1CC(C)CC2 c1(C(N2CC3(CCCC3)C2)=O)cc2cc(Cl)cc(Br)c2[nH]1 N1(C(C(C(C)C)OCC)=O)C(CC(=O)N(C(C)C(F)F)C)C2CCCC12 C1(CNC(C2(F)C(C)OCC2)=O)CN(c2ncnc(=N)[nH]2)CCCO1 C1(COC)(CNC(=O)C(N)=O)CCN(C(c2cc(C(F)(F)F)n(C(F)F)n2)=O)C1 C1(CCOC(C(C)Oc2ccccc2)=O)CCN(C(=O)C(C)(Cl)Cl)CC1O c1(OC(C(=O)NC2CCN(C(C3C(C)CC3)=O)C2)(C)C)ccc(F)cc1 N1(C(C(C)C)=O)CCC2OCCN(C(C34CCC(=O)N3CCS4)=O)C2C1 C1(F)(CNC(=O)CC2CC3CC3C2)CC2CCC(C1)N2C(c1cnc(O)o1)=O C(=O)(C(O)C(C(C)C)OC)NC(C(=O)NCC(C=C)(C)C)CSCC C=C(C)CC(C(=O)NC1CCOC1C(N1CCCC1CNC(N)=O)=O)OC Cc1cc(Br)ccc1C(N1CC(O)(CCNC(=O)CSCC(N)=O)C1)=O C(=O)(CC(C)C(F)(F)F)NC(CCC)CNC(C1CCCN(CC)C1)=O C(CCN=[N+]=[N-])NC(CN(CCOC)C(C1(C)CC1C)=O)=O.CO CC1CN(CC(O)Cc2ccc(C(C)(C)C)cc2)C(=O)N1 CCC(C)(C)CCCC(=O)N1CC(O)CCC1C(N1CCC(C)C1)=O N1(C(c2cc(C(N)=O)c(F)cc2)=O)CC2CCC(NC(=O)CS(N)(=O)=O)CC2C1 c1(C(CNC(CC2(COC)CC2)=O)NC(c2c[nH]nc2C)=O)ccc(C#N)cc1 C1(NC(=O)CCF)CCCCN(C(c2cccc(Br)c2Cl)=O)CC1 c1(C(N(CCCC)C(C)CC)=O)coc2c1CN(C(=O)C(CC1CC1)OC)C2 C1(C)(N(C)C)CCCN(C(C2C=CCCN2C(C2CCOC(C)(C)C2)=O)=O)C1 CCC(CC)C(=O)N(CCOC)CC.C12CCN(C1)CCN2 c1(C(=O)NC2C(CC)CN(C(=O)CC3CCNC3=O)C2)c(Cl)nn(C)c1Cl CCCCC(CNC(=O)C(C)(CC)OC)NC(=O)CCc1ccc(C(C)C)cc1 CC1(C)C(S(=O)(=O)NC(c2cccc3c2CCNC3)=O)C1(C)C N(C(=NCCN1CCCS1(=O)=O)NCC1(N2CCCC2)CC1)CC(C)OC CC(C)CC(CNC(c1cocn1)=O)NC(=O)C1=NOCC1 c1(OC)ccnc(CNc2cc(N3CCCC(C)C3)ncn2)c1OC c1(N2C(CN(C(C(C)c3cccs3)=O)C)CCC2)ncc([N+](=O)[O-])c(=N)[nH]1 CCCCCCCCC(=O)NCC1CC2CN(C(=O)CC(C)(C)OC)CC12 c1(-c2cnc(N3CC(C(=O)OC)C3)c(O)c2)cnn2c1CCCC2 CC(CN=c1[nH]c(=NCc2c(F)cccc2Br)[nH]c2c1CCCCCC2)S(C)(=O)=O CC1CN(C(C2CCCS2)=O)CC1N=c1nc(N2CCOCC2)[nH]c2ccsc12 c1(C(=O)NCCOCCNC(C(C(C)C)OC)=O)ncc(C)cc1Br c1(OC)cc(Br)cc(C(N2CCC3(CCC3)C2)=O)c1NC(=O)C1CC1 c1(N2C(C#N)CN(CCF)CC2)nsc2cc(-c3ccnn3C3COC3)ccc12 [SH](=O)(=O)CC[Si](C)(C)C.CC=C=CCCC.C(=O)C c1(SC)cc(C(=O)NC2CCC2NC(=O)CCc2cncn2C)oc1C N1(C(c2ncn(CC)c2)=O)CCCC(C2CCN(C(=O)COc3ccsc3)C2)C1 C(=O)(CC(C)(C)C(=O)NCC(C)N(C)C(C1CN2CCC1(C)CC2)=O)OC N1(C(C(CC2CC2)OC)=O)CCCCC1CNC(=O)CCCCSC C(CS(=O)(=O)NCC(=O)NC(C)(C)C=CCOC(C)(C)C)OCC=C.CCN c1(CC(=O)N(C2CCN(C(c3ccc(C)n3C)=O)C2)C)nccc2ccccc12 Cc1cc(CN2CCC(C(=O)N(C)CCN3CCCCC3)C2)n(C)n1 c1(C2C(C(=O)NCc3cc(SC)ncc3)CCNC2)cnc(SC)c(C)c1 CCCS(=O)(=O)CC(=O)NC(CNC(c1ccn2ncnc2c1)=O)CCOC C1(C(=O)NC2CCN(C(C)C)C2=O)CC2CN(C(=O)CP(C)(C)=O)CC2C1 C1(C(=O)NCc2occ(C(=O)NC(C#C)CC3CCCO3)n2)CC12CCCCC2 c1(C(=O)NC2CN(C(c3c(C)oc(Cl)n3)=O)CC2(C)C)cc([N+](=O)[O-])ccc1N CN1CC=C(CC(=O)NC2CCCC2NC(=O)C(C)(C)c2cncnc2)CC1 c1(C(N2C(C(=O)NCC(CCC)CCC)CN(C)CC2)=O)cn2ccccc2n1 c1(C(N2CCCC3CCCC23)=O)cccc(S(=O)(=O)C(F)F)c1 O=C(C1c2c[nH]nc2CN1C(=O)Cc1cn[nH]c1)NCCC1CCCCC1 C1(C(=O)NC(C2CCCCC2)CC)C(C)OCCN1C(=O)CN(C)C1CC1 C1(C(=O)OC)CN(C(CC(O)C(C)(C)O)=O)CC12CCC2 C(=O)(C(O)C(C)C)NC1(CC=C)CN(C(c2ccnn2CC#N)=O)C1 C#Cc1cc(NC(C2(NC(=O)C(CCC)NC(N)=O)CCC(C)(C)C2)=O)ccc1C Cc1c(Cl)cc(C(=O)NC2CCC(C(=O)Nc3ncc(C#N)cc3I)CC2)cc1Cl c1(C(=O)NCCN(C(CSC)=O)Cc2ccc(C)cc2)ccc(OCF)cc1 C1(NC(CNS(NC)(=O)=O)=O)CC2CC(NC(C3(C)CC(C)C3)=O)CC2C1 C1(CNC(C(C2CC2)OC)=O)(CNC(c2nc(COC)cs2)=O)CCOCC1 c1(C(=O)NC(C2CCN(C(=O)CSCCN(C)C)C2)C)ncsc1Br CC1CN(C(c2ccncn2)=O)C(C)CN1C(c1nnn2c1CSCC2)=O c1(C(N(C(C2CCC(C)C2)C(=O)NCCOC)C)C2CC2)ccc(F)cc1F C1(C(N(CCNC(c2ccc(C(C)=O)o2)=O)C)=O)CC1C1CC1C c1(CN(CCCC)C(c2cccnc2)=O)cnn2c1NCC(C)C2 C1(CNC(C(CC)NC(N)=O)=O)CN(C(c2cccc(Cl)c2F)=O)CC1(C)C CC1CCN(C(=O)CN(C)C(=O)C2CC2)CC1CNC(=O)C(F)(F)C1CC1 c1(C(N2CCN(C(=O)C(=Cc3cccnc3)F)C3C2C3)=O)ccc2c[nH]nc2c1 Cc1conc1C(=O)NCCCC1CCCN1C(c1ccnn1C(C)(C)C)=O Cc1nc(C#N)c(NCCC(N2CCC(NC(c3cn(C(C)C)cn3)=O)C2)=O)o1 Cc1cccc(C(=O)NCC(CO)NC(=O)C=Cc2cnc(C(C)(C)C)s2)c1 C1(C(N2C(CNC(c3cc(CC)on3)=O)CCC2)=O)CCC(C)(C)CC1 CC1CC(C(=O)NC2(CNC(=O)CCN3CCNC(=O)C3)CC2)CC(C)O1 N1(C(c2ncc(CO)o2)C(=O)NCCCOC)CCn2ncc(CN(C)C)c2C1 C(=O)(C1=CCCCC1)NC(C(C)OC)C(=O)NCC(C)N(C)C C1(NC(C=C)=O)CCCC12CN(C(C1CCC(C)=C(C)C1)=O)C2 N1(C(C(=O)NC(C)C)=O)CC2CN(C(C3CC(F)C(=O)N3C)=O)CC2C1 CCCC(C)(C)C(=O)N1CCC(CCNC(c2cc(C(N)=O)[nH]n2)=O)C1 CC12CC(CCO1)N(C(C1C3CCC(C3)N1C(C1CCCC1F)=O)=O)C2 c1(C(N2CCOCC(CNC(CC3CC(OC)C3)=O)C2)=O)ccc(C)c(C#N)c1 c1(CNC(C2CCN2C(=O)Cc2ccc(Br)cc2F)=O)ccc(Cl)nc1F c1(C(=O)NCC(CC)N(C)C(c2ncnn2CC(C)C)=O)cc[nH]c1C1CCC1 C(C)(CC(=O)N1CC(O)(CNC(c2ccc(CO)s2)=O)C1)(C(F)F)N(C)C N1(CC(=O)NC2(C(F)F)CCNC2)CCN(C(C)C)CC1 C(=O)(C1=C(C)N(C)c2ncnn2C1)N1CC(N(C(CCCC=C)=O)C)C2(C1)CC2 N1(C(CC(C)C2CCCO2)=O)CCCOC(CNC(=O)CC2CCC3(CC2)CC3)C1 C12(CNC(C(C)Sc3ccccn3)=O)CC1CN(C(=O)CCc1ncc[nH]1)C2 Cc1c(C(N2CCOC(CN(C(=O)C(C)C#N)C)C2)=O)nnn1-c1ccn(C)n1 C1(C(=O)NCC2N(CC(=O)OC(C)(C)C)CCC2)CC2(CCCCC2)CO1 C1(NC(C(CCCOC)C)=O)COC2(C1)CN(C(c1ccc(O)cc1OC)=O)C2 C(CC(=O)NCC1CN(C(c2ncc(C)cn2)=O)CC1(C)C)(C(C)C)OCC c1(C(N(CC(C)N(C(CC(CC)(C)C)=O)C)C)=O)cn2c(n1)CC(C)CC2 CN1CCN(CCC(=O)NCCC2CN(C(=O)CCc3cnn[nH]3)CCO2)CC1 c1(C2(C(=O)NC3C(CNC(c4c(C)cn(C)c4)=O)C3)CCC2)c(F)cccc1F C1(O)(C(N(CCN(C(=O)CCCc2ccncc2)C)C)=O)CC1(C)C c1(C(N2CCC(N(C(C(C=C)O)=O)CCC)CC2)=O)ccc(C2=CCCC2)cc1 Cc1ccc2ccsc2c1N1CCCn2cc(C(C)(C)C)nc21 c1(CNC(=O)CC(F)F)cccc(NC(=O)CCCOc2ccccc2Cl)c1 c1(OC)ccc2[nH]nc(C(N3CCCC4CN(C(=O)CCCCO)CC34)=O)c2c1 C1(CNC(C(C)OC2CCCC2)=O)CC2CCC(C1)N2C(=O)Cc1cn[nH]c1 N1(C(C2(F)CCN(c3ncc(Br)cn3)C2)=O)CCC(NCc2ncn(C)c2)CC1 Cc1ccc(C(=O)NCC(=O)NC(C)(C)CN(C2CCC(O)CC2)C)cc1 c1(CNC(C2CC(=C)C2)=O)nnn(C)c1C(=O)NCC1COC(C)C1 Cc1cncc(C(=O)NC(C)CN(C(=O)COCc2nc[nH]n2)C)n1 C1(C(NOCCN(C)C)=O)N(C(=O)C(CO)C(F)(F)F)CC12CCCC2 N1(C(C(CCC)OC)=O)CCC(O)(C(C)NC(=O)CC=C(C)C)CC1 C1(CCC)(OC)CCN(C(c2ccc(CNC(C3CC3CCOC)=O)[nH]2)=O)CC1 CC(C)C(O)C(C)C(=O)NCCC(C)(C)CNC(=O)C(C)(C)CF c1(NC(CN(C(C2CC23CCCOC3)=O)CC)=O)cccc2c1OCO2 N1(C(c2c(CNC(C3C(C)C3)=O)cco2)=O)CCC(C#N)CC12CC2 N1(C(C(C)CC2CCC2)=O)CCCC(CCNC(C2CC23CC3)=O)C1 C1(C(=O)NCC(CCC)OC)CC(C)CN1C(=O)C=Cc1ccncc1 C1(CC)CN(C(C2CC2CN(C)C)=O)CCO1.c12ccncc1NC2=O Cc1c(CN2CCCC(C)(CNC(=O)CC(C)O)C2)cccc1Br C(N=c1ccc(S(=O)(=O)NC2(C)CCCC2O)c[nH]1)c1c(C)noc1C c1(C(=O)NC(C)C)ccccc1NC(N)=O.C12CCN(C1C)C(=O)CC(C)N2 N1(c2nc(NC3CCCC(NCC)C3)nc(C)c2)CCC2CC(=O)NC2C1 c1(C(N2CC(CCNC(C3C4CC4C4CC34)=O)(OC)C2)=O)cccn2ccnc12 N1(C(C(CC)c2ccccc2)=O)CCC(c2cn(Cc3nccs3)nn2)CC1 Cc1nn(C)c(Cl)c1CC(=O)NCC(C1CC1)NC(c1ccc(=N)[nH]c1)=O C#Cc1cn(C)nc1C(=O)NC1CN(C(C2CN(C)CC(C)O2)=O)CC1C C1(N(C(CC(C)SC)=O)C)CCN(C(c2[nH]cc(C)c2C)=O)CC12CC2 O=C1C(C(N2CCC(Oc3ccccc3)C2)=O)C1(F)F C1(C(=O)NC2CC(C)(C)N(C(c3ccsc3Cl)=O)C2)CC12CCC(=O)CC2 c1(NC(c2ccn(CCNC(C(C)OCCCC)=O)c2)=O)cccc(N=[N+]=[N-])c1 C1(CC(=O)NC)(NC(CNC(C2CCC2)=O)=O)COC1.C(=O)(NC)NCCO N1(C(C(C)OC(C)(C)C)=O)CCCC(C)(NC(c2nncnc2N)=O)C1 C12(C(=O)NC3CN(C(c4c(C)c[nH]c4)=O)CC3O)CCC(C)(CC1)CO2 Cc1nc(C(=O)NC2CCN(C(c3cc(C(F)F)ccn3)=O)C2)cn(C)c1=O CC(C)CS(=O)(=O)CCC(=O)NCC12CC(CN1C(=O)C(C)C(C)(C)C)C2 C(CCCCCC(=O)N1CCC(F)(CO)CC1)NC(c1cccc(O)c1)=O N1(C(C(C)C2CC2)=O)CCN(C(=O)C=CC2CCOC2)CC1C c1(C(N(CCCNC(C=C(CCC)C)=O)C)=O)ncc(Br)cc1Cl CCCCC(O)C(=O)N1CCOC(Cn2cc(CCC3CCOCC3)nn2)C1 C1(NC(CC2CCCN(Cc3n(CC)ncc3)C2)=O)CCC2(CCCC2)C1 c1(C(N2C3CCC(NC(C4(CC=C)CCC4)=O)C(C3)C2)=O)n[nH]c2c1CCSC2 c1(C(N2C(C)CC(NC(c3csc(O)n3)=O)C2)=O)cnc2occc2c1 c1(C(N2CCCC(C)(NC(=O)CC3CSCCS3)C2)=O)cc(F)c(F)cc1N c1(C(N2C3CC(NC(CN(CCC)C)=O)C(C3)C2)=O)ccc(S(N)(=O)=O)cc1N C(CCC(CCC)NC(c1cscc1C#N)=O)NC(C1C(=C)C1)=O C1(CC)(NC(=O)C=Cc2cscn2)CCN(C(=O)CC2CCCC(C)(C)O2)CC1 N1(C(c2ccn(C(C)(C)C)c2)=O)CCCC(N(C(=O)CC2CCCCO2)CCF)C1 Cn1nnc2ccc(C(=O)NC3CC(F)(CNC(=O)C(O)CC(F)F)C3)cc12 C1(CNC(=O)NC(C2CCCN2C)C)CCCN(C)C1 C1(CNC(c2ccc(C)cc2)=O)CCC12CCN(C(c1[nH]ncc1C#N)=O)CC2 C(=O)(C(CSC)NC(=O)C(O)CSCC)N(CC=C)CCO Cc1ccc(O)c(C(=O)NC2CC(c3ccc(Cl)cc3)(C(=O)O)C2)n1 C1(NC(C(COC)N(C)C)=O)CCN(C(c2cn(C)cn2)=O)C(C2CC2)C1 Cc1ccc(C(N)=O)cc1NC(=O)COCC(C)NC(=O)CC1CCC(F)(F)C1 N1(C(C2N(C(C3(COC(C)C)CCCO3)=O)CCC2)=O)CCC2CN(C)CCC12 N1(C(C2CC2C(=O)N)=O)CCCN(C(=O)C(F)(F)CO)CC1CC1CC1 c1(NCCNS(C)(=O)=O)cn(C2CCC(C(OCC)OCC)C2)nn1 N1(C(c2c(CNC(=O)Cc3cccc(F)c3)n[nH]c2)=O)CC2(CCCC2)C1 C(=O)(CC(C)C(F)(F)F)NC(C(N1C(C#C)CC1)=O)Cn1cncn1 S(=O)(=O)(c1ccc(C)c([N+](=O)[O-])c1C)N1CC(C=C)C(O)C1 N1(C(C2CCC(OC)C2)=O)CC2CCCC(C1)N2C(c1ccn2ccccc12)=O C(C(=O)NCC#CCNC(C1CCC(F)C1)=O)(c1ccccc1)=C(C)C N1(C(C2C(OCC)C2)=O)CCC2(CCN(C(=O)Cc3coc(C(F)F)n3)C2)C1 C#CC(CNC(=O)CN(C(=O)CC=CCC1CCC1)C)C(C)C CCCC(CC)CC(=O)NCCC1CC(CNC(=O)CC(COC)N=[N+]=[N-])C1 CC1(CCNC(=O)COCc2ccncc2)CCN(C(C2CC2(Cl)Cl)=O)C1 C#Cc1c[nH]nc1C(=O)NCCC1CC(NC(=O)CNC(=O)NC)C1 N1(C(Cc2cc(OC)ncc2)=O)CCC(F)C(NC(c2c[nH]cc2C)=O)C1 CCCCC(CNC(c1ccn(C2CC2)n1)=O)NC(C1CCOC1(C)C)=O Cc1nnn(C)c1C(=O)NCC1CN(C(=O)Cn2cnnc2)CCO1 c1(C(N2CCCN(C(CC(C)C)=O)CC2)=O)cc2ncc(Br)cc2o1 c1(C(N2CC(NC(c3[nH]cc(C#N)c3)=O)C(C(F)F)C2)=O)ncnc(O)c1Cl NS(=O)(=O)CCCCCC(=O)NC1CN(C(c2ncc(Br)cn2)=O)C1 C1(C(=O)NC2(C(C)(F)F)CC2)C(NC(=O)CC#N)C1(C)C C(=O)(C(F)C(C)(F)F)N(C(C(=O)NCC12CC(CCO1)C2)C1CC1)C C(=O)(C(C)CC(C)(F)F)NC(CC)CNC(c1ccc(C2CC2)nc1C)=O CC1(C)CC1(C#N)C(=O)NC1CCC(CC(=O)NCC2(CO)CCCO2)CC1 Cc1ccc(C=CC(N2CCCC(CCNC(c3cnc(N(C)C)o3)=O)C2)=O)o1 c1(C(N(C2CN(C(CC(C=C)(C)O)=O)C2)C)=O)ccc2ccnc(O)c2n1 c1(CC)ncnc(CC)c1C(=O)N(CCCCNc1nccc(C(F)(F)F)n1)C c1(CC(=O)CC2(CNC(=O)COCC)CC2)cccc(F)c1.C(CC(F)(F)F)N C1(C(F)(F)F)(OC)CCc2c(NC(C3C(Cl)(C(=O)OCC)C3)=O)cccc21 c1(CC(=O)NCC(CC)NC(c2cc(CO)ccc2Cl)=O)cnc2ccccn12 C(=O)(CCS(N)(=O)=O)NC(C(C)C)CNC(c1cccc(CC#N)c1)=O N1(C(C2CCOC2=O)=O)C2CCCC1CC(n1cc(CCC3CC3)nn1)C2 C=Cn1nncc1C(=O)NC1CC(F)(CNC(C2CN(C(C)=O)C2)=O)C1 C1(OC)CCC(C(=O)NC2CC(C)(NC(c3cnn(C)c3Br)=O)C2)CC1 Cc1ccc(CSCC(=O)NC2CC(NC(c3cc(C(F)F)[nH]n3)=O)C2)cn1 C1(NC(C(C)OC2CCOC2)=O)CC2CCC1C(NC(=O)CC(C)(C)O)C2 C1(CNC(C2CCN(C)C2=O)=O)CC(O)C(O)CC1C(=O)NOCC1(C#N)CC1 CC1(C(N2CCC(CCc3cccs3)CC2)=O)CCCN(Cc2cnsn2)C1 N1(C(CC=C(C)C)=O)CCCC2CN(C(C3CCOCC3(C)C)=O)CC12 N1(C(CC2(C=C)CN(C(c3cc(CC)ccc3O)=O)C2)=O)CCCCC(CO)C1 N1(c2ccc(=N)[nH]n2)C(=O)CCC(C(=O)N(CC(F)(F)F)CCl)C1c1ccncc1 c1(C(N2CC(NC(C=C(CC)CC)=O)CC(C)(C)C2)=O)cc2c(nc1N)CCC2 c1(C(=O)NC(C2(C(=O)NC3CCCC3(C)O)CC2)C)ccc(C)c(C#N)c1 c1(C(=O)NCC(CN(C)C(C2CCC(C)CC2)=O)O)cc2occc2[nH]1 C(CCS)N(C)CCN(C)CCC1CCC1 C(C(C(F)(F)F)CNc1nc(=N)cc[nH]1)NC(=O)OC(C)(C)C CC1C(=O)N(C)CCN1C(C(=O)NC1CCOC1)C1=CCSC1 N1(C(C(C2CCCC2)OC)=O)CC2CCC(CNC(=O)CN(C)C(C)C)C2C1 N1(C(C2(C)CCCCC2)=O)CC2CN(C(c3c[nH]c(=N)o3)=O)CC2C1CO CC(C)(O)C#Cc1cccc(NC(C2COCCN2C(C2CNC(=O)C2)=O)=O)c1 C1(CC(N2CC(C(CC)C)C2)=O)N(C(C2CCCN2N=O)=O)CCC1(C)C CCCCCC(O)C(=O)NCC1(C)CCCN(c2nc(OC)ncc2Br)C1 C1(CCNC(c2c(C(C)(C)C)[nH]cc2)=O)CCCN(C(=O)COC2CCOC2)C1 Cn1cc(C(=O)NCCc2n[nH]cc2C(=O)N(CCO)CC2CC2)nn1 n1(CC(N2C(CNC(C(C)(C)F)=O)CC2)=O)nc2n(c(=O)c1=O)CCOC2 c1ccc(-n2cc(CNCc3ccc(C4CCCCC4)s3)cn2)cc1 C1(CNC(C2(CC=C)CN(C(=O)COCC3CCCO3)C2)=O)CCOC(C)C1 C(=O)(CCCCCC(C)C)NC(C(C)NC(c1ccc(SC)cc1Cl)=O)CO N1(C(c2ccn(C)n2)=O)CCC2(CC1)CC(NC(=O)CCc1cncn1C)CO2 c1(C(=O)NCCC2N(c3nc(C)nc(=N)[nH]3)CCCC2)cnc2n1CCCC2C c1(C(=O)NC2CC(O)CN(C(=O)Cc3cscn3)C2)nccc2ncccc12 c1(C(=O)NC2CCN(C(C3CC(C)OC3C)=O)C(C)C2)cnc2[nH]cncc1-2 c1(NC(=O)NCC(C)Cc2cn[nH]c2)n[nH]c(-c2ccccc2)n1 c1(C(N(C2CCN(C(CC=CC)=O)CC2C)C)=O)cccc2nc(C)nn12 C(N=c1[nH]c2cccnc2s1)C1CCN(C(CSc2onc(C)n2)=O)C1 C1(NC(C(CC=C)C(C)C)=O)CCC2(CC1)CC(NC(=O)CCN1CCC1)C2 C1(NC(=O)OCC)CCOCC1NC1CCCC1C(=O)NOc1cccc(C)c1 N1(C(Cc2ccc(C)o2)=O)CCC2CCN(C(c3cc(Cl)ccc3F)=O)CC2C1 c1(CC)nc(C)c(C(=O)NCC2CCCCN2C(=O)Cc2ccoc2)c(C)n1 C=Cc1ccc(C(N2CC(F)(CNC(C3CC34CC(OC)C4)=O)C2)=O)cc1 N1(C(C(C)C2CC2)=O)CCC2CCC(NC(c3cc(F)c[nH]3)=O)C1C2 Cc1ccc(C(=O)NC2(C3CCCCN3C(c3csnc3Cl)=O)CC2)c(O)n1 C=Cn1nccc1C(=O)NC1COCC1n1cc(CN2CC3CC3C2)nn1 C1(CNC(C2CCCO2)=O)CCCCN1C(c1csc(-c2cccs2)n1)=O C(N=c1[nH]c(C)cc(=NC2CCCC(F)(F)C2)[nH]1)C1(SC)CCCCC1 N1(C(COCCOCC#C)=O)CCCC1(C)CNC(C1CCC1C(C)(C)C)=O C1(F)(C(N(CCCOCCNC(=O)COCC2CCCO2)C)=O)CCOC1 C1(N(C(CC2CCN(C(Cc3c(C)n(C)cn3)=O)C2)=O)C)CS(=O)(=O)C1(C)C c1(CCC)nc(C(N2CC(O)(CC)C2)=O)co1.c12n[nH]cc1CCN(C)C2=O C1(NC(C2N(C(C)=O)CCCC2)=O)CC2CC1CN(C(=O)CCC1CC1)C2 CC1CC(C(=O)NCCCCN2CCC2)N1C(=O)CC(C)C N1(C(C)=O)CCC(NC(c2c(NC(=O)CCn3ccc(C)n3)c[nH]n2)=O)CC1 C1(NC(CCC=C)=O)C2CC1N(C(c1ncccc1Br)=O)C2 C1(CNc2cc(OC)cc(C)n2)CN(S(C)(=O)=O)CC(F)(F)C1 Cc1cc(Cl)cc2cc(C(=O)NCCC(C)NC(C3(C4CC4)CC3)=O)[nH]c12 c1(CCC(N2CCCCC2c2nc(C3CC3)no2)=O)cnc2n1CCCCC2 Cc1nccnc1C(=O)NC1C=CC(C(N2CC(CS(C)=O)C2)=O)C1 N1(C(=O)OCC)C(C(=O)NC(C(=O)NC(CN(C)C)C(C)O)=O)CCCC1C C1(NC(Cc2cnc(C)s2)=O)CCN(C(=O)CC2CCCOCC2)CCC1(F)F c1(C(N2CCC(F)(CNC(C(CC(C)C)C)=O)C2)=O)ccc(N)c([N+](=O)[O-])c1 C1(CSC)CCN(C(=O)CNC(=O)Cn2cc(C(C3CC3)OC)nn2)C1 Cc1cccc2oc(CCNC(=O)N(C)CCN(C3CCCOC3)C)nc12 c1(OC)c(CC(=O)NCCNC(=O)C(C)(C)C2CCOC2)cccc1F c1(CC)cc(OC)c(OC)c(C(N)=O)c1.C12CCC(CC1)NC(=O)C2(F)F N1(C(C(c2nc(C)sc2)=O)=O)CCN(C(=O)CCNC(C2CCC(=O)N2)=O)CC1 C(C)(CSC1(C)CCCC1)(C(=O)NCc1ncc(Cl)cn1)NC(C)=O C1(NC(c2[nH]cc(C)c(=O)c2)=O)CCC2CN(C(C3CCCC3)=O)CCC2C1 C1(C#N)(Nc2nccc(OCCOC)n2)CCN(C(C2CCNC2=O)=O)C1 c1(CN2CC3CN(C(c4c(C)ncs4)=O)CC32)ccc(S(C)(=O)=O)cn1 c1(CC)c(C(N2CC(CCNC(C3CCCN3C=O)=O)(OC)C2)=O)cccc1F N1(C(Cn2ncc(CC)c2)=O)CCC(C)N(C(c2ccc(Cl)c(C)c2)=O)CC1 Nc1cc(F)ccc1C(=O)NCC1CCN(C(c2cc(F)cc(Cl)c2)=O)C1 Cc1nn2cc(C(=O)NCc3nnn(C)c3C(N3CCOC4CC34)=O)nc2s1 C12(C(N3C(C)(C)C(NC(=O)Cn4ccccc4=O)CC3)=O)CCN(CC1)S(=O)(=O)C2 C(=O)(C1=CC(C)(C)C1)N1C(C(N(C)CC2(OC)CCC2)=O)CC=CC1 C1(C(N)=O)(CNC(C2CC(=C)C2)=O)CN(C(=O)CC2CC2CC)C1 N1(C(Cc2cccc(C)c2F)=O)CC(NC(=O)CCC=CC(C)C)C2CCCC12 c1(OC)cccc2cc(C(N)=O)oc12.c12cccc(c1)CN1CCC(C1)O2 C1(C(N(C)CC2CC2)=O)CC2(CCC2)CN1C(c1ccc2c[nH]nc2c1)=O CC(C)CCCCCC(=O)N1CCC(C)(C)C(CNC(=O)CNC=O)C1 C1(CNC(c2ccccn2)=O)COCCN(C(=O)CC2(O)CCCCC2)C1 CC(C)(CNC(=O)C(Cc1cc[nH]n1)NC(C1CCCSC1)=O)C(F)(F)F Cc1cn2cc(C(=O)NCC3CC(C)N(C(=O)Cc4csc(C)c4)C3)ccc2n1 N1(C(C(N2C(C)CCC2C)C)=O)CC2(CCN(C(=O)C3=CSCCO3)C2)C1 CCCC(CC)C(=O)NC1CCC1NC(c1ccc(-n2ccnc2S)cc1)=O c1(C(N2CCC(N(C(c3cc(C)no3)=O)CCO)C2)=O)cccc(C(=O)N(C)C)c1 N1(C(C(CC)SC)=O)Cc2ccnn2CC(NC(=O)CCC(=O)Nc2nccs2)C1 N1(C(C(CC)SC)=O)CCN(C(C)CNC(=O)CC2C(C)C2(F)F)CC1 n1(CC(N2CCC3(C(NC(C4OCCC(C)C4)=O)C3)C2)=O)cnc2ccccc12 C1(CNC(=O)CNC(C2CCN(C(=O)COC3CCCC3)C2)=O)CCCCO1 C1(C2CCOCC2)(C(N(c2nc3ccccn3n2)C)=O)CCNC1 N1(C(CC(C)Oc2ccccc2)=O)CC2CCN(C(c3cnc(Cl)cc3Cl)=O)CC2C1 Cc1noc(C(F)(F)F)c1C(=O)NCC1CC(F)(CNC(=O)C(O)C2CC2)C1 C1(NC(CSS(C)(=O)=O)=O)CN(C(=O)CN2C(=O)CCC2=O)C2(CCCCC2)C1 c1(NC(C(C2N(C(c3cc(CC)no3)=O)CCC2)(C)C)=O)ccccc1CCO c1(C(=O)NC2(C)CCN(C(C3C(F)(C(=O)OC)C3)=O)C2)ccc(C(C)C)nc1O CS(=O)c1cccc(NC(c2nnnn2C2CCOC2)c2cnc[nH]2)c1 CN1CCC2CCN(C(c3cc(CNC(C4(CO)CCCC4)=O)no3)=O)C2C1 CC(C)CCC(=O)C(=O)N1CCC(NC(=O)CC(C)c2cnn(C)c2)C1(C)C Cc1c(C)c(C)c(C(N2CC(CC(C)NC(C3C(C)C3C)=O)C2)=O)c(C)c1C N1(C(CCCOCCC)=O)CC(C)CN(C(=O)C=CC=C(Cl)Cl)CC1C C1(NC(C2(C)CC(=C)C2)=O)CCC2(CC1)CN(C(=O)CC1CS(=O)(=O)C1)CCO2 N1(C(CCSCC(C)C)=O)CCC2(CC1)CC(NC(=O)CNC(=O)C(F)(F)F)C2 N1(C(C)C)N=C(C(=O)NCC2CCN(C(=O)C3=CCSC3)C(C)C2)CCC1=O C(=O)(C1CCCc2ccnn21)N1CCN(C(CP(C)(C)=O)=O)C(CCO)C1 C1(NC(c2cc(OC)n[nH]2)=O)CC2(C1)CC(CNC(c1ccc(C)nc1)=O)C2 N1(C(C(CCC=C)NC(=O)CC(C)C(F)F)=O)CCC(=O)N(C)CC1 C1(NC(C(CC)N(C)C)=O)CCC12CCN(C(c1csc(S(N)(=O)=O)c1)=O)CC2 C1(CC)(NC(C(C)(C)COC)c2nnnn2C(C)(C)C)CCCSC1 CC(C)CC(C)OC.c1(CC(=O)N(CCCN(C=O)C)C)csc(-c2ncccn2)n1 C1(CNC(C2(CCOC)CC2)=O)C2CN(C(=O)C(F)OC)CC12 N1(C(COCCCCC)=O)CCOC(CNC(=O)CCc2ncc(C)[nH]2)C1 Cc1cc(C(=O)N(CCCOCCNC(=O)C(F)CC2CCCC2)C)nc(O)c1 C=CCCCCS(C)(=O)=NC(=O)c1cc(C)on1 C12(NC(CNC(CC)=O)=O)CCC(CC1n1cc(CCC(OC)OC)nn1)C2 C(CCC(=O)NCc1nnnn1C)(C(C)C)NC(C(CSC)C)=O N1(C(CC(CC)C)=O)CC2(CCN(C(c3cnn4c3OCCC4)=O)CC2)CC1C Cc1cc(C(N2CCCCC2CCC(F)(F)F)=O)c(O)nc1C C(=O)(C1=CCC(F)(F)CC1)NC(C1CCCN1C(C1CC2C=CC1O2)=O)C Cc1ccc(I)cc1C(=O)NCC(=O)NC(C1CCC1)C C1(C(N(C2CC(NC(C3C(C(=O)OC)C3)=O)C2)C)=O)CCCOCC1 C(CC(C)C)(C(=O)N(CCC(=O)NCC1OCCCC1(C)C)CCO)OC N1(C(c2c(CC)non2)=O)CCC(N2CCN(C(=O)C(=O)NC3CC3)CC2)CC1 C1(C(=O)NCCN(C(C(C)SCC(F)(F)F)=O)CC(C)O)COC(=O)N1 C1(NC(COCCC)=O)CCSC12CN(C(=O)C(C)(C(F)F)c1ccccc1)C2 c1(C(=O)OC)cc(O)c(NC(C2CCN(C(C3CC3C)=O)CC2)=O)cc1OC c1(C(=O)NC2C3CN(C(c4nc(Br)c[nH]4)=O)CC23)ccn2cncc2c1 C(N=c1[nH]c2c(c(=NCCNC(=O)C3CC3)[nH]1)CCCCC2)c1cc(OC)ns1 N1(C(C(CC)(C)C#N)=O)CC(C)CN(C(c2csc(-c3ncc[nH]3)n2)=O)C(C)C1 N1(C(C2CCC=CCC2)=O)CC2C(C1)C(F)(F)C2(F)F c1(C(=O)NCC(CC)NC(C2(CC#C)CCC2)=O)c(CC)nn(C)c1CC C(=O)(C(C)C(C)O)NCC(C)=CC(=O)NCc1cc(C(C)C)on1 C1(NC(c2cccc(O)c2F)=O)CCCCN(C(C23CC(C2)C3)=O)C1 C(=O)(CCC1CCc2ccccc21)N(CC(C)NC(C1CC(C)(C)C1)=O)C c1(OC)ccccc1OCC(=O)NCC1(O)CCN(C(c2ccccc2F)=O)C1 CCC(CC(=O)N1CCC(CC(C)NC(c2ccc(N(C)C)cn2)=O)CC1)OC S(=O)(=O)(c1cccnc1NCC1CCCC1C)NCC1(OCC)CCC1 C#CC(C)(C)C(=O)NC1CCCC(CNC(c2ncsc2C(C)C)=O)C1 C1(NC(CC(=C)C)=O)CN(C(c2ccc(OC)c(CC)c2)=O)C(C)(COC)C1 N1(C(C(C(C)C)OC)=O)CC2CCCCC2(NC(=O)C(C)c2ccco2)C1 c1(-c2c(C)c(CO)ccc2)ncn2c1CN(C(=O)Cn1cccc1)CC2 Cc1ccc2cccc(NC(C3CCCN3Cc3ccc(C)n3C)=O)c2c1 C1(C(=O)N(C)Cc2ccccc2)(CC)CCN(C(C2CC2C2CCCC2)=O)CC1 Cc1cc(C(N2CC(NC(c3cccc(C4(C)CC4)c3)=O)C2)=O)c2c(c1)CCO2 c1(C(=O)NCCN(C(c2c(C)nn(C)c2Br)=O)C)ccnc2ccnn12 Cc1csc(=O)n1CC(=O)N(C)C(c1ccc(Br)cc1)C c1(CC2C(C(=O)NCC3(F)CN(C(c4cn(C)nn4)=O)C3)C2)c(Br)cnn1C C1(F)(CNC(CC(C)(C)OC)=O)CCN(C(=O)COc2cccnc2)CC1 N1(c2cccc(C(=O)NCCCc3ncn(C)c3)c2)C(=O)CCCC1=O c1(C(N2C(CNC(C(C(C)C)F)=O)CC2)=O)c(F)ccc2[nH]ccc12 CC1CN(C(C2(C)C=CCCC2)=O)CC1CCNC(=O)CN1CC(=O)NC1=O c1(C(C)=O)cccc(Cl)c1NC(=O)N(C)C(c1ccc(F)cc1)C c1(C(=O)NCC(C(=O)N2CCC(NC(C)=O)C2)OC)ccc2cc[nH]c2n1 c1(OC)ccc2c(c1)C(C(=O)N1CC=CC1CNC(=O)C=CC(C)(C)C)CCC2 C1(CC(=O)NCC2CC(NC(CN(CCC)C)=O)C2)CCC(C)CC1 C1(CNC(c2c(C)sc(C(F)(F)F)n2)=O)CC2(CO1)CN(C(c1cc[nH]c1)=O)C2 O=C(NN1CCCC1C(=O)NC(C(F)(F)F)c1ccco1)c1cc([N+](=O)[O-])n[nH]1 CC1(NC(C2CC(c3ccc(Cl)cc3)C2)=O)CCN(CCN2CCNC2=O)CC1 N1(CC(=O)NCC2CC2NC(C2(CC3CC3)CCC2)=O)CC2CCC1C2 c1(CCNC(CNC(c2cnc(CC)s2)=O)=O)ccc(O)cn1 c1(NC(CC2CCN(C(c3c(CC=C)cccc3)=O)C2)=O)ccc(Br)nc1I n1(CC)cnc2c(N(C)Cc3ccc[nH]3)[nH]c(=NCC(CO)C3CCOC3)nc12 c1(CC(=O)NCC2C(NC(C(Br)=C(C)C)=O)CC2)c(Cl)cnn1C Cc1noc(C(C)NC(c2cc(CNC(=O)C(C)n3ccnn3)no2)=O)n1 N1(C(c2oc(C)c(Br)c2)=O)CCN(C(=O)C2=NOCC2)C(CCO)C1 CCC(C)CCN=c1ccnc(N2CCc3ccc(Br)cc3C2)[nH]1 c1(OC)cc(OC)[nH]c(=NCC2CN(C(=O)CNC(c3ccccc3)=O)C2)n1 C1(N=[N+]=[N-])(C(=O)NCc2scc(C)n2)CCN(C(=O)CC2(C)OCCO2)C1 C(CCC(C)C(=O)N1CCC(n2cc(-c3ccnc(C(F)F)c3)nn2)CC1)OC C(=O)(CCC(C)(C)c1ccccc1)N1CC(COC)(CNC(=O)CC(=O)NC)C1 C1(CC(=O)N(CCOCCC(=O)NCc2c(C)ncs2)C)COCC(C)O1 C1(C2CC2)(C(=O)NCCC2C(C)C2)CN(C(=O)C(F)C2CCCC2)C1 C=CC1OCCC1C(=O)NCC(C)NC(=O)CCc1nc(CC)no1 C1(F)(C(=O)NC(CN(C(c2cncc(SCC)n2)=O)CC)C)CCCN(C)C1 c1(C(C)=O)ccc(C(F)(F)F)nc1NCC1CCCCN1C(=O)Cc1ccoc1 S(=O)(=O)(c1ncc(C(F)(F)F)cc1Cl)NC(c1ncco1)C C1(C)(CNC(c2ccc(OC)cc2)=O)CN(C(=O)CC2CCOC2)CCO1 C=CC1(C(=O)N(CC(=O)NC2CCOC2Cc2ccccc2)C2CC2)CCC1 C1(C(N2CCC(CCNC(c3cc(C(F)F)ccn3)=O)C2)=O)CCCC12CCC2 C12CC(C)(C1)C(=O)N2.S(=O)(=O)(C(C)C)N(CCCNC(C=CCCC)=O)CCO N1(c2ccnc(COC)n2)CCCC(C)(C)C1CNC(C1(C)CCNC1=O)=O N1(C(Cn2ncc(C)c2)=O)CCC(C)(C)C1C(=O)Nc1ccc(C)cc1CO c1(C(N2C(C)(CNC(CCC=C=C)=O)CCC2)=O)nc2nc(C)cc(C)n2n1 c1(C(=O)NC2CN(c3nc(SC)c(C)cn3)C(C)C2)n[nH]c2ccc(F)cc12 c1(C(N2C(CNC(C(c3ccccc3Cl)C)=O)C=CC2)=O)cc(F)c(Cl)cc1Cl c1(-c2cc(OC)ns2)nc(-c2cccs2)nn1-c1ncc(C)cn1 C1(CN(CCCC#C)C(=O)OC(C)(C)C)CC(C)N(C(=O)C(C)C)C1 c1(-n2cc(COC3CCCN(C(C(CC#C)C)=O)C3)nn2)cc(Cl)c(Cl)c(Cl)c1 Cc1csc(CNC(=O)C=CCNC(c2c[nH][nH]c2=N)=O)n1 C(C(=O)NCC1(C)CCCN1C(C1CC(C)(C(C)(C)C)C1)=O)(C(C)C)OC c1(NC(C2C(C(C)NC(CCC=CC)=O)C2)=O)cnc2c(c1)CCC2 C(=O)(CC1=NNC(=O)C1)NC12CC(CNC(c3cnc(CCCC)s3)=O)(OC1)C2 C1(CNC(=O)CSC)CN(C(C23CCC(CC)(CC2)OC3)=O)CCC12CCC2 c1(C(=O)NC2C(C)CCN(C(CCCC(=C)C)=O)C2)c(F)ccc(C)c1F N1(C(c2cc3[nH]ccc3s2)=O)CC2CCC(C1)N2C(=O)C(F)(F)c1cnccn1 C#CCC(C)(CNC(=O)C(CCOC)NC(=O)CSC1CC1)CO S(=O)(=O)(C(F)(F)F)NC(c1ccc(-c2ccnn2C2COC2)nc1)=O C(=O)(CCCC(=O)NC1CC(C(=O)NCc2ccc(OC)cc2)C1)NCCC C1(n2cc(CC(C)O)nn2)C=CCC(CNC(C)COC2CCC2)C1 c1(C(C(=O)NC(CNC(C23OCC(C)(C2)C3)=O)C2CC2)O)cc(F)c(F)cc1F N1(C(C(C2CCN(CC3CC3)C2)F)=O)CCC(CO)CC1.C1(C=O)SCCS1 c1(CC(=O)NCC23CCCC2OCC3)cc(O)nnc1O c1(CC)nncn1NC(=O)C(O)CCCNC(=O)CCCCC(C)=O N1(C(CCC2C(C)(C)C2)=O)CCOC2(CCN(C(c3cc(F)ccc3)=O)C2)C1 C1(NC(Cc2scc(C)c2)=O)CCC(F)(CNC(=O)CCc2ccc(Cl)cc2)C1 CCCC(C(=O)N(CCC(=O)NCCn1ccnc1)OC)OCC C1(NC(C(CCC)OCC)=O)COC2CN(C(c3cccc(OCC)c3)=O)CC12 c1(C(N2CCC(CC)(NC(=O)C(C)CF)CC2)=O)cnc2n1CCOC2 CCC(C(=O)N1CC(Cn2cc(Cn3cnc(C)c3C)nn2)C2(CCC2)C1)C(C)(F)F Cc1cc(C(N2CC(C(N3CC4C(C3)C4(C)C)=O)C(F)(F)C2)=O)ccc1F c1(C(N(C(C(=O)N(C(C=C)C2CC2)C)C)C)=O)cnn(C(C)C)n1 C(C(CC(F)(F)F)NC(=O)CCc1ccc(=N)[nH]c1)NC(COCCCCC)=O c1(CC)ccc(O)cc1C(=O)NCCC1CCN(C(c2csc(C)n2)=O)C(C)C1 N1(C(=O)Cc2cnc3ccnn3c2)CC2CN(C(=O)CSC(F)(F)F)CCC2C1 Cc1cc(Br)cc(C)c1CC(N1CC(C)(NC(c2coc3ccccc23)=O)C1)=O CC1(CNC(C2(C)CCCS2)=O)CCCN(C(c2cnc(N(C)C)s2)=O)C1 N1(C(C(C)C2CCOC2)=O)CCC2(CC1)CCN(C(=O)Cc1sccc1Cl)CC2 Cc1ncc(C=CC(=O)NCCC2CCC(NC(c3cc(O)cs3)=O)C2)s1 C12(C(=O)NC3(C#C)CCOC3)CCCC1N(C(c1cccc3cncn13)=O)CC2 C(=O)(C(F)CC(C)(C)C)N1CCCC(CC(=O)N(C(C)C)Cc2cccnc2)C1 N1(C(CC(C)(F)F)=O)CCC2(CC1)OCCC2NC(=O)CCn1ccnc1 c1(C(C)NC(C(C2CC=CCC2)NC(c2c(C)c[nH]c2)=O)=O)cccc(F)c1 CCCC(C)CC(=O)N(C1CCCCC1NC(c1cc(C#N)n(C)n1)=O)C C(C(C)(C)C#CC(=O)N1CC(CO)CC12CCC2)NC(c1ncc(OC)nc1)=O c1(CCC)nc(C(=O)NC2C=CC(CNC(c3sccc3C3CC3)=O)C2)co1 c1(C(=O)NC(c2ccncc2Br)C)csc(=NCc2ccc(N(C)C)nc2)[nH]1 c1(OCC)ccc(C(=O)N(C(C)(C)C)CC)cc1.C12CC(CN1C)OC2=O C1(NC(C(CSC)C)=O)COC2(C1)CN(C(C1CC3CC1C1CC31)=O)C2 Cc1noc(CCCC(=O)NCC(CNC(=O)Cc2ccn(C(F)F)n2)CO)n1 N1(C(C(C2CCC2)OC)=O)CC(C2(NC(C3CC34CCOCC4)=O)CC2)C1 C(C)(CCCCNC(c1nocc1Br)=O)NC(C(C)SC)=O c1(NC)nnc(-c2ccc(Cl)nc2)n1CC(C)C.c1(C(C)O)cccc(Cl)n1 C1(CNC(COCCCC)=O)CN(C(c2cnc3sccn23)=O)CC1(C)C C12(CNC(C3C(OCC)C3C)=O)CC(C1)C(NC(=O)CC1CCC1)CO2 C12(CC(=O)NC3(CF)CCN(C(c4cccc(N)c4)=O)C3)CCCCC1C2(F)F c1(OC(F)(F)F)cccc(OCC#C)c1.C1(C)CNC(=O)N1 c1(CC(=O)NCC2C(NC(c3cnc(CCC)s3)=O)C2)cc(F)c(F)cc1F c1(C(N2CCN(C(C(CCC)C#N)=O)CC2CC)=O)cc2c(C)c(C)ccc2[nH]1 CC1CC(C)(C(=O)NCC2(O)CN(C(c3c[nH]cc3C3CC3)=O)C2)CCO1 N1(CCNC(C2CCCC(NC(c3ccn(CCF)n3)=O)C2)=O)C(=O)CCC1=O C1(CNC(COCCC)=O)CCC(C)N(C(=O)Cn2ncc(O)nc2=O)C1 CC1(C)CC(NC(C2CCCC23OCCO3)=O)CCN(C(=O)COC(F)F)C1 c1(COC(COCCCCCC)=O)cc2c(cc1Cl)OCCO2 N1(C(c2c(CC)cccc2)=O)CCN(C(c2ncnn2CC)=O)CC1C(C)C c1(NC(C2CC2(C)C)C)nc(N2CCC(Cn3ccnc3CO)C2)nc2sccc12 C1(C2CC2)(CNC(C(CCC)OC)=O)CCN(C(=O)CCc2cnc(C)o2)C1 c1(C(=O)NC2C(NC(CCCCC=C)=O)COC2)cccc2c1NCC(C)C2 C12CCN(N3CC4(CO)CCS(=O)(=O)CC4(CO1)C3)CN(C)C=NN=C2 C(=O)(C1COc2ccc(F)cc21)N1CC(N(C)C(C2CC3(C2)CC3F)=O)C1 C(C)(CCC(=O)NC(CCN(C(=O)CCc1ccsc1Br)C)C(C)C)OC c1(NCCC(N2CC(NC(C34COCC3C4)=O)C2)=O)ccccc1[N+](=O)[O-] n1(CCOC)nnnc1C(C1CC1(C)C)NCCn1cncn1 CC(C(C)C(=O)N1CCC(N(C(=O)C=Cc2ccco2)C)CC1)S(C)(=O)=O c12cccc(c1)S2.C1(C(=O)NCCCC=C)CCC(NC(C2CC(=O)N2)=O)C1 C(=O)(CCC(CF)CF)NC(C)C(C)(C)C(=O)NC(CC1CC1)CO c1(CN(C)C(C2CCC(=O)NC2)=O)cnn2c1CN(C(=O)CCOC1CC1)CC2 C(=O)(CN=c1[nH]c2ccccc2s1)NCCN(C(C1C(C)C1)=O)C N1(C(C2C(Cl)(C(=O)OC)C2)=O)CC(C)(C)CC1CNC(=O)CCc1cnn(C)n1 c1(CNC(CCSCC)=O)ccnn1C.C1(C2CCCO2)C(=O)N1C c1(C(=O)NC2CC(N(C(C3(COCC)CC3)=O)C)C2)cc(Cl)ccc1C C1(C(=O)Nc2cccnc2)CCCN(CC(N2CCCCCC2)=O)C1 C1(C(N2CC(C(=O)NC3CC3)C2)=O)(NC(C(C)(C)C)=O)CC(C)(C)C1 c1(CC(=O)N(CC(CC)NC(=O)C(O)Cn2cncn2)C)cc(OC)nn1C C(=O)(C(C(C)(C)C)C1CCC1)NCc1c(C(N(C(C)C2CC2)C)=O)cnn1C C1(NC(Cc2c(C)ocn2)=O)(CO)CCN(C(=O)C(CO)NC(N)=O)C1 N1(C(CC2CC(OC)C2(C)C)=O)CC2(CCCN(C(=O)C(=O)NCC3CC3)C2)C1 c1(CC(=O)NC(c2cc[nH]c2)CNC(C(C)NC=O)=O)ccc(F)cc1F c1(CC(N2CCN(C(CC)=O)C3C2CC3)=O)ccc(S(=O)(=O)NC(C)C)cc1 C(CC(C(=O)N1CC2CC2(CC)C1)NC(C1CCCC1O)=O)=CC c1(C(N2C(CNC(c3c(COC)nn(C)c3)=O)CC2)=O)c(C)nn(C)c1C C1(C(=O)NCC(CC)(CC)Nc2ncc(Cl)c(O)n2)CC2CCC(C1)N2C Cc1ccc(Cl)c(C(N2CCC(F)(CNC(=O)CCc3scnc3C)C2)=O)c1 c1(C(=O)NC2CC(NC(c3cc(N)c(Cl)nc3)=O)C2)ccc2cc[nH]c2c1 C(C(C)(C)CNC(c1ccoc1COC)=O)NC(C1CC(N(C)CC)C1)=O N1(C(C(C)n2ccnc2)=O)CCCC2C(NC(=O)Cc3cnsc3)C(C)(C)C12 C(=O)(CCC(C)(C)[N+](=O)[O-])NCCC(C(=O)NCc1cccc(C)c1)C n1(CC)c(C)cc(C(N2CCCC2CCCNCc2conc2CC)=O)c1C CC1CC(NC(=O)CN2C(=O)CN(C)C2=O)CCN1c1nc(C#N)c(Cl)s1 Cn1c(CNC23C=CC(CC2)C3)nc2c1CCCC2 c1(C(N2C(CNC(C(C)=C(CC)C)=O)C(C)CCC2)=O)cc2sc(C)cc2s1 C1(NC(c2n[nH]c(C3CC3)n2)=O)CC2CCC(C1)N2C(=O)C1=COCCC1 C1(C(=O)O)C2CCCC1CN(C(c1cnc3c(c1)OCO3)=O)C2 C1(CC)CC(C(=O)NC(C)(C)CCNC(=O)CC2CCN(C(C)C)CC2)CC(=O)N1 NS(=O)(=O)c1ccc(CC(=O)NC2CN(C(C3CCCCC(=O)N3)=O)C2)cc1 N1(C(c2cnc(C)nc2C)=O)CC2CCC(C1)N2C(=O)CN(C1CCC1)C c1(OC)c(CNC(c2ncoc2C(C)(C)C)c2nnnn2C2CC2)cccc1C c1(C(N2CCC(NC(c3n(C)nnc3)=O)C23CC3)=O)cc2c(ccn2C)s1 C(=O)(CC1=CCCC1)NC1CC(C(=O)NCCc2n(C)cnc2)CC1O N1(C(C(CCSC)NC(N)=O)=O)CCCC2(CCN(C(=O)C(Cl)=CCl)CC2)C1 N1(C(CCOC)=O)CCN(C(C2CC3(CC3)CN2C)=O)C(C)C1 C1(CNC(CCSCCCC)=O)C2CCCC1N(C(c1cc(N)ccc1O)=O)C2 N1(C(CCC(=O)NCCC)=O)CC2CCCC2(NC(=O)C=Cc2ccoc2)C1 Cn1nc(C(=O)NC2C3CC2N(C(c2ccc(C(C)(C)C)[nH]2)=O)C3)c(Br)n1 C1(F)(C(=O)NC2CCC(OC)C2)CCCN(C(=O)CC2CCCC(=O)C2)C1 CC(C)CC(C)(C)C(=O)NCC1(CNC(C2CCOCC2)=O)CC12CCC2 C1(C(=O)NCc2ccsc2NC(=O)C(O)C2CCCC2)CCCNS1(=O)=O C(=O)(C(C)CCCC(C)C)NCC(CNC(C1(C)CCCC1(F)F)=O)OC C(=O)(CC(C)P(C)(C)=O)NCCN(C(=O)C(C)(O)CC)CCC c1(C(N2CC(CNC(CNC=O)=O)C3(C2)CC3)=O)cnc2c(c1)CCOC2 C1(C(=O)NCC2CC(C(C)C)C2)CN(C(=O)C(C)CO)CC1C C=CC1(C(=O)NCCC(C)O)CCN(C(=O)C(C2CCOCC2)C)C1 c1(C(N2CC(NC(C3N(CCC)C(=O)CC3)=O)C(O)C2)=O)cc(C)c(N)cn1 C(CCS(C)(=O)=O)C(C1CCCN1C(C1CCC1)=O)C.C1(C=O)CCCN1C(N)=O Cc1cc(-c2csc(C(=O)Nc3nnnn3C(c3ccccc3)C)n2)cc(C)c1 Cc1ccc(C(=O)NCC2CC(O)(CNC(=O)C3=NOC(C)C3)C2)c2c1CCC2 C1(C2CC2)(C(=O)NC2CCCC(CNC(c3cc(Cl)cnc3O)=O)C2)CC=CC1 N1(C(c2c(C)nc(CC(C)C)o2)=O)CCC(CO)(CNC(C2CC2F)=O)CC1 C1(C(N2C(CCC(N3CCN(CC#CC)CC3)=O)CCC2)=O)CCC(C)(O)CC1 N1(CC)CCCC(C(N2CCC(NC(C3CCCN3C(C)C)=O)CC2)=O)C1 c1(OC(C(=O)NC(C2CCN(C(=O)CSCC(N)=O)C2)C)C)ccc(F)cc1 N1(C(C(CC)C#N)=O)C2CCC1C(NC(=O)CCOC1CCCCC1)C2 c1(C(N(C(CCNC(c2ccc(CC)nc2O)=O)C)C)=O)cc(C)c(F)cc1F Cn1ncc(Cl)c1C(=O)NNC(=O)NC1CCN(C(=O)NC2CCCCO2)CC1 C(C(N=[N+]=[N-])C(=O)N1CC=C(C(=O)N(C)CC2COCCO2)C1)OCC c1(NC)cnncc1C(=O)NC1CC1CNC(c1ccn(C)c1)=O CC(CS(C)(=O)=O)C(=O)NCC1CN(C(=O)C=C2SCC(=O)N2C)CC1O Cc1nc(CNC(CSCC(=C2CN(C(=O)CC3CCCO3)C2)F)=O)cs1 N1(C(CCC2C(C)(C)C2)=O)CCCCC1C1(NC(=O)CC2CC3CCC2C3)CC1 C1(C(=O)NC(CN(C(=O)COC(C)(C)C)C)(CO)CO)CC(=O)NC1(C)C Cc1nc2cc(-c3nc(-c4cccc(=O)n4C)no3)cnc2[nH]1 CC(C)CCCCC(=O)N1CCC2(NC(c3cc4cccnn4n3)=O)CC2C1 C1(CC(=O)NCC(C(C)C)NC(=O)CCC2CCCC2)CS(=O)(=O)CCN1C C(=O)(CS(=O)(=O)NCC1CC1)NCC1CN(C(C(C)OCCCC)=O)C1 C1(COCC)CCN(C(=NCC2CCOCO2)Nc2ccc(OC)cc2)C1 Cc1nc(=N)[nH]cc1C(=O)NC1CN(C(=O)CC2CC2c2ccccc2)C1 CCC(C(=O)NCC1CC=CC1)N(C(=O)C1CC1)C(C)=O C1(C(=O)NC2(C)CC(NC(C(C)(C3CC3)OC)=O)C2)OCCCC1(C)C C1(C)(C(=O)NC(C2CCCC2)C#C)C=CCN1C(C1CCC(=O)N1)=O Cc1cnc(CN(C(=O)C(C2CC2)NC(C2CNC(=O)C2)=O)C)cn1 CS(=O)(=O)C1CN(C(c2cccc(O)n2)=O)CC1NC(C1CCCS1)=O C12(CC)CN(C1)C(=O)N2.c1(CC#N)c[nH]cc1-c1csc(C)n1 c1(C(=O)NCC2CCC(C(N3C(C(N(C)C)=O)C=CC3)=O)C2)cc(C#N)cs1 c1(CNC(=O)C(O)C2CN(C(=O)CC3CC4(CC4)CO3)C2)cc(O)ccc1F C(=O)(CC(O)c1cc(C)cs1)N(C1CCN(C(=O)CCc2cnn(C)c2)C1)CC N1(C(C=CSC)=O)CCN(C(c2cn(C)nc2C(F)F)=O)C(C2CC2)C1 N1(C(C=CC=CCC)=O)CCC2(CC1)CC2CNC(=O)C(C(C)(C)C)OCC C(=O)(C(C(C)NC(C1CCNC(=O)C1)=O)C(C)C)NCCCNC(C(C)C)=O Cc1cc(N2CCNC2=O)ccc1C1(N(C(C2(C#N)CCCO2)=O)C2CC2)CC1 c1(C(N(C2CCCC2)CCNC(CC2C(C)(C)CCO2)=O)=O)cc(N)ccc1F c1(CN2C(C(N3CC(C)(CO)C3)=O)C=CC2)ccc(O)c([N+](=O)[O-])c1 C1(OC)CN(C(=O)CSC(C)C)CC1NC(C1CCC(=O)NC1)=O N1(C(C2N(C(=O)OC)CCC2)=O)CC2CC1CC2NC(c1cnn(C)c1)=O C1(C(=O)NCC(C)(O)CO)CN(C(c2cc(Cn3cccn3)[nH]n2)=O)CCO1 CN1CCN(C(=O)CCCCN(C)C(C2(C#N)CC3CC3C2)=O)CC12CCC2 N1(C(CCCCOCCCC)=O)CCCC2CN(C(=O)C(=O)N(C)C)CC12 CC(C)C(CCC(=O)N1CC(CO)C1(C)C)NC(=O)CCC(C)(C)C C(CCCCCCC(F)(F)F)NCc1c(C)ccc(C)c1 N1(C(c2cc(OCC)n[nH]2)=O)CCC(NC(=O)CNC(C2CCOC2)=O)C(C)C1 C1(O)(C(C(=O)N(C(C)C)CCN(C)C(c2cc(CO)[nH]n2)=O)F)CCCC1 C1(CNC(=O)OC(C)(C)C)CCCN(CCc2cc(F)ccc2F)C1=O C1(C(N(CC(=O)N(CCCCO)C2CC2)CCC)=O)CC2(CC2)CO1 c1(C(CC)NC(C2(C(=O)OC)CC2C(F)(F)F)=O)cnn(C)c1 c1(C(N2CC(CC=C)(NC(C34CCC(CC3)CC4)=O)C2)=O)sccc1S(C)(=O)=O C=C=C(C)CC(=O)NCC1(CNC(C2CCN(CCCC)C2)=O)CC12CCC2 N1(C(CN(C)C2CC2)=O)CC(O)(CNC(c2cc(F)n[nH]2)=O)C1 N1(C(CCC#CC)=O)CCCC2(C1)CN(C(C1CCCN(C(=O)OC)C1)=O)C2 c1(OC)ccc(C(N2CCCC(N(C(=O)C(C)=C3CC3)C)CC2)=O)nc1Cl C1(NC(C(C)OCC=C)=O)CCN(C(c2csc(Br)c2C)=O)C(C)C1 N1(C(CCC(C)SC)=O)CCC2CCN(C(=O)C3CCc4c[nH]nc43)CC2C1 c1(C(=O)NC2C(NC(=O)C3=COCCC3)CC2)cc(F)c2ccccc2c1 C1(C(=O)NCC(C)(CO)NC(C2CCC(N(C)C)CC2)=O)CCC(F)(F)CC1 Cc1c(C(N2CC(C)(CCC(N3CC(F)(F)C3C3CC3)=O)C2)=O)ccn1C C1(c2cc(C)cc(C)c2)C2(CCC2)C12CCC2 C1(C(N2CC(O)(CN(C(=O)C(C3CCOCC3)F)C)C2)=O)CCC2(CC2)C1 C1(OC)CCCC(C(N2CCC2Cn2cc(-c3cnn(CCF)c3)nn2)=O)C1 N1(C(CC(C(C)C)O)=O)CCCCC12CC(NC(C1(F)CCOC1)=O)C2 c1(NC(C2C(NCc3nccc(C)c3)CCC2)=O)c(Br)cccc1[N+](=O)[O-] c1(C(=O)NC(C)C(CO)NC(=O)Cn2[nH]cnc2=N)c(Cl)cccc1Cl c1(CC)coc2c1CN(C(=O)C(F)C1CC(NC(C3(OC)CCC(C)C3)=O)C1)C2 C(CCCCC(=O)N1CCC(Cn2cc(COCC(C)O)nn2)C1)OCCOC C=CC1(NC2CCOC(c3ccnn3C)C2)CCCC1 C1(C)(CNC(CCC)=O)CCCN(C(c2c(C3CCC3)cnn2C)=O)C1 Cc1cc(C(N2CCC(NC(=O)CCc3cnc[nH]3)C(F)C2)=O)cc(F)c1 c1(C(=O)NCCC2(O)CN(C(C3CNC(=O)O3)=O)C2)[nH]nc2ncccc12 C1(NC(c2nn[nH]c2Cl)=O)CCN(C(=O)C2=CCCCC2)C12CCC2 C1(NC(c2cc(C)ncn2)=O)CN(C(C2CC=CCO2)=O)CC2(CCC2)C1 Cc1ccc(NC(C2CCCN(C(=O)CC34CCCC3C4)C2C)=O)c(F)c1 CC1(C)Cc2ccc(C(=O)NCCN3CCCN(C(=O)C(O)CF)CC3)cc2O1 C(=O)(C(C)(O)C(F)(F)F)N1CC(NC(C(C(C)C)N2CCN(C)CC2)=O)C1 O=C1C=CC(C(N2CC(NC(c3cc(C(F)(F)F)n[nH]3)=O)C(F)C2)=O)N=N1 C(=O)(C1=NNC(=O)C1C)NC1CC(CNC(C(CC(C)C)N(C)C)=O)C1 C(=O)(C1=Cc2cc(Cl)ccc2OC1)NCC1C(NC(C(CC)(C)C(N)=O)=O)C1 C(CCC(=O)NCC(C1CCCO1)O)N(C(C(C)n1ccnc1)=O)CC1CC1 C#CC1(C(=O)NCc2cn(C(C)C)nn2)CCN(C(=O)C(C)OCC)CC1 S(=O)(=O)(CCC(=O)NCC1CC1CNC(C1(C(F)F)CCCO1)=O)NC C1(NC(C(CC=C)NC(C2CC(CC3CC3)C2)=O)=O)COCC1C1CC1 N1(C(=O)CC2CCN(C(c3ccc(Br)cc3)=O)C2)CCC12CCCCC2 n1(C2(C)CC2)cc(C(N2CC(NC(C3CC=CCO3)=O)CC(O)C2)=O)ccc1=O C1(C(N2CC(CNC(CSC)=O)N(C)CC2)=O)CC12CCC1(CC1)CC2 C1(F)(C(=O)OC)CCN(C(=O)NCCC(O)c2cccs2)CC1 c1(C(CC)N(C)C)cn(C)nc1C(N1CCN(CCC(=O)OC)CC1)=O c1(SC)ncc(C(N2CCC(CN(C)C(C3CCCC(C)C3)=O)CC2)=O)n1C N1(C(CC2C(C)OCC2)=O)CCSCC1C(=O)NCC1(C)CCN(C)C1 C1(NC(CNC(CC)=O)=O)(COC)CCN(C(c2cnn(CC3CCC3)c2)=O)C1 N1(C(CCCC)C)CCC2(CC1)CC2(C)C(=O)NCC1OCCO1 C1(NC(c2n(CC=C)ccn2)=O)CC(C)N(C(=O)C(C)Cc2cnc[nH]2)C1 c1(C(N(CCCNC(C2C(C#C)C2)=O)C2CC2)=O)c(C)c(C)cc(C)c1C c1(C(=O)NCC2(O)CN(C(=O)COC3CC(F)(F)C3)C2)ccnc(C2CC2)n1 C=CC(C)(CC)C(=O)NCC1COCCN(C(c2cc(Br)c(C)s2)=O)C1 N1(C(c2cc(CC)on2)=O)CCN(CC(=O)NCCC2CCC(C)CC2)CC1 C1(OC)CN(C(=O)CCCCN(C)C)CCC1NC(=O)CC(C)n1cccc1 Cc1cccc(N(Cc2ccccn2)CC2CCC2)c1C C(=O)(CCC(C(=O)NC1(CCNC(=O)Cc2sc(S)nc2C)CC1)N(C)C)OC N1(C(CC(C)CC(F)(F)F)=O)C2CCCC1CN(C(C13CCC(C1)C3)=O)C2 C1(OC)CC2CC(C(=O)NC3(C)CCN(C(=O)COC4CCCC4)CC3)CC12 c1(C(N2CC(C)N(C(=O)CN(C3CCSC3)C)CC2)=O)cc[nH]c2nccc1-2 N1(C(C=C(CC)C)=O)CCCC(CC)(NC(c2cccc(C(=O)OC)c2)=O)C1 CC1CCN(C(=O)COCP(C)(C)=O)C1CNC(c1ccn(C)n1)=O N1(c2c(C)cnc(C)n2)CC23CCCC2(CN(C(=O)Cc2ccc(O)nc2)C3)C1 C(C1=NOC2CN(C(c3ccoc3Cl)=O)CC12)NC(c1cc(SC)c(F)cc1)=O C=C(C)C1OCCC1CNC(=O)COC(C)(C)CNC(c1oncc1C)=O c1(CC)cc(C(=O)NCC2CCC(C)N(C(=O)C=Cc3ncc[nH]3)C2)cc(O)n1 c1(C(N(C)CC2(C)C(NC(COC(CC)C)=O)CCC2)=O)nc(C)n(C)c1C c1(C(=O)NCC(CC)NC(C2C(Cl)(Cl)C23CC3)=O)cc(C)cc(C)n1 C(C(O)CN=c1nc(C)cc(C)[nH]1)NC(CN(CCC)C)=O C1(CNC(C(CC)NC(C)=O)=O)CC(F)CN1C(c1ncccc1C(C)(C)C)=O Cc1cc(C(=O)NCC(CNC(=O)C=Cc2ccnn2C)CO)nn1C(F)F C1(C(=O)NC2C(NC(CNC(=O)NC)=O)COC2)CCOCC12CCCC2 N1(C(COC(CN(C)CC)=O)=O)CCN(C(=O)NC2CCC(=O)N2C)CC1 c1(C(N2CCCC(CNc3ncccc3[N+](=O)[O-])CC2)=O)ccc2c(c1)CCC2 CC(C)C(O)C(=O)N(C)CC1CN(C(c2cc(Br)c[nH]2)=O)CC1O N1(C(C(CCC)F)=O)C(C(=O)NCc2nnc(C)s2)CCC12CC2 C=C=CCCC(=O)NCC1(NC(c2cccc(C(C)(C)C#N)c2)=O)CCCC1 C(=O)(CC(C)C(F)(F)F)NC1CC(OC)CN(C(c2cnc(N(C)C)nc2)=O)C1 c1(COC)ccc(C(C(=O)NC(C)C)N(C)CC2CC3CCC2C3)cc1 C(=O)(C1=CCS(=O)(=O)C1)N1CCC(O)(CNC(C2N(C(C)=O)CCCC2)=O)C1 C=CCC(CC)C(=O)NCCC(=O)NCc1nn[nH]n1 C(C(=O)NOCCc1cc(C2CC2)on1)N(C(C)=O)CCO c1(C(N2CC3(CN(C(C4C(CC)OCC4)=O)C3)C2)=O)ccc2[nH]c(=N)[nH]c2c1 C1(CNC(c2ccnc(OC)n2)=O)CN(C(=O)C(C)OC2CCCC2)CCC1C c1(NC(C(C)NC(C=CC(C)(C)SC)=O)=O)ccc(O)c(CO)c1 c1(C(N(C2CN(C(C(C(CC)C)C)=O)C2)C)=O)cc2c(C#N)cccc2[nH]1 N1(C(C)=O)CCC(NC(=O)C(c2cn(C)nc2C(F)F)C)CC1 CC1CCC(NC(=O)CC2CCC(=O)NC2)CN1C(=O)CCC(=O)c1cccs1 O=C(CCC(CF)CF)N1CC(C(N)=O)(CNC(c2cccc[n+]2[O-])=O)C1 CC1(C)CCN(C(C23CCC(C(F)F)(CC2)C3)=O)CC1CNC(=O)CCF c1(NCC2=CN(C(=O)OC(C)(C)C)CCC2)cc2c(Br)cccn2n1 c1(NC(C2CC3CC3N2CC)=O)c(NC(C2CCN(C)C2)=O)cccc1F CC1(O)CCN(C(=O)C(Cc2cn[nH]c2)NC(=O)CC2C=CCC2)CC1O c1(C(N2CCC(c3nnc(C(=O)OCC)s3)C2)=O)c(Cl)cc(F)cc1Br c1(C(N2C3CCC(CNC(C4C(C)(C)C4(C)C)=O)(C3)C2)=O)cc2c(o1)CCCC2 C(CC(C)C(=O)NC1CC2(C1)CC2C(N1CC(CF)C1)=O)=CC Cc1ccc(Br)c(NC(C2CC(NC(=O)Cc3cccc(F)c3)C2)=O)n1 C1(C(=O)NC2CC(NC(C(CC(C)C)O)=O)C2)CCc2c(ncn2C)C1 C1(NC(=O)NCc2c(OC(CC)C)ccc(Cl)c2)(CC)CCCCCCC1 c1(CCNC(c2cc(Cc3ccccn3)no2)=O)ccc(O)cc1 C(=O)(CCCC(=O)N1CCC(NC(=O)CCC2CCCO2)C(CC)C1)NCCC CC(C)(CCCF)C(=O)NC1CCCC1NC(C12CCCC1OCC2)=O C1(NC(C2CCOCC2)=O)CCC2CCN(C(c3cccnc3C3CC3)=O)C1C2 c1(C(=O)NCCCN(C(C(C2CCOC2)OCC)=O)CC)ncn(C)c1C C1(NCc2ccc(C(CC=C)C)cc2)CC2CCC1N2C(=O)OC(C)(C)C c12ccc(cc1)ON1CC3(C(C3)C(=O)NC2)C1.c1(CC2CC2F)ccc(F)cc1 C(C(C)(O)CNC(=O)CC1CCC(=O)N1)NC(CNC(C)=O)=O c1(C(=O)NC(C2CCCN(C(CCCC#C)=O)C2)C)ccc([N+](=O)[O-])cc1[N+](=O)[O-] CCC(C(=O)NC1CC(N(C)C(c2cc(-c3cccs3)[nH]n2)=O)C1)OC c1(CC(=O)NCCCNC(C2(CSC)CC2)=O)c(Br)cnn1C C1(C(N(C2CCOCC2)C(CC)C)=O)CCN(C(=O)C=Cc2cnccn2)CC1 Cc1c(Cl)c(C(=O)NC2CN(C(C3CC4COCC4C3)=O)C(C)(C)C2)nn1C c1(C(N(CCCNC(C(COC)O)=O)C2CC2)=O)ccc2cc(C)ccc2c1 c1(CCCC(=O)NCC2(CNC(C3CCNC3=O)=O)CC2)ccc(F)c(F)c1.CCl C1(C(=O)NC2CCC(NC(C=CC=CCC)=O)CC2)CCC(C)C(C)C1 C(CCF)(C(=O)NC(CCO)C1CC1)NC(C(C)OCCC(C)C)=O C1(C(=O)NC2(CC)CCOC2)(CNC(=O)Cc2csc(OC)n2)CCCCC1C N1(C(c2c(CC)nccc2)=O)CC(NC=O)CC(C)C1.c12ccc(cc1)SC2.CC C(=O)(C(C)(C)S(C)(=O)=O)NC1CCC(C)CN1C(c1cc2c[nH]cnc-2n1)=O CC1CCN(C(C2CC(F)C2)=O)CCN1C(=O)Cc1cnc(C2CC2)[nH]1 N1(C(CN(C(C2(C)CC2(F)F)=O)CC2CC2)=O)CC2CCCCCCC12 C1(NC(C=CSC)=O)CC(CO)N(C(=O)CC2CC3CC3C2)C1 CC1CN(C(=O)OC(C)(C)C)CC1CCOC(=O)C(C)(C)Cc1cnn[nH]1 CCC(O)CC(=O)N1CCCC1CC(=O)NCCCN(C)C N1(Cc2c(C)cccc2Br)CC2(CC(NC(=O)C(F)(F)F)CO2)C1 C1(Nc2cc(OC)ncn2)CCC(C)(C)CC1CNC(=O)CC1CCC(=O)N1 c1(C(=O)NCC2(F)CN(C(C(C)=CC)=O)C2)nc2ccccc2n1CCOC c1(CCC(=O)NCC(CNC(=O)C(C)N2CCC2)OC)cnc(N)[nH]1 C1(NC(c2ccc(C)nc2)=O)CC2CCC1CC2NC(=O)Cc1ncc(C)s1 c1(OC)cc(CNc2cccc(OC)c2OC)c(Cl)cn1 C(c1ccc2ncccc2c1)=CC(=O)N(C1CN(C(c2nccc(C)c2)=O)C1)C c1(NC)ncccc1C(=O)NCCN(C(=O)C(C)n1cccn1)CC(C)O Cc1ccc2c(C(N3CC(F)(F)CC3CNC(C3CC34CC4)=O)=O)ccnc2c1 O(NC(=O)C(C1CC1)NC(=O)CC1CC2(CCC2)C1)C(C)(C)CO N1(C(c2c(CC)nco2)=O)CC(C)CN(C(=O)CCNC(N)=O)CC1C c1(CC(=O)NCC(F)CNC(c2cc(F)ccc2Cl)=O)c[nH]c2ccccc12 N1(C(COCCC)=O)CC(C)(C)CCC1CNC(C1CC(C)=NO1)=O Cc1cc(C(=O)NCC2CN(C(C3(C(C)(F)F)CCC3)=O)CC23CC3)cc(C)n1 N1(C(c2cncc(C3CC3)c2)C(=O)NCc2ccccc2)CCC12CCCSC2 C#CC1CN(C(c2ccc(CO)s2)=O)CCN1C(=O)CC(CN(C)C)C(F)(F)F CC(C)C(C)CC(=O)N1CCC(C(C)(C)C(=O)NC2CCOCC2)C1 C1(NC(Cc2nc(CC)on2)=O)CCCN(C(=O)C=Cc2cnn(C)c2)C1 c1(C(N2CCCC(NC(c3c(C)cco3)=O)C2)=O)cc2c(cn1)OCCC2 C1(O)(CNC(CC(C)CF)=O)CCN(C(=O)OC(C)(C)C)CC1 c1(C(=O)NC2C(C)CN(C(C3(CCO)CC3)=O)CC2)cc([N+](=O)[O-])c(O)cc1N C(CC1=CCCCC1)N(C(=O)NC(C)C1CC1)C CC1(C)CCN(C(c2ccc(Cl)s2)=O)CC1C(=O)NCCn1cc(CO)nn1 N1(C(C2C(CNC(C3CC(O)(CC#C)C3)=O)C2)=O)CCN(CC(C)C)CC1 C1(C)(CNC(CCC)=O)CN(C(c2ccc(Cl)c(OC(F)(F)F)c2)=O)CC1C c1(C(=O)NC2CC(NC(c3cn(CC=C)nc3)=O)C2)sc2nccn2c1C CC12CN(C(=O)CCc3ccc(Cl)s3)CC1(C)CN(C(c1cc(Br)co1)=O)C2 c1(CNC2C(C(=O)Nc3nnc(C)o3)CCC2)c[nH]c2cccc(Cl)c12 c1(OC)ccc2c(=NCCn3cc(Br)nn3)[nH]c(=NCC(=O)N(C)C)[nH]c2c1 c1(OC)cccc(N2CCSCC2)c1C(=O)NC(c1ccc(F)cc1)C c1(-c2ncc(C(=O)NC(CNC(C(CC)NC(N)=O)=O)C)s2)ccc(C)c(C)c1 C1(C(=O)NCC2(CNC(c3c(C(=O)OC)csc3)=O)CC2)CCc2[nH]nc(O)c2C1 N1(C(c2ccc(C)s2)=O)CC(C(=O)NC2CC3CCC(C2)S3)C2(CC2)C1 c1(C2(C)NC(=O)N(CC(C3CC3)C3CC3)C2=O)cccc2ccccc12 N1(C(C(CCCC)=O)=O)CC(NC(=O)CC2C=CS(=O)(=O)C2)CC12CCC2 N1(C(c2cnc(C(C)O)s2)=O)C2CCC1CC(N(C)C(c1ccnc(O)c1)=O)C2 c1(C(=O)NCC2CC(CNC(c3scnc3C3CC3)=O)CO2)ccc(F)cc1 Cc1nn(C(C)C)cc1C(N1CCCC1CN(C)C(c1cnc(Cl)[nH]1)=O)=O c1(OC2CCN(C(N3CC(C(C)C)N(C)CC3)=O)C2)ccc2c(c1)CCC2.C(C)(C)O c1(OC)ccc(C(=O)NCC2(F)CCN(C(=O)CC(C)OC)CC2)c(OC)c1C C1(=CCNC(C(C=C)O)=O)CCN(C(C2CCCN(CC(C)C)C2)=O)CC1 S(=O)(=O)(c1cnn(C(C)(C)C)c1)N1C(c2cc(C)on2)CCCC1 C=CC1(CC(=O)NCC2CCCNC2=O)CN(C(C2(C#N)CC(=O)C2)=O)C1 O=C(C1Cc2ccccc21)NC1CCCCCN(C(=O)CCc2cc(Cl)no2)C1 C[Si](C)(C)C1CCCN(C(=O)CCC2CCC(N)CC2)C1 S(=O)(=O)(C1CCOc2ccc(Br)cc21)N1CCCC(CC)C1C(=O)O c1(C(=O)NCC=CCNC(c2c(CC)ncs2)=O)cccc(C(C)C)c1F N1(C(CN2CCC(C)CC2)=O)CC2COCCC2(NC(=O)CCCN=[N+]=[N-])C1 N1(C(C(C)CN(C)C)=O)CC(C)C(C)(C(=O)N(C)Cc2cn(C)nn2)C1 S(=O)(=O)(c1ccc(Cl)s1)NC(C(=O)NC1CC(CNC(CCC#C)=O)C1)C c1(CCC(=O)NCC2CC(NC(=O)CCSC(F)(F)F)C2)cccc(F)c1 N1(Cc2ccc(C(=O)OC)cc2F)CCC=C(C(=O)Nc2cc(O)ncn2)C1 C1(NC(=O)NC2CCCN(c3ccc(C(F)F)cn3)C2)CC2(CCOC2)C1 C123CCC(CC1)(CC2)C(=O)N3.c1(C2CC(N(c3nnnn3C)C)C2)ccccn1 c1(C(=O)NCC(CC)NC(=O)C(CO)C(C)(C)C)cc2cccc(O)c2[nH]1 c1(C(=O)NC(CC)C(=O)N2CCC(O)C2)c[nH]c2cnccc12 C(CCCCC(=O)NC(C1(CNC(c2ccc(O)c(C(N)=O)c2)=O)CC1)C)OC C(=O)(C1=CC2CCCCCC12)N(CCC)CCNC(=O)CCCCC(C)C c1(C(=O)NCCOCCNC(=O)CCc2cnn[nH]2)ccc(C(F)(F)F)nc1O c1(C(N2CC(C)C(C)(CNC(C3(C)CC4CC4C3)=O)C2)=O)nccc2occc12 N1(C(C(C(CC)C)=O)=O)CCC(C(=O)NCc2cc(C)ccn2)CC1(C)C CCC(CC(=O)N(CC(O)CN(c1cnc(C(=O)OC)cn1)C)C)C1CC1 N1(c2n(CC)c(C3CCC(C(F)(F)F)(OC)C3)nn2)CC2(CC(C)CC(=O)N2)C1 N1(C(c2cc(CSCCC)on2)=O)CCC2(NC(=O)C(=O)NCC)CC2C1 c1(C(N2CCCC(C(C)NC(C=NOC)=O)C2)=O)ncc(Br)cc1N C(=O)(CC1=CCOCC1)NCCOCCCN(C(=O)C(CC#N)c1ccccc1)C N1(C(c2c(Br)nc(C)s2)=O)CCN(C(=O)C(=O)N(C)C)CC1C1CC1.C c1(CC(C(=O)NCCCNC(c2cn(CC)nn2)=O)O)cccc(C)c1 c1(C(=O)NC2C(NC(C3CCN(C)C3)=O)COCC2)cn2ccnc2s1 CN1CCN(C(=O)C(CCOCCO)NC(=O)CCn2ccnc2)C(CCO)C1 c1(C(=O)NCC(C)NC(C(c2ccc(Br)s2)C)=O)cccn2cncc12 C=C(C)C(CC(=O)NCCC1CCCN1C(C1(C)CCC2CC2C1)=O)OCC N1(C(CC2(C)CC(NC(COC(C)=O)=O)C2)=O)CCC(F)(CF)C1 C12(C(=O)NCC(C(C)C)(C)F)CC(CO1)N(C(C1CC3CC1CC31CC1)=O)C2 C(=O)(C1CCCn2nccc21)N1CCN(C(CCCCCC=C)=O)CC1 C1(NC(Cc2c(C)non2)=O)CCCC12CN(C(=O)C(C)(C)c1cc[nH]n1)C2 CC1CN(c2ccncc2)CCN1C(=O)NC1CCC(=O)N1 c1(C(=O)NCC2N(C(C(C)NS(CC)(=O)=O)=O)CC(OC)C2)cc(Cl)ccc1N N1(C(CC2ON=C(CC)C2)=O)CCC2(CCCN(C(C3(Cl)CC3)=O)C2)C1 N1(CC(=O)NC(CCN(C(c2cnc(CC)[nH]2)=O)C)C)C(=O)CN(C)C1=O C(=O)(C1CCCc2c1ncn2C)N1CCN(C(c2c(COC)csc2)=O)CC1C Cc1coc(C)c1C=CC(=O)N(CC(C)O)CCNC(C1CCOC1C(F)(F)F)=O C1(NC(C(C)OCC#C)=O)(CO)CCN(C(=O)Cc2cn(C)nn2)C1 N1(C(C(C2CCCN(C(=O)CNC=O)C2)C)=O)CCCCC1c1nnc(S)n1C CCC(C(=O)NCC(C1CCCN1C(=O)CC(F)F)(C)C)C1CCC(=O)N1 C#Cc1ccc(CC(=O)NC2(CNC(=O)C(O)CN3CCOCC3)CCC2)cc1 N1(C(C(C)S(C)(=O)=O)=O)CCS(=O)(=O)C(CCNC(c2cc(O)nn2C)=O)C1 N1(C(C)C)C(=O)NC(c2ccc(N)c(Cl)c2)C2=C1CC1(CCCC1)NC2=O CC1(C)CCC(C(N2CCOC(C)(CNC(C3CCS3(=O)=O)=O)C2)=O)CC1 C1(CNC(C(CCC)OC)=O)CC2(CCOCC2)CN1C(C1CNC(=O)C1)=O C(=O)(C(C)CC(C)C(C)=O)N(CC(C)NC(c1c[nH]c2cccnc12)=O)CC C1(O)(NC(NC(CC)C)=S)CN(c2nc(C)ns2)C1 N1(C(C(CCC)(C)O)=O)CCc2nc(O)cc(C(=O)NC(C3CCC3)C)c2C1 N1(C(C2(CCC=C)CCCC2)=O)CCCC(CNC(=O)CN(C)CC)CC1 c1(C(=O)NC2COCCN(C(=O)C(O)CF)C2)ccc2oc(N(C)C)nc2c1 N1(C(C(c2ccc(CC)cc2)C)=O)CCN(C(C2CSC2)=O)CC1CC C1(C(=O)NCC2(CO)C(C)(C)C2)CN(C(c2cc[nH]c2)=O)CCO1 C(=O)(CC(F)(F)C(F)(F)F)NCCC1CN(C(C(COC)C)=O)CC1C C1(C(N2CCC(C)C(NC(c3cn[nH]c3)=O)C2)=O)CC2(CCOCC2)CO1 C=CCN=C(NCC1CCCN(C(=O)CCC)C1)NCC1CCSC1 C1(NC(c2cn(C)nc2O)=O)CCN(C(C2COC(=O)N2)=O)CC1F c1(C(N2CC3CN(C(c4cc(Cl)ncc4Cl)=O)CC3C2)=O)cc(F)c(F)c(F)c1 CCC1=NOC(C(=O)NCC2(CN(C(=O)CNC(=O)OC)C)CC2)C1 C1(C(=O)NCC2(CCOC)CC2)CCN(C(=O)C(O)CN(C)C)CC1C C(C(C)(CC(C)C)NC(c1ccsn1)=O)NC(COCCOCC#C)=O C(c1ccc(NC)cc1)=CC(=O)NC1C(CC)N(C(C2CC2C(N)=O)=O)CC1 C1(C(=O)NCc2cc(C(N(CC(C)OCC)C)=O)sc2)CCCN(C)C1 c1(CC)noc(C(N2CCC(NC(=O)C(=CC3CCCC3)C)C2C2CC2)=O)c1C c1(OC)ncc(Br)c(=NCC2CCCN(C(c3cc4cc(F)ccc4[nH]3)=O)C2)[nH]1 C(=O)(C(C)(C)N)N(CC#C)CC=C.C1(CC(=O)NCCSC)CCOC1 N1(C(C(CC)OC)=O)CC2(CCCCN(C(C3(c4cccnc4Cl)CC3)=O)C2)C1 c1(C(=O)NC2C(NC(C=CCOC)=O)CCCC2)c(Cl)cccc1Br CC(C)CC(CC(=O)N1CC(C)(C)C1C(C)C)NC(=O)C(C)n1ccnn1 C1(C(N2C(CC)CC(C)C2)=O)CC1C1CN(C(=O)C=CC2CCCN2C)C1 C(CCCCCC(C)(C)C)O.C1(C(=O)OC)CC2CN(C(=O)OC(C)=O)CC12 CCC(CC)(C(=O)OC(C)(C)C)C(=O)N(CC(C)N(C(=O)C=CS(C)=O)C)C N1(C(C2C(CNC(CC3(C)CCCO3)=O)CCCC2)=O)CCS(=O)(=O)CC1 S(=O)(=O)(c1ccc(F)cc1Cl)NCC1N(C(CCC#C)=O)CCC1 C1(CC(=O)NCC(C2CCC2)NC(Cc2c(C)con2)=O)CCCC(C)(C)O1 c12cccc(c1)C2.C1(C(=O)NCC2C(NC(C=COCC)=O)C2)CC(C)(C)CO1 C12(C(=O)NCC(C)CNC(c3ccccc3CO)=O)CCCC(C1)C(=O)N2 N1(C(CC(=O)OCC)=O)CC2CCC2(C(=O)Nc2cc(C(F)(F)F)c(F)cn2)C1 N1(CC)CCC(NC(C2CCOCC2NC(C2CC2C2CCC2)=O)=O)C(C)C1 Cc1cc(NCCN(C(C(=O)NC(C)(C)C)C2CC2Cl)C)cnc1O CCC(CC(=O)NC12CC1CN(C(=O)C=C=C(C)C)C2)C1CCC1 C(=O)(CCN(OC)C(=O)C1CN2CCN1CC2)NC(CCC(=O)OC)C CCC(C)C(C(=O)NCC(C)(C)C)N(C)C(c1scc(C)c1C)=O C1(CNC(=O)C=Cc2ccc([N+](=O)[O-])s2)C2CCCC1N(C(C1C3CCC13)=O)C2 Cc1ncc(C(=O)NC(C2CN(C(=O)CCc3ccc(O)c(F)c3)C2)C)c(C)n1 C(=O)(C(C)(C)C(F)(F)F)NC1C(CNC(C(C(C)C)(C)O)=O)C1 C(=O)(CC(C)CC(C)C)NCCC1(OC)CN(C(c2ccc3nncn3c2)=O)C1 C1(N(C(C=CC(=O)NCCN(C)C)=O)C)CCC(NC(=O)CCc2cnn[nH]2)C1 c1(NC(c2cccc(C(F)F)c2)=O)ccccc1C(N1CCCC1)=O N1(C(C2CN(S(CC)(=O)=O)C2)=O)CC(NC(=O)CCc2ccoc2)CCC(O)C1 C1(O)(C(=O)NCCC2CCN(C(C(c3cccc(Cl)c3)(C)C)=O)C2)CCSCC1 N1(C(c2cn[nH]c2)=O)CCC(C2CCN(C(C34CC(CN3C3CC3)C4)=O)C2)CC1 N1(C(C2CCC(CCC)C2)C(=O)NC2CCC2)CCCC(COC(C)(C)C)C1 C1(C(=O)N(CCC(=O)N(C)C)C)(CC)CCCN(C(C2CCC(=O)N(C)C2)=O)C1 Cc1ccnc2c(C(=O)NCC3CCC3NC(c3cnc(C4CC4)s3)=O)cnn12 CCS(=O)(=O)CCn1nc(-c2cncnc2)nc1C(CS(C)(=O)=O)c1ccccc1 C(=O)(C1CC=Cc2ccccc21)NC(C1C(OC)CCNCC1)=O Cc1c(F)cc(C(=O)NC2CCN(C(C3CCCO3)=O)CC2)cc1F C(CC1CC1)(C(=O)NCCc1ccon1)NC(C(c1cccs1)SC)=O Cn1c(=O)c(CNc2ccnc(-c3cc(F)ccc3N)c2)cc2ccccc12 CC(C)(CNC(C1CCC2(CC2)N1C(C1CC(=O)NC1(C)C)=O)=O)CC(F)F N1(C(c2c(CCC)n(C)nn2)=O)CCCN(C(C2CC(C3CC3)=NO2)=O)C(C)C1 c12cccc(c1F)O2.N12CC(C1)C(C)NC2=O.C(COC)OC c1(-c2onc(C(CC)COC)n2)ccc(Cl)cc1C N(C(=NCCC(C)C)NCc1cscc1C)Cc1cnc(OC)c(Cl)c1 C1(C(=O)Nc2c3cc(CNC)sc3ncn2)Cc2cccc(OC)c2O1 N1(C(CC(C)OC)=O)CCN(C(c2cccc(F)c2C)=O)C(C2CC2)C1 C1(C(=O)NC2CC(CNC(C(C3CCOCC3)OC)=O)C2)CCCC1(C)C N1(C(C2(SC)CCC2)=O)CCC(CO)(NC(=O)C(C)Sc2nncn2C)C1 C1(NC(CNS(C)(=O)=O)=O)CC1C1CCCN(C(c2nccnc2N)=O)C1 Cc1ccc(C(N2CC(OCCNC(=O)CCc3cc(C)sc3C)C2)=O)nc1 Cc1cc(CN)ccc1F.C(=O)(CC(F)(F)Cl)Nc1ncc(C=O)s1 CCC(CC)C(F)C(=O)N1CCC(C)CC1CNC(=O)CC(C)C1CC1 C1(NC(c2ccc(CCCC)cc2)=O)CCSC12CN(C(C1CC1F)=O)C2 C(=O)(C1=C(C)CCOC1)N1CC(C(=O)NCC2C(OC)CCC2)N(C)CC1 N1(C(C2CCCN(C(C)C)C2)=O)CCC(NC(=O)CCc2ncccn2)C(O)C1 Nc1ccc(NCCC(=O)N2CC(n3cnnn3)C2)cc1 c1(C(=O)NCC2(C)CCC(NC(CSCC=C)=O)C2)coc2cccc(O)c12 c1(C(=O)NC2(CNC(C(CCC)C)=O)CC2)cc(C(=O)OC)c2n1CCOC2 C1(C(=O)NCCCN(C(C2OCC(C)(C)C2)=O)C2CC2)CCn2ncnc2C1 C(=O)(C1Cc2ccc(Cl)cc21)N1CC(O)(CN(C(=O)CCP(C)(C)=O)C)C1 CCC(C(=O)N(C1CC(NC(=O)Cc2cccc(C)c2Cl)C1)C)C(F)(F)F C(Cn1cccn1)(C(=O)N(C)C)N(CC=CC(=O)NCC1(SC)CC1)CC n1(CC(N2CC3CC(C2)N(C(C24CCC(C2)C4)=O)C3)=O)ncc2ncccc12 c1(C(=O)NCC(c2ccc(F)cc2)OC(C)C)c(Br)ccc(F)c1F c1(C(N2CC(C(N)=O)(CNC(C(C)OCC)=O)C2)=O)c(C)cnc2ccccc12 CN1CCN(C(C2(CO)CCC2)=O)CC1CNC(c1cc(C(C)(C)C)nn1C)=O Cn1cccc1C=C(F)C(=O)NCCCNC(=O)C(c1cccc(Cl)c1)O C1(NC(c2ccn3c2CCC3)=O)CN(C(c2cncc(Br)c2)=O)C2(CCC2)C1 c1(CC)ccc(S(=O)(=O)N2C3CC2CN(C(c2cc(Cl)c(F)cc2Br)=O)C3)cc1 C12(C(N(CC(C)NC(C(=O)NC)=O)C)=O)CCC(C(F)(F)F)(CC1)C2 CCC(CC(=O)NCCCN1CCCC1=O)NC(C1CCCN(C)C1)=O CC1CN(C(=O)CCCn2c(O)nnc2O)CCC1NC(=O)CCC1CC1(C)C C(=O)(C1Cc2ccccc21)N1C(CNC(c2cc(C)n(CC3CC3)c2C)=O)CC1 c1(C2C(CC(=O)NCCCC3(CNC(C(C)N(C)C)=O)CC3)C2)nnnn1C C1(CCNC(CCSc2nc(C)[nH]n2)=O)CN(C(c2cnc(O)s2)=O)CCO1 C1(CNC(C2N(C)CC(O)C2)=O)CN(C(=O)Cc2csc(Cl)c2)CCC1(C)C c1c(CNCCC2CCCCCC2)sc2ccccc12 C1(NC(C=Cc2c(C)nsc2)=O)CC2(C1)CC(NC(C1CC3(C1)CC3(F)F)=O)C2 c1(OC)cccc(N2CCC(NCc3cc(-c4ccco4)[nH]n3)CC2)c1 c1(CC)ccc(F)c(CNC2(c3cccc(OC)c3)CCCOC2)c1 N1(C(C(CC)C)=O)CCC2CN(C(=O)CC3CCSC3)CC12 C1(OCC)CC2(C1)CC2C(=O)NC1CCCC(NC(=O)COc2cccnc2)C1 CC(CS(C)(=O)=O)C(=O)NCC1CCN(C(=O)C=CC(C)(C)C)CC1(F)F C(=O)(C(F)C(C)C(F)(F)F)NCC(C)N(C)C(C1COCC(C)(C)O1)=O Cc1onc(C2CC2)c1C(N1CC(NC(C2CC2(C)C(C)C)=O)C1)=O c1(CC)cc(C(N2CCN(CC(F)(F)F)C(C)C2)C(=O)NCCC#N)cc(F)c1 c1(CC(=O)NCC2C(NC(C=C3CCN(C)CC3)=O)CCC2)cccc(F)c1O c1(C(N2C(C)C(NC(c3ncc(F)cn3)=O)CC2)=O)ccc2nc(Br)nn2c1 N#CC1CN(C(c2ccc(O)nn2)=O)CCN1C(c1cc(C2CC2)on1)=O Cc1ccc2c(c1)CCC2C(=O)NC1CCCC1(C)CNC(c1nc(Cl)cs1)=O C1(C(C)NC(=O)Cc2cn[nH]c2)CCCN(C(c2ccc(F)cc2)=O)C1 CCCC(CCC)NC(C1(CC)CN(C(c2ccc(C3CC3)cc2)=O)C1)=O C1(CC)CN(C(c2onc(C)c2C)=O)CCC1NC(c1ccc(CO)c(F)c1)=O C(=O)(N=c1[nH][nH]c2cc(Cl)ncc12)C1NCCN(C(c2cncc(OC)c2)=O)C1 CCC(C)CCCC(=O)N(C1CCCN(C(c2cncc(Cl)c2)=O)C1)CC1CC1 C=Cc1cc(C(=O)NC2CC(O)CN(C(C3(CN(C)C)CC3)=O)C2)cc(F)c1 C(=O)(C1=C(C)N(C)c2nnnn2C1C)N1CC(NC(CCC=CC)=O)(CO)C1 CN1CCC(NC(=O)C(CC2CC2)NC(c2cccnn2)=O)C1=O C(=O)(CP(C)(C)=O)NCCC(C)NC(=O)CCc1nc(Cc2ccccc2)no1 C(=O)(C1CCCn2c(Br)cnc21)N(CCCN(C)C(C1CCNC1=O)=O)C CC(C)(O)CC(=O)NCC(CO)NC(c1cnc(C(F)(F)F)cn1)=O c1(C(=O)NC(C2CCN(C(C3N(C(CC)=O)CSC3)=O)C2)C)c(C#N)cnn1C C(=O)(CCC(N)C(=O)NC1CC2(C1)CN(C)C2)OCC N1(C(C(=O)NCC)=O)CC(NC(c2cncc(-n3ccnc3)n2)=O)CC12CCC2 c1(C(N2CC3CCN(C(CSCC)=O)C3C2)=O)cnc(O)c([N+](=O)[O-])c1 C1(C(N(C2CCN(C(c3cn(C4CCCCC4)nn3)=O)C2)CC)=O)C=CCCC1 C1(N(C(C2(C3N(C(C4CC(C#C)(O)C4)=O)CCC3)CC2)=O)C)CCC(C)(C)CC1 c1(-n2c(CC(C)CC)nc(C(C)OCC)n2)cc(Cl)c(Cl)cc1Cl N1(C(c2nc(C)sc2)=O)CCC2(CCN(C(C(N3CCC(N(C)C)CC3)C)=O)C2)C1 N#CC1CCCC1NC(C1CCC(CNC(c2cn(CCO)nn2)=O)C1)=O c1(C(=O)NCC(=O)NCc2ccc(C)nc2O)nccc2[nH]ccc12 N=c1[nH]cncc1C(=O)NCc1ccc(CNC(=O)C=CC2CCC2)cc1 C1(C(=O)NCC(C2CC2)NC(c2cn(CC(C)C)nc2)=O)CCC(=C(F)F)CC1 N1(C(CCC=C)=O)C2CCC1CC(NC(=O)COc1ccc(F)cc1)C2 c1(C(N2CCCC3(C2)CN(C(=O)C(O)C2CC2)C3)=O)ccc(C#CC2CC2)cc1 C1(C(=O)NOCCC(F)F)CC2(CCC2)CN1C(=O)CC1CCCC12CC2 CCC(C)C(=O)NCC1CC(NC(c2cnn(C(C)C)n2)=O)C1 Cc1cc(CCC(=O)OCC2CN(C(=O)NC(c3ncsc3C)C)C2)cc(C)n1 C1(O)(CCC(=O)O)CCN(C(c2cccc(F)c2)CF)CC1 c1(C(C(=O)NCC)N(C)CCN(C)C(=O)OC)cc(C)c(-c2ccccc2)s1 C(c1ccc(F)nc1)=CC(N1C(CCNC(Cc2nc(C)[nH]n2)=O)CCCC1)=O N1(C(CCc2c(C)noc2)=O)CC(CO)C2(CCN(c3ncc(F)cn3)CC2)C1 C1(C(N2CCC(N(C(=O)C3=CCSC3)CC)C2)=O)CCC(C)(C)CO1 N1(C(C2(COC)CC=CC2)=O)CCC2(CCCN2C(=O)CN(C2CCSC2)C)C1 N1(Cc2c(CC)cccc2)CCN(C(=O)Cc2c(Cl)cncc2Cl)CC1COC C1(NC(C2C(NC(C3C(c4ccc(C)cc4)C3)=O)CCO2)=O)CCCN(O)C1=O CCC(C)(C(=O)N(C)CC1CCN(C(c2cc(-c3cccs3)on2)=O)C1)OC C1(NC(C2(OCC)CCCC2)=O)CC1C1CCCN(C(c2c(C)noc2N)=O)C1 C(=O)(C1CCCc2nc[nH]c21)N1CCC(C)(CNC(=O)CNC(=O)C2CC2)C1 Cc1cc(F)cnc1C(=O)NCC(C1CCN(C(=O)CC(C)(C)C2CC2)CC1)F C(CN=c1ccc(S(=O)(=O)N2CC(C)OC3(CCC3)C2)c[nH]1)OCCC=C Cc1cc(CCNCC(C)COC(C)C)ccc1[N+](=O)[O-] C(=O)(CC(=O)NCC#N)N1CC(N(C(C(C)NC(N)=O)=O)C)C1 c1(C2CCN(C(C3(C#N)CC=CCC3)=O)CC2)nc2c(Cl)cccc2[nH]1 N1(C(CC=CC=C)=O)CCN(C2CN(C(=O)CCOCC3CCCO3)C2)CC1 C1(c2n(C)ncc2)CN(C(=O)OC(C)(C)C)CC1C(=O)OC(c1nn(C)cc1Cl)C1CC1 c1(C(=O)NC(C2OCCN(C(C=CCOC)=O)C2)C)c(C)nn(CC(C)C)c1Cl c1(OC)ccc(C)cc1.c1(C(=O)OC)n[nH]cc1-c1noc(C(C)C)n1 c1(C(N2CCN(C(c3cc[nH]c3)=O)C(CO)C2)=O)cnn2c(Br)cccc12 c1(C(N(C)CC2CCN(C(=O)C3=CSCS3)C2)=O)c[nH]c2ncccc12 c1(CN(C)C)cn(CC2CCN(C(=O)Cn3nnc(-c4cccs4)n3)C2)nn1 N1(C(C2(C)CCC(C)C2)=O)CC2CCC1CN2C(=O)CCc1ccncn1 c1(C(c2ccncn2)=O)cc2c(nc1O)CCC(C(=O)N(c1ccccc1)CCO)C2 c1(CC)nccnc1C(=O)N(C1CCC(NC(=O)COC)C1)C C=CCC(CC)C(=O)N1CCN(C(=O)CCc2ncc(C)[nH]2)CC1CC c1(OC)ccc(Cl)cc1C(C)NC(C1CC(O)CN1C(=O)C1CC1)=O C(=O)(C(C)CC(F)(F)F)NC1(CC=C)CN(C(=O)CCc2ccccc2)C1 Cc1nn(C)cc1CC(N1CSCC1C(=O)N(C)CC1CCCS1)=O Cc1c(C(N2CCCC(O)(CNC(=O)C(O)CC(F)F)C2)=O)sc2cncn12 C=C1CC(C(=O)Nc2csc(Cl)c2)(CNC(c2ccsn2)=O)C1 C1(C(=O)NCCSCCOC)CN(C(C2(n3cnnn3)CC2)=O)CC1(F)F N1(C(c2cc3c(s2)CCC3)=O)CCN(C(c2sccc2F)=O)C2CCCC12 CC1Cn2nc(C(=O)NCC3CCC3NC(C3CCS(=O)CC3)=O)cc2C(=O)N1 N1(C(=O)CN2CCCC2)CCN(C(c2cc(-c3ccccc3)[nH]n2)=O)CC(O)C1 C1(OC)(OC)CCC1C(=O)NCC(C)CNC(=O)C(C)Cc1cccnc1 Cc1cc(C(=O)NCC(C)(C(C)C)NC(=O)C=C2CCC(C)C2)ncn1 C(=O)(CC(O)CC(C)C)N(CCCC(=O)NC(CC)CC(C)CO)C C(=O)(C(O)C1CN(C(=O)C(=O)N(C)C)C1)N1C(C)C1.C(C(F)F)SC N1(C(C2C(OC(C)=O)C2)=O)CCN(C(c2occ(C)c2C)=O)CC12CCC2 C(=O)(CC(O)CC(C)C)NC(C1CC=CCC1)C(=O)NCC1(SC)CCC1 C(=O)(C(O)C1=CCCCC1)NCC1(O)CCCN(C(Cc2ccc(C)o2)=O)CC1 N1(C(=O)CC2NC(=O)NC2=O)CCC(F)(C(N2CCC(c3ccccc3)C2)=O)C1 O=C1CC(=O)N(CCNC2(c3nnnn3C)CC3COCC3C2)C(=O)N1 c1(SC(CCO)Cc2cccc(F)c2)nc2cc(Br)c(F)cc2s1 c1(C(=O)NCC2CCN2C(C2CC2C(F)(F)F)=O)ccn(C2CCC2)n1 c1(C(=O)NCc2cn(CC(=O)NC(c3ccnn3C)C)nn2)cn(C)c(=O)cn1 CC(C)C(C(=O)N1CCN(CC2CN(C(C3OCCO3)=O)C2)CC1)N(C)C c1(C(=O)NC2CCCC(NC(=O)C=Cc3cncs3)C2)cccc2c1OCCN2 c1(C(=O)NC2CN(C(CCC(C)N=O)=O)CC2C)cn2ccc(F)cc2n1 C1(NC(C(C(=O)OCC)CC)=O)CCC2(CC1)CC(NC(=O)CC1CCC1)C2 C1(NC(C2(CC)CCNC2=O)=O)CCCCN(C(=O)CC2(COC)CC2)C1 C1(NC(C(C)N(C(=O)C(c2ccn(C)n2)C)C2CC2)=O)CC1C1CCC1 C1(C(=O)NC(c2ccon2)(C)C)COCCN(C(c2ccc(F)cc2)=O)C1 N(C1c2ccccc2CC1NC(=O)CCCCC(F)(F)F)C(C(C)NC(C)=O)=O C1(OCC(=O)N(C2CC2)Cc2nc[nH]n2)CCN(C(C2CC23CCC3)=O)C1 c1(SC)ccc(CNc2c(C(=O)NCc3nc[nH]n3)cc(C(F)(F)F)cn2)c(I)c1 C1(C(N(CC(CC)NC(=O)CNc2ccccn2)C)=O)CC2(C1)CC21CC1 c1(N(C(c2sc(Br)nc2C)C(=O)NC(CC)(C)C)C)ccccc1SC N1(C(C(CCCOC)C)=O)CCC2CCCC12C(=O)N(C1CN(C(C)C)C1)C C1(NC(CSC)=O)CC(CNC(C2(c3cc(O)ccn3)CC2)=O)C12CCC2 c1(C(=O)NCC(C)N(C)C(C2(C)CCNC(=O)C2)=O)cc2ccccc2c(O)n1 CCC(CC(=O)N(CC(C)C)CCOC)NC(C1CC(C)(O)C1)=O c1(OC)c(F)cc(Br)c(C(=O)NCc2cccc3nn[nH]c23)c1F C(=O)(C1=C(C#N)CCC1)NC(C)CNC(c1occ2c1CCC2)=O N1(C(C2CC(C(F)(F)F)(OC)C2)=O)CCN(C(=O)Cc2cocn2)C(CO)C1 OC1CN(N2CCN(C3CCCOC3)CC2)C2(CCCC2)C1 CCCC(CCCO)C(=O)NC1(CNC(c2cnn(C(C)(C)C)c2N)=O)CCC1 N1(C(c2ccc(OC)c(C3CC3)c2)C(=O)NC)CCN2CC(C)CC2C1 CC1CN(C(C2(NC(N)=O)CC2)=O)CCC1N(C(=O)CC1CC(CF)C1)C C1(C(=O)NC(c2nc(=O)o[nH]2)C)OCCC1CNC(c1cc(C2CC2)[nH]n1)=O c1(C(=O)NCC(CCNC(CCCOC(C)(C)C)=O)(C)C)cnc2ccoc2c1 C(=O)(C(C)(F)C(=O)NCC1CC(C(=O)NCc2cnc(C3CC3)[nH]2)C1)OC c1(C(C(=O)NCC)OC(C)(C)CNC(=O)OC)cncn1C.C1(=O)CN1C C1(C(N2CCC(C#N)C2)=O)C2C3CC4C1C2C34C(=O)Nc1ccnc(C2CC2)n1 C(=O)(C1=CC(O)CCC1)NCC(CCOC)NC(c1ncccc1F)=O N1(C(c2c(C(C)C)n[nH]c2)C(=O)NCc2ccco2)CC2CCC(C1)C2(F)F CC(C)CC(C)(CNC(=O)C(O)c1ccsc1)NC(=O)CC(=O)NCC(F)(F)F N1(C(c2ccc(CCCCC)o2)=O)CC(NC(=O)C(C)OC)C2(CCC2)C1 O(NC(=O)CCC(C)(C)NC(=O)CCCCCCC)CCN=CC=CC N1(C(C(C)OCC2CC2)=O)C2CCC1CC(n1cc(CCCO)nn1)C2 n1(CC)ncc(Br)c1C(=O)NCCCCC(C)NC(=O)CCc1nc(C)no1 N1(C(C(C)NC(N)=O)=O)CCC(NC(=O)Cc2nc(C(C)C)cs2)C1C C1(OC)CC(NC(=O)CCc2cncn2C)CN(C(c2cncc(Cl)c2)=O)C1 CCCC(C)CC(=O)NC(c1ccccc1)C(=O)NCc1ccc(OC)c(F)c1 C1(C(=O)NCC2(NC(CCSCCCC)=O)CCOC2)CCC(C)(C)C1 C12(CNC(COC(CC)C)=O)CC(CN1C(=O)CCCc1nc(C)no1)C2 Cc1c(C(=O)NCC2CNCC(C)(C)C2)sc2ncccc12 c1(C(=O)NCC(C)NC(C(CC)OC2CCCC2)=O)cc2c(=O)[nH]ccn2n1 Cc1ccc(C(N)=O)cc1C(=O)N(CC(O)CNC(C1CCCC1(F)F)=O)C C1(NC(CCNC(C)=O)=O)CN(C(c2cccc(O)n2)=O)CC1C(F)(F)F N1(CC)CCCCC1CNC(=O)CC(C)(C)NC(c1cnc(C)[nH]1)=O CCCC(O)C(=O)N1CCC(OCCNC(C2CCN(C(=O)CCC)CC2)=O)C1 N1(C(Cc2cc(C)on2)=O)CC(CNC(c2ccc(C(C)C)cn2)=O)CCC1C c1(N2CCC(C)C2)nc(N2CCN(c3ccccc3)C(C)C2)c2ccsc2n1 C(C(C)C(=O)N1CC(CC(C2CCCCC2)C)C1)OC.c12coc(c1)CNC2=O C1(=CC(=O)NCC(C(C)C)(C)NC(c2cc(C#N)cn2C)=O)CN2CCC1CC2 Cc1cnc2n1CC(C(c1ccccc1)NCC1=CC(=O)OC1)CC2 c1(CCNC(C2N(C(c3nccc(OC)c3)=O)CC(O)C2)=O)ccc(F)cc1F Cn1ccc2cccc(CN3CCC(O)(C(=O)Nc4ccsc4C(N)=O)C3)c12 CC(CC(C)NC(=O)C(=O)C1CCCC1)NC(c1sccc1Br)=O C(c1ccncc1)=CC(=O)N(CCCN(C(C(C)=CC1CC1)=O)C)C c1(C(=O)OC)[nH]c(C)cc1NC(=O)N(C)Cc1ccc(Cl)cc1.C12CN(C1)C2=O C(CCOC)N.C(=O)(COCC(=O)N(CC#C)CC=C)NCC C1(C(=O)NCC2(CC)CC2)CCCN(C(=O)C(c2ccc(C)o2)C)C1C N1(C(=O)C=C2CCCC2)CC2CCCC(C1)N2C(c1ncc(Cl)c(O)n1)=O C1(OC(C(F)=C(C)C)=O)CCN(OC)CC1 CCC1=NOC(CC(=O)NCCNC(=O)C(O)c2ccsc2)C1 c1(OC)noc(C(N2CCCC2CCCNC(=O)CNC(N)=O)=O)c1Br c1(OC)cc(C(=O)NCCC(C)N(C)C(C2(CC(C)C)CC2)=O)n(C)n1 C(CO)(C(C)NC(C1CCCCS1)=O)NC(CN(CCC)C)=O c1(SC)ccc(C(c2nnnn2C2CCCCC2)NCc2cc(I)nn2C)nc1 N1(C(c2cnc(CC(C)C)[nH]2)=O)CCC2(CCCC2NC(c2ccccn2)=O)C1 C=C(Cl)CC(C(=O)N1CCC2(CCO2)C1)NC(C1CCC(=O)N(C)C1)=O C1(OC)CCC12CC(C(=O)NC1(CO)CN(C(=O)CCC3(C)CC3)C1)C2 c1(N(C)C)ccc(NC(=O)C(F)CC2CCOC2)cn1.C12CC(C1)C(=O)N2 c1(C(N(CCNC(c2c(Cl)cnc(OC)c2Cl)=O)C)=O)cncc2c1CCCC2 N1(C(C(CCC)CCC)=O)CC2COCC(C1)C2NC(c1cc(Cl)cn1C)=O C=CCCC(C(=O)NC1CCOC(C)C1)NC(c1cccc(C)c1C)=O C12CCc3ccccc3N(CC(=O)N1CC1CC1)C2=O.C(CCN)SC CON(CCCO)C(=O)C(C)(CO)NC(c1ccc(C(C)C)o1)=O Cc1cccc2nc[nH]c(=NCC3CN(C(c4cc(C#N)c[nH]4)=O)CCC3C)c12 C(=O)(C(CC(C)(C)C)NC(C1CC1CC)=O)NCCCCCCC n1(CC(=O)NCC=CCNC(C(C)OCC#C)=O)ncc(Cl)c1C N1(C(C2(OC)CCCCC2)=O)CCCC(NC(c2cc(SC)oc2C)=O)CCC1 c1(C(=O)NC2CC(NC(c3c(CC)oc(C)c3)=O)C2)cnc(C2CC2)[nH]c1=N c1(C(=O)NCC(CC)O)n[nH]cc1NC(=O)C(O)C1CCC1 C12(CCCC1)C(=O)N2.C1(CC)CCN(C(=O)CCC2CC(N(C)C)C2)C1 C1(O)(C(=O)NCC(C)NC(COCCCCC)=O)CCc2ccccc2C1 C(N=c1nc(N2CCN(CC3CC3)CC(C)C2)cc(C)[nH]1)c1cc(C)nn1C c1(C(=O)NC2CC(N(C(c3ccc(CC)s3)=O)C)C2)cc2cnccc2[nH]1 C1(CNC(C2(COC)C=CCC2)=O)CN(C(=O)C2=NNC(=O)C2)CCC1C C1(NC(C(=O)NC(C)C)=O)CCCC12CN(C(c1occc1C(C)C)=O)C2 C=CC(C)CC(=O)N1CCC(OCC(=O)NCCc2n[nH]c(C)n2)C1 O=C1CS(=O)(=O)CC(C(=O)NCC2CCC(CNC(C3CC3F)=O)CC2)N1 c1(CNC(C2(NC(CSCCCC)=O)CC(O)C2)=O)cc(O)ccc1C c1(CC(C(=O)OCC)F)ccc(NCCC(C2CCCCC2)O)c(F)c1 C(=O)(C1CC(=O)c2ccccc21)NCC#CCNC(c1cc(Cl)nnc1O)=O C(=O)(C(C(=O)OCC)C(C)C)N1C(COC)C2CCC1C2 C12(C(c3cn(C4CCC(C(=O)N(C)C)C4)nn3)C)CC3CC(CC(C3)C1)C2 c1(C(C(=O)NCC(C)CNC(=O)C(C)(F)F)C)cccc(F)c1 C(C(=O)N1CC(NC(c2ccc(C#C)nc2)=O)C(O)C1)(C(C)(C)C)NC(C)=O C=CCC(C)(C)C(=O)N1CCC(C(F)(F)F)C(CNC(=O)C#CC2(C)CC2)C1 c1(C(N2C(CC(=O)NCCc3cccnc3)COCC2)=O)c(F)cc(Br)cc1F c1(NC(C2(CC)CCN(C(C3C(C)(C)C3(C)C)=O)CC2)=O)cnn2c1CCCC2 c1(C(C)(C)F)cc(C(N2CC(NC(=O)CC3CC4CC4C3)C2)=O)ccc1F c1(C(=O)NC2CC2CNC(C2CN(C3COC3)C2)=O)c(F)cc(Cl)cc1Cl C1(C(=O)NCCCNC(=O)CC(O)c2ccccc2)CC(F)C(=O)N1 C1(N(C(C(CO)OC)=O)C)CC2CCC(C1)N2C(=O)CSc1cc(C)ccc1C c1(OC(C)C)cc(CNC2(C)CCCN2C(=O)C(F)=CC2CC2)ccn1 C1(C(=O)NCC2(C=C)CCC2)CSCCN1C(=O)CC(CC)C1CC1 CC1(CNC(C2=NOCC2)c2nnnn2-c2ccc(F)cc2)CC1(Cl)Cl C1(=O)C#CC2(CCCC2)N1.c1(C(=O)OC)cnn2c1N(C)CC2 C1(n2c(C3N(CC)CCCC3)nc(CCC(C)C)n2)CCCS(=O)(=O)C1 C1(CC)CCCCN1C(c1conc1CNC(=O)CC1CSCCO1)=O CC1(C(=O)OCc2ccccc2OC(F)(F)F)CCCCC1(F)F C(=O)(C1CCc2nnc(C)n21)N(CCCNC(c1cc(C)c(N)c(C)c1)=O)C N1(C(CN(CCC)C)=O)C(C(=O)NCc2n[nH]c(C)n2)CC2CC12 C1(NC(c2cc3ccccc3o2)=O)C2CC(O)C1N(C(=O)Cc1cnns1)C2 N1(C(C(=O)NCCC(=O)OCC)C2COC2)Cc2nc(Br)sc2C1 c1(CNC(=O)NCC2(OCC)CCCC2)ccccc1C.c1(C(=O)N)ccoc1C C(=O)(C1Cc2c(Cl)cccc21)NCC(=O)Nc1c(C)nn(C)c1-n1ccnc1C N1(C(C(NC2CCc3ccccc32)CCSC)=O)CCc2c(CO)nn(C)c2C1 C(C)(CC(C)NC(c1coc(C2CCC2)n1)=O)NC(C(C)C)=O c1(C2C(=O)N2)ccc(C(F)(F)F)cc1.C(C)(C(=O)N(C)C)S.C(C)(CNC)OCC C(=O)(N=c1ccn(COc2ccc(N3C(=O)CCC3=O)cc2)[nH]1)N(C)C C(=O)(CC(F)(F)C(F)F)N1CC(C)CC(CNC(Cc2cc(C)cc(C)c2)=O)C1 N1(C(C(CCCC)=O)=O)CCC2(CC1)CN(C(c1n[nH]cc1C)=O)CC2CO C=C(Br)CC(C)(C)C(=O)N(CCCNC(C1CCN(C(=O)NC)C1)=O)C c1(OCC)ccccc1NC(C1CCN1C(C1CC(CC)C1)=O)=O C(C(CC(=O)N(C(C)COC)C)C1CCC1)NC(C1C(OCC#C)C1)=O C1(NC(C(CCC)NC(c2ccc(CO)cc2)=O)=O)COCC(C)(C)C1 Cc1nn(C)c(N)c1C(=O)NC1CCC(NC(C2CC2c2ccccc2)=O)C1 CN(C(=NCC1CC1)NC1CCOC(C)C1)Cc1cc(F)ccc1N1CCCC1.N(C)C Cc1ncnc(C(N2CCC23CN(C(=O)CC2CCCC2C)C3)=O)c1C c1(C(=O)NC2CCN(C(CCOCCOCC)=O)CC2C)cccn2cnnc12 N1(C(c2c(CC)cns2)=O)CCN(C(=O)CCC2(C)CC2)CC1COC c1(OC)cc(NC(=O)CC2COCCN2C(=O)C(C)c2cccs2)ccc1C#N N1(C(CCSCCC)=O)CC(C2CN(C(=O)CCc3nc(CC)no3)C2)C1 c1(C(N(CCC(C)NC(=O)CCCCc2cnn[nH]2)C)=O)ccccc1CO c1(CNC(CC(CNC(c2c(CC)n(C)cc2)=O)O)=O)cc(C)cnc1F c1(CNC2CCC(NC(Cc3cn(C)nn3)=O)C2)ccc(C(F)(F)F)cc1CO C1(C(N2CCCC2c2ccc(C(F)(F)F)nc2)=O)CS(=O)(=O)CC1CO N1(C(C)=O)CCCC(CNC(=O)C(c2ccc(Br)s2)C)C1 N1(C(CC(CC)OC)=O)CC2(C1)CN(C(c1cncc(CO)c1)=O)CC(C)(C)O2 C1(NC(C2(C(=O)NC3CC=CC3)CC2)=O)CCOCC1CO.C(=O)NCCOCCO C1(NC(C(C)(C)OCC)=O)CN(C(c2c(C)cccc2C)=O)Cc2nccn2C1 Cc1ccc(CN(CC(C)NC(c2ncccc2NCC(C)(C)C)=O)C)cc1 C12(C(N(C(CNC(CN(C(=O)OC)C)=O)C)C)=O)CCN(CC1)C2 Cc1nc(NCCCC2CCN(C)CC2)cc(N2CCOC(C)(C(F)F)C2)n1 c1(CCC(N2CCN(C(C(C(C)C)=O)=O)C3C2C3)=O)ccc2c(c1)OCCO2 N1(C(c2c(N=[N+]=[N-])cccc2)=O)CCn2ncc(S(C)(=O)=NC(=O)C3CC3Cl)c2C1 C1(C(N(C2CCC(NC(C3CC(=O)OC3(C)C)=O)CC2)C)=O)CN2CCN1CC2 CC1CCN(C(c2ccc(F)c(C(F)F)n2)=O)C1CNC(=O)Cc1ccsc1 C1(C(=O)NCCN(C)C2CC2)CCC(C2CC2)N1C(=O)CCc1cn(C)cn1 C1(C)(C(=O)NC2CCC(NC(Cc3cc(C)no3)=O)CC2)CCC(F)(F)C1 c1(CC(=O)NCCC2CCCN2C(=O)CCn2cnnn2)cccc(Cl)c1F Cc1nc(C(=O)NCCC2CC(NC(=O)Cc3nncn3C)C2)c(Br)s1 CC(C)CCC(C(=O)N(CCCC(O)CO)C)NC(c1ccc(CO)s1)=O CS(=O)(=O)CC(CO)NC(=O)Nc1cc(Cc2ccccc2)cs1 C(CCCCC(=O)NCC1CCCN(C(C2(C(F)F)CC2)=O)C1)N(C)C N1(C(C2C(C)(C(F)F)C2)=O)CCC(C)(NC(c2cn(C(C)(C)C)cn2)=O)C1 c1(C(=O)NCC2(COC)CN(C(C3CCCS3)=O)C2)sc2cc(F)ccc2c1Cl CC(CCN(C)C)C(=O)NC1(C)CCN(C(C2CCN(c3ccncc3)C2)=O)C1 Cc1cc(C(=O)N(C(C)C(C)C)C)c(C)n1C1CCOC1 C=CCCC(O)CN(C(=O)CCCN(C)C(c1oc(C)nc1C)=O)C C1(C)(CC)CC(C(=O)NC(C)CCCNC(c2cccnc2C)=O)CCO1 C1(N(C)Cc2nc(CC)on2)CCCN(C(=O)C#CC2CC2)C1 C(C(C(=O)NCC(C)(C(C)C)NC(=O)Cc1ccon1)C(F)(F)F)OC C1(C(C)C)CN(C(C2(C(N)=O)CCC2)=O)CCN1C(=O)CCC1CC1CC1CC1 COn1cnc(C)c1C(=O)NCC12CCC1CN(C(=O)C(=Cc1ccco1)C)C2 C(=O)(C(C(C)NC(C1(CSC)CC1)=O)C(C)C)NC(CCOC)C(N)=O CCCC(C)CC(=O)N1CC2(C1)CN(C(=O)C(C(C)C)OCC(C)C)C2 C1(NC(c2cncc(C)c2Cl)=O)CC2CN(C(=O)C(F)C(F)(F)F)CC2C1 Cc1nc(=N)[nH]cc1C(=O)NCC12CCC(CN1C(c1ccc(C(C)C)s1)=O)C2 C1(NCc2c(OC)nc(Br)cc2)CC2CCC1N(C)C2 CCCCC(C)CCC(=O)NCC1(C)CCN(C(c2ncncc2C)=O)C1 C1(NC2(CCCCNC(CCSC(CC)=O)=O)CC2)CCC(=O)O1 N1(C(c2c(CCC)occ2)=O)CC(NC(c2cc(COC)on2)=O)C(N=[N+]=[N-])C1 c1(N(C)C)ccc(CNC(C2CCC(C(=O)NCc3ccc[nH]3)CC2)=O)nc1 C(=O)(CCS(=O)(=O)c1ccccc1)NCC1(NC(C(C)OCC(F)(F)F)=O)CC1 N1(C(C(C)NC(CC)(C)C)=O)CCCC1(C(=O)NCCc1cccc(O)c1)CC O=C(C1=CCCNCC1)N1CCN(Cc2ccc(C(F)(F)F)cc2)CC1 c1(Cc2ccccn2)nn2c(c1NC(n1cc(COC)nn1)=O)CCC2 C1(n2cc(NC(C)COC(F)F)nn2)C(F)(F)C12CCC2 c1(N2C(=O)CCC2)ccc(NC(N2CCC(CN3CCCOCC3)CC2)=O)cc1 C1(C(N2CC(NC(c3cc(C)[nH]n3)=O)C(O)C2)=O)CCCCC1(C)C Cc1nn(C(F)F)c(C)c1CC(=O)NC(CO)C(C)NC(C12CCC1C2)=O C1(N)CN(C(=O)CCOC)CC1CO.c1(CNC(C(=O)CO)=O)nc(C(F)F)no1 C1(C)(NC(c2ccn(CCN(C)C)n2)=O)CCN(C(=O)CN(S(C)(=O)=O)C)CC1 c1(C(N(CCN(C(C(CC)C)=O)C(C)C)C)=O)ccc(-c2ccon2)cc1 c1(C(=O)NC(C(C)NC(c2nc(C(C)C)oc2)=O)C(C)C)cccc(C#N)c1 C1(C(=O)NCC(C)(CO)NC(c2occ(C(=O)OC)c2)=O)CC(C)(C)CO1 C(CCCCCCO)NC(C1(CCNC(C2OC3CCC2C3)=O)CC1)=O c1(CCN(CCCC#C)C)ccnc(C)n1 c1(C(=O)NC2CC(NC(c3occ(C)c3)=O)CC2O)c(C)ncn(C)c1=O C(=O)(C(C)(C)CF)N1CCC(CN(C(=O)CCN(CC(F)(F)F)C)C)C1 Cc1cccc(C(C)NC(=O)CC2CCCC2NC(C2COCC(C)O2)=O)n1 CCC(CC(C)C)C(=O)NC(C1CCN(C(c2nnc(S)n2C)=O)CC1)C(C)C C(=O)(CCCCCNC(=O)C(C)C(=O)OC)NCCCCOCC c1(C(=O)NC2CC(N(C(CC(C)F)=O)C)C2)cccc2c1NC(=O)CO2 C(=O)(CCC(=O)NCC1CC(NC(=O)C(C)(C)c2nncn2C)C1)OCC N1(C(C2N(C(CC(CC)SC)=O)C(C)CC2)=O)CC(C)N(C)C(C)C1 N#Cc1ccc(F)c(C(=O)NC2CC3(C2)CN(C(=O)CCCN2CCCC2)C3)c1 C1(CNCCCCCCOCCO)Cc2nccn2C1 c1(C(=O)NCC2(F)CC(NC(C3C(C)COCC3)=O)C2)cc(S(N)(=O)=O)c[nH]1 CC1(C)OC2(C(N3CCCC(O)(CNC(c4cccc(F)c4N)=O)C3)=O)CC1C2 c1(C(N2CCC(CNC(CC(C)CF)=O)C2)=O)cc(S(=O)(=O)NCC2CC2)c[nH]1 C(=O)(C(C)(C)S(C)(=O)=O)N1CCCC(N(C(c2[nH]cc(C)c(=O)c2)=O)C)CC1 c1(C(=O)NC)n[nH]c(=NC(=O)N(C(C)C)Cc2ncccc2Cl)s1 C(=O)(CS(=O)CCC(F)(F)F)NC1(CO)CCN(C(c2c(C)n[nH]c2)=O)C1 C1(CNC(C2CC3CC3N2C(=O)C#CC2CC2)=O)CC(C2CC2)=NO1 c1(NC)ccncc1-c1cn(CC2CCCC2NC(c2c(Br)n[nH]c2C)=O)nn1 CC(C)S(=O)(=O)C(C)C(=O)NCCC(C)(C)CNC(c1ccc(N)c(F)c1)=O C(C)(C(=O)NC(C(=O)N(C)CCc1nccs1)c1ccoc1)OC N1(CCNC(C23CC4CC2C3C4)=O)CC2CC(N(Cc3n[nH]c4c3CCC4)CC)C1C2 N1(C(C=CC)=O)CC(CN(c2ccccc2)C2CC(C(F)(F)F)C2)CC1C c1(NC(C23CN(C(CC)=O)C(C2)CO3)=O)ccc(CC)nc1C c1(C(N2CCN(C(C(COC)OC)=O)C(C)C2)=O)ccc(Cl)c(C)c1N N1(C(c2cc(OC)ncc2)=O)CCC12CN(C(C1CCOC(=O)CC1)=O)C2 c1(C(=O)NC2CCN(C(=O)Cc3ccsc3)C2C2CC2)cccc2c1C(=O)NC2 N1(C(C(C=C)(C)O)=O)CC2CC(C1)N(C(c1c[nH]nc1-c1ccsc1)=O)C2 Cc1sc(C)c(C(=O)NC(C)CC(C)NC(C2(CN(C)C)CC2)=O)c1Br N1(C(C(CC)C(=O)OC)=O)CCOCC12COCCN(C(=O)CCSC)C2 C(c1ccc(F)cc1)=CC(=O)N(C1(C2N(C(CC(=C)Br)=O)CCCC2)CC1)CC C1(O)(CNC(C(c2cncnc2)C)=O)CCCN(C(c2cscc2F)=O)C1 c1(CC(C(=O)OCCCC2CCC2=O)O)ccc(O)cc1 c1(C(C)C)cc(N2CCC(C)(CNC(C3(C4CCC4)CC3)=O)C2)n2ncnc2n1 Cc1ccc(CO)cc1C(=O)NC1CCN(C(=O)C(=O)N(C)C)C1(C)C c1(C(N(CCNC(=O)CC2CC(F)(F)C2)CC)=O)cc2n(n1)CCC2 C(C(C)C(=O)N1CCC(CC(N2CCCC2C2CCCC2)=O)C1)OCC C1(CCC)(NC(C2CCCC2C)=O)CCCN(C(=O)CCCCCOC)C1 C12(C(N(CCN(C(C)C)C(c3occc3Cl)=O)C)=O)CCN(CC1)C2 N1(CCC(=O)N(C(CC)CNC(=O)CO)C)CCN(c2ccc(OC)cc2)CC1 C(CC(C)(C)C(=O)N1CC[Si](C)(C)CC1)NC(CCC1N(C)CCC1)=O c1(NCC)c(C(=O)N(C2CN(C(=O)C(CO)N(C)C)C2)C)cccc1F N1(C(c2csnn2)=O)CCCC(C2CCN(C(=O)C=Cc3ccc(F)cc3)C2)C1 c1(NCCN2CCN(c3ccccc3)CC2)cc2c(Cl)cc(Br)cc2[nH]1 N1(CC(C)C)CC(C(N2CCC(CN(C)C(c3ccc(CO)[nH]3)=O)C2)=O)CC1=O N1(C(C(C)NC(c2c(C)ccc(I)c2)=O)=O)CCc2ccccc2C1 c1(CC(=O)NC2CN(C(C(C)=CC)=O)CC(C)(C)C2)ccc2oc(O)nc2c1 C#CC1CC2(CC2)CN1C(=O)CC1CCCC(NC(C2(CC)CCCO2)=O)C1 C1(NC(c2cc[nH]c2C2CC2)=O)CCN(C(c2cc3[nH]ccc3s2)=O)CC1O Nc1cc(C(=O)NCC2CC(NC(C3CC4(CCC4)C3)=O)C23CCC3)cc(F)c1 C1(C(N2CCCC2c2cn(-c3cc(Cl)sc3Cl)nn2)=O)Cc2c[nH]cc2S1(=O)=O C=C(C)C(C)(C)C(=O)NC1CCN(C(=O)COCCc2cccs2)C(C)C1 c1(C(N(CCN(C(=O)C(C2CCOCC2)F)C)C)=O)ccc(F)c(S(N)(=O)=O)c1 c1(C(=O)NCC(CN(C(C(C)NC(N)=O)=O)C)(C)C)ccc(OCF)cc1 C(CO)(CC(C)(C)C)NC(C(CCC1CC1)NC(c1cccc(NC)n1)=O)=O C1(NC(c2cc(C)sc2C)=O)CC(F)CN(C(c2cc(C3CC3)[nH]n2)=O)C1 Fc1cnc(-c2noc(-c3nnc[nH]3)n2)nc1 Nc1cc(C(=O)NCC2CCCCN2C(c2ncnc(O)c2F)=O)cc(Cl)n1 N1(C(C2CC(=C)C2)=O)CC2C(NC(=O)C(C)S(C)(=O)=O)CS(=O)(=O)C2C1 C(C(=O)NC(c1cn(CC2CCC(=O)O2)nn1)C)(C(C)(C)C)NC(C)=O CN1C(=O)NCC1C(=O)NC(CNC(c1cnn(C)c1Cl)=O)C1CCC1 C1(NC(c2[nH]cc(C)c2)=O)CC(CC(=O)NCC(C)C(F)F)C1(C)C C(C(C)(COC)C(=O)NC1CC2(C1)CC(C(=O)NC1(C)CCOC1C)C2)OC c1(CC(=O)NC2C(O)CCN(C(C3(C)CC(=C)C3)=O)C2)coc2ccc(C)cc12 N1(C(c2cnc(CC)nc2)=O)CCOC(C)C1C.C1(CC2CC2)C(=O)N1 C(=O)(C1NCCn2nccc21)Nc1c(Cc2nc(C)cc(C)n2)cccc1 Cc1cc(C(=O)NCCN(C(C2CC3C=CC2O3)=O)CC2CC2)c(F)cc1N CCC(CC(=O)N1CCC(NC(c2ccns2)=O)C12CCC2)C(=O)OC(C)(C)C N1(C(C2C(C)(C(F)F)C2)=O)CC2CC(NC(c3cc4occc4s3)=O)CC(C2)C1 N1(C(COC(CC)C)=O)CCN(C(c2cnc(C(C)OC)s2)=O)CC1C1CCC1 C(=O)(C(CCCC)NC(=O)CCN(C)CCC)NC(C=C)(C)C c1(CN2C3C(C(=O)Nc4cc(C)nc(Cl)c4)C(C3)C2)cnc2ncccn12 CCC(C(=O)N1CC(O)(CCNC(c2ccc(OC(C)(C)C)cc2)=O)C1)C(C)O Cc1c[nH]cc(-c2nc(C3CCOC3)nn2CC(F)(F)F)c1=O C1(C(=O)NC(CC)CCCO)COCCN(C(c2coc(N(C)C)n2)=O)C1 c1(SCC(N2CC(C)(C)OCC2C(F)(F)F)=O)cc2cc(Br)ccc2o1 N#Cc1ccc(C(N2CC3CC2CCC3NC(=O)CC2CCCCC2)=O)c(F)c1 N1(C(C2N(CC)C(=O)CC2)=O)CCC(C)(C)C(NC(=O)CCN2CCCCC2)C1 N1(C(C2C(N(C(C3(C)CCC(=O)N3)=O)C3CC3)COC2)=O)CC(S(N)(=O)=O)C1 CN=c1nc(C(N2CC3C(NC(C45COC(CF)(C4)C5)=O)C3C2)=O)cc(C)[nH]1 CCCCCCOC(C)C(=O)NC(CNC(=O)CC1CCOCC1)C1CC1 N1(C(C(CCC)NC(N)=O)=O)CCN(C(c2ccccc2F)=O)CC1CCOC C(=O)(C(C)(C)CO)NC1(C(C)C(=O)N(CCC(O)C2CCCC2)C)CC1 c1(C(=O)NC2CCN(C(C(C=C)(C)O)=O)CC23CCC3)c(F)c(F)cc(F)c1F C=CCCC(C(=O)OC)NC(C1(CNC(C2COCCN2C)=O)CC(C)(C)C1)=O C1(NC(C2C(C)CN2C(C2COCCN2C)=O)=O)CC(C)(C)C12CC2 C(=O)(C(C)COC(C)=O)N(C1CC(C(=O)NCCOCCC)C1)C C1(C(=O)NCC(CNC(=O)CCN)F)CCCN(C(c2ccc(Cl)s2)=O)C1 C(=O)(C(C)(C)CC1CC1)N1CCC(CN(C(c2nc(CC)oc2)=O)C)C1 CC1(C)CC(NC(C2CN(c3nncs3)C2)=O)CN1C(C1CCC(=O)N1)=O C(=O)(CC(C)(C)C(=O)NCC(C)N(C)C(c1ccccc1C1CCC1)=O)OC Cc1c(NCCCc2nc(C3CC3)n[nH]2)nc[nH]c1=NCC1CC12CCCCC2 C1(C(=O)NCC2(CC)CCCC2)CC(F)CCN1C(=O)CC1CC(C)(C)C1 C(C(C)C(C)C(=O)N(CC(C)(C)NC(c1ocnc1C1CC1)=O)C)OC C1(OC)CCN(C(=NCCNC(C)=O)NCC2(SC)CCC2)CC1(C)OC C1(NC(C2(Cl)C(C)(C)C2)=O)CCCN(C(c2ccc(C(F)(F)F)cn2)=O)C1 C1(C(=O)NCc2ccc(C)cc2)CCN(C(c2cccc(F)c2I)=O)CC1O CCCCC(O)C(C)C(=O)N1CC2(C(=O)N(c3ccc(F)cc3)C)CC1CO2 C1(NC(C2CCC2)=O)CN(C(C2C=CCS2)=O)CC2(CC2)C1 N1(C(C(C2CCCC2)OC)=O)CCCCC(C2CN(C(C3CC34CC4)=O)C2)C1 N1(C(C(C(CCCC)O)C)=O)CCC(C2CCN(C(=O)COCC3CC3)C2)CC1 C(=O)(C1CCOc2c(F)cccc21)N(CCN(C(c1cc(=NC)[nH]cc1)=O)C)C Cc1ccc(C(=O)N(CC(C)NC(c2cc(C(C)C)nn2C)=O)C)nc1C CC(C)C(C(=O)NC1CC(NC(C2CCCCC2)=O)C(O)C1)C1CCC1 Cc1cscc1CNC(=O)CCNC(=O)C(C)n1cccn1 c1(CC(N2CC(OC)C(NC(C3CCCN3N=O)=O)C2)=O)ccc2c(c1)CCO2 c1(OC)c(F)ccc(F)c1C(=O)NCC1CC(NC(=O)Cn2nccn2)C1 C1(C(N2CCC2CC(C)(C)C)=O)(CNC(C(CC2CCC2)OC)=O)CCCCC1 O=C(CS(=O)(=O)c1ccc(Br)cc1)NCC12CC(C1)C(C(F)(F)F)O2 c1(C(=O)NCC2(C(=O)NC3C(C(C)(F)F)C3)CCCCC2)ccc(F)cc1Cl S(=O)(=O)(C1CCc2ccccc2C1)NC1(N2CCN(C)CC2)CC1 [N-]=[N+]=NCCCC(=O)N1CCSCC1CCNC(=O)COCC1CCCO1 c1(C(=O)NC(C=CC(=O)N(C(COC)C)C)(C)C)ncccc1F N1(C(C(P(C)(C)=O)O)=O)CCC2(CC1)CC2NC(c1ccnnc1)=O N1(C(C2CCCC(C)C2)=O)CC2CCC(CNC(c3ncncc3Cl)=O)(C2)C1 N1(C(C2C(C(=O)OC)CCO2)=O)CCC(CNC(=O)CCc2cnc(C)o2)CC1 c1(C(=O)NC2CCN(C(=O)C=CCO)CC2CO)cnc2c(C(F)(F)F)cccn12 N1(C(CCCCCNC(N)=O)=O)CC2(CC(NC(=O)C3=CS(=O)CCC3)CO2)C1 CC1(C(=O)NCc2n[nH]c(=N)[nH]2)C=CCN1C(c1ccc(C#N)o1)=O c1(C(CC)NCC2CCCC3(CCOC3)O2)cccc(S(N)(=O)=O)c1 Cc1cc(OCC(=O)NCC2(O)CN(C(=O)CCC(O)CN(C)C)C2)ccc1Cl c1(OC)cccc(NC(=O)C(C)(C)C2CCN(C(=O)C(C3CCCCC3)=O)C2)c1 C1(CNC(CCC(C)C)=O)CCN(C(c2ccc(Cl)c(F)c2)=O)C1(C)C c1(C(=O)NC2CCN(c3c(C)cccc3)CC2)c[nH]c2cc(Cl)c([N+](=O)[O-])cc12 c1(C(=O)NC2CN(C(c3cnc(OCC)s3)=O)C(C)CC2)cc(F)c(Cl)cc1F C1(NC(CCC#C)=O)CCN(C(C2(c3ccccc3)CC2)=O)C12CCC2 N1(C(c2c(CC)c[nH]c2)=O)CCCC(CO)(NC(=O)C(C)CC)C1 CC1CCC(O)C(NC(=O)CC2CCCCN2C(c2ccc(F)cc2)=O)C1 C1(CC#N)CCN(CC(=O)NCC2CNC(=O)CO2)CC1c1nn[nH]n1 N1(C(c2cnc(OCC)c(Cl)c2)=O)CCC2CN(C(=O)CCCC(C)(C)C)CC12 c1(C(=O)NC23C(NC(CC4(C)CC4)=O)CC(CC2)C3)cccc2c1OCCC2 C(C)(C)(C#Cc1cn(Cc2cnoc2C(=O)OC)nn1)NC(C1(OC)CCC1)=O c1(CNC(C2(NC(CC(C)SC)=O)CCCC2)=O)ccc(C2CCOCO2)cc1 C1(C(=O)NCC(=CC(=O)N(C(CO)CO)CC)C)CCC(C(N)=O)C1 C1(C(=O)NCC(c2ccccc2F)O)(OC)CCN(C(=O)CSC)C1 C(=O)(C1=CCCOCC1)NC(CNC(Cc1nc(C)c(C)s1)=O)CO N1(C(=O)Nc2c(OC(C)C)nccc2)CC2CCC1(CO)CC2 c1(OC2CCN(C(C=CCCC)=O)C2)ccccc1NC(=O)C=CS(C)=O c1(C(=O)NCCCCC(CO)NC(C)=O)ccc2cccc(C)c2n1 n1(CCC(N2CC(NC(=O)CCc3cnco3)C2)=O)nc2ccccn2c1=O N1(C(C2OCCN(C(C(CCOC)OC)=O)C2)=O)CC(C)(C)CCC1CO C1(NC(C2CC(C#C)(O)C2)=O)C2CC3C1C3C2C(=O)NCCCC(C)O N1(C(c2c(C)[nH]c(C#N)c2)=O)CCC2CCC(C1)N2C(c1cccnc1CO)=O N1(C(Cc2onc(COC)n2)=O)CC2(C1)CN(C(c1cnc(OC)c(C)c1)=O)C2 C1(C(=O)NC(COC)C)CCCN(C(=O)CCCC(C)=O)C1C c1(C(N(CCNC(c2ccc(NC(N)=O)cc2)=O)CC)=O)ccc2cc[nH]c2c1F C(=O)(C(O)CC(C)(C)C)NCC1CC(NC(CC(C)SC)=O)C1 c1(C(N2CCC3(C(C(=O)Nc4ncc(F)cn4)C3)C2)=O)cccc(F)c1[N+](=O)[O-] c1(C(=O)NCC2N(C(C(C(CC)C)NC(N)=O)=O)CC2)ccc2c(c1)CC(=O)N2 C=Cc1cnn(C)c1C(=O)N(CC(C)N(C)C(c1cc(C)cc(Br)c1)=O)C c1(C(N2CC(CS(N)(=O)=O)C(C)C2)C(=O)NC)ccc2c(c1)CC(C)(C)O2 c1(-c2ccc(C(=O)NCC(=O)O)cc2)nc2c(s1)CCN(C(=O)CO)C2 CCCCC(CNC(=O)C(C)=C1CCCC1)NC(=O)CC1CCC(=O)N1C Cc1cn(C)cc1C(=O)NC(C(=O)NOCC1CCC1)C1(C)CC1 C1(C)(NC(C2C(CNC(CC3N(C)CCC3)=O)C2(C)C)=O)CC=CCC1 c1(CC)ccc(F)c(C(N2CCOCCC2CC)C(=O)NCC(C)C)c1 O=C(C#Cc1ccccc1)N1CCCCC1CC(N1CCC2(C1)CC2(F)F)=O c1(NC(C2CCCN(C(=O)CSc3nncs3)C2)C)c(F)cc([N+](=O)[O-])cc1F C1(SC)COCC1NC(C1CCN(C(C2CCCO2)=O)C1)=O c1(C(C(=O)NCC2N(C(CC=CC(C)(C)C)=O)CCC2)O)ccc(F)c(F)c1 C1(N(C(c2cnc(C)[nH]2)=O)C)CN(C(c2cc(F)ccc2C)=O)CCC1O c1(OC)cnccc1C(=O)N(CC(=O)NCC1CCC(C)CC1)C c1(CNCC(C)(O)C2CCC2)cc(Br)ccn1 c1(CNC2CC(NC(Cc3c(C)n[nH]c3)=O)C23CCC3)noc2c1COCC2 c1(C(=O)NC(CC2CCN(C(Cc3nnc(C)o3)=O)CC2)C)cc2[nH]ccc2s1 CN1CC(C)(NC(c2ccn(CCNC(c3cnncc3O)=O)c2)=O)CCC1=O Nc1cc(F)c(F)cc1C(=O)NC1CN(C(c2ncc(F)cn2)=O)CC12CC2 CCCC(CC)C(=O)N1CCC(COC)(NC(=O)CN2CCCNC2=O)CC1 C1(CNC(CC(C)OC)=O)CCCCN1C(=O)C(C)Oc1ccc(F)nc1 C1(CCNC(C(C)N(C)C)=O)CCCN(C(c2cc(C(F)(F)F)nn2C)=O)C1 C(=O)(C1=NN(CCO)C(=O)CC1)N(C1CC(NC(c2c(C=C)cnn2C)=O)C1)C C=C(C)C(CC(=O)NC(C)(CNC(=O)CC(CC)OC)C1CC1)OCC c1(N2CCCC(C(C)NC(C3C(CC)OCC3)=O)C2)nc(C(C)C)ccc1C#N CCCC(C(=O)N(C1CCCOC1)C)NC(=O)CC1CCCOC1 C(=O)(CC(C)(O)C(F)(F)F)NCC(C(C)C)NC(CCCCN(C(C)C)C)=O C1(C)(C(N(CC2=CCCOC2)C)=O)CCN(C(C2CC(=O)NC(=O)C2)=O)CC1 c1(C(=O)NC(C)CNC(=O)CN2CCCCC2)ccc2c(c1)CCCS2(=O)=O C1(SC)CN(C(=O)C(n2cc(-c3cnn(C4CC4)c3)nn2)C)C(C)(C)C1 C=CC1CCCC(NC(=O)C(C2CC2)NC(C2CN(C)CCN2C)=O)C1 c1(OC)ccccc1CNC(=O)C(C(C)O)NC(=O)Cc1ccc(F)cc1 Cc1ccncc1C=CC(N1CC(C(C)NC(C2CC(C)(C)C2)=O)C1)=O c1(CC(N2CC(C)C(CNC(c3cccs3)=O)C2)=O)cc2ccccc2o1 Cc1cc(OC(F)(F)F)ccc1C(=O)NC1CCC1NC(C12CCC1C2)=O c1(C(=O)NC2CCC(CCNC(CC3(OC)CC3)=O)C2)ccc2c(n1)CCC2=O C1(NC(=O)NC(COc2c(C)cccc2)C)CCC(=O)N2CCCCC12 c1(C(=O)NCC2(CNC(c3ncn(C(C)C)c3)=O)CC2)nnc(Cl)cc1N C(CC)(C(=O)NCCC(O)CNC(=O)Cc1nncn1C(C)C)OCC Cc1[nH]cc(C(=O)N(CCNC(=O)C=CC(F)(F)F)C(C)C)c(=O)c1Cl c1(C(N2CC3(CCC(NC(c4scc(C)c4)=O)C3)C2)=O)cnc2ccc(F)cn12 N1(C(C(CC)OC)=O)CCC(O)(C2(NC(=O)CNC(=O)CC(F)(F)F)CC2)CC1 N1(C(CC2(CC)CCC2)=O)C(C(=O)NCC2(C)CSC2)CC1C C(C1OCCc2sc(I)cc21)NC(=O)NCCc1cccnc1Cl Cn1nc(C(N2CC(C)(NC(=O)CC3CC(=O)C3)C2)=O)c(=O)c2ccccc12 N1(C(=O)Cc2cccc(OCCF)c2)CCN(C(C2COCC2O)=O)C2CCC12 N1(C(C2N(CC)CC2)=O)CCC2CCN(C(c3ccc(F)cc3C#N)=O)CC2C1 C(=O)(CC(C)NC(=O)C(C)CNC(c1ncoc1C(C)C)=O)OC C#CCC(C(=O)NCc1cncc(C(=O)Nc2cccc(CCO)c2)c1)C1CC1 C#CCCCCCCCC(=O)N(C1CCN(C(=O)COCc2ncnn2C)C1)C Nc1cccc(C(=O)NCC23CC2CN(C(C2CC4CCC4C2)=O)C3)c1F N(C(=NCCN(C)C)NCC1CCOC1=O)Cc1cc(C)on1 N1(CCC2CC(O)C23CCC3)Cc2cccc(-c3ccccc3)c2C1 CCCS(=O)(=O)NC(C)C(=O)N(CC(C)(C)N(C(=O)Cc1csc(=N)[nH]1)CC)C C1(C(=O)NCCN(C(=O)CCS(C)=O)CCCN(C)C)COc2ccc(F)cc2C1 C1(CNC(CC(=C=C)C)=O)CCCN(C(c2cccc(OC(C)C)c2Cl)=O)CC1 C(=O)(C1=NOC2(CCCN(CC3CCCCC3)C2)C1)N(C(=O)C(O)c1ccco1)C c1(C(N2C(C(=O)Nc3c(OCC)nccn3)CC2)=O)nc2c(s1)CN(C)CC2 C(C(C)CC(=O)NCC(C)CN(C(=O)C(C)(C)c1cnco1)C)OC C1(C(=O)NCCOCCCC)(NC(c2ccsc2OC)=O)CCC(C)(C)C1 c1(C(=O)NC(CC)C(=O)NCCN(CCN(C)C)CC)cc(C)c(F)c(C)c1 c1(CNC(c2c(CC)n(C)nn2)=O)cnn2c1CN(C(=O)C1=CCSC1)CC2 C1(C(N2C(CNC(COCc3cccc(OC)c3)=O)CC2)=O)CC12CC(C)(C)C2 C12(C(N3CCC(C4N(C(C(=O)NCC)=O)CCC4)CC3)=O)CCC(C)(CC1)CO2 N1(C(CS(=O)(=O)N(CC)CC)=O)CC(C)CN(C(=O)Cc2cnco2)C(C)C1 N1(C(C(C)Cc2ccncc2)=O)CC(C2CN(C(C3(C)CS(=O)(=O)C3)=O)C2)C1 N1(C(c2c(C)nc(CC)o2)=O)CC(C2(NC(c3ccc(N)c(N)n3)=O)CC2)C1 C1(CO)C2CN(C(=NCCC(C(F)(F)F)N3CCCC3)NC3CCCCC3)CC12 c1(C(=O)NC2C3CCN(C(CCC(=O)N(C)C)=O)C32)cc2cccnc2s1 C(CC(C)N=c1[nH]c2ccc(Br)cc2cc1C#N)NC(c1n(COC)ncc1)=O C#CC1(C(=O)NC(c2ccccc2)CNC(=O)CN(C(=O)C(C)C)C)CCC1 Cc1ccc(C2(C(=O)NCC3(F)CCC(NC(=O)CC(F)(F)F)C3)CC2)cn1 C1(O)(C(=O)OC)CCN(C(=O)CO)CC1.C1(CCCC(C)C)CCCO1 c1(CNC(C2CCCO2)CC)cc(Br)c2c(c1)OCO2 CCC(CCOC)C(=O)N1CCCCCC1C(=O)NCC1CCC2(CC2)C1 N1(C(CCC)=O)CCC(NC(c2ccc(Cc3ccccc3)o2)=O)C1C(C)C C1(C)(C(N2CCC(C(C)NC(CC(C)C)=O)C2)=O)CCNC1=O C12(C)CCN(CC1)C(=O)O2.C1(CCC)COCCN1CC.N(CC)CC C(CC(C(C)C)NC(=O)COCc1cccc(C)c1)NC(c1cc(SC)[nH]n1)=O CC(CC(C)(C)C)C(=O)NC1CCN(C2CCN(C(=O)C3=C(Cl)CCC3)C2)CC1 c1(C(=O)NC2(C#N)CCN(C(c3ccc(O)nc3)=O)C2)cc(F)c(F)c(Br)c1F C(=O)(C(C)C(C)C1CCCC1)NC(CNC(C(c1cccs1)OCC)=O)C(C)C C(=O)(CCC(=O)NCC(O)CNC(c1ccnn1CCF)=O)NC.C12CC1OC2 c1(SC)nc(N2CC3C(CNC(=O)C4=C(Cl)CCOC4)C3C2)c(C)c(Cl)n1 C1(NC(C(c2ccc(F)cc2)C)=O)COCCN(C(c2ccc(=O)n(C)n2)=O)C1 CCN(OC)C(=O)C1CC(O)(CNC(C2(C3CC3)CC2)=O)C1 N1(C(c2cnc(C)nc2C)=O)CC2CCC(C1)N2C(=O)C(C)n1ccnc1 c1(C(=O)NC2CC(O)C2)ccc2ncc(Br)cc2c1.C12CCCC1CNC2=O C1(O)(C(N2CC(c3ccccc3)(N(C)C)C2)=O)CCN(C(=O)OC(C)(C)C)C1 C(=O)(CCCS(N)(=O)=O)NC(CCCNC(Cc1ccc(OCC)cn1)=O)C c1(C(C(=O)NCC(=C)C)N(C2(CNC(C)=O)CC2)C)ccc(Br)cc1C N1(C(CCCOCC(C)C)=O)CCC2CCN(C(=O)CC3CCCC3)CC12 c1(C(=O)NC(CNC(Cc2c(C)n[nH]c2C)=O)C(C)C)cccc2c(C)csc12 C1(C(=O)NCC(c2nccs2)C)CN(C(c2nn(C)cc2Cl)=O)CCN1C c1(C(=O)Oc2ccccc2)cccc2c1oc(=O)n2C.C(C)(CC=O)N(CC)C1CC1 c1(CC)cc(C(=O)NCC2CCCC2NC(=O)C=Cc2cc[nH]c2)nn1C c1(NC(CCCSC)(C)c2nnnn2C2(C)CC2)nc2c(s1)CC(C(C)C)CC2 CCC(CCc1cccc(F)c1)C(=O)O.c12cn(nn1)C1CC(C1)NC(=O)C2 Cn1ncc(CC(=O)NC(C)(C)CNC(=O)CCc2ccco2)n1 S(=O)(=O)(c1ccc(Br)cn1)N(c1nc(C)nc(O)c1)C1CC2CNCC2C1 C(=O)(C#CC1CCOC1)NC1C=CC(NC(CCCC#C)=O)C1 N1(C(C2=C(C)S(=O)(=O)CC2)=O)CCOC2CCN(C(C3CC34CCOCC4)=O)CC12 CC1CCC(NC(c2sc(F)cc2Cl)=O)CN1C(=O)Cc1cccn1C N1(C(c2cnn(CC)n2)=O)C2CCC1C(CNC(=O)C(C)(O)C(C)C)C2 Cc1cc(=NCCc2cscn2)[nH]c(N(C)Cc2ccnc(C(C)C)c2)n1 c1(C(C(F)(F)F)N(C)C)ccc(CN2CC(F)(NC(=O)OC(C)(C)C)C2)cc1 Cc1ccc(CC(=O)NC2(C)CCCN(C(C3CC(=C4CC4)C3)=O)C2)cc1[N+](=O)[O-] Cc1nc(C=CC(=O)NCC(CO)NC(c2c[nH]nc2C2CC2)=O)[nH]c1C c1(CNCC2N(C(C3CCC(CC)CC3)=O)CCOC2)cccc(C)c1Cl N1(C(c2c(C)cnn2C)=O)CCN(C)C(C(=O)Nc2ccc(N(C)C)cc2)C1 C(C(C)(C)CC(=O)NC(c1csc(C)n1)C)NC(C(C1CCOC1)OC)=O c1(C(=O)NC(C(C)NC(CC2N(CC)CCC2)=O)(C)C)cnn2c(N)ccnc12 Cn1nccc1-c1cn(C2(C(=O)NCCC3CC3)CC2)nn1.C12CC(C1)S2 c1(C(C)C)cc(C(=O)NC2CC(NC(c3csc(C(N)=O)n3)=O)C2)on1 CCC(CC(=O)NCC(C)(COC)CC)NC(=O)C(C)SC(C)C C(=O)(C1=C(Cl)CCCC1)N1CCC(COC)(NC(=O)C(c2ccc(C)s2)C)C1 C1(CC(=O)N(C(C)CNC(c2ccc(C(F)F)o2)=O)C)CCCC2(CCC2)O1 Cc1c(C(=O)NCC2(O)CN(C(=O)CC3CCSCC3)C2)[nH]c2c(C)cccc12 C(CCCCCC(=O)NC1CC2CCC1O2)NC(CCCOCCOC)=O c1(CC)ccc(C(=O)NCCC2CCCN2C(=O)COc2ccon2)cc1C CC(c1ccccc1)=CC(=O)NC(CO)C(=O)NC1CC(C2CC2)C1 C1(CN(C(c2cn(CC)nn2)=O)C)COCCN1C(C1CCN(C2COC2)C1)=O N1(C(CC(CC)NC(COC(CC)C)=O)=O)CCOC2(CCC2)CC1 N1(C(C(=O)NCCC)c2ccco2)CCCNC(=O)C1CC CC1CN(C(=O)C(C)n2cccc2)CCCN1C(=O)C(O)CC1CCCCC1 c1(C(=O)OC)sc2nc(C)cc(C)c2c1NC(c1cnc(SC)nc1O)=O n1(CC)nc(C(=O)NCCC2CCCN2C(=O)C(C#N)C2CC2)cc1C1CC1 C(C#Cc1cccnc1)NC(C(c1cn(C)nn1)NC(C=C(COC)C)=O)=O N1(C(CCCC)=O)C2CCCC1CN(C(c1cnc(C)c(C(C)=O)c1)=O)CC2 Cc1c(N)ccc(C(=O)NC(C)CNC(c2ccc(C(N)=O)o2)=O)c1F c1(C(N2CCC(NC(C(CC)SC)=O)C(O)C2)=O)cc(O)cc(F)c1F c1(OC)nc(C)ncc1C(=O)NC(C1CCCN1C(=O)C(C)n1cnnn1)C c1(-c2nc(CC(C)C)nn2C2CC2)ccc2ncc(=O)[nH]c2c1 C(=O)(C1=CCCOCC1)N1CC(CNC(c2c(CC)nnc(C)c2)=O)C(C)CC1 N1(C(C2(F)C(C)OCC2)=O)CC2CC1CC2C(=O)NC(C)C(=O)NC(C)(C)C CN1CCN(C(=O)CC2COC(=O)C2)C(CNC(=O)CCn2ncn(C)c2=O)C1 CCC(CN=c1[nH]c2ccccc2cc1S(=O)(=O)NCc1csnn1)CC(F)(F)F N1(C(C(c2cnn(C)c2)NC(C2OCCN(C)C2)=O)=O)CCC(C2CCCC2)C1 CC1CCCN(C(=O)C(CO)N(C)C)C1CNC(=O)C(=Cc1ccncc1)C CCC(CCC(=O)N1CCN(C(C2CC2c2cccc(C)c2F)=O)CC1)OC C12(CNC(C3CC(CC)C3)=O)CC(NC(=O)CC(C)(C)C(F)F)(C1)C1(CCC1)O2 N1(C(C(C)(C2CC2)OC)=O)CCC(F)(CNC(C2OCCN(C)C2=O)=O)CC1 CC1CN(C(C2CC2Br)=O)CCN1C(=O)CCCCC#N CC1CC(C(=O)N2CC3(CC3)CC2C(=O)Nc2ccc(Cl)cc2N)=NO1 C1(NC(CSC)=O)CC(CO)N(C(=O)CCCN2CCCC2=O)C1 C1(CC(=O)NCCC(C)N(C(CCSCCCC)=O)C)CCCC1C Cn1cc(C(N2CC3CC3(CNC(c3cnc(O)n3C)=O)C2)=O)c(C(F)F)n1 c1(C(N(CCN(C(=O)C(C)Cc2ccco2)CC)CC)=O)cnc(C)c(N)c1 C1(CNC(c2c(C(C)C)scn2)=O)CN(C(C2CNC(=O)N2)=O)CC1(C)C CC1CN(C(=O)CCC2(C)CC2)CCN1C(C1COCC1C(F)F)=O c1(C(=O)NC2C=CCN(C(c3nc(OCC)sn3)=O)C2)cc2nc(Cl)ccc2o1 c1(C(=O)NCC2CC(NC(C3(CCF)CC3)=O)CCO2)cc2c(s1)CCC2 c1(C(N2C(C(=O)NCCOC3CCCOC3)CSC2)=O)scnc1Cl C1(C(N2CC(C(C(=O)NC3(n4cccn4)CCC3)O)C2)=O)CCCSC1 N1(C(C(C)(C)NC(COC)=O)=O)CCC2CC2(C(=O)NCCCCCF)CC1 CC1(C(=O)NC23COC(C(F)F)(C2)C3)CCOC(c2ccccc2)C1 C1(CNC(c2ccc(C)c(F)c2)=O)CC12CCN(C(C1CC(F)C(=O)N1)=O)CC2 CCC(C)(CNC(c1coc(CO)c1)=O)C(=O)N1CCCC(O)(C(N)=O)C1 C1(CNC(c2cc(C)on2)=O)CN(C(=O)Cc2c(C)n[nH]c2C)C(C)(C)C1 Cc1ccc2c(n1)CN(C(=O)C1=NOC(CNC(C3CCOCC3)=O)C1)C2 C(=O)(C1CCc2cccc(O)c21)N1C(C(C)NC(=O)CSC(F)(F)F)CCC1 c1(C(C)NC(=O)C(c2cnn(C)c2)NC(C2CCCC2)=O)cncnc1 C1(NC(c2nccc(C)n2)=O)CC1C1CCN(C(C2CC2F)=O)CC1 C1(NC(C(N2CCC(C(CC)C)CC2)=O)=O)COCC(C)(C)C1 CC(C)CC(C(=O)NCCN1CCOC1=O)NC(C1CC(N(C)C)C1)=O C(C(CC(=O)NCc1cncn1C)C1CCC1)NC(C1CC(C)C1)=O C(=O)(C(CC)C(C)(C)CC)N1CCC(CCN(C(C(CC)OCC)=O)C)CC1 C1(C(=O)NCCSCC=C)CC1C1CN(C(C2CC(O)C(F)C2)=O)C1 N1(C(CCC=C)=O)CC2(CCNC(=O)CCCS(C)(=O)=O)CCC1CC2 CP(C)(=O)CCC(=O)Nc1cn(CC2N(CCc3cccc(F)c3)CCC2)nn1 CCCCCC(C)(C)C(=O)NC1CC(C(=O)N2CCCC2)=CC1O C1(C(=O)NCCc2c(C)ncs2)C2CN(C(C3CC(C(C)C)C3)=O)CC12 c1(C(=O)NCCCC(C)(C)NC(C2CC(CC)C2)=O)ccc2oncc2c1 Cc1cc(C(N2CC(C3(NC(c4nncs4)=O)CC3)C2)=O)c(N)c(F)c1 N1(C(CC2CC(OCC(=O)Nc3cn[nH]c3)C2)=O)CCC2(CCCOC2)C1 C1(C(=O)NCc2ccc(CNC(C3(CC#C)CCC3)=O)cc2)CC(C)CC(C)C1 Cc1cc(C=CC(=O)NC2(C=CC(=O)NCCc3cn(C)cn3)CCC2)on1 C1(C(=O)NCC2(CO)CC(C)(C)C2)(NC(CCCNC(C)=O)=O)CCCC1C C1(C(N2CC(N(C(CCS(=O)(=O)NC)=O)C)C2)=O)Oc2ccccc2OC1C c1(C(=O)OC)cccc(-n2cc(CC(C)NC(c3nn[nH]n3)C3CC3)nn2)c1 Cc1ccnc2nc(C(N3CC(CNC(=O)Cc4nccs4)C3)=O)nn12 C1(NC(CCCC)=O)CN(C(c2cc(C(F)(F)F)n(CC)n2)=O)C2(CCCC2)C1 C#CC1(C(=O)N(C)CC2CCOC2C)CN(C(=O)Cc2ccon2)C1 c1(NCCNC(c2c(CC=CCSC)nc[nH]2)=O)ncnc2c1COC2 c1(-n2cc(CN(C)S(N)(=O)=O)nn2)ccc(S(=O)(=O)C2CC2)cc1 C(C)(C)(CCCNC(=O)CC(O)Cc1ccccc1)NC(C(COC)C)=O C12(C(=O)OC)CC(COc3cccc(N4CCCC4)c3)(CO1)C2 c1(C(=O)NC2CC(O)CN(C(C3CSCCS3)=O)C2)c[nH]c2nc(F)ccc12 c1(C(N2CCC(CC=C)(NC(=O)CC3CC4CC4C3)C2)=O)cccc2c1OCC2 c1(C(N(CCNC(CCn2c(C)ncc2)=O)C2CC2)=O)csc(S(N)(=O)=O)c1 c1(C(N(CCNC(=O)C(C2CCCO2)OCC)CC)=O)cc(C)sc1S(N)(=O)=O Cc1[nH]nc2ccc(C(=O)N(C3CCCN(C(C4CC(C#N)C4)=O)C3)C)cc12 N1(C(C(c2ccc(F)cc2)C)=O)CCCC(F)(CNC(c2ccc(F)s2)=O)C1 C1(NC(C2(OC)CCOC2)=O)CN(C(=O)CCc2ncc(C)[nH]2)CC1C1CC1 CC1(C(=O)NC2CC2NC(c2cnn(C3CCC3)c2)=O)CCOC1 c1(-c2ccc(CC)s2)cc(C(=O)NCC2(CO)COC2)c2cn[nH]c2c1 CC(C)C(O)C(C)C(=O)N1CCCC(O)(CN(C)C(C2(C)CCOCC2)=O)C1 c1(C(N(C2CCN(C(=O)Cc3ccco3)C2)CC)=O)cncc(C)c1Cl C(CCS(=O)(=O)CC)N(C(=O)C=CS(C)=O)CC#C.C12CCN(CC1)C2=O C(=O)(C(C)(C)OC(=O)COc1ccccc1)OCC c1(C(N2CCC(NC(CS(CC)=O)=O)C2C)=O)cccc2c(C#N)c[nH]c12 c1(CC(N2CCCC(CNC(C(CCC)OCC)=O)C2)=O)ccc2occc2c1 Cc1cccc(C)c1CC(N1CC(OCCNC(C2CCCC(C)(C)O2)=O)C1)=O c1(C(CO)NC(C2CC(NC(C(n3ccc(C)n3)C)=O)C2)=O)cccc(Cl)c1 CC(C)(CC(=O)N1CC2CC2(NC(c2ccn(C3CC3)n2)=O)C1)C1CCCCC1 Cc1ccc(O)c(CC(N2CCCC(NC(C3CCCCC(=O)N3)=O)CC2)=O)c1 c1(OCC)ccc2cc(C=CC(C)OC)ccc2c1 C1(C(=O)NCC2CC3(CC3)CO2)COCCN(C(c2cc(Cl)cs2)=O)C1 C#Cc1ccc(C(=O)NC(C)C(C)NC(c2ccc(O)c(OC)c2)=O)nc1 N1(C(c2cn(CCCC)nc2C)=O)CC2CCC(NC(c3ccccn3)=O)(C2)C1 N1(C(=O)NC(c2cccnc2)c2ncc[nH]2)CCc2ccc(F)cc21 c1(C(N2CCN(C(=O)CCC3CCCO3)CC2CCO)=O)ccc2cccnn12 c1(C(=O)NC(CC)CNC(=O)CC2CC(=O)C2)ccnc(S(N)(=O)=O)c1 C#CCC(C)(C)C(=O)NC(C1CCCCC1)CNC(=O)CC(F)(F)F C1(O)(CC)CCCN(C(=O)C(=O)N(C)CCOc2ccc(C)c(C)c2)CC1 c1(N(C)C(C23COC(C)(C2)C3)=O)cc(Cl)ccc1S(N)(=O)=O CC1CCC(c2nc(CCN(C)C)nn2C(C(O)C(F)(F)F)C2CC2)CC1C c1(C(=O)NC2C(NC(C3N(C)CCCC3)=O)CCCC2)ccc2c(c1)COCO2 C1(CC)(CNC(C2CC3CC3N2C(=O)CCCCC2CC2)=O)CC(C)(C)C1 C(=O)(C1Cc2ccc(F)cc21)N1C(CNC(c2c(C)snc2)=O)CC(C)CC1 N1(C(C(CNC(c2cccc(F)c2F)=O)O)=O)CCCC2(CCC2)C1 Cc1cc(C(=O)N(CC(C)(C)NC(c2cnc(O)cc2O)=O)C)c(O)nc1C C(=O)(C(F)CC(CC)CC)NC1(C(=O)NCn2cnc(CC)n2)CSC1 CCCCN=C(NCC1CC12CC2)NCC1(O)CC2C=CC1C2 N1(C2CC(OCC)C2)CC2CCCC2(Oc2ccc(OC)cn2)C1.C(C)NC(=O)OC C1(CC(=O)NCC=CCC(N2C(CCC#C)CCC2)=O)CCC2(CC2)CO1 c1(C(N(C2CCC(NC(=O)CCc3ncco3)C2)C)=O)cccc(C=C(F)F)c1 N1(C(=O)C=C2CCCC2(F)F)CCCN(Cc2ccc(F)cc2)CC1 N1(C(C(C)N2CCCC2)=O)CC(C(=O)N(CC(C)(C)C)C)C(C)(C)C1 CCC(C)(CNC(C1CC(=C2CC2)C1)=O)C(=O)NC1(C2CCCO2)CC1 CC1CCC(CO)CN1C(C(=O)NCC(F)F)C(C)CC1CCC1 N1(C(C=CCCC(C)C)=O)CCC(NC(c2ccsc2C)=O)C(C)C1 CC(C)CC(C)CC(=O)N1CCN(CC(=O)NC2C=CCCC2CO)CC1 C1(CC(=O)N(CCNC(c2c(C)cccc2)=O)C2CC2)CCCC2(CC2)C1 Cc1cnn(C)c1C(=O)NC1CCOC1C(=O)NCC1=CCCOC1 c1(C(=O)NCCOC(CNC(c2c(CC)onc2C)=O)(C)C)cccc2ncnn12 N1C(=O)C(CC2CC2)N(C(O)(COC)C(F)(F)F)C1=O.c1(OC)ccc(C)cc1 c1(C(N2CC3(CC(CO)C3)C2)=O)ccc(NC2CC2)c(F)c1.C12(C(=O)N)CCC(C1)C2 C12(CNC(C3C(=C)CC3)=O)CC(NC(=O)C=CC(=O)OCC)(CO1)C2 C1(NC(=O)NCCCC)CN(C(C2CCCN(C(=O)C3CC3)C2)=O)CC12CC2 C#Cc1ccc(Cl)c(C(=O)NCC2CC2CNC(=O)CC2CCC2)c1 C#CC1(NC(C2C3CCC(C3)N2C(c2ccnnc2O)=O)=O)CCCOC1 C1(C(N2CCC(O)(C(C)NC(=O)C(F)=CC3CC3)C2)=O)CCc2nn(C)cc2C1 N12CCC(C)C(C1)NC(=O)C2c1cnc(CCCC)[nH]1.C(=O)(C(F)(F)F)NCC CCCN=c1nc(N2CCC(C3CCCCO3)CC2)c2ccccc2[nH]1 S(=O)(=O)(c1ccc(F)cc1F)N1CC2(CCN(C(=O)CN3CCCC3)C2)C1 c1(C(N2CCN(C(CNC(C(CC)C)=O)C)CC2)=O)cnc2cccnn12 C1(C(=O)NCC(C)N(C(C(N2CCSCC2)C)=O)C)CC(C2CC2)=NO1 C1(C(=O)NC2(C)CC(C(N(C3C(OC)COC3)C)=O)C2)NC(=O)OC1C C#CCC(CC(=O)N1CCN(C(=O)CCNC(c2scnc2C)=O)CC1)C1CC1 Cc1ccc(N(C)C)cc1.C12C3CN(CC13)C(=O)CCC(=O)Nc1nnnn1C2 C(=O)(C#CC(C)(C)C)NCC(c1cccc(OC)c1)NC(c1cnc(C)[nH]1)=O c1(C(N2CCC(CC)C2CNC(=O)Cc2nccn2C)=O)cccc(Cl)c1F c1(C(=O)NC(C(=O)N(C(C=C)C)C)Cc2ccco2)ccncc1F N1(C(C=C(C)Cl)=O)CCC2CCCN(C(=O)CCOc3ccc(C#N)cc3)C2C1 N1(C(C(CCC)C)=O)CCN(C(C2C3(CC3)C23CC3)=O)CC1CC(=O)NC c1(C(N2CCC(C(N(CCOC)Cc3ccco3)=O)C2)=O)ncccc1C N1(C(Cc2c(CC)con2)=O)CC(NC(c2nnn(CC)c2C)=O)C(C2CC2)C1 N1(C(c2cn(CCC)nn2)=O)CC2CC1C2C(=O)N(C)Cc1c(C)noc1C CC12CCC1CN(C(=O)C(Cn1cncn1)NC(=O)C=Cc1ccco1)C2 c1(N(c2cc(C)c(COC)cn2)C(c2cc(C)no2)=O)cc(F)c(Cl)cc1Cl C1(NC(C2C(C)C2)=O)CN(C(=O)Cc2ccccc2CS(N)(=O)=O)CC12CC2 C12(C(=O)NCC(C)CN(C(=O)CCCCO)C)CCCCC(=O)N1CCC2 CC(C)(C)CCCCNC(=O)C(N1CCOC(Cn2cncn2)C1)=O c1(C(c2n(C(CC)C)nnn2)NC2CCOC2C(C)C)nn(CC)cc1Br c1(C(=O)NCCN(C(=O)C(=O)NC2CC2)CCCOC)ncn(-c2ccccc2)n1 c1(C(N2C(CNC(C3CC(C#C)(O)C3)=O)CC2)=O)c(O)nnc(C)c1C C1(OC)CC2CC1CN(C(C1C(O)C(O)CN1C(=O)OC(C)(C)C)=O)C2 N1(C(c2cc(C(C)=O)on2)=O)CCN(C(C2CCOC2)=O)CC1c1ccccc1 CC(C)C(C(C)NC(c1nnn(-c2ccccc2)n1)=O)NC(c1c[nH]c(C#N)c1)=O CC1(C(N2CC(O)(CNC(c3cccnc3O)=O)C2)=O)CCCCC1 Cc1ncc(COCC(=O)N(CC(O)CNC(=O)C(O)c2ccsc2)C)s1 C1(CNC(C=Cc2cnc(C)s2)=O)CC2CCC(C1)N2C(=O)C(F)CC(C)C c1(C(=O)NCC(CC)NC(C23CC2CCC3(F)F)=O)cc2c(Cl)cncc2s1 CC(C)CCCCCC(=O)N1CC(CCNC(C2(CC(F)F)CC2)=O)OC(C)C1 c1(OCC2CCN(C(CC3CC(C(C)=O)C3(C)C)=O)CC2)ccc(F)cc1C C1(C(N(CC#CC)CC#C)=O)C2CC2CN1C(c1cnc(C)o1)=O c1(C(=O)NCc2c(CNC(=O)CC3(CO)CC3)cccc2)onc2ccccc12 C=CC(C)(O)CC(=O)NCC1(CNC(c2ncccc2F)=O)CCCC1 N1(C(CC23CC(C)(OC2)C3)=O)CCC(NC(c2c[nH]c(C#N)c2)=O)C2(CCC2)C1 c1(C(=O)NCCC(C)NC(CNC(CC(C)C)=O)=O)cc(Br)c(F)cc1N C1(CCNC(c2c(CC)nc(C)[nH]2)=O)CN(C(=O)COC2CCOC2)CCCO1 C(=O)(C(C)C(C)C)N(CCCN(C(C1C2CCCC12)=O)CC)CC C1(CNC(=O)C(C2CCOCC2)O)CC2CC2N1C(=O)CCOCC(F)F C1(C(N(c2ccc(F)cc2)C)=O)CN(C(=O)C=CC2CCOCC2)CC1F N1(C(C)=O)CCC(N(C(=O)COc2ccc(C(C)OC)cc2)C)CC1 N1(C(Cc2c(C)cco2)=O)CC(CNC(=O)C(C)(C)CC2CC2)CC1(C)C CC(C)(O)CC(=O)NCC1(CC(=O)NC2COCCOC2)CC1 N1(C(C(C=C)C)=O)CC(O)CC1CNC(=O)Cc1ccnn1C(C)C c1(-c2cccc(SC)c2)nn(C)c2cc(C(=O)NCc3ccncc3Cl)ccc12 CCCC(C)C(=O)NCC(F)CNC(=O)COCCc1ccc(Cl)s1 N1(C(C(C)N(C(C)=O)CCO)=O)CCC(F)(C(=O)NC(c2cc[nH]n2)C)CC1 C(C1CCCN1C(c1ccncc1CC)=O)=CC(=O)NC(C(=O)N(C)CC)C CCC(C)(COC)C(=O)N(C)CCN(C(C1(c2ccccc2)CC1)=O)C(C)C c1(OC)cc(-c2cn(CC(C)(C)C3CC3)nn2)ccc1O C1(NC(CSCCCCCCC)=O)C2CC(O)C1N(C(c1c(Cl)cnn1C)=O)C2 C1(CNC(c2ncc(OCC)nc2)=O)C(C2CC2)CCN1C(c1cncs1)=O C1(C(=O)OC)CCC(C(=O)SC2(c3cn(C4C(SC)COC4)nn3)COC2)C1 c1(N2CC(NC(C(C)(C)OC)=O)C(C#N)C2)ncc2ccsc2n1 CCCCC(CC)C(=O)N1CCN(C(c2cc(OC)c(C)c(OC)c2)=O)CC1 C(=O)(C(C)(C)CC(=O)NC1(C2CN(C(C3CCn4nccc4C3)=O)C2)CC1)OC c1(C(=O)NC(CNC(C2C(OC)CCC2)=O)C2CC2)sc2cncn2c1C N1(C(CCSCCC)=O)CC2(CCCN(C(=O)CCc3cccc(C)c3)C2)C1 C1(c2cn(CCC=C)nn2)CCCCN1C(c1cccn1C(C)C)=O c1(C(N(CCCCNC(=O)Cc2cnn(C)c2)C)=O)ccnc2c1CCC2 c1(C(C)C(=O)N(CC(O)CNC(c2coc(C(C)(C)C)n2)=O)C)ccc(F)cc1 CC(C)(F)CCC(=O)NCC1CN(C(=O)C(C)(C)c2ccccn2)CC1(F)F c1(C(=O)NC2C(CNC(c3c(SC)snn3)=O)C2)c(F)ccc2nc[nH]c12 Cc1sc(C)c(C(N2CC3CC(NC(c4cnn(C)c4C)=O)C3C2)=O)c1C#N CC1CCCCC1(C)NC(=O)C(CNC(C1CN2CCC1C2)=O)N(C)C N(C(=NCCc1nnc(CCn2ccnn2)s1)N1CCC(C(C)C)C1)C(C=C)C N1(C(=O)NCc2cccc(-n3c(C)ncc3)c2)CC2CC(O)C(O)CC2C1 c1(NC=O)ncncc1C.Cc1nc(C(CCS)NC2CC(N(C)C)C2)n[nH]1 c1(C(N2C(C)CCC(NC(c3ccc(F)c(N)c3)=O)C2)=O)coc2ccccc12 CC1CC(=O)NCC1C(=O)NC(C1(C(=O)NCc2cn(C)nc2C(N)=O)CC1)C Cn1cnc2[nH]c(C(=O)NC3CN(C(=O)CCCC4CC4)CC3C(F)F)cc12 N1(C(CN(C2CCC2)C)=O)CCC(C)(C)C(NC(c2n[nH]c3cccnc23)=O)C1 N1(Cc2cc3[nH]cc(OC)c3cc2)CC(C)NC(=O)c2ccc(F)cc21 C1(CNC(C(C(C)C)N2CCCC2)=O)Cc2ccccc2CO1.C12CC(C1)C2=O CCCC(CNC(c1sccc1Cl)=O)C(=O)NC(C)Cc1cn[nH]c1 N1(C(c2nccc(CC)c2)=O)CCC(F)(C(N2CC3CC2CN3C)=O)CC1 O=S(=O)(c1cccc(N2CCCC2)c1)N1CCNS(=O)(=O)CC1 O=C(C(O)CCn1cncn1)NC1CCCC1NC(c1cc(C2CCC2)[nH]n1)=O C1(c2n(C)cnc2)C(C(=O)NCC2(c3cccs3)CC2)CCC(=O)N1C1CC1 c1(C(=O)NCC2N(C(C(CC)(C)O)=O)C3CCC2C3)ccc(S(C)(=O)=O)c(Cl)c1 C12(CNC(=O)CSCC3CCCCO3)CC(C1)C(NC(C1CCC1)=O)CO2 C1(NC(C(C)O)=O)CCN(C(C23CC(C(F)F)(CO2)C3)=O)CC1O Cn1nc(C2CC2)cc1C(N1CC1CNC(=O)CCC1CCC(C(F)(F)F)O1)=O c1(C(N2CCCC2(C)C2CC2)C(=O)NCC)cc(Br)ccc1C N1(C(CSc2c(C)cccc2)=O)CC(C2CN(C(=O)C=CC3CCCO3)C2)C1 C1(N(C(CC2CCN(CC)C2)=O)CC(F)Cl)CC2(CCNCC2)C1 C1(C(N2C(C)(C)C(NC(c3cc(Cl)c[nH]3)=O)CC2)=O)CCc2cnnn2C1 C(N=c1cc(C(N)=O)nc[nH]1)C1CC2(CC(NC(C(C)OCC)=O)C2)C1 c1(CC)cc(C(=O)NCCC(CNC(=O)CC2CCN(C)C2=O)OC)ccn1 C(=O)(C(F)(F)C(F)(F)C(F)F)N1CCC2CN(C(C3CCCS3(=O)=O)=O)CC21 c1(OC)cc(C(C)ON2CCCC(C(C)=O)C2)ccn1 C1(C(=O)NC2(CO)CCN(C(=O)CCc3cncs3)C2)CC2CCC(C1)O2 N1(C(C(C)OCCN(C)C)=O)CC2(NC(=O)CCC(C)(C)C#N)CCCC2(F)C1 C1(CN(C(CCCOC)=O)C)CCN(C(=O)CCn2cc(Cl)cn2)CC1 C12(C(=O)NCC(C3CCCN3C(C3CC34CCC4)=O)(C)C)CCC(CO)(CC1)C2 c1(C(c2nnnn2C(C)C)NCCCOCC)cc(C(F)F)on1 N1(C(CCSC)=O)CCCCCCC1C(=O)N(C1COCC1O)CCC c1(C(=O)NCC2N(C(c3[nH]cc(C)c3)=O)CCN(C)C2)n[nH]c2c1CC1CC21 C(=O)(CC(C(F)(F)F)N(C)C)NC(c1ccccc1)C(C)NC(=O)C1=CCCC1 c1(C(=O)NC2CN(C(c3ccc(NCC)s3)=O)CC2C)c(OC)ccnc1O c1(C(N2CC(CCCCNC(=O)CC3CC=CCC3)C2)=O)nc(O)nc(O)c1F c1(C(=O)NCCN(C(C(C=C=C)C)=O)CC(C)O)cc(OC)ccc1C C1(C(=O)NC(C2CCOC2)CO)CN(C(c2cc(Cl)ns2)=O)C2(CCC2)C1 C1(C(N2CCN(c3cc(Cl)ccc3Cl)CC2)C(=O)NCC)CCOC2(CCC2)C1 c1(C(=O)NCCCNC(C2C(C)(CC)C2)=O)ccn2c(C)cnc2c1 c1(C(=O)NCC2C(NC(c3ccc(CC(C)C)c(N)c3)=O)C2)ccccc1S(C)=O c1(N2CCC(NC(C(C)CF)=O)C(C)(C)C2)ncnc2cccc([N+](=O)[O-])c12 C1(NC(c2cc(OCC)no2)=O)C2CC1N(C(=O)CC1CC=CCN1C)C2 C=CC(C)C(C)C(=O)NC1CCC(NC(c2cc(Cl)ncc2N)=O)CC1 Cc1ncccc1C=CC(=O)NC1(CNC(=O)CCn2cccc2)CCCCC1 C1(NC(CNC(CC)=O)=O)CN(C(=O)Cc2ccnc(OC)c2)CCC1CO C1(CCCCNC(C(C2CCC2)OC)=O)CCN(C(C2CC=CCC2)=O)CC1 C1(NC(C2(COC)CCOCC2)=O)CC2CC(C1)N(C(C1(COC)CCC1)=O)C2 Cc1nc(=N)[nH]c(C)c1C(=O)NCC1CCCC1NC(C1(O)CCC1)=O Cc1nc(C(C)C)sc1C(=O)NC1CN(C(=O)C(Cl)=CCl)C2CC12 c12nnc(C3CC3C)n1N2CC1(O)CC(OCC)C1.c1(SC)ccccc1 c1(CNC(CCCCF)=O)cn(Cc2ocnc2C(=O)O)nn1 C(CCCCC(=O)N1CC(NC(c2ncc(C(F)F)s2)=O)CC(O)C1)SC C1(C(CC)NC(=O)Nc2cnn(-c3cc(C)ccc3C)c2C)CCC(F)(F)CC1 c1(C(=O)NCCC(C)NC(=O)Cc2cc(C3CC3)no2)noc2ncccc12 c1(C(N2C3CCC2CN(C(C2(Cl)CC2)=O)C3)=O)cc2cccn2cn1 N1(C(C(C)OCOC)=O)CCOCC1CNC(c1cn(C2COCC2F)nn1)=O C=CC1OCCC1C(=O)N(CCN(C(=O)CCCc1nnc(C)n1C)CC)CC CCC(CC)C(F)C(=O)N1CCC2(NC(c3ccc(C(C)C)nc3)=O)CC2C1 C(CC(C)C(=O)N(C(CNC(c1cnc(C)nc1)=O)C1CC1)C)OC c1(CN2C(CNC(c3c(OC)c(Cl)ccc3)=O)CC2)cccc2cccc(O)c12 N1(C(CCc2onc(CSC)n2)=O)CCC(F)(CNC(C2CC(C)CO2)=O)CC1 C1(NC(c2c(C)ccn2C)=O)CCN(C(c2nn(C)c(Br)c2C)=O)C(C)C1 Cc1ccc(N(C)C(C2CC(NC(=O)C3=NOCC3)CCO2)=O)c(C)c1 CC1CN(C(=O)C(N)=O)CC(C)C1NC(C1(C(F)F)CC1)=O c1(C(=O)NCC(C)(O)CNC(=O)C=C(Cl)Cl)cc(Cl)cc2ccncc12 C1(N(C)C(c2cocn2)=O)C2CN(C(=O)CCc3ccc(O)nc3)CC12 C(C(C)(O)C(=O)NCC1(O)CN(C(=O)Cn2cnc(-c3nc(C)no3)c2)C1)OC c1(C(N2C3CC(CNC(c4n(CC)cnn4)=O)C2CC3)=O)nnc2ccccn12 N1(C(c2c(C)cc(Br)cc2)=O)CCN(C(C2(F)CC2)=O)C(C#N)C1 C1(NC(C(C)(O)C2CC2)=O)C2CN(C(=O)Cc3cccc(I)c3)CC12 c1(COC)ccc(C(=O)NC(C2CCOC2)CNC(c2ccnnc2O)=O)cc1 N1(C(CCCSC)=O)C2CCC1C(NC(=O)COc1ccc(C(N)=O)cc1)C2 CC1(C)CCCC(C(N2CC=CC2CNC(c2ccoc2C2CC2)=O)=O)CC1 N1(C(C(CCC)OC)=O)CCC2(C)CN(C(c3cc4cc[nH]c4cn3)=O)CC12 C1(C(N2CC(CN(C(C(=C(C)C3CC3)F)=O)C)C2)=O)Cc2ccncc2C1 c1(N(C(=O)NC2CC(C)(CC)OCC2)C)ccc2cnccc2c1 C(N=c1[nH]cnc(CC(C)C)c1CC)CNC(CCC(=O)NCC)=O.C1C(=O)O1 CCC(C(=O)N1CC(CNC(C2CN(CC)CCO2)=O)OC(C)(C)C1)C(F)(F)F c1(C(=O)NC2CN(C(C(P(C)(C)=O)O)=O)CC2O)cnc2ccnn2c1 c1(CC)[nH]nc(C(N2CC(OCCNC(C3CCCCN3)=O)C2)=O)c1Cl c1(C(N2CC(O)(C(C(=O)NCC3CCCCCC3)F)C2)=O)nnc(O)nc1O C12CN(CCO1)C(=O)CC(C)NC2=O.c1(CC)cc(O)ncn1 N1(C(C2C(=C)CC2)=O)CCC2(COC(CNC(C3CS(=O)(=O)CC(=O)N3)=O)C2)C1 N1(C(C(CSC)C)=O)CC2C(NC(=O)CCc3csc(C(F)(F)F)n3)C2C1 Nc1cc(C(N2CC(C3(NC(c4ccoc4)=O)CC3)C2)=O)cc(O)c1Cl N1(NC(N(C)CCc2cn[nH]c2)=O)CCN(CCNC2CCC2)CC1 n1(CCC(=O)NC2C(NC(C3(S(C)(=O)=O)CC3)=O)CCC2)ccc(O)nc1=O CCC(CC(=O)NCC(C)(C)CC(=O)NC1(C2CCCC2)CC1)C(F)F C(C1CN(C(c2ccc(O)c(F)c2)=O)CC1C(=O)NC(C)(C)CCCF)=CC c1(C(=O)NCC2N(C(=O)CC3CC3(C)C)CCN(C)C2)ccc2c(c1)N(C)CC2 c1(C(=O)NCC(C)(C(C)C)NC(C(C)=C2CC2)=O)ccc2c(c1)NC(=O)CCS2 c1(C(N2CCN(C(C=C(COC)C)=O)CC23CC3)=O)ccc2c(c1)CCCO2 c1(CNC(C2C(C(C)NC(CC)=O)C2)=O)nccn1CC.C(N)(=O)N C=CCCC(F)(F)C(=O)NCCCC(C)NC(C1CCCS(=O)(=O)N1)=O CC(C)C(C(=O)N1CC(O)(C(C)NC(=O)C2=CCSC2)C1)N1CCCCC1 Cc1nn(-c2ccccc2F)c(C)c1CC(=O)N(c1cccc(O)c1)CC(C)C CC1=NS(=O)(=O)NC(C)=C1CC(=O)N1CCCC1c1cn(CCOCCO)nn1 N1(C(CN(CCOC)C)=O)CCOCC1CC(=O)N(C1CCCCO1)C c1(CCC(N2CCN(C(CCC=C)=O)CC2C)=O)ccc2ccn(C)c2c1 C1(CNC(c2ccc3c(c2)COC3)=O)CCC12CCN(C(C1SCCS1)=O)CC2 c1(CCNC(c2c(C)n(-c3ccccc3)nc2)=O)nnc2c(=O)n(C)ccn12 C1(NC(=O)Cn2cnnc2)CCN(c2cc(C(F)(F)F)ncn2)CC1O c1(C(N2CC(C)(CCC(=O)NCCOC)C2)=O)ccc2nc[nH]c2c1 C1(NC(c2n(C(C)C)cnc2)=O)CN(C(c2cc(Cl)no2)=O)C2CC12 C1(C(N(CCn2cc(Cn3ccnc3)nn2)CC)=O)CCc2c(ccnc2C)C1 CC1CC(=O)Nc2c(F)cccc2N1C(=O)CNS(=O)(=O)c1cn(C)nn1 CCC(C)(C)C(O)C(=O)N(CCN(C)C(c1cnn(C(C)(C)C)c1Cl)=O)C(C)C C1(CCC=C)(C(=O)OCCl)CN(C(c2cnnn2C)=O)C1.C1CCN(C(C)=O)C1 CCC(C)C(C)C(=O)N1CCCC1CNC(c1cccc(C(C)C)c1)=O CCCC(C(=O)N(C)C)NC(=O)C(COC)NC(=O)C(O)Cn1cncn1 Cc1nn(C(F)F)c(C)c1CC(N1CCC(C)C1CNC(=O)C(Cl)=CCl)=O c1(CC)noc(C(=O)NCCOC2CCN(C(C3CCC(=O)N3)=O)C2)n1 C1(CNC(CN(C)CCO)=O)CC12CCN(C(=O)C(F)(F)C1CCOC1)CC2 CC1(C)CCCN(C(C2CCSC2)=O)C1C(N1CC(S(N)(=O)=O)C1)=O C12CC(CN1C(=O)OC(C)(C)C)NC2=O.C(=O)(CCOC)NCCOC.OC C1(NC(COCC#C)=O)CCC2(CC1)CN(C(C1CCCC(O)C1)=O)C2 C1(CC)CN(C(c2ccoc2Cl)=O)CCC1NC(c1conc1C1CCC1)=O c1(C(N(CCCCNC(C2N(CC)CCC2)=O)C)=O)c[nH]c2nc(Cl)ccc12 c1(N(C)C)ccc(C(=O)Nc2nnc(-c3ccc(F)cc3)o2)cc1[N+](=O)[O-] c1(CC)occc1C(=O)NC1CCN(C(=O)CC(C)OC)C1 c1(OC)ccc(NC(c2nnnn2C2CC2)CCC2(C)CC2)cc1C(F)F C1(CNC(c2cnc3[nH]cnc3c2)=O)CC2CCC(C1)N2C(c1occc1Br)=O c1(C2(C(=O)NC3(C(N(C4CCCC4(C)O)C)=O)CC3)CCC2)ccncc1Cl N1(CC(=O)NCc2c(C(N(C)Cc3n(CC)ccn3)=O)con2)CCNC(=O)C1 N1(C(Cc2nc(=N)[nH][nH]2)=O)CCC(NC(C2CC(F)C(=O)N2)=O)C(O)C1 C(C(CO)(CO)c1nn[nH]n1)NCC(N1CCCS1(=O)=O)(C)C C=C(C)CN=C(NCc1ccc(F)cc1)NC(C1CC1)C1CC1 N1(C(N(c2cccc(C3CC3(F)F)c2)C)=O)CCCOC(CN=[N+]=[N-])C1 N#CC1CCN(C(c2cncc(-c3cnn(C4CCCCO4)n3)n2)=O)C1 C(N=c1[nH]c2ncnc-2c(NC(C)C)[nH]1)C1(O)CN(C(C(C)NC(CC)=O)=O)C1 C1(NC(C(C2(O)CN(C(CCC(=O)NC)=O)C2)F)=O)CCc2nncn2C1 C1(NC(C(CC)C(C)(F)F)=O)CN(C(=O)C=C(C)Cl)C2(CCCC2)C1 C1(C(=O)NCCN(C(=O)C(C)C(C)O)C(C)C)CCC(C)(F)CC1 c1(C(C(=O)N(CCCCN(C(=O)C2=CSCS2)C)C)(C)C)ccc(F)c(F)c1 C1(C(=O)NC2(CC)CCN(C(C3CC(C)(C)C3)=O)CC2)CC12CCC(F)(F)CC2 Cc1cccnc1C=CC(=O)NCC1CCC(NC(=O)CSc2cnn(C)c2)C1 c1(C(=O)NCC(C)(CNC(=O)C(O)CCC(C)C)OC)cc(F)c(C)cc1F C1(CNC(=O)COCC2CCCO2)CC2(CCC2)CN1C(C1CC12CC(O)C2)=O c1(C(N2CCC(O)C(C)(C)C2)C(=O)NCCOCC)ccnc2ccccc12 Cc1cccn2cc(C(=O)NCC(C3CC3)N(C(=O)CO)C)nc12 c1(C(N2CCCC(NC(C(CC)(CC)CO)=O)C2)=O)cc2ccccc2nc1C c1(C(N(C2CCN(C(=O)C3CC3)C2)CCC)=O)coc2c1N(C)C(=O)CCC2 C#CCC(C)C(=O)NCCCCC1(NC(=O)CCc2csc(=N)[nH]2)CC1 N1(C(C2N(C)CCOC2)=O)CC2CC(NC(C3CNC(=O)N3)=O)CC1C2 C1(OC)CN(C(=O)C2=C(C)CC2)CCC1NC(=O)CC1COC(=O)C1 C1(NC(C2(CSC)CC2)=O)COC2(CCN(C(=O)C=C3CCC(C)CC3)C2)C1 N1(CC(=O)NCC2CCN2C(=O)Cc2cnco2)CCCCS1(=O)=O N1(C(c2ccc(C(C)C)cn2)=O)CCC(NC(c2nnc(S)n2C)=O)C(C)C1 C1(C(=O)NCC(C)(C)NC(C)=O)CCN(c2ccccc2)S1(=O)=O N1(c2cc(C(C)=O)ncn2)CCC(C)C(NC(=O)Cn2nc(Cl)ccc2=O)C1 CCC(CC1CCC1)C(=O)NCC1CC(NC(C2CC2c2cccs2)=O)C(O)C1 C12(CNC(C(C)(CO)OC)=O)CC(CO1)N(C(=O)CC1(CN(C)C)CCC1)C2 Cn1cc(C(=O)NC2CCC2NC(=O)CCc2csc(=N)[nH]2)c(Br)n1 N1(C(c2ncc(C)c(C)c2)=O)C2CCC1CC(NC(C1CCN(C)C(C)C1)=O)C2 c1(-n2cc(CNC(CC3C=NN(C)C3=O)=O)nn2)cccc2ncoc12 C12(C(N3CC4CC(C)C4C3)=O)CC(CCO1)N(C(C1CCCC3(CC3)C1)=O)C2 N1(C(C(C)NC(CC)(C)C)=O)CCC(CO)(NC(c2cc(CF)on2)=O)CC1 N1(C(=O)OC)CCC(NC(=O)CN2CCC(Cc3csc(C(C)C)n3)C2)CC1 c1(-c2cn(C3C(C)CN(C(=O)COC4CCOC4)C3)nn2)ccc(Cl)c(F)c1F C(C(=O)NCC(O)CNC(=O)CCC1CCCCC1)(C(C)(C)C)N(C)C c1(C(N(CC(=O)NCC2(CN(C)C)CCC2)C2CC2)=O)ccc(F)c(O)c1 C(=O)(CC(C)C(C)(C)C)N1CCC(C=C)(C(=O)NC2CN(C)CC2C)C1 N1(C(C2(C)CCOC2)=O)CCC(C2CN(C(=O)CC3=NNC(=O)C3)C2)CC1 N1(C(c2cc(C)cc(O)c2)=O)C2CCC1C(F)C(NC(=O)CNC(=O)C1CC1)C2 C1(CC)C(C(=O)NCC(C)CCCO)CCCN1C(C1CC(CC2CC2)C1)=O CCCC(C)C(=O)N1CCCC(CNC(=O)C(C)COC)C1 N1(C(CCCOCC=C)=O)CC=C(CC(=O)NCC2(C3CC3)CCC2)CC1 C1(CNC(C(CC2CC2)OC)=O)C2CN(C(=O)C(C)(C)NS(C)(=O)=O)CC12 N1(C(c2cn(C(C)(C)C)nn2)=O)CCC(F)(CNC(C2CC(=O)CO2)=O)CC1 N1(C(CCc2scc(C)c2)=O)CCC2CCN(C(=O)C(C)Cc3ccco3)CC12 N1(C(C=CC(C)C)=O)CCC(N(C(=O)Cc2ccccc2Br)C)C(C)C1 N1(C(CCOCC(C)C)=O)CCN(C(C2CC2(C)Br)=O)CC1CCO C(=O)(CCC(C)(C)N1CCOCC1)N(CC(C)NC(=O)C(C)N=[N+]=[N-])CC CCC(CC(F)(F)F)C(=O)N1CCC(F)(CNC(=O)COC2(C)CCOCC2)C1 C1(CC(=O)NOC2CCC2)CN(C(=O)CCC2CCCO2)CC12CC2 N1(C(c2ccc(C(=O)OC)o2)=O)CCC2CCN(C(=O)Cc3csc(Cl)c3)CC12 C=CCCCCCCCC(=O)NCCC1=CCN(C(=O)C=Cc2ccoc2)CC1 N1(C(CCC(=C)C)=O)CC2CC(N(C)C(C3CCCC(C)(C)C3)=O)C1C2 C1(CCC)CN(C(=O)C(Cc2ccco2)NC(c2cc(Cl)no2)=O)CCO1 CC1(C)CCOC(CC(N2CCC(CNC(=O)CC3CC(F)C3)CC2)=O)C1 N1(CC(c2c(C)ccc(C)c2)=O)C2CCCC1CC(O)C2 C1(C)(C(=O)CCNCC(=O)NCCC2CC(NC(=O)OC)C2)CCC(C)C1 N1(C(c2cc(C)no2)=O)CCOCC(CNC(C2CC(C#N)C2)=O)C1 C1(O)(CC#C)CC(C(N2CC(CNC(c3sccc3C(C)=O)=O)C2)=O)C1 c1(C(N)=O)nccc(C(=O)NC2C=CCN(C(C3COCC3C(N)=O)=O)C2)n1 C1(C(=O)NC(CC)CN(C)CC)CC(NC(c2csc(C#N)c2)=O)CCO1 N1(C(Cn2nnc(C)n2)=O)CCCN(C(c2ccc(C(C)(F)F)cn2)=O)CC1 c1(NC(C2COCCN2Cc2ccncc2)=O)nc2cc(Cl)ccn2n1 C1(Nc2nnc(C3(OC(C)C)CCC3)o2)C2CCC1(C)C2(C)C c1(C(C)C(=O)NCCCC2CCCN2C(=O)CCCCCF)ccc(C#N)cc1 N1(C(c2c(C)con2)=O)CCC2CC2(NC(c2cncs2)=O)CC1 C1(NC(C(CN(C)C)(C)C)=O)C2CC3C1C3C2C(=O)NCC1CCCC(CO)C1 C#CCCN=C(NCc1c(Br)nnn1C)NCC(c1ccc(F)cc1)O Cc1nn(C)c(C)c1C(O)CNC(=O)C(=O)NCC1CCNC1 N1(C(=O)Cn2cc(CSCCO)nn2)CCC(C2CCCC2)C1 c1(C(=O)Nc2ccc(C(=O)OC)cc2)c(C)cc(Br)cc1C.C12CC1O2 N1(C(C(C)OCCC#C)=O)CC2CN(C(c3c[nH]nc3C(C)C)=O)CC2C1 C1(C(N2CCC(CN(C)C)CC2)=O)CN(Cc2ncc(Br)cc2F)CCC1O C1(OC)CCn2cc(C(=O)NC(C)CNC(=O)CCc3c(C)noc3Cl)nc2C1 N1(CC(N2CCC(N(C(=O)Cn3ncc(Br)n3)C)C2)=O)CCCNC1=O N1(C(C(N2C(CC)CCC2)=O)=O)CCN(CCCS(=O)(=O)N2CCCCC2)CC1 C(CCC(C)C(=O)N(C)CC1CN(C(c2ccc(COC)o2)=O)C1)OC C1(NC(Cc2cccc(SC)c2)=O)CCN(C(=O)CC2CCCN(C)C2)C(C)C1 N1(C(c2cncc(C)c2C)=O)CC(F)(F)CC1(C)CNC(=O)Cc1cscn1 O=C(CCN1C(=O)COc2ccccc21)N1CC2(CCC(NCc3cncs3)C2)C1 C=Cn1nccc1C(=O)N(CC(=O)NC(C)CC(C)(C)OC)CC(C)C c1(C(=O)NCCC(=C)CNC(=O)CCn2cc(C)cn2)cccc(C(N)=O)n1 C(CCCCCCC(=O)NCC1CN(C(C2CCCCO2)=O)C(C)(C)C1)SC C1(CN(C(=O)CC(O)C2CC2)C)CCCN1C(c1ccnn1CC(F)F)=O N1(C(c2ncn(C)c(=O)c2)=O)CCC2CC2(C(=O)NC2CCCC2)CC1 CC(O)CCCN=C(NCC1CCC1)NC1CC1C(F)(F)F CC(C)(C)C(CO)C(=O)NCc1nc(C(=O)NC2CN(c3ncco3)C2)co1 Cn1cc2cc(C(N3CC4(NC(=O)CCCN5CCCC5)CC3C4)=O)ccc2n1 N1(C(c2ccc(Cl)cc2Br)C)CCc2c(cnn(C)c2=O)C1 C1(CC(N2CCC(C)(NC(=O)C3=CCSC3)C2)=O)CCCC2(CC2)C1 c1(C(=O)NCCCCN(C)C(c2cc(C(N)=O)[nH]n2)=O)csc2ccccc12 N1(C(C(CC#C)C)=O)CCC2C(CCCN2C(=O)Cc2ccc(OC)cc2C)C1 C(c1ccc(F)cc1)=C(C(=O)N(CC(C)CNC(C1(C)CC1(F)Cl)=O)C)C#N C1(C(=O)NCc2cc(C(C)C)no2)CCCC(CNC(=O)C(F)F)C1 O=C(N=c1[nH][nH]c2c1CN(Cc1cc3ccccc3[nH]1)C2)C1=NOCC1 C1(NC(CS(N)(=O)=O)=O)CCC12CN(C(c1cccc(-c3ccncc3)c1)=O)C2 C1(CC(=O)N(CCNC(c2ccccc2)=O)CC)CCC(=O)C1C C=CC(CC)C(=O)NC1CC(CCNC(C2CC=CCC2)=O)C1 C(CC(=O)NCC1CC2C=CC1O2)(C(F)(F)F)NC(=O)OC(C)(C)C c1(CC(N2CC3C(CNC(Cc4n(C)nnc4)=O)C3C2)=O)c(Cl)cccc1Cl N1(C(CN(C(C)=O)CC)=O)CCc2c(ncn2C2CCCN(C(C3C=C3C)=O)C2)C1 N1(C(Cn2c(C)ncc2C(F)F)=O)CCN(C(=O)COC2CC2)CC(CO)C1 C(=O)(C1CNS(=O)(=O)c2ccccc21)NCC1CC(NC(C(C)CC(N)=O)=O)C1 C1(CCNC(C(CCC)C)=O)CN(C(c2nnc(C(F)(F)F)s2)=O)CCCO1 C(=O)(C1CCC(=O)c2ccccc21)NC1CC(NC(C2(OC)CCC2)=O)C1 c1(C(=O)OCC)c[nH]ccc1=NC1CCCC1NC(=O)CCC1CCC(=O)N1 CC1(CCNC(=O)C(CC2CCC2)NC(=O)CN2CCCCC2)CCCO1 C#Cc1cncc(C(N2CC(OCC(=O)NCc3cccc(C)c3F)C2)=O)c1 CCC(CC)C(C)C(=O)NCCCN(C(=O)C=CSCc1ccco1)CC C1(NC(c2cc(C)sc2)=O)CCN(C(=O)CNc2c(C)occc2=O)C1C1CC1 C12(CNC(COCCN(C)C)=O)CC1CN(C(=O)C(=O)NCC(F)(F)F)C2 C1(C(C)C)CCCN(C(C2C=CCN2Cc2sc(Cl)nc2Cl)=O)C1 C12(C(=O)Nc3ccc(F)nc3)CCC(CN(C(c3cnc(C4CC4)o3)=O)C1)C2 CC(C)C(CC1CCCC1)C(=O)N1CC=C(CNC(=O)C(C)c2cc[nH]n2)CC1 Cc1nc(CC(=O)NCc2ccccc2CNC(=O)CC2CCOC2=O)nn1C n1(CCN(C)Cc2cn(CC3(F)CCC(C(=O)O)C3)nn2)nc(O)ccc1=O Cc1c(C(=O)NC2CC2NC(c2nnsc2C(F)F)=O)cccc1N C1(CNC(CC2C(C)CCO2)=O)CC2CC1CN2C(c1cc(C2CCC2)on1)=O C1(C(N2CC(n3cc(CC4CC(C(C)(C)O)C4)nn3)C2)=O)CC2(CCCC2)CO1 N1(C(C2(C)CCCN(C(C3N(C)CC(C)(C)C3)=O)C2)=O)CCCC12CCNC2=O CC1COCC1(c1nnnn1CC1CCOC1)NCC=CCl C#Cc1ccnc(C(=O)NC(C(=O)NCc2ccsc2)C(C)(C)C)c1 C1(C(N2CCC(CCNC(c3cn(CCCF)nn3)=O)C2)=O)CC12CCOCC2 C1(C(=O)NCC(CC)NC(c2ccc(N)c(O)c2)=O)Cc2nnsc2S1 c1(C(=O)NCCN(CCC)C(C2CCC(=O)O2)=O)nccc2cccnc12 C1(CC(N2CC(COC(C)=O)C2)=O)CCCN(C(c2cc(C)c(C)[nH]2)=O)C1 c1(C(C(=O)N(C)CC2CC2(C)C)NC(=O)COC2(C)CCC2)ccnn1C N1(C(Cn2c(C)ccn2)=O)CCOCC(CNC(=O)CCCC(F)F)C1 C1(CNC(c2c(C)nn(CCO)c2C)=O)N(C(=O)C2=CCCO2)CCCC1(C)C c1(CC)ccc(C(=O)NCCC2(O)CN(C(=O)CC3(C)CCCO3)C2)s1 N1(C(CC2C(CNC(C3(Cl)C(C(C)=O)C3)=O)C2)=O)CCN(C(C)C)CC1 C1(C)(CNC(C(CC=C)NC(C)=O)=O)CCCN(C(=O)C(O)CF)C1 N1(C(c2c(C)noc2C)=O)CCCC(NC(c2cnc3[nH]cnc3c2)=O)CCC1 N1(C(Cc2c(C)noc2C)=O)CC2CCCC2(C(=O)Nc2cnn(C)c2Cl)C1 C#Cc1ccc(C(=O)NCC2CCC(C(=O)NCc3csc(C)c3C)O2)cn1 Cc1ncc(C(=O)NCCCNC(C2CC2NC(=O)OC(C)(C)C)=O)[nH]1 c1(CNC(C2(OC)CCN(C)C2)=O)cc(C)cnc1O.c12cc[nH]c1C(=O)NC2 Cc1cc(C(N2CCC(CCNC(=O)CC(C)C3CCCCC3)C2)=O)ns1 N1(C(C(C)CCC(C)(C)C)=O)CCCC(N=c2[nH]c3ncc(Cl)cc3s2)CC1 c1(C(=O)NC23CC(CNC(C(CC)C)=O)(OC2)C3)cc2cccc(C)c2o1 C1(NC(CCCOC)=O)CC(O)CN(C(c2csc(-c3ccc(Cl)s3)n2)=O)C1 C=CCC(CNC(=O)C(c1cnccn1)C)NC(=O)CCCOC1CCOCC1 N1(C(COCCOC)=O)CC(CNC(=O)C(C2CCOCC2)C)C(C)C1 C1(S(N)(=O)=O)(C(=O)NCCC2(NC(C3(C)CCN(C)C3=O)=O)CCC2)CCCC1 c1(SCC(N)=O)ccccc1C(=O)NCC1COCCN1C(C1COC(=O)N1)=O CC1CC(C(=O)NC2CC(F)(CNC(=O)C(C)CSC(F)(F)F)C2)=NO1 N1(C(CNC(=O)NC)=O)CC(CNC(c2csc(Cl)c2)=O)OC(C(F)(F)F)C1 Cc1c(C(=O)N(CC(C)CNC(c2cnn(C(C)C)c2C)=O)C)cnn1C1CC1 N1(C(c2ccn(-c3cccc(F)c3)n2)=O)CC2(CCN2C(c2n[nH]cc2F)=O)C1 CC1(C)C=C(C(=O)N2CC(CNC(=O)Cn3cc(C4CC4)nn3)CCC2C)C1 c1(C(N2CC(CC(C)NC(CC=CC=C)=O)C2)=O)cc([N+](=O)[O-])ccc1SC c1(C(N2CC(N(C)CCO)C(C(F)F)C2)=O)ccc(Cl)nc1OC CC1CCC(C(N2CC(N(C(=O)CC3OCCCO3)C)C2)=O)CC1 CC(C)C(F)C(=O)N1CC2CC1(C(=O)NC1CCCCC1)C2 c1(CC(=O)NC(C)CC2CN(C(=O)C(C)C3CCCC3)C2)ccc(C)o1 Cn1cc(C(=O)NC2CC(CNC(=O)Cc3c(Cl)cnn3C)C2)c(O)n1 N1(C(C(CC)n2cccn2)=O)CCC(C)(NC(c2ccnnc2O)=O)CC1 c1(NC(c2c(CNC(C3(CC)CC3)=O)c[nH]n2)=O)nc2c(C)c(Br)ccc2s1 C1(C(C)C)CCc2sc(C(=O)NC(C)(C)CC3CCC3)cc2C1 C12(CNC(c3cc(C)[nH]n3)=O)CCCN(C(c3cc(Cl)cn3C)=O)C1C2 C1(NC(C=C2CCC(C)C2)=O)CN(C(=O)CN2CC=CC2)C2(CCCCC2)C1 N1(C(c2cccc(OC)n2)=O)CCCC(NC(c2cnoc2C2CC2)=O)CC1 CC1CC(C(=O)NC2CC3CCC2C3)N(C(=O)CCOCC2CC2)C1 c1(C(=O)NCC(c2ccncc2)O)cc2cccc(F)c2s1 c1(-c2nnc(C3CCCS3)[nH]2)cc(-c2ccncc2)cc(SC)c1.CCOC n1(CC)nc(C(N2CCC(N(C(=O)CC3(O)CCC3)C)C2)=O)cc1C c1(C(=O)NC2C(NC(C=CSC)=O)COC2)cccc2nc(O)n(C)c12 Cc1ccc(CN2CCC(CCC(N3CCC(n4ccnc4)C3)=O)CC2)nn1 c1(C(=O)NCC(=O)NC2CC(OC)C2)cccc(NC(C2CCCCC2C)=O)c1 C(=O)(CC(F)(F)C(F)F)N1CCC(CCC(N2C(C)C(=O)NCC2)=O)C1 c1(C(=O)NCCCN(CC#C)C(C2CC2=C)=O)cccc2ccnn12 C(C1=NOC2CN(C(c3ncc(C4CC4)s3)=O)CC12)NC(c1cccc(F)c1)=O c1(C(=O)NCCCCC(C)NC(=O)CC2(C)CC2)cnn2ccncc12 C1(NC(C2N(CCC)CCCC2)=O)C2CC3C1C3C2C(=O)N(CC)CC1CCC1 CCC(C)(C(=O)N1CCC(Cn2cc(-c3ncoc3C)nn2)C1)C(N)=O N1(C(COCCCC(C)C)=O)CCCC(CC(=O)NCC2(CCO)CC2)CC1 C=CC1(C(=O)NCc2ccccc2C#N)CCN(C(c2cnn[nH]2)=O)C1 N1(C(c2n3nc(c2)C3)=O)CCC2CCN(C(=O)CC3CC3)C2C1.CC(O)C1CC1 c1(COC)nn[nH]c1NC(C1(C(N)=O)CN(C(c2nocc2Cl)=O)C1)=O N1(C(C(C)=CC)=O)CC(C2CCCN(C(C3CSc4ccccc4O3)=O)C2)C1 N1(C(CCc2onc(CC)n2)=O)CCC(NC(c2ccnn2C2CC2)=O)C(C)C1 C1(NC(C2CCN(C)C2)=O)CN(C(=O)CC2(C#N)CCOCC2)CC1(C)C CCCCC(CC)N=c1[nH]c(NC2CC(Cl)(Cl)C2)nc2ncn(CC)c12 c1(CC(=O)NCCN(C2CCCCC2)C(C2CC3CC3C2)=O)cc(CO)on1 c1(OC)cc(NC(=O)COC(C)C)cc(OC)c1OC.C1(=O)CC(C)N1 c1(C(N2C3C(C(=O)Nc4cn(CC)nc4)C(C3)C2)=O)ccccc1C#N C=CCC(CNC(c1ccns1)=O)C(=O)NCC1CC2(CCO1)CC2 N1(C(c2ccc(C(C)O)cc2)=O)CCC2(CCCN(C(C3CCC(C)C3)=O)C2)C1 c1(C(C(=O)NCC)N(CC(=O)N(C)C)Cc2ccco2)cnc(C)n1C N1(C(CC(C)=C(C)C)=O)CCC(F)(CNC(C2(C3(C)CC3)CC2)=O)CC1 N1(Cc2ccc(C)[nH]2)CCC2CC(C(=O)Nc3cc(Cl)ncn3)C2C1 C1(NC(c2c(C)c(Br)ncc2)c2nnnn2C(C)(C)C)CC2CCCC(C1)C2 C=CC1(C(=O)NCCc2csc(C)n2)CCN(C(=O)CC2(O)CCCOC2)C1 C(=O)(CCCNC(=O)CSC(F)(F)F)N1CC(CC(C#C)C)C1 Cn1cc(C(N2CCCC(NC(C3C4CC5C(C4=O)C35)=O)C2)=O)c(O)nc1=O c1(C(N(CCNC(c2cncc(C(=O)OC)c2)=O)CC)=O)cnc2n1CC(C)CC2 n1(CC(=O)NCC(C)NC(c2c(C(=O)OC)scc2)=O)nc(C)c2cccnc12 N1(C(c2cnc(COC)s2)=O)CC(NC(C2CCCO2)=O)C(F)C1 Cc1ccc(Cl)cc1CN1CCC(C(O)C(F)(F)F)CC1 C1(C(N2CC(OCC(=O)NC)C2)=O)CCCN1C(=O)CSc1cn[nH]c1 Cc1ccc(CC(N)CC(=O)NCCNC2CCCN(C)C2)c(C)c1 C(C)(CCCCNC(=O)CCn1cccn1)NC(CCCn1ncc(C)c1)=O c1(COC)cc(C)cc(O)c1.C12CCCCC1NC(=O)C1(CC(=C)C1)C(=O)N2 c1(OCC)cccc(C(=O)NCCN(C(=O)C#CC(C)C)CC)c1[N+](=O)[O-] c1(OCC(=O)N(C2CCN(C(C3CCCC34CC4)=O)CC2)CC)cncc(Cl)n1 N(C)(C1CCc2ccccc21)C(C(CC)CC)C(=O)NCCC#N N1(C(CNC(C)=O)=O)CCN(C(C23CC(CO2)C3)=O)CC1c1ccccc1Cl C#Cc1ccc(Br)c(C(=O)NCC(C)(C)NC(C2CCC(C)O2)=O)c1 N1(CCN2CC(C(C(=O)OC)N(C(C)(C)C)CC)C2)CCN(C2CCOC2)CC1 N1(C(c2c(C)[nH]nc2Cl)=O)CCC(CCNC(c2ccc[nH]2)=O)CC1C Cc1cccc(OCC(=O)NCC(C2CCCC2)NC(=O)CCC2CC2C)c1 N1(C(c2c(C)nc(O)cc2)=O)CCC(C2CCN(C(=O)CCP(C)(C)=O)C2)C1 C1(NC(CN(C(C)=O)C)=O)CCN(C(c2cnsc2)=O)C(c2ccccc2)C1 c1(C(N2CC(C(C3(N)CCCC3)C)C(c3ccccc3)C2)=O)cc2c[nH]nc2cn1 Cc1c(C=CC(N2CCN(C)C(C(=O)O)C2)=O)cnn1C S(=O)(=O)(c1cccs1)NCCC(=O)N(CCNC(=O)CC1CC1)CC1CC1 c1(C2(C(=O)NCC(C)N(C(c3c(C)cco3)=O)C)CCCC2)ccc(F)cc1 C1(CC)CN(C(=O)C(C2CC2)N(C)C)CCC1NC(=O)C=CC1CC1 N1(C(C=NOC)=O)CCCC(NC(=O)CSc2c(C)cccc2C)C(F)C1 c1(CC(=O)NC(CCN(C(c2c(CC)c[nH]n2)=O)C)C)cc(Cl)sc1Cl C(=O)(CC(O)C1CCCC1)NCC1C(CC(=O)NCCc2cnn[nH]2)C1 C#CCC(C(=O)NCCCC1(O)CCC1)NC(C12CC(CO)(C1)C2)=O c1(C(=O)NC(CC=CC)C(N2CCN(C)C(C3CC3)C2)=O)cc(N)cc(F)c1 CC(C)(F)CCC(=O)N1CCCC(n2cc(-c3csc(Br)c3)nn2)C1 C(=O)(C(F)(F)CCc1ccccc1)NCC(CNC(=O)C(Br)=C(C)C)OC c1(CC)cc(C(=O)NCC2(OC)CN(C(=O)CC3CS(=O)(=O)C3)C2)n[nH]1 C1(CC(=O)NCc2cc(Br)ccn2)CCN(C(c2ccc(F)nc2)=O)CC1 C(CN=c1nc2scnc2c(NC2CC(C)(C(N)=O)C2)[nH]1)C1COCC(C)O1 N1(C(CC2C(C)CC2)=O)CCC2(CC2NC(C2CC23CC3)=O)C1 C(CCN=c1nc(N2CCOCC2)cc[nH]1)NC1CC2C(O)C(CCC2)C1 C1(CNC(N(c2ccc(OC)cn2)C)=O)CCOCC12CCCC2 N1(C(=O)C=CC(F)(F)F)CC2CC(NC(C3CCOC3C(F)(F)F)=O)C1C2 C12(NC(c3ccc(C)nc3C)=O)CC3CC(C1)CC(NC(C1CC1CF)=O)(C3)C2 c1(C(=O)NC2C=CC(C(N(CCCOC)C)=O)C2)ccc(-c2ccccc2)n1C N12CCC3CN(CC13)N1C(C)C(CCC1)C2=O.C(c1cccc(F)c1)=CC=O CC(C)C(F)(F)CC(=O)N1CCC(CNC(=O)C(c2ccc(Cl)s2)C)C1 C1(C)(C(N(C(C)CN(C)C(c2cnn(CC(F)(F)F)c2)=O)C)=O)CC(C#N)C1 C(CC(=O)N(CC(CO)(CO)NC(c1cccnc1)=O)C)(C(F)(F)F)OC N1(C(c2cccc(OCCN(C)C)c2)=O)CCC(F)(CNC(=O)C(F)OC)CC1 CC1CCS(=O)(=O)CCN1C(=O)CCc1nc2ccc(Br)cc2o1 N1(C(C2CCN(Cc3ccc(OC(F)(F)F)cc3)CC2)C)CC2CCC(O)C2C1 c1(NC(c2ccc(F)c(-c3cccc(F)c3)n2)=O)cc(Br)nc(Br)c1 CN1CCC(NC(=O)CC2C=CC(NC(=O)CC3CCCC34CC4)C2)C1=O C12(NC(C3C(C)CC3)=O)CCC(CN(C(=O)Cc3cnco3)C1)C2 C12(NC(CCNC(=O)OC)=O)CCC1CN(C(=O)C(c1ccccc1Cl)C)C2 N1(C(c2c(C)c(C3CC3)on2)=O)CCN(C(C2CCN(C)C2=O)=O)C(C)C1 c1(C(N(C2CCN(C(CCC(=C)Cl)=O)C2)C)=O)cnc(O)cc1O CC1CCCC(NC(=O)C(c2cnnn2C)N(C)Cc2cccc(Cl)c2)C1C c1(CC(=O)NCC2CCC(NC(C3CC4(CCC4O)C3)=O)C2)csc2ccccc12 c1(NC(C(C(C)C)C)CNC(C2CC23CC(O)C3)=O)ccc(S(C)(=O)=O)cn1 N1(C(CCCC(=O)NC(C)C)=O)CCN(C(C2C(C)(C)OC2(C)C)=O)C2CCC12 n1(C(C)C)ncc2c(NCC(F)(F)COC(C)C)[nH]c(=NCC3CCC4CC34)nc12 N1(C(c2cc(CNC(C(C(CC)C)O)=O)no2)=O)CC(C)CCCC1C N1(C(C(C)C2CCCC2)=O)CC2CC1(CNC(=O)CC(C)c1cccnc1)C2 CCCCS(=O)(=O)NC(C)C(=O)N1CC(N(C(=O)CN(C(=O)C(C)C)C)C)C1 N1(C(C(C2(O)CCC2)NC(COC(C)C)=O)=O)CC(C)OC2(CCC2)C1 C1(NC(C2(C)CC2Br)=O)CC2CC(C1)N(C(=O)Cc1cnn(C(F)F)c1)C2 c1(CCC(=O)NC(C=CC(=O)NC(C)CC2CCOC2)(C)C)ccnn1C CN1CCN(CCNc2nc(Br)c(C3OCCO3)s2)CC1 C1(CC(C(=O)NC(CCO)CN2CCCC(O)C2)O)CC2(C1)CC(C(F)(F)F)C2.OC N1(C(C(c2n(C)ncc2)(C)C)=O)CC2CCN(C(C3(C#N)CC3)=O)CC2C1 C=CCC(C)(CC)C(=O)NCC1(NC(=O)Cn2ccc(=O)n(C)c2=O)CCOC1 CCC(C)C(C(=O)NCC1(C)CCN(C(c2cncs2)=O)CC1)OC C1(C(N(CC=C)CCC)=O)C=CC(NC(=O)CCc2cnccn2)C1 c1(C(N(C2CN(c3ncc(OC)cn3)C2)C)=O)cc(F)c(O)cc1Cl Cc1cnc(C(=O)NC2CC(N(C(=O)CC34CCC(C)(C3)OC4)C)C2)cc1C#N C12(NC(CC3C4CN(C(=O)CC5(CO)CCC5)CC43)=O)CC3CC1(CO)CC3C2 c1(CCC(=O)NCC(CC(C)C)NC(C2(C)CCC(=O)N2)=O)ccc(F)c(Cl)c1 C1(CNC(CC2C(C)CC2)=O)CC2(CO1)CN(C(c1cc(O)ncc1F)=O)C2 c1(N2CCC(N(CCC)C(C3(O)CC4CCC3C4)=O)C2)nc2ccc(F)cc2s1 C1(C(=O)NC(C)CNC(=O)Cc2cnsc2)CCC2CCC12 N1(C(c2ccn(CC)n2)=O)CCCC(C(C)NC(c2nncn2C2CC2)=O)C1 CON(CCC(=O)NCC1COCC(C)O1)C(=O)C1CCCCCC1 c1(OC)ccc(OC(F)F)c(C(=O)NC(C2CN(C(=O)C(C)O)C2)C)c1 CCCC(C(=O)N1CCCC1C(C)(C)CNC(=O)Cc1cncc(F)c1)NC(C)=O c1(C(N(C2CCCN(C(C(CC#C)C)=O)C2)C)=O)cn2ncnc2nc1C c1(C(=O)NCCC2CCN(C(C=CC)=O)C2)ccc(SC)nc1 N1(C(CCN(C(c2cc(OCC)n[nH]2)=O)CCO)=O)CCCC12CCOCC2 c1(CC)cc(NC(=O)CC2CN(C(C3CCSC3)=O)CCO2)cc(O)c1 C(=O)(C(C)(C)C(F)(F)F)N1CC(Sc2ccc(NC(CC(C)C(F)F)=O)cc2)C1 N1(C(=O)CCF)CCC2CCN(C(c3ccoc3C3(O)CCOCC3)=O)CC2C1 C1(CNC(C2(F)C(C)C2)=O)CCN(C(C2CN(CC(N3CCCC3)=O)C2)=O)CC1 N1(C(C(CC)C)=O)CCCC(F)(C(=O)NCc2cccc(C)c2O)C1 C1(C(=O)NC2(CNC(c3cnc4sccn34)=O)CCCO2)CCC2CC2CC1 N1(C(=O)NC(C)Cc2cc[nH]n2)CCOC(c2ccccc2F)C1 c1(OC)cnc(Cl)c(C(=O)NC2CN(C(=O)Cn3ccnc3C)C2)c1 N1(C(C2(C(N)=O)CCC2)=O)CCC(CO)C(NC(c2cc3c(s2)CCC3)=O)C1 c1(C(=O)NCC2N(C(c3nc(C)sc3C)=O)CCC2)cc2c([nH]1)CCOC2 C1(CNC(C2C(C)(C)CC2)=O)CC2(CC2)CN1C(=O)Cc1cc(Cl)cc(Cl)c1 N1(C(C2C(=C)C2)=O)CCN(C(c2c(OC)cccc2O)=O)CC1C1CCCC1 C1(C(=O)NC2C=CCN(C(c3ccc(C#N)cc3)=O)C2)CCC(C2CCCO2)O1 c1(C(C(=O)NC2CC(O)(CNC(c3n[nH]cc3Cl)=O)C2)C2CC2)ccc(F)cc1 C1(CC(=O)NC2(COC)CC2)CCCN(C(=O)C=CC2(C)COC2)C1 C=CCCCCCC(=O)N1CCC(F)(CNC(c2ccncc2OCC)=O)C1 C1(NC(C(C)=C(CC)C)=O)CCN(C(=O)C(C#N)C(C)(C)C)C12CCCC2 N1(C(C(CCC)(C)C)=O)C2CCC1CN(C(c1ccc3c(c1)CN(C)C3)=O)CC2 c1(OC)cc(C(=O)NC2CCN(Cc3cc(C)[nH]n3)CC2O)cc(Cl)c1 S(=O)(=O)(CCN=C(NCC(C)C)N1CCCC1)N1CC(N(OC)C)CC1 C1(NC(c2scc(C)c2C)=O)CN(C(=O)Cn2nccc2C)Cc2ccnn2C1 N1(C(CC(CC)(C)C)=O)CC2CCCC2C1C(=O)NCC(=O)N(CC)CC N1(C(COC(CC)C)=O)CCC2(CC2C(N2C(C)CCC2(C)C)=O)C1 c1(C(N2CCN(C(C(F)=CC)=O)C(CCO)C2)=O)sc2cncn2c1C CC(CC(F)(F)F)C(=O)NC1CC(CNC(=O)Cc2ccc(C(F)F)cc2)C1 Cc1cc(C(=O)NCCC2CCCN(C(=O)C(F)CC)C2)ccc1[N+](=O)[O-] N1(C(C2N(C(=O)NC)CCC2)=O)CCCC(CO)(NC(=O)C(C)=CC2CC2)C1 N1(C(COCCC=C)=O)CCC2(CC1)CN(C(C1NC(=O)OC1C)=O)CCO2 C1(C(=O)NC(C(=O)NCC2CN(CC)C2)COC(C)C)CCC(C)(C)C1 N1(C(c2ccc(CN(C)C)nc2)=O)CC(N(C)C(c2cnc(S)[nH]2)=O)C(C)(C)C1 CCC(C)CC(=O)NC1(C)CN(C(=O)C(C)Cc2ccnn2C)C1 C1(C(N(CCC(C)NC(c2cccc(NC(C)=O)n2)=O)C)=O)COC2(CCC2)C1 c1(C(=O)Nc2c(C)cc(F)nc2)cc2c(F)c(C)ccc2[nH]1 N1(C(c2ccnc(C)n2)=O)CCC(C)(C)C1CNC(C1CS(=O)(=O)C1)=O CC1CCN(C(=O)CN(C2CCC2)C)C(C)C1CN1CCCCCC1.C1(=O)CN1 C1(NC(c2nc(OCC)sn2)=O)CCN(C(c2ccnc(S)c2)=O)CC1C(C)C C(CCC(C(=O)NCCC1CC1)N1CCCC(Cc2ccco2)C1)=C(C)C N1(C(c2c(C)[nH]cc2)=O)CC2CC1CN(C(C1CCCOC1C)=O)C2 C(CC(F)F)(C(=O)NC1CC2C=CC1C2)NC(c1n(CCC)ncc1)=O N1(C(CCOCC)=O)CC(CNC(=O)CC2CCN(C)C2)C(C(F)(F)F)C1 N1(C(CCNC(=O)OC)=O)CC(C2CC2)(C(N2CC3(CCCC3)C2)=O)C1 C1(CNC(C(C)CN(C)C)=O)(NC(=O)CC2COC(C)(C)C2)CCCCC1C C1(NC(CNC(CNC(c2cc(OC)no2)=O)=O)=O)CCOC(C)C1 C1(C)(CNC(c2c(C)c(C3CC3)on2)=O)CCCN(C(=O)Cn2cnc(=N)[nH]2)C1 Cc1ncc(C(=O)NC(CO)C(C)NC(=O)C#CC(C)C)n1C Cc1ccc(NC(C2CC(NC(=O)CCc3ccc(=N)[nH]c3)C2)=O)cc1 C(=O)(CC(O)CC(C)C)NCC(CO)NC(CCCCCOC)=O C1(OCC)CC(N(C(c2cnn(C)c2C(F)(F)F)C(=O)NC)C)C12CCOCC2 O=S(=O)(c1ccc2c3c(cccc13)CC2)N1CC2CCCC12 c1(CC(N2C(C)CCC(NC(=O)C(F)C(C)(C)O)C2)=O)n[nH]c2ccccc12 N1(C(CC=CC)=O)CCCCC1C1CCN(C(=O)C(C)SC)CC1 N=c1[nH]c2ccccc2cc1C(=O)NCC1CC(NC(=O)CC2CC2)C12CCC2 Cc1cc(CC(=O)N(C(CNC(C2CC2C(C)C)=O)C2CC2)C)cc(F)c1 c1(C(N2CCCCC(N(C(C(C)OCC=C)=O)C)C2)=O)c(N)ccc(F)c1C Cc1nc(N2CCCOC(CNC(C3CCCC(F)C3)=O)C2)c(C)c(Cl)n1 N1(C(c2cccc(OCC(N)=O)c2)=O)CCCN(C(=O)CNC(N)=O)CC1CO C1(CNC(c2ccc(F)s2)=O)(CO)CCCN(C(=O)CSC2CC2)C1 c1(C(C)(C)NC(=O)NCC2CC2C(F)(F)F)ccc2c(c1)OCCO2 c1(C(=O)NCC(CNC(C2CC23CC3)=O)OC)csc(C)n1 CC1CCN2CC1N(C)C(=O)C2=O.c1(NC(=O)C=CBr)ccc(F)c(F)c1 C1(C(C)N(CCO)C(=O)NCC2(N(C)C)CC2)CCCC1 NC1CN(C(=O)C(c2ccc(F)cc2F)CF)C2(CCOC2)C1 Cc1cc(C(=O)NC(C)(CO)C(=O)NCC(c2cn(C)cn2)O)cc(O)c1 c1(NC(=O)Nc2cnc(-c3ccccc3)cn2)cc(Cl)cc2cn[nH]c12 c1(NCCNC(=O)NC(C)C2CC2)c[nH]c2cnccc12 N1(CCN=[N+]=[N-])CCC(C(=O)NCC(C2CCC2)Nc2ncncc2Br)CC1 C(C)(C(C)C(=O)NCCCn1ccnc1C)NC(Cn1ccc(C)n1)=O O=C1CCC2(CCCN(C(c3ccc(S(N)(=O)=O)o3)C(=O)NC3CCC3)C2)N1 C#CCC(C(=O)NCc1cc(C)ncn1)NC(=O)Cn1cnnn1 CC(c1ccccc1)=CC(=O)NCC=CCNC(c1nccn1C(C)C)=O CC(C)CCC(=O)C(=O)N1CC2(CCC2)CC1CNC(C1CC2C=CC1C2)=O c1(C(=O)NC2CN(C(C(CC)(C)C)=O)CC2O)cnc2ccc(C)cc2c1 C1(CNC(c2ccc(SC)cc2)=O)C(C)CCCN1C(C1CC(=C(F)F)C1)=O C1(CNC(c2cc(F)cc(Cl)c2)=O)CC2(CCC2)CN1C(=O)Cc1ccncc1 C1(C(=O)NC2CN(C(c3scc(OC)c3OC)=O)C(C)C2)CCCCCCC1 c1(C(=O)NCC(C)(C)NC(C2CCCCC2F)=O)cccc(F)c1N CC1CN(C(c2csc(-c3ncc[nH]3)n2)=O)CCCN1C(C1CCNC(=O)C1)=O CN1CCC(C)(C(=O)NC2CCCCC2CNC(C23CC(F)(C2)C3)=O)C1=O CCC(CC(F)(F)F)C(=O)NC1CC2C(NC(=O)C(=O)NCCOC)C2C1 Cc1cc(N2CCOC(C(=O)OC(C)(C)C)C2)nc(=NCc2nc(O)n[nH]2)[nH]1.C(C)C C1(C(N2CC(CCCCC)C2)=O)CN(C(c2ccc(Cl)o2)=O)CC1OC C1(C2(O)CN(c3ccnc(CO)n3)C2)(CNC(C2C3(CO)CC(C)(C3)O2)=O)CC1 N1(C(C(C)n2cccn2)=O)CCC(NC(c2cn[nH]c2)=O)CC(O)C1 Cc1onc(C(N2CC(CNC(c3cnnc(O)c3)=O)C2)=O)c1[N+](=O)[O-] CCCC(C(=O)NC(C1CN(C(c2cn(C)nc2Br)=O)C1)C)OCC c1(OC)nccc(C(N2CCCC2(C)CNC(=O)C=CI)=O)n1 N1(C(c2ccc3occc3n2)=O)CCC2CC2(C(=O)N=c2ccn(CF)[nH]2)CC1 c1(NC(C2CCCCC2)CC)cc(NCCC2CC(C)(C)C2)nc(C)n1 N1(C(c2c(Cc3cnc(C)s3)cccc2)=O)CC2CC1CN(S(C)(=O)=O)C2 c1(CCC(=O)N(C(CNC(=O)C(C2CC(F)(F)C2)O)C2CC2)C)ncnn1C C1(NC(Cc2ccc(C)cc2Cl)=O)CN(C(c2ccccn2)=O)CCC12CCC2 CC1CCC(O)C(NC(c2cc(CNC(=O)CC3(N(C)C)CCC3)ccn2)=O)C1 C1(NC(c2n(C)ncc2)=O)C2CCN(C(=O)C(N)=O)C12 C(=O)(C1=CCN(C(=O)C(CO)c2ccccc2)CC1)NC(CC(C)C)CCO CC(CC(N)=O)C(=O)N1CC2(CCC2NC(=O)C=Cc2cncs2)C1 N1(C(C(C)S(C)(=O)=O)=O)CCN(C(=O)C=Cc2nc(C3CC3)n[nH]2)CCC1C N1(C(C(=O)N(c2ccc(C)s2)CCNC(C)=O)C)CCP(C)(=O)CC1 c1(C(N2C3CC(CC(NC(c4ccoc4)=O)C3)C2)=O)cc2nn[nH]c2cc1F C1(C(=O)NCC2OCCN(Cc3nccc(C)c3)C2)CCC2CCC(=O)N2C1 c1(C(C(=O)NCC2(CN(C)C(c3cnc(O)o3)=O)CCCC2)O)ccc(F)cc1 Cc1[nH]c(C#N)cc1C(=O)NCC1(F)CCC(NC(=O)C=CC2CCCC2)C1 c1(C(=O)NC2CCC(CNC(C3CCN(C)CC3)=O)C2)nnn2c1C(=O)NCC2 C1(C(=O)NC2CC(C(NOCCC)=O)C2)CC12CCCC2 c1(NC(c2cc(C)c(C)nc2)=O)ccc2c(c1)CN(Cc1nccn1C)CC2 Cc1onc(C(F)(F)F)c1C(=O)NC1CCCC(N(C(=O)CC2CSC2)C)C1 N1(C(C(C)Cc2cnn(C)c2)=O)CCCC(CNC(=O)CCF)CC1 c1(C(N2C(CNC(C3CCCN(C(C)C)C3)=O)CC2)=O)ccc(Cl)c2occc12 N1(C(c2cc(C)c(Cl)cc2)=O)CCC2(C1)CN(C(=O)C=CC1CCCCC1)C2 C1(C(N2CC3C(NC(c4cnn(C)c4N)=O)(C3)C2)=O)Cc2c(F)cccc2O1 CN1CCOCC1C(N1CCCC1CCNC(C1CC2C=CC1C2)=O)=O c1(CC)cc(C(=O)NC2CCC(NC(C3CCOC(C)C3)=O)CC2)ccc1Cl C1(C)(CC)CCCN(C(=O)CC2COCCN2C(C2CC2C(C)(C)C)=O)CC1 N1(C(C(C(C)C)NC=O)=O)CC(C)(C)C(NC(C2COCC2(C)C)=O)C(C)(C)C1 N1(CCC)CC(C(=O)NCC2C3CC2N(C(C2CCCCC2C)=O)C3)CC1=O C(c1ccn(C)c1)=CC(=O)NC(CC=CC(=O)NC(C(C)SC)C)(C)C n1(CC)nnnc1C(C(C1CC(C)=NO1)OC)NCCCCSCCO C1(NC(CCC(=C)C)=O)(CNC(=O)CSCCN(C)C)CCCCC1C C1(CNC(=O)C=Cc2cscn2)CN(C(c2cccnc2S)=O)C2CC12 C#CCCCCC(=O)N(C1CCCC1)CCCNC(c1sc(C)c(C)c1C)=O N1(C(CN(C(C2CCC=CCCC2)=O)CC)=O)CC2(CC(CO)CO2)C1 N1(C(c2ccc(OC)o2)=O)CC2CC2C1C(=O)NC1CN(CC(F)F)C1 N1(c2c(C)c(F)ccc2)C(=S)NC(c2cc(C(=O)O)no2)C2=C1C(C)(C)NC2=O c1(C(=O)NC2CN(Cc3ccc(OC)cc3O)CC2F)c(F)cc(Br)c(F)c1F c1(C(N2CCC(CNC(=O)CC3CCC3)C(O)C2)=O)cccc(F)c1F c1(C(N(C)C(=O)NCC)C)cccc2nsnc12 CCCCC(CC)CCCN(C)C(=O)NCc1ncc([N+](=O)[O-])n1C c1(C(N2C(CNC(C(F)OC)=O)COC(C)(C)C2)=O)cccc2cnccc12 N1(C(C=CCC)=O)CC(CN(C(=O)CCC2CC2)C2CCC2)CC12CCC2 C(=O)(C(C)CC(C)(C)C)NCCCN(C(c1c(C)nn(C)c1N)=O)C c1(OC)cccc(CCC(=O)NCCC2CCN(C(=O)C=CC3CCCO3)C2)c1 C1(C(N(C)CC2CCCN2C(C2C(C)(C)C2(F)F)=O)=O)CCOC2(CCC2)C1 c1(C(N2CCC(C(C)NC(=O)CC(C)(C)C)CC2)=O)ccc2cccnc2n1 C1(N(C(=O)NOCCC(F)F)C(C)=O)CCN(C(=O)C(C)(C)C)CC1 c1(C(=O)NCC2CCC(NC(C3CC=CCC3)=O)C2)c(F)cc(F)cc1Cl N1(Cc2ccc(C)s2)CCC(C2CCCN(C(c3ccc(F)cc3F)=O)C2)CC1 c1(CC(=O)N(CCNC(C(C)C(C2CC2)N)=O)C)cc(Cl)cc(Cl)c1.C=CCCO c1(CNC(N2CC(C(CC)C)C2)=O)cccc(C(F)F)n1 c1(C(C(=O)NCCCC(=O)OCC)N(C(C)CC)C)cnc(N2CCCC2)cc1C C(CCCN=c1[nH]nc(C(=O)OC)s1)C1CCC(NC(C2(OCC)CC2)=O)C1 c1(C(N2CCC(NC(COCC)=O)C(CC)C2)=O)ccc2nc(Cl)nn2c1 CP(C)(=O)c1ccc(C(=O)NC2CCN(C(=O)CN3CCCCC3)C2)nc1 C#Cc1cnn(C(N2CCCCC2CC(=O)NCC2(O)CC2)=O)c1 C12(CN(C)CC3CCN(C(c4cc(CO)ccn4)=O)C3)COC(C)(C1)C2 C(=O)(C1CCCc2c(O)cccc21)NCCOCCCNC(C(C1CC1)SC)=O CC(CN=C(NCc1cccnc1)NC1CC12CC2)NCC(F)(F)F C1(CC(=O)NC(c2cccc(Cl)c2)C)CCCN(C(C2CC(=C3CCC3)C2)=O)C1 C#CCCCCCCC(=O)N(CC(O)CNC(c1cc2c(nn1)CCC2)=O)C C1(CNC(CCN(C)CC)=O)CC(F)CN1C(C1CC1c1nccn1C)=O N(C(=NCCF)NCC(=O)NOCC(=O)OC)CC1CCCC(CC)C1 c1(CC(N2C(C)CN(C(c3coc(Cl)n3)=O)CCC2)=O)c[nH]c2ccc(F)cc12 C1(NC(C(=O)NC(c2ccnc(NC)c2)COC)=O)CC2CC(OC)CC12 C(CC(=O)NCC(O)CNC(=O)COC(F)F)(C(F)F)N(c1nccn1C)C CC(=O)CCCC(=O)N1CC(O)CC1C(=O)NC1CC(C)(N(C)C)C1 c1(C(=O)NCC(CNC(CCCCCC)=O)O)cc(Cl)c(Cl)[nH]c1=N c1(C(=O)N(c2c(F)cc(Cl)cc2Cl)CC(F)F)cc2c(s1)CCN(CCO)C2 Cc1cc(F)c(S(=O)(=O)N2CCCC(c3nnc(C4CC4)o3)C2)c(C)c1 C(CNC(c1ncnc(O)c1F)=O)(C(C)C(C)C)Nc1ccnc(C(C)=O)n1 C1(NC(Cn2cc(CNC(C3ON=C(C)C3)=O)nn2)=O)CN(C)CC12CC2 N1(c2n(CC3CC(O)C3)c(-c3ccon3)nn2)CCCC2COCCC12 N1(C(C2(CCNC(CCc3ccn(C)n3)=O)CC2)=O)CC[Si](C)(C)CC1 N1(CC(=O)N(CCC(F)(F)F)C)CCOC(CN=[N+]=[N-])C1 Cc1ncccc1C(=O)NCc1cn(CCOC2CCC(C(=O)O)CC2)nn1 C(CCCC(=O)NCC(C)CCCO)N(C)C(C1CS(=O)C1)=O n1(CC(=O)N(CCNC(=O)CC(C)OC)CC)ccc(O)nc1=O C1(N(C(c2c(C)nn(C)n2)=O)C)CCCCN(C(c2c[nH]c(=S)cn2)=O)C1 Cc1c(C(N2CC(C(O)C(=O)NCC3C4CCCC34)C2)=O)ncn1C N12CC3CCN(C(C3)C1)C(=O)c1ccc(s1)CC2=O.c1(OC)ccccc1OC C(=O)(CC1OCc2ccccc21)NC1CC2(CC(C)C2)N(C(=O)CNC=O)CC1 C=Cn1nccc1C(=O)N(CCO)C1CC1.N12CCC(C1)OCC2=O C(=O)(CC(O)CC(C)(C)C)NCCCCCC(=O)NCC1CCCC(OC)C1 N1(C(c2ccc(C)cc2F)=O)CCN2CCN(C(c3cccnc3)=O)CC2C1 C12CC(C)N(C1)C(=O)CCN2.CC1C(=O)N1.C1(C(=O)OC(C)(C)C)CCCC1 Cc1c(C(N2CCOC(C(=O)Nc3cncc(O)c3)C2)=O)cccc1Br C12(C(=O)NCC3(O)CCC(C)CC3)COCC1CN(C(=O)CC1CC1(C)C)C2 C1(CCN(CC(N)=O)C)CCN(C(=O)CCC2CCCOC2)CC1 c1(C(=O)NC(Cc2ccc(OC)cc2)(C)CO)ccc(F)c(C)c1 C1(C(N(C)CC2C3CN(C(Cc4c(C)cc(C)s4)=O)CC32)=O)CCCC2(CC2)C1 C12(C(=O)NCCNC(c3ccncc3)=O)CC3CC1C2C3O Cc1cccc(C(N2CC(c3cn(C(C4CCCCC4)C4CC4)nn3)C2)=O)c1I C1(NC(CCC2CCC(C)O2)=O)C2CCN(C(c3cnc(N)c(Cl)c3)=O)CC12 c1(OCC(=O)NCC2CN(C(=O)C=CC=C(Cl)Cl)CCO2)ccc(O)cc1 N1(C(Cc2c(C(C)C)cccc2)=O)CCN(C(=O)CCNC(=O)OC)C(CO)C1 c1(NCCOC(COC)C(C)C)ncc(C)cc1S(=O)(=O)NCC(F)(F)F C1(C2N(C(c3c(C)nc[nH]3)=O)CCC2)CCCN(C(=O)CSC2CC2)C1 N1(C(CC(C)F)=O)CC2CC(C1)N2C(c1ncn(C(C)C)n1)=O C1(C)(NC(C2CC(C)(NC(C)=O)C2)=O)CCN(C(=O)C(n2cc(C)cn2)C)CC1 C1(NC(CCC(=C)Cl)=O)CCN(C(C2CCN(OC)CC2)=O)C(C)C1 C(C(COC)CC(=O)NC1C=CCN(C(=O)CC2CCS(=O)(=O)C2)C1)OC CCCC(CC)C(=O)Nc1cccc(NC(c2oc(CCC)nc2C)=O)c1 Cn1cncc1C(=O)NC1(C(N2CCC(OC3CCCC3)C2)=O)CCCC1 c1(N2CC3CC(NC(c4c(C)nc(CC)s4)=O)C3C2)ncc2c(n1)CCCCC2 c1(COC)n[nH]c(=NCC(c2ccccc2F)NC(=O)C(=Cc2cn[nH]c2)C)s1 C1(CNC(CC=C)=O)CCC(C)(C)CN1c1ncc(C)cn1 C1(C(N2C(C(N(CCCCC)C)=O)C=CC2)=O)CCCC(=O)N1 C1(COC)CCC(C(N2CCC(NC(c3nn[nH]c3C(F)(F)F)=O)C2)=O)C1 C1(CN(C(=O)CCc2ccc(F)nc2)C)CN(C(c2cnn[nH]2)=O)CCO1 C1(C(=O)NC2CCN(C(C)=O)C2)CCCN(C(C2COCC(C)O2)=O)C1 N1(C(c2cc(C(C)C)nn2C)=O)CCC(C)C(CNC(C2CN(C)C(=O)N2)=O)C1 C(=O)(C1=C2CCN=C2NC=C1)NC1CC(OCC(=O)NCC2OCCC(C)C2)C1 N1(C(CCCCOC)=O)CCN(C(=O)CC(C)(C)C2CC2)C(CC(F)(F)F)C1 C(=O)(C(C)CS(C)(=O)=O)NCc1c(C)nn(C2CCC2)c1 c1(OCC)cc(CNC(C)COc2ccnc(OC3CCCCC3)n2)n(C)n1 CCCCCCCC(=O)NCCNC(=O)CN1CCN(c2ccccc2)S1(=O)=O C1(NC(c2cc(CC)nc(Cl)c2)=O)CN(C(=O)CC(C)C)CC2(CCOCC2)C1 N1(CC)CC2CCN(C)CC2C1.N12CCCC1C1(CCC1)C(=O)NC1(CC1)C2=O Cc1c(C(=O)NC(C)CC(C)NC(=O)CC(=O)N(C)C)sc2[nH]cnc(=O)c12 C1(CNC(C(C)Cc2cnc[nH]2)=O)CC2CCC1N2C(=O)CCCC(=O)C1CC1 C1(C#N)(C(N2C(CNC(CC(C)(C)C)=O)CCC2)=O)CC12CCCC2 C1(NC(C2CCCCO2)=O)CCOC2(CCN(C(C3(CO)CCOC3)=O)CC2)C1 CC(CS(C)=O)C(=O)NCC12CC(NC(c3cnc4n3CCC4)=O)(C1)C2 c1(CC(=O)NCC(C)NC(c2nccnc2C(N)=O)=O)ccc2[nH]ccc2c1 Cc1cccc(CN(C)C(C2CCCN(C(c3cc(C)ns3)=O)C2)=O)c1 c1(C(=O)NC2CC(CNC(C3CCC(C)C3)=O)C2)cc2c(cn1)OCCO2 c1(C(=O)NC2CC(CC(=O)NCc3cc(F)cc(F)c3)C2)ccc(F)cc1O C1(C)(CNC(CC(CC)CC)=O)CC(F)(F)CN1c1nc(C(C)(C)C)nc(=N)[nH]1 Cc1[nH]c(Cl)nc(=NCC2(C)CCCN(C(C3(C#N)CC3)=O)C2)c1C#N Cc1cc(C(=O)NCC(C)(O)CNC(c2cn(C(F)F)cn2)=O)cc(N)c1 C1(C(N(C(CC)C)CC)=O)CC=CCC1NC(=O)C1CC1 N1(C(c2c(CC)ocn2)=O)CCC2CN(C(=O)C(C)O)CC2CC1 N1(C(C(C)OC)=O)CCC(O)(C(C)NC(c2ccc(C3CC3)cn2)=O)C1 c1(C(N2C(CCC)CN(C(=O)C#CC(C)C)CC2)=O)cc2cc(C)ccc2o1 c1(CC(N2C(C)C(NC(=O)CN3CCC3C)CC2)=O)ccc2c(c1)OCCO2 C1(C(N(CC(C)CO)C)=O)CCN(C(=O)CC2CC2)C1(C)C C#Cc1ccccc1CC(=O)NC(C)CNC(c1sc(Br)nc1C)=O c1(CCC(=O)NC2CCN(C(=O)C(F)(F)Cl)CC2)ccc(F)c(Cl)c1 C1(OC)CC(C(=O)NC2CC(NC(=O)C=Cc3ccncc3)C2)CC1OC C(N=c1ccc(C(F)(F)F)n[nH]1)C1CCCCN(C(c2cn(CC=C)nn2)=O)C1 C1(CNC(C(C)SC)=O)CN(C(C2CN3CCCN2CC3)=O)CC2(CCC2)O1 CN1CCCC(F)(C(=O)NCC2(C)CN(C(=O)C=C3CCOCC3)CCO2)C1 C1(C(=O)Nc2cncc(CC)c2)CCN(C(=O)CN=[N+]=[N-])CCO1 Cc1cc(C(N2CC3C(CNC(c4snnc4C(C)C)=O)C3C2)=O)c(N)c(F)c1 CCCCCCC(=O)NC1CCC(c2cn(C(CCCSC)C(=O)O)nn2)CC1 C1(NC(CCCCCC)=O)CCCC12CN(c1cc(Cl)nc(C)n1)C2 CCCC(CC)C(=O)NCC1COCCN(C(C2(N(C)C)CCCC2)=O)C1 c1(C(=O)OC)cnc(C(=O)N(C(=O)CCOC2COC2)C2CC2)c(N)c1 CN1CCN(C(=O)C(F)(F)C2CC2)CC1CNC(C1(C2CC2)CC1)=O n1(CC(=O)N(CCC(C)NC(=O)Cc2cncn2C)C)nnc(=N)[nH]1 C(=O)(CC(C)CC(C)C)NC(CC(=O)NCc1nc(C)[nH]n1)C(F)F C(=O)(C1OC(=O)c2ccccc21)NCC1(NC(=O)CC2=CCCC2)CCCC1 N12CCC3C(C3C1)C(=O)NC2.C1(CC)CC1CC(=O)SCCOC.C1(=O)CN1 N1(C(C2CC(=O)NC(=O)N2)=O)CC2(C1)CN(C(=O)CCOCC(F)F)CCO2 C1(C)(CC)C=C(C(=O)NCC2(F)CC(CNC(c3cnncc3NC)=O)C2)C1 N12CC(C3(CC3)C1)NC(=O)C2.c1(CNC(=O)OC)ccc(CO)o1 N(C(=NCCCCC(F)(F)F)N=c1cnc(I)c[nH]1)C(C#C)C(C)NCC CC1(C)c2ccccc2CCN1CCCOc1ccc(F)cc1[N+](=O)[O-] C(=O)(C(O)C(C)(C)CC)N1CC(NC(c2ccc(OCC)nc2)=O)C(OC)C1 Cc1cc(C)c(C(N2C3CCC2C(C)C(NC(c2cnoc2C)=O)C3)=O)c(Cl)n1 S(=O)(=O)(c1ccccc1)CNCCC(=O)NC(CNC(=O)CCF)CO C1(CN(C(C2C(F)(C(=O)OC)C2)=O)C)CCCN(C(c2ccc(N)cn2)=O)C1 c1(C(N2CCCC(N(C)C(c3cncn3C(F)(F)F)=O)C2)=O)cccn(C)c1=O c1(CC)sccc1C(=O)NC1CCC(CNC(=O)C(=Cc2ccco2)C)C1 N1(C(c2c(C)ccc(Cl)c2)=O)CCC(C)(C)CC1C(=O)NOCCC(F)(F)F n1(C(C(=O)NCC(CC)NC(c2sccc2C(C)=O)=O)C)ccc(Br)n1 C1(C(=O)NCCN(C)CCc2ccco2)(NC(C(C)=CCC)=O)CC1(C)C CC1(C)CN(C(=O)CCC2CC2(Cl)Cl)C(CNC(c2cc(Cl)no2)=O)CO1 C1(CC)CN(C(=O)C=Cc2nc(C)c(C)[nH]2)CCC1Nc1ncccc1C#N N1(C(CCc2ccc(C)s2)=O)CCCC(NC(c2cc(C(C)(F)F)n[nH]2)=O)C1C C=CC(C)(O)C(=O)N(CCCNC(c1cnc(C)n1C)=O)Cc1ccccc1 C12(CNC(C3CN(C)C3)=O)CCCC1N(C(=O)CSCc1ccccn1)CC2 c1(COC)ccccc1C(=O)NC1C2CC(NC(c3ccc(C(=O)OC)o3)=O)CC12 c1(OCC)ccc(F)c(C(=O)NC2CS(=O)(=O)CC2NC(C2(O)COC2)=O)c1F C1(CC(=O)NC2(CN(C)C)CC2)CCCN(C(=O)C(F)C2CCCC2)C1 N1(C(CCC(=O)OCC)=O)CC2CCCC(NC(=O)CCC(N)=O)C2C1 N1(C(C2(C#C)CN(C(=O)C(C3CC3)OCC)C2)=O)CCC(C)CC1C N1(C(CCNC(C)=O)=O)CCOCC12CCN(Cc1ccc(C)cc1O)C2 NS(=O)(=O)c1ccsc1C(=O)NCCC1CCCCN1C(=O)C(O)C(F)(F)F C(CN=c1[nH]c2ccc(F)cc2o1)C1N(C(c2cc(C)nn2C)=O)CCCC1C N1(C(c2[nH]cc(CC)c2)=O)CC2C(CNC(=O)C(C)(C)NC(=O)C(F)(F)F)C2C1 C1(C(=O)Nc2c(C)nn(CCF)c2)C(C2CC2)CCN1C(=O)CCc1ncccn1 N1(C(c2c(C)[nH]cc2)=O)CCCC(NC(C2COCCO2)=O)C1C c1(C(N2CC(c3cn(Cc4c(C(=O)OC)scc4)nn3)(O)C2)C)cccc(Br)c1 N1(C(c2csnn2)=O)CC2CC1CN2Cc1ccccc1Br C(=O)(CN=c1[nH]c2ccccc2s1)NC1CN(C(Cc2c(C(C)C)con2)=O)C1 c1(CCN=C(NC(COC)C)NC2CC(OC)C2)cn(C)c2ccccc12 CCCCCC(O)C(=O)N1CC2(CCN(Cc3cc(C)ccc3C)C2)C1 c1(C(=O)NC2CCC2NC(C2CC2(Cl)Cl)=O)c(F)ccc2c1OCO2 N1(C(CCCC)=O)CCCC(C(=O)N(C2CC2(C)C)C)CC1 C1(NC(COc2ccn(C)n2)=O)CC2(CCN(C(=O)CCCC(C)(F)F)C2)C1 C1(NC(CC)=O)CN(C(c2csc(O)n2)=O)CCC1C c1(CC)ncnc(OCc2ccccc2)c1.C1(O)(CO)CN(C(C2CC(=O)N2)=O)C1 CCCCCCCCCC(=O)NC1CCCN(C(c2cnc(O)nc2O)=O)C1C C1(NC(c2ccc(C3CCOC3)s2)=O)CC2CCC(C1)N2C(c1n[nH]cc1F)=O CCC(CC)C(C)C(=O)NCCCC(C)(C)NC(c1ccc(C(C)C)o1)=O C1(C(=O)NC(CNC(CC(C(F)(F)F)OC)=O)(C)C)CCCC2(CCOCC2)O1 C1(N(C)C(C2COC2)=O)CCN(C(C2CCC2)=O)C1.C12(CC1)C(=O)NCC2 CC1(C)C=C(C(=O)N2CCC(C(CO)NC(C3CSCC(=O)N3)=O)CC2)C1 Cc1cc(C(=O)NCCN(C(=O)CCS(C)=O)C)nn1C1CC1 N1(C(C(C2(C)CC2)NC(COCC)=O)=O)CCC(NC(=O)C(C)OC)C(C)(C)C1 N1(C(C2(SCC)CC2)=O)CCC(NC(=O)CC2CN(C)C2)C1(C)C c1(C(N2C(C3CCN(C(COCC#C)=O)CC3)C(C)(C)C2)=O)cccc(N)c1O C(=O)(C(CCC(N)=O)N(C)C)N1C(CCNC(CCCCOC)=O)CSCC1 N1(C(C=CC(C)(C)NC(CCOCC#C)=O)=O)CC2CCC(C1)O2 N=c1nc(N2CCC(N3CCC3)CC2)[nH]c(=NC2Cc3cscc3C2)[nH]1 c1(OC)ccc(C(C)NCc2cccc(CN(C)C(C)C)n2)c(C)c1 c1(C(=O)NC2CCN(C(C(C)CSC(F)(F)F)=O)C2)cncc2ccc(F)cc12 C12(C(=O)Nc3cnc(OC)nc3)COC(C1)C(NC(=O)C(O)C1CC1)C2 Cc1oc(-c2ccc(Cl)cc2)nc1C(=O)NC(C)C(C)NC(c1cnc(O)s1)=O N1(C(C2CCCCC2(F)F)=O)CCCN(C(c2c(Cl)cncc2Cl)=O)C(CO)C1 c1(OC)cc(C(=O)NC2(C(=O)NC(c3cnc(C)s3)C)CCC2)[nH]n1 O=C(CN1CCC=C(Cl)C1)NC(=O)C(CNC(c1ccsc1)=O)c1ccccc1 CON(C(=O)C1CC(C2CC2)=NO1)C1CCOCC1 CCCC(CC)CCC(=O)NCC(C)(C)OCC(N1CC(C2=NOCC2)C1)=O N1(C(=O)CSc2ccccc2F)CCC(C2CCN(C(C3CSC3)=O)CC2)C1 C1(NC(=O)NC(c2c(C)nc(C)[nH]2)C)CCC2(CCC1(F)F)OCCO2 N1(C(c2c(CCC)[nH]cc2)=O)CC(NC(=O)C=CCN2CCCC2)CCC1C c1(C(=O)NC(CNC(CCC#C)=O)CCCC)cnc2c(c1)nc(O)n2C c1(CN2CC(NC(C=CC(=O)NC3CC3)=O)C2)ccc2cc[nH]c2c1 Nc1c(C(=O)NCCC(O)CNC(c2cnc(S)nc2)=O)nc(O)nc1O c1(CNC2CC(C(=O)NC(c3c(O)n[nH]c3C)CC)C2)c(Cl)cc(C#N)cc1Cl c1(SC)ccc(C(N2CCC3CC2CN(C(c2ccc[nH]2)=O)C3)=O)cc1[N+](=O)[O-] n1(C(C)C)ccc2ccc(-c3nc(Nc4cc5c[nH]nc5cc4Cl)cs3)cc12 c1(OC)ncc(C(=O)NC(C2(O)CCN(C(=O)C(F)C3CC3)CC2)C)c(C)n1 CN1C(=O)C(C)(C)c2cc(C(N3CC4CC(NC(=O)CCF)C3C4)=O)ccc21 N1(C(CCC(C)OCC)=O)CCC(CNC(=O)COCc2ncnn2C)C1(C)C N1(C(CC2CCN(C)C2)=O)CCC2CC2(C(=O)NC(C)(CO)CO)CC1 CC1CN(C(=O)COCCCF)CC1(C)CNC(c1cccc(CO)c1)=O C(=O)(C#CC(C)(C)C)NC1(C(N2CC(=C)C2)=O)CC1C Cn1c(C(N2CCCCC(NC(=O)Cc3sc(O)nc3O)C2)=O)cnc1[N+](=O)[O-] C1(C(=O)NC2CCN(C(c3ccccc3Br)=O)C2)CCCCC12OCCO2 N1(C(CS(CC)(=O)=O)=O)CC2(CCC(NC(=O)COC3CCN(C)CC3)CC2)C1 C1(CC(=O)NCCCCNC(c2ccnnc2O)=O)CN2CCN1CC2 C1(C)(CNC(c2c(C)c(C3CC3)on2)=O)COCCN(C(C2(Cl)CC2(C)C)=O)C1 C1(C(N(C)CC2CCCS2)=O)CC12CC(NC(c1ncoc1C1CC1)=O)C2 N1(C(CCC#C)=O)CCn2c(CNC(=O)CSc3ccc(F)cc3)nnc2C1 c1(NC(C2(O)CCN(Cc3ccc(CCC)cc3)C2)=O)ccc(C#N)c(F)c1F CC(C)C(C)(C)C(=O)NC1CC2CC(NC(c3ccc(Cl)nc3Cl)=O)CC12 O=C(C(O)CC1CCCC1)NCC1CCC1NC(=O)C1CC1 C1(NC(c2cc([N+](=O)[O-])n[nH]2)=O)CCC2(CC1)CN(c1nnc(O)s1)CCO2 Cc1cc(C)cc(S(=O)(=O)NC2CCCC2C(=O)Nc2ncc(Br)c(O)n2)c1 N1(C(CC2CC(CC)C2)=O)CCCC(NC(c2[nH]c(C)nc2C)=O)C1C CN1C2CCC1CC(=CC(=O)NCCCNC(=O)C(O)c1ccsc1)C2 CC1CC(NC(=O)C=CC=C(Cl)Cl)CCN1c1cncc(Cl)n1 c1(C(=O)NCC2N(C(C(C)=C3CC3)=O)CCC2C2CC2)cc2c(s1)CC(C)(C)C2 C(=O)(CC(C)(C)CN(C)C)NCC(CCC)NC(C1(CC=C)CCCC1)=O N1(C(C(C)OCCC#C)=O)CCN(C2CCN(C(=O)C(C)O)C2)CC1 N1(Cc2scc(C(=O)OC)n2)CC(O)CC1C(N1CCOC(O)C1)=O C1(C(=O)NCCNC(=O)C(F)n2cccn2)Cc2nccn2C1 N1(C(C)C)CCCC(CC(=O)NC(C)(C)CN(C(=O)CC2CC(F)(F)C2)C)C1 C1(N(C)C)(C(=O)NC2CC2CC(=O)NCC(=O)N(C)O)CCCC1 N1(C(=O)CN2CCOCC2=O)CCC2CC2(C(=O)NO)CC1.C1(C2CC2)CC(=O)N1 C(=O)(C(C(F)(F)F)C(F)(F)F)N1CC(CCNC(CCOCC#C)=O)OCCC1 C1(NC(=O)C(F)CC2CC2)CCN(C(=O)Cc2cnccc2Cl)CC1O N1(C(C2(COC)COC2)=O)CC(NC(=O)Cc2ccnc(OC)c2)CC(O)C1 N1(CN(C(c2c(-c3c(C)nc(C)s3)cnn2C)=O)C)Cc2cnn(C)c2C1 c1(C(N2CC(NC(C(=O)NC(CCOCC)C(C)C)=O)C2)=O)cc(=N)[nH]c(Cl)n1 C(=O)(C1=C(C)CCOC1)N1CCOCC(CNC(C(CCC)OCC)=O)C1 C1(CNC(C(CC)(C)F)=O)CC2(CCN(C(c3cccc(F)c3C)=O)CC2)CO1 N1(C(CCC=CCC=C)=O)CC2(CC(NC(c3ccnc(C)c3O)=O)C2)C1 N12CCSCC1C2=O.C1(CCNC(CC2CC(OCC)C2)=O)CCC(C)(C)C1 CCCCC(C(=O)NCC(CC1CCCC1)C(=O)NC1(C)CC(F)C1)C(C)C c1(OC)ncccc1C(=O)NCC1CC(NC(C2CCCS2=O)=O)C(O)C1 Cc1cccc(C(N2CCCC2CNC(=O)C(C2(O)CCCC2)F)=O)n1 C(=O)(CCCS(C)(=O)=O)NCC(C)CN(C(=O)CNc1cccnc1)C C1(NC(=O)CS)CC2CC1N(C(=O)Cn1cncn1)C2.C1(O)(C)CCC1 c1(NC(c2cc(C)[nH]n2)c2nnnn2Cc2cccs2)c(C)cc(Br)cc1C CCC(C)C(O)CC(=O)N1CCC1c1cn(C2(C(=O)O)CC2)nn1 c1(C(N2CCC(N(C(C(F)=CCCC)=O)CC)CC2)=O)c(F)c(F)cc(F)c1F c1(C(C)O)ccccc1C(N1CC(N(C(=O)C(c2ccc(F)cc2)F)C)C1)=O C(=O)(C(C)C(O)CC(C)C)NC1CCC(C(N(C(C=C)C2CC2)C)=O)C1 c1(CC2(C(=O)NCCN(C(=O)C=C3CCCC3)C)CCC2)ccc(F)cc1 c1(C(C(=O)NCC2(COC)CN(C(C3CCCCO3)=O)C2)C)cccc(O)c1 N1(C(CC2CC(CC)C2)=O)CCCN(C)CC1.C1(=O)CC(C)(C)N1C c1(C(N2CC(n3cc(Cn4cncn4)nn3)C2)=O)ccc(Cl)c(F)c1 c1(C(N(CCC(=O)NC2CCNC(=O)C2)CC)=O)c[nH]ccc1=O N1(C(C(=O)NC2CC(C(=O)OC)C2)CC2CCCO2)CCCN(CCO)C(C)C1 Cc1cc2n(n1)CCN(C(C1CN(C(C34CCN(CC3)C4)=O)CCC1O)=O)C2 C(c1ccc(F)c(F)c1)=CC(=O)NCC(C)NC(C1(O)COC1)=O CC(C)C(CN(C)C)C(=O)N(CCC(=O)NCC(O)CF)C Cc1ccn2ncc(C(N3CC(C)(NC(=O)C=Cc4cnn(C)c4C)C3)=O)c2n1 c1(C(N(C(C)C(=O)NCCc2cnn(CC)c2)CCC)=O)cnn(C)c1 c1(C(=O)NCC(CN(C(CCOCCCOC)=O)C)O)cc(C#N)c(F)cc1F c1(CC(=O)NCCN(C(CN(CCC)C)=O)CC2CC2)c(Cl)ccc(O)c1Cl c1(OC)cc(S(=O)(=O)N(C)CCOCC2CC(c3ccccc3)C2)ccc1OC N1(C(c2ccc(OC)cn2)=O)CCCC(F)(CNC(c2coc(CO)c2)=O)CC1 c1(C(=O)NCCN(C(C=C(CCC)CCC)=O)C(C)C)c(C)ncnc1C C1(O)(CNC(C2CN(S(C)(=O)=O)C2)=O)CC(c2ccccc2)C1 C=CCC(CC=C)C(=O)NCC(C12CCC(CC1)C2)NC(=O)C(C)SCC N1(C(C=COCC)=O)C2CCC1CN(C(=O)C(C)(C)OC(C)C)C2 CC(CC1=CCCCC1)NC(=O)CC1(N(C)C(C2CCN(C)CC2)=O)CC1 N1(C(c2cc(OC)ncc2)=O)CCCC(C)C1CNC(c1ccc(Br)o1)=O Nc1c(C(=O)NCC23CCC2CN(C(C2(CO)CCCO2)=O)C3)cc(F)cc1F C=CCC(CNC(=O)CCOC1CCOCC1)NC(=O)Cc1ncc(C)s1 C1(CC(N2CC3C(NC(C4CC(N(C)C)C4)=O)C3C2)=O)CCC2(CC1)CCC2O N1(C(CCOCC#C)=O)CC2(C1)CN(C(c1cnc(Cl)cc1OC)=O)CCO2 C1(C(=O)NC(CN(C(CSCCC)=O)C)C)Cc2ccccc2N1C(C)=O Cc1ccn2ncc(C(=O)NCC3(C4(O)CN(C(=O)CC#N)C4)CC3)c2c1 c1(CNC(C(CC)Cc2cn(C(C)C(=O)OC)nn2)=O)cc(C2CC2)ccc1C c1(C(=O)NCC(CNC(c2c(C)nco2)=O)O)ccc2ncc(C)n2c1 Cn1cc(C(=O)NC2CCC(CNC(=O)Cc3cccnc3N)C2)ccc1=O C1(C(=O)NC(CNC(C2=C(C)CCC2)=O)CO)CCCN(S(N)(=O)=O)C1 C1(CCC)CCCN(C(=O)CC(C)N(C)C(c2ncn(C)c2C)=O)C1 c1(OC)cc(C(=O)NC2CCN(Cc3c[nH]c(Br)c3)C2)cc(C)c1 C1(CC)C(OC)C(C(=O)OC)CN1C(C1CCCC(=O)C1)=O C(=O)(C1CC(C)Cc2c[nH]nc21)NCCC(C)NC(C12CC3CC1C2C3)=O N12CCC(CC1)NC(=O)C2.C(=O)(C(C)(C)Oc1ccccc1)N(CCC)CC N1(S(CCC)(=O)=O)CC2CCC1CN2C(c1cccc(Cl)c1O)=O N1(C(c2ccc(C)o2)=O)CC(CNC(=O)CSCc2cccs2)CCC1C C(C)(C(=O)NCCCNC(=O)CC12CC(C1)C2)OCC C1(NC(c2cc(C)ns2)=O)CCCCN(C(=O)C(O)C2CCCC2)C1 N1(c2snc(C(C)C)n2)CC=CC(NC(C2CCC(F)CC2)=O)C1 c1(NC(C23C(CN(C(CSc4ccc(C)cc4)=O)C2)C3)=O)c(O)cccc1Br C1(C(=O)NCC2CCN(C(c3c(OC)scc3)=O)CC2C)Cc2ccncc2C1 C#CC1(NC(C2(C)CCN(C(c3cc(C4CC4)on3)=O)C2)=O)CCC(C)(C)C1 c1(N2CCCC(NCC3(C(=O)OC(C)(C)C)CC3(F)F)C2)ncnc2sccc12 C(=O)(C(C)(C)C)NCCC(=O)NCCOCCN(C(=O)C(O)Cc1cnn(C)c1)C c1(CC(=O)NCCCC(C)NC(=O)CN(CC(C)(C)C)C)cccc(Br)c1 c1(C(=O)NCCN(CCC)C(C2C=CC=CC=C2)=O)ccc(OCCF)cn1 C1(CC(=O)NCCCc2cc[nH]n2)CC2(CC2)CN1C(=O)Cn1ncccc1=O Cc1cc(NC2CCC2C2CCCCC2)cc(Cl)c1 Cc1cccn2cc(C(N3CC(N(C)C(c4cccc(=O)o4)=O)C(O)C3)=O)cc12 C(C(=O)NC(CNC(c1ccc(C(=O)OC)s1)=O)C1CC1)(C(C)C)SCC N1(C(C2(COC)CCOC2)=O)CCCC(F)(C(=O)NCC23CC(CN2C)C3)C1 c1(CC)cc(C)nc(N2CCC(CNC(=O)CC3CC4(CC4)CO3)C23CC3)n1 C1(C(=O)NC2CCC(NCc3ccc(C(=O)OC)[nH]3)C2)CCS(=O)(=O)CC1 c1(C(=O)NCCC2CCN(C(C3(C#C)CCC3)=O)CC2)cnc2n1CCCC2 C1(C(=O)NC(CC)COCC2CC2)CCCN(C(c2cocc2C)=O)C1 C1(c2nc(C(C)C)[nH]n2)CN(C(=O)NC(c2ccncc2)CC)CCO1 C1N=C2NC(=NC3CCC4(CC(C4)C3)C(OC(F)F)=CC(F)=CC(F)=CN2)NC(Cl)CC1 c1(C(N(C)CCNC(c2ccc(O)nc2)=O)=O)cc2cc[nH]c2cn1 C1(NC(c2n(CC)c(O)nc2)=O)CC12CCN(C(c1cnc(O)c(C)c1)=O)CC2 C(=O)(CCCCCCNC(=O)C(C)(O)CC(C)C)NCC(CC(C)C)N(C)C c1(SCC)nc(N2CCCCC2CO)cc(C)n1 c1(SC)ccc(Nc2ccc(OC(=O)CSc3ccccc3)cc2)c(C)c1 c1(C(=O)NCC2C(NC(c3c(C)sc(O)n3)=O)CCCC2)cc(O)c(F)cc1N N(C1CC(O)c2ccccc21)CC(n1cc(-c2cc(F)ccc2F)nn1)C C(=O)(C(C)C(C)S(C)(=O)=O)NC1CN(C(C(C2CCOCC2)C)=O)CC2(C1)CC2 c1(C(N(C)CC2N(C(CSc3c(C)cccc3)=O)CCC2)=O)nccc(C)c1N N1(C(c2c(CC)occ2)=O)CCN(C(=O)COC(=O)CO)CC1CCO Cc1nc(C(C)NC(=O)NCC2(F)CN(C(=O)CO)C2)c(C)o1 N1(C(c2c(CC)nc[nH]2)=O)CCCCCC1CNC(c1ccc(CO)cc1)=O CC1CN(C(=O)CCF)CC2(CCN(C(C3CCCS(=O)(=O)C3)=O)C2)O1 N1(C(C(CCC)C)C(=O)NCCC2CC2)CCN2C(=O)OCC2(C)C1 C1(CC(=O)N(CC)Cc2cc[nH]n2)CN(C(c2ccnc(O)c2)=O)CCO1 C1(CC(=O)NC2CCC3(CC3)C2)C2CN(C(=O)CCc3ccccc3)CC12 N1(C(=O)Cc2cccc(F)c2F)CCOC2(C1)CN(C(=O)C(O)CCl)C2 CCCC(C)(C)CC(=O)NCCC(O)CNC(c1cnn(CCF)c1)=O C(=O)(NNC(=O)C(CC)n1cccn1)c1ccc(-c2ncn(C)n2)cc1 N1(C(c2ccc(C(C)(C)C)cc2)=O)CCC2(CC1)CCN2C(C1(Br)CCC1)=O c1(C(N2CCC(C)(CNC(C3CC(=O)N(O)C3)=O)C2)=O)ccc(Br)cc1N C1(C(N2CC(CC(C)NC(=O)C=C3CCCC3)C2)=O)COc2ccc(O)cc2O1 N1(C(C(C2CCC2)OC)=O)CC2CC(C1)CN(C(C1CCC3(CCC3)O1)=O)C2 CCC1CC(=O)c2ccc1cc2.C(=O)(C(C1CCC1)OC)NC1(CN)CC1 N1(C(c2cc(C(C)=O)oc2C)=O)CCC(CO)(NC(c2csnn2)=O)CC1 C=CCC(C(=O)NCC(CC(F)(F)F)NC(c1cc(C2(C)CC2)on1)=O)C(C)C CCC(C(=O)NCCCF)NC(c1csc(CO)n1)=O c1(CN2C(C)(C(N3C(C(=O)OCC)CCC3)=O)CC2)ncccc1Cl C12CCC3CCC1N3C(=O)COC1CN(C1)C2=O.C1(OCC2CC2)CCCC1 CONC(=O)C(=O)N1CCCC1C(C)(C)C(=O)NCC(O)CF c1(-c2cn(CC(=O)OCC)nn2)ccn(C)c(=O)c1.C12CN(C1)C2=O c1(OC)ccc(-n2ccnn2)c(CN2CCOCCC2C(=O)O)c1 Cc1cc(C(=O)NC2CC(NC(=O)COC3CCOC3)C(O)C2)cc(C)c1 c1(C(=O)OC(c2ccccc2N)C(=O)OC)cnc(SC)n1-c1ccccc1 C(=O)(CC(C)P(C)(C)=O)N1CCCC(N(C(c2c(C)oc3ccccc32)=O)C)C1 C1(NCc2ncc(CNC(=O)OC(C)(C)C)o2)CC2C=CC1CC2 N(C(=NCCOc1ncccn1)NCC(F)F)C(c1ccon1)C n1(CC)nc(C)c(C(N2CC(NC(=O)CCC(C)OC)C(C)(C)C2)=O)c1C(F)F N1(C(C(CC2CCOCC2)NC(=O)C(C2CCOCC2)F)=O)CC2(CC(CO)C2)C1 C(=O)(C1=C(Cl)CCOC1)N1C(COC)(CNC(=O)C(C)NS(C)(=O)=O)CCC1 C(=O)(C(O)C(C)(C)C)N1C(C)CC(NC(CNC(c2ccc(OC)cc2)=O)=O)C1 C1(CC(N2C(C(C)NC(=O)CSS(C)(=O)=O)CCC2)=O)C=NN(C)C1=O C1(C(=O)NC2CCC(NC(CNC=O)=O)C2)CC(C2CCOCC2)=NO1 CC(C)(C(=O)NCCCN(C1CC1)CC1CCOC1)C(N)=O CC(C)CC(CC(=O)N(CCNC(c1ncc(F)cn1)=O)CC1CC1)CC(N)=O N1(C(C2C(C)C2)=O)CCCC2(CCN(C(c3ccccc3C(F)(F)F)=O)CC2)C1 C1(NC(C(C)CC2CCC2)=O)CCCC1(C)NC(=O)CSCc1ncc[nH]1 c1(C(=O)NCCCN(C(C)C)C(C2C3CCCC23)=O)cncc(N)c1 C1(CC(=O)NC2CC(NC(CCOCCOCCOC)=O)C2)CCCC=C1Br S(=O)(=O)(c1ccc2nc(O)oc2c1)N1CCC(F)(C(=O)Nc2ncc(Br)c(O)n2)C1 C1(CNC(C2N(CC)CC2)=O)COCCN1C(c1coc(C(F)F)n1)=O c1(C(N(C2CCN(C(=O)COC3CC(F)(F)C3)C2)CC)=O)cnc2[nH]cnc2c1 Cc1nnc(N2CCN(CCNC(=O)CC(C(F)F)N3CCCC3)CC2)nc1C C(=O)(N1OC2CCC1CC2)C1OCCN(C(c2c(C)nc(O)cc2)=O)C1 CC(C)CC(O)C(=O)N(C1CCN(C(c2cccc(O)n2)=O)C1)CC1CC1 C1(C(N(C)CC2CCN(C(C(CC)N(C)C)=O)C2)=O)CC(F)C(=O)N1 CC1CCN(C(=O)C(F)F)C1CNC(=O)CC1(O)CCOC1 c1(C(=O)OC)ccc(CC(=O)NCC(O)CNC(=O)CC(C)(C)CC)cc1F C1(C(N2C(CNC(c3ccns3)=O)CC(F)C2)=O)CNc2ccccc2O1 C1(CNC(C2COCCO2)=O)COCCN1C(c1cccc(C(F)F)c1)=O c1(C(C)C)ncc(Cl)c(C(=O)NC2(C)CN(C(=O)C(c3cccnc3)O)C2)n1 c1(CC)ccc(C(=O)NC2CC23CC(NC(=O)C(c2nc(C)cs2)C)C3)cc1F N1(C(c2cc(OCC)ncc2)=O)CCN(C(C2(C3CCCO3)CC2)=O)C(CO)C1 C(C(C)(C)C(=O)NCCC(=O)NC1(CO)CCC1)NC(CC(C)C)=O.C(=O)(CO)N c1(OC)ccc(C2CCCN2C(c2c[nH]nc2-c2cnccn2)=O)cc1 S(=O)(=O)(CCN=c1[nH]c(=NCCC(C)(C)CO)[nH]c2c1COC2)NC(C)C c1(C(=O)NCCNC(CC(CCC)O)=O)cn(CC#N)c2ccccc12 c1(C(N2CC(NC(c3ccccc3C3CCC3)=O)C(O)C2)=O)cnc(O)c(F)c1 c1(OC)cc(C(=O)NC2C(CNC(c3cc(OC)nn3C)=O)C2(C)C)ncn1 N1(C(c2cccc(C)c2Cl)=O)CCC(CNC(=O)C(C)C2CCC2)C(F)(F)C1 Cc1cn2c(C(=O)N(CC(C)(C)CNC(c3sccc3C(F)F)=O)C)cnc2s1 C1(CNC(C(C(C)C)O)=O)CC2(CCN(C(=O)CCNC(N)=O)CC2)CO1 n1(CC2N(C(=O)Cn3cncn3)CC2)ccc(CNC(=O)CCc2cnco2)n1 C1(C)(CC(=O)NCCC(C)NC(c2nscc2Br)=O)CCCCC1 C#Cc1cnn(C)c1C(=O)NC(C)C=CC(=O)NCC1CCCOC1 C=C(Cl)CC(C(=O)NCCC1CC1)NC(=O)CC(C)F C(=O)(CCCN=c1nccc[nH]1)NC(C1CCCCC1)C(C)NC(=O)C(F)F N1(C(C2CCC(OC)CC2)=O)CC(CC(=O)NC2CCC23CCCC3)C2(CC2)C1 N1(CCCCCCC=C)CCCCCC1C1CCCO1 C1(=CC(=O)NC(C(=O)NCCCCN2CCC2)C2CC2)CCSCC1 N1(C(C(C(C)C)NC(c2cnn(CCF)c2)=O)=O)CCC(C)C(F)(F)C1 N1(C(CCNC(C)=O)=O)CCC2(COCC(CNC(=O)CN=S(C)(C)=O)O2)C1 n1(CC(=O)NCCN(C(c2cncc(OC)c2)=O)C)ccc([N+](=O)[O-])n1 C1(CCC(C)(C)NC(C(C)O)=O)CCN(C(=O)CCc2nc[nH]n2)CC1 N1(C(C(CC=CC)C)=O)CCC2(C1)CN(C(c1cccnc1SC(C)C)=O)C2 c1(OC)cc(CNC(c2ccc(C)o2)c2nnnn2CC2CCCO2)cc(Cl)n1 c1(OC)cccc(C(N2CCCC(C(N3CCC(Br)C3)=O)C2)=O)c1Cl C(=O)(CCC(C)(C)[N+](=O)[O-])N1CCC(c2cn(Cc3nccc(OC)n3)nn2)CC1 C#Cc1cccc(NCC(=O)NCC2CC(F)CN2C(=O)C(C)=C2CCCC2)c1 N1(C(C(CC)N(C)C)=O)CCC2(NC(c3scc(Cl)c3Cl)=O)CCCC12 c1(C(=O)NCCCN(C(CC2CC(=C)C2)=O)C2CC2)ccc2c(c1)CC(C)(C)O2 C1(NC(=O)C=Cc2cscn2)CCSC12CN(C(=O)CSCC1CCCCO1)C2 Cc1cc(=NC(C)c2csc(C)n2)[nH]c(=NCc2ncsc2C)[nH]1 Cc1ccc(N2CCCCC(NC(c3cnn(CC(F)F)c3)=O)C2)c([N+](=O)[O-])c1 C1(OC(c2cn(CCS)nn2)=O)C2CCC(C2)C1CCO N1(C(C2CC(NC(=O)OC(C)(C)C)C2(C)C)=O)CC(C)(C)CC1CC(=O)O C1(C(=O)NCCC(C)CCNC(=O)CNS(C)(=O)=O)CCC2(CC1)CC(O)C2 c1(C(=O)NC2CC(NC(c3c(N)cncc3)=O)C2)cnc(O)c2ncccc12 CC1CCCC=C1C(=O)NCc1ccc(CNC(C2CCS2(=O)=O)=O)cc1F CN1CCC(C(=O)NC2CC3CC2N(C(=O)C(C)(C)N(C)C)C3)CC1=O C(C)(c1ccsc1)=CC(=O)NC(CNC(COCC(=O)OC)=O)C(C)C C1(N)CC2CN(C(=O)C(c3ccc(O)cc3)(C)C)CC12.CC1CC(C(=O)C2CC2)CO1 c1(CN(C(=O)NC)CC2(O)CN(CC(=O)NC3CC(C)=NO3)C2)ccccc1 c1(OC)ccc(C(C)C(=O)N(C2CCN(C(=O)C(C)O)CC2)C)cc1 C1(C(N(CC(CNC(C=C(C)c2cccs2)=O)C)C)=O)CCn2ncnc2C1 C(CCN(C(=O)CC1CC1C)C)(C(C)C)NC(CC(=C)C)=O C1(COC)(CNC(c2cc(C(F)F)ncn2)=O)CCCN1C(C1CSC(C)=N1)=O C1(NC(=O)CN2CCNC2=O)CC2CC(C1)N(C(=O)CCN1CCC(F)C1)C2 Cc1cc(C)c(C(=O)NC(CCC2CC2)C(=O)N2CCOC(CC(N)=O)C2)o1 C12(C(N(C)CC3C4CN(C(C(C)SC)=O)CC43)=O)CC(C)(C1)OC2(C)C C(CCCC(=O)NC1CC(C(F)C(=O)NCCOCCCF)C1)OC(C)=O C(=O)(CCC(C)(C)c1ccccc1)N1C(CNC(CC(C)CN(C)C)=O)CCC1 N1(C(C(CC=CC)C)=O)CCC(NC(=O)CNC(=O)C(C)(C)C)C(F)(F)CC1 c1(C(N2C(CN(C(CC(C=C)(C)O)=O)C)CCCC2)=O)ccc2c(n1)CCOC2 c1(CC)c(C(=O)NC2CN(C(C34CC(F)(C3)C4)=O)CC2O)nnn1C C1(C(N2CCC(NC(=O)CSCC(F)F)C(F)C2)=O)CC12CCCCCC2 C(=O)(CCCCC(N)=O)NC1(C(=O)NCC2CC(OC)C2(C)C)CSC1 C1(C(N2CC(CNC(CCCN(C)C)=O)C(O)C2)=O)CC2CCC1C21CC1 C1(CNC(=O)CCn2cnnn2)CCC(NC(c2coc(C(F)F)n2)=O)C1 N1(C(C(C(C)O)NC(Cn2c(C)ccn2)=O)=O)CCC(O)C(O)C1 c1(C(=O)NCC(C)N(C(CCC(=C)Cl)=O)C)cc2cc(Br)cn2c(O)n1 Cc1cnc(C(N2CCC(C)C2C(=O)NC2(C)CCC(C)(C)C2)=O)cc1C C(=O)(C(F)C1CCC1)C=O.C(C(=O)NCCOCCNC)N(C(C)=O)C Cc1cnn(C)c1C(c1nnnn1C)NCc1nc(Br)cs1 Cc1cccc(-c2cn(CC(=O)N(C)CC3COCCO3)nn2)c1Cl c1(C(=O)NCC(CC)NC(C(C)OCC#C)=O)csc2c(Cl)cccc12 CCCC(C(=O)NCCN(CC(C)O)C(=O)COc1cn[nH]c1)N(C)C C1(N(c2cc(I)c(C)cn2)C(C(C)NC(CC)=O)=O)C(C)OCC12CCNCC2 CCC(CC(=O)N(CC(=O)NCc1cncc(CO)c1)CC1CC1)SC c1(C(N=c2cc(CC)o[nH]2)=O)ccc(Br)c2ncccc12.C12C=CCN1OC2=O C1(C)(CNC(CCC(=C)C)=O)COCCN(C(=O)C(C2CCCCC2)F)C1 c1(C(N(C2CCN(C(C3CCC(O)CC3)=O)CC2)CC#C)=O)ncc(Cl)cc1F N1(C(C2CC(C)C2)=O)CC(NC(=O)C=CC(=O)N(C)C)C(Cc2ccccc2)C1 CS(C)(=O)=NC(=O)C1CCN(C(C2CNCC2F)=O)CC1 N1(CC)CCC(C(N2CC(CC(=O)NC3CC(CCC(N)=O)C3)(OC)C2)=O)CC1 C1(NC(c2ccc(CC)cc2F)=O)CN(C(=O)CCCN(C)C(C)=O)CCC1(C)C C1(c2n(-c3c(OC)cc(F)cc3)nc(CCO)n2)CC2(CCCC2)C(=O)O1 C=CCCCCC(c1nnnn1CC1CCOC1)NCc1coc(C)n1 c1(CN(CC(F)(F)F)C)ccc([N+](=O)[O-])c(F)c1F.C12CN(CC1C#N)C2=O N1(C(c2cnnn2C2CC2)=O)CC2(CCCN(C(C3CN4CCN3CC4)=O)C2)C1 N1(C(c2c(C)n[nH]c2C)=O)CC2(CCC2NC(=O)CCC(F)(F)F)C1 N1(C(CCc2c(C)noc2Cl)=O)CCN(C(=O)CCCN=[N+]=[N-])C(CCO)C1 CN1CC(C(=O)NCC2COCCN(CCS(C)(=O)=O)C2)c2ccccc2C1=O N1(C(CC(CCC)C)=O)CCCC2(CCCN2C(c2ccoc2CC)=O)C1 C1(C(=O)NC(C=C)(C)C)C2CCCC2CN1C(=O)C(C(C)C)C1CCC1 N1(C(C(C)NC(C)(C)C)=O)CCCC2C1CCN2C(c1scc2c1CCCC2)=O C1(C(=O)NC(CNC(c2ccn(C)c2)=O)C(C)(C)C)Cc2cc(Br)ccc2O1 c1(CCC)cccc(C(=O)NC2CCCC2CNC(=O)CC2C(CC)C2(F)F)c1 CC(CC(=O)NCCNC(c1cc2ccncc2[nH]1)=O)CC(F)(F)F C1(NC(c2c(C)n[nH]c2)=O)CCN(C(C2(c3ccccc3F)CC2)=O)CC1O c1(C(N2CC(NC(C3CC4(C(OC)CC4)C3)=O)C2)=O)ccc(F)c(C)c1N c1(C(=O)NC2CCCN(C(c3c(C)oc(CO)c3)=O)CC2)n[nH]c2c1CCSC2 CCCC(CCC)CC(=O)NCCN1CCN(C(=O)CCc2cccn2C)CC1 c1(C(C)(C)C(=O)N2CC(NC(C3CC3Cl)=O)C2)cccc(N=c2cncc[nH]2)c1 N1(C(c2cnc(CC(C)C)[nH]2)=O)CCCC(NC(c2nnc(O)cc2C)=O)C1C c1(NC(C2CCC(NC(Cc3cc(C)[nH]n3)=O)C2)=O)cn(C)c(C(N)=O)n1 c1(CCC(=O)NC(C2CCN(C(=O)CC3CC3C)C2)C)ccc(F)cc1F c1(OC)cc(=O)n(C)cc1C(=O)NC1CCN(C(c2ccn3ccnc3c2)=O)C1 C(=O)(C(C)CC(N)=O)N1CC(C(N(c2cc(C)nn2C)C)=O)NCC1 c1(CC)cnccc1C(N1CCC(C(C)C(=O)NC(C)(COC)COCC)C1)=O C(CCC(N)=O)(C(=O)N(C)CCN(C(=O)C1=COCC1)C)n1cc(CCCO)nn1 C(=O)(CCC(C)(C)C)N(CCCNC(=O)C(C)(CSC)NS(C)(=O)=O)CC c1(C(=O)NCC2N(C(c3c(Cl)cn(CC)n3)=O)CC2)cnc2n1CCC2 O(S(=O)(=O)c1ccnc(CO)c1)c1ccc(C(CC)=O)cc1C c1(C(=O)NCC2C(NC(C3N(CC)CCC3)=O)CC2)cc2c(C)sc(C)c2s1 CCC(C)(C)CC(=O)NCC1CC(C)N(C(=O)CC2(CO)CC2)C1 c1(C(=O)NC(C(=O)NCCCCC=C)CC#C)cccc(C)c1F c1(CNCC2(C(N(c3ccn(C)n3)C)=O)CC2)c(Cl)cccc1Cl C1(C(=O)NCCC2(NC(=O)Cc3cccnc3O)CCCC2)CCC(F)(F)CC1 Cc1conc1C(=O)NCC1COC(CNC(C2CCSCC2)=O)C1 CC(C)(CCCNC(C1CC1)=O)C(=O)N1CCCC(C(C)(C)C)C1 c1(NC)ccc(F)cc1C(=O)N(C1CCC(NC(C2(C(F)F)CCCC2)=O)C1)C C1(C(=O)NCC2CC(NC(C(C)SC)=O)C2)CCCNS1(=O)=O N1(c2cc(N(C)CC3CCC(=O)N3)nc(C(F)(F)F)n2)CCC(C2CCC2)C1 N1(C(C2(CC#C)CCCC2)=O)CC2CC(NC(=O)C(C)(C)CC3CC3)CC1C2 C1(CCNC(=O)CCN2CCCC2)CCN(C(C2SCCCS2)=O)C1 Cc1c(C=CC(=O)NC2(CN(C(=O)CCc3cnc[nH]3)C)CC2)cnn1C N1(C(c2c(C)nn(C)c2)=O)CC2CCC2(NC(C2Cc3nccn3C2)=O)C1 C(=O)(CC1=NNC(=O)C1)NCC(C)(C)CNC(c1ccc2ccnn2c1)=O CC(C)CC(C)CC(=O)NC(C)CNC(c1ncc(Br)cc1O)=O N1(C(CSCCC#N)=O)CC2CCCC(C1)N(C(c1cc3[nH]ccc3s1)=O)C2 c1(CC(N2CC(C)(OCC(=O)NCC(C)N(C)C3CC3)C2)=O)nc([N+](=O)[O-])n[nH]1 C1(C(N2CCC(OCC#C)C2)=O)CCCCN1C(=O)CC1CCC(=O)N1 Cc1ccccc1COCC(=O)NCC=CCNC(C1CCCC(C)C1)=O c1(C(N2CCC(NC(COCC)=O)C(CC)C2)=O)ccc(OC)c2ccncc12 N1(C(CSCCOC)=O)CCC(O)C1C(=O)Nc1sccc1Cl C1(NC(c2cccc(C3(C(=O)OCC)CCC3)c2)=O)CCOCC1(C)C C(C)(CCN=C(NCCC(=O)N(C)C)NCC1(C)CCC(=O)N1)OC c1(NC(c2c(CC)ccs2)=O)cccc(NC(c2cnc(C3CC3)[nH]2)=O)c1 C(=O)(CS(=O)(=O)CCO)NCC1(COC)CCN(C(=O)CC2CCSCC2)CC1 C1(C(N2CC(CNC(c3c(C)nc(C(C)C)o3)=O)OCC2)=O)CNC(=O)CC1C Cc1nc(CC(=O)NCC(C(C)C)NC(C2CCC(C)(C)C2)=O)c(Cl)s1 c1(CC(=O)NCCN(C(=O)C(C)N(C)C)CC)c(N)nc(C)nc1O C(=O)(CC(C)(C)C(C)(F)F)NC(C1CCCCC1)CNC(C(F)OC)=O c1(C(=O)NC2CCN(C(=O)CC3CCOC3)C2)cccc(C(F)(F)F)c1 c1(CCC)c(C(=O)N(C2CCN(C(=O)CS(=O)CC)C2)CC)[nH]c(C)c1CC C1(CC(C(=O)OC)O)CCN(Cc2cn(CC(C)=O)nn2)CC1 N1(C(C2(C#N)CC2)=O)CC2CCC1CN(C(c1cc(O)n[nH]1)=O)C2 N(C1CCC(Nc2ncnc3[nH]cnc23)c2ccccc21)C(CCC(=C)C)=O N1(CCSCC)C(=O)NC(c2nnc(Br)n2C)C2=C1C(C)N(C)C2=O CC1CCC2N1C2=O.c1(N)cc(C(F)(F)F)c[nH]1.C12(CCC1)NC2 CCCCC(CC)C(=O)N1CCOCCC1C(N1CC(O)(c2ccn[nH]2)C1)=O C(=O)(C1CCCc2nn[nH]c21)N1CCC(CNC(CCSCC)=O)C(F)(F)CC1 n1(CCC#C)c2nnc1CCN2C.C1(NC(C)C)CC(F)(F)C1OC C1(C(=O)NC(C(C)NC(=O)C=Cc2cnn(C)c2)CO)CCS(=O)(=O)C1(C)C C(=O)(C(C)C(F)(F)F)N1C(C)CCC1.C1(CC)CC(CNC(=O)N(C)CC)(CC)C1 c1(CC)cc(C(=O)NCC(C2CC2)N(C(=O)C(C)(C)c2cc[nH]n2)C)sc1C C1(C(=O)OCC)CN(C(C2C(CN=[N+]=[N-])C2(C)C)=O)C(C)(C)CO1 CC1CC2(CCO1)CC2C(N1CC2(C1)SCCC2NC(c1cc(C#N)c[nH]1)=O)=O N1(C(c2cc(C)sc2)=O)CCOCC(CNC(=O)CN(c2ncccn2)C)C1 c1(C(=O)NCCN(C(CC2CC(=C)C2)=O)CC)c[nH]c2cccc(Cl)c12 CCC(C)CC(C(=O)N1C2CCC1COC2)NC(=O)C(=O)NC(C)C S(=O)(=O)(c1ccc(I)cc1)N1CC(COC)N(C(c2cccc(CO)c2)=O)CC1 C=C1c2ccccc2C(=O)N1CC(N1C2CCC1CC(NC(=O)COC)C2)=O c1(COC)cc(Cl)ccc1CNCC1CCCC1N(C)C Cc1cc(C(=O)NCC2CCN2C(=O)C2=CC(C)CC2)c(C)n1Cc1cccs1 c1(NC(CC2C(C)CCCN2C(=O)Cc2cnnn2C)=O)ccc2c(c1)CCO2 c1(NC(C(C2CN(C(=O)CC3OCCC3C)C2)OC)=O)conc1C(C)C c1(NC(C2COCCN2C(c2ccc(S)cc2)=O)=O)cc([N+](=O)[O-])c(F)cc1Cl C1(CC(=O)OC)CC(CC)=NO1.C12(CCCC1)CC(=O)N1CC(CO)(C1)OCC2 c1(C(N(CC(Cc2ccccc2)NC(C(C)OCC#C)=O)C)=O)ccn(CC)n1 C(CCC)(C(O)C(=O)N1CCCCC1CO)NC(COCCCCC)=O C(C)(CCC(=O)NC1C=CC(CNC(=O)CC2CCCOCC2)C1)OCC CCCCC(O)C(=O)NCCCN(C)C(c1cn(C)c(=O)cn1)=O C(=O)(CCCCN=[N+]=[N-])NC(C(=O)N(C(C#C)C1CCC1)C)c1cccs1 C1(C(N2CCC(C)(CCO)C2)=O)(CC)CCCN1C(=O)CC1CC2CCC1O2 C1(C(=O)NC2(C)CN(C(c3n[nH]c4c3CC3CC43)=O)C2)Cc2ccccc2O1 O(NC(=O)C(CNC(=O)C=Cc1ccncn1)OC(C)(C)C)CC(C)(C)C CCC(C)(C(=O)NC1COCC1CNC(c1sccc1SC)=O)C(F)F c1(OCC)ncccc1NC(=O)NC(C)(C)C.c12cccc(c1)C(C)(C)N2 C(C(=O)NC(C)C=CC(=O)Nc1ccn(C(C)C)n1)(C(C)C)SCC N1(C(=O)CCc2ccoc2)CCN(C(C2C3(CC3)C23CC3)=O)C(CO)C1 c1(CNC(CCCOC)=O)cc(C(=O)N(C2CCC(C)C2)C2CC2)ccn1 C(=O)(CC(C)C(C)(C)NC(c1sccc1C)=O)NCC(COCC)C C1(NC(C(n2c(C)ccn2)C)=O)CN(C(C2(CF)CC(=O)C2)=O)CCC1C C1(CNC(c2c(C#C)c[nH]n2)=O)CN(C(=O)CC2CC=CCC2)CC2(CCC2)O1 CC(C)(C)C(CO)C(=O)NCCCC1(NC(C2CCc3cncn3C2)=O)CC1 O=C(CC1OCCc2ccccc21)N1CCC1CNC(=O)COC1CCCOC1 c1(C(C(=O)N(C)CCC2CNC2)N)ncc(CC2CCCO2)s1 O=C1CC(C(=O)NCc2cc(C(N3CCOCC3C(F)F)=O)ccn2)CCN1 C1(C(N(C2CCN(C(CC(COC)(C)O)=O)CC2)C)=O)CCC2(CCOCC2)O1 O=C1CCOC(C(=O)NCC2C3CN(C(C4(C(F)F)CCCC4)=O)CC23)C1 c1(C(=O)NC2CCC(CNC(=O)CC3CCOC3)CC2)cc(Cl)ccc1[N+](=O)[O-] C1(C(=O)NC2(COC)CN(C(C3CC34CCC4)=O)C2)CCC(C)CC1 c1(N(CCC)CCNC(c2c[nH]nc2C(N)=O)=O)ncc([N+](=O)[O-])c(=N)[nH]1 c1(C(C)C)cnc(Cl)[nH]c1=NCC1CCCC(NC(c2nc(O)nc(O)c2F)=O)C1 N1(C(c2ccn(CC(C)C)n2)=O)CCCC(C)C1CNC(c1c[nH]c(=O)cn1)=O Nc1c(C(=O)NC2CC2CNC(=O)C(c2ccc(F)cc2)O)ccc(Cl)c1Cl Cn1ccn2c(C(=O)NCC3(C(=O)O)CC(O)C34CCC4)nnc2c1=O C12CN(CCO1)C(=O)Cn1cc2nn1.CS(=O)(=O)N(C1CC1)CC1(F)CC1 CCC(C)C(C)C(=O)NCC1CC(NC(c2ccncc2NC(C)=O)=O)C1 Cc1conc1C(=O)NC(C(=O)NC(Cc1cnc[nH]1)CO)c1ccco1 c1(C(C(=O)NCC2N(C(Cc3c(C)scn3)=O)CC2)(F)F)ccc(F)cc1F CC1=C(C(=O)NCC2(CO)CCN(C(=O)CNC(=O)CC3CCCC3)C2)CC1 C(C(C(=O)NCC1CC1(F)F)C(C)(C)C)NC(Cn1nc(C)oc1=O)=O N1(C(CCCCSC)=O)CC(C2CN(C(=O)C=Cc3ncc(C)[nH]3)C2)C1 CCC(C)(C#N)C(=O)NCC1CC(C(F)(F)F)CN1C(=O)CSC(F)(F)F C1(CNC(=O)CC2CCCC(=O)N2)C(C2CC2)CCN1C(=O)CCCCO C12(C(N3CC(C)=C(C)CC3)=O)CCCC1N(C(=O)OC(C)(C)C)CC2 c1(C(N2C(C(=O)Nc3c(OC)ccc(C)c3)C=CC2)=O)c(Br)cc(Br)c(O)c1Br N1(C(c2n(C(C)C)ccn2)=O)CC2CCCC(CNC(c3coc(Cl)c3)=O)C2C1 c12cccc3c1CN(CC3)CC(=O)N2.c1(C(N(C)C)=O)ccoc1I N1(C(c2c(CC)nc[nH]2)=O)CCC(NC(C2(C)CC2(F)F)=O)CC(O)C1 C1(CNC(CC2(OC)CCC2)=O)CCN(C(c2csc3nnsc23)=O)C(C)C1 C1(C(N2CCC(C(C)NC(=O)CN(C3CCC3)C)C2)=O)CCc2n[nH]cc2C1 N1(C(C(C(CC)CC)OC)=O)Cc2nccn2CC(NC(C2CC(F)(CF)C2)=O)C1 N1(C(CCC(C)=O)=O)CC2CCC1(CNC(c1ccc(CC(C)C)cc1)=O)CC2 c1(CC(=O)N(C(C)CNC(=O)CCN2CCC(F)C2)C)ccc(F)c(Br)c1 C1(CC)CC(C(N2CCC(N(C(c3cscc3COC)=O)CC)C2)=O)CC(=O)N1 N1(CC)CCCC(C(=O)NCC2CC(NC(=O)C(C(C)C)SCC)C2)C1 Cc1cc(Br)cc(C)c1S(=O)(=O)NC(CO)CC(C)(C)C c1(C(N2C(CCNC(C=CC(CC)=CC)=O)CSCC2)=O)cnn(CC)c1Cl C1(CC(=O)N(C2CN(C(=O)C3=CCCSC3)CC2(C)C)C)CCCNC(=O)C1 C1(n2cc(CCOCC(=O)OC)nn2)CCC(C)(C)N(C(=O)C(N)=O)C1 CC(C)C(C(=O)NC1CCN(C)CC1)NC(=O)C=CC1(C)COC1 c1(C(N(CC(C)NC(c2cscc2SC)=O)CC)=O)cnn(CC)c1Cl c1(CC(=O)NC2(CCNC(C3(c4cc[nH]n4)CC3)=O)CC2)c[nH]c2cnccc12 c1(C(=O)OC)cc(C(=O)NCC2(O)CN(C(=O)C(C)N3CCC3)C2)ccc1OC c1(CC)cccc(C(N2CC(NC(c3cccc(-c4cn[nH]c4)c3)=O)C2)=O)c1N C1(NC(C(COC)NC(C)=O)=O)CC2CCC(C1)N2C(C1CC(=C2CCC2)C1)=O Nc1c(C(=O)NC2CCN(C(c3cncs3)=O)CC2)cccc1F C1(CCOC)(NC(C2(F)CCOC2)=O)CCN(C(=O)C(COC)NC(C)=O)CC1 CCCCC(C(=O)NC1C2CCCCCC12)NC(c1cn(C)cn1)=O Cc1c[nH]cc1C(=O)NC1C=CC(CNC(C2CC(n3cnnc3)C2)=O)C1 c1(C(=O)NCC2(OC)CN(C(=O)CCOCC(C)C)C2)cn(C)c(=O)cc1C c1(C(N(C(C)CCNC(=O)C(C)(C)c2ccno2)C)=O)coc(S(=O)(=O)NC)c1 c1(OCC(=O)NCCC2(NC(C3CCCOCC3)=O)CC2)nc(O)nc(O)n1 C1(C(=O)NC(C=CC(=O)N(CCC)CC)C)CN(CC)C1 C(C)(CC(=O)NCc1cccs1)(C(F)(F)F)NC(=O)CSCC1C(C(C)(C)O)C1 c1(C(=O)NCC(C)CN(C)C(C2CC(=O)NC(=O)N2)=O)cccc2c1CCCC2 C(C)(C(C)C(=O)NCCOCCCO)NC(CCSC)=O C1(CNC(C#CC(C)(C)C)=O)COCC2(CCN(C(C3CCNC3=O)=O)CC2)O1 Cc1cccc(C(=O)NC2(C)CCCC2NC(=O)CSCc2ccccn2)c1 c1(C(=O)NC(CN(C(=O)CC2CSC2)CC)C)cc(C)nc(O)c1[N+](=O)[O-] N1(C(c2cc(C)c(Br)o2)=O)CCC(CO)C(NC(=O)C(=O)N(C)C)C1 C12(CNC(CCN(C)C(C3CC(C(C)(C)C)C3)=O)=O)CCC(C1)C2 C=CCCCCC(=O)NC(C)CCCNC(=O)CC(C)(C)COC C1(C(=O)NC(C(C)NC(=O)COc2cccc(Cl)c2)(C)C)CC(S(C)(=O)=O)C1 c1(CNC(C(=O)N(C2CC(OC)C2(C)C)C)=O)ccc([N+](=O)[O-])c(Br)c1 N1(C(=O)NC(C(c2ccc(OC(C)C)cc2)O)C)CC23CCCC2(COC3)C1 S(=O)(=O)(c1cccs1)N(CC(=O)NC1CC(NC(c2cnccn2)=O)C(O)C1)C c1(NC(c2ncc(C)o2)c2nnnn2CC2CC2)cccc(O)c1C C1(OC)CN(C(=O)COCC2CCOCC2)CC1NC(C1(C)CCCCO1)=O N1(C(c2ccc(N)cc2)C(=O)NC2CCCCC2)Cc2ncsc2C1 C1(CCC)CC(C(=O)N(CCC2CCN(C(=O)C3CC3)CC2)C(C)C)CCO1 C1(CC)CCC(C(=O)NC2CCC(C(=O)NCCCC(=O)N(C)CC)C2)CC1 c1(NC2(c3n(CC=C)nnn3)CCCN(C(C)C)C2)ccc(Cl)c2c1CCC2 c1(NC(=O)NCC2CNCCOC2)cc(Br)c(F)cc1I Cc1cccc(C2(C(=O)N(C(C)CNC(=O)C=CC(=O)OC(C)(C)C)C)CC2)c1 N1(CCC(=O)NCC(C)CN)CCN(c2cccs2)CC1 c1(SCCCC(=O)NCC(C)N(C(=O)CSC2CC2)C)nc2ccccc2[nH]1 N1(C(CC(CC)NC(=O)COc2ccsc2)=O)CCCC2C(=O)NCC12 c1(C(=O)NCCC2CN(C(C34CC(CC)(C3)C4)=O)C2)nc(C)ncc1Br Nc1cccc(C(=O)NC2CC(NC(c3cnn(-c4ncccn4)c3)=O)C2)n1 n1(CC)cc2ccc(C(N3CC(NC(c4c(Br)cnn4C)=O)C3)=O)cc2n1 C1(NC(C2C=CC(CNC(CC3(N(C)C)CC3)=O)C2)=O)CCS(=O)(=O)C1 c1(OC)ccc(C(=O)NCC(N2CCC(C)(C)C2)(C)C)c(F)c1F Cc1cncc2cc(C(=O)N(C3CCC(NC(c4ccc(Cl)[nH]4)=O)CC3)C)sc12 N=c1ncn(CCC(=O)NCC2CCC2NC(=O)Cc2nnc(O)s2)[nH]1 N1(CCC(=O)N(CCCN(C)C)C)CCNCC1 c1(OCC(=O)NCCN(CCC)C(c2ccccc2C(F)F)=O)cccc(F)c1 CCCS(=O)(=O)C(C)C(=O)N1CC(CN(C(=O)CS(=O)CC)C)C1 C1(NC(C2N(C(c3c(OC)ccc(C)c3)=O)CC(O)C2)=O)CCc2n[nH]cc2C1 n1(CC(=O)N(CCCN(C(C=CC(CC)C)=O)C)C)nc(C2CC2)cc1C(F)F c1(OC)ccc(CN(C)CCc2nccnc2C)c(Cl)c1OC n1(CC)ccnc1C=CC(=O)NC1CC1NC(c1csc(C2CCCO2)n1)=O N1(Cc2ccc(OC)c(F)c2)CCC(=O)N(CC(F)(F)CN2CCOCC2)C1=O N1(C(COCC(C)C)=O)CC(CN(C)C(C2CCSC2)=O)C2(CC2)C1 C(C(C)(C(=O)NC1CCCC1C(=O)NCC1CC(N(C)C)C1)OC)OC c1(CNC(C=CC(C)NC(CC2CC(SC)C2)=O)=O)oc(C)nc1C N1(C(c2c(CC)non2)=O)CCC(C)(CNC(=O)C(c2cncn2C)N(C)C)C1 C1(C(N(CC(C)NC(=O)Cc2cn(C)nn2)C)=O)CC12C1CC3CC(C1)CC2C3 CC(C)CCCC(=O)N1CC(NC(=O)COCC(F)(F)F)CC1(C)C C1(C(=O)NCCC(C(C)C)OC)COCCN(C(c2c(C)nsc2C)=O)C1 c1(OC(F)(F)F)cc(Br)ccc1CNC1CCC(OBr)CC1.OCCO Cn1ccc(C(=O)NC2(C)CC(NC(=O)C(F)C(F)(F)F)C2)cc1=O CCCCC(O)CC(=O)NC(CCN(C)C)C(=O)NCCC1=CCCCC1 C(=O)(CC1CC(=O)c2ccccc21)NC(C)CNC(c1csc(Cl)n1)=O CCC(CC)CCCC(=O)NC1CCC(NC(=O)C2=CCC(C)(C)CC2)CC1 CCCC1Cc2nnnn2C(C=O)CCC(CC)CCNC(=O)CO1.OC N1(NC(C2CC2C(=O)NOCCCCC2CC2)=O)CCOC(CC2CC2)C1 C1(C(N2C(CN(C(Cc3cc(CC)no3)=O)CC)CCC2)=O)CCCS(=O)(=O)C1 N1(C(C(=O)NCC)=O)CC(CNC(c2c[nH]c(C(N)=O)c2)=O)C(C)C1 c1(NC(CCCN(C)C(C2CCCC(C(F)(F)F)C2)=O)=O)ccc(Cl)cc1F Cn1cnc2cccc(C(=O)NC3CN(C(c4cscc4C(F)F)=O)CC3O)c12 N1(C(c2ccc(C)s2)=O)CC(CNC(c2cc(N(C)C)cs2)=O)C2(CCC2)C1 C(=O)(C1=CC(C)(C)C1)N(C1CCN(C(c2cn(C(C)(C)C)nc2C(F)F)=O)C1)C c1(C(N2CCC(O)C(CO)C2)C(=O)NCC2CCCC2)cnc2ncccn12 C12(NC(CSC)=O)COCCC1CN(C(c1ccnc(OC3CC3)c1)=O)C2 C(C)(C)(CCCNC(C1(C)CS(=O)(=O)C1)=O)NC(Cc1cn(C)nn1)=O CC(C)C(CNC(C1COCC1(C)C)=O)C(=O)NCC1(C)CC2CC2C1 CC1CCOC(C(N2CC(NC(=O)CCCC3CCC3)CC2CO)=O)C1 C(=O)(C(C)(C)CS(N)(=O)=O)NCC1(NC(C2N(C)C(=O)NC2)=O)CCC1 c1(N(CC(=O)N(C(CNC(C2CC2(Cl)Cl)=O)C2CC2)C)C)ccccc1 CC(C)C(CNC(c1cc(O)ccc1F)=O)C(=O)N(CCCO)CCCO c1(CC(N2CC(CC=C)(NC(=O)CSC)C2)=O)cccc(NS(=O)(=O)CCC)c1 C1(CC(=O)NCC2CN(C(c3[nH]cc(C(N)=O)c3)=O)C2)CC2(CC2)CO1 N1(C(c2c(SC)ccs2)=O)CCCCC1CCNC(=O)CC1OCCCO1 N1(CC(=O)Cc2cccnc2Cl)CCCN(C(c2ccccc2)=O)CC1 c1(C(N2CCC(=CCNC(C3(F)CCCCC3)=O)CC2)=O)cc2scnc2[nH]1 C=CC(C)(C)C(=O)NC(CNC(c1cnn(CC)c1C)=O)C(C)C C(=O)(C(C1CCOC1)NC(=O)CNC(C1CCC1)=O)N(CC=C)C c1(OC)ccc(F)cc1C(N1C(CC(=O)NC2CCCC2(C)O)C2CCCC12)=O c1(CC(=O)NCC(CC)NC(=O)CCC(=O)NC2CC2)c(F)cccc1F CC(C)(F)C(=O)N(CC(=O)NCCC1CCC(=O)N1)C1CC1 c1(CC(=O)NCC2CCCN(C(c3ccc(F)c(O)c3)=O)C2)ncc(F)cc1F C1(CC(N2CCN(CC(=O)N(C)CC3CC(=C4CC4)C3)CC2)=O)CC(O)C1(C)C CC(C)(C)CCCCC(=O)NC(C(N1CC2CSCC2C1)=O)c1ccoc1 c1(C2C(C(N3CCN(Cc4ccc(CO)cc4)CC3)=O)C2)ccc(Cl)cc1Cl N1(CCCNC(C(n2cc(C3(O)COC3)nn2)C)=O)CCC(C)(F)C1 C(=O)(CC(C(F)F)c1cccc(F)c1)NC1CCN(C(C2C(=C)C2)=O)CC1 C1(NC(C=C(CC)CC)=O)C2CCN(C(=O)C(C)OCCOCC)CC12 Cc1nn2cc(C(N3CC(NC(c4cn(CC(F)F)cn4)=O)CC3C)=O)nc2s1 C1(C(=O)NCc2nn(C)c(Cl)c2)CC12CCN(c1ncnc3cc[nH]c13)CC2 CC1(C)COC(COCC(=O)NCCCC2CCCN2C(C2CC=CC2)=O)C1 C1(C)(C(=O)NC(C)CCCCNC(c2cnc(C(F)F)s2)=O)CCCC(F)(F)C1 CCC(CN(C)C)CC(=O)NCCC1CCCN1C(c1ccc(N)cn1)=O O(C=CC(=O)NCC(C1CC1)NC(c1cnoc1CCC(F)(F)F)=O)CC c1(C(N(CC2N(C(CCCC=C)=O)CCC2)CC)=O)cccc2c(C)ccnc12 CCCC(CC)N=c1ccc(Br)c(S(=O)(=O)N(CC)CC)[nH]1 CCC(C(=O)N(Cc1ccccc1)OC)NC(=O)CNC(N)=O S(=O)(=O)(c1ccc(NC(=O)CS(C)(=O)=O)cc1)N(C)C N1(C(C(CCCOC)C)=O)CC2(CCN(C(=O)Cn3ccc(C)cc3=O)C2)C1 CC1CCN(C(c2ccc(N3CC=CC3)cc2)=O)C1CO.C12(CC1)C(=O)NC2 C1(COC)CCCCN(C(=O)C(C)(C(C)C)OC)CC1.c12noc(C)c1C(=O)O2 CC1(C)C=C(C(=O)N2CCC2C(=O)NCCCNC(=O)C(C)(C)F)C1 N1(C(C(CC(=O)OC)C)=O)CC2(C1)OC1(C)CC2(NC(=O)CCCSC)C1 C1(C)(CC)C=C(C(=O)NCC2(C(F)F)CCN(C(c3ccccc3O)=O)C2)C1 C(C(C)(F)C(C)(C)F)NC(C(N1CCC(C(F)(F)F)(SC)C1)C)=O C1(CN(C)C)CCCN(c2cc(NC(=O)Cc3cnsc3)ncn2)C1 CC1CC2CN(C(=O)C(=O)NC3CC3)CC2N1C(C1Cc2nccn2C1)=O c1(OCC)cccc2ccc(N3CCN(C(C)=O)CC3)nc12.C1C(F)(F)CC(=O)O1 C1(NC(C(=C(C)C2CC2)F)=O)CN(C(C2(C)CC2)=O)CC(C)(C)C1 N1(C(C2C(C)CCO2)=O)CCC(C2(NC(=O)CC3CCC3)CC2)CC1 C(=O)(CCN=c1ccc(C)c[nH]1)NCCC1CC(OC)CN1C(=O)C(O)C1CC1 C(=O)(CCCCCCC(=O)NCC1(NC(C2CC2[N+](=O)[O-])=O)CCOC1)OC c1(SC)cccc(NC(C2CCN(C(=O)C(c3cccn3C)=O)CC2)=O)c1 Cn1cc2c(n1)CCCC2C(=O)NC1CC(C)(NC(=O)C=C2CCOCC2)C1 CC1CN(C(C2(CO)CCCO2)=O)CCC1NC(c1ccnc(Cl)c1Cl)=O C1(C(N2CCC(NC(CCC#C)=O)CC2)=O)COCC2(CCC2)O1 C(=O)(C(C(C)(C)C)N1CCCC1=O)N(CCCNC(C1(C)CCCC1)=O)C O=C(C1=CCCOC1)NCCC1(NC(c2ccc(-n3ccnn3)cc2)=O)CC1 c1(C(N2CC(C(C)NC(C3CC3C(C)(F)F)=O)C2)=O)ccn2nccc2c1 C(C(=O)NC1CCC1CC1CC1)(C1(O)CCC1)NC(=O)COC1CC(C2CC2)C1 C=CCC(C)(C)CC(=O)N1CC(OC)C(NC(C2(S(N)(=O)=O)CC2)=O)C1 C1(C(=O)NCC2(CNC(C3(C)CC3)=O)CCCC2)CC2(C1)CC(C)(C)C2 C(c1cccnc1)=C(C)C(N1CC(N(C)C(C23CCC(C2)C3)=O)C(F)C1)=O N1(C(c2nn(C)c(C(F)(F)F)c2)=O)CCC2(NC(C3(CO)CCCC3)=O)CC2C1 Cc1ccc2c(c1)CN(C(C1CN(C(=O)CCN=[N+]=[N-])C3(CCC3)C1)=O)C2 N1(C(=O)Cc2nc(Cl)cs2)C2CCCC1CC(NC(c1ccc(Cl)cc1F)=O)C2 Nc1cc(Cl)ccc1C(N1CCCCC1CNC(C12CC(C1)C(C(F)(F)F)O2)=O)=O CC1(CNC(=O)CC23CCC(CC2)C3)CCCN(C(C2CCS(=O)(=O)C2)=O)C1 N(C1CCc2cc(CNC(=O)C(C#N)CC)ccc21)C(c1cnc(CCC)[nH]1)=O C=C=C(C)CC(=O)N1CC(F)CC1CNC(c1cc(C2CC2)nn1CC)=O N1(C(C=Cc2n(C)ncc2)=O)CC2CN(C(C3CC3C(F)F)=O)CCC12 c1(C(C)C(=O)N2CCC2N2CCCCC2C)ccccc1F CC(CC(F)(F)F)C(=O)N1CC2CC(C(N3CCCC(O)C3)=O)CC2C1 C1(C)(CNC(CC(C)(C)OC)=O)CN(C(=O)C(C)CN(C)C)C(C)(C)C1 Cc1nccnc1C(N1CC(CNC(=O)COCCCC(C)C)CC1C)=O c1(CCC(=O)N2CCC2c2cn(-c3cccnc3F)nn2)cc(Cl)ccc1Cl CC1CN(C(c2ccn(C3CC3)n2)=O)CC(C(=O)NCCc2ccco2)O1 C(=O)(C(CCC1CCC1)NC(C1CCC(=O)N1)=O)N1C(C(=O)OC(C)(C)C)CC1 C1(C(=O)NCCC(C)NC(C=CC=CCC)=O)COC(=O)N1 c1(-c2n(C(C)C(F)(F)F)nc(C3CCOC3)n2)cncc2cc(Cl)ccc12 N1(C(C2OCCN(C(C(C)=NOCC#N)=O)C2)=O)CCC2OCCC2C1 N1(C(c2cc(=O)cc[nH]2)=O)CCCN(C(c2cnsc2)=O)C(CO)C1 C1(C(N(CCCC)C)=O)CCCN(C(=O)CCC)CC1.c12cccc(c1)CC2 C#Cc1ccc(C(N2CCC(CNC(=O)C(O)CC)(COC)CC2)=O)nc1 C(C(=O)N1CCCC1CN(C(c1cc(Cl)c(Cl)s1)=O)C1CC1)(C(C)C)NC(C)=O c1(C(=O)NCC(C)(CC)NC(CC(=O)OCC)=O)cnn2c1OCCC2 N1(C(C(F)=CC)=O)CCC(C)(C)C1CN(C)CCOC.c12ccccc1NC2=O C12(NC(C(F)=CC)=O)CCCCCC1N(C(=O)CCC#Cc1ccccc1)CC2 C12(CC(=O)NCC3(NC(c4nc(OC)c(C)s4)=O)CCC3)CCCCC1C2(F)F N#CCCCCC(=O)NC1(CO)CN(C(=O)C(F)CC2CCCC2)C1 C(CCN=c1[nH]c2c(c(=NCc3ccc(N)c(Cl)c3)[nH]1)CSC2)c1cn(C)nc1 C1(C(C)(C)N(C)C(=O)NC)CCN(C(c2ccsc2)=O)CC1.c1(N)cnn[nH]1 C12(CC(=O)NCC3CC(OC)CN3C(c3nc(C)n(C)n3)=O)CC(C)(C1)OC2C C(=O)(CN=S(C)(C)=O)N1CCC(CN(C)C(c2nc(Br)c[nH]2)=O)CC1 C#CCCN=C(NCC1CCCOC1c1ccco1)N(C)Cc1cccs1 C1(C(N2CCC(CNC(c3ncoc3C3CC3)=O)CC2)=O)CCC2(CCCC2)C1 c1(C(=O)NC2CC(CNC(CC(CC)CC)=O)C2)ccc2sncc2c1 C1(CC=C)(NC(c2c[nH]nc2C)=O)CCN(C(C2CC(C(=O)OC)C2)=O)C1 c1(C(=O)NCC(C2CC2)NC(C(CCCC#C)C)=O)cccc2nn(C)nc12 c1(C(=O)NCCCOCCNC(C2N(N=O)CCC2)=O)cccc(Cl)c1[N+](=O)[O-] Cc1c(C(=O)NC(C2CCCN2C(=O)C=CC(F)(F)F)C)cnn1C1CCC1 C(=O)(C(C)(O)C(F)(F)F)N1CC2C(NC(c3c(OC)nccn3)=O)(C2)C1 C1(CNC(COCC(C)C)=O)CN(C(=O)C(O)Cc2ccccc2)CC1(C)C c1(CN2CCCC(C3N(C(CSC)=O)CCCC3)C2)nnc2n1CC(N)C2 N1(C(c2cnc(S(C)(=O)=O)s2)=O)CCCCC2(C1)CN(C(=O)CCC(N)=O)C2 C1(NC(CC=CC)=O)COC2(CCN(C(c3n[nH]c(C4CC4)c3C)=O)C2)C1 C=CC1(CC(=O)NCC(CO)NC(=O)CN(C)CCN(C)C)CCOCC1 CN1Cc2ccc(C(=O)NC3CC(O)CN(C(C4(O)CC4)=O)C3)cc2C1 C1(C(=O)NC(CN(C(C2(COC)CCOC2)=O)C2CC2)C)C(C)(C)C1(C)C C(=O)(C1CCCn2ccnc21)NC1CCCCN(C(C(Br)=C(C)C)=O)C1 Cn1cnc2c(NC(C3CC4CC4N3Cc3cc([N+](=O)[O-])cs3)=O)ncnc12 C(=O)(C1=CCOCC1)NC(C)CCCCNC(c1cnc(C2CC2)o1)=O C1(C(C)(C)NC(C2CC23CCC3)=O)CCCN1C(C1CC1F)=O N1(CC(=O)NCCOC)CCCC2c3ncn(C)c3CCN12 c1(CC(=O)NC2(C)CC(C(=O)NCCCc3ccsc3)C2)ccc(C#N)cc1 C1(CNC(C(CC#C)O)=O)CN(C(c2ccnc(OC)c2F)=O)CC12CC2 CC1CN(CC(=O)NC2CCN(CC(=O)O)CC2)CCO1 C1(C(C)NC(=O)CCc2nc[nH]n2)CCCN1C(C1CC1c1ccnn1C)=O C(CCC(C)CC(=O)NC(C(C)(C)CO)c1ccc(C)o1)=C(C)C c1(C(N2CC(NC(CC(C)C(F)(F)F)=O)C3(C2)CC3)=O)ccc2ncncc2c1 CCC(CNC(c1cnc(C(F)(F)F)s1)=O)N=c1[nH]c2ccc(F)cc2s1 c1(N2C(=O)CC(C(=O)NC(CNC(CC=C=C)=O)C(C)C)C2)ccc(F)cc1F C1(C(C(N2CCC(C)C2CNC(C23CCC(C2)C3)=O)=O)=O)CCC(C)(C)CC1 C(=O)(C(C)(C)c1ccn(C)n1)NCC(CNC(C(C)NS(CC)(=O)=O)=O)C C12(C(=O)NC(C)CCNC(C3CCC(C(N)=O)O3)=O)CCC(CC1)C2 C(=O)(CS(=O)(=O)CCO)NC1(CCC)CCCN(C(=O)Cc2ccco2)C1 c1(NC(C(CC)C2CCOCC2)=O)ncc(C#N)cc1Cl.C12CC(C1)CNC2=O N1(C(C(c2cn(C)nc2)(C)C)=O)CCCC(NCC2CC3CCC2O3)C1 c1(C(=O)NCC23C(CN(C(CC(CC)(C)C)=O)C2)C3)ncn2c1COCC2 N1(C(CN(C)C(N)=O)=O)CC2(CCCC(CNC(c3ccc(CO)cn3)=O)O2)C1 CCS(=O)CC(=O)NCC(C)NC(c1ccc(-n2cncn2)nc1)=O C(CNC(c1cc(C2CC2)[nH]n1)=O)(CC(F)(F)F)NC(c1nn(C)c(F)c1)=O C1(C(=O)NC2C(C3C(C)C3)C2)CC2(CCN(C(=O)OC(C)(C)C)C2)C1 N1(Cc2ccc(CO)cc2)CCc2sc(-c3cccc4ccsc34)nc2C1 Clc1ccc(Br)c2cc(N3CC4COCC4C3)ncc12 c1(C(C(=O)O)NC(c2ccc(C(C)SC)o2)=O)ccccc1F.c1(O)ccccc1 C1(CC(=O)N(C2CCN(C(c3ccccc3)=O)C2)CC)CCC(=O)O1 c1(OCC)ccc(Cl)c(C)c1.C1(CCC)=CC(=O)NCC2CCCC2NC1=O.CCC=C N1(C(C2C(C)(C)CCO2)=O)CC(C(=O)NCC2=NOCC2)C2(CC2)C1 S(=O)(=O)(CCC(=O)NC1CC(F)CN(C(=O)Cn2ccc(C(F)F)n2)C1)NCC C1(C(C)N(C(=O)CNC(c2cccn(C)c2=O)=O)C)COc2ccccc2O1 Cn1cc(CNCCNC(C2CC(c3ccccc3)CO2)=O)c(Cl)n1 c1(CCC(=O)NCCN(C(C2CC=C(C)CC2)=O)C)csc2nc(C)cn12 C1(NC(C2(C)CC2(Cl)Cl)=O)CN(C(C2(F)CCCC2)=O)CC1C1CC1 N1(C(c2c(C)onc2CO)=O)CCCCC(NC(c2cncc(O)c2Cl)=O)C1 c1(NC(=O)NCC2N(S(C)(=O)=O)CCN(C)C2)ccc(S(=O)(=O)C(F)F)cc1Br CC1CN(C(C2CN(C(c3nc[nH]n3)=O)CC2(F)F)=O)CC1(F)F C1(C(N2CCC(N(C(=O)CC3C=CS(=O)(=O)C3)C)CC2)=O)C(F)(F)C12CCC2 N(C(=NCCc1cnccc1C)NC(C)C(=O)NC)Cc1c(CC)ccs1 c1(C(=O)NCc2ccc(CC(C)NC(C(C=C=C)C)=O)cc2)ccc(C)nc1N CC1(C)CN(C(c2n[nH]c3c2CSCC3)=O)C(CNC(=O)CCC(N)=O)CO1 C(=O)(C(O)CC(=O)ON(C)C)N(CC1CC(NC(C(CC)CC)=O)C1)CC N1(C(C2(C)CCCC2)=O)CCC(O)(CCNC(=O)CNC(C2CCC2)=O)CC1 C1(C(=O)NCCSCC#C)C=CCN(C(=O)CCCC2CCCO2)C1 c1(CC)c[nH]nc1C(=O)NC1CC1CNC(c1ccc(C2CCCO2)[nH]1)=O C1(C(=O)NC2CCC(CNC(C3C=C(C)CS3)=O)CC2)CN2CCCC1C2 c1(C(N2CC(NC(c3cccc(OC)n3)=O)C(SC)C2)=O)cn(C)c(C)cc1=O C1(CN(c2ccnc(C(=O)OCC)n2)C)C2Cc3ccccc3C12 Cc1cc(F)sc1NCc1cccc(OCC2CCCO2)c1 c1(C(N)=O)cccc(C(=O)NCCC2CCN(C(=O)CCc3ccccn3)C2)n1 N1(C(c2nn(C)c(O)c2)=O)CC2CN(C(=O)COC(C)(C)C(F)(F)F)CCC12 Cc1ccc(=NCCC(=O)NCCCCC(C)NC(C2C(C)C2(F)F)=O)[nH]c1 c1(OC)cc(C)c(C(=O)NC(CNC(C2(S(C)(=O)=O)CCC2)=O)CO)cn1 C1(C(N2CC(C)(NC(C3(C(F)(F)F)CCCC3)=O)C2)=O)CC2CCC2C1 c1(C(=O)NC2CCC(CNC(Cc3cc(COC)on3)=O)C2)c(C)cnnc1O N1(C(C2(C)N(c3nc(SC)c(F)cn3)CC2)=O)CCc2cccnc2C1 C#CCC(C)(C)C(=O)NC1CC(N(C)C(c2ccc(CCF)cc2)=O)C1 N1(C(c2c(CCC)occ2)=O)C2CCCC1CN(C(C1CC(C)OC(C)C1)=O)C2 CCC(C)C(C(=O)NCc1nnn(C)c1C(=O)N(C1CCOC1)CC)NC(C)=O C=C(Cl)CC(C(=O)N(CC)Cc1nc[nH]n1)NC(=O)Cn1cccn1 c1(C(N2CCC(N(C(=O)CCC(C)(C)C)C)C2)=O)ccc(F)c2cccnc12 c1(N2CCN(C(C3CC34CCC4)=O)CC2CCO)nc2ncc(Cl)cc2o1 N1(CC(=O)NC2CCC(N(C(=O)CNC(N)=O)C)CC2)Cc2ccccc2C1 C1(C(=O)NCC2C(C)OCC2)CSCCN1C(C1CCOC1(C)C)=O c1(C(=O)NCCCCCCN(C(C(C2CC2)OC)=O)C)cccc2nc(C)nn12 C12(C(=O)NCC(C3CN(C(=O)CC(O)C4CCCC4)C3)C)CC(N(C)C)(C1)C2 Cc1c(C(=O)NCC2CCCN(C(=O)C=CCCC(C)C)CC2)cccc1F C1(NC(CCC(C)N(C)C)=O)CCC2CCN(C(C3CCCO3)=O)C1C2 N1(C(C2C(NC(c3n(COC)ncc3)=O)CCC2)=O)CCc2c(cnn2C)C1 N1(C(c2ccc(CCC)cc2)=O)CC2(NC(c3ocnc3C)=O)CCCC2(F)C1 c1(CN)ccc(Cl)cc1Br.C1(C(=O)O)(COC)CC(O)(C(F)(F)F)C1 C1(C(N2CCN(C(c3c(OCC)scc3)=O)C(CO)C2)=O)CC2(C1)CC1(CC1)C2 CC1=NNC(=O)C1CC(=O)NC1CC1NC(c1coc(C2CCCCC2)n1)=O N1(C(C(C=C)C)=O)CC2CC1C2CNC(C1(F)CCOCC1)=O c1(NC(CC2CCN(C(CCCC#CC)=O)C2(C)C)=O)ccc2c(c1)COC2 CC(C)C(CCC(F)F)NC(N1CCC(C)C(F)C1)=O CC1C2CCCCC2CN1C(=O)CC1CCN(C(c2cc(CO)on2)=O)C1(C)C CCCC(O)C(=O)NCC(CNC(C1(C)COC1)=O)OC c1(CN(c2n(CCCOC)nnn2)CC2CC2F)cccc(C2COC2)c1 c1(C(=O)NC(CNC(C2C(=C)C2)=O)C(C)C)cc(S(N)(=O)=O)cc(Cl)c1Cl c1(C(N(C(CNC(C(CC)OC)=O)C)C)=O)cnc(OC)c(C(F)F)c1 CCCCC(=O)NCC1CCN(C(=O)C(C)(C)Nc2ccccn2)C1 n1(CC(=O)OC)ncc(C(=O)NC2CC2NC(C2CCCN2S(C)(=O)=O)=O)c1C c1(C(N2CCC(O)(CN(C(C(C=C)(C)C)=O)C)C2)=O)cccc(F)c1O CC(N)C(=O)N=c1ccn(CC(N2CCCC(CO)C2)=O)c(O)n1 c1(OC)ccc2[nH]c(C(=O)NCC3(C)CCN(C(c4ccc(C)o4)=O)C3)cc2c1 c1(N2C(CNC(c3cnn(-c4ccccc4)n3)=O)CC2)cncc(Cl)n1 CCC(CCC(=O)NCCc1ccccc1)NC(=O)C=CSC c1(C(=O)NC2C(CC(N3C(C(=O)NC)CCC3)=O)CCC2)c[nH]c(=O)cn1 c1(C(=O)OC)cc(C(=O)NC2CCC2NC(=O)Cc2ccc(O)nc2)ccc1Cl c1(OCC(=C)C)ccc(S(=O)(=O)CC(N2CCc3nncn3CC2)=O)cc1 CN(CC(C)(CO)CO)N1CCOC(CNC(=O)NC(C)(C)C)C1 c1(CC)ncc(C(=O)NC2(C(=O)OC)CCCCC2)cn1.N12CC3CC3(C1)C2=O C1(NC(C(c2cccc(C)c2)O)=O)CCSC12CN(C(=O)C(C)NS(C)(=O)=O)C2 c1(C(=O)OC)ncc(NC(C2CCCCN2Cc2coc(OC)n2)=O)cn1 CC1CC2(CC(C(=O)NC3CCCC(C(=O)N(CCF)C4CC4)CC3)C2)C1 C12(C(N(CC(C)CNC(C3CC(C)N(C)C3)=O)C)=O)CCC(C#N)(CC1)CC2 C1(C(=O)NCCOCCCNC(C2(C)CC(=C)C2)=O)CCC(=O)N1C CCCC(F)C(=O)NCC1CC(NC(=O)C(C(C)C)c2ccccc2)C(O)C1 CCCC(CC)C(=O)N1CC(NC(c2cnc(OCC)nc2)=O)C(C)C1 c1(C(N2CC(CCCCNC(c3c(C)snc3)=O)C2)=O)ccccc1F Cc1sc(C(=O)NCC2CC3CCC2N3C(=O)C(C)CN(C)C)c(C)c1C CCC(C)C(C(=O)NC1CC(OC)CN1C(=O)COCc1ccco1)OC c1(CC(=O)NC(C)CCCNC(C2CC2CF)=O)ccc([N+](=O)[O-])cc1F C1(C(N2CCN(C(C(C)OCC=C)=O)C(C)C2)=O)CCC2CCCCN12 N1(C(=O)Nc2cc[n+]([O-])cc2)CCC(C2CCCN2)CC1.c12ncsc1N2 C(=O)(C(F)CC(C)(C)NC(=O)CCC1CC1)N(C)Cc1cccc(C)n1 CON(CCC(=O)NC1CC2CCC(C1)N2C)C(=O)CCN(C)C N1(C(C(=O)Nc2c(C)c(Cl)ccc2)c2csnn2)CCc2nc(Br)sc2C1 Cc1ccc(C(N2CCCN(C(=O)CC3CC3(C)C)CC2C)=O)c(O)c1C c1(N(CCCN2CCCC(C)C2)C)nc2cccnc2c(=NCCN=[N+]=[N-])[nH]1 c1(N2C(C(CNC(C(C)C(C)O)=O)(C)C)CCC2)ncc(Cl)c(O)n1 c1(C(=O)NCCC(CNC(c2nc(C)sc2)=O)O)ccc2[nH]ccc2c1 c1(-c2nnc(C(N3CCC(CCOC)C3)C(=O)NCCC)o2)ccccc1OC N1(C(=O)C(O)Cc2cnc[nH]2)CCN(C(c2coc3c2COC3)=O)CC(CO)C1 C1(CC(N2CCC(NC(=O)CCCn3cccn3)CC2)=O)CC2(COC2)C1 c1(OC)cccc2c(C(N3CCCN(C(=O)C(C)C4CC4)C(CO)C3)=O)cnn12 N1(C(=O)CCC2CCC2)CC(C2CCN(C(C3CC4CC4C3)=O)CC2)C1 N1(C(CN(CC(C)C)C(=O)CCC(C)(C)C)=O)CCC(CCO)C1 Cn1ncc(=NC(=O)N2CCCC2Cc2ccccc2)[nH]1 c1(C(=O)NCC23CCC2CCN3C(C2CCOCC2)=O)ncn2ccccc12 Cc1ccc(C#N)cc1C(=O)N(C(C)C(=O)N(C)CC1CC(O)C1)C1CC1 C#CCCCCC(=O)N(C)CC=CC(N1CCC1CC(C)C)=O C1(C(=O)NCCN(C(C)C)C(C2(C(C)CCO)CCC2)=O)Cc2ccccc2C1 N1(C(CCC)=O)CCCC1C(=O)NC1CCC(N(C(=O)C(F)=C(C)C)C)C1 C1(C(C)(C)O)CCN(C(C2(C)CC(NC(=O)CCN3CCOC3=O)C2)=O)C1 c1(CC(=O)NC(C)C(C)(C)NC(C2CCC(=O)O2)=O)cnccc1Cl c1(NC(C(=O)NCCCC(=O)OC)=O)ccncc1NC(=O)CCc1ccco1 c1(C(=O)NCCC2CCCN(C(CC(=O)OCC)=O)C2)cc(Cl)c([N+](=O)[O-])[nH]1 NC(=O)CCNC(=O)C(=O)NCCC1CN(C(=O)C=CC2CCC2)C1 C(N=c1[nH]c(C)cc(=NCc2ncccc2F)[nH]1)c1nccc(C)c1 C(N=c1nc(N2CCCC(F)C2)c2c(ncn2C)[nH]1)C1CCCN(CC(C)C)C1 C=C(C)CCCC(=O)NC1CC(C(F)F)(NC(=O)C(CC)OC)C1 c1(C(=O)NCCC2N(C(c3c(C)nsc3)=O)CCCC2C)ccc(N)c(C)c1F N1(C(=O)CCc2nc(C3CCCC3)no2)CCN(C(c2ccns2)=O)C2CCC12 c1(C(C)C)nnc(CCC(=O)NC2CC(C)(NC(C3C4CCCC34)=O)C2)o1 C1(C(N(CCOCCC(N2C(CC(C)O)CCCC2)=O)C)=O)CN2CCN1CC2 C1(C(=O)NC(C2(O)CCOC2)C)CC2CCC(C1)N2C(=O)C=Cc1nccs1 N1(C(=O)CCc2cncnc2)CCC(F)(C(=O)NOCC=C(F)Cl)CC1 N1(C(c2ccnc(OC)n2)=O)CC(NC(=O)C#CC(=O)N(C)C)CCC1C C=CC1(C(N2CC(O)(CNC(C3COCCC3C)=O)C2)=O)CCCCC1 C(=O)(C(C(=O)N(CC(C)Cc1ccccn1)C)C1CC1)OCC c1(CC(=O)NCCC2CCCN(C(COCCSC)=O)C2)cc(F)cc(F)c1 C#CCCCCCC(N)C(=O)NCC1COCCC1C N1(C(c2cccc(C#C)c2)=O)CC2CS(=O)(=O)CC2(CNC(=O)CC(CC)CC)C1 C12(C(N3C(COC)CC3)=O)CC(CO1)N(C(C1C3CCC(C3)C1C)=O)C2 c1(C(N)=O)ccnc(NC(C2CCCC(NC(=O)Cc3ccccc3O)C2)=O)c1 c1(-n2c(C(C#N)C(C)(C)C)nc(CC)n2)cccc(C#N)c1 Cc1ccc(C=CC(=O)N(C2CC(NC(c3cc(C)nn3CC(F)F)=O)C2)C)o1 Cc1ncc(C(=O)NCC2C(C(=O)N(C3CCOC3)CCF)C2(C)C)s1 N1(C(c2snc(C)c2N)=O)CCCC(O)(CCNC(c2nscc2C)=O)C1 C1(CC(=O)NC(C)C2CC2)CCN(C(c2ncccc2F)=O)CC1 N1(C(C(C)SC)=O)CC2CCOC2(CNC(c2nnn(C)c2N)=O)C1 c1(C(N2C(CO)CC(NC(C(CCC)OC)=O)C2)=O)cccc(OC)c1C n1(CCC(=O)NC(C)CCNC(=O)C2=COCCO2)nc(O)c2ccccc12 N1(C(C2N(C(C)=O)CCC2)=O)CC(NC(C2(CF)CC(F)(F)C2)=O)CCC1C Cc1n[nH]c2cc(C(N3CCC(C)CC3CNC(=O)CC(C)(F)F)=O)ncc12 c1(NC)cnc(C(C(=O)NCCC(C)C)N(C)CC2(OC)CCC2)s1 C1(CC)CN(C(=O)CCCCN(C)C)CCC1NC(C1CC(C)=NO1)=O CCN(CC(=O)OC(C)(C)C)N1CCCCCCC1C N1(C(C(C(C)C)NS(C)(=O)=O)=O)CCN(C(c2cncc(F)c2)=O)C(C)C1 Cc1cc(C)c(C(=O)N(C)CC2CCN(C(C3CCCC(=O)N3)=O)C2)s1 N1(C(CCCn2ncc(C)c2)=O)CCN(C)CC1CNC(c1conc1CO)=O C1(OC)CC(CNC(=O)C(C)OCCN(C)C)N(C(=O)C2=C(C)CC2)C1 CCC(C)C1C(=O)N2CCC(C2)CON1C.C1(C(=O)NC)OCCC1C c1(C(=O)NC2CC(CC(=O)OC)(C(F)(F)F)C2)cc(Br)cn1C c1(CC)nn(C)cc1C(=O)NCC(O)CNC(=O)Cc1cncn1C N1(C(C(CC)Sc2nc[nH]n2)=O)CC(O)CC1CNCCNC(=O)C1CC1 C1(CC=C)(C(=O)NC(CNC(=O)C(C)=CC(C)(C)C)CCC)CCOCC1.C1(CO)CC1 c1(C(=O)O)cn(CC(=O)NN2CC(CO)CC(CO)C2)c2ccccc12 N1(C(C(CC2CC2)NC(=O)C(C2CCCCC2)F)=O)CCOC(CCCO)C1 C12(C(=O)OC)COC(C(=O)NC3CC(CCNC(C4CCCCC4C)=O)C3)(C1)C2 C1(N(C(c2c(C)ccnn2)=O)C)CN(C(c2cnc(Cl)n2C)=O)CC1(C)C Cc1c(C(=O)NC(C)CCCNC(c2ccccc2F)=O)ccc2cncn12 C1(C(=O)NCC=C(C)C2CC2)CC(O)CCN1C(c1cn[nH]c1)=O c1(C(=O)NCC2C3CN(C(C4CCCS4(=O)=O)=O)CC23)cc(Cl)cc(F)c1F C1(N(C(C2CCCN(CC)C2)=O)C)(CSc2cccc(C(N)=O)c2)CC2(CCC2)C1 N1(C(CN(S(C)(=O)=O)C)=O)CCC2(CC(NC(=O)C3=CCC(F)(F)CC3)CO2)C1 CN1CC(C(N2CCCC(C(=O)N(c3cccc(O)c3)C)C2)=O)CCC1=O CC1CCCCC1CC(=O)NCc1cc(C(N2CCN(C)CC2)=O)cs1 c1(CC)cc(CC(=O)NCC2CCOC2C(=O)NCC(C)(C)n2ccnc2)on1 C(=O)(C1=CS(=O)(=O)CCC1)NCCCCCNC(c1c(CC)[nH]nc1Cl)=O c1(N(C)C)cccnc1C(=O)NCCNC(C1CC1C(F)(F)F)=O CC(C)C(C#N)C(=O)N1CC(C2(NC(=O)C(C)COc3ccccc3)CC2)C1 C#CC1(NC(=O)C(CC2CC2)NC(=O)C(C)NC(=O)CC)CCC(C)(C)C1 N1(C(C(CC)OC)=O)C2CCC1CN(C(=O)CCC1CCc3ccccc3C1)C2 N(C)(C1CCCc2ccccc21)C(=O)NCC1C(Cl)(C(=O)OC)C1 N#Cc1c[nH]c(=NC(=O)C2CC(F)CN(C(=O)CCN(C)C)C2)cc1F O=C(NN=c1cncc[nH]1)C1CCC12CCCNC2 c1(C(c2n(CC=C)nnn2)NCc2scnc2C)c(Br)nc(C)n1C CCC(CC)C(C)C(=O)NC1CN(C(=O)CCc2cncc(OC)c2)CC1F C(=O)(C(F)C(=O)NCC1CN(C(c2ncccn2)=O)CCO1)OCC c1(CNC(c2ccc(C)c(C)c2)=O)cnn2c1CN(C(=O)C(C)(Cl)Cl)CC2 Nc1cccc(C(N2CCC2CNC(=O)CCC2CC2(F)F)=O)c1F N1(C(CNC(C(CC)CC)=O)=O)CCC2(C1)CN(C(c1ccc(Cl)cc1)=O)C2 C(CNC(c1ccc(C(F)F)cc1)=O)(C(C)C(C)C)NC(CCCOC(C)=O)=O c1(CC(=O)NC(CN(C(c2c(CC)non2)=O)C)C)noc2ccc(F)cc12 CC1CCN(C(=O)CC2CCO2)C1CNC(=O)CCc1cc(Cl)cs1 C12(NC(c3cocn3)=O)CCOCC1CN(C(c1ccc(Br)s1)=O)C2 C(C)(CC(C)(C)O)NC(C(CC1CN(C(C=CCOCCOC)=O)C1)F)=O c1(CS(C)(=O)=O)cn(CC(=O)NC2C(CNC(C3(CF)CC3)=O)CCC2)nn1 c1(OCC(=O)NC2CN(C(c3c(OC)cccc3)=O)CC2O)cc(C)ccc1F C1(NC(c2cn(CCNC(C3C(C)(C)COC3)=O)nc2)=O)C2CCC(F)(F)C12 C(CCCCCC(=O)NC1CN(C(=O)CCC2CCCC2)CCC1(F)F)NSC Cc1cc(C(=O)NC2CCN(C(C3(N(C)C)CCC3)=O)C(C)C2)cc(C)c1 c1(C(N2CCC(CNC(CN(C)C(N)=O)=O)(CO)C2)=O)cc2ccccc2o1 C(C(C)(C)C(C)(C)C)NC(c1cccc(Cn2cc(CN(C(C)=O)C)nn2)c1)=O c1(C(=O)NCC(=O)NCc2ccc(Cl)cc2)ccc(O)nc1 C1(COC)CN(C(c2cnn(C)c2C2CC2)=O)CCN1C(=O)Cc1cnoc1 CCCC(C(=O)N1CCC(CF)(NC(C2CCCOC2C)=O)C1)N(C)C Cc1cc2scc(CC(=O)NC3CC(F)CN(C(=O)CNC(N)=O)C3)c2s1 Cc1cccc(Cl)c1C(N1CC2C(NCc3cnco3)C2C1)=O Cc1cccc(Cl)c1C(c1ccc(CN2CC(NC(=O)C=CCF)C(F)C2)o1)=O C1(C(=O)NCCN2CCN(C(c3ccc(COC)nc3)=O)CC2)CCC(C2CC2)C1 CCCCC(C(=O)N1CCC(=CCNC(=O)Cc2cnn(C)c2C)CC1)N(C)C O=[N+]([O-])c1cccc(Br)c1NCc1cnn(-c2ccccn2)c1 CCCCC(CNC(=O)CCNC(=O)C=CCl)NC(c1ccc(F)cn1)=O C1(C(N2CCC(CNC(CC=C)=O)C(C)C2)=O)CC2C=CC1C21CC1 N1(C(CCC=C)=O)CCC(CNC(=O)CNc2ncccn2)(COC)CC1 N1(C(c2ccc(C)cc2F)=O)CCCC2C1CCN2c1nccc(C(C)C)n1 N12CCC(C1)C2=O.C1(C(CNC=O)NC(C)=O)CCCCC1.C1(C(=O)N)(N(C)C)CC1 c1(C(=O)NC(C)(C)CCCNC(C2CCC3CCC23)=O)coc(S(C)(=O)=O)c1 C(C(=O)NC1CN(C(=O)CCC(C)C)CC1C(F)F)(C(C)C)SC c1(C)ccc(C(F)(F)F)cc1C#N.N(C(=NCC(C)C)N)C(C)C.N1S(=O)(=O)N1 Cc1ccc(F)cc1NC(=O)CC(C)CNC(=O)CCc1ncccn1 C1(N(C(CCOC)=O)C)CCCC(N(C(=O)CCOc2cccnc2)C)C1 C1(NC(=O)CCCC2CCCC2)CC12CCN(C(=O)C(=O)NC1CC1)CC2 c1(C(C)(C)NC(C2CCC(c3ccccc3)CC2)=O)ccc(F)c(Cl)c1 C(CCC(=O)NC1CC(C(=O)NCC2(CO)CCOC2)C1)OCC c1(C(=O)NC(C(CO)NC(C2C(=C)C2)=O)C)ccccc1Cn1ccnn1 C1(CCNC(C2(COC)CCCC2)=O)COCCN1C(=O)CC1C(C)C1(F)F c1(C(=O)NC23CC(C2)N(C(=O)CCn2ccnc2)C3)ccn2nnnc2c1 O=C(N=c1cncc[nH]1)C1CCC(C)N1Cc1cc(O)cc(Cl)c1 CC(C(F)C(=O)NC1CCN(CCNC(C2CCCC3CC23)=O)CC1)C(F)(F)F c1(N2CCOCC(C)C2)ccc(S(=O)(=O)N2CCn3c(C(F)F)nnc3C2)cc1F CC1Sc2ccccc2N(C(c2ccc(Br)cc2-n2cnnn2)=O)C1C C1(C)(COC)CC(NC(=O)OC(C)(C)C)CN1C(=O)C1CC1 C(CCCCCCO)c1cc(N2CCC(N(C)Cc3c(OC)cncc3)C2)ncn1 Cc1cc(NCC(=O)NC(CNC(c2ccc(Cl)cc2)=O)C(C)(C)C)cc(F)c1 CC(C)C(F)C(=O)N1CC2C(C(N3CCSC(C)C3)=O)C2C1 C1(CNC(CCN(C(=O)OC)CC)=O)CCC(C(F)(F)F)CC1.C1CCC1 Cc1nc(Cl)sc1C(N1CCN(CC(=O)NCC2CNC(=O)CO2)CC1)=O c1(NC(C2(C)N(C(C3CCC(=C)CC3)=O)CCC2)=O)nc(Cl)c(Cl)cc1Cl N1(C(CCc2onc(C)n2)=O)CCCC2(CC(NC(=O)C(F)=CCCF)C2)C1 c1(CNCC2N(c3ccc(OCC)nc3)CCC2)cc(OC)cc(F)c1 C(=O)(C1=CCCSC1)N1CCCC(C(=O)N2CCCO2)C1 C1(NC(CCN(CCC)C)=O)CN(C(C2CCC(CN(C)C)O2)=O)CC1O c1(C(N(CC)CC2CCCN2C(=O)CCc2nncs2)=O)cnc2scnc2c1 C12(C(N(C)Cc3cn(CCCc4ccncc4)nn3)=O)OCCCC1C2(F)F C(c1ccc2occc2c1)=CC(=O)NCC1C(C)CN(C(C2CCS2(=O)=O)=O)C1 Cc1c(N2CC(CS(C)=O)C2)ncnc1N1CC2CC1C2 N1(Cc2ccc(CC)cc2)CC2(CN(C(c3ccccc3I)=O)CC2C(=O)O)C1 CC(C)CC(C)(C(N)=O)NC(=O)CN(C(C1CC(=O)N(C)C1)=O)C(C)C c1(C(N2CCCC(c3onc(C(C)C)n3)C2)=O)ccc(Cl)c2ccccc12 c1(CN(C2CCOCC2)CCC)nc(O)nc2ccccc12 c1(OCC)ccc(C(N2CCCC2CN(C(=O)C(C)SC(C)C)C)=O)cc1C C(c1cccnc1)=C(C(=O)N(CCCNC(C1C=CCS1)=O)CC)C c1(-c2nc(CSC)nn2CC(F)(F)F)ncn2cc(C)cnc12 C(=O)(C1=NN(C)C(=O)CC1)N1CCC(C(N2CC(C)OCC2)=O)C1 C(=O)(CCCS(C)(=O)=O)NC(C1CN(C(C(C)OCCCC)=O)C1)C C1(CNC(c2cscn2)=O)CC2CC(C1)N(C(c1cc3n(c1)CCCC3)=O)C2 C=CC1(C(=O)NCCc2nnc(C)n2C)CCN(C(c2cc[nH]c2CCC)=O)C1 C1(C(=O)NCc2ccccc2Cl)CN(C(=O)C(O)c2ccco2)CCC1O c1(OC)ccc(C)cc1C=CC(=O)NC(C)C(C)NC(c1csc(C#N)c1)=O C1(NC(c2ccc(C(C)=O)o2)=O)CN(C(=O)C(C)(F)F)CC1n1ccnn1 C(=O)(CCCCC(C)CC)NC(CC=C)CNC(=O)CC1=CCCCC1 CC1CCC(Nc2ncc(F)cn2)CN1C(=O)CCc1cncnc1 C=C1CCC(CNC(C2CC(NC(c3csnc3Cl)=O)CCO2)=O)CC1 CCCCCCCCN(C)C(C1CCCN(C(=O)C(C)C(O)C(C)C)C1C)=O CC1(C)C(C(F)(F)F)CCN1C(c1cn(C2CCNC2=O)nn1)=O c1(CC)nc(C(N2CC(CNC(=O)CC(CN(C)C)CC)C2)=O)c2ccccn12 Cc1nc2cc(C(=O)N(CCN(c3cc(=O)n(C)cn3)C)C(C)C)cnc2[nH]1 Cc1c(C(N2C(C(=O)NC(C)(C)C)CCC2C)=O)sc2cncn12 Cc1ccc(CN(C2CC2)CC2CCN(C(C3(C)CCNC3=O)=O)CC2)nc1C c1(C(CC)N(C2CC(n3ccnn3)C2)C)cccnc1.C12CN(C1)C2=O C1(NC(c2c(C(C)C)ccs2)=O)CC(NC(=O)CN(C)C(=O)C2CC2)C12CCC2 N1(C(=O)C=Cc2ccco2)CCC2CN(Cc3cccnc3O)CC2CC1 N1(C(c2scc(C)c2Cl)=O)CC(NC(C2CCCC2)=O)CC2(CC2)C1 CCCC(C(=O)N(C1CCCN(C(c2cc(C(C)(F)F)on2)=O)C1)CC)OC c1(CCC)nc(=NC(C)C2CCN(C(=O)CC3CCCOCC3)C2)s[nH]1 C1(NC(C(CCC)C)=O)CC2CCC(C1)N2C(=O)CNS(=O)(=O)c1cn(C)cn1 CC1CC(C(=O)NCC2(CNC(C3CCCC(O)C3)=O)CC2)CCS1(=O)=O Cc1[nH]nc(C(=O)N(CCCN(C)C(C2CC2C#N)=O)C)c1C(F)(F)F C1(C(N2CCOCC2CNC(C2(F)CCOCC2)=O)=O)CC2(CCCO2)C1 N1(C(c2cc(OC)n[nH]2)=O)CC(O)(C2CCN(C(C3C=CCC3)=O)CC2)C1 C#Cc1ccc(C(=O)NC(C2CCN(C(c3cccc(CO)c3)=O)C2)C)c(C)c1 C1(CN(C(C(c2scc(CC)n2)(F)F)=O)C)COCCN1C(=O)COCC(F)F C1(NC(CC(C)C)=O)CC2CCC(C1)N2C(c1ccc(NC(C)C)nc1)=O C(=O)(C1=CC2C=CC1C2)NC1C(C)CN(C(C2CCCC2O)=O)C1 C1(NC(C(N2CCN(C)CC2)C)=O)COC2(CCN(C(C3CC(O)C3)=O)CC2)C1 c1(CNC(=O)NCC(c2ccc(Br)cc2)F)cnc2ccccc2c1 n1(CC)cc(CC(=O)NC2(CN(C(=O)Cc3cc(C)on3)C)CC2)cn1 O=C(CCCC#Cc1ccccc1)NCC12CCC1CCN2C(=O)C=CCO CN1CCOC(C(=O)NCC2CCC2NC(=O)CN2CCC(CN(C)C)CC2)C1 CC1(NC(=O)CSc2ccc(F)cc2)CCCN(C(C2CCO2)=O)C1 C(=O)(C1=C(Cl)CCOC1)N1C(CNC(=O)C=CC(F)F)CC1 C12(C(N(CCN(C(C)C)C(c3cc(C4CC4)cs3)=O)C)=O)CC(C(C)(C)C)(C1)C2 c1(OC)cnccc1CNC(=O)CCC(C)NC(=O)CC(C)(C)OC C=CCCC(C)N=c1[nH]c(N(CCC(N)=O)C)nc2cc[nH]c12 c1(C(=O)NCC(CO)NC(C(CCC)O)=O)csc2c(F)cc(F)cc12 N1(CCC(=O)NCC(CN(C(C2CC2CN(C)C)=O)CC)(C)C)CCNC(=O)C1 N1(C(c2c(CC)ocn2)=O)CC2CC(NC(C34CCC(OC)C3C4)=O)C1C2 C12(C(=O)NC(CC(C)C(F)F)C)CC(CCO1)N(C(=O)C=Cc1cc[nH]n1)C2 n1(CCC)cc(NC(C2(NC(=O)CCCc3cnn[nH]3)CCSC2)=O)cn1 C1(NC(=O)Cc2ccc(O)nc2)CN(C(c2sccc2F)=O)CC12CC2 C1(CNC(=O)CC2CC(F)C2)COCCN(C(C2CCC3(CC2)CC3)=O)C1 CC1(C(=O)NC2CC=CCC2C(=O)NCc2cnc(C(C)C)[nH]2)CCCCO1 N1(C(CCCSC)=O)CC(CNC(=O)CCc2nncs2)C(F)(CO)C1 c1(C(=O)NCC2(NC(c3ccc(COC)o3)=O)CCOC2)cc2ncccc2o1 c1(C(=O)NCC2(C(C)NC(=O)CC(F)F)CC2)ccc(Cl)c(S(N)(=O)=O)c1 C1(C(=O)NCCOCCNC(C(C)c2cc[nH]n2)=O)CC(C)N(C)C1 C1(C(N2C(CNC(COCCOC)=O)CC2)=O)Cc2ccc(F)cc2O1 C1(C)(C(=O)NCC#CCNC(c2ccc(CCCCC)o2)=O)CCCNS1(=O)=O C12CCOC1CNC2=O.C1(C(N)=O)CCC(CNC(C2(O)CCC2)=O)O1 c1(CC2CCOC2)ccc(C)cc1-n1cc(C(=O)Nc2cncc(SC)c2)nn1 N1(C(c2n(CC)ncc2)=O)CCC(NC(C2CC2CCOC)=O)C1C C1(C(=O)OCC)CCN(C(=O)C2(CCNC(=O)C=C(C)C(C)C)CC2)O1 c1(NC(C(CC2CN(C(C(C)C3(O)CCC3)=O)C2)F)=O)ccccc1CC1CC1 C1(NC(c2c(OC)cc(C)cc2)=O)CN(C(c2nnc(C)s2)=O)CC2(CC2)C1 Cc1nn(C)c2c(NC3COC4(CCC4)C3)nc(N3CCSC(C)(C)C3)nc12 c1(CC)cccc(N(CC)CC2CC2)c1.N1(C=O)CCOCC1CO C1(CNC(=O)NCC2(C(F)F)CCCCC2)CC2CCCC2C1 C1(NC(Cc2c(C)ccs2)=O)CC2CN(C(C3(C#N)CC(C)C3)=O)CC2C1 CCCC(C)(O)CC(=O)NC(C)(CC)CCNC(=O)CNC(=O)CCC C=CCCCC(C)(C)C(=O)NC(CNC(=O)Cc1cnn(C)c1)C1CCC1 c1(C(C)NC(CCOCCOCC)=O)csc(CNC(c2ccn(C)c2)=O)n1 c1(OC)ccc(C(=O)N(C2CC3CNC2C3)CCO)c(NC(C)CCO)c1C N1(C(c2nc(-c3cn(C)nc3)oc2)C(=O)NCCC2CC2)CCCC2COCC12 c1(C(=O)NC(C)CCN(C(=O)CSC2CCOC2=O)C)cncc(F)c1 CC1CC2CN(C(C3C4COCC34)=O)CC2N1C(c1ccc2c(c1)N(C)CC2)=O S(=O)(=O)(c1ccc(NCc2cc(C3CC3)on2)c(Cl)c1)N1CC(C)CC(C)C1 c1(C(=O)NCC2(C)CCCN(CC(=O)N(CC(F)(F)F)C)C2)nc[nH]c2nccc1-2 CC1(C)C2CCC1(C)C2C(N1CCCC(NC(=O)COCCN2CCCC2)C1)=O C1(C(=O)NC(C)(C)CNC(C2COC2)=O)CCCCC1c1ccc(F)cc1 N#Cc1cnn2cc(C(=O)NCC3CCN3C(=O)C3=CC4(CCOC4)C3)cnc12 N1(c2ccc(C)cn2)CCCC(C)(C(=O)NCC2CC2(C)C)C1 C1(C)(C(=O)NCCC2(OC)CN(C(=O)C=C(C)Cl)C2)COc2ccccc2O1 N1(C(C(C(C)C)n2cnnn2)=O)CCC2CCC(C1)N2C(C1CS(=O)C1)=O N1(C(=O)NC(C(=O)OC)C)CCC2CC(C(=O)NCc3nnn(C(C)C)n3)C2C1 Cc1cccc(C(=O)NC2CCC2CNC(C2CCC(C)(C)O2)=O)c1Cl C(C#Cc1cnn(C)c1)NC(CNC(C1CCC(C)C1)=O)=O N1(C(C2(C(=O)O)CC2c2ccc(C(F)(F)F)cc2)=O)CC(O)CC1C1(CO)CC1 C12(N(C3CCSC3)CC)CCN(CC1)C2=O.c1(C(=O)O)cscc1C(F)(F)F C(=O)(CC(C(F)F)NC(N)=O)N1C2(C(N(C(C)C(C)(C)C)C)=O)CC(C1)C2 C12(C(=O)NC(C(N3CC4C(CC)(C4)C3)=O)(C)CSC)CCC(CO)(CC1)C2 N1(C(c2cc(C#N)cc(F)c2)=O)CCCC2CN(C(C3C4COCC34)=O)CC12 N1(C2CCC(NC(C(=O)NC(C)C)=O)C2)CCN(C(c2cnc(Cl)[nH]2)=O)CC1 CCCCC(C(=O)N(C)CC1(NC(c2nc(C)n(C)n2)=O)CC1)C(C)C C(=O)(NN1CCCC1C(=O)NC1CCC(=O)NC1C)c1c(C)cncc1C c1(C(N(C(C)CCNC(C2CC(C)(F)C2)=O)C)=O)ccc(S(=O)(=O)C2CC2)cc1 c1(Cn2cc(C(=O)OCCN(CCC)CC3CC3)nn2)ccc(Cl)cc1 Cc1c(F)cc(CNC(=O)NC2CCC(CSC3CC(=O)C3)CC2)cc1[N+](=O)[O-] C1(CNC(c2c[nH]cc2Br)=O)CCCN1C(=O)CC1CC2CC1C2 C1(C(N2CCC(N(C(C=Cc3cn(C)nc3)=O)CCO)C2)=O)CN2CCN1CC2 C1(NC(=O)NCC(O)CF)CCCc2ccccc2C1 c1(NCCc2cccc(OC)c2)cc(=NCC2CCC2)[nH]c(C)n1.C(C(C)C)S C1(C(=O)NC)CN(CC)CC1C1CC1.C1C(C(=O)OC)NC(=O)CCOCCO1 C(CN=C(Nc1ccc(NC(C)=O)cc1)NC1CSCC1C)OCC=C n1(C(C(N2CCCC(CN(C(CC=CC=C)=O)C)C2)=O)C)c(C)cc(O)cc1=O c1(N(C)C)ccc(C(N2CCN(C(=O)C(F)F)CC2)=O)cc1.C1(C(=O)N)CCC1CF C(=O)(C1CCc2nccn21)N1CCCCC(C(=O)NC(c2nc[nH]n2)(C)C)C1 C#CCC(CC(=O)N1CCC(O)(CC(C)C)C1)NC(C1CC2CC1CC2O)=O CC1(C)CN(C(=O)CCc2ncc[nH]2)CC(CNC(c2cnc3n2CCS3)=O)O1 c1(CC)ncc(C(=O)N(CCCNC(C2(CO)CCC2)=O)C2CC2)s1 c1(OC)ccc(F)c(-c2nc(C3CC3)nn2CC(C)C2CC2)c1 C1(C(N2CCC(CCCC)C2)=O)CC2(CCN1C(=O)CCCNC(N)=O)CC2 c1(C(CN(CC(C)(C)C)C(C)=O)N(c2nnc(C3CC3)s2)C(C)C)ccccc1 C(CN=c1nc(N2CCC(C)C(C)(C)C2)c2ccc(C)cc2[nH]1)c1cc(C)no1 C1(OC(=O)CCC(=O)NCCCCOc2c(C)noc2C)CC(C)CN(CC)C1 Cc1csnc1C(N1CCCC1Cc1ccco1)=O N1(C(C2C(C(C)C)C2)=O)CCSCC1CC(=O)NCCCCCF Cc1cc(C(N2CCC(O)(C(C)NC(c3ccc(Br)cc3)=O)C2)=O)c(C)n1C C(=O)(CC(CCCC(C)C)NC(C1(C)CCCS1)=O)OCC C1(CNC(C(C2CC2)OC)=O)CC2CCC(C1)N2C(=O)CC(=O)NC1CC1 C1(C(F)(F)F)(C(=O)NCCCCNC(CCN(C(CC)CC)C)=O)CC=CCO1 c1(OC)cccc(Cl)c1C(=O)NCCC1(NC(C2CC3(C2)CC32CC2)=O)CCC1 N1(C(CCC=C)=O)CCC(N(C)C(c2c[nH]c(C#N)c2)=O)CC1 C1(C(N2CC(C(=O)NC(C)CCCOC)(CC)C2)=O)CCOCC1(C)C C(C(CC(=O)NC(C)CC1(n2cccn2)CC1)NC(c1ccccc1C)=O)OC C1(CC)CCC(C(=O)NC2CC(O)(CNC(=O)CCCN3CCOCC3)C2)C1 Cc1cc(=NC(C)C2CCN(C(c3nc(Cl)sc3Cl)=O)C2)[nH]c(S(C)(=O)=O)n1 C1(CC)C(N)CCCN1C(C1CCN(CC(N)=O)CC1)=O O(NC(=O)C(c1ccnn1C)NC(C1CN(C)C(=O)N1)=O)C(C=C)C C(=O)(CC(C)C(F)(F)F)N1C(C=CC(=O)NC(C2CC(F)(F)C2)C)CCC1 C1(C(N(CCNC(CCN(CCC)C(=O)OC(C)(C)C)=O)CC)=O)CCSC1C C1(N(C(CC(C)c2cccnc2)=O)CCF)CCCN(C(c2cncc(N)n2)=O)C1 Cc1ccc(NC(c2ccccc2Br)c2nnnn2Cc2ccccc2)c(Cl)c1 C(C)(C(CC(=O)NCC1CC12CC2)NC(c1n[nH]c(C)c1O)=O)OC N1(C(c2nccs2)=O)CC2CCCN(C(c3cc4ccccn4n3)=O)C2C1 CC1CC(CNC(=O)C(F)=CCCF)CCN1C(=O)CSc1nnnn1C1CC1 CCC1=NOC(CC(=O)NC(C)CCCCNC(c2cnn(CCO)c2N)=O)C1 C1(NC(=O)C2=C(Cl)CC2)CS(=O)(=O)CC1NC(c1cscc1Cl)=O c1(C(N2CC3C(CNC(CCn4c(C)nc(C)n4)=O)(C3)C2)=O)cc(C#N)cn1C c1(CN(C)C(c2cc(C(N)=O)no2)=O)ccc(CNC(=O)CSS(C)(=O)=O)cc1 N1(CC)CC(NC(C23CC(CO2)N(C(c2cn(C)c(C)n2)=O)C3)=O)CCC1=O CC1(C)CC(CN2CCCC(CNC(=O)CC3CCCC3)C2)CC(C)(C)C1 CCC(CC)CC(=O)NC1(C(F)F)CCN(C(=O)C(F)(F)c2csc(C)c2)C1 Cc1nn(C)c(Cl)c1C=CC(N1CCCCC(NC(C2CC2(C)C)=O)C1)=O C1(C)(C(=O)NCC2N(C(C(C)CC3CC3)=O)CCCC2C)COC(C)(C)OC1 n1(CCN2CC3C(NC(c4cnn(C(F)(F)F)c4)=O)C3C2)cc([N+](=O)[O-])cn1 N1(C(CC=CC=C)=O)CCCCCC1CNC(C12CC(CO1)C2)=O C(=O)(C(C)(C)C(C)(C)N(C)C)N1CC(CCNC(C(C)NC(N)=O)=O)OCC1 C(=O)(C1Cc2c(Cl)cccc21)N1CCC(C)(NC(c2cnc(C3CC3)[nH]2)=O)CC1 CC1(C(=O)NC(c2ccccc2)C#N)CC12CCN(C(C1(C(=O)O)CC1)=O)CC2 Cc1nc(C(=O)NC2CC(O)(CNC(=O)Cc3cncnc3)C2)ccc1Br c1(C(=O)NCC2C(C(N3CC(C)(CC=C)C3)=O)CCCC2)cncn(C)c1=O C12(NC(c3c(C(=O)OC)ccnc3)=O)CCN(C(c3cnn(C)c3N)=O)CC1C2 N1(C(c2n[nH]cc2[N+](=O)[O-])=O)CC(C(N2CCCC3(CC3)C2)=O)C(F)(F)C1 CC1C(NC(=O)C(C)(C)N(C)C)CCCN1C(c1cccc(Cl)c1F)=O N1(C(C(n2cc(Cn3ncc(C)c3)nn2)C)=O)CCc2cc(F)cc(Br)c2C1 CCS(=O)(=O)c1ccc(CC(N2CCN(C(=O)CCCCCF)CC2C)=O)cc1 CS(=O)C1CN(C(=O)CCNC(C2CCCC(F)C2)=O)C1 c1(C(N2CCCC(C)(CNC(=O)C=CC(F)F)C2)=O)cc2nccnc2cc1F CC(C)C(CCNC(C1CC12CCC2)=O)NC(=O)CC1C=CS(=O)(=O)C1 C(=O)(N=c1nc(C(CC(F)(F)F)NC(COc2cccc(OC)c2)=O)[nH][nH]1)OC c1(C(=O)NC2C(C)CN(C(C3COCCO3)=O)C2)ccc2c(c1)NC(=O)C2(C)C c1(SCCNC(N2CC(c3cn[nH]c3)C2)=O)ccc(Cl)c(Cl)c1 c12cc(on1)C2.C1(n2cccn2)(C(=O)NCC2(NC(C)=O)CC2)CCC1 C=CCC(C(=O)N1CC(NC(c2cn3c(n2)CCC3)=O)C2(CC2)C1)C(C)C C(=O)(CCCCCF)NCC1(CNC(c2c(C#N)scc2)=O)CC12CCC2 N12CCC(C1(C)C)C2=O.C12COCCC1C(=O)N2.C(C(C)=CC(=O)OC)OC C1(C(=O)NCCC(C)NC(CNC(=O)OC)=O)CCCc2ccccc2C1 Cc1cc(N)c(C(=O)NCC(CNC(C2CC3CCC2O3)=O)C(F)(F)F)cc1F Cc1ccc(S(N)(=O)=O)c(NC(=O)NCC(C)(C)S(C)(=O)=O)c1 C1(NC(CC)=O)CCCN(C(=O)Nc2nc(-c3ccc(F)cc3)sc2C)C1 Cn1cnc2c1CCC(C(N1CCCC1C(C)(C)NC(=O)COC(F)F)=O)C2 c1(C(=O)NCC2CC(C)N(C(=O)C3=COCC3)C2)ccc2nc[nH]c2c1F c1(CC(C)NC(=O)NC2CC3CC3C2)cn(C)c2ccc(F)cc12 CCC(C(=O)N1CCC(Cn2cc(C3(F)COCCOC3)nn2)C1)C(C)(F)F C1(CC)CCC(C(=O)NCCOC2CCN(C(=O)Cc3ccc(Cl)cc3)C2)CC1 N1(C(C2CCC2C(=O)O)=O)CC(CNC2(CC3CC3)CC2)c2ccccc21 C1(C(C(=O)NCCCC=C)(C)C)CN(C(=O)CC23CCCC2C3)C2(CCC2)C1 C1(OC)Cc2ccccc2N(C(=O)C(C2CCCO2)C2CC2)C1 C(C(CC(F)(F)F)NC(c1c(F)cccc1F)c1cc(=O)n(C)o1)NC(C)=O CC(C)C(CCN(C(=O)CCN1CCCS1(=O)=O)C)NC(C1CC1C(F)F)=O Cc1ncc(CC(=O)N(CC(O)CN(C)C(c2coc(C3CCCC3)n2)=O)C)s1 c1(C(N2CCC(O)(C(N3CCCCC(C)(F)C3)=O)C2)=O)ccc2c(c1)NC(=O)C2 CC1CCC(NC(=O)CSC(F)F)CN1C(=O)C(O)C1CC1 N1(C(c2c(C)c[nH]n2)=O)CCCCCCC1C(=O)NOCC1(C)CC2CCC1C2 c1(C(=O)Nc2nc(Cl)ccc2I)c[nH]c2ccc(-c3ccc4ccoc4c3)cc12 N1(C(C(C)CF)=O)CCn2c(CNC(c3scnc3C(F)(F)F)=O)nnc2C1 C1(C(=O)NCc2cccc(CNC(=O)CC(F)(F)F)c2)CCn2ncnc2C1 c1(CC(C#N)N(C(c2ccccc2)C)CC)cc(F)c(F)cc1F CC(CC(C)(F)F)C(=O)NC1CCCC1CNC(c1cc(Cl)no1)=O N1(C(C2CC(=O)C2)C(=O)NCCCC2OCCO2)CCOCC1 C1(NC(c2cc(CCC)[nH]n2)=O)CN(C(c2cc(C)c(CC)o2)=O)C(C)(C)C1 c1(CC(=O)OC)sccc1C(=O)NCC1C=CC(NC(=O)C(C)N(C)C(C)=O)C1 C1(NC(C(C)C)=O)CN(C(C23CC(C)(C2)OC3C)=O)C2(CCOCC2)C1 CC1CCCC(CC(=O)N(C)CCN(C(c2nc(C3CC3)cs2)=O)C(C)C)C1 Cc1ccc(Cl)c(C(N2CC(O)(CNC(=O)CC3CC4C=CC3CC4)C2)=O)c1N C1(C)(CC(=O)N(C(C)CNC(=O)CCC2CC2)C)CCCO1 CN1CC(O)CC1(C)C(=O)NCC1CC(NC(c2ccc(C#N)o2)=O)C1 C(c1sc2ccccc2c1Cl)=CC(=O)NC1(C)CN(C(C(COC)(F)F)=O)C1 c1(C(=O)NC2CC3CC(NC(c4c(C)oc(Cl)n4)=O)CC32)cnc2cc[nH]c2c1 N(C1COc2ccc(F)cc21)C(C(=O)NC(C#C)CC1CCOCC1)=O Nc1cncc(C(=O)NCC2(F)CCC(CNC(=O)Cc3csnn3)C2)c1 c1(C(=O)NCCn2cc(C(=O)NC(CC=C)C)nn2)cc(CO)ccn1 c1(C(=O)OC)nc(C(N2CCCC2CNC(=O)C(C)Cn2cccn2)=O)sc1C c1(C(N2C(C)CN(c3cccc(F)c3)CC2)=O)cc2c(nc1O)CCC(C)(C)C2 C(CC(C(=O)NCC1CCN(C(N)=O)CC1)NC(=O)Cc1ccon1)OC C(=O)(C(CCF)OC(C)(C)C)NC.C(CCC(=O)C1(NC(=O)NC2CC2)CCC1)=CC S(=O)(=O)(c1ccccc1)NC(=O)C=CC1CC1.C12COCC1CNC(=O)C(F)=CC2 C1(CC(=O)NCCOC(C)(C)CNC(=O)CC2CNC(=O)O2)CCCS1(=O)=O c1(C(N2CCN(C(C3CC3(Cl)Cl)=O)CC2)=O)nccc(Br)c1O Cc1ccnc(C(=O)NC2CC(CNC(=O)Cc3ccccc3Cl)CC2O)c1N CN1CC(C)(C)CC1C(N1CCC(Nc2ccc(C#N)cn2)C1)=O N1(C(c2ccc(C)nc2Cl)C(=O)NC2COC2)CCOCC12CCCCC2 O=C1CCc2cc(N(c3nc(NC(=O)CCCCC4CCS4)cs3)CCO)ccc21 C(=O)(CC(C)C(F)(F)F)NCc1ncc(C(N2C(COC)CC2)=O)cn1 C1(CC(=O)NC(c2cccc(OC(F)(F)F)c2)CNC(C)=O)CCC12CCC2 C1(NC(C(C)OCCC=C)=O)COC2(C1)CN(C(c1cscn1)=O)C2 C(=O)(CC(C)C(C)(C)C)N1C(CNC(c2c(Br)c(C)n(C)n2)=O)CC1 C(=O)(C1=C(Cl)CCCC1)N(CC(CO)(CO)NC(=O)CCC1CCCN1C)C c1(C(C(=O)NCCC2(NC(CCOCCOCC)=O)CC2)O)cccnc1 C(=O)(C(C)CC(C)(F)F)OCC(=O)NCC1(NCc2ncc(C)o2)CCCC1 c1(C(N(C2CCCC2)CCNC(CCCSC)=O)=O)cnc[nH]c1=N c1(NC2(C)CC2(F)Cl)nc2c(c(=NCC3(c4ccc(C)cc4C)CC3)[nH]1)COC2 c1(CC)nc(C)c(C(=O)NCCOCCCNC(C2(C(N)=O)CCC2)=O)s1 CC1SCCCC1C(=O)NC(Cc1cn[nH]c1)C(N1CC(C)(C)C1C1CC1)=O N1(C(c2[nH]c(=NC)sc2)=O)CC(F)(F)CC1(C)CNC(c1ccc(=O)n(C)n1)=O C1(NC(=O)NCCC(=O)NC)CCN(C(=O)C2(CF)CCC2)O1 c1(CN(C)C(C2(NC(=O)Cn3cnnn3)CCSC2)=O)cnn(C)c1 C1(C(=O)NCC2(F)CCC(NC(C3CCOCC3)=O)C2)COC2(CCC2)C1 CC(C)(F)CCC(=O)N1CCC(n2cc(CNC(=O)CN3CCOCC3)nn2)C1 N1(C(c2ncc(OC)cn2)=O)CC(CNC(=O)CC(C)(C)C)C2(CC2)C1 C12(CNC(C(C=C)(C)O)=O)CC(C1)C(NC(c1sc(OC)nc1Cl)=O)CO2 C1(C(C)=O)CC2CCC(C1)N2N(C(=O)Nc1ccccc1OC(C)(C)C)C C1(NC(N2CCC(c3onc(C)n3)CC2)=O)CC(C)(C)OC1(C)C C(CC(=O)O)(C(F)F)NC(CCC1C(C)C1)=O c1(C(=O)NC2CCCCCN(C(c3ccsn3)=O)C2)cnc2c(c1)OCC(=O)N2 C12(CC(=O)NCCc3cccs3)CCC1CN(C(=O)Cn1ccnn1)C2 C(=O)(CCC(C)(F)F)NCCOCCCNC(CCc1cncc(OCC)c1)=O CC(C)(CS(N)(=O)=O)C(=O)NCC1CCCC(NC(c2ccc(O)nc2Cl)=O)C1 C(=O)(CCN(OC)C(=O)C(C)N1CCCCC1)N(C)C(c1nc(=O)o[nH]1)C C=C(Cl)CC(C(=O)NCCNC(=O)NC)NC(=O)CCn1ccnc1 C1(CCCCC(=O)O)NC(=S)N(CC2CC2)C(Cc2ccccc2)=C1C(=O)OC c1(C(N2C(CNC(c3nnc(C)s3)=O)CC(OC)C2)=O)c(F)cc(Cl)cc1Cl C(=O)(CCCC(F)(F)F)NC1CCC(F)(CNC(c2ccc(Cl)cn2)=O)C1 C12(NC(=O)CO)CCCC(CN(C(C34CCCC3CS(=O)(=O)C4)=O)C1)C2 c1(OC)ccccc1C(=O)NC1CC(CNC(c2cnc(CC(C)(C)C)s2)=O)C1 c1(CC(C)=O)ccc(C(=O)NC(c2cccc(Cl)c2)CF)cc1 C1(C(=O)NC2CCN(C(=O)OC(C)(C)C)CC2(C)C)CCn2c(O)nnc2C1 c1(N2C(C3CCN(S(CCC)(=O)=O)CC3)CCC2)cnc(F)c(C)c1 C1(C(C)C)CN(C(=O)C=Cc2ccoc2)CC1C(=O)NC(c1cnn(C)c1)CO C(N=c1nn[nH]n1C(C)C)C1(O)CN(C(C(C)c2ccsc2)=O)C1 [N-]=[N+]=NCCCCCC(=O)NC1CC=C(C(=O)N2CC(c3nn[nH]n3)C2)C1 CCCC(C)CCCC(=O)NC1CCC(NC(C2CC=CCC2C)=O)C1 c1(CCC)ccccc1C(=O)NCC(C(C)C)NC(=O)C=CCCC(C)C c1(C(N2CC(OCCNC(C3CC(CCC)C3)=O)C2)=O)coc(C#C)c1 c1(CC(N2CCC(F)(COC)C2)=O)ccc(Br)c(C)c1 c1(CNC(N2C(C(=O)NCCCCCl)COCC2)=O)cccc2ccoc12 S(=O)(=O)(c1cccnc1N1CC2CCCC12)N(C)Cc1c(C)cc(Br)cc1 Cc1ccc2oc(C(=O)N(C(C)CNC(c3nnsc3C)=O)C)cc2c1 C1(NC(Cc2ccc(C(C)=O)nc2)=O)CCCN(C(=O)C(=O)C2CCCC2)C1C C(N(C)N1CCN(CC(=O)NCC2CC2)CC1)c1ccc(C)cc1OC.C(=O)(C)NC N1(C(c2cncc(C#N)n2)=O)CCN(C(=O)Cc2ccccc2C#N)CC(O)C1 O=S(=O)(c1ccc(NCC2(CO)CC3CC3C2)c(Cl)c1)NCCC1CCC2(CC2)C1 N1(C(CC2(OCC)CCC2)=O)CC2(C)CC1(C(=O)NCC(C)(C)CCCO)C2 N1(CCOC)CC(C(=O)N(C2CN(C(c3ccsc3OC(C)C)=O)C2)C)CC1=O N1(C(=O)NC2C(C)SCCC2)CCc2ccc(O)cc2C1C Cc1csc2c(N3CCOCC(NC(C4C(C)C4C)=O)C3)ncnc12 Cc1ccc(C(C)C(O)C(=O)NCC#CCNC(c2cnc(C(C)C)[nH]2)=O)cc1 N1(C(C=C(CCC)C)=O)CCCC12CCN(C(c1cccc(Cl)c1)=O)CC2 C(c1ccncc1C)=CC(=O)N(CCCCC(=O)N1CC(O)CC1CN)CC Cc1cc(C(N2CSCC2C(=O)NC(C)CCC(C)C)=O)ncc1F C1(NC(C(C)N2CCC2)=O)CN(C(=O)CCc2cscn2)CC2(CCC2)C1 C1(NC(=O)C(F)F)CN(C(=O)CC(=O)NCCc2ccccn2)CC1C(F)(F)F Cc1c[nH]c2ncc(C(=O)N(C)CCNC(c3ccc(C4CCC4)cc3)=O)cc12 C1(CC#C)(C(N2CCOC(C3CC3)C2)=O)CCN(C(=O)CCc2nccn2C)C1 Cc1csc(=O)n1CCC(N1CCCC1C(C)(C)NC(=O)C(O)C1CCCC1)=O c1(CC(=O)NCCC2N(C(C3C(=C)CC3)=O)CCCC2)ccc(OC)cc1Cl C(CC(=O)N1CC(CF)C1)C(=O)NC1(C(O)CO)CC1 N1(C(=O)NCC(C)CC(F)(F)F)CC2CC1CN2C(=O)OC(C)(C)C C(=O)(CC(F)(F)C(F)F)N1CCCC(CC(=O)NCCC2CCCC23CC3)C1 N1(C(CCC#C)=O)C2CCC1CC(CNC(c1cc(C(N)=O)cc(F)c1F)=O)C2 C1(NC(c2cc(CC)on2)=O)(COC)CCN(C(c2cc(C(F)F)on2)=O)CC1 C(C(COC)C(=O)NCc1csc(CNC(=O)CC2COC(C)(C)C2)n1)OC C(CC(=O)N(C)CCC1CCCC1)(C(F)F)NC(c1c(C)coc1)=O Cc1cc(S(C)(=O)=O)ccc1NC(=O)CC1CCCN1C(=O)CC(F)(F)F N1(C(C(C2CC2)NC(C2=CCC(C)(C)C2)=O)=O)Cc2cccc(F)c2C1 c1(C(C(=O)N(CCC)CCNC(C2CC2(C)COC)=O)C)ccc(C#N)cc1 C1(CC(=O)NCCC2CCCN(C(C3C=CC=CC=C3)=O)C2)CCCC(CF)C1 N1(C(CN(C(C)=O)C)=O)CC(CNC(=O)CCc2nccn2C)C2CC12 N1(C(C(C)C(F)(F)F)=O)CC2(CCC(CNC(=O)C(F)(F)C(F)F)O2)C1 Cc1nn(CC(N2CCCCC2CNC(=O)C(C)n2cccn2)=O)cc1Br N1(C(C(C)OCOC)=O)CC(CNC(c2ccc(OC)cc2)=O)CC1(C)C c1(C(CNC(C2CC23CCC3)=O)NC(C2(C3CC3)CCC2)=O)ccc(Cl)c(F)c1 CCCC(C)(O)CC(=O)NC1CCOC1C(=O)NCC1CCC(CC)O1 C1(CC(=O)NCCOCCN(C(C(C2CCCC2)OCC)=O)C)CC2(CC2)CO1 c1(OC)ccc(CNC(=S)NC(C)C(=O)Nc2ccsc2)cc1 c1(OC)ccc(C2CCN(C(=O)CNC(=O)CCn3ccnn3)C2)cc1F C1(NC(CCC2CC(OC)C2)=O)C2COCC1CN(C(c1cc(O)nn1C)=O)C2 C1(NC(C23CC(C)C2C3)=O)CCCN(C(=O)CCC2NC(=O)NC2=O)C1C C12(C(N(C)CC3N(C(C4OCC(C)C4)=O)CCC3)=O)COCC(C1)OC2 CCC(C(=O)NCC(C)(O)CNC(=O)CNc1ncccn1)SC C(=O)(C(CCC1CC1)NC(c1scc(C)c1C)=O)NCC(CC)(C)OC c1(C(=O)NC2C(C)CN(C(=O)C(C)(C)C3CCC3)C2)ncc2n1CCCC2 c1(C(=O)NC2CCN(C(C3CC(=O)OC3)=O)C23CC3)cc2cccnc2o1 CON(Cc1cn(CCN(C2(C(N)=O)CC2)C)nn1)C(=O)C(C)N1CCCCC1 N(C1CN(C(=O)C2=CCOC2)Cc2ccccc21)C(c1cc2cnccc2[nH]1)=O c1(C(=O)NC2C(NC(c3c(COC)cccc3)=O)CC2)nn(C)c2c1CCC2 C1(C(=O)NC2CN(C(=O)Cc3ccoc3)CCC2CO)CCC(=C(F)F)CC1 c1(CC)ccc(NC(c2cc(C(F)(F)F)cc(Cl)n2)=O)c(OC)n1 c1(C(=O)NCC(C)NC(c2ccc(F)cc2Cl)=O)ccc(Br)nc1N c1(C(=O)NC2(CNC(c3cc[nH]c3)=O)CCC2)ccc2c(c1)NS(=O)(=O)C2 C#Cc1ccc(C(=O)NC2(CO)CN(C(=O)Cc3ccsn3)C2)c(F)c1Cl c1(C(N(C)CC2(CNC(=O)C3=CCCC3)CC2)=O)ccc(=O)n(O)c1 c1(CC)ccc(C(=O)NCCCCNC(c2ccn(C)n2)=O)cc1C#N N#Cc1nnc(N(C)CC2CCN(C(=O)CNC(c3ccc(F)cc3)=O)CC2)s1 Cc1cncc(C(=O)NC2CC(NC(=O)CC3CCNC3=O)C2)n1 C(=O)(C(C)C(=O)NCC12CC(CNC(C3CCC(C(N)=O)C3)=O)(CO1)C2)OC c1(NC(c2[nH]c(C)c(C(=O)NC3CNC(=O)C3)c2C)=O)ccc2ncnn2c1 c1(NC(=O)NC(C(C)C)Cc2nccn2C)ccccc1Sc1ccccn1 C1(C(=O)NCC2CC(F)(CNC(=O)CCn3cc(Cl)cn3)C2)CC12CCSCC2 c1(CNCc2c(C)nc(C)[nH]2)ccc([N+](=O)[O-])c(-n2ccnc2)c1 C=CCC(C(=O)N(C)Cc1cccc(CNC(C2CNC(=O)C2)=O)c1)OC C(C)(C(C(=O)N(C)Cc1ccc(O)cc1)C(C)C)NC(c1c(C)cco1)=O C1(C(=O)NCC2C(C)(C)C2(F)F)(CNC(CCc2n(C)ccn2)=O)CC12CCC2 N1(C(c2cccc(CC)c2)=O)CCC(NC(=O)CC2CCC(=O)C2)CC1C C(=O)(CCCCCC(C)(C)C)N1C(CNC(CC(=O)N(C)C)=O)C(C2CC2)CC1 CS(=O)(=O)CCCCCCCC(=O)NC1CCC1NC(=O)C1=COCCO1 CC(CO)(C(=O)NCC(O)C(F)(F)F)NC(=O)CCOC1CCC1 c1(OC)ccc(C(=O)NC2CC(NC(=O)C3=C(C)CC3)C2)cc1OC c1(COc2nnc(C(C3C(SC)C3(C)C)c3ccccc3)o2)ncc(NC(C)=O)s1 CC1CCn2ncc(C(=O)NCCC3(NC(=O)C=C(Cl)Cl)CCCC3)c2C1 c1(CNC(C(=O)Nc2nc(SC)sc2)=O)ccc(C(F)(F)F)cc1[N+](=O)[O-] CC(CCN(C)C)C(=O)N(CCC(=O)NCc1cccc(O)n1)C CC1(C)CN(C(=O)CC2C=CCC2)CC1NC(=O)CCCC(F)F CCC(C)C(C(=O)NCc1nn(C)cc1C)N(C(=O)CCc1cnco1)C Cc1cc2occ(C(=O)N(C3CCN(C(=O)C(C)C(C)O)CC3)C)c2cc1C CC(C(C)(C)C(=O)N(C(C(N)=O)C1CC1)C)NC(=O)CCc1ccnn1C Cn1ncc(C#N)c1C(N1CCC(O)(CNC(=O)CC2CCS(=O)(=O)C2)C1)=O c1(CNC(C2CC(C(=O)Nc3ccc(C4CC4)cc3)C2)=O)ccncc1F C#Cc1ccc(C(N2CCCC(N(C(c3cc(Cl)ns3)=O)CC)C2)=O)c(C)c1 C(=O)(C1=CCCCC1C)N1CC(OC)C(C(=O)NCC2(C3CCC3)CC2)C1 c1(-c2ccc(CC)nc2)ccc(C(=O)NCc2csc(C3CC3)n2)c2[nH]ccc12 C1(NC(c2cnsc2)=O)CCC2CCN(C(C34CC3Cc3c[nH]nc34)=O)C12 C(=O)(CCN=c1[nH]ccs1)N1CCC(NC(c2c(C)snn2)=O)C(F)C1 C12(CC(=O)Nc3cn(CCC#C)nc3C)CCC1CN(C(C1CC(C)=NO1)=O)C2 c1(C(N2CC(CCCNC(=O)CCF)OCC2)=O)cc2c(Cl)nccc2o1 CC(C)CCCC(C)C(=O)NCC1CCNCC1O CC1CN(C(c2cccnc2O)=O)CCCN1C(=O)Cc1nnc(S)n1C C1(C(=O)NC(c2nc(C)[nH]n2)C)CC2(CCN(C(=O)C=CCO)CC2)C1 Cc1ccc(OCC(=O)N(C)CCNC(=O)C(C)C=Cc2ccccc2)c(C)c1 c1(CNC(CC2CCN(C(COCCOC)=O)C2)=O)ccc(Br)cc1 CCCCCC(F)C(=O)N1CC=C(C(=O)NC2(COC)CC2(C)C)C1 c1(OC)cc(F)c(F)cc1C(=O)NCC(C)NC(c1nc(C(=O)OCC)sc1)=O C1(CN=C(NNC2(c3nc(C)on3)CCC2)NC2CC2)C(F)(F)C12CCCC2 CCC(C)CCC(O)CC(=O)NCC1CC(NC(c2cn(C)nc2C2CC2)=O)C1 C1(=CC(N2C(C)CCC(NC(C3COC(C)C3)=O)C2)=O)C2CC3CC(C2)CC1C3 C1(NC(C(C)CC(F)F)=O)CCC2(CC1)CN(C(=O)Cc1cnccn1)CCO2 c1(C(N2CC(CN(C)C(C3COCCO3)=O)OCC2)=O)ccnc(F)c1N C1(C(=O)NCC2CN(C(c3nc(C)sc3)=O)C2)CSc2ccccc2O1 c1(C(=O)NC2C(CNC(C=CCOC)=O)CCCC2)ccc2ncccc2c1 CN1CCC=C(CNC(C23CCC(CC2NC(C2CC4CC4C2)=O)C3)=O)C1 N1(C(c2n(CC)cnn2)=O)CCC(N(C(=O)C2=COCC2)C)C(C)C1 c1(C(C(N2CC(NC(CCCC)=O)C(C)C2)=O)C)ccc(C)c(Br)c1 c1(C(=O)NC2C(CNC(CCS(C)=O)=O)C2)cc2cccnc2cc1F C(=O)(C1c2ccccc2CN1c1ncccn1)NC C1(N(C(c2c(C)cccc2)=O)C)CN(C(=O)Cc2c(C)cnn2C)CC12CC2 c1(CC(=O)NC2C3CN(C(C4CC(C)(CC)C4)=O)CC32)c[nH]c2ccncc12 c1(N2Cc3c(=N)[nH][nH]c3CC2)nc2ccccc2c(=NC(CF)CF)[nH]1 N1(C(C2(CCF)CC2)=O)CCC(C(C)(C)CNC(C2(C)CC2Br)=O)CC1 c1(CN(C(C(=O)OC)C)C(C2CC3CC2CC2(CC2)C3)=O)cc(Br)cc(C)c1OC C(=O)(C1CCCc2nccn21)N1CC2(CN(C(=O)C(F)n3ccnc3)C2)C1 C1(C(=O)NC(c2cc(Br)c(Cl)s2)C)CCC12CNC2 c1(CC)ccnc(C(N2CCCC(N(C(=O)Cc3csnc3C)C)C2)=O)c1 C#Cc1cc(C(=O)N(C(C)CNC(C2CC2CN(C)C)=O)C)cc(F)c1 Cc1ncc(-c2cnc(C(=O)NCc3cc(Cl)ccc3F)cc2C)cc1C#N N1(C(CCc2onc(CC)n2)=O)CCCN(C(C2CC3(C2)CC32CC2)=O)CCC1 C1(N(C)C(c2ncc[nH]2)=O)CCCC(C(=O)NCCc2ncc[nH]2)C1 C1(C(=O)NC(C)CCCNC(c2cnn(C)c2C(F)(F)F)=O)CCC=CCCC1 C=CC1CCCCN1C(=O)N(CC(O)CF)C1CC1 N(C(=NCc1nc(C(C)O)n[nH]1)N1CC2C(CF)C2C1)Cc1cccc(CC)c1 c1(CC(CN(C)C(C2COC2)=O)NC(C(C)OCCC(C)C)=O)ccccc1 C12(C(=O)NCCC3CCN(C(C4(CC)CCCC4)=O)C3)CC1CNC2=O C1(CN(C(=O)C=Cc2ccco2)C)CCCN(C(=O)C2=COCC2)C1 CN1CCc2cc(CC(=O)NC3CCCC3NC(=O)CC3COC(=O)C3)ccc21 C(C(=O)NOCC(=O)NCCC(=O)N(C1CC1)CC1CC1)(C1(C)CC1)OC C(=O)(CCCS(C)(=O)=O)NC1C(NC(CCC(=O)NCCC)=O)CS(=O)(=O)C1 C12(NC(CCCCSC)=O)CC(CNC(c3cnoc3C)=O)(C1)OC2C N1(C(C2OCCN(CC)C2)=O)CCC2CCC(C1)N2C(c1cnoc1C1CC1)=O C#Cc1ccc(Nc2cccc(CNc3ncc(Cl)cc3F)c2)cc1 c1(C(N2C(C)CC(CNC(c3ccoc3Br)=O)C2)=O)nccc2ccn(C)c12 Cc1cnn(C(C)C(=O)NCC(F)(F)C2CNC2)c1 O=C(CCCC(=O)N1CCN(C(=O)CCS(N)(=O)=O)CC1CC(F)F)NC1CC1 N1(C(Cn2c(C(F)F)cc(C)n2)=O)CCC(C)C(CN(c2ccccc2)C)C1 c1(C(N2CC(O)(CNC(C(CC)N(C)C)=O)C2)=O)c(C)coc1C CC1(C)CCCN(C(=O)C=CC(=O)NCCCN2CCCC2)C1NC(=O)CCF Cc1cc(CN(C2CCCC(O)C2)C=O)cc(O)c1 Cc1ccc(C(=O)NC2C3CN(C(=O)CCc4nc(C5CC5)no4)CC23)cc1F C1(O)(C(=O)NCC2CC2CNC(c2ccc(OC)nc2)=O)CN2CCC1CC2 C=CC(C)(C)CCCNC(c1c[nH]nc1CNC(=O)C(C)NC(N)=O)=O N1(C(C(C)(N(C(c2c(CCC)nco2)=O)C)C2CC2)=O)CC(C)CC(O)C1 c1(CC(N2CC(c3cn(CCC)nn3)(C)C2)=O)ccc2nc(OC)ncc2c1 Cc1nc(CC2CN(C(c3coc(N(C)C)n3)=O)C2)sc1C(=O)OCC.C(C)(C)(C)O C1(C)(C(=O)NCCCC(C)NC(c2c[nH]c(Br)c2)=O)CCCC1(F)F c1(CC(N2CCC(N(CCC)C(c3cc(Cl)no3)=O)C2)=O)ccc2[nH]ccc2c1 N1(C(CCC(=O)NCCC2CC2)=O)CCc2c(Cl)cc(F)cc2C1 c1(C(N2C3C(NC(C4(OCC)CCCCC4)=O)C(C3)C2)=O)nc(C)n(C)c1C c1(C(=O)NCC2(O)CCCN(C(C3CC(CCC)C3)=O)C2)ccc2c(c1)OCC2 N1(C(c2cc(C(C)=O)oc2)=O)CC(NC(=O)CSc2ncccn2)C(C)C1 C1(NC(C2(C(N)=O)CC2)=O)CCC2(CCN(C(C3(N4CCCC4)CC3)=O)CC2)C1 N1(C(Cc2c(C)nn(C)c2C)=O)CCN(C(C23COC(C2)C3)=O)C2CCC12 Cc1cnc(C(=O)NCC2CCN(C(=O)CCc3cccc(C(N)=O)c3)C2)nc1 c1(C(c2n(CC)nnn2)NCC(CO)OC)cccc(OC)n1 N1(C(CNC(=O)NCCOC)=O)CC(N(C(=O)COC)C)CCC1C c1(N(C)C)nc(C(=O)NC2CCOC(CNC(C3CC(C)(C)C3)=O)C2)cc(O)n1 C12(CCCN(C(=O)C(CC)=CC)C1)C(=O)NC2.c1(CCC)ccccc1OC C1(C(=O)NC(C(=O)NC2(C(N(C)C)=O)CC2)CO)CC(=O)CC12CCC2 c1(C(=O)NC2(CO)CN(C(=O)CN3CC4CC4C3)C2)cc(Cl)cc2c1CCC2 c1(C(=O)OCC)nn(C)cc1C(N1CC2CC2(CNC(c2coc(Cl)c2)=O)C1)=O C1(C(=O)NC(CN(C)C)C(=O)NCCN2CC3CC3C2)CC2CC1CC2O C1(C(N(C2CC(NC(c3c(OC)ccs3)=O)C2)C)=O)Cc2ccccc2O1 N(C1CCCc2sccc21)C(c1n(C(C)(C)C)nnn1)CC1CCCOCC1 C(=O)(C1=CCCN(C(c2ccnn2CCF)=O)C1)NC(C)Cc1ncn(C)n1 Nc1cc(C(=O)NC2CC(F)CN(C(c3ccoc3)=O)C2)ccc1S(N)(=O)=O C1(C)(CC)CN(C(=O)C=CC2CCN(C(=O)Cn3cnc(C#N)n3)CC2)CCO1 C1(NCCC(=O)NCC)CCC(n2cc(CCc3nn[nH]n3)nn2)CC1 C1(CCC(=O)NC(C(C)C)CN(C)C)CCCCN1C(c1ccccc1)=O CS(=O)c1ccccc1CC(=O)NCCC(C(C)(C)C)N(C)C.C(=O)(CCC1CC1)N C(=O)(C(F)C(=O)NCC(C1CCCC1)NC(c1sc(C(C)C)nc1C)=O)OCC c1(C(N(C)CC2CCCN2C(=O)CC2CCCO2)=O)ccc2c(c1)CCCC2 N1(C(C(CCC#C)O)=O)CCn2c(CNC(=O)C(CC)CC(F)(F)F)nnc2C1 CCS(=O)c1ccccc1C(=O)NC(C(N)=O)C(C)O C1(NC(c2nc[nH]n2)=O)CCN(Cc2ccc(O)c(I)c2)CC1F N1(C(C2CCC(C3CC3)N2C(=O)CCCCC2CC2)=O)CCCC2CCCCC12 c1(C(=O)NCC(C)NC(c2coc(Cl)c2)=O)c(N)cc(Br)cc1Cl C1(C(N2CC(NC(CC(C)F)=O)C2)=O)CCC(F)(COCC2CCOCC2)C1 c1(C(=O)NCC2(CN(C(CCSC)=O)C)CCC2)cc(C(N)=O)c[nH]1 CC1(C)CCN(C(c2sccc2C(F)F)=O)CC1CNC(=O)CC1CCC(=O)N1 C(=O)(C#CC1CCOC1)NCC(CNC(Cc1cc(C)sc1)=O)(C)C CCC(CC(F)F)C(=O)N1CCCC(F)(CNC(=O)CC23CCC(CC2)OC3)C1 CN1CCC2CCN(C(C3CN(C(=O)C=Cc4ccsc4)CC3C3CC3)=O)CC12 C(=O)(C1Cc2ccc(Cl)cc21)N1CCC(C)(NC(c2c(Cl)cnc(C)n2)=O)C1 c1(S)ccc(Cl)cc1.CCC(CNC(=O)COCCF)NC(=O)CC N1(Cc2ncn(C)c2)CCN(C(c2ccc(Br)cc2)C(=O)NC2CCCC2)CC1 C=CC1CCCCN1C(C1CC(NC(c2c(C)ccn2C)=O)C1)=O N1(C(C2(N(C)C)CCOCC2)=O)CC(NC(C2COC(=O)N2C)=O)C(C)(C)C1 C1(F)(CN(C(C2CC(NCc3sccc3Cl)C2)=O)CC)CCOCC1 C1(N(C(CN(CCC)C)=O)CC(C)C)CCN(C(C2OC3CCC2C3)=O)CC1 C1(O)(C(N2CC(C(C)NC(c3cccc(-n4cccn4)n3)=O)C2)=O)CCCOC1 C12(C(=O)NC(CCOC)COC)CC(CCO1)N(C(c1cnn(C)c1)=O)C2 c1(C2(O)CC(NC(c3c(C)coc3)=O)C2)ccc(F)cc1 C1(C(C)C)C(C(=O)N(CCCN(C)C)C)CCN1C(=O)CCc1cn(C)nn1 C1(C(=O)NCCCCNC(c2cccnc2)=O)CCCCC12CC2 CCC(C)(C#N)C(=O)N1CCC(OCCNC(=O)C(C)(C)c2ccc(Cl)s2)C1 N1(C(CCOCCCNC(C(C)S(C)(=O)=O)=O)=O)CCC(O)CC(C)(C)C1 S(=O)(=O)(c1ccc2ccccc2n1)N1CCCC(C)(C(=O)OC)C1 c1(CCC)ccccc1C(=O)NC1CC2C(NC(C3CCCS3)=O)C2C1 C1(CN(C(CCSCCCC)=O)CC)CCN(C(=O)CC(C)N(C)C)CC1 c1(CNC(C2(F)CCN(C(CCc3nccc(C)c3)=O)C2)=O)cc(C)ccc1C c1(C(=O)N(C2CCN(C(C(CC)n3ccnc3)=O)C2)CC)c(C(F)(F)F)coc1C c1(C(=O)NCC(COC)C(=O)O)cc(N)cnc1Cl C=CCC(C)(C)C(=O)N1CCCCC(CNC(C23CCC(OC)C2C3)=O)C1 N1(C(CCC=CC(C)C)=O)CCCC(OC(C)C)C1.C1CC(=O)N1C1CC1 N(C1CC(C)n2ccnc21)C(C1(CC=C)CN(C(c2cc(C)ccc2F)=O)C1)=O C12(C(N(C)CCn3cnnc3)=O)CCC(CN(C(=O)CC3CC3C3CC3)C1)C2 C(CCC(C(=O)N1CCC(C(C)(C)C)CC1)NC(=O)Cc1ccc(F)nc1)OC c1(N(CCOC)CCNC(C2CC23CCOC3)=O)ncnc2ccc(O)cc12 c1(C(=O)NCCC(C)NC(=O)CS(N)(=O)=O)cc(Cl)c(N)c([N+](=O)[O-])c1 CC#CCCC(=O)N(C1CC(NC(c2ncc(C(F)(F)F)s2)=O)C1)C CC(CC(=O)c1ccccc1F)C(=O)NC1(CCNC(C2CCC2)=O)CC1 CC(CC(C)NC(c1cnoc1C1CC1)=O)NC(c1cn(CC(N)=O)nn1)=O C(=O)(C1c2ccccc2C2CC1C2)NC(CNC(c1ccc(CSCC)o1)=O)C C1(CNC(c2c(C(=O)OCC)c[nH]n2)=O)CC2CCC(C1)N2C(C1CCOC1)=O N1(C(C(C)(C)n2cccn2)=O)C2CCCC1CC(NC(C1CCCCO1)=O)C2 C(=O)(CCC(C)OC(C)C)NC(COC)C(=O)NC(c1nncn1C)CO CC(C)(CCC#N)C(=O)NC1CCC(NC(=O)Cc2cc3ccccc3s2)CC1 N1(C(CN(C)C(C2CCCCN2C(=O)C(N)=O)=O)=O)CCCN(C2CC2)CC1 C(=O)(C(C1=NOC2COCC12)N1CCN(C)CC1)C(=O)C(F)(F)F.C1(CN)CCCC1 CCCCC(CC)CCC(=O)NCCC(C)(C)NC(=O)CCc1cscn1 CC1(C)CCN(S(=O)(=O)c2cccs2)C2CCOCC12 c1(C(N2CC(C(C)NC(c3cnn(CC(F)F)n3)=O)C2)=O)cc2c(s1)CCC2 C1(O)(C(N2CCC(C3N(C(C=NOC)=O)CCC3)C2)=O)Cc2ccccc2C1 c1(C(=O)NCC2(C)CCC(NC(CN3CCC(C)CC3)=O)C2)cn(C)c(=O)cn1 N1(C(C2(COC)CCCO2)=O)CC2C(CNC(c3cc(C(C)=O)c(C)[nH]3)=O)C2C1 C12(NC(C3(N(C)C)CC3)=O)CCCC1N(C(c1cnns1)=O)CC2 c1(Nc2cc(O)c(F)cc2F)ncnc2[nH]cc(I)c12.CC12CN(C1)C2=O O=C(O)CCC(CN1CCC1C1CCC(=O)O1)C(=O)O N1(C(C(CC=C)CC)=O)CC2CC1CCC2NC(C1(CC2CC2)CCCO1)=O c1(C(C)C)ncncc1NCC1CN(C(=O)CC(C)n2cccn2)C1 C1(CNC(C2CC(=C)C2)=O)CC2CC(C1)N(C(c1nc(NC3CC3)sn1)=O)C2 C(C1CSc2ccccc21)n1cc(C(O)C2CC2)nn1 N1(C(C=C(C)C2CC2)=O)CCCC2(C1)C(NC(=O)Cc1csnn1)CCN2C C1(CN(C(=O)CS(=O)(=O)NC2CC2)CC)CCCCN1C(C1CC1C)=O CCC(CC)CC(=O)N(C)CC1CCN(C(c2cnc(C)o2)=O)C1 Cc1c(Cl)ccnc1C(=O)N(CCCNC(=O)CCCc1nncn1C)CCO C1(NC(CC(CNC(c2cnc(CC)s2)=O)OC)=O)CCOC(C)(CC)C1 C(=O)(C(C)C(O)CC)NC(CC)CNC(c1ccnc(N2CCOCC2)c1)=O CCC(C)(C)CCCC(=O)N1CCCCC1C1CCN(Cc2cccc(Cl)c2F)C1 C1(NC(=O)COCC2CCCO2)CC2CCC1C(NC(c1ccccc1F)=O)C2 N1(C(=O)OC(C)(C)C)CCCC2(CC(C(=O)OC(C3CC3(Cl)C(=O)O)=O)C2)C1 C1(NC(C2CC(N(C)C)C2)=O)CCC(C)(CNC(c2cc(O)cs2)=O)C1 Cc1cc(F)c(CCNC(=O)NCC(CCO)CC(C)C)cc1Br C1(CC)CCC(C)CN1C(c1cc(CNC(=O)C(C)(CC)CO)no1)=O c1(C(=O)NCC2OCCC(NC(CC(=C)C)=O)C2)ccc2ncsc2c1 C1(F)(CNC(CN(CC(C)(C)C)C)=O)CCN(C(C2CC=CCC2)=O)C1 CCCCC(C(=O)NCC(CC)N(C(=O)CNS(=O)(=O)NC)C1CC1)NC(N)=O C1(C(=O)NCCOC(CC)CC)C=CCN1C(=O)CC1C=CCCC1 c1(C(N2CC3C(NC(c4cccc(C(F)(F)F)c4)=O)(C3)C2)=O)ccc(O)c(Cl)c1 c1(C(N2CCC(OC)(CNC(C3CCC(C)O3)=O)C2)=O)c[nH]c(C#N)c1C c1(-c2cncc(OC)n2)ccn2nc(C(=O)Nc3ccc(Br)nc3C)cc2c1 N1(C(CSC(C)(C)C)=O)CC(NC(c2ccc(Br)o2)=O)C(O)C1 Nc1ccccc1COC(C1(C2CCC2)CC1)=O Cc1ncc(C(N2CCC(CCOC(=O)CC3COCCO3)CC2)=O)n1C c1(C(C)C)cccc(C(=O)NCCC(O)CNC(=O)C(C)(C)N2CCOCC2)n1 C1(C(=O)NCC(CC=C)NC(c2cccc(C(N)=O)c2C)=O)CCC2CC2CC1 CC1(CO)CN(C(c2ncc(-c3ccc(C#N)nc3)cn2)=O)CCC1O N1(C(C(C)OCCC=C)=O)CCCC(C)(C(N2CCCSCC2C)=O)C1 N(C(=NCCOC(C)C)NCC1CCCCC1)C(C1CCCCC1)C#C c1ccc(COCCCc2cccnc2)cc1.C12(CCOC1)CNC2 CCC(C)(C(=O)NCC(C)(C)CN(C)C(c1c(C)ccc(C)c1C)=O)C(N)=O c1(CC)cc(C)c(C(=O)NC2CC(CCNC(=O)CCc3cnco3)C2)o1 N1(C(C2CN(C(C)=O)C2)=O)C(C)CN(C(=O)C(C)n2cnnn2)CC1C C1(C(=O)NCC)CCC(c2nc(CC(CC(C)C)OC)no2)CC1 CC1CCN(C(=O)Cc2cn3ccsc3n2)CC1NC(=O)C1=CCC1 c1(C(=O)NCC2CC3CC3N2C(=O)Cc2ccns2)cc(F)c(F)c(F)c1F C(=O)(C1CCCc2ncnn21)N1CCC2(N(C(CCC(C)(C)O)=O)CCC2)C1 n1(CC=C)cc(C(=O)N(C(C)CNC(c2nc(C(C)(C)C)no2)=O)C)nn1 C1(NC(CCCn2c(C)ncc2)=O)CC2CCC(C1)N2C(=O)CC1CCCCC1 c1(CNc2ccc(C(C)O)cc2)cc(F)ccc1C(F)(F)F CN1CC(O)CC1(C)C(=O)NCC1CC(NC(=O)CCCCN(C)C)C1 c1(CC(=O)NCC(CC=C)NC(c2c[nH]nc2OCC)=O)ccc([N+](=O)[O-])cc1 CCCCC(CC)C(=O)N1CCN(C(c2cnn(C)c2C(C)C)=O)C(C2CC2)C1 C1(OCC(=O)NCc2c(C(=O)NC3C(CCOC)C3)occ2)CCCCC1C C1(NC(C)=O)CCCN(C(=O)NC)C1.N1(CC)CCOC(c2n[nH]c(C(F)(F)F)n2)C1 CC1(C)CC(CNC(C2CC(F)C2)=O)N(C(=O)Cn2ccc(Br)n2)C1 C1(CNC(c2c(C)nn[nH]2)=O)CN(C(c2csc(O)n2)=O)CC1c1ccccc1 Cc1ccc(=N)[nH]c1C(=O)NC(C)(CNC(=O)C(c1ccc(F)cn1)(F)F)CO c1(CNC2CCN(C(c3ccc(Cl)cc3)=O)C2)cc(Br)ncc1F C(=O)(NN=c1cc[nH]c(=N)[nH]1)OCC(c1cc(C)n(CC(C)C)c1C)=O CCCCC(CC(=O)NCC(C)CC1CCC1)NC(=O)C=CC1CCCC1 c1(OC)ccc(C(=O)NC23CC2CN(C(=O)COc2ccncc2)C3)cc1OC C(=O)(C1CCCc2c[nH]nc21)N1C(CNC(c2cscc2Cl)=O)CC1 c1(C(N2CCC(NC(c3cn4c(n3)CCC4)=O)C2)=O)cc2ccncc2c(O)n1 c1(C(N2CC(CNC(C(C)CC3CCC3)=O)OCC2)=O)ccnc2c1CCC2 C(CC(CNC(c1scnc1Br)=O)NC(C1(OC)CCC1)=O)OC C1(C#N)(C(=O)NCCN(C(CNS(CC)(=O)=O)=O)C)CC2(CC2)C1 C1(C)(CC(=O)NCCCN(CCCCNC(C(C)O)=O)C)OCCO1 c1(N(C(C2CCCC2)C)C)ccc2nccnc2n1.CC(C)CC(C)(C)C(=O)N c1(CC)ccc(C(N2CCN(C(=O)Cn3ccnn3)CC2C)=O)c(Br)c1 C1(C)(CC)CC(CN)C1.C12CC(C1)C(=O)NCCCO2.n1(CC)ccnn1.C1CO1 C1(NC(COCC=C)=O)C(C)CN(C(c2coc3c2COC3)=O)CC1C C1(CNC(c2n(C)ncc2)=O)CCC2CN(C(c3cnoc3)=O)CCC2C1 C1(C(=O)OC(C)C)CCCN(C(C)(C)CNC(N2CCCC2c2ccc(Br)s2)=O)C1 c1(C(=O)NCC2C(CNC(CCCC#CC)=O)C2)cnc2sc(C)cn2c1=O C1(C(N2CC(NC(c3ccccc3CO)=O)CC(C)C2)=O)CC2C=CC1C21CC1 CCCC(CCC)CC(=O)N1CCCC1C(C)(C)NC(=O)CC1(O)CCCC1 N1(C(c2ncc(C)c(C)c2)=O)CCN(C(C2CCN2S(C)(=O)=O)=O)CC2(CC2)C1 C1(C(=O)NC(CC(C)NC(c2c(OC)c[nH]n2)=O)C)CCC(C(=O)OC)CC1 C=CCCC(C(=O)NCC1CC(NC(=O)CC2(C)CC2)CCO1)c1ccccc1 CC1CN(C(C2C3CN(C(C4CCC(C#N)CC4)=O)CC23)=O)CC(=O)N1C CN1CCOC(C(N2CCCC2C(C)(C)CNC(C2CC3C=CC2C3)=O)=O)C1=O Cc1ccc(C(=O)NCCC(C)(C)NC(=O)C(c2nc(F)ccc2Cl)C)c(C)c1 c12ncc(s1)CN(Cc1ccccn1)C2=O.N(CCOC)(CC)CC C1(NC(CC=CCC)=O)CCN(C(=O)Cn2nnc(C(C)(C)C)n2)CC1CC N1(C(c2cnc(CS(C)(=O)=O)s2)=O)CCCCC1C(O)C(F)F CC1(C)COC(CC(N2CC(CNC(c3c[nH]nc3C(F)F)=O)C2)=O)C1 c1(CC)ccc(-c2cn(CC3CCN(C(c4cnc(Br)o4)=O)C3)nn2)s1 N1(C(C)C)CCOC(C(=O)N(C)CC2(NC(=O)CCc3ccccc3F)CC2)C1 C1(NC(C(C)CC2CC2)=O)CC2CCC(C1)N2C(C1CN(CC(F)(F)F)C1)=O C(CC(C(=O)NCC1(C)CCCC1O)NC(=O)C(c1ccccc1)F)OCC n1(CC(=O)N(CCCNC(C(C(CC)O)C)=O)C)nc(C)c([N+](=O)[O-])c1C c1(CC(=O)NC2(C(N(CC(CCC)C)C)=O)CCCC2)ncccc1F Cc1ccc(C2(C(N3CCOC(CNC(C4(O)CCC4)=O)C3)=O)CC2)cc1Cl c1(C(N(CC(C)NC(C2(C)CCCO2)=O)C)=O)cc(F)c(F)cc1O C1(C(=O)NC(C2CC=CCC2)C#C)CCN(C(c2cnn(C)c2N)=O)CC1 C1(C(N2CCCC(O)(CCNC(C=CSC)=O)C2)=O)COCC2(CCC2)O1 N1(C(c2cc(F)c[nH]2)=O)CC2(CCN(C(=O)C(F)(F)CC3CC3)C2)C1 C1(CNC(C(C)OC(NOCCC(C)C)=O)=O)CCCCCCO1 c1(C(=O)NC(CC(C)NC(CC(=C=C)C)=O)C)ccc2nnc(C(F)F)n2c1 C(=O)(C(C)C(=O)N1CCCC(CCNC(=O)COc2ccccc2)C1)OC Cc1cc(C=CC(=O)NC(CC(=O)NC(C)Cc2ccccn2)C2CC2)on1 CC(C)CC(CC(C)C)NC(=O)NC(CCN1CCOCC1)C(C)C c1(C(C(=O)NC)N(C)Cc2cc(OC)ncc2Br)ccc(C(=O)OC)cc1C Cc1cnn(CC(C)NC(=O)CCN(C(=O)C(C)OCCN(C)C)C)c1 N(C1CCc2c(O)cccc21)N1C(C2C(O)CCC(C)C2)CCC1 N1(C(C(c2ccccc2)OCC)=O)CCN(C(=O)C(O)CC2CCCC2)CC1C N1(CCS(C)=O)CCC(c2ccc(Cl)cn2)CC1 C(=O)(CN=c1cc[nH]cc1)NC(CC=CC)C(=O)NCc1cc(C)ccc1F c1(C(=O)NCCN(C(CN2CC(COC)C2)=O)C)cn2ccccc2n1 C(=O)(CC(C)(O)C(F)(F)F)N(C)CC1CCC(NC(CC(=O)NCC)=O)CC1 n1(CCC(=O)NC(CN(C(CN(C(=O)OCC)C)=O)C)C)ncc2c1CCCC2 C1(C)(CC(=O)N(CC)Cc2cnn(C)c2)CCN(C(c2ccc(C)cn2)=O)C1 CCCCC(O)CC(=O)N(C1CN(C(c2cnccn2)=O)CCC1O)C N1(C(C2CCC(=O)O2)=O)CCC(F)(F)C(CNC(=O)C(O)CC2CCCCC2)C1 CCCC(C)(C)C(=O)N(C1CC(NC(C2CCCN(C(N)=O)C2)=O)C1)C Cc1cc(CCC(=O)NC(C)C(C)(C)NC(=O)CC2COCC2O)on1 Cc1c(C(=O)NCC2CCCC2NC(=O)CC(C)F)cnn1-c1ccccc1Cl c1(C(=O)NCCO)cn(C2COCC2CNC(C)C)nn1.C1(NC=O)(CO)CCCC1 c1(C(=O)NC(C2C3CCC(C3)N2C(=O)COC2CC2)C)cn2cccc(F)c2n1 C(C(=O)N1CCC(CNC(c2ccoc2-c2ccccc2)=O)CC1)(C(C)C)OC c1(N2CCN(S(CC)(=O)=O)CC2)nccn2nc(C)cc12.C(C(=O)O)N N1(C(C=CC(CC)=CC)=O)CCC2CC2(NC(=O)COCCOCCO)CC1 c1(CC(=O)N(CCC(C(C)C)NC(C2(C)CC(=C)C2)=O)C)cc(C)cc(F)c1 c1(C(N2CCCC2Cc2ccc(Br)cc2)=O)noc2ncccc12 c1(NC(c2cn(CC)nc2)=O)cc(-c2ccc(SC)cn2)cnc1OC c1(C(=O)NCC2C(NC(c3c(CC)cccn3)=O)COC2)cc(Cl)c(O)cc1C c1(C(N2CC(CNC(CCC(=C)Br)=O)C2)=O)ccc2c(c1)C(=O)NC2=O C1(C(=O)O)C2CC3C(C2NCc2c(N)cccc2Cl)C13 CC(C)CCCC(C)C(=O)NC1CN(C(C2CCc3nccn3C2)=O)CC1CO C1(CNC(C2(CN(C)C)CC2)=O)CC(O)CN1C(=O)CCC1CCCOC1 c1(C(N2CC3C(CNC(=O)CCc4ccccc4)(C3)C2)=O)nnn2ccccc12 c1(CC)sc(C(=O)NCC2CCCN(C(C3CC3F)=O)C2)cc1Br Cc1cc(Cl)ccc1CC(=O)NCCC1CN(C(=O)C=CC2CCCC2)CC1C C=CC1CCN1C(=O)CC1(C)CCN1C(c1conc1CC)=O S(=O)(=O)(c1cn(C)cn1)NCC(=O)NCC1N(C(C(C(C)O)N(C)C)=O)CC=C1 c1(OCCC)cccc(CNC(c2ccc(-n3cnnn3)cc2)=O)c1 C(=O)(C(CSC)OC)NC1C(C(N(CCCO)CC#C)=O)C1 N1(C(=O)C2=CCCOCC2)CC2(C1)CN(C(C13CCC(CC1O)C3)=O)CCO2 C(=O)(C1CSc2ccccc21)NCC1(OC)CN(C(=O)CNS(C)(=O)=O)C1 Cc1cncc(C(=O)NC(C)CCCNC(=O)C(O)CC2CC2)c1C N1(C(C2(CC)CC2)=O)CCC2(CC1)CN(C(C13CCCC1COC3)=O)C2 C1(COC)CC(CNC(c2cnn(C)c2SC)=O)N(C(c2cn(C)cc2C)=O)C1 C1(F)(CNC(c2csc(-c3nc[nH]n3)n2)=O)CCN(C(=O)C(O)C2CC2)C1 N1(C(C(C=CC)O)=O)CCCC(CNC(c2cc(C)on2)=O)CC1 O=C(C1=Cc2cc(F)ccc2OC1)Nc1ccc2c(c1)CC(O)C2 C1(NC(C(CSC)O)=O)CN(C(=O)C(C)(C)CCSC)CC1S(C)(=O)=O CC(C)C(C(=O)N1CCC1c1cccc(C(F)(F)F)c1)N(C(C1CCC1)=O)C1CC1 c1(CC)cccc(C(N2CCOC(CN(C)C(c3cnc(C)o3)=O)C2)=O)c1 N1(C(c2c(CC(=O)OC)scc2)=O)CC(CNC(=O)C2=CCOCC2)CCC1C N1(C(C(C)CN(C)C)=O)CC(Nc2cc(C(N)=O)ncn2)CC(F)C1 C1(CC(=O)NC(CNC(=O)CC(C)n2ccc(C)n2)C2CC2)(OC)CCCCC1 C(=O)(CCC(C)(C)C(=O)NC1CCC1CNC(c1cc(C2CC2)nn1C)=O)OC N1(CCC(=O)N(CCCCCNC(c2coc(Cl)c2)=O)C)CCP(C)(=O)CC1 C1(C(N2CC(NC(C)=O)C2)=O)N(C(=O)CC2CC3(CC3)CO2)CC12CCCC2 C(=O)(C(CC1CC1)CC)N(C)Cc1cc(C(=O)NCC2CC2c2ccccc2)[nH]c1 C1(CCC)(C(=O)NC(COC)C2(C)CC2)CCN(C(=O)CCC2CCCOC2)C1 C1(CC)CC(N=c2nc(N3CCC(CC(F)F)C3)c3ncn(C)c3[nH]2)C1 C(C(=O)NCCC1CCCCO1)(C(C)(C)C)NC(C1C(C)CC1)=O CC(O)(C(=O)N1CC2CC1C2C(N1CCN(NC(=O)C2CC2)CC1)=O)C(F)(F)F c1(C(N2CC(NC(C(CC)COC)=O)C(C(F)F)C2)=O)cc(Cl)cc2c1OCC2 C1(C(=O)NCc2ncc(C)s2)CN(C(=O)CNc2ncccn2)CC1(F)F C1(C(=O)NC2CC(C)(NC(c3cnc(N)c(Cl)c3)=O)C2)CC12CCN(C(N)=O)CC2 C(=O)(C1CCCn2ccnc21)N1C2CCC(NC(CCCSC)=O)(C2)C1 CC(=O)C(C(C)C)(c1ccccc1)NC(=O)CNC1CC1 N1(C(c2c(C)noc2)=O)CCC(CO)(NC(c2cc(C#N)cs2)=O)CC1 c1(OCCCOC)ccc(C(C)(C)C)cc1.C(=O)(C(C)N(C1CC1)C)OC C(CCCC(CO)NC(=O)Cc1sccc1Cl)NC(C(CC)N(C)C)=O N1(C(c2n(C=C)ncc2)=O)Cc2nccn2CC(NC(=O)Cc2cn(C)nn2)C1 O=C(C(CO)C(F)(F)F)N1CCCC(C(N2CC(F)(F)CCC2C)=O)C1 c1(SC(F)(F)F)ccc(-c2csc(-c3csc(-c4cccnc4)n3)n2)cc1Cl c1(C(=O)NC(C(=O)N(CC(F)C2CCC2)CCO)c2ccoc2)cc(CO)no1 N1(S(CC(C)c2ccc(F)cc2)(=O)=O)Cc2ccccc2OCC1(C)C c1(OC)ccc2c(c1)OCC(CN1CCN(C(c3nnn(C)c3C)=O)CC1)=C2 C1(CNC(c2cn(C)nn2)=O)CC(C)(C)CCC1NC(c1cnc(C2CC2)s1)=O C1(O)(CNC(=O)C=CCO)CCN(C(C2C=CCC2)=O)C1 C(=O)(CN1C(=O)Cc2ccccc21)NCC1OCCN(C(CCS(C)(=O)=O)=O)C1 c1(C(N(C(=O)CNCC(C)C)CC)C)ccncc1.n1(CC(=O)C(=O)C)nccc1C c1(OC)ccc(I)cc1C(N1CC2C(C1)N2c1ncc(-c2ccccc2)cn1)=O CC1CC(CNC(=O)C(N2CCCCC2)C)CN1C(c1nocc1C(C)(C)C)=O CCC(C)C(C(=O)N1CCCCC1CNC(=O)CC1CC2CCC1O2)OC Cc1cnc2n1CCC(C(=O)NCCCCN(C(=O)CC1COC(C)(C)C1)C)C2 c1(OC)cc2c(C(=O)OCCC(=O)OCC3(NC4CC4)CC3)c[nH]c2cc1Cl c1(NC(C)=O)ccc(C)c(C(=O)NC2CCCN(C(=O)Cc3csc(C)n3)C2)c1 C1(C(=O)NCC23CC(NC(CSc4c(C)n(C)nc4)=O)(C2)C3)Cc2nncn2C1 CCCCCC(=O)NC(C1CCCN(C(=O)Cn2nc(C3CC3)cc2N)C1)C CCCC(CC)C(=O)NCCC(C)NC(C1CCN(CC(C)C)CC1)=O c1(CNCCC(C)(C)NC(=O)OC(C)(C)C)cn(CC(F)(F)F)c(=O)nc1O c1(-c2n(CC(=O)N(C(c3ccccc3)C)C3CC3)c(=O)on2)cc(Cl)ccc1Cl c1(C(N(CC(O)CNC(=O)C(c2ccccc2)F)C)=O)nnn(C)c1N N1(C(C2C=CC(NC(C3CN(C)C3)=O)C2)=O)Cc2ccncc2C1 CC1(C)CCCOC1C(=O)NC(CCC1CC1)C(=O)NCCc1cnn[nH]1 C#Cc1cc(C(=O)NC2CCN(C(c3cnn(C(C)(C)C)c3C)=O)C2)cc(F)c1 N1(C(C2C(C)CC(=O)CC2)=O)CCCN(C(=O)CCCn2ccnc2)CC1C C(=O)(C(C(C)C)NC(=O)CC12CCCC1C2)N(CC)CC1CC1 Cc1ccc(S(=O)(=O)N2CCCN(Cc3ccc(N(C)C)nc3)C(C)C2)c(C)c1 C=C(C)C(CC(=O)N1CCCC(N(C(=O)CCn2cnc(=N)[nH]2)CC)C1)OCC N1(C(C(CO)NC(CC2CC(=O)NC2=O)=O)=O)CCn2ccnc2C1 Cc1nc(NCC(C)N(C)C(c2sc(F)cc2C)=O)c2cnn(C)c2n1 c1(OCCC#C)ccc(C(=O)NC2CCCC2NC(=O)C(C)C2(O)CCC2)cc1 c1(CC(=O)N(CCCN(C(C=CSC)=O)C)C)ccnc(O)c1 NS(=O)(=O)c1sc(NC(=O)Cc2cccc(F)c2)nc1SCC(=O)NCCCO N1(C(C(C=C=C)C)=O)CC(C(=O)N(C2COC2)C)C2(CC2)C1 C1(F)(NC(CCSCCC)=O)CC(NC(=O)C(C)OC2CCOC2)C1 n1(CC)cc(C(=O)NC2COCC2NC(=O)CC2COC(=O)C2)c(C(C)(C)C)n1 Cc1cc(F)c(C(=O)NCC2C3CC2N(C(C2CC4(CCC4)CO2)=O)C3)cc1F C1(C(N2CC(C)(CCO)C2)=O)(SC)CN(C(C2CC(C)=NO2)=O)C1 c1(CN2CCC(F)(C(=O)Nc3ccc(I)nc3)C2)ncn2ccccc12 c1(CN2CC3CN(C(c4cccc(Cl)c4)=O)CC32)cc2cccnc2s1 C1(C)(C(N(CC(C)NC(c2cccc(C(C)C)c2N)=O)C)=O)CC(C2CC2)=NO1 c1(C(N2CCCC(N(CCO)C(C3CC3F)=O)C2)=O)nccc(Cl)c1F Cc1cccn(C(=O)N2CC(S(C)(=O)=O)C2)c1=NC1CCC2(COC(C)(C)C2)C1 CC1CN(C(=O)CCS(C)(=O)=O)C(C)CN1C(=O)CCn1ccnn1 CC1CN(C(=O)Cn2ccc(C(N)=O)n2)CC1CNC(=O)COC(F)F N1(C(C(c2cccc(Cl)c2)C)=O)CCC(CO)(NC(c2csc(Cl)c2)=O)C1 c1(C(N2CCC(NCC3CCN(C(CC(C)C)=O)CC3)C2)=O)cc(=O)n(C)cn1 N1(C(C2C(C)(C(F)(F)F)C2)=O)CCC(NC(=O)CC23CC(C2)C3)C1C(C)(C)C n1(COCC)nc(C)c(CC(=O)NCC2(F)CCN(C(=O)C3=NOCC3)C2)c1C c1(C(=O)NCC(CC)NC(=O)Cc2scnc2C)ccc(O)cc1[N+](=O)[O-] N1(C(CCc2scc(C)n2)=O)CCN(C(c2cnc[nH]2)=O)C(C(C)(C)C)C1 N1(C(C(c2ccoc2)NC(c2cnc(C)nc2)=O)=O)CC2CC1C1CC21 Cc1nn(C)c2c(NCC3CCCCC3)nc(=NCCn3cnccc3=O)[nH]c12 c1(CN(CCNC(CCc2cc(C)no2)=O)CCN(C)C)c(C)n[nH]c1C C12(C(=O)NC3CCN(CC)C3)CC1CCN2C(c1cccc(CO)c1)=O N1(CC#N)CCCC12CCN(C(c1ccc(-n3cncn3)nc1)=O)CC2 C(=O)(C1=Cc2ccccc2OC1C(F)F)NCC(C1CCC1)NC(C(C)(C)F)=O N1(C(C(=O)N2CCC2CC(=O)N2CCC2)=O)CCOC(c2cccnc2)C1 N1(C(C(CC)F)=O)CC23CCCC2(C1)CN(C(=O)CC1CC1)C3 C1(CC=C)(NC(=O)C(C)CNS(=O)(=O)CC)CN(C(=O)C(C2CCC2)OC)C1 c1(C(=O)N(C2CC3C(C2)C3(F)F)CCO)ccc2nc(O)oc2c1 C1(C(=O)NC(C)CN(C)C)(CC)CCCN1C(=O)CC(Cl)Cl CCC(C)C(O)C(C)C(=O)N(CCN(C(=O)CC(CN(C)C)CC)C)C(C)C CC1CN(C(=O)COCCc2ccccc2)CC1CNC(c1cnccc1Cl)=O N1(C(C=C(C)Cl)=O)CC2(CCN2C(=O)C(C)(C)C(F)c2ccccc2)C1 N1(C(CNC(C)=O)=O)CCC2CN(C(C3(NC(C)C)CC3)=O)CCC2C1 C1(CNC(CCCn2ncc(C)c2)=O)CC2CCC1N(C(=O)COCC(C)C)C2 CC(C#N)C(=O)NC1(C(=O)NCC(F)Br)CCSC1 C1(C(N(CC(COCC)O)C)=O)N(C(=O)CC2C(=O)NN=C2C)CCC1(C)C c1(C(N(C2CCC(NC(c3ccc(CC)nc3)=O)C2)C)=O)cc(C)ccc1F Cc1cnc(N2CCOC(C(=O)Nc3cc(O)nn3C)C2)nc1 c1(C(=O)NC2CCCN(C(=O)CCNc3ccccn3)CC2)cc2ccsc2s1 C1(C(N2CC(C(C(=O)NC3CC(C)CC3(C)C)O)C2)=O)CCC2(CCC2)CC1 C1(O)(CNC(c2ccc(C#C)nc2)=O)CCCN(C(=O)CCC(C)N(C)C)CC1 N1(C(c2c(C)cncn2)=O)CC(CNC(=O)Cn2nnnc2C)CC(C)C1 c1(OC)nnc(Cl)cc1NC(=O)C(C1CCN(C(C2(C)CCOCC2)=O)CC1)C C1(NC(CCOC)=O)CN(C(c2ccc(CO)nc2)=O)C(C)(C)C1 C(=O)(C1=C(Cl)CCOC1)NCC1C(NC(C(C)(C)OC)=O)CC1 c1(NC(C)=O)cccc(C(N2CCC(F)(C(=O)Nc3nn[nH]n3)C2)=O)c1 N1(C(CSCC2CC2)=O)CC2(C1)C(NC(c1ccc(C(F)F)o1)=O)CCS2(=O)=O Cc1ccc(C(O)C(N2CCC(O)(CCNC(c3csc(Cl)n3)=O)C2)=O)cc1 C=C(C)CCCC(=O)NCCC(O)CNC(C1CC(C(=O)OC)C1)=O CC(N=c1cc2c(n[nH]1)ncn2C)C(O)c1cc(F)cc(F)c1 N1(C(c2ccn(C)c2)=O)CCCC1(C)C(=O)NC1CCCC(CO)C1 C(C(C(=O)N(CC(C1(O)CCCC1)C)C)NC(=O)CSC1CCC1)SCC c1(C(=O)NC2C(CNC(C3C(OCC)C3)=O)CC2)cccnc1-n1cnnn1 n1(CC(=O)NC(C)CCN(C(=O)CC(C)(C)O)C)ccc2ccc(F)cc12 C1(COC)(NC(=O)C=Cc2ccccc2C)CCCN(C(C2(C)COC2)=O)C1 CC1(C)CC(NC(=O)Cc2cnc[nH]2)CN1C(C1CCOC(=O)CC1)=O C(=O)(CC(F)(F)C(F)(F)F)NC1C2CN(C(c3c(CC)nccc3)=O)C1C(O)C2 C1(CNC(C2C(C(=O)OC)CC2)=O)CC(F)CN1C(=O)CC(C)(C)O C#CCCCCC(=O)N1CCCC(F)(CNC(=O)Cc2cn(C)nn2)C1 c1(SCCC(=O)NCCCCCNC(C2CCNC2=O)=O)cccc(F)c1 CCC(CC)(C(N)=O)NC(c1[nH]ccc1CNC(C1CCCC(C)CC1)=O)=O C1(F)(C(=O)NCC(CCOC)NC(c2ccc(C#N)s2)=O)CCS(=O)(=O)C1 C1(CNC(CC2(OC)CC2)=O)CN(C(c2nnc(C)cc2O)=O)CCC1(C)C C12(CC(=O)N(C3(C(=O)OC)CC3)C)CCC1CN(C(C1(C)COC1)=O)C2 N1(C(CCCOCC)=O)Cc2ccccc2CC1CNC(=O)CC(C)C(F)(F)F N1(C(CN(S(CC)(=O)=O)C)=O)CCC(C2CC(NC(=O)CO)CCO2)CC1 C1(NC(C2CC2C(=O)CCO)=O)CCCC12CCN(C(=O)Cn1cnnc1)CC2 c1(C(=O)N=c2cc(Cl)[nH][nH]2)cnc2n1CCN(C(=O)C=Cc1ccc(Cl)cc1)C2 N1(C(C(C)CF)=O)C2CCC1CC(NC(c1ccc(N3CCC3)nc1)=O)C2 CC1CN(C)CC(C(=O)N(CCCn2cc(C3(n4nccn4)CC3)nn2)C2CC2)O1 CCCCN=C(NCCOC(F)F)NC1CC2CCCCN2C1 C1(CNC(c2n(CC)ccc2)=O)CC2CCC(C1)N2C(=O)C(C)NC(=O)C1CC1 C=CCC(CC(F)F)C(=O)NCC(CCCC)NC(c1cccnn1)=O C(C)(N=c1nc2scnc2c(NC2CC(=O)NC(C)C2)[nH]1)c1cn(C(C)C)nc1 CN1CCC(C)(C(N2CCC(NC(C3(Cl)CC3(F)F)=O)C(O)C2)=O)CC1 C(=O)(CCC(C)CN(C)C)N(C(C)C(=O)NCc1n[nH]cc1C)CC C1(CNC(C(C2CC(C)(C)C2)OC)=O)CCCN(C(=O)Cn2ncn(C)c2=O)C1 c12coc(c1)NC2=O.C(=O)(CCNC(=O)COC)NCC1C(C(=O)OCC)C1 CCCC(=O)NNC(=O)N1CCC(C(=O)OCc2ccc(C)c(C)c2)C1 c1(C(=O)NCC(CCNC(CCCCOC)=O)(C)C)ccc(Cl)c([N+](=O)[O-])c1 c1(CC(N2C(CNC(=O)CCCC3CC3)C=CC2)=O)cnccc1Cl OC12CCCCC1CN(Cc1sccc1Cl)CC2 CC(C(=O)N1CCOc2cc(Br)cnc21)C1OCCc2sccc21 C(C)(c1ccc(OC)cc1)=CC(=O)NCC1CN(C(C(CC#C)C)=O)C1 Nc1c(C(=O)NC2CC(NC(=O)CCNC(c3ccc[nH]3)=O)C2)cc(F)cc1Cl c1(C(=O)NC(CNC(CCc2n(C)ccn2)=O)CO)cc(OC(F)F)n(C)n1 c1(C(N2CC(NC(CCC=C(C)C)=O)CC3(C2)CC3)=O)cccc(P(C)(C)=O)c1 Cc1c(Cl)ccc(C(N2CCSC(C(=O)NC3CCC(F)(F)C3)C2)=O)c1Cl c1(CNC(C(N2CC(C)C(N)C(C)C2)=O)=O)cnc(O)c2ccccc12 Cc1[nH]nc2ncc(C(=O)NCC(C3CC3)NC(=O)C3=NOC(C)C3)cc12 C(CO)(C(C)(C)c1cccc(F)c1)NC(=O)NC(C)Cc1ccnn1C C(=O)(C1=CCCC1C)NC(CCSC)C(=O)NOCC1CCOCC1 C1(NC(c2cnc[nH]2)=O)CN(C(c2cccc(F)c2Br)=O)CC1C1CC1 N1(C(c2ccc(F)c(C)c2F)=O)CCC2(CC1)CC(NC(c1nc[nH]n1)=O)CO2 N1(C(c2cc(OC)ns2)=O)CCCC(C2(NC(c3ccco3)=O)CC2)C1 N1(C(c2c(C(C)C)ncs2)=O)CCC(C2(O)CCN(C(=O)C=CC3CC3)C2)CC1 N1(C(COCC=C)=O)CC=CCC1C(=O)NCCC(C)C(C)C CCCCS(=O)(=O)c1ccc(C(=O)NC2CC(NC(=O)CC(C)SC)C2)cc1 c1(OC)ccc(OC)c(CNC2CC2C(=O)Nc2ncc(Br)s2)c1F c1(C(=O)NC2CCC(NC(C(CCC)OCC)=O)C2)scc2c1CCCC2 C1(NC(c2cccc(OC)n2)=O)Cc2ccccc2C1NC(c1cc(C)ns1)=O c1(C(=O)NCC(CNC(C2(C)CNC(=O)N2)=O)O)nccc(Cl)c1Cl CCCCS(=O)(=O)CC(=O)NCC1(O)CN(C(c2cc(O)cc(=O)o2)=O)C1 CC(C)CCCC(C)C(=O)N(C(CC(C)C)C(=O)N1CC2CC1C2)C C1(NC(c2nc(C)c(C)n2C)c2n(C(CC)C)nnn2)CCC12CCCC2 C1(C(=O)NC(C=C)CC)CCC2(CC2)N1C(C1CC(=O)C1)=O C1(C)(C(N(CCCCN(C(c2nc(C)n(C)n2)=O)C)C)=O)CC2C=CC1C2 N1(C(C(C)n2cccc2)=O)CCOC(C(N2CCOC(CCF)C2)=O)C1 CC(C)(CCF)NC(=O)Cn1cc(CNC(=O)CC2CCCC2O)nn1 Cc1ccc(C(=O)NCC=CCNC(c2cn(C3CC3)cn2)=O)c(F)c1F C(=O)(CC1OCc2ccccc21)NCC(CC(C)C)NC(=O)CC(C)C1CC1 C1(C(=O)NC(C#C)CC2CCOC2)CCCN(c2cccc(F)c2)C1=O C1(C(=O)NCCSC)CC2C(C1)C2(F)F.C(=O)(CC1=CCCC1)N C1(C(=O)NCCC(C)NC(c2cccc(F)c2C(F)F)=O)OC2CCC1CC2 c1(C(N(CCCNC(=O)CC2CCC(F)(F)CO2)C)=O)c[nH]c2cccc(F)c12 C(=O)(CC1C(=O)N(C)c2ccccc21)N1CC(OC)(CNC(C2CC2C)=O)C1 Cc1cc(CNC(=O)CCn2ccnc2)oc1C(N1CC(C)(C)C1C1CC1)=O N1(C(CN(CCC#C)C)=O)CCC2(CCCCC2NC(C2CCCSC2)=O)CC1 c1(C(N2C(CN(C(=O)CCC3CCC3)C)CCC2)=O)cc2c(s1)COCC2 Cc1cc(C(=O)N(C)CCOCCN(C)C(c2[nH]nc(C(F)F)c2C)=O)ncn1 CC(O)(C(=O)N1CC2C(NCc3cnc[nH]3)C2C1)C(F)(F)F c1(C(=O)NCC2C=CCN2C(=O)Cc2cnc[nH]2)ccc2nccn2n1 C12(CC(=O)NC3CC(NC(C4C(C(=O)OC)CS4)=O)C3)CCCN1CCC2 CC1(C)CN(C(=O)CSCCC#N)CC1C(N1CCC(CCCO)CC1)=O c1(N2CCC(OC)C(F)C2)nc(N(CCCS(C)(=O)=O)C)nc2ccsc12 C(C1=CCN(C(=O)CC2(O)CCCC2)CC1)NC(c1ncoc1-c1ccon1)=O C#CCC(O)C(=O)NCC(C)NC(c1ccc(NC(N2CCCC2)=O)cc1)=O c1(C(=O)NC23CC2CN(C(C2CCCC2C2CC2)=O)C3)cc2c(cc1Cl)NCC2 c1(OC)c(C(N2CCNC(C(=O)Nc3cnccc3C)C2)=O)cccc1C c1(C(=O)NCC(C)NC(C2CCC(=O)CC2C)=O)cc(Cl)cc([N+](=O)[O-])c1O C1(CNC(c2cc[nH]n2)=O)CCN(C(=O)CC2(O)CCOC2)C12CC2 C1(CC=C)(NC(c2cc(C)ns2)=O)CCCN(C(c2cc(SC)c(C)o2)=O)C1 C1(NC(C2CCC(C)O2)=O)C2CC1CN(C(=O)Cc1ccc(F)cn1)C2 C(CC(C)C(=O)NCCOC1CN(C(c2nc(C(C)C)oc2C)=O)C1)OC C(CC(C)C)(C(=O)NCc1ccc(C(=O)NC2CCN(OC)CC2)cc1)OC CC1OC2CCC1(NC(C1CC(F)(F)CN1C(c1cnnn1C)=O)=O)C2 C1(C)(CC)C=C(C(=O)NCC(C)(C2CCC2)NC(c2cccnc2S)=O)C1 c1(OC)ccc(CC(=O)NC2CC(C)CN(C(c3cncc(C)n3)=O)C2)c(F)c1 N1(C(COCC)=O)CCC12CN(C(c1cccc(C(C)C)c1)=O)C2 c1(C(N2CCCN(C(C3(OC)CC3)=O)CC2C)=O)ccc([N+](=O)[O-])cc1N N1(Cc2cc(C(=O)O)on2)CC2(CC(NC(=O)CCCc3ccccn3)CO2)C1 c1(OC)cc(F)cc(C(=O)NC(C)CCNC(C2CCCOCC2)=O)c1N CC(N=c1[nH]c2c(c(=NCc3cccc(OC(F)F)n3)[nH]1)SCC2)c1csnn1 N1(C(C2COC(=O)O2)=O)CCC2CN(C(c3cnn4c3OCC4)=O)CC12 C1(O)(C(=O)NCCCCNC(c2cnc(NC3CC3)s2)=O)CCOCC1 C1(C(=O)NC(CNC(C2N(CCC)CCC2)=O)C(C)C)CCCN1N=O c1(COC)nc(NCc2cccc(Br)c2F)cc(N2CCCC(NC(C)=O)C2)n1 C1(CCC(=O)NC2CC(CNC(C3N(NS(C)(=O)=O)CC3)=O)C2)CCC(=O)N1 N1(C(C2CC(CC)C2)=O)C2CCCC1CN(C(=O)CC1CSCCO1)C2 N1(C(CNC(CCC)=O)=O)CC(O)(C2CCCN2C(c2cc(COC)on2)=O)C1 N1(C(c2cnco2)=O)CC(NC(C23CCC2C3)=O)C2(CCC2)C1 c1(CC(N2CC(c3ccc(Br)cc3)(C)C2)=O)cncnc1N C(=O)(C(C)(C)C(O)c1cc(Cl)cc(Cl)c1)NC(C(=O)OC)C(=O)OC Cc1oc(-c2ccccc2)nc1CNC(=O)NNC(=O)c1sccc1Cl C(CCC(O)CC)N(C(C(=O)Nc1ncc(C(=O)OCC)s1)=O)CCO c1(CCC(N2CCCC(OC3CC3)C2)=O)ccccc1F Cc1ccc(C(=O)NCC2CN(C(C3(N(C)C)CCC3)=O)CCC2C)c(C)c1 c1(CC(N2CC(CN(C(C(C=CCCC)O)=O)C)OCC2)=O)ccnc(Cl)c1F N1(C(CCC#CC)=O)CCN(C(=O)COCc2ccccc2)C(CC(=O)NC)C1 Cc1cc(C(=O)NCCCN(C)C(c2cnn(CC(F)(F)F)c2)=O)c(C)o1 c1(C(=O)NCC2(COC)N(C(CC=CCC)=O)CCC2)ccc(Cl)c(CC)c1 CCC(O)(CN(C)C(C1(F)CCN(C(=O)CCC2CCCOC2)C1)=O)CC C(CCCC(=O)N1CCOCC1CNC(C1CC1(F)F)=O)OC Cc1cc(Cl)cc(N)c1C(N1CC(NC(=O)COc2ccc(F)cc2)C(C)C1)=O Cc1cnc(NCC2CC(F)(F)C2)c(S(=O)(=O)NC(c2ccccc2C)C)c1 CCC(C)CC(C)CC(C)C(=O)Nc1ccc(C(=O)O)cc1C N1(C(Cc2n(C)cnc2)=O)CCC(C(=O)NC(CO)CCO)C1(C)C N1(C(C)=O)CCCC12CCN(C(C1CCc3cc(O)ccc3C1)=O)C2 CCCCC(F)C(=O)N(N1CCN(C(=O)C(C)(CC)OC)CC1)CC1CC1C1CC1 c1(C(C)=O)cc(NCC(C)N(C(=O)CCCCC(F)(F)F)C)ncc1[N+](=O)[O-] Cc1oc(C#N)cc1C(=O)NC1CC=CCC1NC(=O)CC=C(Cl)Cl N1(C(COCCC)=O)CCC(C2CCN(C(C34COC(CF)(C3)C4)=O)CC2)CC1 Cc1c(Cl)sc(Cl)c1C(=O)NC1CCN(C(c2ccc(N)c(F)c2)=O)CC1C c1(CC(N2CC(NC(C(CC)OC)=O)C2)=O)c(F)cc(Br)cc1F c1(CC)c(C(=O)NC(C2CCOC2)CNC(c2c(C)ncn2O)=O)csc1C C1(CNC(C=CCC)=O)CN(C(c2cccnc2S)=O)CC2CC12 C1(NC(c2cc(COC)on2)=O)CCN(C(=O)Cn2cc(N)cn2)C(C)C1 CC1CC(CCNC(=O)COC2(C)CCC2)CCN1C(=O)Cc1cccc(O)c1 N1(C(CC(CC)(C)C)=O)CCC2(CC1)CC(N=c1[nH]cnc3cnccc13)O2 n1(CC)cc(C#N)c(=NC(=O)C2CN(c3ncc4cccnc4n3)CCO2)[nH]1 Cc1cc(Cl)c(C(=O)NCCC2CN(C(c3cnn(C(F)F)c3)=O)CCO2)cn1 C=CC(C(F)(F)F)NC(=O)NCC(CC(C)C)OCC c1(C(N2C(CNC(CC(C)O)=O)CC(O)C2)=O)cnc(O)c2c1NCCC2 C1(O)(c2cccc(C(F)(F)F)n2)CCN(CCCn2ncnn2)CC1 Cc1cc(C(=O)NC(C)Cc2cn[nH]c2)cc2c[nH]nc12 c1(C(=O)NC2CC(CCNC(C(C)OC(C)(C)C)=O)C2)cccc(Br)c1F CCCCCC(O)C(=O)NC(CC(=O)N1CCN(C(=O)NC)CC1)C(C)CC c1(CC2CCC(CNC(c3nnnn3C)(COC(C)C)C)C2)c(F)cccc1F c1(CCC(=O)NCC2CCCN2C(C2CCCO2)=O)nc(-c2ccccc2)no1 N1(C(CN(C(=O)CC2CCC(=O)C2)CCOC)=O)CCC(C)(CCO)C1 Cc1ccc(C(=O)NC(C(=O)NC2CCCC3(C2)N=N3)C(C)C)nc1C C1(C(N(CC(O)CN(c2nc[nH]c3ncnc2-3)C)C)=O)CCCC12CCOCC2 C1(=O)CCOCCN1C1CC1.CC(CN(C)C(=O)N(C)C)O.C1(C(=O)N)CCC1 c1(C(=O)NC2CCCC(CN(C(CSCCOC)=O)C)C2)c(C)ncn1OC C=CCCCCC(=O)NC1CCCC1CC(=O)NC(CC)(CC)CCO N1(CC(=O)NCC(C)C)CCC(C)(NC(=O)C(C)c2ccco2)CC1 Cc1cc(C)n2cnc(C(=O)NCCOC3CCN(C(C4CCC(=O)N4)=O)C3)c2n1 c1(C(=O)NCC(CNC(c2nc(OC)oc2)=O)(C)F)nnc(O)nc1O CC1COCCC1N(C)C(C1CC(CNC(=O)CCOCC(C)(C)C)C1)=O N1(C(C=CCN(C)C(C2CC3CC3C2)=O)=O)CC2CCC1C(O)C2O C(CCCCC(=O)NCCN(C(=O)Cc1nc(C2CC2)n[nH]1)C)=CC C1(C(=O)NC(CC=C)CNC(=O)Cc2ccoc2C)CN(C)C(=O)CCO1 C1(NC(=O)NCCC)CN(C(=O)Nc2cccc(CSC)c2C)CC12CCC2 Cn1nc2c(c1C(=O)NCC13CCC(C1)N(C(C1CCC(=O)O1)=O)C3)COCC2 C(=O)(C(CNC(c1cnnn1C1CC1)=O)CC(C)C)NC(CC#CC)C c1(C(=O)NCCN2CCCN(C(C(CC)C(C)C)=O)CC2)ncnc2sccc12 C(=O)(C1CN(C(C2CCC2(F)F)=O)c2ccccc21)OC C(=O)(C1Cc2c(Cl)cccc21)NCC(CNC(c1ccnnc1)=O)C(F)(F)F C(=O)(C(C)(CO)NC(C1CC2(CC2)CO1)=O)NC(CC)Cn1cncn1 C=C(C)CC(C(=O)N1CCC(O)C1)NC(=O)C(=O)C(C)CC c1(NCC2(OCC)CCC2)nc(C)cc(=NC(C)CS(=O)(=O)CC)[nH]1 N(C1COc2cc(F)c(Br)cc21)CC(C1CCC2(CC1)OCCO2)=O N1(C(=O)OCc2ccccc2)CCCC(OCCc2coc(C3CCC3)n2)C1 N1(C(C2CC2Br)=O)CCCC2(C1)CN(C(=O)C(O)CC1CC1)C2 C1(NC(c2c(C)nc(C)[nH]2)=O)CC2CCC(C1)N2C(c1ccc(Cl)c(Cl)c1N)=O c1(C(=O)NCC2CC(NC(C=CC(C)C)=O)CC2O)noc2cc(F)ccc12 CN1CCN2C(C1)C2=O.c1(C(C(=O)NC2CSC2)=O)cnn(C)c1 C(=O)(CC(CC(C)C)NC(c1cncc(O)c1)=O)N1CCC(C(=O)OC)C1C N1(C(C=CC(=O)NC(c2cccnc2)CO)=O)CCC2CCCC12 C(N=c1[nH]cnc2c(F)cccc12)c1ccc(CNC(C2CCCS2)=O)cc1 N1(CCNC(C(COC)NC(=O)CCN(C)C)=O)CCCNC1=O c1(C(C)=O)ccc(N(C)C)nc1.c12n[nH]cc1C(=O)NCC(F)CNC2=O C1(NC(c2ccc(COC)s2)=O)CC2CCC1CC2NC(c1cc(C)co1)=O N1(C(c2nnn(C(C)(C)C)n2)=O)CCCN(CCNC(C2CC2(Cl)Cl)=O)CC1 C(CC(C(=O)N1CC(CC)C(O)C1)NC(c1nc[nH]n1)=O)=CC c1(SCc2nc(C(CC(N)=O)NC(C3CNC3)=O)on2)cc(F)c(F)c(F)c1 N1(C(C=C(C)Cl)=O)CC(NC(c2cnc(N(C)C)nc2)=O)C(C)C1 N1(C(C(CC)n2cccn2)=O)CCSCC1CCNC(C1(C)CC(F)(F)C1)=O C(=O)(CCCC(N)=O)N(C)CC1CN(C(=O)C=Cc2cccnc2)CCO1 C1(CC(=O)N(CC(=O)N(C(c2cccs2)=O)CC)CC)CCOC1C N1(CCN(CC(=O)N(c2ccccc2)C2CC2)C)CCC(C)(O)C1.C(C)(C)(C)O C1(C2CC2)(C(N2CCN(C(CC(C=C)C)=O)CC2COC)=O)CCOCC1 C1(OC(=O)NC2CC3(C(C(=O)OC)C3)C2)COCCN(C(=O)CC(C)C)C1 CC(C)CC(CNC(=O)COC(C)C)NC(c1cncc(I)c1)=O Cc1ccc(=NCCC(=O)N2CCC(CCNC(c3nc(O)sc3C)=O)C2)[nH]c1 CN1CC(O)(CC(=O)NCCc2ocnc2CNC(C2(N(C)C)CCCC2)=O)C1 C(=O)(C(C(C)C)C(C)C)NC12CC(C(=O)NC(C(=O)OC)CCF)(C1)C2 Cc1c(C(=O)NCCC2CSCCN2C(=O)Cc2cncnc2O)cccc1CO C1(N(C(CCCCC)=O)C)CCC2CN(C(c3coc(C(C)(C)C)n3)=O)CC12 Cc1ccc(C=CC(=O)NC(C)CC(C)NC(c2cnn(C(F)F)c2)=O)nc1 C(=O)(C(C)C(F)(F)F)NCCCN(C(c1cnc(CCCC)s1)=O)CC N1(C(C2CCC(=C)CC2)=O)CCCC(C2CCN(C(=O)CCCOC)C2)C1 c1(N2CCCC(NC(Cc3n(C(C)(C)C)ncc3)=O)C2)ncncc1Cl c1(C(=O)OC)cccc(CNC(=O)C(=O)N(C2CCCCC2C)C)c1S(C)(=O)=O N1(CC(=O)NCCC(C)N(C)C(C2CCC23CCC3)=O)CCOCC1=O C1(C)(CC)CN(C(c2cc(Cl)ccn2)C(=O)NC2CC(F)(F)C2)CCO1 S(=O)(=O)(c1ccccc1Br)NC1C(C#N)CN(C(c2c(F)cccc2Br)=O)C1 C1(CC(=O)NC2(CNC(C3(C#N)CCCC3)=O)CCOC2)CCCS(=O)(=O)C1 Cc1ccc(C(F)(F)C(N2CC(CNC(=O)C(C#N)C3CC3)C(O)C2)=O)cc1 N1(C(CCn2c(C)nc(C)n2)=O)CC2CCC(C1)C(NC(=O)C(C)C(C)(C)C)C2 C1(C(N2CC(C3(NC(c4c(C)c(F)ccc4)=O)CC3)C2)=O)CS(=O)(=O)CC12CC2 c1(CNC(C23CCC(CO2)C3)CNC(Cc2nc(C)sc2)=O)ccc(F)cc1 C1(NC(C2(C#N)CC3CC3C2)=O)CN(C(c2cnsc2)=O)C2(CCOCC2)C1 n1(CC(=O)NC2(C)CCN(C(CCCC)=O)C2)cnc(C)c1C(=O)OC(C)(C)C C(=O)(CC(C)C(F)F)NCC1CCN(Cc2c(C)nn(CCO)c2)C1 N1(C(C=C(C)Cl)=O)C2CCC1CC(NC(c1c(C)nc3sccn13)=O)C2 c1(C(C(N2C(CNC(CC(CC)(F)F)=O)C=CC2)=O)C)ccc(S(N)(=O)=O)cc1 CN1Cc2cccc(NC(c3cccnn3)c3nnnn3CC(F)F)c2C1=O CC1(CC(=O)NCC2(CO)CCC2)CCN(C(=O)CC2CC3CCC2C3)C1 C1(NC(CNC(=O)OCC)=O)(CNC(C2CC=CCO2)=O)CCCC1 S(=O)(=O)(c1cccc(N2CCC2)n1)NCCCCN(C)C C(=O)(C(CC(C)C)OC)NC(CC(C)NC(C(C)=C(CC)C)=O)C Cc1cc(=NC(=O)C2CC2(c2ccc(Br)cc2)NC(=O)CCN2CCOCC2)[nH]o1 CC1CCN(CCC(N2CCOC(CCNC(=O)CCS(C)=O)C2)=O)CC1 c1(CC(N2CCC(CNCc3ccc(C(C)O)cc3)CC2)=O)ccnc(Cl)c1F CC(C)(C(=O)N1CCC(C(F)C(N2CCCC(C3CC3)C2)=O)C1)C(F)(F)F C1(NC(COCC)=O)CC2CN(c3ccnc(SC)n3)CC2C1 c1(CCC(=O)NCCCC(C)NC(C2CCCSC2)=O)n[nH]c2ccccc12 C1(NC(c2c(OC)cccc2)=O)CN(C(c2cc(=N)[nH]c(Cl)n2)=O)CC1C1CC1 N1(C(COCC)=O)CCCC(C)C1CNC(C1(c2cncnc2)CCCC1)=O Cc1c(F)ccc(C(N2CC=CC2C(=O)NCCCN(C)C)=O)c1Cl N1(C(C(C)CC2CCC2)=O)CC2C(NC(c3ccc(OCCF)cn3)=O)C2C1 CCC(C)(C)C(O)C(=O)N1CCC(C(C)NC(=O)CCCC(=O)N(C)C)C1 C(c1cc(OC)c(O)c(OC)c1)=CC(=O)NC(CCCC)CNC(C1CC1C)=O N1(C(c2noc(CC)c2C)=O)CC(CCNC(=O)C=CCF)OC(C)C1 O=C(CC1=NNC(=O)C1)NCC(C1CCN(C(c2ccn(C(F)F)n2)=O)CC1)F C1(CNC(c2ccsn2)=O)CC(F)CN1C(=O)CC(O)Cc1ccccc1 C1(c2cn(C3C(O)CC3)nn2)CCCCN1C1CC1 CC1COCC(CC(=O)NC(C2(O)CCN(C(=O)CN3CC4CC4C3)C2)C)O1 C12(N(C)C(C3CCCC(C#N)C3)=O)CCC(CC1)CC2 c1(C(N2C3CC(NC(C4CN(C(C)=O)C4)=O)C2CC3)=O)ccc2nnn(O)c2c1 C(=O)(CC1=Cc2ccccc2C1)N1C(CNC(C23C(C)OC(C)(C2)C3)=O)CCC1 CC(C)C(C)C(C)CC(=O)NC1(CNC(c2ccn(CC(F)F)n2)=O)CC1 N1(C(Cc2c(C)cco2)=O)CCC(O)C(NC(C2CCCCN2C)=O)C1 C1(CCC)(CO)CCN(CCC(N2CCC(N3CCCCC3=O)CC2)=O)CC1O N1(C(C(CO)N(C)C)=O)CCCC2(NC(c3ccn4nccc4n3)=O)CCCC12 c1(OC)ccc(F)c(C(N2CCC(N(C(=O)CO)C)CC2)=O)c1F c1(C(=O)NC(CNC(CC=CC)=O)(C)CO)cc(COC)ccn1 c1(OCC)ccc(N)c(C(=O)NC(C)(C)CNC(C2CCC(C)S2)=O)c1 C=CCN(OC)C(=O)C1(C)CC(O)CN1C(c1cnn(C)c1C)=O N1(C(c2ccc(C)cc2C)C(=O)NC(CC)C)CCN(C)C(c2ncc[nH]2)C1 N(C1CCNc2cc(F)ccc21)S(=O)(=O)Cc1c(Br)ccc(Cl)c1F C=CC1CN(C(=O)Nc2ccn(C(C)(C)C(=O)OC(C)(C)C)c2)C1 c1(NC(=O)NC(c2cccnc2)CC)ccc(C)c(OCCC(C)C)c1 CN1C(C(=O)NCC2CCC2NC(c2n[nH]cc2[N+](=O)[O-])=O)CCS1(=O)=O CN1Cc2cc(C(=O)NC3CC3CNC(c3cn(C)nc3O)=O)ccc2NC1=O c1(C(N(C2CCCN(C(c3cnc(C)s3)=O)C2)CC)=O)nn2cccnc2c1Cl S(=O)(=O)(C(F)(F)F)NCCC(=O)NCCC(=O)N(C(C)CC1CC1)C c1(C(=O)NCC(C)NC(CS(=O)(=O)NC)=O)nc(C)ccc1C CC(=O)C(C)(C)CC(=O)N(C1CC1)CC1CC1CC(=O)NCC1CC2(CCC2O)C1 Cc1ccc(CN2CCCC(NC(c3[nH]cc(C)c3C)=O)C2)c(Cl)c1 S1(=O)(=O)c2cnc(c(Cl)c2)CN1.c1(C(CC)NCC2(SC)CC2)ccccc1Cl c1(C(=O)NCC(CN(C(C2(C)C(C)CCC2)=O)C)(C)C)cc(O)cnc1Cl c1(C(=O)NC(C(C)C)CNC(c2cncs2)=O)ncncc1N c1(SCC)ccc(Cl)cc1C(N1CCCC(N(C(=O)C(C)(C)C2CC2)C)CC1)=O C1(CNC(c2cc(C)sc2)=O)CCCCC1NC(C1(C(F)(F)F)CCOCC1)=O C1(NC(CCC=CC)=O)CCN(C(=O)COc2cc(C)ccc2Cl)CC1CO N1(C(c2cnc(OC)s2)=O)C2CCC1CC(NC(C1CC13CCC3)=O)C2 C1(NC(C2C(C)(C)C(F)(F)C2)=O)CN(C(=O)C(F)F)CC(C)(C)C1 c1(CC)nc(C)n(C)c1C(=O)NCCN(C(=O)CN1CCC1C)CC1CC1.SCC C#Cc1cc(C(=O)NC(C(=O)NCc2nc(C)no2)C2CCCO2)ccc1C Cn1cnc2[nH]c(C(=O)NC3CN(C(c4ccc(Br)o4)=O)C4(CCC4)C3)cc12 C12(CC(=O)NC3CC(C)N(C(=O)Cn4cc(N)cn4)C3)CCC(CC1)CC2 C(=O)(C1=C(Cl)CCCC1)NC(C(=O)NCC(C)OC(F)F)Cc1cc[nH]n1 C1(SCN(C(C2(SC)CCC2)=O)C)CCCCN1C(C1CCN(C(C)C)CC1)=O C1(C(=O)NC2CC2C(=O)NCC(C)(C)O)(COC)COC1 N1(C(C(c2cccnc2)OC)=O)CC(C)(C)CC1CNC(=O)CC(C)(C)C#N N1(C(CCC=C)=O)CC23CCCCC2(C1)CN(C(c1n[nH]c2c1CCC2C)=O)C3 N1(C(C2C(C(=O)OCC)C2)=O)CCC(C(C)NC(=O)C=Cc2ccsc2)CC1 C(=O)(CS(=O)(=O)C(C)C)N1CCCC(N(C(=O)Cc2coc(C)n2)CC)C1 C(C(C)(C)C(=O)NCCCC(=O)N(C)C)NC(C(CCOC)C)=O c1(C(=O)N(C23CCC(C)(C2)CO3)N2CCC(=O)NC2=O)cc2n(c1)CCSC2 Cc1c(C(=O)NCCC2(O)CCN(C(=O)CN3CCC(C)(C)C3)C2)cnn1C N1(C(=O)CN2CCCCC2)CCN(C(c2cc3[nH]ccc3s2)=O)C2(CC2)C1 C1(C(N2CCC(N(C)C(C3CCC(C)CC3)=O)CC2)=O)CN=C2N=CNN2C1 c1(OCC)ccc(-c2nc(-c3ccc(OC)cn3)oc2NC(=O)CCSC)cc1 N1(C(C2COCCN(C(C3(OC)CC(C)(C)C3)=O)C2)=O)CCC(C2CCCC2)C1 Cc1cc(N2CCOCC2CNC(c2conc2C2CCC2)=O)nc(CO)n1 c1(C(N2CC3C(CC(=O)NC(C#C)C(C)C)C3C2)=O)ncc(C#N)cc1C C1(CCC=C)(C(=O)NCC2C(C)C2C)CN(C(=O)Cc2cc(C)cs2)C1 c1(C(N2CC(C)CC(NC(c3n(C(C)C)ccn3)=O)C2)=O)ccc(C#N)c(F)c1 C1(CNC(C2(C)CC(C)C2)=O)CC2(CCOCC2)CN1c1ccnc(Cl)n1 N1(C(CSCC)=O)CCCC1(C)CNC(=O)C(c1ccccc1)c1ccccc1 Cc1nc(C#N)cc(=NCC(C2CCCC2)NC(c2cn(C)c(=O)n2C)=O)[nH]1 C1(NC(C(C)=CC2CC2)=O)(CNC(C2COC3(CCC3)C2)=O)CCC(F)(F)CC1 C(=O)(CCCCC(=O)NOC(C)(C)C)NC1CCCN(C(CCCC#C)=O)C1 c1(-c2cc(NC(c3cc(C(=O)OC)nn3C)=O)ncc2)cc(C)ccc1C c1(C(=O)NCC(CO)NC(C=Cc2nc(C)c(C)[nH]2)=O)ccc(C#N)cc1O N12CCC1(CC(C(C(C)N(C(C1C=CCCC1)=O)C1CC1)=O)CO)CC2 C#Cc1ccc(C(=O)NC2CCN(C(C3CC(=C(F)F)C3)=O)C(C3CC3)C2)cn1 c1(C(=O)NC(C2(O)CN(C(=O)CC3CCCO3)C2)C)c[nH]nc1C(F)F c1(C(=O)NC2(COC)CN(C(=O)CCCn3ccnn3)C2)cccc(N)c1C N1(C(Cc2cc(C)c(O)cc2)=O)C2CCC1CC(N(C)C(C1(F)CCOC1)=O)C2 c1(OC)ccc(C(=O)NCCC2(C(=O)NC(c3ncc[nH]3)CO)CCC2)s1 c1(C(C)(F)F)ccc(CC(=O)NCC2(NC(=O)COCCF)CCCCC2)cc1 N1(C(C)=O)CCN(C(c2n[nH]cc2C(C)C)=O)CC1CS(C)(=O)=O N1(C(C(CCC)CCCO)=O)CCCC(C2CCN(C(C3CC3F)=O)CC2)CC1 N1(C(c2c(OC)ccs2)=O)CCN(C(=O)CCC(F)(F)F)CC1C(C)(C)C CCC(C)(CNC(c1cc(C)c(C)cn1)=O)C(=O)NCC1(n2nccn2)CC1 c1(C(N2CCC(NC(C(CC=C)C)=O)C(O)C2)=O)nc2ncc(CCO)cn2n1 CN=c1[nH]nc(CC(=O)NCC2(F)CC(NC(=O)C(c3ccc(Cl)cc3)C)C2)s1 Nc1cc(F)c(CC(=O)NCCCNC(C2CCC2c2ccccc2)=O)cc1F CCC(C)(C)CCCC(=O)NC12CC(CNc3nc(Cl)ncc3SC)(C1)OC2C c1(OCC)ccc(C(=O)N(C)CCNC(C2(F)C(C)(C)C2(C)C)=O)cc1C N1(C(CC(C=C)CCC)=O)C2CC=C(C(=O)N3CCOC(CC)C3)C1CC2 Cc1ncc(C=CC(N2CCC(NC(c3cscc3C(F)(F)F)=O)C2)=O)c(O)n1 C12CC(C)(C1)OC2C.C1(NC(CNC(CNC(C)=O)=O)=O)CCC(CNC=O)CC1 C(CC(C)(C)C(=O)NCC1(F)CC(NC(C2(C)CC(O)CN2C)=O)C1)NC(C)=O C12(C(N(C3CCCOC3)CC)=O)CC(C)(CN1C(=O)CCC(=O)NCC#C)C2 C1(NC(C2(F)CCC(C)CC2)=O)CN(C(c2ccc(=O)oc2)=O)CC(C)(C)C1 c1(C(=O)NC(CNC(C2(CC=C)CCOCC2)=O)(C)CC)cc(CC)ccc1Cl C1(CNC(c2ccc(C)s2)=O)CCC(F)(CNC(C2(C#N)CCCO2)=O)CC1 c1(OC)ccc2nc(C)cc(C(=O)NC3CCCC(c4ccc(F)cc4)C3)c2c1 c1(NCC(Cn2c(C)ncc2)C)sccc1S(=O)(=O)N1CCOC(C)C1 N1(C(C2CC(C(=O)OC)C2)=O)CCCC(CO)C1.c1(N)ccccn1.C1(=O)C(C)N1C c1(C(=O)NC2C(NC(CCC)=O)CCCC2)ccc(=O)n2c1CCC2 N1(C(CCc2nnc(C)o2)=O)CC2(CCN(C(C3(O)CCCC3)=O)CC2)C1 CC1CN(C(C2CC(=O)N(c3nccs3)C2)=O)CC1NC(=O)C1=COCC1 CC(C)C#CC(=O)N(C)Cc1ccnc(C(N2CC(SC)C2)=O)n1 CC1CCC(NC(=O)COC2CC2)CN1C(c1cccc(Br)c1Cl)=O Cc1cccc(C(=O)NC2CCCC2CC(N2CC3CC3(CO)C2)=O)c1C c1(C(C)C)nc(C(=O)NCC23CC(NC(=O)CCc4cnc[nH]4)(C2)C3)cs1 C1(CNC(C(C(C)C)C2CCC2)=O)CC2(CCN(c3nccn3C)CC2)CO1 c1(OC)ncc(F)c(=NC(=O)c2cncc(NCc3c(Br)cc(F)cc3Br)c2)[nH]1 CC(CNC1CCCCN(C(=O)Cc2cncn2C)C1)CS(C)(=O)=O C1(NC(C(CC=C)C)=O)CN(C(c2ccnc3c2CCC3)=O)CC2CCCC12 N1(C(=O)NC2CC(C)C2(C)C)CCCc2cc(C(=O)OC(C)(C)C)ccc21 N1(C(CC(=O)OCC)=O)CC2CC(C(=O)NC(C(C)CC)c3ccccc3)(C2)C1 C1(CC(=O)NCC2(C)CSC2)CN(C(c2ccc(O)cn2)=O)CCO1 C1(CNC(c2c(C)nns2)=O)CC2COCC2N1C(=O)CC1CC(F)(F)C1 c1(C(c2nnnn2C(C)C)NC(c2scc(C)n2)C)cccc(C(C)C)c1 C12(CCNC(c3n(CCCSCC)nnn3)c3sncc3C)CC(CCO1)C2.OC c1(CN2C3CN(C(c4ccnnc4O)=O)C(C3)C2)cccc2nc[nH]c12 c1(CC)nc(C#N)cc(=NCC(C)N(C)C(C2CCc3ncncc3C2)=O)[nH]1 c1(C(=O)NCC2(O)CN(C(C(C(CC)C)C)=O)C2)cc(OC)c(F)c(F)c1 c1(C(=O)NC(C2COCCO2)C)ccc(CNC(C2CC2(C)C)=O)cc1 c1(OC)ccc(Cc2nc(-c3cc(C(C)C)c[nH]3)n(CC(N)=O)n2)cc1 C1(CNC(c2cccc(OC)c2)=O)CC2(CO1)CN(C(=O)CCC(=O)C1CC1)C2 N1(C(c2ccc(F)c(F)c2)=O)CCC2CN(C(c3ccc[n+]([O-])c3)=O)CCC2C1 S(=O)(=O)(c1cc(Br)ccc1Cl)N1CCC(NC(c2cccc(C)n2)=O)C1 c1(C(=O)NCC(C)NC(c2cnc3occc3c2)=O)cc(Br)cc2c1OCO2 Cc1ccc2sc(=NCC(C3CC3)NC(=O)CC(C)C(F)(F)F)[nH]c2c1 Cc1ccccc1OCC(=O)N(C1CN(C(=O)CCN2CCC2)C1)C N1(CCC(C(=O)OCC)NC(CCCCC=CC)=O)CCCN(C)CC1C CCCC(C)CCCC(=O)NC1(CNC(=O)CC2CCCCC2(C)C)CC1 c1(C(C)=O)ccc(CN2CCOC(C3CCCC3)C2)nc1OC c1(C(=O)NCCN(CCCCCC)C(=O)C=CCO)cccc(CC(F)(F)F)c1 c1(C(N2C(CN(C(Cc3cn(CC)nn3)=O)CC)CCC2)=O)ccc(N)c(F)c1 C1(C(=O)NCC(CC=C)NC(c2ocnc2CCC)=O)CC2CCC(C1)C2O c1(CC)ccc(C(=O)NC2CCC2NC(c2cc(N(C)C)nc(Cl)c2)=O)c(F)c1 C12(C(N3CC(C(C)(C)C)OCC3)=O)CCCN1CCC2.c12ccc(s1)C(=O)NC2 C(c1cccn1C)=CC(=O)NC(C(C)NC(C(C1CCCC1)OCC)=O)C CC1CCCC1(C)C(=O)NC1CN(C(c2n[nH]cc2Br)=O)CC1C c1(COCCCN(C(C2C(Cl)(C(=O)OC)C2)=O)C)cccnc1.C1CO1 N1(C(c2c(C)c(F)ccc2)=O)CCCC(C2CCCN(C(=O)COC(F)F)C2)C1 c1(C(N(CC(O)CNC(c2ccn(C)n2)=O)C)=O)cc(Cl)c(F)cc1F N1(C(c2cc(CC)no2)=O)CCC(C2CC(NC(C3C4CC5C(C4)C35)=O)C2)CC1 C12(C(=O)NCc3c(CC)nn[nH]3)CCCC1N(C(C1OCCC1(C)C)=O)CC2 N1(C(C2(OCC)CCCCC2)=O)CC(NC(C2CC3CCC2C3)=O)C(C2CC2)C1 N1(C(C=Cc2c(C)nccc2)=O)CC2CN(C(=O)Cc3conc3C)CC2(C)C1 c1(C(N2CCOCC2)C(=O)N(c2cnn(C)c2C)CCCC)ccc([N+](=O)[O-])s1 c1(C(=O)NC(C(=O)NCC(C)CN2CCCC2)C2CC2)ccc(N(C)C)cc1Cl c1(CN(C)C)ccccc1C(=O)NCc1cnc(CC(=O)N(C)C)s1 C1(C(=O)NC2(C)CN(C(=O)CCC3CCC(C(N)=O)O3)C2)COCCN1C=O c1(C(=O)NCC(CO)NC(C2C(CCC)C2)=O)cnc([N+](=O)[O-])cc1C C12(C(N3C(C(=O)OC)CC(F)(F)C3)=O)CCCC1CN(C(C1CCC(=O)O1)=O)C2 C(=O)(CCCCC(=O)N(C(C)C(=O)Nc1ccc(F)cc1C)C)OC n1(C(C)C)cc(C(=O)OC(C)C)ccc1=O.N12CCCC(C1)OC(=O)C2=O C1(CNC(c2ccoc2Cl)=O)COCCN(C(c2coc(C3CC3)n2)=O)C1 c1(C(N2CCC(C(=O)NC3(C=C)CCC3)C2C)=O)c[nH]c2ncccc12 C(C(C)C(=O)NC(C)CC1CN(C(c2ccn(C3CC3)n2)=O)C1)OC C1(C(=O)NC(CSC)CO)CN(C)CCN1C(=O)CC1(N(C)C)CC1 N(C1COc2c(Cl)cc(Cl)cc21)C(=O)CN1C(=O)C2CCCCC2C1=O Clc1cc2ccnc(Nc3ccccc3)c2cn1.c12ccc(cc1)OC2 c1(C(N2CCC(CNC(C(C)CO)=O)C23CC3)=O)ccc2[nH]c(=N)[nH]c2c1 Cc1cc(C(=O)NC23CCC(C(N4CCCC4C(C)(C)C)=O)(CC2)C3)nc(O)n1 c1(C(=O)OC)csc(C(=O)NCC(C)(O)CNC(=O)C(C)n2ccnc2)c1 c1(CC(C(=O)N2CCC(NC(=O)C(F)(F)C3(O)CCC3)C2)O)cc(Cl)cc(Cl)c1 N1(CC)CCN(CC(N2CCCC3(CCC3)C2)=O)C(=O)C1=O Cc1nc(C(=O)NCC2CC3(CCC3)CN2C(C2CC2C#N)=O)c2n1CCCC2 S(=O)(=O)(c1ccc(NC(c2ccc(F)cc2)C)c(F)c1)NCC(CC)O C1(NC(C2(NC(=O)C=CCn3cccc3)CCCC2)=O)CC2(CCC2)C1O N1(C(Cn2ncc(CC)c2)=O)CCN(CC(=O)NC2CC3CCC2O3)CC1 Cc1cc(C(=O)NC(C)CCCCNC(=O)CCC2CC2C)cc(N)c1 CN1CCN(C(C2(C)CCCS2)=O)C(C(=O)NC2CC(F)(F)C2)C1 C(CCCC(C)NC(=O)CCN1CCCCCC1)NC(C(CC1(C)CC1)C)=O N1(C(c2c(C)ccn2C)=O)CCCN(C(C2CCCC2C2CC2)=O)C(CO)C1 C1(NC(c2n(C)c(S)nn2)=O)CCCN(C(=O)CCc2ccc(Cl)cc2)CC1 CC1CC(C(=O)NCC(C(=O)NC2CCN(C(N)=O)C2)N(C)C)CC(=O)N1 N1(C(Cc2cnc(C)s2)=O)CC2CCC(NC(c3cc4cccnc4[nH]3)=O)C2C1 N(C1CCCn2nccc21)C(CC(C)N(C(=O)C(O)C(F)(F)F)C)=O N1(C(=O)NCC(c2c(C)cccc2C)N(C)C)CC2(CC2)C(=O)c2ccccc21 C1(C(N2CC(C#C)(O)C2)=O)CN(C(=O)CN2CCC(C)CC2)CC1C1CC1 Cc1cccc(Cl)c1OCC(=O)NC1(C)CC(NC(=O)Cc2cncn2C)C1 C(CCCCC(=O)N1CCC(F)(CNC(c2c(C)nc(C)n2O)=O)C1)OCC N1(C(CN(C(=O)C2=NNC(=O)C2)C2CC(C#N)C2)=O)CC2(CCC1CO)CC2 N1(C(c2n(CC)ccn2)=O)CCC2(CCCCC2NC(c2ccncc2Cl)=O)C1 CC1COc2c(C(N3CCC(C)(NC(C4(n5cnnn5)CC4)=O)C3)=O)cnn2C1 Cc1ccc(C(=O)NC(CNC(C2CCC(=O)N(C)C2)=O)C2CC2)c(F)c1 CCC(C)(COC)C(=O)N1C(C(=O)Nc2cccc(CCO)c2)CC1C c1(C(N(CCN(C(c2c(CC)c[nH]c2)=O)CC2CC2)C)=O)c(Cl)n[nH]c1C1CC1 c1(C(N2CCN(C(C3C(c4cn(C)nc4)C3)=O)CC2)=O)n[nH]c2cccnc12 C1(NC(C=C(COC)C)=O)CN(C(C2CC2(c2ccco2)C)=O)CC1(C)C CCCS(=O)(=O)OC(C)C(c1ccc(C(C)N)cc1)=O C1(NC(C2C(c3cn(C)nc3)C2)=O)CC2(C1)CC(CNC(C1CCC1)=O)C2 C(=O)(CCCC(C)(C)C)N(CC(CC)NC(c1nccn2nccc12)=O)C c1(C(C(=O)NCCOC)N(CCC(=O)NC)C)cc(OC)c2c(c1)OCO2 c1(C(=O)NC2C(NC(c3cnc(CC)[nH]3)=O)CS(=O)(=O)C2)c(F)ccc(F)c1N C1(NC(=O)Cc2ccc(O)c(O)c2)CC(O)CN(C(c2csc([N+](=O)[O-])c2)=O)C1 C1(NC(c2cnc(C)[nH]2)=O)CN(C(C2(C)CC(C(C)C)=NO2)=O)CC1N=[N+]=[N-] C1(NC(N2CC(C(N3CSCCSC3)=O)C2)=O)CCSC1c1ccccc1 C1(C(=O)OCC)CCCCN1C(N1CCN(CCc2nn[nH]n2)CC1)=O C1(CC(=O)N(CC(O)CNC(c2nc(O)[nH]c(=O)n2)=O)C)CCC2(CCC2)CO1 c1(C(=O)NCCCC(CO)NC(C2(CC)COC2)=O)cc2c([nH]1)CCCC2 C(CCCC(=O)NCC1CC(C)(C)CO1)NC(CC(=O)NCC)=O c1(CCCC(=O)NC2CC(CNC(C3CC3Cl)=O)C2)ccc(F)c(F)c1 C(=O)(C1=C(Cl)CCC(C)C1)NCCNC(C=Cc1occ(C(=O)OC)c1)=O C1(CNC(C=C(C)C)=O)CCC12CCN(C(=O)C(C)Cc1ccc(Cl)cc1)CC2 N1(C(C(CC2CCC2)OC)=O)CCC(C(CO)NC(c2ccc(F)cc2)=O)CC1 N1(C(c2c(C)n(C)cn2)=O)CC(N(C(=O)C=CC2CCCC2)C)C2(CC2)C1 N1(C(C(C2CCCN(C(c3c[nH]c(=N)o3)=O)C2)C)=O)CCC12CCN(C)C2 c1(C(=O)NC2CCC(NC(c3n(C)cc(Cl)c3)=O)C2)cc(F)c(F)c(Br)c1F N1(CCC)CCC(N=c2[nH]c(=NCCc3nccnc3C)c3[nH]ccc3[nH]2)C1 C(=O)(C(C(C)OC)N(C)C)N1CCC(C(N(C(CC)CC)CC)=O)C1 c1(NCC(N2CCN(CC(C)(C)C)CC2)=O)cc(N)ccc1F c1(CCNC(N2CC3(CN(CC)CC)N(CC2)C3)=O)cccc([N+](=O)[O-])c1 c1(C(C(=O)NCC)N2CCC2COc2cnsn2)nc(C)c(C)s1.C1(C)C(=O)N1 CC1(CNC(=O)CCF)CCC(NC(=O)C=CCN2CCCC2)C1 C=CC1(C(=O)O)CCN(C(=O)CCCc2cn(-c3cnccc3Br)nn2)C1 C1(CNC(C(CC)OCC)=O)CC2(CC2)CN1C(c1cncc(C(C)(C)C)c1)=O CC(C)CN=c1[nH]c(N(C)C(c2ccccc2)C2CC2)nc2ccc(Cl)cc12 C(=O)(C(F)(F)CCn1cc(-c2ccsc2)nn1)N(C(c1ccccc1)CO)C CC1CN(C(C2CN3CCN2CC3C)=O)C(C)CN1C(=O)COc1ccccc1 CC1(C)COC(CCC(N2CC(N3CCN(CCCO)CC3)CC2=O)=O)C1 C1(CNC(C(C(C)C)C2CCCO2)=O)CCC12CCN(C(C1CCN1C)=O)CC2 c1(C(=O)NCC(CC)NC(C2(c3ccc(O)nc3)CC2)=O)nc2ccc(Cl)nn2n1 C#CCC(C)(C)C(=O)NCCC1CN(C(=O)C(F)CC)CCO1 c1(NC(C)=O)ccc(C(=O)NCCC(C)NC(=O)C(F)C)cc1F.C1(C)CC1 C=CCCCCC(=O)NC1CCN(C(c2cc(Br)c(C)s2)=O)C1CC N1(C(c2cc(C)nc(C)n2)=O)CCCC(C2CC2NC(C2CCC(F)C2)=O)C1 N1(C(c2cc(C#N)no2)=O)CCCCCC1CNC(c1[nH]ccc1C1CC1)=O c1(C(N(CC)CC2CCN(C(=O)COC(C)=O)CC2)=O)ccc(C)c(O)n1 C1(CCNC(C2(C#C)CC2)=O)CCCN(C(=O)CC2CSCCO2)C1 N1(C(C(c2ccccc2Cl)C)=O)CCOCC1CNC(=O)CSCC1CCCS1 N1(C(C(C)OCCCC)=O)CC(N=c2cc(Cl)nc(C(F)(F)F)[nH]2)C(C)(C)C1 N1(C(CSCC#C)=O)CC2CC2(NC(c2ccnc(N(C)C(C)C)c2)=O)C1 c1(C(=O)NC2(CCOC)CCN(C(=O)C#CC(C)C)C2)nc(C)n2c1CCCC2 c12cnc(nc1)OCNC2=O.C1(CSC)CCC(NC(CCN(CC)CC)=O)C1 c1(CNC(=O)CC(C2CC2)NC(=O)C2=CCCC2)cnc2n1CCC2 C1(C(N2CCC(C(C(NOCC(=O)OC)=O)C)CC2)=O)CCC2(CCCC2)C1 c1(C(C)(C)C)ccc(-c2cnc(C(=O)N(C3CC3)CC3CCC3)cn2)cc1 C(N(CC(C)C)N1CCC(N=[N+]=[N-])CC1)c1c(OC)cccc1 C1(CNC(c2nccs2)=O)CN(C(c2scnc2C2CC2)=O)CCO1 C(CCCCCC(=O)N(CCN(C(=O)Cc1csc(C)n1)C)C(C)C)SC CC(C)(C)C1CNC(=O)N1.c1(C(CNC(N)=O)OC(C)(C)C)ccccc1Cl C1(NC(C(=Cc2cccnc2)C)=O)CC(C)CN(C(=O)Cn2ncn(C)c2=O)C1 C1(NC(=O)C=CC2CCCCC2)COCCN(C(=O)C(O)Cn2cncn2)C1 C(C(C(C)C(C)C)NC(c1ccc(O)nc1)=O)NC(C12CC(CSC)(OC1)C2)=O C(CCC(=O)NCC(C)(C)CN(C(=O)Cc1ccnn1C1CC1)C)OCCOC C1(CC(=O)NCCC(=O)NCC)CC(O)CN1C(=O)C(n1nccc1C)C c1(SC)cncc(C(N2CCC(NC(c3nccc(OC)n3)=O)C2C)=O)c1 C#CC1(C(=O)NCC(C(C)C)NC(C2CCC(=O)N2)=O)CCCC1 C(=O)(C1CCCc2cncn21)NCCC(C)NC(=O)CC1(C)OCCO1 Cc1ccc(C)c(C(=O)NCCC(C)(C)NC(C2CCCOCC2)=O)n1 N1(C(c2c(C)nsc2)=O)Cc2ccnn2CC(NC(c2cc(C(C)C)[nH]n2)=O)C1 C(C)(CNC(C1(C)CC2(CCC2)C1)=O)(CC(C)C)NC(c1cc(C)n(C)n1)=O O=C1Cc2c(-c3nc(NC(c4ccsc4CO)=O)cs3)cccc2N1 Cc1cc(Br)cc(C)c1CC(=O)N(C)CCNC(=O)C(C)O CCCCC(C(=O)N1CCOC(CF)C1)NC(c1ccc(O)c(C)c1)=O c1(C(=O)NC2C(NC(=O)CC3CCCCO3)C2)ccc(CNC(=O)C2=CCOC2)cc1 O=C(CCn1cccc1)N(CCC(=O)NCCCC1CCC1)CCCO N1(C(CC(C)C2CCCCC2)=O)CC2CCCC(C(=O)O)C2C1 N1(C(CCCCNC(C(CCC=C)(F)F)=O)=O)C2CCCC1CC(O)C2 N1(C(CC(CC)C2CC2)=O)CCC(C2CCN(C(=O)C3=C(C)OCC3)CC2)C1 c1(C(=O)NCC2C3CN(C(CSC)=O)C(C3)C2)ccc2c(c1)C(=O)OCC2 N1(C(C=CCCC)=O)CCOCC(CNC(C2(c3cccs3)CC2)=O)C1 c1(CNC(CCCCCC2(CC=C)CCC2)=O)cccc(OCC(=O)N)c1.OCC CC1(C)OC2(CO)CC1(C(=O)NC1CCCCC1NC(=O)C1=COCC1)C2 c1(N(C2(C=C)CCCC2)C(CC)CCOC)c(C)cc(C)cc1C c1(SC)ccc(C(=O)N(CC(C)(C)NC(C2CCC(O)C2)=O)C)c(Cl)c1 C#Cc1ccc(NC(=O)C(C2(O)CN(C(=O)C=Cc3cc(C)no3)C2)F)cn1 C(=O)(C(F)(F)C(C)(C)O)NCCOCCCNC(c1cc(C)no1)=O c1(C(=O)NC2CC(C)(CNC(C(C(C)(C)C)OC)=O)C2)cccc2[nH]ncc12 Cc1ccc(F)cc1CC(=O)NCC(N1CCCC(CNC(=O)C=CCO)C1)=O CC1(C)CCC(CCNC(N2CCCC(c3nc[nH]n3)C2)=O)O1 N1(C(CC2C(CC)C2)=O)CC2CC1CN2C(=O)C=CC(=O)N(C)C C1(C(=O)NC2C(CN=c3nnn(C)[nH]3)CCCC2)CC12C1CC3CC(C1)CC2C3 c1(OC)ccccc1C(N)CC(=O)NC(C)Cc1ccnn1C C12(NCc3ccc(C(=O)OC)cc3)CC1CN(C(=O)Cn1cnnn1)C2 c1(CNC(C(C)N(C(=O)Cc2cnc(CC)[nH]2)CC)=O)cc(C)cc(C)c1 C(C)(C)(CC(F)C(=O)NC1(CCO)CCCC1)NC(C(C)C1CCCO1)=O C1(CNC(C=CCC)=O)CCC(C(N2CCC(CC(N)=O)C2)=O)O1 N1(C(C=CSC)=O)CCCN(C(c2ccc(CC)c(F)c2)=O)C(C)C1 N1(CCS(CCCC)(=O)=O)CCC2(CC1)CN(C(c1cccn1C)=O)CC(C)O2 c1(CN)c[nH]c2cc(C(N3CC4CC4C3)=O)ccc12 C1(NC(c2ccc(C(OC)OC)o2)=O)CN(C(=O)CCC2CC2(Cl)Cl)CC1OC C1(NC(c2c(C)ncnc2)=O)CN(C(c2cc(Cl)ccc2F)=O)CC(F)(F)C1 C1(NC(c2c(CC)oc(C)c2)=O)CN(C(=O)C(C)(C)C2CC2)CC2(CCC2)C1 N1(C(CCc2ccc(C)o2)=O)CCOC(C)C1C(=O)NCCOCC(F)F C1(C(N2CCC(Nc3ccnc(Cl)c3)CC2)=O)CCOC2(CCS(=O)(=O)CC2)C1 CC1CN(C(C2COC(C)C2)=O)CC1CNC(=O)CSC(F)F N1(C(Cc2nc(CC)sc2)=O)CCOCC(NC(C2CC(C)(C(C)(C)C)C2)=O)C1 c1(C(=O)NCC(CNC(c2cccc(OC)n2)=O)(C)O)c2c(nn1C)CCC2 C1(CC#C)CCN(C(=O)CN(C(=O)Cc2cnccc2C)C(C)C)CC1 C1(C(N(CCNC(c2nocc2Br)=O)CC)=O)CCC2(CCC2)CO1 C1(C(=O)NC(C)CN(C(=O)Cc2ccccc2F)C)CCS(=O)(=O)C(C)C1 C1(NC(C(CC)c2ccccc2)=O)C=CCN(C(=O)CNC(=O)CC)C1 C1(N(C(C(COC)O)=O)C)CCCN(C(=O)CNS(N)(=O)=O)C1 Cc1cc(C)nc(NC2CC(C)CN(C(c3cc(N(C)C)ccc3F)=O)C2)n1 c1(C(N2CCCC(C)(NC(c3ncn(CC)n3)=O)C2)=O)noc2c1CCCCC2 C1(Nc2ccc(C(=O)NCCC3(C)CCCC3)cc2)CCCCC1(C)C CC1OC2(CO)CC1(C(=O)NC(CNC(C1CCC=CCC1)=O)CO)C2 Cc1cc(I)ccc1C(=O)NC1CN(C(c2cncnc2C)=O)CC1(F)F N1(Cc2cc(OC)cc(F)c2)CC2(CCC(NC(c3ccc(=O)oc3)=O)CC2)C1 Cc1cc(C(N2CC(N(C)C(c3cc(Cl)ccn3)=O)C(O)C2)=O)ccc1Cl C1(C(=O)NC2CN(C(C3OCC4CCCC34)=O)C2)CCC2(CCC2)CC1 C1(CC)CC(C)CN1C(C1OCCC1CNC(C1CC(=C2CC2)C1)=O)=O C(CC)(CC(=O)N1CC2(CC2)C1)N(C(CN1CCC(OC)C1)=O)C c1(C(=O)OC)cccc2c1CCN(C(C1CC1CNC(c1cn(C)cn1)=O)=O)C2 C(=O)(C(C)(C)CC(C)C)NC(CCOC)CNC(=O)CCCc1cnn[nH]1 C1(CNC(C2(CC)CC2)=O)CCCCN(C(c2cc(OC)ncc2F)=O)CC1 C(CC(=O)N(C)C1CC1)(C(F)F)NC(c1c(C)oc(Cl)n1)=O C(=O)(C#CC(C)(C)C)N(C1C(N(C(Cc2c(C)n[nH]c2C)=O)C)CCCC1)C CC(C)(CCC(=O)N1CCCC2(NC(c3ccc(C(N)=O)s3)=O)CC2C1)[N+](=O)[O-] C1(C(=O)NCC(C)C2CC2)(CO)CN(C(c2ccc[nH]2)=O)C1 C(CCC(C)(C)C(=O)NC1CCC(C)CC1)NC(C(C(=O)OC)C)=O C=CCCCCCC(=O)NC(CN(C)C(c1cc(F)cs1)=O)CC c1(C(=O)NCc2onc(C)n2)nccc(Cl)c1C CCC(CC(=O)NC(c1cnc(C)s1)C)N(C(=O)COCC1CC1)C C=CCCCC(=O)NCn1c(-c2ccccc2)nnc1.C12(CC3(CC3)C1)C(=O)OC2 c1(-n2cc(NC(N(c3ccn(C)c3)CCN(C)C)=O)nn2)cc(F)c(N)c(F)c1 N1(C(c2nc(C)sc2C)=O)CCN(C)C(C(=O)Nc2cccc(O)c2)C1 N1(C(C(CC)C)=O)CCCC(C2CC2NC(=O)C(c2cccc(F)c2F)(F)F)C1 N1(C(CCOC)=O)CCCC(C)C1CNC(c1ccsc1C#N)=O C(C)(CCCC(=O)NC1C2CCC(C2)C1CO)NC(C(CC)=CCCC)=O S(=O)(=O)(c1ccc(-c2ccc(O)c(Cl)c2Cl)cc1)NCCN=[N+]=[N-] N1(C(C)=O)CCN(Cc2cn(CCC=C(C)C)nn2)CC1CC(C)C Cc1cc(C(N2CCC(C(C)NC(=O)C(O)CF)CC2)=O)c2c(O)n[nH]c2n1 N1(C(C)C(=O)NC(N)=O)CCC(C)(NC(c2cnc(C3CC3)[nH]2)=O)C1 C1(c2ccc(Br)cc2)(CNC(=O)OC)CCN(C(=O)C(F)(F)c2csc(Br)c2)CC1 Cc1nc(C2CC2)sc1C1CCCN1C(=O)OC(C)(C)C.c1ccn(C)n1 N1(C(CCCCc2ccc(OC)cc2)=O)CC2=C(C1)CN(C(=O)C(C)C1CC1)C2 c1(NC2(c3n(CCOCC)nnn3)COCC(C)(C)C2)cc2cnccc2o1 c1(CNCCN2CCN(C(c3c(C)scn3)=O)CC2)cc2ccccc2cn1 C1(NC(C2CCC(CNC(c3[nH]cc(C)c3)=O)CC2)=O)CN2CCC1(C)CC2 N1(C(c2cccc(OCCOC)c2)=O)CCC(C2CCCC2(C)C)C1 c1(OC)ccc(C(=O)NC2CC(C)CN(C(=O)CC3OCCO3)C2)cc1C N1(C(=O)C(F)C2CC2)CCC2(CC1)CN(C(C1CC3CCC1C3)=O)C2 c1(OC)ccc2c(c1)C(C(=O)OC1CCCC1)CC2.c12ccc(F)cc1NC2=O Cc1ncoc1C(N1CCC1)C(=O)NCCCOC(C1CCOC1)C1CC1 c1(C(N(C(C)CNC(C)=O)CC)=O)cnn(CCc2cc(COC)on2)c1 N1(C(c2c(OC)cccc2)=O)CCC(C)C(CNC(c2ccc(OC)s2)=O)C1 C1(C)(CNC(COCCOC)=O)CN(C(c2cc(C(F)F)ccn2)=O)CCO1 c1(C(N(CCCCNC(c2cc(CC)c(CC)o2)=O)C)=O)cnc(C)c(C)c1 Cc1ccc(Br)c(C(=O)NCC(C2CC2)NC(=O)C2=CCCCO2)c1 N1(C(C)=O)CCC(O)(C(=O)NCCCOc2ccccc2)C1.C1(C)CC1(C)C CC1CC(=O)CCC1C(N1C(C(N2CCC23CCCC3)=O)CCC12CC2)=O c1(CNC(COCC#C)=O)cccc(NC(c2cnn(C)c2CC)=O)c1 C12(C(N3CC4C(NC(c5ccn(C)c5)=O)C4C3)=O)CC3CC(CC1C3)C2 c1(CCOC)ccc(CSC2CC2)cc1CCN(CCN(CCCC)C)C C1(NC(Cn2ccc(C)n2)=O)CC12CCC(NC(=O)CCc1ccn(C)n1)CC2 c1(OC)cc(F)c(CNC(N2CCCC2(C)Cc2cccc(Cl)c2)=O)cc1OC C(=O)(C1=CC2(CN(C(=O)C(C)(C3CC3)OC)C2)OC1)NC1(C#C)CCCCC1 N1(C(c2cccc(SC)c2)=O)CC2COCC2C1 C(C(COC)CC(=O)N1CCOCCC1C(=O)NC1C2CCCCCC12)OC N1(C(c2ccn(C)c2)=O)CCCC(O)(CNC(c2cnsc2)=O)C1 N1(C(c2c(C)c(C3CC3)on2)=O)CC(NC(C2CC(F)C2)=O)CC(C)(C)C1 c1(C(=O)NC2CCN(C(=O)CCc3cccc(O)c3)C2)cn2ccccc2n1 c1(OCC(=O)NC2CC3(C)N(C2)C3=O)cc2n(n1)CC(C)(C)CO2.CCSC N1(C(C(CNC(C(CC=CC)C)=O)C)=O)CCn2nc(C)cc2C1 N1(C(C=COC(c2cc(-c3cccnc3)no2)=O)=O)CC2CC1CN2C(=O)OC C1(C(=O)NC(C2(OC)CCC2)C)CC2(CC2)CN1C(C1CC1(F)F)=O C(=O)(C(C)CCCC(C)C)NCCOC(CNC(C(CCC(=O)OC)OC)=O)(C)C C(=O)(C(=O)N=c1nc[nH]n1C)NC(c1cn(CCN(C)C)nn1)C N1(C(C(F)=CC)=O)CCC(C2CCN(C(=O)COc3cccnc3)C2)C1.C1CN1 c1(-c2cn(C(C)C(=O)N3CC(CCF)C3)nn2)ccc(CCC(N)=O)cc1 c1(CC)ccc(C(N2CC(O)(CN(C(=O)C(C)(C)C3CCCC3)C)C2)=O)o1 c1(CC)ocnc1C(=O)NC(C1CN(C(c2cc(Br)sn2)=O)C1)C c1(C(=O)NC(CN(C(=O)C=Cc2ccc(CC)o2)CC)C)cccnc1OC CC1(CCO)CCN(C(=O)CC2CCN(C(=O)CC(=O)NCC3CC3)CC2)CC1 C(CC(CC)(CC)NC(C1CC1[N+](=O)[O-])=O)NC(C1(CC=C)CCOC1)=O c1(CN2C(NC(c3ccc(O)cc3F)=O)CC(OC)C2)cc2ccc(Br)cc2[nH]1 C(=O)(C(O)C(F)F)NC1CC(CCNC(CSc2cn(C)nc2)=O)C1 C1(COC)(NC(c2cccs2)=O)CCN(C(c2ccc(O)c(Cl)n2)=O)CC1 c1(CN2C(C(N3C(C(=O)OC)CNC(=O)C3)=O)COCC2)ccc2c(c1)CCC2 CC1CN(C(C2CCC(NC(=O)CC3CCC(=O)C3C)CC2)=O)CC(C)O1 c1(N2CCC(CN(C)C(c3c(Cl)nsc3Cl)=O)CC2)ncc(Cl)cc1[N+](=O)[O-] O=C(CCCC(F)(F)F)NC1CC(CO)N(C(c2nscc2Br)=O)C1 Cn1nc(CCCCC(=O)N2CCC(CF)C2)c2ccccc2c1=O N1(C(C=C(CCN(C)C)Cl)=O)CC(NC(=O)C(c2cncnc2)C)CCC1C Cc1ccc2c(CC(=O)NC3(CO)CCN(C(c4ccncc4)=O)C3)c[nH]c2c1 C1(NC(CNC(c2n(CCSC)nnn2)(CCSC)C2CC2)=O)CC(F)(F)CO1 C1(CC(=O)NCC2CN(C(=O)CCc3cccnc3)C2)CC(=O)N(C2CC2)C1 C#CC(CC(C)C)NC(C1(COC)C=CCN1C(=O)CC(O)C1CCCC1)=O Cc1cc(Br)ccc1S(=O)(=O)NC(c1cncc2c1CCC2)=O c1(C(=O)NC2CC3(CN(C(CCc4ccc(C)s4)=O)C3)C2)cnc2nccn2c1 C1(CNC(c2cn(C)nc2Cl)=O)CN(C(c2ncncc2Cl)=O)C(C)(C)C1 c1(C(N2CCCC(CCNC(C3CCC(COC)C3)=O)C2)=O)cnc(C)c(Cl)c1 CC1COC2(CCCC2)CN1C(C(=O)NCC(F)F)C(C)CC1CCC1 C12(C(=O)NCC34CC(NC(c5ccnc(C)c5C)=O)(C3)C4)CCC(C)(CC1)OC2 CC1OC(C)CC1C(=O)NCC1CCC(NC(=O)C(F)(F)c2csc(=N)[nH]2)CC1 C(=O)(C(CC)C(F)(F)F)N1CC(COC)N(C(C2CC3(CSC3)C2)=O)CC1 c1(OC)cc(OC)c(NC(C2(C)CCCN(C(=O)CC3(O)CCC3)C2)=O)cn1 N1(C(c2ccc(CCC)s2)=O)CCC(C)(CNC(c2ccnn2CCF)=O)C1 C(=O)(CC1=CCOCC1)NC(C(N1CCC(C)C(CC(F)(F)F)C1)=O)=O C1(C)(C(N(C2CCCCC2)CC(C)NC(C2C3COCC23)=O)=O)CCCN1CC c1(C(N2CC(NC(C(C)SCC)=O)(COC)C2)=O)nc(OC)c(OC)o1 c1(C(N(C2CCN(C(c3ccc(F)o3)=O)C2)CC)=O)ncc(C(F)(F)F)cc1N C1(C)(CCC)CCN(C(C2(F)CN(C(c3ccncn3)=O)C2)=O)C1 C1(NC(c2cn[nH]c2)=O)CC(O)(CNC(c2nnsc2-c2ccccc2)=O)C1 c1(C(=O)NCC(CN(C(=O)CC2CC2(Cl)Cl)C)O)ccc(C(C)(C)C)cn1 Cn1cnc2c(C(=O)NCC(CO)NC(=O)Cc3csc(S)n3)ccnc12 Cc1ccc2cc(C(=O)NCC(CO)NC(=O)C(c3ccnn3C)O)cnc2c1 C1(=O)C(CC(C)C)CN1.N1(CC(=C)Br)CCC(OC)C1 c1(C(=O)NCCN(C(CCSC)=O)C2CC2)ccc(-n2nc(C)cc2C)nc1 N1(C(=O)CCc2ccncc2)CCOCC1Cn1cc(Cn2cccn2)nn1 c1(NC(c2n(CCC)nnn2)(C)COC)ccc(-n2nccn2)cc1 N1(C(c2c(CCC)nco2)=O)CC2CC2C1C(=O)Nc1ccc(OC)cc1 c1(C(=O)OC)nc(=NC(=O)c2cccc(C(O)C(F)(F)F)c2)[nH]cc1F C1(CN(C)C(c2cc(Cl)cn2C)=O)CCCN(C(=O)C=C(C2CC2)C2CC2)C1 CCCC(CCCNC(c1cc(C)c(Cl)s1)=O)NC(C1(n2ccnn2)CC1)=O C#Cc1c(NCC(=O)N(CC)Cc2ccc(Br)cc2Cl)cc(Br)cc1F N1(C(C2N(C)CC(F)C2)=O)CC(CNC(c2cnsc2)=O)OC(C)(C)C1 S(=O)(=O)(c1cnc(N2CCCC(O)CC2)c(Cl)c1)N(C(CCSC)=O)C c1(C(=O)NC(c2cccc(C)c2)CNC(C(C=C)(C)O)=O)cccc2c1CCO2 N1(C(C2(C)N(C(CCCOCC=C)=O)CCC2)=O)Cc2n[nH]cc2C1CO c1(C(=O)NC(C2(NC(=O)C(C)OCCN(C)C)CC2)C)cc2c(cn1)OCCC2 N1(C(C=CC)=O)CC(O)CC1(C)C(=O)N(C)CCN(C)C N1(C(C(C)NC(=O)CC2CCOCC2)=O)CCCC1(C)Cc1nccs1 Cc1cc(C(=O)NCC(C)N(C(=O)CCc2c(Cl)cncc2Cl)C)ccc1Cl c1(C(=O)NCCC2CN(C(CS(CC)=O)=O)C2)cc([N+](=O)[O-])cc(C)n1 c1(C(=O)NC(CNC(Cc2ccc(OC)nc2)=O)C)ccc(N)c(F)c1Br c1(CC(=O)NCC2CCCC2NC(C2(Br)CC2)=O)cc(F)cc(Cl)c1 C(CCCCCC(=O)NC(C)CC(C)O)NC(C=CCN(C)CC)=O c1(C(=O)NC(C2CN(C(C3CCCN3C3CC3)=O)C2)C)cccc2c1OC(C)C2 C1(C(=O)OC)CCC(C(N2CC(OCCNc3cc(C)on3)C2)=O)C1 c1(NC(=O)NC(C)CCC(=O)O)cccc2[nH]ncc12 CC1CCC(NC(c2nnc(O)nc2O)=O)CN1CC(=O)NCC(F)(F)F c1(CNCC2(CO)CC(C)(C)C2)ccc(F)cc1F C(C(C)(C)C(=O)Nc1ccnc(Br)c1)NC c1(CN2CCOCC(NC(C=Cc3cnc(C)s3)=O)C2)c(F)ccc(O)c1F c1(C(N2C(CN(C(c3c(CC)ocn3)=O)C3CC3)CCC2)=O)ccc(O)c(N)n1 c1(OC)cc(C)c(NC(C2CN(C(c3ncccc3Cl)=O)CCO2)=O)cn1 C1(NC(C(n2ccc(C)n2)C)=O)CCC2(CC1)CN(C(=O)C1CC1)CCO2 CCC(C)C(C)C(=O)NCC=CCC(=O)N(C)Cc1ccncn1 C12(COCC)CN(C(C3CCOCC3)=O)CC1CN(Cc1ccccc1OC)C2 c1(C(=O)NC(C(C)NC(c2ccc(COC)c(F)c2)=O)C)ccc([N+](=O)[O-])cc1 N1(C(C(=C)CC)=O)CC(C2CN(C(c3cn(CCCOC(C)=O)nn3)=O)C2)C1 c1(C(CNC(=O)NCC(C)N(C)CC2(OC)CCC2)=O)ccccc1.C(CO)O C1(NC(CONC(=O)OC)(C)OC)C2CCCC(F)(F)C12 c1(C(=O)OC)ccc(C(=O)NC2CCC(CN(C)C(C)=O)CC2)cc1O c1(C(=O)NC2(C(=O)O)CCCCC2)cnc2[nH]cnc2c1 CCCCC(C)(F)C(=O)NC1CC2CC(C1)N(C(=O)CN(C1CCSC1)C)C2 C(=O)(C(C)CC(F)(F)F)NC(CNC(C(C=C)(C)O)=O)C(C)C CC(CCCCNC(c1cc(Br)no1)=O)NC(=O)C(C1CCOCC1)F C(=O)(C1CCCc2nccn21)NCCCCNC(C1(CC)CC(F)(F)C1)=O c1(C(=O)NCC(CC)(C)NC(=O)C(C)N2CC(C)C2)cccc(C)c1NC c1(C(=O)NC(C)CN(C(=O)Cc2ccc(Cl)s2)C)cnc2ccc(F)cn12 c1(C(=O)NCCCOCCCNC(C2(CC(C)C)CCC2)=O)cnn(C)n1 N1(C(C2C(OC)CC2)=O)CCN(C(c2cccc[n+]2[O-])=O)C(CCO)C1 c1(N2C(=O)CC(C(N(C)CC3CCN(C(=O)C(N)=O)C3)=O)C2)cc(Cl)cc(Cl)c1 c1(C(=O)NC(C(C)NC(c2nc(C)sc2)=O)C)cc(Br)c(C)o1 Fc1ccc(-c2nc(CC3CC4CCC3C4)n(-c3cccnc3)n2)cc1 CCS(=O)(=O)c1ccc(CC(N2CC(C(C)NC(=O)C(C)(F)CC)C2)=O)cc1 CCCCC(O)C(C)C(=O)NC1CN(C(c2ccnc(F)c2N)=O)CC1CO C(=O)(C(F)C(C)(C)O)N1CCC(N(C(c2ccn(CCO)c(=O)c2)=O)CC)CC1 c1(C(=O)NCC(CN(C(c2c(OC)csc2)=O)C)O)cc2c(C)c(Cl)ccc2[nH]1 C#Cc1cncc(C(=O)NC2CC2CNC(C2CCCN2c2ncccn2)=O)c1 C1(NC(C(C)(C)n2cncn2)=O)CC2(C1)CC(CC(=O)NCC1(F)CCOC1)C2 C(=O)(CC(C(F)(F)F)OC)NC1CCCN(C(=O)Nc2ccc(NCC)nc2)C1 CC1Cc2cc(F)ccc2N1C(=O)NCC(c1ccc(Cl)s1)O N1(C(C2CC2F)=O)CC2CCC1C1CN(c3ncncc3Br)CC21 c1(N2CCCC(NC(C3C(OCC)C3)=O)(CO)C2)nc2ccc(O)cc2s1 c1(C(=O)NC(C(C)NC(=O)COC(F)(F)F)C)cc(Cl)ccn1 c1(OC)ccc(C)c(C(=O)NC(C)CC(C)NC(=O)COCCCC(C)C)c1 CCC(C(=O)N1CC(C(N2CC3(CCC(=O)NC3)C2)=O)(COC)C1)C(C)(C)CC c1(C(=O)NCCCN(C(CCC=CC(C)C)=O)C2CC2)ccc(F)c(F)c1C CCC1=NOC(C(N2CCOCC2CNC(c2cnc(C)s2)=O)=O)C1 CN1CCOC(C(=O)NCCCCNC(c2[nH][nH]c(=N)c2Br)=O)C1 C1(C(=O)NCCOC2CCN(C(c3cn(C)nc3Cl)=O)C2)CN(CP(C)(C)=O)C1 N1(C(c2c(C)cco2)=O)CC2CC(C1)C2NC(C1CC2(CC2)CO1)=O c1(-c2c(-c3n(CC4OCC(C(=O)O)C4)ccn3)csc2)ccccc1F FC1(F)C(CNCCN2CCCN(c3nccs3)CC2)C12CCCC2 c1(C(C)=O)ccc(C(N2CC=CC2CNC(C2CC(=C3CCC3)C2)=O)=O)cc1C c1(C(C)C)ocnc1C(=O)NCC1(F)CC(CNC(=O)CC2OCCO2)C1 c1(OCC)ccc(-c2cn(CCCCCCCNC(=O)CNC=O)nn2)cc1F c1(C(C(N2CCC(OCCNC(=O)CC3CC=CC3)C2)=O)CO)ccc(Cl)cc1 C(=O)(NNc1cccc2c1CCCC2)c1ccc(-c2cccc(N=[N+]=[N-])c2)nc1 CCC(C)C(CC(=O)N1CCOCC1CO)NC(=O)CC1CCCCC1O N1(C(c2c(C)nccn2)=O)CCC2(CCCC2C(N2CCCNC(=O)C2)=O)C1 C(C1CCCCC1)=CC(=O)N(C(C)C(=O)Nc1cnn(C)c1C)CC c1nc(NC2(CSc3ccc(C4CCCCC4)cc3)CC2)cc(N2CCOCC2)n1 c1(CONC(=O)NC(C)(C)Cc2ccccc2Br)c(Br)cc(Br)cc1Br N1(C(C2CCC(O)CC2)=O)CCC2C(C1)CN2C(c1cn(CCO)nn1)=O CC1CCN(C(=O)CCC2CCC(NC(C3CCC(N(C)C)C3)=O)C2)CC1(F)F c1(C(N2CCC(C(C)NC(=O)CC(C)(C)C#N)C2)=O)ccc(F)cc1O C1(C)(C(N2CC(N(C(c3c(Cl)c(C)n(C)n3)=O)C)C2)=O)Cc2ccccc2C1 C(C1CN(C(=O)C(C)N(C)C)Cc2ccccc21)NC(c1c(C(C)C)c[nH]n1)=O C1(C(=O)NCC2(CNC(CC(C)=C(C)C)=O)CCCC2)CCCC(C)C1 c1(OCC)cncc(C(=O)NCC(C)(O)CNC(c2ccc(C)cc2)=O)c1 c1(C(N2C3(CNC(C(F)OC)=O)CC(C2)C3)=O)ccc2c(c1)CCCC2 C=C1Cn2c(OC3CCC(NCC)C3)nnc2S(=O)(=O)CC1.c1(OCC)cccc(OC)c1 N1(C(c2cncc(C)n2)=O)CCCCC12CC(NC(C1CCCC(=O)C1)=O)C2 c1(C(N(CC(CO)(CO)NC(C(C)SCCCC)=O)C)=O)cc(F)ccc1O C1(OC)CN(C(=O)C(=O)NCC(C2CC2)SC)CC1Oc1ccccc1 C(CC(C(=O)N(C)CCc1cc[nH]n1)NC(=O)Cc1cc[nH]n1)OC Cc1conc1CC(N1CCC(CCC(=O)NC(C(N)=O)C2CCCC2)C1)=O N1(C(C2N(C(C)C)CCC2)=O)C(C(N2CCC(C(C)(C)C)C2)=O)CCC1C N1(C(CC=CC=C)=O)CCCCC1C(C)NC(c1oc(CO)nc1C)=O C1(CC)C(CC(=O)NCC2CCC(NC(c3n[nH]cc3C)=O)C2)C1(F)F c1(Cn2cc(C(CNC(C3C(CCOC)C3)=O)C)nn2)nc(C)ccc1C CCCCCCCCC(=O)NC(CC(=O)NC1CCCN2CCCC12)C(F)F Cc1ccc(C(=O)N(C2CN(C(=O)CN3CC4CC4C3)CC2(C)C)C)nc1O C(=O)(CC(P(C)(C)=O)P(C)(C)=O)N1CC(C)C1.CO.CC Cc1nccc(N(C)CC2CCCO2)n1.c12ccc(cc1)NCC2 C(CC(F)F)(C(=O)N1CCCC1CNC(C)=O)N(C(c1c(CC)nn(C)c1)=O)C c1(OC)ccc(CN2CCC(F)CC2)cc1.N1CCC(C(F)C=O)C1 n1(C(C)CC(N2CCN(C(=O)CS(N)(=O)=O)C3CC23)=O)cnc2ccccc12 C1(CNC(c2sccc2Cl)=O)CN(C(=O)C2=CCCOC2)C2CCCCC12 C(=O)(CC(C)(C)N(C)C(c1ncncc1C)=O)NCCNS(CC)(=O)=O CCC(C)C(O)C(=O)NC1C=CC(CNC(c2cnc3sccn23)=O)C1 C(=O)(C(C)CC(C)C)N1CC(O)(CN(C(C(C(C)C)n2ccc(C)c2)=O)C)C1 CC(C(=O)N1CCCC1CCCNC(C12CCC1CC2)=O)C(C)O c1(CC)nnsc1CNC(=O)CNC(=O)CNC(=O)CC12CCCC1C2 C(c1cccc(-c2cccnc2)c1)=CC(=O)NC(c1nc(C)cs1)CC C1(C(=O)Nc2cccc(NC(=O)CC3(CO)CC3)c2)CCCCNC1=O C(=O)(C#CC1(C(F)(F)F)CC1)N1CCCC(NC(c2nnc(C)s2)=O)C1 C(C(C(F)(F)F)N1CCN(C(=O)C=CSC)CC1)NC(C1C(CC)CCO1)=O N1(C(c2cc(Cl)ncc2Cl)C(=O)NC(CC)(C)C)CCS(=O)(=O)C(C)(C)C1 CCC(C(=O)N1CCC(OC(C)(C)C)C1)NC(N)=O.C12CCCC1NC2=O C(=O)(C1=CS(=O)CCC1)N1CCC(OCCN(C(=O)COCC(F)(F)F)C)C1 c1(C(=O)NCC(CC=C)NC(c2ccc(C(F)F)o2)=O)cc(C2CC2)nc(O)c1 N1(C(=O)OC(C)(C)C)CCC(C(=O)OCCC2CCC2(C)C)CC1 Cc1ccc(-c2ccc(-c3nccn3C(C3CCS(=O)(=O)C3)n3ccnc3)s2)nn1 c1(COCC(CC)N(C(=O)OCC(F)(F)F)CC)ccc2c(=O)cc[nH]c2c1 Cc1cccc(F)c1C(=O)NCC1CC2CCC1N2C(C1CCCC1C)=O C(C(C)(CC(C)C)NC(c1cc(C2CC2)no1)=O)NC(c1c(C)onc1)=O c1(CC)ccc(C)cc1C(=O)N(C1CCCN(C(=O)CCCC(N)=O)C1)CCF CC1OC(C)CC1(c1nnnn1CC1CC1)NCCCCSC(C)(C)C C1(C(=O)NCC2(C#C)CCCC2)CC2CC1CC2NC(=O)CC1CSC1 N1(C(C2(OCC)CCC2)=O)C2CCC1C(NC(C1CC1c1ccccc1)=O)C2 Cc1ccc(C(N2CCC(C)C2)C(=O)NCc2ccccc2)cc1I c1(C(CNC(CN2CCCC(COCC)C2)=O)OC)c(C)nn(C)c1C Cc1cc(C)nc(CNC(C)C#CC(=O)OCC(=O)N(C)C)n1 c1(C(=O)Nc2ccc(F)cc2)cc(F)cnc1O.O=C1CCOCCN1 CCCC(CC)CCC(=O)N1CCC(CCC(=O)NCCC(F)=C(F)F)C1 C(=O)(C(F)C(C)CNC(C1(CF)CC(=O)C1)=O)N(C1(SC)CC1)C C1(C(N2CC(C3OCCN(C(CC(CC)C)=O)C3)C2)=O)CC2C(C1)C2(F)F N1(C(c2ccnc(F)c2)=O)CCC2(CCCC2N=c2[nH]nco2)CC1 N1(C(C2C(OC)CCCC2)=O)CCCN(C(c2ccn(C(F)(F)F)n2)=O)CC1 c1(C(=O)OC)cc(C)nc(N(CC(C)NC(C2CCS(=O)(=O)C2)=O)C)n1 C12(C(=O)NCC=CCNC(=O)CCCC3CCC3)CC3CC(C(=O)N1)C2C3 Cc1ccccc1CC(=O)NCCC(C)N(C)C(c1c[nH]nc1C1CC1)=O N1(C(c2nc(CC)sc2)=O)CCOC(CCNc2cnc(C(=O)NC)cn2)C1 N1(C(C)C)C(=O)COCC1C(N1CCC1C(=O)NC1CCN(C(=O)CO)CC1)=O c1(SC)ncc(C(=O)NCC2(C)CC(NC(=O)C3=CCSC3)C2)c(O)n1 C1(OC)(OC)CCC1C(=O)NCC=CCC(=O)NC1CC(n2ccnn2)C1 Cc1ccccc1Oc1ccc(NC(C2(N)CC(F)C2)=O)cc1 C(C)(C)(CN=c1cc(Cl)nc(C2CCCO2)[nH]1)NC(CC1C(C)(C)C(O)C1)=O C1(CN(C2CCN(C(CCN(C)C)=O)C2)C)CCC(C(N)=O)O1.c1(N)nnco1 c1(NCC2(C(C)O)CC2)ccc(S(=O)(=O)NC(C)(C)C(C)(C)C)c(Cl)c1 C(=O)(C(C)C(O)C(C)CC)N(C1CC(NC(c2ccc(CC)c(CC)c2)=O)C1)C N1(C(C2CC(OC)CN2C(C)(C)C)=O)CCCCC(CNC(=O)C=CCOC)C1 N1(C(CC2(CC(=O)OC)CC2)=O)CCCC(NC(c2ccc(Cl)nc2)=O)C1C C1(CCCCC)CCC(C(=O)NC(C)C(CO)NC(=O)CCCCOC)CC1 c1(C(N(CCNC(c2ccnc(Cl)c2)=O)CC)=O)ccn(C)c(=O)c1O C(C)(C(O)C(=O)NCC1(F)CC(NC(c2ccc(CCN(C)C)cc2)=O)C1)SC C(CC(CC)C(=O)NC(C)CCC=CC(=O)Nc1ccc(F)cc1CO)=CC C1(CC=C)(C(=O)NCCCCCCOC)CCN(C(C2CC=C(C)CC2)=O)C1 CCC(O)(CC(=O)N1CCC(CCNC(=O)C2CC2)CC1)c1ccccc1 c1(C2(C(=O)NCC(CC)NC(C3(OC)CCOC3)=O)CCC2)cccc(Cl)c1Cl CC(C#N)CCC(=O)NC1CCC(N(C(=O)CC2CC3(CC3)C2)C)CC1 C1(n2cc(-c3cn(CCC)nc3)nn2)CCCCN(C(c2c[nH]c(=O)cn2)=O)C1 c1(C(N2CC(C)C(NC(=O)Cc3n[nH]c(=N)s3)CC2)=O)occ2c1CCCC2 C1(C(=O)NCC2N(C(CC3CC(=C)C3)=O)CCN(C)C2)CN=C2N=CNN2C1 C1(NC(CC)=O)CC2(CCCN(C(=O)CCc3cc(C)ncn3)C2)C1 C=C(C)C1OCCCC1C(=O)N(C(C)CCNC(C1(C(F)(F)F)CCO1)=O)C Cc1ccc(C(=O)NCC2(F)CCN(C(C3CN(C)C(=O)N3)=O)C2)cc1C c1(C(N2CCC(N(C(C(CCC)=CCC)=O)C)C(C)C2)=O)cc(Cl)c(F)c(Cl)c1 C1(C(N2CC3(OCC(NC(CCCC#C)=O)C3)C2)=O)COc2ccc(O)cc2O1 N1(C(COCC(=O)NC)=O)C2CCC1CC(NC(c1cncc(C)c1C)=O)C2 c1(C(N(CCNC(=O)CCc2cscn2)CC)=O)[nH]c(O)nc1C c1(CC(=O)NCC(C)(C)Cn2ccnc2)cc(C(N)=S)ccn1 N1(C(c2c(C)ncs2)=O)CC2CN(Cc3cc(C(=O)CBr)ccc3O)CC2C1 C(C)(C(C(=O)N1CCCC(CCF)C1)C(C)C)NC(c1c(C)csc1)=O Cc1ccc(OCCN(C(=O)CC2CCCCCC2)CC2CC3CCC2C3)c(C)c1 c1(NC(C2N(Cc3cc(C)[nH]c3C)CC2)=O)cccc(C)c1F N1(C(C(C)O)=O)CCN(C(=O)C=Cc2cnn(C)c2)CC1C(F)F C#CC1CN(C(=O)CC2CCCN(C(=O)C(c3ccn(C)c3)C)CC2)CCO1 C#CCC(C)(C(=O)N1CCCC(CCC)C1)NC(c1scnc1CC)=O c1(C(=O)N(C2CC2)CC2CCCN2C(=O)CC2CC3(CC3)CO2)cnn2ccsc12 C1(NC(=O)NCc2c(C)ncs2)CN(C(=O)CC(C)P(C)(C)=O)C2(CCCC2)C1 n1(COC)cc2c(n1)C(N=c1cc(C)c(C#N)c[nH]1)CCC2 c1(C(=O)NC2CCN(C(c3cnc(CC)nc3)=O)C2)cc2c(Cl)cccc2s1 Cc1[nH]nc2c(C(N3CC(CCCCNC(c4c[nH]nc4Cl)=O)C3)=O)cccc12 C12(OC)CCC(C(=O)NCC3CC3CNC(c3ccc(F)cn3)=O)(CC1)CC2 C1(COC(C2N(C(CCCC)=O)CSC2)=O)CCCC2(CC2)C1 N1(C(CCSCCCC)=O)CCC2C1CCCN2C(=O)Cc1ccccc1O Cn1cc(CNC(=O)CCN(C(=O)C(c2cnn(C)c2)O)CC2CC2)nn1 C12(CO)COCC1CN(S(C)(=O)=O)C2.C12(COC1)C(C)N2 c1(C(=O)NCCCCCCN(C(=O)CC2CC2(C)C)C)ncc([N+](=O)[O-])n1C c1(C(N2CCCC(CNC(C3=C(C)CCC3)=O)C2)=O)ncnc2ccsc12 C1(C(F)(Cl)Cl)CN(c2ccnc(NCC3(c4ccccc4Br)CCC3)n2)CCO1 C1(C(=O)NCCNC(c2ccnn2C2CCC2)=O)CCC2(CCC2)C1 c1(C(=O)NC2C(NC(C(C)(C)NC(=O)OC)=O)COCC2)ccnc2c1CCC2 c1(N(C2CCCN(C(C3C(C)CC(=O)NC3)=O)C2)C)ccn2c(Br)cnc2n1 Cc1ncc(C=CC(N2CCCN(C(c3coc(Br)c3)=O)CC2)=O)c(O)n1 C1(CNC(COCC#C)=O)CCC2(CN(C(c3ccc(CO)o3)=O)C2)O1 C1(CC)CC(C(=O)NC2CC3(CCC3)C2O)CCN1C(=O)CCC(C)C C12CN(CC1C(=O)O)CC(=O)N2.c1(CS(=O)(=O)NC(CC(C)C)=O)ccc(Cl)cc1 n1(CC(N)=O)cc(C2(O)CN(C(c3nc(Cl)cs3)=O)C2)nn1 CCC(C)(CO)C(=O)NCCOCCCN(C)C(c1ccnc(Cl)c1N)=O C#Cc1cccc(C(=O)NC2CCN(C(=O)C(=O)C(F)(F)F)C(C)C2)c1 Cc1ncsc1C(=O)NCC1(O)CC(CNC(c2scnc2C2CC2)=O)C1 CC1(C)CCCC(CC(=O)NCC23CC(CN2C(=O)CSc2nncs2)C3)C1 C1(C(=O)NCC2(O)CC(O)C2)(NC(C(C)CC2CCCC2)=O)CCC(C)(C)C1 c1(C(N2CC(CC(C(=O)N(C3CCC4CC34)C)F)C2)=O)cccn2cncc12 C1(C)(CNC(C2(CC#C)CCOC2)=O)CC(F)(F)CN1C(=O)C(C1CC1)OC C1(C)(CNC(C(C)(C)NC(C2N(CCC)CCC2)=O)=O)CCCCC1O C1(CC(N2CCC(OCC3CCOC3)C2)=O)CCN(C(=O)C=CCF)CC1 n1(CC(=O)NC(C2CCN(C(c3cc(C)no3)=O)C2)(C)C)c(C)c(C)sc1=O c1(C(=O)NC2CC(CCNC(C3C(C(C)C)(CC)C3)=O)C2)cncc2nc[nH]c12 c1(C(N(CCOCCN(C(CCSCCC)=O)C)C)=O)cc(NC)cc(Cl)c1 N1(C(Cc2ccn(C)n2)=O)CC2(CCC(NC(c3coc(Cl)c3)=O)CC2)C1 C1(c2c(C)nc[nH]2)CCN(N(C)Cc2c[nH]ccc2=N)CC1 C1(C)(C(=O)NC2(CNC(C(C)n3ccnc3)=O)CCCC2)CC2(CC2)C1 c1(C(N(CCOCCCN(C(C(C2CC2)SC)=O)C)C)=O)ccccc1F c1(OC)ccc2cc(C(=O)NCc3nc(C)ccc3O)ccc2c1 C1(C)(CCC)CCCN(C(C2(CNC(=O)C(F)(F)C3CC3)CCC2)=O)C1 C1(CCCNC(CCC=C)=O)CN(C(=O)C(C)OCCCCCC)CCO1 C(=O)(C(F)C(F)(F)F)NCC1(CNC(c2ncc(OC)nc2)=O)CC1(F)F N1(C(CCCC)=O)CC=CC(NC(C2CC(N3CCCC3)C2)=O)C1 N1(C(C(C)N(C(COCCCC)=O)C2CC2)=O)CCOC(CCN2CCCC2)C1 N1(C(C(C)C)=O)CCC(NC(c2cnc(OCC(F)F)cn2)=O)C(O)C1 c1(OC)nccc(N2CCCC(CCNC(c3ccc(CC(C)C)nc3)=O)C2)n1 Cc1cc(CC(N2CC(NC(c3ccnn3C(C)C)=O)C(C)(C)C2)=O)ccc1Cl C(C(C)N=c1cc(C)nc(S(C)(=O)=O)[nH]1)NC(c1c(CNC(C)=O)cco1)=O CCCCC(CNC(c1ccnc(C(F)(F)F)c1)=O)NC(c1ncncc1Cl)=O C(C(F)(F)C(=O)NCC1CN(C(C2(Br)CC2)=O)CC1C)OC N1(C(c2ccc(SC(F)F)cc2)C(=O)NC)CCC2(CCN(C)CC2)C1 N1(C(c2ncn(CC)n2)=O)CC(CNC(=O)C=CCCC(C)C)CC(C)C1 C1(C(N(CCCN(C)C)CCNC(=O)C=Cc2cn[nH]c2)=O)CCC(=O)N1 C1(C(=O)NCC2CN(C(C3CCCO3)=O)C2)(CSc2ccccc2)CCOCC1 CC1C(C(=O)N2CC(CO)(NC(C3CC34CC(F)(F)C4)=O)C2)=Cc2ccccc21 Cc1nn(C)c(C)c1CCC(=O)NCC1CCCN(C(c2csc(O)n2)=O)C1 N1(C(C2CC(CC)C2)=O)CCCC(C(C)(C)C(N2CCC(C)(C(N)=O)C2)=O)C1 C1(C(N(CCC(C)C)C)=O)N(C(=O)C=CC2(C)COC2)CCC1(C)C c1(C(N2CCN(C)CC2C(N2CC(S(C)(=O)=O)C2)=O)=O)cnn2cccc2c1 C1(CC)C(NCCCCOCCOCCSC)CCN1C(=O)CCc1nncs1 C1(C(=O)NC(CC=C)CC)CCC2(CC2)N1C(c1cc[n+]([O-])cc1)=O c1(C(=O)NC(C(C)OC)C(=O)NC2CN(C)CC2(F)F)cc(F)ccc1O C1(NC(C2(CO)CC2(F)F)=O)C2COCC1CN(C(=O)CCC(F)F)C2 CN1CCOC(C(N2CCN(C(=O)CCn3ccnc3)C(CF)C2)=O)C1=O CCC(CC)C(F)C(=O)N1CCC2(CC2C(=O)N(C)CCN2CCCC2)C1 C(CC1=NOC2CCCC12)COC(C(C)C(C)C(C)(C)C)=O C1(NC(c2nnn(C)n2)=O)CN(C(C2CCn3ncnc3C2)=O)CCC12CCC2 CC1=C(C(=O)NC2(CCNC(=O)CCC3CCCC(O)C3)CC2)CCS1(=O)=O Cc1cc(C(F)(F)F)nn1CC(N1CCCCC1CC(=O)C1CC1)=O c1(C(=O)NC(CNC(c2cc(CC)ncn2)=O)(C)C2CC2)cncc2ccsc12 N1(C(C2C(OC)CN(C(c3ccc(O)cn3)=O)C2)=O)CC(CO)CC12CCC2 N1(C(Cn2cc(C(C)=O)nn2)=O)CCC(C)(NC=O)C1.c1(C(C)OC)nn(C)cc1O c1(OC)ccc(C)cc1CC(=O)NCC#CCNC(=O)C(C)S(C)(=O)=O Cn1ccc2cc(C(=O)NC3CC4CC3CN4C(c3csc(Cl)n3)=O)cnc12 C(=O)(C(C)(C)C(=O)N1CCOCC1)N(CC(CNC(C=C(CC)CC)=O)(C)C)C c1(OC)ccc(OC)c(C(=O)NCCC2CCC2C(F)(F)F)n1 C1(NC(=O)CCOC2COC2)CCSC12CN(C(c1ccc3nonc3c1)=O)C2 c1(CNc2cccc(-c3c(OCCCC)ccc(F)c3)n2)cc([N+](=O)[O-])c(C)s1 C(=O)(C1CCCn2nccc21)NCC(CC=C)NC(=O)CN1CC(C)C1 c1(NC(N2CCC(C(C)(C)O)C2)=O)cccc(-c2ccc[nH]2)c1 N1(C(CC(=O)OC)=O)CCC2CC2(C(N2CCCC2)=O)CC1 C12(NC(=O)C=CCC(C)(C)SC)CCCC1N(C(=O)C(C)C1CCCC1)CC2 c1(C(=O)NC2CCCN(C(c3c(CC)c[nH]c3)=O)C2)ccc(Cl)cc1C C1(C(N2CCCC(NC(C3CSCC(=O)N3)=O)CC2)=O)CCCCC12OCCO2 C1(NC(CN2C(C)CCC2)=O)CCC2(CC1)CN(C(C1CC(C3CC3)=NO1)=O)C2 C1(CN(C(C2CC(=C)C2)=O)CC)CCCN(C(=O)Cc2ccc(CO)cc2)C1 N1(C(CCc2cn(C)nc2)=O)CCCCC(C(=O)NCCC(=O)NCC(F)F)C1 N1(C(COC(C)=O)=O)CC(NC(C2(C)CSC2)=O)CC12CCOC2 N#Cc1ccc(C(N2CCC2CNC(C2CC23CC3)=O)=O)c(F)c1 CCCCC(C)NCC1CCCN1C(=O)CNC(CC(=O)OC)C1CC1.c1ccccc1 Cc1cc2ccc(C(=O)NCC3CC3NC(=O)C3=CC(C)(C)C3)cn2c1 c1(OC)ccc2c(C(=O)NC3CC3CNC(C3CCC4CC34)=O)c[nH]c2c1 N1(C(C2CC(=C)C2)=O)CCC(NC(=O)C(F)C(F)(F)C(F)(F)F)C2(CCC2)C1 Cc1cc(O)ccc1C(=O)N(CC(C)NC(C1C(C)C1C)=O)C Cc1cccnc1C=CC(=O)NC1CC(CO)N(C(=O)C2=COCCO2)C1 C(=O)(CCCC(C)CC)NC(C(=O)NC(CCCC)C(=O)NC)CCC C12(C(N3C(C(C)(C)NC(c4ccc(Cl)s4)=O)CCC3)=O)CCOC1CCOC2 c1(C(C(N2CC(C)(OCC(=O)NC)C2)=O)=O)ccc(O)cc1 C(=O)(CCC(=O)NC(C1CCCCN1C(C1CS(=O)(=O)C1)=O)C)NCCC N1(C(C(CC)OC)=O)CC(C)(C)OCC1CNC(c1cc(C(=O)OC)nn1C)=O C1(NC(C=CSC)=O)COC2(C1)CN(C(C1CC1C(C)C)=O)C2 CCC(O)C(=O)NC(c1ccccc1)CNC(C1(CF)CC1)=O n1(CC(N2C(CNC(CSCCC#N)=O)CC(O)C2)=O)ncn2nccc2c1=O c1(CC(=O)NC(CC)CN(C(=O)C(C)OC)C)ccc(NC(N)=O)nc1 C12(NC(c3ccco3)=O)CCCC(NC(=O)CN3CCCC3=O)(C1)C2 c1(CC(=O)NC(C)C(C)(C)NC(=O)CN=S(C)(C)=O)ccc(F)c(Cl)c1 CCCCC(C(=O)NCC1(O)CC(CNC(c2cc(Cl)ccc2C)=O)C1)N(C)C C=CCC(C(=O)NCC(O)CN(C)C(C1(c2ccc(Cl)nc2)CC1)=O)OC c1(C(N(CCNC(c2cccc(F)c2)=O)C2CC2)=O)cc2ccncc2cc1F c1(CNC(C2CC(OCC)C2)=O)cc(C(=O)NC2CCC2O)on1 CC1CN(C(C2Cc3nccn3C2)=O)CCCN1C(C1CC(N(C)C)C1)=O N1(C(CC(C)SC)=O)CCOC2CCN(C(c3ccc(Cl)cc3Cl)=O)CC12 C1(CC(=O)N(CCCNC(C2(C)CCCO2)=O)CC)COc2ccccc2O1 C1(C(=O)NCC(CC)CC)CC(NC(=O)CN2CCCC2)C12CCC2 C123CCC(CC1)(CC2)C(=O)N1CCN(CC1)C(C)CNC3=O.c1(N)cccs1 CC1Oc2ccc(C(=O)NC3CN(C(C4CCC(=O)N4)=O)CC3(C)C)cc2C1C c1(CCC(=O)NCC2N(C(C(C)c3ccco3)=O)CC2)nc(=N)[nH][nH]1 N1(C(C(n2cc(-c3cc(Cl)ccc3F)nn2)C)=O)CC2(CCC2)C2COCC12 C(=O)(C1COc2ccc(F)cc21)N(C)CCNC(=O)C=CC=C(Cl)Cl Cc1ccc(C(C)C)cc1C(N(C1CN(C(=O)C(C)CF)CC1O)C)=O C(=O)(CCCCCO)NC(C1CN(C(c2ccc(C(F)(F)F)cn2)=O)CCO1)C N1(C(C(C=C)(C)O)=O)CCN(C(C23CC(C2)C3)=O)C(CCO)C1 N1(C(CN(C(C)=O)C2CC2)=O)CCC(C2CC(NC(c3ccccc3F)=O)C2)C1 c1(CNC(C(N2CC(C)(C(C)C)OCC2)=O)=O)ccc2c(c1)CCCC2 N1(C(=O)OC(C)(C)C)CC2CC2C1C(=O)O.c1(Nc2ccc(F)cc2)cccc(O)c1 C1(NC(C(F)=CC)=O)CCC2(CCCN(C(=O)Cc3cnn4ccccc34)C2)C1 CC1CN(C(=O)C(C)CC(N)=O)CC2(CCN(C(c3cc(Cl)ccc3Cl)=O)C2)O1 c1(CC)c(F)ccc(S(C)(=O)=O)c1F.c1(C2CN(C(C)=O)C2)cn(CCCO)nn1 C1(C2CN(C(=O)C=Cc3ccco3)CCO2)CCn2cncc2C1 C1(C)(NC(C=CC(=O)NC(C(=O)NCC=CC)C)C)COCCO1 N1(C(CC2ON=C(C)C2)=O)CC2CCN(C(c3cnn(C4CCCC4)c3)=O)CC12 c1(C(=O)NCc2scc(C)n2)cccn2c(-c3cccn3C)cnc12 CN1C(C(N2CCC(NC(=O)CCCCNC(N)=O)C(O)C2)=O)CCS1(=O)=O N1(C(C(C)c2ccco2)=O)CC2CN(C(c3ccc(C(N)=O)o3)=O)CCC12 Cc1cc(C=CN2CCN(C(=O)CC(=O)N(C)C)CC2C)ccc1F N1(CC)CC(NC(=O)C(C)(C)C2CCCN2C(C2CC(F)(CF)C2)=O)C(C)C1 Cc1ccc(C)c(C(N2CCC(NC(=O)C(F)(F)c3csc(C)c3)C2C)=O)c1 C1(C#N)(C(=O)NC2C(C)CN(C(=O)CCC3CCCC3)CC2)CC12CCCC2 C(C(N=[N+]=[N-])C(=O)NC1CC(C(F)C(N2CC(OC)CC2(C)C)=O)C1)OCC N1(C(COCC(=O)NC)=O)CCC2C(CCN2C(c2cncc3c2CCC3)=O)C1 C(CNC(c1conc1C)=O)(C(=O)N1CC(CC(F)F)C1)OC C1(OCCNC(C2COCC2O)=O)CCN(C(=O)CCc2cc[nH]n2)CC1 CC(C)(O)C(C(N)=O)NC(C1(CCNC(c2ccc(C(F)F)o2)=O)CC1)=O c1(C(=O)NCC2C(NC(C(C(C)O)N(C)C)=O)COC2)c[nH]c2nccc(Cl)c12 c1(-c2nc(CC)nn2C2CCCOC2)ccc(O)cc1Cl C(CN=c1ccnc(N2CCC(c3cncn3C)C2)[nH]1)SC c1(C(=O)NC(C2CCCN2C(=O)CC2(C)CCCC2)C)nccn2ccnc12 c1(CN(CC(=O)NCCCNC(=O)C=CC(F)(F)F)C)ccc(Cl)c([N+](=O)[O-])c1 c1(C(=O)NC(CC)CNC(=O)C(C)N(C)C)ccc(C)c(S(=O)(=O)N(C)C)c1 c1(C(=O)NC)cc(OC)c(C)c(OC)c1.C1(NC2C(SCC)C2)CC(CC=O)C1 c1(C(N2C(CO)CC(NC(c3cnc(OC)s3)=O)C2)=O)cc2cccnc2s1 C1(C(N2CC(NC(CCN3C(C)CCCC3)=O)C(O)C2)=O)OCCN(C)C1=O CC(C)(O)C(C(=O)NCC1CCSC1)NC(=O)C=Cc1cc[nH]c1 C1(C(=O)OC2CC2(F)F)CCCCC1OC(C(C(=O)NC)SC)=O N1(C(C=Cc2ccc(CC)cc2)=O)CC2CCC(NC(=O)C3=C(Cl)CCC3)(C2)C1 C1(COC)(NC(=O)CSC2CC2)CCCN(C(=O)CN2CCCNS2(=O)=O)C1 S(=O)(=O)(c1cc(Br)c(F)cc1F)N1C(C(N=c2[nH][nH]c(C)c2C)=O)CC1 C12(C(=O)NCCCCNC(C(COC)(C)C)=O)C3C(=O)C4C5CC(C14)C2C35 N1(C(C(CCCC)O)=O)CCC(C)(C)C(CNC(=O)CCN2CCC(C)CC2)C1 c1(CC(=O)NCC(C)NC(C(c2cccc(Cl)c2)OC)=O)n[nH]c(=NC)s1 C1(O)(C(C2CC2)NC(N2CC(CC#C)C2)=O)CCCCC1 c1(CNC(C2CCN(C(C(=O)OC)C)CC2O)=O)cc2n(n1)CCCC2 c1(NC(C2(C)CN(Cc3cc(O)cc(F)c3)C2)=O)cc(F)c(Cl)cc1F c1(OC)ccc(C(=O)NC(CCNC(C2CCOCC2)=O)C(C)C)c(C(=O)O)c1 C12(CNC(C=CCOC)=O)CC(CN1C(=O)CC(C)OC(C)=O)C2 c1(CC)cnc(C(N2CCC(C(C)C(N3CCC(OC)(OC)C3)=O)CC2)=O)nc1 CC(C)(C)C(CC(=O)N(CCCO)CCO)NC(c1cccc2c[nH]nc12)=O C(N=c1[nH]c(=NCC2COc3ccccc3O2)c2[nH]ccc2[nH]1)C1OCC(C)(C)C1 Cc1nc(CC(=O)NCC2CC(C)N(C(=O)C=Cc3cc[nH]n3)C2)sc1C Cc1[nH]nc(C(=O)NCc2ccc(CNC(=O)CCc3nc(O)n[nH]3)cc2)c1Br C1(C(=O)OC)CCC(CCOC(C2CN(C(=O)Nc3csnn3)C2)=O)CC1 N1(C(C2CC(n3cc(OCCOCCOC)nn3)C2)=O)CCCC2(CCCO2)C1 N1(C(CN2C(C)CC2)=O)CC2CCCC(C1)C2C(=O)NC1C2COCC12 N1(C(C(C)OCCC(C)C)=O)C2CCC(C2)C1CC(=O)NC(C)CCCl C1(NC(C(OC)OC)=O)CC(C)N(C(C2(c3cccc(Br)c3)CC2)=O)C1 C1(NC(=O)CC2CCCC2)C2CCC(F)(F)C12.C12CCCC1CNC2=O CCC(Cc1cccc(C)c1)C(=O)NC(c1cccc(Cl)c1)CN1CCCC1 C(=O)(C(C)C(C)S(C)(=O)=O)NC1(CO)CN(c2cc(C)nc(C3CC3)n2)C1 c1(C(=O)NC(C(C)NC(C2=NOC(C)C2)=O)CO)cc(N)cc2ccccc12 c1(NCC2CCN(C(c3cnn(C4CC4(F)F)c3)=O)C2)ccc(C(F)(F)F)cc1 N1(C(C(CO)OC)=O)CCOCC1C(=O)NC(CCO)C1CC1 C(=O)(C(CC)SC)N(CC(CC)NC(=O)CC1COC(=O)C1)CC N1(C(CCOC2CN(C(C(CC)SC)=O)C2)=O)CCC(C)(O)C1 c1(-c2n(C)nnn2)cc(Nc2sccc2C(N2CCC3(N)CC3C2)=O)ccc1F c1(COC)ccc(C(=O)N(CCCCNC(=O)Cc2cc(OC)no2)C)cc1F c1(CC(=O)NCCC(=C)CNC(=O)C(O)CN(C)C)c(OC)cccc1F C(=O)(C#CC1CCCOC1)N1CCC(CCN(C(C(C)C)=O)C)CC1 C1(NC(C(CC)Oc2ccccc2)=O)CN(C(C2(C3CC3)CC2)=O)CC(C)(C)C1 N1(C(c2n[nH]c3c2CCC3)=O)CCCCC12CC(NC(C1(O)CCSCC1)=O)C2 C1(NC(c2cc(C3(C)CC3)n[nH]2)=O)CCCC(NC(=O)CSS(C)(=O)=O)C1 c1(CC)ccc(NC(=O)CN(C(=O)CCc2cc(C)no2)C2CC2)c(C)c1 N1(C(CC2(C(=C)F)CCC2)=O)C2CCC(C(=O)N(CC#CC)C)C1CC2 C1(C)(n2c(CCCCCSC)nc(-c3ccc(C)o3)n2)CCS(=O)(=O)C1 C1(=CC(=O)NC(C2CN(C(=O)CC3COCCO3)C2)C)CCC(C)(C)CC1 C1(N(C(c2occc2C(C)C)=O)CC)CCN(C(c2cn(C)nc2C)=O)CC1 N1(C(C2(C#C)CC2)=O)CCOC(CCNC(=O)CC2CCC(C)(C)O2)C1 C1(NC(C(C=C)O)=O)(COC)CCN(C(c2ccnc(N3CCC(C)C3)c2)=O)C1 C1(C(=O)NC(C)C(C)NC(=O)CN(C2CCSC2)C)(OC)CCC(C)(C)C1 N1(C(=O)OCC)CCN(C(C2CCC(NC(c3ccn(C)n3)=O)C2)=O)CC1 C1(C)(CNC(CC2CC(SC)C2)=O)CCCN(C(c2scnc2C(C)(C)C)=O)C1 C1(CNC(C(C)NC(C(OC)OC)C)=O)CCCCC1 CCCCC(F)C(=O)NCC(c1ccccc1)(c1ccccc1)O Cc1nnn(CC(=O)NCC#CC(=O)N2CCC(C(=O)N(C)C)C2)n1 C1(C(=O)NC23CC(CNC(C4=CC(C)(C)C4)=O)(C2)C3)CCCCC12CCC2 N1(C(CCCOCCC)=O)CCC(CO)C(NC(C2(CCF)CCC2)=O)C1 N1(C(CCOCC#C)=O)CCOC(CCNC(=O)C=CC2CCOC2)C1 c1(CNC(CC(C)CNC(c2ncccc2N)=O)=O)cc(F)ccc1F C1(NC(=O)CC2CCC(F)(F)C2)CCN(C(=O)CSc2nc[nH]n2)CC(O)C1 n1(CC(Cc2ccccc2)NCCC(C)n2cccc2)cnc2ccccc12 c1(CC(C(=O)O)Nc2ccccc2)cn(C2CC2)nc1C.c1(OC)cccc(Cl)c1 N1(c2cc(C)[nH]n2)CC2C(C(=O)NCC3CCN(C)C3)C2C1 N1(C(CCN(C)CC)=O)CCCC(C(=O)NCc2csnc2OC)CC1 Cc1ccc(C(=O)NC(CCNC(=O)C(C)(Cl)Cl)C(C)C)c(Br)c1 N1(CC(=O)NCC2(CNC(C3CCCC(OC)C3)=O)CCC2)CCCNS1(=O)=O C(c1cncs1)=CC(=O)NCCCC1(NC(C2CC3CC3C2)=O)CC1 CC1CN(C(=O)COc2ccc(Cl)c(C(F)F)c2)CC(C)CN1C(=O)C=C1CC1 C1(NC(=O)NC(c2ccccn2)(C)Cc2ccc(C)cc2)CCOC12CCOCC2 CC(C)(C)C(C(=O)NCCCC1(NC(C2CCCOC2)=O)CC1)C1CCCC1 Cc1nn(CC(=O)NC2CC2NC(c2nc(C(F)(F)F)sc2C)=O)cc1Cl CN1N=C(CC(=O)N(C2CCN(C)CC2(C)C)CC)CC1=O.C(=O)(C1CC1)OC N1(C(c2ccc(OC)cc2Br)C(=O)NC2CC2)CCS(=O)(=O)CCC1C C#CC1(O)CCN(C(=NCCC(=O)N(C)C)NCc2ncc(CC)o2)C1 CC(CC(F)(F)F)C(C(=O)NC(C)(C)C)N1CCC(O)C(C2CCCC2)C1 C(C(C)(C)CC(=O)NCC1C2CC3C(C2)C13C(=O)NCC(C1(C)CC1)OC)OC Cc1cc(C(=O)N(C)CC2COCCN2C(=O)C#CC2CCCO2)cn(C)c1=O CN1C(=O)CC(C(=O)NC2CCCC(NC(=O)C3=CCCCO3)C2)NC1=O C(=O)(C(C)CC(C)C(C)=O)N(C(C(=O)NC1CCN(OCC)CC1)CC(F)F)C C1(CNC(C=COCC)=O)COCCN(C(c2ccccc2CCC(N)=O)=O)C1 CC1CN(C(=O)CSCO)CCN1C(=O)COCC1CCCCO1.C1(SC)CCCO1 O=[N+]([O-])c1cc(F)cc(Cl)c1N1CCCC(c2cc[nH]n2)C1 C1(NC(c2c(CC)nn(C)c2)=O)CC2CC(NC(C3CC4(CCCO4)C3)=O)CC12 C1(C)(OC)CC(NC(c2c(CNC(=O)CC3CCC4CC34)nnn2C)=O)C1(C)C c1(C(N2CCC(C(N)=O)CC2)=O)cc(S(=O)(=O)N2CCCCC2)ccc1O CC1CCC2CN1C(=O)CNC2=O.C(=O)(CCP(C)(C)=O)NCc1ccc(Cl)s1 c1(C(N2CC3C(N(C(CCC#CC)=O)C)C3C2)=O)c(C)ccc2ncccc12 Cc1nnc(CC(=O)NC2CCN(C(c3ccn(C4CC4)n3)=O)C2)s1 Cc1nn(CCO)c(C)c1C(=O)NCCC(C)N(C(=O)C(F)=C1CCCC1)C c1(C(=O)NC(C)(CNC(=O)CCC2CCCO2)C2CC2)nnn2c1COCC2 C(C(C(=O)N(CC(F)F)C)C(C)C)NC(C(C(=O)OCC)F)=O N1(C(C23CCC(OC)C2CC3)=O)CC2N(C(=O)C(F)CC3CCC3)CCC2(C)C1 c1(C(N2CC(CNC(CCOCCC)=O)C(C)CC2)=O)cnc2sccn2c1=O Cc1cccc(C(=O)NC(c2ccccc2)C(=O)NCC(C)(C)F)c1N c1(C(=O)NC2CCC(C(N(CCCC)CCO)=O)C2)ccc(C)c(CO)c1 N1(C(C(C(C)C)O)=O)CCCN(C(c2ccn(C3CCCC3)n2)=O)CC1C Cc1cc(=N)[nH]cc1C(=O)NCC1(C)CCN(C(c2nc(O)[nH]c(=O)n2)=O)C1 N1(C(c2cn(CCCC)nn2)=O)CC(C2(NC(=O)CCOC3COC3)CC2)C1 C=CCC(C)C(=O)NCC1(CNC(c2ccccn2)=O)CCCC1 n1(CCCOCC(C)C)cc(CCCCCO)nn1 C1(F)(CNC(C(CC)NC(N)=O)=O)CCCN(C(=O)C(C)(C)NC(C)=O)C1 C12(C(=O)NCCN(CCCC)C)CC(CCO1)N(C(=O)CC(=O)OCCCF)C2 N1(C(c2cc(CC)cc(C)c2)=O)CC(C2CN(C(C3(Cl)CC3)=O)C2)C1 N1(C(c2c(F)ncc(OC)c2)=O)CCC2(C1)CN(C(=O)CNS(C)(=O)=O)C2 C1(C(=O)OC(=O)CCc2ccsc2Br)CC(=O)N(Cc2cccs2)C(=O)C1 C1(Cc2ccoc2)C(=O)N1.c1(C(N2CC(=CC)C2)=O)ccn(CCC)n1 CC1(C)COCCC1C(=O)NCC1CC2CCC1N2C(c1cnns1)=O CC1CN(C(=O)C(C)(C)CN(C)C)CCN(C(=O)C(F)CC2CCOC2)C1 C1(NC(c2nnn(C)n2)=O)CCN(C(c2ccnn2CCF)=O)CC1(C)C C1(NC(c2nc(C)oc2)c2nnnn2CCOCC2CC2)CC12CCCC2 CC1CC(NCC(c2ccccc2)N)c2ncnn21 CC1(C)CC(=O)OC1NC(=O)Cn1ccc(-c2ccco2)n1 Cc1cc(C(=O)NCCOC2CCN(C(C3(C)COC3)=O)CC2)c(O)nn1 CC(C)CC(C(=O)NCCC1CCCN(C(=O)CCCSC(C)(C)C)C1)C(N)=O c1(C(N2CCC(CNC(c3cnn4cnnc4c3)=O)C2)=O)cc(O)cc(F)c1F C(=O)(C#CC1(C(F)(F)F)CC1)NCCN(C(Cc1n[nH]c(=NC)s1)=O)C c1(C(=O)NC(C2CCN(C(=O)Cn3ncnn3)C2)C)cc2n(n1)CC(F)C2 N1(C(C=CC(=O)OCC)=O)CC2CC1C2CNC(c1cncc(C(F)(F)F)c1)=O C1(CC)CN(C(=O)CSCCc2ccccc2)CCN1C(c1ccc(C)cn1)=O C1(C(N(OCC)CC)=O)CN(CC)C(C)(C)C1.C1(=O)CCCN1 C=CC(C)(O)CC(=O)N(CCC(C)NC(C1(c2cccc(C)c2)CCCC1)=O)C CC1(C)CCCN(C(=O)CC2CCCOC2)C1CNC(C12CCC(CC1)CO2)=O C#CCCCCCCC(=O)NC1CN(C(=O)CCn2ccnn2)CCC1F C(=O)(CC(C)(C)CC(F)F)NCCC(C)N(C(C(CC)CC(C)C)=O)C C(=O)(C(C)(C)N(C)C)NCCCN(C(c1c[nH]nc1-c1cccnc1)=O)CC.C c1(C(=O)NC(CNC(c2cnn(COC)c2C)=O)C)cc2cccc(OC)c2o1 C1(CO)(CN2CCC(=O)CC2C2CC2)Cc2ccccc2C1 C1(CNC(CCC(C)O)=O)CN(C(c2cc(C3CC3)no2)=O)CCC1(C)C C1(CNC(C(C)N(C)C)=O)CCC(C)(C)CN1C(C1COC(=O)O1)=O c1(C(=O)NCC(C)(C)NC(Cc2c(C)ocn2)=O)cc2c(C)n[nH]c2nc1O c1(C(=O)NC2C(NC(CC3CCC(=O)NC3=O)=O)C2)ccccc1C#CC1CC1 C1(C(=O)NCCOc2ccc(C(CC)=O)cc2)CC2C=CC1C21CC1 Cc1nn(CC(=O)NCC(C2(O)CCN(C(c3ccnn3C)=O)C2)C)c(C)c1C Cc1ccc(C)c(C(N2CC3CN(C(c4cc(C)c(C)o4)=O)CC23)=O)c1 N1(C(CNC(C2C(C)C2)=O)=O)CCC(F)(C(=O)N(C)CCn2ccnc2)C1 c1(OC)ccc(S(=O)(=O)N2CCN(C(c3occc3Cl)=O)CC(O)C2)cc1 C1(N(C2CCS(=O)(=O)C2)CC(C)C)CCCN(CC(=O)NCCc2ccco2)C1 N1(C(C=CC(C)(C)SC)=O)CCCCC1C(N1CCC(C2(C)N=N2)C1)=O C1(CC)CCC(C(=O)NC2C=CCC(C(=O)NCCOCCF)C2)CC1 c1(Cc2nc(C3ON=C(C4CC(=C)C4)C3)on2)ccc2ccc3ccccc3c2n1 Cc1nc(C)n(CCNC(=O)CC2CC2C2CN(C(C3OCCC3(C)C)=O)C2)n1 C1(CNC(=O)Cn2cnnc2O)CCCCC1C(=O)NCC1CNC(=O)CO1 CN1CCN(C)C(C(=O)NCC2CC2NC(c2ncoc2C2CCC2)=O)C1 Cc1nn(C)c(Cl)c1C=CC(=O)NCCCCC(C)NC(=O)CC(C)CF C1(C(=O)NC2C(CC=C)COC2)CCN(C(c2cccc(=O)o2)=O)C1CC c1(C(N2CC(N(C(c3c(OCC)scc3)=O)C)C(O)C2)=O)ccn2c1CCCC2 N1(C(CCC2C(C)=NOC2=O)=O)CCC(C2CCCN(C(=O)C#CC(C)C)C2)C1 N1(C(c2c(C)cc(CO)o2)=O)CCN(C(=O)CCCn2cccn2)C(CCO)C1 C(CCC(=O)NCCC1(O)CCOC1)(C(C)C)NC(Cc1c(C)con1)=O c1(CC(=O)NCC2(NC(c3[nH]cc(C)c3)=O)CCC2)cn2c(n1)CCCC2 c1(C(=O)NC(C2CN(C(CC(=C)C)=O)C2)C)cc(O)cc(Cl)c1 c1(CC(=O)NC2C3N(C(C=C(CC)C)=O)CC(CC3)C2)ccc(S(C)(=O)=O)cc1 N1(C(CC)=O)CCN(C(c2cnc3snc(C)c3c2)=O)C(C)CC1C n1(C(C)C)ncc(C(=O)NCC2(NC(=O)CC3CC=CCN3C)CCC2)c1Cl Cc1cc(C(=O)NC2CCN(C(c3cnn(C(C)C)c3N)=O)C2)cnn1 C(C)(C(=O)NC1CCC(NC(=O)CCC2(C)NC(=O)NC2=O)CC1)(C(C)C)OC C1(NC(CCC=C(C)C)=O)(CO)CCCN(C(=O)Cc2csnn2)C1 c1(NC(C2(F)CCN(C(CC3CC(=O)C3)=O)C2)=O)cccc([N+](=O)[O-])c1 Cc1cc(C(=O)NCc2ccc(C(=O)NCc3cc(C)ns3)s2)c[nH]1 c1(C(=O)NCC(C2CCOC2)NC(C=CCOC)=O)sc(CO)nc1C C(=O)(C(F)C(C)CNC(c1nnccc1C)=O)N1CCC(COC)CC1 c1(CC(C)C(=O)NC2C=CCN(C(=O)CCS(N)(=O)=O)C2)nc2cccnc2[nH]1 C1(CNC(c2n(C(C)C)ncc2)=O)CC2COCC2N1C(c1csc(C#N)c1)=O CC(CCNC(=O)CCn1cnnn1)CCNC(c1nccnc1C(N)=O)=O c1(OC(C)C)ccccc1CC(=O)NCC(C)(C)CNC(=O)C(F)=CC1CC1 C=CCC(C(=O)NC(c1ccccc1F)CNC(=O)CCSC)NC(C)=O N1(C(C(SC)SC)=O)CCC(C)(C)C(CNC(=O)CC2CCCCC2(F)F)C1 C1(C)(NC(C(CC)N(C2CN(C(=O)OC(C)(C)C)CC2F)C)=O)CCCCC1C C1(C(NOCCC(C)O)=O)CC(O)(CNC(=O)CC2CC(N(C)C)C2)C1 c1(C(=O)NCCCCNC(CCCn2c(C)nc(C)n2)=O)c(O)nnc(C)c1C c1(OC(CC)C)cccc(C(=O)NCC(CNC(C2CC(Cl)(Cl)C2)=O)OCC)c1 c1(OCCC)ccc2cc(-c3nc(Cc4ccccc4)no3)[nH]c2c1 c1(C(=O)NC(c2cn(-c3ccc(C)cc3)nn2)(C)C)cncn(C)c1=O C1(CNC(=O)NC2CCC2CC2CC2)C=CCN1C(n1cc(Br)cn1)=O c1(CC(N2CC(C)C(NC(c3cc(O)no3)=O)C2)=O)nc([N+](=O)[O-])n[nH]1 CC(C)C(C(=O)N1CCCC1CN(C(=O)CC1CCC2CC12)C)n1ncc(N)n1 N12CCCC1C2=O.C1(COCCCN(C(C)=O)C)CCCN1c1cnccn1 N(S(=O)(=O)N1CCC(CO)C1)CC1CCCS(=O)(=O)C1 C=CCN=C(NCC(C)(C)C(=O)OC(C)C)NCc1ccc(I)cc1 c1(C(=O)NCC2CC(NC(C(C)OCCC#C)=O)CC2O)ccc(F)c(Cl)c1 N#Cc1cc(CN2CCC(C(=O)Nc3c(Br)cc(F)cc3Br)C2)cc(F)c1 C1(O)(CN(C)C(c2cc(N)cc(F)c2)=O)CCN(C(C2(O)CCOC2)=O)CC1 c1(C(=O)NC(C2CCN(C(=O)C3=NNC(=O)C3)CC2)C)cc2ccc(F)cc2s1 CC1NC(=O)OC12CCN(C(C1CCC3COCCC3C1)=O)CC2 c1(C(N2CC=CC(NC(c3n(CC)ccc3)=O)C2)=O)cccc(F)c1C(F)(F)F C1(C(=O)NCC(CCC)CCO)C(C2CC2)CCN1C(C1CC(=O)OC1(C)C)=O C(CCOC(C)C)(C1CC1)SC.C1=CC=NC(=O)C2(CC2)N(C)C1=O C1(C(N(CCCC(F)(F)F)C)=O)CN(C(=O)C(C)(C)F)C2(CCC2)C1 N1(C(c2cncc(OC)c2C)=O)CC2CCC1CC2NC(C1CNC(=O)N1)=O C(C)(c1ccco1)=CC(=O)N(CC(=O)NC1C(CSC)C1(C)C)CC C1(C(N(CCC(C)NC(CC(CC)(C)C)=O)C)=O)C2CCC1(C)C2(C)C N1(CCNC(C(c2cc[nH]n2)N(C(c2ccccc2)C)C)=O)CCOCC1C C1(O)(C(C)NC(=O)COC2CCC2)CN(C(=O)Cc2c[nH]nc2O)C1 C(c1cccc(F)c1)=CC(=O)NCC(N(C)C(C1(C(C)(C)C)CCC1)=O)C1CC1 S(=O)(=O)(c1cc(C(=O)NCCC(C)NC)c(C)c(C)c1)NCC C1(CN(C)CC2CC(=O)N(C(c3c[nH]c(=NC)s3)=O)C2)CCCCCCC1 C12(CNC(CC3CC(=C)C3)=O)CC(NC(=O)C(C)n3cccn3)(C1)C2 c1(CC(=O)NCC(c2ccccc2)NC(C(CC)OC)=O)ccc(F)cc1Cl O=C1C=C2CN(c3nnc(C4CC4)s3)CCC2CC1 c1(OCC)ccc(COC(C2(O)CCCCC2)=O)cc1OC c1(CC)cc(C(N2CC3CC3(CNC(=O)C(F)=CCCF)C2)=O)ccc1Cl C(=O)(C(CCS(C)=O)NCc1ccccc1)OCC(CC(C)C)C c1(C(N2CC(C(C)(C)O)(CNC(c3cc(C)[nH]n3)=O)C2)=O)n[nH]c2c1CCC2 C1(C#CC(=O)NC2CC3CC(NC(c4c(Cl)cnn4C)=O)C2C3)(CC)CC1 c1(C(N(CCC2N(C(CC(CC)C)=O)CCCC2)C)=O)cccn2cc(C)nc12 C1(C(N(c2ccccc2)C)=O)CN(C(=O)CCC2CCCOC2)CC12CC2 S(=O)(=O)(c1c[nH]c(=NCCn2ccnn2)cc1C)NC1C(C=C)CCCC1 C(=O)(C1CCc2c[nH]nc21)N1CC2C(Nc3c(C)cnc(C)n3)C2C1 C=CCCCCCC(=O)N1CC(F)CC1C(=O)NC1(CO)CCCCC1 c1(CC)cc(C(=O)NC2CC(CNC(=O)Cc3ncoc3C)C2(C)C)ccc1F n1(CCSC)nnnc1C(c1ccon1)NCCC(c1ccc(C)s1)O C1(CNC(C=CC)=O)COCCN1C(=O)C=Cc1sccc1C N1(C(CN2C(C)CCC2C)=O)CC2CC(C1)N(C(C13CC1C3)=O)C2 N1(C(C#CC2(CC)COC2)=O)CCCC(C2CN(C(=O)Cn3nnc(=O)[nH]3)C2)C1 C(=O)(CC1=CCCCC1)N(C(N1C(C(c2ccc(Cl)cc2)C)CCC1)=O)C C1(C(C(=O)OC)O)CCN(C(=O)NC2CC2(C(C)C)CO)CC1 Cc1nnc2n1CCN(Cc1cn(C3CCC(C(N4CC(F)(F)C4)=O)C3)nn1)C2 C1(CC(=O)NC(C#C)C2CCC2)CCN(Cc2cc[nH]n2)CC1 C(=O)(C(C)(C)CN(C)C(c1cscc1OC)=O)N(C1CCCOC1)CC N1(C(C(F)=C(C)C)=O)CCC2CN(C(C3CCN(S(C)(=O)=O)C3)=O)CC2C1 C1(C(=O)NC(C2CC2(C)C)C)OCCC1NC(C1CC(N(C)C)C1)=O c1(NC2CC(CNC(Cc3ccc(OC)c(O)c3)=O)C2)nccc(S(C)(=O)=O)n1 N1(C(c2c(C)[nH]c(C(F)(F)F)c2)=O)CC(NC(C2(C)CCC(=O)N2)=O)CC(F)C1 c1(C(N(C)CC2(NC(c3cc(Br)co3)=O)CC2)=O)cc2cc[nH]c(=O)c2s1 c1(C(N2CC(O)(CCNC(c3cnc(OC)s3)=O)C2)=O)cc(S(N)(=O)=O)oc1C c1(-c2cc(C(C)NCc3ccc[nH]3)n[nH]2)cccc(C(F)(F)F)c1 Cc1cc(C(=O)NC2CC(CNC(c3ccc(Cl)cn3)=O)C2)ccc1C#N N1(C(c2nn(CC)c(=O)cc2)=O)C(C)C2CC1C2NC(=O)C(C)OCC(C)C c1(C(=O)NC2(C)CCCN(C(c3cccnc3)=O)C2)cc(F)c(F)c(N)c1Cl C1(CN(CCC(=O)NC(C)C2CC2)CC)OCCN(C)C1c1cnn(C)c1 C1(CC(c2nncn2C)OC)(CC(=O)N(C2CCOC2)CCC2CC2)CCCC1 Cc1ccc2c(c1)CCC(C(=O)N(C(CNC(C1CCSCC1)=O)C1CC1)C)O2 C1(NC(c2ccnc(CC(C)C)n2)=O)CCN(C(c2cnc(=N)[nH]c2)=O)CC1C C(=O)(C(C)(C)CN(C)C(c1cn(C(C)C)cn1)=O)N(C)CC1CCCO1 N1(Cc2cn(C(C)C(=O)Nc3ccnc(Br)c3)nn2)CCOCCC1=O C(=O)(C(Cc1ccsc1)NC=O)NCCN.C(=O)(C=CCF)CC C1(NC(C)Cc2cc(F)ccc2F)CN2CCC1(C)C2 C1(NC(CC(=O)N(C)C)=O)CCC2(CN(C(N3CCc4ccccc43)=O)C2)O1 Cc1cc(-c2cn(C3CCC(C(=O)NC(Cc4nccs4)C(=O)O)C3)nn2)cnn1 C(=O)(C1(C)OCCc2ccccc21)N1CC(CCCC)N(C(=O)COCC)CC1 C1(C(N(C)CC2CCCN2C(=O)C=CC2CCCC2)=O)OCC2COCCC12 c1(C(N2CCCC(N(C(CNC(=O)OCC)=O)C)C2)=O)cc(C(N)=O)ccc1F N1(C(COC(CC)C)=O)CC2(CC(NC(C3(F)CCCCCC3)=O)C2)C1 c1(OC)ccc(F)c(C(=O)NCC#CCNC(c2ncc3n2CCCC3)=O)c1F N1(C(c2cc(C)oc2C)=O)CC2CC(NC(c3ccc(C(F)F)cn3)=O)CC1C2 C1(c2cn(CC(=O)N(CC(C)NC(C)=O)CC)nn2)CCC(F)(F)CC1 C1(NC(CCC2(C)CC2)=O)CN(C(c2cccs2)=O)C2(CCCOC2)C1 c1(C(=O)NC2(C(N3CCCC(N(C)C(N)=O)C3)=O)CC2)cnn2c1CCC2 CC(C)CC(C)(CNC(C1CCCCC1(F)F)=O)NC(=O)Cn1ccnn1 c1(NC(c2n(CCCC)nnn2)c2cnn(C(F)F)c2)ccc(Br)nc1 CN1CCN(CC(=O)NCC(CC2CC2)C(=O)NC2(C(N)=O)CCC2)CC1 c1(C(=O)NCCOC2CCN(C(C3C(C)(CC)C3)=O)C2)n[nH]c(C)c1Br c1(C(=O)NCC2(Cc3ccccc3)CCCO2)ncc2c(n1)CCCCC2 C1(CNC(CCCNC(C)=O)=O)CCN(C(=O)Cc2nc(C)cs2)CC1O c1(OCC)ccc(C(C(=O)NCC2CC2)N(C2CCCN2C)C)cc1 CCC(C)(C)CCCC(=O)N1CCSCC1C(=O)N1OC2CCC1CC2 C1(CNC(c2c(C)cno2)=O)CN(C(=O)Cc2cccc(Cl)c2F)C(C)(C)C1 S(=O)(=O)(c1ccccc1)NC(C(=O)NCCNC(C(CC)(CO)OC)=O)C(C)O N1(C2CN(C(C(C3CN(C(CCc4nc(C)sc4)=O)C3)O)=O)C2)CC(C)OC1=O C1(C(N2C(CC=C)(C(=O)NCCc3cnn[nH]3)CCC2)=O)CCCCC1(F)F C1(C(=O)NC(COC)(C)CCO)(CF)CCN(C(=O)CCC(C)OC)C1 c1(SCC2(CC(=O)NCC(=O)NCc3ccco3)CCC2)c(F)cccc1F C12(C=O)CCC(Cn3cc(C)nn3)(CC1)CC2=O.C1(Cc2nn[nH]n2)CCCN1C N1(C(C2(C)CCCS2)=O)CCN(C(=O)COc2ccc(F)c(F)c2)C2(CC2)C1 C(C)(CN=c1cc[nH]cc1S(=O)(=O)N(C)C)NCCc1c(C)cc(C)n(C)c1=O CCN(CCCF)N1CC(c2cccc(Br)c2)C1 C(=O)(C1CCc2cccnc21)NCC1C(NC(c2c(OCC)ccs2)=O)CCC1 C1(SCC(=O)NCC)CC2CCC1C2.n12cc(nn1)CN(C)C(=O)CC2 Cc1ncn(C)c1C(=O)NC1CCCN(C(c2cc(Cl)sc2Cl)=O)C1 C1(NC(C(CCOC)C)=O)COC2C(NC(c3nc(C)nn3C)=O)COC12 c1(C(C(=O)N(CC(C)NC(c2ccccc2)=O)CC)(F)F)cccc(Cl)c1 C1(C(=O)OC2CN(C(=O)OC(C)C)C2)CCc2nncn2C1 c1(C(N2C(CNC(C=C(C)Cl)=O)C(C)CCC2)=O)ncnc2[nH]cnc12 c1(OC)nc(C(=O)NCC2C3CN(C(c4cccn(O)c4=O)=O)CC23)cc(O)n1 N1(C(c2ccc(OC)c(OC)c2Cl)=O)CCC2(CC1)CC2(C)C(=O)NC(C)CO N1(C(CCOCCCOC)=O)CCC(F)(CNC(c2cn(C)nc2C(C)C)=O)C1 c1(C(=O)NC2C3CN(C(C(c4c(C)cccc4)C)=O)C2C3)n[nH]c2c1CCOC2 c1(C(=O)NC2C(C)CCN(C(C3(C)CCCO3)=O)C2)cc2nc(=O)ccn2[nH]1 N1(C(CC(CC)C)=O)CCOC(C(=O)NCCN=S(C)(C)=O)CC1 c1(C(N2CC(NC(C3(C)CC(=C)C3)=O)CC23CCC3)=O)n[nH]c2c1CCCCC2 C1(OC)C(NC(C2(NC(=O)CCN3CCCC3)CCOCC2)=O)CC12CCC2 N(C1C(=O)Nc2ccc(C)cc21)C(c1ccc(OC)cc1F)=O C(=O)(C(C)(C)C#N)N1CCC(N(C(C=CCCC(C)C)=O)C)C1 N(C(=NCc1ccc(CO)cc1)N1CCC(O)C1)CC(N1CCN(C)CC1)C c1(C(=O)NC(C)CNC(=O)C(O)C(C)(C)C)ccc(S(C)=O)cc1 c1(C(N(CCOC)CCN(C)C)=O)cc(-c2ccccc2OC)c2n[nH]cc2c1 Cc1cnc(S(C)(=O)=O)nc1N1CCC(F)C(NC(c2ccc(Br)c(Cl)c2)=O)C1 CC(C)CC(C(=O)NC1CCCN(C)C1)NC(c1cc(Cl)c[nH]1)=O C#Cc1cccc(OCC(N2CCC3C(NC(C4CCOC(C)(C)C4)=O)C23)=O)c1 Cc1ccc(C(=O)NCC(F)CNC(=O)C(c2ccccc2C)(C)C)nn1 c1(C2(C(C=CC(=O)NCC(F)(F)F)=O)CC2c2ccccn2)ccc(Cl)cc1 C1(C(=O)Nc2cncc(C(N)=O)c2)CC(F)(F)CN1Cc1cnccc1C#N C1(C(=O)NCc2cc(C)no2)COCCN(C(=O)CCCC2CCCCC2)C1 C1(F)(CNC(C2C(C)(C)C2)=O)CN(C(C2(C(N)=O)CC2)=O)C1 C=C(C)CC(C(=O)NC1CC(OCC(=O)Nc2cnc(F)c(C)c2)C1)N(C)C C1(C(=O)N(CCO)C2CNC2=O)COc2ccc(Cl)cc2C1=O C1(C(=O)NC(C#C)C2CCC2)CC(O)CN1C(=O)CCCN1CCCC1 N1(C(C2(NC(c3cn(C4CC4)nn3)=O)CC(F)C2)=O)CC2CC1C1CC21 C1(CNC(CCCCC=C)=O)CC2(CCOCC2)CN1C(c1c[nH]c(=NC)s1)=O Cc1[nH]c(=N)ccc1C=CC(=O)NCC(C)NC(c1ccccc1Br)=O c1(OC)nc(C)ccc1C(N1CC2(CC(NC(=O)CN3CCCC3=O)C2)C1)=O C1(NC(CC2CN(C)C2)=O)CN(C(c2sccc2OC(F)F)=O)CC1(C)C N1(C(CC(C)CN(C)C)=O)CCC2(CCC(NC(=O)CC(O)CN(C)C)C2)C1 c1(CN2CCC(N(C(=O)Cc3c(Cl)ccc(O)c3Cl)C)C2)ccc2c(c1)CCO2 c1(NC(C2(CNC(=O)C(F)C(C)(C)O)CC2)C)ccc(Cl)cc1[N+](=O)[O-] CC(C)(C)C#CC(=O)N1CC2(CCC2CNC(c2ncn3c2CCC3)=O)C1 N1(C(c2c(C)c[nH]n2)=O)CC(C2CCN(C(c3cc(Cl)c[nH]3)=O)CC2)OCC1C C(CN=c1[nH]c2c(c(=NCC(Cl)(Cl)Cl)[nH]1)SCC2)c1cnc(C(C)C)[nH]1 N#CC1CC(C(N2CCC2CNC(C2CC(O)C2)=O)=O)C1 c1(C(N2CCC(CNC(C(C)OCCOCC)=O)C2)=O)nn(C)c(=O)cc1C n1(CC)nc(C(=O)NCC2CCCN2C(=O)C(N2CCOC2=O)C)ccc1=O C12(NC(CC(C)(C)N(C)C)=O)CCOC(CNC(c3ccoc3Cl)=O)(C1)C2 c1(C(N2CCC(N(C(C3CC(C)C3(C)C)=O)C)CC2)=O)cc(S(N)(=O)=O)ccn1 C(=O)(C#CC1(CC)CC1)NCCCOCCNC(C(C(C)C)SC)=O c1(C(N2C3CC(CNC(C=CCC)=O)C2CC3)=O)ccc2c(c1)CCCCN2 C1(C(=O)NCCC2(CC)CC2)CCC2(CN(C(c3cc4scc(C)c4[nH]3)=O)C2)O1 C1(NC(c2ccc(C#C)cc2)=O)C2COCC1CN(C(=O)C(=O)NC1CC1)C2 C(=O)(C1=NN(C)C(=O)CC1)NC(C(=O)NCC(CC)(C)CO)C(C)(C)O O=C1CCC(C(N2CCN(C3CCCN(C(=O)CSC(F)F)C3)CC2)=O)CCO1 C1(C(N2CCC3(CC3C(=O)NCC34CCC(CO3)C4)C2)=O)CN2CCC1CC2 Cc1noc(C2CC2)c1NC(=O)C(C1CCN(C(c2ccc(F)cc2)=O)C1)F O=C(C(CO)c1ccccc1)NCCCN(C(C1CCCOC1)=O)CC1CC1 C(=O)(CC(=O)NC(CC1CC(N(C)C)C1)=O)NCC1(N(C2CC2)CC)CCC1 C1(C)(CC)CC(NC(C)=O)CN1C(=O)Nc1ccc(CC(C)(F)F)cc1 N1(C(C(C)CN(C(=O)Cn2ncn(C)c2=O)C)=O)CC2CCC(C1)N2C C(=O)(C1=C(C)NC2=NCCCC2=C1)NCCN(C(C(CC)OC)=O)C1CC1 O=C1C=C2CN(C(C3CCCC(NCc4ccccn4)C3)=O)CCC2S1 c1(C(C(=O)NC2(C)CN(C(COCCSC)=O)C2)C2CC2)ccc(O)cc1 C1(NC(c2nc(C)sc2C)=O)CC(F)CN(C(C2CCS(=O)CC2)=O)C1 C=CCCCN=C(NCC(=O)NCCF)N1CCC(CNC(N)=O)C1 C(=O)(C(C)(C)C(=O)NCCC1CCCCN1C(=O)Cn1ccccc1=O)OC c1(OC)ccc(Br)c(CN2CC(CNC(=O)Cn3nc(C)cc3C(F)(F)F)C2)n1 CC(C)(CO)C(=O)NCCCOC1CN(C(=O)CN(C2CCC2)C2CC2)C1 C(CC(=O)N(CC(CC)NC(=O)C(C)c1ncco1)C)N(CCC)C Cc1nccc(Cl)c1C(=O)NCC(C1(O)CCN(C(C2(O)CC(C)(C)C2)=O)C1)C N1(C(c2ccc(C(=O)NC)nc2)=O)CC(OC)CC(NC(=O)C#CC2(C)CC2)C1 C1(NC(C(CC(C)C)C)=O)C(C)(C)CN(C(=O)CCC(CF)CF)CC1(C)C c1(OC)c(C(=O)NC(C)Cc2cccc(O)c2)ccc2ccccc12 C1(CC(=O)NC2C(CCC)C2)CCCN(C(=O)C(C)CC)C1 C=C(C)CC(C(=O)NCC(C)(C)C(=O)OC)NC(C1CC(CC)C1)=O N1(C(COCc2nnc(C)s2)=O)CCN(C(=O)C2=NNC(C(F)(F)F)C2)CC1C N1(C(C(C)C(F)(F)F)C(=O)NC)CCn2c(cnc2C)C1 Cc1n[nH]c(C)c1CC(=O)NC1CCCC(N(C)C(C2CCC3CC23)=O)C1 C(=O)(C1CSc2ccccc21)N1CCCC2(CN(C(Cc3n(C)cnc3)=O)C2)C1 C(=O)(C(C)CCCOC)N1CCCC(N(C(Cc2ccc(CC)cc2)=O)CC)C1 CN1C(=O)CCCC1C(=O)NCC(C1CCC1)NC(c1csc(C(N)=O)n1)=O c1(C(=O)NCC2CC(NC(CC(COC)C)=O)C2)cn2c(n1)COCC2 Clc1cc(Br)c2ncnc(NC3CNC4CCCOC34)c2c1 C(=O)(C1=CNS(=O)(=O)N=C1C)N1CCN(C(C(CCC)C(=O)OC)=O)CC1C c1(C(N2CCN(C(C(OC)OC)=O)C(C(F)(F)F)C2)=O)ccc2nn[nH]c2c1 C1(CC(=O)NC(CNC(c2c(C)n(C)nc2)=O)CO)CCCC2(CC2)C1 Cc1nc2sccn2c1C(N1CCC(NC(=O)C(C)c2cccs2)C(O)C1)=O C1(C(=O)NC(C(=O)NC(C)CSC(F)F)c2ccco2)CCCC(CF)C1 N12CCC(CC1)C2.C1(Nc2ccnc(C(C)C)n2)CC(CC#N)C1(C)C C1(NC(CCNC(C)=O)=O)CN(C(=O)CC#N)CC1F N1(C(C2CCN(C)C(=O)C2)=O)CCN(C(=O)CC2(C)CC2)CC(O)C1 N1(C(c2ccc(C)[nH]2)=O)CCCC2CN(C(=O)CCNC(C3CCCO3)=O)CCC12 C(=O)(C(Cc1ccoc1)NC(=O)CC(=O)NC1CC1)NCC(CC)N1CCCC1 N1(C(C(CC)(C)C#N)=O)CCC2(CC(NC(C3CC3c3cnn(C)c3)=O)C2)C1 C1(NC(CCCOCC)=O)CC2CCC1CN(C(c1cc(Cl)ccn1)=O)C2 N1(C(=O)CSC(F)F)CCCCC(C(N2CCC(c3ccco3)C2)=O)C1 c1(C(=O)NC(C(C)NC(c2cc(C)nn2C)=O)C)c(Cl)c(Cl)cc(Cl)c1Cl c1(CSCC(=O)N(C(C)CNC(c2cocn2)=O)CC)ccccc1 C(=O)(N1OC2CCC1C(O)C2O)C1CN(C(=O)OC(C)(C)C)CC(F)C1 C1(c2cc(C)no2)CCCCN1C(c1csc(NC(c2ccccc2Cl)=O)n1)=O N1(C(CCC#C)=O)CCCC(NC(=O)CSCc2cccc(C)c2)C(F)C1 C1(C(=O)Nc2cnc(OC)nc2)(NC(c2c(OC)cccc2)=O)CCC(C)(C)C1 C(=O)(C1=CC2CCC(C1)C2)N1CC(C)CC(C(=O)NC(CC)(C)C(N)=O)C1 c1(OCC)cccc(NC2CCN(C(C3CN(C)C(=O)N3)=O)C2)c1[N+](=O)[O-] Cc1c(C(N2CC(O)CC2C(=O)NCc2ccc(I)cc2)=O)cccc1[N+](=O)[O-] CCC(C(=O)N1CC2(CCCC2NC(c2cc(C3CC3)[nH]n2)=O)C1)C(F)(F)F C#CC1CCCN1C(=O)CCCNC(=O)CC(C)(F)F C(=O)(C1=COCCC1)NC(C)CNC(=O)C(C)(Cl)Cl N1(C(CCOCCC)=O)CCC(C2CC2)(CNC(=O)C(O)C(F)(F)F)C1 C1(C(C)(O)CNC(C2CC3C=CC2C3)=O)CCN(C(c2n[nH]cc2Cl)=O)CC1 c1(C(N2CCC(C(=O)OC)(CO)C2)C(=O)NCC(=C)C)c([N+](=O)[O-])ccc(Cl)c1Cl N1(c2n(CC(=C)C)c(-c3ccccc3)nn2)CCOC(C)CC1 O=C(CC(C(F)F)N1CCOCC1)NCC1CC(NC(C2(O)CCC2)=O)C1 N1(C(CCC2CCN(C(C(CNC(C)=O)(C)C)=O)C2)=O)CCCCC(F)(F)C1 c1(CC)cc(C)ccc1C(=O)NC1(CCNC(=O)COCCCF)CCC1 C(=O)(CC(C(C)C)c1ccccc1)NC1C(NC(C(CO)OC)=O)C1 C(=O)(CC(C(F)F)N(C)C)N(C(CO)C(=O)NC(C)(C)CC1CCOC1)C C#CC1(O)CCCN(C(=O)C(CCCC=C)NC(=O)C(C)CO)C1 C(=O)(C1=CC2CCC1C2)N(CCCCN(C(C(C)Oc1cccc(C)c1)=O)C)C c1(CC)cnc(Cl)[nH]c1=NC1CC2CC(C1)N(C(c1cn3c(n1)CCCC3)=O)C2 CC(CC(F)(F)F)C(=O)N(C(C)CN(C(=O)C(C)(C)c1cccs1)C)C c1(C(C)C(=O)N(CCCn2cc(-c3ccccc3I)nn2)C)ccc(F)cc1 c1(C(=O)NCCC2N(C(CC(CC)C)=O)CC(F)(F)C2)c(C)nc2cccnn12 N1(CC(=O)N(C)C)CCNC(=O)C1C(C)(C)C.n12cc(nn1)C1CC1NC(=O)C2 C(CN=c1[nH]cnc2cc(F)c(F)cc12)C1CN(CC2(C)CCN(C(C)=O)C2)C1 c1(C(N2C3C(NC(CC4CC(=C)C4)=O)CC(C3)C2)=O)n[nH]c2c1CCSC2 C1(NC(CCn2ccc(C)n2)=O)CN(Cc2ncc(C)s2)CC1O C=C1CC2(C1)CC(C(=O)NC1CCN(C(=O)C(C)Sc3nncn3C)C1C)C2 C1(C(=O)NCc2c(C(=O)NCC(C)C#N)nco2)CNC(=O)CC1C N1(C(CCCCC#C)=O)CC2(CCCC(CNC(=O)CC3COCCO3)O2)C1 C1(C(=O)NC2CC(C)N(C(C3C4COCC34)=O)CC2)CCc2ncn(C)c2C1 C1(CNC(c2ccon2)=O)CCC2(CCC2)CN1C(=O)Cn1cnnc1O N1(C(c2ccnc(C(C)C)n2)=O)CCC(NC(C2CCCS2)=O)C(O)C1 N1(C(c2c(OC)scc2)=O)CCC2CC2(C(=O)NCC2(S(C)=O)CC2)CC1 Cc1ccnn1CC(N1CCC(C(C)C(=O)NCC2(O)CCSC2)C1)=O CCCCC(CC)CC(=O)N1CC2CC(NC(c3ccc(Cl)nc3F)=O)CC2C1 CC1CN(C(c2cc(Cc3cccs3)on2)=O)CCN1C(=O)Cc1cncnc1 CCC(C(=O)NCC1CCCN1C(=O)CCc1nccn1C)C(C)O N1(C(Cc2cc(C)no2)=O)CCN(C(C2CC2C2CCCC2)=O)C(C)C1 C(=O)(C(CO)C(C)(C)C)NCC(CC)(CC)NC(=O)CCC(=O)c1ccccn1 N1(C(C(N)=O)=O)CCOCC2(COCCN2C(=O)CCc2cncc(F)c2)C1 C(=O)(C(C1CN(C(=O)Cn2cccn2)C1)N(C)C)N(C(CC)C)C C(C(=O)NC(CO)CCOCc1ccccc1)(C(C)C)n1c(C)nnc1 C1(NC(CN(CCOC)C)=O)CN(C(C2CCCC(=O)N2)=O)CC1S(C)(=O)=O C1(F)(C(N(C2CCCCC2O)C)=O)CCCN(C(C2CCCC2F)=O)C1 c1(OC)cc(C)cc(C(=O)NC(C)CNC(c2c[nH]nc2-c2ccoc2)=O)c1O N1(C(C(CC2CC2)OC)=O)CCN(C(C2CCCC2C(C)C)=O)C(CO)C1 c1(C(=O)NCC2OCCC(NC(C(C)SC(C)C)=O)C2)cccc2c1OCCN2 CCC(C)CCCC(=O)N1CCC(C2CC2)C1C(=O)N(C1CCCC1C)CC CC1CC(C(=O)NCCC(=O)OC(C)(C)C)CN(C(c2ccc[nH]2)=O)C1 C12(C(=O)NC(C(CO)NC(c3ccc(C(=O)OC)cc3)=O)C)CC3CC1C2C3O N1(C(C2OCCN(C(c3c(C)c(C#N)[nH]c3)=O)C2)=O)CCCC2(C=CCO2)C1 c1(C(N2C(CNC(C(CC)OCC)=O)C=CC2)=O)cc(OC)ccn1 C(c1cc(F)cc(F)c1)=CC(=O)Nc1nc(-c2ccc(OC)c(F)c2)sc1C c1(C(N2CCN(C(c3c(OC)nsc3OC)=O)CC2)=O)occ2c1CCC2 N1(C(C2CC(CC)C2)=O)CCN(C(=O)CCCN2CCCC2)CC1CCOC C=CCC(C)(C)CC(=O)NC(Cc1ccco1)C(=O)NOCC(=O)N(C)C c1(OC)nc(C(=O)NCCN(C(C2CCC(O)CC2)=O)C2CC2)cc(O)n1 Cc1cc(CNC(=O)C=CC2CCC2)oc1C(=O)NC1(C)CSC1 C1(c2ccccc2)(CC(=O)NCCC2CC(NC(C(C)C#N)=O)C2)CS(=O)(=O)C1 Cc1csc(C(=O)NCCC2CCN(C(C3CCN3C)=O)C2)c1Cl C(C(CC(=O)NOCCCO)C1CC1)NC(=O)OCC(F)(F)C(F)F S(=O)(=O)(c1[nH]c(=NCC2CC23CC3)ccc1Br)c1n(C2CCS(=O)(=O)C2)ncc1 C1(C)(CNC(c2c(OC)nsc2)=O)CCN(C(C2CC(N3CC(O)C3)C2)=O)C1 c1(N(C)C)ncccc1C(=O)NCCn1ccc(C(=O)NC2CC(O)C2)c1 c1(C(=O)NCCOC2CN(C(c3c(C)ncs3)=O)C2)ccc(P(C)(C)=O)o1 c1(C(=O)NCc2cc(C(=O)NCc3nc(C#N)sc3)on2)cnn2ccccc12 c1(C(N2CC(N(C(CC(CC)C)=O)C)C2)=O)ccc(OC)c(OC)c1Cl CC(C)C(F)(F)CN=c1[nH]c(N(CCCS(N)(=O)=O)C)nc2cc[nH]c12 C1(OC)CN(C(=O)C(=O)Nc2cn(C)nc2C2CCCO2)CC1n1ccnn1 Cc1cc(C(N2CCCC2c2ccnn2C(C)C)=O)c(N)c(Cl)c1 N1(C(CC2CC(=C)C2)=O)CC(NC(C2CCN2C(C)(C)C)=O)C(C)(C)C1 CC(C)C(C)CC(=O)NCCC(C)CCNC(c1cccc(C2COC2)c1)=O Cc1nc(C(=O)N(CC(=O)NC2CNC(=O)C23CC3)C)c(=O)[nH]c1C N=c1[nH]cc(C(N2CCOCC2c2nc[nH]n2)=O)c2occc12 C1(CCNC(C)=O)(NC(C(SC)SC)=O)CCN(C(=O)CCCn2ccnc2)C1 C1(CC=C)(C(=O)NC2CC(C)N(C(=O)OC(C)(C)C)C2)CCOCC1 N1(CC(=O)NCCCN(C(C)C)C(c2ccc(O)cn2)=O)CCC(N(C)C)CC1 CC(C)C(C)C(C)CC(=O)N1CCC(CNC(=O)CN2CCC(C)CC2)C1(C)C C1(C)(C(N(CCC(C(C)C)NC(c2ccc(CC)nc2)=O)C)=O)CC2C=CC1C2 C1(C(=O)NC(C)CN(C)C(C2CCCCC2n2cccn2)=O)CC2CCC(C1)S2 C1(CNC(C=COCC)=O)CCN(C(C2CC2c2ccc(Br)cc2)=O)CC1 c1(C(N2CC(CN(C(c3nccc(C)c3)=O)C)C2)=O)ccc2c(c1)CNC2=O C(C)(C(CC(=O)NC1CCOCC1C)NC(=O)CC1CNC(=O)O1)OC CCCS(=O)(=O)NCC(=O)NC1CC(C)(NC(c2cnn[nH]2)=O)C1 c1(C(=O)NCC2(OC)CN(C(c3ccnc(F)c3Cl)=O)C2)cnc2cccnn12 N1(C(C2(C)CC(=C)C2)=O)CCOC(C)(CNC(c2cncc(F)c2Cl)=O)C1 N1(CC(=O)NC(CN(C(=O)C=CC(C)(C)C)C)(C)C)CCCS1(=O)=O Cc1cc(C#N)sc1C(N1CCOCCC1CO)C(=O)Nc1ccc(F)cc1 CCS(=O)(=O)CC(=O)NCC1CC2CCC1N2C(=O)C(C)(O)c1ccccc1 N1(C(C)CN(C)C(C23CC(CO)(C2)C3)=O)CC(NC(=O)C(C)C2CC2)CC1=O c12cc3ccccc3n1c2=O.c1(OC)c[nH]nc1C(=O)NCC1(CCC)CC1.C1(S)CC1 Cc1ccc(F)c(C(=O)NCC2CN(C(C3C(C)CC3C)=O)C2)c1F c1(C(=O)NC2CC(c3ccc(Cl)cc3)C2)ccc(-n2cccn2)nc1 CN1CCCC(CC(=O)NCC2C=CC(NC(=O)CC(F)(F)Cl)C2)C1 c1(C(=O)NCC2(F)CC(NC(C3CCC(C)C3)=O)C2)ccnc(P(C)(C)=O)c1 C(=O)(CCC(F)(F)F)NC1CN(C(c2cccc(C(N(C)C)=O)c2)=O)CC1O C(C)(CC(=O)NC(CCO)C1CC1)N(c1ccccc1)C(C)=O N1(C(COC2CC(n3cc(C(CC(C)C)(C)C)nn3)C2)=O)CCN(C)CC(O)C1 C1(NC(c2n(C)ncc2)=O)CC(=O)N(C2CN(C(=O)Cc3nc(=N)[nH][nH]3)C2)C1 C1(C(N2CC(O)(CCNC(c3c(C)ncs3)=O)C2)=O)CS(=O)(=O)CCO1 N1(C(CC=CC=C)=O)C2CCC1CC(NC(C1Cc3ccccc3S1)=O)C2 N1(C(C=COCC)=O)CC(C)CN(C(c2cncc3c(Cl)cccc23)=O)C(C)C1 N1(C(C2(CC)COC2)=O)CCc2nc(CNC(C3CC(=O)N(C)C3)=O)sc2C1 N1(C(C(C)SC)=O)CCC(F)(C(=O)NCc2cccnc2OC2CCCC2)C1 N1(C(c2cc(C)n(C)n2)=O)CCCN(C(=O)CCn2cccc2)CC1C CS(=O)(=O)CCC(=O)N1CCC(NC(=O)NCCCl)C(C(F)(F)F)C1 C1(CCN(C(C(CC)NC(N)=O)=O)CC)CCCCN1C(=O)C(CC)n1ccnc1 N1(CC(COCC)O)CCN(C(=O)NCc2cccc(Cl)c2F)C(C)(C)C1 Cc1nc(CC(=O)Nc2cn(CC(=O)NC(C)(C)C)nn2)oc1-c1ccccc1 N1(C(C(C)OCC)=O)CCOCC1CCNC(c1cc(-c2csc(C)n2)c[nH]1)=O C(C(=O)NC(c1ccccc1)CNC(c1cnccc1Br)=O)(C(C)C)OC Cc1nc(NCC2CCCN(CC(C)C)C2)cc(=NC(C)c2nnc(CO)s2)[nH]1 c1(CC(N2C3CCN(C(C4CC(OC)C4)=O)C(C3)C2)=O)cccc2ccncc12 c1(C(=O)NC(CNC(Cn2ccc(C)n2)=O)C)ccc(F)c(C(=O)NCCC)c1 CCC(C)C(C(=O)NCCCC(C)NC(C1(n2cc(Cl)cn2)CC1)=O)NC(C)=O c1(SC)nnc(SCC(N2CCCC(N)C2)=O)n1CC(C)C C1(C(=O)NCC2(NC(CSCCCC)=O)CCOCC2)CC2CC(=O)C1C2 N1(C(c2c(C)cccc2O)=O)CCCC(C2CCN(C(=O)CO)C2)C1 c1(C(N2CC(C)CC(NC(Cc3cnc(C)[nH]3)=O)C2)=O)oc2ccccc2c1C CCC(CC(C)C)C(=O)N1CCN(C2CN(C(C3CCC(F)(F)CO3)=O)C2)CC1 N1(C(c2c(C)nc(C)n2O)=O)CC2CCCC(C1)N2C(=O)C(=O)N=S(C)(C)=O C(C(C(C)C(C)C)NC(C1CCC1C#N)=O)NC(CCC(=O)NC)=O c1(C(=O)NC2C3(CCN(C(C4C(C)CN(C)C4)=O)CC3)C2)ccc2nc[nH]c2c1 C12(C(=O)OC)CCC(C1)OC21CN(C(c2cnc(C(F)(F)F)o2)=O)C1 C1(C(N2CC(CC=C)(C(=O)Nc3cnc(SC)nc3)C2)=O)CCOC2(CCC2)C1 CN=c1cc(C(N2CCCC(C(=O)NCCc3cc(C)no3)CC2)=O)cc[nH]1 N1(C(CCC#C)=O)CC2CCC2(CCNC(c2c(C)noc2N)=O)C1 Cc1cc(Cl)ccc1CN(C(c1cnn(CCO)c1)c1nnnn1C1CCC1)C c1(-c2nc(CC(CC)C)nn2CC)ccc(=O)n(CC2CCC2)c1 c1(C(=O)NC2C(NC(C3(CC)CC3(F)F)=O)CC2)ccccc1OCCCC#N c1(Oc2c(C(N3CCC(C(=O)OC)CC3)=O)nccn2)cc(F)c(CO)c(F)c1 C1(CCC)CCC(C(=O)NC2CCCCC2NC(=O)C(C)C(=O)OC)CC1 N1(CC=CC)CCC(N=c2nc(N3CCC4(CC3)CC4CO)c3c([nH]2)CCOC3)C1 CCC(CC)CC(F)C(=O)N1CCC(C)C(CC(=O)NC2CC3CCC2O3)C1 C1(C(N)=O)CC12CN(C(C1(NC(=O)CCCn3ccnc3)CCC1)=O)C2 N1(c2ccnc(C)n2)CC2CC(NC(c3ccc(C4CC4)nc3O)=O)CC2C1 C(=O)(C1=CC2(CCOC2)C1)N1C2C(C(N3C(CN(C)C)CCCC3)=O)C(C2)C1 c1(C(=O)NCc2cccc(NC(CCC#C)=O)c2)c[nH]cc(C)c1=O C1(C)(C(=O)NCC2(CNC(C3(C)N(C)CCC3)=O)CC2)CCCNC1=O N1(C(c2ccc(F)c(C)c2C)=O)CCC2(CC1)CC(NC(c1cc[nH]n1)=O)CO2 C=CCC(CC=C)C(=O)NC1CC(O)CN(C(=O)Cc2csc3nccn23)C1 Cc1cnc(C(=O)NC(CNC(c2scnc2C(C)C)=O)C2CC2)cc1Br N1(C(C2CCN(C(C)=O)C2)=O)CCOC(CN(C(=O)CCCN(C)C)C)C1 c1(C(C)=O)cc(C(N2CCC(C3CCCN3C(=O)CSC)C2)=O)[nH]n1 CC1CCc2nc(C(N3CCCN(C(=O)Cn4cc(Cl)cn4)CC3)=O)ccc2C1 c1(CS(=O)(=O)NC2C(C)CN(C(C)(C)C)C2)ccc([N+](=O)[O-])cc1 CC1(O)CCCC1NC(=O)CN(C1CCC1)C(c1cncc(CO)c1)=O N1(C(c2c(C)n[nH]c2C)=O)CC23CCCC2(C1)CN(C(c1cnccc1F)=O)C3 c1(CN2Cc3c(-c4c(C)onc4)n[nH]c3C2)ccc(S(=O)(=O)C2CC2)cc1 C1(CC)(NC(=O)CNC(c2cccc(C)c2)=O)CCCN(C(=O)C=C(C)C)C1 C=C(Cl)C(C)(C)C(=O)N1CC(O)(CCNC(c2sc(C(C)C)nc2C)=O)C1 Cc1nnc(C(C)N)s1.c1(C(CCCOCC)C2CC2)nnnn1C(C)C c1(C(N(C2CCCCC2)CCNC(C2(C)CCCC2)=O)=O)cn2cccc(F)c2n1 Cc1nc(CC(=O)N(C(C)(C)C2CC2)C)n[nH]1.C(CS(N)(=O)=O)N CCCCCCC(=O)NC1(C(=O)N(C2CCC(O)CC2)CC)CC1 c1(N(CC(F)C2CCC2)C)nc(N2CCC(c3nc[nH]n3)C2)nc2c1CSC2 N(C(=NCCCSC)NCC1(C2CCC2)CCC1)C(CC)C(F)F C1(C(=O)NCC2(O)CN(C(C(CC)OCC)=O)C2)CCc2ncccc2C1 C(=O)(CCCCCC(C)C)NC(CC(C)NCc1c(Cl)cccc1[N+](=O)[O-])C N1(C(C2(N(C)CC)CC2)=O)CCC2(C=C(C(=O)N(C3CCC3)C3CC3)C2)C1 N1(C(=O)NCCn2ccccc2=O)CCc2cc(F)ccc2C1 c1(C2C(N(CCN3CCC(NC(COC)=O)C3)C)C2)cccc(C#N)c1 N1(C(=O)Nc2sc(C(=O)OC)c(C)c2)Cc2nc(Br)sc2C1 C(=O)(C(CC)C(=O)NC(C1(CNC(c2cc(Cl)ccc2C)=O)CC1)C)OCC c1(C(=O)NCC(N(C)C(C2CCCC2)=O)C2CC2)ccc2c(c1)C(=O)NCC2 c1(C(N(C(CCCC)C)C)=O)ccc(-c2ccccc2)c(Cl)c1 CSC1=C(C(=O)N=c2ccn(CC3CCCO3)[nH]2)CCCC1 C(=O)(C(C)(C)C(C)(C)C)NCC(C)(CC(C)C)NC(Cc1ccc(C#C)cc1)=O C1(NC(C2(OC)CCOC2)=O)CN(C(=O)CN(c2ccccc2)C)CC1OC N1(CC(C2CCOC(C(C)(C)C)C2)(C)C)CCOC(CS(N)(=O)=O)C1 c1(CNC(=O)NC2C(C(=O)OCC)C3CCC2C3)cccc2ccc(Cl)cc12 c1(CC(C(=O)N(C2CN(C(=O)CC3COC(=O)C3)C2)C)NC=O)ccc(F)cc1 C(=O)(C(O)P(C)(C)=O)NCC(N(C(CCc1ccc(N(C)C)cc1)=O)C)C1CC1 c1(C(N(CCNC(=O)C(C)N(CC(F)(F)F)C)CC)=O)cnn(CCO)c1C C#Cc1cccc(CC(=O)NC(C2CC2C(=O)NC2CNC(=O)C23CC3)C)c1 C(=O)(C(C)(C)C(C)(F)F)NCc1c(CN(C(C2CCN(C)CC2)=O)CC)nco1 Cc1ccc(=N)[nH]c1C(=O)NCC1CN(C(c2n[nH]cc2C)=O)C1 C12COC(C1)NC2.c1(C(=O)NCC2(CC(=O)OC)CC2)coc(-c2cc[nH]n2)c1 C1(CCNC(=O)CC(Cl)Cl)CSCCN1C(c1cc(C2CC2)on1)=O N1(C(C(c2scc(C)n2)C)=O)CCN(C(C2COC(=O)N2)=O)CC1C(C)(C)C C1(O)(C(=O)OC)CCCN(C(=O)C(C2CCC(NC(=O)Cc3ccoc3)CC2)C)C1 C1(NC(=O)CCC2CCC2)CN(C(=O)Cn2cc(CO)nn2)CC12CC2 C(=O)(CCC(=O)NC(c1ccc(NC)cc1)=O)N1CC2C(N(C(=O)CO)C)C2C1 C1(NC(c2ccnc(Cl)c2)=O)CCC2CCN(C(C3(CO)CCC3)=O)C1C2 c1(C(=O)NC2C(NC(CCCN=[N+]=[N-])=O)CCCCC2)csc2ccc(F)cc12 c1(N2C(C)CCC(NC(C3CCC(=O)N3C)=O)C2)ncc2cccnc2n1 N1(C(CSCCC)=O)CCN(C(=O)CSCC(F)F)CC1C1CC1 c1(C(N(C2CCC(NC(C(C)=CC)=O)CC2)C)=O)ccc(OC)c(Br)c1 N1(CC)CCCCC1C(=O)NCC1(F)CC(NC(=O)CSc2cn[nH]c2)C1 c1(C(N(C2CN(C(=O)CN(S(C)(=O)=O)C)C2)C)=O)ccc2c(c1)CCC2 c1(OCC)cccc(C(=O)N(CC(O)CN(C)C(c2cc(C)n(C)c2)=O)C)c1F c1(COC)ccc(C(=O)NCCCOCCN(C(=O)Cc2ccn(C)n2)C)s1.NCO c1(C(=O)OC)cc(N2CCC(C)(NC(=O)C=CC3CCCO3)C2)nc(SC)n1 N1(c2nc(C3CC3)nc(=N)[nH]2)CC(NC(C2CCCC23CC3)=O)CC2(CC2)C1 c1(C(CC)NCc2nnc(-c3cccc(C)c3)o2)ccc([N+](=O)[O-])cc1O N1(C(C2CCN(CC)CC2)=O)CCC2(CCN(C(=O)CN3CCCC3C)C2)C1 Cc1ncsc1CCC(=O)NCC1(O)CN(CCOCF)C1 N1(C(c2ccc3c(n2)NCCO3)=O)CCOC2(CC1)CCS(=O)(=O)C2 c1(C(N2C(C(N3CCC(F)CC3)=O)CCC2)=O)cc(OC(F)(F)F)cc(Br)c1 N1(C(c2ccc(C(C)C)nn2)=O)CCN(C(=O)CCC(=O)NC2CC2)C2CCC12 c1(C(=O)NC(C)CC(C)NC(=O)Cc2ccc(Br)cc2)cc(O)cc(C#N)c1 CCCCCCCC(F)C(=O)NCC(C)(CNC(c1c[nH]nc1CCC)=O)OC C1(CC=C)(NC(CCCCCF)=O)CCN(C(=O)C(c2ccn(C)n2)C)C1 C1(C(=O)NC(=O)Nc2ccc(CC)cc2)CCN(c2nnn(C)n2)CCC1CO C(=O)(C(C)(C)CSC)N1CC(OCCNC(c2nc(C(C)OC)sc2)=O)C1 Cc1[nH][nH]c(=N)c1C(=O)NC(C)CN(C)C(c1ccc(C(C)C)nc1)=O C(=O)(CS(=O)C(F)(F)F)N1CCC(C(C)NC(C2(OC)CCSC2)=O)CC1 C12(CNCC(C3CC(F)(F)C3)OC)COC(CCO1)C2 C(CN=c1[nH]c(N2CCCOC(CCO)C2)nc2cccc(F)c12)OC C=CC(C)(CCOC)C(=O)NCCN1CCN(C(c2cc(CC)n(C)n2)=O)CC1 c1(NC(c2nc(-c3ccc(OCCC)cc3F)sc2)=O)c(O)cccc1[N+](=O)[O-] n1(CCC(=O)NC(C)CNC(C2(C)COCCO2)=O)cc([N+](=O)[O-])cn1 N(C(=NCC(C)C)NC1CC1)CCc1cc(OC)c(NC2CCCC2)cc1 N1(C(CCN(C(=O)CC2CCCOCC2)CCO)=O)CCC2OCCC2C1 Cn1cc([N+](=O)[O-])c(C(N2CC(Cn3cc(CN4CCCOCC4)nn3)C2)=O)n1 c1(CC(=O)NCCN(C(=O)CC2OCCCO2)C)ccc2c(c1)CCOC2 C1(CCNC(COC)=O)CSCCN1C(c1cccc(N2CCCC2=O)c1)=O C1(C)(CNC(CCOC)=O)CCN(C(c2ccc(C(O)CF)cc2)=O)C1 C(CNC(c1cscc1-c1ccccc1)=O)(C(C)C(C)C)NC(C(C(C)C)O)=O CCC(CC(=O)N1CCC(N(C(c2ccc(C)c(Cl)c2)=O)CC2CC2)C1)C(C)C CCCCN=c1ncc(-c2nccn2CC2CN(C(N)=S)C2)c[nH]1 C=C1CC(C(=O)NC23CC(F)(C2)C3)(CNC(C2CS(=O)C2)=O)C1 c1(OC)ccc2c(C(=O)NC(C)C(C)(C)NC(C3CC3C(N)=O)=O)coc2c1 c1(CC(N2CCC(CN(C(=O)Cc3cncn3C3CC3)C)C2)=O)cccc(O)c1 c1(C(=O)NC2CN(C(C(C)SCC)=O)C3(C2)CCC3)cccc(C)c1[N+](=O)[O-] C1(C(=O)NCC2CCC(NC(COCCOC)=O)CC2)CC12CCS(=O)(=O)CC2 c1(CC)nnc2cc(N3CCC(C)(NC(=O)C(c4csc(C)n4)=O)CC3)ncn12 N1(CC(=O)N(CCC(=O)NCc2ncsn2)C(C)C)C(C)CCC1C C(=O)(C(CC(C)(C)C)OC)N(CC(C)(O)NC(=O)Cc1ncoc1C)CC c1(C(C)C)ccc(CCC(=O)NCC=CCNC(C2CC(F)C2)=O)cc1 C1(C(=O)OC)(C(=O)NC2CC(NC(C3CC4C=CC3O4)=O)C2)CC1S(N)(=O)=O c1(NC(C2CCN2C(=O)CCc2ccco2)=O)ccc(CCO)cc1 Cc1cnnc(O)c1C(=O)NC1CC(C)(NC(c2cnn(C3CC3(F)F)c2)=O)C1 c1(C(=O)NCC(C2CCCC2)NC(Cc2cc(C(C)=O)sc2)=O)c(C)csc1Cl C1(NC(=O)COCCCC(=O)NC(c2ccnn2C)C)CC(C2CC2)C1 c1(C(=O)NCCCCCC(=O)OCc2ccccc2)ccc2[nH]nc(Cl)c2c1 Cc1ccn2cc(C(=O)NCC(O)CNC(=O)CC(C)CC(F)(F)F)nc2c1C N1(C(CC(=C=C)C)=O)CCCCCC1C(=O)N(C(C)C(N)=O)C N1(C(Cc2nc(CC)sc2)=O)CC2CS(=O)(=O)CC2(NC(=O)CCCF)C1 c1(C(=O)NCCCN(C(CN(C2CCCC2)CC)=O)C)cccc(N)c1 N1(C(CC=CC)=O)CCCCC(NC(=O)CCP(C)(C)=O)CC1 C(=O)(CC(C(C)C)C(C)C)Nc1ccc(-c2ccc(OCCC)nc2F)nc1 N1(C(c2cc(C(=O)OC)no2)=O)CCSCC1CCNC(=O)CCCSC C1(C)(NC(C=Cc2c(C)ncs2)=O)CCCN(C(c2ccco2)=O)C1 CC1CC(CNC(c2ccc(F)c(Br)c2)=O)CCN1C(c1ccon1)=O N1(C(C2CC(SC)C2)=O)CC2(CCN(C(=O)CC(O)C3CCCC3)CC2)C1 N1(C(C2(C)CCCCC2)=O)CC2CC1CC2NC(=O)Cn1cncn1 Cc1ccc(Br)cc1CC(=O)NC1(CNC(=O)C(CCO)N2CCC2)CCC1 N1(C(CCn2c(C(C)C)ncc2)=O)CC=CC(NC(=O)CSc2cccs2)C1 c1(CC)c(OC)cccc1C(=O)NCC(CO)NC(=O)CCF c1(NC)ccc(C(=O)Nc2cccc(NC(=O)Cc3ccn(C)n3)c2)nc1 c1(C(=O)OC)cc(C(=O)NC2CC(CNC(C3CCCC3(F)F)=O)C2)ccn1 CCCC(C(F)(F)F)NC(=O)C(=O)CCNC(=O)C(CN(C)C)CC C1(NC(=O)C(CO)c2ccccc2)CCOCC1C(=O)NC12CC(F)(C1)C2 C1(C(=O)NCC2(N(C)C)CC2)(CNC(c2cccc(C3CC3)c2)=O)CC12CCC2 Cc1ccncc1CC(=O)NCCC1(O)CN(C(c2cc(N)ccn2)=O)C1 C1(C(N2CCOCC(CNC(CCC3C(C)C3)=O)C2)=O)CS(=O)(=O)CC(=O)N1 C(CC(C)C(=O)NC(CN=[N+]=[N-])C(=O)N(CC1=CCSC1)C)=CCC CC1CN(C(=O)C(O)CN2CCCC2)CC1CNC(=O)C(C)(C)C1CC1 c1(CNC(CCCC)CC)cc2c(Br)cc(OC)cc2[nH]1 N1(C(C2(C=C)CCC2)=O)CCCC(C)(CNC(=O)CCOc2cccc(Cl)c2)C1 N1(C(=O)OC(C)(C)C)CCC2(CC2NC(c2cnn3c2CCC3)=O)C1 c1(C(=O)NCC2(F)CC(NC(c3c(C)nsc3)=O)C2)cccc(CO)c1 C1(C#N)(C(=O)NCC2(NC(C3C(C)C3)=O)CCC2)CCC(=O)CC1 N1(C(COc2ccc(-c3nc(C(=O)OC)c(C)o3)cc2)=O)CC(C)OCC12CCC2 N1(C(C2(C)CCN(C(C3C(C=C)OCC3)=O)C2)=O)CC2CCC(C1)N2C N1(C(c2nc(C)sc2)=O)CCOCC12COCCN(C(C1COC(=O)C1)=O)C2 CC1(C)OCCC1C(=O)NC(CNC(c1ncncc1F)=O)Cc1ccccc1 Cc1cccc(C(=O)NC2CCCC(NC(C3CCCS3)=O)C2)c1Cl N1(C(CC2CN(C)C2)=O)CCN(C(C2(O)CCCCCCC2)=O)CC2(CC2)C1 c1(C(=O)NCC(CNC(Cc2nc(C)[nH]n2)=O)C)c[nH]cc(Br)c1=O C=CCC(CC=C)C(=O)N1C2CCC1CC(CNC(C13CCCCC1C3)=O)C2 N1(CN)CC2CN(Cc3ccn(C4CC4)c3)CC2C1 C1(CNC(CNC(C)=O)=O)CCCN1C(=O)Cc1ccoc1C c1(C(N2CCC(C(C)NC(=O)C(C)(C)C(F)F)CC2)=O)cncc2cccnc12 C(c1cccc(F)c1Cl)=CCNC1(CO)CCC(C)C1 N1(C(C(=O)OCC)C)CCN(C(C2CCCN2C(=O)C(C)CC)=O)CC1 N1(c2nccc(C)n2)CC(NC(=O)CCc2cncc(F)c2)C2CCCCC12 c1(NC(c2nccc(C)c2)C)nccc(=NC(C)COc2ccc(C)c(C)c2)[nH]1 CCCC(CNC(=O)CSCC)C(=O)NCC(c1cccs1)O Cc1nc(N(C)C)sc1C(=O)NC1C=CCN(C(c2n[nH]cc2Cl)=O)C1 Cc1oc(C#N)cc1C(=O)NCC(C)(C(C)C)NC(=O)CCCC(=O)NC(C)C N1(C(c2nc(CC)oc2)=O)CCCC(C(C)(O)CNC(c2ncn(CC)n2)=O)C1 n1(CCC(N2CC(c3cccc(C)n3)C2)=O)ccn2nncc2c1=O C=CCCC(C(=O)OC)NC(=O)C(CNC(=O)C#CC1CC1)C(C)C c1(NC(C(c2cn(CCC)nc2)N(C)CC)=O)nccc(OC)c1OC c1(NC(C2CC(F)CN(C(C3CCC(F)(F)C3)=O)C2)=O)cccc(S(=O)(=O)O)c1 N1(C(c2ccc(C)s2)=O)CC2(CC(NC(=O)C(C)(C)C)C2)C1 C12(OC)CCN(C1)C2=O.c1(C(=O)OC)ccc(CC2CC2)s1.C1CO1 CCC(CNC(c1cncs1)=O)(CC)NC(=O)Cc1nc[nH]n1 N1(c2cc(N(CC(N3CCOCC3)=O)C)ncn2)CCCC(NCCO)C1 c1(C(=O)NCc2ccc(F)cc2)ccc(C(F)F)cc1-n1cccn1 C=C(Cl)CC(C(=O)NCC12CCC(CC1)C2)NC(c1cccn1CC)=O c1(CC)nc(=N)[nH]c(=NCC2CCCC(NC(C3(c4ccncc4)CC3)=O)C2)[nH]1 CC(C)C(O)CC(=O)NCC(CNC(c1ccc(N2CCOCC2)nc1)=O)CO S(=O)(=O)(c1cc(C)cnc1NCC1(C)CCN(C)CC1)NC(CSC)C Cc1ncnc(C)c1CC(=O)N(CCCNC(C1CCCN1C)=O)CCO C1(NC(C(C=C)O)=O)COCCN(c2nnc(C(N)=O)s2)C1 C(=O)(CCCN(C(=O)C=CC(C)NC(=O)C(c1ccccc1)O)C1CC1)NC CC(C)CCCC(C)C(=O)N(CC(N1CCC(CCN(C)C)CC1)=O)C N1(C(C(C2(O)CN(C(C3C(C)CCO3)=O)C2)F)=O)CCCCCCCCC1 C(=O)(C1=CCC(NC(c2cnn(C)c2C#N)=O)C1)NCCC(CC)C C1(N(C(CC)=O)CC(=O)OC(C)(C)C)CC(=O)N(n2c(C)csc2=O)C1 CCC(C)C(C(=O)N(C)Cc1csc(=N)[nH]1)N(C)C(C1CC(O)C1)=O C12(C(=O)NCc3cn(CC4CNC(=O)O4)nn3)CCCN1CCC2.NC(=O)C1CS1 C(=O)(CCCCC(C)(C)C)NC(C(=O)NC(CCC(=O)OC)C(C)C)C1CCCC1 CC1CCN(C(=O)C(C)C2CCC2)CCN1C(=O)COc1c[nH]nc1Cl c1(C(=O)NCC(CNC(c2cc(C)nc(Cl)c2)=O)O)cc2c(F)cccc2s1 Cc1ncc(Cl)cc1C(=O)NC(C)CNC(c1cc(-c2csc(CO)n2)c[nH]1)=O N1(C(c2ncc(F)cc2F)=O)CCCC2(C1)CN(c1ncnc3ccsc13)C2 C1(CNC(C(C)(C)C)=O)CC2(CCN(C(=O)C3=CCCC3)C2)CO1 Cc1cnn(C)c1C(=O)NCC1CC(NC(=O)C(c2ccccc2F)C)CCO1 C12=NC=C(Br)C(=NCC34CC(CO3)(C4)NC1=O)N2.c1(C(C)C)cc2n(n1)CCO2 c1(NC2CC(O)C2)nc(=NCC2CCCN2c2ccccn2)[nH]c2c1COCC2 C1(CCNc2onc(C)c2Cl)(NC(c2ccc(N(C)C)cc2)=O)CCN(C)CC1 Cc1cnc(C(C)NC(c2cc(CNC(=O)Cn3cncn3)cs2)=O)s1 CC(C)C(CCC(=O)NC(C)Cc1ncn(C)n1)NC(C1CCC(C)(C)OC1)=O CCCCCC(O)C(=O)N1CSCC1C(=O)NCC1CC(O)C1 C(=O)(NNC(=O)CCC(C)N(CCOCC)CC)NCC.C12(CCOC1)C(=O)O2 C1(NC(CCCCCC)=O)CCN(C(=O)CC2OCCC2(C)C)C(C)(C)C1 c1(C(=O)NC2CN(C(c3ccnc(Cl)c3O)=O)CC23CC3)ccnc2c1CCC2 N1(C(c2c(C(C)C)occ2)=O)CCC2CN(C(=O)CNC(N)=O)CCC12 C(C(C)(CC(C)C)NC(C1C=CCC1)=O)OCC(=O)Nc1c(OCC)cccc1 Cc1ccc(C(N2CC3CC3(CNC(=O)CC3CC3(C)C)C2)=O)c2c1CCC2 N1(C(C2(NC(c3cc(C)ncc3)=O)CCCC2)=O)CCCC(C)C1CO CC(C)(C#N)CCC(=O)N1CC(C(N2CC(C)(F)C2)=O)C(F)(F)C1 Cc1ccc2c(C(N3Cc4cccc(CNC(=O)C(F)F)c4C3)=O)ccnc2c1 Cc1csc2nc(C(=O)NCC(O)CNC(=O)CC3CCC4(CCC4)CO3)cn12 CC1(C)CC(C(=O)NC2(CCC(N3CC(F)(CO)C3)=O)CCC2)=NO1 C1(O)(CNC(C(C=CC)O)=O)CC2CCC(C1)N2C(=O)Cc1ccc(O)cn1 N1(C(C(CC)(C)C)=O)CCCCCC(NC(=O)Cc2cncnc2O)C1 CC#CCCCC(=O)N(C)CC1CC(F)CN1C(c1cnc(C2CC2)nc1C)=O c1(CNC(CC2(C)CCN(C(c3ccc(CO)cc3)=O)C2)=O)ccc(F)nc1F C1(N(C(CCN(CCC)C)=O)C)C2CN(C(c3cc(CC)n(C)n3)=O)CC12 CCCCCC(CC)C(=O)NCC=CCC(N1CCC2(CCC(O)C2)C1)=O C1(CC)(CC)CC(NC(C2CC(C(C)C)=NO2)=O)CN1C(=O)CC(F)(F)F C(CC1=CCN(C(=O)C=CC(N)=O)CC1)N(C(Cn1cc(C(C)O)nn1)=O)C1CC1 c1(NC(CCC)COCC)cc(S(=O)(=O)NC(CC)CC#N)ccc1C#N CC1CCN(C(=O)Cc2csc(C(F)(F)F)n2)CC1NC(c1n[nH]cc1Cl)=O C1(C(N2C(CNC(C34OC(C)C(C3)C4)=O)CCCC2)=O)C2CC3CC(C2)CC1C3 c1(OC)ccc2c(c1)CCN(C(c1cc3n(c1)CCOC3)=O)C2 N1(C(COC)OC)C(=O)CCN(CCC2CCN(C(C3CCCO3)=O)CC2)C1=O C1(CC=C)(C(=O)NCC(C)(C)CN(C)C(C2CC2c2cccs2)=O)CCCCC1 C12(NC(=O)C=CC3CCC3)CCCC1CN(C(=O)C(F)(F)C1CCOCC1)C2 Cc1nc(Cl)ccc1NC(C1(NC(C2CCOC2(C)C)=O)CCCC1)=O C1(CNC(CC2CC(OC)C2(C)C)=O)CN(C(=O)CNC(=O)COC)CCCO1 c1(SC(C(=O)NC2C(CNC(CCSC)=O)CCC2)C2CC2)ccc(C#N)cc1 c1(C(N(C)CC2CCN(C(c3cn(C)nc3C(N)=O)=O)C2)=O)ccc(CO)c(F)c1 C1(C(=O)NCC(CN(C(C=CC)=O)C)C)CCc2n[nH]c(C)c2C1 C1(N=c2[nH]nc(-c3ccccc3)s2)(CNC(C(C)CS(C)(=O)=O)=O)CCCC1 C1(C(N(C2CC(NC(c3cncc(C)n3)=O)C2)C)=O)CCCN(CP(C)(C)=O)C1 c1(C(=O)NCCC(CCNC(C(C(C)C)SCC)=O)C)ccc(C#N)c(C)n1 C1(C(=O)NC(C2CCN(C(c3ccc(C(C)C)cn3)=O)C2)C)CCC(F)(F)CC1 N1(C2CCN(C(CCNC(C)=O)=O)CC2)CCN(C(=O)C(F)C(C)C)CC1C C(=O)(CC(C)CC(=O)OC)N1CCCC(CCC(=O)N(CCCN(C)C)CC)C1 C12(C(N3CCCC(N(C(=O)COCc4nc[nH]n4)C)C3)=O)CCN(C1)S(=O)(=O)C2 c1(C(N2C(C(=O)NCC3CCCCC3)CC(O)C2)=O)cccc(Br)c1F O=C(C1=CCCCCC1)NCCC1CCN(C(=O)C=Cc2cocn2)C1 c1(C(=O)NCC2CN(C(C3(CC(F)F)CC3)=O)CCO2)c[nH]c2cccc(F)c12 Cc1cc(C(N2CCCC(NC(C3CC4(CC4)C3)=O)CC2)=O)c2[nH]cnc2c1 CC(C)(C)CC(O)CC(=O)N1CCC(C2CCCCN2C(=O)C=CCO)CC1 c1(C(=O)NC2CCCC(CNC(CSCCC)=O)C2)ccc2c(=N)[nH]cnc2c1 C1(CNC(C2CCCN2CC(F)(F)F)=O)COCC2(CCNC2)O1 c1(C(N2CCCC3(NC(=O)CC(F)(F)F)C(C2)C3)=O)cc2nc(F)ccc2o1 C1(CNC(CC2OCC(C)(C)C2)=O)CN(C(c2sccc2C#N)=O)CC12CC2 c1(OC)cc(F)c(C(=O)NCC2CCCC2NC(c2snnc2C)=O)cc1N c1(CC(N2C3C(NC(c4nc(OCC)sn4)=O)C(C3)C2)=O)nc2ccccc2s1 C12(CNC(CC(C)(C)N(C)C)=O)CCC1CN(C(=O)CN(c1ccccc1)C)C2